SMILES N1(C(C(Cc2cc(C)[nH]n2)NC(=O)OC(C)(C)C)=O)CCC(C)(F)CC1 c1(C(N2CC(O)(CCNC(C3N(C)CCCC3)=O)C2)=O)ccc2c(c1)CCC2 c1(N2CCC(CC)(CO)C2)ncnc(NN(CC(N2CCCC2)=O)C2CC2)c1C C1(OC)CN(C(=O)CN2CCC(C)CC2)CC1NC(C1CCCN(C(C)C)C1)=O Cc1nn(C)nc1C(=O)NC1COCC1CNC(=O)CC(C)c1ccccc1 C1(O)(C(C(=O)NC(c2cnsc2)C)NC(CCCOCC=C)=O)CCCCC1 C(=O)(N=c1[nH]c(Cl)c(I)nc1Br)C1N(C(c2cccc(N)c2)=O)C2C(C1)C2 c1(C(=O)NCC=CCNC(C2C(C)(C)CC2)=O)ccc2cc(Cl)ccc2n1 C(=O)(C(C(C)O)N(C)C)NC(c1cn(CCCOC(c2cccs2)=O)nn1)C(C)C c1(NCC(C(CC)C)OC)ccc(S(=O)(=O)NCC2(CC#N)CC2)c(Br)c1 c1(C(C)C)cc(C(=O)NC2CCCC(NC(=O)CN(CC(C)(C)C)C)C2)nn1C Cc1nccnc1C(C)NC(C1CSCN1C(c1c[nH]nc1Cl)=O)=O Cn1cnnc1CCC(=O)NC1CCN(CC(F)(F)F)C1.C12CCN1C2=O N1(C(CSCCC#N)=O)CC(NC(=O)C=Cc2cncs2)CC(F)(F)C1 c1(C(N2CCCCC(Nc3c(C#N)c(Cl)ncn3)C2)=O)cc2cccc(F)c2o1 Cc1cc(-c2cncc(C(=O)Nc3nc(C4CC4)c(Br)s3)n2)cc(C)c1 C1(C(=O)OC)CC(C)N1C(=O)CCC1(NC(C2CCC2C)=O)CCC1 CCC(CN=c1[nH]c(=NCC2=CCCC2)[nH]c2ccc(Cl)cc12)n1cccn1 c1(OC)cc(Cl)ccc1CN=C(NC(C)C)NCC12CC(CN1C1CC1)C2 C1(O)(C(=O)NC2CN(C(c3c(OC)c(C)cs3)=O)CC2O)CCC(C)(C)CC1 c1(CC(=O)NC2C(C)CCN(C(C(C)=C3CCC3)=O)C2)nnc2n1CCOC2 N1(C(=O)NC(C)Sc2nnc(C3CC3)n2C)CCn2ncc(C(F)(F)F)c2C1 C(=O)(CC(O)C(C)C)NC1(C(=O)NCc2ccn(CCC)n2)CC(F)(F)C1 c1(CC(C)C)ncc(C(=O)NC(C)(C)CNC(C2CC2(F)Cl)=O)s1 c1(C(=O)NC23CN(C(c4c(CC)c(C)ccc4)=O)C(C2)C3)cc2ccccn2n1 C1(NC(c2cn(CCC(C)C)nn2)=O)CN(C(=O)C=Cc2ccoc2)CC12CC2 c1(CC)cncc(C(=O)NC2COCC2CNC(=O)C(C)(C)C)c1 c1(C(=O)NCCCC2CCN(C(C(OC)OC)=O)CC2)cn2ncccc2n1 Cc1csc2c(N3CC(C(C)NC(=O)Cc4cccs4)C3)ncnc12 N1(C(c2nccnc2Cl)=O)CCC(NC(C2(F)CCC2)=O)C(F)C1 N1(C(CCC=C)=O)CCC2(C=C(C(=O)NCC3(N(C)C)CCCC3)C2)C1 O=C(CCCSc1ccccc1)NCCCN(C(=O)Cc1cccnc1)C1CC1 CC1(C)CC(NC(C2CC(O)C2)=O)CN(C(c2cc(N)cc(F)c2Br)=O)C1 N1(C(C2=C(C)OCCC2)=O)CC2CCCCC2(NC(=O)C=C(Cl)Cl)C1 c1(OC)ncc(F)c(N(C2CC3(CNC3)C2)C(c2cc(F)c(C)s2)=O)n1 C1(C(N2CCCC(CC(=O)NCC(c3ncon3)C)C2)=O)CCCC1C1CC1 N1(C(C2(CC)CC2(F)F)=O)CCCN(C(=O)C(C)(F)CC)CC1 CCC(C)(COC)CNC(=O)CCC1(C)CN(C(c2ncncc2OC)=O)C1 c1(C(=O)NC(C2CN(C(=O)C(C)(F)C(C)(C)F)CCO2)C)cnc2ccnn2c1 C1(C(N(C2CCC2O)C)=O)CCCN(C(c2cnnc(O)c2)=O)C1 CS(=O)(=O)c1cncc(C(=O)NC2CCCN(C(C34CCC3C4)=O)C2)c1 N1(C(COC(CC)(C)C)=O)CCC2CCN(C(c3c(O)cc(F)cc3F)=O)CC2C1 N1(C(C)C(N)=O)CCC(CCNC(c2ccc(-c3cnn(C)c3)s2)=O)C1 c1(OCC(=O)OCC)cc([N+](=O)[O-])ccc1NC(c1ccc(Cl)cc1)C N1(C(CCOC)=O)CCC(O)(C(=O)NC(Cc2ccccc2)C(=O)OC)CC1 C1(C(N2CC3C(CNC(c4cc(C)sc4)=O)(C3)C2)=O)CC2(C1)CC(C)C2 c1(CNCc2cn(-c3c(C)ccnc3)nn2)ccc2nnnn2c1 N1(C(CNC(C)=O)=O)CCC(NC(=O)Cc2scnc2-c2ccccc2)C(F)C1 Nc1cc(C(=O)NCC2(NC(=O)CC3(O)CCC3)CC2)cc(F)c1 C1(CC(=O)NCc2cc(C(=O)NCC3(O)CCC3)ccn2)CC(=O)NC1=O N1(C(CNS(NC)(=O)=O)=O)CC(CNC(=O)Cc2nonc2C)N2CCC1C2 c1(OC)ccc(Cl)c(C(N2CC(N(C)C(C3CCCN3C)=O)C3(CC3)C2)=O)n1 c1(OC(F)F)cc(CCNc2ccnc(OC)c2)cc(F)c1OC.CO CC1(C)C(NC2CCC23CCC3)CC1O N1(C(C2(CCC)CC(=O)C2)=O)CC2(CC(CC(=O)NCC(C)C3CC3)C2)C1 C(C(CC(=O)NCC1C2CCCC12)NC(=O)CN1CC(=O)NC1=O)OC CC1=NOC(C(N2CCCC2C(C)(C)CNC(C2(N3CCOCC3)CC2)=O)=O)C1 C1(C(=O)NCC2(O)CCN(C(CP(C)(C)=O)=O)C2)CC1C1(C)COC1 N1(CC(=O)NC(C(C)C)CNC(C2CC(C)(F)C2)=O)CCNC(=O)C1 S(=O)(=O)(c1cnc2ccccc2c1)N(C1CCCC(C)C1)C C1(C(=O)NCC(C)(C)SC)CCN(C(c2ccc3[nH]ccc3n2)=O)CC1(C)C N1(C(=O)OC(C)(C)C)CCCC(COCC(N2CCC3CC23)=O)C1 c1(C(=O)NC(CC)CN(C(=O)CC2CC(F)C2)CC)cnn(-c2ccncc2)c1C CC1CC(NC(C2(C)CCN(C)C2=O)=O)CCN1C(=O)Cc1cc(Cl)cc(Cl)c1 C(=O)(C(CCCCN)CC(F)(F)F)N1CC(NC(Cc2cc(C)on2)=O)C1 C(C(N=c1[nH]c(C2CC2)nc(Cl)c1C)C(C)C)NC(C(CC)(CC)C(C)(C)C)=O N1(C(C(CC#C)O)=O)CCCC2(CCN(C(=O)Cn3nc(O)ccc3=O)C2)C1 C1(NC(C(C)(N(C(c2nc(OCC)oc2)=O)C)C2CC2)=O)CC2COCC2C1 c1(CN2CCC3(C(C(=O)NC(C(=O)NC)C)C3)C2)c(OC)cc(Cl)cc1F C(CCN=C(NCc1ccc(SC)o1)N1CCC(C(F)(F)F)(CO)C1)OC Cc1ccc(N2CCCC2C(N2CC(N3CCNCC3)C2)=O)cc1 N1(C(C(C)C(F)F)=O)CC2CC(C1)C(CO)C2NC(C1C2C3CCC(C3)C12)=O C(=O)(C(C#N)C(C)(C)C)NC(C)(C)CCNC(=O)Cc1cncc(O)c1 N1(C(c2c(C)cc(F)cc2)=O)CC(C)N(C(c2cc(Br)c(Cl)cc2C)=O)CC1C C(C1=CCN(C(C2CCCC23CCC3)=O)CC1)NC(=O)CCC1CCOC1 c1(C(N(C2CCN(C(=O)CC3CC34CC4)C2)C)=O)ccnn1CC1CCC1 CC1CCN(C(c2csc(CNC(C3(N4CCCC4)CC3)=O)c2)=O)CCO1 C1(C2CCN(C(=O)C(C)(C)CS(C)(=O)=O)CC2)(NC(C(CC)CCOC)=O)CC1 N1(C(c2c(CC)c[nH]c2)=O)CC2CCN(C(=O)C(CO)NC(=O)C(F)(F)F)CC12 C1(C(=O)NCc2occ(C(N3CCC(N(C)C)(CC)C3)=O)n2)CC2COCC2C1 N1(Cc2c(C)nn(C)c2C)CCN(C(c2ccc(O)cc2)=O)C2(CC2)C1 N#CC1CN(Cc2cnn(C3CCOCC3)c2)CC1NC(=O)CCBr C1(NC(c2c(Cl)cn(CC)n2)=O)CC(CNC(C2SCCS2)=O)C12CCC2 C#Cc1ccc(C(=O)N(C)CCOCCNC(C2CC2CC)=O)cc1 C(=O)(CC(C)(C)C(=O)NCC1(NC(=O)CS(N)(=O)=O)CCOCC1)OCC c1(CC(C(=O)NCC(N(C(COCCCC)=O)C)C2CC2)O)ccc(Cl)cc1 C1(CCC)(NC(c2ncccc2SC)=O)CCCN(C(C2CCOC2)=O)C1 C1(C(=O)NCC2N(C(C3C(C)CCOC3)=O)CCC2)CC(=O)NC(=O)C1 C1(NC(C2C(C(C)NC(C(CC)CN(C)C)=O)C2)=O)CC2(CCCCO2)C1 CCC(C)CCCC(=O)NC(C1CCCN1C(c1cccc(C#N)c1C)=O)C Cc1ccc2c(CCNC3CCCN(c4ncnc5ccsc45)C3)cn(C)c2c1 C=Cc1cc(C(=O)NCC2CC2N(C(c2cc(C3CCC3)on2)=O)CC)cc(F)c1 CC1CCCC(C)N(C(c2conc2CNC(=O)C(C)n2cccn2)=O)C1 C1(C(=O)NCC(=C2CN(C(C3(CC=C)CC3)=O)C2)F)CCCCN1CC c1(C(N2C(CNC(CC(C)OC)=O)C(C)(C)CC2)=O)cccc2c1C(=O)CC2 c1(C(N2CC(O)(CN(C(c3ccc(C(C)=O)cn3)=O)C)C2)=O)cc(O)nc(O)n1 CC(O)C(=O)NNC(=O)NCc1cccc(F)c1I C1(NC(C2N(C(C(NOC)=O)=O)CCOCC2)=O)CCOCC12CCC2 N1(C(C(C(C)CC)N(C(CC=CC)=O)C)=O)C2CCC1CC1(CC1)C2 c1(C(=O)NC(C(C)C)C)sc(Br)cc1Br C1(CC(=O)NC(CNC(C2(CSC)CC2)=O)C(C)C)CCCCCO1 C1(NC(C2C(C(=O)OC)C2)=O)C2COCC1CN(C(c1n[nH]cc1C)=O)C2 C=CC1CN(C(C2C3CC4C(C3)C24)=O)CC1NC(=O)C(C)CC(N)=O CC1(C(N2CC(OCCNC(c3ccnc(C4CCC4)c3)=O)C2)=O)CC=CCO1 CC(C)=C=CC(=O)NCCCN(C(=O)CC(C)C)C1CC1 C1(SCC)CCC(C(N2CC(c3cn(C4CCCC4C(=O)O)nn3)C2)=O)CC1 CCC(CC)(CO)C(=O)NCCC1CN(C(c2cc(Br)n(C)c2)=O)C1 CC(C)(C)C(C(=O)Nc1cccc(NC(=O)C2=CCCS2)c1)c1cc[nH]n1 C1(NC(=O)OC(C)(C)C)CC(Nc2cnn(-c3ccncc3)c2)C12CCC2 N1(C(Cc2cc(C)sc2C)=O)CCN(C(=O)CNC(c2cccs2)=O)C2CCC12 C(=O)(C(C)CCCCCC)N1CC(C(N2CC(C#C)(F)C2)=O)C(C)(C)C1 c1(C(=O)NCCN(CCC)C(C2CCC(C)C2)=O)csc(-c2cnc[nH]2)n1 C1(C(N(C(CCCC)C)C)=O)CN(C(=O)Cc2c(C)cnn2C)CCN1C c1(OC)c(Cl)cc(C(=O)NC23CCCC2CN(C(c2cnccn2)=O)C3)nc1Cl Cn1cnc(CCC(N2CC(O)(C(C)(C)CNC(=O)CCc3ccc[nH]3)C2)=O)c1 CCCC(CCCNC(c1cc(CC)nn1C)=O)NC(c1coc(C(N)=O)c1)=O N1(C(C)=O)CCCC1(C)C(=O)NCC1(O)CCN(C(=O)CCCC2CC2)C1 C#Cc1c[nH]nc1C(=O)NCC1CC(F)CN1C(c1ccoc1Cl)=O c1(C(=O)NC(CC=C)CNC(c2ncn(CC)n2)=O)ccc(C2CC2)cc1C c1(CC)ccc(C(=O)NC2CCC(C)N(C(c3cc(C)ns3)=O)C2)cc1CC N1(C(c2nn(C(C)C)nc2Br)C(=O)NCC=C)C2CCC1CC(C)C2 c1(N2C(CNC(C(C(CC)O)C)=O)CCC2)nc2c(F)cc(Cl)cc2s1 C(CC(CC)C(=O)NCC(O)CC(=O)NC(C)C(C)C(=O)OC)=CC C(=O)(CCCC(C)(C)C)N1CC(C(=O)NCCCC(=C)Cl)C(C)C1 n1(CC)cc(C(=O)NC23CC2CN(C(C2CCN2C)=O)C3)c(C)n1 c1(C(N2CC(CCNC(C(CC)(C)CO)=O)C2)=O)ncc(P(C)(C)=O)cn1 C1(N(C(c2coc(Cl)n2)=O)CC)CCCN(C(=O)Cn2ncc(Cl)c2C)C1 c1(C(=O)NCC2C(C)CCN(C(=O)C(C)(C)CO)C2)ccc(S(N)(=O)=O)nc1 C(=O)(C(C)(C)C1=CCSCC1)N(CC(C)(C)NSC1CCCC(C(=O)OC)C1)C CCCC(CCCNC(=O)CC1CCCO1)NC(C1(C(F)F)CCCCC1)=O CC1(C)CCCOC1C(=O)NC1CN(C(=O)Cc2ccc(Cl)cc2)CCC1CO CCC(CC)C(c1nnnn1C(C)CC)NCc1cscn1 CC1OC2(CNC(C3CC3(Cl)Cl)=O)CC1(NC(=O)COC1CCCC(C)C1)C2 CN1C(C(N)=O)CCC1C(N1CCOC(CCNC(c2cnc[nH]2)=O)C1)=O C1(CNC(CC(C)(C)NC(=O)CCNC(=O)CO)=O)CC2(CCCO2)C1 c1(C(=O)OCCN2CCN(C(c3c(OC)ccs3)=O)CC2)cc(F)c(Cl)c(Cl)c1 C#CCC(CC(=O)NCCC(C)(C)COC)NC(=O)C=CCOC c1(C(=O)NCC2CCC(C)CN2C(=O)Cc2ccon2)cncc2ccccc12 CC1CN(C(=O)CC2CC(=O)C2)CCN1C(c1c[nH]nc1-c1ccco1)=O c1(C(C(=O)NC2CCCCC2)N(C(c2ncc[nH]2)C)CC)ccc(S(N)(=O)=O)o1 c1(CC)nc(C)oc1C(=O)NCC(=O)NCC(=O)NCC(O)CO C1(C(N2CC(O)CC(NC(C(CCSC)(C)C)=O)C2)=O)CCc2c[nH]nc2C1 c1(C(C(CN2CCC(NC(C(=O)OC)=O)C2)O)C)ccc(C(F)(F)F)cc1 c1(OC(CC)C)ccc(CN2CC3C(CNC(c4cscc4C)=O)C3C2)cc1 c1(C(=O)NC2C(NC(=O)CSC3CCCO3)C2)cc(C(F)(F)F)ccc1F C12(C(N3CC(CNC(CC4(C)CC4(F)Cl)=O)C3)=O)CC3CC(C1)CC(F)(C3)C2 C(CCCC(=O)NC(C1CC1)C1CC1)NC(CC(C)C)=O N1(Cc2cc(C(=O)OC)n(C)n2)CC2CN(C(C3CC(O)CN3)=O)CC12 C(C(=O)NC1CN(C(c2cc(CCC(=O)OC)on2)=O)CC1C)(C(C)C)OC c1(NC(C2C(NCc3cn(CC)nc3)C2)=O)cc(F)ccc1C c1(C(N2CC3OCC(NC(CC4C(C)(C)C4)=O)C3C2)=O)cncc2ccccc12 C(CC(N)=O)(C(=O)N1CCC(C)(C)CC1)NC(c1c(OC)scc1)=O C(=O)(CCCCO)N(C1(C)CN(C(=O)CNC(=O)CNC(=O)CC(C)(C)C)C1)C C1(NC(c2n[nH]c(C)c2Cl)=O)C2CC3C(C2)C13C(N1CC2CCC1CC2)=O c1(OC)ncc(NC(C23CC2CN(C(c2cncc(C#N)c2)=O)C3)=O)cc1C C=CCCCC(=O)N1CCCC1C(C)NC(C1(OC)CC(C)C1)=O Cc1ccc(Br)cc1CC(=O)NCC1CCCN1Cc1ccc(Br)cc1Br N1(C(C2(F)CCN(C(CC3(OCC)CC3)=O)C2)=O)CC(C#N)C2(CCC2)C1 C(=O)(C#CC1(C)COC1)N1CCN(C(CN(C(C2C(C)OC(=O)N2)=O)C)=O)CC1 C1(CNC(=O)C=Cc2ccco2)CC2(CCC2)CN1C(c1ncc(Cl)nc1Cl)=O c1(C(C)=O)[nH]c2ccccc2c1C(=O)NC(C1CCCC1)CNC(=O)C(N)=O N1(C(CC2(C)CCC2)=O)CCC2(CCN(C(=O)CC3(C)CCS(=O)(=O)N3)C2)C1 C(=O)(C#CC1CC(F)(F)C1)N1C(CNC(C(CCCCC)O)=O)CCCC1 C1(CCC)(NC(=O)CCc2cc(C)[nH]n2)CCCN(C(=O)CS(=O)(=O)CC)C1 c1(C(=O)Nc2c(SCCC(=O)OC)cccc2)cc(F)c(O)c(Cl)c1 C1(C(=O)NCC(CC=C)(C)C)CC(C)(C)CN1C(c1ccnc(O)c1F)=O c1(CC)ccc(CC(=O)N(CC(C)(C)CNC(=O)CCC2CCOC2)C)cc1 C1(NC(C2CCCC2)=O)COC2(CCCN(C(=O)COc3cncc(Cl)n3)C2)C1 CCCC(C)CC(C)OCCSc1cccc(NC(C)C)c1 c1(CC(N2CCC(C)C(NC(c3cc(Cl)ccn3)=O)C2)=O)cccc2ccoc12 CCCCC(CNC(c1ccc(SC)cc1)=O)NC(c1n[nH]cc1C1CCC1)=O C1(CC(=O)NCC(C)(O)C2CCC2)C2CN(C(c3csc(Cl)c3)=O)CC12 CC(C)CC(O)C(C)C(=O)N1CCC(C(=O)NC2(c3cc[nH]n3)CC2)(C(C)C)C1 N1(C(C)C)CCCC1C(=O)NC1CCC1CNC(=O)Cn1cnnc1 c1(C(N2CCOCC(NC(C(CC)(C)C)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 c1(OCCC(=O)NCC=CCNC(CSCC)=O)ccccc1F N=c1[nH]cnc2c(C(N3CCCC(NC(=O)C=CC4CC4)CCC3)=O)cnn12 c1(OC)cc(Br)ccc1CCC(=O)NC1CN(C(=O)CNC(C)=O)CC1C Cc1c(C(=O)NC(C)(CNC(C2CC(C(F)F)C2)=O)CO)ccn1C c1(N2CCC(CCNC(=O)CCN3CCCS3(=O)=O)CC2)ncc2ccnc-2[nH]1 N1(C(C2C(C)OC(=O)N2)=O)CCC(F)(C(=O)NCC2CCSC2)CC1 C(=O)(CCN=C(NCCc1cnn(C)c1)NCC1CCCC1OC)NC C#Cc1ccc(NC(C2CCC(CNC(c3coc(SC)c3)=O)O2)=O)cc1 c1(COCCC(=O)N(CCn2ccc(C)n2)C)ccccc1Br CC(C)(CC(=O)NCC1CCC1NC(c1cc(F)ccc1F)=O)CC(F)(F)F C(CC(C)C)(C(=O)N1CCC(N(C)C)CC1)ONC(c1c(CCC)n[nH]c1)=O N1(C(C2(CC)CCCO2)=O)C(C)CN(C(c2nc3ccccc3[nH]2)=O)CC1C CC(C)(C#CC(=O)NCc1nc(C(C)(C)C)ns1)CNC(=O)OC(C)(C)C CC1CN(C(=O)C=Cc2cc[nH]n2)CCC1NC(=O)CN1CCNC(=O)C1 c1(C(=O)NCC2(C)CC3CC3C2)c(-c2cccnc2Br)ccc2c1OCO2 N1(C(c2n(CCC)ncc2)=O)CCCC(NC(c2cncc(C(C)(C)C)c2)=O)C1 C1(CC(=O)N(CC(CNC(c2c(C)cc(F)s2)=O)O)C)CC(C)CC(C)(C)C1 C12(CNC(C3N(CC)CCCC3)=O)CCC(CC1)CN2C(=O)C(C#N)C(C)C CC1(C)CCC(CN2CCC(c3ccccc3Br)C2)OC1 C#CCCN=C(NCC1CC(OCC)C1)NCC1CC(F)(F)C1 C1(C(C)C)CC(C(N2CC3CC2C3NC(=O)Cn2cccnc2=O)=O)CCO1 C1(CNC(C2C(CC)CCC2)=O)CC(O)CN1C(=O)CCCc1ccsc1 C1(C(N(C)CC2CN(C(=O)C=Cc3ccnn3C)CCO2)=O)CC(C)(C)CCO1 CC(C)(CNC(C1(C)CC2CCC1O2)=O)CC(=O)NCCc1ccnc(O)c1 C12(NC(C(CCCC)C)=O)CC(C)(C1)OC21CN(C(=O)CCCC(N)=O)C1 CC1=C(CNC(=O)C(N)Cc2ccc(OCC(C)C)cc2)C(C)(C)CCC1 C1(NC(C(F)=CCC)=O)CCCC(N(C)C(c2cc(Br)cn2C)=O)C1 C1(NC(CC)=O)CCCN(C(=O)N(C2CC2)CC2(C(C)(C)C)CCCCC2)C1 N1(C(c2c(C)nc(C3CC3)[nH]2)=O)CCN(C(=O)Cc2occc2C)C(CO)C1 CC1(C)COC(C(=O)NCC(C2CCC2)NC(=O)CCN2CCOC2=O)C1 CC1(C)CCN(C(C2CCC3(CCC3)C2)=O)CC1NC(=O)C1=CCCSC1 c1(C(N2CCC(CC)(CO)C2)=O)cc2c(cc1F)NC(=O)CC2 S(=O)(=O)(c1ccc(Cc2ccccc2)cc1)N1CCN(CC(CC)O)CC1 N1(C(C2CC(n3cc(C4CC45CC5)nn3)C2)=O)CC2C(C1)C2(F)F C1(C(N2CCC(OC)(CNC(c3ncccc3O)=O)C2)=O)CNC(=O)C(C)(C)C1 C(=O)(C(C(C)CC)N(C)C(c1ccncc1O)=O)NC(C#C)C(C)(C)C CCC(C#N)C(=O)NCC(C1CC1)N(C(=O)CC1CCC(C)C1)C N1(C(C2CCC(n3ccc(C#N)n3)CC2)=O)CC2COCC(C2)C1 C1(C(=O)NC(c2c(C)nns2)C)CC(C)(C)CCN1C(=O)CC12CCCC1C2 N1(C(=O)C=CSc2ccccc2)CCN(C(c2cnns2)=O)C(CC2CC2)C1 CCC(C)CC(C(=O)NC1CCCCCC1)NC(=O)CC1(N(C)C)CCC1 C1(NC(C2(CSC)CCC2)=O)CCOCC1C(=O)NCCc1ncnn1C N1(C(C2(F)C(C)C2)=O)CCCC2(CCCN2C(c2ccsc2Cl)=O)C1 N1(C(c2cc(SC)n(C)n2)=O)CCC2CN(C(C3CC3F)=O)CCC12 c1(C(=O)NC2CN(C(C=CCCC)=O)CC(O)C2)cc(F)c(F)cc1OC C1(c2cn(-c3cc(F)ccc3F)nn2)(NC(C2CSCCS2)=O)CCCCCC1 C(=O)(C1CCc2c[nH]nc21)NCC(C(N1C(C)CCCC(C)C1)=O)CC1CC1 c1(OCC)ccccc1NC(=O)C=CC(=O)NCCN(C)CC1CC2C=CC1C2 CC1CN(C(c2nscc2I)=O)CCCN1C(=O)CCF n1(CC)cnc(C(N2CCC2CC(=O)NCc2ncc(C)o2)=O)c1 c1(C(N2CC(C(C(=O)NCc3ccco3)OC)C2)=O)cncc(F)c1C C(=O)(C1CCc2ccccc21)NC1C(C)(C)C(C(N2CCC3(CCC3)C2)=O)C1 C=CC(O)C(C)(C)C(=O)N1CCCC(C)(C(=O)N(C2CCN(C)C2)C)C1 c1(C2(C(=O)NCCC(CC)O)CC(N)C2)ccccc1F CC1CN(C(=O)CC2(O)CC2)CCN1C(c1ccc(-n2cccn2)cc1)=O C12(C(=O)NC(CN(CC)Cc3ccncc3)=O)CC(c3ccccc3)(C1)C2 C(C(C)(C(=O)NCC(C)(Cn1cccn1)NC(C1CCCN(C)C1)=O)OC)OC c1(OC)ccccc1-n1ncc(C(=O)N(c2cccc(F)c2)C)c1C C(CC(C(=O)N(C)CCc1ccccc1)NC(=O)C(CC)OC)OCC C1(CCNC(C(C)OCC=C)=O)COCCN1C(c1cc(C2CCCC2)[nH]n1)=O C1(F)(C(N(CC(C)O)CC(F)F)=O)CCN(C(=O)CSC2CC2)CC1 Cc1cnc(C)c(NC(=O)C(O)C2CN(C(C3CCCC(=O)N3)=O)C2)c1 CC12CN(C(c3cnc(-c4ccoc4)[nH]c3=N)=O)CC1CS(=O)(=O)C2 C1(C(=O)NC2CC(F)(CNC(C3CCN(CC)C3)=O)C2)CCN(CC(F)F)CC1 C=CC(CCC)CC(=O)N1CCC2(C(=O)NC3C=CCC3)CCCC12 N1(C(C(C2CC2)OC)=O)CC2(NC(=O)Cc3csc(Br)c3)CCC1CC2 C1(CN(C(=O)CCSc2ccc(C)cc2)CC)CCCN(C(=O)CS(C)(=O)=O)C1 N1(C(C2(CCCC)CC2)=O)CCN(C)CC1C(N1CCC(SC)C1)=O C1(N(C(c2ccc[nH]2)=O)Cc2ccccc2)CCCN(CCCn2ccnc2)CC1 C1(CC(N2C(CNC(C3(O)CCC3)=O)CCC(C)C2)=O)CCCC2(CCC2)O1 c1(C(=O)NC(C)CN(C(=O)CCC2CC2)C)ccc(P(C)(C)=O)cn1 S(=O)(=O)(c1cnc2sccc2c1)N1CC(NC(c2cccc(C)c2)=O)C1 C12(CNC(C3(C)C(C)(C(=O)OC)CC3)=O)CCC(CC1)N(C(=O)C(C)=C1CC1)C2 c1(NC(C2C(C(=O)NC3CN(C)C3)C2)=O)ncccc1OCC(F)(F)F C(C(=O)NCC(C)(O)CNC(c1ncnn1CC)=O)(C(C)C)OCC CC(C)CC(C(=O)NCC1C=CCOC1)NC(c1cnc(S)nc1)=O C1(N(C(C23CC(C2)C3)=O)CC)CCCN(C(=O)CC(=O)N(C)C)C1 CC1CCn2cc(C(=O)NC3CCN(C(C4(C#N)CCOC4)=O)CC3F)nc2C1 CN1C(=O)CCC1(C)CNC(C1(CO)CCN(C(C2CCCC2C2CC2)=O)C1)=O c1(CS(C)(=O)=O)cccc(CNC(C2CCCN(c3ccccn3)C2)=O)c1 C(=O)(CCCS(C)(=O)=O)NCCC(C)CCNC(=O)CN(c1ccnc(Cl)n1)C CCC(CC)CC(F)C(=O)NCC1CC(NC(=O)Cc2cc(C)on2)C1 c1(CC)nc[nH]c1C(=O)NCC(C)(C1CC1)NC(=O)CCc1ccc(C)s1 C1(O)(C(N2C(C(=O)NCCC(F)(F)F)CC2)=O)CCOCC1 C12(C(=O)NCC(CC)NC(C3(SC)CC3)=O)CCN(CC1)CC2 C=CCC(C(=O)N1CC(C(N)=O)(N(C)C)C1)NC(=O)Cc1cn[nH]c1 C(=O)(C1=CCC(C)(C)CC1)N1C(CN(C(c2c(C)nsc2C)=O)C)COCC1 N(C1CCCOc2ccc(Br)cc21)C(=O)NC1CN(C)CC1c1ccccc1 C1(CC(=O)NC2C3CCN(C(c4ccnnc4)=O)C23)CCS(=O)(=O)CC1 C1(NC(c2cnc(NC3CC3)s2)=O)CC2CC(C1)N(C(C1(S(N)(=O)=O)CC1)=O)C2 C1(C(=O)NCCOCCC(=O)NC(C(CCC)O)C)CCC2(CCC2)O1 C1(CC(=O)NCC(CC)NC(c2cc(O)ccc2N)=O)CCCC(C)(C)O1 c1(C(C)C)ccc(C(N2CC(O)(CNC(c3ccc(-c4ccco4)s3)=O)C2)=O)o1 CN1CCN(C(c2cccc(CNC(=O)CSc3ccccc3)c2)=O)C(CO)C1 c1(C(=O)NCC2(C)C(C)CN(C(=O)C(C)(C)C(C)O)C2)c[nH]c2c(Cl)cccc12 c1(OC)cc2c(cc1OC)CC(C)(C(=O)NC1CC1NC(C1(CCO)CC1)=O)C2 c1(CC(C)C)ccc(CCC(=O)NCC23CC(NC(C4CC(O)C4)=O)(C2)C3)cc1 c1(C(N2CCC(NC(C(COCC)C)=O)C2CC)=O)ccc2ccsc2c1 C1(C(=O)NCC(CC(C)C)NC(c2cc(O)cnc2Cl)=O)(OC)CCC(C)CC1 C(CN=C(NCC(=O)Nc1cn(C)c(=O)cn1)NC(C)C1CC1)OCC c1(OCC)cc2ccccc2cc1C(=O)NC1CC2(CCC2)CN1C(C)=O c1(C(N2CC3CC(NC(=O)C(F)(F)F)CC3C2)C(=O)NC)ccc([N+](=O)[O-])c(Cl)c1 C(=O)(CCCCCn1cnnn1)NC1(CNC(C2C(C)C2)=O)CCOCC1 c1(OC)ccc(C(N2CCCC(CO)(NC(C3CC3F)=O)C2)=O)cc1S(C)(=O)=O N1(C(C(C)CC2CC2)=O)CCN(C)CC1CNC(C1CCOC1C(N)=O)=O N1(C(CC2CCC(NC(C3ON=C(C)C3)=O)C2)=O)CCCC(C)(C(N)=O)C1 CCCCC(CC(=O)N1CC=CCO1)NC(c1cc(C)nn1CC)=O C1(C(=O)NC2(CNC(c3nc(OCC)oc3)=O)CC2)OC2CCC1C2 C(=O)(C(C)Cc1ccccc1)NCCN(C(=O)Cc1nccn1C)CC c1(C(N2CC(NC(CCC(=O)NC)=O)C(F)C2)=O)cccc(S(=O)(=O)C(C)C)c1 c1(C(N2CC(C)N(C(=O)C(C)CN3CCOCC3)CC2)=O)cccc2occc12 C12(COCCC(=O)NCCC)CC(CC)(CN1C(=O)C(C)NS(=O)(=O)CCC)C2 C1(CN(CC(C)NC(=O)CCn2cccn2)C)CCC1C(F)(F)F C(C(F)(C(=O)N1CC2CCC2(CO)C1)C(C)C)NC(C1=C(C)CC1)=O C(C(CC(=O)N1CCOC(CC(C)C)C1)C1CCC1)NC(CNC(CC)=O)=O N1(Cc2nc(C)on2)CCN(C2CCSC2)CC1.N1(C)C(=O)N1 C(C(C(C)(C)C)NC(=O)CNC(=O)CC(F)(F)F)NC(Cc1onc(C)n1)=O C1(c2n(C(c3ccc(C(F)F)nc3)C)cnn2)CCCN(C(=O)CCC(C)C)C1 C1(CNC(C(CC=C)CC)=O)CC2CCC1N(C(=O)CC(O)C(C)CC)C2 C1(NC(c2c(CC)cc[nH]2)=O)C2CCC1N(C(=O)Cc1cnc[nH]1)C2 C1(OCC(=O)NC(C)(C)CCNC(=O)Cc2nc[nH]n2)CCCCCC1 N1(C(C(c2c(C)cccc2)C)=O)CC(F)(F)CC1CNC(C1CCSC(C)C1)=O Cc1[nH]nc(C(N2CC3(NC(=O)C(C)N(C)C(=O)OC(C)(C)C)CC2C3)=O)c1C N1(C(C2(C)CC2)=O)CCC(C2(NC(c3sc(Cl)cc3Br)=O)CC2)C1 C1(CN(C)C(C2(F)CC=CC2)=O)CCN(C(=O)CC2COCC2O)C1 O=S(Cc1ccccc1)CCNc1ccnn1Cc1nn[nH]n1 c1(C(=O)NC(C(CO)NC(c2c(F)ccc(OC)c2)=O)C)cc2c(s1)CCCC2 C1(NC(C(C)=CC2CC2)=O)CCCC1CC(=O)NC(c1ncc(C)s1)C c1(OC)n[nH]c(C(=O)N(C)CCOCCNC(C2CCC(O)CC2)=O)c1Br C1(N(C(CCOC)=O)C)CCCN(C(C2CCOC2(C)C)=O)C1 C1(NC(C2CN(C)C(=O)N2)=O)CCC2CN(C(=O)COCC3CCCO3)CC2C1 c1(C(=O)NC(CNC(=O)C=Cc2ccccc2Cl)CO)c[nH]c2cccnc12 C1(C(N(CC(C)CNC(=O)CSCC(F)F)C)=O)CCCN1CC(F)F NS(=O)(=O)c1ccc(C(N2CC(NC(=O)C3=CCCC3)CC(F)C2)=O)o1 C(=O)(CC(C)(O)CC(=O)O)N1CCCC(C(=O)NCc2ccnc(C)n2)CC1 C(=O)(C(C(C)(C)C)C1CCC1)N1CC(N(C(c2cnc(CC(C)C)s2)=O)C)C1 c1(C(=O)NCC2C(OCC)CN(C(c3cc(Cl)no3)=O)C2)c(Cl)ccc(C)c1O N1(C(c2c(CC)nn(C)c2Cl)=O)CCCC(N=c2[nH]nc(CC(C)C)s2)CC1 N1(C(CC2CCCN(C)C2)=O)CC=C(CNC(C2(O)CCCCCC2)=O)CC1 c1(CCC)cc(C(=O)NC(C)CNC(c2ncccc2C(F)F)=O)sc1C c1(-c2cn(CC3N(C(CCC=CC=C)=O)CC3)nn2)ccnn(CC2CC2)c1=O CCC(CCCC(=O)N1CC2CC2(C(=O)OC)C1)NC(C1CC12CCC2)=O c1(C(=O)OC)cccc(CNC(C)(C)CCCF)c1Br N1(C(CC2(SCC)CC2)=O)CCCC(NC(C23OCC(C(=O)OCC)(C2)C3)=O)C1 N1(C(c2c(C)cns2)=O)CC2CC2(C(=O)NCC2=NOC(C)C2)C1 C1(C(N2CC3N(C(C(CCCCC)O)=O)C(CC3)C2)=O)CC2(CCOCC2)CO1 c1(COC)cc(=NCCC2CCC(NC(c3csnc3C)=O)C2)[nH]cn1 CC(CC(F)(F)F)C(=O)NCCCOCCNC(=O)C(O)C1CCC1 N1(C(c2cccc(OC)c2C)C(=O)NC2CC(F)(F)C2)CCC2CCC(O)C1C2 C(=O)(CCCC(F)(F)F)NC(C1CC=CCC1)C(=O)NCc1cc(C)oc1 N1(C(C(CC(F)F)NC(COCC=C)=O)=O)CC2(COC(=O)C2)C1 Cc1cc(Cl)c(C(=O)NC2CC2NC(c2ccnc(CO)c2)=O)cc1N C(C(=O)N(C)CC1CCCC1)(C(C)O)NC(C(C)CO)=O CC(N=[N+]=[N-])C(=O)NC1CCCCC1C(N1CC(N2CC(O)C2)C1)=O n1(C(C)C)cc(C(=O)NCCC2CCN(C(=O)COC(F)F)C2)c(Br)n1 C(=O)(C1CCCc2nc[nH]c21)N1CC2(CC(CNC(C(C)OCCCC)=O)C2)C1 C(=O)(CS(=O)(=O)CC(=O)NC1CCCCC1NC(c1cnc[nH]1)=O)OC C=CCC(CC(=O)N(C1CSC1)C)NC(=O)CC1CCCCC1 C1(NC(Cn2ncn(C)c2=O)=O)CC2CC(C1)N(C(C1COC(=O)C1)=O)C2 O=C1CCC(C(=O)NCCCC2CCOC2=O)CN1 NS(=O)(=O)N1CCC(C(=O)NCCNC(c2coc(C(F)(F)F)n2)=O)CC1 C(=O)(C(C)n1cncn1)NCCCN(C(C1(CC)CC1)=O)C CC1CN(C(=O)C(=O)NCCOc2cccnc2)CCC1C c1(OC)ccc(C(=O)NC2CC(C(=O)Nc3cc(Br)cnc3O)C2)c([N+](=O)[O-])c1 N1(C(Cc2cc(CC)no2)=O)CC(CNC(c2sccc2C)=O)CC(C)C1 Cc1ccc(CC(N2CCC(OCc3noc(C)n3)CC2)=O)cc1 c1(C2(NC(C3(SC)CCC3)=O)CC2)ccc(F)cc1.C12(CCC1)C(=O)NC2 C1(C2(C)CC2)CCN(C(=O)C(Cc2cnc[nH]2)NC(=O)CN2CCNC(=O)C2)CC1 CCC(CC(C)C)C(=O)N1CCC(CCNC(c2ncncc2F)=O)C1 N1(C(c2cn(CCC)nc2C)=O)CCN(C(c2cc(OC)cs2)=O)C2CC12 C(=O)(C1=NN2CCCN=C2N1)N1C(CNC(C(C)SC)=O)CCC(C)(C)C1 c1(CN2C(C(=O)Nc3cccnc3C(F)(F)F)CC(=C)C2)ccc(C#N)c(Cl)c1 Cc1cc2cc(NC(C3CCN(C(c4ccncc4Br)=O)CC3O)=O)ccc2[nH]1 C(C(CO)(CO)NC(=O)Cc1nocc1C)N(C(C(COC)NC(C)=O)=O)C C(CCCCCCC(=O)N1CC(CNC(c2ncc[nH]c2=O)=O)C(C)(C)C1)SC N1(C(c2c(C)nn[nH]2)=O)CC2(CCCC2NC(C2CC(=O)N(CC3CC3)C2)=O)C1 C1(C(=O)NCC(C2CC2)SC)CCC(NC(=O)CC(C)N(C)C)CC1 C1(CNC(C(CC)SC)=O)CN(C(C2(CCF)CCC2)=O)CCC1(C)C c1(C2C(C(N(CCNC(c3nocc3Br)=O)CC)=O)C2)ccc(OC)cc1 n1(CC)cc([N+](=O)[O-])c(C(=O)NCC2CN(C(=O)COC(C)C)CC2C)n1 C(=O)(CC(O)CC(C)(C)C)NCC1C(C(N2C(C(N(C)C)=O)C=CC2)=O)CCO1 c1(C(N2CC(C(N3CCN(CC#C)CC3)=O)SCC2)=O)c(C)cc(Br)cc1F c1(C(N2CCC(NC(C(CCC)CC)=O)C(O)C2)=O)ccc(O)c2c1CCCC2 S(=O)(=O)(c1cccnc1N(C)Cc1ccc(C)s1)NC(c1cc(C)on1)C C1(NC(C2CC2F)=O)CCCN(C(C2CCCO2)=O)C1.CC1C(=O)N1C1CC1 C1(O)(C(=O)NC2CCN(C(=O)OC)CC2)CCN(C(C2CC23CCCC3)=O)CC1 c1(C(=O)NCCCCN(C)C(C2CC2F)=O)c(O)nnc2c1CCCC2 C12(C(=O)N)C3C4C1C1C2C3C41CO.C1(C=O)C2CCC(O2)C1C(F)(F)F C1(C(=O)NCCN(C(CCc2cc(C)no2)=O)C(C)C)CCC2C1C2(F)F C1(N(C)C(C2(F)CCC2)=O)CC2CC1N(C(C1CCC1)=O)C2 c1(C(=O)NCC2(F)CC(NC(C3C(C)CC=CC3)=O)C2)ccc2ncsc2c1 N1(C(c2cncc(C(C)C)c2)C(=O)NC(C(=O)OC)C)CC(C)CCC12CC2 c1(N2CCC(CNC(C3C(C)=C3)=O)C2)nc2c(cc1C#N)CCC2(C)C c1(CC(=O)NC(C2(CNC(CCc3cnc(C)s3)=O)CC2)C)cccnc1Cl c1(OC)cccc(CCC(N2CCCC(NC(=O)C(C)(C)C(N)=O)C2C)=O)c1F c1(CN2CCC(C(=O)Nc3nccc(N4CCC4)n3)CC2)ccc2ccoc2c1 C1(=O)C(C)(CNC(c2cnc(=N)[nH]c2)=O)N1.N(C)(CCSC)CC C(CCC(=O)NCC1C(C)(C)C1(C)C)(C(C)C)NC(C1C(C(=C)C)OCC1)=O c1(C(N(C(C)C(=O)NC2CC2)CC)=O)oc(CNC(c2ccc[nH]2)=O)cc1C c1(C(N2C(CCC)CCC2)C(=O)NCC(F)F)cc2c(cc1Br)OCO2 C1(NCC(=O)NC(c2ncccn2)CC)CCOC(c2cccc(F)c2)C1 c1(OC)ccc(OC)c(CN=C(NCC(F)F)N(C)Cc2ccc[nH]2)c1 N1(CCNC(C2C=CCN2Cc2cocn2)=O)C(=O)c2ccccc2C1=O NC(CCc1c[nH]nc1C(F)(F)F)C(=O)NC1CN(c2ccccc2)C1 C1(CNC(CCC)=O)CCN(C(=O)COCc2nc[nH]n2)C1(C)C c1(Nc2ncc(C(N(C3CCNC3)CC)=O)cn2)cccc([N+](=O)[O-])c1[N+](=O)[O-] c1(N2C(C3(NC(=O)C=CC4CCCO4)CC3)CCC2)ncnc2c1CCCC2 CC1(C)CC(C(=O)NC2CC3(C2)CC3NC(c2ccc(C3CC3)o2)=O)CNC1=O Cc1[nH]c2c(CN3CCC(C(=O)OCC(C)(C)C)CC3)cccc2c1C N1(C(C(C2CC2)OC)=O)CCC2C(C1)CN2C(c1ccn2nccc2n1)=O C1(NC(C(C)CN(C)C)=O)(CO)CCCN(C(=O)C(C)(C)C2CC2)C1 CN1C(=O)C2CC1CCN2C(N1CCCC1c1ccc(F)nc1)=O C1(CC(=O)NC(C(=O)NCC2CC(OC(C)(C)C)C2)C2CCCC2)COCCO1 Cc1cccc2cc(NC(=O)Nc3nc4cc(Cl)ccc4n3C)cnc12 N1(C(c2[nH]cc(C(C)=O)c2)=O)CCOC2CN(C(C3(C)CC=CCC3)=O)CC12 N1(C(C(n2c(C)ccn2)C)=O)CC(NC(c2cnc(C(N)=O)s2)=O)CC1CO c1(C(=O)NC2CCN(C(CCOC(C)C)=O)CC2CO)cc(Cl)c(N)cc1F Cc1sc(N)c(C(=O)NC2CCCC(NC(C3(C)CC(C)(C)C3)=O)CC2)c1C C(C(=O)NCCC(C)N(C(=O)CCc1cc(C)n(C)n1)C)(C(C)(C)C)SC N1(C(CC2C(C)(C)C(O)C2)=O)CC2(C=C(C(=O)NOCCCF)CO2)C1 Cc1nc(NCCc2ccsc2Cl)cc(N(C)Cc2ccco2)n1 C1(C(=O)NCCC(C)N2CCCC2)CC=CCN1C(=O)C=C(C1CC1)C1CC1 C(=O)(C1=CC2(CCOCC2)C1)N1CCC(CNC(CC(C)F)=O)C(F)(F)CC1 Cc1cc(C)nc(-c2cn(CC(=O)NCc3nnnn3C)nn2)n1 c1(OC(N(CC(=O)NC(C(C)N(C(C)=O)C)(C)C)C)=O)ccccc1C C1(NC(C(C)OCCN(C)C)=O)CC(F)(NCC(C2CC(SC)C2)=O)C1.C1(C)CC1 N1(C(c2ccc(CC)s2)=O)CCC(CNC(c2cc(N)nc(Cl)c2)=O)CC1C Cn1ncc(C(N2CCOC(CCNC(C3CC4CCC(C3)C4)=O)C2)=O)c1C#N CC1(C)C2CN(C(c3sccc3NC(C3(Br)CCC3)=O)=O)CC12 c1(OC)cc(C(=O)NCC2C=CCN2C(C2CCCOC2)=O)ccc1C(F)F C(=O)(CCC(=O)C1CCc2ccccc21)NC(c1cc(F)c(F)c(F)c1)(C)C CCC(CC)C(C)C(=O)NCCCN(C(=O)CC1CCCS1(=O)=O)C1CC1 c1(CNC(=O)NC(C#C)(C)CC)nn(C)c(C)c1Br C(C(C)(C)CNC(C1(F)CCOC1)=O)N(C(=O)C(C)c1ncco1)CC C1(CNC(C=C(CC)C)=O)CCN(C(C2CC2C2(C)COC2)=O)CC1(F)F Cc1cccc(CC(=O)NC(CO)CCCNC(=O)Cc2ccn(C)n2)c1 C1(CC(C)C)CC(C)CN(CCNC(=O)CS(=O)(=O)N2CCCCC2)C1 c1(C(N(C2CCS(=O)(=O)C2)CC)=O)ccccc1C(N)=O C=C1CCC(C(N2CCCC(N(C(=O)CC3CNC(=O)C3)CC)C2)=O)CC1 C1(CNC(CNC(C)=O)=O)CCN(C(c2c(C)nsc2C)=O)CC1CO c1(C(CC#C)=O)coc(CCC)n1.C1C(=O)N(C)CC(C)OCCOCCO1 c1(C(N2CC(F)(CNC(CCOCCC)=O)C2)=O)ccc(C)c2c1NCCC2 C1(NC(C(C)=C(CC)C)=O)CCCC12CN(C(=O)C(c1c(F)cccc1F)C)C2 c1(C(=O)NCCC(=C)CNC(=O)CN(C)CCO)cc(S(N)(=O)=O)cs1 c1(C(=O)NC(CNC(C(C)SCCCC)=O)C(C)(C)C)cnc2cc(C)nn2c1 c1(SCCC(=O)NCC2(C)CCCN2C(C2CCC(=O)N2)=O)ccc(C#N)cc1 c1(C(CNC(c2c(NS(CC(C)C)(=O)=O)cccc2)=O)O)ccc(Cl)cc1Cl c1(C(=O)NC(C(C)NC(c2nccc(CC)c2)=O)C)nccc2ccn(C)c12 c1(NC(C2CC2C(=O)NCC(c2ccccc2)O)=O)ccnc2c1CCO2 N1(C(c2ncc(Cl)s2)C(=O)NCCSCc2ccncc2)CCC(CO)CC1 c1(C(=O)NC2(C)CN(C(C(C3CCCO3)OC)=O)C2)[nH]cnc1C#N c1(C(=O)OC)n[nH]c(SC2CC(Cl)(Cl)C2)c1Cl N1(C(C(C)CC2CC2)C(=O)NC(C)(C)C)CCc2cc(F)cc(Br)c2C1 c1(C(N(C2CCCCN(C(=O)C(C)(F)F)C2)C)=O)ccc(Br)c(Cl)c1 N1(C(=O)Nc2csc(C(F)(F)F)c2)CC(CO)OCC12CC2 c1(C(=O)NC(C(C)NC(C2CN(C)CCO2)=O)(C)C)ccc2c(O)ncnc2c1 CC(C)C(CC(=O)N(CC(C)C(F)(F)F)C)NC(c1cscn1)=O N1(C(C2CC(NC(C(C3CCCC3)OC)=O)C2)=O)CCC(=C(F)F)CC1 Cc1cnc(CNC(=O)C(C)CNC(C2CC2C(F)F)=O)[nH]1 N1(C(C(CN(C)C2CC2)N)=O)CCOCC(n2ccnc2)C1 N1(C(C(C)(C)O)=O)CCC(C2CCCN2C(=O)Oc2cccc(Br)c2)CC1 c1(C(=O)NC(CNC(=O)CC2OCCCO2)C2CC2)cccc(=O)o1 C1(C)(CC)CCCN1Cc1cccc(-c2nnn(C)n2)c1 c1(CNC(c2cnc(-c3ccccc3)s2)=O)cccc(OCC2CCCO2)c1 C(C(CNC(=O)CC1CCSC1)S(C)(=O)=O)NC(C1C(C)(C)C1C(F)F)=O C#CC(CNC(C1CCN(C(=O)CCCC2CC2)C1)=O)CC(C)(C)C n1(CC(=O)NCC(CCOC)NC(C2C3CCOCC23)=O)ncccc1=O c1(C(N2CCN(C(CC(=O)OC)=O)C(CC#N)C2)=O)c2c(nn1C)CCC2 c1(C(=O)NCCC2C(C)CN(C(=O)C(=O)NC3CC3)C2)ccc(O)c(C(N)=O)c1 c1(C(N2CC(C)(NC(C(CCC)C)=O)C2)=O)cc2cc(N)ccc2s1 C(CNC(C1C(C)CCN1C(=O)CCc1conc1C)=O)(CC(C)C)OC C1(N(CCC(F)(F)F)C(c2c(C)nn[nH]2)=O)CCC2(CC1)CNC2 C1(N(C(CC(OCC)OCC=O)=O)C)CCN(c2ccccc2Cl)C1=O.OCC c1(C(C(C)C)=O)ccc(OCC2(S(C)(=O)=O)CC2)cc1 N1(C(C2(C(C)(C)OC)CC2)=O)CCN(C(C2C3C4CCC(C4)C23)=O)C(CF)C1 c1(C2C(C(=O)NCC(C(C)C)NC(C3CN(C(N)=O)C3)=O)C2)c(F)cccc1Cl C1(C(N2CCCC(N(C(c3ccc(Cl)cn3)=O)CC)C2)=O)CCC2(CC1)CC2 c1(OCC(CN(CCOC)CCN(C)C)O)cccc(Cl)c1 C(=O)(C1=CC2(CCOC2)C1)NCC(CCCC)NC(C1(C2CCCO2)CCC1)=O c1(NC)nc(C(=O)N(C)CC2CCCCN2C(C2CCSC2)=O)ccc1[N+](=O)[O-] c1(OC)cc(C(N2CC(NC(=O)C=C(C)C(C)(C)C)C(O)C2)=O)c(O)c(Cl)c1 c1(CC(N2CC(NC(C(C(CC)C)O)=O)C2)=O)c(Br)sc2ccccc12 N1(c2nc(C)nc(N3CC4CC3CS4=O)c2)C2CCC1CC(c1nccn1C)C2 C1(C(N2CCC(C)C(F)(F)C2)=O)COCCC12CN(C(=O)C(C)(C)C#N)C2 c1(C(=O)OC)sc(N2CCCC2c2c(C)n[nH]c2C)nc1C(C)C C1(C)(C(=O)NCCC(C)C)CCN(Cc2ccccc2C(=O)O)C1 N1(C(C2(CC)CCN(C(C3CCCN3C(C)C)=O)C2)=O)CCN(C)C2(CC2)C1 N1(C(CN(CCOC)CC2COC(C)C2)=O)CC(C)(C(F)(F)F)C1 N1(C(C(C(C)C)OC)=O)CCC2(C)CN(C(C3CCC(C(C)(C)C)O3)=O)CC12 c1(OC)ccc2oc(C(N3CCC4CCC34CNC(C3(C)CC3)=O)=O)cc2c1 CC1CN(C(=O)CNC(C2CCC(C)(O)CC2)=O)CC(=O)N1 Cc1cn2c(n1)C(C(=O)N(CCCCNC(=O)CC1(O)CCCOC1)C)CCC2 c1(N2CC3CC(NC(c4cc(CCC)[nH]n4)=O)C3C2)cc(C)c(C#N)cn1 N1(C(C(C)=CC)=O)CCN(C(C2CCC(=O)N(C(C)C)C2)=O)C(CC(F)F)C1 c1(C(=O)NCC2N(C(C(COCC)(C)C)=O)CCC2)cc2cccnc2[nH]1 c1(C(=O)NC2CN(C(Cn3nnc(C)n3)=O)C(C)(C)C2)cnc2ncccc2c1 c1(COC(C(C)(O)Cn2ccccc2=O)=O)nc2nc(O)c3ccccc3n2n1 c1(C(N2CCN(C(C(c3cccc(F)c3)(C)O)=O)CC2)=O)nc2ccccc2s1 N1(C(c2cn(C)nc2N)=O)CCN(C(=O)CCS(N)(=O)=O)C(CO)C1 Cc1cc(C(=O)NC2CN(C(C3CC4CCCCC34)=O)CC2O)n2nccc2n1 C1(C(=O)NC(CCNC(CCc2cc(C)n(C)n2)=O)C)CCc2c(nnn2C)C1 CCCCS(=O)(=O)CC(=O)NC12CCCC(NC(c3ccns3)=O)(C1)C2 C1(F)(CN(C(=O)NC(C)CCC2CCCO2)C)CCCC1 Cc1nc(C)c(C(=O)N(C)CC2COCCN2C(=O)CNc2ccccc2F)[nH]1 c1(NCC(C)(C)C(=O)N2CCCC2C2CCC(N)CC2)ncc(C(F)F)cc1Cl c1(N(CCC)Cc2ccnc(Cl)c2)ccc(CO)cc1[N+](=O)[O-] CCC(O)C(C)(C)C(=O)NCC1C=CC(NC(=O)CC2CC(C)C2)C1 C12(NC(C(CSC)C)=O)CC3CC(C1)CC(NC(C1CCCCN1C)=O)(C3)C2 C1(C(=O)NCC(NOC)=O)CCN(C(C2CCCC(C#N)C2)=O)CC1(C)C C1(NC(CC)=O)CN(C(c2ccc(-c3sccc3C)s2)=O)C2(CCCOC2)C1 C1(C(N2CC(NC(C3(C)CCNC3=O)=O)C(CC3CC3)C2)=O)CCS(=O)(=O)CC1 Cc1cc(NC(C2CCCN(C(c3nc[nH]n3)=O)C2)=O)n(C(C)C)n1 C1(CCNC(C=CC(CC)=CC)=O)COCCN1C(=O)Cn1cccn1 N1(C(c2cc(C(N)=O)no2)=O)CCCC2(CC(NC(=O)C(F)=C3CCC3)CO2)C1 CCC(F)(C(=O)OC)C(=O)N1CC2C(N(C)C(c3cc(F)cnc3O)=O)C2C1 Cc1cnc(C(=O)NC(CCNC(C2(CF)CC2)=O)C(C)C)c(O)c1 C(c1ccc(F)cc1)=CC(=O)NCC(C)NC(=O)C=Cc1ccsc1 c1(CC)oc(C)cc1C(=O)NC(CO)C(=O)N(C1CC2CC2C1)C Cc1nc(C(N2CCSCC2CCNC(=O)C(N2CCCCC2)C)=O)c(C)s1 c1(C(=O)NCC(N2CCN(C(=O)Cc3cnns3)CC2)=O)ccc(O)nn1 c1(C(N2CCC(c3n(C)ncc3)C2)C(=O)NCC2CCOC2)ccc(Cl)cc1Cl C1(CNC(Cc2cn(CC)nc2)=O)CN(C(=O)CC2COC(=O)C2)CC(C)(C)C1 C1(NC(=O)CSCc2cscn2)CCCCN(C(=O)CCC2CCCO2)C1 N1(C(c2ccn3ncnc3c2)=O)CC2(C1)CN(C(c1ccsc1Cl)=O)CC2CO N1(C(C2CN(C(C)=O)C2)=O)CC2(C(N3CCSC(C)(C)C3)=O)CC1CO2 C1(N(C(=O)C=CC(C)(C)NC(=O)CNc2cccnc2)C)CCCOC1 Cc1ncnc(C(=O)NCCC2CCCN(C(=O)CC(C)F)CC2)c1C c1(C(=O)NC(c2ncc(C)cn2)C)nccc2c(Cl)cccc12 c1(NCc2occ(C(=O)OCC)c2)cccnc1Sc1ccncc1 C1(O)(CNC(C(CC)N(CC)CC)=O)CCCN(C(c2cnn3c2CCC3)=O)C1 c1(C(N(CC(C)NC(c2c(C)cns2)=O)C)=O)nccnc1N C(c1ccoc1)=CC(=O)NCCN(CCC)C(C1CC1OCC)=O Cc1oc(C(C)C)nc1C(=O)NCCC1CCN(C(=O)CC2C=NN(C)C2=O)C1 N1(C(c2cccc(CC)c2)=O)CCC2(CCN(C(C)C)C2)C1 C1(N(C(C23C(CN(C(C(CC)N(C)C)=O)C2)C3)=O)C)CN2CCC1CC2 c1(N2CC(CN(CC(=O)NC)C)C2)ncnc2ccc(OC)nc12 Cc1cc(C(=O)NC2CCC(C)(CNC(=O)CC3CCCC3O)CC2)ccc1Cl Cc1cnc(C(=O)N(C)CCNC(c2csc(-c3ccccc3)n2)=O)cc1Cl C(=O)(CC(C)C(F)F)N1CCC(NC(C2(C=C)CCC2)=O)C1C(C)C c1(C(=O)O)cc(S(=O)(=O)N(C2CCCCCCC2)c2ccccc2)ccn1 CCCC(CC)C(=O)N1CC(O)CC1CNC(c1sc(Cl)cc1Cl)=O C1(NC)CCN(CC2CC(O)C2(C)C)CC1 C(=O)(CCCCC(N)=O)NC(CC)CNC(=O)C=CC(c1ccccc1)=O C12(C(=O)NCC(c3ccccc3)NC(CN(C)CCO)=O)CC(F)C1C2 O=C(N=c1ccc(-c2ccccc2F)n[nH]1)c1cccc(Cl)c1Cl c1(NC(c2nc(Cc3ncccc3F)cs2)=O)cc(F)ccc1Br c1(C(N(C2C(NC(C(C)S(N)(=O)=O)=O)CCCC2)C)=O)cnc2c(c1)CCCO2 C=CCC(C)(CC)C(=O)NCC1C2CN(C(C3(OC)CCS(=O)(=O)C3)=O)CC12 C(CCC(=O)NO)NC(CC1CCN(C(C2N(C(C)C)CCC2)=O)C1)=O N1(C(C(=C(C)C2CC2)F)=O)CCCCC1CNC(=O)CCNS(C)(=O)=O N1(C(CNC(CNC(C)=O)=O)=O)CCC(OC(C)C)CC1.C1(=O)C(C)(CO)N1 CC1CCCN(C(=O)CCC2CC(F)(F)C2)C1CNc1ccncn1 c1(C(=O)N)conc1C1CC1.CC1C(=O)NC(C)CCN1C.N(C)C Cc1ccc([N+](=O)[O-])c(C(N2CC(NC(C3(O)CC3(C)C)=O)C(O)C2)=O)c1 c1(C(=O)NCCC2(NC(C(F)OC)=O)CC2)cc2cccc(Br)c2o1 C1(NC(c2c(C)cc(SC)o2)=O)CC2CC(NC(=O)C(F)n3ccnc3)CC12 C(=O)(C(C)C(C)S(C)(=O)=O)NC(C1(O)CCN(C(c2c[nH]c(Br)c2)=O)CC1)C c1(C(N(C(C)CNC(=O)CCCC(F)F)CC)=O)sc2nccc(C)c2c1C C=CC(O)C(C)(C)C(=O)N1CC2CC1C2C(=O)NCc1ncccc1C C1(C(=O)NCC(CN(C(C2C(C(=O)OC)C2)=O)C)O)CC2(CC2)CN1C N1(C(C(CCC=C)NC(=O)COC2(C)CCCC2)=O)CCC2(CCCC2)CC1 C1(N(C(=O)CC2(C)CC2)C)CN(C(c2ccccc2OCC(F)(F)F)=O)CC1F C1(OC)CN(C(=O)CNC(c2ccccn2)=O)CC1NC(=O)CC1(O)CCOC1 c1(OCC)nc(C(=O)NC(C)CNC(c2nc(O)sc2C)=O)cc2ccccc12 c1(NC(CC)CN(C)C)[nH]c(=NCC(C)(CC)OC)nc2c1ncn2C(C)C Cn1nc(C(=O)NCC2CN(C(=O)C=C3CCCCC3)C3CC23)cc1C(F)F C1(C)(C(N(C)CC2OCCN(C(C3C(C)(CC)C3)=O)C2)=O)CC(OC)CN1C N1(C(CCOCC#C)=O)CC(C(=O)N(C)CC2CCCC2(C)C)C(C)C1 c1(OC)cc(C(=O)NCCC2CCC(NC(=O)Cc3cccs3)C2)cc(Cl)c1O N1(C(c2c(C)cc(=N)[nH]c2)=O)CC(NC(C2CC3C=CC2C3)=O)CC(F)(F)C1 n1(CC)cnc2[nH]c(=NCC3CCCOC3)[nH]c(=NC(C)CCCC(F)(F)F)c12 CC1CCCC(C(N2CCC(OCCNC(c3cc(CC4CC4)on3)=O)C2)=O)C1 C12(C(=O)NCC3C(C)CN(C(=O)COCCCF)CC3)C3C4C1C1C2C3C41C Cc1[nH]cc(C(=O)NCC2CCN2C(=O)C=C2CC2)c(=O)c1Br c1(C(N2C(CCCNC(C3C(C)C3C)=O)CCC2)=O)cccc2c1COCCN2 CC1CN(C(=O)CN(C)C2CC2)CC(C)N(C(c2cc3c(s2)CCSC3)=O)C1 C1(c2nnnn2CCN(C)C(=O)OC(C)(C)C)(NC(CC)CO)COCCOC1 N1(C(C(C)CF)=O)CC(NC(c2ccc(-c3cccs3)o2)=O)C(O)C1 C1(C(N(CC=C)C)=O)CCCN(C(=O)CN(CC)CC)C1 N1(C(CCC(C)C)=O)CCC2(CCCN(C(=O)CCCc3nccs3)C2)C1 n1(CC(=O)NC2CC(NC(C(=O)NC(C)C)=O)C(O)C2)ccc(=O)n(C)c1=O c1(OC)cc(C(=O)NCC(O)CCNC(C2OCC2(C)C)=O)cc(Cl)c1 c1(C(N2CCn3c(C)cnc3C2)=O)ccnc2cc(Cl)ccc12 Cc1cc(C(=O)NCCN(C(=O)CC(C)c2ccccc2)C)nn1C N1(C(c2ccnc(Br)c2)=O)CCC(C2CN(C(c3cc(Br)cnc3F)=O)C2)CC1 Nc1cc(F)c(F)cc1C(N1C2CCC1CC(NC(=O)CN1CCCCC1)C2)=O N1(C(CCSCC(N)=O)=O)CCC2CCN(C(c3nnc(O)nc3O)=O)C2C1 c1(CNC(C=CC(C)(C)SC)=O)cnn(C)c1C(=O)NOCCCC1CC1 C#Cc1ccc(NC(=O)CCN(CC=C)C(c2cccc(OC)c2OC)=O)cn1 c1(COC)ccoc1C(N1CCCC1C1CCN(C(=O)CCC2(C)CC2)C1)=O C1(C(N2C(C(N(CC(C)CO)C)=O)CC2C)=O)CC2CC(=O)C1O2 Cc1ccc(C(=O)N(C)CC2CN(C(=O)C(F)C3CCC3)CC23CC3)c(N)c1 N1(C(C(C)C#N)=O)CCC(NC(c2cnn3ccc(Br)cc23)=O)CC(C)(C)C1 C(CCC(C(=O)NCC(O)CCC1CC1)NC(c1cc(F)ccc1O)=O)OC C(C1CCCCc2ccccc21)NC(c1c(OC)nc(N(C)C)cc1)=O C#CC1(O)CCCN(C(C2C3CCC(C3)C2NC(=O)COC2CCCOC2)=O)C1 N1(C(C(CC=C)CC)=O)CCN(C(c2csc(C(C)C)n2)=O)C2CCC12 c1(-n2cc(CC(C)N(C)C(C3(C)CC3C(=O)O)=O)nn2)cccc(C(F)(F)F)c1 C(C#CC(=O)N(CC(CO)(CO)NC(=O)Cc1cnn(C)c1)C)(OCC)OCC c1(NC(=O)NCc2ccc(OC)c(Br)c2)nc2ccc(C)cc2[nH]1 C(=O)(C(O)C(C)(C)C)NCC1(CN(C(=O)C(c2ccccc2)O)C)CC1 C1(CNC(c2ccn(CCN(C)C)n2)=O)C2CN(CCC3CCCCO3)CC12 C1(NC(c2cc(C)n(C)c2)=O)CCN(C(=O)CCc2cc(Cl)no2)CC1C(C)C N1(C(c2ncn(CC)n2)=O)CC(NC(c2cnncc2O)=O)C(O)C1 Cn1cnc(N2CCC(CCNC(c3cccc(F)n3)=O)C2)c(Br)c1=O c1(C(N2CCCC(NC(C3CCSC3)=O)C2)=O)c(Cl)nc2cc(Cl)ccn12 O=C(C1c2ccccc2CN1C(c1nc(Cl)ccc1Cl)=O)N1CC2CC2(CO)C1 C1(CNC(C2CCCS2(=O)=O)=O)CC12CCN(C(C1C=CCS1)=O)CC2 c1(OC)c(C(=O)Nc2cc(C(F)F)ncn2)nc(O)nc1O.N12CCCC(C1)C2 C1(NC(c2cc(C)no2)=O)CCCC1(C)CNC(=O)C(c1ccccc1Cl)C c1(CNC(C(C2CCC2)NC(COCCC)=O)=O)ccc(CC)o1 C(=O)(C1=CCC(NC(c2csc(=N)[nH]2)=O)C1)NCC(CC(=O)NC)C N1(C(C2(CCCC)CCCC2)=O)CC2CN(C(C3CCC=CCC3)=O)CC(C1)O2 C1(OC)CN(C(C2(C)CCC(C)CC2)=O)CCC1NC(=O)CC1CCOC1 N1(C(COc2cccc(C)c2)=O)CCCCC(CNC(=O)CC2CCCC2C)C1 N1(C(C2CC(C)(O)C2)=O)CC2CC(C1)N(C(=O)CCC1CC1CC1CC1)C2 CC1CN2CCN1CC2C(=O)N(CCCNC(C12CCC(CC1)OC2)=O)C1CC1 N1(C(=O)CC2CCCO2)CC2CCN(C(c3snc(Cl)c3Cl)=O)CC2C1 c1(OC)c(C(=O)NCC(CNC(=O)C=Cc2ccncc2)OC)cc(F)cc1F C1(C(=O)NCC(C)(Cn2cccn2)NC(CNS(C)(=O)=O)=O)CCS(=O)(=O)N1 c1(OC(C(=O)NCCCC2(NC(C3C(CC)C3)=O)CC2)C)ccc(C)cc1C C#Cc1cccc(CC(N2CC3CC2C3NC(=O)C(N2CCSCC2)C)=O)c1 C(=O)(CC(O)(C(F)(F)F)c1ncco1)NCC=CCNC(c1c(C)cncc1)=O C(=O)(C1COc2ccccc21)N1CC2C(CNC(c3n(C)nnc3)=O)C2C1 N1(C(C2(C=C)CCCCC2)=O)CC=C(CC(=O)NCc2cc(C)ncn2)CC1 c1(-n2cc(O)nn2)ccc(F)cc1Cl.N1(C(=O)CCO)CCC(CO)(C)C1 CC(C)CC(C)(C)C(=O)NCCn1cnc(C(N2CCOCCC2C2CC2)=O)c1 c1(C(N)=O)ccc(C(=O)NC2CCCC2NC(C2CC3CC3C2)=O)cc1 N1(C(C2C(CC)OCC2)=O)CC2=C(C1)CN(C(c1ccc(F)cc1F)=O)C2 C(=O)(C1=COc2ccccc2O1)NCCCCC(C)NC(=O)C=CC(=O)NC1CC1 C(=O)(C(C)CC(=O)NCC1(C(=O)NCCC(C)N2CCCC2)CC=CC1)OC O=C1NCCOc2ccc(CNCC3CCCN(Cc4ccccc4)C3)cc21 Cc1ccc(C(=O)NC2CC(O)CN(C(c3ccc(O)cc3)=O)C2)cc1C c1(NC(C(C)(C)C)C2CCCCC2)cc(Cl)cc(Br)c1 C1(NC(CC2(N(C)C)CCC2)=O)CCN(C(=O)CC2CCC=CCC2)CC1 c1(COCC)nc(Cl)cc(=NC2CC(CNC(=O)CS(=O)CC)C2)[nH]1 c1(CNC(CC2N(C(C3(C(N)=O)CCC3)=O)CC2)=O)ncccc1O N1(C(CCC)=O)CCC(C2CCCCN2C(=O)Cn2cc(C(C)O)nn2)CC1 Cc1csc2cc(C(=O)NC3CC3CNC(=O)C(N)=O)[nH]c12 C(=O)(C(CCC(N)=O)n1cc(CO)nn1)N1CCC(SC(c2cnn[nH]2)C)CC1 c1(NC(C(=O)Nc2cccc(-c3ccncc3)c2)=O)ccc2c(c1)CCNCC2 N1(C(CN(C(CC2ON=C(C)C2)=O)C)=O)CCN(C(=O)C=CCF)CC1 N1(C(C=CC(CC)=CC)=O)CC2CN(C(=O)C(C3CCOCC3)OC)CC2(C)C1 C(=O)(CC(C)C(C)(C)NC(=O)CCC(=O)C1CC1)N1CCC(C=C)C1 C=CC1(NC(=O)C(Cc2ccoc2)NC(=O)Cc2cc(C)nn2C)CCOCC1 Cc1ccc(C(=O)N(C2CCCC(N(C(=O)COCC(F)F)C)C2)C)nn1 c1(C(=O)NCCCN(C(=O)C(C)C2CCC2)CC)cc2ccncc2s1 N1(C(N2CCC(OCC)C(C)C2)=O)CCCc2ccc(C(=O)OC)cc2C1 Cc1ncc(CCC(=O)NC2(CNC(c3csc(-c4ncccn4)n3)=O)CC2)o1 C1(CC(=O)OC)CCCN1C(C1C=CC(NC(C2CCCS2)=O)C1)=O Cc1noc(C2CC2)c1C(=O)NCC1(C)CCCN1C(=O)CC1(C)CCCCC1 c1(C(N2CC(NC(c3c(C)sc(CC(=O)O)n3)=O)C2)=O)sccc1S(N)(=O)=O N1(C(COC)=O)CCC(CON(C2C3CCC23)C)CC1 N(C(=NCc1ccc(F)cc1)N1CCC(F)C1)CC1N(CC)CCC1 C1(C(=O)NCC2(C)CCCN2C(c2cnc3sccn23)=O)NC(=O)C2CCC12 N1(C(C=C(CCC)C)=O)CC=CC1CNC(c1n[nH]cc1C1CC1)=O c1(C(=O)NCCC2(CNC(C3CC4CCC4C3)=O)CC2)ccnc2ccsc12 CC1CCCn2cc(C(N3CC(O)(CNC(=O)CCc4cccnc4)C3)=O)nc21 C1(C(=O)NCC(C2CC2)NC(c2cc(OC)ns2)=O)CCC2(CC1)CNC(=O)C2 CC(C)(CS(C)(=O)=O)C(=O)NC1CN(C(=O)CCCCC2CC2)C2(CCOC2)C1 C1(NC(C2N(CC)CCC2)=O)CCCCN(C(c2cc3ccccc3[nH]2)=O)CC1 CC1CCC(C(N2CCN(C(N)=O)CC2)=O)CN1C(c1ccncc1O)=O Cc1ccc(-n2nnnc2N2CCC(C(=O)OCc3ccccc3)C2)cc1 c1(C(=O)OCCC2C(C)(C)CCO2)ccc2c(=O)[nH]ccc2c1 Cc1noc2cc(C(N3CC4CC(NC(=O)CC(C)(F)F)CC4C3)=O)ccc12 C1(CNC(COCCOCCOC)=O)CN(C(c2c(C)nsc2N)=O)CC1(F)F c1(C(=O)NC2C(C)N(Cc3ccccc3)CCC2)cnc2cnccc2c1 c1(C(=O)NC2C3OCC(NC(C4CCC(C)O4)=O)(C3)C2)cccc(O)c1[N+](=O)[O-] N1(C(C(=O)Nc2c(C)ccc(F)c2)C)CC(C)C(C2CCC2)C1 N1(C(CCOCC#C)=O)CCC(C(C)(C)C)(NC(=O)CC2(C=C)CCC2)C1 c1(C(N(C)CC2(NC(C=C(CC)C)=O)CC2)=O)nccc(Cl)c1C N1(CCOc2c(C(=O)NC3CC3)cc(Br)cc2)CC2C3C=CC(CC3)C2C1 c1(-c2cn(CCC(N3CC(OC)C(OC(C)(C)C)C3)=O)nn2)nnc2n1CCC2 C(=O)(C1=COCCO1)N1C(CNC(c2ccc(CN3CCOCC3)o2)=O)C=CC1 C(c1ccc(=N)[nH]c1C)=CC(=O)NCC1C(NC(CCSCC)=O)CC1 C(=O)(C1=CNC2=NCCCC2=C1)NCCN(C1CCCCCC1)C(C(CC)C)=O C1(C(N(C(C)CC(N)=O)C)=O)CC2CCC(C1)N2C(C1CC1(C)C(F)F)=O C(=O)(C1=CCCCC1)N1C(CNC(c2csc(O)n2)=O)CCCC1 N1(C(CN(C(COC)=O)C)=O)CCC(C(=O)NCCC2CC(C)C2)CC1(C)C c1(CC(=O)N(CC(CNC(CC2CC(C)C2)=O)O)C)cccc(C(F)(F)F)n1 C(CN=c1[nH]c(N(CC(c2nccs2)C)C)nc2c1CCCC2)OC(C)C C1(C(=O)NCCCCC(C)NC(CC(CC)CC)=O)CCCCN(C)C1=O C1(C)(CNC(CC2(C)CCOC2)=O)CCCN(C(=O)Cc2nccs2)C1 N1(C(c2c(C(C)(C)C)c[nH]c2)=O)CCCCC(NC(C23COCC2C3(F)F)=O)C1 CC1(C)C2CCC1(C(=O)NC13CC(NC(c4cc(Cl)ns4)=O)(C1)C3)CC2 CC1=C(F)CN(C(=O)C(C(C)(C)O)NC(=O)COC(C)(C)C)CC1 C1(CCC)CN(C(=O)CC(C)(C)N(C)C)CCN1C(C1CCCN(C)C1)=O C1(N(C(=O)C(=O)NCC(F)(F)F)CC#C)CCN(C(=O)Cn2nnnc2C)C1 Cn1cnc(CC(=O)NC(C)(C(=O)N2CC(O)(CCO)C2)C2CCC2)c1 C1(C(N2C(CN(C(=O)Cn3ccc(C4CC4)n3)C)CCC2)=O)CC12CC(C)(C)C2 Cn1cccc1C(=O)C(=O)NC1CC(CNC(c2ccnn2C2CCCC2)=O)C1 CON(CCO)C(=O)c1cc(CNC(c2c(O)cccc2F)=O)[nH]n1 C(=O)(CC(C)C(=O)NC(C(=O)Nc1cnn(CCF)c1)C1(C)CC1)OC N1(C(CN2CC(C)(C)C2)=O)CC2(CCC2)CC1CNC(C1CC2CCC(C1)N2C)=O c1(CNC(CCC=C(C)C)=O)cccc(C(=O)NC2CCCC(C(N)=O)C2)n1 CC(C)(C)CN=C(NCC1(O)CCOC1)NCC(C)(O)c1ccsc1 c1(C(N2C(C)C(NC(=O)CCC3CCC3)CCC2)=O)ccnc2ccnn12 C(=O)(C(C)(C(C)C)OC)N(C(CC(=O)NC1CC(CC)OCC1)CC)C CCC(C)(C)CCCC(=O)N1C(CC(=O)NC(C(C)C)C(C)C)C2CCCC12 C1(C(N2CC(C)(CC=C)C2)=O)CC2(CC(NC(=O)Cc3scnc3C)C2)C1 O=C(CCC(=O)c1ccc(F)cc1)NCCOCc1cn(CC2CCCO2)nn1 Nc1cc(F)c(C(=O)NC(CNC(=O)CCC2CC2)CO)cc1F c1(OC(CCC)C(=O)OC2CC(F)(F)C2)cncc2ncccc12.n12cc(cn1)C2 C1(N(C(=O)COCc2cccnc2)C)CCCN(C(C2CC(F)(F)C2)=O)C1 c1(C(N(C2CCN(C(=O)CN3C(=O)CNC3=O)CC2)CC)=O)ncc(F)cc1F C1(C(=O)NCC(C)NC(c2cnn(CC)c2C)=O)CCC(S(C)(=O)=O)CC1 C(CCOCC)(C(=O)NCc1occc1C)NC(CC1CC(=C)C1)=O C1(NC(CC(C=C)CC)=O)CN(C(c2cc(CC)[nH]n2)=O)CCC12CCC2 C1(CNC(=O)CCc2cnc(O)[nH]2)CN(C(c2cc(C(F)(F)F)no2)=O)CC1O CCC(O)C(C)C(=O)N(C1CCC(NC(=O)CCCc2csc(=N)[nH]2)CC1)C C=CCC(CNC(c1sccc1F)=O)NC(=O)C(n1ccc(C(F)(F)F)n1)C N1(C(CCc2ccc(C)cc2)=O)CCC(C)C(NC(=O)CNc2ccccn2)C1 N1(C(C2CN(C(c3n(C=C)ncc3)=O)CC2C=CC)=O)CCC(C)CC(C)C1 CC1(C)CC(NC(=O)C=C2CCC2)CN(c2ncc(C#N)cc2F)C1 c1(C(=O)NCC23CC2CN(C(=O)CCn2ccnn2)C3)cncc2nc(O)[nH]c12 n1(CC)ncc(C(=O)NC2CCOCC2NC(=O)COC2CC2)c1C C(=O)(C1=CC2CCCCCC12)N1CC2CCC(NC(=O)CCCCF)CC2C1 C(=O)(C(C)(O)C(C)C)NC(C1CCCN(C(=O)Cc2cnc(C3CC3)[nH]2)C1)C c1(C(=O)NCCCN(C(Cc2cn(C(C)C)nc2)=O)C)ccncc1C(F)F c1(C(=O)NC(C)CCN(C(=O)C(F)(F)c2ccncc2)C)cccc(Cl)c1 C(=O)(C1=C(Cl)CCC1)NC1(CCCC(=O)NCC2N(C(C)=O)CCC2)CCC1 N1(C(C(C)(C)C2CC2)=O)CCN(C(C2C=CCC2)=O)C(C2CC2)C1 c1(C(N2C(C)C(NC(C3CCCN(C)C3=O)=O)CC2)=O)ccc2nccn2n1 c1(OC)cncc(CC(N2CC(NC(C3CCC(CN(C)C)O3)=O)C2)=O)c1 Cc1ccc(OCC(=O)NCC2(C)CN(C(=O)CCCC(N)=O)CC2C)cc1C c1(C(c2n(CCOC)nnn2)NC2(C)CCC2)cccc(C(=O)NC2CC2)c1F N1(C(C2CN(CC(C)C)C2)=O)CCCC(CN(C(=O)CCNS(C)(=O)=O)C)C1 C(=O)(CCC(=O)c1ccc(Cl)s1)NC(CNC(c1nc(COC)sc1)=O)(C)CO CC(c1ccccc1F)=CC(=O)NC(C)(C)C(C)NC(c1c[nH]cc1Br)=O c1(C(=O)NC2CN(C(=O)CN3CSCC3=O)CC2F)oc2ccccc2c1Cl C12(NC(Cc3c(CSCC)cccc3)=O)CCCC1N(C(c1cocn1)=O)CC2 c1(C(=O)NC2CCC(NC(C(C)P(C)(C)=O)=O)CC2)c[nH]c2cccc(C#N)c12 C1(C(=O)NCC(C)(F)F)CC12CCN(C(=O)C=Cc1cc[nH]n1)C2 c1(C(=O)NCC(C)N(C(C(CCC)OC)=O)C)cccc(C2=CCOCC2)c1 Cc1cn2nc(C(=O)NC3(CO)CCN(C(=O)CC4CCOC4)C3)cc2c(=O)[nH]1 C1(C(=O)NC(CCC)C2CC2)CC(C)(C)CCN1C(=O)CC1CC=CCC1 c1(C(=O)NC2(CNC(c3ccc(O)nc3Cl)=O)CCC2)ccnc2ncnn12 Cn1ncnc1CCCNC(c1cn(CCNC(C2CCCCC2)=O)cn1)=O C1(C)(CNC(CC2(CSC)CC2)=O)CCCN1C(=O)Cc1ccc(C)nc1 CCC(C)(CC)C(=O)NC(C)C(C)C(=O)Nc1cnc(Cl)nc1C c1(C(CC(=O)NCC(n2cc(C(=O)OCC)nn2)C)C)ccc(F)c(F)c1 N(C(=NCCc1ccn(CC)n1)N1CCC(c2ccccc2F)C1)C(CC)C c1(C(=O)NCCC2COCCN2C(C2CCCCO2)=O)c[nH]nc1[N+](=O)[O-] c1(OC)cc(F)c(CCNCc2ccoc2C)c(F)c1 C=CCCC(C)(C)C(=O)N1CC(NC(=O)CCc2c(Cl)cccc2Cl)C2(CC2)C1 CCCCCCn1cc(CC2CCN(C(=O)CC(C)c3ccco3)C2)nn1 Cc1nc(C(=O)NCC(C)(CO)NC(c2cscc2Cl)=O)nn1-c1ccccc1 c1(OC)ccc(CC(O)C(=O)NC(CO)C(C)NC(=O)Cc2c[nH]nc2O)cc1 C(N=c1[nH]cncc1Br)C1(CNC(C(C)(C)c2cncnc2)=O)CCCC1 N1(C(CSC)=O)CCCCC1CN(C)C(c1ccnc(C(N)=O)c1)=O N1(C(c2c(C)cccn2)=O)C2CCC1CC(C(N1CC(C)C1(C)C)=O)C2 c1(C(C)C)ccc(CC(=O)NCC2(O)CC(NC(C3COC(=O)C3)=O)C2)cc1 N1(C(c2c(C)nc(C(C)C)o2)=O)CCN(C)CC1CNC(C1CC12CC2)=O C#Cc1ccc(F)cc1NC1CCCC1CNC(=O)OC(C)(C)C N1(C(C2CN(CC)C2)=O)CCCC(CN2CCN(C(=O)CSS(C)(=O)=O)CC2)C1 c1(CCC)cc(C(N2CC3CC2C3NC(=O)C(C)C(=O)OC)=O)c(C)o1 N1(C(C(C2CCCC2)NC(CC)=O)=O)CCCCC1CNC(=O)CN(C)CCO c1(CC(=O)NC(C(C)(C)C)CNC(c2cncc(F)n2)=O)ccc(C#N)cc1F C1(NC(=O)CC(O)c2ccccc2)(CNC(=O)C(O)C2CC2)CCCCC1 Cc1cc(C(N2CCCC2(C)C(N2CCn3cnnc3C2)=O)=O)cc(C)c1O CCC(CC)(CO)C(=O)NCC(C)NC(C1(C)CC(C(=O)OC(C)(C)C)C1)=O C1(C(=O)NC2(C(C)C)CCCC2)CC12CCN(CC1CCNC1)CC2 CC(C)CC(CNC(=O)C(CC1CC1)CC1CC1)NC(=O)Cc1ccccc1Cl c1(NC(=O)NC(C)CO)onc2ccccc12 N1(C(c2scc(C(N)=O)c2)=O)CCN(C(C2CC2CF)=O)C(c2ccccn2)C1 c1(CNC(C2C(C3C(C)C3)C2)=O)cccc2c1CCN(C1CCN(C)C1=O)C2 N1(C(C(C)CC2CC2)=O)CC(C(N2CCC(c3cnn[nH]3)C2)=O)CC(C)(C)C1 C1(NC(C(CC)OCC)=O)CC2CN(C(c3ncc(Br)cc3O)=O)CC12 Cn1cc(Cl)cc1C(=O)NCC1CCCCC1NC(c1cnccc1Cl)=O c1(C(=O)NCC2C(NC(c3cnc(C(F)(F)F)s3)=O)COC2)cnc(O)cc1F C1(C(=O)NC(CC=C)CNC(=O)Cn2ncnn2)CCC2(CCC2)C1 C1(C(N2C(CC)CC(C)C2)=O)CCC2(CC2)N1C(c1cc[nH]c1C)=O n1(CCC)nnnc1C(C1CC1C1CC1)NCCNC(=O)C(C)C C12(CC(=O)NC(CNC(C(C(=O)OC)C)=O)(C)C)CCC(CC1)OC2 C12(C(=O)NC3C(NC(C4(OC)CCC4)=O)CCCC3)CCCN(CC1)S2(=O)=O C1(C(=O)NCC2CN(C(C(CCNC(=O)C3CC3)O)=O)C2)CCc2ncnn2C1 C(C(F)(F)C(=O)N1CC(NC(c2sccc2-n2cnnn2)=O)C(C)C1)OC CCC(CC)C(F)C(=O)N1CCCC(F)(C(=O)NCC(n2cccn2)C)C1 C1(C2CCC2)(C(=O)NCC2(C(C)NC(=O)C=CI)CC2)CCC1 C1(CCC)CN(CCC2CCOC2)CCO1 C(=O)(CC(C)(O)C(F)(F)F)N1C(C)CC(NC(C2(C=C)CCC2)=O)C1 N1(C(C(C)OCC=C)=O)CC(=O)NC(=O)C1 N1(C(C=NOC)=O)CCC(C)N(C(=O)CCOc2ccc(Cl)cc2F)CC1 Cc1cc(C(=O)NC2CCC(C)N(C(c3cc(C#N)c[nH]3)=O)C2)cnc1C C1(NC(c2cc(C)nc(C)n2)=O)CCC2CC1CN2C(c1nc(Cl)ccc1N)=O N1(C(c2n(C)nc(C(F)F)c2)=O)CC(NC(c2ccc(F)s2)=O)C2(CC2)C1 C(=O)(N=c1ccc(C2CCOC2)n[nH]1)NCC1(OC)CCC(C)C1 CCCCC(C)(C)NC(C1CC(C)CN1C(=O)C(F)CC1CCOC1)=O C1(C(=O)Nc2ccc(CC(=O)OC)cc2)CC2(CCOCC2)CO1 c1(OCCC#C)ccc(CNC(=O)NCC2(O)CCC(CC)C2)cc1 CCN=c1ccc(C(N2CCCCC(NC(=O)C(C)OCC3CC3)C2)=O)c[nH]1 N(C(=NCCSC)NCc1nncn1-c1ccccc1)C(C=C)C Cc1nn(C(C)C)cc1CO.c12ccc(cc1)CC(=O)NC2=O c1(C(=O)NCCN(C(=O)C(CC)n2cccn2)CCC)cnncc1C C(N=c1[nH]c(=NC2CC2C(C)C)c2c(ncn2C)[nH]1)c1cc(C)ncc1 c1(C(N2C(CNC(=O)COC3CCCC3)CCCC2)=O)ccc(Br)c(O)n1 N1(C(C(=O)NCC2(OC)CCCCCC2)=O)CCC(C)CC(C)C1 n1(-c2scc(CC(=O)NCC(CN(C(CSC)=O)C)O)n2)c(C)ccc1C C(=O)(C1CC(=O)Nc2ncn(C)c21)OC.C12(C)CC(F)(F)CN1C2=O C1(CC(N2C(C(C)O)CC2)=O)CN(C(=O)CCCn2cccc2)CCO1 Cc1nccnc1C(=O)NC(C)CCN(C(=O)Cc1cncs1)C C(C(C)(C)C#CC(=O)NCc1csc(C)n1)NC(C(C)=CCC)=O CC1CN(C(C2(C#N)CC3(CC3)C2)=O)CCC1NC(C1(C2CC2)CCC1)=O CC1(C(=O)NCC#CCNC=O)CC12CCN(C(c1ccon1)=O)CC2 c1(CC)c(C(N2CCC(C)(Cn3cncn3)C2)=O)cnn1-c1ccc(Cl)cc1 N1(C(CCC(C)OC)=O)CC(N(C)C(c2ccnc(C(F)(F)F)n2)=O)C2(CC2)C1 c1(NC(C(C)SCCCC)=O)cc(C(=O)O)c(CC)cc1OC C1(C#N)(C(NNC(=O)OC(CC)C)=O)CC2CCC1CC2 N#Cc1c([N+](=O)[O-])cccc1S(=O)(=O)N(CC(O)CO)C1CC1 N1(C(=O)NC2CCC(C)C2)CCN2CCCC2C1 C1(C(NOCC=C)=O)CN(C(=O)COCC2CCC2)CC12CC2 CCCC(CC1CCCCC1)C(=O)OCC(=O)NC(=O)NCC(C)C c1(SC)cccc(NC(=O)Cc2ccc(C3CCNCC3)cc2)c1 Cc1ccoc1CC(=O)NCCC1(CNC(C2COC(=O)C2)=O)CC1 c1(C(N2C(C)(CNC(C3C(CC)OCC3)=O)CCC2)=O)cc(O)cc(O)c1 C=CC(CC(=O)NCCNC(c1sc(F)cc1Br)=O)c1ccccc1 C1(NC(C2N(C(C(COC)N(C)C)=O)CC=CC2)=O)CC(C)(C)OC1=O Cc1csc(=O)n1CC(=O)NC1COCC1N1CCN(C(=O)CCC2CC2)CC1 c1(OC2CC(NC(C(C)N(C)CCc3nn[nH]n3)=O)C2)cccc(Br)c1 N1(C(CC2N(C(C)C)CCC2)=O)CCC(NC(C2COC(=O)N2)=O)C1C C(=O)(C(C)C(C)c1ccccc1Cl)NCCCN(C(c1c(CC)noc1)=O)C c1(CCN)nccc(C(=O)N(CC2CC2)CC2CCCO2)n1 C1(NC(c2c(C)nc(C3CC3)o2)=O)Cc2ccccc2C1Nc1cncc(Cl)n1 N1(C(C(C)O)=O)CCC(NC(=O)COC2CC2)CC1.N12CC(C1)C2=O c1(C(N2C(c3ccc(OC)cc3)CC(C)C2)=O)ccc(I)c(Cl)c1 C(C)(C(=O)NCC(C1CC1)OCC)N(C(CSCCC)=O)C1CC1 CC(C)CCC(F)C(=O)NCCOCCOCCCNC(=O)C(C)C#N C1(CC=C)(NC(=O)CC2CC(SCOC)C2)CCOC1.C12CCC1CC(=O)N2 c1(OC)ccc2c(CC(=O)NCC=CCNC(c3cnc(Cl)n3C)=O)c[nH]c2c1 C1(C2CCN(C(=O)CC(O)CN(C)C)CC2)(NC(C2C(C)CC(C)O2)=O)CC1 C1(CC(=O)NCC2CC(NC(Cc3cn(C)nn3)=O)C2)CCCCCC1(F)F C1(C)(C(=O)NCC2(NC(c3c(SC)ccs3)=O)CCOC2)CCC(=O)N(C)C1 C(=O)(CCS(=O)(=O)Cc1ccncc1)NCCCNC(CSC(C)(C)C)=O C1(CNC(=O)CCc2c(C)n[nH]c2C)COC(C)(C)CN1C(CCC(=O)OC)=O CC(C)C(N=[N+]=[N-])C(=O)NC(Cc1cn[nH]c1)C(N1CC2(CCCN2C)C1)=O c1(-c2cc(OCC)cc(OC)c2)n[nH]c2c1CN(C(=O)C(C)O)CC2 CCCCCC(C)(CC)C(=O)NCCC1(O)CN(C(=O)CC2CC2(Cl)Cl)C1 c1(C(=O)NC(C)CN(C)C(C2CC2C2CC2)=O)cc2ccccc2n1C C1(F)(CNC(C(C2CC2)OCC)=O)CCC(CNC(=O)C=CSC)CC1 c1(C(=O)NCC2CN(C(c3n(C(CC)C)ncc3)=O)C2)nn(C(C)C)cc1Br C1(C(N2CC(NC(=O)CCCCN(C)C)C2)=O)(COC)CCCCO1 c1(C(=O)NCC2C(OCC)(OC)CC2)ncoc1-c1cc(C)no1 C(CCSC)(C(=O)NOCc1ccccc1)NC(Cc1cc(CC)no1)=O c1(OC)ccc2cc(C(N3CCC(C)(NC(c4ncoc4C)=O)C3)=O)n(C)c2c1 N1(C(CSc2nc(C)cc(C)n2)=O)CCC2CCN(C(c3cc[nH]c3)=O)C2C1 C=CC1OCCC1C(=O)NC(C1(O)CN(C(=O)CC2(C(F)(F)F)CC2)C1)C C(=O)(C(C)OCCCN(C(COCCCN(C)C)=O)C)NCC=CCNC(N)=O N1(C(CSS(C)(=O)=O)=O)CCCCC1C1CCN(C(=O)C2=C(Cl)CC2)C1 C1(CNC(C(n2cc(Cl)cn2)C)=O)CCN(C(c2ccc(F)c(F)c2)=O)C1(C)C c1(CN2CCC(O)(C(=O)Nc3cccnc3Cl)C2)ccc(Cl)c(I)c1 C1(C(=O)NCC2CN(C(=O)Cn3cnccc3=O)CC2O)COC2(CCC2)C1 Cc1nn(C2CCCN(c3nnnn3C3CCC(C(=O)N(C)C)CC3)C2)c(C)c1Cl C12(C(=O)NC(CNC(c3ccc(CC)[nH]3)=O)C)CCC(C1)OC2 c1(C(N2C(CNC(C(C(C)C)F)=O)C(C)CCC2)=O)nccc2ncccc12 CC1C(NC(=O)NCCCCc2ccccc2)CCCN1C(=O)OC(C)(C)C C#CCC(CC#C)C(=O)N1CCCCC(N(C(=O)CC(C)C(F)(F)F)C)C1 Cc1cccc(N)c1C(=O)NC(CNC(=O)C(C(C)C)c1ccccc1)CO N1(C(c2c(CC)noc2)=O)CC2(CC(NC(=O)C(N3CCCC(C)C3)=O)CO2)C1 Cc1[nH]c2ccccc2c1CCNC(=O)NC1CCCC1CO c1(N2CC(CCC)OCC2)[nH]c(=NC2CC(N(C)C)C2)nc2c1cnn2C(C)C N1(C(CCNS(CC)(=O)=O)=O)CCCC1C1CCN(C(=O)CNC(=O)C2CC2)C1 C(=O)(C(F)C(F)(F)F)N(C)CC1CCCN(C(=O)Cc2ccn(C(F)F)n2)C1 N1(C(C2(C#C)CC(=O)C2)=O)CCC=C(C(=O)N2CCC=C(C)C2)C1 c1(C(CNC(c2cc(C)[nH]n2)=O)NC(=O)C(F)(F)c2cscn2)ccc(F)cc1 C1(CC)(NC(=O)C(O)C2CCC2)CCN(C(=O)Cc2cccc(C)c2F)CC1 C1(C2(C(=O)NC(C)Cn3cncn3)CC2)CCCN1C(c1cccnn1)=O CCCCCC(=O)N1CCCC(N(C)C(C2CC2Br)=O)C1 C1(CNC(Cn2ccc(C)n2)=O)CN(C)CCN1C(c1ccc(C(C)C)cn1)=O c1(C(=O)NC2CC(N(C(=O)CSC(F)(F)F)C)C2)cccn2ccnc12 C1(C(=O)NC(CNC(c2c(CC)n(C)nn2)=O)C2CC2)C2CCCCCC12 N1(C(C(COC)OC)=O)CC(NC(c2ccoc2)=O)CCC(O)C1 C1(C(N2C(CCNC(=O)C(F)C3CC3)COCC2)=O)CC2CCC1CC2 c1(C(C(=O)Nc2n(CC)ncc2)O)ccc(CC(=O)Nc2cc(C)[nH]c2C)cc1 NS(=O)(=O)c1ccc(C(=O)NC2CC3(C2)CN(C(=O)Cc2cncnc2)C3)[nH]1 C1(NC(c2conc2C2CCCC2)=O)CCN(C(=O)C(O)CC2CCOCC2)C1 C1(C(=O)NCCOCC#C)CCC2CCC1N2C(c1cnn(CCO)c1)=O C12(C(N(CCCNC(=O)Cc3cc[nH]n3)CCO)=O)CCC(F)(CC1)CC2 N1(C(c2cn(C)nc2)=O)CCC(NC(c2ccc(C#N)o2)=O)C(CO)C1 Cc1cc(C(N2CCC(N3CCN(C(=O)CC4CC4(C)C)CC3)C2)=O)c(O)nn1 CC(CC(=O)NCC(C)CN(C)C(C1CC(C)(C)C1)=O)c1ccco1 N1(C(c2c(CC)nc[nH]2)=O)CCC2CN(C(=O)C(O)CC[S+](C)C)CC2C1 C1(N(C)C)(CC)CCN(C(=O)C(C)CNC(=O)CC2(C)CCCCC2)C1 CN1CCN(c2ncc(C(=O)NCC34CC3CN(C(=O)C(=O)N(C)C)C4)s2)CC1 c1(NC(CC)(CNC(=O)C(C)CF)CC)ccc(C#N)c(C)n1 c1(C(N2C(C(=O)Nc3cc(OC)cc(F)c3)CC2)=O)c[nH]c2ccc(F)cc12 C1(NC(CC2N(C)CCCC2)=O)CCCCCCC1NC(=O)CCC1CCCO1 CS(C)(=O)=NCC(=O)NC1CCN(C(c2ncsc2C(F)(F)F)=O)CC1CO c1(OC)ccc(C(N2CCN(C(=O)Cn3cnnc3O)C3CC23)=O)cc1Cl C(CCCC(C)NC(=O)C(CC1CC1)CC1CC1)NC(c1c(C)con1)=O C(=O)(CC(C)CC(C)(C)C)NC1CN(C(c2cnc(C)n2C)=O)CC1O CC1CC(NC(=O)C(=O)Cc2ccccc2)CCN1C(c1cocn1)=O CCC(CC)C(=O)N(C(CC)CC(=O)NCCC1(COC)CCC1)C c1(C(=O)NCC(CC)NC(c2cnc(C)[nH]2)=O)c(C)oc(C)c1Br c1(C(C(C)C)NC(C2(c3ncon3)CC2)=O)ccccc1Cl C(=O)(CCCNC(=O)CCOC(C)CC(C)C)NC(CC)Cn1cncn1 C(CCCNC(=O)CCC1CCCOC1)(c1ccccc1)NC(C=C(C)Cl)=O CCCC(C(=O)N1CC(CCNC(=O)CSC(F)F)C1)S(N)(=O)=O c1(CCC(=O)NCCN2CCN(C(C3C(=C)CC3)=O)CC2)ccc2ncsc2c1 C1(C(N2C(C(C)C)CCC2)=O)CCN(C(=O)COC2CC=CC2)O1 C1(CC)(NC(=O)C(C)CC(F)F)CCN(C(c2ccncc2)=O)CC1 c1(CC)sc(C(=O)NCC2CCN(C(=O)CCC3CCOCC3)C2)cc1C c1(N(CC=C)C)ccc(Br)c(S(=O)(=O)NCCc2c(F)cncc2F)n1 c1(CC(=O)NCCC2(C(=O)O)CC2)ccccn1 C1(CNC(C2(OC)CCCCC2)=O)CC2CCC(C1)N2C(=O)C(C)C1CC1 N1(C(Cc2c(OC)c(F)ccc2)=O)CC2CCCC(C1)N2C(=O)C(=O)NC(C)C Cc1cccc2[nH]c(C(N3CCC4CCC(NC(=O)C(O)CN(C)C)C34)=O)cc12 C1(C)(C(=O)NC2C(NC(c3n(C)ncc3)=O)COCC2)CCC(O)CC1 C(C(C)(CC(C)C)n1cc(C(F)(F)S(=O)(=O)CCl)nn1)c1cccc(C)c1 C12(NC(c3nn(CC)c(C)c3)=O)CCCC1CN(C(c1cc(C)oc1C)=O)C2 C(=O)(C(C)(C)CC(C)C)NCC1OCCC(NC(c2c(Cl)cnc(CC)n2)=O)C1 C1(C(=O)N(CC)CC2CCN(C(=O)CC3CCCC3)C2)COCCN1CC(F)(F)F Cc1cc(Br)c(Cl)cc1C(=O)N(c1ncccc1F)C C1(C)(NC(C(C)CCN(C)C)=O)CCCN(C(=O)CC2CCC(C)C(C)C2)C1 C1(CNC(C(COC)C)=O)CC2CCCCC2N1C(=O)CCn1cccnc1=O N1(C(CC(C)OC)=O)CC(NC(c2[nH]nc(C(F)(F)F)c2C(C)C)=O)C(C)C1 c1(C(=O)NC23CN(C(CCNC(=O)OC)=O)C(C2)C3)c(C)[nH]c2ccccc12 Cc1ccc(C(=O)NC(C2CCN(C(=O)CC3COCCO3)CC2)C(C)C)c(C)c1 c1(OC)ccc(CNC(C2CN(C(C3CCCCO3)=O)CC23CC3)=O)c(OC)c1 C(=O)(C#CC1CCCCO1)NCCCN(C(c1c(Br)ccc(C)n1)=O)C(C)C Cc1cc(CO)oc1C(=O)NC1CN(C(c2nc(Cl)cs2)=O)CC1C c1(C(C)C(=O)NCC2(F)CN(C(=O)CCN3CCCC3)C2)nc(F)ccc1Cl N1(C(C(C(CC)O)C)=O)CCc2cc(CNC(c3ccc(F)cc3)=O)ccc2C1 N1(C(CCC)=O)C2CCC1CC(CNC(c1ccc(OC(F)F)cc1)=O)C2 c1(C(=O)NCC2(NC(C(C)OC3CCOC3)=O)CCC2)ccc(N)cc1Cl C(=O)(C(CNC(c1ccn2nccc2c1)=O)CC(C)C)NCCN(C(=O)OC)C C1(CNC(C2CCC(=O)NC2)=O)CC2(CCN(C(c3cc(Cl)cnn3)=O)C2)CO1 CN1CC(C)(C)CC1C(N1CCCC1(C)c1cn(-c2c(F)cccc2Cl)nn1)=O Cc1cc(C(N2CCCCC(NC(c3ccc(Cl)nc3O)=O)C2)=O)nc(C)c1 C(=O)(C1=NOCC1)N(CC(CC)NC(=O)Cc1cccc(OC(F)F)n1)CC N1(C(=O)CS(=O)(=O)N2CCOCC2)CCC2CCN(C(=O)C(F)C3CC3)C2C1 CN1N=CC(CC(=O)NCC2CN(C(C3CCS(=O)(=O)C3)=O)C2)C1=O CCC(C#N)C(=O)NC1(C)CC(NC(c2cc(CCCO)on2)=O)C1 c1(CNC(CC(C)c2ccccc2)=O)ccc(CNC(c2cnsc2)=O)c(F)c1 c1(NC(CNCC2CC(OC)(CN)C2)=O)ccc(C)c(Br)c1 C1(CC(=O)NC2(COC)CN(C(=O)C(CO)N(C)C)C2)CC2(CC2)CO1 C(=O)(C1=CCc2ccccc21)N1C(CNC(c2cc(CCOC)on2)=O)C=CC1 c1(C(=O)NCC2C(NC(C(CC(C)C)O)=O)CCC2)ccc2c(c1)CC(C)O2 Cc1nn(C2CC2)cc1C(=O)NC1CC(NC(C2(C(=O)OCC(C)C)CC2)=O)C1 c1(C(N2C(CN(C(C3CN(CC)C(=O)C3)=O)CC)CCC2)=O)cncc(Cl)c1C N1(C(C(COC)(C)O)=O)CCN(C)C(CNC(=O)Cn2nc(C)cc2C(F)F)C1 c1(NC(C2C(C(=O)OC)C2)=O)cc(C(=O)NCCCC(F)(F)F)cnc1Cl C#CC1CC2(CC2)CN1C(=O)NCC(C(C)C)c1ccccc1 N1(C(C(C)N(CC)CC)=O)CCC2CCCC12C(=O)NCC1CCC(C)(CC)O1 C(=O)(CCCCCCC(=O)NC(CO)C(C)NC(=O)C(=O)NCC(F)F)OC N1(C(C2CC(O)CN2C2CC2)=O)CC2(CC2)CC1C(N1CC2CC1C2)=O C(=O)(CC1=CCCCC1)N1CC(C=C)C(NC(C2CC(C)CC(=O)N2)=O)C1 CN1CC2CC1CN(C(C1N(C(=O)COC(C)(C)C)CCC1(C)C)=O)C2 C1(NC(CC2CCCC(C)C2)=O)CC2CCC1N(C(c1coc(Cl)n1)=O)C2 C1(CNC(c2c(CNC(CCC#C)=O)ocn2)=O)CCC(=O)NC1C C1(CNC(C(C)CCN(C)C)=O)CC2(CCN(C(C3(C)CCCN3C)=O)CC2)C1 c1(C(C)C)ncc(Br)c(=NC(CNC(C2CCC(=O)N(C(C)C)C2)=O)CO)[nH]1 C1(C)(C(N(CCOCCNC(C(C)CSc2ccccc2)=O)C)=O)COCCO1 c1(NC(=O)NCC(=O)NCC(CC)NC(=O)C(O)CF)ccc(F)cc1F c1(N(C)CC2CCCO2)nc(N2CCN(Cc3ccco3)CC2)c2c(n1)CCS2 N1(C(c2ccc(OC)cc2)=O)CC(C(N2CC(C(C)C)C2)=O)CCC1(C)C C(C1CCCC1)=C(C)C(=O)NCC1CN(C(C2(n3cc(C(C)C)nn3)CC2)=O)C1 N1(C(C(CSC)O)=O)CC(NC(=O)CCc2csc(C)n2)C(C2CC2)C1 CCC(C)(C(=O)NCCOCCCNC(=O)Cc1ccoc1)OC N#Cc1cnn2cc(-c3nc(CC4CCCS(=O)(=O)C4)no3)cnc12 C(=O)(CCCCC(C)C)N1CC(N(C(C=C(CCC)C)=O)C)C(C)(C)C1 C(C(O)C(C)(C)C)N(C(c1scc(CNC(CC2C(CC)C2)=O)c1)=O)CC c1(C(N)=O)cc([N+](=O)[O-])cnc1NC1CCCC(NC(=O)C(C)(F)C(C)(C)F)C1 CCC(C)(C)C(O)C(=O)N(CCC(=O)N(CCO)C)C.C(C(C)(C)OC)OC C#Cc1ccnc(C(=O)NC(CCC)C(=O)N2CC(CC3CC3)C2)c1 c1(C(=O)NC(CN(C(C2N(CC)CCC2)=O)C)C)[nH]c(C)nc1C c1(C(=O)NCCCC(CCC)NC(C2CCN(C)C2=O)=O)cn2cccnc2n1 Cc1noc(C)c1CC(=O)NC1CCCCN1C(=O)C=CCOC1CCCCC1 C1(C2CCC2)(CNC(C(C#C)(C)C)=O)CCN(C(=O)CC(C)c2ccco2)CC1 C1(N(C(c2cc(C)cc(F)c2N)=O)C)CCCC2CN(C(=O)C3=CCSC3)CC12 C#CCC(CC(=O)NCC1C(CO)C1(C)C)NC(C1(C)CCCCCC1)=O C(=O)(C1CCc2nccn21)NC1(COC)CCCN(C(=O)C=CCO)C1 C(=O)(C(CC(C)C)NC(=O)NC(C)C(C)n1cncn1)NC c1(C(=O)NC2CCN(C(c3nc(=O)n(C)[nH]3)=O)CC2)cc(N(C)CC)nc(C)n1 N1(C(CC(C)=C(C)C)=O)CCCCC1CC(=O)NCCCCC1CC1 C1(C(N)=O)CCCC2(CCN(c3nnc(CC4CCCC4)n3CC(C)C)CC2)O1 C1(O)(C(C)NC(=O)CC2(C)CC2)CN(C(=O)CCCc2ccccc2)C1 C1(C)(CNC(CN(CCOC)C)=O)CCC(NC(=O)C(C)=C(C)CC)C1 c1(-c2ccc(C)c(CO)c2)ccc(S(=O)(=O)C2CC2)cc1 c1(OC)c(Br)ccc(F)c1C(c1nnnn1CCC1(C)CC1)NCCC1C=CCC1 C(C(CC(=O)NC1CN(C(=O)CC2(C)CC2)CC(C)(C)C1)C(F)F)N(C)C C(=O)(C(C)CC(F)(F)F)NC1C(CCC)CN(C(C2C=CC=CC=C2)=O)C1 c1(OCC(=O)NC2(CNC(C3(OC)CCCC3)=O)CCCC2)cccc(C#N)c1 c1(C(N2CC(CC=C)(NC(c3nc(C)sc3C)=O)C2)=O)cc(C#N)ccc1O C(=O)(CCC(O)C(C)(C)C)NCC(C)N(C(c1cc(SC)ncc1)=O)C N(C(=NCCCF)NCC(C(=O)OC(C)(C)C)C1CC1)C(CC)CC C1(F)(CNC(c2c(C)cnn2C)=O)CC2CCC(C1)N2C(C1CCC(C)(C)C1)=O CC1CN(C(c2cccc(C#N)c2)=O)CCC1N(C(=O)C1=CCOCC1)C N1(C(CC(=O)NCC)=O)CC(NC(=O)COC2CCOC2)C(c2cnn(C)c2)C1 c1(OCC)cc(Cl)ccc1C(=O)NC1CN(C(C2CCCC2(F)F)=O)C1 c1(C(=O)NCC2CCC(C)N(C(c3cc(Cl)ns3)=O)C2)cccc2c1OCCN2 c1(OC)ccc(CN2CC3CN(C(c4ccc(Cl)o4)=O)CC23)cc1F C1(NC(C(CC#C)NC(=O)CCCCCF)=O)CC2(C1)CC(C#N)C2 N1(C(COCC)=O)CCN(C(c2scnc2COC)=O)CC1CC CCCCC(C(=O)N1CC(CNC(=O)CC(C)(C)O)CC12CCC2)C(C)C C(CC1CC1)(CC(=O)N1CCOCC1CCO)NC(c1ccn(COC)n1)=O N1(C(C2C(C)CCC2)=O)CCC(C(C)(C)C)(CNC(=O)COC(F)F)C1 CCC(CCC(=O)N(C(C)CN(C)C(c1ccc(C(=O)OC)s1)=O)C)OC C(=O)(C1=CC2CCCC12)NC1(CNC(CNC(C(C)(C)C)=O)=O)CC1 C1(CC(=O)NC2(C(C)O)CC2)CCCN(C(C2CC(F)C(=O)N2)=O)C1 C12(CNC(C3CC(C#N)C3)=O)CCC(NC(=O)Cc3cccc(Cl)c3)(CC1)CO2 CC1=C(C(=O)Nc2ccc(-c3ccc(OC(C)(C)C)cc3F)nc2C)CCO1 N#CC1CN(Cc2cc(Cl)ncc2Br)CC1NC(=O)C(=O)c1ccco1 N1(C(C2(S(C)(=O)=O)CC2)=O)CC2CCCC2(CNC(=O)Cc2ccc(O)cc2)C1 c1(NCCOCCNC(Cc2c(CC)cccc2)=O)ncc2ncnc-2[nH]1 CC1CN(C(c2cnnn2C)=O)CC1NC(C1(C)C=CCC1)=O N1(C(C2N(C(c3c(CC)nn(C)c3)=O)CC(C)C2)=O)CC2CC2C2CC12 C1(NC(C2CCSCC2)=O)CCCC(CC(=O)NCC(CN(C)C)O)C1 C1(C(=O)NCC2CC(F)(CNC(Cc3n[nH]c(=N)s3)=O)C2)CCCN1C=O C#CC1CN(C(=O)CC2CN(C)C2)CCN1C(c1ccnc2c1CCO2)=O N1(C(c2c(C)cnnc2)=O)CC2CCCC(C1)N2C(C12CCC(C)(CC1)CC2)=O c1(OC)cncc(C(=O)NCC2(F)CCC(CNC(C3(CCF)CCC3)=O)C2)c1 c1(C(=O)NCCC2(O)CCN(C(=O)CCC3CC3(F)F)C2)cc(Cl)cnc1O c1(C(N2CCC(N(C(=O)C3=NOCC3)CCC)CC2)=O)cn2c(n1)CCC(C)C2 C1(NC(C#C)CC2CCOC2)CCOC2(CCC2)C1 C(C(C(=O)NC1(CO)CC(F)C1)C(C)(C)C)NC(CCCC#C)=O CC(C)CC(C)(CNC(c1csnc1Cl)=O)NC(=O)CCCCN(C)C Cc1cnn(C)c1CC(N1CC(N(C(=O)CN2CC(C)C2)C)C(O)C1)=O C(=O)(C1c2c[nH]nc2CN1C(=O)CSC(F)F)NCc1cc(OC)ncn1 N1(C(c2ccc(CN=[N+]=[N-])o2)=O)CCC(NC(=O)CCSC2CCCC2)C(O)C1 c1(SC)cc(F)ccc1C(N1CC(C)(NC(C2CCC(N(C)C)CC2)=O)C1)=O C1(C(=O)NC2CC(CNC(c3c(C)cc(Br)cn3)=O)C2)CCC2CCC(=O)N12 O=C1NCC2(CCN(c3nc(N4CC5CC4CS5)nc4cc[nH]c34)CC2)N1 CC1(F)CCN(C(C2(C)CN(C(=O)CCn3cccc3)CC2C)=O)CC1 Cn1ccc(C(N2C3CCC2C(CNC(C2(c4cccs4)CC2)=O)C3)=O)cc1=O Cc1ccn(CC(=O)N(CCNC(=O)C=CCl)CC2CC2)n1.C1(=O)CCN1CCO C1(CC(=O)N(CC(C)O)CCNC(c2c(C)n[nH]c2)=O)CC(C)(C)CO1 C1(O)(C(C)C)CCN(C(=O)CC2CCCN2C(=O)CC2CCOC2C)C1 Cc1n[nH]c(=NC(C)CNC(=O)COc2cnn(C)c2)o1 C(=O)(CCC(=O)c1ccc(F)cc1)NC1C(CNC(C(C)(F)F)=O)CCC1 C1(C(N(C)CC2N(C(CCSCC(C)C)=O)CCOC2)=O)Cc2cccnc2C1 C1(Cn2cc(C(C)OC)nn2)N(C(C23CSCC2C3)=O)CC1(C)C c1(C(=O)NCC2=CCN(C(C(C=C)(C)CC)=O)CC2)c(Cl)cc(Cl)c(Cl)c1F c1(NCC2C(C)CN(C(C3CNC(=O)CC3C)=O)C2)c(C#N)c(=O)n(C)c(=O)n1C N1(C(CCNC(=O)OC)=O)CC2CC1(CNC(c1cc(C3CC3)[nH]n1)=O)C2 n1(CC)cc(CC(=O)NC2CC(CNC(=O)C(C)C(C)(F)F)C2)c2ccccc12 c1(C(=O)OCC)ncc(Br)cc1NCC1(c2cccs2)CC1C C1(C)(NC(C2(CC#C)CCCO2)=O)CCN(C(=O)C#CC2CC2)CC1 N1(C(c2c(S(C)=O)cccc2)=O)CCC(C2CCCN(c3nnno3)C2)CC1 CC1(C)C2CCC1(C(N1CCN(C(c3cc4scnc4[nH]3)=O)CC(O)C1)=O)CC2 c1(OC)c[nH]c(C(=O)NCCCCCCNC(c2cncn2C2CC2)=O)cc1=O Cc1cccc(C(=O)NCCC(C)CCNC(=O)C(F)n2ccnc2)c1C C1(CC)(CC)CC(NC(c2sc(C)cc2Cl)=O)CN1C(=O)C=CS(C)=O C1(CCNC(c2ccc(=O)n(O)c2)=O)CC(N=c2nn[nH]n2-c2ccccc2)C1 C1(NC(C(CC)NC(N)=O)=O)CCN(C(=O)C(Cl)=CCl)CCC1(F)F C1(O)(CCNC(C2CC(OC)C2)=O)CCCN(C(=O)CCCc2nncn2C)C1 C12(c3ncn(C)c3)CC(CN1C(=O)Nc1cccc(C(=O)N)c1)C2.C1CC1 c1(C(C(=O)NCC(C)NC(C2C3CCC23)=O)C)ccc2c(c1)OCCO2 CN1CC(C)(C(=O)N(CCCn2cc(CCC3CC3)nn2)C2CC2)CCC1=O N1(C(C(C(C)C)O)=O)CCOC2(CCCCC2NC(C2CNC(=O)C2)=O)C1 C1(NC(C(CCN(C)C)O)=O)CC2CC1N(C(C1(CCO)CC1)=O)C2 c1(C2C(CNCc3nc(CC)on3)C2)ccc(Br)cc1 C1(C(F)(F)F)(NC(N2CCN(CCOCCO)CC2)=O)CC2CCC1CC2 CC(C)P(=O)(CC(=O)N(C)CC1(O)CCN(C(=O)C=C2CCOCC2)C1)C(C)C CCCC(C(=O)NCc1ccc[nH]1)NC(c1cc(C(=O)OC)ccn1)=O c1(C(=O)NCC(CC)NC(=O)CCC=CBr)cc(N)cc([N+](=O)[O-])c1 CCC(CCC(=O)NCC1(CO)CCN(C(=O)CCCn2ccnn2)C1)OC c1(C(=O)NC2C(NC(c3c[nH]c(C)c(Br)c3=O)=O)CC2)cccn2c(O)nnc12 C1(CC)CN(C(=O)CCNC(c2cc(CO)c(C)o2)=O)CCN1C C1(NC(CSCCC)=O)CCCCC1CNC(C1C2CCCOC12)=O N1(C(c2cncc(C)c2Cl)=O)CC2(C1)CN(C(C1(C)CC1F)=O)CCO2 C(=O)(C(CCCC)C(C)C)NCC(C(=O)N(C1CCCC1)CC#CC)CC1CC1 N1(C(c2nncs2)=O)CCOC2(CCN(C(C3(n4cccn4)CC3)=O)C2)C1 C(=O)(C(C)(C)CF)N(C)CC1C(NC(C(CC)OC)=O)CCC1 c1(C(N2CCC(NC(=O)CCC(F)F)CC2C2CC2)=O)ccc(Cl)c(F)c1F CCC(CN=c1ccc(S(=O)(=O)NC2CCC3(CCC3)CC2)c[nH]1)n1cccn1 Cc1cccc2[nH]c(=NC3CC(CNC(=O)C4=CCCC(C)(C)C4)C3)sc12 N1(C(=O)NCCn2nnc(C)n2)CCC(OC)C1(C)C C1(C(N2C(C)CC(CNC(c3ccncc3)=O)C2)=O)CC2C=CC1C21CC1 CC1CSCCCN1C(C1CNC(=O)CN1C(C1CCCC1)=O)=O C1(C(=O)NCCn2cc(C(N3CC(OCC)C3)=O)nn2)OCCC1(C)C N1(C(c2c(CCC)nns2)=O)CCC(F)(F)C(CNC(c2sc(F)cc2C)=O)C1 C1(C(=O)NCC=CC)CCN(C(=O)Cc2cccnc2)C1C N1(C(=O)Nc2cc(C)[nH]c2C)CCCc2cccc(OC(F)F)c21 N1(C(=O)OC)CCOC(C)C1CNC(C)(C)C.c12cn(nn1)C1CC(C1)NC2=O CC(C)CC(C)CC(=O)N1CCC(F)C(NC(=O)C(C)(C)n2cnnn2)C1 c1(C(=O)NC2C(OC)CN(C(=O)CC(C)N(C)C)C2)cccc(C)c1O N1(CC)N=C(C(=O)NCC2CCN2C(c2cc(C3CCC3)[nH]n2)=O)CCC1=O N1(C(C2(C(=O)OCC)CC2)=O)CC(COC)CC(C)C1 C1(C(=O)NCC2N(C(c3cc(C(C)C)n(C)n3)=O)CC=C2)CN(C)C(=O)CCO1 CC1C(NC(C2CCCS2(=O)=O)=O)CCCN1C(=O)CC1CN2CCN1CC2 CCCC(CCO)NC(=O)Nc1ccnc(N2CCC(C)C2)c1 c1(-c2nnc(C)o2)ccccc1C(=O)N(C(CNC(C12CCC1C2)=O)C1CC1)C c1(C(=O)NCC2CC(NC(CCOC)=O)C2(C)C)ccc2nnn(C)c2n1 C1(CC(C)C)(C(=O)NC2CCC(CNC(C3(C#N)CC3)=O)C2)CCNC1=O c1(C(=O)NCC(CC=C)NC(=O)CSC(C)C)cn(C)cc1C(F)(F)F c1(C(=O)NC2CC(CNC(C(C)NC(=O)OC)=O)C2)cnc(SC)nc1O N1(C(CC2(C=C)CN(C(C3(C(N)=O)CC3)=O)C2)=O)CC(C)OCCC1C N1(C(C(c2nc(C)sc2)=O)=O)CC2CC(C1)C2NC(C1CCCC1C)=O c1(CC)ccc(C(=O)NCCC2CC(F)(F)CN2C(c2cnsn2)=O)cc1F C1(C)(C(N2CC(F)(CNC(CC(n3c(CC)ncc3)C)=O)C2)=O)CC2CC2C1 C(=O)(C(C(C)NC(c1ncccc1Cl)=O)C(C)C)Nc1c(OC)cc(F)cc1 C12(CNC(c3ncn(C)c3)=O)CC1CN(C(=O)CCCC1CCOCC1)C2 C1(CC(=O)Nc2n(C(C)C)nc(-c3ccccc3)c2)CN2CCC1CC2 C(=O)(CCCC(C)(C)C)N(CCCNC(C1CCC(C)S1)=O)CCO c1(CCOC)oncc1C(=O)NC1CCC(CC(N2C(CO)CC2CO)=O)C1 C=C(C)c1ccccc1NC(=O)CCOCCCNC(C1CCCN1C)=O c1(CC)nc(N2CC3CC2(CNC(=O)CC(C)(O)COC)C3)c(F)c(Cl)n1 CC1(C)CCC1C(=O)NCC1(CCNC(c2ccn(C3CCCCC3)n2)=O)CC1 N1(C(C(CC)SC)=O)C(C)C2CC1C2NC(=O)CNC(C1CCCC1)=O C1(NC(C2(CCC)CC2)=O)CC2CCC(C1)N2C(=O)C1=C(C)CCCC1 c1(C(=O)NC2C(C)N(C(=O)CC3CCSCC3)CCC2)cnc(O)n(C)c1=O c1(C(C)=O)cccc(C(N2CCOC(CNC(=O)CSCC(N)=O)C2)=O)n1 N1(C(c2c(C(=O)OC)scc2)=O)CCCCC(Cn2cc(CNC(N)=O)nn2)C1 C1(NC(C2CCN(CCF)C2=O)=O)CN(C(=O)COC2CCOC2)CC1C(F)F c1(C(C)(C)C)scnc1C(=O)N(CCNC(C1CCCN1C1CC1)=O)C1CC1 C1(C(N(CCCN(C(CC=C)=O)C)C)=O)CC2(C1)CC(F)C2 C1(OC)CC(NC(c2cncnc2)=O)CN(C(=O)Cn2ncc(Br)n2)C1 C1(NC(C(n2c(C)ccn2)C)=O)CCN(C(=O)COc2ccc(O)cc2)CC1 C(=O)(CCN=C(NCC1CCC2(C1)OCCO2)N1CCN(CCOC)CC1)NC CCCCC#CC(C)(C)NC(C1CC(O)CN1C(C1CCC(=O)N(C)C1)=O)=O Cc1cc(=NC(C)c2ncnn2C(C)C)[nH]c(=NCc2nccc(O)n2)[nH]1 C(CC(O)C(=O)NCC(CC1CCCC1)C(=O)NCC(c1ccccc1)C)SC C1(c2onc(CN(C)C)n2)CN(CC2(C)CSCCO2)CCO1 N1(C(c2cc(C)[nH]c2C)=O)CCCC(CO)(NC(C2CCSC(C)C2)=O)C1 c1(CC)occc1C(=O)NC1(C(=O)N(CCF)CCOC)CC1(C)C c1(C(N2CCC(CNC(Cc3c(C)scc3)=O)CC2)=O)ccc(F)c(C2CC2)c1 c1(N2CCC(OC(C(C(C)C)N(C)C(=O)N(C)C)=O)CC2)c(F)cccc1F C(=O)(C(O)CCCNC(=O)CC1CSC1)NC(C1CCOC1)C#C N1(C(c2cc(C)on2)=O)CCCC(C2CN(C(=O)C(C3CC(F)(F)C3)O)C2)C1 c1(OCC(=O)NCC(CC)NC(c2cncc(F)c2)=O)cncc(Br)c1 C1(C(N(C2CCCN(C(=O)Cc3ccc(C)nc3)C2)CC)=O)CCN(C)C(C)C1 C1(C(N2CCC(NC(CN(C(C)C)C)=O)C2)=O)CC(c2ccccc2)=NO1 C1(C(=O)NC(CC=C)(C)C)C(C)CCN1C(=O)C=Cc1cocn1 N1(C(=O)NCc2c(CC)nn[nH]2)c2c(Br)cccc2CCC1C N1(C(c2ccc(C(C)C)s2)=O)C2CCC(C2)C1CNC(=O)C(C)C#N Cc1cncc(C(=O)NC2CCCC(NC(=O)CCc3ccccc3Cl)C2)c1 N1(CC)CC(C(N2CCC(C)(NC(=O)C(F)=CCCF)C2)=O)NC1=O c1(C(=O)NC2CCN(CC(Cl)=CCl)C2)ccccc1C1CC1 c1(C(=O)NC2(C)CN(C)C(=O)CC2)cc2n(c1)CCCNC2=O c1(CC(=O)NCC(CNC(C2(CC=C)CCC2)=O)C)ccc(F)c(Br)c1 CC1CC=C(C(=O)NC2CCCCC2NC(=O)COc2ccc(Cl)nc2)CC1 N1(C(c2ccc(N(C)C)cn2)=O)CCCCCC(Nc2ccccc2[N+](=O)[O-])C1 c1(C(N2C(Cc3cn(-c4ccc(OC)cc4)nn3)CC2)=O)ccc(Br)c(F)c1F O=C(N=c1[nH]sc2ncccc12)C1CC(O)CN1C(c1c(Cl)cncc1Cl)=O N1(C(c2nc(C)ccc2OC)C(=O)NCCC)CCSC2CCCCC12 CCCC(C)(CCC)C(=O)NC1C2CC3C1C3C2C(=O)NCC(C)(COC)CC C(c1ccc2c(c1)COCC2)=CC(=O)NCC1CC(NC(CN(C(C)C)C)=O)C1 N1(C(C2N(C(c3cc(C)c(C)nn3)=O)CC(O)C2)=O)CC2(CCC1CO)CC2 C(=O)(C1=CCCCCC1)NC(CN(C(C(C(=C)C)(C)C)=O)C)C N1(C(CC2OCCC(C)(C)C2)=O)Cc2ccccc2C(NC(=O)CC2CCC2)C1 c1(CC(=O)NCC(CC)NC(=O)CC(C)(C)COC(C)=O)ccc2[nH]ccc2c1 N1(C(c2c(C=C)cnn2C)=O)CC=C(C(C)(C)C(=O)NCC)C1 c1(OC)cc(CNC(Cn2cncn2)C(=O)O)cc(C#N)c1 CC(C)CC(O)C(=O)N1CCOCC1CNC(=O)CCN1CCCCCC1 c1(C(=O)NCCC2CC(OC)CN2C(C2CCOC2)=O)c(F)cc(Cl)cc1F C1(CNC(c2c(C)nsc2)=O)CC2(CCOCC2)CN1C(=O)C1=CCCC1C c1(C(N2CCC(C(C)NC(=O)Cn3cc(Cl)cn3)C2)=O)ccc2nc(O)oc2c1 C1(CNC(c2scnc2C(F)(F)F)=O)COCCN1C(=O)CC1(O)CCC1 C1(NC(C(C)SC)=O)CC2(C1)CC2NC(=O)CCc1cccc(Cl)c1 S(=O)(=O)(c1ccc(NC2CC(O)C2)cc1Br)N1C(COC)CC(F)C1 c1(CC)ccc(C(N2CCCC(c3cn(C)nn3)C2)C(=O)NCC2CC2)cc1 N12CCOCC1C2=O.C1(NC(CC2CC(NS(C)(=O)=O)C2)=O)CCCCO1 Cc1cc(Cl)c(Cl)cc1C(N1CCSC(NC(=O)Nc2c(C)cccc2C)C1)=O Cc1ccc(S(=O)(=O)C2(C(=O)NC3CCNS3(=O)=O)CCCC2)cc1 C1(COC)CN(C(C2CC2c2cnc[nH]2)=O)CCN1C(C1(F)CCCC1)=O c1(C(N(C(C)C)CC2CCC2)=O)c[nH]nc1CNC(=O)CC1OCCC1C C1(NC(C2C(CC)CCCN2)=O)CCC2(CCNCC2)C1 c1(CC)noc(C(N2CCOCC2CN(C)C(C2(COC)CCCC2)=O)=O)c1C Cc1cc(C)c(C(=O)NCc2nnn(C)c2C(=O)NCc2cncn2C)s1 CCCCCC(CC)C(=O)NCC(=O)NCC(=O)NC12CC1COC2(C)C C(=O)(C#CC1(C)CC1)NC1(CN(C)C(C2(C)CC2c2ccccc2)=O)CC1 CCC(CN(C)C)CC(=O)NCC(C)CNC(c1nc(OC)ccc1C)=O C(CC(C)C(=O)NC(C)CCN(C)C(c1cn(C2CCC2)nn1)=O)=CCC CC(C)CC(C(=O)NCC1(O)CCCN(C(=O)Cc2ccco2)C1)C(N)=O C(=O)(C(C)CS(C)(=O)=O)N(C)CC1CCCN(C(c2cncc(C(C)C)c2)=O)C1 N1(C(c2cc(C(C)=O)c(O)cc2)=O)CCC(C2(NC(=O)CC3CC3(Cl)Cl)CC2)C1 N1(C(CCOCCOCC)=O)CCC2(CCN(C(c3ccc(C#N)[nH]3)=O)C2)C1 N1(c2nnc(CC)o2)C(CNC(=O)C=Cc2cocn2)CC2COCC12 c1(OCCC(=O)N(C2CC2)CC2CCNC2)ccccc1Cl c1(C(N2CCC(CC=C)(NC(c3cc(C)sc3C)=O)C2)=O)cccc(F)c1F c1(CC)noc(C)c1C(=O)NCC1(F)CC(CNC(C2CC2(C)Br)=O)C1 N1(C(C2CC(C)(C)CN(C(=O)CC3CCC(=O)N3)C2)=O)CCc2ncncc2C1 Cc1nc2ccccc2n1CC(=O)NC1CN(C(C2CCSC2)=O)CC1O C(C)(C(=O)N1CC(c2ncccn2)C1)(C1CCC1)NC(COCCN(C)C)=O c1(COC(C2OCCN(C(CC(C)C)=O)C2)=O)cc(F)cc2c1CCC2 c1(C(=O)NC(C)C(C)NC(=O)C=Cc2ccccc2)ncc(Cl)cc1Cl c1(OC)ncnc(OC)c1C(N1CC(CN(C)C(C2CCCCC2(C)C)=O)C1)=O CP(C)(=O)CC(=O)NCCOCCNC(C1CCN(c2nc(=N)[nH][nH]2)C1)=O CC1(C(=O)NC2CCCN(C3CCCCC3)C2=O)CC(c2ccccc2F)=NO1 c1(C(N(CCN(C(c2cc(C)on2)=O)C(C)C)C)=O)cc(F)cc(Cl)c1N c1(CC)cc(C(=O)NCC2CC2C(=O)NC2CC(CC)(CC)C2)on1 C=Cc1ccc(C(=O)NCCC2CC(C(N3CC(N(C)C4CC4)C3)=O)C2)cc1 c1(C(N(CC(CN(C(C2C(OC)CC2)=O)C)O)C)=O)cccc(C)c1[N+](=O)[O-] c1(NC(C2CC3CC3N2C(=O)C(c2ccccc2Cl)(F)F)=O)ccc(F)cc1O c1(CNc2c(NC)ccc(F)c2)cc(=O)n2c(n1)CCCC2 c1(CC(N2CCCC(c3cn(C4CC(O)C4)nn3)C2)=O)cnc2cccnn12 C#CCCCCCCC(=O)NCC1CCCN(C(C2(CC)CCCCO2)=O)C1 n1(CC(=O)NCCC2CCC(NC(=O)CN(C3CCCC3)C)C2)nnc(=O)[nH]1 c1(C(=O)NCCCCCCN(C(=O)CC2CCC(F)(F)C2)C)ccc([N+](=O)[O-])s1 CC1CC(NC(c2occ3c2CCC3)=O)CN(C(=O)Cc2cnns2)C1 O=C(Nn1nnc2c1CCCC2)C1CCN(CC(F)F)C1 C1(CC(=O)NCCNC(C2C=CCCC2)=O)COCCO1 C1(F)(CNC(C(C)O)=O)CCC(CNC(=O)Cn2cc(CO)nn2)C1 C1(C(=O)NCC2N(C(C3(C(C)(F)F)CCOCC3)=O)CCC2)CCCCN1N=O C1(C(N2C(COC)(CNC(c3ncc[nH]3)=O)CCC2)=O)CC2C(C1)C2(F)F C1(COC)CCC(NC(=O)CC2CCCN2C(=O)CC2CC(SC)C2)CC1 c1(CS(C)=O)cccc(NC(=O)NCC(c2ccc(F)cc2)F)c1 C1(NC(c2c(C)nc[nH]2)=O)CCCCC1C(=O)NCC1(O)CCOC1 O=C(NNc1cc(F)cc(F)c1)N1CC(F)CC1CO C1(C(N2CCC(C(N)=O)C2)=O)CC2CCCCC2N1Cc1ccccc1 c1(NC(c2ccc(C(F)(F)F)cc2)C)cccn2c(O)nnc12 C1(NC(c2cccc(CC)n2)=O)(CC)CCCN(C(C2CCC2)=O)C1 N1(C(c2n(C(C)C)nnc2)=O)CCC2CCN(C(c3nncs3)=O)C2C1 C1(C2CN(C(=O)C(C)(C)C3CCCC3)C2)(NC(C(n2c(C)ncc2)C)=O)CC1 CCCCC(=O)NC(C(C1CC(C2(C3CCCCO3)CC2)C1)F)=O C1(NC(c2ncc(C)cn2)=O)CCN(C(=O)COCC2CCC2)CC1CO C1(C(N(C)Cc2n(CC)ncc2)=O)COCCC1NC(C1(CO)CCOCC1)=O C12(CNC(C3CCC4(CC4)C3)=O)CC1CN(C(=O)C=CCO)C2 c1(C(c2nnc(-c3ccccc3)s2)SCCN(C)C)ccc(Cl)cc1 c1(C(=O)NCCN(C(C2CCC(C(C)C)NC2=O)=O)C)cn2cc(Cl)cnc2n1 C(=O)(C1CCc2c[nH]nc21)NC(CCC=C)C(=O)Nc1cc(Cl)ccc1C C1(CNC(=O)C(N2CCC(C3CC3)C2)=O)CCC2(CCCCCC2)O1 N1(C(c2c(C)[nH]nc2Cl)=O)CCCC(C)C1CNC(C1CC(=O)NC(=O)C1)=O Cc1cc2c(cc1C)C(C(=O)NCCCCC(C)NC(C1CCCSS1)=O)CO2 C1(C(=O)OC)CCC1(C)C(=O)N(CCCNC(=O)C(C)CC)C1CC1 C1(C(CC)C(=O)N(CCCN(C)C(c2ccnn2COC)=O)C)CCC(C)CC1 C(=O)(C(C)CN(C(=O)CC1CSC1)C)N(C1CCCOC1)CCC N1(C(C(C)(C)C(N)=O)=O)CCN(c2ncc([N+](=O)[O-])cn2)CC(O)C1 CCCN(C1CC1)N(C)Cc1cn2ccccc2n1 CC(C)C(F)(CNC(=O)CC1OCCCO1)C(=O)NC(C)Cc1cccs1 N1(CCC)CC2CCN(C(=O)C(C)CCC(C)(C)C)CCC2C1 c1(C(N2CCC(CC)CC2C(N2CCC=C(Cl)C2)=O)=O)cccc2ccccc12 c1(-c2cc(C(N(C3CN(C(C(CSCC)O)=O)C3)C)=O)no2)ccc(OC)cc1 N1(C(C=C=C(C)C)=O)CCCC(C)C1CNC(c1cn(C)ccc1=O)=O N1(C(c2cccc(C(C)C)n2)=O)CCCC12CCN(C(c1cncs1)=O)CC2 N1(C(C(C(C)(C)C)NC(C)=O)=O)CC2CC(C1)N(C(=O)CCC1OCCO1)C2 Cc1cc(N2CCN(C(C)(C)C)CC2COCc2ccccc2)cnc1O N1(C(c2c(SCC)cccc2)=O)CCCOC(CNC(C2C3CCC(=O)C23)=O)C1 N1(C(C(C)CC(F)F)=O)CC2COCCC2(NC(c2ccc(Cl)cc2Cl)=O)C1 C(c1ccsc1)=CC(=O)NCC(CC)NC(C1(N2CCNC2=O)CC1)=O C1(OCC)COCCC1CC(=O)NCC(C)N(C)C(c1ccoc1Br)=O c1(C(N2CCN(C(C(=O)NC(C)C)=O)C(C)C2C)=O)nnc(O)c2ccccc12 c1(NC(C2CC(F)CN2C(c2c(F)ccnc2Cl)=O)=O)ncc([N+](=O)[O-])cc1Br C(CN=c1[nH]cnc2c1COC2)C1CC(NC(C2C(C)c3c[nH]nc3CC2)=O)C1 C1(NC(C(C)OC)=O)CCC2(CCN(C(=O)C3Cc4ccccc43)C2)C1 C1(CNC(C2N(CC)CCCC2)=O)CCCC12CCN(C(=O)C(OC)OC)CC2 c1(NC(c2n(C(CC)C)nnn2)c2scnc2Cl)cccc(OCCCC#N)c1 CC1(C)CC(C#N)(CNC(=O)CCNC(C23CCCCC2C3)=O)C1 c1(C(=O)NCC(CC)NC(C2OCCO2)=O)ccnc(C(C)(F)F)c1 c1(C(=O)NCC(=C)CCNC(=O)C2=CCCOC2)oc2ccccc2c1OC N1(C(C(C#C)(C)C)=O)CCCC(C(=O)NCC2(CO)CC3CC3C2)CC1 N1(C(C(CN(C)C)(C)C)=O)CC2(NC(=O)C(C3CCCCCC3)O)CCC1CC2 C(=O)(C(C)(C)CS(C)(=O)=O)NCC(C)N(C(=O)Cc1cc(F)cc(F)c1)C O=C(C1=CCCC1)NCCN(C(=O)Cc1cccc(O)c1)C1CC1 c1(C(N2C(CNC(c3c(SC)ccs3)=O)CC(C)(C)C2)=O)cc2ccncc2[nH]1 Cc1cc(Br)cnc1C(=O)N(C)C1CC1C1CCN(C(C23CC(C(=O)O)C2C3)=O)C1 C(C)(C(=O)N1CCCC(NC(=O)CCn2ccnc2)C1)(C(C)C)OC CC(C)(C)C1=NOC(C(=O)NCC(c2ccccc2F)NC(=O)C(C)(C)F)C1 Cc1cccn(CC(=O)N(C)CC2(O)CCN(C(C3CCCC(=O)N3)=O)C2)c1=O N1(C(CC(CC)O)=O)CCn2ncc(C(=O)NCc3cccc(C)c3O)c2C1 N1(CC2(CN=c3c(C(=O)OC)cc(Cl)n[nH]3)CC2)CCC(C2CCCC2(C)C)C1 CC(C)C(C(=O)OCS(=O)(=O)C1CC1)NC1(C)CS(=O)(=O)C1 N1(C(C(=O)NCCNC(C)=O)=O)CCOCC(C(=O)NCC2CCC(F)(F)C2)C1 C(CCCCC(=O)NC1CCN(C(c2cnc(OC)c(Cl)c2)=O)CC1C)OCC C(=O)(C1=CC2(CCOC2)C1)N1C(C)CC(NC(=O)CC2CC(=O)C2)CC1 C1(C)(CC)C=C(C(=O)NC(C(=O)N(C)CC)C2CCC2)C1 CC1(C#CC(=O)NCC23CC2CN(C(=O)C(c2cc(Cl)cc(Cl)c2)=O)C3)CC1 C1(NC(C(C2CN(C(C(C3CCCC3)OC)=O)C2)OC)=O)CCCCC1 C1(CC(=O)NCC2(F)CN(C(=O)COCCc3ccccc3)C2)CC=CCC1 C(=O)(CC(CC)C(C)C)NCC(CCCC)NC(c1ccsc1Br)=O N1(C(COC2(C)CCC2)=O)CC2(CC(C(=O)N(CC3CC3)CC3CC3)CO2)C1 N1(C(CCC=C)=O)CCCC(C)C1CCNC(=O)CC(C)(C)c1ccc(F)cc1 c1(OC)ccc(C(O)C(=O)NCC(C2CCC2)NC(c2n[nH]c(C)c2C)=O)cc1 C1(C(=O)NC2C=CC(CC(=O)NCCOCCC)C2)CC2OC1C1CC21 N1(C(c2c(CC)nccn2)=O)CC2CC1CN2C(=O)Cc1cccc(C(N)=O)c1 C1(C)(C(N2CCCC(CN(C(C(C(=O)NC)(C)C)=O)C)C2)=O)CCC(C)C1(C)C N1(C(C2C(C=C)CC2)=O)CCN(C(c2ccc(CNC(N)=O)cc2)=O)C2(CC2)C1 Cc1ccc(S(=O)(=O)NCC2CC(OC(C)(C)C)C2)c(C#N)c1 C1(C(N(CCN(C(c2cc(OC)no2)=O)CC)CC)=O)CCS(=O)(=O)C(C)C1 N1(CCC)CCCC(C(=O)NC(C)(C)CNC(C2CCCCN2CCC)=O)C1 Cc1ccc(NC(c2nc(C(c3cccnc3)C)n(-c3ncnn3C)n2)=O)cc1 Cc1cccnc1-n1cc(-c2ncccc2C)nn1 C1(NC)CCN(CCNC(c2cn(Cc3csnc3N(C)C)nn2)=O)CC1 N1(C(CC(C)(C)O)=O)CCC2(CCC2)C(NC(C2CCC(=O)NC2)=O)C1 N1(C(C2(C#C)CCN(C(=O)C(CC)SC)C2)=O)CC2CCC(C1)C(=O)N2 c1(C(=O)NCCC(CNC(C(CC)F)=O)O)cc(OC(F)F)ccc1F c1(COC)cccc(C(c2nnnn2CC2CC2)NCc2c(C)cnn2C)c1 c1(C(=O)NC2CN(C(c3c(CC)n(C)nc3)=O)C2)cc(OC)c2c(c1)CC(C)O2 c1(OCC)cccnc1C(=O)NCC1C2CN(C(=O)CC3CCC(F)(F)C3)CC12 C1(C(C(=O)NCC(CC)CO)(C)C)CCCN(C(c2cscc2C)=O)C1 N1(C(C(=O)NCC2C3CN(C(c4cc(C)sn4)=O)CC32)C)CCc2ccccc21 C1(C(=O)NCC(COC)(C)CO)CCOCCN1C(=O)Cn1ncnn1 c1(CC(N2C(CN(C(=O)CC3(N(C)C)CC3)CC)CCC2)=O)ccccc1O C(c1ccncc1)=CC(=O)NC12CC(CNC(C(C)OCC(F)(F)F)=O)(C1)C2 CCCC(C)(O)CC(=O)NC(CC(=O)NCCc1cnc(C)cn1)C1CC1 c1(C(=O)NCC2N(C(C(CC=C)C)=O)CCCC2)c[nH]c2cccc(F)c12 C1(C)(CNC(c2c(CC)con2)=O)CCCN(C(c2nn(C)cc2C(C)=O)=O)C1 C1(NC(CC2CCC(=O)NC2)=O)CCS(=O)(=O)C12CN(C(=O)CCC[N+](=O)[O-])C2 c1(N2CC(C)OCC2)nc(N2CCC3(CCCC3)CC2)nc2c1CSC2 c1(C(C2CCCC2)OC(c2nc(COC)oc2)=O)ccc(Br)cc1 C12(CNC(CC=C=C)=O)COCCN1C(=O)CN(C(c1cccc(Cl)c1F)=O)C2 N1(C(C2(C)CC=CCC2)=O)CCCC(C(=O)N(C2CC2)C2CC2)CC1 C(=O)(CC(C)(C)F)NCC1C(NC(c2cc(OC)ns2)=O)CCC1 C1(NC(c2csc(Br)c2)=O)CCN(Cc2cc(Br)c[nH]2)CC1F C(=O)(C1CCCc2nc(C)[nH]c21)N1CCN(C(c2nccc(C)c2)=O)CC12CC2 O=C(CCC1=CCCCC1)NCCNC(c1ccsc1)=O C1(C(=O)NC(C2CN(C(c3cnc(SC)s3)=O)C2)C)COC2COCC12 c1(OC)cc(F)cc2[nH]c(NC(N3CC4CN(C5CCC5)CC4C3)=O)cc12 c1(CC(=O)N(CC(CN(C(Cc2nnc(C)o2)=O)C)O)C)ccc(C)c(C)c1 C1(C(N2CC(F)(CNC(Cc3c(C)nc(S)s3)=O)C2)=O)CC2CSCC(C1)C2 c1(CC(=O)NCC)ccc(-c2ccnc(CC(N3CC4CC4C3)=O)c2)cc1 N1(C(c2c(COC)n(C)nc2)=O)CC2(C)CN(C(c3ccoc3Cl)=O)CC2(C)C1 N1(C(=O)OC(C)(C)C)CCC(N=c2[nH]c(C(F)(F)F)nc3c2CCC3)C(F)C1 c1(OC)ccc(CC(N2CC(F)(CNC(c3cn(C(C)C)nc3C)=O)C2)=O)cc1 C(C(C)C(=O)NC1COCC1NC(c1c[nH]nc1C(C)C)=O)OC(C)=O c1(OC)ccc(C(=O)NCC2CN(C(=O)C=CSC)CC2C(F)(F)F)c(C)c1 C12(CNC(C3C(OC)(OC)CC3)=O)CC1CN(C(=O)CCN1CCOCC1)C2 N1(C(CC)=O)CC(NC(c2csc(Br)c2)=O)CC12CCCCCC2 N1(C(C(C2CC(F)(F)C2)OCC)=O)CCN(C(=O)C#CC(C)(C)C)CC1C N1(C(c2nc(C)c(C)[nH]2)C)CCC(O)(Cc2cn(C3COCC3O)nn2)CC1 CC1CCCN(C(=O)C=Cc2cnn(C)c2)C1CNC(=O)CCCC#N C(=O)(C(O)CCC(C)C)NCC(COC)NC(=O)CCCN1CCOC1=O C(C(C)(C(=O)NCC1C(C)CCN1C(c1ccn(CCO)c1C)=O)OC)OC c1(N2CCC(C=C)CC2)[nH]c(=NCc2c[nH]nc2C2CC2)nc2scnc12 n1(C(=O)NCC(C)(CC2CCC2)OC)ccc2c(C)cccc12 c1(NC(N(CC(O)C2CC2)C)=O)ccc(N2CCOCC2)nc1C C(=O)(CCCCCCCC1CC1)N(CCCN(C)Cn1cc(CN)nn1)C1CC1 C1(C2CCN(C(=O)Cn3ccnn3)C2)(NC(C(C)C(C)(F)F)=O)CC1 C1(C(N2CCC(NC(c3c(C)[nH]nc3C(C)C)=O)CC2)=O)CCCC1S(C)(=O)=O c1(CC)nn(C)c(CC)c1C(=O)N(C)CC1CCCN1C(=O)CSC(C)C C1(NC(C(C2CC2)SC)=O)COCCN(C(C2(C)CCN(C(C)=O)CC2)=O)C1 C1(C(=O)NCc2c(COC)noc2)CN(C(=O)CC(C)(F)F)CC12CC2 C(=O)(C(C)CC(F)F)NCC(CCC)NC(C1(C)CC2(CC2)C1)=O c1(N2CC(C)(NC(CCC(C)SC)=O)C2)ccnc2ncnn12 CCCCCCCC(=O)NC1CC(N(C)C(C2CC(F)(F)C2(F)F)=O)C1 CCC(CC(=O)NC1(C)CCN(C(=O)CCn2ccnc2C)C1)C(C)(C)C N1(C(c2cccc(OCC)c2)=O)CC2CCN(C(c3ccc(O)nc3)=O)CC2C1 c1(C(=O)NCC2CCN(C(c3ccc(C(N)=O)s3)=O)C2)ccc(O)c(CO)c1 Cc1ccc(OCC(N2CCN(C(=O)CC3(C)CC3)C3CC23)=O)c(Br)c1 C1(CC)C(N)CCCN1Cc1ccc(N2CCCC2)o1 CC1CN(C(C2(N(C)C)CCC2)=O)CC1CNC(c1c(C(F)(F)F)cnn1C)=O Cc1n[nH]c(C)c1CC(N1CC(C(C)NC(=O)CCCc2cccnc2)C1)=O c1(SCCNC(=O)OCC(C)(C)C)ccc(OC(F)(F)F)cc1.ON c1(C(N2CC3C(CNC(C4CCC(CC)CC4)=O)(C3)C2)=O)nccc(Cl)c1O C(=O)(CS(=O)(=O)C(C)(C)C)NC(C)CC(C)NC(C1(c2ccccc2)CCC1)=O C1(CC(N2C(C)CC(CNC(C3(C)C(C)CCC3)=O)C2)=O)CN2CCC1CC2 Cc1c(C2OCCC2NC(=O)NCC2CCNC2=O)cnn1C CCC(CN(C)C)CC(=O)N(C(C)CCC=C(C)C)C.c1c(=O)n1 CCCC(C(F)(F)F)NC(=O)CC1CCCN(C(=O)COC2(C)CCC2)C1 Cc1n[nH]c(C)c1C(C)CC(=O)NCC(F)CNC(=O)COCC1(F)CC1 Cc1ccc(C(=O)N(C2CN(C(=O)CCCC(C)(F)F)C2)C)c(N)c1C C12(NC(C(CCC#C)O)=O)CC3CC(C1)CC(CNC(c1ccnn1C)=O)(C3)C2 Cc1ccc(C(N2CCN(C)CC2C(=O)NCCC(=O)NC2CC2)=O)c(F)c1F C(=O)(C(C)C(C)(F)F)NCC(C)NC(c1ccc(-c2cn[nH]c2)cc1)=O N1(C(C=C(C)Cl)=O)CC2CCC(C1)N(C(c1cncc(F)c1C(F)(F)F)=O)C2 C#CCCCCCCC(=O)NC1(C(N2CCOC(C)CC2)=O)CCOCC1 C1(NC(COC2CCCC(C)C2)=O)CN(C(=O)CS(N)(=O)=O)C(C)(C)C1 C12CCCN(C1)C(=O)NCCCC2.N1(C(C2CCC2)=O)CCC1CO.C1CC1 CC1(C)CC(CNC(=O)CC2(CNC(=O)Cc3cccn3C)CC2)CO1 c1(C(N2CC(COC)N(C(=O)CCCCCF)CC2)=O)ncnc2c(C)csc12 CC12CC(C(N3CCN(C(C4CC5CCC(C4)S5)=O)CC3)=O)(C1)C1(CCC1)O2 c1(C(=O)NCC2(C)CCCN(C(C(C)OCCCC)=O)C2)cn2c(n1)CCCC2 N1(C(C(COC)(C)O)=O)CC2CC(NC(c3ccc(OC)nc3Cl)=O)CC2C1 N1(C(c2cncc(CC)c2)C(=O)NCC(F)F)CCOC(CC)C12CCC2 c1(C(C)C(=O)NCCOCCNC(C2CC2C(F)F)=O)ccc(Br)s1 c1(C(N2C(C)CC(CNC(c3ncc(C)nc3)=O)C2)=O)cc(N)cc(N)c1 C=CCC(CNC(=O)CCNc1ccccc1)NC(=O)C=C(Cl)Cl c1(CNC(C(C)OC(C)=O)=O)ccc(C(N2CCC2(C)C(C)C)=O)s1 c1(OCC(=O)NC(CC(=O)OC)C)cnc(SC)nc1O N1(C(C2=NOC(CNC(C(COCC)N=[N+]=[N-])=O)C2)=O)CCn2cc(C)nc2C1 C1(C)(CC)C=C(C(=O)NC2COCC2NC(c2ccc(F)cc2)=O)C1 C1(C(=O)NCC(CC=C)NC(=O)C=C2CCCC2)CCN(c2nncs2)CC1 C(CCC(C)C(=O)NC1CCCC(NC(=O)CCCNS(C)(=O)=O)C1)OC CCC(CNC(=O)CCCn1cc(-c2ccc(C)cc2C)nn1)CC(F)F C1(C(N2CC(NC(C(C3CCC3)OC)=O)C(SC)C2)=O)CS(=O)(=O)CC(=O)N1 S(=O)(=O)(c1ccc(NC(C2CCC(C)CC2)=O)nc1)N(C(C)CSC)CC Cc1cc(C(=O)NCC2CC3CC3N2C(=O)CC2(NC(C)C)CC2)n(C)n1 C1(C(=O)NCc2ccn(C)n2)(CNC(=O)C(C2CCCCC2)F)CC2(CC2)C1 Cc1cc(C(=O)NC2CS(=O)(=O)CC2NC(c2sccc2C(F)F)=O)cc(O)n1 C1(OC(CCNC(CC(=O)OCC)=O)COC)CC(C)(C)C(C)(C)C1 Cc1cc(NC(C23CC2CN(Cc2[nH]c(C)nc2C)C3)=O)cc(Br)c1 c1(C(=O)NCC2CC(C)N(C(=O)CCC3CC3)C2)csc(N=S(C)(C)=O)n1 c1(C(C2(NC(=O)NC3(C(C)C)C(CC)C3)CC2)OC)ccc(C#N)cc1 CP(C)(=O)c1cnc(C(=O)Nc2cc(Br)cc3c2OCO3)nc1 C1C(C)N=C2C=CC=C(S(=O)(=O)N1)N2.c1(C(CN(C(C)C)C)(C)C)ccccc1 N1(C(CCC)=O)CC2(CC(C(=O)NC(C)CCC(F)(F)F)CO2)C1 N1(C(c2c(OC)cc(C)cc2)=O)CC2CCCC(CNC(=O)C(C)OC)(C2)C1 N1(C(C(=O)NCc2ccc(OC)cc2)C(C)C2CCCCC2)Cc2ncsc2C1 C1(NC(C2(C)CS(=O)(=O)C2)=O)CCC2(CCCN(C(c3cc(Cl)c[nH]3)=O)C2)C1 C#Cc1cncc(NC(=O)C(CCF)NC(=O)Cc2cn(C)cn2)c1 c1(C(N2CC(C(C)NC(=O)Cn3cnnn3)C2)=O)cccn2c(O)nnc12 CC(C)C(F)C(=O)NCC(C1CCN(C(c2cnn(C(C)(C)C)c2)=O)CC1)(C)C c1(C(=O)NC(C(C)NC(c2cnc(CC)[nH]2)=O)C(C)C)ncc(C)cc1C C1(NC(c2ocnc2C(F)F)=O)CCN(C(C2CCCC23CC3)=O)CCC1CO C(=O)(CC(O)CC(C)(C)C)N(CC(=O)NC(c1cc(C)on1)C)CCOC C1(CNC(=O)NC2(C(F)(F)F)CC(O)C2)CCC2CC2C1 C1(CNC(c2scc(OC)c2)=O)CCCCN(C(=O)Cc2cc(C)cc(F)c2)C1 c1(CNC(C2(F)CN(C(CC(CC)SC)=O)C2)=O)ccc(C(C)C)cc1F c1(C(N2C(CNC(c3c(C)ccs3)=O)CC(F)C2)=O)cc2c(Cl)cncc2s1 C1(CNC(=O)CCc2ccncn2)COCCN1C(=O)Cc1cnccn1 C(=O)(C1Cc2ccccc21)N(CCC(=O)NC1C(C#C)CCC1)C1CC1 C(=O)(CCC(F)(F)F)NCCC1(C)CCN(C(c2c(C(C)C)ncnc2)=O)C1 C1(NC(CC(C)(C)C2CC2)=O)COC2CN(C(c3cnc(=N)[nH]c3)=O)CC12 N1(C(Cc2ccc(C)o2)=O)CCC(C)N(C(c2n[nH]c3c2COCC3)=O)CC1 c1(C(=O)NCC2(NC(C(C3CCC3)OC)=O)CCC2)ccc(Cl)cc1 Cc1nc2ncc(C(=O)NC3CC3CNC(=O)C(C)Cc3ccccn3)cc2o1 c1(C(N2CCC(NC(C3C=C(C)CS3)=O)CC(F)C2)=O)ccc2[nH]nc(Cl)c2c1 N(C(=NCCC1COC(C)(C)OC1)NCC1CC1)CC1C(C(=C)C)CNC1 C12(C(=O)NCC(CCNC(=O)C3CC3)O)CCC(CO)(CC1)CC2 c1(NC(N2CCC2C2CCOC2)=O)ccc(F)c(F)c1 C1(C(C(=O)NC2(C(C)NC(c3occc3C3CC3)=O)CCC2)C)CCOCC1 c1(N2C(CNC(=O)Cc3ccco3)CC3(CC3)C2)ncc2ccccc2n1 N1(C(c2c(C)n[nH]c2C)=O)CCCC(C(=O)NCc2cccc(Cl)c2)CC1 C1(CNC(C2C(OCC)C2C)=O)CCCN1C(C1CCCN1c1ccccc1)=O c1(C(=O)NCC(=C2CN(C(CC3(OC)CC3)=O)C2)F)sc(C)nc1C C1(C(=O)OC)(OC(C(=O)NCCF)C2CC(NC(=O)OC(C)(C)C)C2)CCOCC1 CN=c1[nH]nc(CC(=O)NC2CC2NC(c2ccc(SC)cc2)=O)s1 C1(O)(CNC(C2(CCS(N)(=O)=O)CCC2)=O)CCCN(C(=O)C2=NOCC2)CC1 C(=O)(C(F)CC(C)C)NCC1CCCC(NC(c2scc(C(=O)OCC)c2)=O)C1 N1(C(c2cc(C(F)F)no2)=O)CCC2OCCN(C(=O)CC3COCCO3)C2C1 N1(C(c2[nH]cc(C#N)c2)=O)CC2CCC2(NC(=O)CSc2ccncc2)C1 c1(C(=O)NC2(C3CN(C(C4C(C(C)C)C4)=O)C3)CC2)ncccc1N=[N+]=[N-] C1(C(=O)NCC(C#C)OC)CN(C(=O)C(O)CSC)CC1C=CC CC1CCN(C(C2CCCN(C(c3cc(=O)cc[nH]3)=O)CC2)=O)CC1(F)F c1(C(N2CCC(C)(CNC(c3cc(F)c[nH]3)=O)C2)=O)ccc(O)c2c1CCCC2 c1(C(N(C2CCCN(C(CC)=O)C2)C)=O)cccn2c(O)nnc12 N1(CC)CC(C(N2CC(CNC(=O)CCc3ccc(C)o3)C(O)C2)=O)CCC1=O C1(C(N2CCCC2(C)CO)=O)(NC(CC(=O)OCC)=O)CC(F)(F)C1 Cc1nc(CS(C)(=O)=O)sc1CN1CC(C(=O)N(C)C)C1 c1(C(N2CCC(NC(c3cc(Cl)cnn3)=O)C(O)C2)=O)ccn2ccccc12 c1(C(N(C2CCN(C(c3cc(CCC)n(C)n3)=O)C2)C)=O)[nH]cc2c1CCCC2 c1(CC)cc2c(NCC3CCCC3NC(C3(O)CC(C)(C)C3)=O)nc(C)nc2s1 Cc1ccc(F)cc1C(=O)NC(c1nocc1C(=O)NC1CCCCCCC1)C CCCCCCCCCn1cc(CN2CCCC(F)(F)CC2)nn1 N1(C(C(=O)NC(C)C)=O)CCC(NC(=O)CC2CCOC2)C1(C)C S(=O)(=O)(c1cc(C(=O)NC2CC(CCNC(C3(C)CCC3)=O)C2)c(C)o1)NC C1(NC(Cc2ccc(OC)c(O)c2)=O)CCOC2(CCS(=O)(=O)CC2)C1 Cc1nc(O)nc(S)c1CN1CCCC1Cn1ccnc1 C1(C(=O)NCCCCC2N(C(C3CCC(C)C3)=O)CCC2)CC2C=CC1C21CC1 n1(CC(=O)N(CC(CNC(C(CC)(F)F)=O)C)C)ncc(C)cc1=O C(=O)(C1=C(Cl)CCC1)NCCN(C(c1nc(C#C)sc1)=O)C1CC1 CCCCC(C)C(=O)NCC(CNC(c1ccc(Br)cc1Cl)=O)CO C12(C(=O)NCC(CNC(C(C(C)C)n3cccc3)=O)C)CC(C)(C1)OC21CCC1 CC1(C)COCC1CNC(=O)NC1CC1c1ccc(C(F)(F)F)cc1 c1(N(C(=O)NC(C2CCSCC2)C(=O)OC)Cc2cnn(C)c2)cc(O)ccc1F C1(N(C)C)CC(C(=O)NC(C2CCOC2)CNC(=O)C(=O)NCC(F)F)C1 Cc1cc(F)ccc1S(=O)(=O)N(CC(C)C)C(=O)CC1OCCCO1 c1(C(=O)NCC(C)NC(C=C(C)c2ccsc2)=O)cc2c(ccn2C)[nH]1 N1(C(CSCC=C)=O)CC2CC2(CNC(C2CC(C(F)F)C2)=O)C1 N1(C(CC#C)=O)CC2CCC2(CNC(c2ccsc2Cl)=O)C1 C(=O)(C(CO)C(F)(F)F)N(C)CC1CCN(C(c2cncnc2C2CC2)=O)C1 C1(CC(=O)NCC2(CNC(CCc3ccn(C)n3)=O)CCC2)CCOC(C)(C)C1 C1(N(C(C2C(C)C2)=O)C)CCN(C(=O)COCc2nc(C3CC3)no2)C1 c1(C(C(=O)NCC2CN(C(C=NOC)=O)C2)O)cccc(Cl)c1 CCCCC(C)(F)C(=O)N1CC(CCNC(C2CC23CCCC3)=O)(OC)C1 Nc1cc2c(cc1C(=O)NCCCCCNC(=O)CCc1cncnc1)OCO2 N1(C(C2(CC)CCN(C(c3c[nH]nc3C)=O)C2)=O)CCOC2COCC12 C(=O)(C(C)(C)C(=O)N1CCC(CC(=O)NCC2CC3(CC3)C2)C1)OCC c1(C(N(C2CCS(=O)CC2)CC)=O)cccc(-c2ccccc2CN(C)C)c1 N1(C(=O)NC(c2scc(C(=O)OC)n2)C)CCOC(c2cccc(O)c2)C1 N1(C(C(C)(C)OCC)=O)CCCC(CCC(=O)NCC(C)CC2CCC2)C1 C1(NC(C(Cc2cnc[nH]2)NC(CP(C)(C)=O)=O)=O)CCn2ncnc2C1 C(CNC(=O)Cc1cnc(C)s1)(C(C)C(C)C)NC(c1ccn(CCCC)n1)=O Cc1nc(CC(=O)N(CCC(C)NC(C2CCCO2)=O)C)c(Cl)s1 c1(CN(C)C(C2(C(C)(F)F)CCC2)=O)ccnc(C(=O)NC2(CCF)CC2)c1 c1(C(=O)NC(CC)CNC(=O)C(c2c(C)n[nH]c2C)C)cc2ccnc(Cl)c2[nH]1 c1(CC(N2CC(C(C)NC(=O)CC3CCC4CC34)C2)=O)c[nH]c2ncccc12 C1(C(=O)NCCC2(O)CCN(C(c3cccnc3O)=O)C2)CN2CCCN1CC2 S(=O)(=O)(c1c(OC)noc1CC)NCC1(F)CC(C(=O)OCC)C1 CC1CCN(C(c2ccon2)=O)CC1NC(=O)Cn1cc(Br)ccc1=O CCCCCCC(=O)NC(C)(C)CC=CC(N1CC(C(N)=O)C(C)C1)=O N1(C(CSCCC)=O)CC2(CCN(C(c3cnccc3N3CCOCC3)=O)C2)C1 c1(C(C(C)NC(C(=O)Nc2ccc(OC)cc2OC)=O)O)ccc2c(c1)OCO2 C(C(C(=O)NCC(C)NC(=O)CN(C)Cc1ccccc1)OC(C)(C)C)SC C1(CNC(C(C)SCC)=O)CC2(CO1)CN(C(c1c(Cl)nn(C)c1C)=O)C2 C(=O)(CC1=CCCC1)NC1CCC(NC(C(CC)(O)c2cccc(Cl)c2)=O)CC1 C(=O)(C#CC1(C)COC1)N1CCCC(C)(C(N2CC(C(CC)C)C2)=O)C1 C1(C(C)C)Cc2cc(F)ccc2N(C(c2cc(Cl)ccc2C(F)F)=O)C1 c1(C(N(c2nc(OC)c(C)cn2)C2CNCCC2(F)F)=O)cc(F)cc(F)c1OC N1(C(CCOC)=O)CC(CNC(c2cncnc2)=O)(OC)C1 c1(C(=O)NC(C2(C(=O)NC3CC(N4CCC4)C3)CC2)C)cccnc1 C(c1sc(Cl)nc1Cl)=CC(=O)NCC1C2CN(C(CNC(=O)NC)=O)CC21 c1(C(N(CCCCN(C(=O)C(F)CC2CC2)C)C)=O)cnc(O)cc1C(F)(F)F c1(OCCOC)cc(O)ccc1NC(=O)Cc1ncccc1O C(=O)(C1=Cc2ccccc2C1)NC1CC(C(=O)NC2CN(c3ccncc3)C2)C1 C(CCCC(=O)NC(C12CCC(CO1)C2)C)N(C(c1cc(C(C)=O)[nH]n1)=O)C Cc1c(C(=O)NCC(O)CN(C)C(C2CCCN2C)=O)cnn1CC(C)C.CC C1(CNC(c2c(-c3cn(CC)nc3)n[nH]c2)=O)COCCN1C(c1cn[nH]c1)=O C12(NC(C3C(C)C3C)=O)CCC1CN(C(=O)CCc1cc(Br)ccc1F)C2 CC1CN(C(=O)CC2CN(Cc3cccc(-n4cncn4)c3)CCO2)CC(=O)N1 C(=O)(C(CC=C(Cl)Cl)c1ccccc1)N1CCCC(C)(CN)C1 C(C)(CC(=O)N1CCC(CC(=O)NC(c2ncc(C(C)(C)C)o2)C)C1)OC C1(C(N2C(CN(C(c3c(C)occ3)=O)C3CC3)CCC2)=O)CCC12CCC2 C(CCCC(=O)NC1CC(F)(CNC(c2cnccc2Br)=O)C1)SC C12(CNC(Cc3cc(COC)on3)=O)CC1CN(C(=O)CCNC(C)=O)C2 c1(NC(C2N(c3cc(SC)ncn3)C3C(C2)C3)=O)cc(F)c(O)cc1Cl n1(CC(=C)C)nnnc1C1(CCOC)C(c2noc(C3CC3)n2)N1.CC.OC CCCC(CNC(=O)C(CC)CCOC)C(=O)N1CCC(NC(N)=O)CC1 C(=O)(CCn1cccn1)NC1C(NC(N(C(C)(C)C)CCN)=O)C1 c1(NC(c2cncc(NCc3nc(C)c(Br)cc3)c2)=O)cccnc1[N+](=O)[O-] C1(NC(Cc2c(CC)cc(F)cc2)=O)CN(C(=O)CC2CC2)C2(CCC2)C1 N1(C(C(C2(C)CC2)NC(=O)COC2CCC2)=O)CC2CC2(CO)C1 Cc1nn(C)cc1NC(c1cn(CC(F)(F)F)nn1)C(=O)NC1(C2(C)CC2)CC1 c1(CC)ncncc1C(=O)NCC12CC1CN(C(=O)C(=Cc1cccnc1)C)C2 C(=O)(CCCC(N)=O)NC1(C)CCN(C(Cc2c(C)cco2)=O)C1 C(=O)(C(C(=O)NCC1CCC1)OC)OCC.C1(=O)C(Cc2ccc(C)cc2)CN1 C#CC12CCC(C(=O)NCC3CCN(C(=O)C(C)C4CCC4)C3(C)C)(CC1)CC2 CCCC(CC)CC(=O)NC1(CN(C(=O)COc2ccc(F)cn2)C)CC1 c1(C(=O)NC2CC(CNC(CC(=C)C)=O)C2(C)C)ccc2cc(O)ccc2n1 N1(C(c2c(C)cno2)=O)CCC(F)C(NC(C2(C)CCCOC2)=O)C1 C1(CC=C)(NC(=O)C=Cc2cc[nH]n2)CCCN(C(C2CCC3CC2CO3)=O)C1 N1(C(c2nnc(-c3ccccc3F)s2)C)CCCC2CN(CC3CCCO3)CC12 C=CC1CN(C(=O)C(c2cncn2C)O)CC1NC(=O)CN1CCCCC1=O N1(C(c2c(C)nc(C)o2)=O)CCCC(C)(CNC(=O)C(c2ccccc2)F)C1 C1(N(C(=O)CN2CC3CC3C2)C)CN(C(c2cc(C(F)F)nn2C)=O)CC1F CCCCC(O)C(=O)N1CC(NC(c2cncc(C(C)(F)F)c2)=O)CC1(C)C c1(OC(C)C)ccccc1CC(=O)N(C)CCN(C)C(C1C(C)(C)C1(C)C)=O CCC(C)C(C(=O)N1CC(OC(F)F)C1)NC(=O)Cc1cnsc1 c12ncccc1NC2=O.O=C(CC(C1CC1)C1CC1)NC(C1CCC2CC12)C1CC1 c1(COC)cnc(OC)c(C(=O)NC2COCC2NC(C2C=CCCC2)=O)c1 c1(CN2CCN(C(=O)CCc3ccc(C(=O)O)nc3)C3C2C3)ccc(O)c(O)c1 CC(C)C(CC(=O)NCC1CCCOC1(C)C)NC(c1nnc(S)n1C)=O C12(NC(CNC(C3C(C)C3)=O)=O)CC(C(=O)NC3(CCO)CCC3)(C1)C2 N1(C(CONC(c2c(C)ocn2)=O)=O)CC=CC1(C)CO c1(C(=O)NCCN(C(C(C2(O)CCCCC2)CC)=O)C)ccc2c(c1)CC(C)O2 CC(c1ccccc1Cl)=CC(=O)NC(C)CCCNC(c1c[nH]ccc1=N)=O C1(NC(c2c(SC)ccs2)=O)CCC2CC1CN2C(=O)CC1(O)CCCOC1 C=CCC(CC=C)C(=O)NC1CCN(C(C2CCOCC2)=O)C12CCC2 C(N=c1nc2ncn(C)c2c(NCc2cccnc2Cl)[nH]1)c1cccc(C)c1F C1(COC)(CNC(C2CC23CC(O)C3)=O)CCCN1C(=O)C(C)(C)F c1(OC)ccc(C2CSCCN2C(=O)CCCN2CCOC2=O)cc1 C(=O)(CC(C)C(=O)N1CCN(C2CN(C(c3ccc(F)cc3Cl)=O)C2)CC1)OC c1(C(N(C2CN(C(c3occc3C3CC3)=O)C2)C)=O)ccc2[nH]nc(O)c2c1 C1(NC(CC=C)=O)CN(C(c2nnn(Cc3ccncc3)c2C)=O)CC(C)(C)C1 CC1CN(C(c2sccc2Cl)=O)CCC1NC(=O)Cc1cnn(C(F)F)c1 N1(C(C=C(CCC)CCC)=O)CCN(C(C2(C)SCCCS2)=O)CC12CC2 C1(C)(C(N(CCC(N)=O)C)=O)C=CCN1C(=O)CNC(N)=O CCCCC(C)CCC(=O)NCC1C=CC(NC(c2ccoc2Br)=O)C1 c1(OC(=O)NCCC2C(CCN(C)C)COC2)cccc(F)c1 c1(C(=O)NC(C2CCCN(C(c3cscc3C(F)F)=O)C2)C)ccc(=O)n(C)c1 N1(C(C=CCN(C)CC)=O)CCC2(CC1)CN(C(=O)C1=CCCC1)CC(C)O2 c1(-c2cc(NC(C(N3CC(C)N(C)CC3)=O)=O)n[nH]2)ccc2c(c1)OCCO2 N1(C(CC(C)NC(=O)OC(C)(C)C)=O)CCC(C(=O)NCC(N(C)C)C2CC2)C1 Cn1nnc2cc(C(N3CCCC3(C)CNC(=O)CC3CC4CC4C3)=O)ccc12 c1(CC)ccc(C(N2CCCC(NC(=O)CCC(C)CN(C)C)C2C)=O)c(O)c1 N1(C(CC2(CNC(CN(CCC)C)=O)CC2)=O)CC(CO)CC1CO c1(C(=O)NC2CC(CCNC(CC3CC(=C)C3)=O)C2)conc1C(F)(F)F c1(C(=O)NCCC(C)(C)CNC(C2CCOC2)=O)ccc2ncnn2c1 CC1(CCC(=O)NCC(=O)NCC(=O)NC2CC2)CN(C(=O)CC(N)=O)C1 C1(C(=O)NC(c2ccccc2)CNC(C(C)NC(CC)(C)C)=O)CC(C2CC2)C1 C#Cc1cc(C(=O)NC2CCC(C)N(C(=O)C=Cc3cnc(C)s3)C2)ccc1Cl CCC(CC(=O)N1CCN(C(c2cc(C)nc(O)n2)=O)C(CF)C1)C(F)F C1(C(N(CC(=O)NC(c2cncnc2)C)CC)=O)CCCC(C#N)C1 CC(C)CC(CNC(=O)C(N1CCCCC1=O)C)NC(c1ccccc1)=O CCCCC(CC(=O)NOC1CCCC1)NC(=O)CCCCC1CC1 c1(C(=O)NC(CCCC)CNC(=O)CC)[nH]cc2c1CCC2 C(=O)(C(C)(CCC)CCC)N1CCC(N(C(CCC)=O)C)C(C)C1 N1(C(Cc2c(C)nsc2)=O)CC2CCCN(C(C3CC4C=CCC(C3)C4)=O)C2C1 c1(OC)cccc2c1C(C(=O)NCC1CSCCS1)CC2 C1(CNCC2CC(C(F)F)OC2)CC12CCCCC2 C(c1cnn(C)c1)=C(C(=O)NC1CCC(CNC(c2c(CCC)[nH]cc2)=O)C1)C c1(CC)nc(C)c(C(=O)NC2CCC(CNC(=O)CC3CSC3)C2)o1 C(CC1=CCN(C(c2c[nH]nc2C(C)(C)C)=O)CC1)NC(C1(C)ON=C(C)C1)=O C1(NC(Cn2cc(CNC(C=C(C)C(F)F)=O)nn2)=O)CC2(C1)CC(C)C2 N1(c2c(C)c(NCCc3nnc(CO)s3)ncn2)CCOC(C)(C)CC1 C1(NC(CNC(C(CC)C)=O)=O)COC2CN(C(=O)C=Cc3ccncc3)CC12 C1(CC)CN(C(c2ccccn2)=O)CCC1NC(c1ccc(OC)s1)=O C=C(F)CN=C(NCC(c1ccc(Cl)cc1)NC(=O)OC(C)(C)C)NCC NS(=O)(=O)c1c[nH]c(C(=O)NC2CC(C(=O)O)C2)c1 c1(CN2CCC(C(N3CCCCC(C)(F)C3)C)C2)cccc(N=S(C)(C)=O)c1 c1(OC)ccc(C(=O)N(C2CCCC(NC(=O)CC3CCSCC3)C2)C)c(C)c1 C(C(C)(C)CC(=O)NC(C)CC(=O)NCC1CCC2(CC2)CO1)OC C(=O)(C1CCc2c[nH]nc21)NC(CCNC(C(=Cc1ccccc1)CC)=O)C C1(NC(CN(S(CC)(=O)=O)C)=O)CCC(C)(CNC(C2(C(F)(F)F)CC2)=O)C1 N1(C(c2c(NC(C)=O)cccc2F)=O)CCC2(NC(=O)C(CO)OC)CCCC12 CC1CC(NC(C23CC(C(F)(F)F)(CO2)C3)=O)CN1C(=O)C=CC1CCCCC1 C(CCC(=O)NCCCCC1CC1)NC(=O)OC(C)(C)C.C12CC1N2.C1(=O)CN1 N1(C(Cc2n(C)nnc2)=O)CC2CCC2(CCNC(=O)CC2(CO)CC2)C1 CC(C(=O)NCC(C)NC(C1CC(N2CC(O)C2)C1)=O)C1CCC1 c1(C(=O)NCC2(F)CN(C(CCCCNC(N)=O)=O)C2)cc2cc[nH]c2cn1 c12cccc(c1)N(C1CC3CNC1C3)C(=O)N2C.N1(C(=O)CC#N)CCSCC1 N1(C(C=Cc2c(C#N)cccc2)=O)CCC2C(CCN2C(C2CC2C(F)F)=O)C1 C(COCC)(C(=O)NC1(CC)CCCO1)NC(CSCC#C)=O c1(CC(N2CCC(C)(NC(c3cn(C)c(=O)cn3)=O)C2)=O)c[nH]c2ccccc12 c1(C(N2CC(C)C(NC(C3(O)CCSCC3)=O)CC2)=O)cc2c(ccn2C)s1 C(CCC(O)C(=O)NCC(C)(C)CC(F)F)NC(C(C)c1cccs1)=O c1(C(N2CCN(C(CN3C(=O)CSC3=S)=O)C3C2C3)=O)c(F)cc(F)cc1Cl Nc1cc(F)c(C(=O)N(CCNC(c2cn3ccncc3n2)=O)C2CC2)cc1Cl N1(C(c2cc(C)sc2)=O)CCCC(C)C1CNC(C1(O)CCCC1)=O c1(C(N(CC(CC)NC(C(C(CC)C)O)=O)C)=O)c(F)cc(C)cc1Br c1(CC)cc(C(N2CCC(COC)(NC(=O)CC(C)(C)N(C)C)C2)=O)cc(O)n1 C1(CC=C)CCCCN1C(C1C(C)CN1C(=O)C=CCC)=O C1(C(N2CC(C)CC(NC(C(CCC)NC(C)=O)=O)C2)=O)CC2C=CC1C21CC1 c1(OC(C(=O)N(CCCN(C(C(CC#C)C)=O)C)C)C)ccccc1C#N Cc1c(F)ccc(C(N2CC(C3CN(C(C4CC4[N+](=O)[O-])=O)C3)C2)=O)c1C C1(CCC)(NC(c2cnc(CC)nc2)=O)CCCN(C(=O)CC2CC2(C)C)C1 CCC(CC)C(C(=O)N1CC(C(=O)NOC(C)(C)C)C2(CCC2)C1)OC C(=O)(CCCCCCNC(=O)Nc1cccc(-c2n[nH]c(O)n2)c1)OC(C)(C)C CCC(O)CC(=O)NC1CCC1NC(c1ccc(-c2ccc(C)cc2)cc1)=O CCC(CNC(c1cccc(OC(F)(F)F)c1)c1nnnn1C1CC1)(CC)CO C1(NC(C2CN(C(=O)NC)C2)=O)CC(NC(C2CC(C(F)F)C2)=O)C12CCC2 N1(C(c2c(C)nc(C)o2)=O)CC2CCN(C(=O)C(F)(F)c3nccn3C)CC2C1 C=CCC(CC(=O)NCc1cc(C)c(C)s1)NC(c1cc(C(C)C)no1)=O N1(C(C(CC(C)C)C)=O)CCCC(C2(NC(=O)Cc3ncc(Cl)s3)CC2)C1 c1(CC)c(C(=O)NC23CC2CN(C(=O)C=CC)C3)cnn1C1CCCC1.CCC(C)C c1(CCC)nc(CS(=O)(=O)Cc2cc(C)on2)n(-c2ccn(C)n2)n1 C(C(C)(CC(C)C)NC(c1nsnc1O)=O)NC(Cc1c(C)cnn1C)=O CC1CCCn2ncc(C(N3CC(F)(CNC(=O)CCc4ncc[nH]4)C3)=O)c21 C1(F)(C(N(CC(C)NC(=O)C(c2ccc(Cl)cc2)(C)O)C)=O)C(C)(C)C1(C)C C(CCC)(C(=O)NC1CC(NC(=O)C(c2ccccc2F)C)C(O)C1)=CCC N1(C(C(CC)C(C)O)=O)CCCC(C2CCN(C(C3COCCO3)=O)CC2)C1 c1(C(=O)NC2CCN(C(CSCCCC)=O)C(C)C2)cccc2cccnc12 Cc1nc(CN(C(C)(C)C)C(C2CCCC2(C)C)=O)nn1-c1nc[nH]n1 C1(C(=O)NC23CC(C2)C3)(CC)CCCN(C(=O)CC2CCCOC2)C1 C(CN=C(NCC(C)C)NC1C2(CC2)C12CC2)c1c(OC)cccc1 C(=O)(CCCCCc1cccc(O)c1)NCC1C(NC(C=C(C)C(C)(C)C)=O)C1 c1(C(=O)NC(CC)(C)CNC(c2cscc2C)=O)cc2c(cc1C)OCO2 C(C)(C)(CC(F)C(=O)NCC1CSCC(=O)N1)NC(C(C1CCCCC1)C)=O C(=O)(CC(F)(F)C(F)F)N(CCCNC(=O)CCC(F)(F)F)CC c1(OC)cccc(C(=O)N(CC(C)C(=O)N(C)C(c2nc(C)no2)C)C)c1 C(=O)(C1=CC2(CCOC2)C1)NC(C=CC(=O)N(CC(C)O)CC)C c1(C(=O)NC(c2ccc(OCC)c(OC)c2)C)c(C)ccc(Cl)c1O C1(CNC(=O)CCOC2CCCC2)CCCN(C(=O)CCC2OCCO2)C1 c1(CC(=O)NC2C(NC(CC3ON=C(CC)C3)=O)C2)ccnc2ccccc12 CCC(CC(=O)N1CCC(C(=O)NCC(C)C(C)(F)F)(CC)C1)CC(C)C c1(NC(C(c2nc(CC(C)C)sc2)N(CC)Cc2ccoc2)=O)cccc(Cl)c1 N1(C(C2CC(C#C)(O)C2)=O)CCC(NC(=O)C(CSC)OC)C(O)C1 Cc1sc(Cl)nc1C(=O)NC(CNC(C1(Cl)CC12CCC2)=O)C(C)(C)C c1(CC)ccc(O)c(C(=O)N(C)CC2CCCN(C(=O)C(=O)NCC(F)F)C2)c1 c1(OC)cc(-c2cncc(NC(=O)C(c3ccccc3)C)c2)ccc1O c1(C(=O)NC2(CC(=O)Nc3ccc(Cl)nc3Cl)CCC2)ccc(F)c(Br)c1 C1(NC(c2c(C)oc(Cl)n2)=O)CCN(C(=O)CCC(C)(C)C)C(C2CC2)C1 C(=O)(CCC(F)(F)C(F)(F)F)NCC1N(C(=O)C(O)CC2CC2)CCN(C)C1 N1(C(c2nnc(C)s2)=O)C2CCC1CC(CNC(C1CCSCC1)=O)C2 C1(C(=O)NC(c2ncccc2C2CC2)OC)CCCN(C(N)=O)C1 C=CCCC(C(=O)NC1CCOC1)NC(=O)CC1(C)CC1 N1(C(CSC(C)C)=O)CC(C)CN(C(=O)Cc2ccc(F)cc2Cl)C(C)C1 C1(C(N2CC(F)(CNC(c3cc(CCCO)on3)=O)C2)=O)CN2CCC1CC2 C(=O)(CCCCC(C)C)N1C(CO)CC(NC(c2ccc(C)cc2Cl)=O)C1 C1(N(C(=O)CCC(N)=O)C)CC2CCC(C1)N2C(=O)CC1CCCC(C2CC2)O1 CC(C)CC(C)(C)OC(=O)NC(C)CC1CCCCO1 Cc1ccncc1-n1cc(C2(O)CN(C(C3CCC(C(N)=O)CC3)=O)C2)nn1 C1(NC(C(C2CCN(C(=O)C3=CCCOC3)CC2)C)=O)CC2(CCCO2)C1 c1(C(N(CCNC(C2(C)C=CCC2)=O)C2CC2)=O)cccc2nc(O)oc12 C1(OC)CC(C(=O)N(C)C(c2cnn(C)c2)C)N(C(=O)C(CO)NC(N)=O)C1 C1(O)(CCNC(CSCC#C)=O)CCCN(C(c2nocc2C(C)C)=O)C1 c1(NC(C(=O)N(CCCOCCN(C(CC)=O)C)C)C)ccccc1N.C(N)(=O)N C1(CNC(C2N(CCC)CCCC2)=O)(NC(=O)CNC(=O)NC)CCCCCC1 Cc1cc(C)c(C(N2CCC3CC23C(=O)NCc2nccn2C(C)C)=O)cn1 c1(C(=O)NCC2(COC)CCCN2C(=O)CNS(N)(=O)=O)ccc(F)c(O)c1 C12(C(=O)NC(CNC(=O)C(F)CC3CCCC3)C3CC3)CCC(CC1F)C2 C1(F)(CC)CN(C(=O)C#CCNC(=O)COC2CC=CC2)C1 c1(C(N2CCCN(C(C=C(COC)C)=O)C(CO)C2)=O)ccc2nc(O)[nH]c2c1 c1(C(=O)NC2CC(CNC(c3cccs3)=O)C2)c(F)c(F)cc(F)c1F N1(C(C(C)NC(c2ccccc2)=O)=O)CC2(CCCO2)C1 N1(C(CC2(C)CCC(=O)C2)=O)CCCC(O)(c2cn(-c3ccccn3)nn2)CC1 Cc1ccc2c(C(=O)NC3CN(C(=O)C(C)CC4CC4)CCC3O)cnn2c1C c1(C(N2CCC(O)(C(C)NC(=O)C(O)C3CCC3)CC2)=O)ccn2c1CSCC2 c1(C(N(CC(=O)NC(c2cn(CC)nc2)C)C(C)C)=O)ccncc1Cl C(CC(C(=O)N1CC([N+](=O)[O-])C1)NC(=O)C(C)CN(C)C)SC n1(CC)nc(C)c(C(N2CCOC(C)C2c2nc(C)no2)=O)c1C(F)F C1(C(C)(C)O)(CNC(c2ccnnc2)=O)CN(C(C2COCOC2)=O)C1 N(C(=NCCc1nc(C2CC2)n[nH]1)NCCc1cccs1)C1C(C)CCCC1 C1(C(=O)OC)CC(C)N1C(c1cnn(CCNC(C2CS(=O)C2)=O)c1)=O C1(=O)CCCCCn2cc(nn2)-c2cccnc2N1C.CC1CC1CO N1(C(C(C2CCC2)OCC)=O)CCCCC1CCCNC(=O)CCc1cnc[nH]1 C1(C(C)NC(=O)C2=CCC2)CN(C(c2cc(C3CC3)cs2)=O)CCO1 c1(C(N2C(C(=O)Nc3scc(C(C)(C)C)n3)COCC2)=O)cc(I)ccc1Cl C(=O)(C(F)CC(C)(C)NC(c1cn(C)c(C)n1)=O)NC(CC=C)CC C(CC(C(=O)Nc1cccc(Cl)c1)NC(c1n[nH]c(C)c1Cl)=O)=CC c1(CN2C(C)(C(=O)Nc3ncc(Br)nc3I)CC2)c(F)cc([N+](=O)[O-])cc1F c1(C(=O)NCC2CN(C(C3(CC)CCC3)=O)C2)ccc2nc(O)oc2c1 c1(N2C(C)CNC2)c(Oc2cccc(Cl)c2)ccc2ccccc12 c1(C(N2CC(N(C)C(C3CCC34CCC4)=O)C2)=O)ccc(C(F)F)c(F)c1 c1(CC)c(C(N2CCCC2C(C)(C)C(=O)NCC(C)O)=O)nnn1C CCCC(C(=O)N1CCOCC1)OC(C1(C(=O)OC)CCC1)=O C1(C(N2CCN(C(c3ccc(C)c(C)n3)=O)C(C)C2)=O)CCc2n[nH]cc2C1C Cc1cccc(C(=O)Nc2ccsc2C(N2CCOCC2C(C)C)=O)c1C Cc1ccc(Br)cc1C(N1CCCC(C(=O)NCCc2cscn2)C1)=O C(=O)(C#CC(C)(C)O)NC(C(C)NC(c1cn(C(C)C)nc1)=O)C(C)C c1(C(=O)NC2(CC=C)CCN(C(C3CCN3CC)=O)C2)coc2c1CCCC2 N1(C(Cn2ccc(C)n2)=O)CCC2(CC1)CCN(c1ncnn3ccc(Br)c13)C2 c1(C(C(=O)NC2CN(C(c3occ(C)c3)=O)CC2F)(F)F)ccc(F)c(F)c1 CCC(CC)C(C)C(=O)NCC(C1CCCC1)NC(c1cc2c([nH]1)CCC2)=O N1(C(c2cccc(CCC)c2)=O)CCN(C(=O)C(F)CC2CCCC2)CC(O)C1 C(=O)(C(COC)NC(C1CCN(CCF)C1)=O)N(C(C(=O)NC)C)C c1(C(N(CCN(C(CC(COC)C)=O)C(C)C)C)=O)cc(Br)ccc1OC N1(C(C2C=CC(C(=O)OC)C2)=O)CCC(F)(CNC(=O)C=CBr)C1 N1(C(=O)OC(C)(C)C)CCn2c(CNC(C3(C)CCCNS3(=O)=O)=O)nnc2C1 c1(C(=O)NC(CCN(C(C(CC)OC)=O)C)C)ccc(C#CC2CC2)cc1 CC1CN(C(=O)CCOC2CC2)CC1CNC(c1csc(C(N)=O)n1)=O n1(CC(=O)OCC)c(N2CCC(C)C2)nnc1-c1cc(Br)no1 N1(C(C(c2cn(C)nc2)(C)C)=O)CCC2(CC1)CC(NC(C1(N=[N+]=[N-])CC1)=O)C2 C(=O)(CCC(C)(C)[N+](=O)[O-])N(C1CCN(C(c2c(OC)c(Cl)ccc2)=O)C1)C c1(C(N2C(C)C(NC(C3CC(F)C(=O)N3)=O)CC2)=O)cncc2c(O)nccc12 CN1C(=O)CC(C(=O)NCC(=O)NC2CCC2O)C1c1ccc(Cl)c(F)c1 CC1(C)CN(CC2CCC(C(F)(F)F)C2)C(C)(C)C1O N1(C(c2ccc(OCC)cc2)=O)CC2(CCC2NC(=O)C=C2CCSCC2)C1 c1(C(N2CC(CNC(CCC(C)SC)=O)C(N(C)C)C2)=O)ccc(CO)c(F)c1 C#CCCCC(C)C(=O)NC(CCC1CCC1)C(=O)NCC(C#N)CC c1(C(=O)NCC2N(C(C=C(CCN(C)C)Cl)=O)CC2)c(Br)ncn1C CC(CC(=O)NC1CN2CCC1CC2)C(C)(C)NC(C1C=CC=CC=C1)=O Cc1cc(C(N2CC(CNC(C3(C(F)F)CCOCC3)=O)C3CC23)=O)c(C)n1C Cn1ccc2cc(NC(C3COC4CN(C(C5CCCCO5)=O)CC34)=O)ccc12 c1(C(N2C(CNC(CCn3c(C(C)C)ncc3)=O)CC2)=O)nn(C)cc1N N1(C(C2(CC)CNC(=O)C2)=O)CC2(CC(C(N3CC(=O)NC(C)C3)=O)CO2)C1 Cc1ccc2c(c1)C(C(=O)NC1(CCNC(=O)C(c3ccc(F)cc3)O)CC1)C2 C1(NC(c2ccc(SC)s2)=O)CN(C(c2cc3ccoc3s2)=O)CC(F)(F)C1 c1(C(=O)NC(C2CCN(C(CC=C)=O)C2)C)cc(C(F)(F)F)cnc1N C1(C(N(C(C)C)C(C)C)=O)CN(C(=O)C2=NOC(c3ccccc3)C2)CCC1O C1(CC)C(C(N2CCN(C)C(C)C2)=O)CCCN1C(=O)CCOCC1CCC1 c1(OCC)ccc(C(=O)NCC2CCC(C)CN2C(=O)C2=COCCC2)cc1N C1(C(=O)NCC(CC(C)C)C)CCN(C(C2CC(F)CN2C)=O)CC1C C(=O)(C(C)(O)C(F)(F)F)N1CCC(OC)(CNC(C23CCCC2C3)=O)CC1 CC(C)CCCCC(=O)N(C)CC1CN(C(C2CCC3CCC2O3)=O)CCO1 C1(C)(C(N(CC(C)NC(c2csc(C3CCCC3)n2)=O)C)=O)CC2(CCC2)C1 N1(C(c2cncc(SC)c2)=O)CCC2(CCC2NC(=O)Cn2nnc(C)n2)CC1 c1(N2CCCN(Cc3cc(O)c(Cl)cc3)CC2)ncnc2[nH]ccc12 C#Cc1cc(F)c(C(=O)N(C)CCOCCN(C(=O)C(N)=O)C)c(F)c1 C(=O)(C(C(C)C)N(C(=O)CC1(C)CCCC1)CC)NCC.C1C(C)N1 N1(C(C23CC(COC)(OC2)C3)=O)CCCN(C(c2cnns2)=O)C(C)C1 C(=O)(C(CC(C)C)N1CCCCC1=O)NCCCN(C(=O)CC1CC12CC2)CC c1(C(N2CCC(CNC(c3c(COC)ncs3)=O)C2)=O)cc([N+](=O)[O-])ccc1C c1(C(=O)NCC(CNC(C2(C)CC=C(C)CC2)=O)(C)C)coc2c1C(O)CCC2 C12(C(N(CCC)CCNC(C3CCCN3C(C)=O)=O)=O)CCCC1CCC2 C12C(C)CCCN1C(=O)C(=O)N2.Cc1cccc(SCC(c2ccccc2)C)c1 N1(C(C(c2cn(C)nn2)NC(C=C(C)C(C)(C)C)=O)=O)CCC2(C1)CN(C)C2 C1(C2CCC2)(C(N2CC(O)(CNC(C(c3ccccc3)OC)=O)C2)=O)CC1(F)F c1(OC)ccc(Cl)c(CC(=O)NCC(C2CCC2)NC(C2CC2F)=O)c1 Cc1cccc(C(=O)ON)c1.C1(C)C(=O)N(CC(F)F)CCOC(=O)N1.C1C(=O)N1 C(=O)(C1=NOC(C)C1C)N1C(CC)C(NC(c2ccnn2C(C)C)=O)CC1 c1(NCCC(Cc2cccs2)NC(c2ccc(C)[nH]2)=O)cnc(Cl)c(Br)c1C C1(CC(N2CCC(O)(C(C)CNC(C3CSCCS3)=O)C2)=O)CCC(C)(C)CC1 C#CC(C)(C)C(=O)NCCC(C)NC(c1c(Cl)noc1C)=O c1(Cc2cc(=NC)[nH]cc2)cc(=NCCC2CCN(C(=O)NC(C)C)C2)[nH]cn1 C#CCC(O)C(=O)NC1CC1CNC(=O)Cc1csc(-c2ccc(Cl)cc2)n1 CCC1=C(C(=O)NC2CCC(C(=O)NCC3CC(C)=NO3)C2)CCCO1 c12c(cnn1C)N(C)C(=O)CN(C)CCCn1cc-2nn1.c1(CO)c[nH]nc1F C#Cc1cc(NC(=O)C(CC2CCC2)NC(C2CCCC(C#N)C2)=O)cc(F)c1 Nc1cccn(CC(=O)NCC2(NC(C3SCCS3)=O)CCCCC2)c1=O C1(CNC(C(C)OCCOCC)=O)CCC(C(N2CCC(F)(CF)C2)=O)CC1 N1(C(C2(C)CC(=C)C2)=O)CCC=C(C(=O)N2CCCC(OC)CC2)C1 c1(C(=O)NC(CNC(C(CC)(C)OC)=O)C)ccc(C(F)(F)F)c(F)c1 C1(C(N(C(CNC(=O)CCCCO)C2CC2)C)=O)CC(=O)NC1(C)C N1(CCNC(C2CCN(Cc3ccncc3)CC2)C)CCC(CC2CCC2)CC1 C1(C(=O)NCC(C)NC(=O)CC2CS(=O)(=O)CCN2C)Cc2n[nH]cc2C(=O)N1 C1(C[Si](C)(C)C)CCC(N=c2nc(-c3cc(Cl)cc(Cl)c3)[nH]o2)C1 CC1CN(C(=O)C(F)C(C)(C)O)CCCN1C(c1cc(Cl)ncc1N)=O CCCC(C)CC(=O)NCC(C1CCCCC1)NC(C12CC(C1)C(C)O2)=O N1(C(C(C2CC2)OCC)=O)CC2(CCC2NC(c2ccc(OC)s2)=O)C1 c1(NCC)cncc(C(N2CC=CC2CNC(c2ncn(C(C)(C)C)n2)=O)=O)c1 S(=O)(=O)(c1cccc2c1OCCCO2)NC(c1ccc(=NC)[nH]c1)=O CCCC(C)C(C)(c1nnnn1C1(C)CC1)NCCOCC(F)(F)C(F)F.CCO Cn1cc(C(=O)NC(CNC(C2(S(C)(=O)=O)CCC2)=O)CO)n(C)c1=O c1(C(=O)NCC(CC)NC(c2cnc[nH]2)=O)cc(S(N)(=O)=O)co1 c1(C(=O)Nc2cc(Cl)cc(Cl)c2Br)n[nH]c2cccc(-c3cnn(CCF)c3)c12 N1(C(c2cncc(C(C)C)c2)=O)CCN(C(C23CCCC(C2)OC3)=O)C(CO)C1 CC1=NOC2(C1)CC(C(=O)NCCCNC(=O)CC(Cl)Cl)C2 c1(C(=O)NCC(CC)NC(=O)C(F)(F)C2(O)CCC2)ccc(COC)s1 C1(NC(CCOC)=O)CCCC1NC(=O)COCC1CCC1 Cc1cc(C)c(C(=O)NCC(C2CCCN2C(=O)COC(F)(F)F)(C)C)c(O)n1 c1(C(=O)NC2C(NC(CCc3cc(C)on3)=O)COC2)cnc2[nH]ncc2c1 CCC(COC)C(=O)NC1CCCC1CC(=O)NCC1CC(C(C)C)C1 CC(C)(CO)CC(O)CNCC(C)(C)C1(O)CNC1 Cc1cc(C(=O)N(C2CCCN(C(=O)C(N3CCNC3=O)C)C2)CCO)n(C)n1 Cc1ncc(C(=O)NC2CC(C(N3CCC(CC(N)=O)C3)=O)C2)cn1 N1(C(c2c(OC)scc2)=O)CCN(C(=O)C(C)(C)C#N)CC(C)(C)C1 CC(C)C(C(=O)NCC(C)CNC(c1ccon1)=O)NS(N)(=O)=O N1(C(c2ccc(CC)cc2)=O)CC(C)N(C(=O)CCCCC(C)C)CC1C N1(C(C)=O)CCN(C(=O)CCN(C(=O)C(CCOC)OC)CCO)CC1.CCCO c1(CN2CC(C(=O)NCCn3c(C)ncc3)SCC2)cc(F)ccc1Br CC1(CNC(=O)CCN2CCOCC2)CCN(C(c2cnc(C3CC3)s2)=O)C1 c1(COCC#N)cccc(C(=O)N(CC(C)NC(=O)CC2CC=CCC2)NC(C)=O)c1 C1(NC(C=Cc2n(CC)ccn2)=O)CN(C(C2CCCCC2(C)C)=O)CCC1O N1(C(c2ccc(C(C)=O)o2)=O)CC(NC(=O)C(C)Cc2ccccc2)CC1C C(N=c1nc(N2CCC(CO)CC2)c2sccc2[nH]1)c1ccc(C2CC2)cc1 C(CC(=O)NCC1(C)CCN(C(c2ccc(CO)cc2)=O)C1)(C(C)C)OCC C1(C(C)C)CN(C(=O)CC(C)c2ccccc2)CCN1C(=O)C1=COCCO1 N1(C(c2cc(C)on2)=O)CCC(C)(CNC(=O)CCc2ccc(Br)cn2)C1 n1(CCC)ncc(C(=O)NCC2CN(C(c3cc(F)cs3)=O)C2)c1C C(=O)(C1=NN(C)C(=O)CC1)N1C(CC)C(NC(c2cncn(C)c2=O)=O)CCC1 c1(C(N(CCCNC(c2[nH]cc(C(=O)OC)c2)=O)C)=O)cnnc2ccccc12 c1(CCC)ccc(NC(N2CCCC(NC(c3ccccc3)C)C2)=O)c(C#N)c1 N1(C(c2c(N)cnc(Cl)c2)=O)CC2CCCN(C(c3cnn[nH]3)=O)C2C1 C1(CC(=O)NCC2=C(C)CCC2)N(C(C2CCN(C)C2C)=O)CCC1(C)C C1(C(N(C2CCN(C(=O)CCC3CC(F)(F)C3)CC2)CC#C)=O)CCS(=O)CC1 N1(C(C2(C)CN(Cc3ccc(C#N)c(Cl)c3)C2)=O)CCN2CCCC2C1 CC(Cc1ccccc1)C(=O)NCCC(C)(C)NC(c1cc(C(N)=O)no1)=O c1(C(=O)NC(C2CCN(C(c3c(C)ccc(O)c3)=O)C2)C)c[nH]c2cccnc12 CC(F)(F)C(C)(C)CCCN.C1(CC(=O)NC(c2cccnc2)C(=O)N)CCC(=O)N1 CCCC(CCC)=CC(=O)N(CCC)CCNC(=O)Cn1nccn1 CC1(C)CCCN(S(=O)(=O)N2CCC(C(N)=O)CC2)C1C(=O)O CC1CCC(CNC(c2nccnc2-n2ccnc2)=O)N(C(=O)CNS(N)(=O)=O)C1 C1(NC(c2cc(C(F)F)on2)=O)(CNC(C2(O)CC2)=O)CCOC1 O=C(C#CC1CCCO1)NCC1CN(C(=O)C2=CCCS2)CC12CCC2 CON(CCC(=O)NCCc1ccoc1)C(=O)C1=C(C)OCC1 C(=O)(C(CC1CCOCC1)NC(=O)CC1(CO)CC1)N(CC)CC1CCCC1 C(=O)(CC(C(F)(F)F)N(C)C(c1csc(O)n1)=O)NCC(COC)OC N1(C(=O)Cc2ccccc2F)CCCC2C1CCN2c1ncnc2sccc12 C1(CC)CN(C(C2CC(F)(F)CS2)=O)CCN1C(=O)CC12CCC(CC1)C2 C1(NC(CSCCCC)=O)CCC12CN(C(c1ccco1)=O)C2 c1(NC(C2CC(C)(C(=O)OC(C)(C)C)C2)=O)ccc2c(c1)C(O)CC2 c1(NC(C(CCC#C)NC(=O)Cc2nc(=N)[nH][nH]2)=O)cccc2c1CCO2 N1(C(C(CC(N)=O)NC(CCCCN=[N+]=[N-])=O)=O)C2CCCC1CC(O)C2 c1(C(N(CC(F)(F)F)CC(C)C)=O)cnc2ccccc2c1Br Cc1cc2ncn(CCNC(=O)C=Cc3ccc(F)c4ccccc34)c2cc1C N1(C(c2c(C(C)C)nns2)=O)CC2CCC1CN2C(c1cnc2ncccn12)=O C1(CCNC(CC)=O)CCN(C(=O)C(CC(C)(C)C)OC)C12CCC2 N1(C(C2C(OC)CN(C(c3cnc(CC)nc3)=O)C2)=O)CCC(CO)C(C)(C)C1 N1(C(CC2ON=C(C)C2)=O)CCC12CN(C(C1CCN(C)CC1)=O)C2 C#CC1CCN(C(=O)C(F)C2CC(NC(C3(N(C)C)CC3)=O)C2)C1 C(=O)(C(CCF)NC(C1C=CCN(C(c2oc(C)cc2C)=O)C1)=O)OC C(=O)(CC(C)C(C)C(C)C)N1CCC(CNC(c2c(OC)scc2)=O)C(C)C1 c1(C(N(CC(C)NC(C(C2CCC2)OC)=O)C)=O)c(C)cncc1F C1(CNC(c2ccncc2)=O)CC(F)(CNC(C23CCC2C3)=O)C1 c1(OC)ccc(C)c(NC(c2cc(NC(=O)C#CC(=O)O)cn2C)=O)c1 C(=O)(C1=CNC2=NCCCN12)N1CC(CN(C(=O)C=CC(F)(F)F)C)OCC1 c1(C(=O)NC(CN(C(=O)C(C)CC(N)=O)CC)C)cc(Br)c2c(c1)CCO2 c1(CNC(=O)CN2CC(NC(C34CNCC3C4)=O)C(=O)N2)ccccc1CO C1(O)(CNC(C=CC(C)C)=O)CCN(C(C2CCN(CC(C)C)C2)=O)C1 C1(OC)CC(NC(=O)CCc2cc(C)on2)CN(C(C2CC(C)(O)C2)=O)C1 N1(C(C=C(C)C2CC2)=O)CCOC2(CCC(N=c3nc(C(C)C)[nH]s3)CC2)C1 C(C(C(C)(C)C)NC(=O)CC(C)O)NC(C1N(CC)CCC1)=O C1(C(=O)NCC=CCC(=O)NCC2CCC(=O)O2)CC12CCCC2 Cc1ccc2cc(C(=O)NC(C)(C)CN(C(=O)C=Cc3cn(C)nn3)C)[nH]c2c1 n1(CCC(=O)NC2(CNC(C(CC)(C)OC)=O)CCCC2)ccc(O)nc1=O c1(C(=O)NCC(CC)(CC)NC(C=CCOC)=O)ccc2c(c1)CCC(=O)N2 c1(C2C(C(N3CC(C)(NC(c4n(CC)ncc4)=O)C3)=O)C2)ccc(Cl)nc1 C1(c2n(C)nnn2)(NC(CC2CC2)C2CC2)CC2(CCCOC2)C1 CCCCC(CC)C(=O)NCc1occc1C(=O)NCC(CC)n1cccn1 c1(CC(N2CC3C(CNC(c4c(C)ncnc4)=O)C3C2)=O)cccc2c1OCO2 N1(C(c2ccc(CC)o2)=O)CCN(C(=O)C2=C(Cl)CCOC2)CC(O)C1 C(=O)(C1CCCn2c(Br)cnc21)NC(C)CNC(=O)Cc1cc(F)ccc1O N#CC1CN(c2ncc(I)cn2)CCN1c1ncncc1F C=C1c2ccccc2C(=O)N1C(C)C(N1CCC(C)S(=O)(=O)CC1)=O N1(C(C=CCN(C)C)=O)CCN(C2CCN(C(c3csnn3)=O)C2)CC1 CCCCCCC(C)C(=O)NCC1CCC1NC(C1(CC)CCC1)=O C(=O)(C(F)C(C)(F)F)NCC1(COC)CCCN1C(c1cccc(C(C)C)n1)=O O=C(CC(C1=CCCC1)NCc1ccnnc1)Nc1ccccc1F c1(SC(CC)C(=O)NC(c2ccc(C(C)C)cc2)CO)ccc(Br)cc1 C1(NC(C(CC=CC)NC(c2ccn(C(F)F)n2)=O)=O)CCC(=O)NC1C CC1CC(c2cn(-c3ncc(Cl)cn3)nn2)CCN1C(c1cc(N)cc(F)c1)=O c1(C(=O)NCc2ncccc2C(N2CCC(F)C2)=O)cnc2c(Cl)cccn12 C1(NC(CCOc2ccc(OC)cc2)=O)CCN(C(C2CCCSC2)=O)CC1F C1(COC)(NC(c2ccc(OC)s2)=O)CCCN(C(=O)C(C)SC)C1 CC1(C(=O)NCC2CN(C(=O)C(C)(C)c3ccccc3)CC2O)CC(F)(F)C1 c1(N(C(=O)CC2COCCO2)C)cccc(Oc2ncns2)c1 N1(C(Cc2c(C)noc2C)=O)CCC(NC(c2ccnn2C)=O)C(C)(C)C1 N1(C(c2nc(CC)sc2)=O)CC(CNC(=O)C(=O)NCCC(N)=O)CC1C C1(OC)CC(C)CN(C(c2ccc(OC3CCC3)cc2)C(=O)NCCCF)C1 N1(C(=O)OC(C)(C)C)CC(C(=O)NC2CC23CCCC3)CC(F)C1 C1(C(C)C)CN(C(c2ncn(C)n2)=O)CCN1C(c1cc(Br)n(C)n1)=O n1(CC)nc(C(=O)NCC2CC(C)N(C(=O)Cc3ncoc3C)C2)cc1C Cc1ccc2cc(C(=O)NCCCn3cc(-c4coc(C)n4)nn3)sc2c1 c1(SC)cn(C)nc1C(=O)NC1C=CC(CNC(C2CC=CCO2)=O)C1 C(CC)(C(=O)NC1CC(CSC2CCCN2C(=O)C=CC(=O)NC2CC2)C1)=CC C1(CC=C)(C(=O)NC(c2nc(C)no2)C)CCCN1C(=O)Cc1ccn(C)c1 C1(C(N(C)CCNC(c2ccccc2OC2CC2)=O)=O)CCCCC12CCC2 N1(C(C2CC(OC)(OC)C2)=O)C2CCC1CC(NC(c1ccsn1)=O)C2 c1(C(=O)NCC(C)NC(C(C)OCc2ccc(C)cc2)=O)ccc(C)nc1N CC1=NOC(C(=O)NC(CNC(=O)CNC(c2cccc(F)c2)=O)C2CC2)C1C N1(C(CCc2ncc(C)[nH]2)=O)CC2(CCOCC2)C1c1cn(-c2nccs2)nn1 c1(C(N(CC2CC2)CC2CC(O)C2)=O)cnccn1.O=CCN c1(-c2ncc(C(=O)NC(CC=C)CO)nc2)cc(SC)cc(F)c1 N1(C(c2scc(C)c2)=O)CC2CCCC(NC(c3cnoc3)=O)C2C1 N1(C(CCC)=O)CCC2(CCC(NC(C3CCC(O)CN3C)=O)CC2)C1 C1(NC(C(N2CC(C)C2)C)=O)CCN(C(c2cc(Cl)n[nH]2)=O)CC1O CC1(C2(C(=O)NCCc3cc(C(=O)O)no3)CC2)CC1 C1(C(N(CCC(C)NC(=O)C(C)(C)C2CCCO2)C)=O)CCC(N(C)C)CC1 n1(CCC(=O)NCC(CN(C(Cc2cc(C)n(C)n2)=O)C)C)ccc(O)nc1=O c1(NC(C(C)OC(C2CN(c3ncccn3)C2)=O)=O)cccc2ccoc12 c1(C(N2C(CNC(C3C(C)C3C)=O)C(O)C(O)C2)=O)cc(=O)c2ccccc2[nH]1 C1(NC(CC(=O)NC)=O)C2CN(C(=O)Cc3csc(NC=O)n3)CC12 c1(C(N(C(C(=O)NC)CO)C2CC2)=O)nc(C(=O)OC)co1 C1(NC(C(COC(C)(C)C)N(C)C)=O)CCC2(CC1)CC(NC(C1CC1F)=O)C2 C=CCC(C)(C)CC(=O)NC1COCC1NC(C1CCCN(C(=O)N(C)C)C1)=O Cc1nn(C)c(C)c1C(=O)NCc1cc(C(=O)O)ccc1C(F)(F)F N1(C(C)=O)CCCC(OC(=O)C(C)(C)C2CC2)C1.C(=O)C(C)C N1(C(CS(CC)(=O)=O)=O)CC(C)N(C(c2ccc(C)c(Cl)c2)=O)CC1C C(C(=O)N1CC(C)(O)CO1)OCCN(C(=O)CC1=CCCCC1)C.C1CO1 C1(N(C(C=CCCC)=O)CC(=O)NCC2(O)CC2)CC(C#N)C1 C(=O)(CCCS(=O)(=O)N1CCCC1)NCCN(C(C(CCC)C)=O)CC N1(C(C(CC#C)NC(c2cccc(CO)c2)=O)=O)CCCC(C)(C#N)C1 Cc1ncnc2c1CC(C(=O)N(CCC(C(C)C)NC(c1ccoc1)=O)C)CC2 N1(C(=O)OCC)CCCC(C2CCCN(C(=O)CCC3OCCC(N)C3O)C2)C1 C1(C(N2CC(CNC(C3(C)CC(=C)C3)=O)OCCC2)=O)Cc2c(C)cccc2N1 S(=O)(=O)(c1cccc2cnccc12)N1C(C(C(F)(F)F)NCC2(C)CCC2)CC1 C(CCCC(=O)N(CC(C)(C)CNC(C1CCC1c1nc[nH]n1)=O)C)(OC)OC c1(C(N2CCCC(NC(CC3CCC(C)C3)=O)CC2)=O)c2c(nn1C)CCCC2 c1(OC)cnc(Cl)nc1N1CC2C(NC(=O)C(C)OC3CCCC3)C2C1 CCCC(C)(O)C(=O)NCCCC(C)NC(C12CC(C1)C2)=O N1(C(CN2CCC(C)(C)C2)=O)CC2ON=C(CNC(=O)CCNC(=O)CO)C2C1 CCCCC(O)C(=O)NC1(C)CC(C(=O)NC2(C)CCOCC2)C1 n1(CC(=O)N(C(C)CCNC(c2nc(C3CC3)cs2)=O)C)nc(O)ccc1=O C(CCS(C)(=O)=O)(C1CC1)NC(NC(C1CC2C=CC1C2)C(=O)OC)=O Cc1nc(C)c(C(=O)NC2CCN(C(=O)CC3CCN(C)C3=O)CC2O)c(C)n1 N12CC(C(F)C1)NCc1cc([nH]c1)C2=O.c1(C=O)c(C)ncn1C.CO c1(C(=O)OC)ccc(C)nc1N1CCCC(C(N2CCNC(=O)C2C)=O)CC1 c1(C(N2C(C)CN(C(c3ccc(N)cn3)=O)CC2)=O)ccc(Cl)c(S(C)(=O)=O)c1 C(=O)(C1COc2ccc(Cl)cc21)N1C(Cn2cc(CCC(=O)O)nn2)CC(O)C1 c1(C(N(C2CC(NC(CCc3cc(C)[nH]n3)=O)C2)C)=O)nccc2occc12 C12(C(N3CC(CNC(c4cnc(CC)s4)=O)OCCC3)=O)CCCCN1CCC2 CC(C(=O)NCC1=CCCN(C(C2(F)CCOC2)=O)C1)S(N)(=O)=O C(C(=O)NNC(=O)COc1c(Cl)cccc1Cl)c1ccc(OC)c(OC)c1 C1(C(N(CC(C)NC(C23CCN(CC2)CC3)=O)CC)=O)CN(C)C(=O)CCO1 Cc1cc(C(=O)NC2CC(C)N(C(c3cn(-c4ccn(C)n4)cn3)=O)C2)ccn1 N1(C(CCCCCC)=O)CC2=C(C1)CN(C(C1CC3CCC1C3)=O)C2 c1(C(C(=O)O)NC(N(C)CCC2CCCN2C)=O)ccccc1Br C(=O)(C(C)(F)C(=O)NCCCC(C)NC(=O)CN1CCCNS1(=O)=O)OCC N1(C(=O)NCC(C)CN2CCOCC2)CCCC1Cn1ccnn1 C12(C(N3CC(C)C(CC(=O)NCC4CNC(=O)C4)C3)=O)CCCC1OCC2 C#CCC(C)(CC)C(=O)N1CCCC(NC(c2sc(SC)cc2C)=O)CC1 Cc1ccccc1COCC(=O)NC(C)C(C)NC(c1ncccc1O)=O C(=O)(C(F)CCC(C)(C)C)NC(C(N1CCC(OC)C1(C)C)=O)Cc1cnc[nH]1 N1(C(CC(n2c(CC)ncc2)C)=O)CC(O)CC1CNC(c1csc(=NC)[nH]1)=O N1(C(c2cn(CC)nn2)=O)CCC2CN(C(=O)C(F)(F)C(O)C3CC3)CC2CC1 C1(C(N2CC(c3cn(-c4nccs4)nn3)C2)=O)CCCCC1C1CC1 Cc1ccc2cc(C(N3CCC(NC(C4CCC(C)CC4)=O)C(C)C3)=O)cn2c1 C1(C(=O)N(C(C(C)C)C2CCC2)CCO)CN(C(=O)C2CC2)CC1C(C)C c1(C(=O)NC2(C)CCN(C(CC(C)(C)OC)=O)C2)cccc(S(N)(=O)=O)c1 c1(C(=O)NCC(CC)(C)NC(c2n[nH]c(C)n2)=O)cccn(CC(=O)NC)c1=O C1(C(N2CCC3(CN(C(C4CC5CC5C4)=O)C3)C2)=O)COc2cc(F)ccc2O1 c1(CCOC(CCNC(C)=O)=O)cc(C)c(F)cc1Cl C1(C(=O)NCc2c(C(=O)NC3COC(C(F)F)C3)c[nH]n2)CC12CCCC2 c1(CNCc2c(C)nns2)cccc(N2CCOC2=O)c1 c1(Cc2cn(CCNC(C(CN(CC)CC)F)=O)nn2)cccc(S(C)(=O)=O)c1 c1(C(=O)NCC2CC3CC3N2C(=O)CC2CC=CC2)[nH]nc2ncnc(O)c12 C(=O)(C1CCc2scnc21)NCC(C1CCCCN1C(=O)CC1CCSC1)(C)C c1(CC(N2CCCCC(NC(C3(Cl)C(C(C)=O)C3)=O)C2)=O)cnc2cccnn12 C1(CC(=O)NCC=CCNC(c2c[nH]nc2-c2ccncc2)=O)CCOCC1 c1(OCC(=O)N(C(C)CNC(c2ccc(C(C)O)cc2)=O)C)cc(F)cc(F)c1 C1(CNC(c2cc(C)on2)=O)CCN(C(C2(C)CCC(O)CC2)=O)CC1(F)F C1(F)(CNC(c2ccc(C)s2)=O)CCN(C(c2cccc(OC(C)C)c2)=O)CC1 c1(C(N(CCOC)CCNC(C23CC(C)C2C3)=O)=O)cccc(C(C)C)n1 c1(C(N2C(CC(=O)NCC(CCOC)O)CCC2)=O)ccn2nccc2c1 N1(C(C(CC)(C)OC)=O)Cc2ccccc2C(NC(C2(C(N)=O)CCC2)=O)C1 C12(C(=O)NCC(C3CC3)NC(C3(C)CC(C)C3)=O)CC(C)(CCO1)C2 Cc1cc(N)cnc1C(=O)NCC12CCC1CN(C(C1CCS(=O)(=O)C1)=O)C2 C#CCCCCCCCNC(=O)C(C1CCC1)NC(=O)CC(O)CC(C)C C(=O)(CC1=CCCC1)NC(C1N(C(C(SC)SC)=O)CCC1)C c1(C(N(C)CC2N(C(C3(CC(C)C)CCCC3)=O)CCC2)=O)cccnc1O c1(CN(C(C2C(N)(CC)C2)=O)C)ccc(SC)c(C2CC2)c1 c1(C(=O)NC2C(NC(c3ccnnc3O)=O)CC2)nccn2ccnc12 N1(C(C2=CC(C)(CC)C2)=O)CCC2CCN(C(c3sc(C)nc3C)=O)CC12 c1(OC)ccc(OC)c(C(=O)NC(CCN(C)C(C2CC(F)C2)=O)C(C)C)c1N c1(NC(C2(C)CN(C(c3n(C)ncc3Br)=O)C2)=O)ncc(C#N)cc1I CCCCCCC(C)(C)C(=O)N1CC(O)(CCNC(=O)C=CC=C(Cl)Cl)C1 c1(C(=O)NC2(CNC(c3cc(CC)sc3)=O)CCCC2)oc(C)nc1C c1(C(=O)NC2(CNC(COC)=O)CCC2)cc2c([nH]1)CCOC2 C=CCC(CC)C(=O)NC1(c2cn(CCSCCO)nn2)CCOC1 N1(C(=O)Nc2c(OCC)c(Cl)ccc2)C(C)CS(=O)(=O)CC1C CC1CCC(C(=O)N2CC(n3cc(CN(C4CC4)CC4CC4)nn3)CO2)CC1C n1(C(CC)CC)nc(C)cc1C(=O)NCC1CN(C(=O)C=CCn2cncn2)C1 c1(C(=O)NC(CC(C)C)CNC(=O)C(C)S(N)(=O)=O)ccc2cc[nH]c2c1F C1(CC(=O)NCCCOCCNC(CCCN(C2CC2)CC)=O)CCCC12CC2 C1(NC(=O)CSCC(F)F)COCC1C(=O)NCC1(O)CC(CO)C1 C1(C(C)NC(C2(C3CCCO3)CC2)=O)CCN(C(=O)C(c2ccnn2C)C)CC1 N1(C(C2C(SC)CCC2)=O)CCCOC(CCNC(c2nnsc2C)=O)C1 CC12CCCN1S(=O)(=O)C(C(N1CC(CCO)(NC(=O)C(=O)NC3CC3)C1)=O)C2 C1(C(N2CCC(CNC(CC=C)=O)C(C)C2)=O)C2CCC1(C)C2(C)C N1(C(Cc2c(CC)cccc2)=O)CC2OCC(NC(C3CC3(C)C(F)F)=O)C2C1 C(=O)(CCC(C)(C)OC)NC1CC(N(C(=O)CCOC2CCCC(CO)C2)C)C1 N1(C(c2c[nH]c(=NC)s2)=O)CCC(NC(=O)C2=C(C)CCOC2)CC(C)(C)C1 C=C(C)C(O)CC(=O)NCC(C1CCCC1)NC(c1cc(-c2csc(C)n2)c[nH]1)=O N1(C(CC(=O)OC(C)(C)C)=O)CC2CC1C2NC(C12CCCCC1C2)=O C(=O)(C1=CCC(F)(F)CC1)NCCN1CCC(NC(C(C(C)SC)O)=O)CC1 C1(C(=O)NCc2ccc(C(C)NC(c3cscn3)=O)cc2)CCc2c[nH]nc2C1 c1(NC(C2CCC(c3ccc(OC)cc3)CC2)C)ccc2c(c1)C(C)(C)C(=O)N2 c1(OC)cc(C(=O)NCc2ccc(CNC(=O)C(F)OC)cc2F)cc(C)c1 Cc1ccc(Cl)c(O)c1C(=O)N(C)CC1CCCC(NC(=O)C2=CC(C)(C)C2)C1 c1(C(N2CCC3CC(C2)CN(C(C2(Cl)CC2)=O)C3)=O)ccc2cnccc2n1 CC1(C)CCC(F)(F)CC1C(=O)NCC=CCNC(=O)C1=CCCC1 CON1CC(C(N2CCCC2C(=O)NC2CCCOC2)=O)CC1=O CC1(C)CN(C(=O)CCCn2cccn2)CC(CNC(=O)C=CC2CCOC2)O1 N1(C(Cc2ccc(C)cc2)=O)CCN(C(=O)C(C)n2ccnc2)C2CC12 N1(C(C2CC(=C)C2)=O)CCC(NC(=O)C=C(C)C(F)F)C(CC)C1 Cn1cc(C(=O)NCCCCCNC(=O)C(C)(C)C2CCC2)c(-c2nccs2)n1 C1(C(=O)NC2(C)CN(C(=O)C#CC(=O)N(C)C)C2)CCn2cnnc2C1 c1(C(=O)NCCN(C(=O)CC2CCC(C)(O)CC2)C)cc(=O)c2ccncc2o1 C(C(F)(C(=O)N1CCCC(C)(C#N)C1)C(C)C)NC(C(C(=O)OCC)OC)=O N1(C(CCc2n(C)c(S)nn2)=O)CC2CCN(C(C3(F)CCCOC3)=O)CC2C1 Cc1cc(=NC(=O)CN(Cc2ccccc2)Cc2cnc(C3CCC3)nc2)[nH]o1 c1(C(N(C)CC)=O)ccoc1CCC1(NC(=O)C(C)(C)OC(C)=O)CC1 CCC(C)C(=O)NCC1(NC(=O)CN2CCSCC2)CC(OC)C1 N1(C(CC(C)c2ccsc2)=O)CCCC(CO)(CNC(C2CN(S(N)(=O)=O)C2)=O)C1 O=C(C1=CC2(CCN(C(=O)CCOCC(F)F)C2)C1)NCC1CC(F)(CF)C1 C1(C(N2CC(OC)C(NC(C3CC4CCC3O4)=O)C2)=O)CC2(C1)CS(=O)(=O)C2 N1(C(C2(C#C)CCC2)=O)CCC2CCN(C(c3cccc([N+](=O)[O-])c3C)=O)C2C1 C1(C(=O)NCC(C)(C2CC2)NC(c2c(CC)occ2)=O)CCN(C)C1C N1(C2CCN(c3c(OC)cnc(SC)n3)CC2)C2CCC1CN(C)C(=O)C2 C1(C(=O)NC(C)CC(C)O)(COC)CN(C(=O)CCNC(N)=O)C1 c1(C(=O)NCC(C2CC2)NC(CCSC)=O)cc(C#N)c(F)cc1F CCC(C(=O)NCCOC1CCN(C(=O)Cn2ncnn2)C1)N(C)C C1(NC(c2c(-c3c(OC)cccc3)c[nH]c2)=O)C2CCC1N(C(=O)CN(C)C)C2 C1(NC(C2C(NC(C(C(C)C)=O)=O)CCC2)=O)CCCC2(CC1)CC2 CN1C2CCC1CC(=CC(=O)NC13CCC1CN(C(c1cccc(F)c1)=O)C3)C2 c1(C(C)=O)ccc(CN2CCC(C(N3CCC(OCCNC(C)=O)C3)=O)C2)cc1 CC1CC(C(N2CCC2(C)CCO)=O)CCN1C(c1csc(F)c1)=O C1(CNC(c2occ(C(N)=O)c2)=O)CCCCN(c2ccc(C#N)nc2)C1 N1(C(C2C(c3n(CC)ccn3)C2)=O)CCC2(CC1)CCN(C(C1CC(C)C1)=O)C2 C1(C(N(C2CCOC2)C)=O)C2CN(C(C3(C(F)(F)F)CCC3)=O)CC12 N1(C(C(C)SC(F)(F)F)=O)CCC(CNC(=O)CC2CCCC(C)C2)C12CCC2 C1(N(CC=C(C)C)C(=O)NC2(c3ccccc3)CC2(C)C)C(C)CCC1C c1(N2CC(NC(C(C)OCCC(C)C)=O)(CO)C2)ncc(I)cn1 C1(C(=O)NCc2n(CC)cnn2)CCN(C(c2snnc2C)=O)C1C C(=O)(CCCN=[N+]=[N-])N1C(CC(=O)NC(C=C)C2CCC2)CC1 CC(C)CCC(=O)NCCCC(C)NC(c1ccc(CC2CC2)s1)=O c1(C(N2CCC(OCCNC(c3ccc(CSC)o3)=O)C2)=O)cncc(O)c1Cl C1(CC#C)(C(N2CC(N=[N+]=[N-])C2)=O)CCN(C(=O)CC2CCCO2)C1 N12CCN(CC1)CCN(CC)C(CC)C2=O.C1(C(=O)NC)CC(n2cnnc2)C1 C12(NC(c3cnc(C(C)C)[nH]3)=O)CCCC1CN(C(C13CCC(CC1=O)C3)=O)C2 C(=O)(C#CC(C)(C)CNC(c1nc(O)sc1C)=O)N(CCSC)CC C1(CC(=O)NC(C)C(=O)N(C23CC(C2)C3)C)CCOC1=O CC(C)C(O)CC(=O)N1CC(NC(c2ncc[nH]c2=O)=O)CC(O)C1 C(=O)(C1CSc2ccccc21)N1CCC(O)(CN(C(CCC(=O)NC)=O)C)CC1 N1(C(C(C(C)C)C#N)=O)CCC(C2CC2)C1C(=O)Nc1ccc2nncn2c1 CC1CC2CN(C(=O)C(O)CC(F)(F)F)CC2N1C(=O)CN1CCC(=O)NC1=O c1(C(N2C(C(=O)Nc3c(OC)cc(O)cc3)CC2)=O)cc2cccn2cn1 C1(NC(Cc2n(C)nnc2)=O)CC2CC1CN(C(C13CCC(CC1)OC3)=O)C2 N1(C(CCC(C)OC)=O)CCC2(CC1)CN(C(C1CCCC(F)(F)C1)=O)C2 c1(C(=O)NCC(CC)NC(C2(C(=O)OCC)CCC2)=O)coc(CC)n1 c1(C(=O)NCCOC2CN(C(=O)Cn3cc(Cl)cn3)C2)cc(O)ccc1F c12cc(cc(C)c1)NC2.C1(NC(=O)NCc2ccn(CC)n2)(CC)CCCCC1 N1(C(c2nn(CC)c(O)c2)=O)CC2(CC2)CC1CC(=O)NCCCS(C)=O C1(NC(C2CN(C(CCOCC)=O)CC2C)=O)COCCN(C)C1 C1(N(C(CCOC(C)C)=O)C)CN(C(=O)CC2CCCN2C(C)C)CC12CC2 CC(C)C(C)CC(=O)NC1(CCNC(C2(F)CCCOC2)=O)CC1 N(C1CCOc2cc(F)cc(F)c21)C(N(CCC(C)C)C(C)C)=O CC(C(=O)N1CC(O)(CN(C)C(c2cc(C3CCCC3)[nH]n2)=O)C1)C(C)O c1(OC)cc(OC)nc(NC2CC2C(=O)Nc2ncc(Cl)nc2Br)n1 N1(C(C(CC=CCC)C)=O)CCC(CNC(c2nnsc2C)=O)C12CC2 N1(C(CC(CNC(COCC(=O)NC)=O)O)=O)CC(=O)NCC1C(N)=O c1(NC(C2CC(NC(c3ccsn3)=O)C2)=O)cc(Br)c([N+](=O)[O-])cn1 C1(CC)CC(c2nnnn2C2CC(F)(F)C2)(NC2CSC2)CCO1 C1(NC(C)=O)CC2(C1)CN(C(c1cccc(C(N)=O)c1F)=O)C2 N1(C(=O)CCOc2ccc(F)cc2)CCC2CN(C(=O)C3=CCCC3)C2C1 c1(C(C(=O)NC2CN(C(C(CC)SC)=O)C2)O)ccc(Br)cc1 CC(C)C1=NOC(C(N2CC(O)CC2C(=O)Nc2cnn(C(C)C)c2)=O)C1 N1(C(C=CC)=O)CC(NC(c2cnc(C)n2C)=O)CC2(CCC2)C1 N1(c2n(CC(=C)C)c(-c3cnn4cc[nH]c34)nn2)CCCC(C2CCC2)C1 C1(C(N2C(C)CN(C)CC2)=O)CCN(C(=O)C(C)N=[N+]=[N-])CC1(C)C C(=O)(C1=CC2CC=CCC12)NCCC1CC(NC(c2cc(C)c(Cl)c(N)c2)=O)C1 C1(NC(c2[nH]nc(OC)c2Cl)=O)CC2CC1CN2C(=O)CC(C)(C)C C1(NC(c2[nH]c3ncn(C)c3c2)=O)CCN(C(c2cc(Cl)no2)=O)CC12CCC2 C1(CNC(C(CC)F)=O)CN(C(=O)CSc2ccc(Cl)cc2)CC1C c1(C(=O)NCC(C2CCCC2)NC(C(C)(C)N(C)C)=O)cccc2c1CCN2 Cn1cc(-c2cccs2)cc(OC(=O)CC(=O)OC(C)(C)C)c1=O C=CCCCCC(=O)N1CCOC(CNC(C2CC(Oc3ccccc3)C2)=O)C1 CC(C)(CC(F)(F)F)C(=O)N1CCC(OCCNC(=O)CN2C(=O)CCC2=O)C1 CC(CC(=O)N(CCCOCCN(C(=O)C1=CCCSC1)C)C)C(F)(F)F c1(C(=O)NC2CCC(C(=O)NCc3occ(C)n3)CC2)ccn2nccc2c1 C(=O)(CC(C)(C)C(F)(F)F)NCCCN(C(=O)C(c1cccc(F)c1)(C)O)CC CC1=C(C(=O)NCC2CC3CN(C(=O)C(C)Cc4ccnn4C)CC23)CCCO1 c1(C(=O)NCCCC2(NC(CCCCC)=O)CC2)cc2n(n1)CCNC2=O C1(C)(C(N(CC)CC2CCCN2C(=O)CSc2nncs2)=O)CCCNC1=O Cn1c(CO)nc2cc(C(N3CCC4CC4(NC(=O)CC4CC4)CC3)=O)ccc12 c1(C2C(C(N(CCCNC(C(CC)(C)O)=O)C)=O)C2)c(Cl)cccc1Cl C(CC(C)C)(C(=O)NCC(CC(C)C)NC(c1coc(C2CCC2)n1)=O)OC C1(O)(CNC(C2(COC)CCC2)=O)CCCN(C(=O)CCn2ccc(C)n2)C1 c1(C(N2CC=CC(C(N(C3CCCOC3)CC)=O)C2)=O)cc2ccncc2[nH]1 Cc1nn(C)c2nc(O)cc(C(=O)NC(C)CC(C)NC(=O)CC3CC=CC3)c12 N1(C(C(C)C2CCCC2)=O)CC2(C(=O)NCCCC(C)(F)F)CC1CO2 N1(C(CC)=O)CCN(C(c2ccc(CC)nc2)=O)CC(O)C1 C(C(C)(COC)C(=O)NC1C=CCN(C(=O)C(O)Cc2ccccn2)C1)OC C1(N(C(=O)C(C2CCOCC2)O)C)CCCCN(C(=O)CN2CC3C=CC2C3)C1 C1(C(C(=O)NCC2CC(CNC(C3(CCOC)CCC3)=O)C2)C)CCC(=O)N1 C(C1CCc2cc(F)ccc21)NC(=O)C1CC1c1ccc(C(F)(F)F)cc1 C1(C(=O)NCC2C(CC(=O)NCC3(C)CC3)C2)CN2CCC1C2 N1(C(C2C(C)C2)=O)CC(CNC(c2cn(C(F)F)cn2)=O)CC1(C)C N1(C(C(C=C=C)C)=O)CCN(C(=O)CSc2nnnn2C)C(CC(F)(F)F)C1 FC(F)(F)C(C(F)(F)F)Sc1nc(C2CCC2)nn1-c1cncc(Br)c1 N1(C(C2CC(OC)C2)=O)CC=CC1(C)C(=O)NCCCC1CCCCO1 C(c1ccncc1)=CC(=O)NC1CC(CNC(c2nnc(C(F)(F)F)s2)=O)C1 C1(CCNC(COCCC#C)=O)CCN(C(c2ccnn2C(F)F)=O)C(C)C1 N1(C(CCN(CCC)C)=O)CCC(NC(c2[nH]cnc2C)=O)C1C N1(C(CC(CNC(=O)OC(C)(C)C)OC)=O)CC2CC1CS2=O.c12occc1N2 C12(CNC(Cc3cccc(OCC)c3)=O)CCCC1CCN2C(=O)CN(C)C N1(C(C23N(C(=O)Cc4ccco4)CCC2C3)=O)CCC([N+](=O)[O-])CC1 N1(C(c2c(N)nccn2)=O)CCCC(NC(c2nn[nH]c2Cl)=O)C(F)C1 C1(NC(CNCC(N2CCOCC2)(C)C)=O)CCN(CC(F)(F)F)CC1 C#Cc1ccnc(C(=O)NC(CNC(c2cc(=O)n(C)cn2)=O)C(C)(C)C)c1 c1(-c2cn(CCOCCNC(=O)C(=O)C3CCCC3)nn2)ccc(F)cn1 N1(C(=O)Cn2ncnn2)CCC2CN(C(C3(n4cccn4)CC3)=O)CC2C1 CCC(C)(F)C(=O)N1CCC(NC(=O)C(O)Cc2[nH]cnc2C)CC1 CCC(CC)(C(=O)NC1CC(C)N(C(=O)Cc2cnsc2)C1)OC N1(C(CN(C(=O)C(=O)O)C)=O)CCC12CCCOC2.c12cccc(c1)NC2=O Cc1ncc(N)cc1C(N1CC(O)(CNC(=O)C(C)Cc2cccc(F)c2)C1)=O N1(CC(C)C)CC2(CN(C(=O)CC(C)C3CC3)CCO2)C1 C1(NC(c2c(C)nc[nH]2)=O)CCN(C(c2cnn(C3CC3)c2Cl)=O)CC1(C)C C1(C(CNC(=O)CC2OCCO2)NC(CN(C)C(N)=O)=O)CCCCC1 C1(NC(NCc2cc(C)on2)=NCCCCl)CCn2c(C(F)(F)F)nnc2C1 C#Cc1ccnc(C(N2CC(NC(=O)CCc3ccc(F)cc3)CC2C)=O)c1 c1(NC(C(=O)NC(C)(C)C2CC2)=O)cnc(N2CCOCC2)ccc1=O N1(CCSc2scc(C)n2)CCOC(C)(CNC(=O)C(C)(C)C(F)F)C1 C1(NC(C(COC)O)=O)CCOCC1NC(C1(C(F)(F)F)CCCC1)=O CN=c1c(C(=O)NC(C)C(C)NC(=O)Cn2cncc2C)c[nH]c2ccccc12 C1(C(=O)NCC(CCC)OCC)C(C)OCCN1C(=O)C(C)N(C)C N1(C(C(C)OCCOC)=O)CCC2C(NC(=O)CCc3cnc[nH]3)CC12 c1(CC)ccc(CCC(=O)NCCN(C(=O)C(C)(C)C2CCCCO2)C)cc1 c1(N2C(CNC(c3c(CC)noc3)=O)CC3(CC3)C2)nc(O)c2ccccc2n1 C(c1ccc(O)cc1)=CC(=O)NC1CC(C(N2CCC(N(C)C)C2)=O)C1 C1(C(=O)NC(C)CC(C)NC(=O)CC2CCC2)(OC)CCOCC1 c1(C(=O)NCCC(CC)(C)NC(=O)CN(C)C2CC2)cccc(C)c1C N1(C(C(CC)(CO)OC)=O)CC2(CC(C(=O)NCc3cncc(F)c3)CO2)C1 N1(C(c2cncc(C)c2)=O)CCC2(CCN(c3cc(C)ncn3)C2)C1 CC(C)C(C(=O)NC1CCN(C(C2(C)CCCCC2)=O)C1)c1cccnc1 C1(CCC)CN(C(C2CC23CC3)=O)CCN1C(=O)CCCCCSC C1(C(=O)Nc2cccc(OCC)c2)CCc2nc(-c3cccc(C)c3O)sc2C1 c1(C(=O)NC(CC)CNC(=O)C(c2ccc(C)cc2)O)cc(C(N)=O)ccc1C N1(C(COCCC=C)=O)CCC(C2CC2)C1CNC(c1ccc[n+]([O-])c1)=O C(=O)(C1=NNC(=O)C1)N1CC2C(NC(c3ccc(C(=O)NC(C)C)cc3)=O)(C2)C1 C#CCCCC(=O)N(C1CCN(C(=O)C=C2CCCO2)CC1)CCOC Cc1n[nH]c(C)c1CCC(=O)NC1CN(C(=O)CC2CCC(=O)N2)CC1O c1(-c2cc(C(=O)OCC3CCCCC3)on2)cccc(Br)c1 c1(CNC2C(C(=O)Nc3c(Cl)cc(C)c(O)c3)C2)cccc2cnccc12 C1(NC(c2n(C)nc(CC)c2Cl)=O)CC2CCC1N(C(=O)CC(C)C(C)C)C2 S(=O)(=O)(c1cc(Br)c(F)cc1F)NCC1N(C(C2C(C(=O)O)C2)=O)CCOC1 c1(C(N(CCCCNC(C(C)NC(CC)=O)=O)C)=O)cccc([N+](=O)[O-])c1 N1(C(C(C)OCCOCC)=O)CCCN(C(=O)C=CC(C)(C)C)CC1C CCCCC(CC(=O)NC1CC(C(F)F)C1)NC(C12CCCN1CCC2)=O C(=O)(CCCCCNC(=O)Cc1n[nH]c(C)n1)N1C(CC)(CC)CC1 C(=O)(C(C)(C(C)C)NC(C)=O)NCC(C1CCN(C(C(CC)(C)O)=O)CC1)(C)C C(=O)(CS(=O)(=O)C(C)C)N1CCC(NC(CCn2ccc(C)n2)=O)C(F)C1 C1(CNC(C2(CC)CCN(C(=O)C(c3cnn(C)c3)C)C2)=O)CC2CCC(C1)C2 N1(C(c2c(CC)nnc(C)c2)=O)CCCCC2(CCN(C(=O)C(C)(C)SC)C2)C1 C(=O)(C(F)CCC(C)C)NCC1ON=C(C(=O)NCC2OCCN(CC)C2)C1 c1(C(N2CC=CC(c3ccccc3)C2)C(=O)NC2CCC2)cc(F)ccn1 c1(N2CCC(C)C(NC(c3c(C)onc3)=O)C2C)ncc2ncn(C)c2n1 c1(C(=O)NCCCN(C)C(C2CSCCS2)=O)ccc(C2CCC2(C)C)cc1 Cc1ncccc1NC(C1CSCCN1Cc1cncc(-c2ccccc2)c1)=O C1(NC(CC=CC(C)(C)C)=O)CCCC(C(=O)NC2(CC(C)(C)C)CC2)C1 c1(C(=O)NCC2(F)CCC(NC(C(C)=CC)=O)C2)cc(=NS(C)(=O)=O)cc[nH]1 c1(OCC(=O)NC2C(CCC)CCC2)cncc(C)n1.N12CC(C1)OCC2=O C1(C2CCOCC2)(C(=O)NC(CNC(c2c(Cl)ccc(C)c2)=O)C)CC1(F)F C1(C(=O)NCCSCCC=C)CCC(O)CN1C(c1ccn(C)c1CC)=O N(C1CCCc2ccc(Br)cc21)CC(C)(C)C N1(C(C2CC3(CC3)C2)=O)CCC(CO)(CC2CCCNC2)CC1 c1(C(N2C(CNC(c3cn(CC)nc3)=O)CC(O)C2)=O)cc(F)cc([N+](=O)[O-])c1 c1(CNC(=NCC=C)NC(CC)C(F)F)ccc2c(n1)CCCC2 CCC(C)C(O)C(=O)N1CCCC(C)(NC(c2nc(=O)n(C)[nH]2)=O)C1 c1(C(C(F)(F)F)NC(=O)C(N2CCCC2CN2CCCC2)=O)ccc(Br)cn1 C1(C(=O)NC2CC(CNC(C3C(C=C)OCC3)=O)C2)C(C)(C)CCCC1(C)C CC1CN(C(=O)C(CN(C)C)NC(=O)C(C)n2ccnn2)C(C)C1C N1(C(C2(SC)CC2)=O)CCC2CN(C(=O)CC3CNC(=O)O3)CCC2C1 C1(NC(C(C)c2ccsc2)=O)CCC(O)CN(C(=O)CP(C)(C)=O)C1 C(CC(=O)NC1CCC(NC(=O)CCC#N)C1)(C(F)(F)F)N(C)C1CC1 N1(C(CC(CC)(C)C)=O)CC2(CNC(c3ncsc3NC)=O)CCC1CC2 C1(C(=O)NC2CCN(C(c3ccn(CC)n3)=O)C2C2CC2)CS(=O)(=O)CC12CC2 C1(NC(c2cnco2)=O)CC(C(=O)NCC2(CO)CC23CCC3)=CC1O C1(CC(N2CC(CNC(C3C(C)C3)=O)N(C)CC2)=O)CC(C)CC(C)(C)C1 c1(N(C)CC2CCN(C(C(C)OCCCCCC)=O)C2)cc(C)ncc1C#N N1(C(Cc2nccc(OCCC)n2)=O)CC(C)CN(C(=O)C=C(C)Cl)C(C)C1 c1(C(=O)NC(C(C)C)CNC(=O)CC2CCN(C)CC2)cc(C#N)c(N)cc1O N=c1[nH]c(=NCc2ccc3c(c2)OC(F)(F)O3)[nH]c(=NC2C=CCCCC2)[nH]1 Cc1cc(N)c(C(N2CCCCC2CCNC(C2(C)CCCO2)=O)=O)cc1C c1(CC(=O)NCC(C)(O)CNC(c2cnoc2-c2ccoc2)=O)cnc(O)nc1O CC1(C)CN(C(C2CC3(C2)CC(F)C3)=O)CC(CNC(c2cnccn2)=O)O1 C1(CC(=O)N(C2CCCN(C(Cn3c(C)nnn3)=O)C2)C2CC2)CCCCC1(C)C C1(CCCNC(c2c(C)coc2)=O)CN(C(=O)Cn2ccnc2C(C)C)CCO1 C1(C)(CNC(C(CCOC)(C)C)=O)COCCN(C(C2(C)C=CCCC2)=O)C1 N1(C(c2c(C)[nH]nc2CO)=O)CCOCC(C(=O)NCC2CC23CC3(F)F)C1 N1(C(C2CCC(=O)C2)=O)CCC(C2(NC(C3(Cc4cccnc4)CC3)=O)CC2)C1 c1(CSCCC)ccc(C(N2CC(C(C)N(C(c3cnc(S)[nH]3)=O)CC)C2)=O)o1 C1(C(=O)NCC2(O)CN(C(c3nn(C)c(F)c3)=O)C2)CC2OC(=O)OC2C1 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)N1CCC(CNC(C(C)(C)OCC)=O)C(C)C1 C1(CC(=O)NC(C(=O)NC(C=C)(C)CC)CSCC)CCCC12CC2 C=CC(CC)CC(=O)NCCC1(O)CCN(C(c2cnc(OC)c(C)c2)=O)C1 N1(N2CCC(n3cc(CC(c4cc(CC)[nH]n4)=O)nn3)C2)C(C)CCCC1C C1(C2CCN(C(=O)CNC(=O)NC3CC3)C2)(NC(=O)CC2COC(=O)C2)CC1 c1(NC(C=CC(C)NC(=O)C2=CCN(C)C2)=O)cnn2ccccc12 C=CCC(C)(C(=O)N1CC(C)(C)CC1CNC(c1ccncn1)=O)N(C)C C1(=CC(=O)NCCC2COCCN2C(c2ncccc2F)=O)CN2CCC1CC2 c1(C(N2C3C(NC(C(NOC)=O)=O)CC(C3)C2)=O)ccc2n[nH]cc2n1 C(CC(C)C)(C(=O)NCC1(COC)CCC1)ONC(C(C)NC(CC)=O)=O c1(C(CSC)NCC(C)CCc2ccccc2)cccc(C)c1 C(=O)(CCCCC(C)C)N1C(CCCNC(CCSCCC)=O)CCC1 C1(CNC(C(C=CC)O)=O)CC2(CO1)CN(C(C1CSC1)=O)C2 N1(C(C2CC(N(C)C)C2)=O)CCC2(CCC(NC(C3CSCC(=O)N3)=O)C2)CC1 C(=O)(CCCS(N)(=O)=O)NC1CCN(C(c2ccc(C)nc2)=O)CC1C N1(C(c2nnc(C)s2)C)CCC(C)(NC(=O)CC2CC=CC2)C1 Cc1cc(C(=O)COC(=O)C(C)(C)C2CCCC2O)cnc1Br N1(C(=O)Nc2nccc(-c3ccc(Cl)cc3)n2)CCCC2(CCNC2=O)C1 Cc1ccc2[nH]c(C(=O)Nc3cccc(Cn4nc(C)cc4C)c3)c(Cl)c2c1 Cc1cc(=O)oc2ccc(OCC(=O)NCC(O)CCNC(=O)CN(C)C)cc12 c1(CN(C(=O)Cn2ncnn2)C)csc(CNC(c2cnn(C)c2)=O)n1 Cc1cc(=NCc2nc3ccccn3c2Cl)[nH]c(N2CCC3(CC2)CSC3)n1 C1(C(N(CCCNC(CCC=C(C)C)=O)C2CC2)=O)CC1C1CCCC1 c1(C(=O)NC2C(NC(=O)CCc3ccon3)CC2)ccccc1OC(F)F c1(C(=O)NCCC(O)C(=O)N2CC(N3CC(F)C3)C2)ccn2nccc2c1 N1(C(C)=O)CCCC1C(=O)N(C1CCN(C(=O)CSc2ccccn2)C1)C c1(OC)c(C(N2CCCCC2c2cccs2)C(=O)NCCC2CC2)cccc1F N1(C(C=CCOC)=O)CC(CO)C2(CCN(C(=O)C(C)(C)CC3CC3)CC2)C1 N1(C(COCP(C)(C)=O)=O)CCC(NC(=O)CCc2cccs2)C(O)C1 Cc1c(C(=O)NCC2N(C(c3ccc[nH]3)=O)CCC2(C)C)c[nH]c1C#N c1(C(N2CC(F)(C(=O)NC(CN(CCCC)C)C)C2)=O)cncc(CC)c1 C1(C(=O)NC(C)(C)CNC(=O)C(c2cccc(Cl)c2)(C)C)CC1C1CCCC1 C1(N(C(CC(OCC)OCC)=O)C)CCCN(C(=O)C(C)(C)C)CC1 c1(C(=O)NC2C(CNC(CNC(=O)NC)=O)CCC2)cnn(C(C)C)c1Br C1(OC)CN(C(c2ccns2)=O)CCC1NC(=O)CN1CC2CC2C1 S(=O)(=O)(c1cc(F)c(F)c(F)c1)NC1CC(C(=O)Nc2cnc(C#N)c(Cl)c2)C1 n1(CC(=O)NCC(C2CC2)NC(=O)CC2CC2(Cl)Cl)nnc(-c2cccs2)n1 C1(C(=O)NC(C2CCCN2C(c2cc[nH]n2)=O)C)(COC)CCOCC1 c1(C(C(=O)NC2CC2)N(C)CCOCCO)cccc(C2CCCC2)c1 c1(OC)cc(N2CC(O)(CO)C2)nc(C(F)(F)F)n1.C12CCC(CC1)C(=O)NC2 C1(C(N2C(CC(C)C)CC2)=O)N(C(C2CCC(=O)CC2)=O)CC12CCCC2 C1(C(=O)NC(c2ccc(F)cc2)CNC(CCCOC(C)=O)=O)CCCC1(C)C N1(C(C(COCC)NC(c2cncnc2C)=O)=O)CC(N(C)C)C2(CCC2)C1 CCCCC(CCC)NC(=O)CC(C)(C)NC(C1CC(F)C1)=O C12(CNC(C(C=C)O)=O)CCCCC1N(c1ncc([N+](=O)[O-])cc1Cl)CC2 N1(C(=O)C=CCN2CCOCC2)CCC2CC(C1)CN(C(=O)C(O)C1CCCC1)C2 c1(C(=O)NC(C)C)c(C(=O)NCCN(CCOC)C(C2CC2F)=O)cnn1C C(C(C)(C)C(=O)NC1CC(CC(=O)Nc2cnc(SC)nc2)C1)N(C)C N1(C(c2ccsc2C)C(=O)NC(c2ccc(F)cc2)C)CCC(C(F)(F)F)C1(C)C CC1(C)CC(CC(=O)NCCC2CCCC23CC3)CN1C(=O)Cn1cnc(=N)[nH]1 C12(C(=O)NCc3nc(C4CCCOC4)n[nH]3)CCCCN1CCC2 Cc1cc(C(N2CCCC(O)(CNC(=O)CN3CC=CC3)C2)=O)c(C)cn1 c1(C(N2CCC(C)(NC(C3CN(CCC)C(=O)C3)=O)C2)=O)ncc(C)cc1OC c1(C(=O)NCC2N(C(CC3(C)CCCO3)=O)CCC2)ccc(Br)cc1F C1(NC(C(c2cnn(C)c2)C)=O)CCCCCC1NC(c1cnc(O)n1C)=O C1(CNC(C(C=CC)O)=O)CN(C(=O)Cn2cc(C#N)cn2)CCC1C Cc1c(C(=O)NC2CC(CC(=O)NC34CCC(CC3)C4)C2(C)C)ncn1C C12(NC(c3ccc(-n4cccc4)cc3)=O)CC1CN(C(=O)Cn1cc(Cl)cn1)C2 Cc1cnc(NC(CC2CCOC2)CO)c(S(=O)(=O)NCCc2ccnc(Cl)c2)c1 c1(C(=O)NC2CCCN(C(=O)C(F)OC(F)(F)F)C2)ccc2ccccc2c1F C1(C)(CC(N2CCC(OCC(N3C(CC)(CC)CC3)=O)C2)=O)CCOCC1 Cc1nc2sccn2c1C(=O)N(C(C)CNC(C1(Oc2cnn(C)c2)CC1)=O)C c1(C(C(=O)Nc2cccc(OC)c2)N(C)Cc2cccs2)cc(S(N)(=O)=O)co1 c1(NC2N(CC)CCC2)cc(=NCCCOCCOC)[nH]c(CC)n1 C1(C(=O)NCCc2onc(CC)n2)CCC(C(C)C)N1C(c1cccc(F)c1)=O N1(C(C2C(C)OCCC2)=O)CCC(NC(c2ccc(CO)c(F)c2)=O)CC1C N1(C(C(=O)NC)C2CC(NC(=O)OC(C)(C)C)C2)CCCC1C(C)(C)CO C1(NC(C(C)N2CCC2)=O)CCCCCC1n1cc(CC(C)(C)O)nn1 c1(OC)c[nH]c(C(=O)N(CCC(C)NC(=O)CC2CC=CC2)C)cc1=O C1(c2cn(CC3(O)CCN(C(CC)=O)C3)nn2)CC2(C1)OCCO2 C(=O)(C1=NOC2(CCC2)C1)NC1(CC=C)CN(C(=O)CC2CCCN(C)C2)C1 c1(C(=O)NC2CCN(C(c3ncccc3F)=O)C2)cc([N+](=O)[O-])c(O)cc1F C1(NC(c2c(C)n[nH]c2)=O)CCN(C(=O)CC(=O)OC(C)(C)C)CC1F c1(CCCC)ccc(NC(c2cnn(C(C)C)c2C)=O)cc1 Cc1onc(C(N2CCC23CN(C(C2CCC(=O)N2C)=O)C3)=O)c1[N+](=O)[O-] CC(C(=O)NC1COC2(C1)CN(C(c1cc(N)ccn1)=O)C2)C1=CCCC1 N1(Cc2ccc(-c3nc(C)c(C)s3)cc2)CC(C)(C)OCC1C N1(c2ncc(OC)cn2)CCN(C(c2cc(Br)cnc2Cl)=O)CC12CC2 N1(C(COCCOCC)=O)C2CCC1CC(O)(CNC(c1cc(C)ns1)=O)C2 c1(CC)cn2c(n1)CCC(C(=O)NCC1CC(F)(F)CN1C(C1CC1C)=O)C2 N1(C(C2CC2F)=O)CC2CCC(C1)N2Cc1ccc(Br)nc1Br c1(C(N2C(CCC)(C(=O)NC)CCC2)=O)cc2c(F)c(F)cc(F)c2[nH]1 c1(C(=O)NCC2OCC(CNC(=O)CC3CC3)C2)ccc2ncnn2c1 c1(C(N2C(CN(C(C(C3CCCOC3)OC)=O)C)CCC2)=O)cnc(N)cn1 c1(CC(N2CCC(N(C(C(C(C)C)C)=O)C)CC2)=O)cc(Cl)cc2ccccc12 C1(CC)CCN(C(=O)CCOCC(C)(C)C)C1C(=O)NCc1cnn(CC)c1C c1(NCC(CNC(=O)CC2CCC(F)(F)C2)O)ccccc1[N+](=O)[O-] c1(NC(=O)NC2C(C)C2C)cccc(Oc2ccccc2)c1.C(CN(C)C)O C1(CC(N2C(c3cn(-c4ccc(C)nc4)nn3)CC3CC32)=O)CCC(C)(O)CC1 N1(CCC)CCCN(C(C2COCCC2NC(=O)C(F)(F)CC)=O)CC1 c1(N2CCC(C)(CSC)CC2)nc(NC2CC2Cl)c2c(n1)c(C)nn2C C1(NC(C(C)SC)=O)CCN(C(c2[nH]ccc2C2CC2)=O)C1 C1(NC(c2ccns2)=O)CN(C(C2CCCOC2)=O)CC2(CC2)C1 C1(C(=O)NC2CN(C(c3c(OC)n[nH]c3)=O)C(C)(C)C2)CC(C)(C)OC1(C)C c1(SC)cccc(C(=O)NC2CCOCC2NC(=O)C(C)(C)C(N)=O)c1[N+](=O)[O-] c1(CC(C)(C)CNCC2COCCO2)ccc(C(F)(F)F)cc1 N1(Cc2nc(Cl)sc2)CCC2CCCC(C2)C1 N1(c2n(C)c(CC(c3ccccc3)(C)O)nn2)CCc2c(cnn(C)c2=O)C1 CC1(C)CN(C(=O)NCC2CCCC3(CC3)C2)C(C)(C)C1 N#Cc1cc(C(N2CC(CCn3cc(C4CCCCO4)nn3)C2)=O)ccc1F CS(C)(=O)=NCC(=O)N1CCN(C(c2cc(C3CC3)nc(O)c2)=O)C2CC12 CC1(C)CC(NC(=O)C2=CSCCO2)CCN(C(C2CCn3cnnc3C2)=O)C1 c1(SCC)ccccc1N(C)C(C1CN(C(=O)C(C)NC(=O)C2CC2)CC1F)=O c1(C(C)(F)F)ccccc1C(N1CCN(C(=O)CC2CCC3CC23)CC1)=O N1(C(CCC(C)C)=O)C2CC1CN(C(=O)CNC(=O)COc1ccccc1)C2 N1(C(C(CCC)OC)=O)CCN(C(=O)COc2ccon2)CC(O)C1 N1(C(C(C(C)C)C2CCC2)=O)CCC(C)N(C(C2CN(C3CCOC3)C2)=O)CC1 CCCCC(C)C(=O)N(C(C)CNC(=O)CC(C)N(C)C)C(C)C c1(C(N2CC(C)C(CNC(C3(O)CC3)=O)CC2)=O)nc[nH]c2nccc1-2 N1(C(C(CC)F)=O)CCCC(C)(C)C1CNC(=O)CCN1CCCCC1=O C(=O)(C(C)SC(F)(F)F)NC(CNC(=O)C1CC1)C1CCC1 N1(C(CC2(C)CCOCC2)=O)CCC2(CC1)CC2CNC(=O)C(F)(F)C(F)(F)F c1(C(=O)NCC2(CNC(CCN(C)CC)=O)CCCC2)cccc(C(C)C)c1N O=C(C1CCCc2n[nH]cc21)NC1CN(C(c2coc(Br)n2)=O)C2CCCCC12 S(=O)(=O)(c1ccc(NCCCC2CCOC2)cc1Cl)N1CCC(CCC)(CO)C1 CC1(NC(c2ccccc2)=O)CCN(C(=O)CC2(O)COC(C)(C)C2)CC1 N1(C(c2c(F)cc(OC)cc2Cl)=O)CCc2[nH]nc(CNC(=O)C(C)(C)F)c2C1 C1(CNC(C=CCOC)=O)CC2(CCOCC2)CN1C(c1cc(O)nc(C)n1)=O C(=O)(C(CC(C)C)ONC(C1CC(=O)NC1(C)C)=O)NC(CCC)CO c1(CC)nnc(C)cc1C(=O)NC(c1ccccc1)CNC(C1CC(C)(O)C1)=O c1(SC)ccc(O)c(C(=O)N(C)CC2CN(C(C3CCCC3O)=O)CC23CC3)c1 C1(NC(C(CC)N(C)C)=O)CN(C(=O)C(O)CCC(F)(F)F)CCC12CCC2 CCC(N)CCC(=O)N1CCCC(C(=O)N(C)Cc2occc2CC(=O)O)C1 Cc1cc(C)c(C(=O)NCC(C)CNC(c2cn(C(C)(C)C)nc2C)=O)[nH]1 C(=O)(C(C)CC(F)(F)F)N1CCC(C#C)(C(=O)Nc2ccccc2OC)C1 C1(O)(CN(C(CCCSC)=O)C)CCN(C(c2cnoc2-c2ccoc2)=O)CC1 C1(CS(=O)(=O)N(C(C2OCCCO2)CC)CC)CN(C(=O)OC(C)(C)C)CCO1 C(=O)(C1NCc2n[nH]cc21)NC(CC(=O)OC)c1ccccc1 C12(NC(c3ccnc(CO)c3)=O)CCCC1CN(C(c1ccc(F)c(F)c1)=O)C2 C1(C(=O)NC(CCC)C(=O)NC(COC)CCOC)CCCCC1(C)C CN1CCCC(C(C)(C)C(N2CCC(F)(CF)C2)=O)C1.C12=CC(COC)(CC1)C2 c1(OC)ccc(C)nc1C(=O)NC1(CO)CN(C(c2cc(CO)[nH]n2)=O)C1 N1(C(c2ncc(OC)cn2)C(=O)Nc2ccccc2)CCC(C)(O)CC1 Cc1nc(N)cnc1C(=O)N(CCNC(=O)C=Cc1ccc(Cl)cc1)C1CC1 C1(N(C)C(c2cc[nH]c2)=O)CCCC2CN(C(C3(n4cnnn4)CC3)=O)CC12 C1(NC(c2nc(-c3cccnc3)cs2)=O)CCNCC1CO N1(C(CC(CNC(C2CC(OC(C)C)C2)=O)OC)=O)CC2CC(O)CC1C2 c1(CNC(C2C3CN(c4c(OC)c(C)ncn4)CC32)=O)ccc2oc(C)nc2c1 CC(CC(=O)NC1CCC(N(C(=O)CCC2(C)N=N2)C)CC1)C(F)(F)F N1(C(CC=CC)=O)CCC2(CO)CN(C(=O)CSc3ccc(O)cc3)CC2C1 c1(C(CNC(=NC)N(C)CC2CCCC(C)(C)C2)OC)ccc(F)c(F)c1 c1(C(N2CCCC(C)C2CCNC(C2(O)CCC2)=O)=O)noc2cc(F)ccc12 C1(C#N)(C(=O)NCC(CNC(CC(C)OC)=O)OC)CC(=O)C1 c1(N2C(CC#N)CN(Cc3cc(I)ccc3O)CC2)ncc2cc(Br)cnc2n1 C(=O)(C1=CC2CCCC12)NC1CCCN(C(c2ccc(=NC)[nH]c2)=O)C1C Cc1ccc(C(=O)NC2(CF)CN(C(c3cc(C(F)F)nn3C)=O)C2)nc1C CCCC(C(O)C(=O)NCC(C)(C)CO)NC(C1(C)CCOCC1)=O N1(C(=O)Nc2c(CC)nco2)CCC(Cc2ccnn2C)CC1 C(C(C)(C)CC(=O)O)NC(c1cnn(C(C)C)c1N)=O C12(NC(c3ccnnc3O)=O)CCCC1N(C(=O)C=CSc1nc[nH]n1)CCC2 C(=O)(C1=CS(=O)(=O)CCC1)N1C2CC(NC(=O)C=CCN3CCCC3)CC1CC2 N1(C(C(CCOC)(C)C)=O)CCN(C(=O)C(C(C)C)Nc2ccccc2)CC12CC2 N1(C(C2N(CC)CC2)=O)CCC2(CCCC2NC(C2CCCC3CC23)=O)CC1 C1(CNC(CSCC#C)=O)N(C(C2CCC(=O)N2CCC)=O)CCC1(C)C C1(C(N(C2CCN(C(C=CC(C)(C)SC)=O)CC2)C)=O)Cc2nccn2C1 CC(CNC(C1CN(CC(F)(F)F)C1)=O)CN(C(=O)CCc1cn[nH]c1)C CN1C(=O)C(=O)N(CC(=O)NCc2ccnc(N3CCNCC3)n2)C1=O C1(C(N(C2CCSC2)C)=O)(CNC(C2CCC2)=O)CC2(CC2)C1 N1(S(CC=C)(=O)=O)C(C(=O)Nc2ccnc(C3CC3)n2)CCC1C c1(C(=O)NCC(C2CCN(C(CS(CC)=O)=O)CC2)(C)C)ccnc(F)c1F C(CCCCCNC(=O)CCc1cnn(C)c1)NC(C1C(CC)CCC1)=O c1(N(C2CCCCCC2NC(=O)CC#N)C(C(F)OC)=O)cccc2cccnc12 C1(CNC(CC(C)OC)=O)CC2(CO1)CN(C(=O)C(C)(F)c1ccon1)C2 Nc1nc2c(cc1C(N1CC3CCC(C1)N3C(C1CCCCO1)=O)=O)CCCC2 N1(C(C2(CC)CC2)=O)CCC2CCCN(C(c3c[nH]c(=O)c4ccnn34)=O)C2C1 N1(C(C(C)=CC2CC2)=O)CCC(CC(C)N(CC(=O)NC2(C)CCOC2)C)CC1 c1(CC(=O)NCC=CCNC(C2CCC(=O)NC2)=O)c[nH]c2ccccc12 Cc1ccc(O)c(C(=O)NC(c2ccnn2C)C(=O)NC(CO)C(C)C)c1 C1(CN(C)C(C2CCCN2C(=O)CCc2cnccn2)=O)CCCC2CC12 C(C(C)(C)CC1CN(C(c2nocc2C)=O)C1)NC(C(=O)NCCOC)=O N1(C(c2ncc(CC)s2)C(=O)NC2CCC2)CCOCC(C2CCC2)C1 C(C(C)(C)CNC(=O)CC1CC1(Cl)Cl)N(C(=O)Cn1ccc(C(F)F)n1)C NS(=O)(=O)CCCCCC(=O)N1CC(NC(c2cnco2)=O)CC(O)C1 c1(NC(CNC(c2cnc(C(C)O)s2)=O)C2CC2)nc2c(cc1C#N)COCC2 N1(C(c2cc(OC)nn2C)=O)CC(C2(NC(=O)Cn3cc(C(C)O)nn3)CC2)C1 c1(CC)c(C(=O)NCCN(C2CCCC2)C(=O)CC2CCCC2(F)F)ccn1C CC1CCC(CC(=O)NC2(CF)CCN(C(=O)COCCN(C)C)C2)CC1 N1(C(CC2(C)CCCO2)=O)CCC(C2(NC(=O)C(F)=CCCF)CC2)CC1 c1(OC)cc(OC)c(C(=O)NCC(C)N(C(=O)C(C2CC2)OC)C)c(OC)c1 N#CC1(O)CC(C(=O)NC2CCCN(C(=O)Cc3cscn3)C2)C1 C1(CC(=O)N(CC(C)C)C)CC2(CC2)C1.C12CC(C1)CO2.C1C(=O)N1 CCCCC(CNC(C1CC1C)=O)NC(c1ccoc1C(C)C)=O Cc1c(C(=O)N(CC(C)(C)NC(=O)CC(C)C(F)F)C)cc(C(C)C)n1C c1(NCc2ccc(CC)o2)cc(=NCc2ccc(C)cn2)[nH]cn1 N1(C(C2(NC(C)=O)CC2)=O)CC(C(=O)NCCOCC(F)F)C1 Cc1onc(Br)c1C(=O)N(CCC(C)NC(C1CC1F)=O)C N1(C(c2c(CC)nns2)=O)CCCN(C(c2ccc(C)cc2)=O)C(CO)C1 N1(OCCC)CC2CC1CN2C(=O)CNC(c1ccco1)=O C(C(=O)NCCCCc1ncc[nH]1)(C1CCCO1)NC(C1CC(CF)C1)=O N#Cc1ccc(C(N2CC3CC2C3NC(=O)CCN2CCCCC2=O)=O)c(O)n1 C(=O)(C#CC1CCCCO1)NCC1C(NC(c2ncc(C)cc2F)=O)CC1 C(=O)(C(O)C(F)F)N(CCN(C(c1cccc(Br)c1)=O)CC)CC CC(C)(O)C#CC(=O)NC(CNC(=O)C(C)(C)CC1CCOC1)CO N1(C(c2cncc(C)c2)=O)CCCC(C)C1CNC(c1cn(C)nc1Br)=O C1(NC(c2n(CC)nnc2)=O)(CC)CCN(C(=O)Cc2ccc(C)cc2)CC1 C1(CNC(COCC(=C)C)=O)CC(C)CN(C(=O)C(C)(C)CSC)C1 CC(C)C(C(=O)NOCC(F)(F)F)NC(=O)CCCCC1CC1 N1(C(CC(C(C)C)O)=O)CCC2(CC1)CN(C(c1cccc(N)c1)=O)CCO2 CC1(C)CN(C(=O)C=Cc2cc[nH]n2)C(CNC(=O)CNC(=O)C(F)(F)F)CO1 C1(C(N(CCOCCNC(=O)C(CN(C)C)NC(C)=O)CC)=O)CCCNS1(=O)=O N#Cc1cc(Br)ccc1C(=O)NC1CCN(C(C23CC(CO2)C3)=O)C1 C(=O)(CC(C)(C)CC(=O)N1CCC2C1CCCN2C(=O)Cn1nnnc1C)OC N1(C(c2cnc(CC)[nH]2)=O)CCC2CCN(C(=O)Cn3ccc([N+](=O)[O-])n3)C2C1 n1(CCSCCOCC=C)ncc(C#N)c1N C(N=c1[nH]c2c(c(=NC(C)C3CCOCC3)[nH]1)COCC2)C1(C(C(C)C)O)CC1 c1(COC)nc(C)c(C(=O)NCC(C)(C)NC(c2nc(Cl)c(Cl)s2)=O)s1 N1(C(C(C(C)C)O)=O)C2CCC1CN(C(c1cccc(C(C)(C)C#N)c1)=O)C2 C#CC(C)(C)C(=O)NCC(C1CC1)N(C(=O)C(C1CCOCC1)F)C C1(N(C(=O)Cc2cnns2)C)CCN(C(=O)C(c2ccccc2)O)CC1 CC(C)(C)C(C(=O)N1CCC(F)(CO)C1)NC(c1ccncc1O)=O C(=O)(C(C)(F)C(C)(C)F)N1CCN(C(CCCCC)=O)C(CC(=O)NC)C1 C1(C(N2CCC(C)(NC(=O)C(=O)N=S(C)(C)=O)C2)=O)CCCN(S(N)(=O)=O)C1 c1(C(=O)NC(C)CCCNC(C2(c3cccnc3)CCC2)=O)ccncc1F O=C1CCCc2nc(N3CCCC4(NC(=O)Cc5cc[nH]n5)CC4C3)ccc21 CC1CN(C(=O)CCCNC(C2CC=CCC2)=O)CC1NC(=O)CCC1CCC1 n1(CCCNC(C(N)CC2CCS(=O)(=O)C2)=O)c(=O)oc2ccccc12 C1(NC(C(CC)SC)=O)CN(C(=O)CCN(C)C(=O)OC(C)(C)C)CCS1 C1(C(=O)NC(C)CCN(C)C(c2cncc(N)c2)=O)CCS(=O)(=O)C1(C)C c1(C(N(CC(C)NC(=O)C(C)(c2ccccc2)N(C)C)C)=O)cncn1C C(C)(CCCCNC(=O)Cc1cn(C)nc1C)NC(COCCC)=O CC1C(NC(=O)C(C)(C)CC(F)F)C2CCN1CC2 N1(C(CN(CC)CC)=O)CC(CC(=O)N(C)CC2CN(C)C2)C(C)C1 C1(CNC(=O)C2=CCCCCC2)CN(c2ccncc2Cl)CCC12CCOC2 O=C(CC1C2CN(C(=O)CCN=[N+]=[N-])CC12)N1Cc2ccccc2CO1 CC(C)C(C#N)C(=O)NC1C=CC(C(=O)NCCc2cc[nH]n2)C1 C(=O)(C(C)C(C)COC)NCc1c(C(N(CC(=C)C)CC(=C)C)=O)cccn1 CCC(C)C(C)C(=O)N1CCC(C)(CNC(c2cc(Cl)ccc2N)=O)CC1 C1(N)CC2CC(C1)N(C(=O)C=CC=C(Cl)Cl)C2.CCCCCC=CCC=O c1(SC2CCN(c3nc(Cl)ncc3F)C2)ccc(F)c(F)c1.C(CCO)N1C(=O)N1 CCC(CCC(C)C)N1CCCC(C(=O)NCC2CCC(=O)N2C)C1 Cc1ccc(CCC(=O)NC23CC2CN(C(=O)Cc2cccnc2O)C3)cc1 O=C(C1CCCc2nnnn21)NC1CCOCC1NC(C1(C2CC2)CC1)=O C(=O)(C(C(C)(C)C)OC(C1(c2cc(OC)cc(F)c2)CCCC1)=O)OC C(CC(C)C(=O)N1CSCC1C(N1CCC(C(F)F)C1)=O)=CCC CN1C(=O)CCCC1C(=O)NC1CCCC1CNC(c1csc(O)n1)=O c1(CNC(c2cnsn2)=O)ccc2c(c1)CCCC2NC(c1cccnc1O)=O c1(C(N(C2CCN(C(c3cccc(CO)n3)=O)C2)C)=O)ccc(C#N)c(Cl)c1 C1(C)(C(=O)NCCC(C)N(C(c2cnc(OC)nc2)=O)C)CCCNC1=O C(C(C(C)C)NC(=O)C(F)(F)c1cnn(C)c1)NC(C1C(CCC)C1)=O C1(CCOC)COCCN1C(C1(Cc2ccccc2)CCCN1)=O C1(NC(c2c(C)cco2)=O)CCCCC1NC(=O)C(=O)N(C)C c1(CC(=O)NCc2cccc(NC(=O)C(Cl)=CCl)c2)ncc(F)cc1F CC1(C)CC(CO)CN(CC(=O)Nc2cnc(Cl)c(F)c2)C1 C1(CNC(c2c[nH]nc2Cl)=O)CC2(CC2)CN1C(C1CC2CC2C1)=O CCC(CNC(C1CCN(C2CC2)CC1)=O)(CC)NC(c1ccsn1)=O C1(F)(CNC(C=NOC)=O)CCN(C(=O)C(C)(C)CSC)C1 CCC(CC)(CO)C(=O)NCC(F)CNC(=O)CC1(C)CC1(Cl)Cl N1(C(c2c(CCC)n(CC)nn2)=O)CCCN(C(=O)C=CC2CCOC2)CC1 C1(C(N(CC(=O)NOCCCOC(C)C)CC)=O)CCOC(C)C1 C=CCC(C(=O)N1CCCCCCC1C(=O)NCC1(O)CC1)C(C)C C(=O)(C#CC(C)(C)C)N(C)CC1CCN(C(c2cncc(NC)n2)=O)C1 Cc1cc(=NCC(C)N(C(=O)C(C)c2ccco2)C)[nH]c(C(C)(C)C)n1 C(C)(C)(C(=O)NCCC(C1CCC1)NC(c1cn(CC(=O)N(C)C)nn1)=O)OC c1(CNC(C(=O)Nc2ccc(C)c(Cl)c2F)=O)sc(Br)c2c1OCCO2 n1(CCC=C)cc(C2CCCN2C(=O)CC2CCC2)nn1 C1(OC)CC(CNC(=O)C(C(C)C)c2cc(C)no2)N(C(=O)Cc2ccsc2)C1 c1(C(=O)NCCCCCCCn2cc(CC=C)nn2)ccc(S(C)(=O)=O)c(C)c1 c1(C(=O)NC(CC(C)C)CNC(c2cccc(O)c2)=O)coc2c1C(=O)NCC2 N1(C(=O)NOCC2CCOC2)CC(O)C(O)C1 C1(C(N(C)CC2CCN(C)C2)=O)C2CC1N(C(=O)CC1CCCN1C)C2 C(C(=O)N(C1CCN(C(C2(c3ncco3)CCC2)=O)C1)CCO)(C(C)C)OC N1(C(c2nc(COC)[nH]n2)=O)CCOCC(CNC(C2CCS2(=O)=O)=O)C1 CCC(CO)C(=O)NCCCCC(C)NC(c1scnc1C1CCCC1)=O C1(NC(c2ccc(Cn3ccnn3)o2)=O)CN(C(C2(Cl)CC2)=O)CC2(CCC2)C1 C1(CCOC)CN(C(c2sc(=N)[nH]c2C)=O)CCN1C(c1ccns1)=O C(CCF)(C(=O)NCc1cc(OC)ns1)NC(c1c(CC)c[nH]n1)=O N1(C(C(CCC2CC2)NC(Cc2n(C)nnc2)=O)=O)CCC12CCCSC2 N1(C(C2C(=C)C2)=O)CCCC(C2(NC(C3CC(O)C3)=O)CC2)C1 N1(C(c2nocc2C)C(=O)NCCCCCC)CCc2c(Cl)cccc21 N1(C(C2(C)C(C(=O)OC)C2)=O)CCC2(CC1)CC(NC(=O)CCCC(C)C)C2 C(=O)(CCCCC(F)F)N1CCC(N(C(=O)COCC2CCCCO2)CCC)C1 CCC(CC(F)(F)F)C(=O)N(C(C)CN(C(=O)C(F)C(C)(F)F)C)C N1(C(C(CC)CCc2ccccc2)=O)CC2CCC1CN2C(=O)C1=CC(C)(C)C1 N1(C(C2N(C(C)=O)CC(O)C2)=O)CC2CN(C(=O)CSc3nccn3C)CCC12 C1(CCNC(=O)Cc2ccccn2)CCN(Cc2cccc(OC(F)F)c2)CC1 C(=O)(CC(C=C)CC)NC1(CC=C)CCN(C(c2nccnc2Cl)=O)C1 c1(-c2n(CC=C)nc(-c3ccnn3C)n2)cc(OC)c(O)cc1C O=C(C1=CC2(CCN(C(=O)C3CC3)C2)C1)N1CCC(CSC)C1 CN1CCc2cc(CC(=O)NCCC3CN(C(=O)C4=CCCC4)C3)ccc21 C1(CNC(C2(CC)CCC2)=O)CC(O)(CNC(=O)CC=CC(C)(C)C)C1 C(=O)(CC(COC)COC)NC(CC)C(=O)NCC1CCOC1C C(=O)(C#CC1CCOC1)NCC(c1ccc(C)cc1)NC(C1CC(O)C1)=O C1(C=O)CC12CC(F)(F)C2.N1(C2CN(C(CCC#C)=O)C2)CC(NCC=C)CC1=O N1(C(CC(C=C)(C)O)=O)CCC(O)(C2(NC(=O)CN(C3CCSC3)C)CC2)CC1 C12(CNC(CN3C(C)CC3)=O)CCC(CC1)CN2C(=O)C(O)CCn1cncn1 c1(CC(N2CC3(C2)CN(C(=O)Cc2sc(O)nc2O)C3)=O)ncc(Cl)cc1Cl C1(C(N(CC)CC)=O)CC(NC(c2c(N)c(C(=O)OC)nn2C)=O)C12CCC2 c1(C(=O)NC2CC(C)(CC)N(C(=O)C=Cc3cnc[nH]3)C2)cc(C#N)ccc1N c1(CC(=O)NCC(CN(C(CSCCCC)=O)C)O)noc2ccc(OC)cc12 c1(SC)ccc(O)c(C(=O)N(CCNC(C2CCSC(C)C2)=O)C2CC2)c1 C(c1c(Cl)cccc1Cl)=CC(=O)NC1C(F)CCN(C(COCCN(C)C)=O)C1 c1(OC)cc(C(N2CCC2CNC(=O)CC23COC(C)(C2)C3)=O)ccn1 C(C)(C)(CN1C(=O)CCc2ccc(Br)cc21)C1CCC(C(=O)OCC)CC1 C(=O)(C(C)C(CC)CC)N1CCC(C#C)(C(=O)NCC2(N(C)C)CC2)C1 c1(NC(C(=O)NCC2OCC(Cc3n[nH]c(=N)s3)C2)=O)ccc(Br)cn1 N1(C(=O)C2CC2)CCCC(COC2(C)C(C(NOC(C)(C)C)=O)CC2)C1 N1(C(CCOC)=O)C2CCC1C(CNC(=O)Cc1cccc(NC(C)=O)c1)C2 c1(CCCC)ccc(C=CC(=O)NC2CC2CNC(c2cc(C)nn2CC)=O)o1 N1(C(C(C=C)OC)=O)CCCC1C=CC(=O)NC(CC)C(C)CN(C)C C(=O)(C1c2c[nH]nc2CN1C(c1cnc(=N)[nH]c1)=O)NCC(C(=O)NC)(C)C N1(C(C(C(C)C)O)=O)CC(NC(=O)CCCOc2cccnc2)CC2(CC2)C1 C1(NC(=O)Cn2cncn2)CCSC12CN(C(C13CCC(F)C1CC3)=O)C2 C(CN=c1[nH]c(C2CCCC2)nc(=N)[nH]1)(C(C)(C)C)NC(C(C)O)=O c1(C(=O)NCCC(C)(C)NC(c2occ(C)c2)=O)cc2n(n1)CC(F)C2 n1(CC(=O)NCC)cc(CNC(=O)CN(C(=O)C(CC)OC)C2CC2)nn1 c1(C(N(CC(C)NC(=O)CC(=O)c2cnn(C)c2)C)=O)ccc(O)cn1 N1(C(c2cc(SC)oc2)=O)CCSCC1CCNC(=O)CC1CCCO1 CN1CC(NC(C2(NC(c3ccncn3)=O)CC2(C)C)=O)C(=O)N1 C1(OC)(OC)COC(NC(N2CCC(SC)CC2)=O)C1 C1(C2CCN(C(=O)CC3C=CCCC3)C2)CCCCN1C(=O)C(F)CC1CC1 Cc1cc(C(=O)NC2(C)CC(NC(=O)Cc3ccc(F)c(F)c3)C2)cc(F)c1 C1(NC(C(c2ccco2)NC(CCN(C)CC)=O)=O)CCCCC1NC(C)=O c1(C(N(C2CC(NC(=O)CC3CCCOCC3)C2)C)=O)cc2cccnc2[nH]1 Cc1cc(Cl)cc(C(=O)NCCN2CCN(C(c3cc(=O)cc[nH]3)=O)CC2)c1O CC(=O)CCCC(=O)NC1CC(F)CN(C(=O)CCN2CCN(C)CC2)C1 N12CCC(O)(CC1)C(=O)N1CCC(CC1)C2=O.N1(CC)CCCC(C(F)(F)F)C1 CCC(CC)C(C)C(=O)N(CCCCCC(=O)N1CC(OC(C)C)C1)C N1(C(c2ccc(CC)cn2)=O)CC2CC(NC(c3ccn(CCOC)n3)=O)C1C2 N1(C(CC=CCC)=O)C(C(=O)NCc2ccns2)CC1C C1(CNC(COc2ccc(C)cc2)=O)CCC(C)CN1C(=O)Cc1cnns1 N1(C(C(C)=C(C)C)=O)CC(NC(c2nn[nH]c2Cl)=O)CC2(CCOCC2)C1 c1(C(=O)NCC(C2CCOC2)NC(c2nc(C(N)=O)sc2)=O)nnn2c1CCC2 CCC(N=c1ccnc(NCCC2COCCO2)[nH]1)c1ccc(F)cc1F c1(CNC(CC=C(C)C)=O)nccc(C(=O)NOCCC2COCC(C)O2)n1 N1(C(C(C)S(C)(=O)=O)=O)CC2CCN(C(=O)C(C)(Cl)Cl)CC(C2)C1 C1(N(C(=O)CO)C)CCN(C(=O)CCc2nc(C3CC3)no2)C1.C(c1cnc[nH]1)=C(C)C N1(C(CCSCC)=O)CCC(C)(C)C(C(=O)NC(c2ccco2)CO)C1 N1(C(=O)Nc2cc(Cl)ccc2Cl)CCN(Cc2cc(Cl)ccn2)CC12CC2 C1(CC)CCCCN1C(=O)C(CNC(=O)CCCN(C)C(C)C)CC1CCCC1 C1(CCNC(C(=Cc2ccncc2)C)=O)CCN(C(=O)CN(C)C(C)C)C(C)C1 CCCCCC(O)C(=O)N1CC2C(CC(=O)NC3CCCC4(C3)N=N4)C2C1 CC(CCNC(=O)C(C)n1ccnn1)NC(=O)Cc1cnoc1 C1(C)(CCOC)CN(CC(C2CCC(F)(F)CC2)C)CCO1 c1(C(=O)NCC(CNC(C(C)n2cccn2)=O)O)cc2c(o1)CCCNC2=O c1(NC(C2CCN2C(c2ccc(OC(F)(F)F)c(F)c2)=O)=O)ccc(Br)cc1Cl n1(CC)cc(CO)nn1.c1(CNC(C2CC(C(C)C)C2)=O)cnn(-c2nccs2)c1 c1(C(=O)NCCN(C(C(CC)F)=O)CCOCCO)oc(C)nc1C Cc1cc(N)ccc1C(=O)NCC(C)(C)CN(C)C(C1CCN1C)=O c1(C(N2CC(OC)(CNC(=O)C(O)Cn3cncn3)C2)=O)cncc(N)n1 C12(NC(c3cc(C)cc(C)c3)=O)CCCC1N(C(=O)CC1CCCCO1)CCC2 C(=O)(C(C)C(O)CC)NCCCC(C)(C)NC(c1c(CC)cco1)=O C(=O)(C(C)CC(C)(C)C)NCCC(C)(C)NC(CSc1ccc(C)cc1)=O N1(CC(N2CC(n3cc(C(C4C(C)OCC4)=O)nn3)C2)=O)CCS(=O)CC1 CC(N=c1ccnc(NC(c2cc(F)c(F)c(F)c2)C)[nH]1)c1ccc(O)nc1 Cc1nc(C2CCCN(C(C3CN(C(C4CCC4)=O)CCO3)=O)C2)oc1C(=O)O CC(CC(=O)OCC1CSCN1C(=O)C(C)(C)F)N(C(=O)C(C)(C)C)C C1(CCNC(CN(C)C(=O)C2CC2)=O)CCCN(C(C2CC(CF)C2)=O)C1 N1(C(CCc2ccn(C)n2)=O)CCC(CCC(=O)NC2CCSCC2)CC1 C1(C(N2CC3CCCC3(CNC(=O)C(F)(F)C(F)F)C2)=O)Cc2ccccc2C1 CC1CC(NC(c2cccc(Cl)n2)=O)CCN1C(c1cc(O)n[nH]1)=O C1(CC(C)C)(C(=O)NC2CCCC2CNC(c2ccco2)=O)CCCC1 N1(C(C23CC(CO2)C3)=O)CC2CN(c3nnc(O)s3)CC2C1 N1(C(C)C)CCN(C(=O)NCC(C2CCOCC2)F)CC1C C1(CCC(=O)NCCNC(C2CN(C(c3cnn[nH]3)=O)C2)=O)CCCCC1 N1(C(c2cc(COC)cn2C)=O)CC2(CC(NC(C34CC(OC)C3C4)=O)CO2)C1 C(=O)(C(=O)N=c1nc(-n2cccn2)[nH]o1)N(c1cc(Br)ccc1C)CCC C1(CCN(C)C(C2CCN(C)C2=O)=O)CCCCN1C(=O)CC1(C)CCC1 C1(NC(Cc2c(C)nc[nH]2)=O)CN(C(=O)Cc2ncccc2C2CC2)CC1(C)C n1(CCOC)nc(C2Cc3ccccc32)nc1C1CCCN(c2ncccn2)C1 S(=O)(=O)(c1cccc2nsnc12)NC1CCN(CCN(C)Cc2cccnc2)C1 c1(C(N2CCN(C(C3(COC)CC3)=O)CC2C)=O)cc(P(C)(C)=O)cs1 c1(CC(=O)NCC(CNC(C2CCN(CCC)CC2)=O)O)nsc2ccccc12 N1(C(CN(C2CCC2)C)=O)CCC2(CC1)CC2C(=O)NCCC(O)C(F)(F)F c1(CN=C(NCC(C=C)(F)F)NC2CC(=O)N(CCC)C2)cc(Cl)ccc1OC N(C(=NCCc1cc(OC)ccc1C)NC1CCCC1)CCOC c1(OC)ccn2c(C(N3CC(CNC(=O)C(O)CF)C3)=O)cnc2c1 CCC(Cc1ccccc1)CC(=O)NC(COC)CNC(=O)C(F)(F)N(C)C N1(C(COCC(C)C)=O)CCCCC(N(C)C(C2CN(C(C)C)C2)=O)C1 C1(NC(c2cnc(C3CCCC3)s2)=O)CCCCN(C(=O)CC2CCOC2)C1 N1(C(C(CSC)OC)=O)CC(C2CCCCN(C(c3ccc(Cl)c(F)c3)=O)C2)C1 CN1CCCC1(C)C(=O)NCC(c1ccccc1OCc1ccccc1)N(C)C C1(CNC(C2CCCCO2)=O)CC12CCN(C(c1cc(F)n[nH]1)=O)CC2 C=Cn1nncc1C(=O)NCc1cc(Br)n[nH]1.c12cn(nn1)C1CN(C1)C2=O c1(C(N2CC3C(CN(C(c4c(C)cccn4)=O)C)C3C2)=O)ccc2nncn2c1 Cc1nc(C)c(CC(=O)NC2C=CCN(C(=O)CC3(O)CCOC3)C2)s1 CC1(C)CN(C(C2(O)CCCCCC2)=O)CC(C)(C)S1(=O)=O S(=O)(=O)(c1ccc(F)c(Cl)c1)N1CC(F)CC(C(=O)Nc2cnc(CO)nc2)C1 C1(CNC(C(C=C)O)=O)CC2CCC(C1)N2C(=O)C(c1cccc(Cl)c1)C c1(C(N2CC(N(C(C=CCOC)=O)C)C2)=O)cccc2nc(COC)[nH]c12 c1(CN2CCC(=O)N(Cc3ccccc3)CC2)cc2cc3c(cc2[nH]1)OCCO3 C(=O)(CC1C(=O)Nc2c(F)cccc21)NC(CN(C(c1csc(C)n1)=O)CC)C c1(C(=O)NC(CNC(c2c(C)coc2)=O)CO)ccc(-c2nnc(O)o2)cc1 C1(C(N(CCNC(C(CCC)O)=O)CC)=O)CC2CCC(C1)N2 C12(CNC(CCCCC)=O)CCCCC1N(C(c1cccnc1F)=O)CC2 Cc1csc2c(CC(N3CCCC3C(=O)N(C)C3CC3)=O)cccc12 N1(C(C(C)OCCCC)=O)CCC2CN(C(c3cc(C#N)ccc3F)=O)C(C)C12 c1(C(C)C)ccc(OCC(=O)NCC(C)(CO)NC(C2CCC23CCC3)=O)cc1 C(=O)(CCCCCF)NC(C1CCN(C(c2ccc(CC)cc2)=O)C1)C Cc1ccncc1C(N1CC(NC(c2cccnc2O)=O)C(C)C1)=O C1(CNC(C=CC)=O)COCC1NC(=O)CSc1nncn1C(C)(C)C Cc1cc(C(=O)NC2CCN(C(=O)CCn3cccn3)C(C)C2)ncc1Br C1(F)(CNC(=O)OC)CCC(NC(C2(NC(=O)CCS(C)=O)CCCC2)=O)C1 C1(C(=O)NC2CC(CCNC(CSCCOC)=O)C2)CCOC(C(C)C)C1 CC1CN(C(=O)CCOCC(F)F)CCN(C(c2cc(C(C)(C)C)on2)=O)C1 N1(C(c2c(OC)nccc2)=O)CCC(NC(c2csc(C)n2)=O)C(F)C1 N1(C(CCCCC)=O)CCCOC(CNC(c2n[nH]cc2Br)=O)C1 N1(c2nc(C)nc3c2cc[nH]3)CCC2(CN(C(C3CCCC3O)=O)CC(C)O2)C1 C(CN=C(NCc1nc(-c2ccccc2)n[nH]1)NCC1CC1)C1CCC(C)C1 C(=O)(C1Cc2ccc(F)cc21)NCC1(C2(O)CN(C(C(CC)(C)C)=O)C2)CC1 C1(NC(C(CC)OC)=O)CN(C(c2c(Cl)ccc(O)c2Cl)=O)CC2(CCC2)C1 c1(C(N2C(CNC(c3cnc(Br)s3)=O)CCC2)=O)nc2ncccn2n1 c1(C(=O)NC(CC=C)CNC(=O)C(C)CN(C)C)cc2nccnc2[nH]1 c1(C(=O)NC(CC)(C)CNC(c2n[nH]cc2[N+](=O)[O-])=O)ccc(C)c(Cl)c1F N1(C(CC(C)NC(c2ccn(CCC)n2)=O)=O)CC(=O)NC(=O)C1C c1(OC)ccc([N+](=O)[O-])c(C(N2CC3C(NC(=O)CC#N)C3C2)=O)c1 CC1(C(=O)NC(CNC(C2CCCN2N=O)=O)C2CCC2)CS(=O)(=O)C1 C1(C(C(=O)N(CC=C)C)C)CCCN(C(C2CN(C(C)=O)C2)=O)C1 c1(C(N2CC=CC(NC(C(C)SC)=O)C2)=O)c[nH]c2ncc(Br)cc12 CC1CCC(CNC(=O)C(C)(C)C(F)F)CN1C(c1coc(C#N)c1)=O C1(NC(c2ccc(=N)[nH]c2)=O)CCN(C(c2scnc2C2CC2)=O)CC1CO C(=O)(C(C)CCC(C)(C)C)NCC(C)(C)OCCNC(C1(CC=C)CCOC1)=O CC1CC(NC(C2CCC3(CC2)CC3)=O)CCN1C(=O)COC1(C)CCCC1 C1(CC=C)(C(=O)NC2CCC2C(=O)OC)CN(C(=O)CCCNC(C)=O)C1 Cc1cccc(C)c1C(=O)NC1CC2(C1)CC2NC(=O)CC1CC2(CC2)C1 C(=O)(C1=CC(O)CCC1)NC1(CNC(c2nc(C(C)=O)sc2)=O)CC1 c1(OC)ccc(C(=O)NC(C)COCC(F)(F)F)c(Br)c1F c1(N(CC(=O)NCC)C)cc(C)nc(NC2CCCOC2c2ccnn2C)n1 C1(NC(C2CCC(C(C)C)CC2)=O)CCN(C(=O)CC2COC(C)(C)C2)CC1O C1(CC(N2CCC(NC(c3c(C(=O)OC)c(C)[nH]n3)=O)C2)=O)CCC(F)(F)CC1 CC1(C)OCc2c1n[nH]c2C(=O)NC1CC(NC(c2cnc(S)nc2)=O)C1 N1(C(C2CCCN(C)C2)=O)CCC(C(=O)NC(c2ncc(F)cn2)C)C1(C)C C1(NC(C(CC)C2CC2)=O)CCCCC1CC(=O)N(C1CC(CCF)C1)C C#Cc1ccnc(C(=O)NCCN(C(=O)CCc2nncs2)CC(C)O)c1 N1(C(c2c(C)nc(C(C)C)s2)=O)CCOCC(NC(=O)C(C)(O)C(C)C)C1 C1(F)(CNC(=O)Cc2cnns2)CCC(CNC(=O)CN2C(=O)CCC2=O)C1 c1(C(N2C(C)CN(C(c3ccncn3)=O)CC2)=O)c(F)ccc(F)c1Cl C1(CNC(CC(CC)C2CC2)=O)CCC2(CN(C(c3cc(CC(C)C)c[nH]3)=O)C2)O1 CC1(C)CC=C(C(=O)NC23CCC2CN(C(c2ocnc2C2CC2)=O)C3)CC1 C(CCCCNC(C12CCC1CC2)=O)NC(=O)CCF CC(C)(O)CC(=O)N1CCCC1CCNC(c1cccc(C2CNC(=O)C2)c1)=O C1(F)(C(N2CCC(CC)(CC)C2)=O)CCCN(C(c2cccc(OC)n2)=O)C1 N1(C(c2n(CC)nc(C)c2)=O)CC2CCN(C(c3cnn4ccccc34)=O)CC12 c1(OC)cc(C)cnc1C(N1CCCC(CNC(=O)C(O)CSC)CC1)=O C1(C(C)(C)C)CC(CNC(=O)CCc2ccsc2)CN(C(c2ccon2)=O)C1 N1(C(C2CCCCN2Cc2cccnc2)=O)CCC(C2CCOC2)CC1 C(=O)(C1=NN(c2ccccc2)C(C(=O)NCc2coc(C)n2)C1)OC C(=O)(C(C)(F)C(C)(C)F)N1CCC(C2NCCCC2)C1.c1(CC)c(F)ccnc1F C(=O)(C(C)CCCC(C)C)NCC(CC(=O)Nc1c(C)ccc(OC)c1)(C)C Cc1ccc(CNC(=O)COC2CN(C(c3ncccc3N)=O)C2)c(F)c1 CCC(C)(CNC(=O)COCCOC)C(=O)N(C)Cc1cc(C)nn1C CCCC(C)(CC)C(=O)N1CC(C)C(C)(CNC(=O)CCCc2ccccc2)C1 N1(C(C=CC(=O)N(C)C)=O)CC(F)(F)CC1CO.c12cc(no1)C(=O)NC2 c1(C(=O)OCC)ccc(C(N2CC(NC(c3cccc(C)n3)=O)C(C)C2)=O)cc1 CN1CCCCC1CCC(=O)NCC1CCCC1NC(=O)C(O)c1ccco1 c1(C(N2CCC(CNC(C(COC)OC)=O)CC2C)=O)ccc2ccccc2c1 C=CCC(CC=C)n1cc(CONC(=O)CCc2cccc(C)c2)nn1 CCCC(C)(O)CC(=O)NC1C=CCC(C(=O)NC2CCN(C(C)=O)C2)C1 C(=O)(CCCC(C)(C)C#N)N1CCC(C)N(C(c2cn(C)nc2Br)=O)CC1 C1(C(N(C(C)C)CCN(C)C(C2(C)CCC(=O)CC2)=O)=O)CCCCCC(=O)C1 C1(NC(CC2(C)CCN(C(CCCC)=O)C2)=O)CC2CCC(C1)N2C Cc1nnc(CC(=O)NC(C)(CNC(=O)C(F)(F)c2cnn(C)c2)CO)o1 c1(CC)ccc(C(=O)NC(C2CCN(C(=O)CNC(c3ccccc3)=O)C2)C)s1 N1(C(C2C=CCC2)=O)CCN(C(=O)C=CC2CC2)C(c2ccncc2)C1 C(CC(C)C(=O)NC(C1CCN(C(=O)CCc2cccnc2F)C1)(C)C)OC c1(C(=O)NCC2(O)CCN(C(c3cc(C4CC4)sn3)=O)C2)cnc2c(c1)CCC2 Cc1cc(O)c(C(N2CC(N(C(=O)CN3C(=O)CCC3=O)C)C2)=O)nn1 C(=O)(C(C(=O)NCC1CCC1NC(=O)CCSc1ccccn1)C(C)C)OCC c1(C(N(CCNC(=O)COCCN(C)C)CC)=O)ccc(-n2ccnn2)cc1 C1(NC(CC(CC)(C)C)=O)CN(C(c2cc(C(F)F)ncn2)=O)CC12CCC2 N1(C(CCC=C)=O)CCC(C2CC2)C1CNC(c1ncn2cccnc12)=O C=CCC(C(=O)NCCN(C)C(c1[nH]c(=N)sc1CC)=O)C(C)C c1(C(=O)NCC2N(C(C=C3CCN(C)CC3)=O)CC=C2)csc2nccn12 c1(CCC)nc(C)c(C(N2CCCC2C2(NC(c3cnn(C)n3)=O)CC2)=O)o1 c1(C(N2CCCC(N(C)C(C3CCCC3(F)F)=O)C2)=O)ccc(N)c(Br)n1 C1(CNC(C2C(C)(C)CO2)=O)CN(c2nnc(C(F)(F)F)s2)CCCO1 C(C(=O)N1CC(F)(CNC(C2CC2C(F)(F)F)=O)C1)(C(C)C)c1cc(C)no1 C(C(=O)N(C)C)(C(C)C)c1cc(C)no1.c12ccnc(n1)C(=O)O2 c1(C(=O)NC(C(C)NC(c2c(C)con2)=O)CO)cnn(-c2ccccn2)c1C C1(NC(C2N(C)C(=O)CCC2)=O)CCC2CCN(C(C34CCCN3CCC4)=O)C12 C1(C(N2CC(OC)(CO)C2)=O)CCCN(C(=O)C(n2cc(C)cn2)C)C1 N1(Cc2cccc(N(C)CC)c2)CCC2(CCCOC2)C1 CC1(C)CC(C(N2CCC(C3CCC3)C2)C(=O)C)CC(C)(C)C1.CNC=O c1(C(N2C3CN(C(CC(C)=C(C)C)=O)C(C3)C2)=O)cc2ccc(N(C)C)cc2[nH]1 c1(NC(CC)=O)ccc(Nc2ccncc2F)cc1.C12CCN(C1)C(=O)C2 N1(C(C2=CC(C)CC2)=O)CCCC2(C1)OCCCO2 C(=O)(C(F)CC(C)(C)C)NCc1cc(C(N2CCCC(C=C)C2)=O)sc1 Cc1cc2n(n1)CCN(C(c1ccc(-c3ccccc3F)cn1)=O)C2 c1(CC(=O)NCCN(CCOC)C(C2CCCCC2OC)=O)c(C)cnn1C N1(C(c2c(NC)cnc(Cl)c2)=O)CCC(NC(=O)C(CO)N(C)C)C12CCC2 c1(OC)nccc(C(=O)NCCCCN(C)C(c2sccc2CC#N)=O)c1F N#Cc1c(F)cc(C(=O)NCC2(NC(c3cnc(O)o3)=O)CCC2)cc1F C1(C(=O)NCC(CCO)OC)CCCN(C(C23CSCC2C3)=O)CC1 c1(NC(CC)(C)CNC(C2CC(C(=O)OC(C)(C)C)C2)=O)ccc(Cl)cn1 C(C1(C)CCOCC1)=CC(=O)NCC(C)CNc1ncc(Br)cn1 c1(C(N2CCCC3(NC(CC(C(C)C)O)=O)C2C3)=O)c2ccccc2nn1C CN(C)S(=O)(=O)N1CCCC1CNC(=O)NCC1CCCN1CCCO CCCCC(CNC(c1cc(C2CC2)ncn1)=O)NC(c1cc(CC)c[nH]1)=O C(=O)(C1CCCc2ccccc21)N1C(C)CCC(NC(c2c(CC)cco2)=O)C1 C1(CC=C)(NC(=O)C=CC(C)CC)CCN(C(=O)CCS(N)(=O)=O)CC1 c1(CCCCC)nc(CSCc2ncccn2)n(-c2ccc(Cl)cc2)n1 C1(NC(COCC=C)=O)CCN(C(=O)CN2CC(=O)NC2=O)C(C2CC2)C1 c1(N(C(C(=O)OC)(C)C2CC2)C)ncc(C#N)cc1F N1(C(C2(COC)CC2(F)F)=O)CCC(F)(CNC(c2cccnc2C)=O)CC1 C1(C(=O)NCC2N(C(c3c(C)cncc3)=O)CC(O)C2)CCCCC1(F)F Cc1cc(C(N2CCCC(CN(C)C(C3CCCSS3)=O)C2)=O)cc(C)c1 Cc1c(C(N2CC3(CCC3NC(c3sccc3F)=O)C2)=O)cncc1Br N1(C(c2cnc(CCC)s2)=O)CCC(NC(c2cnoc2CC(C)C)=O)C(O)C1 Cc1cc(C(=O)NCC(Cc2ccccc2)NC(=O)C=CCO)cn1C(C)C C1(C)(CC(=O)NCC(C)N(C(C2CC(C#C)(O)C2)=O)C)CCS(=O)(=O)N1 Cc1cc(O)ccc1CC(N1CC2CC2(NC(=O)CCNC(=O)C2CC2)C1)=O C1(C(=O)NC2(CO)CC2)CC2(CC2)CN1C(=O)CC1CCCOC1 N1(C(CCc2ccn(C)n2)=O)CC(CNC(c2ccc(Cl)c(N)c2)=O)C(C)(C)C1 CCCCCCCCCCCC(=O)N1CC2CC1CN2C(C1CCOC(=O)N1)=O N1(C(C(C)CN(C)C)=O)CCCCCC(NC(=O)COCC2CCCC2)C1 C1(CC(=O)OC)CCCN(C(N2CCC3(CC2)CC3)=O)CC1 c1(C(N2CCC(N(C(CCNS(CC)(=O)=O)=O)C)C2)=O)ncccc1C(F)(F)F c1(C(C)C)ccc(-n2cc(CNC(=O)C(C)C3CCOC3)nn2)cc1 CCC1=C(C(=O)NCC2CCN2C(=O)CC(C)OC)CCCO1 C(=O)(CC(O)C(C)(C)C)NC1CN(C(C(c2ccc(F)cc2)OC)=O)CC1O N1(C(CNC(=O)Cn2nccn2)=O)CCC(OCCS(C)(=O)=O)CC1.C(CCN)O C1(CNC(CCC=C)=O)CN(C(c2ccncc2-c2ccccc2)=O)CC1(F)F C1(CNC(c2c(C)ccc(Br)c2)C(=O)O)CC2OC(C)(C)OC2C1 N#Cc1ccc(C(=O)NCC=CCNC(c2ncsc2-c2ccccc2)=O)o1 N1(C(C2CN3CCC2C3)=O)CCC2(C1)CN(C(C1CC=CCO1)=O)C2 C1(C2CCN(C(=O)CNC=O)CC2)(C(=O)NCC(CCC)O)CCOCC1 C12(NC(=O)CCC(F)(F)F)CCCC1(F)CN(C(=O)CCC1CC1(F)F)C2 c1(C(=O)NC2CCCC(CNC(C(C)=C(C)C)=O)C2)c(F)ccc(F)c1O c1(NC(C(CC)NC(=O)Cc2cc(C)cs2)=O)cc(C)c(C)cc1C C(=O)(C1Cc2ccccc21)N1C(C(=O)NCC(C(CC)C)CO)CCC12CC2 Cc1ccc(CN2CC(C(=O)NC3CN(C(c4ccnnc4)=O)C3)CC2=O)cc1 C1(CNC(C2CC(CSC)C2)=O)CN(C(c2cc3ccsc3s2)=O)CC(C)(C)O1 c1(-c2nc(-c3c(OC)n(C)nc3)on2)c[nH]c2nccc-2c1 C(=O)(CS(=O)(=O)C1CC1)NC12CCC(CNC(C(C)=CC3CC3)=O)(OC1)C2 N1(C(c2c(OC(F)F)cccc2Cl)=O)CCC2CN(C(c3cnc[nH]3)=O)C2C1 CCC(CCC(=O)Nc1cnc(C)c(Cl)c1)NC(C1CC(C)(C)CO1)=O C1(CC=C)(NC(=O)CC=C(C)C)CCN(C(=O)C(C)N(CC)CC)CC1 C1(C)(CC)CC(NC(=O)CSCC(N)=O)CN1C(c1cccc(CCO)c1)=O c1(COC(N2CC(CC(C)OC(C)(C)C)C2)=O)ccc2ccc(F)c(F)c2n1 N1(CCc2cn(NC(C3CCC(=O)N3)=O)nn2)CCCC(CC2CCOCC2)C1 Cc1cnn2ccc(C(N3CCCC3C(C)NC(C34CC(C)C3C4)=O)=O)nc12 c1(C(=O)NCC2N(C(CC3N(C(C)C)CCC3)=O)CC2)[nH]nc2ncnc(O)c12 c1(N(CC#CC)C)nc(=NCC2CCC(F)C2)nc(N2CCOCC2)[nH]1 CC1COCC1(c1nnnn1C)NCCCCn1cc(CO)nn1 C(=O)(C(C)C(CC)CC)N1CCC(C#C)(C(=O)NCC(C)(C)CC2CC2)C1 C(C(N=[N+]=[N-])C(=O)N(C)CC1CN(C(c2cc(C)cnc2C)=O)C1)OCC C(CCNC(c1ccc(O)nn1)=O)(C(=O)N1CC2CC2C1)OC c1(-c2nn(C(COC)COC)c(CCC(F)(F)Cl)n2)cc(F)c(N)c(F)c1 CC1CCC(C(F)(F)F)CN1C(c1ccc(CCN)cc1F)=O C1(C(=O)NC2CCC(NC(C3CC3c3cccs3)=O)C2)(C(F)F)CC(F)(F)C1 C1(CNC(c2c(C)ccnc2)=O)CN(C(=O)Cc2ccoc2)CCC12CCC2 C(CCOCCO)(C(=O)NC(c1ccn(C)n1)C)NC(C(CSC)O)=O c1(C(N(CC(CC)NC(=O)CC2C=CS(=O)(=O)C2)C)=O)nc2nc(C)ccn2n1 c1(CC)ccc(C(N2C(CNC(c3n[nH]c(C)c3Cl)=O)CC3CC23)=O)cn1 Cc1cccnc1C=CC(=O)NC1CCN(C(=O)CC2(O)CC2)CC1F N1(C(C2CN(CC)CC(F)C2)=O)CC(F)(F)CC1C#N.c12csc(n1)CNC2=O C#Cc1cc(C(=O)NCC(C(C)C)NC(=O)C(C)(O)COC)ccc1C C1(C(=O)NC2(CCNC(c3cncn(C)c3=O)=O)CC2)CCC2(C1)CC2(F)F N1(C(C2CCCC(C)C2)=O)C(C)CC2CN(C(c3ccc(CO)nc3)=O)CC12 C12(NC(C(=O)NCCOCCOC)=O)CCCN(C(=O)CCC(C)(C)C)CC1C2 c1(NCC(CSC)OC)ccc(S(=O)(=O)NCc2cncs2)c(Cl)c1 Cn1c(C(c2nnnn2CC)NC2CCc3[nH]c(=N)sc3C2)nc2c1CCCC2 c1(C(N(C)CC2CCN(C(CCOCC)=O)C2)=O)ccc(OC)c(OC)c1C C(CCCC(C)NC(=O)Cn1ccsc1=N)NC(C=C(C)Cl)=O c1(C(C(=O)NCCCC2CC2)N(CCC(=O)OC)CC#N)csc(Cl)c1Cl C1(C(=O)NCC23CN(C(Cc4c(CC)cccc4)=O)C(C2)C3)CC2(CCCC2)CO1 c1(OC(C)C)ccc(Cl)c(C(N2CCCC(O)(CNC(c3ccco3)=O)C2)=O)n1 C1(C2CC2)(CNC(c2cc(OC)c(O)nc2)=O)CCN(C(c2ccsc2C)=O)C1 N=c1ccc(C(=O)NC2C=CC(CNC(c3cn(CC(F)F)cn3)=O)C2)n[nH]1 c1(NC(C2CS(=O)(=O)CC2N2CCOCC2)=O)nc2cccc([N+](=O)[O-])c2s1 c1(C(C)NC(C(=O)NCCCC)CC)ccc(OC)cc1 c1(C(=O)NC(CNC(C(C=C)(C)C)=O)(C)C)cc(C)cc2c1NCCC2 Cc1cccc(N)c1C(=O)NC1CC(O)CN(C(=O)CC2CSCCS2)C1 C1(C(=O)NCC2C(C(F)(F)F)CCN(C(CSC)=O)C2)CCc2nn[nH]c2C1 Cc1cc(C)c(NC(=O)CCC2CC(NC(=O)C=CC(=O)NC3CC3)C2)s1 c1(OCC(=O)NCC(C2CC2)NC(Cc2c(C)ccnc2)=O)ccc(Cl)c(F)c1 N1(C(c2cc(C)no2)=O)CC2CC(C1)CN(C(c1ccnc(Cl)c1N)=O)C2 c1(C(=O)NC2CCN(C(=O)Nc3c(Cl)cccc3Cl)CC2)ccc2c[nH]nc2c1 CC(C(=O)OCc1nccnc1O)C(C)NC(=O)OC(C)(C)C c1(CC(=O)NCC2CN(C(C=CCOC)=O)C3C2C3)c(C)nn(C)c1Cl C1(C(N2CCC(NC(CCC(=C)Br)=O)C2)=O)CCC(C)(O)CC1 c1(C(C(=O)NC2CC2)N(CCOC)CCNC2CCCCC2)cc(I)ccc1F c1(CCC(=O)NCCCN(CCCNC(C2CC23CC3)=O)C)ccnn1C C(=O)(C(C)CCOC)NC1(CCCNC(C2C(=C)CC2)=O)CC1 Cn1ccc(=O)c(C(N2CC=CCC2C(=O)NC2CC(O)C(F)C2)=O)c1 CCCCCC(C(=O)NC1CCN(C(=O)C(C(=O)OC)OC)C1(C)C)C(C)C c1(C(N(C2(CO)CN(C(=O)CCOCCOCCO)C2)C)=O)ccon1 Cn1cc(S(N)(=O)=O)cc1CC(=O)Nc1ccc(OCCO)cc1 CC1CN(C)CC1NCCC(C)(C)c1ccccc1 C1(CC=C)(NC(C2CC(C(F)(F)F)C2)=O)CCN(C(=O)C(O)C=C)C1 C1(NC(CCCC#CC)=O)CCOC12CCN(C(=O)CC1NC(=O)NC1=O)CC2 C1(C(=O)OCC(=O)OCC2CC(F)(F)CO2)(OCC)CCOCC1 C1(NC(C(c2c(C)cccc2)(C)C)=O)CC2CC1N(C(=O)C=Cc1cnc[nH]1)C2 N1(C(c2ccc(C#N)cc2)=O)CCN(C(C2CCSCC2)=O)CC(CO)C1 CCC(C)C(C)C(=O)N(C)CC1(O)CN(C(c2ccc(SC(F)F)cc2)=O)C1 Cn1cccc(C(=O)NCC2(F)CN(C(=O)C(C3CCCCCC3)O)C2)c1=O N1(c2cc(SC)nc(C)n2)CCC2CN(C(=O)CCc3ccccc3CO)CC12 N1(C(C(CC2CCOCC2)NC(c2c(C)scc2)=O)=O)CC(CO)C1(C)C CSC1=C(C(=O)NCCC2(O)CCCN(C(=O)Cc3cnnn3C)C2)CCCC1 c1(-c2ccc(CNCCN3C(COC)CC(C)CC3)s2)n[nH]c2c1CC1CC21 c1(CN2C(C)CC(c3cn(-c4cncc(Cl)c4)nn3)CC2)c2c(nn1C)CCC2 c1(CC(=O)NCC2CN(C(c3cc(O)no3)=O)CCCO2)n[nH]c2c1CCCC2 C1(NC(c2ccc(Cl)s2)=O)COC2(CCN(C(c3cnc(Cl)s3)=O)CC2)C1 c1(C(=O)NC2(C)CC(C(N3C(C(=O)OC)C=CC3)=O)C2)ccc(C#N)c(C)n1 N1(C(c2c(SC)cccn2)=O)CCCCC(C2CN(C(=O)C(C)=C(C)C)C2)C1 N1(C(c2cc(Br)co2)=O)CC2CCC(C1CO)N2C(C1CC1[N+](=O)[O-])=O CC1CC(NC(=O)C(c2ccc(F)c(F)c2)=O)CN(C(c2cc[n+]([O-])cc2)=O)C1 CCC(CCCC(=O)N(C1CCCC1(C)O)C)NC(=O)C(C1CCCCC1)O N1(C(C(CCN(C(=O)OC(C)(C)C)CCO)(C)C)=O)CC2(CCCO2)C1C1CC1 C1(NC(c2ccc(Cl)cn2)=O)CCN(C(c2csc(Cl)n2)=O)C12CC2 CC1OCCC1CN(C(=O)C=CCC1(NC(=O)Cc2ccoc2)CCC1)C c1(C(N2C3CN(C(c4cnc(O)[nH]4)=O)C(C3)C2)=O)c(Cl)cc(Cl)cc1Cl c1(C(=O)NC(CNC(C=C(C)C)=O)CO)cc2cc(C)ccc2[nH]1 C(=O)(CC(C)C(=O)NC(c1ccccc1)C(N1CCC(F)(F)C1)=O)OC C1(O)(CCNC(C(C)N2CCC2)=O)CCCN(C(c2cc(=O)c(O)c[nH]2)=O)C1 C(=O)(CC(C(F)(F)F)NC(=O)CCCc1cnn[nH]1)N1CC(C)(COC)C1 N1(C(COCCCCC)=O)CC(NC(=O)C(C)(C)c2ccno2)C2CC12 CC1(F)CN(C(=O)CN2CCOCC2)CCN(C(C2(C(F)(F)F)CCCC2)=O)C1 C1(C2(NC(C3CCN(C(=O)c4occc4C)O3)=O)CC2)(OC)CCC1 N1(C(c2c(C)occ2)=O)CCC(C)(C)C(C(=O)NC(C)(C)CCF)C1 N1(C(CC(CC)NC(CCCC#C)=O)=O)C2CCC1COC2 CC1=CCCN(C(C2(F)CN(C(=O)CC3CCCC(C)O3)C2)=O)C1 c1(OC)ccccc1CC(C)(C)C(=O)NCC(CNC(C1CC1(F)F)=O)CO c1(CNC(c2cnn(CC)c2C)=O)c(Cl)c(C)nn1C Cn1ncc(C(=O)NC(CC2CCC2)C(=O)NC2(c3nc[nH]n3)CC2)n1 C(=O)(CCS(=O)(=O)CC(C)C)N1CC(NC(c2ncnc(C)c2C)=O)C1 C(=O)(C(C(C)(C)C)C1CCC1)N(C)CC1(NC(c2ccc(OC)cn2)=O)CC1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CCN(C(=O)CC(=O)NC)CCC1C C1(CCC)NC(=O)CCN(CC2=C(C)OCCS2)C1=O C(CN(C)C)(C(=O)N1CC(CC2CC2)C1)NC(C1C(C)C1)=O C1(C(N(C(COC)COC)C)=O)C=CCCN1C(=O)CC1CCC(C)(C)C1 C1(C)(C(=O)NC(C)C(=O)NCCC(Cl)Cl)C=CCCC1 CC1CC(C)C1CCCNC(=O)COCCO.c1(SC)cn(CC(C)(C)O)nn1 N1(C(C2CC(C(C)C)OCC2)=O)CC=C(CCNC(C2(C)CCCOC2)=O)CC1 C1(C(N(CC(COCC)O)C)=O)CN(C(=O)CCCn2ccnn2)C(C)(C)C1 C1(CN(C(C2(COC)CCC2)=O)C)CCN(Cc2ccccc2)C1 C1(CNC(CCOC)=O)C(C2CC2)CCN1C(c1nc(Cl)cs1)=O C=C1Cn2c(C(N3CC4CCC4(NC(C4CC4(C)CC)=O)C3)=O)nnc2S1 c1(CCC(=O)NC2CC(NC(COC(CC)C)=O)C2)ccc(F)cc1Br C1(NC(c2cc(C)n(C(F)(F)F)n2)=O)CC(C)CN(C(c2ccc(O)nc2)=O)C1 Cc1cc(C(N2CCCC(C(=O)NCC3CC(C)C3)C2)=O)cc(C)c1F c1(OCC)ccccc1C(N1CCC(C(=O)NC(C)CCC)CC1)=O c1(C(=O)NCC(CC)O)cccnc1CNC(=O)COCC1CCOC1 c1(C(C(=O)OCC=CC)C)cccc(NC(Cc2ccccc2)CO)c1 CC(C)C(C#N)C(=O)NCC(C)N(C)C(c1ccc(C(F)(F)C(F)F)cn1)=O N1(C(c2c(OC(F)F)cc(C)s2)=O)CCN(C(C2CC(C)C2)=O)CC(O)C1 c1(C(=O)NC2C(C)(C)N(C(=O)Cc3ccsn3)CC2)noc2c1COCC2 CC(C)CCCC(=O)NCC1CN(C(=O)C2=CCCCO2)CC1O C(=O)(C1CCC(=O)c2cccn21)N1CCN(C(C(C(C)C)NC=O)=O)CC1C C(CN=C(NCC1CCC1)N1CCOC(C2CCCO2)C1)c1ncc(C)cn1 Cc1nocc1CNC(=O)C(C1(O)CCC1)NC(=O)C(C1CC1)C1CC1 Cc1c(C(N2CC(CCNC(=O)C(C)C#N)C2)=O)cc([N+](=O)[O-])cc1Br C=C(CNC(=O)CC(C)C(C)(C)NC(=O)Cc1cnc(C)s1)c1ccccc1 N1(C(c2cnc(C)s2)=O)CCC(C(CO)NCC2(c3ccncc3)CC2)CC1 C12(C(=O)NCC3(CC(=O)NC(c4nc(C)on4)C)CC3)CCC(CC1F)C2 C1(NC(C(CCCC)C)=O)CCC2(CC1)CN(C(c1ccc(OCC)cc1)=O)C2 C1(NC(c2cnc(CCCC)s2)=O)CCN(C(c2oncc2CC)=O)CC1(C)C C1(C(N(C)CCN2CCCCC2)=O)N(C(=O)CCCC#N)CC12CCCC2 c1(C(N2C(CN(C(C(n3cc(Cl)cn3)C)=O)C)CCC2)=O)nnn(C)c1N C1(CC(=O)NCCCN(C(C2CCCCO2)=O)C(C)C)(OC)CCOCC1 N1(C(c2cnccc2)c2nc[nH]n2)CCCN(CC2CCCOC2)CC1 C(=O)(C1=CS(=O)(=O)CCC1)N(CCCCCCNC(C1CCCCNC1=O)=O)C CCCCC(C)C(=O)N1CCCOC(CCNC(c2c(C)ccnc2O)=O)C1 C(=O)(C(C)C(C)C)N(CCN(C(Cn1ccc(C(=O)OC)n1)=O)C)C(C)C c1(C(N2CCC(CCNC(C(C#N)C3CC3)=O)CC2)=O)cnc(O)c(Cl)c1 CC1CN(C(C2CN(C(c3c[nH]nc3C(F)F)=O)CC2(C)C)=O)CC1(C)CO N1(c2cc(C)nc(CO)n2)CCC2(COC(CNC(=O)C=C3CCCCC3)C2)C1 C1(C(N(CC=C)CC)=O)CC(O)CN1C(C1CCNC1=O)=O Cc1cnc2n1CCC(C(=O)NC1(Cc3ccccc3)CCNCC1)C2 Cc1ccc(O)c(C(=O)NCCCCCCNC(c2cc(C)[nH]n2)=O)c1 c1(COC)nn(C)cc1C(=O)NCC1C=CCN1C(=O)C(O)COC N1(C(c2on(C)c(=O)c2)=O)CC2(CCN(C(C3(c4cccs4)CCCC3)=O)C2)C1 c1(C(N(CC(C)(C)NC(C23CCCC2C3)=O)C)=O)n[nH]c2c1CCC2 Cc1cc(C(=O)NC(C)(CNC(=O)CC2CCCC23CC3)C(C)C)[nH]c1C CCC(C)(C)C(=O)C(=O)N1C(OC)CCC1c1ccccc1 C(C(O)C(=O)NCC(C)CNC(=O)CCN1CCC(F)C1)=CC N1(C(C2(C)CC(F)C2)=O)CCN(c2ccc(C(F)(F)F)cn2)C(CCO)C1 c1(OC)c(Cl)ncnc1NNC(=O)NC1CC1(F)F C(Cn1ccnn1)(C(=O)NOCCF)NC(C1CCNC1=O)=O c1(C(=O)NCC=C)ccc(C(=O)NC(C)(CNC(C2C=CCC2)=O)C(C)C)cc1 c1(-c2cc(NCc3c(C)cccn3)ncc2)cccc(O)c1C C1(CNC(C(C)NC(CC)=O)=O)(NC(=O)CC2CCCCC2)CC=CC1 CCCC1C(=O)NCCCN1CC(C)C.C1(C(=O)N)(OC)CCC1.O(CC)CC C1(CC)C(C(=O)NCCCN(CCCNC(C23CC(CO2)C3)=O)C)CCN1C c1(NCC(=O)NC(C2CCCC2)CNC(=O)CSC(F)F)cccnc1 N1(C(c2cc(CC)[nH]n2)=O)CCC(C)(NC(=O)C(C)COC(C)=O)C1 C1(CNC(c2cc(C(C)(C)C)on2)=O)CN(C(=O)C(O)CC(N)=O)C2(CCC2)C1 c1(C(CNC(=O)C(=O)N(C)C)NC(CCn2c(C)ncc2)=O)cccc(C(F)F)c1 N1(C(c2n(C(CC)C)ncc2)=O)CC(NC(=O)Cc2nocc2C)C(SC)C1 C1(OC)CN(C(=O)Nc2cnn(-c3ccc(Br)cn3)c2C)CCC1F c1(OC)ccc(Cl)c(C(=O)NCC23CC2CN(C(c2cc(N)nc(Cl)c2)=O)C3)n1 C(=O)(C(C)(C(F)F)SC(C)(C)C)NC(C)=O.CC(CC(C)NC(=O)COC(C)(C)C)N c1(C(N2C(C)(C)C(CNC(=O)Cn3ccnn3)CC2)=O)ccc(N)c(F)c1F Cc1[nH]c2ncccc2c1C(=O)NCC1CN(C(=O)C(C)CS(C)=O)CCCO1 c1(N2CCCCC(C)C2)nc2c(c(=NCCS(=O)c3ccccc3)[nH]1)SCC2 N1(C(COCC=C)=O)CCCC(O)(CNC(c2cc[nH]c2C2CC2)=O)C1 C#CCCCC(C)C(=O)NC12CC(C1)C2.C1CC(=O)N2CC(C2)N1C(C)=O C12(CNC(c3cc(CC)n(C)n3)=O)CC(CO1)N(C(=O)Cc1n[nH]c(=NC)s1)C2 c1(CNC(C2CC(CCC)C2)=O)nc(C(=O)N(C2CCCC2C)C)c(C)o1 CCC(CC)C(=O)OCCn1cc(CN2CC2=O)nn1.C(C)(C)(CC(N)=O)NC N1(C(C)=O)CCc2cc(N(C(=O)C(=O)N=c3[nH]nc(C4CCCC4)s3)CC)ccc21 N1(C(CC2CCC(=O)O2)=O)CCCC(NC(=O)COCc2cccnc2)C1 c1(C(=O)NCCC(C)N(C(=O)CSc2n[nH]c(O)n2)C)cc2cccc(F)c2s1 C12CCOCC1NC(=O)N2.c1(NC(=O)OC(C)(C)C)nonc1CC1CCCO1 c1(OCC)cncc(C(=O)N(C(CNC(c2ccnn2CCF)=O)C2CC2)C)c1 C1(C(=O)NC2(COC)CCCCC2)COCCN(C(C2(C)CC2C)=O)C1 N1(C(CC2CC(OC)C2(C)C)=O)CCC(NC(c2cc(Cl)n(C)n2)=O)C(C)C1 N1(C(c2cc(C)ns2)=O)CCC(C)(C)C1CNC(=O)Cc1cccs1 N1(c2nc(C)cc(OC)n2)CC2(CCOCC2)CC1CNC(C1CCCOC1)=O CC1(NC(C2CC2F)=O)CCCN(C(C2CC(O)C2)=O)C1 c1(C(=O)NCCNC(=O)NCc2csc(Br)c2)cccc(OC2CCCC2)c1 C1(C(=O)NC(C)C(C)(C)CO)(NC(c2oc(C)c(CO)c2)=O)CCC(C)(C)C1 n1(CC(=O)OCC)cc(C(=O)NCC(O)CN(C(=O)C(C)n2cncn2)C)nn1 N1(C(N(CCF)CC)=O)CCCC(CC2CC2(F)F)C1 N1(C(C(CC2C(C(=O)O)C2)(C)C)=O)CC2CCC1CN2C(=O)OC(C)(C)C C(=O)(C1=NOC2(CCNCC2)C1)N(C)Cc1n(CC2CCC(C)N2C)ncc1 C(CCCC(=O)NCc1ncnn1C)N(C(c1c(C(C)C)onc1)=O)C Cc1c(C(C)N(C(=O)C(C)S)C)cccc1-c1nn[nH]n1 C(CC(F)F)(C(=O)Nc1cc(N(C)C)cc(F)c1)N(C(c1n(C=C)nnc1)=O)C c1(NC(C2(C)CN(C(=O)Nc3ccccn3)C2)=O)nnc2ccc(Cl)nn12 C#CCC(O)C(=O)N(C1CCCN(C(=O)Cc2coc(-c3ccccc3)n2)C1)C CC1(C(N2CCC(CNC(c3cc(F)ccc3Cl)=O)C2)=O)CCC(F)(F)C1 CC1CCC(NC(C2CCC3(CC2)CC3)=O)CN1C(=O)C1=NOC(C(C)(C)C)C1 C1(CCC)CN(C(=O)CC2CC=CCN2C)CC1NC(c1nocc1C)=O C12(NC(C3N(CCC)CCC3)=O)COC(C1)C(NC(=O)CCC(=O)OC)C2 C(=O)(C(C(C)(C)C)NC(=O)CC(F)(F)CC)N1CCC(O)(CC)C1 N1(C(C(C2CCCCC2)OC)=O)CC2(CCN(Cc3sccc3C)CC2)C1 CC(C(=O)N=S1(=O)CCC2(CCCN2)CC1)C1CCS(=O)(=O)C1 Cc1ccc2scc(C(N3CCN(C(=O)CC45COCC(C4)C5)C(C)C3)=O)c2c1 C1(CNC(c2c(OC)ccc(Br)c2)=O)Cc2cc(C)cc(Br)c2O1 c1(C(N2C(CNC(C3(C(C)C)CC3)=O)CCC2)=O)cc2ccccc2[nH]1 c1(CNC(C(=O)OCC)C(O)c2ccc(Cl)cc2)cc(C)c(Cl)c(C)c1 N1(C(C(C2CCOCC2)C)=O)CCN(C(c2cnc(S)nc2)=O)CC1CO O=S(=O)(c1cccnc1NC1CCS(=O)CC1)NCCn1ncc2ccccc12 c1(C(=O)NC(C(=O)OC)(C)C(F)F)ccnc2[nH]c(C(F)F)nc12 C(=O)(C=CS(C)=O)NCCNC(C1CN(C(C2C(C)OCC2)=O)C1)=O c1(C(N2CC3CC(NC(c4ccc(CC)s4)=O)C3C2)=O)c(C)ccc(F)c1N Cc1cccc(CNC(=O)CC2CN(C(c3cncc(F)c3C)=O)CC2C)c1O N1(C(C=Cc2n(C)ncc2)=O)CCC(NC(=O)CO)C(CO)CC1 C(=O)(C1=C(C)CC(C)(C)CC1)NC1C(CO)CCN(C(C2C(=C)C2)=O)C1 c1(CC)ccc(C(C)CC(=O)NCC(O)CNC(c2coc(OC)n2)=O)cc1 c1(C(=O)NCCC(=C)CNC(c2ccnc(O)c2)=O)cc(S(C)(=O)=O)ccc1O C(=O)(CC(C)(O)C1CC1)NCC(C)CN(C)C(C1(N(C)C)CC1)=O C1(NC(C=CCOC)=O)CCN(C(C2(C(=O)C3CC3)CC2)=O)CC1F CC1OCCC1C(=O)NCC1CCCC1NC(=O)CCc1nccs1 C1(C(N(CCC(=O)NC(C2CCCC2)C#C)CC#C)=O)COCCN1CC C(C(C(=O)NC1CCN(C)CC1C)C(C)C)NC(C1(CCOC)CCC1)=O c1(CC(=O)NC2CC(CCNC(c3cc(OC)no3)=O)C2)cc(F)ccc1F C(C)(CC1CCCCC1)(C(=O)NC(C)CN(C(=O)Cn1nnnc1C)C)OC c1(C(=O)NCC2(OC)CN(C(C3(C)CCCN3C)=O)C2)ccc(F)c(C(F)F)n1 c1(C(=O)NC(C2(CNC(c3cn(CC)nc3)=O)CC2)C)ccc2c(c1)CN(C)C2 CC(C)C(O)CC(=O)NC1CCCN(C(c2coc(C(F)F)c2)=O)CC1 c1(C(=O)NC2CC(NC(C3(C)CCC(C)C3)=O)C2)n[nH]c2cccnc12 c1(OC)cccc(C(C)C(=O)NC2CCCCC2NC(c2cnc[nH]c2=N)=O)c1 CCC(C(=O)NC(C)C(C1CCCCC1)NC(c1cnsc1)=O)OC n1(CC(=O)NC2CN(C(C3(C(N)=O)CCC3)=O)CCC2O)cnc2c1CCCC2 c1(C(N(C2CCN(C(=O)CC(C)(C)OC)C2)CC)=O)c(C)nn(C)c1OC C=Cc1ccc(C(N2CC(NC(C3CN(C(N)=O)C3)=O)C2)=O)cc1 CN1CCC(C)(C(=O)NC2(C)CCCN(C(c3nscc3N)=O)C2)C1=O N1(C(C(C)CC2CC2)=O)CC(C(=O)NC(C)(C)CC2CC2)C(F)C1 CC(CC(=O)NCC(C)NC(c1cnn(-c2ccccc2F)c1)=O)C(F)F C1(COC)(NC(C2(c3cc[nH]n3)CC2)=O)CCN(C(=O)Cn2nc(C)cc2C)C1 C(=O)(CCC(C)CN(C)C)NC1(CNC(Cc2ccc(OC)cn2)=O)CCOC1 C(=O)(CCCC(C)CC)NC(CC#C)CC(=O)NCCCN1CCOC1=O N1(C(CCC#C)=O)CCC2(CC2)CC1C(=O)NC(C=C)C1CCC1 N1(C(c2c(N)sc(C)c2C)=O)CC2CCC(C1)C(NC(C1(C)CCNC1=O)=O)C2 Cc1ccc(C(N2CCC(C)C2CNC(=O)Cc2cc(Cl)ccc2F)=O)cc1Cl C(=O)(C(C)N=c1cc[nH]cc1)N1CCCN(C(C(C)C(F)F)=O)CCC1 C1(COC)(NC(=O)Cc2ccsc2)CCN(C(c2cn(C3CC3)cn2)=O)CC1 C#Cc1cccc(C(=O)NCC(C2(O)CN(C(=O)C=CC3CC3)C2)(C)C)c1C CC1(CNC(c2ccccc2C(N)=O)=O)CCCN1C(=O)COC1CC(F)(F)C1 c1(OC)nc(Cl)ncc1OC(=O)NC(=O)N(C)C CC1(C)CCN(C(C2CCC3(CC3)C2)=O)C1C(=O)NCC1=CCCCCC1 CCCCCC(F)C(=O)NC(CCCC)C(=O)NCCc1cc(CC)no1 c1(CNC(CC2(C)CCN2C(=O)COc2ccsc2)=O)n[nH]c2c1CCC2 C1(C(=O)NCC(C)C(=O)NCC(c2ccncc2)C)CCCCNC1=O N1(C(C(c2n(C)cnn2)(C)C)=O)CCN(C(C2(CF)CC2(F)F)=O)CC12CCC2 Cc1nc(C(=O)NC2CCC2NC(=O)COC2(C)CCCC2)c(C(F)(F)F)[nH]1 CC(C(C)(C)NC(c1cnn(-c2ccccn2)c1)=O)NC(=O)C(=O)N(C)C C1(C2CCCCC2)(NC(C2=NOC(C3(C)COC3)C2)=O)CC1 N1(C(C=CC=CC)=O)CC2C(C(F)(F)F)CC2(NC(=O)C2=CCCSC2)C1 C(=O)(CC(C)(C)C=C)N(C1CCN(C(c2ccc(F)c(CC)c2)=O)CC1)CC#C C1(CC(=O)NCC2N(C(c3cncn(C)c3=O)=O)CCC2)CCC2(CC1)COC2 C#Cc1ccc(C(N2CCC(NC(c3cc(F)ccc3F)=O)C(O)C2)=O)cc1C c1(CN2CCC(C(=O)Nc3c(OC)ncc(Cl)c3)C(O)C2)ccccc1[N+](=O)[O-] C1(C(N(CC(O)C2CCC2)C)=O)CCC2CCC1N2C(c1ncn(C)n1)=O O=C1NC(CN=c2ccnc(N3CCCCC3)[nH]2)C2(OCC(O)CO)CCC12 N1(Cc2cc(OC)c(I)cc2)CCC2(CC1)CC2C(=O)NCC1(C)OCCO1 C1(C(=O)OC)COCC1C(=O)N(C(C)C(N1CCCC1C1CCOC1)=O)C(C)C Cc1cc(-c2cn(C3CCN(C(c4c(C)ccn4C)=O)CC3)nn2)ccc1F c1(C(N(C)CCN(C)C(C2CCc3nccn3C2)=O)=O)cc(F)cc2nc[nH]c12 C1(CC)CN(C(c2ccsc2NC(C)=O)=O)CCC1NC(c1nnn(C)c1C)=O C(=O)(C(C)(C)CC(C)(C)C)NC(CC)CN(C)C(C1COC2(CO)CC1C2)=O C1(C(=O)NCC(C(C(=O)OC)F)C)CCN(C(=O)C=C(C)C(C)(C)C)C(C)(C)C1 C=CCC(C(=O)NCC1CCC(C(=O)NC(c2cn[nH]c2)C)C1)C(C)C n1(CC)cnc2[nH]c(=NCC3CC(=O)N(C(C)(C)C)C3)[nH]c(=NC3CCOC3)c12 c1(CN2C(C)(C(C)NC(C3CC(F)C3)=O)CC2)cccc(C(F)(F)F)c1F CC(C(=O)OC(C)(C)C)C(=O)N1CC2C(CNC(=O)CCC(=O)N(C)C)C2C1 C=CCC(CNC(=O)C(C1(O)CCC1)NC(=O)CC(CC)C1CCC1)CC(C)C N1(C(=O)NCCc2ccc(Cl)cc2C(C)C)CCCC1C1CCCO1 c1(C(C)=O)cc(NCCCNC(C2CCC(=O)N2)=O)ncn1 c1(CC(=O)NC(CCCNC(CC=C)=O)C)coc2cc(Cl)ccc12 c1(C(N2C(C)CC(CNC(C3CCC4(CC4)C3)=O)C2)=O)ccn2ncnc2c1 c1(C(=O)OCCc2ccccn2)ccc(NC(c2ccon2)=O)cc1 c1(OC)cc(O)c(CN(C)CC2CN(C(c3ccc(Cl)c(F)c3F)=O)C2)cc1Cl c1(C(N(CC(CC)NC(CC=CC=C)=O)CC)=O)cnc(O)c2cncn12 Cc1cccc(CC(=O)NCCCCN(C(=O)COc2cnc(Cl)cn2)C)c1 c1(-c2ccc(C)c(CO)c2)nn(C)c2ncccc12 C(=O)(C(CC)CCCC)NC(CCC)CNC(c1ccc(C)nc1O)=O N1(C(C23CCC(OC)C2C3)=O)CC(NC(c2cnc(C)cc2C)=O)CC(C)C1 N1(C(CNC(=N)N)=O)CC2CCC1CN2C(=O)C(=O)NC1CC1 c1(CNC(CC)Cn2cncn2)cc(OC)c(C)cc1F CC1CN(C(C2CCC3(C2)CC3(F)F)=O)CC2(CCN(C(C3CC3F)=O)C2)O1 N1(C(c2n[nH]c(C)c2C)=O)C(C)CN(C(c2cnccn2)=O)CC1C CN1C(=O)CN(CC(N2CC(NC(=O)CCCCN(C)C)C(F)C2)=O)C1=O C1(=CC(N2CC3C(CNC(=O)CN4C(=O)CCC4=O)(C3)C2)=O)CN2CCC1CC2 C(=O)(C#CC(C)(C)CNC(=O)C(C)CC(C)C)NCCC(=O)NC(CC)C c1(CC)cc(C(=O)OCC2CC2c2ccc(Br)cn2)c(Br)s1 N1(C(C(C)(C)F)=O)CC2CCC1C(NC(C1(c3ccccc3)CC(O)C1)=O)C2 C1(NCC2C(C(C)C)C=C2)CN(C(=O)OC(C)(C)C)CCC1CO Cc1ncn2ccc(C(=O)NC(C)(C)CN(C(=O)C3=CCCC3)C)cc12 N1(C(CC(=O)OCC)=O)CCCCC1C1CN(C(=O)C(C)(C)COCC)C1 c1(C(N2CC=CC(NC(CCCC#C)=O)C2)=O)ccn2c(C)cnc2c1 C1(C(N(CC(C)(C)CNC(c2ccnc(CO)c2)=O)C)=O)OCC2CCCC12 C1(OCCC)CCCN(C(=O)CCCCNC(c2ccnnc2O)=O)C1 N1(C(CC=CC)=O)CC2CC1CCC2NC(C1(CC)CCC(O)CC1)=O C1(C(N(CC(CN(C)C(c2n[nH]cc2[N+](=O)[O-])=O)O)C)=O)CCCCC(F)(F)C1 C1(C(=O)NCC2(F)COC2)COCCN(C(c2ccnnc2O)=O)C1 N1(C(C(C(C)C)O)=O)CCC(C2CC2)C1CNC(c1cccc2nsnc12)=O CCCC(CNC(c1cccc(O)c1F)=O)C(=O)N1CC(C)CC1CC C(C(C(=O)NC1(c2ncc(C)s2)CC1)C(C)(C)C)NC(CCCSC)=O C(CCCCC(=O)NCC(C)C1CCC1)NC(Cc1c(C)noc1C)=O C#CCCCC(C)C(=O)N1CC2=C(C1)CN(C(=O)C(C)(C)CF)C2 C(c1ccccn1)=CC(=O)NCC1CC(O)(CNC(C2(C3CC3)CCCO2)=O)C1 C12(C(=O)NCC(C)(CO)NC(=O)C#CC3CCOC3)CCCN(CCC1)C2 C(=O)(C1=NOC(C)C1C)N1C(C(N(CC)Cc2ccoc2)=O)C=CC1 C(=O)(C(=O)C(C)(C)C)N1CC2C(C(=O)NC(C3CCOCC3)C)(C2)C1 C(=O)(C(C)CC(F)(F)F)N(CCNC(c1c(C)n(C(C)(C)C)nc1)=O)C.C(C)(=O)O N1(C(CCC)=O)CCC(C(=O)NC2(C)CCN(C(=O)OC(C)(C)C)C2)CC1 c1(C(N(CCOCCN(C(C(CC)OC)=O)C)C)=O)ncc(OC)cc1F.C1CC1 c1(C(=O)NC2CN(C(c3ccnnc3)=O)CC3(CC3)C2)cnc2ncccc2c1 O=C(C(C1=NOCC1)N1CCCC1C1CC1(F)F)NCc1ccc(Cl)cc1 C(=O)(N1CCC(C(N2CC(CO)C2)=O)O1)c1nc(CCC)oc1 C(=O)(C(CNC(c1nc(C)oc1C)=O)CC(C)C)NC(c1nc[nH]n1)CC CCC(C)(C(=O)N1CCN(C(=O)CCc2ccnc(Cl)c2)C(C)C1)C(N)=O CC(C)C(C)(CNC(=O)CC1(N(C)C)COC1)NC(C1CC1(C)C)=O c1(C(C)NC(C2OCCC2CNC(=O)C(CO)N(C)C)=O)cccnc1O c1(C(N2C(CC(=O)N(C)CC3COCCO3)CC2)=O)ccnnc1O CCCCCCCCC(=O)NC1CCC(C)N(C(c2cc3c(ncn3C)[nH]2)=O)C1 CCC(C)C(O)C(C)C(=O)NC(CC(F)F)C(N1CCC2(CCCC2)C1)=O C1(C(N2CCC(CN(C(=O)C(C)(C)n3ccnn3)C)C2)=O)CCCC(C)(C)CC1 C=CCCCCNC(=O)C(C)(C1CCC1)NC(=O)C(C)N(C)C(C)=O N1(C(=O)C=CCF)CCC2(CCCN2C(C2SCCCS2)=O)C1 c1(C(=O)NC(C(=O)NC(c2nnc(O)n2C)C)C2CCOC2)ccnnc1O c1(C2(NC3C(c4n(CC)ccn4)OCC3)CCC2)ccccc1Br C12(CNC(C3(CC)CC3(F)F)=O)CC1CN(C(C1(CO)CCCCC1)=O)C2 C1(NC(=O)COC(F)F)CCC(F)(CNC(c2cncc(N3CCCC3)n2)=O)C1 c1(NC(c2ncn(C)c2)=O)sc2c(c1C(=O)Nc1ccc(Cl)cn1)CCC2 C1(CNC(c2cc(C(C)C)on2)=O)CCN(C(C2CC(F)(CO)C2)=O)CC1(F)F c1(C(N(CC(CNC(c2nccc(C)n2)=O)C)C)=O)cc(N)c(C)cc1C N(C1CCCn2ccnc21)C(C(C1CCCN(C(=O)CC(C)(C)C#N)C1)C)=O n1(CCOC)cc(C(=O)NCCC2CCCN2C(C2CC(CF)C2)=O)nn1 N1(C(C2(N(C)C)CC2)=O)CCC(F)(F)C(CNC(c2nc(Cl)sc2Cl)=O)C1 N1(C(Cc2c(C)ccs2)=O)CC(C)CCC1CNC(c1ccc(NC=O)cc1)=O N1(C(C2C(C=C)C2)=O)CC2CCC1CN2C(C1(C#N)CCOC1)=O n1(CC(=O)N(C(CCNC(C2N(CCC)CCC2)=O)C)C)cc(C#N)cn1 C(=O)(C(C(C)(C)O)OC1CC(C)(C)C1)NC(CCOCC)C Nc1ccc2nc(NC3(CNC(=O)CN4CCCC4)CCC3)sc2c1 CC1(C)CC(NC(C2(F)CCC2)=O)CCN(c2nccnc2C#N)C1 C(c1ccc2ncccc2c1)=CC(=O)NC1(CO)CN(C(c2ccc[nH]2)=O)C1 Cc1cc(C(C(=O)NCc2ccco2)N(C)CC2(O)CCOCC2)cc(F)c1 c1(C(N2C(CNC(C3C(CN(C)C)C3)=O)CC(F)C2)=O)cc2sccc2[nH]1 C1(C(=O)NCCNC(=O)CCc2nnc(-c3ccccc3)o2)CCCS(=O)(=O)C1 C1(NC(c2nc(CC)oc2C)=O)CC2CC1CN(C(c1cc([N+](=O)[O-])c[nH]1)=O)C2 CN=S1(=O)CCN(C(=O)C(c2ccc3c(c2)OCO3)=O)CC1 N1(C(c2cc(Br)ccn2)=O)CC2CCN(C(c3cccc(=O)n3O)=O)CC2C1 CCCCC(C)CCC(=O)NC(C)CN(C(=O)CC=CCc1ccccc1)CC N1(Cc2c(OCC)cccc2)C(=O)CN(CC(C)CC(F)F)C1=O C1(C(=O)NC2CCCC(OC)C2)CCOCCN1C(c1ccc(Cl)o1)=O c1(C(=O)NCc2nc(CC(=O)OCC)on2)cnn(CC)c1C1CCCC1 c1(NC(C(n2ncc(C)c2)C)=O)ccc(C(N)=O)cc1 C1(C(=O)OCC)(CC)CCCN1C(C12CC(CCO1)C2)=O CCCC(CNC(=O)Cc1ccsc1C)C(=O)NCCOCC C(=O)(C(CCNC(=O)C(C)OCC1CC1)OC)NCCC(=O)OCC c1(C(=O)NCC(CC)NC(=O)C(C)NC(C)(C)CC)cccc2c1C(=O)CC2 N1(C(C(CC)C)=O)CCCOC(CNC(c2cnc(CO)nc2C)=O)C1 C1(NC(c2ccoc2)=O)C2CC(O)C1N(C(c1cc(Cl)c(F)c(Cl)c1)=O)C2 N1(C(C(CN(C)C)O)=O)CC(NC(=O)COCP(C)(C)=O)CC1CO C1(C(=O)NC2(CNc3cccs3)CCC2)OCCCC1c1ccccc1 c1(OC)cc(C(=O)NCC2CCN2C(=O)CN2CCN(CC)CC2)cc(N)c1O C1(C(=O)NC(C2CCN(C(c3cc(C)on3)=O)C2)(C)C)CCc2n[nH]cc2C1C C1(NC(=O)CCNC(C2CNC(=O)C2)=O)CC2C=CCC(C1)C2 C1(NC(C2C(CC)OCC2)=O)CCCN(C(C23CC2CNC3=O)=O)C1 Cc1ccncc1COC(C1CC=CCC1NC(=O)OC(C)(C)C)=O C(CN=c1ccn2ncc(I)c2[nH]1)c1ccc(C)c([N+](=O)[O-])c1 c1(C(=O)NCCCC(C)(C)NC(COCCN(C)C)=O)ccc(O)c(=O)cc1 c1(OC)ncnc(C(N2CCC(NC(=O)CSC(C)C)C23CC3)=O)c1F Cc1nc(CN2CCCC(C(=O)OC(C)(C)C)C2)c(C)s1 Cc1ccnc(NC(C)(CCCO)c2nnnn2CC2CCCO2)n1 C1(CCCNC(c2cn(CCO)nn2)=O)CCCCN1C(=O)C=CC1CC1 c1(C(N2CCC(CNC(CN(C(COC)=O)C)=O)C2)=O)c(C)oc2ccccc12 Cc1[nH]nc2c1CCC(C(=O)NCCCNC(C1CCN(C3CC3)C1=O)=O)C2 C1(C(=O)OCC)CC(C)N(Cc2ccc(Br)cc2OCC)C(C)C1 C1(CC)CN(C(C2CC2C)=O)CCN1C(c1cc(C2CCCC2)nn1C)=O C1(NC(C(c2cn(C)nc2)=O)=O)CCCC(NC(=O)COC2CC=CC2)CC1 C1(O)(CNC(C2C(C(=O)OC)C2)=O)CCCN(C(=O)CC2(OC)CCC2)C1 CC1CC(NC(=O)CC2=CCCC2)CN(C(=O)CCCN2C(=O)CCC2=O)C1 CC1CN(C(C2CCC2)=O)CC(CCNC(c2cnn(-c3cccnc3)c2)=O)O1 C1(C(C)NC(=O)Cc2ccns2)CCN(C(=O)CCC2CCC2)C1 N1(C2CCC(=O)CC2)CCN(C(C2CCN(CCF)CC2)=O)C(=O)C1 Cc1cc(CCC(=O)NCC(C)CNC(C2CCC2(C)C)=O)on1 C1(NC(C(c2ccc(Cl)cc2F)C)=O)CC2CCC1N2C(C1CCOC1)=O C1(CN(C(C(C)Cn2ccnc2)=O)C)CN(C(c2c[nH]nc2C(F)F)=O)CCO1 c1(C(N2CC(CC(=O)NC(CC)CO)C2)=O)cc(C(F)(F)F)cc(F)c1 c1(C(=O)NCC2(F)CC(NC(C3(C#C)CCC3)=O)C2)c(C)c(C)c(C)c(C)c1C C(=O)(C(CC(C)(C)C)NC(=O)C=Cc1cncn1C)NCC(=O)N(C)CC c1(C(=O)NC2CCCS2)nnc(C)cc1NC(C1CCC(CNC(C)=O)CC1)=O C(CCCCC(=O)NC1C2CC3C1C3C2C(=O)NCC1(SC)CC1)OC c1(C(N2CCOCC2)C(=O)NCCSC)ncccc1Cl C1(CCNC(C2C(C=C)C2)=O)CN(C(=O)COCc2ccnn2C)CCS1(=O)=O N1(C(c2cnn(C)c2Cl)=O)CC(NC(c2nncs2)=O)CC1(C)C N1(C(C(COC(C)=O)C)=O)CCOC(CCC(=O)NC2(CCO)CCCC2)C1 c1(C(C(=O)NCCCCCC)N(C2CCCOC2)CC)cccc(Cl)c1Cl N1(C(CC2N(C(c3c(C)ocn3)=O)CCC2)=O)CCCC(OC2CCC2)C1 c1(C(=O)NC(CC2CCN(C(C3(C#C)CC3)=O)CC2)C)cccc(F)c1CC n1(CCC(=O)OC)cnc2c(cnn2C)c1=O.C(=O)(C1(N)Cc2cn1nn2)OC N1(C(COCCC)=O)CCN(C(=O)Cc2cccc(Br)c2C)CC1CO N1(C(CC2C(C)CCN(C(Cc3ccn(CC)n3)=O)C2)=O)CC2(COC(=O)C2)C1 C(C(C)(O)CC(=O)NC1CCCC(C(=O)NC2CCC3(CC2)N=N3)C1)OC C(=O)(C#CC1CCC1)N1CC(CCNC(C2(C)CC(C(F)(F)F)C2)=O)C1 Cc1ccoc1C(N1CCCC1CNC(=O)CCNC(=O)CC1CCCCC1)=O N1(C(CC(C)(C)C#N)=O)CCC2(CC2)CC1C(=O)NCc1cccc(O)c1F Cc1cc(F)c(Cl)cc1C(=O)NC1(C)CCC(NC(=O)C2=CCCOCC2)CC1 C1(C(=O)NCC(C)(C2CCC2)NC(c2nn(CC)c(C)c2)=O)COC(C)(C)CO1 CC1COCCN(C(=O)C(F)(F)F)C1.S1(=O)(=O)CCN1 C(=O)(CCC(=O)c1ccc(Br)cc1)NC(CNC(=O)C(F)=CCCF)CO C(C(=O)NC1CC(F)(F)C1)(C1=CCSC1(C)C)N(CC(N1CCCC1)=O)CC n1(CC)ncc(I)c1C(=O)NCCNC(c1cccc(N(C)C)c1)=O C1(C(=O)NCC2CCN(C(c3c(C)nc[nH]3)=O)C2(C)C)CCCCCC1(F)F C(=O)(C(C)C(O)C(C)C)N(C1CCN(C(c2cc(CC)[nH]n2)=O)C1)CC C(=O)(CCN=c1ccc(C)c[nH]1)N1C(CCNC(CCCCC)=O)CC(OC)C1 c1(C(=O)NCC(C)CN(C(=O)C(O)C2CCC2)C)cccc(C(C)(C)C)n1 c1(C(CNC(=O)CCNC(C2CCOCC2)=O)N(C(CCC)=O)C)ccccc1 C1(C(=O)NCCCOCCCC)C2CCC(C2)N1Cc1ccc(C#N)s1 c1(CN2CC3C(C(=O)Nc4c(CO)ccc(OC)c4)(C3)C2)c(Br)cc(Br)cc1Br C1(C(=O)NCC2(CO)CCCC2)CC2CC2N1C(=O)Cc1cnns1 c1(CC)cncc(C(=O)NC2(C3CCCN3C(c3ccnnc3)=O)CC2)c1 CCC(COC)C(=O)NCCCN(C)C(c1cnn(CCC#N)c1C)=O c1(C(N2C(C)(C(=O)NCCCS(C)(=O)=O)CCC2)=O)cnn2cccc(F)c12 c1(NC(=O)N(C(CCOCCOC)C(C)(C)C)C)ccc2cc(O)ccc2c1 CN1CC2CN(C(C3(c4ccccc4)CCC3)=O)CCN2C1=O N1(C(c2cnn(CC3CCCCC3)c2)C(=O)NCCCF)CCOCC(CO)C1 C1(C)(C(N(OC)C)=O)CCCN1C(c1ccccc1C)=O c1(-c2c(C)ccc(CO)c2)cc(C(N2CC(NS(C)(=O)=O)C2)=O)c2cc[nH]c2c1 c1(CC(=O)NCc2ccc(C)cc2OCC(F)(F)F)ccc2c(c1)NC(=O)C2 N=c1ccc(C(N2CC3C(NC(c4csc(-c5nc[nH]n5)n4)=O)C3C2)=O)n[nH]1 C1(C(=O)NCCN(CC(C)O)C(=O)Cc2csc(C(F)(F)F)n2)CC(C)OC(C)C1 C1(C(C)C)CN(C(=O)CC2CC2)CCC1NC(C1(N(C)C)CCCSC1)=O C1(Nc2c(NC)c[nH]c2C)CC2CCC(C1)N2CC(=O)NCc1ccccn1 c1(C2C(C(N3C(CNC(c4csc(S)n4)=O)CC3)=O)C2)c(F)cccc1F CCN=c1[nH]c(C(N2CCOC(CCNC(=O)COC3CC(F)(F)C3)C2)=O)cs1 N1(C(CCCC)=O)CC23CCCC2(C1)CN(C(=O)CCCCCN=[N+]=[N-])C3 c1(C(=O)NC(CCC)C(=O)NC2CN(CC)CC2C)ccnc(F)c1Cl c1(CNC(C(C#C)(C)C)=O)cc(C#N)ccc1Cl C(CC(=O)N(CCN(C(=O)C(C)CO)C)C(C)C)(C1=CCCC1)OCC C1(C(=O)NC2C(CNC(=O)C=Cc3cncc(F)c3)CC2)CCn2nncc2C1 CC(CCCC(=O)Nc1cncc(F)c1)NC(c1ncc[nH]1)=O c1(CNCC23C(CN(C(c4n[nH]c(C)c4C)=O)C2)C3)cccc(F)c1C#N c1(CC(C)C(N2C(C(=O)NCc3cccc(Cl)n3)CC3CC23)=O)ccc(O)cc1 c1(N(C2CN(S(=O)(=O)C3CCCCC3)C2)C)nccc(=NC(=O)c2sccc2N)[nH]1 N1(C(C23C(CCN(C(=O)C=CC(F)(F)F)CC2)C3)=O)CCC2C(=O)NCC2C1 C1(CC(=O)N(C(C)C)C2CC2)CCN(C(=O)CC2CC3(CC3)CO2)CC1 c1(C(N(CC(CC)NC(c2csc(C)n2)=O)C)=O)nc(C(C)C)oc1C C1(NC(c2c(CCC)n(CC)nn2)=O)C(CNC(=O)C=C(C)Cl)CCC12CCC2 c1(C(N2CCC2C(c2cn(C(C)(C)C)nn2)N2CC3CC3C2)=O)nc(=N)cc[nH]1 C1(C(N(CC(=O)NC(C)Cc2cnc[nH]2)C2CCC2)=O)CC2(CC2)C1 c1(NCCCC(=O)NCCCN(C)C(c2cc[nH]n2)=O)ccc([N+](=O)[O-])cc1 Cc1nccc(F)c1NC(=O)Nc1sc(-c2ccccc2)cc1C(C)C N1(C(CCC(=C)Cl)=O)CCN(C(c2cn3c(n2)SCC3)=O)CC1C Cc1oc(=O)oc1COC(C1CCCC1CC(=O)OC(C)(C)C)=O CC1SCCCC1C(=O)NCC1CC(C(=O)NOCC2(C)CCC2)C1 c1(C(N2CC3C(CNC(=O)Cc4ccsc4)C3C2)=O)c(Cl)ccc(Cl)c1O C1(CC(N2CC(O)(C(C(=O)N(CC=C)CCO)F)C2)=O)CCOC1(C)C N1(C(CSc2cccc(C)c2)=O)CCN(C(=O)Cc2sc(C)nc2C)C2CC12 c1(C(=O)NCC(C(=O)NC2COCC2CO)N(C)C)ccc2c(c1)CC2 N1(C(CN2CCC(C)CC2)=O)CC(C)(C)OC2(C1)CN(C(C1OCCC1C)=O)C2 c1(NC(C2(CCNC(=O)Cc3ccsc3)CC2)=O)csc(Cl)c1 C1(C(=O)NCc2cc(C)[nH]n2)CC(C)CN(C(c2occ3c2CCC3)=O)C1 CN1CC2CCN(C(c3csc4ccccc34)C(=O)NCC3CCCO3)C2C1 N1(C(c2nccc(OC)c2OC)=O)CC(C(=O)NC2CC2)C2(CCC2)C1 N1(C(C2(OC)CCSC2)=O)C2CCCC1CC(NC(=O)CSc1n[nH]c(O)n1)C2 S(=O)(=O)(c1ccc(NCCC2CCSCC2)c(F)c1)NCC(CCC)OC.OC N1(C(C(CC2CCC2)OC)=O)CC2CC1(C(=O)NCC(C)C(F)F)C2 N(C1COc2ccc(F)cc21)C1CCC(C)NC1=O N1(C(C(CC2CC2)NC(C2CC(O)(CC#C)C2)=O)=O)CC(CN(C)C)C2(CC2)C1 C(=O)(NN1CCCCC1C)c1cccc(NC(=O)OC)n1 C12(C)CCCN1C2=O.C(C(C(=O)NCc1cnns1)NC(C)=O)OC c1(NCC(CCC)O)ncccc1S(=O)(=O)NCC1CCC1c1ccc(F)cc1 N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCC2C(C1)CN2C(C1CCS1(=O)=O)=O c1(C(=O)NC2CCN(C(c3nc(C)sc3C)=O)CC2CO)cc(C)c(N)cc1Cl C=C(C)CCCC(=O)N1CC(NC(C2CCCN2N=O)=O)CCC1C N1(C(c2ncc(C3N(C(=O)OC(C)(C)C)CCC3)s2)=O)CC2CC(O)C2C1 c1(C(=O)NCCN(CCCN(C)C)C(c2c(OC)n[nH]c2)=O)cnn2c1OCC2 c1(-n2cc(C(CNC)=O)nn2)ccc2[nH]c(C(=O)OC)c(C)c2c1.N(C)C CC(CN(C)C)CCC(=O)NC1(CF)CCN(C(=O)CN2CCOC2=O)C1 c1(C(=O)N=c2cc[nH][nH]2)cnc2cccc(Br)c2c1 C1(OC)CC2CC1CN(C(=O)C(CNC(=O)CCCCN(C)C)CC(C)C)C2 c1(C(=O)NC2CN(C(c3c(C)cn(C)c3)=O)C(C)CC2)cn(C)c2ncccc12 C(CC(=O)NCCn1cc(C)cn1)(C1CC1)NC(CC1(OCC)CCC1)=O C1(C(=O)NC2C(C)CN(C(C3CCOCC3)=O)C2)CCn2ccnc2C1 Cc1ccc2cc(C(=O)NCCCN(C)C(c3cc(=O)c(C)c[nH]3)=O)[nH]c2c1 C(=O)(CC(C)(C)CC(=O)NC(C)CC(C)NC(=O)CCc1cccnc1Cl)OC C(=O)(C(F)C1=CCCCC1)NCC1CCN(C(C2CCCCN(C)C2=O)=O)C1 C1(n2c(C(CCCOC)NCC3(CC)CC3)nnn2)CC(NC(=O)C2CC2)C1(C)C c1(C(=O)NCC2C(NC(COCCC=C)=O)COC2)cc(N)ccc1F C1(C(=O)NC2C(SC)CN(C(c3coc(SC)c3)=O)C2)COc2ccccc2C1 c1(C(=O)NCC2(O)CCN(C(c3cnc(Cl)s3)=O)C2)nc[nH]c2nccc1-2 C(=O)(C1CCc2ccccc21)NC(CNC(C(C1CC1)OCC)=O)CC(C)C C(c1nc2ccccc2o1)=CC(=O)NCC(CO)NC(=O)COCC1CC1 N1(C(C(CC)COC)=O)CCN(C(c2ccsc2OC)=O)CC(O)C1 N1(C(C(CC)NC(N)=O)=O)CC(C)(C)CC1CC(=O)NC1CC(CN(C)C)C1 C1(C(C)(C)NC(CSCC#C)=O)CCN(C(C2CCCCO2)=O)CC1 C1(CNC(CC(CSC)(C)C)=O)CN(C(=O)C(C(C)C)SC)CC2(CCC2)O1 C1(CNC(C2C(CC)C2)=O)CCCN(C(C2CC2c2cccnc2)=O)C1 N=c1[nH]c2c(s1)CCCC2C(=O)NCC(CO)NC(=O)C=Cc1ccoc1 c1(CC(=O)N(CCN(C(Cc2nc(COCC)sc2)=O)C)C)ccc(OC)nc1 c1(C(=O)NC(CCNC(C=CC)=O)C)cnoc1-c1ccoc1 N1(C(COCCOCCOC)=O)CCN(C(C2CC23CC(O)C3)=O)CC1CO c1(C(=O)NCC(=C)CCNC(c2cc[nH]c2C)=O)ccc(CC2CCC2)cc1 N1(C(c2cc(OC)cc(OC)c2)=O)CC(NC(C2CCC2)=O)CC2(CCC2)C1 C1(NC(=O)Nc2c(F)cc(C)c(F)c2)CCOC2(CCSCC2)C1 N1(C(CC(=O)NCC)=O)CCC2(CC1)COCC(CNC(C1CCOC1)=O)O2 c1(SC)ccc([N+](=O)[O-])cc1NC(N1CC2NCCOC2C1)=O c1(C(C)C(=O)NCC2(NC(c3ccc(F)cc3)=O)CCOC2)nc(F)ccc1Cl O(CP(C)(C)=O)CC(=O)NC(C1CCCCC1)CNC(C1C(CCC)C1)=O c1(C(N(CCNC(c2scc(C(C)=O)c2)=O)C)=O)n[nH]c2c1CCCC2 c1(CC(C(N)=O)NC(C2C(NC(c3c(C)scc3)=O)CCC2)=O)ccc(O)cc1 C(=O)(C1=C(Cl)CCC1)NCCN(CC(C(N1CCN(C(C)C)CC1)=O)O)C N1(C(CCc2onc(CCC)n2)=O)CCC(NC(c2snnc2C)=O)C(F)C1 c1(SCC(=O)NCC2C(C(=O)NC(CSCC(=O)OC)=O)C2)nc(C)cc(C)n1 C(=O)(CS(=O)(=O)C(C)C)N1C2C(NC(CCCC=C)=O)C(CC2)C1 C1(C(=O)NCC(=CC(N2C(CC)COCC2)=O)C)CC(C)(C)CN1C c1(C(N(CC(CNC(CC(C=C)CC)=O)O)C)=O)cc(Cl)c(C)cc1Br C1(N(C(C2C(CC)C2)=O)C)CCCN(C(C2(n3cccn3)CC2)=O)CC1 c1(OC)cc(C(N2CC3(C2)CN(C(C2(C)CC2)=O)C3)=O)c([N+](=O)[O-])cc1OC C12(C(=O)NC3CN(C(c4c(C)sc(C(F)(F)F)n4)=O)CC3C)CC1COC2(C)C c1(COC(CONCC)=O)nn(C)cc1C#C[Si](C)(C)C C(C)(CC(=O)NCC1CCCN1CC(=O)N(C)C(c1nc(C)no1)C)OC N1(C(C2OCCN(CC)C2)=O)CCN(C(c2snnc2C)=O)CC(CO)C1 N1(CC(=O)N(C(C)C)C(C)C)CCOC(CNC(=O)CCc2cn(C)nc2C)C1 N1(C(CC2(C=C)CCC2)=O)CCC(C)(NC(=O)C(c2ccccn2)C)C1 c1(C2(C(N3CC(N(C(C=C4CCC(C)C4)=O)C)C3)=O)CC2)ccc(F)cc1Br C(=O)(C1=CC2CCC(C1)N2)NC(C(=O)NC1CC(CC(C)C)C1(C)C)=O c1(C(=O)NC2(C)CN(C(c3ccn4nccc4n3)=O)C2)cc(O)c2ccoc2c1 N1(C(C2N(C)C(=O)OC2)=O)CCS(=O)(=O)C(CCNC(c2ccc(O)nc2)=O)C1 CC(C)C(C(=O)CN1CCCC(CC(F)F)C1)OC(=O)NC(C)(C)C C1(C(N2CCC(CC(C)NC(C(=O)NCC)=O)CC2)=O)CS(=O)(=O)CC(=O)N1 C(CC(C)C(=O)NCC1CC1NC(c1cnc(C2CC2)o1)=O)=CCC Cc1ccc(C(CNC(C2(C)CC2(Cl)Cl)=O)NC(c2cccnc2)=O)cc1 C1(C(NC2CCn3ccnc32)=O)CCCC(C2CCC2)C1 c1(CCC)cc(C(N2CCC(CN(C(=O)C3=CCCC3)C)C2)=O)sc1C c1(C(=O)NCC2C(NC(C=C(CCC)C)=O)CC2)cc2c(C)ccc(Cl)c2[nH]1 c1(C(N(CCn2cc(C3(O)CCOCC3)nn2)CC)=O)cc(Cl)cc2[nH]ncc12 N1(C(c2cccc(CC)c2F)C(=O)NCC2CCOC2)CCCC(C)(C)CC1 c1(CCCC(=O)NCCN(C(C2(Cl)CC2)=O)Cc2ccccc2)ccc(O)cc1 C(=O)(CCS(C)(=O)=O)NC1CC(N(C)C(c2n[nH]cc2Cl)=O)C1 C(=O)(C1=CC2(CN(C(c3csc(Cl)c3)=O)C2)OC1)N1CC(C)(C(F)(F)F)C1 C=CCC(CNC(c1cn(C)c(C)n1)=O)C(=O)NC1CCCCNC1=O O=C(CCN=c1[nH]c(=NCCCF)[nH]c2c1CCCCC2)Nc1ccccc1 N1(C(CC=CCC)=O)CCC(NC(c2coc(S(C)(=O)=O)c2)=O)C12CCC2 Cc1nc(F)ccc1CNC(=O)CC1CCCC1NC(C1CC(O)C1)=O C1(CNC(C(c2ccc(Cl)cc2)OC)=O)CCC(C)(C)CN1C(c1ccoc1)=O c1(-c2ccc(C)cc2)nc(C)cc(=NC2CN(C(=O)C(F)C(C)(C)O)C2)[nH]1 N1(C(c2c(SCC)nccn2)=O)CCC2C1CCCN2C(=O)CCC(C)(F)F N1(C(c2c(C)nn(C)c2C(F)F)=O)CC(NC(c2cccn2C)=O)C(C2CC2)C1 CC(C)(F)CCC(=O)NC12CC(C(N3CC(CF)OC(CF)C3)=O)(C1)C2 N(C1CCOc2ccc(Br)cc21)C(=O)NCC1C(=O)OCCC1 n1(C(C)(C)C)nccc1C(N1CCC(OCCNC(=O)Cc2csnn2)C1)=O C1(CNC(CCc2cccc(OC)c2)=O)C(C)CCCN1C(c1coc(Br)c1)=O C1(NC(CCC(C)(F)F)=O)CN(C(=O)CC2CCCCC23CC3)C2(CCCC2)C1 C1(NC(c2cccc(N)c2O)=O)CCCCCN(C(=O)CCCC2CC2)C1 N1(C(C2CCN(C)CC2)=O)CC(C(N2CCC(CO)C(C)(C)C2)=O)CC12CCC2 c1(C(c2n(CCN3CCCC(CSC)C3)nnn2)NC(C)=O)cccc2c1OCC2 Cc1cc(C(=O)N(C2CCC(NC(c3ccnnc3C)=O)CC2)C)nc(C)c1 C(=O)(CC(F)(F)C(F)F)NCCC(C)N(C)C(C1C(F)(F)C12CC2)=O C1(NC(COC(CC(C)C)C)=O)CC2(C1)CN(C(=O)C=CCN1CCCC1)C2 N1(C(C(C)C#N)=O)CCC(NC(C2CCC(c3ccccc3)C2)=O)C(C)(C)C1 C(=O)(C1=CCC2(COC2)OC1)NC(CCCNC(CSCc1nc(C)[nH]n1)=O)C N1(CCCCCNC(C2CC3C=CC2C3)=O)CCN(C(=O)COCC(F)F)CC1 N1(C(c2cc(C)c(Cl)cc2)=O)CC2OCCN(C(=O)CC3CCCN(C)C3)C2C1 C1(C(=O)NC2CCCCC2CNC(=O)COCCC(C)C)(OC)CCOCC1 CC(CN(C)C)CCC(=O)N(CCC(=O)NCC1(F)CCN(C)C1)C1CC1 C(=O)(CCC(C)(C)NC(C1C(C(F)F)C1(C)C)=O)Nc1cn(CCC)nc1 c1(C(=O)NCC#CCNC(C=CC(CC)=CC)=O)nnn(C(C)C)c1C c1(N(C)CCN2CCCCCC2)[nH]c(=NCCc2cn[nH]c2)nc2c1cnn2C Cc1csc2ncc(C(=O)NCC3(NC(=O)C(C)CC4CC4)CCCC3)n12 c1(OC)cc(CC(=O)NC(C)(C)C(C)NC(=O)CCc2ccsc2)c(F)cc1O CP(C)(=O)C1CCC(C(=O)OCc2cc(-c3ccco3)on2)C1 C(CCC(c1ccccc1)NC(=O)C(C)NC(C)(C)C)NC(C=C(CC)CC)=O C(C(=O)NCC(C)C)(C1CCSC1)N(CCC)C C=CCC(C)(C)C(=O)NCC1CN(C(=O)C(F)(F)CO)CC1O C1(C(C)C(=O)N(C)C2CC2)CCCN(C(=O)C(C)(C)N(C)C)C1 C(=O)(CCCC(=O)NCC)NCCCC1OCCN(C(C(COCC)C)=O)C1 Cc1cc(C(=O)NC(CNC(=O)C(C)O)C2CCC2)c2cccc(C)c2n1 C1(NC(c2cc(Cl)c(Br)c(Cl)c2)=O)CCc2nc(NC(=O)C(F)F)sc2C1 CC1(C)CN(C(c2ccc(Cl)s2)=O)CC1NC(=O)C1=NNC(C(F)(F)F)C1 c1(C(C(=O)N(c2cncc(N)c2)CC)(C)C)cc(Br)ccc1C N1(CC(N2CC(O)(CNC(c3ccc(Br)o3)=O)C2)=O)Cc2ccccc2C1=O CCCCS(=O)(=O)NCC(N1CCOC(CNC(=O)C(C)(CC)OC)C1)=O C1(CNC(c2n(CC)ncn2)=O)CCC(C)N(C(c2c[nH]cc2Br)=O)C1 C1(N(C(C=CC=CCC)=O)C)CCCCN(C(C2CC=C(C)CC2)=O)C1 C1(CC)C(NC(=O)C=Cc2ncc[nH]2)CCN1C(C1CCS(=O)CC1)=O Cc1nc(=NC2CN(C(c3cc(C(N)=O)cs3)=O)CC(C)(C)C2)s[nH]1 N1(C(C(CCC)C#N)=O)CCC2(CC1)CC2CNC(=O)Cn1cc(C)cn1 N1(C(CC2CC(C)(C)C2)=O)CC(F)(F)CC1CCNC(C1CC1CF)=O N1(Cc2c(C)cccn2)CC2(C1)CN(c1ncc(Br)cn1)C2 C1(C(N2C(C(N(CCCCCC)C)=O)C(O)CC2)=O)CCC2(CC1)CC2 Cc1ccc(Cn2nc(-c3nc[nH]n3)nc2CC2CCCOCC2)cc1 C1(N(C(=O)C(C)=CC(C)(C)C)CC)CCCN(C(c2ccc(N)c(N)n2)=O)CC1 C1(CNC(C2C(NC(c3nc(C)oc3)=O)CC=CC2)=O)CCC(C)(C)CC1 C1(C2CN(C(=O)CC34CCCN3CCC4)C2)(NC(CC(CC)C)=O)CC1 C1(NC(N2CCNC(c3cccc(F)c3)C2)=O)CCCC2(CC1)CC2 Cc1ccc2nc(C(N3CC(CN(C)C(c4ccnn4C(F)F)=O)C3)=O)cn2c1 N1(C(C2(C#N)CC(C)C2)=O)CCC(NC(=O)CC2(C)CCCC2)C(C)(C)C1 C1(CNC(CC2CCN(C(C34CC(CCC)(C3)C4)=O)C2)=O)CC(=O)N(CC)C1 C1(NC(=O)OC(C)(C)C)CN(C(=O)NCCc2cc(Cl)cc(Cl)c2)CC1C1CC1 C(=O)(CC(C(C)CC)NC(c1cncc(OC)n1)=O)Nc1cccc(CC)c1F c1(C(N(C)CC2CN(C(=O)CC3CCSCC3)C2)=O)ccc(C(F)(F)F)cc1 c1(C(N2CCC(CNC(C(C(C)C)N(C)C)=O)CC2)=O)cnn2c(=O)cc[nH]c12 C(N=c1[nH]nc(C(N)=O)s1)C1C(NC(C2(C)CNC(=O)C2)=O)CCCC1 N1(C(=O)C2=CCCCC2)CCC(C2CCCN(C(C3COCCO3)=O)C2)CC1 Cc1ncnc2c1CC(C(=O)NC1(CCNC(=O)C(CO)N(C)C)CC1)CC2 C1(C(=O)NC(C)(C(N2CCC=C(Cl)C2)=O)C2CCC2)CCCCC(=O)N1 C(=O)(N=c1ccn(CC(F)(F)F)[nH]1)N1CCC(C(C)C)C1 N1(C(CC)=O)CCC(C(=O)OC)(CC)CC1.c1(C)nn[nH]n1 C1(O)(C(C)NC(CCCc2scc(C)n2)=O)CCN(C(=O)CSC(F)(F)F)CC1 c1(OC)ccc(-n2nc(Cc3cccnc3)nc2C(O)CC(F)(F)F)cc1 S(=O)(=O)(C1CCOC1)Nc1cc(C(=O)OC)nn1-c1ncccc1Cl C1(CC)(CO)CCN(C(C2(C)CCCN(C(C3CC(C)=NO3)=O)C2)=O)CC1 c1(OC)ccc2cc(C(N3CC(CNC(=O)C(C)O)CC(C)(C)C3)=O)n(C)c2c1 C=CCCC(C(=O)OC)NC(c1cc(OC)c(-c2cc(F)cc(F)c2)cn1)=O c1(CC(=O)NCC2N(C(CCNC(=O)NC)=O)CCC2)ccc(C#N)cc1 N1(C(c2cc(C)[nH]c2)=O)CC2(CC2)CC1C(=O)NCCc1ccon1 CC1CC(C(=O)NC(C)CN(C)C)N(C(C2CN(c3ncccn3)CCO2)=O)C1 Cc1ccc2nc(C(=O)NC(C)CN(C)C(C3CCC4(C3)N=N4)=O)cn2c1 CC1CCC2(CCC2)CN1C(=O)NC1CC1(c1ccc(Br)cc1)C c1(OC)ncc(C(=O)NCC2CCCCCN2C(=O)CCNC(C)=O)cc1C C1(CNC(C2(S(N)(=O)=O)CC2)C)CC2(C1)CC(F)C2 Cc1cnn(CC(=O)NC2CCC(CNC(C3CCOC3=O)=O)C2)c1 CCC(C)C(CC(=O)N(CCC(C)OC)C)NC(=O)C(O)CC(N)=O n1(CC(=O)NC(CC(C)C)c2cccs2)ccc2ccc(F)cc12 C1(CNC(c2c(C)snc2)=O)CN(C(C2CC2C(=O)OC)=O)CCN1C c1(NC(C)CC2CCCC2)ncccc1S(=O)(=O)N1CCCC1c1ccncn1 N1(C(c2c(N)nccn2)=O)CCOC2CN(C(=O)CNc3ncccn3)CC12 c1(NC(C2CC(CNC(c3csc(C(F)(F)F)n3)=O)C2)=O)cccc(F)c1F Cc1nc(CC(C)C)c(C(=O)NC(C)C(CO)NC(=O)CSC(F)(F)F)s1 N1(C(C(CC)n2cncn2)=O)CC2CCN(C(=O)Cc3ccccc3C)CC12 n1(CC)ccnc1C(=O)NCCCCCN(C(=O)CC1CC1(Cl)Cl)C c1(C(=O)NCC(C2CCCC2)NC(C(C)CF)=O)c[nH]c2ccncc2c1=O C1(C(N(CCN(C(=O)CC(C)N2CCCC2=O)C(C)C)C)=O)CCCC(C)(C)O1 C(CC1=CCN(C(c2csnc2Cl)=O)CC1)NC(c1c(OC)ccs1)=O C(=O)(CC(=O)NCC(CNC(=O)CC1CCCOC1)CO)OCC c1(OC)cccc(C(C)=CC(N2CCN(C(c3ccc(C)s3)=O)C(C)C2C)=O)c1 CN1CCC12CN(C(C13CC(CN1C(C1CCCCC1(C)C)=O)C3)=O)C2 N1(C(=O)CCNC2(CO)CCC2c2cccs2)CCNC(c2ccc(Br)cc2)C1 N1(C(C2CCC(C)(C)OC2)=O)CCCC12CCCN(C(=O)C=CC=C(Cl)Cl)C2 c1(CCC(=O)NCC2CN(C(C(C=C)(F)F)=O)CC2C)ccc(Cl)c(OC)c1 N1(C(C(C)OCC)=O)CCC(NC(c2cnc(F)c(Cl)c2)=O)C(CC)C1 c1(OCC)ncc(C(=O)NC(CN(C(=O)CC2CC2(C)C)C)CC)s1 N1(C(CC=CCC)=O)C(CNC(C2CC(n3ccnn3)C2)=O)CC2CCCC12 CC1CN(C(c2cc(Br)ccc2O)=O)CCN1C(c1cc(F)cn1C)=O C(CCS(C)=O)(C(=O)N1CC2(C1)CN(C(C1(c3ccncc3)CC1)=O)C2)N(C)C c1(OC)ccnc(C(=O)NC(C)C(CO)NC(=O)C(C)P(C)(C)=O)c1OC N1(C(c2c(CC)onc2C)=O)CCN(C(=O)C(C)CF)C(c2ccccn2)C1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC(CO)C(NC(=O)Cn2cnc(C(N)=O)n2)C1 N1(C(C2N(C(C(C)NC(=O)OC)=O)CCC2)=O)CCOCC2(CC2)C1 C1(NC(CC(CC)C2CCC2)=O)CN(C(c2cc(C)cc(C)c2)=O)CCC1F C(C(CNC(=O)NC1C2COCC12)C(F)(F)F)NC(=O)CCc1ncccn1 c1(C(=O)NC(C)CN(C)C(C2CCC(=O)N2)=O)cncc([N+](=O)[O-])c1 c1(C(N(CC(C)O)CC)=O)ccc(CNC(=O)CC2CC(C)=NO2)s1 c1(C(=O)NCC(C)(CO)NC(CC2(COC)CC2)=O)cccc2nc(C)nn12 c1(C(N(CCNC(c2cccc(CC)n2)=O)C)=O)ccc2c(c1)COCO2 Cc1ccc(Br)c(F)c1CNC1CCC(=O)NC1=O c1(C(=O)NCc2nc(CNC(COC)=O)sc2)cnn(CCN)c1C Cc1ccc(C)c(CC(N2CC(NC(=O)CC3(C)CCOC3)C(O)C2)=O)c1 c1(C(=O)NCC(C2CC2)NC(C2(OCC)CCOC2)=O)cnc(=NCCF)[nH]c1 C(C(=O)N(C)OCC)NC(CNC(C(C1CCCC1)OCC)=O)=O N1(C(c2c(CC)ncnc2)=O)CC2CC(NC(C3(C4CCC4)CCC3)=O)CC2C1 C=CC(C(=O)N(C1CCN(C(c2csnc2C)=O)C1)CCO)c1ccccc1 C12C(C1C(=O)OC)C(=O)NC2=O.C(CCN(CCCN(C1CCC1)C)C)OC N1(C(CCOCC#C)=O)C(C(=O)NCC2CCCSC2)CC2CCCC12 c1(C(=O)NCC(C)N(C(CNC(C(CC)C)=O)=O)C)c(C)cncc1F c1(C(N(CC(C)N(C(=O)C(N2CCOCC2)C)C)C)=O)csc(S)n1 C1(C)(NC(C(CNC(c2cncnc2)=O)N(C)C)=O)CC(C)(C)C1 Cc1ccc(C(=O)NC2CC(C(N3CC(OCC(N)=O)C3)=O)C23CCC3)nc1O CC(C)C1=CCC(C(=O)NCCC2CC(NC(C3(C)CCCOC3)=O)C2)CC1 c1(CC)oc(C)cc1C(=O)NCc1nnn(C)c1C(=O)NCC1CCCSC1 Cc1cn2ccc(C(=O)NC3COC4C(NC(c5cnco5)=O)COC34)cc2n1 c1(C(=O)NC(C)CNC(c2c[nH]nc2-c2ccoc2)=O)ccc(Cl)cc1O C(=O)(CCCC(=O)N(C)C)NCC1(CN(C(CC(c2scc(C)c2)O)=O)C)CC1 C(CCCN=c1[nH]c(Cl)nc2c1CCOC2)NC1(C(C)(C)OC)CC1 O=C(C(F)C(F)(F)F)NCC1(CO)CCN(C(=O)CC2CC3(CC3)C2)CC1 C#CCC(C)(C(=O)N1CCCC1CNC(C)=O)NC(=O)CC1CCOC1(C)C c1(C(=O)NC(CC=C)CNC(C2CN(C(C)=O)C2)=O)ccc2cc(Cl)ccc2c1 C(=O)(C(C(C)C)CN)OC1COCC1Cc1cnn(C(=O)OC)c1 c1(C(=O)NC2CCN(C(C3(C)CCCCC3)=O)CC2)cc(C(F)(F)F)ncc1N N1(C(C(c2cccc(Cl)c2)C)=O)CCC(NC(c2n[nH]cc2C2CC2)=O)C1C c1(CC(=O)NCC(O)CCNC(c2ccc(C(F)F)nc2)=O)cncnc1O N1(C(C2(OC(C)=O)CC2)=O)CCC(F)(C(=O)NC2(C3CCCO3)CC2)C1 c1(OC)ncnc(OC)c1C(=O)NC1CCN(C(=O)CN2CSCC2=O)C(C)C1 c1(C(=O)NCC(c2ccccc2F)NC(CCC#C)=O)cnc2nccn2c1 c1(C(=O)NC(CC(C)C)CNC(C2(C)CC(=O)C2)=O)c(F)ccnc1Cl C(=O)(C#CC(C)(C)CNC(c1ccn2ccccc12)=O)N(C1CCN(C)C1=O)C N1(C(CCN(C)CC)=O)C2CCC1CC(CCNC(=O)C(C)(C)NC(C)=O)C2 CC(c1cccc(Cl)c1)=CC(=O)NC1CCN(C(=O)CCc2cncs2)C12CC2 C1(c2cn(CC)nc2)OCCCC1CC1COCCN1C(=O)NC1COC1 c1(OC)cccc(C2CC(O)CN2C(=O)C(N)Cc2cncs2)c1 N1(C(c2ccc(C#N)cc2)=O)CCC(C2CCCN(C(c3ccoc3Cl)=O)C2)C1 N1(C(c2ccc(CC)o2)=O)CCC(NC(c2cnn(CC(F)(F)F)c2Cl)=O)C1C C1(CN(C(=O)CSCCC#N)C)CCCN1C(=O)CCc1ccncc1 c1(OC)ccc(Cl)c(-n2cc(CCCCNC(C3CCC3C(=O)O)=O)nn2)c1 C(CC1CCC1)(C(=O)N(CC(C)NC(=O)CC1(OC)CCC1)CC)OC Cc1cc(C(=O)NCC2CN(C(=O)C=CC3CCCO3)CC2O)cc(F)c1 S(=O)(=O)(c1cnn(C)c1)NCC(=O)NCC1(F)CCC(NC(C(C)N(C)C)=O)C1 N1(C(c2nn(CC)nc2C)=O)CCC(C)C(CNC(c2cc(F)cnc2Cl)=O)C1 C#CC1(C(=O)NC(C=C)COC)CCN(C(c2ccc(C(F)F)o2)=O)C1 C(C(C(=O)NCC(O)C(=O)NC(Cc1cn(CC)nn1)=O)N(C)C)NC C=C(C)CCC(=O)NCC(C)(C1CC1)NC(=O)COCCNC(=O)OC(C)(C)C C1(C(N2C(CNC(=O)Cc3csc(S)n3)CC(OC)C2)=O)CCc2ccnn2C1 N1(C(c2c(OCC)cccn2)=O)CCN(C(c2ccc(C#N)[nH]2)=O)C2CC12 c1(CC(=O)NC2C(CNC(c3cc(OC)no3)=O)CCC2)cnn2c1OCCC2 c1(CC(=O)NCC(CC)NC(=O)CC2CC3CC3C2)cnn2ccccc12 C1(NC(CCCc2onc(C)n2)=O)CC2CN(C(c3nc(Cl)oc3C)=O)CC12 C=C(CNC(=O)CSCC1CCCO1)CCNC(=O)Cc1ccccc1 C(C1=Cc2ccccc2OC1)=CC(=O)NC1CN(C(C2CCC(F)(F)CO2)=O)C1 C1(CC(=O)NC(CNC(=O)CC2CC(C3CC3)C2)C2CCC2)CCC(=O)NC1=O C1(CNC(CCN2CCC(C)CC2)=O)CCN(C(=O)CCS(N)(=O)=O)C1(C)C c1(C(N2CCC3(C(=O)NCC4(F)CCC4)CC3C2)=O)ccnc(Cl)c1F N1(C(C(N)CCSC(F)(F)F)=O)CCCC(c2ccncc2)CC1 N1(CCC)CCC(C(=O)NC2CN(C(=O)CN(C)C(C)C)C3CC23)CC1 c1(CC)oc2ccccc2c1C(N1CCOC2(C1)CN(C(=O)C(C)(F)CC)C2)=O C#Cc1ccc(C(=O)NCC(C)(O)CNC(=O)CN2CC(=O)N(C)C2=O)cc1C CCCC(C(=O)OC)C(=O)N(CC(O)CN(C(=O)COCC)C)C N1(C(c2nn(C)c(F)c2)=O)CCC2(CCN(C(C3CCCCS3(=O)=O)=O)C2)C1 CCC(C)C(C(=O)NCC(O)C(C)C)NC(C1CCC1C(C)(C)C)=O c1(CC(N2CCC(C(=O)Nc3cncc(C(N)=O)c3)CC2)=O)ccc(Br)c(F)c1 Cc1ocnc1CNC(=O)C(c1ccnn1C)NC(=O)COC1CC=CC1 c1(CC(=O)NCC(CC)NC(c2nocc2Cl)=O)csc(C2CCOCC2)n1 C1(N(C(=O)CC2CC2)CC)CCCN(C(c2ccc(C3(C#N)CC3)cc2)=O)C1 Cc1cc(F)cnc1C(=O)NCC(C1CCCN1C(c1cnc(C)n1C)=O)(C)C C#CCC(C)(C(=O)NC(CO)CC(C)CC)NC(c1nonc1C)=O CC1CN(C(=O)C=CCF)CCN1C(C1CCCN1CC(F)(F)F)=O CC1(C)CCCCCC1NC(=O)CCCCNC(C1(CCCF)CC1)=O C(C)(CCNC(C1(OC)CC1)=O)N(C(C=C(CC)C)=O)C N1(C(C(C)S(N)(=O)=O)=O)CCC2C1CCCN2C(c1nccc2n[nH]cc12)=O C1(CNC(c2cc(OCC)ns2)=O)N(C(C2CCC(C)O2)=O)CCCC1(C)C C(=O)(C1CCc2c[nH]nc21)N1CC2CN(C(c3c(C(C)(C)C)c[nH]c3)=O)CC2C1 CC1CC2(CO1)CN(C(=O)CC1(C)CCN(C(=O)C(C)(C)C(=O)N(C)C)C1)C2 O=C1CSC(C(N2CCC2C(N2CCC(n3ccnc3)C2)=O)=O)C1 Cc1cc(Cl)ncc1S(=O)(=O)N1CCOC(C(N2Cc3ccc(Br)cc3C2)=O)C1 CCC(C)(C(=O)O)NC(c1ccc(C2(C)CC2)cc1)=O CCCCS(=O)(=O)CC(=O)N(C)CC1(O)CCN(C(c2ccccc2CO)=O)C1 CC1(C)CN(C(c2ccccc2O)=O)CC1NC(=O)Cc1cccc(F)c1 CC(C(=O)NC1CCN(C(=O)Cc2nc(C3CC3)nn2C)C1C1CC1)C(C)(C)C Cc1ccc(C(N2CC(CC(=O)NC3CC(C)OC3=O)C3(CC3)C2)=O)c(O)c1 Cc1nccc(C(N2CCCCC(C(=O)N(C)Cc3cncn3C)C2)=O)c1N N1(C(C(CSC)C)=O)CC(NC(=O)C(C2CCCCC2)O)C(CC(C)(C)C)C1 c1(C(N2Cc3cccnc3C2)C(=O)NCCCC2CC2)nc(Br)c2ccccn12 c1(CNCC(n2cnnc2)C)ccc(C(O)COCc2ccccc2)cc1 C(CC(=O)N(C)CCOCCCC(F)(F)F)C=CC(=O)NCCCOCCOC N1(C(c2cccc(OCC)c2)=O)CCC(C)N(C(c2c[nH]ccc2=O)=O)CC1 c1(NC)cnncc1C(=O)NCC1CCC1C(=O)NC(c1ccoc1)C c1(C(=O)NC2CCC(C)N(C(=O)COc3cn[nH]c3)C2)cncc2ncn(C)c12 c1(C(=O)NCCn2c(C)ccc2C)c[nH]c2ccnc(Cl)c12 c1(C(=O)NC2CN(C(COC)=O)CC(O)C2)nn(C)c(=O)c2ccccc12 C(=O)(C(CNC(c1ccc(F)cc1)=O)CC1CC1)NCCC(C)N1CCCC1 C1(C(=O)N(CCC(C)(C)NC(=O)CSC(F)F)C)(OC)CCSC1 c1(C(=O)NCC(C)NC(C2CC(C)(C)CC(C)(C)C2)=O)cnc2nccnc2c1 C1(CC(=O)NCCC(C)(C)NC(c2cc(OC)n[nH]2)=O)CCCCN1C c1(C(=O)NC2CC(CCNC(c3c(COC)noc3)=O)C2)[nH]cc2c1CCCC2 N1(C(c2cncc(OCC)c2)=O)CCCC2(CCC(NC(=O)CC(F)(F)Cl)C2)C1 CCC(CC(=O)NC(C)(C)C(C)NC(=O)C=C(C)c1ccco1)c1ccccc1 C1(C(=O)NCC(C)(C2CC2)NC(C(C)C(F)F)=O)C2CCN(C)CC12 c1(OCC(N2C(CNC(C(C)OC)=O)C3CC3C2)=O)cccc(F)c1F c1(C(N)=O)ccccc1-n1ccc(-c2cnc(C3CC3)nc2)n1 N1(C(c2cnc(C(C)C)nc2)=O)CCC=C(CNC(=O)CC(C)(C)CN(C)C)C1 c1(C(N(C(C2CCCCC2)C)C)=O)cccc(CNC(=O)C(F)C2CCOC2)n1 C1(C(=O)NC(C)CNC(=O)CCc2cnco2)CCC(=O)N1 CC1(C)CC(NC(C2(C)CCC(=O)N2)=O)CN1C(C12CC(F)(C1)C2)=O C1(C(=O)NC(C)(C)CCNC(C2CCCN2C(N)=O)=O)CCCCC1(F)F N1(C(c2c(C3(C)CC3)c[nH]c2)=O)CC(C)(C)C(NC(=O)C(Cl)=CCl)C(C)(C)C1 C(=O)(C(CNC(c1cc[nH]n1)=O)CC1CC1)NC(C#C)CC1CCC1 N1(C(C2CC(SC)C2)=O)CCCC(C)(C)C1CNC(c1cncn1C1CC1)=O C1(CNC(c2c(CC)nns2)=O)CCC(C)N(C(c2ccc(O)nn2)=O)C1 CN=S(=O)(c1ccc(Sc2ccnc(C(F)(F)F)c2)cc1)N(C)C Cc1cccc(F)c1C(=O)NC1CN(C(=O)Cc2ccc(F)cc2)CC1CO c1(C(=O)NCC(CNC(C2CC(F)(F)C2)=O)C(F)(F)F)cccc2c1COC2 c1(C(=O)NC2CC(C)CN(C(=O)C(C)(C)N(C)C)C2)n[nH]c2c1CC1CC21 O=S(=O)(c1cnc(NCc2sncc2Br)c(Cl)c1)N1CCCC2(C1)OCCO2 CC1CCN(C(C2(C)CCN(C(c3ccc(CO)cc3F)=O)C2)=O)CC1(F)F Cc1ccc(C(N2CCC(C)(NC(c3cc4sc(C)nc4[nH]3)=O)C2)=O)c(F)c1F c1(C(=O)NC2CC(NC(c3c(-c4n(C)ncc4)n[nH]c3)=O)C2)cncc(N)n1 C1(NC(c2c(OC)cc(C)cn2)=O)CCN(C(=O)CCCCCF)CCC1CO C(=O)(CCCC(F)(F)F)N1CC(C)C(C(=O)NCc2ccnc(O)c2)C1 n1(CCOC)nc(-c2ccc(Cl)s2)nc1CCN1CC(Cc2ccccc2)C1 c1(C(N2CC3CC(O)CC2C3)=O)cc(Br)c2nccnc2c1 N1(CC(=O)N(CCNC(C(C(C)SC)O)=O)C(C)C)C(=O)CCCC1=O N1(C(C2C(CC)CCO2)=O)CCCCC1C(=O)NC1(C)CC1(C)C CCC(C)C(C(=O)N1CCCC1CNC(C1OCCC1C)=O)OC N1(C(c2cc3n(n2)CCC3)C(=O)NCCOC)Cc2ccc(OC)cc2CC1C c1(C(N(CCC(C)NC(C(CC)OC)=O)C)=O)cc2cc(F)cc(F)c2[nH]1 N1(C(c2cccc(C)n2)=O)C2CCC1CC(NC(C13CCC1C3)=O)C2 c1(C(N2C(CN(C)C(c3nnsc3N)=O)CCC2)=O)ccc(O)nn1 C1(NC(c2cccnn2)=O)CCCC12CN(C(c1cc3nc[nH]c3cn1)=O)C2 C1(CNC(c2c(C)cns2)=O)CCCC(NC(=O)Cn2ncnn2)C1 C1(SC)CCC(N=c2ccnc(N3CCCN(Cc4ccsc4)CC3)[nH]2)C1 C(c1nc2ccccc2[nH]1)=CC(N1C(CNC(C(C(C)C)(C)O)=O)CC(O)C1)=O C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CNC(CC(C)O)=O)CC(F)(F)F Cc1cn2c(C(=O)NC3CN(C(=O)C(C)CC(N)=O)C4CC34)cnc2s1 c1(C(N(C(CNC(C(CCC)C)=O)CC)C)=O)ccnc2cc[nH]c12 C1(C(NOCCOCC)=O)CN(C(=O)C(C)(C)CF)CC(C)O1 c1(C(=O)NC2C(NC(CCCC)=O)CCC2)ccc(C(C)C)cn1 c1(OC)cccc2ccc(C(=O)NCC(C)NC(c3cc(=O)n(C)cn3)=O)nc12 CC1CN(C(=O)CCc2nncs2)CC1(C)CNC(=O)C(c1cccn1C)=O C1(NC(=O)COC2CCOC2)(CO)CN(C(C2CC2c2ccncc2)=O)C1 C1(C(=O)NCCNC(c2cncc(C#C)c2)=O)CC2(CCOCC2)CO1 N1(C(CC)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)C1Cc2c(Cl)cccc21 O=S(=O)(c1cc(Cl)c(I)s1)N1CC(O)CC1c1cc(F)c(F)c(F)c1 C(CC(CC)C(=O)N(CCCCNC(=O)CC(C(F)F)n1ccnc1)C)=CC C1(C(=O)NC(C)CCO)CCCN(C(c2cc(Cl)c(Cl)s2)=O)C1 Cc1cc(CNC(=O)C(CCF)NC(C2CC2(C)C(F)F)=O)cnc1F C1(C(N2C(C(=O)NC3CC(C)(CC)C3)C3CC3C2)=O)CC2OC1C1CC21 c1(C(N(CCCNC(c2cnn(C(F)F)c2)=O)CCO)=O)ccc2c(c1)CCO2 N1(C(Cc2c(C)n[nH]c2C)=O)CC2CCN(C(C3C4CC5C(C4)C35)=O)CC12 C(=O)(C(C)CC(C)(C)C)NCCC1CC(OC)CN1C(=O)CC(C)(C)C(F)F C(CCC(=O)NCCNC1(n2cc(-c3c[nH]nc3F)nn2)CC1)OC(C)=O CCCC(O)CC(=O)NCCCCNC(c1scnc1C(F)F)=O N1(Cc2cnc(CCOC)s2)CCCC(c2cccc(C(=O)OC)c2)C1 N1(C(C2CC(C)CN2C(=O)C=Cc2ccccc2)=O)CCC(O)C(C)(CO)C1 Cn1cc(C=CC(=O)NCCOCCC(=O)NOCCCF)nn1 c1(C(=O)OCC)cc2cn[nH]c2cn1.c12ncc(nc1OCC)N1CCC2CC1 C(=O)(C(CC(C)C)NC(c1sc(C)cc1C)=O)N(CCC#C)CC N1(C(C2N(C)CC2)=O)CCCC2(CCCN2C(C2CCc3c[nH]nc3C2)=O)C1 c1(CNC(C(C)Cn2ccnc2)=O)ccc(CNC(C2CC2C(F)(F)F)=O)cc1 CC(C(=O)NCC1(O)CN(C(c2ccc(F)cc2F)=O)C1)S(C)(=O)=O c1(C(=O)NCC2OCCC(NC(C3CCN(C)C3)=O)C2)cc2c(Cl)nccc2o1 C1(C(=O)NOCCO)(CC#C)CCN(C(=O)C(C)CCN(C)C)C1 C1(NC(C(CC(=C)C)C)=O)CC2(C1)CC1(CC(NC(=O)C(CC)(CC)CC)C1)C2 CC1(C)CCN(C(c2cccc(F)c2F)=O)C1CNC(C1(C)CCCS1(=O)=O)=O c1(C(N2CC(NC(c3cocn3)=O)C(O)C2)=O)cnc2ccccn2c1=O c1(CNC(c2ncncc2Cl)=O)ccccc1CNC(c1cscc1Cl)=O C(C1=CCN(C(=O)CC2CC2C)CC1)NC(C(C(C)C)N(C)C)=O O=C1CC2CCC1C(C(=O)Nc1nc(-c3c[nH]c4ccccc34)cs1)C2 C(=O)(CCCCC(=O)NCC1CC1NC(=O)COCCc1cccs1)OC c1(OC(C(=O)NCC(C)NC(C(CC)N2CCCC2=O)=O)C)cccc(C#N)c1 CON(CCC(=O)NC1C=C(C)CCC1)C(=O)Cc1c(C)cnn1C N1(C(C=COCC)=O)CCC2C(CCN2C(C2C(C(=O)OC)C2(F)F)=O)C1 C(=O)(CS(=O)(=O)C1CC1)NC(C)CN(C)C(C1CCCCN1S(C)(=O)=O)=O C1(NC(=O)Cc2ccccc2)CCN(C(C2CCCC23CC3)=O)CC1 N1(C(c2ccccn2)=O)CCN(CC2CN(C(c3scnc3Cl)=O)C2)CC1 Cc1cnc(N2CCOC(C(C)NC(c3cc(Cl)n(C)n3)=O)C2)nc1 c1(OC)ccc(C(=O)NCCC(C)CCNC(c2cc(SC)oc2C)=O)c(F)c1 C(C(C)(C)CNC(c1ccoc1Cl)=O)N(C(C1C(CC)C1)=O)CC Cc1nc(Cl)ccc1CC(=O)NCC1CCCCC1NC(=O)C(C)n1cccn1 N1(C(CNC(CC)=O)=O)CC2CCC1C(CNC(=O)C(C)CNC(=O)C(C)=O)C2 C1(SCC(=O)NCCC(Cn2cc(C(C)(C)S(C)(=O)=O)nn2)F)CCC(=O)NC1 C1(CNC(C(C)S(N)(=O)=O)=O)CN(C(c2cccc(CO)c2)=O)CC(C)(C)O1 C(=O)(CCC(CC)CC)N1CCC2(C(C(NOONC(=O)COC)=O)C2)C1.CC N1(C(c2cnn(C(F)F)c2)C(=O)NCCCC)CCC(O)CC12CC2 C1(CN(C(C2CC(SC)C2)=O)C)CCCN1C(=O)C(C)=C1CCCC1 N1(C(C2CC(OCC)C2)=O)CC2(CCC2)CCC1CNC(=O)CC1(C)CCCCC1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC(C)N(C(c1ccnc(Cl)c1O)=O)CC c1(C(=O)NC23CN(C(C(COC)(C)OC)=O)C(CC2)C3)cc(F)c2[nH]nnc2c1 C(=O)(CCCCCF)NCCn1ccc(C(=O)NCC(COC)C(C)C)c1 c1(C(N(CC(CC)NC(c2cccc(N)n2)=O)C)=O)ccccc1NCCO c1(C(=O)NCC(C)N(C(=O)CCN(S(C)(=O)=O)C)CC)ccc2nc(O)[nH]c2n1 c1(OC)cccc(C(F)(F)C(=O)NC(CNC(=O)C=CC(=O)N(C)C)C2CC2)c1 N1(Cc2c(OCC)cccc2)CCC(=O)N(CCc2cnoc2)C1=O Cc1cc(CC(N2CC(=C(F)CNC(=O)C(n3nccc3C)C)C2)=O)ccc1O c1(C(=O)NC(C(C)NC(CCCCC)=O)C)c[nH]c2cc(C(=O)OC)ccc12 N1(C(c2cc(CNC(c3cnc(C)s3)=O)no2)=O)CC(F)CC1CO c1(OC)ccc(-c2csc(NC(=O)NCCCC3(O)CCOCC3)n2)cc1 N1(C(=O)OCC(=O)N(C(=O)C(F)F)C(C)C)CCC(C)(C)C1 C1(NC(C(C)n2ccnc2)=O)CC2C(NC(=O)CCCn3cncn3)C2C1 c1(C(N(CCOCCN(C(=O)CC#N)C)C)=O)cccc(S(C)(=O)=O)c1 C(=O)(C(=O)N=S(C)(C)=O)N1CCC(C(C)NC(=O)CC2COC(C)(C)C2)CC1 N1(C(c2c(CC)cc[nH]2)=O)CC(C(=O)N(C2CNC(=O)C23CC3)C)CC(C)(C)C1 c1(CC(C(=O)NCC(C(C)(C)C)NC(CCC(=C)Cl)=O)C)ccc(C#N)cc1 CC1(C)CN(C(c2cc(F)c(F)cc2F)C(=O)NC2CCOCC2)Cc2ccccc21 c1(C(CC(=O)OCC)NC(c2ccc(NS(C)(=O)=O)cn2)=O)ccc(Cl)c(F)c1 Cc1nc2ccc(Br)cc2cc1NC(=O)CCCCCCCO c1(C(CNC(=O)NC(c2ccccc2)CC)=O)ccc(C)cn1 N1(C(C2(COC)CCCC2)=O)CCN(C)C(CNC(C2CC2(C)C(F)F)=O)C1 c1(-c2cccc(NC(Cc3cc(C)no3)=O)n2)cc(N2CCCCC2)ccc1F c1(C(=O)NCCC(C)N(C)C(c2ccc(C3CC3)o2)=O)snnc1C1CCC1 C(C(C(C)C)NC(=O)Cc1cc(C)on1)NC(C1(C(C)(C)OC)CC1)=O C1(NC(C(C)SCCCC)=O)CN(C(=O)COc2ccn(C)n2)C(CC)(CC)C1 c1(OC)c(Cl)ccc(C(N2CC(NC(=O)CC3(C)CC3)CCC2C)=O)c1F C1(O)(CNC(c2ncn(CCNC(CCCOC(C)C)=O)c2)=O)CCOC1C c1(C(=O)NC2CC(C(N(CCO)CC)=O)(COC)C2)ccccc1 C12(C(=O)NCC(=O)NCC(C)C)CC1CCN2C(=O)CC=C(Cl)Cl C=CC(C)(C)CC(=O)N1CCC(NC(c2cccc(OC)c2C)=O)CC1C C1(C(N(C2CCCCC2)CC)=O)CSC(C)(C)C(=O)N1C(=O)CN1CCCC1=O C1(CNC(=O)COCC2CC2)CC12CCN(C(c1ccsc1Br)=O)CC2 c1(C(N2CC(OC)C(NC(=O)CCc3nc[nH]n3)C2)=O)cc(F)c(C#N)c(F)c1 N1(C(CSCC)=O)CCCC(C)(C)C1C(=O)NC1CN(C(N)=O)C1 CC(CN=c1c(C#N)c[nH]c2c(F)ccc(F)c12)N(C)C(c1cc(O)ncn1)=O c1(C(=O)NCC2N(C(C(COC)COC)=O)CC2)ccnc(S(N)(=O)=O)c1 N1(C(C2(OC)CCC(C)C2)=O)CCCC(C(=O)NCCCCN2CCC2)CC1 C1(NC(CC2(C)CCN2C(=O)CCc2nncs2)=O)COC2(CCC2)C1 c1(C(N2CC(C(=O)OC)(C(C)C)C(O)CC2)=O)nc2cc(F)cc(F)c2[nH]1 C1(CC(=O)NC2CC(n3cc(C(CC)(C)O)nn3)C2)(CO)CCCCC1 C(C)(C)(CC(=O)NC1(C(C)(C)C)CCN(C(=O)C(C)OCC2CCCC2)C1)OC N1(C(c2ccc(C3CC3)o2)C(=O)Nc2c(C)cccc2C)CCCC2CCCC12 CC1=C(C)CC(C)(C(=O)NC(C)CNC(C2(C)CCC(C)C2)=O)CC1 c1(-c2c(NC(C)=O)cccc2)cccc2[nH]c(C(=O)NCC(O)C(F)(F)F)cc12 C1(C)(C(=O)NCCCCCC)CCN(c2ccnc(N(C)C)n2)C1 CCC(CC)CCC(=O)N1CCCC(C(C)NC(=O)CSS(C)(=O)=O)C1 c1(OC)cc(O)ncc1C(=O)NC1CCC(Nc2cc(C(C)(C)C)ncn2)C1 N1(C(Cc2nc(C)oc2)=O)CCN(C(c2nc(C(F)(F)F)ccc2F)=O)CC1C C(=O)(CCCc1ccccn1)NC(C1CCCN1C(C1CC1c1ccco1)=O)C CCC(C)C(=O)NC(CC(=O)N1CC(N2CCC2)C1)C1CC1 C1(C(=O)NCC2COCCN2C(C23CCCC2C3(F)F)=O)CN2CCCN1CC2 CC(C)CCC(O)C(=O)NC(c1cn(C)nn1)CNC(c1cc[nH]c(=N)c1)=O C1(NC(=O)CC2CCC(=O)N2)CCN(C(=O)CC2(N3CCCC3)CC2)CC1O N1(C(CC(C=C)C)=O)CC2CCC1C(CNC(C1(O)CCOC1)=O)C2 N1(C(COC2(C)CCC2)=O)CC(C)(C(=O)NCC2(C)CC(O)C2)CC1(C)C CCS(=O)CC(=O)NC(c1ccccc1CO)CNC(=O)C(C)OC(C)(C)C CC(C)CCC(O)C(=O)NCCC1CCN(C(=O)CCCn2cnc(C#N)n2)C1 N1(CC(=O)NC2(CNC(CCCNC(C)=O)=O)CCC2)CCC(F)(F)C1 n1(CCOC)c(C)cc(C(=O)Nc2ccnn2Cc2cccc(CC#N)n2)c1C FC1(F)CC1C1CCCN(c2nc(Cl)nc3ccccc23)C1 C1(CNC(c2cccnc2Cl)=O)CCN(c2ncc(I)cn2)CC1(F)F C1(n2cc(C(C)N(C(=O)C(C)(C)F)C)nn2)CCCCC1=O C(C)(C)(C(C)CC(=O)NC1CC(n2cncn2)C1)NC(Cn1c(C)nc(C)n1)=O N1(C2c3ccnn3NC2=O)CCN(CC(O)C2CC2)CC1.C1(CO)CCCCC1 C1(C(=O)N2CC(O)CO2)CC12CCN(C(=O)CC1(O)CCOC1)CC2 c1(NC(N2CCC(C#N)(CC)CC2)=O)ccc2nn(C)cc2c1 N1(C(c2c(C)cco2)=O)CCC2CN(C(c3ccncn3)=O)C2C1 C1(CNC(c2cccc(C(=O)NC)n2)=O)CN(C(=O)C(F)CC2CC2)CCCO1 c1(NC(C2(OC)CCSC2)=O)ccc(NC(=O)C(C)CC(C)C)cc1C C1(NC(CNC(CC)=O)=O)C(CNC(c2ncccc2Cl)=O)CCC12CCC2 C12(C(=O)NC3(CC=C)CN(C(C4CCCN4CCC)=O)C3)CC1COC2(C)C C1(NC(C=CC(CC)C)=O)CCC2(CCN(C(c3cnn(C)n3)=O)C2)C1 C1(N(C(N2C(C)(COC)CC2)=O)C)CCS(=O)(=O)C1 c1(CC(=O)NCC(C)(C2CCC2)NC(C(CC(C)C)C)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NC2C(OC)CN(C(=O)C(C3CCOCC3)C)C2)cc(S(N)(=O)=O)co1 C1(NC(CCC(C)O)=O)CCSC12CN(C(=O)CC(C)(C)C1CCCCC1)C2 c1(C(N2CC(C)C(C(=O)NCC3CCC(C)CC3)C2)=O)cncc(C#N)c1 Cc1ccc(C(C(=O)NCCC2CCCN2C(=O)CCCF)C2CC2)cc1 Cn1cnc2ccc(CN3CCOCC3CCN)cc12 C1(C(N2CCN(C(C=CC)=O)CC2)=O)Cc2nn[nH]c2C(C)C1 Cc1cccc2c(C(N3CCCC(F)(CNC(=O)C(Cl)=CCl)C3)=O)n[nH]c12 CCC(C)C(C(=O)NC1CCCC1CN(C)C)NC(=O)CCOC c1(C(N(CCNC(=O)CSc2nncn2C)CC)=O)cnc2cccnn12 C1(NC(=O)CN2CCSCC2)CCCCC1N=c1[nH]c2cc(Br)cnc2s1 C1(C(=O)NCC2CCN2C(c2coc(O)n2)=O)CCc2nnc(O)n2C1 N1(C(CN2C(=O)CCC2)=O)CC2CCN(Cc3ccc(Cl)s3)C2C1 CCC(CC)(CC)C(=O)NCC(CC(C)C)C(=O)N(C(C)CC1CC1)C N(C(=NCCc1ccnc(Cl)c1)NCC(c1ccc(F)cc1)(F)F)C1C(C)C1 C1(C(N2CC(CNC(C3C(C)(Br)C3)=O)C2)=O)Cc2cc(F)ccc2C(=O)O1 c1(COC)cc(C(=O)NC2CCCC2NC(=O)C=Cc2cc[nH]c2)n(C)c1 C1(OC)C(n2cc(-c3cc(Cl)ccn3)nn2)COC1(C)C c1(C(=O)NC2CCC(NC(C(C)CF)=O)C2)noc2c1COCC2 C1(CCOC)(C(=O)NCC(C)(O)CSC)CCN(C(=O)CCc2csnn2)CC1 N1(C(C2(CCC)CC2)=O)CCOC(C)(CNC(=O)CCS(C)=O)C1 c1(C(=O)NCCn2cc(-c3nccc(OC)c3)nn2)ccc2c(c1)C(C)C(C)O2 n1(C(C)C)cc([N+](=O)[O-])c(=NCC2CCCN(C(C3CC=CCC3)=O)C2)[nH]1 n1(CC(C(=O)C(C)(C)C(F)F)=O)ccc2ccccc2c1=O.C1(C)CCN1CC N1(C(C(C)(C)Nc2ccccc2)=O)CCC(CO)(NC(c2occc2F)=O)CC1 C1(NC(C2C(C)OC(C)C2)=O)(CO)CCCN(C(c2cn(CCO)nn2)=O)C1 N1(C(CC2C(C)CCO2)=O)CC(CNC(=O)CCc2ccn(C)n2)C(C)(C)C1 N1(C(Cc2ccc(C)cc2)=O)CC(C(=O)NC(C(N)=O)C2CC2)OC(C)C1 c1(C(=O)NCC(CNC(C2(C)CC2)=O)F)sc2cccc(Cl)c2c1Cl c1(C(=O)OC)cccc2oc(=NCCCCNC(=O)C(C(C)C)NC=O)[nH]c12 N1(C(=O)OC(C)(C)C)CCC2(CCC(CNCc3ccnc(Cl)c3)C2)CC1 C12(CNC(C(C=C)(C)C)=O)CC(CC)(CN1C(C1(c3cccc(OC)c3)CC1)=O)C2 C1(CNC(C(C)OCCCC)=O)CC(O)CN1C(c1nc(C)nn1C)=O C(CC(C)CC(C)(C)C)NC(c1ccccc1COC)c1n(CCC)nnn1 C1(CNC(c2ncn(C(C)C)n2)=O)CN(C(c2cc(CO)ccn2)=O)CCN1C CCC(C)(COC)C(=O)N1CCCCC(C(=O)NCC(C2CCC2)OC)C1 N1(C(c2cnn(-c3cccc(Cl)c3)c2)C(=O)NCCC)CC(C)CCC12CC2 c1(C(=O)OC)cc(NC(=O)NC2CC(NC(=O)NC(C)(C)C)C2)c(F)cc1C C12(C(N3CCC(CNC(C=C4CCC(C)C4)=O)CC3)=O)CCC(F)(CC1)CC2 CC1(CNC(C2CCCOC2)=O)CCN(C(=O)CCCCN2CCCC2)C1 C1(C(N(C)CC2(NC(CC3C(C)OCC3)=O)CC2)=O)CC2(C1)CC(O)C2 C=C(Cl)C(C)(C)C(=O)NCC1CCCCN(C(C2CCN(S(C)(=O)=O)C2)=O)C1 c1(C(C(=O)NCC2(O)CN(C(C(CC)n3ccnc3)=O)C2)C)nc(F)ccc1Cl C1(C(N2CCCC(N(C)C(c3cnn[nH]3)=O)CC2)=O)CC(=O)C12CCCC2 c1(NC(C(C)CC2CCCO2)=O)ccc2ccn(CC(=O)N(C)C)c2c1 C1(C)(C(=O)NC(C(=O)NC)CO)CCCN1C(=O)CC(C1CC1)C1CC1 N1(C(c2c(C)occ2)=O)CCC2CCN(C(C3CCC(N=[N+]=[N-])CC3)=O)CC2C1 N1(C(C(N2CCCC(C(C)C)C2)=O)=O)CCc2cc(Br)cc(F)c2C1 N1(C(CSCCN(C(c2sccc2F)=O)CC)=O)CCC(CCNC)C1 Cc1c(CCC(=O)NC(C)CCN(C(=O)C=CC(C)(C)N(C)C)C)cnn1C N1(C(C=Cc2ccn(C)c2)=O)CC(C)(C)CCC1CNC(c1cnco1)=O c1(CC)c(C(=O)NC(CNC(C2CN(C(C)=O)C2)=O)CC)sc2ccccc12 CCC(C)CCC(=O)NCc1ccc(CN(C)C(C2(F)CC=CCC2)=O)cc1 CC1CN(C(=O)C(Cl)Cl)CC1(C)C(=O)N(C)CC1(CO)CC1 CC1(C(=O)NC(CNC(C2(C(F)(F)F)CCOCC2)=O)C(C)(C)C)CC(F)(F)C1 C(C(C)C(C)C(=O)N(C)CC1CCN(C(C2CC(OC)C2)=O)CC1)OC N(C1CC2(CN(C(c3ccc(F)s3)=O)C2)n2ccnc21)C(c1ccc(C)nn1)=O c1(C(=O)NCC2=CCN(C(c3[nH]c(=NC)sc3)=O)CC2)cccc2sccc12 N1(C(C(CC)n2ccnc2)=O)CCN(C(=O)Cc2ccc(Cl)s2)C(CO)C1 c1(OCC)cccc(CNC(C2CC(C)(C)O2)=O)n1 C1(NC(c2cnc(OC)nc2)=O)CC2CC(NC(C3COC3)=O)CC2C1 C1(CNC(C(CC)N(C)C)=O)CCCCC1NC(=O)COc1ccccn1 C1(NC(CCc2nc(C)c(C)[nH]2)=O)CC2CCC(C1)N2c1cc(C2CC2)ncn1 N1(C(c2scc(C)c2C)C(=O)NCCCSCC)CCC(O)C(C)(C)C1 c1(CCC(=O)NCC2(CNC(c3c(C)scc3)=O)CC2)ccc(Cl)cc1Cl N1(C(c2c(CC)csc2)=O)CC2(C(=O)NCC(c3nccs3)C)CCC1CC2 N1(C(=O)OC)CC2(CCC(CO)O2)C1.CC(C)(C)OC(=O)COCC(N)=O Cc1ncc(NC(=O)C(C(C)(C)C)NC(c2cc[n+]([O-])cc2)=O)c(C)c1C N1(CC)CCOC(C(=O)NC(CNC(=O)CCOC2CCOCC2)C(C)(C)C)C1 N1(C(c2cc(OC)c(O)cc2)=O)CCCC2(CCC2NC(C2CC2F)=O)C1 C(=O)(C(CC(C)C)C(C)C)NCC1C2CN(C(c3c(C)cc[nH]3)=O)C1C2 N1(C(CSCC=C)=O)CCC(C)C(CNC(c2nc(OC)cc(OC)n2)=O)C1 C(=O)(C#CC1CCC1)NC1CC(C(C)NC(C2CC(=O)N(C(C)(C)C)C2)=O)C1 C(=O)(C(Cc1ccsc1)N(C)C)OCC(C)=O CCCCC(CNC(c1snc(Cl)c1Cl)=O)NC(c1cnc(C(N)=O)cn1)=O CC(Cc1ccccn1)C(=O)NCCC(C)NC(c1cc(Cl)cs1)=O C(=O)(C(C)(F)C(C)(C)F)NCC(C(C)(C)C)NC(c1ccc(C#N)cn1)=O c1(C(N2CC(CCOC)C2)=O)cnn(CCNC(=O)C(C)C2CCCO2)c1 c1(OC)cccn2ncc(C(=O)NCC3(C)CCCN(CC(C)O)C3)c12 CN1CC(C)(C(=O)NCC2CCCN2C(c2cc(C(F)(F)F)ncn2)=O)CC1=O C(=O)(CC(C)(O)COC)NCC(C1CC1)NC(c1nnn(CC)c1C)=O C#Cc1ccc(CC(=O)N(CCC(C)(C)NC(c2nc(O)sc2C)=O)C)c(F)c1 Cc1c(C(N2CCCC(O)(CNC(=O)CO)C2)=O)ccnc1Cl CCC(CC(=O)N1CC(CNC(c2ccc(-c3cccs3)cn2)=O)C(O)C1)OC c1(C(=O)NCCC(CNC(=O)CC2C=CCC2)O)nc2c(s1)COCC2 CC1CC(C)N(C(=O)CSc2ccccc2)CCN1C(c1cc(O)nc(Cl)c1)=O C1(CC=C)(NC(c2cnc(C3CC3)nc2)=O)CCN(C(=O)C(C)n2cncn2)C1 c1(C(=O)NC2CCN(C(COC)=O)C2)cnc2c(c1)CCC(=O)N2 N1(C(=O)OC)CSCC1C(=O)NCC1(F)CC(C(C)(C)C)C1 N1(C(CC(CC)OC)=O)CCC(C2CC2)(CNC(C2CCCN2C(C)=O)=O)C1 C1(C(=O)NC2CC(C(C)O)C2)CCC(O)CN1C(c1cccc(F)c1)=O c1(OC)cc2ccccc2cc1C(N1CC(CNC(=O)CC2CCC(=O)N2)C1)=O N1(C(C(CCCC)F)=O)CCC2(CC1)CC2NC(c1cccc(C)c1)=O c1(NC(C(C2CCN(C(c3ccncn3)=O)CC2)C)=O)nc(Cl)ccc1I N1(C(C(C=C=C)C)=O)CCCCCC(NC(c2cc(C)cc(C)c2C)=O)C1 Cc1cncc(C(=O)NC2(CCNC(=O)CSCc3cscn3)CCC2)c1C CC1(C)CC(CNC(=O)C=Cc2cnc[nH]2)CN1C(c1cccc(N)c1)=O c1(OC)cc(C(=O)NC2CN(C(=O)CCC3CC3(F)F)CC2OC)ccc1Cl C12(C(N3CCC(OCC(N)=O)C3)=O)CCC(NC(c3ccsc3)=O)(CC1)C2 N1(C(C(C)C2CCCC2)=O)CC(C2(NC(=O)CCN3CCC3)CC2)C1 n1(CC(N2CC3C(CNC(c4cc5sccc5[nH]4)=O)(C3)C2)=O)ccc(O)nc1=O Cc1nccn2ncc(C(N3CC4CC(NC(=O)C=C5CCN(C)C5)C3C4)=O)c12 N1(C(C2N(C(C(CC)n3cncn3)=O)C3(CC2)CC3)=O)CC(O)C(O)C12CCC2 C1(C)(C(=O)NCC(C)(F)CNC(C2CC3CC3C2)=O)CCC2CC2C1 Cc1cc(C)n(CCC(=O)NCC2(C)CCC(NC(=O)CCOC3CCC3)C2)n1 c1(C(N2CCOC(CN=c3[nH]nco3)C2)=O)ccn2ccccc12 CC1CN2CCN1CC2C(N(CC(C)(C)NC(c1csc(C(F)F)n1)=O)C)=O c1(C(=O)NCC2C3CN(C(C4CC(=C)C4)=O)CC32)cc(F)c(C)cc1F N1(C(C(C(C)NC(c2cc(C(N)=O)co2)=O)C)=O)CC(O)(C2CCC2)C1 c1(OC)ccc2c(c1Br)CN(S(=O)(=O)N1CCC(C)CC1)CC2 C(=O)(CC(=O)N1C(C(=O)NC(c2ccncc2)CC)CC1C)NCC#C c1(CNC(C2CCC2)=O)ccccc1C.N1(C(COCCOCC)=O)CC(C)C1 n1(CCC(=O)NCC(C)N(C(=O)C(C)NC(C)(C)C)CC)cccnc1=O N1(C(CNS(N)(=O)=O)=O)CCC2(CCN(C(c3n[nH]cc3OC(F)F)=O)CC2)C1 c1(CC(N2CC(N(C(COCCOCC)=O)C)C2)=O)c[nH]nc1O c1(NC(CCC2(C)N(C(C3C(C(=O)OCC)C3)=O)CCC2)=O)cnc(Cl)nc1C c1(C(N2CCCC(C)(NC(CNC(=O)NC)=O)C2)=O)cccc2nc(C)nn12 C1(CC(=O)NCC(N(C)C)C2CC2)CCC(NC(=O)C=Cc2ccco2)C1 C=Cn1nccc1C(N1CC(NC(=O)CCN(CC(C)C(C)C)C)CC1C)=O C1(NC(c2c(C)noc2)=O)CC(F)CN(C(=O)C(C)Oc2ccc(Cl)cc2Cl)C1 CC(CC(=O)NC1CCC(C(=O)NCCCF)C1)C1CCCC1 N1(C(C(C)=CC2CC2)=O)CCSCC1C(N1CCC1(C)C(C)C)=O C1(CC(=O)NC(CC)(C)CNC(c2cscc2F)=O)CC=CCN1C CC1CCC(NC(c2ccnc(C(F)F)c2)=O)CN1C(=O)CNC(=O)C(F)(F)F C1(C(=O)NCc2n(CC)cnc2)CCCCC1NC(C1(O)CC(CF)C1)=O C1(CNC(C(=O)NC(C)C)=O)CC2CC(C1)N(C(c1noc3ncccc13)=O)C2 c1(C(N(CCN(C(C2SCCCS2)=O)CC)CC)=O)cnn2c1N(C)CC2 C(=O)(C(C)N(C(C1CN(c2ncco2)C1)=O)CCOC)NCC N1(C(C2CCC(=O)N2)=O)CCC2(CC1)CC(n1ccnn1)CCO2 C1(CC(=O)NCC2(F)CN(C(C(OC)OC)=O)C2)NC(=O)NC1=O C=CCCCCCC(=O)NCC1(CO)CCN(C(=O)CC2CCC2OC)CC1 n1(CC(=O)NC(c2oc(C)nc2C)c2ccc(C)o2)cc(C(N)=O)c2ccccc12 N1(C(C2C(COC)C2)=O)CC2CC1CN(C(c1cc3occc3n1C)=O)C2 C1(NC(CC2(C(=C)F)CCC2)=O)CC2(CCN(C(c3cccc(N)n3)=O)C2)C1 C(=O)(C#CC12CC3CC(CC(C3)C1)C2)N(C(C12CCC(CC1)C2)=O)Cc1n(C)ccn1 C1(NC(C=CCC)=O)CN(C(=O)Cc2ccsc2Br)C2CC12 CC1(C)NC(=O)CC1C(=O)NC(C)(C(=O)NCc1ccc(Cl)nc1)C1CC1 c1(OC)nc(C)ncc1C(=O)NC1CN(C(c2cnn(C)c2SC)=O)CC1C CCCC(CC)CC(=O)N1CCCC(CNC(c2ncc(C(N)=O)cc2Cl)=O)C1 Cc1cn2nc(N3CC=C(CCNC(=O)CCc4nnc(C)n4C)CC3)sc2n1 C1(NC(c2c(OC)ccs2)=O)CN(C(c2cc(O)nc(Cl)c2)=O)C2(CCOC2)C1 CCCC(CC)CCC(=O)NC1CCN(C(=O)CCSCC(N)=O)C1C CN1CCCCC1C(=O)NCC(F)CNC(=O)CC(c1ccccc1)C1CC1 C1(C(N(C2CCOC2)CC)=O)CC2(CCN(C(c3ccc(C(C)=O)o3)=O)C2)C1 c1(C(=O)NCC(CC)(CC)NC(=O)Cc2cncs2)nccc2n[nH]cc12 C(c1cn(C)cn1)=CC(=O)N(C)CCNC(C1(O)CCSC1)=O N1(C(C(C(C)C)C(C)C)=O)CCC(C2(NC(=O)CCc3ccoc3)CCC2)CC1 C=C(Cl)CC(C(=O)NC)NC(=O)C(C(C)(C)C)NC(=O)CCC(C)(C)F NS(=O)(=O)c1cc(C(N2CCCC3(C2)CN(C(c2cnsn2)=O)C3)=O)c(Cl)o1 N1(C(CCCC)=O)CCS(=O)(=O)C(CCNC(=O)CC(C)C(F)(F)F)C1 CC(C(=O)NC1CC2(C1)CC(NC(C1OCCN(C)C1=O)=O)C2)C(C)(C)C c1(C(=O)NCC(CNC(CCc2ccc(C)o2)=O)C)cc(Cl)cc(F)c1F Cc1cc(C(N2CCCC(C(=O)NC3(C)CCOCC3)CC2)=O)nnc1C C(CC(=O)N(CC(O)CN(C)C(c1sc(COC)nc1C)=O)C)(C(C)C)OCC C1(NC(c2sccc2Cl)=O)CN(CC(=O)Nc2ccc(F)cc2)CCC1COC N1(C(c2ccc(OC)cc2F)=O)CCC2(CC1)CN(C(=O)CC1CCSCC1)C2 C1(NC(c2cc(CCC)[nH]n2)=O)CC(O)CN(C(C2(CO)COC2)=O)C1 c1(C(c2nnnn2Cc2nnn(C)n2)NC(c2ccccc2)C)csc(Cl)c1Cl C(=O)(CCCCCCC(=O)NC(Cc1ccccc1[N+](=O)[O-])C(=O)O)OC CCC(C)C(O)C(=O)NCC1(C)CCN(C(c2ccc(=O)n(CCO)c2)=O)C1 c1(NC(C2N(C(c3cn(CCC)nc3)=O)CCC2C)=O)ccc(O)c(=O)cc1 N(C1CCCc2n[nH]cc21)C1(CCCC)CO1.C1(CC(=C)C)CCOC(=O)N1 C1(O)(CNC(Cc2scc(C)c2)=O)CCN(C(C2CC(CN(C)C)C2)=O)C1 c1(NC(C(CCCC)NCCCC(=O)OC)=O)ccc2c(c1)OC1(CCCC1)O2 C1(C(=O)NC2(CC)CCN(C(=O)C(Cl)=CCl)CC2)CCc2c(ncn2C)C1 S(=O)(=O)(c1cccs1)NC(C)C(N1CCC(C(=O)O)C(C)C1)=O C1(CNC(=O)C(O)CC(F)F)CC2(CCN(C(=O)CCn3ccnc3)CC2)C1 N(C1CC(C)(C)Oc2cc(F)ccc21)CC(=O)N(CC(=O)OC)C Cc1cc(C(=O)N(C)CC2(NC(=O)C(C)c3cncs3)CC2)cnc1C(F)(F)F c1(C(=O)OC)ccc(SCCCC(=O)Nc2nnc(CO)s2)cc1 CS(=O)(=O)C1CN(C(C=Cc2ccc(Br)cc2)C(=O)NC2CCC2)CC1C(N)=O C(=O)(CCCC(C)(F)F)NCC1(O)CN(C(C2CC(C)OC(C)C2)=O)C1 N1(C(C(CC=C)CC)=O)CCOCC(C)(CNC(=O)CCc2cc(Cl)cs2)C1 N1(C(c2c(C)nc(O)[nH]2)=O)CC2CC(NC(c3cc(F)ccc3Cl)=O)CC1C2 c1(C(=O)NCC2CCN(C(c3ccco3)=O)CC2)cccc2c1CCO2 CCCC(C)(C)CC(=O)N1CCC2CC2(C(N2CCC3CCCC23)=O)CC1 c1(CC(=O)NC(C)(CNC(=O)C(F)=C2CCC2)C2CC2)ccc(Br)s1 C(CCC(C)C(=O)NC1CCC(CNC(c2occc2C(C)C)=O)CC1)OC Cc1cc(C)c(CC(=O)NC2CCN(C(c3cn(C)c(O)n3)=O)CC2)s1 Cc1cncc(C(=O)NCC2(CO)CN(C(c3ccc(OC(F)F)cn3)=O)C2)n1 C(C)(CN=c1[nH]c(C)cc(=NCc2nc(C)ccc2Cl)[nH]1)OC N1(C(CC2(COC)CC2)=O)CCC2(CCCCN(C(C3CC3C3CC3)=O)C2)C1 C1(COC)CN(C(C2CCS2(=O)=O)=O)CCN1C(=O)CC1(C)CC1 N1(C(c2csc(-c3cnc[nH]3)n2)=O)CCN(C(c2ccc(O)c(F)c2)=O)C2CC12 c1(CN(C(=O)NC(Cc2scc(C)n2)C)CC2CC2)ccc(O)cn1 C1(CN(C(C(C)OC)=O)C)CC(F)CN1C(=O)C(C)Cc1cnco1 c1(C(N(C(C)CNC(=O)CN2CCCOC2=O)C)=O)ncc(P(C)(C)=O)cn1 c1(C(N(C2CCN(C(C3CC(O)C(F)C3)=O)CC2)CC)=O)cc(OC)ncc1F CC(C)C(C)C(CNC(c1cnc2n1CCC2)=O)N=c1cnc2ccccc2[nH]1 C12CCN(CC1)CC1CCC21.C1(c2cn(C3CN(C)C3)nn2)(CO)CCN(C)C1 N1(C(COCCCC)=O)CCOC(C(C)NC(=O)Cc2ccc(OC)s2)C1 C(C)(C)(CCCC(=O)NCC1CCCC(OC)C1)NC(C(C)=CCC)=O c1(C(=O)NCC2(C)CCCN(c3nc(C)nc(Cl)c3)C2)cc2c([nH]1)CCCC2 CC1(C)CCOC1CCC(N1CCC(NC(=O)Cn2ccnn2)C1)=O N1(C(COC(CC)C)=O)CC2(CC(NC(=O)C=C(C)c3ccccc3)CO2)C1 c1(C(=O)NCC(=C)CCNC(=O)C=CC(=O)NCC2CCCC2)ccc(F)cc1 c1(C(=O)NCC2(F)CCN(C(COC(C)C)=O)CC2)cccc(C#CC2CC2)c1 Cc1cn2c(C(N3CC=CC3CNC(=O)COCC(C)C)=O)cnc2s1 C1(NC(C(CC)C)=O)CN(C(c2ncccc2O)=O)CC2(CC2)C1 N1(C(CC(=C)Br)=O)CC(CNC(C2(CCCC)CCCC2)=O)C(O)C1 C1(C(C)C)CCOCCN1C(C1CC2CCC1CC2)C(=O)NC1COC1 c1(C(C)C)ncc2c(n1)CCN(N1CCN(CCNC(C3CCCO3)=O)CC1)C2 Cc1cc(F)ccc1NC(C1CC(O)CN1C(c1ccn(C(C)(C)C)n1)=O)=O CCCC(C(=O)NCC1CC1CO)NC(=O)C(Cl)Cl C1(OC)CCC(C(=O)NC(C2CCCN(C(c3ccnnc3)=O)C2)C)CC1 S(=O)(=O)(c1cccnc1NCC1CCCCCC1)NC(C1CCCCC1)CSC C1(C(=O)NC(C(C)(C)C)CO)C(C2CC2)CCN1C(=O)Cc1ncccc1F C(c1c(Cl)nc2sccn12)=CC(N1C(CNC(=O)C2=CCCCO2)CCCC1)=O C(CC(C(=O)NC(CO)C1CCC1)NC(=O)Cc1cnn(C)c1C)SC C(=O)(C(C)(C)CC(F)F)N1CC(OCCNC(C(C(C)C)NC(COC)=O)=O)C1 C1(NC(C(C=C)OC)=O)CCN(C(=O)COc2ccccc2)C1(C)C c1(CCC(=O)NCC(CCOC)NC(c2nc(C)nn2C)=O)ccccc1C C1(CC)CCCN(C(=O)COC2CCN(C(c3sccc3C)=O)C2)C1 Cc1nn(C)c(C(=O)NCC2(NC(=O)C(C)(C)n3cnnn3)CC2)c1[N+](=O)[O-] C1(C(=O)NCCC2CC(C)C2)CC2CN(C(=O)C(F)(F)c3nccs3)CC2C1 C1(CC(C)NC(=O)C(O)C(F)F)CCN(C(c2ccc(F)s2)=O)CC1 N1(C(C(CC)COC)=O)CC2(CC2)CC1CNC(=O)Cc1ccccc1C(N)=O N1(C(C(C)=O)=O)CC2(C1)C(NC(c1nc(C)c(C)nc1O)=O)CCS2(=O)=O C(C)(C(=O)OC(C)(C)C)(C(=O)N1C(C)COCC1C)SC C1(NC(c2cc(COC)c(F)cc2)=O)CC2CN(c3ncc(OC)cn3)CC2C1 Cc1cc(C)c(CCC(=O)OCC2(CC(=O)OC(C)(C)C)COC(C)C2)c(O)c1 C1(NC(C2(CC=C)CCCC2)=O)CC2CCCC(C1)N2C(=O)Cc1cnoc1 N1(C(CCC(CC)NC(c2nnsc2C)=O)=O)CCC(O)C(F)(F)C1 c1(C(=O)NC2CN(C(C=CC=CCC)=O)CC(O)C2)cc2nccnc2cc1F N(C1CCCc2c1cnn2C(C)(C)C)CC(=O)NC(C)(C)C CC1CN(C(C2CCC=CCC2)=O)CC1CC(=O)NC1CCC1(C)C C#Cc1cccc(C(N2CCN(C)C(CNC(C3CS(=O)(=O)C3)=O)C2)=O)c1 C(C(C(=O)NCCc1cscn1)NC(=O)CC1CC=CCC1)N(C)C C(CC(C(=O)N1CCC(C)(O)C1)NC(C1CC2(CC2)CO1)=O)N(C)C C=CC(F)(F)C(=O)NC1CC(C)N(C(c2cccnc2NC)=O)C1 c1(C(=O)NCC2CC3(CN(C(CC(CC)OC)=O)C3)C2)n[nH]c2ccc(Cl)cc12 c1(C(N2C(C)C3CC2C3NC(=O)CCCNC(N)=O)=O)c(F)ccc(N)c1F CC1(C)C2CCC(C2)C1C(=O)NCCC1CCCN1C(=O)COC1CCCC1 CN1CC(C(N2CCCC(CNC(=O)Cc3ccc(C4CC4)cc3)C2)=O)NC1=O C1(C(N2CC(F)(CNC(C(COC)C)=O)C2)=O)CNC(=O)N1C c1(CNC(C(C=CC)O)=O)ccc2c(c1)CN(C(c1ccc(F)c(F)c1C)=O)C2 CCCC(C)(O)CC(=O)NC(CC(=O)N(C1(c2cc[nH]n2)CC1)C)C(C)OC C(=O)(C(COC)CC(C)C)N1CCC(O)(C(C)NC(CC2(C=C)CCC2)=O)CC1 N1(C(c2cccc(OC(F)F)c2)C(=O)NC(CC)(C)C)CC2CCC(C1)C2(F)F c1(OC)cc(C(N2CC(C(C(=O)NC(COC)C(C)C)OC)C2)=O)[nH]n1 C(=O)(C(C)C1=CCCC1)NC1(CO)CCCN(C(c2cncc(OC)c2)=O)C1 N1(C(Cc2cc(C)on2)=O)CCC2(NC(=O)OC(C)(C)C)CCCCC12 N1(CC(c2ccccc2)C)CCCC(NC(=O)CCNC(N)=O)C1 CCC(CC(F)F)C(=O)N1CC(NC(c2ccc(C(F)(F)F)c(O)c2)=O)C(C)C1 N1(C(C(N2CCCC(O)C2)C)=O)CCCC1(C)CNC(c1ccoc1Cl)=O C1(C(=O)NCc2n(CC)ccn2)CCC2CCC1N2C(=O)CC1CNC(=O)O1 c1(-c2nc(CO)nn2CCCN2CCOCC2)ccnc(Cl)c1Cl C12C=CCN1C2=O.c1(CN(C)C)coc(CNC(=O)C=CC(=O)OC(C)(C)C)c1 N1(C(CC(=C=C)C)=O)CCN(C(c2scnc2Cl)=O)CC1CC(F)F c1(CN(C)CC2CNC(C)(C)C2)cccc(OCC(F)(F)F)n1 C1(C(=O)NCCC2CCSC2)CCCN(C(C2(Cl)CC2(F)F)=O)CC1 c1(C(=O)NCCN(C(c2c(C)[nH][nH]c2=N)=O)C)cc2cccc(F)c2o1 CC1(C)OCc2cc(NC(=O)Nc3cnn(-c4ccccc4F)c3N)ccc21 c1(C2(C(=O)NCC3CCC(NC(c4c(C)nc[nH]4)=O)C3)CCC2)ccccc1Cl c1(C(NNC(C2OCCN(CCN3CCCC(C)C3)C2)=O)=O)ccccc1[N+](=O)[O-] O=C(C1CCSc2ccccc21)NC1C2CC1N(C(C1CC3CC3C1)=O)C2 C(=O)(C(C)(COC)CC)NC(CCN(C(c1c(CC)occ1)=O)C)c1cccs1 C(=O)(CC(C)CC(=O)N1CCC12CN(C(=O)COC1CCCC1)C2)OC N1(CC2(C)CC(C)(C)C2)C2CCC1CC(n1cc(NC(=O)C(F)(F)F)nn1)C2 c1(CC(=O)NC(CNC(c2cc(C(C)(C)C)n[nH]2)=O)CO)cnn2c1CCCC2 C12(C(=O)NCC3N(C(c4n(CC)nnc4)=O)CCOC3)CC1COC21CCC1 c1(C(N2C(C)CCC2C(N2CCC(C(=O)N(C)C)C2)=O)=O)ccnc2ncccc12 C1(C(C)C)C(NC(C2(c3cccc(F)c3)CCC2)=O)CCN1C(=O)C1=CCSC1 Cc1ncccc1-c1cn(CC2CCCC2NC(C2CS(=O)C2)=O)nn1 c1(CC(=O)N(C2CCCN(C(=O)Cc3cccs3)C2)CC)cc(F)c(F)cc1F C1(CNC(CC=CC)=O)OCC2CCC1C2.C12C(C1(C)C)NC2=O CCC(C(=O)NCC1CC(F)(CNC(=O)Cn2nnc(=N)[nH]2)C1)C(F)(F)F c1(C(=O)NCC2CCC(NC(C3CCCSC3)=O)CC2)c[nH]nc1[N+](=O)[O-] c1(OC)cccc(C(c2ccc(F)cc2)(c2nnnn2C)NC2CC3CC3C2)c1 c1(CC(=O)NC(C)CN(C)C(C2(C#N)CCC2)=O)nn(C)c2ccccc12 C12(C(=O)NC3C(NC(c4nc(COC)sc4)=O)CCCC3)CC3CC(CC1C3)C2 c1(C(N2C(C)C(C(=O)NC3COC3)CC2)C(=O)N(C)C)cc(Cl)c(Cl)c(Cl)c1 C1(NC(c2n(C)ncc2)=O)CCN(C(=O)CC2CCCC(=O)N2)C1(C)C C1(NC(C2N(CC)CC2)=O)CC(F)(CNC(=O)C(c2ccccn2)OC)C1 C=CCC(C(=O)NC(CCC)C(O)C(=O)NCCN1CCCC(O)C1)C(C)C c1(C(=O)NCC2CN(C(C(C)Nc3scc(C)n3)=O)C(C)C2)cc(F)cnc1Cl c1(CCC(=O)NCC(CNC(CCC(=C)Br)=O)F)ccc(O)c(Cl)c1 C1(NCCN(C)C)CC2(CC2)C(=O)O1.C12(CCCC1)N(C(C)C)C2=O C12(CC(C)CNC(=O)C(=O)NCCOc3cccc(F)c3)CCC(CC1)C2 c1(C(N2CC(C)C(NC(c3cnc(N)c(Cl)c3)=O)C2)=O)cccc2c1CNC2=O N1(C(c2c(C)con2)=O)CCC2(CCCC2NC(C2(F)CCCCC2)=O)C1 O=S(=O)(c1ccnn1C1CC1(F)F)Nc1cnn(-c2ccccc2)n1 CC(O)C(C)C(=O)NCC1CCN(C(=O)CSC(=N)N)C1 C(=O)(C1=Cc2ccccc2C1)NC(C(=O)N(C(C#C)C)C)CCCOC C1(c2n(CCCCCCC)nnn2)(NCC(C)(C)C2CCC2)CC2CCC1CC2 c1(C(N(CC(C)NC(C(C=C)O)=O)CC)=O)ccc(-c2nnc(O)n2C)cc1 C1(C(N(CCC)CCNC(C2(C)CC(C)C2)=O)=O)CC(O)CN1C(=O)OC(C)C C(N=c1[nH]c(=NCCCc2nc(C3CC3)n[nH]2)[nH]c2c1CSC2)c1cnco1 N1(C(C2C(C)=C2)=O)CC(NC(C2(C)CC=C(C)CC2)=O)CC12CCOCC2 C1(NC(c2cc(C)sc2)=O)CC2(CCN(C(C3CC(=O)CO3)=O)C2)C1 c1(C(=O)NC(C)CCCNC(c2ncoc2C(C)(C)C)=O)cnc(Cl)c(F)c1N CCC(C)CC(=O)C(=O)N1CC2CC(C1)N2C(=O)C=CCF CCCCCCCCCC(C)CC(=O)N1CC2CCC(C1)N2C(C1SCCS1)=O C1(=CCNC(C(COC)O)=O)CCN(C(C2COC(=O)N2)=O)CC1 C(C1c2ccsc2CCN1C(C1CCCCC1)=O)NC(CC1(C)CCC1)=O C1(C(=O)NC2(C)CN(C(c3cnc(OC)s3)=O)C2)CC2CCCCN2C1 N1(C(CNC=O)=O)CC2CCC2(CC(=O)NC2(c3nn[nH]n3)CC2)C1 C1(CC(=O)NCC(C)=CC(=O)N(CC(C)(C)C)C2CC2)CCOCC1 Cc1ccc2c(c1)CCC(C(=O)NCC1CCN1C(c1cnsc1C)=O)O2 N1(C(C2(CCNC(C(C)OCCOC)=O)CCC2)=O)CCC(C)(C#N)C1 c1(C(N2CC3CCN(C(c4c(C)nn(C)c4)=O)C3C2)=O)cc(F)cc([N+](=O)[O-])c1 Cc1c(C(=O)N(C)CC2CCCN(C(=O)C(F)=CC3CC3)C2)ccc(F)c1F C1(N(C(c2c(C)sc(Cl)n2)=O)C)CCCN(CC2CC(C)(C)C2)CC1 C1(NC(c2cc(C)c(C(F)F)nc2)=O)CCCN(C(c2sccc2Cl)=O)CC1F c1(CCC(=O)N(CCNC(=O)Cc2cnco2)CC)cc(C)cs1 CC1CCN(C(=O)C(C)(C)CN(C)C)CCN1C(C1CCCCC(C)(C)C1)=O Cc1nn(C)c(C)c1C(=O)C(=O)NCCNC(=O)CN1C(=O)CCC1=O N1(C(C2C(CC)C2)=O)CC2(C1)CN(C(=O)C(O)c1ccsc1)CC(C)(C)O2 CC1CN(C(=O)CCCN2CCOCC2)CC1CNC(c1cccs1)=O N1(C(c2cccc(CCC)c2)=O)CCC(C)C(NC(=O)CN(C)C(C)=O)C1 N1(C(C2CC=CCN2C(c2cc(CO)[nH]n2)=O)=O)CCC(CO)C(O)C1 C(=O)(CC(O)(C(F)(F)F)c1ccccc1)Nc1ccc(OCC#N)nc1 Cc1ccc(F)c(CC(=O)NC(C)(CNC(C2(O)CCCCC2)=O)C2CC2)c1 C(=O)(C1=CC2C=CC1C2)N1CC(CC(=O)NC(C)C(C)(C)O)OCC1 Cn1ncc(C(=O)NCCC2CCCN2C(C2CCCCO2)=O)c1C(F)F C12(C(=O)NC(C(C)NC(C(CC)(C)OC)=O)CO)CC3CC(C1)CC(C)(C3)C2 c1(N2CCC(OCCOC)C2)nc(C)cc(=NC(C)CN2CCOCC2)[nH]1 N1(CCOC)CC(C(=O)NC(C)(C)CNC(c2csnc2C2CC2)=O)CC1=O C1(NC(=O)CCOC2CCC2)CC2(CCN(C(=O)CC3CCCCCO3)CC2)C1 N1(C(C(=O)N(C(C)C)C)C)CC2CCC1CN2C(c1c(Cl)nn(C)c1Cl)=O CC(C)CC(C)C(=O)N(C1CCN(C(c2coc(C3CCCC3)n2)=O)C1)C c1(C(C)NC(=O)C(C2CCN(Cc3occc3C(=O)O)C2)C)cc2ccccc2o1 c1(C(=O)Nc2c(-c3cn(C(CCC)C4CC4)nn3)n(C)nc2)c(C)cccc1Cl c1(N2CCC(OCC)C2)nc(=NCCC(C(F)(F)F)C(F)(F)F)[nH]c2c1CCC2 c1(C(=O)Nc2cccc(C)c2)ccc2c(c1)CN(C(c1nc(Br)ccc1C)=O)C2 c1(C(=O)NCC(CC)NC(=O)C(C)C23CC(C2)C3)c(F)cccc1F C1(NC(c2c(CNC(=O)CN3CCOC3=O)ocn2)=O)CC2(CCC2)C1O C1(CC(=O)NCC(C)(C)C(N)=O)CCCN(C(=O)CCc2cn[nH]c2)CC1 c1(C(=O)NC(C(C)NC(C2CC(OCC)C2)=O)C(C)C)cc(C)nc(Cl)c1N c1(C(=O)NCCNC(=O)Cc2ccc(F)cc2C(F)(F)F)cnc2n1CCCC2 CC(C)C(CO)C(=O)NCC1CCC(NC(=O)CC2CCC(C)(C)CC2)CC1 CN1CCCc2ccc(NC(c3cc(S(=O)(=O)CC4CC4)ccc3F)=O)cc2C1 Cc1ncc(C(=O)NCC2CC2NC(=O)Cn2cccnc2=O)n1C N1(C(c2c(C)coc2)=O)CCCC(N(C(=O)Cc2nc(=N)[nH][nH]2)CCO)C1 CC(C(=O)NC1(CNC(C2C(C)(C)C2(F)F)=O)CC1)S(=O)(=O)c1ccc(F)cc1 c1(CNC(CN(C2CC2)CC)=O)ccccc1CNC(C1C=C(C)CS1)=O N1(C(C2CCC(=C)CC2)=O)CCC2C(CCCN2C(C2CCC(O)CN2C)=O)C1 Cc1ccc(CNC(C2CCC(C)N2C(=O)C2=NOCC2)=O)cn1 CC1(C)CCCCC1C(N1CCC(C(O)CNC(C2CCC3(CC3)C2)=O)CC1)=O c1(C(=O)NC2C(OC)CN(C(C(CC)F)=O)C2)cc2n(n1)CCNC2=O O=C1NC2(CO1)CC(C(=O)NCC1CCN1C(=O)C1=COCCC1)C2 C1(C2CCCCN2C(=O)C=C2CCCC2)(CNC(C2CC2(F)F)=O)CCOCC1 C1(C)(C(=O)NCC(CCOC)NC(=O)C(CO)OC)CC2C=CC1C2 C1(C(N2C(C)(C)C(NC(=O)Cn3ccccc3=O)CC2)=O)Cc2nccnc2C1 C1(C)(C(=O)NC2CC(CCNC(c3c(C)cn(C)n3)=O)C2)CCOC12CC2(F)F Cc1onc(C(=O)N(C)CCN(C)C(C2CC2CC(C)C)=O)c1Br N1(C(C2(CC)CCCC2O)=O)CC2(C1)CN(C(c1[nH]c(C)cc1C)=O)CCO2 C(=O)(CC(C(F)(F)F)NC(=O)C(CC)CCC)O.O(CP(C)(C)=O)C(CC)CC C(=O)(CC(O)C(Cl)(Cl)Cl)N1CC(OC2CCN(C(C(C=C)O)=O)CC2)C1 c1(NC(=O)C(N2CC3C4CCC(C4)C23)=O)cc2cc(Br)ccc2o1 N1(C(COCCCC)=O)CCC(NC(=O)CC2CC2C2CC2)C1C1CC1 C1(C(c2nnnn2C)NCC2CN(C)CCO2)(OCCC)CCCCC1 C(CC(C)(C)C(=O)N1CCN(C)C(CNC(C2CCCO2)=O)C1)SC CCCC(C)(C)C(=O)N1CCN(C(=O)CCc2nncs2)C(c2ccccn2)C1 C1(CC(=O)NCC#CCC)CC(NC(c2nc(C)oc2C)=O)C1(C)C C1(NC(CNC(=O)CCF)=O)C2CCCN(C(C3CCC4(CC3)CC4)=O)C12 N1(C(C2C(CC)CCC2)=O)CC2CC3CC2C1C3NC(c1ccncc1OC)=O N1(C(c2ccn(C(C)C)n2)C(=O)NCC2CCCO2)CC(C)CC1C c1(CNC(N(C(C)CC(N)=O)C)=O)ccccc1OC1CCC1 C(C(C)(CC)C(=O)Nc1cnc(C)c(Cl)c1)NC(C1C(CC)CCO1)=O N1(C(=O)CN2CCCC2)CCOC2(C1)CN(Cc1cc(O)ccc1[N+](=O)[O-])C2 C1(CC)CCCCC1C(=O)Nc1ncc(CCNC(=O)CSc2ccccc2)s1 c1(N2CC(NC(C(CC)SC)=O)(COC)C2)ncncc1OC N1(C(C(COCC)C)=O)CCC(NC(=O)CCC2CCC2)CC(O)C1 c1(CC)ccc(C(C)CC(=O)N(CCCN(C(=O)Cn2cc(N)cn2)C)C)cc1 CC(C)C(C(=O)N1CCC(OCCNC(c2cccn2C)=O)C1)NC=O c1(CCNC(c2c(OC)ccc(C(N)=O)c2)=O)c[nH]c2ccc(C)cc12 c1(OCCC(=O)NC(C)C(C)NC(=O)C=Cc2cn[nH]c2)cc(Cl)cc(Cl)c1 c1(CNC(c2c(Br)n[nH]c2C)c2n(C(CC)C)nnn2)ccc2ccccc2n1 C1(C(=O)NCC2CCCC(CNC(C3(C(N)=O)CC3)=O)C2)CC2(C1)CC21CC1 c1(OCC(=O)NC2CC(C)(CNC(c3c(C)nn(C)c3)=O)C2)ccc(F)c(F)c1 C1(C(N(CCOC)CCNC(C2(S(C)(=O)=O)CC2)=O)=O)CCn2cc(C)nc2C1 C(C(C(C)C(C)C)NC(c1n[nH]c(C)c1Br)=O)NC(C(F)=CCC)=O C1(COC)(CNC(C2CCOC(C)(C)C2)=O)CCN(C(=O)Cc2ccco2)CC1 c1(C(N2CCN(C(CC3CC(C(=O)OC)C3)=O)C3C2C3)=O)cccc2nccn12 c1(-c2ccc(OCC)c(OC)c2)nc2c(s1)CN(C(C1CCCCCC1)=O)CC2 c1(OC)c(C(c2ccccc2)NC(=O)N(C2COC2)C(C)C)cccc1Cl C(=O)(C1CCOc2ccc(Cl)cc21)N1C(CNC(c2cnn(C)c2N)=O)CC1 Cc1cc(C(=O)N(C)CC2CCCC(NC(C3CC(OC4CC4)C3)=O)C2)sc1Cl N1(C(C=COCC)=O)CCC(O)(CCNC(c2cn(C)nc2C(=O)OC)=O)C1 C=CC(F)(F)C(=O)N1CCOC(CCNC(c2cn(C(F)F)cn2)=O)C1 N1(C(CN(C)CC)=O)CCCN(C(=O)CSc2cn[nH]c2)C(C)C1 Cc1conc1CC(=O)NCC1CC(CNC(=O)CNC(=O)C(F)(F)F)CO1 C1(NC(c2ccc(OC)c(F)c2)=O)CC2CN(C(=O)CN3CC(C)(C)C3)CC2C1 CC1(C)C(CNC(=O)CCC2CC(NC(=O)CN3CCC(F)CC3)C2)C1(F)F C1(O)(CNC(C2(C)CN(C(CN3CCC(C)C3)=O)C2)=O)CCCCC1 C1(NC(C(c2cnn(-c3ccccc3)c2)N(C2CCCC2)CC)=O)CC(F)(F)C1 C1(NC(c2c(C)[nH]nc2Cl)=O)CCCCCC1NC(c1cc(O)cc(Br)c1)=O C1(C)(NC(c2n(CC)ccc2)=O)CCCCC1C(=O)NC(C)(C)CC(=O)OC C1(CC(=O)NCCOCCCC)CN(C(c2cnc(C)s2)=O)CCO1 C1(CC(=O)NC2(CC)CC2)CCN(C(=O)CNC(=O)NC)C1 CCC(C)(C)CC(=O)NN1CCCC1C(=O)NCC(C)(C)CO Cc1cc(C(=O)NC(C)C(CO)NC(=O)CCOCC2CC2)cs1 N1(C(=O)CC(F)(F)F)CCC2C(C1)CN2C(c1cnn(CC(F)F)n1)=O C(=O)(C1CCc2ccc(OC)cc21)N(C)CC1N(C(CSCC)=O)CCC1 c1(OC)cc(C(N2CCC(NC(=O)Cc3cnsc3)C2)=O)ccc1C#N C1(CC(=O)NC(c2cccnc2O)C)CN(C(c2cnn(C)c2)=O)CC12CC2 O=C(C1Cc2ccc(Cl)cc21)NCC12CC1CN(C(=O)CCC(F)F)C2 c1(OC)cccc2ccc(C(=O)NCC3(F)CC(NC(C)=O)C3)nc12 C1(C(=O)NCC2CCN(CCC)C2)CCCCN1C(C1(CO)CCC1)=O N1(C(C(C)C(C)(C)C)=O)CC2CCCC(N(C)C(C3CCCCN3N=O)=O)C2C1 C#CCC(C(=O)N1CCCCC1CF)NC(c1oc(C)nc1CC)=O C1(CN(CC(C)O)C)CCCN1C(=O)CCCC1CCC1 C1(CC)CN(C(=O)C(CCF)NC(=O)C2=C(C)CCC2)C(C)CO1 c1(CC)nc(C)c(C(=O)NCC2(NC(=O)C(C)Cc3cnco3)CCOC2)o1 c1(OCC(C)C)cccc(C(=O)N(C(C)CNC(=O)C=C(Cl)Cl)C)c1 C(C(C)C)(C(O)C(=O)NCC1(NC(C2CC2(C)C(F)F)=O)CCC1)OC C12(C(=O)NCc3nnc4n3CCC4)CCC(CC1)N(C(=O)C=C1CCOCC1)C2 C1(NC(c2c(O)ccc(SC)c2)=O)CN(C(=O)C(C)SC(C)C)CC2(CCC2)C1 C1(C(N(C(c2c(C)ccc(C)c2)C)C)=O)CC2(CCCC2)CO1 CCC(C)CCCCC(=O)N(CCCCCC(=O)NC1(C)CC(F)C1)C N1(C(c2c(C)ocn2)=O)CCCC2(CCN(C(c3cc4n(n3)CC(F)C4)=O)C2)C1 C#CCC(C)(C(=O)N=c1cc(C)n(C)[nH]1)NC(=O)CC(O)CC(C)C c1(COC)ccoc1C(=O)NCC1CCN(C(C2CCC(C(N)=O)C2)=O)C1 C(=O)(CCCC(C)(C)C)NC1C(C)CN(C(=O)C2=C(Cl)N(CC(F)(F)F)C2)CC1 N1(C(c2cncc(N)n2)=O)CCN(C(C2CC(F)(CO)C2)=O)C2CCC12 C1(C(=O)OC(C)(C)C)(CCC(N2CCC(O)C2)=O)CCCO1 CC1C(NC(c2cccc(F)n2)=O)CCN1C(=O)Cc1ccccc1Cl CCC(C(=O)N(C1CCCC1C)C)NC(c1scnc1Cl)=O CC1CC(CCNC(c2cnc(N)c(Cl)c2)=O)CCN1C(=O)Cc1cnoc1 C1(C(=O)NCCCCC(N)=O)(CC)CCCN(C(=O)C2=C(C)CCC2)C1 N1(C(C(N)Cc2ccc(SC(F)(F)F)cc2)=O)CCCS(=O)(=O)CC1C1CC1 Cc1cc(NC(C2CCN(C(=O)C(C)CC(F)F)CC2O)=O)cc(F)c1 c1(C(=O)NC2(CC(=O)NCCn3c(CC)nnc3)CCC2)ccc(C#N)[nH]1 C(=O)(N1CC2COCC2O1)C12C(CCN(C(Cc3n(C)ccn3)=O)CC1)C2 c1(-n2cc(CN(C(C)(C)CO)CC)nn2)c(C(C)C)cccc1C c1(C(=O)NCCCCNC(c2cn(CCC=C)nn2)=O)[nH]c2c(c1C)CCCC2 N1(C(C(CC)NC(C)=O)=O)CC2CCC(NC(c3ccc(C)nc3SC)=O)C2C1 C1(C)(CNC(C2(C(=O)OC)CC2C)=O)CCN(C(=O)CCN2C(=O)CCC2=O)C1 N#Cc1ccc(CSCC(=O)NC2CC2NC(C2(C3CCC3)CCC2)=O)cc1 C(C)(CNC(c1ccc(O)c(N)n1)=O)(CC(C)C)NC(Cc1c(C)n[nH]c1C)=O N1(C(C2(CC)CC2)=O)CCC(O)(CNC(=O)C(c2ccc(Cl)s2)C)CC1 C1(COC)(NC(c2cc(C(F)(F)F)c[nH]2)=O)CN(C(c2coc(C(C)C)n2)=O)C1 N(C1CCCn2ncnc21)C(C(CC#C)NC(c1c[nH]c(C#N)c1)=O)=O c1(C(C(N2CCC(N(C(Cc3ccn(CC)n3)=O)C)C2)=O)(C)C)cccc(F)c1 c1(CC2(C(=O)NCC(C)NC(c3cnc(C(C)OC)s3)=O)CC2)cccc(Cl)c1 O=C1NCC2(CN(C(=O)NC3(c4ccc(F)cc4F)CC3)C2)N1 CCC(C)C(C(=O)NCC1CC(O)CN1C(c1csc(-c2ccsc2)n1)=O)OC c1(NC(c2c(-c3cccc(OC)n3)nccc2)=O)c(C)ccnc1C c1(C(=O)NCC(c2ccccc2)NC(C(C)(CO)OC)=O)ccc([N+](=O)[O-])[nH]1 c1(C(N(CCCNC(CSCC)=O)C)=O)nc(N(C)C)nc(=N)[nH]1 c1(N2CCC(CC(N)=O)C2)ccc(S(=O)(=O)NCCn2ncc(Br)n2)cn1 C(=O)(C(CC)C(=O)N1CCCC1C1(O)CN(C(c2cnc[nH]2)=O)C1)OCC c1(C(=O)NC(CNC(C(C(C)C)F)=O)(C)C(C)C)cncc2cc(Cl)ccc12 c1(C(=O)NCCN(C(C)C(=O)NC)CCOC)cccc2ccncc12 C(=O)(C(CC1CCC1)NC(C1CC(C(C)(C)C)C1)=O)N(CC(F)F)C CCCCCC(=O)NC1CCC1C(=O)NC(=O)CSCC(=O)N(C(C)C)CC N1(C(C(C2CC2)OCC)=O)CCC(C(N2CC(C#N)C2)=O)C1CC N1(C=O)CCC2CN(C(C3C4CC5C(C4=O)C35)=O)C2C1.c1ccc(C(C)(C)C)[nH]1 N1(C(c2c(C)nc[nH]2)=O)CCN(C(=O)C(C)N(CC(F)(F)F)C)C(COC)C1 N1(C(c2c(C)c(Br)cnc2)=O)CC2(C1)CN(C(=O)C#CC1CC1)CC2CO CC(C)CC(O)C(=O)N1CCC2CC12C(N1CC2(CC=CC2)C1)=O C1(CC(=O)NCC2C=CC(NC(CC=C)=O)C2)CCCC(F)(F)C1 c1(C(=O)NCCCNC(c2c(C)nc(C3CC3)o2)=O)coc2ccc(Cl)cc12 N1(C(CN(C2CC2)CC)=O)CC(NC(=O)C=CC=C(Cl)Cl)C(c2ccccc2)C1 C1(NC(CS(N)(=O)=O)=O)COCCN(C(c2cccs2)=O)C1 c1(C(=O)NCC2C=CC(NC(c3c(C)nco3)=O)C2)ccc(F)c2[nH]ccc12 C1(C(=O)NCC2CCN(C(C3(OC)CCCC3)=O)C2)CCOCC12CCCCC2 c1(C(N2C(Cn3cc(-c4c(C)cncc4)nn3)CCC2)=O)cc(Cl)nnc1O CCN=C(NCC(=O)NOCc1ccnn1C)NCCc1ccc(Cl)cc1 CCC(CC)C(C)C(=O)NC1CCC1C(=O)NC1CCN(C(C)C)CC1 N1(CCOC)CC(C(=O)NCC2C(C)CCN2C(=O)Cc2n[nH]c(C)n2)CC1=O c1(CC)ccc(OCC(=O)NC(C)(C)C(C)NC(=O)C(CSC)OC)cc1 C1(OC)CCC(C(=O)NCc2nnnn2C)CC1.C12CC(C1(C)C)CC(=O)N2 Cc1ccc(Br)c(C(=O)NCC2COCCN2C(C2CC2(C)C)=O)c1F c1(OC)cc(C)cc(C(N2CC=C(CCNC(=O)CC3CC(F)C3)CC2)=O)c1O c1(C(N2CCNC(=O)C23CCC3)C(=O)NC(CC)C)ccc([N+](=O)[O-])c(Cl)c1 c1(C(N(CC(CNC(c2c(COC)cco2)=O)C)C)=O)c(O)cccc1Cl C1(C(C)C)COCCN(C(=O)C(O)Cc2cnc[nH]2)C1.c12ccc(Cl)cc1S2 N1(C(c2ccc(OC(F)F)cn2)C(=O)NCCC)CCC2OC(=O)OC2C1 c1(SCC(N2CC(C)C(NC(=O)COC3CC3)C2)=O)nc2ccccc2s1 c1(CC(=O)NCCN(C2CCCC2)C(C2C(CN(C)C)C2)=O)ccc(O)c(Cl)c1 C1(NC(c2cc(C)ncn2)=O)CC2CN(C(c3cscn3)=O)CC12 C(CC(=O)N1CCC(C#N)(CC)CC1)(CC(C)C)NC(C(C)NC(CC)=O)=O C1(O)(CNC(CCC(N)=O)=O)CCN(C(c2ccsc2)=O)CC1 C1(C(N(C2CCN(C(C3CCCC3)=O)CC2)CCC)=O)Oc2ccccc2C1C Cc1ncc(CNC(C2(c3cc(F)cc(F)c3)CCCC2)=O)c(=N)[nH]1 [N-]=[N+]=NCCCCC(=O)NC(Cc1ccco1)C(=O)NCC1CN(C(N)=O)C1 c1(CCC(=O)NC2CCN(C(CSCC#C)=O)C2C(C)C)c(C)nn(C)c1C C1(C(=O)OC)CCCN(C(C2CCN(C(=O)Cc3cccc(Br)c3)C2)=O)C1 c1(OCC(=O)NCCC2CN(C(C3C(C)(COC)C3)=O)C2)c(C)occc1=O C(=O)(C1=CCC(NC(C2(C)COC(=O)N2)=O)C1)N(C1CC(CO)C1)C C(CCC(=O)NC(C)C(C)NC(c1cnc(-c2cccs2)s1)=O)NC(=O)OCC C1(O)(CCNC(C2(C)CNC(=O)C2)=O)CCN(C(C2CCCCC2)=O)CC1 c1(Cn2cc(C3CCN(C(C(CN(C)C)O)=O)C3)nn2)ccc(N)cc1 C1(N2CCC(O)CC2)C2CCC1CN(C(=O)C=Cc1cccs1)C2.CC(C)N(C)C N1(C(C(C(C)(C)C)OC(C)(C)C)=O)CC(C2CN(C(=O)C(Cl)=CCl)C2)C1 Oc1ncnc2c1CCN(Cc1nnc3ccccn13)CC2 c1(N(C)C)cnc(CNCC#CCCO)cn1.N12CCC(C1)n1cc(nn1)C2=O N1(c2nccc(OC)n2)CCC(C2CCN(C(C3CCC(F)(F)CC3)=O)CC2)C1 C(=O)(CC(C)CC(=O)OC)NCc1c(C(=O)NCCc2cn(CC)nn2)con1 c1(C(=O)NC(C)C(C)NC(c2n[nH]cc2[N+](=O)[O-])=O)cccc2ncn(C)c12 c1(CC(C)NC(=O)C(O)(C(F)(F)F)c2ccccc2)c[nH]c2ccc(F)cc12 CCC(C)(C)C(O)C(=O)N1CC2(C1)CN(C(c1nnn(C)c1C)=O)C2 C1(C)(C)CC(F)C(=O)N1.C(C(O)C(C)C)N(C(C(SC)SC)=O)C C#CC1(O)CCN(C(C23CC(CO)(CN2C(c2csc(O)n2)=O)C3)=O)C1 C(=O)(C1=CCN(C(=O)CC2CC3CC3C2)CC1)NCC1(O)CCC(C)C1 N1(C(c2nn[nH]c2Cl)=O)CCC2CN(C(c3ccc(-c4ccon4)cc3)=O)C2C1 C(=O)(CC1=CCOCC1)NCCCC(C(=O)N1C(CN(C)C)C=CC1)O c1(C(N2C(CN(C(=O)C(CO)C(C)(C)C)C)COCC2)=O)c(F)ccc(N)c1F c1(C(=O)NC2CCC(F)(CNC(C(CC=C)C)=O)C2)ncc(C)cc1Br C1(C(N(C(C(C)SC)C)C)=O)C(C2CC2)CCN1C(C1Cc2ccccc2C1)=O c1(C(N2CC(C(C)NC(C(C(=C)Cl)(C)C)=O)OCC2)=O)ccc2c(c1)CC(=O)N2 C1(Cc2cccc(C)c2)CC1C1CCCC1.c12ccnc(c1)C(=O)OC2 N1(C(COC(C)=O)=O)CCCC2(CCCCC2NC(c2nc(Cl)sc2C)=O)C1 C1(CCC(=O)NC2CC(CNC(CN(C3CCC3)C)=O)C2)CCC(=O)N1 c1(NCC(N2CCCCC2)=O)cc(=NCc2ncc[nH]c2=O)[nH]cn1 Cc1nc(C(N2CC(C)(C(=O)Nc3cccnc3C)C2)=O)ccc1F CCCCC(O)CC(=O)N1CCC(C)(C(=O)NCCN(C(C)C)CC)CC1 N1(C(CC2N(CC)CCOC2)=O)C2CCCC1CN(C(C1CCS(=O)(=O)C1)=O)C2 c1(C(=O)NCC(CCNC(c2c(CC)cco2)=O)O)cnncc1C c1(C(C)N(C)C(C2CC(C(C)(C)C)C2)=O)nn[nH]n1.C1(C2CC2)CN1C c1(C(C(=O)NCC(C)C)N(CC(CCC)C)C)ccc(F)c(C)c1 N1(CCNC(C(C)N(C(=O)C=Cc2ccc[nH]2)C2CC2)=O)CCCOC1=O C#CC1CCCN(C(=O)C(C2CCCCC2)NC(C2CCC2C#N)=O)CC1 c1(OCCCOCC)cnc(C(=O)NCCNC(C2CCCC(O)C2)=O)c(Cl)c1 C1(CC)CN(C(=O)CCN(C(=O)Cc2cn(C)cn2)C)CCN1C C(=O)(CC(O)CC(C)(C)C)NC1(CC(N2C3CN(C(C)C)C(C3)C2)=O)CCC1 C1(CNC(C2CC(=C)C2)=O)CN(C(c2ccc(=O)n(C)c2)=O)CCC1C c1(OC)ccc(CN(C(=O)C=CC(F)(F)F)C(C2CCC(C)CC2)C)c(OC)c1 CC1CC(NC(c2cc(C#N)cs2)=O)CCN1C(=O)C=Cc1ccc(Cl)s1 CC1(CO)CCC(N=c2[nH]c(=NCc3cncs3)[nH]c3c2SCC3)CC1 c1(C(N2C(CCNC(C(C(CC)O)C)=O)COCC2)=O)ccc(C#N)nc1O C(=O)(C(CCC1CCC1)NC(c1cocn1)=O)NC(CC)C c1(C(=O)NCC(CC(C)C)NC(=O)C(F)F)cc(C(F)(F)F)cc(O)n1 C1(NC(CC2CC(=O)C2)=O)CCN(C(c2csc(Cl)n2)=O)CC12CCC2 C(CNC(=O)Cc1csnn1)(CC(F)(F)F)NC(C(N1CC(C)C1)C)=O C1(C(=O)NCC2(C(=O)NC(CC)C3CCC3)CCCC2)CCN(C)CC1 N1(C(C2(C(N(C)C)=O)CC2)=O)CCN(C(c2cc(S(N)(=O)=O)cs2)=O)CC(O)C1 C(C(=O)NC1(CNC(C2(C(N)=O)CC2)=O)CCOC1)(C(F)(F)F)OC(C)=O C12(C(N(CCNC(C(CCC)O)=O)CCC)=O)CC(c3ccccc3)(C1)C2(F)F c1(CC2(CC(=O)N(CC(C)(C)NC(COCC(=C)C)=O)C)CC2)ccccc1 N1(C(CC(C)F)=O)CCC2CN(C(c3csc(-c4cnc[nH]4)n3)=O)CC12 C1(NC(C2(COC)CC(F)(F)C2)=O)CN(C(c2cn(C)[nH]c2=N)=O)C2(CCC2)C1 N1(C(=O)CC2CCCN(C(c3ccc(O)cc3)=O)CC2)CCC2(CCCC2)C1 Cc1cc(CC(N2CCC(C(C)NC(C3CC(O)C3)=O)C2)=O)ccc1Cl C(=O)(C#CC1CCCCC1)NCCN(C(c1cn(CC(C)O)c(=O)cc1)=O)C1CC1 CC1CCOC(C(=O)NC(C2CCCN2C(=O)CCNC(=O)CO)C)C1 c1(C(N2CCC3(NC(c4nn(C)c(O)c4)=O)C(C2)C3)=O)ccc(Cl)c(N)c1Cl CCCC(O)C(CO)NC(=O)C=CC(C)NC(=O)CCN(C)C1CC1 c1(C(=O)NC2(CO)CCN(C(C3(C)CCCC3)=O)C2)ccc(NC(N)=O)cc1 c1(C(=O)NCC(C)N(C(=O)CCC2CCCCO2)CC)cc(C)nc(O)n1 C(=O)(C1=CCCC1(C)C)N1CCN(C(c2nn(C)c(F)c2)=O)CC1CCO C(CCCC(=O)N(C(CNC(=O)CC1CCCCC1O)CC)C)OCC CCN=c1ccc(C(N2CC(NC(C3(C)CC(F)(F)C3)=O)CC3(CC3)C2)=O)c[nH]1 C(c1ccc(S(N)(=O)=O)cc1)=CC(=O)N(C(C)CNC(C1C(C)C1C)=O)C CN1CCC2CN(C(c3conc3CNC(C3CCCCC3)=O)=O)CC12 Cc1cc(C(N2CC(O)(CCNC(=O)Cc3cnnn3C)C2)=O)c(C)cn1 c1(C(N2CC(OC)(CNC(C3CCSC(C)C3)=O)C2)=O)cc2ccccn2n1 C(=O)(C1CCc2nccn21)N1CC2(CC(NC(C(C)C(=O)N3CCOCC3)=O)C2)C1 C1(C2CCN(C(=O)CC3CCC(=O)NC3=O)C2)(NC(c2c(C)coc2)=O)CC1 C12(C(N3CCC(NC(CNS(CC)(=O)=O)=O)C(F)C3)=O)CCOC1CCOC2 C1(Nc2cc(C(=O)NC(CC)CN(C)C(C)=O)ncc2)CCN(C)C1=O N1(C(c2c(C)cn(C)c2)=O)CC2CC(C(=O)Nc3cn(C)nc3C)C(C2)C1 C(=O)(C1CCCn2nccc21)NC1CC(C(C)NC(=O)CS(=O)(=O)N(C)C)C1 N1(C(C2C(C)CCO2)=O)CCCC2C(NC(=O)CCc3n[nH]c(=N)s3)C(C)(C)C12 c1(OC)c(C(N2CCC2CNC(c2ccnc3[nH]ncc23)=O)=O)cc(Cl)cc1Cl c1(NC(C(c2scc(C)c2C)N(c2scc(C)n2)CC2CC2)=O)ccccc1C N1(C(C)C2CC2)CCCC(C)(C(N2CCOCC(NC(C3CCC3)=O)C2)=O)C1 CS(=O)CCC(=O)NCCCNC(c1scnc1Br)=O c1(C(N(CC#C)C2CC2)=O)ccn(CCNC(=O)Cc2ccc[nH]2)c1 CCCCC(O)C(=O)N1CCC(CNC(=O)CC(C)(F)F)C1(C)C C1(CCC(=O)NC(CC)CNC(c2cnn(CC(F)(F)F)c2)=O)C(=O)ON=C1C C1(N(C(C(C2CN(C(C(C=C)C)=O)C2)OC)=O)C)CCOC(C)C1 c1(C(C(=O)NC2C(NC(C3CC4CC4C3)=O)CC2)CO)ccc(Cl)cc1 CC(C)S(=O)(=O)CC(=O)N1CCCC1CCNC(c1cc(C(F)(F)F)cs1)=O c1(SCC(=O)C2CC2)ccc(Cl)cc1.C12CCC(CC1)NC(=O)C1(CC1)C2 N1(C(c2c(F)ccc(F)c2Cl)=O)CCC2(CCCN2C(C23CC(F)C2C3)=O)C1 Cn1cc(S(C)(=O)=O)c(C(=O)NCCCNC(c2ccc(C3CC3)cn2)=O)n1 Cc1cn2c(C(=O)NCC3CCC(C)CN3C(=O)C=CCN(C)C)c(Cl)nc2s1 C(=O)(C#CC1CCC2(CC1)OCCO2)N1CC(NC(C(C(C)C)C)=O)(CO)C1 c1(N2CC(NC(C3(C(C)C)CCC3)=O)CC(F)(F)C2)ncnc2c(Br)c[nH]c12 C(=O)(C1Cc2ccc(F)cc21)N(C1CCN(C(C2CCc3nncn3C2)=O)C1)C c12ccc(cc1)S(=O)(=O)N(C(C)C)C2.C1(C(N(CC)CC)=O)COC(C)(C)CN1 c1(C(N(CC(C(=O)NCC)OC)c2ccccc2)=O)n[nH]c2c1CCOC2 Cc1ccccc1C=CC(N1CCC(NC(C2(C)CC=CCO2)=O)C1)=O C12(CNC(c3csc(Br)c3)=O)CCC1CN(C(=O)C(O)CN1CCCC1)C2 c1(C(=O)NCCCN(C(=O)C(c2cnn(C)c2)C)C(C)C)cnc(O)cc1O c1(C(C(=O)NC(C(C)NC(C=CC(C)C)=O)(C)C)=O)ccc(F)c(F)c1 C1(C(N2CCCC(NC(c3c(CC)ocn3)=O)(CO)C2)=O)CCCC(C)(C)CC1 c1(CC(=O)NCCCNC(COc2c(C)c(Cl)ccc2)=O)cnc2n1CCOC2 c1(C(=O)NC2CCC(C)N(C(=O)CC3CCSCC3)C2)cc2cc(F)ccc2s1 CC1(CNC(C2COCCO2)=O)CCCN(C(C2CC3(CCO2)CC3)=O)C1 C1(C(N(CCC(C(C)C)NC(c2cnco2)=O)C)=O)C2Cc3cc(Cl)ccc3C12 C12CCN(CC1)CCc1csc(n1)C2.C1(C)(C(C)(C)C)CC(C(=O)O)C1 c1(C(=O)OC)ccc(S(=O)(=O)NCCC2CCC(F)(F)C2)c(Cl)c1 c1(C2C(C(=O)NCC3CCN3C(=O)C(=O)NC3CC3)C2)c(F)cccc1Cl c1(SC)nccc(N2CC3C(NC(c4cnoc4-c4ccco4)=O)C3C2)n1 N1(C(c2[nH]cc(C(=O)OC)c2)=O)CCOCC12CCN(C(C1(CO)CC1)=O)C2 N1(C(c2ccc(C(C)C)cc2)=O)CCCC(C)(C(N2CCCC2C#N)=O)C1 CC1CC(CO)CCN1C(C12CC1CCN2C(=O)CNC(=O)C(C)(C)C)=O N1(C(CC=CC=C)=O)CCC2(CCOCC2)C(CNC(=O)Cn2[nH]cnc2=N)C1 C1(C(=O)NCC2CC(NC(C3CCS3(=O)=O)=O)C2)(OC)CCC12CCC2 C(CC1=CCCCCC1)NC(C1C2(CCN(C(C3=C(C)OCC3)=O)C2)C1)=O C1(CC(=O)NCC(CC=C)NC(c2cnc(N(C)C)nc2)=O)COC(C)(C)C1 c1(CCC(=O)NCC2(F)CC(NC(=O)CC3CCC(=O)N3)C2)ccc(Cl)nc1 C1(NC(CN(C(COC)=O)C)=O)CCCC1NC(=O)C(F)(F)C1(OC)CCC1 c1(CC)c(C(=O)NCC2CC(COC)CN2C(=O)CC)nnn1CC.C(C)=O c1(NC(C2CC3(C2)CN(Cc2cnccc2C(F)(F)F)C3)=O)nccc(Cl)c1I N1(C(c2c(C)[nH]c(C#N)c2)=O)CC(C(=O)NC(C)C(C)C)CC12CCC2 C(C)(N=c1nc(Cl)[nH]n2c(Br)cnc12)c1ccc(OC)cc1OC c1(C(=O)OCC)cncc(NC(C2CCCN2Cc2nccn2C)=O)n1 C1(NC(c2ccc(C)nc2C)=O)CCN(C(=O)Cc2cccnc2O)CC(O)C1 Cc1cc(Br)ccc1S(=O)(=O)NC12CC(C(=O)N=c3cc(Cl)cn[nH]3)(C1)C2 N(C(=NCc1ccc(C(F)(F)F)cn1)N1CCC(CNC(N)=O)C1)OC(C)C c1(C(=O)NC2CN(Cc3c(Br)ccc(OC)c3)CC2C#N)ccc2nc[nH]c2c1 C1(C(=O)NC2(CC(=O)NC(C(CC)C)CN(C)C)CCC2)CCC(=O)N(C)C1 c1(C(=O)NC2C(C)N(C(c3nc(=N)cc[nH]3)=O)CCC2)cc([N+](=O)[O-])cnc1O Cn1c(S)nc2cc(C(=O)NCCCNC(C3CCC3CF)=O)ccc2c1=O CN1CCN(c2nnc(-c3ccon3)s2)C(CNC(c2cc(F)cnc2O)=O)C1 N1(C(CC2CCN(C(c3c(NC)cncc3)=O)C2)=O)CC(C)CC1(C)C c1(C(=O)OCC)c(NC(=O)NC(C2CCN(CC)CC2)C)cnn1C C1(NC(CNC(CC)=O)=O)CC2CCC(C1)N2C(=O)Cc1occc1C c1(CC)nc(C)[nH]c1C(=O)N(C1CCCC(NC(c2c[nH]nc2Br)=O)C1)C N(C1CCSc2ccc(F)cc21)C(C(C(C)(C)C)n1cc(CCC(CC)O)nn1)=O C1(C(N(C(CCC)C)C)=O)CN(C)CCN1C(=O)COC(C)(C)C c1(C(N2C(CC(=O)NCC(C)(C)C(N)=O)COCC2)=O)ccc2ncoc2c1 S(=O)(=O)(c1ccc(C(N2CC(NC(=O)COCC3CC3)C2)=O)cc1)NC CC1CC(=O)NCC1C(N1CCN(C(C2CCN(C)CC2)=O)C(CO)C1)=O c1(C(=O)NC2CN(C(=O)C3=CCSC3)CC23CC3)cc(Cl)c(F)cc1F C(=O)(C(CN(C)C)NC(C)=O)N1C(C(=O)NC2(CC#C)CC2)CC1.OCC C1(C)(C(N(CCCNC(CN(C)C(N)=O)=O)C)=O)Cc2ccccc2NC1=O C(=O)(C1=CCCCCC1)N(C)CC1N(C(CC(C)O)=O)CCCC1 N1(C(=O)CCc2cnccn2)CCN(C(c2cnn3c2CCCC3)=O)C2CCC12 C1(C(=O)NCc2cncc(C(=O)NC(CO)C3CCC3)c2)CCC(=O)NC1 C12(C(=O)NCc3nccc(C(=O)NC4(C(=O)OC)CC4)c3)C(=O)C3CC1C2C3 C1(NS(Cc2ccc(C)cc2)(=O)=O)CCCCN(Cc2ccc(O)c(C(=O)O)c2)C1 N1(C(c2c(C)ccnc2O)=O)CCC2(CC1)CC2NC(c1ccc(O)nc1Cl)=O N1(c2ncc(C)cn2)CCCC2(CCCN(C(C3CCSCC3)=O)C2)C1 c1(CNC(C2(C=C)CCC2)=O)cnn2c1CN(C(c1cc(C)on1)=O)CC2 C(=O)(CCCCCNC(=O)COCCOC)NCC(=O)N(CCC(F)(F)F)CC c1(CNC(CC(=C)C)=O)nnc2n1CCN(C(c1cnc3sccn13)=O)C2 Cc1coc(C)c1C=CC(N1CC(CNC(C2(C)CCOCC2)=O)C(O)C1)=O CC(C)CC(C(=O)NCC1CCOC1)N(C(=O)CC1CC2(CC2)C1)C C(=O)(CC(C)C(C)(C)NC(=O)C(CC)C(=O)OCC)N(CCC#C)CCO N12CCCC(C1)C(=O)N2.C(=O)(C(C)(C)CO)NC(c1ccccc1)C(C)N(C)C c1(C(N2CCC(NC(CC3(C)CC3(Cl)Cl)=O)C2)=O)nc(O)nc(O)c1F C1(C(N2CC(O)(CNC(=O)CC3CCCSC3)C2)=O)CCC(=O)N1C1CC1 C=C(C)CC(C(=O)NCCCN(C)C1CC1)NC(c1cc(OCC)ns1)=O.OCC c1(C(=O)NC23CC(C(N4CC(O)C(F)C4)=O)(C2)C3)c(F)ccc2[nH]ccc12 C(=O)(C(CC(F)F)C1CCC1)NCCOC1CN(C(COc2cc(C)on2)=O)C1 N1(C(C2(C#N)CCCO2)=O)CC2CC(C1)CN(C(=O)CCc1cc(Cl)cs1)C2 N1(C(C(=O)NCCOC)CCC2CC2)CCC(C(=O)OC)C12CC2 Cc1ccc2cc(C(N3CCC(c4nnc(S)n4C)CC3)=O)cnc2c1 c1(-c2n(C3CCCC(C)C3)nc(C3CC34CC4)n2)cnc(Cl)c(Br)c1 c1(C(C)=O)cn(CC(=O)NCC(C2CCC2)NC(C2CCC3CC23)=O)nn1 N1(c2cc(OC)ncn2)CC2(CCC(C(=O)Nc3cccc(Cl)c3C)O2)C1 c1(-n2ncc(C(=O)NCC3N(C(COC4(C)CCCC4)=O)CC3)c2)ncc(Cl)cn1 Cn1cnn(CC(=O)NCC2CN(C(=O)CN3CSCC3=O)C2)c1=O C=CC(C)(O)CC(=O)N(CC)CC1CCN(C(c2nccc(Cl)c2C)=O)CC1 C1(C)(C(=O)NC2CCC(CNC(C3(OC)CCOCC3)=O)CC2)CCC(=O)CC1 C1(CNC(c2n(CC(=C)C)nnn2)(C2CCOCC2)C)CC2CCC1CC2 CC(C)=C=CC(=O)NC(C(=O)NC(c1n[nH]c(CO)n1)C)C1CCC1 C1(C(=O)NCc2c(CNC(C3(C)COCCO3)=O)cccc2)CC12CCOCC2 C1(C(N2CC3C(CNC(CCNC(=O)C=CCl)=O)C3C2)=O)CC2(C1)CC(CO)C2 N1(C(CC(C)(C(F)F)N(C)C)=O)CCC2(CCCCN(C(c3csnn3)=O)C2)C1 c1(N)cn2c(n1)CCC2.N1(C(C=C(C)Cl)=O)CC(F)C1 c1(C(=O)NC(c2ccncc2)CC=C)cc(Cl)nc(Cl)n1 N1(C(c2n(CCC)ncc2)=O)CCC(C(=O)NCC2CCCN2CC)=C(F)C1 C(=O)(C1=CS(=O)CCC1)NC1C(NC(C(C)CN2CCCCC2)=O)C1 c1(NC)ccc(C(=O)NC2CC(N(C)C(C3CC(C(F)(F)F)C3)=O)C2)c(Cl)c1 CCS(=O)(=O)c1ccc(-c2cc3cc[nH]c3cc2C(=O)Nc2nc(Br)cs2)cn1 C1(NC(C(c2ccc(C)cc2)F)=O)CC(O)CN(C(=O)CCCN2CCCC2)C1 c1(C(=O)NC(CCCNC(COCC)=O)c2ccccc2)c2c(nn1C)CCC2 N1(C(=O)CC2(O)CCC2)CCC2CCN(C(=O)COc3cccc(Cl)c3Cl)C2C1 c1(CC)nc(C)sc1C(=O)N(C)CCOCCN(C(=O)Cc1ccccc1F)C c1(C(=O)NC(C)(CNC(C2CCNC2=O)=O)C2CC2)nc(C2CC2)n2ccccc12 c1(C(N2CC(NC(C3CCCC(CC(F)(F)F)C3)=O)(CO)C2)=O)ccccc1F c1(C(=O)NC2CC(CNC(CCC(C)OC)=O)C2)ccc(Br)cc1N C12(NC(=O)CC(=O)NCC(F)(F)F)CCCN(C1)C2=O.C1(C)(CC)CCCCC1 O(P(=O)(CCC1CCCCO1)OCC)CC c1(C(=O)NC(CC)CN(C)C(C2CC(=O)NC2(C)C)=O)cc(Cl)cc(Cl)c1N CC1(C)CCN(C(=O)C(C#N)CCCc2ccccc2)CC1NC(=O)C=C(Cl)Cl c1(C(=O)OC)ccc(NNC(=O)C(C)NS(=O)(=O)c2cccc(Cl)c2)cc1 N1(C(C(CC(F)F)NC(c2cc(C)sc2)=O)=O)CCCCCCCC1 C1(NC(C2(C#C)CCCC2)=O)CC2(CCN(C(=O)CCc3cccc(C)c3)C2)C1 n1(CC)nc(C)c(C(=O)NCCC2CC(NC(=O)C3=CCCCO3)C2)c1C CC1CN(C(=O)CCC(=O)N(C)C)CCC1CNC(c1ncccc1F)=O C(=O)(CC(C)(C)N(C)C)N(CCC(=O)NCC(CC)O)CCCO c1(CNC(C(CC)(C)CC)=O)nc(C(F)(F)F)n2c1CCCC2 c1(C(N(C)Cc2nnc(C)o2)=O)ccc(O)c(Cl)n1 C(=O)(C(CO)C(C)(C)C)N1CC(N(C(CS)=O)CCC)C(O)C1.SC N1(C(c2cnc(CCCC)s2)=O)CCOC(C)(CNC(C2(CO)CCCO2)=O)C1 CC(CCNCc1ccccc1OCC(F)(F)F)C(F)F CC1(C)CCCCCC1NC(C1C2CCCC2CN1C(C1CCSC1)=O)=O c1(C(=O)OCC)[nH]cc(C)c1C(=O)NC1CN(C(C2(C)CS(=O)(=O)C2)=O)CC1C CC1=C(C(=O)N2CCOC(CCNC(c3cncc(Cl)c3Cl)=O)C2)CCCO1 c1(C(N(CC(C)O)CCNC(C(C)SC(C)C)=O)=O)nc2ccccc2nc1O C1(CNC(c2onc(C)n2)=O)CCC(NC(=O)C(C)CF)CC1 C(N=C(NC(C)C)N1CCC(OC(C)C)C1)Sc1cc(OC)cc(C(F)(F)F)c1 Cc1cccn2cc(C(N3CCCC(F)(CNC(=O)CCCN=[N+]=[N-])C3)=O)nc12 C1(CNC(COC2CCC(C)CC2)=O)CC2(CC2)CN1C(=O)C(C)N(C)C C1(CC(NOCCCC)=O)CCC(C(NC(C)(C)C)OC)CC1 c1(C(=O)NC(C(C)(C)C)CNC(C2CCCSC2)=O)cc(F)c(F)cc1Cl C1(C(N(CCNC(CCC#CC)=O)CC2CC2)=O)CCC(O)(C(F)(F)F)CC1 N1(C(Cc2cc(C)no2)=O)CCC(C)C(CC(=O)NC2(C)CCSC2)C1 Cc1cccn2ncc(C(=O)NC(C)CCN(C(=O)C=C3CC3)C)c12 C(=O)(CC(CC(N)=O)CC(C)C)NCC1N(C(C(CC#C)CC#C)=O)CC=C1 n1(CC(=O)NC2CC(N3CCNCC3)C2)ccc(C(=O)O)n1 N1(C(C2C(=C)C2)=O)CCC(CNC(c2cscc2C2CC2)=O)CC1C c1(-n2cc(CONC(c3cnc(C4CC4)s3)=O)nn2)cc2ccc(Br)cc2[nH]1 C1(NC(C(C)n2cnnn2)=O)CCCC2CN(C(=O)C(O)CC(C)(C)C)CC12 c1(NC(=O)NC(c2ccc(F)c(Br)c2)(C)C)cncc(P(C)(C)=O)c1 C1(CNC(c2c(Cl)cn(CC)n2)=O)CN(C(C2CCC23CCC3)=O)CC12CCC2 c1(CC)cc(C(=O)OCc2ccc(Cl)cc2)cc(Cc2ccc(OC)cc2)c1 C1(CNC(CCCNC(C)=O)=O)COCC2(CCN(C(=O)C=CC=C(Cl)Cl)CC2)O1 c1(C(N2CC3CCN(Cc4cocn4)C3C2)=O)cc(I)ccc1[N+](=O)[O-] c1(CCNC(C2(COC)CN(C(=O)C=C(C)C3CC3)C2)=O)cccnc1O N1(C(c2c(OC)noc2C)=O)CC2(CCC(NC(=O)CC(C)C)CC2)C1 N1(C(CCC(CC)C)=O)CCC2CN(C(=O)CCC(C)(C)N(C)C)C2C1 C1(CNC(Cc2cncc(C)c2)=O)CCN(C(c2nccc(Cl)c2C)=O)CC1C c1(C(N2CC(C)C(CNC(C3(CF)CC3)=O)C2)=O)csc2c1CCC(C)(C)C2 N1(C(c2ccc(OC)cn2)=O)CCN(C(=O)CCCCC2CCCCC2)C2CC12 C1(NC(=O)NC(Cc2cccnc2)CO)COCC1C(=O)O c12cncc(c1)N1CC(O)CC(C1)C(=O)NC2.C1(N(CC)CC)CSC(C)C1 Cc1cc(=O)n(CC(N2CC3CC(CNC(c4ccon4)=O)C3C2)=O)cn1 C(c1ccc2c(c1)NC(=O)CO2)=CC(=O)NCC(CC)NC(CSCCC)=O c1(CC(=O)NC(CC)(C)CNC(c2ccsc2OC)=O)ccc2c(c1)CCCO2 CCCC(C(=O)NCC(F)(F)C(F)F)NC(c1cn(CC)nn1)=O c1(CNC(C=CC(C)NC(C(C)NC(C)=O)=O)=O)nc(C)c(C)[nH]1 N1(C(=O)CC2CCCOC2)CC2CCC1CN2C(c1cc2ncccc2o1)=O C1(C(=O)NC(COC)COC)(CC)CCCN(C(=O)CP(C)(C)=O)C1 C1(C(=O)NCCc2ccc(CNC(=O)OC(C)(C)C)cc2)CCCCC12CCC2 C(=O)(C(CNC(C)=O)C(C)C)NCC(CC(=O)NC(CCC)C(=O)N(C)C)C c1(NCC(=O)NCC2C(CNC(C=CC=CC)=O)C2)ccc(C)cc1 C1(CC(NOCCCOC)=O)CC(C)(C)CN1C(=O)Cn1c(O)nnc1O N1(C(=O)C2CC2)CCCCC1NCc1cnc(C(C)C)s1 Cc1cccc2ncnc(N3CC(NC(c4cncn4C(C)C)=O)CC3C)c12 C(CC(=O)O)(c1cccnc1)N(C(N(C(COC(F)F)CO)C)=O)CCN c1(C(=O)NC2(CNC(C(C)=C(CC)C)=O)CCC2)cnn(CC(F)(F)F)c1 c1(CC)cc(Br)ccc1C(N1CC(NC(c2cc(I)ccc2F)=O)C(O)C1)=O C(=O)(CC(F)(F)C(F)(F)F)N1CCC(N(C(c2ccnc(C)n2)=O)C)C2(C1)CC2 C1(NC(c2c(C)nn(C)n2)=O)CCC2CCN(C(c3cnsn3)=O)C1C2 c1(C(N2CC(C(C)NC(C3CCN(C)CC3)=O)C2)=O)cc2n(c1)CCCC2 N1(C(C(C)(C)NS(C)(=O)=O)=O)C2CCC1CN(C(c1cncc(N(C)C)c1)=O)C2 CC1(C)CN(C(=O)CCNCCCOc2ccc(Cl)cc2)C1C1CC1 N1(C(CC2C(C)CCO2)=O)CCC(C2CC2)C1CNC(=O)C(c1ccncc1)C CC1CN(C(C2(C)CC2(F)Cl)=O)CC(C)N(C(c2n[nH]c(C3CC3)n2)=O)C1 CC1c2cc(Br)ccc2CCN1CC(=O)NCC1CCc2ccccc21 N1(C(C(CSC)O)=O)CC(C2CN(C(=O)C(C(C)C)NC(C)=O)C2)C1 N1(C(c2scc(OC)c2)=O)CCC(CF)(NC(=O)C(F)C(C)C)C1 CC1Cc2cc(S(N)(=O)=O)ccc2N1C(=O)CSCc1cc(Br)cnc1Cl C1(C)(CC)CC(C(=O)NC(C)CNC(c2ccc(NC(=O)NC)s2)=O)CCO1 CC1CCN(C(c2cccnc2C(F)(F)F)=O)CC1CNC(C1(C)CCCO1)=O n1(CCOC)ncc(C(=O)NC2CN(C(=O)CCCN3CCCC3)CC2F)c1C N1(CCCC)CCOCC1C(=O)NCC(C)NC(=O)CCc1ccc(C)s1 c1(CN(C(=O)C(C)(O)CC)c2cc(C(=O)OC)[nH]c2)cn(C)nc1-c1ccccn1 N1(C(c2ccc(OC)cc2)=O)C2CCCC1COC2.N12CC3C(C3C1)OCC2=O C1(CCNC(C23CC(CO)(C2)C3)=O)(OC)CN(C(c2cnc(C(C)C)[nH]2)=O)C1 c1(C(=O)NCC2(C)CCN(C(C3(c4cc[nH]n4)CC3)=O)C2)cnn2c1OCCC2 N1(C(CCC=C=C)=O)CCCCC(C2CN(C(=O)CC(=O)NCC(F)(F)F)C2)C1 C(=O)(C(O)CC(C)(C)C)N1CCCCC(C(=O)Nc2ccc(CN(C)C)cc2)C1 C#Cc1ccc(C(N2CCN(CC(N3CC4CC3CN4C)=O)C(=O)C2)=O)cc1 c1(C(N2C3CCN(C(c4c(C)onc4)=O)C3CC2)=O)ccc2nc(Cl)ccc2c1 CC1CCC(N(C(c2cn(CCNC3(C)COC3)nn2)=O)C2CC2)CC1 N1(C(CC(CC)C)=O)CCOC(C)(CNC(c2c(Cl)c(C)nn2C)=O)C1 c1(C(=O)NCCC(C)N(C)C(C2CC3CCC2O3)=O)cc(Cl)c(Br)[nH]1 c1(OC)c(C(=O)NC23CCC(CC2NC(C2CNC(=O)C2)=O)C3)cc(Cl)cc1Cl c1(OC)ccccc1C(CNC(C1CCCN1c1ccccc1)=O)NC(C)=O C1(C)(N(C(c2cccs2)C)Cc2ccc(F)cc2)CCC(O)CC1 N1(CC(C)C)CCC(C(=O)NC(C2CN(C(C3(CF)CCOCC3)=O)C2)C)CC1 C1(CNC(=O)Cn2cnnc2)CC2CCCC2N1C(=O)CSC1CCS(=O)(=O)C1 c1(OC)ccc(C(=O)NCC2CC(C)N(C(c3ccccc3C)=O)C2)c(OC)c1 N1(C(CC(CC)CC)=O)CCN(C(=O)C(C)Cc2ccnn2C)CC(O)C1 c1(OC)ccc2c(c1)C(NC(=O)C(N1CC3CC(O)CC1C3)=O)CCC2 c1(C(N2CCN(C(Cc3ccc(C)cc3)=O)C(C)C2)=O)c(C)ccc(C)c1N C(=O)(CC(C)(C)C(=O)N(CC(C)NC(c1cncc(Cl)n1)=O)C)OC C1(CNC(CC(CN(C)C)(C)C)=O)CC2CCCCC2N1C(C1CCC1)=O c1(CCC2(CNC(CC)=O)CC2)cncc(C(=O)OC)c1.C12CC1CNC2=O c1(C(=O)NCC(CNC(c2cccc(C3CC3(F)F)c2)=O)O)cc(F)ccc1O c1(C(=O)NC2(CNC(C(C)(C)CO)=O)CCOC2)cncc2cccnc12 c1(NCc2ncc(OC)nc2)nccc(=NCc2nnc(C)n2C)[nH]1 C1(OC)CCCC(CNC(=O)CN(C)C(c2nc(C)oc2OC(C)C)=O)C1 Cc1nn(C)c(C)c1C(=O)C(=O)N(C)CCOCCN(C)C(c1cnsc1)=O c1(C(N(C2CC(NC(C3(C(F)F)CC(F)(F)C3)=O)C2)C)=O)cnc2n1CCC2 C1(OC)CCCC(NC(=O)CC2(N(C(=O)C=C3CCCCC3)C)CC2)C1 CS(=O)(=O)c1ccsc1C(=O)NCCCCC(CO)NC(=O)Cc1cnccn1 C(=O)(CCN(OC)C(=O)C1CCN(C(=O)CC2CC(OC)C2)C1C)OC CC1CN(C(C2(O)CCC2)=O)CC2(CCN(C(C3CCCOC3C)=O)C2)O1 C1(CC(=O)NCC2(OCC)CC2)CC(F)CN1C(=O)C=CC1CC1 C(=O)(C(O)C(CCC)NC(C1CCS1(=O)=O)=O)NC1(C#C)CC(F)(F)C1 C=CC1CCN(C(C2(OC)CCN(C(=O)Cc3cn(C)cn3)C2)=O)C1 C1(CNC(C(C)(C)C)=O)CN(C(C2CCCCCC2)=O)CCC1C(F)(F)F N(C1CCc2cccnc21)C(C12C(NC(c3c(C)nccn3)=O)C3CC1C2C3)=O N1(C(C2(n3cc(C(c4cccc(C)c4)O)nn3)CC2)=O)CCCC2C(O)C(C)(C)C12 Cc1c(C(N2C(C(=O)NCC(F)CO)CC2C)=O)cccc1C#N C1(NC(C2CCCCC2)=O)CCCC12CCN(C(c1cc(Br)cs1)=O)C2 c1(C(N2C3(CNC(C4CCCC(C)C4)=O)CC(C2)C3)=O)csc([N+](=O)[O-])c1 Cc1ccc(CCC(=O)NC2CCC(NC(C3SCCCS3)=O)C2)cn1 C1(CN(C(C(C)c2ccsc2)=O)C)CCCN(C(c2cn(C)nc2C2CC2)=O)C1 N1(C(CNC(CC(C)C)=O)=O)CC(NC(C2CC=CC2)=O)CCC1C C1(N(C(C(C(C)O)N(C)C)=O)C)CCCCN(C(c2ccc(O)cc2)=O)C1 Cc1cc(CN2CCC(CO)CC2)n2nc(C)cc2n1.N12CCCC1CCC2=O CC12CCCCC1CN2C(C(=O)NC1CCC1)C1CC1 N1(C(Cn2ccc(C)n2)=O)CCC(CCNC(=O)C(c2c(C)n[nH]c2C)C)CC1 c1(OCC)cc(C=CC(=O)NCc2ccc(C3CC3)cc2C)cc(Cl)c1O N1(C(C2ON=C(CC)C2)=O)CCC2C(CCCN2C(=O)C(C)=C2CCC2)C1 c1(C(C)=O)ccc(C(N2CCCC2CC(C)NC(=O)C(O)C2CC2)=O)c(C)c1 C1(C(C(=O)NCc2cccs2)N(C)Cc2cn(CC)nc2)CCC2(CC1)CC2 N1(C(CC2(C)CC2(Cl)Cl)=O)CCOC(CNC(=O)Cc2cccc(C(N)=O)c2)C1 C1(C(=O)NCC2C(NC(c3cn(C)nc3C(F)F)=O)C2)CCC2(CCC2)O1 c1(C(N2CC(C)C(NC(=O)C=CC(C)(C)C)C2)=O)cc(Br)ncc1F C1(C(=O)NC(C)CN2CCN(C)CC2)CC12CCN(C(c1cnns1)=O)CC2 N1(C(C=CC)=O)CCC(C2(NC(c3cccn3CCC)=O)CC2)C1 Cc1cc(C(=O)NC(C)CC2CCN(C(=O)CC(C)(C)F)C2)ccc1C(N)=O C1(CNC(C2C(C)COCC2)=O)CC2(C1)CC(N)CCO2 c1(C(=O)NC2(CCNC(Cc3n(C)ncc3)=O)CCC2)cccc(C(F)F)c1 N1(C(CNC(COCC(=C)C)=O)=O)CCCN(C(c2nn[nH]c2Cl)=O)CC1 CC1CCC(NC(c2cncc(-n3cnnn3)c2)=O)CN1C(=O)CCC(C)(C)C N1(C(CCNC(C)=O)=O)CC2CCC1C(CNC(=O)CSc1nncn1C)C2 C1(NC(c2cncc(CC)c2)=O)CCCN(C(=O)Cc2ccnn2C)CC1 c1(C(=O)NCC(O)CCNC(C2(F)CCC2)=O)cnc2ccc(F)cn12 N1(C(CN(C(C(C)N2CCCC2)=O)CC2CC2)=O)CC(N(C)C)C(C)(C)C1 N1(C(c2ncn(C)c(=O)c2)=O)CC2(C1)CN(C(c1csc(Cl)c1)=O)CC(C)(C)O2 N1(C(c2cc(C)n(C)n2)=O)C2CCC1C(NC(=O)CCOCC1CCCO1)C2 C1(C(=O)NCC2(CCNC(=O)C(O)c3ccsc3)CC2)CC12CCOCC2 CC(C)(C)C(CNC(c1ncc(F)cn1)=O)NC(=O)C(F)C1CC1 c1(C(=O)OCc2ccc(O)cc2)cnn2c1OCC2 N1(C(CN(C)C(=O)C2CC2)=O)CC2(CCN(C(c3csc(Cl)n3)=O)CC2)C1 C(=O)(CC(C)CN(C)C)NCC(CC)NC(=O)CCc1ccc(C(C)C)cc1 C1(CNC(c2ccc(OCC#C)cc2)=O)CN(C(C2CCCN2C)=O)CC12CC2 c1(C(Cn2cccn2)NC(C(=O)N(C23CC(C2)C3)C)=O)ccccc1 C1(OC)CN(C(=O)CCCNC(=O)C(C)(C)C2CC2)CC12CC2 S(=O)(=O)(c1c[nH]ccc1=NCc1nc(Cl)cs1)N1CCCC(C)(CCC)C1 c1(C(=O)NCCCCC2CCCN(C(C(C)(C)SC)=O)C2)cnc(O)n(C)c1=O C1(OC)(CNC(=O)Cc2cncn2C)CCN(C(=O)C(c2ccc(F)cc2)=O)C1 Cc1csc2ncc(C(N3CC4CCN(C(=O)CC5CCCO5)C4C3)=O)c(=O)n12 C1(NC(Cc2n(C)ccc2)=O)CC2CCC1(C(=O)NCCCC(C)(C)O)C2 N1(C(c2ccc(C)c(Cl)c2Cl)=O)CC2COCC(C1)C2NC(=O)C(Cl)=CCl C(=O)(CC(C)CC(C)(C)C)N1CC(O)(CNC(C(C)N(C)C)=O)C1 C=CCCC(C(=O)NCCCNC(=O)NC)NC(=O)C=CCCC c1(CCC(=O)N(C)CC2N(C(CC(CC)C)=O)CCCC2)cccc(C#N)c1 C1(C(=O)NC(CC)CNC(c2cc(Cl)c(Cl)s2)=O)CCc2nncn2C1 Cc1cnc(CN2CC(C(N3CC(O)C(F)C3)=O)CC(F)C2)c(F)c1 c1(C(N2C(C)CC(NC(c3cc(CCC)[nH]n3)=O)C2)=O)coc2c(C)cccc12 CN1CCN(C(C2CCCN(C3CCC(=O)NC3)C2)=O)CC1 c1(C(=O)OCC)c(C)sc(CNC(CC2CCCN2C)C2CC2)c1Cl N1(C(C2CC2C2CCC2)=O)CC2CCCC(C1)N2C(C1CCC2CC2CC1)=O c1(CC)cc(C(N2CC=CC2CNC(C2CC(N(C)CC)C2)=O)=O)ns1 Cc1cc(OCC(=O)NC2(CNC(c3cc(Cl)cn3C)=O)CCCC2)cc(C)c1 c1(CN2CCN(C3CN(C(C4C5COCC45)=O)C3)CC2)ccc(O)cc1O O=S(=O)(c1cccc(C(F)F)c1)N1CCN(CCNCc2cc(Br)ncc2Br)CC1 CC1CN(C(C2(S(N)(=O)=O)CCC2)=O)CCC1NC(=O)C(C)CC1CCC1 C1(CNC(c2c(OC)ccs2)=O)CN(C(C2C3(CC3)C23CC3)=O)CC2(CCC2)O1 C1(C(=O)NCC2C(NC(C(c3nc(C)sc3)=O)=O)CCC2)CCCCCC1 N#Cc1cccc(C2CCCN2Cc2ccc(-c3ccc(F)cc3)nn2)c1 Cc1sc(C(=O)NC2CC(O)CN(C(c3coc(N(C)C)n3)=O)C2)c(C)c1C c1(C(N(C(C(=O)NCCC(O)C(F)F)C2CC2)C)=O)ccc(C(N)=O)cc1 C1(CCNC(C(C)(O)C2CCC2)=O)CSCCN1C(c1cccnc1N)=O N1(CCNC(COC2CC(NC(C3(CC=C)CCOC3)=O)C2)=O)CCCC(C)C1 c1(C(=O)OC)ccc2ncc(N3CCCC(C4CC4(F)F)C3)nc2c1 C1(C(=O)NCCCOCCNC(n2cnc(C(C)=O)n2)=O)CC(C(C)C)=NO1 Cc1nc(C(N2CCN(C3CN(C(=O)C=CCF)C3)CC2)=O)c2ccccn12 Cn1c(C(=O)NCCC2CN(C(c3nc(C4CC4)cs3)=O)C2)cnc1S C1(NC(CS(=O)(=O)NC)=O)CC2CCC1CN2C(=O)Cc1ccccc1O CC1C(NC(c2cnc(Cl)c(C3CC3)c2)=O)CCCN1C(C1CC2(CSC2)C1)=O C1(C(=O)NC(COC)C)C2CCCC1CN(Cc1c(Br)cc(Br)c(O)c1Br)C2 S(=O)(=O)(CCCNC(C)(C(C)(C)C)c1nnnn1C1CCOC1)N(C)C c1(C(=O)NC(CNC(C(CC)OC)=O)C2CC2)cc2nc(Cl)ccc2o1 CC(C)C(C(=O)NCCc1ocnc1CO)C(C)NC(=O)CNC(N)=O CC1(C)CC(CNC(c2ccccc2)=O)CN(C(c2nnn3ccccc23)=O)C1 Cc1ccc(COCC(=O)NC2CC(CCNC(=O)CCC3OCCO3)C2)cc1 C1(C(C)NC(c2ccn(C(F)F)n2)=O)CCCN(C(=O)C=C2CCCC2)C1 N1(CCONC(C2ON=C(C)C2)=O)CC(O)CC1CO c1(C(=O)OC)ccc(C(=O)NCC2CCCCCN2C(c2cnco2)=O)cc1Cl C(=O)(CCCCCCNC(c1coc(C2CC2)n1)=O)N1C(C)CC(O)C1 c1(OCC)ccccc1C(=O)N(C(C)CNC(=O)C(F)(F)c1ccccn1)C c1(C(N(C2CCN(C(=O)CCCC(C)=O)C2)CC)=O)n[nH]c2c1CCOC2 N1(C(CSCCC#N)=O)CC(C2(NC(C3(Sc4ccccc4)CC3)=O)CC2)C1 C(c1ccc(Br)cc1)=CCCNC(c1c(C)nccc1)=O c1(C(N2CCC(NC(c3ccns3)=O)CC2C2CC2)=O)cccc2c1COCC2 C#Cc1cccc(C(=O)NCCNC(c2cc(O)nc(OC)n2)=O)c1F C(=O)(C(C)CN(C(=O)CCc1cnco1)C)NC(C#C)CC CC1CCC(NC(=O)CCCSC(C)(C)C)CN1C(c1cc(C(F)F)ncn1)=O C1(CC(=O)NCCN(C)C2CC2)CCN(CC2CCC2C(=O)NC(C)(C)C)CC1 C12(C(=O)NCc3nccc(C)c3)CC(CO)(CN1C(C1CC3COCC3C1)=O)C2 C1(C(=O)NC(C2OCCC2C)C)(CCNC(=O)CCc2cn(C)nn2)CCCC1 c1(NC2CC(C)N(C(C3(CN(C)C)CC3)=O)C2)cc2nncn2cn1 c1(OC)cccc(Cl)c1CNC(N1CCC(C)C(NC(=O)OC(C)(C)C)C1)=O C(=O)(CC(C)CN=C(NCC1CCCCO1)NCC(C)(C)C(F)(F)F)OC C1(C(=O)NCC2CC(F)(F)CO2)(COCC)CCCCO1 C1(NC(c2cc(-c3ccncc3)ccn2)=O)CC2CN(C(=O)CSC3CC3)CC2C1 C1(CNC(C2(CC)CCCO2)=O)CC(C(=O)Nc2cc(C)ccc2O)=NO1 C1(CNC(CC(C)(C)C#N)=O)CN(C(c2ncc(F)cn2)=O)C2(CCOCC2)C1 Cc1nc(C(N2CC(NC(c3ccccc3OC(F)(F)F)=O)C3CC23)=O)c(C)s1 c1(CNC(c2cccc(C(=O)NC(C(=O)OCC)C)c2)=O)cncc(OCC)n1 Cc1cc(=NCCOc2ncccn2)[nH]cc1S(=O)(=O)NCC(C)C(F)(F)F C#Cc1ccc(C(N2CC(C(=O)O)CC(C(=O)O)C2)=O)cc1C N1(C(c2cnc(SC)n2C)=O)CCC(NC(C2CC2C)=O)C(F)C1 C1(NC(COCCOCC)=O)CN(C(C2CCC(O)CC2)=O)CC1C C(=O)(C(F)C(=O)N1CCN(CCNC(=O)CCc2ccnn2C)CC1)OCC Cn1cc(Cl)c(CC(=O)NC2CCCCC2NC(=O)C(O)C(F)F)n1 C1(NC(c2sccc2F)=O)C2CC1CN(C(C1COCCC1(F)F)=O)C2 CN=c1[nH]cc(C(=O)NCC(C)C(=O)NCCc2c(C)n[nH]c2C)s1 c1(N2CCN(C(c3ccnc(OC)n3)=O)CC2C)nc(Cl)nc2[nH]cnc12 c1(CNC(NC2C(C)(C)CC2)=NCCOCCO)cccc2c(Cl)c[nH]c12 c1(C(=O)NCC(C)NC(=O)C2=CCCC2)cc2ccnn2cn1 c1(C(N2CC(C(N3CCC(OCC)C3)=O)(SC)C2)=O)cnncc1O c1(OC)ccc(CN2CC(C)(CNC(=O)COC3CCOC3)C2)c([N+](=O)[O-])c1 Cc1cc(C(=O)NCC23CC2CN(C(=O)C#CC2CC2)C3)ccc1F C1(CNC(CCCOCC)=O)(OC)CCCN(C(=O)C(C)C(F)F)C1 C1(C)(CNC(CC2CCCC(C)O2)=O)CC(F)(F)CN1C(c1cnn[nH]1)=O CCC(C)C(O)CC(=O)NCC(C)(C)C(=O)N(C1CCC1C)C C1(F)(C(=O)NC2CCC(CC(=O)N(C)Cc3cncnc3O)C2)C(C)(C)C1(C)C Cc1ccc(S(=O)(=O)NC(CCC(N)=O)C(=O)NC2CCCCC2(F)F)c(F)c1 C1(CC=C)CC(O)CCN1Cc1ccc(C)cc1C CCCC(CC)C(=O)NC1CCCCC1CNC(c1ccc(F)s1)=O N1(C(Cc2c(C)cco2)=O)CCC(CO)(NC(C2CC23CC3)=O)CC1 C(Cn1nnnc1C(C(C)(C)C)c1ccccc1)(C(C)C)OC.C1CCS1 c1(OCC)cc(NCC2CC(NC(C3CC3F)=O)C2)nc(C)n1 Cc1nc(Br)ccc1C(C)NC(=O)C(N1CCN(C(C)CN)CC1)=O N1(C(c2c(C)snn2)=O)CC(NC(c2cn(C)cc2C(F)(F)F)=O)CC(O)C1 c1(CCC(=O)NC2C(CNC(C3N(CC)CCC3)=O)CC2)nc2ccccc2s1 Cc1cc(N2CCOCC(CNC(=O)CCCC3CCC3)C2)nc(S(C)(=O)=O)n1 C1(C(N2CCC(CNC(c3cncc(SC)c3)=O)(CO)C2)=O)CCN(C)C(=O)C1 c1(C(N2CCN(C(CC(CCC)C)=O)CC2CCO)=O)cc(F)c(C#N)c(F)c1 C1(NC(C(C)=CC2CC2)=O)COC2(C1)CN(C(C1CC(=O)N(CC3CC3)C1)=O)C2 CC(C)CCC(F)C(=O)NCC(CC1CC1)C(=O)Nc1cccc(C(N)=O)c1 C12(NC(C3CC3c3cccnc3)=O)CCCC1N(C(=O)C=CBr)CC2 N1(C(c2c(C(C)=O)ccs2)=O)C2CCC1CC(NC(C1C=CCC1)=O)C2 Cc1cccc2cc(C(=O)NC(C3CN(C(=O)CSCc4ncc[nH]4)C3)C)oc12 CC(C)CC(C)(C)C(=O)NC1CCCC1NC(c1ccccc1SC(F)(F)F)=O C1(NC(CC(C)F)=O)CCC(NC(c2nccnc2N)=O)CC1 C(=O)(C(C)CO)N(C(C(=O)NCCOC(C)C)C1CC1)C N1(C(c2cc(OC)c(Br)nc2)=O)CCC(C)(C)C(NC(C2CCC2)=O)C1 CCCC(CC1CCCC1)C(=O)NC(C)(CNC(=O)C(C)(C)CO)C(C)C C1(NC(C(CC=C)OC)=O)COC2(C1)CN(C(=O)CC1OCCO1)C2 c1(CNC(C2C(NC(=O)Nc3cccc(OC)c3)C2)=O)cc(C)ccc1F N1(C(CC2CCC(C)CO2)=O)CC2CC(C1)CN(C(C13C=CC(CC1)C3)=O)C2 c1(C(N2CC(NC(C3C(CCC)CCC3)=O)(CO)C2)=O)cnc2c(c1)COC2 c1(OC)ccccc1CNC(=O)C(c1ccsc1)N(CC(=O)N(C)C)C Cc1ccc(C(N2CCCC(N(C(=O)CC3CCC(C)CO3)C)C2)=O)cc1C C1(C(N2CCCC(C=C)C2)C(=O)NCC(=C)C)Cc2ccccc2C1 c1(C(N2CC(CC(N3CCC(c4ccccc4)C3)=O)C2)=O)ccc(F)c(I)c1 C1(NC(C(CC2CCC2)OC)=O)CCC(C)(CNC(C2CCC(=O)O2)=O)C1 Cc1cc(Cl)c(Cl)cc1C(=O)NC1CN(C(=O)C(O)CC(N)=O)C2(CCC2)C1 N(C1CCCc2occc21)C(C(c1ccco1)NC(C(=CC1CCCC1)C)=O)=O C1(C2CCCN(C(=O)CN(c3ccncc3)C)C2)(NC(CN(C)C(N)=O)=O)CC1 c1(C(=O)NCC(c2ccccc2)NC(C2CC23CCCC3)=O)ncc(Cl)cc1Cl C1(NC(C2CCNC2=O)=O)CC=CCC1C(N1CC(c2nn[nH]n2)C1)=O C=C1CCN(C(C2COCOC2)=O)C(C(N2CCC(OCCO)C2)=O)C1 N1(C(Cc2c(C)nc[nH]2)=O)CC2CCC1CN2C(C1C=CCS1)=O c1(C(=O)NC(C2CCCC2)CNC(=O)C=Cc2ccc[nH]2)cc2c(s1)CCC2 N1(C(COCCN(C)C)=O)CC(C)(C(N2CCC3(CCC3)C2)=O)CC1(C)C c1(C(N2CCC(O)(CNC(CC(C)OC)=O)C2)=O)cnc(=NCCF)[nH]c1 C1(NC(C(CC)OC)=O)CCSC12CN(C(c1cc(O)ncc1Br)=O)C2 c1(C(=O)NC(CNC(C=C(C)c2cnn(C)c2)=O)(C)CO)ccc(S(C)(=O)=O)s1 c1(CNC(c2scc3c2OCCO3)C)c(Br)sc2ccccc12 C(=O)(C1=CS(=O)CCC1)N1CC(C)C(CNC(C2(C)CNC(=O)C2)=O)C1 C1(C(C(C)CCO)=O)COC2(CCN(c3ncc4[nH]ccc4n3)CC2)C1 C1(C(=O)NCC(CC2CC2)CO)(CNC(=O)Cn2ccnn2)CCCC1 N1(C(c2c(SC)scc2)=O)CCOC(C)(CNC(C23CC(C)(CCO2)C3)=O)C1 CCC(C)(C)CC(=O)N1CCOCC(C(N2CC(CO)(OC)C2)=O)C1 CCCC(CNC(c1cc(C)nn1C)=O)C(=O)NC1CC12CC(OC)C2 C1(CC=C)(CNC(=O)Cc2cnoc2)CCCN1C(=O)C(O)CCN(C)C Cc1nc(C(=O)NCC2(F)CC(CNC(=O)Cc3cnn(C)c3)C2)c(C)s1 c1(C(N2CC(NC(C3N(C)CCC3)=O)C(F)C2)=O)cc2nnn(C)c2s1 CN1N=C(C(=O)N2CCC3CCN(C(c4ccc(=N)[nH]c4Cl)=O)C3C2)CCC1=O c1(OC(C2=NOC(C)C2)=O)cnc2ccc(Br)cc2c1 C(CC(=O)N1CC(O)CCO1)NC(=O)CCc1ccccn1 c1(CCC(N2CC(C(N)=O)(CNC(=O)CNC=O)C2)=O)cccc(Cl)c1Cl c1(C(N2C(CC)C=CCC2)=O)ccc(S(=O)(=O)N2CCCC(CC#N)C2)cc1 Cc1ncc(NC(C2C3CN(C(C4CC5CCC4O5)=O)CC23)=O)cc1F c1(OC)ncc(-c2sccc2C)cc1C(=O)Nc1sccc1CO C(CCC(C(=O)N(C)Cc1cocn1)NC(c1cc(CCO)on1)=O)OC C(=O)(C1=CCN(C(=O)C(F)C2CCOC2)CC1)N(C)CCn1cncn1 CC1CC2CC2CC1C(=O)NCC1CN(Cc2ccc(SC(F)(F)F)cc2)C1 S(=O)(=O)(c1ccc(Br)cc1)N1C(C)CC(=O)C1 c1(C(N2CC3C(NC(C4CCC(C#N)CC4)=O)(C3)C2)=O)ccn2cccc2c1 N1(CC(=O)N(C2CCN(C(COCC(=C)C)=O)C2)CC)CCN(C)C(=O)C1 C12(C(=O)NCc3c(C)noc3)C(NC(c3ncc(F)cc3C)=O)C3CC1C2C3 CCCC(CC)CC(=O)NCCCN(C(=O)C(c1cccnc1F)(C)C)CC C1(c2cn(CCN(C)C(c3sccc3Cl)=O)nn2)(COC)CCCCC1 c1(C(=O)NCC(C)NC(C=Cc2ccc(SC)s2)=O)ccc2nc(O)n(C)c2c1 c1(C(=O)NCC(C)N(C(=O)C(C)OCC(C)C)CC)cnsc1C C#Cc1cc(C(=O)NCC(C)CN(C(=O)C(C)NC=O)C)cc(F)c1 C(=O)(C(C)CC(=O)c1ccc(F)cc1)NCCN(C(C(C)(C)SC)=O)CC(C)O C1(C(=O)NCCC(C)NC(c2c(C(=O)OCC)c[nH]c2)=O)CCN(C)C1C c1(CC(=O)NC2(CNC(C(CC)O)=O)CCOCC2)cc(F)c(F)cc1F CC(C(=O)NCC(C1CC1)NC(C1CC(=O)C1)=O)S(C)(=O)=O C(=O)(CCCCCn1cnnn1)N1CC2C(CNC(Cc3cnn(C)n3)=O)C2C1 c1(C(N2CC(NC(C3CC3(C)C)=O)CC(OC)C2)=O)n[nH]c2c1CCOC2 C1(C(=O)NCC=CCNC(C2(OCC)CCCCC2)=O)CCn2ncnc2C1 c1(CC)ccccc1CC(=O)NCC1CN(C(C2CC2CC(C)C)=O)CC1O c1(C(=O)NC(C)CCN(C)C(C2CC23CCC3)=O)cncc(S(C)(=O)=O)c1 Cc1cc(C(=O)NC2CCC(C)(N3CCOCC3)CC2)nnc1O c1(C(N(CCCNC(c2nccc(OC)c2F)=O)C)=O)nc2n(c1Cl)CCCC2 C1(CNC(C2CCOC2c2ccccc2)=O)CN(C(C2CC3CC2C3)=O)CCO1 N1(C(CC=CC=C)=O)CCCC(C)(C)C1CNC(C1CCC(C)(C)OC1)=O Cc1nsc(N2CCCOC(c3ccccc3)C2)c1C#N C(=O)(C(C)(C)CCCO)NCC(C)(C1CC1)NC(C1CN(C)C(=O)CC1)=O Cc1ccc(Cl)c(F)c1C(=O)NC1CC(C(=O)O)C2CC12 N1(C(=O)CNC2CCCC(Cl)C2)CCCC(F)(c2ccccc2)C1 c1(C(N2CC(N(C(c3nc(COCC)sc3)=O)C)C2)=O)cc(C(N)=O)cn1C c1(C(=O)NCCC2CN(C(CN(C)C)=O)C2)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1 c1(C(=O)NCC(CNC(C(C)OCCOC)=O)O)sc2ncccc2c1Cl Cc1nc(O)c2cc(C(=O)NCC3CC3NC(C3CC4CCC3O4)=O)ccc2n1 C(C(CC(F)(F)F)NC(C1CCC(NC)CC1)=O)NC(Cc1ccn(CC)n1)=O N1(C(c2c(F)ncc(OC)c2)=O)CC2CCC1CC2NC(C1(Br)CC1)=O c1(C(N(C2CCN(C(=O)Cn3nccn3)CC2)C)=O)cc(C(F)(F)F)cc(O)c1 CCCCCC(O)CC(=O)N(CCC(C(C)C)NC(c1ccc(N)c(F)n1)=O)C n1(CCN(CC)CC)nc(C)c2c1CC(NC(c1onc(CC)c1C#N)=O)CC2 CCCCC(CC)CC(=O)N(CCC(=O)NCC(C)(COC)CO)CCO Cc1ccc(C(N2CCCC(C(=O)NC3CN(C)CCC3O)C2)=O)cc1O C(=O)(C(F)CC(C)(C)NC(=O)C(CC(C)(C)C)OC)Nc1cn(CCC)nc1 C1(CCNC(C(C)c2ccsc2)=O)CN(C(c2cn(C)cn2)=O)CC1C C(CCCCCCC(=O)NC(CNC(C1CCC(C)(C)O1)=O)C(C)(C)C)SC C1(NC(CN(CC#C)C(c2ccc(SCCCO)cc2)=O)=O)CCCCC1O c1(-c2cn(C)nc2)ccncc1COC(C1NC(=O)C2CC12)=O C1(NC(c2c(C)nc(N(C)C)s2)=O)CN(C(=O)C(C)(C)CF)C2(CCOCC2)C1 C1(NC(c2ccc(F)cc2Cl)=O)CC(C2CCN(C(=O)C3=C(Cl)CCCC3)C2)C1 CCCC(CC(=O)NC(C)COCC)NC(=O)CC1CCC(=O)NC1 CCCC(CCCNC(c1ccc(CN(C)C)o1)=O)N=c1nc(C)[nH]s1 C(=O)(C1CCc2c[nH]nc21)NCC(CCOC)NC(c1ccc(F)c(C)c1)=O N1(C(=O)CCc2ccncc2)CCC(F)(C(N2CC(c3ncccn3)C2)=O)C1 CC(CS(C)=O)C(=O)NCCC1(NC(c2cccc(N3CCNC3=O)c2)=O)CC1 c1(CC(=O)N(C(CN2CCCC(CC3CC3)C2)=O)C)cn2ccccc2n1 c1(C(=O)NCC2CCC(NC(c3c(C)ncs3)=O)C2)nc(O)c(C)s1 N1(C(CNC(CCCCC)=O)=O)CCC(NC(c2ccoc2)=O)C2(CCC2)C1 C1(C#N)(C(N(CCN(C(=O)CCOC2CCC2)C(C)C)C)=O)CCCOC1 C(=O)(C1CCc2nccn21)N1C(CNC(C(CC)CCOC)=O)COC(C)(C)C1 n1(CC(C)N(C2CCCNC2)C2CC2)cc(Cl)cn1 Cn1[nH]c(C(=O)NC2(CN(C(=O)CC3CC(CF)C3)C)CC2)nc1=O N1(C(c2c(C)nc(O)cc2)=O)CCC2(NC(=O)Cc3ccco3)CCCC12 C12(CCSC1)C(=O)N2.C(CC(=O)NC1CC1)N(C(=O)CC1OCCO1)C C1(NC(=O)COCCOCCNC(=O)C(O)c2ccsc2)CCC2(CC2)C1 CC1(C)C=C(C(=O)NC(C)(C)C=CC(=O)NCCC2CCC(C)(C)O2)C1 N1(C(c2c(OC)csc2)=O)CCC(O)C(C(N2CCCCC2C)=O)C1 c1(CC(=O)NC(CNC(C(C=C=C)C)=O)(C)CO)ccc2[nH]ccc2c1 c1(C(N(CC(C)NC(C2CN(CCOC)C(=O)C2)=O)C)=O)sc(C#N)cc1Cl C1(C)(C(N2C(C)CC2CO)=O)CCN(C(=O)C(F)C2CCCC2)CC1 C1(NC(c2c(C)onc2-c2ccccc2Cl)=O)CCN(C(=O)C(C)C)CC1F N1(C(C(F)=CCC)=O)Cc2ccccc2CC1CNC(=O)CC1CNC(=O)C1 C(=O)(C(C)S(N)(=O)=O)NCc1occ(C(N2C(CSC)CCC2)=O)c1 n1(CC(=O)NCC(c2ccccc2)N(C(C=CCCC)=O)C)c(C)ccc1C c1(COC)ccc(C(=O)N(C2CCN(C(=O)CO)CC2)C)cc1OC C(=O)(C1=CCCSC1)NC(C(C)O)C(=O)N(C1(CCO)CC1)C C=CC(C)CC(=O)NCC(C1CCCCC1)NC(c1cc(C(C)(F)F)on1)=O C1(CN(C(C2CCCC2F)=O)CC)CCCCN1C(=O)CCSCC(N)=O C(=O)(C1=CCCC1C)NCC(C)NC(c1cn(C)nc1C1CCOCC1)=O CC(F)(F)CC(=O)NC1CCC(CNC(c2ccc(NC=O)cc2)=O)CC1 S(=O)(=O)(c1cccc(S(=O)(=O)NC(C)(C)C)c1)NCC(=C)CC c1(C(N(C)CC2N(C(COCCC)=O)CCC2)=O)cc(O)cc(=O)o1 N1(CCNC(=O)CC2CCC(O)C2)CCN(C(C2CCS2(=O)=O)=O)CC1 c1(CNC(C2CC(OC)CN(C(CCOCC#C)=O)C2)=O)ccc2ncsc2c1 c1(C(N2CCN3CCOCC3C2)=O)cc(F)ccc1[N+](=O)[O-] c1(C(N2CC(F)CC(C(=O)NC(C)(C)CO)C2)=O)cc(F)c2cc[nH]c2c1 C1(C(=O)NCC(CC(=O)N2CC(COC(C)=O)C2)O)C2CC(=O)CC12 N1(C(c2nc(C(C)OC)oc2)=O)CCCC(O)(CCNC(c2cnns2)=O)C1 N1(C(C(C)CO)=O)CCN(C(c2cn(C3CCCCC3)nn2)=O)CC1CO N1(C(C=CC)=O)CC2CCC1CC2NC(=O)CC(C)(C)O N1(C(c2nc(CCC)oc2)=O)CC(NC(C2CCC=CO2)=O)CC2(CC2)C1 c1(C(=O)NCCCC(C)NC(C2CC3C=CC2C3)=O)cnn2cc(C#N)cnc12 N1(C(c2cn(C)nc2)=O)CC(CNC(=O)Cc2cccc(OCC#N)n2)C(O)C1 C1(C(N(CC(C)C#N)C)=O)CC2CC1CC2NC(=O)CCC(N)=O n1(CC(=O)NCC2C(CNC(c3c(N)cn(C)n3)=O)C2)cc([N+](=O)[O-])cn1 C=CC(CC)C(=O)N(C)CCC1CCN(C(C2CC(N(C)CC)C2)=O)CC1 C1(C(=O)NCC(C(=O)NC2C=CCC2)N(C)C)(OC)CCOC1 c1(C(N2CCCC(CNC(C(C)c3ncco3)=O)C2)=O)cc(Cl)cc(Cl)c1 c1(C(=O)NCC(CN(C)C(c2ccnn2C2CCOCC2)=O)O)cccc(Br)c1 N1(C(C(CC=C)C)=O)CCCN(C(=O)CCOCC(F)(F)C(F)(F)F)CC1C N1(C(=O)Cc2ccno2)CCN(C(c2cc([N+](=O)[O-])n[nH]2)=O)C2(CCC2)C1 N1(C(C2(CC=C)CCOC2)=O)CCCC2(CCCN2C(c2cnn(C)c2C)=O)C1 C(C(=O)NCC1(F)CCN(C(=O)Cc2c(C)cnn2C)C1)(C(C)C)NC(C)=O Cc1cccc(N(c2ccnc(N(C)C)c2Br)C(=O)CC(C)(C)C)c1C Cc1ccc(C(=O)NC2CC(C)CN(C(c3ccnc(C)c3C)=O)C2)cc1Cl C1(C(N(C2CCCOC2)CC)=O)COC(CNC(=O)CCCOC(C)=O)C1 C#Cc1c[nH]nc1C(=O)NCc1cncc(C(=O)NC)c1 C(=O)(CS(=O)(=O)C(C)C)NCC1C(CNC(C2(OC)CCCCC2)=O)C1 c1(C(=O)NC2COC3CN(C(CCOC(C)C)=O)CC32)cnc(O)c2cncn12 CC(C)C(C)CC(=O)NC(C1CN(C(=O)C(O)CN(C)C)C1)C n1(CC)nc(C)c(C(=O)N(CCCCCNC(c2n[nH]c(Cl)c2Cl)=O)C)c1C C(=O)(C(CC(F)(F)F)NC(=O)Nc1cccnc1OC)OCCCC C(=O)(CC(F)(F)F)NCCCCCN(C(=O)CSc1ccccc1Br)C n1(CCCn2c3ncnc(CC(=O)NCC(=C)Cl)c3nc2)c2ccccc2c(=O)c2ccccc12 C(CCN=c1ccnc(SC)[nH]1)NC(C(CC)F)=O c1(C(N2C3CC(NC(CCCC(C)=O)=O)(C3)C2)=O)cnc2c(F)cc(C)cc2c1 N1(C(C2CCN(C(C)=O)C2)=O)CC2CC2(CNC(c2csc(C)n2)=O)C1 C1(NC(c2n(C)nc(CC)c2Br)c2nnnn2C2CC2)CCS(=O)(=O)C(C)(C)C1 C1(C(=O)NCCN(C(c2c(C(=O)OC)c[nH]n2)=O)C2CC2)C(O)C(=O)N(C)C1C C12(C(N(C(C=C)C)C)=O)CC(NC(C3CCCSC3)=O)(C1)C2 c1(CC(=O)NCCN(C(=O)C2=NOCC2)CC)cc(C(F)(F)F)cc(Cl)n1 CCCCC(C)C(=O)NCc1csc(CCNC(=O)C=CCOCCOC)n1 N1(C(C2C(C)C2C)=O)CC2(CCC(CNC(c3cc(C4CCC4)no3)=O)O2)C1 c1(CCNC(C(C2CCC2)OC)=O)cnccc1C n1(CC(OCC)OCC)cc(C(=O)N(C)CCN(C)C(C2CC(C)CO2)=O)nn1 CCC(CNC(=O)C(C)CN(C(=O)CN(C)CC)C)CC(C)C C(=O)(C1CCCc2nc[nH]c21)NCc1nc(O)cc(CNC(C(C=CC)O)=O)n1 Cc1nc2ncnn2c(C)c1CC(=O)NC1CN(C(c2csc(O)n2)=O)CC1C c1(-c2c(C(N3CCC(NC(C4C(OC)C4)=O)C3)=O)c[nH]n2)ccc2c(c1)OCO2 C1(NC(c2ccnnc2)=O)CN(C(=O)Cc2ccc(Br)s2)CCC1CO C1(C(=O)O)(NC(c2cnc(-c3ncccn3)s2)=O)CCNCC1 c1(N(CC=CCl)C)cccnc1N(C)C(c1ccc(NCCO)cc1)=O C(c1ccc(F)cc1)=CCC(=O)NCCCCN(C(c1cc(SC)oc1)=O)C N1(C(C2(C)CC2)=O)CC2(CC(NC(c3cn(CC(N)=O)nn3)=O)c3nccn32)C1 C(=O)(C(F)CC(CC)CC)NCCOCC(N1CC(CCC)C(CO)C1)=O c1(C(N2CC(C)N(C(=O)CCC3CCCCO3)CC2)=O)nncc2c1CCCC2 C(C(O)CC(=O)NC1COCC1CO)NC(Cc1n(C)nnc1)=O N1(C(=O)NC(c2cnc(C3CC3)nc2)C)CCN2C(=O)COCC2C1 S(=O)(=O)(c1ccc(NC2CCN3CCCC23)c(Br)c1)NCCNC(=O)OCC C(=O)(C1=CCC(NC(C2CC(C3CC3)=NO2)=O)C1)NCCCSC c1(C(=O)NC(C2CCCC2)CNC(C(C(=O)OC)OC)=O)cc2sc(C)cc2s1 N1(CCCc2c(C)nccc2)CCC(=O)N(Cc2cccc(C(C)(F)F)c2)C1=O N1(c2ccnc(NCc3c(O)nc(=N)[nH]c3)n2)CCC2(CC1)CC2CO C(CC(=O)NOC1CCCCC1)N(CC=C)C(C1CCCN1CC)=O c1(CCC(N2CCOCC(NC(C(N)=O)=O)C2)=O)ccc2c(c1)OCCO2 C(=O)(CS(=O)(=O)CC(=O)N1CCC(O)(C(C)NC(c2ccoc2Cl)=O)C1)OC N1(C(c2ccncc2)=O)CCC(C(N2CC(F)(C3CC3)C2)=O)C(O)C1 C(=O)(C1=CCSC1)N1C(CCNC(C(C)OCCC(C)C)=O)CCC1 c1(C(C)C)cnn(C)c1C(=O)N(CC(O)CN(C(=O)C(C)(C)CO)C)C C1(NC(C=CCCC)=O)CCN(C(=O)C(F)n2ccnc2)CC1C(N)=O c1(C(C)CC(=O)N(CCNC(C2COC2)=O)C2CC2)ccccc1Br C1(C(=O)OC)CCC(NC(=O)OC(C)(C)C)CN1C(=O)NCc1cn(C)nc1I N1(C(CCc2c(C)cccc2)=O)CCC2(CC2NC(C2CCCC(=O)N2C)=O)C1 S(=O)(=O)(CC#Cc1ccccc1)NC(CCC1CC(C)OC1=O)=O C1(NC(C2(CC)CC2(F)F)=O)CCC2CN(C(c3ccc(O)c(F)c3)=O)CC2C1 C1(C(NC[Si](C)(C)C)=O)CC2CC2N1C(=O)C=Cc1ccsc1 N1(C(C2OCCC(C)C2)=O)CCC2(CCCN(C(C3C=CC=CC=C3)=O)C2)C1 CCN=C1NCCOCCN1.C(CCC)ON.OC n1(CC(=O)NC2CC(NC(Cc3cc(C)nn3C)=O)C(O)C2)nc(O)ccc1=O Cc1ccc(C)c(NCC(C2CCC2=O)C)n1 C1(SCC(=O)NCC(CN(C)C(C2(c3ccsn3)CC2)=O)O)CCCCO1 CN1CC2CCN(C(C3CCN(C(c4nonc4N)=O)CC3(C)C)=O)CC2C1 c1(C(N2CC(NC(C3(C#N)CC4CC4C3)=O)C2)=O)cc2c([nH]1)CCCC2 CC(C)C(C)C(C)CC(=O)NCCOCCN(C)C(C1CCCCC(F)(F)C1)=O c1(COC)ccoc1C(=O)NC(C)C(C)NC(c1ncccn1)=O n1(CC)ncn(NC(=O)c2cc(CNC(=O)C(C)(O)C3CCC3)[nH]n2)c1=O Cc1cc(C(N2CCC(NC(c3cc(CO)c(C)o3)=O)C2)=O)c(C)s1 C(=O)(C1=CCCOC1)N1CC(C)C(CNC(=O)CCc2ncc[nH]2)C1 N1(C(CN(CCOC)C)=O)CCN(C)CC1CNC(=O)CCc1nncs1 CCC(CC)(CC)C(c1ccccc1)N(S(=O)(=O)CC(C)OC)C C1(NC(Cn2ncc(C)c2)=O)CCN(C(=O)CS(=O)(=O)NC(C)(C)C)C1C N1(C(C2C(C)(Br)C2)=O)CCC2(CC1)CC(NC(c1ccnc(O)c1)=O)C2 N1(C(C(C)NC(=O)C(C)(C)C)=O)CCCC(NC(c2cnc(C#N)s2)=O)CC1 Cc1oc(Cl)nc1C(=O)N(C1CCN(C(=O)CC2CCOC2C)CC1)CCO Cc1cc(C#N)cnc1N1CCC(C)C(NC(C2CC(n3ccnc3)C2)=O)C1 C1(OC)CC(CCNC(=O)Cc2nc[nH]n2)N(C(=O)CC2CCC(=O)N2)C1 C(C)(CNC(=O)C(O)Cn1cncn1)(CC(C)C)NC(c1nc(C)n(C)c1)=O C12(C(N(CCC(=O)N(C)CC3(C#N)CC3)CCO)=O)CCC(CC1F)C2 C1(C(=O)NC(C)COC(F)F)(NC(=O)C(c2cncnc2)C)CCCC1C C1(C(=O)NCC2CN(C(=O)CC(O)C3CCCC3)C2)C2CC3C(C2=O)C13 c1(C(N2CCN(C(CCC(C)C#N)=O)C(CO)C2)=O)ccc2sncc2c1 C1(CC(=O)NC2CC(C)(CNC(c3cnc(C)[nH]3)=O)C2)CCCCC1O c1(C(=O)NC(CC)CNC(=O)COC(F)(F)C(F)(F)F)c(C)[nH]cc([N+](=O)[O-])c1=O C1(CC(=O)NCC2CCC(NC(=O)Cc3ccno3)CC2)CN2CCN1CC2 C(=O)(CC(=O)NCC(C1CC1)NC(=O)Cc1cncn1C)OC N1(C(C2C(=C)CC2)=O)CCC2(CCCN(C(=O)CCc3cnc(OC)s3)C2)C1 Cc1ncnc(C(=O)NCCC(C)N(C)C(C2CC(=O)NC2(C)C)=O)c1C C(CC(C)(C)C)N(C(C(C)N(C(C1CCCOC1)=O)C1CC1)=O)CCO CC(C)CC(C(=O)NCc1cccs1)ONC(=O)C(C)(O)C1CCCC1 C1(N(C(C2(CNC(C(CC)C)=O)CC(F)C2)=O)C)CCOCC1C C(=O)(N=c1cc(C)n(C)[nH]1)C1N(C(C2CC2C(C)(C)C)=O)CCC(=C)C1 N1(C(C(CCSC)NC(C2CC(F)(F)C2)=O)=O)CCn2nc(C)cc2C1 N1(C(c2nc(C)oc2C)=O)CCCC(C2CCN(C(=O)C(C)(C)CO)CC2)C1 CC(C)C(C)C(=O)N(CCCOCCN(C(=O)CC1CCCSC1)C)C c1(OCCN(C)C)cncc(C(=O)NC(C)(C)C(O)c2ccccc2)c1 c1(NCC2(CNC(c3cc(C)c(C)s3)=O)CC23CCC3)ncnc2cnn(C)c12 C1(NC(c2cnn(CCF)c2)=O)CN(C(c2cccc(F)c2)=O)CC12CC2 C(=O)(N=c1ccn(-c2ccccc2)[nH]1)c1cc(NC2C(COCC)C2)c(Br)cc1 C(=O)(C1CCc2cc(Cl)ccc21)NC(C)CNC(=O)CSCCC#N C1(CC(=O)NC(CC)CNC(c2cnc(O)o2)=O)CC2(CCO1)CC2 c1(C(N(CC(=O)NCCN2CCCC2=O)C)=O)cc2cccnn2c1 c1(OC)ccc2c(c1)N(C(=O)C(C1CCOCC1)O)CC2C C1(NC(CCCC#CC)=O)CN(C(=O)CC(=O)N(C)C)C2(CCC2)C1 Cc1ccc(C(=O)NCCNC(N2CCCC(Cc3ccc(O)cc3)C2)=O)cc1 C1(C(C(=O)NCCC)N(C2CCC2)C2CC2)CCC2COCCC2C1 c1(C(N2CC(CCC=C)(C(=O)NC(CC)C(C)(F)F)C2)=O)c[nH]c2cnccc12 N1(C(C2CC3(CCC3O)C2)=O)CCC2CN(C(=O)CC3CCCC3)C2C1 C(=O)(C(CC)CCOC)N1C(CCNC(C(CC)CC)=O)CCC1 C1(C(=O)NC2C(C#C)CCC2)CC2CC1CC2NC(c1ccn(CC)n1)=O C1(CNC(=O)C=CC2CCCO2)COCCN(C(c2ccc(Cl)nc2)=O)C1 C1(NC(C2C3(CN(C(=O)OC(C)(C)C)C3)C2)=O)CCC2(CC1)CC2C#N C=CCCCCCC(=O)N(C1CCN(C(=O)C=C2CCSCC2)CC1)CC(C)C C(=O)(C1CCOc2c(F)cccc21)N1CCCCC(NC(C(=O)NC2CC2)=O)C1 N1(C(C2CC(C)(CC)C2)=O)CC2CCCC(N(C(=O)CC(C)C(F)F)C)C2C1 N1(C(C2N(C)CCCC2)=O)CCC2(CC(NC(=O)C=CCF)C2)C1 C1(C(=O)NCC(C)(F)F)CC(NC(c2ccc[nH]2)=O)C12CCC2 C1(CNC(C(CC)(C)CC)=O)CCN(C(=O)Cc2nncn2C)CC1(F)F C1(C(=O)NC2C(NC(c3ccn(C)c3)=O)COC2)CCOC1(C)C c1(OC)cc(C(=O)N(C2CCCN(C(=O)CN(S(C)(=O)=O)C)C2)C)nn1C C12(C(=O)NC3C4CC(NC(CC(C)SC)=O)CC43)CC1COC21CCC1 c1(C(N2C(Cn3cc(-c4c(C)cccc4)nn3)CCC2)=O)coc2ccccc12 c1(COC)cc[nH]c1C(=O)NCCn1cc(C(=O)NC2(C3CCCCO3)CC2)nn1 C(=O)(C(O)CCCNC(c1c(OC)noc1C)=O)N(CC(CC)OC)C N1(CC)OCC(NC(C2CCC2NC(c2ccnc(O)c2)=O)=O)C1=O N1(C(CNC=O)=O)CCCCC1C1CCCN1C(C1CCC(=C(F)F)CC1)=O CCS(=O)(=O)c1cccc(C(=O)NCC2(Cn3cc(C(O)C4CC4)nn3)CC2)c1 C(CC(C(=O)NCCn1ncnn1)NC(=O)C(c1cnn(C)c1)=O)=CC CC1(C)CC1(C(=O)O)NC(c1ccoc1CN)=O c1(NC(c2ccncn2)C)ccnc2ccnn12 N1(C(CN(C)CC)=O)CC2CCCC(C1)N2C(=O)C1=NOC(C(C)(C)C)C1 c1(C(=O)NCC(CNC(c2ncccn2)=O)F)c(Cl)sc2nnsc12 C1(C2CCC2)(C(=O)NCC2(C)CCCN(C(C(C3CCC3)OC)=O)C2)CC1(F)F C1(CCC)CC(C(N2CCC(OCCNC(=O)COC(C)CC)CC2)=O)CCO1 c1(C(C)C)conc1CC(=O)NC(CNC(=O)CCc1ncnn1C)C1CCC1 c1(C(N2C3C(NC(c4ccn(C(C)C)n4)=O)CC(C3)C2)=O)cnn2c1NCCC2 [N-]=[N+]=NC1(C(=O)NC(c2ccc(Br)cc2)CO)COC1 c1(-c2nc(C3OCC(C)C3)on2)ccc(-n2cccn2)cc1 CCCCC(CC)C(=O)NCC1(NC(=O)C(C(C)(C)C)C2CCCC2)CCCC1 C1(CN(C(c2nocc2C(C)(C)C)=O)CC)CCN(C(=O)C(C)CC2CC2)CC1 N1(C(=O)C2CC2)CCCC1C(=O)NCC12CCCC1C2.C12(CCCC1)C(=O)NC2 C1(n2cc(-c3c(C)cnn3C)nn2)CC(C2CC2)=NO1 c1(OC)ccc(C(=O)NCCNC(C2CCN(C)C(=O)C2)=O)c(Cl)c1 c1(CC(=O)NC(C2CCCC2)CNC(C(C)=CC)=O)cc(F)ncc1Br N1(C(C(CCC)O)=O)CC(C2CCCCN(C(=O)CC3CCC(=O)N3CC)C2)C1 C(C(=O)N=c1[nH][nH]c2ccnc(O)c12)(c1ccc(F)cc1)N(C)C C1(NC(C(C)NC(c2cccs2)=O)=O)CCC(NC(=O)C(C)(F)F)C1 c1(C(N2CC(N(C(COC(C)=O)=O)C)C(C)(C)C2)=O)c(Cl)nc2cc(Cl)ccn12 N1(C(CNC(CCC)=O)=O)CC2CCC(C1)N2C(=O)CN1CCC1C N1(C(C2(C)CN(C(C3CCN(C)C(=O)C3)=O)C2)=O)CCOCC12COCCN(C)C2 CC(C)CC(C)C(=O)N1CCCC(C)(CNC(c2cc(CO)ccc2Cl)=O)C1 CCC(CC(=O)N1CCC2C(NC(c3cccc(OC)n3)=O)C12)SC C1(C)(CNC(C2CC(NC(C3C(COC)CC3)=O)C2)=O)CCCO1 C1(C(=O)NCC2CN(C(=O)Cc3ccccc3)CC2(F)F)(OC)CCCCCC1 c1(C(=O)NC(CNC(c2c(C)cc(CC)o2)=O)C)sccc1S(C)(=O)=O c1(C(N2CCN(C(C(CCC)NC(C)=O)=O)C(CO)C2)=O)cnn2ccn(C)c12 Cc1cnc(NCC(C)N(C(=O)CC2C(C)(C)C2(C)C)C)nc1S(C)(=O)=O C(=O)(C(C)(C)C(C)O)N1CC(OC)C(NC(=O)Cc2ncccc2C)C1 c1(CC(=O)N(CCC(=O)NCCSCCO)CC=C)ccncc1C C1(NC(=O)NC2C(CCC(=O)OC)CCC2)CC(=O)N(c2ccccc2OC)C1 CC1CNc2c(C(=O)NCCc3nc(-c4ccccc4)ns3)cnn2C1 N1(C(C=CC=CC)=O)CC2(CC(C(=O)NCCSC)CO2)C1 n1(CCC)cc(C(=O)N(CCN(C)C(c2cc(CC)cs2)=O)C(C)C)cn1 N1(CCC)CCC(C(=O)NC23CC2CN(C(=O)C=CC(C)(C)SC)C3)CC1 N1(C(CC2(CN(C)NC(=O)CN)CC2)=O)CCCC(CC2(CC)CC2(F)F)C1 c1(C(=O)NCc2c(F)cc(C)c(F)c2)c(F)cncc1C1=CCN(C)CC1 C1(CC(=O)N(C(CN(C(c2ncn(CC)c2)=O)C)C)C)CC(C)(C)CCO1 C=C=C(C)CC(=O)N1CCC(F)(CNC(=O)CCn2cncn2)C1 N1(C(c2cc(CCCC)no2)=O)CCCCC1Cc1cn(CCCC(=O)O)nn1 N1(C(CCCCC#N)=O)CCC2(CC1)CC2(CO)CNC(=O)C=C1CCCCC1 CCC(CCC(=O)N1CCN(C(C2CC(F)(CSC)C2)=O)C(C2CCC2)C1)OC C1(CNC(Cc2c(C)n(C)cn2)=O)CN(C(c2csc(O)n2)=O)C(C)(C)C1 c1(C(N2CC(CC(=O)NC(C(=O)NC(C)C)C)OCC2)=O)ncc(F)cc1F C(=O)(CC1=CCCCC1)N1CCCCC(CCC(=O)NC2(C)C(C)CCCC2)C1 C1(C(=O)NC(CCC)C(F)(F)F)C(C2CC2)CCN1C(=O)CN1CCNC(=O)C1 C1(C(N(C)CCNC(=O)OC(C)(C)C)=O)(Cc2nccs2)CCc2ccccc2O1 c12c(ccnc1OC)NC2=O.C(C(C)C(=O)N(CCOC)CC)OCC c1(CNCc2ccc(CC)cc2)cccc(S(=O)(=O)N(C)CCO)c1 N1(C(C(Cc2ccccc2)OC)=O)CCCC(CNC(c2cc(CF)on2)=O)C1 C1(CC(=O)NCC(C(=O)OCC)(C)C)CN(C(=O)C(C(C)C)OC)CC12CC2 C12(NC(CC3(C(=O)OCC)CCC3)=O)CC(NC(c3cnccn3)=O)(C1)C2 N1(C(CCNC(N)=O)=O)CCC(CN2CCN(C(C3CC3C(N)=O)=O)CC2)CC1 C(=O)(C(O)CC(C)(C)C)N(CCCCCC(=O)NCc1nc(=O)o[nH]1)C Cc1cc(C(=O)NC(C2CN(C(c3cc(C)[nH]c3C)=O)C2)C)n(C)n1 CCC(C(=O)NCC(F)CNC(=O)C=CSC)OC1CCCC1 CCCC(CNC(C1(COC(C)C)CC1)=O)C(=O)NC1CCOC(C)C1 N1(C(C2C(C(C)C)CCC2)=O)CC(C2CC2)(C(=O)N(C)CC2(F)CCC2)C1 C1(NC(CSC)=O)CCC2(CCCN2C(=O)C(C(C)C)c2ccc(Cl)cc2)CC1 CC(COCc1ccco1)N=c1ccnc(NC2CCCC(C)(C)C2)[nH]1 C#Cc1cccc(C(N2CCCCC2)C(=O)NCC(F)F)c1 CCC(C(=O)N1CCC(CNC(c2sc(C3CCCC3)nc2C)=O)C1)C(C)C C1(NC(=O)CCSC(F)(F)F)COCCN(C(=O)CC2CC3CC3C2)C1 N1(C(C(c2ccc(Cl)cc2)C)=O)CCC(C)C(NC(=O)Cc2ccc(F)cn2)C1 C=CC(C)CCNC(c1occc1CNC(=O)C(c1cnn(C)c1)O)=O N1(C(CN2CC(C)(C)C2)=O)CC2(CCC(CNC(C3CC=CCO3)=O)O2)C1 c1(NC(c2ccc(Cl)c(C#N)c2)c2n(C(C)(C)C)nnn2)ccc2nncn2c1 N1(C(CC(C=C)C)=O)C2CCC1(CNC(=O)C(C)CCCOC)CC2 c1(CC(=O)NCC2CC(F)(CNC(=O)C(O)C(F)F)C2)cc(F)ccc1Cl C1(NC(c2c(C)nn[nH]2)=O)CC(NC(=O)COCCC(C)C)C1(C)C CN=c1ccc(C(N2CCCC(C(C)NC(=O)COC(C)C)C2)=O)c[nH]1 C12(NC(CC3CCN(OC)CC3)=O)CCC(CNC(C3(Cl)CC3)=O)(CC1)OC2 C1(CC(=O)N(CCC(=O)N(C(C(=O)NC)C)C)C)CCCCN1C c1(C(N(CCCCN(C(C2N(CC)CC2)=O)C)C)=O)ccc(S(=O)CC#N)cc1 C(=O)(C1=NNC(=O)CC1)NCC1(CNC(c2cccc(NC)n2)=O)CC12CCC2 c1(CN(C(C(CC)C)=O)C)cccc(CNC(C2(CC)CC2(F)F)=O)c1 CC(C)C(C(=O)N1CC2C(CNC(C3C4COCC34)=O)C2C1)c1cccc(Cl)c1 c1(C(=O)NC2C(C)CN(C(=O)CC3CCCCO3)C2)cc(C#N)c2n1CCCC2 C=CC1CCCN(C(=O)NC2CC2C(=O)Nc2cnccc2C(=O)OC(C)(C)C)C1 N1(C(c2ccc(CNC(C3CCC(C)(CC)O3)=O)s2)=O)CC2(CCCC2)C1 n1(CCC(=O)OC)cc(CC2(O)CN(C(C3(CCS(N)(=O)=O)CCC3)=O)C2)nn1 N1(C(C2CCC(C)(CC)O2)=O)CC(C)N(C(=O)CCc2cccc(C)n2)C(C)C1 n1(CC)nc(C(=O)OC(C)C(=O)Nc2ccc(CC#N)cc2)c2c1CCOC2 C(=O)(CC(C)(C)C#N)N1CC(=C(CNC(C(C)Sc2ncccn2)=O)F)C1 c1(CC)cc(Cl)ccc1C(=O)NCc1ccnc(C(=O)O)c1 C(=O)(CS(C)(=O)=O)NC(C(=O)N1CC(CC(=O)OC)C1)COC C1(C(=O)NCCC2(CNC(C(CC)(C)C)=O)CC2)Cc2cccnc2C1 Cc1nc2c(s1)CCCC2C(=O)NCC1CN(C(C2(C)CCCO2)=O)CCCO1 CCCC(C)C(=O)NCCOCCOCCNC(=O)CC1CCC(O)C1 C1(C)(CNC(c2cn(CCC)nn2)=O)CCN(C(=O)CC(=O)NC)CC1 c1(CN(C(c2ccc(C(F)F)o2)C(=O)NCc2ccc(Cl)s2)CC)ccccc1 C(C)(C)(CC(=O)NCC1CCN1C1CC1)n1cc(CN(C(C)C)C)nn1 C1(CC)CCN(C(=O)CSC(C)(C)C)C1NC(=O)COC C1(N(C(Cc2ncc(C)s2)=O)C)CN(C(c2ccnc(C(C)(C)C)c2)=O)CC1O C1(CC)CC(O)CN1C(=O)C=CCOC.C1(=O)C(C)N1C C(=O)(C1=CCN(C)C1)NCCC(C)NC(c1cnc(CC)o1)=O CC1=C(C(=O)N2CCCC(NC(c3ccc(CO)cc3)=O)C(F)C2)CCCO1 CC1CN(C(c2nncn2C2CC2)=O)CC1CNC(=O)C(F)=CC1CC1 Cc1nn(C2CC2)cc1C(N1CCC(CNC(C2(C(F)(F)F)CCCC2)=O)C1)=O N1(C(C(COCC)NC(C2CC2(C)C)=O)=O)CCC2C(=O)NCC2C1 N(C1CCCc2cn(CC(F)(F)F)nc21)C(c1c(C)cc(F)c(F)c1)=O N1(C(C2C3CN(C)CC32)=O)CCC(NC(=O)Cc2cnc[nH]2)C(F)C1 N1(CC(=O)O)CCN(C(=O)C=CC2CC2)CC1.c12nc(no1)C2 C1(C(C(=O)NCC(C)N(C)C(C2CC2(Cl)Cl)=O)C2CC2)CCCCC1 C=CCC(CC(C)C)C(=O)N1CCCC(CC=C)(NC(=O)CC2CCC2)C1 n1(C(CC)CC)nc(C)cc1C(N1CCCC1CNC(=O)CN1CCCC1C)=O c1(OC)noc(C2CC2)c1C(N1CCC(N(C(=O)CCC2CCCO2)C)CC1)=O c1(CC(N2C(CCNC(CCC3C(C)C3)=O)CCC2)=O)ccc2c(c1)CCCC2 c1(C(CNC(c2n[nH]cc2Br)=O)NC(CC=C=C)=O)ccccc1F N1(C(C2COC(=O)O2)=O)CCCC2(C1)CN(C(c1cc(Cl)nc(Cl)c1)=O)CCO2 C(=O)(C1CC=Cc2ccccc21)NCC(CNC(C1(F)CCCCC1)=O)O c1(C(=O)NCC2(CC(=O)NC3(c4nccs4)CC3)CC2)cccn2ccnc12 c1(CC)oc(C(N2CC=CC(NC(=O)C=C(Br)Br)C2)=O)cc1C C12(CCCCC1)CC(=O)OC2.C1(C(=O)OC)(C(=O)N(C)C)CNC1 C1(NC(c2c(CNC(C(CC)n3ccnc3)=O)ocn2)=O)(COC)CCOCC1 CC(CC(=O)NC1(CF)CCN(C(=O)CN2CCCCC2=O)C1)C(F)(F)F c1(CC)ccsc1C(=O)NC(C)CN(C(=O)CCc1ncco1)CC C1(CCNC(C2C=CCCC2)=O)CN(C(c2sccc2Cl)=O)CCO1 c1(C(C(N2C(C)(Cc3cccc(Br)c3)CCC2)=O)O)ccc(F)c(F)c1 CC(O)CC(C)N=c1cc(NCc2ccc(CO)c(F)c2)nc(C(F)(F)F)[nH]1 N1(C(C2OCCN(C(c3cc(OC)c(Cl)nc3)=O)C2)=O)Cc2ccc(F)cc2C1 N1(C(C(C2CC2)OCC)=O)CCOC2(C1)CN(C(C1CC1C(C)(F)F)=O)C2.C1(C)CC1 N1(C(c2c(C)cc[nH]2)=O)CCCC(NC(C23CC(C2)C(C)(C)O3)=O)CC1 C12(NC(C3CC(OC(C)C)C3)=O)CCC(CC1)N(C(=O)CC1(O)CCCOC1)C2 O=C(CC1NC(=O)c2ccccc21)NCC1(NC(C2CCC3C2C3(F)F)=O)CC1 C1(C(=O)NCCC(=O)OC)CCN(C(C2CC(SC)C2)=O)CC1 C#CCC(CC(F)(F)F)C(=O)N1CCC(C(=O)OC)(CO)C1 CC1(C)CC(CNC(c2cncc(F)c2Cl)=O)CN(C(=O)CCCS(N)(=O)=O)C1 Cc1cc(C(=O)N(C(C)CNC(c2ccn(C)c2C)=O)C)cc(S(N)(=O)=O)c1C c1(C(=O)NC(C(C)NC(C(CC)N2CCCC2=O)=O)(C)C)cc(OC)n(C)n1 S(=O)(=O)(c1csc(C(=O)N(CC(C)NC(=O)Cn2ncnn2)C)c1)NC N1(C(C=CC)=O)CCc2c(CNC(=O)CCCN3C(=O)CNC3=O)cccc2C1 c1(OC)ccc(-c2ccnc(NCCNC(C3COCC3C)=O)n2)cc1 Cc1ccc2c(cnn2C)c1-c1cc(C(N2CC3C(CO)C3C2)=O)n[nH]1 CC1(C#N)CCC(N=c2cc[nH]cc2S(=O)(=O)NCC2CSCCS2)CC1 CC(C)CC(=O)N(CCCC1CCNCC1)CCO C1(c2n(C3C(F)(F)C3)ncc2)NC(=S)N(C2CC2)C2=C1C(=O)NC2c1ccccc1 Cc1cccnc1C=CCNc1cn(C)nc1C(F)(F)Cl C(=O)(C(Cc1ccccc1)C(C)C)NCC1CN(C(=O)C(C)(C)CF)CC1C c1(CC(=O)N(C2C3CN(C(CC4CN(C)C4)=O)CC32)C)c[nH]c2cc(F)ccc12 c1(C(=O)NCC2N(C(C3C(C(N)=O)C3)=O)CCCCC2)cc2cccnc2o1 N1(C(C(N)=O)=O)CC=CC(NC(C2(O)CCC2)=O)C1 c1(-c2cc(OC)cc(COC)c2)ccc2nnc(C(N3CCOCC3C)=O)n2c1 c1(C(N2CC(O)(C(C)NC(=O)C(C)n3cncn3)C2)=O)cc(CO)n(C)n1 C(CO)(CCCCNC(=O)C(F)=C1CCCC1)NC(=O)CCC1CCC(O)CC1 C(CC(C)C)(C(=O)N1CCC(F)C(F)C1)ONC(C1C(CC(C)C)C1)=O c1(C(C2CC2)NC(CN(CCOC)C(c2cnn(CC)c2)=O)=O)ccc(C)cc1 CC(C)CC(O)C(=O)NCCCC1(O)CCCN(C(=O)C(F)(F)CN(C)C)C1 C1(C(=O)NCC23CC(NC(c4cnc(C)s4)=O)(C2)C3)CCCN2CCCCC12 C(=O)(C(O)C1=CCCCC1)NC1(CNC(C(c2cncnc2)C)=O)CC1 C(=O)(CC(C(F)(F)F)NC(=O)C(c1ccccc1)F)N1CC(N(C)C)(C(N)=O)C1 c1(CC(=O)OCC2(COC)CCC2)cccc(F)c1Nc1ncccc1OCC c1(C(=O)NCC2CC(OC)CN2C(C2OCCC2C(C)C)=O)cc2occc2[nH]1 C1(C(=O)NCc2c(CC)nn[nH]2)CN(C(=O)C(C(C)C)n2cccc2)C(C)(C)C1 c1(C(=O)NCC(CC=C)NC(c2c(Cl)cnn2C)=O)ccccc1CC C(=O)(C#CC(C)(C)C)N1C(C(C)NC(=O)C(F)(F)Oc2cnn(C)c2)CCC1 CCCCCCC(C)C(=O)NC1CN(C(=O)C=Cc2cnc(C)s2)CC12CCC2 C1(NC(C(c2cccc(F)c2)(C)C)=O)CCC2CCN(C(=O)CCCF)C1C2 C(=O)(CC(C)(C)CCC)NC(C1(O)CCN(C(C2(CC=C)CCOC2)=O)CC1)C CC(C)CC(O)C(C)C(=O)N1CC2(CCC2OC(C)(C)C)C1 N1(C(c2c(SC)cccc2)=O)CC(CNC(=O)C(C#N)C(C)(C)C)C2(CCC2)C1 C1(C)(CC(N2C(COC)CC2)=O)CCN1C(c1cnnn1C)=O C1(NC(N(CCOc2ccc(OC)cc2)CCO)=O)CC2CC1CC2=O N1(C(CCC2N(C(c3c(C)cc[nH]3)=O)CCCC2)=O)CCOCC(O)C1 C1(C(=O)NCCC(C=C)C)CC(NC(C2(COCC)CCC2)=O)C(O)C1 Cc1cc(CN=c2[nH]c(C(=O)NCCCN3CCCC3)cs2)cc(Br)c1 CC1(C)CC(NC(c2c(F)cccc2Cl)=O)CN(C(=O)C(C)(O)C2CCC2)C1 Cc1cc(C(=O)C(c2cccc(C(F)(F)F)n2)C#N)c2ccc(F)cc2n1 N1(C(C(CCC(C)C)=O)=O)Cc2n[nH]cc2C1C(=O)NC1CCn2ncnc2C1 c1(N(C)C)nc(Cl)c(C(N2CCOCC2CNC(=O)CCc2cnc(O)[nH]2)=O)s1 C=CCC(C)(C)CC(=O)NCC(C)CN(C)C(C12COC(CF)(C1)C2)=O N1(C(C(=O)N(C)C)=O)CCCC(C(=O)N(c2ccncc2)CC(=O)NC(N)=O)C1 N1CCC(S(=O)(=O)F)CC1.c1(CNCC)cccc(C)c1 CC1CC(C(=O)NC2(CNC(c3cc(O)nn3C)=O)CCC2)CCN1C C1(CCNC(CSCC(C)C)=O)CCN(C(=O)C(C)(C)n2ccnn2)CC1(F)F c1(OC)ccccc1OCC(N1CCC(NC(c2scnc2Cl)=O)C1)=O C1(CCO)(SC)CN(C(=O)OCC2(O)CCC2)C1.C(Cc1ccccc1)(C(=O)O)N CC1(C)C=C(C(=O)NC2CCN(C(c3csnc3Br)=O)C2)C1 C=CC1CCCN(C(=O)C(CCSC)NC(=O)COCCOC)C1 C12(C(=O)NCC(CC)NC(C3CCC(=O)N(C)C3)=O)CCCN1CC(OC)C2 C1(CC)CN(C(c2cnc(Cl)c(C)c2)=O)CCN1C(c1cc(I)ccc1C)=O C1(C(=O)O)COCCN1C(C12CC1CN(C(=O)Cc1ncccc1F)C2)=O C1(CC)CCC(C(=O)N(C)CC2COCCN2C(C2CCOC2)=O)CC1 c1(C(N2CCC(C)(CNC(=O)C(F)C3CC3)C2)=O)cc2ccccc2s1 c1(CC(=O)NCC(C)N(C(c2c(CC)onc2)=O)CC)cn2cc(F)ccc2n1 CCCCC(O)C(C)C(=O)NC1CC(CC(N2CCC2(C)COC)=O)C1 c1(C(N2C(CNC(C(C)NC(=O)CC(C)(C)C)=O)CC2)=O)cnn2c1OCC2 C(c1c(Cl)cccc1Cl)=C(C)C(=O)N(CCCNC(=O)CCc1cn(C)nn1)C C1(C(=O)NCC2C(NC(c3cccc4c3COC4)=O)C2)CCc2ccccc2C1 c12ccc(F)c(c1)C(=O)Nc1cncc-2c1.c1(C(=O)OCC)n[nH]cc1C(C)C c1(CNc2ccc(C(C(F)F)F)cn2)cccc2ncnn12 N1(C(Cc2c(C)n[nH]c2C)=O)CC(NC(C2CC(C(F)(F)F)C2)=O)C(C)(C)C1 N1(C(C2C(C(=O)OCC)CC2)=O)C(C(N2CCC(O)(CC)C2)=O)CCC12CC2 c1(NC(C(c2cn(C)nc2)NC(=O)CCCCCO)=O)cccc(C#N)c1 c1(-n2cc(CCNC(c3c(C)nc(Br)s3)=O)nn2)cccc2ncccc12 c1(C(N(CCCN(C(C2C(C)C2)=O)C)C)=O)cn2c(n1)COCC2 N1(C(C(=O)NC)C)CCOCC(C(=O)N(c2ccc(C)cc2)C(C)C)C1 C1(C)(C(=O)NCCCCC(C)NC(C(C)CCO)=O)CCN(C)C1=O c1(C(C)(C)C)ncn(CCC(=O)NCCNC(=O)NC2COC(C(F)(F)F)C2)n1 c1(C(=O)NC2C3CC(CNC(CC(=C)C)=O)(C3)OC2)ccc2c(c1)CC(C)O2 C1(CNC(C(CC(=O)OC)C)=O)CC2CCC1N(C(=O)CC1COCCN1C)C2 Cc1[nH]c2ccccc2c1C(=O)NC1CCC(CNC(C2CCCC2(C)O)=O)C1 C1(CNC(C=CC=CC)=O)CN(C(c2cncc(NCC)c2)=O)CC2(CCC2)O1 c1(C(=O)NC2C(NC(C3CC(C)C3)=O)CCCC2)cc(C2CC2)nc2ccnn12 C1(C(N(C)CCc2nccs2)=O)CCCC(NC(=O)COC2(C)CCC2)CC1 c1(C(=O)NCC(CCC)CCC)c(Cn2cc(CC(C)O)nn2)nn2c1CCC2 c1(C(N2CCCC(CCNC(=O)C(O)C(F)F)CC2)=O)cc2ccc(F)cc2o1 C1(NC(C(C=C=C)C)=O)CN(C(c2cccnc2SC(F)F)=O)CC12CC2 c1(C(=O)NC(C)C(=O)NC2CCCC(NC(C3CC3CF)=O)C2)ccc(F)cc1 C1(CNC(C(F)=CCC)=O)CC(C)N(C(c2cncnc2C)=O)C1 C1(NC(=O)CCn2ccnn2)CC2(C1)CN(C(=O)C=Cc1cnccn1)C2 CN1CCC(NC(C2CCC(F)CC2)=O)C12CCCN(C(C1(C(N)=O)CC1)=O)C2 c1(C(N(CCOCCCNC(C(CC)(C)CO)=O)C)=O)n[nH]c2ccc(C)cc12 N1(C(C(C(C)C)F)=O)CCC2(CCCC2CNC(=O)C=C2CCCC2)CC1 C(=O)(CC(O)C(C)(C)C)N(CCCCNC(C1CCC(=O)N(C2CC2)C1)=O)C Cn1c(O)nc2c(C(=O)NC3CCC(P(C)(C)=O)C3)cccc12 Cc1nnc(NC2CCCCN(C(=O)C(C)CC3CCC3)C2)c(C#N)c1C c1(C(C(=O)NCCCF)N(C)Cc2cncs2)ccc(F)c2c1CCC2 C1(C(=O)NC(C)CCCNC(=O)COCC(C)(C)C)CC2(C1)NC(=O)NC2=O CCCCCCC(F)C(=O)NCCC1(C)CCN(C(=O)Cc2ccc(F)cc2)C1 C(c1cccc(O)c1)=CC(=O)NC1CC2(C1)CC2Nc1cc(O)ncn1 C1(CC(=O)NC(CCC)CO)CCCN(C(=O)CN2CCNC2=O)C1 O=C(CC1CC(C(F)(F)F)CO1)NNC(=O)N1CCC(c2cc[nH]n2)C1 O=C(CCC(F)(F)F)NCc1csc(C(=O)NCCCOCCCO)c1 Cc1cc(Br)cc(CN2CCC(N(C)C(c3cnc(O)c(Cl)c3)=O)C2)c1O C1(Nc2c(C)n(C3CC3)nc2)CC(CNC(=O)OC(C)(C)C)C12CCC2 C1(C(=O)NC2(CC=C)CN(C(=O)Cc3n[nH]c(=NC)s3)C2)CCN(C)C(=O)C1 C1(C(=O)NCC(CC)N2CCCC2)CCCCCN1C(=O)C(CC1CC1)OC c1(OCCCOC)ccc(C(N2CC(NC(C3(CO)CCC3)=O)C3CC23)=O)cn1 N1(C(C2C(C)(Br)C2)=O)CC2(C1)C(NC(=O)Cc1cccc(F)c1)CCS2(=O)=O N#Cc1cncc(NC(=O)CC2CN(C(=O)C(c3cccc(Br)c3)O)CCO2)n1 C1(CC=C)(NC(C2CC2(C)C(C)C)=O)CCN(C(=O)CSc2nncn2C)C1 c1(OC)nn(C)cc1NC(C1COCCN1C(=O)CCc1cnn[nH]1)=O C=CC1(C(=O)NC23CC4CC(CC2C4)C3)CCN(C(=O)C#CC2CC2)CC1 c1(C(N2CCC(C)(CO)CC2)C(=O)NCCC2CC2)nnc2n1CCNC2=O c1(CC(=O)NCC2CCN(C(CC(C)C3CC3)=O)C2)ccc(-n2cnnc2)cc1 c1(CC(=O)N(C2CCN(C(C3CCN3S(C)(=O)=O)=O)C2)C)cc(F)cc(Cl)c1 c1(C(N2CC(SC)C(NC(=O)CC3(C)CC(F)(F)C3)C2)=O)cc(C)c(C)nc1C c1(C(=O)NC2CC(C)N(C(c3ccn(O)c(=O)c3)=O)CC2)cnn2ncccc12 C1(C(=O)NC2(C)CN(C(C3(COC)CC=CCC3)=O)C2)CCC2(CCOCC2)C1 Cc1ccc(NC(=O)OC(C)(C)C)cc1CNC(=O)CCC(=O)c1cccnc1 C1(C(N2CCC(Nc3ncnc(O)c3Br)C2)=O)CC2(C1)CS(=O)(=O)C2 Cc1scc(C(N2CCC(C)(NC(=O)CCCC3CCCO3)C2)=O)c1C C12(NC(COCC(C)C)=O)CC(CNC(=O)COCC(c3ccccc3)C)(C1)C2 C(=O)(CCCN(C)N=O)NCCCN(C(=O)Cc1cnn(C)c1)CCC N1(C(Cc2nn(C)c(Cl)c2)=O)CC(NC(=O)Cc2cnoc2)CC12CCOCC2 Cc1ccc(CC(=O)NCC2CCN(C(=O)CSc3nncs3)CC2)cn1 C1(C(N(C(C)CSC)CC)=O)CCN(C(=O)CCOCC(C)C)C1C Cc1ccc(C=CC(=O)NC2CCCC2NC(c2ncoc2C2CC2)=O)cc1C c1(C(N(C2CC(=C)C2)C)=O)conc1CNC(C1(CCC)CCC1)=O C1(C(=O)Nc2cscn2)CC2(CCCC2)C1.C12(C)CCCN1N(C)CC(=O)NC2 c1(N(CCN)CC)ccc(S(=O)(=O)N(C)C)cc1.C1(C(C(CC)=O)=O)CC(CSC)C1 N1(C(c2c(C)cncc2C)=O)CCC2CCC(C1)N2C(c1ccc(Cl)cc1F)=O CCCC(C)(CCC)C(=O)N1CCOC(CC(N2CC(CO)C(O)C2)=O)C1 c1(C(C)N(C(CC2CCCC2)C(=O)NCC(F)F)C)nc(C2CC2)no1 c1(C(=O)NC(C(C)NC(CC(n2ccc(C)n2)C)=O)C)ccc2c(c1)OCCO2 c1(C(N2CC(NC(C3CCCO3)=O)CC(C)(C)C2)=O)ccc2c(O)n[nH]c2c1 C1(CCNC(C(C)OCC(C)C)=O)CN(C(C2(N(C)C)CC2)=O)CCS1(=O)=O C=CCC(C)(C)CC(=O)NC1CCN(C(=O)CCCc2ccc(Cl)cc2)CC1F Cc1ccc(CNC(=O)C(c2ccccc2)C2CCCNC2)nc1-c1nn[nH]n1 c1(OC)ccc(C(=O)NC2CC2CNC(=O)CN2CCC(C)C2)cc1O c1(C(N2C(CNC(c3c(C)cn(C)n3)=O)CC3(CC3)C2)=O)ccc2cccnn12 c1(C(N2CC3C(CC(=O)OC)(CC3)C2)=O)cc(Cl)nc(Br)c1N CCC(CC)(C(=O)N(C1CCCC1)C(=O)CN(C1(n2cccn2)CCC1)C)OC C1(NC(c2c(C)nc(CC)o2)=O)CN(C(c2ccc(C)cc2O)=O)C2(CCC2)C1 c1(NC(C2CC(NC(C3CCCO3)=O)C2)=O)cc2ccccc2c(Br)n1 Cc1cc(C(N2CCN(C(c3c(C)ncn3C)=O)CC2C)=O)c(O)c(C)c1 C(=O)(C1=CC2(CN(C(C3CCC(F)C3)=O)C2)OC1)NCCc1n(C)cnc1 C(=O)(CC(C)CC(C)C)NCCC1N(C(CCCc2nnc(C)n2C)=O)CCC1 C(C(CCC)C(=O)NCCNC(=O)OC)NC(COCC(=C)C)=O N1(Cc2cccc(OC)c2Cl)CC2OCCN(C(=O)CNC(=O)C(F)(F)F)C2C1 c1(CNC(C23CC(C(=O)Nc4cnc(Cl)cn4)(C2)C3)=O)ccc([N+](=O)[O-])cc1 C1(NC(c2c(Br)ccc(N)c2)=O)CC2CCC(C1)N2C(C1CC2(CCC2)C1)=O N1(C(c2c(C)sc(O)n2)=O)CCCN(C(c2cc(N)cc(O)c2)=O)CC1 N1(C(CSCC=C)=O)CCOCC1CN(C)C(C1COCCN1CCC)=O.C(=O)NC N1(C(C(N2CCOCC2)C)=O)CCC(CN(C(=O)COc2ccon2)C2CC2)C1 c1(C(N(C(C)C)CCNC(C2CC2c2ccccc2)=O)=O)cc(C(F)F)nn1C CC1=C(C(=O)NC2CCN(C(=O)Cc3ccc(F)cn3)C(C)C2)CCS1(=O)=O CC1(C)CCCCC1CC(N1CCSCC1CCNC(=O)CCC1CCCCC1)=O c1(NC(C2C3(CN(C(Cc4ccc(C)nc4)=O)C3)C2)=O)c(F)cc(Br)cc1Br C(=O)(C1CC(=O)Nc2cc(F)ccc21)NC1(C)CN(C(C2COC(=O)N2C)=O)C1 c1(NC(C)C)cncc(C(=O)NCC2(C)CCN(C(c3cc(CF)on3)=O)C2)c1 c1(C(N(CCCCCNC(COC(CC)C)=O)C)=O)cncc(CO)c1 O=C1CC(C(N2CCC3CC23C(N2CCC3CCCC23)=O)=O)C2(CCC2)C1 c1(CCC(=O)NCC2(O)CCN(C(c3cc(F)cs3)=O)C2)ccccc1Cl C12(CNC(C3(OC)CCCC3)=O)CC(CN(C(=O)CC3CC(SC)C3)C1)C2 CC1(C)CCCC(C(=O)NC2CC(C(N3CC(F)(F)CC3C(N)=O)=O)C2)C1 C1(NC(C2CC(OC)C2)=O)CN(C(=O)CC(C)c2ccccc2)CC12CC2 Cc1cc(C(N2CCC(C(C)NC(=O)COCC3CC3)C2)=O)ccc1O C(=O)(C(O)C(C)(C)CC)NC(CN1CCN(C(C(CC=C)(F)F)=O)CC1)C N1(S(C)(=O)=O)CCc2c(NC(=O)CC(F)(F)c3ccccc3)cccc2C1 c1(C(=O)NC2C(NC(C3(C)CCCCC3)=O)CCC2)cccc(C#N)c1 C1(C(N(C2CCCC(O)C2O)C)=O)CN(C(=O)CCOCC2CC2)CC1(C)C c1(C(N2CC(COC)(CNC(=O)C(CO)N(C)C)C2)=O)cc2n(n1)CCCO2 CC1(C(=O)NC2CC(NC(C3(c4cccnc4)CC(F)(F)C3)=O)C2)COC(=O)C1 CCC(CC(=O)NC(c1n[nH]c(CO)n1)C)NC(C1CCN1CC)=O C=CCC(CNC(c1cc(C#N)cn1C)=O)C(=O)N1CCC(C(=O)OC)O1 Cc1sc(C(=O)NC2(C3CCCN3C(c3cc(O)n(C)n3)=O)CC2)nc1O N#Cc1cccc(C(=O)NC(CNC(C2CC2C2CCOCC2)=O)CO)c1Br CCCC(O)CCN=c1ccnc(NC(c2nccn2CC)C)[nH]1 N1(C(C(=O)NCc2cncc(OC3CCCCC3)c2)=O)CCC2(CC1)CC2 Cc1cc(=O)n(C)nc1C(N1CC(Oc2ccc(Cl)c(F)c2)C1)=O C12(C(=O)NCC3(C#C)CCC3)CC(C)(CN1C(=O)C(C(C)C)SCC)C2 C1(C(N2CCC(O)(CC)C2)=O)CN(C(C2CC3CCC2CC3)=O)CC12CCC2 c1(C(C)C)cc(C(N2CCN(C(=O)C(F)C(C)(C)O)CC2C)=O)cc(F)c1 O(NC(=O)C(C)N(C)C(c1c[nH]nc1CC)=O)CCC C1(N(C(=O)N(C)CCF)CC)COCC1O CCCC(CNC(c1ccnc(C)n1)=O)C(=O)N(C)CC1(OCC)CCC1 Nc1cc(C(N2CCOC(CNC(C3Cc4nncn4C3)=O)C2)=O)cnc1Cl C(=O)(C1CCCc2sccc21)NC(C(C)NC(C(C)C)=O)CO C=C(C)CCC(=O)N1CCN(CC2CCCN(C(C3CC3C(C)C)=O)C2)CC1 N1(C(CN(C(C(COC)OC)=O)CC2CC2)=O)CC2(CCC(=O)O2)C1 CC(C)P(=O)(CC(=O)NCCC1CN(C(C2CCn3ncnc3C2)=O)C1)C(C)C N1(C(C(=Cc2ccc(F)cc2)C)=O)CCC2(C1)CN(C(=O)Cn1nnc(=O)[nH]1)C2 N1(C(C(C)n2cnnn2)=O)CCC(CCNC(=O)C(c2cccc(O)c2)C)CC1 c1(NC(C2CCN(C(C(COC)OC)=O)C2(C)C)=O)cccc2cccnc12 C=CC1CN(C(=O)C2=C(Cl)CC2)CC1NC(c1ccnc(C)c1)=O C1(CC(C)N(C(=O)C(=O)NCC2CCCC2C)CCO)CCCCC1 C1(CC)(NC(=O)CCNC(=O)C=CCl)CCCN(C(c2cnn(C3CC3)c2)=O)C1 C1(CC(=O)OC)CN(C(c2cc(C)c(OC)c(I)c2)=O)CCC1(F)F c1(C(=O)NCC2(C(N)=O)CN(C(c3cnsn3)=O)C2)ccc2c(c1)C(=O)NC2 N1(C(C(CSC)C)=O)CCCC2(C1)CN(C(C1(C#N)CCCOC1)=O)C2 c1(N(CCN(C)C(C2(c3ccc(S(N)(=O)=O)o3)CC2)=O)C)nc2c(F)cccc2o1 CC(C)C(C#N)C(=O)NCC1CN(C(=O)CCCNC(=O)C2CC2)CC1C c1(OC)ccc(CC(=O)NCC2CCN2C(=O)CC2CCOC2(C)C)cc1 Cc1ncc(C(=O)NCc2cc(C(=O)NC3CC3O)on2)c(=N)[nH]1 N1(CC(=O)N(CCOC)CCNC(C2CCCN2CC(C)C)=O)CCN(C)CC1 Cc1cc(C(F)(F)F)c(C(N2CC3CC2CN3C(c2cncn2C)=O)=O)c(O)n1 CCC(C)(C(=O)NCC1CC2(CO1)CN(C(C13CC(F)(C1)C3)=O)C2)C(F)F c1(C(N2CC(O)(C(C)NC(C(C)C3CCCC3)=O)C2)=O)ccc([N+](=O)[O-])cn1 Cn1cncc1C(=O)NC1(CO)CN(C(C2CCNC2=O)=O)C1 c1(C(C)=O)cc(-c2csc(NC(=O)CCC3CC3)n2)n(C)n1 C12(C(N(CCCCN(C(=O)CCc3ncc[nH]3)C)C)=O)CSCC1C2(F)F CCCCCC(O)C(=O)NC1CC(NC(C2(C(C)C)CCC2)=O)C1 Cc1cn2ccnc(C(=O)NCCC(C)N(C(=O)CN3CCC3C)C)c2n1 C(CC(C)C)(C(=O)N1CCC(O)(C(C)C)C1)NC(c1cc(OCC)no1)=O N1(C(CC2N(CC)CCOC2)=O)Cc2ccccc2C1CNC(=O)C(C)COC c1(C(=O)NC2CN(C(C(CCC)OCC)=O)C2)cc(Cl)c(Cl)cc1N N1(C(=O)Cc2ccc(O)cc2)CCC(NC(C2(O)CCCCCC2)=O)C(CO)C1 C(=O)(CC(C(F)(F)F)NC(C1CCOC1(C)C)=O)N1CCC(CCCC)C1 C1(NC(c2ncc(OC)nc2OC)=O)CCCC12CN(C(=O)CCCF)C2 c1(-c2nc(COC)nn2-c2ccc(F)c(F)c2)cc2cccc(Cl)c2s1 O=C(CCCCC1CCCC1)OCCCN1CCC1 C1(C(=O)NC2(CC=C)CCOC2)C2CC3C(C2NC(=O)C(=O)NCC)C13 c1(OC)cc(NC(C2CCC3(CCC3)CN2)=O)c(C)cc1C c1(CC(C)Nc2nccc(N3CCSC(C(F)(F)F)C3)n2)ccc(C#N)cc1 N1(C(N)=O)CCCC1C(=O)NC1CC(CCNC(=O)C(c2ccccc2)O)C1 CC1OCCCC1C(=O)NCC1C2CC1N(C(c1cnsn1)=O)C2 N1(C(C(CC)C)=O)CCOC(CNC(=O)CC2CC3(COC3)C2)C1 C12(C(=O)NC3CC(C)CN(C(=O)CNC(=O)C4CC4)C3)CCC(O)(CC1)CC2 c1(CC)ccc(C(=O)N(C)CCNC(=O)CCc2cc(C)on2)s1 N1(C(C2(SCC)CC2)=O)CCCC2(CCN(C(=O)C#CC3CCCOC3)C2)C1 c1(CC(=O)NCCN(C(=O)C(C)C(F)(F)F)CC(C)O)cc(O)nc(O)n1 CCCCCCCCNC(=O)C(N1CC2CC2(CNC(=O)CCC2CC2)C1)=O c1(C(C(=O)NCCCOC)N(CC(C)OC)C(C)C)cc(C)cc2c1CCC2 N1(C(C2CC(F)CN2Cc2cc(C(F)(F)F)ccc2Br)=O)Cc2ccncc2C1 c1(-c2ccc(C(=O)NCC(CNC(c3c(CC)scn3)=O)O)s2)ccc(Cl)cc1 C(=O)(CS(=O)(=O)C(C)C)N1CC=CC(NC(c2cc(COC)sc2)=O)C1 c1(CC(=O)NC2C3CC2CN(C(=O)CC2C=CCC2)C3)ccc2c[nH]nc2c1 CS(=O)CCC(O)C(=O)NCCC1CN(C(=O)CC2(C)CC2)C1 c1(C(N(C)CC2OCCN(C(C(CCC)O)=O)C2)=O)nn(C)c(=O)cc1C CN1N=C(CC(=O)NC(c2ccnn2C)C(=O)NCC2(C)CCOCC2)CC1=O C(=O)(C#CC1CCOCC1)N1CC(NC(CCOC)=O)C2(C1)CC2 C1(C(=O)NC(C=C)(C)CC)CCC(NC(=O)CC2(C)CCCCC2)CC1 Cc1ccc2c(c1)CN(C(C1CCC(NC(C3(C#N)CC3)=O)C1)=O)C2 C1(CC)CN(C(=O)CCc2ccc(F)cc2F)CCC1NC(c1csc(O)n1)=O C1(C(=O)NC(C#C)(C)C2CCCO2)CCC(CNC(=O)CCc2nc[nH]n2)C1 c1(OC)c(F)cccc1NNC(=O)NCc1nc2ccc(Br)cc2o1 C1(C(=O)NC(C2CCCC2)CNC(C2(CC)CCC2)=O)(OC(C)C)CCCC1 c1(NC(C2CCC(CC)CC2)=O)cc(NC(C)(C)C)ccc1P(C)(C)=O C(=O)(C(C)S(=O)(=O)Cc1ccc(C#N)cc1)N1CCC(N(C)CC)CC1 c1(C(N(CC(CC)NC(=O)C(C)CSC)C)=O)cc(-c2ccccc2)oc1C CC1(C)CN(C(c2n[nH]cc2Cl)=O)C(CNC(=O)C(C2(O)CCCC2)F)CO1 c1(C(=O)NC2CC(C)(NC(=O)Cn3cnnc3O)C2)c(F)cc(Cl)cc1F C(=O)(C(C)(F)C(C)(C)F)N(C(CNC(c1cccc(C(F)F)n1)=O)C1CC1)C C(=O)(C(CC(=C)C)NC(C1CCC(=O)N(C)C1)=O)NCC(C#C)CC C1(CC)CCN(C(=O)C=CC(C)NC(c2ncoc2C2CC2)=O)CC1 c1(OCC(N2CC(NC(C3(COC)COC3)=O)C2)=O)cncc(Cl)n1 N1(C(c2scc(C)c2)=O)CCCC1C1CCCN1C(=O)CCN(C)CCO c1(CNC(C(=O)NC(c2ccnn2C)COC)=O)nn(C)cc1Cl C1(NC(C(C=C)C)=O)CCC(CC(=O)Nc2cnc(SC)nc2)CC1 C12(C(=O)NCC3(OC)CN(C(C(CC)(CC)OC)=O)C3)CCCCC1C2(F)F c1(C(=O)NCC2CCC2C(=O)NCC2CCCO2)cccs1 C(=O)(C1Cc2ccc(Cl)cc21)N1CC2C(NC(=O)CC3(CO)CC3)(C2)C1 c1(NC(N(C(CC)C)C)=O)cnn(CCOC)c1 C1(C)(CNC(C2(C(=O)OCC)CCC2)=O)CN(C(=O)C(O)C(C)CC)CC1C Cn1ncc(C(=O)NC2CCC2NC(=O)C(O)C2CCC2)c1Br N1(C(C(COC)(C)C)=O)C2CCC1(CNC(C1CCC(F)CC1)=O)CC2 C1(CN(C(C2(CSC)CCC2)=O)C)CC(F)CN1C(c1cc(C)c(Cl)s1)=O Cc1nnc(O)c(C(=O)N(C)CC2(NC(=O)C(C)SC(F)(F)F)CC2)c1C c1(C(=O)NC2C(NC(c3cc(OC)nn3C)=O)COCC2)cccc2nccn12 C1(C)(CCC)CCCN(C(C2(C)CN(C(=O)Cc3cnnn3C)CC2C)=O)C1 C1(CC=C)(CNC(=O)C(=O)Nc2ccnn2CC2CCOC2)CCOCC1 C1(SC)CCC(N=c2[nH]c(Cl)nc3c2CCCC3)C1 CCC(C#N)C(=O)NC1CC(N(C(=O)C=Cc2cnccn2)C)C1 C1(CC(=O)OC)C2CN(C(C3(N)CCC4CC34)=O)CC12 c1(C(N2CC(COC)(NC(=O)C(C)=O)C2)=O)ccccc1OC c1(C(N2CC(CNC(c3cncc(C)n3)=O)C2)=O)nc2n(c1Cl)CCCC2 c1(C(=O)NC2CN(C(COCCC)=O)C(C)(CC)C2)cc2ccccc2cc1Cl C(=O)(C1CCCc2nc[nH]c21)NCC(CNC(=O)CC(c1cccc(F)c1)O)O N1(C(c2cccc(NC)n2)=O)CC(NC(C2(CC(C)C)CCC2)=O)C(C2CC2)C1 C1(C(N2CCC(NC(c3cc(Br)c(Cl)s3)=O)C2)=O)CCC=CCC1 N1(C(C2C(OC)CC2)=O)CCCN(C(C2CC3C=CC2CC3)=O)CC1 N1(C(C(CC2CC2)OCC)=O)CCCCC(C(=O)NCc2ccc(CC)o2)C1 C1(NCCCC2CCN(C(=O)OC(C)(C)C)CC2)CCOC12CCCCC2 CC1CCN(C(=O)COCCCF)C1C(N1CCC1)=O C(=O)(C1CCCc2sccc21)N1CC(C)(NC(c2onc(C)n2)=O)C1 CC1CC(c2ccccc2)CN(C(C2CCCN(C(c3cccnc3)=O)C2)=O)C1 C(=O)(CC(O)CC(C)C)N1CCC(C)(C(=O)NC(CCC)C(F)(F)F)CC1 Cc1cc(C(=O)NC2CCCCC2NC(c2cn(C3CCOC3)nn2)=O)nn1C C(=O)(C(O)C1=CCCCC1)NCCC(CC)(C)NC(C1CC12CCC2)=O C1(NC(c2cnn(C(C)C)c2F)=O)CC2CN(C(=O)C(C)(C)C3CC3)CC2C1 N1(CC(C)O)CCN(C(=O)CCCn2cc(CCN(C)C)nn2)CC1 Cc1ccc(CCC(=O)NC2CCN(C(=O)C=C3CC3)CC2C)cc1C C1(CNC(C(CCCOC)C)=O)CC2(CCC2)CN1C(C1CCCN1C=O)=O c1(CC(OC)OC)csc(CNC2CC2CN(C)C2CC2)n1 c1(C(=O)NCCN(C(C(C)OCc2ccc(F)cc2)=O)C(C)C)cn2ccnc2s1 C(=O)(N1CCC(C(N(C)CC2(O)CCOC2(C)C)=O)O1)c1cncc(C(N)=O)c1 N1(C(c2c(N)non2)=O)CCC(C2CCN(C(=O)C(=O)NCC(F)F)C2)C1 C(=O)(CC(C)C(C)C(C)C)N1CC(N(C(=O)CCc2cc(C)cc(C)c2)CC)C1 c1(C(=O)NCCC(C)CCNC(=O)C=Cc2ccco2)cc2c(s1)CC(C)(C)C2 N1(C(Cn2ncc(C)c2)=O)CCC(C)(CCNC(=O)CC23COC(CF)(C2)C3)C1 Cc1oc(CO)cc1C(N1CCC(C(C)C(=O)N(C)CC2CCOC2)C1)=O C(=O)(CCC(=O)NC(C(C)NC(c1csc(O)n1)=O)C(C)C)NCCCOC Cc1noc(NC(C2CN(C(c3cccc(=O)n3C)=O)CCN2)=O)c1C#N S(=O)(=O)(C=Cc1ccccc1)NC1CCC(NC(c2ccsc2)=O)C1 N1(C(c2c(C)nns2)=O)CC2(CCC2)CC1CNC(c1ccc(CCO)cc1)=O N1(CC(C)C)CCC(C(N2CC=CC2CNC(C2CC2(Cl)Cl)=O)=O)CC1 CC(CC(=O)NCCC(N)=O)NC(=O)Nc1ccccc1 N1(C(C(CC)(C)CO)=O)CCCC2(CCN(C(=O)CC(C)(O)C(F)(F)F)CC2)C1 C(=O)(CC(CN(C)C)C(F)F)N(C1(NC(CN(C(C)C)C)=O)CC1)C C(CC(CC)C(=O)N1CC=CCC1C(=O)NCC1CCC(C)C1)=CC C(C(=O)NC(CNC(c1cccc(SC)c1)=O)C1CCC1)(C(C)(C)C)OC N1(C(=O)C2=C(Cl)CC2)CCCC(C2CN(C(=O)COCCO)C2)C1 c1(CC(=O)NCCN(C(c2cnc(C3CC3)[nH]2)=O)C2CC2)ccc(F)cc1 N1(CCC)C(=O)CCC1C(=O)N(C)CC1CCCCN1C(c1coc(CO)c1)=O C1(CC)CCN(C(c2cnn(C(C)C)c2)=O)C1C(=O)N(CC)Cc1cn(C)nn1 N1(C(COCCC#C)=O)CCC2CCN(C(=O)CCCCCCCSC)CC2C1 C1(NC(CC2(C)CC2(F)F)=O)C2CC3CN(C(c4cc5occc5s4)=O)C1C3C2 CC1CN(C(C2(CNC(C3CC(O)C3)=O)CC3(CC3)C2)=O)CC(CO)O1 c1(CCC)cc(C(N2CC(CNC(=O)CCc3nncn3C)CC2C)=O)n(C)n1 c1(C(=O)NCCCN(C)C(C2(CF)CCC2)=O)cncc(C(F)F)c1 C(CC(F)F)(C(=O)NC(C)CN1CCOCC1)N(C(Cc1c(C)nccc1)=O)C C(C)(c1ccccc1C)=CC(N1CC(OCC)(CNC(c2c[nH]cc2Br)=O)C1)=O N1(C(COCCCOC)=O)CCN(C2CCN(C(C3CCC(=O)N3)=O)CC2)CC1 c1(C(N2CC(CNC(C(CC)(C)F)=O)OCC2)=O)ccc([N+](=O)[O-])cc1Cl C1(C(N2CCCC(CCNC(C(C)=C(C)C)=O)CC2)=O)CC2CSCC(C1)C2 C(Cc1cc[nH]n1)(C(=O)NCC1COCC1O)NC(CN(C)C1CC1)=O C=CCN=C(NCC1CCOC1(C)C)N1CCC2(OC)CCCCC2(OC)C1 c1(C(N2CCC(NC(c3cnc(OC)c(Cl)c3)=O)C2)=O)c(Cl)cccc1[N+](=O)[O-] C1(CNC(=O)C(=CC2CCCCC2)F)CC2(C1)CN(C(C1CCCC1(F)F)=O)C2 N1(C(C(C)OC)=O)CCC2(CCCCC2NC(c2cc(C)no2)=O)C1 C(CCCCCN=[N+]=[N-])NC(C(C(C)NC(C1C(C)(C)C1(F)F)=O)(C)C)=O C1(O)(C(C)NC(=O)CCc2cn[nH]c2)CCN(C(=O)C(N2CCC(O)CC2)C)C1 CCC(O)C(C)(C)C(=O)N1CCC(CNC(c2sccc2F)=O)(OC)C1 c1(CC)ncc(Cl)c(C(=O)NCC2CN(C(=O)CC3(C4CC4)CC3)CCN2C)n1 C(=O)(C1=NOC(C(=O)NCC(CC(C)C)NC(C2(SC)CCC2)=O)C1)OC c1(C(=O)NCC2C(CNC(=O)C=C3CCCCC3)C2)ccccc1-n1nccn1 C1(C(N2C(COC)C=CCC2)=O)CCN(C(=O)C(C)O)C1(C)C O=C1Cc2cc(C(N3CC(NC(C4CC=CC4)=O)C(F)C3)=O)c(Cl)cc2N1 N1(C(c2c(C)ccs2)=O)CCCC(CNC(c2c(C)cnn2C(C)C)=O)CC1 CCC(CC(=O)NC1(CNC(c2sccc2-n2ccnn2)=O)CCC1)C1CC1 C12(C(N3CC(C)C(O)CC3)=O)CCCC1CCN2C(=O)CNC(=O)CN(C)C CC1N(C(=O)CC2(NC(c3ccc(F)c(O)c3)=O)CC2)CCCC1(C)C CC12CC(NC(=O)C(C3CCCCC3)O)(C1)C1(CN(C(c3ccc(F)s3)=O)C1)O2 c1(C(=O)NCC(C)N(C)C(c2ccc(F)o2)=O)c(Cl)cc(Cl)cc1Cl N1(Cc2cccc(NC(C)=O)c2)CCC(C)(CNC(c2cnc(C)s2)=O)CC1 C(CCOCCO)(C(=O)NC1COCC1CO)NC(C1CCC(F)(F)C1)=O C1(CNC(C=CC(C)(C)NC(=O)Cc2ccnc(O)c2)=O)CC2CCC1C2 c1(C(N2CC(OC)CC2CNC(=O)C(C)(C)CO)=O)cccc(OC)c1C.CCO c1(CC(=O)NC(C2N(C(CNC(=O)NC)=O)CCC2)C)ccc2nc[nH]c2c1 c1(OC)cc(OC)c(OC)cc1CN(c1cc(NCCOC)ncn1)C N1(C(=O)C=CCN2CCCC2)CCN(C(=O)COCCN(C)C)C2CC12 Cc1cccc(C(=O)NC2CC2C(N2CCC(O)C2)=O)c1 Cc1ncn(C)c(=O)c1C(=O)NC1CN(C(C2(C#N)CC3(CCC3)C2)=O)CC1O C1(C2CCCCN2)(C(N(CC(C)CO)C)=O)CCOCC1 CC1(C)CN(C(C2CCCC3CC23)=O)CC(CNC(=O)Cn2ccc(O)nc2=O)O1 N1(C(C(C)OCc2cccnc2)=O)CCC2CN(C(C3(CF)COC3)=O)CC12 CC(CCC(=O)NC1CC(NC(C2CN(C)C(=O)N2)=O)C(O)C1)N(C)C C1(c2scc(C(N3CCN(C)CC3CC3CC3)=O)n2)Cc2ccccc2O1 CCCCC(C)C(=O)N1CC2(C1)CN(C(c1ccc(NS(C)(=O)=O)cc1O)=O)C2 C1(C(N2C(CC(=O)NC3CCC(N(C)C)C3)CC(O)C2)=O)CCCC12CCC2 N1(C(=O)CO)CCCC2(C1)CN(c1ccnc3cc(Br)nn13)CCO2 Cc1cc(NC(c2cc(Cl)n(C)n2)c2nnnn2CCCF)cc(C(F)(F)F)c1 C1(C(=O)NC2(CO)CCN(C(=O)C=CCF)C2)(OCC)CCSCC1 C(=O)(CC(F)(F)CNC(=O)OC(C)(C)C)NC1CC(C)(NC(CC(=C)C)=O)C1 N1(C(CC(=O)NCC#C)=O)CC2COCCC2(NC(c2ccc(F)cc2C)=O)C1 N1(C(c2c(F)ccc(C)c2)=O)CCC2(NC(c3cc4n(c3)CCC4)=O)CCCC12 Cc1cnn(CC(=O)NC2CCC(NC(c3cscn3)=O)C2)c1 c1(C(=O)NC2C(NC(C=C(C)C(F)F)=O)CC2)ncnc2c1CCC2 C1(C(=O)NC(c2ccccc2)CNC(C2(CO)CCC2)=O)CN2CCN1CC2 CCCCC(C)CC(=O)NC1C=CC(C(=O)NC(C)CCC)C1 Cc1nc(O)c(C(N2CC(NC(C3CC4CCC(C3)C4F)=O)C2)=O)nc1C n1(C2CN(c3c(Br)cnc(C)n3)C2)ccc(=NC(=O)C2(c3cccs3)CC2)[nH]1 C=CC(C)(CC)C(=O)N1CCC(CCCCNC(c2ccc(C)c(F)c2)=O)CC1 C=CCCCCCN(C)C(C1CSCCN1C(=O)Cc1cc(C)no1)=O C(=O)(CCCCC(F)(F)F)NCCN(C(=O)C(C(C)C)C1CC1)CCOC C12(C(N(CCCCO)CC)=O)CCN(C(c3nc(O)sc3C)=O)CCC1C2 c1(C(N(CC(CC)NC(=O)CNS(=O)(=O)N(C)C)C)=O)cccc(Cl)c1C c1(C(N2CCC(F)(CNC(Cc3cn(C)nn3)=O)C2)=O)cccc2cnn(C)c12 c1(CN(C(C(c2cccs2)NC)=O)C)ccc(OCC(=O)OC)cc1 C(C1=NOC2CCCC12)NC(C(C1CN(C(CCC=C)=O)C1)O)=O C1(C(=O)NCC2C(CNC(COc3cccc(CC)c3)=O)C2)OCCOC1(C)C C(=O)(C(C)(C)CCF)N1CC2C(C(=O)NCCC(C)N3CCC3)(C2)C1 c1(NC(CN(C(C2CCN2CC)=O)NC(CCSCC)=O)C)ccccc1Cl C1(C(=O)NC(c2nc(C(N3CCC3C3CCCC3)=O)co2)C)(CO)CC=CC1 c1(OC)ccccc1-c1ncc(C(=O)NC2CC2CNC(C2OCCC2C)=O)s1 CC(C)(C)C(C(=O)NCc1ncccn1)NC(c1nsnc1O)=O N1(C(c2c(OC)cncn2)=O)CC2(C1)CN(C(=O)C(C)(C)S(C)(=O)=O)CCO2 C#CC1(C(=O)N(CCC(C)O)C)CCN(C(C2CCCCO2)=O)C1 c1(-n2cc(CCCCCCNC(C(C)(CO)OCC)=O)nn2)cnc2ccnn2c1 N1(C(CSCc2nc(C)sc2)=O)CCC(C)C1CNC(=O)CCc1cc(Cl)no1 CCCCCC(CC)C(=O)NC1CCC(C(=O)NCc2ncsn2)C1 CC1CCCC2CCCN(CC3CCN(Cc4ccccc4)C3)C12 c1(OC)cnc(Cl)[nH]c1=NC(=O)C1CC1Nc1ncncc1Br c1(N2CC(CC)C(O)C2)cc(NC(c2ccc(OC)nc2C)C)nc(C)n1 C12(C(N3CC(CNC(CCNC(=O)OC)=O)C3)=O)CCCCC1CCCC2 CCC(C)CC(C)C(=O)N1CCC(C(C)(C)O)C1 c1(CC)nn(C)c(NC(C2CCCCN(C(=O)COC(C)=O)C2)=O)c1Cl CCC(CCC(=O)N(C(C)CC(=O)Nc1ccc(OC)c(O)c1)C)OC CCCN(OC)C(=O)CC(CCC)NC(=O)C(N)CC(C)C C(=O)(C(C)(C)C(=O)N1CCC(NC(=O)C=C2CCN(C)C2)C(O)C1)OCC Cc1c(C(N2CC(=C(F)CNC(=O)C(F)C(F)(F)F)C2)=O)oc2ccc(F)cc12 C1(CC#C)(C(=O)NCC(=C)CCNC(=O)CCC2CCCOC2)CCOC1 Cc1n[nH]cc1CN(C)C(c1ccoc1CNC(C12CSCC1C2)=O)=O C1(NC(c2nc(C(C)OC)sc2)=O)CCN(C(C2(CSC)CC2)=O)CC12CCC2 c1(SC(CC)C(=O)N2CCCC2CC)ccnc(N(C)C)n1.C12CCCN1C2=O C(CC(CC)C(=O)NCC1CCCN(C(=O)CCc2ccc(O)nc2)CC1)=CC C1(C(N(CC(O)CO)CC)=O)CC2CN(C(c3cccn4cncc34)=O)CC2C1 Cc1nc(C(N2CC=CC(NC(=O)CCCCNC(N)=O)C2)=O)nn1C c1(CC(C(C(=O)NCCN(C(CCC(C)C)=O)C)F)C)c[nH]c2ccccc12 c1(CC)ncc(C(N2CCC(NC(c3csc(Cl)n3)=O)CC2C)=O)c(C)n1 CC1CN(C(=O)C(c2cnn(C)c2)NC(c2ccc(F)cc2)=O)CCN(C)C1 N1(C(C(=C)Cc2ccccc2)=O)CCSCC1C(=O)Nc1oncc1C#N C(C(CO)(CO)NC(C1OCCC1(C)C)=O)N(C(C1(CC)CC1)=O)C c1(OC)ccc2c(c1)CCC2(O)CNC(=NCC1CCC1)NCC1OCCO1 c1(C(=O)NCC2(NC(CCCCOCCC=C)=O)CC2)nc2sc(C)cn2c1C C1(NC(CSC)=O)CN(C(c2cc(O)nc3c2CCCC3)=O)CC12CCOCC2 CC(CC(N)=O)C(=O)N1C(CNC(=O)CCc2nnc(C(F)F)o2)CC2CC12 C(C)(CCCCNC(c1cccc(Cn2cccn2)n1)=O)NC(C1C(=C)CC1)=O N1(C(C(C)OCCOC)=O)CC2CC(NC(c3ccnc(C4CCC4)c3)=O)CC1C2 N1(C(C(COC)O)=O)CCN(C(c2ccn(C3CC3)n2)=O)C(C(F)F)C1 n1(CC(=O)NC(CN(C(C(CC)(C)F)=O)C)C)cc(F)ccc1=O c1(C(C)C)cccc(F)c1C(=O)NCCC(C)NC(c1c(Cl)cnn1C)=O N#Cc1c(NC(C2CC23CCN(C(C2(O)CC2)=O)C3)=O)cccc1F N1(C(c2cc(SC)c(C)o2)=O)CC(C)C(NC(=O)CC2(O)CCC2)C(C)C1 N1(CC)CCN(CC(N2CCC(C(=O)NC3CCN(C(N)=O)CC3)C2)=O)CC1 c1(C(N(C(C)CCNC(=O)CNS(C)(=O)=O)C)=O)ccc(-c2cnco2)cc1 C(=O)(C1=CC2CCCC12)NCC1CCN(C(c2c[nH]c(=NC)s2)=O)CC1 C1(CCOC)CN(C(=O)C2=NOC(C(C)(C)C)C2)CCN1C(=O)CS(N)(=O)=O C1(NC(C(C2(O)CCCCCC2)(C)C)=O)CC2CCC(C1F)N2C(C1CSC1)=O N1(CC(=O)NCC2(C(C)(C)O)CN(C(C(CC)F)=O)C2)CCN(C)CC1 c1(C(N2CCCC(CC=C)(NC(C3CC3C)=O)C2)=O)cc2c(nn1)OCCS2 c1(OC)nc(N2CC3C(NC(=O)COc4ccc(C(C)C)cc4)C3C2)ncc1Br Cc1ccc(C(=O)OCC2CC=CCC2)nn1 C1(C(N2CCN(C(C)=O)C3C2C3)=O)CC2(CCCCC2)C1 Cn1c(C(=O)NC2CC(NC(C3(CO)CCCO3)=O)C2)cnc1S CC(O)C(C(=O)NC1CCC1)NC(C1CC1C(N)=O)=O c1(SC)c(Cl)ccc(C)c1NC(c1cccc(Br)c1)C1CC1 C1(C(=O)Nc2ccc(Cl)s2)CSCCN1C(=O)NC1(c2cccnc2)CC1 c1(C(=O)NC(CNC(C(c2ccccc2)OC)=O)CO)c[nH]c2cccc(Cl)c12 C(=O)(C1=CNS(=O)(=O)N=C1C)NCCN(C(C(C)OCC#C)=O)CC(C)O C1(C(N2C(CNC(C3C(C)(C)C3C#N)=O)CCC2)=O)CC(=O)CC(=O)C1 C1(NC(CCc2ccn(C)n2)=O)CN(C(=O)Cc2cnn(C(F)F)c2)CC1F Cc1ccc(CC(=O)NC2CCN(C(c3cc(O)nc(Cl)c3)=O)CC2F)c(C)c1 c1(C(=O)NC(CC(C)C)(C)CNC(C2CC=CCO2)=O)ccc2cncn2c1 O=C(C1=Cc2ccccc2C1O)NC1C=CCN(C(c2csc(Cl)c2)=O)C1 N1(C(C2CC(OC)(OC)C2)=O)CC2(C(=O)NCCCCCCOC)CC1CO2 N1(C(CSCC(C)C)=O)CCCC(CN(C)C(c2cc(C(N)=O)cn2C)=O)C1 c1(C(=O)NCC(CN(C(=O)CC2CCC(C#N)C2)C)(C)C)cn(C)nc1Br Cc1cc(C(=O)NC2CC(O)CN(C(c3ccccc3C(C)C)=O)C2)cc(C)c1 N1(C(C(C)=C(CC)C)=O)CC2(COC(CNC(c3nccn4ccnc34)=O)C2)C1 C1(C(N2C(C(=O)Nc3ccc(OC)nc3C)CC3CC32)=O)CCc2ccccc2C1 C1(CNC(C(C)c2cccs2)=O)CCCCN(C(C2(C#N)CCOCC2)=O)C1 c1(CC(=O)NCCC2CCN(C(c3ccc(CO)s3)=O)C2)nnc2n1CCCC2 c1(N2CCCC(CC)CC2)nc2ccsc2c(=NCC2(CO)CCCOC2)[nH]1 c1(C(=O)NCC(CC(C)C)NC(CS(=O)(=O)NC)=O)ccc2c[nH]nc2n1 c1(OCC(N2CC(NC(c3nc(CC)oc3)=O)C(C)C2)=O)c(C)cc(C)cc1C c1(C(N2C(C(CNC(C(C)(C)F)=O)(C)C)CCC2)=O)cnc2cc[nH]c2c1 CCCC(O)CC(=O)NCC12CC(CNC(=O)CSc3n[nH]c(O)n3)(CO1)C2 CCN=C(NCCc1cnc(Cl)c(C)c1)N1CCC(O)C1 C(CCC(C)NC(c1cccnc1)=O)NC(C(c1ccccc1)C)=O c1(CC)cc(C(=O)N(CC)CC2CCN2C(=O)CC2CCCO2)ns1 C1(CNC(CC(CC)C2CC2)=O)N(C(=O)C=CCOC(C)(C)C)CCCC1(C)C C=Cn1nncc1C(=O)NC(COCC)C(=O)NCCC1COCCO1 N#CC1CCCC(CC(=O)NC2C3CC2CN(C(=O)Cc2ccc(Cl)cc2)C3)C1 c1(C(=O)OC)ccc(Cl)nc1NC(CCSC)C(=O)Nc1ccccc1C c1(NC(c2ccc(F)c(F)c2Br)=O)ccc2oc(Cl)cc2c1 Cc1ccc2c(c1)ncn2CC(=O)NC1CCC(NC(=O)CC(C)C(F)F)C1 Cc1cc(C(N2CCC(C(CO)NC(=O)CCc3cnn[nH]3)CC2)=O)c(C)s1 N1(C(C(C)=C2CCCC2)=O)C2CCC1CC(NC(C1CC1c1ccccc1Cl)=O)C2 C(=O)(CS(=O)(=O)C1CC1)NCC1CCN(C(C(Cc2ccccc2)N(C)C)=O)C1 C(CNC(=O)CC=CC(C)(C)C)(CC(F)(F)F)NC(C(C1CC1)OC)=O c1(CC(C(=O)OC)NS(=O)(=O)CC2CCOC2)cc(Br)sc1Br C1(NC(c2c(COC)scc2)=O)CC2CCC(C1C)N2C(=O)Cc1cc(C)on1 c1(CC(=O)NCC(CN(C)C(C2C=CCS2)=O)O)cncnc1O N1(C(CC2(C=C)CCC2)=O)CCC(C2CC2)C1CNC(C1C2C3CCC(C3)C12)=O C1(C)(NC(C=CC(C)NC(C2CC3CCC3C2)=O)=O)C(C)(C)C1(C)C c1(C(CC)C)nc(C)c(CC(=O)NC(C)CCCNC(=O)C(C)CO)c(C)n1 C1(C(=O)NC(C2CCN(C(=O)OC(C)(C)C)CC2)C(F)(F)F)CC(O)C12CCC2 O=Cc1cccc(-c2cccc(CN3CCOCC3)c2)c1Br C1(C(=O)NC(=O)CCC2CC(C)C2)OCCC1C(N(CCF)CC)=O CCCC(C(=O)OC)C(=O)NCC(C)N(C(=O)COc1cccc(Cl)c1)C c1(C(N2CCC(O)(C(CNC(C(F)=CC)=O)C)C2)=O)nc(O)nc(O)c1F CCCCCCCCOCC(=O)NCC1(NC(C2CC2C(=O)OC)=O)CCCC1 C1(NC(c2c(C)nccc2)=O)CN(C(=O)CCc2ccncc2)C2CCCCC12 N1(C(=O)OC(C)(C)C)CCC2C(NC(=O)Cn3cccc3)C12 c1(C2(OC)CCN(C(c3n(CC)ccn3)=O)C2)cc(Br)ccc1F C(=O)(CC(O)C(C)C)N1CCC(OCCNC(c2nc(C)c(C)s2)=O)CC1 N1(C(COCC(=O)OC)=O)CC2CCC1CC2NC(c1cc(C)oc1C)=O N1(C(c2c(C)oc(C#N)c2)=O)CCC2(CC1)CCN(C(=O)C1=CCN(C)C1)C2 CCC(O)C(C)(C)C(=O)N(CCCNC(c1cc(-c2cccnc2)on1)=O)C c1(C(=O)NC2C(C(N3CCC(OC(C)=O)C3)=O)COC2)nccc(C)c1N CCC1(CNC(=O)NC2CN(C)CCN2C)OCCc2ccccc21 C=CCC(CC(=O)NC(C)(CSC)CO)NC(=O)CCCOC(C)C N1(C(C(CC)(CC)OC)=O)CC(NC(=O)CCCCCOC)C(C2CC2)C1 Cc1cccc(C(O)C(=O)NCC(c2ccccc2)NC(C2CCCN2C)=O)c1 N1(C(c2c(C)noc2)=O)CC2CC1CN(C(=O)C(C(C)C)c1cnn(C)c1)C2 C(CCC(=O)NCC1CCCN1C(C1CC2CC2C1)=O)N(C(C)=O)C CC(C)(CCCNC(c1sccc1F)=O)NC(=O)COc1ccccc1C(N)=O c1(CC)nsc(CNC(=O)C(C)CN(C(=O)CCC2CCCCC2)C)n1 N#Cc1ccc(C(=O)Nc2ccc(SCc3nc(=O)o[nH]3)cc2)nc1 C(=O)(C1=NOC(C)(C)C1)NCC1(CN(C(=O)C#CC2CC2)C)CC1 CCCCC(CNCc1cccc(C#N)c1F)CCC c1(C(=O)NCC(CNC(c2ccccc2F)=O)OC)cc(S(N)(=O)=O)oc1C C(=O)(C(C)(C)C(=O)NCC1CC(C)(C)CN1C(=O)C(CC(C)C)N(C)C)NC CN1C(=O)C2CC1CCN2C(=O)CC1CC2(C1)CN(C(c1ccc(F)s1)=O)C2 Cn1nnc2cc(C(=O)NCC3(NC(C4CC(C)(O)C4)=O)CC3)cc(Br)c12 C1(COC)(NC(c2cc(Cl)cnn2)=O)CCN(C(=O)CCCn2cccc2)C1 C(=O)(C(=O)CCC(C)C)NC1C(CC)CN(C(=O)COC2CCOCC2)CC1 C1(CC)CN(C(c2cc(C)ccc2I)=O)CCN1C(c1cnc(Cl)s1)=O c1(C(N2CCC(O)(CNC(C3CCCOC3)=O)C2)=O)cccc2cc(Cl)ccc12 c1(C(CNC(CSC)=O)NC(=O)C(O)CF)ccc2ccccc2c1 C(CCN(C1CCCCCC1)N1CCCC12CCS(=O)(=O)C2)N(CC)CC c1(OC)cc(Br)ccc1CN1CC2CC1CN2Cc1ccc(C(=O)N(C)C)nc1 C#Cc1ccc(OC)c(C(=O)NC2COCC2NC(c2conc2C2CC2)=O)c1 C1(C(=O)NCC(=O)NC(CN(C(c2cncnc2)=O)CC)C)CCOCC1 C1(C(C(=O)NCC(=C)C)N(CC(C)C(=O)OC)C)CCC12CCOCC2 C#CCCCCC(c1nnnn1C)Nc1cccc(C(O)CC(F)(F)F)c1 C1(C(F)(F)C(=O)NC2CC(NC(=O)Cc3cnsc3)C2)(OC)CCOCC1 C1(C(=O)NC2CCC(C)CC2)CN(C(=O)C2=CCSC2)CC1C1CC1 C12(CNC(c3cnn(C)c3Cl)=O)CC(C1)C(NC(=O)C(O)c1ccsc1)CO2 CN=c1[nH]c(=NCCS(=O)(=O)N2CCCC2)[nH]c(=NC2CC2)[nH]1 Cc1cc(C(=O)NCC(C)(CO)NC(C2CC(n3cccn3)C2)=O)ncc1F c1(C(C(N2CC(OCC)(CNC(c3cc(F)c[nH]3)=O)C2)=O)(F)F)cccc(C)n1 c1(C(N2CC(NC(C3(O)CCC3)=O)CC(O)C2)=O)cccc2ccccc12 C(=O)(C(C)CC(=O)OC)NCC(CC)NC(c1ccc(OC)nc1C)=O Cc1nc(S)nc(C)c1CCC(=O)NCCC(C)N(C)C(c1ncccc1Cl)=O N(C1CN(C(C23CC2C3)=O)CCc2ccccc21)C(C(CC)OC)=O C1(C(C(=O)NCC)N(CC)CC)CC(OC)OC1OC N(C1CN(C(=O)C(C)SC)Cc2ccccc21)C(CC1(OC)CCCCC1)=O c1(C(=O)NC2CC(CN(CCOC)C)C2)c(C)nn(-c2ccc(F)cc2Cl)c1C C(c1cnc(C)nc1O)=CC(=O)NC1CCN(C(c2cn(CC)nn2)=O)C12CC2 C(=O)(C(=O)N=S(C)(C)=O)N(CC(CC)NC(=O)CCC(=O)c1ccc(Cl)cc1)C c1(OC)ncc(F)cc1C(=O)NC(C)(C)CNC(=O)C(C)c1ccon1 CN1CCC(CO)(CNC(=O)C(CCC2CC2)NC(c2coc(C(N)=O)c2)=O)C1 c1(C(N(CCNC(=O)CCc2cccnc2Cl)CC)=O)c(C)cccc1C c1(CC)ccc(C(=O)NCc2cc(C(=O)N(C)OCC3CCCO3)on2)s1 C1(NC(c2ncoc2C2CC2)=O)CCCC(CNC(C2CC(O)C2)=O)C1 c1(CC(=O)NC2C3CN(C(CC4OCC(C)(C)C4)=O)C2C3)cc2ccccc2o1 c1(C(N2C3C(NC(=O)C=CC=C(Cl)Cl)C(CC3)C2)=O)cc2c[nH]cnc-2n1 N1(C(CCc2scc(C)n2)=O)CCC(O)(C(C)NC(c2cccc(F)n2)=O)C1 C1(NC(C2C(C)C2C)=O)CCOCC1C(=O)NC1(CCO)CCCCC1.CCO C(=O)(C1=Cc2ccccc2C1O)N1C(C(C)NC(c2cc(OC)no2)=O)CCC1 CCCCC(=O)C(=O)N1CC(N(C(=O)Cc2ccc(OC)cc2)C)C(O)C1 CC1CC(NC(=O)C(=O)N(C)Cc2ncccc2F)CN1C1CC1 Cc1nn(C)cc1CN(C1CC2CNC1C2)C(=O)C(CN)c1ccccc1 c1(C(C)(F)F)ccc(C(=O)NCC(C)(O)CNC(C2CCCO2)=O)cc1 C1(CC(=O)N(CCN(CCC)CC)C)CCCN(C(=O)CCCNC(=O)OC)C1 CCC(C)(CO)C(=O)NCCC1CCN(C(c2csc(=N)[nH]2)=O)C1 C(C(F)(F)CNC(=O)CCC1OCCO1)(C1CC1)OC c1(C(=O)NCC2(OC)CN(c3ncc(C#N)cc3F)C2)sc2nccn2c1C N1(C(C(CCOC)C)=O)CCC(C2(NC(=O)C(C)O)CC2)C1 c1(C(N2C(C)CC(NC(c3csc(C(F)F)n3)=O)C2)=O)ccc2c(c1)CCCC2 c1(CNC(C(C2CCCOC2)OC)=O)cccn1C(c1ccncc1)C C(=O)(C(C#N)(CC)CC)N1CC2CC(C(N3CC(C#C)OCC3)=O)(C1)C2 Cn1nc(C(=O)OCC(=O)NCC(C)(Cn2cccn2)NC(=O)C(C)(C)C)cc1O CC1=C(C(=O)NC2C=CCN(C(=O)CN3CC4CC4C3)C2)CCC1 C(CC(N)=O)(C(=O)NCCc1cc(C)n(C)n1)NC(CCC=C=C)=O c1(CCNC(CNC(C2CC(OC)(OC)C2)=O)=O)cccnc1F O(NC(=O)CSCC(=O)NC(=O)NCCOCCN)CC(CC)C c1(COCC(=O)NCC(C)NC(c2ccc(CCC)s2)=O)cccc(OC)c1 c1(C(=O)NCC2N(C(CCC3CC(OC)C3)=O)CC2)ncccc1O c1(C(=O)NC2C(NC(C3CC(=C)C3)=O)CCOC2)cc(=N)[nH]c(Cl)n1 c1(C(N2CC(CNC(C(COC)C)=O)C(C)(C)C2)=O)cnc2[nH]cc(C)c2c1 Cc1cc(CNC(=O)C(N2CCC(c3nncs3)C2)=O)cs1 c1(CC)cc(C(=O)NCC(C)CN(C(=O)CC(C)OC)C)n[nH]1 c1(COCCNC(CC(CN(CC(N)=O)C)O)=O)ccc(C#N)c(C)n1 Cc1c(C(=O)NC(C)(CNC(=O)CSC(C)C)C(C)C)cnn1CCC(C)C N1(C(C2C(CNC(C(C)n3ccnn3)=O)CC2)=O)CCN(C(C)(C)C)CC1 N1(C(C2C(CC)C2)=O)C(C(=O)NCCc2nccn2C)CC2CC12 c1(C(=O)NC(C2CCCN(C(c3cc(F)n[nH]3)=O)C2)C)ccc2nsnc2c1 C(=O)(CS(=O)CCC(F)(F)F)N1CC(C)C(NC(c2cc3ccccc3o2)=O)C1 C1(NC(C=CCCC)=O)CCC2(CCCN2C(c2cccn(C)c2=O)=O)CC1 N1(C(c2c(CC)c[nH]n2)=O)CCCC2(C1)CN(C(=O)CN1OC(C)(C)CC1=O)C2 C#Cc1cccc(N(C(=O)C(C)N(C(=O)CCC(C)N(C)C)C(C)C)C)c1 N1(C(C(c2n(C)ccc2)=O)=O)CCOC2(CCN(C(C3CC(F)(F)C3)=O)C2)C1 c1(SC)cc(NC(=O)C(=O)Nc2ccc(C(=O)OCC(C)C)cc2)c(C)cc1F c1(C(=O)NC(CN(C(CC(c2ccc(F)cc2)C)=O)C)C)ccc2ncnn2c1 c1(C(N2CCN(C(C(c3c(C)cncc3)C)=O)CC2)=O)cc(Br)cc(N)c1C Cc1ncc(NC(=O)CC=CCNC(C2CN3CCC2CC3)=O)c(C)n1 c1(NC(=O)C=Cc2cccnc2)cc(Cl)c(I)cc1[N+](=O)[O-] c1(C(=O)NC2CC(CNC(C(C)CC3CCCO3)=O)C2)ccsc1C#N CC1C(NC(c2ccc([N+](=O)[O-])s2)=O)C(C)CCN1C(=O)Cn1cccc1 CC1(C)COC(Cc2cn(CCCC(=O)NCC3CC(F)(F)CNC3)nn2)C1 N1(C(C2(NC(CC3CCN(C)C3=O)=O)CC(F)C2)=O)CCN2CCC1CC2 C(=O)(CC(F)(F)C(C)C)NC1CCC(CCNC(C2(OC)CCSC2)=O)C1 C1(NC(C(CC)(F)F)=O)CCC2CC1CN2C(=O)C=Cc1ccccn1 CC1CN(C(=O)CCCCCNC(C2CCNC(=O)C2)=O)C(C)(C)C1 C(CC1=CCN(Cc2cncs2)CC1)NC(C(c1c(C)noc1C)C)=O c1(N(CC(F)F)C)nnc(-c2ccc(Br)s2)n1CCCCCCN1CCCC1 C=C(Cl)C(C)(C)C(=O)N1CCN(CCNC(=O)C(C)NC(N)=O)CC1 C1(CC(=O)NC23CC(NC(CC4(C=C)CC4)=O)(C2)C3)C=CS(=O)(=O)C1 c1(CNC(C)=O)ccc(C(=O)NC23CC(NC(C4CCC(F)C4)=O)(C2)C3)cc1 C1(C(N2C(CN(C(CSCC=C)=O)C)CCC2)=O)CCc2ncccc2C1 C(=O)(C(C)(C)C)NCCC1CC(C(=O)OC(C)(C)C)C1 C1(CCNC(c2c(C(=O)OC)coc2)=O)C(C)CCCN1C(c1c[nH]nc1F)=O c1(CC(=O)NC(CC(C)NC(=O)C=CI)C)c(Cl)cnn1C c1(CNC(CC)=O)cn(C2CCN(C(=O)C(C)(C)c3ccno3)C2)nn1 c1(C(=O)NC(CCCCNC(c2c(NC)cccc2)=O)C)cc2n(c1)CCC2 n1(CCNC2(C(C)=O)CC2C(=O)C(c2coc(C)n2)=O)cc(CO)nn1.C(CO)O c1(N2CCN(C)C(CNC(C3CC4CCC3O4)=O)C2)ncnc2c1COC2 N1(C(C(CO)N(C)C)=O)CC(F)(F)CC1CCNC(c1cc2n(c1)CCC2)=O c1(C(=O)NC2(CN(C(=O)Cc3c[nH]ccc3=O)C)CC2)cc2c(Br)cccc2[nH]1 N1(C(c2cccc3nc(O)[nH]c23)=O)CCCC2(CNC(C3(F)CC3)=O)CCCC12 CC(N=c1cc2n([nH]1)CCOC2)c1nc(Cl)ccc1Cl C1(NC(=O)COC(F)F)C=CCN(C(=O)CNc2ccc(O)cc2)C1 Cc1cc(=NC(=O)C2CCCN(Cc3cccc(OC(F)(F)F)c3)CC2)[nH][nH]1 C1(C(N2CC(C)N(C(C34CCC3CC4)=O)CC2)=O)COc2ccc(Cl)cc2C1 C(C1=CCN(C(c2scnc2Cl)=O)CC1)NC(C1C(C)C1C)=O c1(C(N(C)CC2N(C(CC=C)=O)CCOC2)=O)c[nH]c2ncnc(O)c12 C12(NC(C(CC(C)C)O)=O)CCCCC1CN(C(c1nc3cnccc3s1)=O)C2 c1(C(=O)NC(C(C)NC(=O)Cn2nccn2)C)cnc2sccn2c1=O N1(C(C(CC#C)O)=O)CCC2CN(C(=O)C=Cc3nccs3)CCC12 C1(NC(c2coc(Cl)n2)=O)CC2CCC1N(C(c1ncc(F)cn1)=O)C2 C1(NC(C(Cc2ccccc2)OC)=O)CCCCCN(C(=O)C(F)=C(C)C)C1 N1(C(C(c2cccc(O)c2)C)=O)CC2CCC(C1)N2C(C1CCC2(CCC2)C1)=O c1(C(N2CCC(CN(C(=O)CN(S(C)(=O)=O)C)C)C2)=O)c(O)nnc2c1CCC2 Cc1c(CNC(C2CC(C)N2C(=O)CCCCN(C)C)=O)cccc1O C#CCCCCCC(=O)NC1(C)CCC(C(=O)NOCC(C)O)CC1 C1(C)(C(=O)NC2CCCCN(C(c3c(CC)non3)=O)C2)CC2(CC(O)C2)C1 C1(NC(c2cnc(C(C)C)[nH]2)=O)CCCC(NC(=O)C(F)(F)c2ccnn2C)C1 CC(C)(C)C(O)C(N)C(=O)N1CCCC(N2CCNCC2=O)C1 C(CC(CC)C(=O)N1CC(CF)(NC(=O)C(C)CO)C1)=CC N1(C(C2C(O)CCN2C(C2CC2c2ccc(F)cc2)=O)=O)CC2CCCCC2C1 C12(Nc3nc(CC)cc(CC)n3)CCCC1CN(C(C1(COC)CC=CC1)=O)C2 c1(C(N(C(c2ccccc2)CC)CC)=O)cc(Br)cc([N+](=O)[O-])c1C c1(NC(C2N(C(Cn3ccc(C)n3)=O)CC(F)C2)=O)c(O)ncnc1O C1(C(=O)OC2CCC(OC)C2)CC(C)N(C(=O)OC(C)(C)C)C(C(F)(F)F)C1 C1(NC(C2OCCN(C(CCCOCCC)=O)C2)=O)CCCCC1C#N c1(C(N2CC(CNC(=O)CCCc3nccs3)C3C2C3)=O)ccc(O)c(Cl)n1 C(CCSC)(C(=O)NC(C)CCC=C)NC(CCC#C)=O c1(C2(C(N3CC(NC(=O)CC45CCCC4C5)C3)=O)CC2)cccnc1Cl C1(CNC(c2c(CC)c[nH]n2)=O)C2CN(C(=O)CC3CCC(=O)CC3)CC12 S(=O)(=O)(c1cc(Cl)c([N+](=O)[O-])cc1F)NC(c1cccc(NS(C)(=O)=O)c1)C CC(C)S(=O)(=O)CC(=O)N1CC(F)(CNC(=O)CC2CCCCC2(F)F)C1 CCC(Cc1cccc(C)c1)C(=O)NC(CNC(c1c(C)[nH][nH]c1=N)=O)CO N1(C(C=CC(=O)OCC)=O)CCCC(C(=O)NCCC(=O)Nc2ccccc2)C1 C1(CNC(CN(CCC#C)C)=O)CN(C(=O)C(O)CCSC)CC1F c1(C(C)=O)cc([N+](=O)[O-])ccc1C(=O)NC(C)CNCc1ccc(CO)cc1F C(=O)(C(F)CC(C)(C)C)N1C(C(C)C)CN(C(=O)C(C)n2cccn2)CC1 N1(C(c2c[nH]c(=NC)o2)=O)CCCC1C1CCCN1C(=O)CN1CCCCC1 C1(C(N(CCCC=C)C)=O)CCC(O)CN1C(c1cnc(=N)[nH]c1)=O C1(C)(C(=O)NCCn2ncc(CC)c2)CCCN1C(c1ccsc1C#N)=O CC1CC(NC(=O)C2=CCCCO2)CN(C(c2cc(=N)[nH]cc2Br)=O)C1 c1(NC(C2C(Nc3cc(C)ncn3)C2)=O)nc(C)c(C)cc1Br N1(CCCOCC)CC2CN(C(c3cnn(C4CCC4)c3)=O)CC2C1 N1(C(C2C(CCC)C2)=O)CC(N(C(=O)CCOCc2ccccc2)C)C(O)C1 C1(NC(CS(=O)(=O)NCC)=O)CC2(CCN(C(=O)C(C)=O)C2)C1.C(=O)C(C)SCC C(C(CC(=O)NC1CCN(C(c2ccc3oncc3c2)=O)C1)C(F)(F)F)N(C)C c1(C(N)=O)ccc(C(=O)NC2CC(NC(C3CCCC3c3nc(S)n[nH]3)=O)C2)o1 C=CCC(C(=O)NCC=C(C)C)NC(=O)OC(C)(C)C.C1(=O)C(COC)O1 C1(N(C)C(C2COCCO2)=O)CCC(NC(c2sccc2C#N)=O)CC1 N1(C(c2ccc(=O)oc2)=O)CCC2CCN(C(n3nnc4ccccc34)=O)C2C1 N1(C(c2cc(C(=O)NCC)no2)=O)CCC(C)N(C(=O)COc2cn[nH]c2)CC1 c1(CC(C)NCC(c2cccc(C)c2)OC)c(F)cccc1Cl C1(C(=O)NC2C3(CC(NC(C(CN(C)C)(C)C)=O)C3)C2)CCC(N=[N+]=[N-])CC1 C1(C(=O)NC2CSC2)(C(C2CC2)NC(C2C(Cc3cnccn3)C2)=O)CCCC1 Cc1nc(O)ccc1C(=O)NCCN(CCCN(C)C)C(=O)Cc1cc[nH]n1 C1(CC(N2CC(NC(c3nc(C)oc3)=O)C(C)C2)=O)OCCCC1(C)C O=S(=O)(NCC1CNC1)N1CCC2(CCCCC2)CC1 C1(CN(C)C(c2cc(CCCO)on2)=O)CCCN1C(c1ccc(C(N)=O)[nH]1)=O c1(NC(C23C(CN(C(C4(Br)CC4)=O)C2)C3)=O)cc(Cl)ccc1[N+](=O)[O-] N1(C(C2C(C)(C)COC2)=O)CC2(C=C(C(=O)NC34CCC(CC3)C4)CO2)C1 C(=O)(CCCC(=O)NC1CC(F)(CNC(C2CCC3(CCC3)C2)=O)C1)OC N1(CC=CCCC)CC(Nc2cnc(-c3cccc(C(=O)OC)c3)nc2)C(C)C1 c1(CC)cc(C(=O)NCc2nc(C(=O)NCC34CCCCC3C4)cs2)ccn1 N1(C(C=C(C)C)=O)CCOC2CN(C(=O)C=Cc3ccco3)CC12 Cc1ccc2nc(SCC(N3CC(CNC(=O)CC4CCCCO4)C3)=O)[nH]c2c1 C1(N(C)CCc2ccc(Cl)s2)CCCN(c2ccnc(N(C)CCS(C)(=O)=O)n2)C1 Cc1cc2nccnc2cc1C(=O)NC(C)CCNC(C1CC2(CCC2)C1)=O C=CC1(C(N2CC(OC)CC2CNC(C2COCCO2)=O)=O)CCCCC1 Cc1cnc(N(C2CCCNCC2)C(c2ccc(CO)o2)=O)nc1 CCCCC(O)CC(=O)N1CCOC(CCNC(c2ncc([N+](=O)[O-])n2C)=O)C1 c1(OC)ccnc(CNC(c2cn(CCNC(C3CC4C=CC3O4)=O)cn2)=O)n1 NS(=O)(=O)c1ccc(NC(C2CC23CCN(S(=O)(=O)C(Cl)(Cl)Cl)C3)=O)c(Cl)c1 c1(CC)cc(C(=O)NC2CN(C(=O)CCc3cncs3)C2)no1 N(C1CCCOc2ccc(F)cc21)S(C1=NOC(C(=O)O)C1)(=O)=O C1(NC(c2nc(OC)c(C)s2)=O)CN(C(C2(C#N)CC=CC2)=O)CCC1C c1(C(N(C2CCN(c3cc(CC)cnn3)C2)CCC)=O)ccc2c(c1)OCO2 CC1CC(C)(NC(=O)C=CCN(C)C(C2CNC(=O)N2)=O)C1 c1(OC)ccc(Cl)cc1C(=O)NCCC1CC(NC(C2CC23CCCOC3)=O)C1 C1(C(=O)OC)(CNC(C23CCCC2C3(F)F)c2ccccc2)CCC(OC)CC1 C1(C(=O)NCCN(C)C(C2(C)CC3CC3C2)=O)CCCC1C1CC1 c1(C(C(=O)NCCCC)N(CCc2cccs2)C(C)C)scnc1Br c1(C(=O)NCC2N(C(C3C(CC)C3)=O)CC(O)C2)cc(Br)ccc1OC Cc1ccccc1C(c1nnnn1C)NC(c1cccc(Br)c1)C1CCCCC1 N1(c2nnc(CCO)n2CC2(Sc3ccccc3)CCC2)CCSC2CCC12 C(=O)(CCC(CF)CF)N(CC(=O)NCCC1CCOCC1)CC#C C(=O)(CCCC(F)(F)F)N1CC(C)C(CNC(c2nc(Cl)cc(N)c2Cl)=O)C1 c1(-c2ccc(CCc3onc(C(CC)(O)CC)n3)s2)cn2ccsc2n1 c1(COC2CN(C(c3cnc(-c4ccccn4)s3)=O)C2)cccnc1 c1(C(=O)NCC(C)CNC(C2CC3OC2C2CC32)=O)onc2ccccc12 C(=O)(C1=CC2C=CC1C2)N1CC(C2(NC(c3cc[nH]n3)=O)CC2)C1 C#CC1CN(C(=O)CN(C)C2CC2)CCN1C(c1ccc(OC)nc1)=O c1(C(N2CCC(C)C(NC(=O)CSc3nnnn3C)C2)=O)ccc2nccn2c1 c1(C(N2CCOCC2)N(C(C(=O)NCCC(C)SC)=O)C)cc2ccccc2o1 CC(C(C)(O)C(=O)N1CC(O)(CNC(=O)CN(C)C)C1)c1ccccc1 N1(C(c2cnc(C(C)O)s2)=O)CC2(C1)CN(C(=O)CC1NC(=O)NC1=O)CCO2 C1(NC(C(C)NC(CC)=O)=O)CC12CC(NC(c1cnn(C3COC3)c1)=O)C2 c1(C(=O)NCC(C(N2CCC(O)(COC)C2)=O)C)nc(C)ccc1F N1(C(C2C(OC(C)(C)C)C2)=O)CC2(C1)CN(C(=O)C1=CCCOC1)C2 c1(C(N2CC(=C)C2)=O)oc(CNC(c2ccc(CO)s2)=O)cc1C N1(C(C(C)SC(C)C)=O)CCC(F)(CNC(=O)C=Cc2ccc(C(N)=O)o2)C1 N1(C(CC2(C=C)CC2)=O)CCN(C(=O)C(n2cc(C)cn2)C)C(CC(F)(F)F)C1 c1(NCc2c(CC)nco2)nccc(=NC(C)c2ncc(C)s2)[nH]1 N1(C(C(=O)NC2CC(N(C(c3ncc(OC)cn3)=O)C)C2)C)CCP(C)(=O)CC1 C(c1ccc(N(C)C)cc1)=CC(N1CC(O)(CN(C(c2scc(C)c2)=O)C)C1)=O C1(C)(NC(C(COCC)C)=O)CCN(C(C2CCCS2)=O)CC1 N1(C(C2C(C(N)=O)COC2)=O)CC2(CC(NC(C3CC(F)C(=O)N3)=O)CO2)C1 C1(NC(c2cc(COC)on2)=O)CN(C(=O)CC2CC3(CCC3)C2)C2CCCC12 C1(C(=O)NC2C3C=CC(C3)C2CO)CC2CCC(C1)N2C(=O)C1=CCCCO1 C1(C(CNC(CCOC(C)C)=O)C)CCN(C(=O)C(C2(O)CCCC2)F)CC1 c1(C(=O)NCC(=O)NCC(=O)N(C(C)CO)C)ccc(C#N)o1 N1(C(Cn2cc(C(C)OCC)nn2)=O)CC2CN(S(C)(=O)=O)CC2C1 C(C1c2ccccc2CCN1C(C1(OC)CC1)=O)NC(C1CCC(CC)O1)=O c1(C(=O)NC2CC(C)CN(C(=O)C(F)CC3CCCC3)C2)ccc(N=[N+]=[N-])cc1 C1(O)(C(N(C2CN(C3CC3)C2)C)=O)CCN(C(=O)C(C)C#N)CC1 Cc1nc(O)ccc1C(N1CCC1C(=O)NC1(c2ccccc2)CC1(C)C)=O C1(C(N2CC(OC)(CNC(=O)CCN(C)C(C)=O)C2)=O)CCN2CCOCC12 C1(C(N2C(C(CC)C)CCC2)=O)CN(C(=O)CC(C)O)CC1(F)F NS(=O)(=O)c1cc(C(=O)NCCCCNC(=O)C=CC2CCCC2)c(Cl)o1 N1(C(C(C)C2CCCC2)=O)CC(CC(N2CCC(C(C)(C)C)CC2)=O)C2(CC2)C1 Cn1cc(C(N2CCN(C(=O)C(C)(F)F)C3CCC23)=O)c2cccc(Cl)c12 c1(CC(=O)NC2CCN(C(CC(CC)CN(C)C)=O)C2C)ccn2cncc2c1 C1(=CC(=O)NC2(C)CCN(C(C(Br)=C(C)C)=O)C2)CCCCCC1(F)F C(C(C(C)C)NC(C1CCN(C(=O)Cn2ccc(C3CC3)n2)C1)=O)OC N1(C(CC(CCC)C)=O)CCOC2(C1)CN(C(=O)C1=C(C)OCCS1)C2 C(=O)(C1Cc2ccccc21)N(C(C)CNC(c1c(C)nc2sc(C)cn12)=O)CC CC(C)C(O)C(F)(F)C(=O)NCCC1(CNC(=O)C(c2ccccc2)C)CC1 C(=O)(C(C)CC(F)(F)F)NCC1(NC(C=Cc2c(C)n[nH]c2)=O)CCCC1 C1(CNC(C=CCCC)=O)CCC(C)CN1C(=O)C(C)=C1CC1 C1(CNC(C2CC(=C)C2)=O)CCCC(NC(=O)CCCc2ccc(Cl)cc2)C1 N1(C(c2c(C)ncs2)=O)CC(F)(F)CC1CNC(=O)C(C)S(N)(=O)=O n1(CC(N2CC(NC(=O)CC3CCC(O)C3)C(O)C2)=O)cnc2c1CCCC2 CC(O)(C(=O)NC1COCC1CNC(C1(CO)CCC1)=O)C(F)(F)F c1(C(C)C)nc2cc(NC(C3(C)COCCO3)=O)ccc2o1 c1(CCC(=O)NCC2CCN(C(C3CC34CC(F)(F)C4)=O)C2)ccc(F)c(F)c1 C1(C)(NC(C(CCC)O)=O)CCCN(C(=O)CCCOc2ccc(C)cc2)C1 C(CNC(c1ccc[nH]1)=O)(CC(F)(F)F)NC(C(C(C)C)n1ccnc1)=O C1(=CCNC(CC2CC(SC)C2)=O)CCN(C(C2CCC(C)C2)=O)CC1 Cc1nc(C)n(CC(=O)NCCC2(O)CCN(C(C3(C#N)CCCO3)=O)C2)n1 C12(NC(C3CC(=C)C3)=O)CCN(C(=O)Cc3cccc(OCCCC)c3)CC1C2 N1(C(c2cncc(C#C)c2)=O)CC2=C(C1)CN(C(C1(C)CC1Br)=O)C2 c1(C(c2n(C(CC)C)nnn2)NCC2(S(C)(=O)=O)CC2)ccc(C)cc1Cl c1(C(=O)NC2(C)CCC(NC(C(C=C=C)C)=O)CC2)cccc2cnsc12 C1(CNC(C2(C(C)=O)CC2)=O)CC2(CCN(C(c3cccn3C)=O)C2)CO1 Cc1ccc([N+](=O)[O-])cc1C(=O)NCC(CO)NC(=O)C(C)SC(F)(F)F C(=O)(CC(C)C(F)(F)C(F)(F)F)N(CCCNC(C(CC(C)C)OC)=O)C1CC1 c1(CC)nn(C)cc1C(=O)NC1CCC(C(=O)NCCC2CCCC(C)C2)C1 N1(C(C=Cc2cc(OC)ns2)=O)CCCC(C)(CNC(=O)CCC(C)(C)F)C1 c1(-c2cn(CC(C)NC(=O)CC3CCOC3=O)nn2)ccc2ncsc2c1 CC(CCCC(=O)NCCCCC1CC1C)NC(=O)Cc1cc[nH]c1 c1(C(=O)NC(COC)CNC(=O)CC2C(C)C2(F)F)ccc(C)cc1 c1(OC)ccc(CCC(=O)N(CC(C)O)CCNC(c2occc2C)=O)c(F)c1 Cn1cnc2c(N3CCCC(C(N4CCc5ccccc54)=O)C3)nc(Cl)nc12 C1(C)(C(=O)NCCN(C(C(C)OCc2c(C)cccc2)=O)C)CCC12CCC2 c1(CCC(N2C3C(NC(C=C(C)C)=O)C(C3)C2)=O)cc(Br)ccc1C C(=O)(CCC(C)(C)F)NCC(c1ccc(N(C)C)cc1)NC(C1C(C)C1)=O C1(C(CN2CCCC2(C)NC(C)=O)OCC)CCC(F)(F)CC1 C1(C(=O)NCC(C)CNC(C2COC2)=O)CCC(F)(F)CC1 C=CC(CC)C(=O)NC1CC(CNC(C2(CCC)CCC2)=O)CC1O C(=O)(C(CCC1CC1)NC(C1C=CCS1)=O)NC1(C)CC(O)C1 Cc1cncnc1C(=O)NC1CCC1C(=O)NCC(C)(C)C(N)=O c1(C(=O)OCC2C(=O)O2)cc(C)n(C2CC2)c1C.C(CC)OC C1(NC(Cc2onc(C)n2)=O)CCN(C2CCN(C(=O)C(F)CC3CC3)C2)CC1 CC(C(=O)N1CC(CCNC(C2(Cl)CC2)=O)C1)N(C)C Cc1c(C(=O)N(C2CCCN(C(=O)C3=CCCO3)CC2)C)cncc1Cl CC1=C(CNC(=NCCCCl)NCC2(C)CCCC2(F)F)S(=O)(=O)CCO1 C1(n2c(CC(N)=O)ncc2)CCC(F)(F)CC1.c12cccc(c1)c1nc2no1 c1(C(=O)NCCN(C(Cc2scc(C)c2)=O)CC(C)O)cc(C(F)F)nn1C c1(C(=O)NCC2CCCC(NC(CCCOCC)=O)C2)cc2cccc(F)c2o1 N1(C(c2c(OC)cncc2)=O)CCN(C(=O)CCC(F)(F)F)C(CC(C)(C)C)C1 c1(C(N2CCC(O)(CNC(C(CC)SC)=O)C2)=O)ccc2ncc(=O)[nH]c2c1 C1(CNC(C2(CCC)CCNC2=O)=O)CN(C)CCN1C(=O)Cc1nc[nH]n1 N1(C(c2c(CNC(C=CC(=O)N(C)C)=O)nnn2C)=O)CCCC(N=[N+]=[N-])C1 c1(C(=O)OC(C)C=O)c[nH]c2ccc(Br)cc2c1=N.CCCC(O)C(=O)NC1CC1 N1(C(c2cc(CC(C)C)nn2C)=O)C2CCC1CN(C(C1C(C)(C)C1(F)F)=O)C2 CC1SCCC1N=c1nc(N(C)Cc2cn(C)cn2)c2c([nH]1)CCCCC2 c1(C(=O)OC)cc(C(=O)NCC(F)CNC(=O)CC2(C)CC2)cc([N+](=O)[O-])c1 C(CC(C(C)(C)C)NC(C1(c2ccccc2Cl)CC1)=O)N(C(CC(C)SC)=O)C C1(NC(C2=C(C)CCC2)=O)CCOC2(CCN(C(c3cc(CO)[nH]n3)=O)CC2)C1 N1(Cc2c(C)nc(C)s2)CCS(=O)(=O)C(CCNC(c2cc(C)n(C)n2)=O)C1 c1(CC(C(=O)NC(C(=O)OCC)CC2CC(F)(F)C2)C#N)ccc(C#N)cc1 C1(C(C(=O)NCC2(CO)CCCC2)F)CCN(C(c2ccoc2)=O)C1 CC1CCCC(C)N1C(=O)NCC.N12CC3(CCN3C1=O)C2.C(C)(C)C c1(OC)cc2nc(NC3CCCN(Cc4cccs4)C3)nc(O)c2cc1OC CCC(CC(F)(F)F)NC(=O)CC(CNC(=O)Cc1cnoc1)C1CCC1 c1(C(=O)NCC(C)(CC(C)C)NC(C(CC)F)=O)ccc2occc2n1 c1(C(=O)NCC2CN(C(c3nnn(C)n3)=O)CC2O)c(F)ccc(C#N)c1F c1(C2(C)COC2)cn(CCCC(=O)NC(C2CCC2)C2CC2)nn1 c1(C(N2CC(c3c(CNC(c4ccc(OC)s4)=O)nco3)C2)=O)cnnc(C)c1 C1(CN(C)C(c2cncc(C3CC3)c2)=O)COCCN1.C1(C=O)COCCN1C C1(CNC(Cc2c(C)noc2Cl)=O)CN(C(=O)CCC(C)N(C)C)CC1(C)C c1(CSCC(=O)NC2(COC)CN(C(C=NOC)=O)C2)ccc(Cl)cc1 N1(C(c2ccc3cncn3c2)=O)CC2C=CCC(C2)C1.C1(CC)CN2CC1C2=O N1(C(c2c(CC(=O)OC)scc2)=O)CC2CCN(C(=O)CCC(C)N(C)C)C2C1 CCC(CCOC)C(=O)N1CCC(C(=O)NC(c2cncnc2)C)(CF)C1 Cc1ccc(CNC2CCN(Cc3cn(C)nc3C(F)F)C2)c(Cl)c1 C1(NC(CCc2ccc(CC)cc2)=O)CCN(C(C2CC23CC3)=O)CC1F C12(C(=O)NCC3(F)CCN(C(=O)COc4ccsn4)CC3)CCCCN1CCC2 Cc1oc(C2CC2)nc1C(=O)NC1(CCO)CN(C(C2(F)CCOC2)=O)C1 N1(C(C(n2cc(Cl)cn2)C)=O)CC2CCCC(C1)N2C(=O)C(C#N)CC1CC1 C1(CNC(C2CC(=O)OC2)=O)CN(C(C2(CF)CCOCC2)=O)CCO1 C1(NC(C2N(C(C)=O)CC(O)C2)=O)CCN(C(c2cccc(N)c2N)=O)CC1F CCC(CC(C)C)C(=O)N1CC(C(=O)NCC2CCC2CO)C(F)(F)C1 CCC(C)(CC)C(=O)N1CCOC(CNC(C2(C#N)CC3(CC3)C2)=O)C1 C(=O)(CC1=CCCCC1)NCC1C(CNC(c2c(C(C)C)noc2)=O)C1 CC(C)C(=O)C(=O)NC(c1ccccc1)CNC(C1CC(F)C1)=O CC1CCC(=CC(=O)NC2(CCNC(c3cn(CCN(C)C)nn3)=O)CC2)C1 Cc1ncc(C(=O)NC(C2(CNC(C3CC34CCSCC4)=O)CC2)C)c(C)n1 c1(OCC(=O)N(c2ccccc2O)CC)cc(O)ccc1OC C1(C)C(C)C(=O)N1C1CC1.c1(OCC)cc(C(=O)NCCC(C)C)on1 C1(N(C)C)CCCC(C(=O)OCN2CCCC2NC(=O)C(c2ccccc2)F)C1 CCCC(C)C(C)N=c1[nH]c(=NCc2cc(F)ccc2Cl)[nH]c2ncn(C)c12 C1(NC(N2C(c3c(OC)cccc3)CCCCC2)=O)CC2(CCC2)C12CCC2 Cc1nc(N2CCCC(CNC(c3ccno3)=O)CC2)c(C)c(Cl)n1 C=CCCCCCCCC(=O)NC1CN(C(=O)Cn2ncn(C)c2=O)C(C)(C)C1 N1(C(c2c(C)nccn2)=O)CCCC2(NC(c3nc(Cl)ccc3F)=O)CC2C1 N1(C(C=CC(C)NC(=O)C2=C(Cl)CCOC2)=O)C2CCCC1CN(C)C2 c1(CCNC(=O)C=Cc2cccs2)ccc(-c2cn(CCC(F)(F)Cl)nn2)cc1 c1(-n2c(CCC(CC)C)nc(CN3CCC(O)CC3)n2)ccc(F)cc1CO C=CCN(OC)C(=O)C(F)CC(C)(C)NC(c1ncccc1Cl)=O CCC(C)(COC)CNC(=O)COC(C)(C)CNC(=O)CCCCSC C1(F)(C(=O)NCC(O)Cn2cccn2)CCCN(C(c2cc3n(n2)CCC3)=O)C1 N1(C(CC(C=C)CC)=O)CC(C)CN(C(c2cnn(CC)c2)=O)CC1C Cc1ccc2ncc(C(=O)NC(C)C(C)NC(c3cnc(N)c(Cl)c3)=O)cc2c1 CCCC(CNC(C1CC1C1CC1)=O)C(=O)NC(C(C)C)C(C)C Cc1nn(CC(F)F)cc1C(=O)NC1CCC1NC(C1(O)CCC1)=O c1(C(=O)NC(CCNC(c2nc(C)oc2)=O)C)cc(S(N)(=O)=O)co1 CC1C(NC(=O)C2=CCC2)CCN1C(c1cc(C(F)(F)F)cs1)=O C1(NC(CC(CCC)C)=O)CC(C(=O)NCCCc2ccccn2)=CC1O c1(C(N2CC(C)(CCC(N3C(C(N)=O)CC3)=O)C2)=O)cc2ccccc2[nH]1 N1(c2ncnc(C)c2Br)CCC2CCC(C1)N2C(C1CCOCC1(C)C)=O C1(N(C(C=CCCC)=O)C)CN(C(c2sccc2CO)=O)CC1O c1(N(C)C)ccc(C(=O)NCC2(CCNC(=O)C(C)(C)C3CCC3)CC2)cc1F c1(CC)nnc2cc(N3CCC(NC(c4ccnc(C)n4)=O)CC3C)ncn12 C1(c2cn(C)nc2)CN(C(c2cc(C(N)=O)co2)=O)CCN1C(=O)CCC1CC1 N1(C(CN(C(C)=O)C)=O)CCC(C2CC2)(NC(=O)CN2CCN(C3CC3)C2=O)C1 n1(CCOC)nc(C(N2CC(N(C(=O)Cc3nc[nH]n3)C)C(F)C2)=O)ccc1=O N1(C(=O)NC2C(C(C)(C)C)C2)CCC2CC(O)CCC2C1 c1(C(C(=O)NCC=C)N(C)Cc2ccc(NC(C)=O)cc2)ccc(Cl)cn1 O=C(O)C1CCCc2nc(C(=O)NC(c3ncco3)Cc3ccccc3)cn21 C1(C(N(CC=C)C)=O)C2CC(O)C(C2)N1C(C1CC2CCCC2C1)=O C1(NC(c2cc(CC)no2)=O)CC(NC(C2(COC)CC(F)(F)C2)=O)C12CCC2 CC(C(F)(F)C(F)(F)F)=CC(=O)NCCCN1CCN(C(C2CCO2)=O)CC1 C1(C(=O)NCC2(COC)CCC2)CN(C(c2c[nH]nc2C)=O)CCO1 C(CN=c1[nH]ncs1)NC(CNC(CS(=O)(=O)N(C)C)=O)=O Cc1ccc(NC(=O)CC2CC(F)CN2C(=O)C(=O)C(C)C)c(F)c1F N1(C(CC#N)=O)CCC2(CC1)CC(NCc1cccc3c1CCCC3)C2 CCCC(C)(C)CC(=O)N1CC(NC(=O)C(C2CCC2)C2CCC2)CCC(O)C1 C1(Sc2ccc(C(=O)NC(CC=C)CNC(=O)CSC)nc2)OCC2CCCC12 CC1=C(C(=O)NC2(CC(=O)NCC(C)N(C)C)CCCCC2)CCC1 C=CCCCC(C(=O)NCC(C1CCCCC1)O)NC(C1CC(=O)N(C)C1)=O N1(C(c2cnc(CC)s2)=O)CCN(C(c2cc(C3CC3C)on2)=O)C(CCO)C1 C1(O)(CC)CCCN(C(C2(NC(=O)C=CCCC(C)C)CCSC2)=O)C1 C(=O)(CCC=CBr)N(CCC)CCNC(=O)Cn1ccc(C(F)F)n1 c1(C(=O)NCC(CO)NC(CNC(C)=O)=O)cc2c(ccn2C)s1 C1(CC(=O)NCC2CCN(CP(C)(C)=O)C2)Oc2ccccc2NC1=O C1(C#N)(NC(CCCC#C)=O)CCN(C(=O)Nc2cc(F)ccc2C)C1 C=CC1(C2(C(=O)NCC3CCN(C(c4c(C)cnn4C)=O)C3)CCC2)CCC1 CCCC(CCC)=CC(=O)NC1(CF)CCN(C(=O)C(C)(C)C2CCO2)C1 c1(C(=O)NC2CCN(C(C(C)S(C)(=O)=O)=O)CC2F)nc2ccccc2[nH]1 c1(C(N2CC(CNC(=O)CN3CSCCSC3)C2)=O)cccc2occc12 C1(C(N(C2C3CN(C(=O)CCC(F)(F)F)CC23)C)=O)CC2(C1)CC2(F)F N1(C(C(C)SC)=O)CCOC(CNC(=O)CC(c2c(C)n[nH]c2C)C)C1 c1(-c2cn(CC3CN(C(CN(C)C(N)=O)=O)C3)nn2)ccn(C)c(=O)c1 c1cc2c(C3CN(CCS)CCO3)[nH]nc2cn1 N1(C(CC2(C)CC2(Cl)Cl)=O)CC2CCC2(CNC(C2(C(N)=O)CC2)=O)C1 C(CCCCCC(=O)NC(c1ccccn1)CO)NC(c1ccc(SC)o1)=O c1(C(=O)NCC2(F)CC(NC(CC(C)C)=O)C2)cccc(C(C)C)c1F C(=O)(C(C)(C)CCS(C)(=O)=O)N(CCCN(C(C(=C(C)C1CC1)F)=O)C)C c1(OC)ccc(C=CC(=O)N(C2CCN(C(C3CC(SC)C3)=O)C2)C)c(OC)c1 CN(CC(=O)c1cccnc1)N1CCN(C(C2C3CCCC23)=O)CC1 N(C1CCCc2occc21)C(C1(n2cnnn2)CCOCC1)=O C(=O)(C(F)(F)CCNc1ccccc1)NCCC(C)NC(CSCC(C)C)=O c1(C(N2C(C)C(C(=O)NCC(C)(O)CCO)CCC2)=O)ccc2ccoc2c1 n1(C(N(CC2N(C(=O)NC3CC(C)(CC)C3)CCCC2)O)=O)ncc(O)nc1=O c1(C(C(=O)NC(CNC(C2(CC(=O)OC)CC2)=O)CO)C)ccc(Br)s1 c1(CC(=O)NCC(CC)NC(c2ccc[n+]([O-])c2)=O)nccc2ccccc12 CC(=NO)C1CC(C(=O)NCC2CCCN2C(=O)C=C2CCSCC2)C1(C)C C1(C(F)F)(OCCOC)CCN(CSCc2ccn(C3CCCC3)n2)CC1 C1(NC(CCN(C(CCC)C)C)=O)CC2(CCN(C(C3COCCO3)=O)C2)C1 C(=O)(CS(=O)(=O)N1CCN(C2COCC2c2ccccc2)CC1)OCC C12(C(N3CC(CNC(=O)CCc4ccsc4)C(O)C3)=O)CCC(CC1F)C2 N1(C(c2cc(Br)ccc2C)C(=O)NCCOC)CCC(F)(F)CC1C C#CCC(CC(=O)NC(C)CCC(=C)C)NC(C1(OC)CCC(C)C1)=O C(=O)(C#CC1CCCO1)N1CC(O)CC(NC(c2cc(=O)cc[nH]2)=O)C1 Cc1nc(O)ccc1C(=O)NCC(CNC(c1ccc(C(C)C)c(F)c1)=O)CO c1(C(=O)NC2CC3(C(C(N4CC(COC)OCC4)=O)C3)C2)ccc(C)c(C)n1 C1(C)(C(=O)NCC(C)(C(C)C)NC(CCc2c(C)nccc2)=O)CCC(=O)NC1 C1(C(=O)NCC2(NC(COC(CC)(C)C)=O)CCOC2)CCCC(N(C)C)C1 C12CCCCN1C(=O)C(=O)NCCC2.c1(C(=O)NCC2CC2)nocc1Cl CC1(C)CCC(CNC(=O)CC2CCCCN2C(=O)COC2CCOC2)CC1 c1(CC(C)C)n[nH]c(=NCCC2CCN(C(=O)C(c3cc(F)cc(F)c3)O)C2)s1 C1(NC(c2n(C)ncc2Cl)=O)CCN(C(c2ncc(Br)cn2)=O)C12CC2 C(CC(C)C(=O)NCC1CC(O)CN1C(c1[nH]c(O)nc1C)=O)=CC C(=O)(C(C)C(C)NC(CC=CC)=O)NC(=O)CN(CC(=O)NCC1CCCC1)C c1(N(CC(CN(C(c2c(C)noc2C)=O)C)O)C)cc(Cl)nc(C(F)(F)F)n1 c1(CNC(C2C(NC(C(CCC)O)=O)CCC2)=O)ccc(OC)cc1Br CC(C)(C)CC(O)CC(=O)NC1CC(C)(NC(=O)C=CCOCc2ccccc2)C1 C12(NC(c3ccc(C)s3)=O)CCC(CN(C(c3csc(C)c3C)=O)C1)C2 CC1OCC2(CCN(C(=O)Cc3ncccn3)CC2)C1N1CCOC(CO)C1 Cc1nn(C(C)C)c(C)c1COC(=O)C(C)SC1CC1.C1C(=O)N(S(C)(=O)=O)C1 N1(C(CCNCCCCC)=O)CC2CCN(C(=O)CN(C)CCOC(C)=O)CC12 c1(C(=O)NC2C(NC(c3c(C)nsc3)=O)CC2)cccc(-c2nnco2)c1 C(C(C(=O)OC(C)(C)C)NC(=O)CC=CCNC(C1CC1[N+](=O)[O-])=O)N(C)C C1(C(=O)NC2C=CCN(C(c3nc(COC)sc3)=O)C2)Cc2ccncc2C1 C12(C(N(C(CC#C)C)C)=O)CCCC1CN(C(=O)C(C)(C)C#N)C2 c1(OC)cc(Br)ccc1CC(=O)NC1C=CC(C(=O)Nc2ccc(Cl)cc2O)C1 C1(F)(CNC(C2(C)CC(=C)C2)=O)COCCN(C(C2CN3CCCN2CC3)=O)C1 c1(CO)cncc(-c2nc(CSc3ccccc3)nn2C2CCSCC2)n1 C12(C(N3CC(N(C)C(C4CCCCC4F)=O)C3)=O)CC(CO)(C1)OC21CCC1 C1(CNC(C2COC2)=O)CC2CCC1N(C(c1ncnc(O)c1Cl)=O)C2 c1(CC)ccc(C(=O)NCc2c(C)sc(C)c2Br)c(Br)c1 Cc1ccc(NC(=O)C(C)(O)C(F)(F)F)c2[nH]ncc12 Cc1nn(C)c(C)c1CC(=O)NCC1(C)CCC(NC(=O)C(O)C2CCC2)CC1 Cc1ccc(C=CC(N2CC(NC(C3CCC(=O)C3)=O)C2)=O)cc1Cl c1(C(=O)NC(C2CCN(C(C3CCCC3O)=O)CC2)C)snc2ccccc12 C(C1=NOC2CN(C(c3nnc(O)cc3O)=O)CC12)NC(C1(SC)CC1)=O c1(CNC(C2CCN2C(=O)C(c2ccc(Cl)cc2)O)=O)c(F)ccc(F)c1F Cc1c(NC(c2c[nH]nc2CCNC(=O)C(C(C)O)N(C)C)=O)cnn1C c1(CC(N2CCC(NC(C(CC)n3cncn3)=O)(CO)C2)=O)c(F)cccc1Cl C1(CNC(CCC)CC)CCC(F)(CC(=O)OC(C)(C)C)C1 C1(CC(C)NC(C2COC(C)(C)C2)=O)CCN(C(=O)CC(C)n2cccn2)CC1 C1(C(=O)NCC(N)=O)COCCN(C(=O)C(c2cc(C(F)(F)F)c(O)nn2)=O)C1 c1(NCCC2N(C(=O)C=CBr)CCC2)ccnc2ncnn12 N1(C(COC2(C)CCC2)=O)CCC(CCNC(C2OCC2(C)C)=O)CC1 C1(NC(c2nncc(C)c2)=O)CCC2CN(C(=O)CCc3cnn[nH]3)CC2C1 C1(C(=O)NCC2(CNC(c3ccc(C#C)o3)=O)CCOCC2)CC(=O)NC1(C)C N1(C(CNS(C)(=O)=O)=O)CCC(N2CCC(NC(=O)CCC(F)F)CC2)CC1 N1(CC(=O)NC2CCC(NC(C3(CC)CC3)=O)C2)CCC(=O)NC1=O C(=O)(C1=CS(=O)(=O)CCC1)NCC(C)NC(C1(n2cccn2)CCC1)=O C1(CNC(CC(C)(C)OC)=O)CN(C(c2ccc(C)nc2O)=O)C2CCN1C2 c1(-c2c(C)cc(C#N)cc2)ccc2c(C(=O)N(C)CCN(C)C)nsc2c1 C1(COC)CCC(NC(=O)C(=O)NCC2CN(Cc3ccccc3)C2)C1 CCC(C)C(O)C(=O)NCC1C2CN(C(=O)CC(F)(F)CC)CC12 C1(C(=O)NCCCN(C(=O)Cc2ccoc2)C)CC(c2cccc(Cl)c2F)=NO1 C1(C)(CNC(COCC)=O)CC(F)(F)CN1C(C1CCc2n[nH]cc2C1)=O c1(C(=O)NC2(C)CCCN(C(CNC(CC)=O)=O)C2)ccc(S(=O)(=O)CC)cc1 c1(C(N2CCC(C)(COC)C2)C(=O)NC(C)C(=O)OC)cc(Br)ccc1C C1(C(=O)NC2CCN(C3CC3)C2)(CNC(=O)CCOCC(F)(F)F)CC12CCC2 c1(C(=O)NC2(CC=C)CCN(C(C3CCC(=O)O3)=O)C2)cc2ccccc2cn1 Cc1cccn2cc(OC(N3CCC(NC(=O)NC(C)(C)C)C3C(C)C)=O)nc12 Cc1cc(C(=O)N(C2CC2)CC2CCCN2C(c2ccc(CO)o2)=O)nc(C)n1 c1(C(N2C(CC(=O)NCCCC3(O)CCC3)COCC2)=O)occ2c1CCC2 c1(N(CCNC(=O)Cc2ncsc2Br)CC)ccc(C(=O)OC)cc1 c1(C(N(C2CCCN(C(=O)CN(C3CCSC3)C)CC2)C)=O)cc(F)cc(F)c1 Cc1c(-c2cnc(CNC(c3ncnn3C)=O)nc2)cccc1F N1(C(C2N(CC)CC2)=O)CC(CCNC(=O)CC2CCC(C)(C)O2)C(C)C1 CCC(C)C(O)C(=O)NCc1nnn(C)c1C(=O)NC1(c2nc[nH]n2)CCC1 c1(C(N(C2C(C)CC2)C)=O)cnc(C2CC2)nc1.c1(C(C(=O)NC)SSC)cccnc1 c1(C(=O)NC2CCC(CNC(c3cc(Cl)c(Cl)[nH]3)=O)CC2)ccc2cccnn12 CS(=O)c1cccc(C(N2CC=C(CNC(C3(O)CC4CCC3C4)=O)CC2)=O)c1 C1(CC)CCN(C(=O)CC(C)C2CC2)C(C(=O)NC2CC(CCF)C2)C1 C1(CNC(c2ccn(CC)c2C)=O)CN(C(=O)CNC(=O)C(C)(C)C)CCC1C c1(CNC(CCCCC#C)=O)nnc2n1CCN(C(=O)C(O)CCCC)C2 C1(C(N(C2CCN(C(=O)CCc3nc(C)no3)C2)CCC)=O)CCCC1C(C)C c1(C(N(CCCCNC(C2CCCCC2(C)C)=O)C)=O)c(F)ccc(O)c1F N1(C(COC(CC)(C)C)=O)CCN(C(c2ccn(CCO)c(=O)c2)=O)CC1CO c1(C(=O)NCCC2CCCN(C(C(C)CN(C)C)=O)C2)cn(C)c(=O)n(C)c1=O N1(C(COCCCCC)=O)CC2CCC1CC2NC(c1cnncc1O)=O C#Cc1cn(C)nc1C(=O)N(C1CCCC(NC(c2cncs2)=O)C1)C CC(C)(C)C(O)CONC(=O)C1CC(NC(c2ncc(F)cn2)=O)C1 C(=O)(CC(C)(O)C(F)(F)F)N1CC(C(C)NC(c2ccccc2F)=O)OCC1 N1(C(C(C)n2ccnn2)=O)CCOCC(NC(=O)C(O)CC(N)=O)C1 C1(NC(c2nnc(CC)s2)=O)CCCN(C(=O)CCc2cc(C)[nH]n2)CC1 C1(NC(CN(C2CCC2)C)=O)CCOCC1NC(=O)CCn1cnccc1=O c1(CCC)nc(C)c(C(N2CC(F)CC2CNC(c2cnn(C(C)C)c2)=O)=O)s1 c1(CNC(c2nnnn2C2CCC2)(C)CC2CCCCO2)nocc1C1CC1 C1(CNC(C(c2cccnc2)NC(CCOCCCOC)=O)=O)CC(C#N)C1 C1(C(N2C(C)(C(C)C)CC2)=O)CCCCN(C(=O)C(C)S(C)(=O)=O)C1 N1(C(CCC#C)=O)CCC(C(N2CCC(c3cnco3)C2)=O)CC1(C)C c1(C(=O)NCC(CNC(c2cc(C)[nH]n2)=O)(C)C)ccc2c(n1)CCC(C)(C)C2 c1(C(=O)Nc2ccc(O)c(F)c2)cnc2ccncc2c1 c1(CC)ncccc1C(=O)NC1CCCC1C(=O)NC(C(F)(F)F)C1CC1 c12cccc(c1)CN(C)C(=O)CC1(CC1)NC2=O.C1(N(C)C)CCOCC1 N1(C(c2ccc(CCCCC)o2)=O)CCC(O)(C(C)CNC(C2(CO)CC2)=O)C1 C1(C2CCN(C(=O)C(O)C3CCC3)CC2)(NC(=O)CNc2ccccc2Cl)CC1 C=CCC(CC(=O)N1CC2CC2C2CC12)NC(=O)CC1CC(OCC)C1 C=CCC(C(=O)N1CC(NC(c2ccc(OC)cc2C)=O)C1)C(C)(C)C c1(CCC(=O)N(CC(N2CC(NC(CC)=O)C2)=O)C)ccccc1 N1(C(C(CC=CC)C)=O)CCC2CN(C(=O)C=Cc3ccco3)CC2CC1 c1(C(=O)OC)cccc(CN(CC(C2CCOC2)O)C)c1O C(CCCCC(=O)NC1CCCC(NC(C2(C)C=CCC2)=O)C1)OCC Cc1nc(C2CC2)ccc1C(N1CCOCC1CNC(=O)CC1CCC2CC12)=O c1(C(N2CCSC(C(N3CC4COCC4C3)=O)C2)=O)c[nH]c2nccc-2c1 c1(C(C)C)nccc(CNC(CCO)c2nccs2)n1 C1(NC(c2n[nH]c(C)c2O)=O)C2CC1CN(C(=O)Cc1cc(F)ccc1Br)C2 C1(C(=O)NC2CCN(C(c3c[nH]nc3C)=O)C2)(OC)CS(=O)(=O)C1 c1(N2C(C(=O)NC(CC)C(=O)OC)COCC2)ncnc2c1ncn2C C1(COC)CN(C(=O)CNC(C2CCSC2)=O)CCN1C(=O)Cc1nc[nH]n1 c1(OC)ccccc1C1(CNC(C2CCC(N3CCCC3)CC2)=O)CCC1 Cc1cccc(C(=O)NC2CN(C(=O)CC3SC(=N)NC3=O)CC2O)c1Cl C(CN=c1[nH]c(=N)[nH]c(=NCC(C)NC(=O)OC(C)(C)C)[nH]1)N(CC(C)C)C Cn1cc(C(=O)NCCN(C(C2C=CC=CC=C2)=O)C2CC2)c(-c2ccco2)n1 C1(C(=O)NC2(C)CCCN(C(=O)COCCF)C2)OCC2CCCC1C2 c1(C(=O)NCC(CNC(c2cc(C)nn2C)=O)O)nc(O)c2ccccc2c1C CC1(C)CCCN(c2ncccc2-c2ccccc2)C1C(N)=O C1(C(=O)NC2CC(N(C(=O)Cn3cnc(=N)[nH]3)C)C2)CN2CC3CC2(CO1)C3 CCC#CCN=c1nc(N2CCCC(N3CC(O)C3)C2)c2ccccc2[nH]1 Cc1cc(C(c2cccnc2)NC(=O)NC2CC3(C2)CC(CO)C3)cc(O)n1 N1(C(C2CN(C(c3c(OC)csc3)=O)CC(C)(C)C2)=O)CCCC2(CCCO2)C1 Cn1cc(C(F)(F)F)nc1C(N1CCC(C(C)(O)CNC(C2(O)CC2)=O)CC1)=O N1(C(C(C(C)C)NC(Cc2c(C)n[nH]c2C)=O)=O)CC2CCCCC2C1 S(=O)(=O)(c1ccc(F)cc1F)N(C)CCNC1CCC1(F)F c1(NC(=O)NC2CCC(CC34CC(C(=O)OC)(C3)C4)CC2)ccc([N+](=O)[O-])cc1 N1(C(=O)N(c2cccc(F)c2F)C2CCCO2)CCCc2cncc(Cl)c21 N1(C(c2csc(C)c2C)=O)CCCC2C(NC(=O)CCC(C)(C)F)C(C)(C)C12 CC1(C)CC1(C)C(=O)NCC1(CNC(c2cc(Br)n[nH]2)=O)CCC1 c1(CC(=O)N(C2CN3CCC2CC3)CCO)ccc(S(=O)(=O)N2CCOCC2)s1 N1(C(c2cc(CC)oc2C)=O)CCC(C(=O)NOCCC(C)O)CC1(C)C C(C(=O)N1CCC(F)(c2cn(C(C)C(=O)N(C)C)nn2)C1)(C(F)(F)F)OC(C)=O c1(C(=O)NCC=CCNC(c2c(CC)occ2)=O)nccc(Br)c1C C#CCC(C)(C(=O)NCCOCC(N)=O)N(C(=O)C(C)C1CC1)C1CC1 Cc1nn(C)c(C)c1COC(=O)C(O)Cn1cncn1 c1(Cn2c(C)cc(C)n2)c(Cl)cccc1Cl.c12cn(nn1)C(C)C(=O)N(C)C2 Nc1nc(Cl)ccc1C(N1CC2CC1C2NC(c1ccc(Br)o1)=O)=O Cc1ccc(C(=O)NC2CCCCC2C(=O)Nc2ncncc2F)nc1O C1(C(=O)NC2(CCOC)CCCC2)CC(C)(C)CN1C(C1CC1C(C)C)=O CC1CN(C(=O)CC2CCCC2NC(c2ccncn2)=O)CC(C)(C)O1 c1(C(=O)NC2CCN(C(CCC(C)C)=O)CC2O)cn2c(n1)CCC(C)C2 N1(C(C(C)OCC#C)=O)CCCC1CN(C)C(C1CCC(F)C1)=O C1(CNC(CNC(CCNC(C)=O)=O)=O)C2CCCC1N(C(=O)CSC(C)(C)C)C2 C1(C(=O)NC(C)C#N)CN(C(c2cc(F)c(F)cc2I)=O)CCC1(F)F C(=O)(C1CCCc2sccc21)NCCN1CCN(C(C2C(C)C2C)=O)CC1 Cc1cc2c[nH]nc2cc1C(=O)N(C1CC(NC(c2cnnn2C2CC2)=O)C1)C CCCC(O)(CCC)CC(=O)N1CCN(C(=O)C(C)NC(=O)NC)C(CCO)C1 CC(C)C(F)C(=O)NC(C1CN(C(c2cn[nH]c2)=O)CCO1)C n1(CC)nc(C(=O)NC2CC(O)C2CC(=O)NCc2cc(C)cs2)cc1O C12CCN(C(c3ccccc3)C1)C2=O.c1(NC(C=CCOC)=O)cnc[nH]c1=N C1(C(=O)NC(C)CN(c2cc(Cl)nc(C3(C)CC3)n2)C)CNC(=O)CC1C N1(CC(=O)NCC2CC(NC(C3(COC)CCC3)=O)C2)CCCNC1=O C1(NC(C2C(NC(Cn3c(C)nc(C)n3)=O)CCOC2)=O)CC2(C1)CN(C)C2 C(=O)(CC(C)C(F)(F)F)N1C(Cn2cc(CCCC=C)nn2)CC(C(C)C)CC1 CC(CC(F)(F)F)C(=O)N(CCCNC(=O)C(F)(F)C(C)(C)O)C Cc1c(C(=O)NCC23CCC(CC2)N3C(=O)C(O)C2CC2)c(C(F)(F)F)nn1C Cc1nc(Cl)ccc1CC(N1CCC(C(F)CNC(C2(C)CC2)=O)CC1)=O c1(CC)cc(C(=O)NCc2csc(CNC(C3CCC(OC)C3)=O)n2)nn1C N1(C(c2c(C(C)C)cco2)=O)CCC2(CC1)CC2NC(=O)CN1CC=CC1 C1(NC(C=CCOC)=O)CCN(C(=O)C2=CC(C)C2)CC1CO N1(C(CC2(C)CC2(F)F)=O)CCCC(C(=O)NCC(N2CCCCC2)=O)CC1 c1(NC(C)(C)CC(=O)N2CCCC2)ccc(S(C)(=O)=O)cn1 C(=O)(C1=CC(O)C(NC(=O)COC(C)(C)C)C1)NCCNS(CC)(=O)=O c1(C(C(=O)NCCCSC)N(C)CC2CC2(C)C)ccc(Br)c(C)c1 C=CC1CCC1C(=O)NCCC1CCN(C(c2ccn(CC(F)F)n2)=O)C1 c1(OC)ccc([N+](=O)[O-])c(C(N2CCC(NC(c3cnns3)=O)C(CO)C2)=O)c1 C12(NC(c3cn4cc(C)nc4s3)=O)CCOCC1CN(C(C1(C(F)F)CC1)=O)C2 C(=O)(CC(C)CC(C)C)NCCC(C)N(C(c1ccc(C#C)cc1)=O)C C1(NC(c2cnc(CC)s2)=O)(COC)CCN(C(C2(F)CC3(CCC3)C2)=O)CC1 CCCCCC(CC)C(=O)N1CCC2(C1)CN(C(=O)Cc1ccc(F)cc1Cl)C2 C12(CNC(c3ccns3)=O)CCCCC1N(C(c1ccc(F)nc1)=O)CC2 C#CCCCC(C)C(=O)NC(C1(C(=O)NC(C)CCOC)CC1)C C1(C(N2C(C)COCC2)=O)CCN(C(=O)C2CCC2C#N)O1 c1(CNC(C(C)C)=O)nnc2n1CCN(C(=O)Cc1ccc(Cl)cc1)C2 c1(C(=O)NCC2(NC(C3CCCN3C3CCCC3)=O)CC2)ccncc1Br c1(NC(C2CN(Cc3cc(B(O)O)co3)C2)=O)nc2cc(Cl)ccc2s1 C=CC(C)(O)CC(=O)N1CC(N(C(=O)CS(=O)(=O)N2CCCCC2)C)C(O)C1 Cc1cc(-c2cn(CCC(=O)NCC3OC(=O)NC3(C)C)nn2)cc(C)n1 C12(CC)CCC(C(N3CCC(CNC(c4ccncc4F)=O)(OC)C3)=O)(CO1)C2 C#Cc1ccc(NC(=O)Nc2n[nH]cc2C(=O)OC(=O)C2CC2)cc1 C(=O)(C(F)(F)C(F)(F)F)NCC1CCCC(NC(c2ccc(N(C)C)cn2)=O)C1 N1(C(C=COCC)=O)C2CCC1CN(C(=O)CC1CCC(=O)O1)C2 c1(OCCC)ccccc1CN1CC2C(C1)N2C(C1CCC(F)(F)C1)=O C1(C(=O)NCCCC(C)(C)O)CC2(CC2)CN1C(C1CC2(CCO1)CC2)=O C(=O)(CS(=O)(=O)C(C)C)N1C2(CNC(c3c(C)c(N)ccc3)=O)CCC2CC1 c1(C(N(CC(C)N(C)C(C2(C#N)CC2)=O)C)=O)ccc(Cl)c(Br)c1F C1(C(=O)NC(CC)CNC(c2cc(C)c(C)s2)=O)CCCN(S(N)(=O)=O)C1 CC1(CNC(C2CCC(=O)N2)=O)CCN(C(c2ccsc2N)=O)CC1 N1(C(C=CCC)=O)CCCCCC1CNC(c1c(Cl)cncc1Br)=O C1(NC(C)=O)COCCC1NC(c1ccc(-c2ccccn2)nc1)=O C1(NC(CNC(c2ccc(C)s2)=O)=O)CCOCC1NC(=O)Cc1cncnc1O C1(N(C(CN(CCC)C)=O)CC)CCN(C(=O)CCC)C1.C(C)(C)(C)OC(C)=O C#Cc1cccc(C(=O)NCCC(C)NC(C2CC3(C)CC2CO3)=O)c1 N1(C(C(F)OC)=O)CCN(C(c2csc(C(N)=O)n2)=O)C(CCO)C1 Cc1cnc(Cl)cc1NC(C1(C)CCN(Cc2ccc(F)c(O)c2)CC1)=O CC(CC(C)(C)O)N1CCC(CNC(C2(c3ccc(F)cc3)CCCC2)=O)C1 C(CCCC(=O)N1CCC(O)C1C(C)(C)C)N(C(C(C)SCC)=O)C C=CCCCCN=c1nc2ncn(C)c2c(NCC2(Cl)CC23CCC3)[nH]1 Cc1cc(C(=O)NC2(CNC(=O)CNC(=O)CC(F)(F)F)CC2)nc(O)n1 c1(C(=O)NCC2(NC(C(CCOC)C)=O)CCC2)ccc2[nH]c(=N)oc2c1 N1(C(C2CCCC(C)CC2)=O)CCCN(C(c2ncccc2N)=O)CCC1 C(=O)(C1=CCCCCC1)NCC1N(C(C2CC(C)OC(C)C2)=O)CC=C1 N1(C(C2C(CNC(C(C(C)C)OC)=O)CCC2)=O)CCC2(CC1)CN(C)C2 C=CC(CCC)CC(=O)N(C1CN(C(c2ccc3c(c2)COC3)=O)CC12CC2)C c1(C(=O)NC2CC3CN(C(C(CC)C)=O)CC(C2)C3)cnc(O)c([N+](=O)[O-])c1 CC(F)CN=c1nc2c(cnn2C)c(NCC2CCCC2N2CCCS2(=O)=O)[nH]1 C1(CC)CN(C)CCCN1C(C1CN(C(=O)C(Cl)Cl)C(C)(C)C1)=O C=CC1CCN(C(=O)CC2CC3(C2)CN(C(=O)Nc2cc(C)ccc2C)C3)CC1 CCC(CNC(=O)C(F)(F)c1ccsc1Cl)(CC)NC(=O)CSCCN(C)C C1(C(=O)NCC2C(C=C)C2)CCC(n2cc(-c3ccccn3)nn2)CC1 C1(C(=O)NCC(C)NC(C2CC(OC)C2)=O)CC12CCOc1ccc(F)cc12 C(C(=O)NC1CCC1NC(c1c[nH]cc1C1CC1)=O)(C(C)C)OC c1(CC(N2CCN(CC(=O)NC(CC)C(C)O)CC2)=O)cc(C)ccc1C C=CCC(CC(C)C)C(=O)NCC1(NC(=O)CCN2CCCCC2=O)CCC1 CC(C)(C)C#CCCNC(C1COCCN(C(=O)C=CC(F)F)C1)=O N1(C(CC2(C)CCCCC2)=O)C2CCC1CC(CNC(=O)C=CC1CCOC1)C2 c1(C(=O)NCC(N2CCN(C(C3CCCCS3)=O)CC2)C)cc(O)ccc1F C12(CNC(CCCCSC)=O)CCC(C1)N(C(=O)Cc1cc(F)ccc1F)C2 Cc1cccc2cc(C(=O)NCC(n3cc(C4(C(C)C)COC4)nn3)C)[nH]c12 c1(C(=O)NC2CC(C)N(C(c3csc(=N)[nH]3)=O)C2)cccc([N+](=O)[O-])c1 c1(C(=O)NCC(C)O)c[nH]c2ccc(-c3cccc(NC(N)=O)c3)cc12 n1(CC)nc(C)c([N+](=O)[O-])c1NCC1CCC(NC(C2CCCS(=O)(=O)C2)=O)C1 c1(C(=O)NC23C(CN(C(CS(CC)(=O)=O)=O)C2)C3)cc(F)c(C#N)c(F)c1 C1(CNC(C#CC(C)C)=O)(CO)CCN(C(=O)C(C)COc2ccccc2)CC1 C(=O)(C=C1SCC(=O)N1C)N1CCCC(CCC)(NC(c2nc(Cl)oc2C)=O)C1 CC(C(=O)NCC1CN(C(=O)C(C)(C)n2cccn2)C1)C(F)(F)F c1(OC)c(CNC2CCS(=O)(=O)C2C)cc(Cl)cc1Cl c1(C(=O)NC(CCC)CO)coc2c1CN(C(=O)CN(C)CC)C2 N1(C(=O)NC2C(c3n(C)ccn3)OCC2)CCCC2CCC12 c1(C(N(CCC)CCNC(=O)C(c2nc(C)cs2)C)=O)cc2c(ncn2C)[nH]1 C1(C)(CNC(CCSC)=O)COCCN(C(c2c(C)noc2C2CC2)=O)C1 C(CC(F)(F)F)NC(c1cn(CC2CCCNC2)nn1)=O c1(OC)cncc(C(=O)N(C(C)C(=O)NCc2csc(C)c2C)C2CC2)n1 c1(OCC(=O)NCC2CC(NC(c3c(C)nsc3)=O)C2)cccc(Cl)c1 C1(NC(c2cc(C)nnc2O)=O)CCCCN(C(=O)C(C)(Cl)Cl)CC1 N1(C(CC2CCCN(C(C(C)CC3CCC3)=O)CC2)=O)CC2(CCCCC2)C1 C1(C(N2CC(C(N)=O)(CNC(C3(C)CCCCC3)=O)C2)=O)Cc2ccccc2O1 c1(N2CCN(C(=O)Nc3ccc(C)nc3)CC2)cc(C)nc(C(F)(F)F)n1 c1(C(=O)NCC(C)(C)NC(CSCCC)=O)cc(O)cc(Cl)c1 CCCCC(CNC(c1nncs1)=O)NC(=O)C(C)Cc1ccc(N)cc1 n1(C(CC)C)nc(C(=O)NCCC2CCCN(C(=O)CCNC(N)=O)C2)cc1C C(=O)(C(C1=CCCSC1)N1CCCC(c2ccccc2)(CO)C1)NCCCOC CCCC(CNC(=O)CCOCC)NC(c1cc(=N)[nH][nH]1)=O CCC(CC(=O)N1CC(CC(C)NC(c2sccc2S(N)(=O)=O)=O)C1)C(F)F c1(NC(C)=O)ccc(N)c(C(N2CC(N(C)C(C3CCCO3)=O)C(C)(C)C2)=O)c1 c1(C(=O)OC)sccc1C(=O)NCC1(O)CN(C(C2(CN(C)C)CC2)=O)C1 C(C(C(=O)N1CCCC1CCCNC(c1cn(CCO)nn1)=O)NC(C)=O)OC N1(C(CCSCC)=O)CC2(CCC2)CC1NC(=O)CC(C)NC(=O)OC(C)(C)C C1(C(=O)OC(c2ccc(Br)c(Cl)c2F)=CCl)CCC2CN(C(=O)C(F)(F)F)CC2O1 CC1(C)CN(C(=O)C(c2ccoc2)NC(c2ncc[nH]2)=O)C2CCCC12 C12(NC(c3cc(SC)ncc3)=O)CCCC1N(Cc1nc3c(o1)CCCC3)CC2 c1(SCC(N2CCC(O)(CN(C(C3(C=C)CC3)=O)C)C2)=O)ccc(C#N)cc1 C1(NC(CC2CC(CC)C2)=O)CCC(NC(c2ccn(C)c2)=O)CC1 c1(C(=O)NC2C3(NC(CCC(C)(C)C)=O)CCC(C2)C3)scc2c1CCCC2 CC1(C)CC(NC(C2CN(C(=O)CC3OCCCO3)CC2C2CC2)=O)C(C)(C)O1 C(=O)(C1CCCn2cncc21)NCC(CCCC)NC(=O)C(Cl)=CCl C1(NCC(=O)N(CC(=O)Nc2cc(C)no2)C)CCCCC12CCC2 N1(CCN(C(C2(CC)CCCO2)=O)C)CCN(C(=O)CCc2ccccc2)CC1 N1(C(c2cc(C(N)=O)[nH]n2)=O)CC2CC(C1)CN(C(C1CCC3CCC13)=O)C2 C1(NC(c2c(CNC(C(CN(C)C)(C)C)=O)occ2)=O)CCCC(F)(F)C1 C1(CNC(=O)C=CCF)CCC2(CCC2)C1NC(=O)COc1ccccc1[N+](=O)[O-] Cc1cc(N2Cc3c[nH]nc3C2)nc(N2CCCC(n3ccnn3)CC2)n1 Cc1ccc(Cl)c(OCC(=O)NCC2(F)CC(NC(=O)CC3(O)CCC3)C2)c1 C12(CNC(C(C=CCCC)O)=O)CC1CN(C(c1cnn(CC)c1Cl)=O)C2 C1(C(=O)NCC2CC(NC(Cc3c(C)cco3)=O)C2)CC(C)(C)CO1 c1(NC(c2n(C(CC)C)nnn2)c2coc(C)n2)cccc(C#N)c1C c1(C(=O)NC2(CN(C)C(C3CC4CCC3O4)=O)CC2)cc(=O)n(C)o1 C1(C#N)(CC(=O)N(C)CCOCCN(C)C(c2cccc(Cl)c2)=O)CCOCC1 CC1CC(C(=O)Nc2ccc(C(C)(C)C#N)cc2)N(C(=O)CC(F)(F)F)C1 Cn1ncc(CNC(=O)CCc2nncs2)c1C(=O)NC1CC(O)C1 C(=O)(CCCCC(F)(F)F)N1CCN(CCNC(c2c(CC)cncc2)=O)CC1 Cc1cc(Cl)ccc1-n1nc(CCC(C)C)nc1C1CCCN1c1ncccn1 c1(C(=O)NC2CCN(C(c3ccc(COC)o3)=O)C2)ccc2cnccc2n1 c1(C(N2CCC(OC)(CNC(c3ncccc3C)=O)C2)=O)ncc(C)cc1C CC(C)C(O)CC(=O)N(CCNC(c1csc(NC(N)=O)n1)=O)C(C)C N1(C(C2CCC(=O)N(C)C2)C(=O)NCCSC)CCc2cc(CO)ccc2C1 c1(C(=O)NC(C(=O)NCCC)C)ccnc(CNC(=O)CN2CCCCC2)c1 N1(C(C2Cn3c(C)nnc3C2)=O)CCCn2nncc2C1 c1(CNC(N(CCC[Si](C)(C)C)CC)=O)ccc2c(n1)CCO2 Cc1cccc(C(CNC(c2c(C)n[nH]c2C)=O)NC(C2(C)C=CCCC2)=O)c1 c1(C(=O)NC2C(NC(C3N(C)CC(C)(C)C3)=O)CCOC2)ccc(Cl)c(F)c1N CCS(=O)CC(=O)NCCC1CC(NC(=O)CN2CCC(O)CC2)C1 CN1CNC(=O)C12CN(Cc1ccc(-c3ccsc3)nc1)C2 N1(C(c2ccc(NS(C)(=O)=O)cc2)=O)CCC2CCC12CNC(c1ccc[nH]1)=O C=CCCCC(=O)NC1(C)CN(C(C2(c3ccccc3)CC(C)C2)=O)C1 N1(C(=O)OC(C)(C)C)CC=C(C(C)(C)C(=O)Nc2cc3cccnn3n2)C1 N1(C(C=C(CC)C)=O)CCC(CF)(NC(c2ccc(C3CCOC3)s2)=O)C1 C1(F)(CNC(C(C)OCC)=O)CCN(C(c2cc(C3CCCCC3)n(C)n2)=O)C1 C(C)(C(O)C(C)C)NC(c1nc(CNC(c2c(C)snc2)=O)oc1)=O C(=O)(C(C)(C)Cc1cccc(Cl)c1)N(CCNC(C1CC2CC2C1)=O)CC c1(C(N(CCCCCC)CCNC(C2CCCS2)=O)=O)nccc2ncccc12 CC1CC(NC(c2cc(O)cc(O)n2)=O)CN(C(C2(C)CC2Br)=O)C1 c1(OCC(=O)NC(CC)(CNC(=O)C=CC2CCC2)CC)c(F)cccc1F N1(C(C(C)N(C(C)=O)CCO)=O)CCC(O)C(C(=O)NCC2CC3CCC2O3)C1 Cc1ccc(C(=O)NC2CCCC(NC(c3c(CO)cccc3F)=O)C2)cc1F Cc1ccc(F)cc1C(N1CCCC1C(C)(C)C(=O)N(C1CCSCC1)C)=O c1(C(C)C)ccc(C(N2CC(F)(CNC(C3CCC3C)=O)C2)=O)c(F)c1 N1(C(CC(=C=C)C)=O)CCC(C)C(CNC(C2(COC)CCCCO2)=O)C1 c1(N2CC(=O)NCC2)ccc(NC(C2C(F)(F)C23CCC3)=O)cc1Cl N1(C(CCCCCCC)=O)CC(NC(=O)C2=CCCOCC2)C2(CCCC2)C1 C1(NC(CC2(N(C)C(c3csc(F)c3)=O)CC2)=O)CC2CCC1O2 C1(NC(C(CSC)OC)=O)CCCC(NC(c2cncc(C(F)F)c2)=O)C1 C1(C(N(CCC(=O)NC2CCC2(C)C)CC#C)=O)C(C)(C)C1(F)F C(=O)(C(C)CCC(C)(C)C)NCC(C)(C)NC(c1c(C)cc(OC)nc1)=O N1(C(=O)CCOC2CCC2)CC2CC1CN2C(=O)C=Cc1cncs1 C1(CNC(c2ccc(OC)nn2)=O)CC2(CC2)CN1C(=O)C(C)(F)F c1(OC)ccc(OC)c(C(=O)NC2CC(CNC(=O)C=CC=C(Cl)Cl)C(O)C2)n1 N1(C(c2c(C)cccc2[N+](=O)[O-])=O)CC2CN(C(C3CC3F)=O)CC2C(F)(F)C1 c1(OC)ccc(O)cc1NC(C1CC(N(C)C(c2[nH]cc(C)c2C)=O)C1)=O c1(C(=O)NC2CCN(C(c3c(C)[nH]nc3Cl)=O)C2)nccc2cccnc12 C(c1ccccn1)=C(C)C(=O)NCCCC1CCCN1C(=O)C=C1CCOCC1 N(C1CCCc2ccc(Cl)cc21)C1C(C)CNC1 c1(C(N(C(C(=O)OCC)C)C)=O)csc(CNC(C2(C#N)CC2)=O)c1 C1(NC(C(COC)(F)F)=O)CC2CCC(C1)N2C(=O)CC1CCCCCC1(F)F C(=O)(CCNC(N)=O)N(CC(=O)N(CCSC)C)C1CC1 C1(O)(CC(=O)NN2CCCCC2)CCCC1.C1(C2CNC(=O)CS2)CCCCC1 C1(CCn2cc(CO)nc2)CN(CCC2CCCC3CC23)CCO1 C1(O)(CNC(c2c(CC)cns2)=O)CCN(C(C2C(C)(C)C2(F)F)=O)C1 N1(C(CCC(=C)Cl)=O)CCCCCC1CNC(C1CCN(C)C1CC)=O CC1CN(C(=O)C#CC2CC2)CC(C)C1NC(c1ccc(Br)cc1O)=O C1(C)(NC(C2(CCNC(c3cn(CC)nc3)=O)CC2)=O)CCC(=O)N(C)C1 c1(-c2cn(CC=C)nn2)nc(Cc2ccccc2C)nn1C1CCCCC1 N1(C(C(C#C)(C)C)=O)CCN(C(c2cc[nH]c2C2CCC2)=O)C2(CC2)C1 CC1CCC2(CCN(C(=O)CN(C(=O)CCc3ncccn3)C)C2)C1 C1(CNC(c2ccc(C)nc2O)=O)CN(C(c2cc(C)[nH]n2)=O)C2(CCC2)C1 C1(OC)CCC(NCC2(c3noc(C)n3)CC2)CC1 c1(CC(=O)N(CCC(=O)N(C(CC)C)CC)CCCO)ccc(C)cc1C c1(NC(c2ccc(CCNCc3ccc(C)nc3)cc2)=O)cnn(C)c1C#N C(=O)(C(CC(C)C)NC(c1ccc(F)c(C)c1)=O)N1CCC(SC)C1 c1(-c2cc(C(N(CCNC(C(C)OC)=O)C)=O)n[nH]2)ccc(Br)cc1 C1(NC(c2ccc(I)c(Cl)c2)=O)CC12CCN(C(C13CC(C1)C3)=O)CC2 C=CCCC(CC(C)C)C(=O)NCC(C(C)C)NC(c1cc(C)n(C)c(=O)c1)=O N1(C2CCN(C(C(C)CF)=O)CC2)CCN(C(=O)C=CC2CC2)CC1=O c1(C(=O)NC2CN(Cc3nnc(C4CC4)n3C3CC3)C2)cc2cc(Cl)ccc2[nH]1 N1(C(c2nc(O)cc(OC)n2)=O)COC2CCCCC2C1 N1(C(CNC(C2CCC2)=O)=O)CCCC(O)(CNC(C2CC2C2CC2)=O)CC1 C(=O)(C(CC)CC(C)C)NC(CCCC(=O)N(CC)Cc1cnn(C)c1)C c1(C(=O)NCCC2CC(NC(CC(CN(C)C)O)=O)C2)ccn2cc(C)nc2c1 c1(OC(C)C)ccc(CC(=O)NCC2(F)CC(NC(c3ccsn3)=O)C2)cc1 N1(C(COC(C)(C)C)=O)CC2CCC1C1CN(C(=O)C=Cc3ncc[nH]3)CC21 CC1(C)CC(CNC(C2(C3CC3)CCC2)=O)N(C(=O)CCCn2ccnc2)C1 c1(CNC(C(COCC)NC(CC=CC=C)=O)=O)ccc(O)cn1 c1(CSCCC(=O)OC)ccc(NC(=O)C(=O)Nc2cccc(I)c2)cc1 Cc1nncc(C(=O)N(C(C)C(N2CC(C)C2(C)C)=O)C)c1C c1(C(=O)NCC2(CCNC(c3ccc[nH]3)=O)CC2)nccc2c(F)cccc12 c1(C(C)(C)C(=O)NCC2CCN(C(=O)CS(=O)(=O)N(C)C)C2)ccc(F)c(F)c1 c1(C(=O)NC(C2CCN(C(c3c(CC)occ3C)=O)C2)C)cc(C)ccc1C Cc1cc(O)c(Cl)cc1C(=O)NC(C)CN(C)C(c1ccc(Cl)[nH]1)=O N1(C(CCOCC)=O)CCC(F)(CNC(C2CC(O)(CC)C2)=O)C1 C1(C(=O)NCCCN(C(c2nc3cnccc3s2)=O)CC)CCc2nnnn2C1 CC1(C)CC(C(=O)NCc2ncc[nH]2)CN(C(C2COCC2(C)C)=O)C1 C1(c2nnnn2CCCN(C(=O)C(=O)NCC(C)OC)C)(N)CCOCC1.CO C(=O)(C(C)(C)C(O)C(C)C)NCC(CC(=O)N(C(C(=O)NC)C)C)C1CCC1 C1(NC(C(CC)SC)=O)CCCCN(C(c2ccc(O)cn2)=O)C1 c1(CC(=O)OC)csc(=NCC2CCCCC2C(=O)O)[nH]1 c1(C(=O)NC2CC(C)N(C(c3cc4c(ccn4C)s3)=O)C2)cc2occc2n1C Cc1cc(C(=O)NC(C)CC(=O)NC2CCCC2)nn1-c1ccccc1 C(=O)(CCCCCN=[N+]=[N-])N(C(C(N1CC(C(=O)OCC)C1)=O)C)C N1(C(C2C(N(C(C3OC4CCC3C4)=O)CCO)CCCC2)=O)CC=CC(O)C1 C1(C(F)(F)F)(C(=O)NCC(C)(C)NC(c2n[nH]c(C)c2O)=O)CC2CCC1C2 CCCCN=C(NCC1CCNC(=O)C1)N1CCN(CC(C)C)CC1 C1(C(N2CC(C(C)NC(C(C)Sc3ccccn3)=O)C2)=O)CC(=O)N(C2CC2)C1 c1(NC(C=C)=O)ccc(Br)cc1NC(=O)Nc1ccc(Sc2ccncc2)cc1 N1(C(c2c(C)cns2)=O)CC(C)C(C)(CNC(=O)C(O)C(F)F)C1 c1(OC)nccc(C(N2CCC3CC23C(=O)NC(C)Cc2cn[nH]c2)=O)n1 C(=O)(C1=CCCCCC1)NC(C)C(c1ccccc1)NC(c1cccc(O)n1)=O CCCC(F)C(=O)NC1(C)CN(C(c2cn(CCC)nc2C)=O)C1 C1(NC(c2cc(C)nn2C)=O)CCN(C(=O)Cc2cc(Br)cs2)CC1(C)C N#Cc1cncc(C(N2CC3CC2C3CNC(=O)CN2CCc3ccccc32)=O)c1 C1(CC)(NC(=O)C(O)C(C)C)CCN(C(c2cn(CC)nc2C)=O)CC1 C1(S(N)(=O)=O)(C(=O)NC2CCCN(C(C(F)OC)=O)C2)CCC1 c1(C(=O)NC2(CCOCC)CC2)nnc(O)cc1C.C12(CC1)CC(=O)NC2 N1(C(COCCCCC)=O)CCCC(N(C(=O)CC2C=CCCC2)CCOC)CC1 C#Cc1cnn(C)c1C(=O)NCC1CCC(C)N(C(=O)Cn2nc(C)nc2C)C1 C1(NC(C(C)OCC(C)C)=O)COCCC1NC(=O)CCC1CC1 C1(CC)CN(C(=O)Cn2nccn2)CCC1CNC(c1c[nH]c(=N)o1)=O N1(C(c2ccc(Cl)c(F)c2)=O)CCC2(CCN(Cc3cc(O)cc(Br)c3)CC2)C1 Cc1cc(C(=O)NC2CCC(CNC(=O)CC(C)(C)O)C2)nn1C N#Cc1c(Cl)nsc1N1CCC(C(N2C3CCC2(CO)CC3)=O)C1 c1(C(=O)NC2CN(C(C(CC=CC)CC)=O)C(C)C2)cc(Br)c([N+](=O)[O-])[nH]1 N1(C(C2(CC)CN(C(=O)C(C)=CCO)C2)=O)CCC(CC(N)=O)CC1 C=CCCCC(C)NC(=O)C(COCC)NC(c1ccco1)=O C(=O)(C1=C(c2ccc(OCOCC)cc2)CCCC1)OC1COC1 C1(C(N2CC(OC)(CO)C2)=O)CC(CC)CCN1C(c1cc(CO)oc1C)=O Cc1cc(C(=O)N(CCNC(C2(C)CC3CC3C2)=O)C2CC2)c(O)c(C)n1 C=CC(O)C(=O)NCC1CCC(C(=O)NC2CN(C(=O)C3CC3)C2)O1 C(=O)(C1=Cc2cc(F)ccc2OC1)NC1CCN(C(C=C2CCN(C)C2)=O)CC1 C1(C(=O)NC2CCN(C(C3(CC=C)CCOCC3)=O)C2)CCCC2(CCC2)O1 c1(C(=O)NC2CC3(CC(C)C3)C2)nc(Cl)c(=O)[nH]c1N C1(C(=O)NCCCCC(C)NC(c2n(CC)nc(C)c2)=O)OCC2COCCC12 Cc1nccc(C(C(=O)NC2COC2)NC(C2CC(OC(C)(C)C)C2(C)C)=O)n1 C=C(C)C1OCCC1C(N1CC2(C=CCO2)C1)=O.C12CC(C1)OCC(=O)N2 N1(C(C(C2CCC2)OC)=O)CCOCC1CNC(C1(n2ccnc2)CCCC1)=O Cc1cc(C(=O)N(C2CC(C#N)C2)CC(=O)NCCN2CCCC2=O)c(C)s1 C1(CC(C)C)CN(C(C2CCCN2Cc2cn(Cc3csnn3)nn2)=O)CCO1 Cc1cc(F)c(NC(=O)NCC2CC2Cc2ccccc2)c(F)c1 Cc1nc2cc(NC(c3cc(F)ncc3NCc3cn(C)cn3)=O)ccc2o1 Cc1ncc(CC(=O)NCC(C)NC(C2CC3(CC3)C2)=O)s1 C1(C(=O)NC(C2CCCO2)(C)C)CCCC(NC(C2(F)CCOCC2)=O)C1 c1(SC)ccccc1-n1nc(-c2cncc(F)c2)nc1CN(C)C N1(C(CC(CCC)O)=O)CCC(C)N(C(=O)C(O)CN(C)C)CC1 CC1SCCCC1C(N1CC=CC1(C)C(=O)NCCN(C)C)=O c1(NC(c2nnnn2C)C)[nH]c(=NCc2coc(CO)c2)nc2c1ncn2C C(=O)(C(C)(C)C1=CCN(C(=O)C(O)CN2CCCC2)C1)N1CCC(C)(C)C(O)C1 C#CC1CCN(C(C2CCN2C(=O)CN2CC(C)(C)C2)=O)C1 C(=O)(CC1NC(=O)c2ccccc21)NC1CCN(C(C(COC)(C)O)=O)C1C Cc1nc2c(o1)CCCC2CC(=O)N1CC(NC(c2ccc[nH]2)=O)CC(F)C1 C(=O)(CS(=O)(=O)C1CC1)NCC1(C(C)NC(C)=O)CC1 C1(C(N2CC(C(N)=O)(CNC(C3(CC)CC3(F)F)=O)C2)=O)CC(C)CCO1 C(CCC(C)NC(c1cnc(CC)o1)=O)NC(COCCC=C)=O C1(CNC(c2nc(CC)sc2)c2nnnn2CCCSC)CCCC(F)C1 Cc1nn(C)c(C)c1CC(C)C(N1CC2(CC2)CC1CNC(c1cnoc1)=O)=O c1(C(=O)NC2C(NC(C(CCCC)CC)=O)C2)cc2cccc(OC)c2o1 C(=O)(CS(=O)(=O)CCO)N(C)CC1CCCN(C(=O)CC2CC3(CC3)C2)C1 C(N=c1nc(-c2ccsc2)c(F)c[nH]1)C1CCC(NC(CC2(C)CCCO2)=O)C1 Cc1ccc(C)c(CN2CC3CC(C2)N3C(=O)C=Cc2ccc(F)cc2F)c1O c1(C(=O)NC(C(CO)NC(c2oc(CC)c(C)c2)=O)C)coc2c1COC2 c1(CCCNC(CCN(C(CCOCCOC)=O)C(C)C)=O)cccnc1 N1(C(CCCc2onc(CCC)n2)=O)CCCN(C(C2CN(C)C2)=O)CCC1 C1(CC=C)CCCCN1C(C1CSCCN1C(c1cc(C)nn1C)=O)=O C=C(C)c1cncc(CNC(=O)C(n2cc(-c3cnc(F)c(C)c3)nn2)C)c1 CC1CCC(C(N2CC(CCCCNC(=O)C3=CCCCO3)C2)=O)C(=O)N1 N1(C(CNC(C)=O)=O)CCC(C(=O)NCC2CC2(F)F)(CO)C1 Cc1cc(C(F)(F)C(=O)NCC(O)CCNC(C2CCCN2N=O)=O)cnc1Cl C(=O)(CC(C)C(=O)OC)NCc1c(C(=O)NC(c2ccccc2)CC)cccn1 C(=O)(C1=NN(C)C(=O)CC1)N1CC(CCNC(=O)C=Cc2csc(C)n2)(OC)C1 CC(C)C(C)(CNC(=O)CSCc1cscn1)NC(=O)CC1CCCC1O C1(c2ccc(C(=O)OC)cc2)CCCN(Cn2cnc(-c3ccccc3)n2)C1 N1(C(C(c2ccnn2C)NC(CCC=CCC=C)=O)=O)CCCC2(C=CCO2)C1 C1(CNC(c2c(CCC)nsc2N)=O)CC2CCC1N(C(c1cncn1C)=O)C2 c1(C(N2CC(CN(C(C3N(C)C(=O)CC3)=O)C)C2)=O)nnc2ccccn12 C1(CC(=O)NC2CCC(F)(CNC(c3c(C)ncn3O)=O)C2)(OC)CCOCC1 N1(C(COC)=O)CCCC(C2CN(C(=O)Cc3ccccc3C#N)C2)C1 C1(OC)CC2(CCC(C(=O)N(CC(C)NC(c3n[nH]cc3Br)=O)C)CC2)C1 N1(C(C2=CC(C)CC2)=O)CCCC2CN(C(=O)CCn3cc([N+](=O)[O-])cn3)CC12 Cc1occc1CC(=O)NCCOCCCNC(=O)C(c1ccccc1)O C12(CC)CC1CN(C(C1(c3cscc3Br)CCCO1)=O)C2 c1(C(=O)NCCCC2N(C(Cn3c(C)nc(C)n3)=O)CCC2)cc(O)ncc1F Cc1ccsc1C(=O)NCC1CC(F)(CNC(=O)CCc2nncs2)C1 N(C(=NCCCCl)N1CCN(C(c2ccco2)=O)CC1)CC(CC)C(C)C C(CN=C(NCC)N1CCC2(CCCC2)C1)OCC12OCC(C(=O)OCC)(C1)C2 C1(NC(c2cc(O)cs2)=O)CCCC(NC(c2cc(F)ccc2F)=O)CC1 CC1CCCN(C(=O)C(C2CC2)NC(=O)CS(C)(=O)=O)CC1 C1(NC(CC2CC(SC)C2)=O)C2CC(NC(c3ccc(Cl)cn3)=O)CC12 C(C1CCC(C)CC1)=C(C)C(N1CC(C)(NC(c2c[nH]cc2Br)=O)C1)=O C1(C(=O)N(CCCNC(=O)Cn2cc(Br)cn2)C)(COCC)CCCC1 C1(NC(C(CC(C)C)F)=O)CN(C(c2cocn2)=O)C2(CCCCC2)C1 Cc1ccc(CSCCC(=O)NCC2CCN2C(=O)Cn2nc(C)nc2C)cc1 CCC(CC)CCC(=O)N1CC2CC(C(=O)N(CC)Cc3cccnc3)CC2C1 N1(c2ncc(C(=O)OCC)cn2)C2CCC1CC(NC(=O)Cn1cncc1C)C2 c1(CNC(C2N(C(C(CC)n3cncn3)=O)CC2)=O)nnc(O)n1C CC1CC(NC(C2CCCCCC2)=O)CCN1C(c1nccc(C(F)(F)F)n1)=O Cn1cc([N+](=O)[O-])c(C(=O)NC(CNC(=O)C=CC2(C)CCOCC2)CO)n1 c1(-c2n(-c3ccn(CC)n3)nc(-c3ccsc3)n2)cc(F)ccc1F C1(CCOC)CN(C(c2cc(F)ccc2Br)=O)CCN1C(=O)C=CCO c1(C(NNC(=O)NC(c2sccc2C)CC)=O)cccc2ccccc12 S(=O)(=O)(CCC(F)(F)F)NC1CCN(C(=O)CC2CC3CCC2C3)C1 c1(NC(C2(CCNC(c3cscn3)=O)CC2)=O)cccc(NC(=O)C2CC2)c1 C1(CCNC(C23CCOCC2C3)=O)CCCCN1C(=O)CNc1nccs1 c1(C(=O)NCCCN(C)C(C2(F)C3CCCCC23)=O)ccc(F)c2ccccc12 N12CC3CC(CC(C3)C1)C2=O.c1(SC(C)C(=O)NCC2CC2CO)ccccc1 c1(NCC(CCOC)(C)C)nc2ccccc2nc1N1CC2CSCC(C2)C1 C1(C(=O)NCc2scc(C(N(C3CC(OCC)C3)C)=O)c2)OCCCC1(C)C c1(NC(CCCN(C(c2ccc(OCC)nc2)=O)C)=O)cnnc(O)c1Cl C1(C(=O)NCCN(C(Cc2cn(CC)nc2)=O)C)CCCCC1(F)F c1(CCC(=O)NC2CC(NC(c3c(C)nn(C)c3F)=O)C2)nc2ccccc2[nH]1 C1(C)(NC(C(CCC)=CCC)=O)CCN(C(=O)C(O)Cc2ccc(F)cc2)CC1 c1(C(N(C)CCNC(C2COC2)=O)=O)cc(Cl)c(Cl)s1 C1(c2ccn(C)n2)CCN(C(C2CCN2C2CCNCC2)=O)CC1 Cc1occ(-c2ccccc2)c1C(N1CCC(NC(=O)CC2CC23CC3)C1)=O CC(C)(CNC(=O)C(N1CCC(CC(N)=O)C1)=O)CC1CCC1 Cc1c(C(=O)N(C(C)CCNC(C2CCC2)=O)C)csc1Br N1(C(c2n[nH]c(CC)c2Cl)=O)CCC2CN(C(c3ccc(F)c(C)c3)=O)CCC12 c1(Cn2cc(C(N3CCCCC3(C)C)C)nn2)ccc(Br)cc1[N+](=O)[O-] CC1CC(C(=O)N2CCCC2C2CCN(C(=O)CC3CCCCC3(C)C)C2)=NO1 C(C(=O)Nn1nnc2c1CCCC2)(C(C)(C)C)NC(c1c(C)cns1)=O CC(O)(CNC(=O)CC1CCCC1NC(=O)C=CC(F)(F)F)CCO C(=O)(CCC(C)CN(C)C)NCCC(CCNC(c1nn(CC)c(C)c1)=O)C C(=O)(C(C#N)C(C)(C)C)N1C(C)CC(CC(=O)NCC2(OCC)CC2)C1 N1(C(C2OCC(C)C2)=O)CCC(CNC(=O)C(C)(C)N(C)C)C(F)(F)CC1 c1(CC)oc2ccccc2c1C(N1CCCC(C)C1CNC(C1(O)CC1)=O)=O CC1CN(C(=O)Cc2csnn2)CC1(C)CNC(=O)C(C)(C)Oc1ccccc1 N1(C(C(C2CCOCC2)C)=O)CCN(C(C2CC(F)C(=O)N2)=O)CC12CC2 c1(CNC(CC(C)SC)=O)cccc(NC(c2ccns2)=O)c1 N1(C(c2nc(C)[nH]n2)=O)CCCCC1CN(C)C(C1(c2ccncc2)CCC1)=O CC1OCC2(CCC(CNC(N3CC(C)(C)OCC3CO)=O)O2)C1C N1(C(C2(COC)CCCC2)=O)CCC(NC(=O)CC23COC(C)(C2)C3)C(C)(C)C1 C1(C)(C(N(C)CC2(O)CN(C(C(c3cccc(F)c3)C)=O)C2)=O)CCSCC1 N1(CCOC)CCC(NC(=O)CN(C2CC(C#N)C2)C(=O)C=CC2CCOC2)C1 N1(C(C(COC)(C)OC)=O)CC2(CC(CNC(=O)CCc3ccn(C)n3)C2)C1 CCC(CC)C(=O)N(CCC(C)NC(=O)C(C)(C)c1cnco1)C N1(C(CSC)=O)CC(O)(C(C)NC(=O)CCOCC2CCCO2)C1 c1(C(=O)NC(CNC(C(CCCC)CC)=O)CO)ccc2c(c1)COCO2 N1(C(c2ccc(F)cc2)=O)CCC2CCCN(C(c3cc4[nH]ccc4s3)=O)C2C1 C1(OC)CCCCC1C(=O)NC12CC(C1)N(C(c1ccc(C(N)=O)nc1)=O)C2 n1(CC#C)cccc1C(=O)NC(C1CCCN1C(c1cnc(C2CC2)s1)=O)C N1(C(C(c2cncc(F)c2)C)=O)CCC(CNC(C2CC3CCC3C2)=O)CC1 C1(CNC(Cn2c(C)c(Cl)cn2)=O)C(C2CC2)CCN1C(=O)C(N=[N+]=[N-])C(C)C C(CCCCNC(=O)CC1CC(F)C1)N(C(=O)CCN1CCOC1=O)C C1(OC)CC(CNC(=O)CCCNC(N)=O)N(C(=O)Nc2[nH]c(O)nc2C)C1 C12(NC(C3CCC(OC)C3)=O)COC(CNC(=O)CCc3cccc(F)c3)(C1)C2 C1(CC(=O)NCC2(OC)CN(C(=O)C(F)=C(C)C)C2)CCCC(O)C1 N1(C(c2c(C)n(C)cn2)=O)CCC(NC(c2ccccc2F)=O)C(O)C1 C1(NC(=O)Nc2ccc(CC(=O)OC)cc2)C2Cc3c(Br)cccc3C12 C1(C(=O)OCc2cn3ccsc3n2)CC(O)(C2(O)CCC2)C1 N1(C(C(CNC(c2cnc(C)s2)=O)(C)C)=O)CC(C)OC(C)(C)C1 c1(C(N2CCC(NC(C3CCSCC3)=O)CC2)=O)ccc2cnnc(O)c2c1 S(=O)(=O)(c1cc(Cl)ccc1OCC1CCC1)NC(C)(CO)C1CCCO1 CC1(CNC(=O)CC2(CO)CCC2)CCN(C(=O)CCCN2CCCC2)CC1 C(=O)(C(F)(CNC(=O)C=Cc1cn(C)nn1)C(C)C)N1CC(CCCCC)C1 Cc1cnc2cccc(C(N3CC(NC(=O)Cn4cncn4)CCC3C)=O)n12 c1(C(=O)NC(C2CCCN(C(CCC(=O)NC)=O)C2)C)ccc(F)c(F)c1F c1(NC(C2(C)CCN(C(CC(CC)O)=O)C2)=O)cccc(C#C[Si](C)(C)C)c1 N1(C(C2C(C=C)C2)=O)CCN(C(c2c(C)cccc2F)=O)CC1CS(C)(=O)=O N1(CCCNC(C2CCC(C(N)=O)C2)=O)CCN(C(=O)CCc2ccco2)CC1 N1(C(CN2CCN(CC)CC2)=O)CCC(C)(NC(c2nnn(C)c2N)=O)CC1 c1(CC(=O)NCC2COCCN2C(=O)C2=CSCS2)c(Cl)cccc1Cl N1(C(Cc2cc(COC)on2)=O)CC(NC(C2CC(C)=NO2)=O)C(C(F)(F)F)C1 n1(CCNC(=O)Cn2cnnn2)ccc(C(=O)NCCC2CCC3CC23)c1 CC1=C(C)CC(C(=O)NCC(O)CCNC(=O)CC23CCC(CC2)CC3)CC1 C1(C(=O)NCC2C(NC(c3cccc(C(=O)NC)c3)=O)C2)CCN(C)C(C)C1 c1(C(=O)NC(CC=C)CNC(=O)Cc2cncs2)c(C)nc2ncnn2c1C CN1CCN(C(=O)CCOCC2CC2)C(C(=O)NCCc2ccccc2)C1 C(=O)(CC(O)CC(C)(C)C)N1CC(OCCNC(C(CCC=C)(F)F)=O)C1 c1(SCc2n(CCSC)c(-c3ccccc3)nn2)cc(F)c(OC)cc1Cl NC(=O)CCCC(=O)NCC1C=CC(NC(c2ccc(C3CC3)cc2F)=O)C1 C(CC(C)(C)C)(C(=O)NCc1nc(C(C)C)no1)NC(CN(CCOC)C)=O N1(CC(=O)NCCCC(C)NC(=O)CCNS(C)(=O)=O)CCCCS1(=O)=O C1(CC)CC(NC(=O)C(c2ccnn2C)NC(=O)C=C(C)c2ccco2)CCO1 C1(CC(=O)NCC(O)CNC(c2cnoc2-c2ccco2)=O)CCCS1(=O)=O Cc1ncnc(C(=O)NC2CC=C(C(=O)NCC3C4CCCCC34)C2)c1C Cc1ccc(O)cc1C(=O)NC1CCC(CNC(=O)C#CC(C)C)CC1 Cc1csc(C=CC(=O)NCC(C(C)C)NC(=O)COc2ccon2)n1 c1(CN(C(c2nc(CC)[nH]n2)C(=O)NCCCF)C)cc(Br)nn1C Cc1cc(C)c(C(N2CC(C)(CNC(C3(C)CCCC3)=O)C2)=O)c(Cl)n1 c1(C(=O)NC(=C2CCCC2)CNC(C(C)=CC2CC2)=O)c(Cl)cc(Cl)nc1N C(C(F)(F)CNC(=O)C(CNC(=O)C(C)OCC1CC1)OC)OC c1(C(=O)OCC)cc(C(=O)NCC2CN(C(c3ccon3)=O)C2)no1 c1(C(=O)NC23CC(CNC(c4ccc(Br)s4)=O)(C2)C3)cccc2nc[nH]c12 C1(NC(c2noc(CC)c2C)=O)CCCC12CN(C(=O)CC1COC(C)(C)C1)C2 CON(CCC(=O)NC1CN(C(c2ccc[nH]2)=O)C(C)(C)C1)C(=O)OC(C)(C)C C1(c2cn(C(CNC(COCCCOC)=O)C)nn2)CN(C(C)=O)CC(C)(C)C1 C1(CCOC)CN(C(=O)CCC(=O)c2ccccn2)CCN1C(C1CC=CC1)=O Cc1cc(F)cnc1C(=O)NCCCCCCNC(=O)CCc1nc[nH]n1 N1(C(c2ncc(CC)s2)C(=O)NCCCF)CCCC2(CCCCC2O)C1 CC(C)CC(C(=O)NC(C)CNC(=O)Cc1coc(C(F)F)n1)N1CCCC1=O c1(C(N2CCC(CC)(CO)C2)C(=O)NC(CC)C)ccc(N2CCCCC2)cc1 c1(C(=O)NC2C(CC(=O)NC3CN(CC)CC3C)C(O)C2)cnn2ccccc12 c1(C(N2CCN(C(COC(C)C)=O)C(C3CC3)C2)=O)cc2cn[nH]c2cn1 c1(C(=O)NCC(CNC(CCCn2ncc(C)c2)=O)O)cncc(C(F)F)c1 N1(C(CCSCC(C)C)=O)CCCC2(CCCN2C(C2OCCOC2C)=O)C1 c1(C(C)C)nnc(C=CC(=O)N(C)CCN(C(C2(F)CCCC2)=O)C(C)C)o1 C1(F)(CNC(c2cnns2)=O)CCC(CNC(=O)C(F)(F)c2ccncc2)C1 C1(NC(c2ccccc2CO)=O)CCC2CN(C(=O)CCOC3CC3)CC2C1 N1(C(c2cnc(C)s2)=O)CCC(C=CC(=O)NC2CC(=O)N(C)C2=O)CC1 c1(OCC)ccc2cccnc2c1.N12CCCCCC1C(=O)NC1CC(C1)C2=O C1(C(=O)NC(c2ncc(C)[nH]2)CC)CCCN(C(C2CC3(CSC3)C2)=O)CC1 CCCC(C(=O)N1CCN(CCC)CC1)NC(c1cccc(C)n1)=O CC(CN(C)C)CC(=O)NCc1cn(CC(=O)NC(c2ncccc2F)C)nn1 C1(CNC(C(CC)F)=O)CCCCN(C(=O)CCc2c(C)nc(C)nc2O)CC1 c1(N(C)CC2CCS(=O)(=O)C2)ncccc1S(=O)(=O)N(C1COCC1O)C c1(CC(=O)NCCC(C)(C)NC(C2C(C)C2)=O)c[nH]c2cc(Cl)ccc12 S(=O)(=O)(c1cc(C)ccc1C)NCC(N1CC(NC(C2C(C=C)C2)=O)C(C)C1)=O C1(C)(NC(N2CCCC(NC(C(C)(C)C)=O)C2)=O)CCC(F)(F)C1 c1(CNC(C2(C)CCCN2Cc2cc(Cl)nc(Cl)c2)=O)ccc(C#N)cc1F CCCCC(C)C(=O)NC1(COC)CCCN(C(c2c[nH]c(=N)cc2C)=O)C1 c1(N(C(C)=O)C)cccc(C(=O)N(CCCN(C)C(c2cn[nH]c2)=O)C)c1 C(=O)(C(CC(N)=O)NC(C1CC12CCC2)=O)N1C(C)(CCO)CC1 C1(C(=O)NCCC2CN(C(C=C(CC)CC)=O)C2)CCC(NC(=O)C2CC2)CC1 C1(C(c2n(CC)nnn2)Nc2cccc(OC)c2S(N)(=O)=O)CC(C)(C)OC(C)(C)C1 N1(C(C(N)=O)=O)CCC(OCC2CCN(C(=O)CC3CC4CCC3O4)C2)CC1 N1(C(c2c(CC)n(C)nn2)=O)CCC(C)(C)C(C(=O)NCC2CC(F)C2)C1 CC1=C(C(=O)N2CCCC(N(C(=O)C3=CCC3)C)CC2)Cn2nnnc2N1C c1(C(N2CCC(CC=C)C2)C(=O)NC2CC2)ccc2nc(C)ccc2c1 CCC(C(=O)NC(c1cn(C2COC2)nn1)C)C(F)(F)F C#Cc1ccc(OC)c(C(=O)NCCC(CNC(=O)C(C)(CO)OC)OC)c1 C1(NC(=O)C=CBr)COCCN(C(=O)CCc2cccc(F)c2Cl)C1 c1(C(=O)NC(CC)CN(C)C(c2cc(C)no2)=O)cncc(C(=O)OC)c1 c1(N2CC(NC(CC)=O)C(O)C2)nccc(C#N)n1 c1(CC)ccc(C(=O)NCC(C)(C)NC(c2ccc(O)nc2)=O)cc1C#N C(=O)(C(CC)C(F)(F)F)NC(CC(N1CCC(C#C)CC1)=O)C1CC1 C1(CC(=O)NC(c2nc(C(=O)NCC3CCCC(C)C3)co2)C)C(C)(C)C1(C)C c1(C(N(CCN(C(C(CC)COC)=O)C)C)=O)c(Cl)c(C)nn1C Cc1cc(C(C)C(=O)NC2CN(C(=O)C(C)CCO)C2)cc(C)c1 c1(OC)cncc(CNC(=O)CN(C(=O)C(C)C#N)C(C)C)n1 C(C)(CC(=O)NCCC1CCC(NC(=O)Cc2cccnc2)C1)OC C1(NC(C(CC)O)=O)CCOCC1NC(c1cccnc1OCC)=O c1(C(N2C(CCNC(c3ccnn3CCF)=O)CCC2)=O)cn2ccsc2n1 CC1(C)CCCCC(C(N2CC(NC(c3ncccc3O)=O)C2)=O)C1 c1(OC)c(Br)ccc(-c2ccc(-c3nccn3CCN3CCCCC3)cc2)c1F N1(CCCCCNC(C(CC)SC)=O)CCN(C(C2OCCOC2C)=O)CC1 c1(C(=O)NCC2(OC)CN(C(CCCCC=C)=O)C2)ccc2c(Br)cnn2c1 C(=O)(C(C(C)C)n1cncn1)N(CCN(C(=O)C(C)(C)C)CCOC)C1CC1 C1(OC)CCCC1C(N1CCCC1CNC(=O)C=CC1CCCO1)=O N1(C(COCC=C)=O)CCC2CC2(NC(c2cc(OC)cnn2)=O)CC1 c1(-c2cn(CC(CCNC(C(C)C3CCCO3)=O)F)nn2)cccnc1Cl c1(C(=O)NC2C(NC(c3n(C)c(S)nn3)=O)C2)cnc(O)c2cccnc12 C1(CC#C)(C(=O)NCC2CC2[N+](=O)[O-])CCN(C(c2sc(F)cc2C)=O)C1 CC1(CNC(=O)Cc2cscn2)CCCN(C(=O)CCC2NC(=O)NC2=O)C1 c1(C(=O)NC(c2ncc(CC)s2)C)cccc(S(=O)(=O)N2CC(=O)NC(C)C2)c1 c1(C(N2C(c3cn(Cc4c(C)c[nH]n4)nn3)CCCC2)=O)cc(=O)n2ccsc2n1 Cc1c(C(N2CC3(CCN3C(=O)CC3CCCC(O)C3)C2)=O)sc2nnc(S)n12 C1(NC(Cc2ccc(C)s2)=O)C(C)CCN(C(c2cc(O)cc(N)c2C)=O)C1C c1(-c2occ(C)n2)ccc(C)c(NC(C)CC2CCNC2=O)c1 Cc1ccc(C(=O)NC(C(=O)N(C2CCOC2)CCO)C2CC2)o1 C=CCC(CC)N=c1nc(N(C)Cc2nocc2CC)c2cnn(C)c2[nH]1 c1(C(C)NC(c2n(CCOC)nnn2)c2ccoc2C2CC2)ccccc1Br c1(C(=O)NC(CNC(C=C(COC)C)=O)CO)cc2sc(C)c(C(=O)OC)c2[nH]1 c1(CC(=O)NC(CCOC)CNC(C)=O)sc(C2CCC2)nc1C Cc1cc(=NC(=O)C2CCCC23CN(C(=O)CCC2CCOC2)C3)[nH]o1 N1(C(C=COCC)=O)CC(CNC(c2ccnn2CC#N)=O)CC1(C)C C1(C(=O)NC(CC)C)CC2(CCN1C(C1C=CC1C(=O)OC)=O)CC2 N1(C(CC2C(C)OC(C)C2)=O)CCCC(N(C)C(c2ccc([N+](=O)[O-])s2)=O)CC1 C1(NC(Cc2cnc(C)s2)=O)CN(C(c2cc(F)c(N)cc2F)=O)CC(C)(C)C1 C12(CNC(C3CCCC3)=O)CC(CCO1)N(C(c1cccc(CO)c1)=O)C2 c1(NC(C(C)Oc2ccccc2)=O)cccc2c1C1CN(C(C3CCC3)=O)CC1O2 C1(NC(C(c2ccn(C)n2)(C)C)=O)CC2CC(NC(c3cc(Cl)c[nH]3)=O)C2C1 C1(CNC(C(CCOC)C)=O)CC(NC(=O)C(=O)NC2CC2)C12CCC2 N1(C(c2cncc(OC)c2)=O)CCC(C2CC2)C1CNC(C1CCCC(F)C1)=O c1(OCC2C(C)(C)C2)cnn(OCC(N)=S)c1 CN1C(=O)CCCC1C(=O)NC1CC2CC(NC(C3SCCS3)=O)C2C1 CCCC(C(=O)NC1CCN(C2CCOCC2)C1=O)N1CCCCC1 C1(CCOC)(NC(=O)CC2(C)OCCO2)CCN(C(=O)C=C=C(C)C)C1 c1(C(=O)NC2C(NC(C3(C)CC3)=O)CCCC2)cc(Cl)c(Cl)c(Cl)c1 c1(NC(C(CO)NC(C2CCC(OC)CC2)=O)=O)ccc2nncn2c1 C(C(C)(CC)C(=O)NCCn1ccc(=O)cc1)NC(CCC(=O)NCC)=O N1(C(C2(SC)CCC2)=O)CCC(F)(F)C(CNC(=O)CCCc2ccccc2)C1 C(CCC(=O)NC(C(=O)NCCCSC)C1CCSC1)OCCOC c1(C(=O)NCC2(F)CCCN(C(c3nc(=N)[nH]cc3)=O)C2)ccnc2cc[nH]c12 N1(C(c2nc(COC)oc2)=O)CC(C)CN(C(c2cc(Cl)no2)=O)CC1C C1(C(=O)NCC(C)NC(=O)C(C)c2ccsn2)CC(F)(F)C1 c1(CC)cccc(-c2ccc(CN3CCN(c4ccc(F)cn4)CC3)cn2)c1 C(=O)(C1CCCn2ncnc21)N1CCCC(CNC(C(C(C)C)(C)C)=O)CC1 C1(C(N2CCC(CCNC(c3cccc(OC(F)F)c3)=O)C2)=O)CC2CC1CO2 N1(C(c2cccc(Cl)c2OC)C(=O)NCCCCCC)CC2OC(=O)N(C)C2C1 N1(C(c2cnn(CCC)c2C)=O)CC(NC(c2cc(C)nnc2O)=O)CC(C)C1 N1(C(c2nc(COC)oc2)=O)C2CCC1CN(C(=O)CCC=CBr)C2 C12(SC)CCC(CN1Cc1scc(CC(=O)OCS(C)(=O)=O)n1)C2 C(=O)(C(C)(C)C(=O)NCC1C2CN(C(=O)CC3COCCO3)CC12)OCC C=CC(C)(CCOC)C(=O)N1CC2(CNC(C3CC3C(=O)OC)=O)CC1CO2 C1(C(C)C)CCCN(C(C23CC2CN(C(=O)C(C)N2CCCC2)C3)=O)CC1 c1(C(N)=O)ccc(CNC(C2C=CCCN2C(=O)CC2CC(=O)C2)=O)cc1 c1(C(=O)NCC2CCCN(C(c3c(C#C)c[nH]n3)=O)C2)cnc(C)cc1Cl Cc1ccc(C(CNC(C2CCCSC2)=O)NC(C2CC(C)(C)C2)=O)cc1 C1(F)(CNC(C2CCCO2)=O)COCCN(C(=O)C=CCN2CCOCC2)C1 C12CC(C1(C)C)NC2=O.c1(CNC(CSCCN(C)C)=O)cnn(CCF)c1 c1(C(=O)NC(CCNC(c2c(CC)nc(C)o2)=O)(C)CC)ccc(OC)c(C)c1 Cc1ccc(NC(C2(C)CCN2C(c2cc(C(F)(F)F)cc(Br)c2)=O)=O)c(Br)n1 C(CC(C(=O)N(C)Cc1nc(C)ns1)NC(c1nn(C)cc1C)=O)=CC c1(C(C(=O)N(CCNC(=O)CN(C)C(N)=O)CC)C)c(F)cccc1F N1(C(C(CC)C)=O)CC(NC(c2ccc3nncn3c2)=O)CC(F)(F)C1 C(=O)(C(C)CC=CC)N(CC(=O)NC(CC=C)CC)CCC O=C(C1CSc2ccccc21)OCC(c1ccncc1C1=COCC1)=O CC(CC(C)(c1ccccc1)NC(=O)CCCC(=O)N(C)C)C(=O)O CC1CCN(C(=O)COc2ccsc2)CCN1C(c1ccnc(O)c1)=O c1(C(=O)NC(C)CNC(C2COC(=O)O2)=O)ccc(C(=O)N(C)C)cc1 c1(C(=O)NCC#CCNC(C(C)OCC#C)=O)cc(C)n(-c2cc(C)on2)c1C Cc1cccc(C(O)C(=O)NC2CC(CNC(=O)CCc3ccco3)C2)c1 Cc1cc(C(N2CC3(CC(CC(=O)N(C(C)C(C)N(C)C)C)C3)C2)=O)ccc1O N1(C(Cc2ccc(C)cc2)=O)CCC(C(=O)N(C2CCC2)CC2CC2)=C(F)C1 Cc1ccc(C(=O)NC2CCCCC2NC(C2CCN(C)C2)=O)c(OC(F)F)c1 C1(C2CN(C(=O)C=C(C)Cl)C2)(NC(C2CC(C(F)(F)F)(OC)C2)=O)CC1 N(C1CCCCc2ccc(Br)cc21)C(N1C2(CO)CN(C)C(C2)C1)=O c1(N2CCC(CCOC)CC2)nc2c(c(=NCC3CCOC(C)C3)[nH]1)CCC2 C=CCC(C)(O)C(=O)NCC1CCOC1C(=O)NCCC(O)C(F)F c1(C(=O)NCC(CNC(CC2N(CC)CCOC2)=O)(C)O)cc(F)ccc1F C1(C(N(CC(C)NC(c2coc(O)n2)=O)C)=O)COCOC1 CCC(C(=O)N1CC(N2CCN(C(=O)Cn3nnc(C)n3)CC2)C1)C(C)(C)CC C(CN1C(=O)Cc2ccccc21)NC(c1cc2cccc(OC)c2o1)C c1(C(N2CC(CCCCNC(C(CNS(C)(=O)=O)OC)=O)C2)=O)ccc(Cl)c(Cl)c1 CCC(CC)C(C(=O)OC)Nc1ccc(NC(=O)C(C)C)cc1 C12(C(=O)OC)CC(C(N3CC(NC(=O)C(C)C4CCOC4)C3)=O)(C1)C2 Cc1c(C(N2CCC(CNC(=O)C(c3ccc(Cl)cc3)=O)CC2)=O)cccc1F Cc1cc(F)cnc1C(=O)N(C1CCN(C(C2CC(C)(F)C2)=O)CC1)C C1(C(=O)NCCC2CCCCN2C(=O)C=Cc2cscn2)CCOCC12CCC2 Cc1ccc(CNC(=O)CC2CC(C)N(C(C3CC(N(C)C)C3)=O)C2)cc1O c1(C(=O)NC2(CNC(=O)COCC3CC3)CCC2)oc2ccccc2c1CO Cc1nc(N(C)CC2CCCN2C(C2(C)CCC(F)(F)C2)=O)ncc1Br N1(C(C2N(C(c3c(NC)cccc3)=O)CCCC2)=O)CCN2CCCCC2C1 c1(C(N2CCC(C(C)NC(C(C)=CC)=O)C2)=O)ccc(Br)cc1O c1(OC)cc(C)c(C(=O)NC(CNC(=O)C2=CCCS2)C2CCC2)cc1OC CC(C)(CCCNC(=O)CNC(=O)C1CC1)NC(=O)CCOC1CCOCC1 C1(O)(C(C)NC(C(CC=C)C)=O)CCN(C(=O)COc2cncc(Cl)n2)CC1 c1(C(N2CCCC(CN(C(=O)CC3CCCO3)C)C2)=O)ccc(C2CC2)nc1O c1(C(N2CCC(C)C2C(N2CCSCC2)=O)=O)cc(O)cc(F)c1 C1(CNC(C(CC)C2CCOCC2)=O)CCC(C)(C)CN1c1nncs1 c1(C(N2CC3=C(CN(C(C(CCSC)O)=O)C3)C2)=O)ccc(F)c(C)c1C#N S(=O)(=O)(c1ccc(NC2COCCOC2)cc1Br)NCC1CC(C)(C)OC1(C)C CCC(CCC(=O)NC(C)(COC)CC)NC(C1CC1c1ccco1)=O c1(C(=O)NC(CC=C)CNC(=O)Cc2ncc(C)o2)cc(C)c2[nH]cnc2c1 C12(C(N3CC(NC(C(C)OC)=O)(CO)C3)=O)CC(C)(C1)OC2C N1(C(c2c(C)ccs2)=O)CC(C(N2CCSCC2C2CC2)=O)C2(CCC2)C1 O=C(CC(F)(F)Cl)NCCC1CN(C(=O)CSc2cccc(F)c2)C2CC12 c1(C(=O)NCCC(CNC(=O)CC2CC(F)(F)C2)O)cc(Cl)ccn1 Cc1cc(C(N2CC(NC(c3ccc(C)s3)=O)CC(C)C2)=O)n2ncnc2n1 N1(C(=O)NCCNC(=O)OC)CCOC(c2ccccc2)C1 C1(CC)C(C(=O)N(C)CC2CCCCC2)CCN1C(C1COCC1C(N)=O)=O C1(C(=O)Nc2ccc(SC)cc2)CCC(C)N(C(=O)Cc2cc(F)ccc2F)C1 C(=O)(C1=CCCCO1)N1CCC(NC(c2c(C)nn[nH]2)=O)(CF)C1 c1(N(CC(C)NC(=O)CN2CC3CC3C2)C)ccnc(C2CCCC2)n1 Cc1cc(C(=O)N(C)CC2CCCN2C(c2cscn2)=O)ns1 CCCCC(C(=O)N(C)CCOCCNC(=O)Cc1cncn1C)C(C)C N1(C(C2(COC)C=CCC2)=O)CCN(C(=O)C(C)N2CCCC2)C(CF)C1 c1(C(=O)NCCN(CC(C)O)C(c2cc(C(C)C)nn2C)=O)cnn2c1OCC2 C1(CC(C)NC(=O)COCC2(F)CC2)CN(C(=O)CC2(O)CCC2)C1 CC(C)C(C)(O)C(=O)NCCn1cc(C(=O)NOCCOC2CC2)nn1 N1(C(CCC(C)OCC)=O)C2CCC1CC(N(C(=O)C(=CC1CCCC1)C)C)C2 N(C(=NCCc1ccccc1)NCC(c1cn(C)cn1)(C)C)CCOCC#C Cc1ncc(F)c(N2CCN(C(C3CC(=O)N3)=O)C3CC23)n1 Cn1c(C(=O)NC2CC2NC(C2CC=CCC2)=O)nnc1S c1(CC(=O)NC2(C)CC(NC(CC(C)(C)O)=O)C2)c(F)cccc1F c1(N2CC(CNC(CC(C)n3cccn3)=O)OCC2)ncnc2[nH]ccc12 C(=O)(CCC(CF)CF)NC1C2CC(C(=O)NC(C)(CO)C3CC3)C(C2)C1 C#CCCCCCCC(=O)NC1CCCN(C(=O)CC(O)CCC)CC1 C(C(O)CC(=O)NC1CCC(=O)NC1)NC(C=C(CC)CC)=O C#CCC(C(=O)N(C(C)CNC(c1snc(O)c1Cl)=O)CC)C1CC1 C(N=c1[nH]c(=N)[nH]c(=NCC(F)(F)CC2CC2)[nH]1)C1N(C)CC(O)C1 c1(C(=O)NC2C(CNC(c3ccsc3)=O)CCCC2)nc2cncnc2nc1O CC(C)C(C)C(=O)NC1CCOC1C1CCN(C(C2(O)CC(F)(F)C2)=O)CC1 c1(C(=O)NCC2N(C(C=CC=CC)=O)CCOC2)ccc(F)c(Br)c1 C12(CNC(C3CC34CCOCC4)=O)CCCC1CN(C(c1sccc1Cl)=O)C2 S(=O)(=O)(c1ccc(F)cc1)N(C)CCNC1CN(C(=O)CC(F)(F)F)CCN1 N1(C(C(C)C2CCOC2)=O)CCOCC(NC(=O)CCOC2CCOCC2)C1 C1(c2nnnn2C2CC2)(Nc2ccc(CN(C)C)c(F)c2)COCC(C)(C)C1 Cc1cc(=NC(=O)C2c3ccccc3CN2S(=O)(=O)CCBr)[nH]n1C N1(C(c2c(CC)ncnc2)=O)CC(C(=O)NCC(C)CC(=O)OC)CCC1(C)C CCC(C)C(C(=O)NCC1(C(N2CC3C=CC3C2)=O)CCC1)N(C)C c1(C(=O)NC(C(C)NC(C2C(CC(C)C)C2)=O)CO)ccc(N2CCCC2)c(F)c1 c1(C(=O)OCC)cnn(C)c1C(=O)NCC1(NC(=O)CCN2CCC2)CCOC1 N1(C(CC2C(C)(C)CCO2)=O)CC(NC(C2CCC3CC2CO3)=O)C2CCCC12 N1(C(C(F)OC)=O)CCN(C(=O)CCSC(F)(F)F)C(C(F)F)C1 C(=O)(C1=C(F)CN(C(=O)C(C)(F)F)CC1)N1CC(C)C(CCO)C1 Cc1ccc(NC(C2OCCC2CNC(c2ccccc2)=O)=O)cc1C Cc1ccc(C(=O)NCC2C(C(=O)NCC3CCOC3=O)C2(C)C)nc1O N1(C(CCC(=O)NC)=O)CC(C(=O)O)C2(C1)CN(C(=O)C(c1ccccc1)O)C2 c1(C(N2CCC(O)(CNC(C(C(C)C)SC)=O)C2)=O)cccc2cc[nH]c12 N#Cc1c(NC(=O)CCC2CCCN2C(=O)C2=NNC(=O)CC2)cccc1Cl C1(C(=O)Nc2c(C)noc2C)COC2(CCN(C(=O)C=CC(C)(C)C)CC2)C1 C(C(CCC)NC(=O)Cc1nnc(C)o1)NC(C(C)OCC=C)=O CCCCC(CC)C(=O)N1CC(C(C)NC(c2ccc(C(C)=O)o2)=O)C1 C(CC(=O)N1CC2CCC1CC2)(C(F)(F)F)NC(C(C(=O)OC)C)=O c1(OCC(=O)NC2C3CN(C(c4cc(CC)oc4C)=O)C2C3)ccc(Cl)cc1Cl N1(C(C2=NOC(C)C2)=O)CC2(CCN(C(C3CCOC(=O)CC3)=O)CC2)C1 C1(C(=O)NCCC2OCCN(C(C3(C)CS(=O)(=O)C3)=O)C2)CCC2(CCC2)CO1 c1(C(=O)NCC2N(C(C3ON=C(C)C3)=O)CCCC2C)ccc([N+](=O)[O-])cc1Cl C(=O)(C1=CS(=O)CCC1)NC1CCCN(C(c2n(CC)ccc2)=O)CC1 Cc1ccc(NC(C2CN(C(C3CCCC34CCC4)=O)CC2F)=O)c(O)n1 c1(OC)cc(C(=O)NCCC(F)Cn2cc(Cc3cccnc3)nn2)ncc1Br c1(NS(=O)(=O)CCc2cnoc2)cccc2c1OCCC2 C1(C(C)(C)NC(=O)CCNC(=O)C=CCl)CCN(C(=O)CN2CCOCC2)C1 N1(C(C=CC)=O)CCN(C(c2conc2Cc2ccccc2)=O)CCC1C N1(C(C2C(C)C2)=O)CCN(C(C2CN(C)C2)=O)C(CC2CC2)C1 C12(CNC(c3c(C)nc(C(C)OCC)s3)=O)CCC(C1)N(C(C1(O)CCC1)=O)C2 C1(CC(=O)NC(c2ccc(C)s2)CO)CCn2cncc2C1 CCCCC(C)CCC(=O)NC1CCC1C(=O)Nc1cccc2c1CCO2 CC1CN(C(=O)CC(C)(C)c2ccc(F)cc2)CC1NC(c1cc(C#N)cs1)=O c1(OC)ccc(C(F)F)cc1C(=O)NCC12CC1CN(C(C1CCC(=O)C1)=O)C2 C1(C(=O)NC2(CCCC)CC2)COCCN(C(c2ccnc(OC)c2)=O)C1 N1(C(C(C(CC)CC)C)=O)CCC(NC(=O)Cc2c(C)cnn2C)CC(C)(C)C1 CC(C)C(C(=O)N1CCCCCC1CNC(=O)C(C(C)O)N(C)C)C(C)C C#Cc1cccc(NC(=O)NC2CC3(CSCc4ccccc4)COC2C3)c1F C=C=C(C)CC(=O)N1CCC(N(C(C2(N3CC4CC4C3)CC2)=O)CC2CC2)CC1 Nc1cnc(C(N2CCC(O)(CCNC(c3cnncc3O)=O)CC2)=O)c(Cl)c1 C1(COC)CN(C(=O)C(C2CCOCC2)F)CCN1C(c1nc(Cl)cs1)=O C(=O)(CN=c1ccc(Cl)n[nH]1)N1CCN(C(CS(CC)=O)=O)C2(C1)CCC2 C1(C(=O)NCC(CC)N(C)C(c2[nH]nnc2C)=O)CC2(CCO1)CC2 c1(OC)ccc(C(N2CC(C)(NC(C3CCCC(F)C3)=O)C2)=O)cc1 Cc1cc(O)cc(C)c1NC(C1CCC(NC(=O)CCC(F)(F)F)C1)=O Cc1cc(C(N2CC(NC(=O)CCCc3ccc(Br)cc3)C(F)C2)=O)c(C)o1 CC1(C)CCC(CO)N(C(C2CN(C(=O)Cn3cnc(=N)[nH]3)CC2(F)F)=O)C1 C1(C(=O)NCC(CNC(=O)C(c2cccnc2)O)CO)CC12CCSCC2 CC1(C)OCCC1CNC(c1cccc(O)c1)Nc1ccc(CO)cc1 N1(C(CN(S(CC)(=O)=O)C)=O)CCN(C)C(CNC(=O)COC2CCOCC2)C1 N1(C(C(C)OCCC=C)=O)CCOCC(F)(CNC(c2cc(C(F)F)cs2)=O)C1 C1(CNC(c2nn(CC)nc2C)=O)CC2(CC(NC(C34CCC(CC3)C4)=O)C2)C1 C1(NC(C2(COC)CC(F)(F)C2)=O)CCN(C(c2snnc2C)=O)CC1O C(=O)(C(O)CCCc1ccccc1)N(CCCNC(C1N(CC)CC1)=O)C N1(C(c2ccc(C#C)cc2)=O)CC2OCCN(C(C3CC3(C)C(F)F)=O)C2C1 C=CC(CC(=O)N1CC(NC(c2csc(C#N)c2)=O)C(O)C1)c1ccccc1 c1(C(=O)NCCNC(c2cccc(OC)n2)=O)cccn(C2CC2)c1=O C1(N(C)C(c2ccoc2C2CC2)=O)CN(C(C2CCCC23CC3)=O)CC1O C#CCCCC(C)C(=O)N1CCCC1C(=O)NCCc1ncc(C)o1 C(c1ccccc1)=CCOCC(=O)NCCN(C(CC1(CC)CC1)=O)C1CC1 c1(C(N2C3C(NC(CCNC(C4C(C)=C4)=O)=O)C(C3)C2)=O)ccc([N+](=O)[O-])c(C)c1 O=C1CCc2cc(CC(=O)NC3CC3c3ccc(F)cn3)ccc2N1 C1(NC(c2cc(SC)oc2C)=O)CCSC12CN(C(=O)C(c1ccccc1)F)C2 N1(C(c2nnc(CC)s2)=O)CCN(C(=O)C(CC(C)C)OC)C(CO)C1 C1(C(N2C(C)CCCC2)=O)CC(c2ccccn2)=NO1 N1(C(C=CC)=O)CCCC(C2CCN(C(=O)C(CC3CC3)CC3CC3)C2)C1 c1(-c2n(CC=C)nc(COC)n2)ccc(CC)c(CCCC)c1Cl C1(N(CC)CC)CCN(C(c2ccc(CNC(C3CCC3(F)F)=O)o2)=O)C1 C(C(C(C)(C)C)NC(=O)CCc1ncccc1C)NC(C(=O)NCC)=O CCC(C(=O)N1CC2CCC2(NC(=O)CCc2nnc(O)nc2O)C1)C(C)C CC1OC2(C)CC1(C(N1CCC(CNC(c3ccnc(F)c3Cl)=O)C1(C)C)=O)C2 C1(C(=O)NCC(C)(CO)NC(c2cccc(C3CC3)c2)=O)CCN(C2CC2)C1=O c1(C(N(CCC(C(C)C)NC(C(C)OCCC=C)=O)C)=O)ccnc(F)c1OC c1(OC)ccc(CC(N2CCC(C)C2CNC(=O)CS(N)(=O)=O)=O)cc1O c1(NC(C2C3CN(S(CC)(=O)=O)C2C3)=O)ccc(S(C)(=O)=O)nc1C c1(CC)nc(O)c(C(=O)NCC2CCN2C(=O)CC2CC3(CCC3)C2)cc1C N1(C(CCCSC)=O)CCC(NC(c2cnccc2C(C)(C)C)=O)C(F)C1 C1(NC(C(C)SC(C)C)=O)CCN(C(=O)CCNC(=O)CO)CCC1(F)F C(C(O)CC(=O)N1CC(F)CC1CN(C)C(c1cc(CO)n(C)n1)=O)N(C)C C1(C(N2CC(CC(=O)NCCc3cscn3)OCC2)=O)CC2(CCO1)CC2 N1(NC(=O)OC(C)(C)C)CCCC1CNC1CCCN1S(C)(=O)=O C1(C(=O)NCCC(C)(C)OC)CCCC(NC(=O)C=Cc2cccc(C)c2)CC1 c1(CC)cc(C(N2CC(NC(c3cc(F)c[nH]3)=O)C(F)C2)=O)cc(C)c1 c1(C(=O)NC2C(NC(c3nc(C(C)C)sc3)=O)COC2)ccnc2ccccc12 O=C(C(F)C(F)(F)F)NCc1ccc(NC2(C3CCCO3)CC2)cc1 N1(C(C(C)C(C)(C)C)=O)CC(NC(c2ccccc2[N+](=O)[O-])=O)CC(C)(C)C1 c1(CCCC(=O)NCC2CC(F)(CNC(CC(=C)Br)=O)C2)nnc(C)n1C c1(OC)c(Cl)ccc(C(N2CCCN(C(=O)CC3C=CCC3)C(CO)C2)=O)c1F C1(NC(CCNC(=O)NC)=O)CC2C(NC(c3cc(C)oc3C)=O)C2C1 c1(C(N2CC(OCCNC(C(CC)Sc3ccncc3)=O)C2)=O)nnn(CC)c1C c1(CC)cccc(C)c1NC(=O)Nc1ccc(-n2cccc2)nc1 C(=O)(CCCCCC(C)O)NCC1CC(O)(CNC(c2cc(CC)nn2C)=O)C1 C1(C(=O)NC(CCNC(C(C2CC2)OC)=O)C)CNC(=O)N1 C1(F)(C(=O)NCC2C(C)(C)C2CO)CCCN(C(=O)CC2CCC(=O)N2)C1 c1(-n2cc(CCC(=O)C(C(N3CCC(SC)C3)C)=O)nn2)c[nH]c2ccccc12 c1(C(=O)NCC2CC(CNC(CCC)=O)OC2)cc(F)c2[nH]nnc2c1 c1(CC)cn2c(C(=O)NCCC3CN(C(=O)C(C)=O)CC3C)cccc2n1 N1(C(=O)OCC)CCCC(C(=O)N(CC#CCNC(=O)C=CS(C)=O)C(C)C)C1 CCC1=C(C(=O)NCC2(O)CC(CNC(=O)C(C)(C)CC#N)C2)CCCO1 C1(C)(C(N2CCC(C)(CNC(Cc3c(C)cco3)=O)CC2)=O)CCC(=O)N(C)C1 C(=O)(C(CN(C)C)C(C)C)NC(C(N1C(CC)(CC)CC1)=O)CC1CCCC1 c1(C(N2CC(O)CC2COC)C(=O)NCC(=C)C)c(Cl)ncn1C c1(C(=O)NC2CC3CN(C(CCOC)=O)C(C2)C3)cccc2cccc(OC)c12 N1(C(c2c(CC)nco2)=O)CCOC(C(C)NC(c2ccccc2C2CC2)=O)C1 CC#CCCC(=O)NC(CNC(C1CCC(COC)CC1)=O)(CC)CC c1(C(=O)NC(CNC(c2cnn(CCC)c2Cl)=O)(C)CO)ncnc2c1CCC2 C1(C)(C(=O)NCCC(=C)C)CCN(C(=O)C=C(C)c2ccccc2)CC1 CC1OC2(C(N3CC4CC(NC(c5cnnc(O)c5)=O)C3C4)=O)CCC1CC2 C(c1nc2ccccc2o1)=CC(=O)NC1CCN(C(C=C(CC)C)=O)CC1CO c1(SCC(CC)N(C)C)nnc(-c2ccc(OC)cc2)n1CCC#N N1(C(c2c(SC)scc2)=O)C2CCC1C(CNC(=O)C(C)CC(F)F)C2 Cc1ccc(C23CC(C(=O)NCCc4cc(C)n(C)n4)(C2)C3F)cc1 n1(C(C)C)ncc(F)c1C(N1CCCC(C(C)NC(=O)C=Cc2ccco2)C1)=O c1(C(N2C(CNC(C3(O)CC3)=O)CC(C)(C)C2)=O)cc(Br)c2c(c1)OCO2 C12(NC(=O)NC(=O)C(F)(F)Br)CCOC1CCOC2 N1(C(CCOCCCOC)=O)CC2CCC(C1)N2Cc1ccc(C)cc1F N1(C(c2cnc(CC)s2)=O)CCC(C)(NC(c2n[nH]c(C(C)(C)C)n2)=O)C1 N1(C(CCC(C)OC)=O)CCN(C(c2ccc(C)cc2N)=O)CC1C1CC1 c1(CNC(C(C(C)SC)O)=O)c(C)nn2c1CN(C(=O)CCCSC)CC2 c1(C(=O)NCC2CCC(NC(Cc3cc(C)on3)=O)C2)c(Cl)ccc(F)c1C N1(C(c2c(CC)nn[nH]2)=O)CCC(C)(CCNC(=O)C=Cc2ccoc2)C1 N1(C(c2c(C)nccn2)=O)CCCC12CCCN(C(=O)Cc1ccc(Cl)cc1)C2 C1(C(F)(F)F)(C(=O)OC)CCN(C(=O)NC(c2occc2C)C)CC1 CCC(C(=O)NCC1(NC(C2(C)CCCCC2)=O)CCOC1)C(C)(F)F C1(CC(=O)NC(CC#C)C)CC(C)N(C(=O)CSCCCC)C1 C1(C(=O)NC(CNC(C2(C=C)CC2)=O)CC)CC(F)C(=O)N1C C1(C(=O)NCC23CC(C)(C2)C3)CCCN(C(C2CCCN(S(C)(=O)=O)C2)=O)C1 C12(NC(c3nc(CNC(C)=O)sc3)=O)CC1CN(C(=O)CC(O)CN(C)C)C2 C1(F)(C(=O)NC2(CC)CCOCC2)CCCN(C(c2cc(C)c(C)o2)=O)C1 CC(C)CN=C(NCC1(CC(F)(F)F)CC1)N1CCCC(NC(=O)CO)C1C C=Cn1nccc1C(=O)NCC1CC(NC(=O)CCNC(=O)CO)C1 C1(O)(C(=O)NC(CCC)CNC(c2c[nH]nc2Cl)=O)CCC(C)(C)CC1 C1(NC(C2CC(O)(CC#C)C2)=O)CN(C(=O)Cc2ccsn2)CC(C)(C)C1 C1(NC(N(CCC)CCC)=O)CC(CN2CC(CF)C2)CO1 C1(NC(c2cc(C)on2)=O)CCN(C(C2CCC=CCC2)=O)CCC1CO c1(CC(=O)NC2(CN(C)C(C3CCCC(F)(F)C3)=O)CC2)cc(Cl)cc(Cl)c1 c1(C(=O)NCC2CC(NC(=O)CCF)C(O)C2)cccc2c1COC2 C1(CC(=O)N(CC)Cc2cccnc2)CCCN(C(=O)CP(C)(C)=O)C1 c1(C(N2C(CCNC(c3n(C)ncc3)=O)COCC2)=O)cnc2c[nH]nc2c1 CC1CCC(NC(=O)CCC2CC(C)(C)CO2)CN1C(=O)CCn1cncn1 c1(C(=O)NCC(CO)NC(c2c(C)occ2)=O)ccc(F)c(C)c1N C1(NC(CCc2cn(C)nc2)=O)CC2(C1)CC2C(=O)N(C1COCC1O)C1CC1 N1(C(C(CC)=CCCC)=O)CC(NC(c2cc(COC)on2)=O)C(C(F)F)C1 CC(C)CC(CNC(C1(O)CC(C)(C)C1)=O)NC(=O)CCC(C)N(C)C c1(NC(c2c(C(=O)N=c3ccn(C(F)(F)F)[nH]3)n[nH]c2)=O)ccc([N+](=O)[O-])cc1Br C1(C2CC2)(CNC(C(CCCC)N(C)C)=O)CCN(C(c2cc(C)c(C)[nH]2)=O)C1 O=S(=O)(c1ccc(NC2CC(n3ccnn3)C2)nc1)NC(CO)C1CC1 N1(C(C2(C)CCC(=O)C2)=O)CC23CCCCC2(C1)CN(C(=O)Cc1ccsn1)C3 c1(SC)ccc(C(N2CC(F)CC2C(c2cc(C3CCCCC3)no2)=O)=O)cc1 c1(NC2C(NC(c3c(CC)ccs3)=O)CS(=O)(=O)C2)cc(C#N)nc(C)n1 CC(CCCNC(c1cc(Cl)cs1)=O)NC(=O)Cc1nc(C(C)C)n[nH]1 C1(NC(CC(CCC)CC)=O)CC2CCCC(C1)N2C(=O)C(C1CCOCC1)F C(c1ccccc1C)=CC(=O)NC(C1CCCC1)CNC(c1c(C)cn(C)c1)=O C1(NC(CCOCC#C)=O)CCC(C)(NC(=O)C(F)Cc2ccccc2)CC1 N1(c2cc(NC(c3ccc(F)cc3)C)ncn2)CCc2ncn(C)c2C1 CCCC(C)(CC)C(=O)N1CCN(C(=O)CCn2cnnn2)C(COC)C1 C=C1Cn2c(C(N3CCN(C(c4c(C)ccn4C)=O)CC3CC)=O)nnc2S1 c1(CC(N2CCCC(C)(NC(c3c(CC)nns3)=O)C2)=O)ccc2nsnc2c1 C1(C(=O)NCC(CNC(=O)CCCn2ccnc2)O)CCCC2(CCOCC2)O1 c1(CC(=O)NC(CCNC(C(COC)N(C)C)=O)C)ccc2c(c1)COC2 C12(C(=O)NC(c3ccc[nH]3)C)CC(c3cccc(C(C)O)c3)(C1)C2F C1(NC(C(C)=C(C)C)=O)CC2(CCN(C(c3cccc(C4(C)CCO4)c3)=O)C2)C1 C1(C(=O)NCCCc2c(C)n[nH]c2)CN(C(=O)Cc2cnoc2)CC(C)O1 C1(C(N(CC)CC2CCCN2C(c2snc(C)c2N)=O)=O)C2CN(C)CC12 C12(CNC(CN(C)C(N)=O)=O)CC(C1)C(NC(c1cnc(S)n1C)=O)CO2 c1(C(N2CCC(C(C(C)C)NC(C3CCNC3=O)=O)CC2)=O)ccc(Cl)nc1O C1(C(C)C)CN(C(c2nc(Cl)cs2)=O)CCCN1C(c1cc(C2CC2)[nH]n1)=O N1(C(CC2(N(C)C)CCCC2)=O)CCC(CCCNC(C2CCOC2)=O)CC1 c1(C(=O)NC2CC(C)NC2)ccc(S(=O)(=O)N(C)CCC2CCCCN2C)cc1 C1(C(=O)NC2(CCCNC(C3C(CC)CCC3)=O)CC2)CC(F)C(=O)N1 Cc1nnc2n1CCN(C(C1CC(F)(F)CN1C(c1cc(Cl)n(C)n1)=O)=O)C2 c1(C(C)NC(=O)C(=O)NCc2cc(Br)ccc2O)nc2ccccc2n1C(F)F CC1CCOC(C(=O)NC(C)(C(=O)NCC(c2cnc[nH]2)C)C2CCC2)C1 C1(CC=C)(C(=O)N(CC(O)COC)C)CCN(C(=O)CCOCC)C1 n1(CC)cc2ccc(C(=O)NCC(C)NC(c3cncc4ccsc34)=O)cc2n1 c1(CNC(=O)NCC)ccc(S(=O)(=O)NCC2(CC(F)(F)F)CC2)cc1 C1(CC(=O)NCC(CCC)C)CN(C(c2cccc(CC#N)c2)=O)CC12CC2 CC(C)C(O)C(C)(C)C(=O)NC1CC(CNC(c2ccc(F)c(F)c2)=O)C1 Cc1cc(-n2ccc(C(=O)N(CCC(C)(C)O)C)n2)ccc1Cl CC1(C)CCC=C1C(=O)N1CC2CCCC2(NC(=O)Cc2ccccc2Br)C1 N1(C(C(C2CCOCC2)OC)=O)CCN(C(=O)CCCN=[N+]=[N-])C(C2CCC2)C1 C(=O)(C1CS(=O)(=O)c2ccccc21)N(C1CCCC1)CCNC(c1csnn1)=O C12(CC)CN(C(C3(SC)CC3)=O)C(CNC(=O)CC3CCCC(=O)N3)(C1)C2 CN1CC(O)CC1C(=O)NC(C)(C)CN1CCN(C(C2CN(C(N)=O)C2)=O)CC1 c1(C(=O)NC(CC)CNC(=O)C(C)CC2CC2)noc2cc(F)ccc12 c1(C(=O)NC(Cn2cc(CNC(C(CC)F)=O)nn2)C)cccc(Cl)c1O N1(C(CSCC(C)C)=O)CC2CCCC(C1)N2C(=O)CSc1ccccc1Cl CCCC(C(=O)NC(Cn1ccnn1)C(=O)NCCCCS(C)=O)OC c1(C(=O)NC(c2ccc(F)cc2)C(=O)NC)cn2c(n1)CCCC2C(=O)O N1(C(C(CC)OC2CCCC2)=O)CCc2c(ncn2C)C12CCN(CCOC)C2 N1(C(c2occ(C)c2)=O)CCN(C(=O)CC2(O)CCCC2)CC1C(C)(C)C C12(C(=O)NC3(C)CCOC3)C(NC(=O)C(c3ccccc3)=O)C3CC1C2C3 C(=O)(CC(C)(CC)C(=O)OC)NCc1cccc(NC(C(F)=CC)=O)c1 C#CCC(CC(=O)NC(C1CSC1)C)NC(=O)CNC(C1CC1C)=O c1(CN2CC3N(C(c4cccc(O)n4)=O)C3C2)c[nH]c2ncc(Br)nc12 Cn1nc2c(c1C(=O)NC1CCCCC1NC(c1ccc(=N)[nH]n1)=O)CCC2 N1(C(C(C)=CC2CC2)=O)CC(F)(F)CC1CCNC(=O)Cc1scnc1C c1(CC(=O)NCC2(NC(C3CC3F)=O)CCC2)ccccc1Br c1(OC)cc(C(=O)NC2CN(C(C3CCCC3)=O)C2)cc(Br)c1OC(C)C c1(C(N(CCCNC(C2(C)CCCN2C)=O)C)=O)cnc(S(C)(=O)=O)s1 c1(C(=O)NC(CNC(C(C)N2CCC2)=O)C2CCC2)cc(C(N)=O)co1 c1(C(=O)NC(CNC(C(C)NC(c2ccoc2)=O)=O)C2CC2)cc(Cl)cnn1 C1(C(=O)NCc2c(CC)noc2)CC(NC(=O)C(C)(C)NC(=O)OC)CCO1 C(=O)(C1=CC2(CCN(C(C3CCSC(C)C3)=O)C2)C1)NC1CCC(CC)CC1 C1(C#CC(=O)N2CCC(C(C)(O)CNC(=O)Cc3cc(C)on3)CC2)(CC)CC1 C1(CNC(C(=O)NCC2(CCC)CC2)=O)CC(C)(C)CN1 C1(NC(c2cc(Cl)c(Cl)[nH]2)=O)CN(C(=O)C(F)F)CCC1c1ccccc1 c1(C(N2CC(O)(CNC(Cc3scc(C)n3)=O)C2)=O)cc2c(F)ccc(F)c2[nH]1 C1(NC(CCOc2ccc(C)cc2)=O)CCN(C(c2ncc(F)cn2)=O)CC1C C1(CCC(=O)OC)CCC(C(=O)NCC(C)(O)CNC(=O)C(C)C)O1 C(=O)(C1CCc2c[nH]nc21)NC(CC=CC)C(=O)O C1(NC(=O)CC2CC=CCC2)CC(F)CN(C(c2cc(Cl)ccc2O)=O)C1 N1(C(C(CC2CN(C(C=C(CC)CC)=O)C2)F)=O)CC(O)CC(C)(C)C1 c1(NC(C23N(C(C(C)NC(CC)(C)C)=O)CCC2C3)=O)cnc(C)c(C)c1 N1(CC(=O)N(CC(N2CC(C)(C(=O)OC)C2)=O)CCC)CCCCC1=O c1(C(=O)NCCC2CN(C(c3[nH]nc(OC)c3Cl)=O)C2)n[nH]c(C)c1[N+](=O)[O-] Cc1cc(C(=O)Nc2cccc(NC(c3cc[nH]c3C(C)C)=O)c2)cn1C c1(OC)cc(CNc2ccccc2N2CCC(CO)C2)ncn1 CC1CCC(NC(c2ccnc(S)c2)=O)CN1C(=O)CN1CCN(C)CC1 c1(C(=O)NC(CC(C)C)C(F)F)c2ccccc2nn1C CCCC(C(=O)OC)C(=O)N1CC(NC(c2cc(C(C)C)[nH]n2)=O)C(N=[N+]=[N-])C1 N1(CCC)CCCC1C(=O)NCC(c1cn(C)nn1)NC(=O)COCCCOC N1(C(C2ON=C(CC)C2)=O)CC(N(C(=O)C(c2ccccc2)=O)C)C2(CC2)C1 CN1CCOC(C(=O)N(CCCNC(C2CNC(=O)N2)=O)CC2CCCC2)C1 c1(CC2(Cc3nc(-c4ccc(OC)cc4)oc3C)CCC2)cc(Br)cc(Cl)c1F CC(C)C(CNC(c1cccnc1O)=O)C(=O)NC(C(N)=O)C(C)O N1(C(c2cc(CC)oc2C)=O)CCC2CCN(C(=O)CCCN(C)C(C)=O)CC12 N1(C(CNC(CNC(C)=O)=O)=O)CCC(F)(CNC(c2cscc2Cl)=O)C1 C(c1ccc(C)cc1)=CCC(=O)NCCN(C(=O)CCC(C)N(C)C)CCOC N1(C(C2(SC)CC2)=O)CCC(n2cc(-c3csc(N(C)C)c3)nn2)C1 C(CCC(C)C(=O)N1CCC=CC1C(=O)NCCCC(=O)NO)OC C1(CC(=O)NCC2(OC)CN(C(C3CCCS3(=O)=O)=O)C2)CCN(C(C)C)CC1 CCC(C(=O)NCCCC(C)NC(C1(N(C)C)CC1)=O)C(C)C O=C(CCCC(F)(F)C(F)(F)F)NC1CCN(C(C2(F)CCC2)=O)CCC1CO N1(C(c2c(C)nccc2)=O)CCC(C)C(NC(c2cc(C)n(CC(F)F)n2)=O)C1 C1(NC(CCCOC(C)C)=O)CC2CN(C(=O)CCc3ccc(F)cc3)CC2C1 c1(C(=O)NCCCCN(C(CS(=O)(=O)NC)=O)C)cc(F)ccc1C(F)F c1(C(=O)NCC(C2CCCC2)NC(=O)CCc2ncc[nH]2)cc(Cl)ccn1 c1(C(=O)NCCCCCNC(C2N(CC)CC2)=O)cnc(C(F)(F)F)cc1C C1(NC(=O)NC(C)C(C)(C)F)CCN(c2ccccc2C(F)(F)F)C1=O c1(C(=O)NCCC2CCCC2)ccc2cnn(Cc3ccccc3)c2c1 N1(C(CC=C=C)=O)CC(NC(=O)CCc2ccccc2OCC)CC2(CCC2)C1 C(=O)(C(C(C)(C)C)N(C)C)N1CC(F)(CNC(C(C)(C2(C)CC2)OC)=O)C1 c1(C(N2CCC(N(C(CC)=O)C)C2)=O)cccc2c1CCCCC2 C(CCC)(C(=O)N1CC(O)(C(F)C(=O)NCC(=O)N(C)C)C1)=CCC C1(NC(C2(C=C)CCC2)=O)CCCCC1NC(=O)CCN(C(CC)CC)C C1(C)(C(=O)NCC2CCN(C(CC(C)(C)OC)=O)C2)COCC1(F)F C(N=c1nc2[nH][nH]cc-2c(O)n1)C1(NC(CC(n2ccc(C)n2)C)=O)CCCC1 N(C1CCc2cc(CNC(C3(C#N)CC(=O)C3)=O)ccc21)C(C1(C)CC1(Cl)Cl)=O C=CC1(C(=O)NCCC2(O)CN(C(c3ccc(CCC)[nH]3)=O)C2)CCC1 N1(C(C(C=CC)O)=O)C2CCC1CC(NC(c1ccc(OC)c(CC)c1)=O)C2 N1(C(CCCC#C)=O)CCCC2(CC(NC(=O)C=CC(=O)N(C)C)C2)C1 c1(C(=O)NC2CN(C(c3[nH]cc(CC)c3)=O)CC2C(F)F)cccc2[nH]ccc12 C1(CC)C(=O)N(C)CCN1C(C1CN(C(c2ccc[nH]2)=O)CCC1O)=O CCCCC(C)CCC(=O)N1CCC2C(C1)CN2C(c1cc(Cl)c(F)c(Cl)c1)=O N1(C(c2cn(CCC)nc2)=O)CCCC(NC(C2C=CC=CC=C2)=O)C1 c1(C(=O)NCC(CNC(C2(CC=C)CC2)=O)F)cc(Cl)ccc1Cl C1(C(=O)NC2CC(OCC(=O)Nc3cccc(F)c3)C2)CC2CCCC2C1 C#CCC(CC(=O)NCC1CC2(CC2)C(=O)O1)NC(c1cc(Cl)c[nH]1)=O CCC(C)(C#N)C(=O)NCC(=O)NC(CCO)CC(C)C N1(C(CNC(c2cn(-c3ncc(Br)s3)nn2)C)=O)CCN(C(=O)C2CC2)CC1 c1(C(N2C(C)(CNC(C3C(C)(C)C3)=O)CCC2)=O)cc(Br)cnc1N c1(CC)[nH]nc(C(=O)NC2CC3CC2CN(C(=O)C(CSC)OC)C3)c1[N+](=O)[O-] c1(CC(=O)NC2C3CN(C(C(C(=O)OC)OC)=O)CC32)cc(C)cc(F)c1 C1(NC(CCCOCC=C)=O)CC=C(C(=O)NC2(C)CCC(C)(C)C2)C1 N1(C(C2(O)CC(C)(C)C2)=O)CCCC(CCNC(c2cccnc2F)=O)CC1 C1(NC(c2ccc(CO)o2)=O)CCN(C(C2CCCCC2O)=O)C12CCCC2 Cc1cc(=NCCCCC#N)[nH]c(=NCCOCCS(N)(=O)=O)[nH]1 c1(C(=O)NC2(CO)CN(C(COCc3cc(C)no3)=O)C2)cc(Cl)c(C)cn1 C1(C(=O)NCC2C(C)CCN(C(CCCC(C)O)=O)C2)CS(=O)(=O)CC(=O)N1 C(=O)(C1=CCc2ccccc21)NCCCC(C)NC(C(CC(C)C)NC(C)=O)=O C(=O)(C(CO)C(F)(F)F)NC1CCCC(C(=O)NC2(CCC)CCC2)CC1 Nc1nccnc1C(N1CCCC1C=CC(N1CCCC(CCCO)C1)=O)=O N1(C(CSCCC)=O)CC(NC(=O)C=CC(=O)OC(C)(C)C)C(C(F)(F)F)C1 C1(C)(C(N2CCC(C(N3CCN(C(=O)OCC)CC3)=O)CC2)=O)CNCCC1O Cc1cc(N(C(C)CCNC(=O)COCc2cc(C)on2)C)n2nc(C)cc2n1 N1(C(CN(C(C(CC)C)=O)C)=O)CCN(C(C2C(C)(C)C2(F)F)=O)CC1 CC1CC=C(C(=O)N2CCC2CNC(=O)Cn2ccc(Br)n2)CC1 C1(NC(CSCCC)=O)CCN(C(=O)CCc2n[nH]c(=N)s2)CC1O C(C)(C)(CC(F)C(=O)N(C)CCC1CCC1)NC(c1cncc(C)n1)=O C1(CNC(C=CSC)=O)CC2CCC1N2C(=O)COC1CCCCC1 c1(OC)ccc(CC(=O)NCC2CC(NC(=O)CC=C(C)C)C2(C)C)c(F)c1 C12(CNC(CN(C(COC(C)C)=O)C(C)C)=O)CCC(CC1)CC2 Cc1cc(C(C)C(=O)NCCCCN(C)C(C2C3CCC(F)(F)C23)=O)cc(F)c1 c1(CC(=O)NC2CCN(C(C=CC)=O)CC2O)nnc(O)c2ccccc12 Cc1cc(CN2CC3CC3(C(=O)NCc3cccc(C4CC4)c3)C2)cc(C)c1Br C1(C(=O)NC2CN(C(c3c[nH]c(=NCC)s3)=O)CC2(C)C)CCCC2C1C2(F)F N1(C(C(CC)COC)=O)CCCC(C)(C)C1C(=O)NC1CCC2CCC12 C12(C(=O)NCCc3ccc(C(=O)NCc4cnc[nH]4)cc3)CC=CCN1CCC2 N1(Cc2ccc(OC)c(SC)c2)CCC2(CCC(O)C2)C1 CCCCC(O)C(=O)N1CCOCC(NC(c2cc(C(=O)OCC)n(C)n2)=O)C1 C1(NC(c2nc(CCC)oc2)=O)CC(N=c2nc(CCN(C)C)[nH]s2)C1 C(=O)(C(C)(C)C1CCN(C(=O)CC2CC3(CC3)C2)C1)NCC(CC)N(C)C c1(CC(=O)NC(C2(O)CN(C(=O)CCC(C)(C)O)C2)C)ccc2c(c1)OCCO2 Cc1ccnn1C(C)C(=O)NC1CC(CNC(c2csc(C(C)(C)C)n2)=O)C1 Cc1cc(C(N2CC3CC2C3C(=O)NCc2ccccc2O)=O)nc2nccn12 O=C(CCCCCn1cc(-c2ccc(Cl)cn2)nn1)NC1CC2CCC1(C(=O)O)C2 C1(NC(CC2(OC)CN(C(CCSCC)=O)C2)=O)CCCN(C)C1C c1(C(=O)NC(CC)CNC(=O)Cn2cn[nH]c2=N)snc2c1CC(C)(C)CC2 C(CCCCCC(C)C)n1cc(C2N(C(CC(C)(C)OCC)=O)CCCC2)nn1 N1(C(Cn2ncc(C)c2)=O)CC2CCN(C(C3COCC3C(F)F)=O)CCC2C1 c1(C(=O)NC2C(NC(C(C#C)(C)C)=O)CCCC2)cc([N+](=O)[O-])c(C)cc1Cl c1(C(=O)NC2CC3CC2N(C(C2CCO2)=O)C3)cc2c(nc1O)CCCCC2 C1(NC(Cn2nc(C)c(C)c2C)=O)CC12CCC(NC(C1CC1C(F)F)=O)CC2 n1(CC(=O)NC(C2CN(C(C3CC3c3ccco3)=O)C2)C)nnc(C2CC2)n1 C=CC(C)(CCOC)C(=O)NC(C)C(=O)NC(C)CCC1CC1 C(=O)(CC(C)(C(F)F)N(C)C)N(C)CC1CCCN(C(=O)CC2=CCCCC2)C1 C1(NC(C(C)OCC2CCCO2)=O)CN(C(c2c(F)cncc2Cl)=O)CCC1F c1(NC(CC)=O)ccccc1C(=O)NCC1CN(C(C2(C)CC=CCO2)=O)C1 N1(C(=O)NCCC2CN(C)CC(C)O2)CC(c2ccccc2)C2CCCC12 c1(-c2nn(CC)c(C(F)(F)F)c2)ccc(N(C)C)cc1F C=CCC(CC(C)C)C(=O)N1CC(NC(c2cn3cc(Cl)cnc3n2)=O)C(C)C1 CCCC(C)(O)C(=O)NC(CNC(C1(C)CCN(C(C)=O)C1)=O)C(C)C c1(OC)ccc(C2(CNC(=O)Nc3cnc(OCCO)cn3)CC2)nc1 Cc1[nH]nc2c1CCC(C(=O)N(CCCCNC(C1CC3COCC3C1)=O)C)C2 C1(OC)CN(C(=O)C(F)(F)c2cnccn2)CCC1NC(C1CCSC1)=O C(=O)(CC(C(C)(C)C)NC(=O)CC1(N(C)C)CC1)NC1(CC)CC(C)(C)C1 c1(C(=O)NC(C#C)C)noc2c1CC(NC(c1nc(C)c(C)[nH]c1=O)=O)CC2 Cc1ncc(C(=O)NCC2CCN(C)C2)c(Cl)c1Br c1(C(=O)NCCOCCCNC(C(CCSC)O)=O)ccc(S(C)=O)cc1 C1(C)(NC(C=C(C)CN2CCOCC2)=O)CCN(C(c2ccno2)=O)C1 N1(C(c2c(C)ncs2)=O)CC(NC(c2ccsc2Br)=O)C(O)C1 c1(-c2nc(CCCCCCNS(C)(=O)=O)on2)ccc(F)c(S(C)(=O)=O)c1 CC1CC(NC(=O)CNC(=O)C2CC2)CCN1C(c1c(Cl)nsc1Cl)=O N1(C(C2(OCC)CC2)=O)CCCC(C(=O)NC2CC(=O)NC2=O)CC1 CC1(C(=O)NCC2(O)CC(NC(C3(N4CCCC4=O)CC3)=O)C2)CC=CCC1 c1(C(N2C(C(=O)Nc3c(CC)cc(Cl)cc3)CSCC2)=O)ccn2ccccc12 c1(OC)ccc(CN2C(C(N3CCC(N4CCCC4)CC3)=O)CC3CC23)cc1F c1(C(=O)NCC(C)(C2CC2)NC(C#CC2(C)CC2)=O)ncn2cc(Cl)ccc12 c1(C(N2CC(NC(c3cnc(CCCC)s3)=O)C(C)C2)=O)nccn2nccc12 C1(CCSC)NC(=O)CCN(CC2CC(F)(F)C2)C1=O c1(OC)ccc(F)c(C(N2CCCC(C(=O)Nc3ccnc(Br)c3)C2)=O)c1 C1(CN(C)C)CCCN1C(=O)CC1(O)CN(C(C2(Br)CC2(C)C)=O)C1 C1(CNC(C(CCC)OCC)=O)CN(C(=O)CCCC(F)F)CC12CC2 CCC(C(=O)N1CCOCC1CNC(c1c[nH]nc1C(C)(F)F)=O)C(C)C N1(C(c2cc(OC)no2)=O)CC(C(N2CCC3C(C(N)=O)C3C2)=O)C2(CC2)C1 c1(NCC(=O)NC)nccc(=NC(C)c2nc(O)n[nH]2)[nH]1 N1(C(C2CCC(C)O2)=O)CC2CCC(C1)N2C(c1cscc1C(F)(F)F)=O N1(C(c2c(Cl)cc(C)c(C)c2)=O)Cc2ccccc2CC1CNC(=O)CC(C)F Cc1c(O)ccc(C(=O)NCC2CCN(C(c3ccc(Cl)nc3)=O)C2)c1C C1(CNC(C(C(C)C)OC)=O)CC2CCC1N(C(=O)CN1CCCC1=O)C2 N1(C(C(C(C)C)NC(=O)Cn2ccnn2)=O)CCC(O)CC(C)(C)C1 CP(C)(=O)CC(=O)NCCC1CN(C(c2cc(O)n(CCBr)n2)=O)CCO1 N1(C(CNC(CCCCC)=O)=O)CCCCC(CNC(C2CCC2(C)C)=O)C1 C(CC(=O)NC1CC(=O)N(C2CC2)C1)(C(F)F)NC(C1(OC)CCC(C)C1)=O C1(C(CC)NC(=O)NCCCC(C)(C)OC(C)=O)CN(C)CCO1 C1(C(=O)NC2CCC(CCNC(C(CC)(F)F)=O)C2)CCc2nccn2CC1 Cc1cc(C(=O)N(C)CCOCCCN(C(=O)C(F)n2cccn2)C)ccn1 c1(C(N(C)CCNC(C2C=CCC2)=O)=O)ccc(NCCO)cc1 C1(NC(C2CC(CCC)C2)=O)CCC(NC(C2CC3C=CC2O3)=O)CC1 C1(NC(COCCN(C)C)=O)CS(=O)(=O)CC1NC(=O)C=CC1(C)CCOCC1 N1(C(CC2ON=C(C)C2)=O)CC(C)CC1C(=O)NC(c1cccnc1O)C CN1CCC(C(=O)NCCCn2cccn2)(NC(=O)C(F)=CC2CC2)C1 C#Cc1ccc(C(=O)NC2CC3CC2N(C(=O)C#CC2CC2)C3)cc1C C1(Cn2cc(C3C4CN(C(C5C(CC)CCO5)=O)CC43)nn2)CCCCC1(C)C N1(C(CC2(C)CN(C(=O)CNS(C)(=O)=O)C2)=O)CCC(C2OCCO2)CC1 C(=O)(CCC(=O)NCc1cc(C(=O)NCc2cnco2)n[nH]1)NCC c1(OCOC)cc(Br)ccc1CNCCCCCN N1(C(C(C=C)O)=O)CCCC2CN(C(c3[nH]nnc3COC)=O)CCC12 C1(NC(CN(CC)CC)=O)CC(OC)CN(C(C2CCC(=O)N2C)=O)C1 c1(NC(=O)N(CCCc2c(C)n[nH]c2)C2CC2)ccc(I)c(CC#N)c1 C1(C(=O)NCCCOCCO)CC1C1CCC1.C1C(=O)N1CC Cc1oc(C2CC2)nc1C(=O)NCCC1CCCCN1C(C1CCCC(O)C1)=O c1(CNC(CCNC(COC)=O)=O)cn(CC(=O)NCC2(n3ccnn3)CC2)nn1 c1(C(=O)NC2C(CNC(c3cn(C)nn3)=O)C2)ccnc(-n2cncn2)c1 C1(CNC2C(C(=O)NC(C#N)C(N)=O)CCC2)CCNC(=O)C1 c1(C(=O)OCC)nc(NC2CCN(C(=O)Cc3cnn(CC)c3)CC2)ncc1Cl N1(C(c2cc(OC)c(Cl)cc2)=O)CCC2C(CCN2Cc2ncc[nH]2)C1 C1(C(=O)NC2CN(C(c3c(OC)nn(C)c3)=O)CC2C)CCn2c(cnc2C)C1 CC1(C)Cc2cccc(C(=O)OCC(=O)NCC34CCCC(C)(C3)OC4)c2O1 N1(C(C=CC(CC)C)=O)CCC(C)(CC(N2CCC3CC23C)=O)C1 c1(C(N2CC(NC(c3c(C)ccs3)=O)C(C)C2)=O)cc(F)cc(C)c1N CCCCC(=O)C(=O)NCC(C)NC(=O)CCNC(=O)COC C1(NC(c2c(C)scn2)=O)CCCC(NC(=O)Cn2cc(Cl)cn2)C1 c1(CSCC(=O)NCC#CCNC(C2C(C)(C(=O)OCC)C2)=O)ccc(F)cc1 CC1CCN(C(C23CC(C)(CO2)C3)=O)CC1NC(c1cccc(=S)n1O)=O C1(CNC(=O)C=CCF)CC2COCC2N1C(=O)C(O)CC1CCCCC1 N1(C(C(C)OC)=O)CCN(C(=O)C(c2cc(Cl)ccc2Cl)(C)C)CC1C(F)F N(C1CN(C(=O)CCCC2CC2)Cc2ccccc21)C(CC1C(=O)NCCC1)=O c1(CC)cccnc1C(=O)NCCCC1CCCN1C(=O)CN1CCCC1=O Cc1cn2c(C(=O)NCC3(NC(C4CCC(=O)N4C)=O)CCCC3)c(C)nc2s1 CCS(=O)(=O)CC(=O)NCCCCCN(C(=O)C(C)(C)C1CCCO1)C c1(C(=O)NC2(C(N(OC)CCO)=O)CCSC2)cccc2cncn12 CC1=NOC2(C1)CN(N1CCC(N)(C(=O)N(C)C)C1)C2 c1(CNCC(C2CCCCC2)O)nccc(Br)c1Br CC1CN2CCN1C(C(=O)NCC1CCN(C(=O)CCCC(N)=O)C1)C2 N1CCC2(CCCC2Nc2ncc(C#N)cc2F)CC1.c1(C=O)coc(Br)n1 c1(C(=O)NC2CN(C(C3C(C(C)C)CCO3)=O)CC(C)C2)c(F)cc(F)cc1F C1(C(CC)C)CCN(C(c2nc(C)co2)C(=O)NCc2ccco2)CC1 C1(CNC(C(CCC)NC(C)=O)=O)(CO)CC12CCN(C(=O)C(C)N(C)C)CC2 C1(NC(c2cc(C)ncn2)=O)CC2CCC1(NC(=O)CC1(N(C)C)CCC1)C2 Cc1ccc(NC(c2cnn(C3CCC3)c2)=O)cc1.C1(=O)C(C)CC2CN1C2 N1(C(C2(c3cc(C)on3)CC2)=O)CCN(C(C2CC3CCCC3C2)=O)CC1CO CCCCCCC(F)C(=O)N1CC(N2CCN(C(=O)CC3CCCCO3)CC2)C1 C1(C(N(C)CC2CCC2)=O)CN(C(c2ccc(CO)cn2)=O)CCO1 O=C(N=c1ccn(C2CCSCC2)[nH]1)c1ccc(C2CCCCC2)c(Cl)c1 C1(NC(C(C)CC(F)F)=O)CN(C(=O)Cc2cc(Br)cs2)C2(CCC2)C1 Cc1cc(C)c(C(=O)NC2CC3CC(C2)N(C(=O)CN2CCC(C)C2)C3)c(N)c1 C#Cc1cc(F)c(C(N2CCC(NC(=O)C=CSC)C2C)=O)cc1F N1(C(CN(CC#C)C(c2ccn3ccccc23)=O)=O)CCC2CCC(C2)C1 CC(C)(C)CCC(F)C(=O)NC(Cc1ccoc1)C(N1Cc2c[nH]nc2C1)=O N1(C(C(Br)=C(C)C)=O)CC(CNC(c2cc3n(n2)CCO3)=O)CCC1C C1(C(=O)NCC#CCC)CCCCCCN1C(c1ncc2ccccn12)=O c1(C(C(=O)NC2CCCN(C(c3cnc(C)[nH]3)=O)C2)C(C)C)ccc(C#N)cc1 c1(C(C)C)nc(NCC2CCCS2)cc(N2CCC(c3cc[nH]n3)CC2)n1 N1(C(C(N2CC(C)OCC2)=O)=O)CCCC2CCC(C)CC12 c1(C(=O)NC2(CNC(Cc3cc(C)sc3)=O)CC2)cc2oc(Br)cc2[nH]1 c1(C(N(C)CC2CCN(C(c3cc(Cl)no3)=O)C2)=O)cc2ccc(F)cc2s1 c1(C(N2CC(F)CC(NC(CC(COC)(C)O)=O)C2)=O)ccc2c(c1)C(=O)OC2 C1(NC(C(CCOC)C)=O)CCN(C(c2cnc(-c3ccsc3)s2)=O)CC1(C)C Cc1ncncc1C(=O)NC1CC2(C1)CC2NC(c1n[nH]cc1F)=O N1(C(c2cncc(OC(C)C)c2)=O)CCCN(C(=O)C(C)CF)CC1C C1(CN2CCC(C(=O)NCCc3cn(C)nc3)C2)COC(C)(C)O1 c1(-n2cc(C(C)NC(c3ccc(C(=O)NC)nc3)=O)nn2)ccc(Cl)c(F)c1 CCC(C)(C)C(O)C(=O)N1CCC(C)C(NC(c2cc(C(C)C)oc2C)=O)C1C Cc1cn2cc(CC(=O)NCCC3CCCN3C(=O)CN3CCNC3=O)nc2s1 C(C(C)(C)C(=O)NC1CCC1NC(c1cc(I)on1)=O)OC c1(CC)ccc(S(=O)(=O)NC2CN(Cc3cccc(OC)c3)CC2(F)F)cc1 CC1CCCN(C(=O)C(=O)N(CCCCNC(C2CCCN2N=O)=O)C)C1 N1(C(c2[nH]cc(C)c2)=O)CCC(NC(c2ncccc2C(F)F)=O)C(CO)CC1 C1(CCNC(CCNS(CC)(=O)=O)=O)CCCN(C(c2[nH]c(C)nc2C)=O)CC1 C(=O)(CC(C)CC(C)C)N1CCC(NC(c2n(COC)ncc2)=O)C(CO)C1 C12(CNC(CC(C=C)C)=O)CCCC(CN1C(=O)COc1cccc(C)c1C)C2 c1(C(C)C)ccc(CC(=O)NCC2CN(C(=O)CCCC3CCC3)CC2O)cc1 C(=O)(C1Cc2ccc(F)cc21)NC(CC=C)CNC(c1ccc(C)nc1CC)=O c1(C(=O)NC(C(=O)NCc2cnc(C)[nH]2)C2CC2)ccc([N+](=O)[O-])o1 c1(C(N2C(C(C)NC(Cc3nnc(C)o3)=O)CCC2)=O)ncn2c1CCC2 Cc1ncc(Br)cc1NC(=O)C(O)C(F)F C(=O)(C(=O)N=S(C)(C)=O)NCC(CNC(C(c1cc(F)cc(F)c1)C)=O)CO CCCCC(C)C(=O)N1CCC(C(=O)NCc2nnc(C)s2)(CO)C1 C(=O)(C(C)(O)CCC)NC(CCC)C(=O)NC(c1ncc[nH]1)C Cc1c[nH]c(CC(N)=O)c1C(=O)NCC(C)NC(=O)C(C)Cc1ccc(F)cc1 c1(NC(C2CCCN2C(C2CC=CCC2)=O)=O)nc(NCC2CC2)c(Br)cc1Br C1(COC)CCCCN1C(=O)C(=O)NC1CCCNC1=O c1(NC(=O)NC(C#C)(C)C)ccc2c(c1)c(=O)c(Br)cn2C C1(NC(CN(C(=O)C=Cc2cscn2)CCC)=O)CCCC1(C)O c1(C(CC)NC(=O)CN(C(c2cnns2)=O)CC)nccn1C CCS(=O)CC(=O)NC1CN(C(c2c[nH]nc2I)=O)CC1C C(N=c1[nH]c(N2CCC(c3nncs3)C2)nc2c1SCC2)c1cccc(CC)n1 C(C(C)(C(C)C)NC(C1CCN(C(C)=O)C1)=O)NC(C(C)(C)OC)=O C(=O)(C(C)(C)c1cscn1)NCC(C)NC(c1cnc(CC(C)(C)C)s1)=O C1(NC(c2c(C#C)c[nH]n2)=O)CC1C1CCN(C(=O)CCOCCCOC)CC1 Cn1nc(C(=O)NC(Cc2cn[nH]c2)C(=O)NCCc2ncccc2F)cc1O N12CC3CCN(C3C1)C(=O)c1c[nH]c(c1)C2=O.c1(COC)c(C)cc(C)cc1C C1(c2nn[nH]n2)(OC(C)=O)CC1CSC.C12(CC1)C(=O)N2 c1(NC(=O)CC2CCCN2Cc2cnn(CCF)c2)ccc2c(n1)CCCC2 N1(C(CCCCOCC)=O)CCC(NC(=O)CCSCC(N)=O)C(F)C1 C1(NC(CSCCCC)=O)COCCN(C(=O)CCC2COC(C)(C)O2)C1 N12CCC(C(F)C1)C2.c1(NC(CSC(C)=O)=O)ccc(C)c(-c2ccccc2)c1 c1(NC2(C)CC(NC(=O)CCC3CC(F)(F)C3)C2)nc(C2CC2)nc2[nH]ccc12 C=CCC(CC)C(=O)NC(C1(O)CN(C(c2ccc(CCC(N)=O)cc2)=O)C1)C N1(C(C(CC)C)=O)CC(CNC(c2cn(CC3CCOCC3)nn2)=O)C(O)C1 C1(CNC(c2cc(C)ns2)=O)CC(C)(C)CN1C(c1nn(C)c(Cl)c1Cl)=O C1(NC(c2c(CC)cccc2)=O)CCC(C)(NC(=O)CCN2CCOC2=O)CC1 CC1CN(C(=O)CC(c2ccc(F)cc2)C)CC1CCNC(=O)C(C)(C)CF Cn1cc(Br)c(CS(N2CC(C(=O)O)C(C(F)(F)F)C2)(=O)=O)n1 CC1CCCC(C(N2CCCC2C(=O)NCCC(=O)Nc2nccs2)=O)C1 CN1CCn2cc(C(N3CCOC(CNC(=O)CCP(C)(C)=O)C3)=O)nc2C1=O N1(CC)C(=O)CCC1CC(=O)NCC(CO)NC(c1n[nH]cc1OC)=O c1(C(N(C(c2cnn(C)c2)C(=O)O)C)=O)cc2ccccc2n1CC#N c1(N2CCC(CC)(CO)C2)nc(NCC(C2CC2)OC)c2ccsc2n1 N1(C(c2c(CC)n[nH]c2)=O)CCOC(C(=O)Nc2cnsc2)CC1 Cn1cc(C(=O)NCC(CNC(=O)CC2(n3ccnc3)CC2)S(C)(=O)=O)n(C)c1=O C1(COC)(CNC(=O)Cc2c(C)noc2C)CCCN1C(C1CC1(C)C(C)C)=O C1(NC(C(C2CCN(C(c3c(OC)n[nH]c3)=O)C2)C)=O)CCc2ncnn2C1 n1(CC(=O)NCC2C3CN(C(C(CC)(C)O)=O)CC32)c(NC)nc2ccccc12 CCCS(=O)(=O)C(C)C(=O)NCC(C)(CC)NC(=O)C1=C(C#N)CCC1 c1(C(N2CCCC(C)(C(=O)NCCNC(C)=O)C2)=O)cn2c(Cl)cccc2n1 N1(C(c2c(C(C)C)ocn2)=O)C(C)CN(C(=O)C(C)N2CCC2)CC1C C1(CNC(CC2(C)CC2(F)F)=O)CC(O)CN1C(=O)CSc1ccc(O)cc1 Cc1cc(C(=O)NCC2(F)CCN(C(C3CCCCCCC3)=O)CC2)nc(C)n1 c1(C(=O)NCC(Cn2cc(C(CC)O)nn2)(C)C)cc2c(C)n[nH]c2cn1 C12(CNC(Cc3cc(C)no3)=O)CN(C(C3CCCCS3)=O)CC1CCO2 N1(C(Cc2ccc(OCCC)cc2)=O)CC2(CCCCN2C(=O)C(C)CF)C1 N1(C(C(C)(C)F)=O)CC(CC(=O)NC2C(O)CC2O)C2(CC2)C1 Cc1cccc(SCC(=O)NCC2CCN(C(C3CCCCS3)=O)C2)c1 C(C(CC(C)C)C(=O)NC1CC(=O)NC1=O)NC(c1cncc(C)n1)=O C1(CNC(C=COCC)=O)CCC2(CCC2)C1NC(c1cccc(O)c1C)=O CCCC(O)C(=O)NCCC(C(C)C)NC(=O)C(F)=C(C)C1CC1 C=CCC(C)(CC)C(=O)NCC(CO)NC(=O)CSC C1(C(=O)NCC(COC)C)CCN(C(C2(SC)CC(=O)C2)=O)CCO1 C(N=c1ccnc[nH]1)C1NC(=O)N(CCc2ccc(Cl)cc2)C1=O C1(CNC(N2CCC(C3CCCCO3)CC2)=O)CC2CCC2C1 Cc1c(C(N2CCN(C(=O)CCCCCF)CC2C)=O)cccc1Cl c1(C(N2CCCC(CC(=O)Nc3cn(CC)nc3C)C2)=O)ncc2[nH]ncc2n1 C(C(C)(O)CC(=O)N1CCC(CNC(=O)C(C)(C)c2ccccn2)C1(C)C)OC N1(C(c2c(C)cno2)=O)CCCC12CCN(C(c1ccnc3[nH]c(O)nc13)=O)C2 C1(C(=O)NCC2CN(CC)C(=O)O2)CC2CCC(C1)N2C(=O)CCC1CC1 CC(CC(=O)N(C)CCN(C)Cc1nncn1C1CC1)N1CCOC1=O NC(=O)CC(N=c1ccnc(NC2CC3CCCC3C2)[nH]1)c1ccccc1 CC1C(NC(=O)C=Cc2ccc(Cl)nc2)C(C)CCN1C(C1(C(N)=O)CC1)=O CC(C)CC(CC(C)C)(c1nnnn1C1CCOCC1)NCc1cccc(Cl)c1 c1(C(=O)NCCCCNC(CC2N(C)C(=O)CC2)=O)cc(F)cc(Br)c1F Cc1ccc2c(=NC(C)c3ccc(Br)cn3)[nH]c(=NCC(C)CO)[nH]c2c1 CC1CN(C)C(=O)CN1C(=O)CCC(C)NC(c1cncc(F)c1)=O N1(C(CCN(C(C2CC(C)(O)C2)=O)CC2CC2)=O)CC2(COC(=O)C2)C1 C=CC(C)CC(=O)NC1CCC(N2CCN(C(=O)C=Cc3nc[nH]n3)CC2)CC1 c1(SC)nc(=NCC2CCCN2C(c2cccc(C(N)=O)n2)=O)s[nH]1 C1(C(N(C(C)C)CC)=O)CC(NC(=O)C(C)NC(C2CCC2)=O)C1 c1(OC)cccc(CN2CCCC(C(=O)NCCC3CCCCO3)C2)c1C C1(COC)(NC(=O)CC(F)(F)F)CCCN(C(c2ccccc2C(C)(C)C)=O)C1 C(CC)(CCC(=O)N(CC(O)CF)C)NC(c1[nH]cc(C(C)=O)c1)=O C1(C2CCN(C(C3COC(=O)N3C)=O)C2)(NC(CN(C(C)C)C)=O)CC1 N1(C(C2(C)CCNC2=O)=O)CC2(C1)CN(C(=O)C=Cc1cn[nH]c1)CCO2 c1(C(N2CCN(C(C3CCCCC3)=O)C3CC23)=O)ccc2c(O)nnc(O)c2c1 c1(NC(=O)NCCCN2C(=O)CCC2=O)cc([N+](=O)[O-])n[nH]1 CC(C)CC(O)CC(=O)NC1C2CCC(=O)C12.c12ccc(cc1F)CNC2=O C1(C(N2C(CC(=O)N(CCn3c(C)ncc3)C)CCC2)=O)CC2C=CC1C2 C1(NC(c2cc(SCC)ncc2)=O)CC2(CCCN(C(c3occc3Br)=O)C2)C1 Cc1cc(C(=O)NC(CNC(C2CCCC2O)=O)C(C)(C)C)nn1CCO CC1CCN(C(c2nccn2C)=O)CC1NC(C1(C(F)(F)F)CC1)=O n1(CCC(=O)N(C2CN(C(C3C(=C)C3)=O)CC2(C)C)C)c(C)nc2ccccc12 c1(C(C)C)ccc(C(=O)N(c2ccccc2)CC2CC(=O)N(C3CNC3)C2)nc1 CC(C)(Cc1ccc(Br)cc1)C(=O)NC1CC1NC(C1CC(C)(C)CO1)=O C1(C2CN(C(=O)CCCC3CCCO3)C2)(NC(Cc2c(C)cc(C)s2)=O)CC1 N1(C(CN(c2ccccc2)C)=O)CC(NC(=O)C(CC(N)=O)N(C)C)C(C)(C)C1 c1(C(=O)NC(CNC(Cc2scc(C)c2)=O)C(C)(C)C)cnc2ncnn2c1C C12(NC(CCNC(C)=O)=O)CC(C1)N(C(c1ccco1)=O)C2.c12sncc1C(=O)N2 c1(C(N2C3CN(C(c4c(OC)nsc4)=O)CC2C3)=O)ccc2cncn2c1 C1(C(=O)NCCCC(C)NC(=O)CO)CC2(CCC2)C1 C(=O)(CC(C)C(=O)NCC(C)(F)CNC(C1CN(C)CCO1)=O)OC C1(COC(CCNC(=O)NC(C2CC(C(=O)OC)C2)=O)=O)CCCOC1 N1(C(C2CN(C(C)=O)C2)=O)C2CCC1C(C(=O)Nc1cccc(Cl)c1C)C2 C1(OC)CN2CCCC2(C(=O)NCC(C(C)C)N2CCOCC2)C1 C(c1ccc(Cl)cc1)=CC(=O)NC1CCC(NC(CC2C(C)(C)CCO2)=O)CC1 c1(OCC)n[nH]cc1C(=O)NCCCCCNC(=O)C(C)OCC1CC1 C#Cc1ccc(C(=O)NC(CNC(=O)C(C(C)C)N(C)C)C2CCC2)c(C)c1 O=C(CC1CN(C(C2CN(C3COC3)C2)=O)CCO1)N=c1cc[nH]c(CCO)c1 C1(C(C)NC(c2ccn(C(F)F)n2)=O)CCCCN1C(=O)CC1CS(=O)(=O)C1 C(CCCCC(=O)N1C2CCC(C2)C1CC(N1CCC(n2ccnc2)C1)=O)OC C(CNC(C1(C)C=CCC1)=O)(CC(=O)N1CCC(F)C1)OC c1(C(=O)NC(CC)CNC(=O)CC2(O)CCC2)cc2cc(OC)ccc2nc1C c1(C(=O)NC(CNC(C2(COC)CC2)=O)(C)CC)ccc(F)cc1[N+](=O)[O-] C1(NC(c2ccco2)=O)C=CCN(C(=O)C=Cc2ncc[nH]2)C1 c1(CONC(C(C)(O)c2n(C)ccn2)=O)ccc2ccccc2c1 c1(C(=O)NCCN(CCC)C(C2(F)CCOC2C)=O)cc(C)nn1C(C)(C)C c1(CCNC(C2(C)CSC2)=O)ccc(CNC(=O)CC2CCC(=O)N2)cc1 C1(C(=O)NC2CC(OCC)C2OC)CCc2nncn2CC1 c1(C(N2CC(C)N(C(=O)Cn3ncnn3)CCC2)=O)cnc2sccn2c1=O CC(C)=C=CC(=O)NCC1CCC(C(=O)NCCSC(C)C)CC1 C(=O)(CCN=c1cc(C)[nH]c(=NCC2CC3CCCCC3O2)[nH]1)NC(CC)C C1(C(=O)NC(CC#C)C(=O)NCC2CC3(CCC3)CO2)CC(C)(C)CCO1 C1(C(=O)NCCCCN(C(=O)CSc2ccncc2)C)CC2(CCC2)CO1 C=CCC(C(=O)N1CCC(CC)C1C(N1CCC1CC1CC1)=O)NC(C)=O C(=O)(CC(O)CC1CC1)N1CCC(OCC)C1 N1(C(COCCOC)=O)CCC(NC(c2c(SC)cccc2F)=O)C1(C)C c1(C(N(CC(CNC(CC(C)(C)OC)=O)O)C)=O)cnc2cc(Br)ccn12 C(C(C)(C)CCNC(=O)C=C(C)C1CC1)NC(CCN(C(CCC)C)C)=O c1(-c2cn(CCN(C(C34COCC3C4(F)F)=O)CC)nn2)ccccc1[N+](=O)[O-] CC1(C)CCCC(C(N2CC3CC2C3C(=O)NC2CC3CCC(C2)S3)=O)C1 c1(C(N(C(CNC(C(C=C)(C)CC)=O)C)C)=O)c[nH]c2c(Br)cccc12 c1(OC)c(Br)cc(C(N2CCC(F)(c3ccccc3)C2)=O)cc1Br C1(C(=O)NCCCCCO)CC12CN(C(C1CC(O)CN1)=O)C2 CC1C(C)N2CCN1C(=O)C1CC(C1)C2=O.c1(CCN(C)C)ccc(O)c(F)c1 C1(C)(CNC(CCOC)=O)CCN(C(=O)C(C)Cc2ccc(N)cc2)C1 c1(CNC(=O)Nc2c(C(C)(C)C)con2)cccc(N2CCOC2=O)c1 C1(CCOC)(NC(C2CCC3(CC3)C2)=O)CCN(C(=O)CCOCC2CC2)C1 C1(OC)CC(NC(c2cscn2)=O)CN(C(=O)C(C)(O)c2ccccc2)C1 c1(OC)cccc(-n2cc(CC3CCCN3CC3CC(F)(F)C3)nn2)n1 C1(CC)CC(C(=O)NCC2C=CCN2C(=O)CCc2csc(C)n2)CC(=O)N1 C1(NC(C(C)CN2CCCCC2)=O)CCN(c2nnc(C(F)F)s2)C12CCC2 Cc1ncc(C(=O)NC(C2CCCN(C(C3(S(C)(=O)=O)CC3)=O)C2)C)cc1N CC1(C)CCC=C(C(=O)NCC2CC(F)(F)CN2C(=O)CCc2nc[nH]n2)C1 C12(NC(COCCCC)=O)CCCC(CN(C(=O)CCCCN(C)C)C1)C2 C1(C2C(C)(C)CN2)CCN(C(=O)C(=O)NCC2CC2c2ccccc2F)CC1 C1(C(=O)NCC(C2CCN(C(CC3(C=C)CC3)=O)CC2)C)CN2CCC1CC2 C(CC(C(=O)NCc1ccco1)NC(c1cc(Br)cs1)=O)SC N1(C(CCC#CC)=O)CC2(CC(CNC(c3ccc(OC(C)CC)cc3)=O)C2)C1 C1(c2n(CCCOC)nnn2)(NCc2cccc(F)c2)CCC2C3C=CC(C3)C12 C1(C(=O)NCc2c(C(=O)NC(C)C(=O)NC3CC3)[nH]cc2)CC2(CCO1)CC2 C(CC1=CCOCC1)NC(C(CCC)NC(=O)CCOC(C)C)=O C(CC(C)(C)NC(c1cc(-c2ccc(C)o2)on1)=O)NC(C1CC(SC)C1)=O C(CCCCCNC(C1C2CCCC12)=O)N(C)C(C1CC(=O)N(C)C1)=O c1(CNCC2CCN(C(=O)Cc3ccccc3)C2)cc2ccccc2cc1O C1(CCC(=O)NC(c2cccs2)C)CCCCN(C(=O)CCCF)C1 C12(C(=O)NC3(CNC(C4CSC4)=O)CCCCC3)CCCC1CC(F)(F)CC2 C#Cc1cc(C(N2CCC(NC(=O)C(C)NC(C)(C)C)C2)=O)cc(Br)c1 Cc1cc2c(cc1NC(c1ccc(Cl)c(O)c1)=O)C(=O)NC2=O c1(C(N)=O)cc(C(N2CCC(O)(CNC(=O)C(O)CF)C2)=O)ccn1 c1(C(=O)NC(CNC(CCC)=O)C2CCC2)ccn2ccnc2c1 CC1CC2(CC(C(=O)NCCCCC(=O)N3CCOCC3C3(C)CC3)C2)C1 C(C)(C)(C(C)CC(=O)NCc1cn(C)nc1C(C)C)NC(CCC(C)=O)=O CC(C)CCC(O)C(=O)N1CCCC(CC(=O)NC2C(O)CC2O)C1 c1(N2CCC(SC)C2)ncc(-c2cn(-c3cncc(F)c3C)nn2)cc1Cl N1(C(CC)=O)CCC(CNC(=O)CCNC(c2ccccc2OC)=O)(OC)C1 N1(C(CCCNC(=O)OC)=O)CCCN(C(=O)CN2CCC(C)CC2)CC1CO N1(C(C2C(C)(C)CC2)=O)CCn2c(CNC(C3(C)C=CCCC3)=O)nnc2C1 c1(OC)ccc(CN2CCC(C(=O)Nc3c[nH]nc3Br)C(O)C2)c2ccccc12 c1(C(=O)NCC(CNC(C(C)OCC(F)(F)F)=O)CO)cnc2ncccn12 C1(CNC(c2ccc(C)n2C)=O)CN2CCCCC2CN1C(=O)COCC(C)C N1(C(c2nn(CC)c(C)c2)=O)CCC12CN(C(c1cc(C(F)(F)F)n[nH]1)=O)C2 C1(CC(=O)NC)CN(C(=O)CN(c2ccccc2)C)CCN1C(=O)CP(C)(C)=O c1(OCC)oc(C)nc1C(N1CC(CNC(=O)C=CC2(C)COC2)C(O)C1)=O C1(OC)CCN(C(=O)C=CCC(C)(C)NC(=O)CCCn2cncn2)CC1 c1(CC(CNC(=O)NCCC2CC3C=CC2C3)CO)ccccc1F c1(C(C(=O)O)NCc2ccn(C)c2)cc(F)c(Br)c(F)c1 C#CCCC(C(=O)NC12CCCN(CC1)C2)NC(=O)C=C(CCC)CCC c1(C(=O)OC)ccc(Cl)c(Cl)c1NC(=O)CCc1ccncc1Br c1(OC)cccc(N(C(=O)CNC(=O)CNC(c2cc(C)sc2N)=O)C)c1 c1(CC)cscc1C(=O)NC1(CNC(c2cnsc2C)=O)CCOC1 CC(C)CCC(F)C(=O)N1CC(NC(C2CCC(CO)CC2)=O)CC(F)C1 C(C)(CNC(=O)CSc1nncn1C(C)(C)C)(C(C)C)NC(C(CC)F)=O C(CC(=O)NCCC(C(C)C)NC(C1CCC1)=O)(C(N)=O)NC(C)=O c1(C(=O)NCCN(C(CCCc2ccc(C)s2)=O)C)cccc(CO)c1C O=C1CC(C(=O)NC2CCC(CO)C2)CN1CC(F)(F)F O=C(NOC1CCCCC1)C1=CCN(C(c2cn(C3CC3)nn2)=O)CC1 C=CC1(CC(=O)NC2CC(NC(=O)C(C)c3cccs3)C2)CCOCC1 Cc1ccccc1C(=O)NC1CCC(CC(=O)NOCCOCCF)C1 Cc1ccc(C(N2CC(C(C)NC(C3C=CC=CC=C3)=O)C2)=O)cn1 C1(C(N(C2CCN(S(C)(=O)=O)C2)C)=O)CC2CC1CO2.c12csc(n1)NC(=O)C2 C(CCC(=O)N1CCC(C(C)NC(c2cc(C(=O)OC)on2)=O)C1)=CCC=C Cc1c(O)c(=O)ccn1CC(=O)N(C)CCN(C(=O)C(C)N1CCC1)C C1(NC(C2(CCOC)CCN(C(=O)C(C)CC(N)=O)C2)=O)CC2C(C1)C2(F)F c1(C(N2C3CN(C(Cn4c(C)csc4=O)=O)C(C3)C2)=O)ccn2c1CSCC2 c1(NC2CCN(C(Cn3ccc(C)n3)=O)C(C)C2)ncnc2c1nnn2C(C)C c1(C(=O)NCCCCNC(c2ccn(C3CC3(F)F)n2)=O)cscc1F CCCCCC(C)(C)C(=O)N(CC(C)NC(c1ccc(F)nc1F)=O)C Cc1ccnc(Cl)c1CN1CC(C)(C(=O)NC2CC2c2ccc(Br)cc2)C1 C1(N(C(=O)COC(C)=O)C)CCN(C(=O)CC2CCC2C)CC1 c1(C(N(C)CC2CCCN2C(=O)CCF)=O)cc2cccc(Br)c2[nH]1 CCC(CC(=O)N1CC(NC(c2nnsc2C(F)F)=O)C(C)C1)c1ccccc1 N1(C(C2C(C)=C2)=O)CCN(C(C2CC3(C2)CC3(F)F)=O)C2(CCC2)C1 Cc1ccc(NCC(N2CC(CNC(c3c[nH]cc3C3CC3)=O)C(C)C2)=O)cc1 c1(N2CCC(NC(C(CCC)N(C)C)=O)C(F)C2)ncc([N+](=O)[O-])cc1C N1(C(c2cc(CNC(C=CCCC)=O)sn2)=O)CC(C2CC2)C1C1CC1 C(C(N)=O)(C(F)(F)F)NC(c1cc(-c2nc(C)sc2)oc1)=O c1(OCC(=O)NCC(CC)N(C(=O)CC2CC(OCC)C2)C)cccc(C)c1 C1(NC(C23C(C(=O)OC)C(CC2)C3)=O)CCCCN(C(C2COCCO2)=O)C1 C1(NC(CC23CC(C)(OC2)C3)=O)CCC2CCN(C(C3(C)CCCO3)=O)C1C2 S(=O)(=O)(c1ccc(C)cc1C)N1CC(NC(c2cncc(C)c2)=O)CC(F)(F)C1 c1(CCC(=O)NCC2C3CC2N(C(=O)C=Cc2ccoc2)C3)ccc(F)cc1F N1(C(c2cnc(C(C)C)nc2)C(=O)NCC=C)CC(C(F)F)CC1(C)C c1(C(=O)NC2CN(C(C3CCS3(=O)=O)=O)CC2O)cc(Br)c2nccn2c1 c1(N(C(C)=O)C)ccccc1C(N1CCC(CNC(=O)Cc2ccsc2C)C1)=O C(=O)(C1=Cc2ccccc2C1O)N1CCC(NC(CCC(=C)Cl)=O)(CC)CC1 c1(C(=O)NC2CC(C)(NC(CC3C(C)CCO3)=O)C2)ccccc1O N1(C(C(C)O)=O)CCC(NC(=O)Cc2ccc(-c3ccccc3)cc2)C(F)C1 C1(C(N)=O)CC(CC(=O)NC(C2CCCC2)CNC(C2(Br)CC2)=O)C1 c1(N2CCCC(CCC)CC2)nc2c(c(=NC(C)C3CC3)[nH]1)SCC2 C1(CNC(C(C(C)C)N(C)C)=O)CC2CN(C(c3cc(O)cc(Cl)c3)=O)CC12 c1(C(=O)NCC(C)NC(c2c(C)nc(COC)s2)=O)ccc(C(F)(F)F)cc1N c1(CC(N2C(CNC(C3C(C=C)OCC3)=O)CCCC2)=O)ccc2c(c1)CCOC2 c1(C(N2C(CNC(C(C)C3(O)CCC3)=O)CCC2)=O)coc2c1CS(=O)(=O)C2 n1(CC(=O)NC2(C)C(C)CCC2)cc(Br)c([N+](=O)[O-])n1 N1(C(=O)NC(C)COc2ccccc2Br)CCCC(C(C)N)C1 C1(NC(C2(COCC)CC2)=O)CC2CCC1N2C(C1CCCC1CC)=O N1(C(C=CSC)=O)CC2(CCC(CNC(=O)CNC(=O)Nc3ccccc3)O2)C1 C(C)(CCCCCO)NC(C1(C2N(C(c3nc(C)oc3C)=O)CCC2)CC1)=O C(CN=c1[nH]c(=N)[nH]c(=NCCCC2(C)N=N2)[nH]1)c1nc(C)nc(O)c1 C1(NC(c2cc(C(C)=O)sc2)=O)CC(NC(=O)C=C2CCOCC2)C12CCC2 c1(C(=O)NC2CN(C(C3(SCC)CC3)=O)C2)cccc(CC)c1F c1(C(=O)NC2C(CNC(CC=C)=O)C2)nn(C(C)C)nc1Br CCC(C#N)(CC)C(=O)N1CCCCC(CNC(=O)Cn2nc(C)n(C)c2=O)C1 c12cccc(Cl)c1NC(=O)COC2=O.n1(CC(=O)NC(C)(C)C)ncccc1=O N1(C(c2cc(C)cc(OC)c2O)=O)C2CCCC1CN(C(=O)CN=S(C)(C)=O)C2 Clc1ncccc1-n1cc(CNCC(c2ccccc2)N2CCOCC2)nn1 N1(CC(CNC)O)CCN(C)CC1.c1(OC)ccc(C(C)(C)N)cc1 c1(OC)cc(-c2nc(C)nn2C2CCC2)cc(Cl)n1 C1(NC(C2(C)CC=CC2)=O)CCCCN(C(=O)CCN2CCCC2=O)CC1 C(=O)(CCC(=O)NC1CCCN(C(=O)C(C2CC(F)(F)C2)O)C1)N(C(C)C)C CCC(CNC(C1CCN(C)C1)=O)(CC)NC(c1ccc(C(N)=O)nc1)=O N1(C(CSC)=O)CCC(C2CC2)(CNC(=O)C(C2CCOCC2)F)C1 c1(C(=O)NC(C)CN(C(=O)Cc2nc(C(C)C)n[nH]2)C)cnn(C)c1N CCC(CC)C(=O)N1CC(NC(c2ccc(Oc3ccccc3)o2)=O)CC1C C=CC1CCCC(NC(=O)C(C)(CNC(c2cc(OC)no2)=O)CC)C1 C1(CNC(CCc2cc(C)[nH]n2)=O)(NC(=O)CC(O)CN(C)C)CC(F)(F)C1 c1(C(CF)NC(=O)Nc2ncc(-c3ccccc3F)s2)ccccc1Br CCS(=O)(=O)CCn1cc(NC(N2CCC2C2CCCCC2)=O)cn1 C(CCC(=O)NC1CCC(CNC(=O)OC(C)(C)C)C1)=CC(C)C Cc1cc(C(=O)NCC2N(C(=O)CS(N)(=O)=O)CCCC2(C)C)c(N)c(Cl)n1 c1(OC)cc(C(=O)NC2CC(C)N(C(C3CCC(C)CC3)=O)C2)cc(N)c1N C1(NC(C2CC(OC)C2)=O)CCN(C(=O)CCSC2CCCC2)C(C)C1 C#Cc1ccc(C(N2CC(CNC(=O)C(F)(F)C(F)(F)F)OC(C)C2)=O)cc1C C12(NC(C3CC(C)OCC3)=O)CC(C)(C1)OC21CN(C(c2ccc(O)nn2)=O)C1 n1(CC(=O)NC2C(C)(C)CN(C(=O)C(O)C(F)(F)F)C2)ncn2cccc2c1=O O=C1CCc2cccc(C(=O)NC34CC(C3)N(C(=O)CN3CCSCC3)C4)c2N1 C1(N(C(CC(=C)C)=O)CC)CCCN(C(c2ncoc2-c2ccccc2C)=O)C1 CN1CCN(C(c2cncc(C#N)c2)=O)CC1C(N1CCC(C)(C)C1CO)=O c1(C(=O)NC2(CCCNC(C(C)O)=O)CC2)sc(C(C)(C)C)nc1C(F)F N1(C(CCc2cc(C)[nH]n2)=O)CCCC(NC(c2csc(Cl)c2Cl)=O)CC1 C1(c2ccc(C(c3ccccc3)=O)c(F)c2)CN(N2CC3CCCCCC3C2)C1 CC(C)C(O)C(=O)N(C(=O)OCC1CCCCN1S(C)(=O)=O)C1CC1 c1(C(N(C(CN(C(c2c(CC)nco2)=O)C)C)C)=O)cc2nc(C)[nH]c2cc1F N1(C(C(=O)N(CCCC2CCCNC2)C)=O)CCC(C(C)(C)C#N)CC1 c1(CN(c2ccc(OC)c(C)c2)C)cc(Br)cc(C)c1F C1(COC)CCN(C(=NCCc2ccc(F)cc2)NCCc2nc(C)cs2)C1 C(=O)(C(CN=[N+]=[N-])NC(c1cnsc1)=O)N1CCN(CCC#C)CC1 c1(CNC(C(=O)NCCC(C)OCC)=O)cnc(OC(C)C)cn1 c1(OC)ccc(C(C)C(=O)NC(C)CCNN2CCCCC2=O)cc1F N1(C(c2cc(C)[nH]c2C)=O)CC2CC(NC(C3Cc4cccnc4C3)=O)CC1C2 C1(Cn2cc(CCNC(=O)OC(C)(C)C)nn2)CC2CN(OC)CC12.C1CNC1=O C(CCC(=O)O)(C(N)=O)OC(=O)NC1CCN(C(=O)OC(C)C)CC1 n1(CC=C)cc2ccc(NC(=O)NC3(C4CCC4)CC3(F)F)cc2n1 N1(C(C2(NC(C)=O)CC2)=O)CC(O)(c2cn(Cc3ncoc3C3CC3)nn2)C1 O=S(=O)(c1ccc(Br)s1)N1CCCC(Nc2ccccc2OC(F)(F)F)C1 c1(C(=O)NC(CC)CNC(c2cnccn2)=O)ccc2c(C)cc(Cl)nc2c1 C1(CN(C)C)CN(C(C2OCCC2CNC(c2nocc2Cl)=O)=O)CCO1 c1(CC(=O)NCC(CN(C)C(C2CC2c2ccco2)=O)O)nc2c([nH]1)CCCC2 C1(C(N2CC(O)(CC=C)C2)=O)CNC(=O)CN1C(=O)CSCC(N)=O C1(C(N2CC(C=C)C(NC(c3cncc(OC)n3)=O)C2)=O)CCCCC(C)(C)C1 n1(CC)ncc(C(N2CCC(C)(CNC(C3(F)CCOC3)=O)C2)=O)c1Cl c1(C(=O)OCC)cnc(C(=O)NCC2C(C(C)NC)C2)o1 c1(-n2c(CNC(c3n(CC=C)nnn3)C3CCSC3)ncc2)ccc(F)cc1 Cc1ccc(Cl)c(C(N2CCCC(NC(c3csc(-c4nc[nH]n4)n3)=O)C2)=O)c1 CCC(F)(F)C(C)(C)C(=O)NC1CCCC(NC(=O)CCn2cncn2)CC1 C(=O)(NNC(=O)C(C)(C)CCCCNC(c1cnc(Cl)s1)=O)C1(CC=C)COC1 Cc1ncnc(C(N2CCN(C(c3cc(C4CC4)[nH]n3)=O)C(C(F)F)C2)=O)c1C c1(NC(C2CN(Cc3cccs3)CCO2)=O)ccc(I)c(Br)c1 C(=O)(C1Cc2ccccc21)NCCCCCNC(C(CNC(C)=O)(C)C)=O C(C1=CCN(C(c2ccc(C(C)C)o2)=O)CC1)NC(C(C)SC)=O Cc1ccc(F)c2oc(C(=O)NCC3(NC(c4ccnc(S)c4)=O)CCC3)cc12 c1(C(=O)NCCn2cc(C(N3CC=CC3)=O)nn2)ccc(O)cc1 C=CC(C)C(C)C(=O)NCC(c1ccc(F)cc1)NC(=O)C1=CC(C)(C)C1 c1(C(=O)OC)cc(C)cnc1C(=O)OC.C12(CCCCC1)CCC(=O)N2 C12(NC(C3CC(N(C)C)C3)=O)CCCC1CN(C(=O)CC1CCCCC(=O)N1)C2 c1(NC2CN(C)C2)[nH]c(=NCc2c(Br)cccc2Br)nc2scnc12 C#CCCN=C(NCC1(CC2CCC2)CC1)N1CC(C)CC(C)C1 N1(C(C2(NC(=O)CC(=O)N(C)C)C(C)CCC2)=O)CC2CCC(C1)C(=O)O2 c1(CC)cccc(C(=O)NC(C2CCN(C(c3[nH]ccc3C)=O)C2)C)c1 C1(C(N2CC(OCC(=O)NCc3n(CCC)ccn3)C2)=O)CC2(CC(=O)C2)C1 c1(CC(=O)NCC(C)NC(c2cc3ccncc3[nH]2)=O)ccc2c(c1)CCOC2 N(C)(C(=NCc1cc(Cl)cs1)NCC(F)F)CC1CCN(C(C)=O)C1 c1(C(=O)OCC)cnccc1NC(C1(C)CCCN1C(=O)C(C)N=[N+]=[N-])=O Cc1cc(=N)[nH]cc1C(=O)NCC(C)(C1CC1)NC(c1cccs1)=O c1(C(=O)NC2(CCNC(C(CC(C)(C)C)O)=O)CC2)cc2ccoc2cc1F N1(CC2CCC(=O)N2Cc2ccccc2)CC(=O)NC2(CC2)C1 CCC(CO)CCNCc1cc(CC(C)C)ncn1 C1(C(N2OCC(=C)C2)=O)C(C2CC2)CCN1C(c1cc(C2CC2)[nH]n1)=O Cc1cc(S(N)(=O)=O)ccc1CNC(=O)C(=O)N(CC(c1ccnn1C)O)C c1(C(=O)NCC2C(NC(c3nnn(CC)c3C)=O)C2)cncc2ccc(F)cc12 Cc1cc(Br)cc(C(=O)NC(C)(C)CN(C)C(C2CCC(F)C2)=O)c1F C1(C(=O)NCCC#CCC)C(CC)CCN1C(=O)Cc1ccoc1 C1(C(=O)NC(CNC(c2c(C)cc(C)[nH]2)=O)C)CCC(F)(F)CC1 c1(C(N2CC(CC(C(=O)N(C3CC(=C)C3)C)F)C2)=O)ccc(C)nc1C C(CN=C(NCCC1CC1)NCC1(F)CCCCC1)=CC N1(C(CC(CN(C)C)O)=O)CCc2[nH]nc(CNC(C3(C)CC=CCC3)=O)c2C1 CC(C)CCCCC(=O)N1CCCC(CNC(=O)C(C)CCn2cccn2)CC1 CCC(O)C(C)C(=O)NCC1C2CC1N(C(c1cc(F)ccc1C(F)(F)F)=O)C2 C1(N=[N+]=[N-])(C(=O)NCc2c(C)cc(C)s2)CCN(C(C2CN3CCC2CC3)=O)C1 C12(NC(C3CC4(C3)CC(F)C4)=O)CCCC1N(C(c1ccc(O)cc1)=O)CC2 c1(C(C(N2CC(CCCC(=O)OC)C2)=O)NC2(F)CC2C)ccc(Br)cc1 Cc1cncc(CC(=O)NC(C)(CNC(C2CC2(F)F)=O)CO)c1 N1(C(CC(C(C(C)C)C)C)=O)CCC(O)(C2CCC2)CC1 C1(C2CC2)(NC(Cc2n(C)ccn2)=O)CCN(C(=O)COc2cccnc2)C1 N1(C(C(COC)O)=O)CC2CC(NC(c3occ4c3CCC4)=O)C(C2)C1 C12(NC(=O)CCn3cnccc3=O)CCCC1N(C(C1CSC1)=O)CC2 c1(C(=O)NCCC(C)NC(c2ccc(CC(C)C)s2)=O)ccc(F)c(CO)c1 CC(C)C(O)CC(=O)NC1CN(C(=O)C(O)C(C)C)CC1O N1(C(CCC=CCC=C)=O)CCCCC2(C1)CN(C(c1cnccn1)=O)C2 c1(C(=O)NC(CC(C)C)CNC(c2nccn2C)=O)ccnc2cc[nH]c12 C=C(C)CC(C)C(=O)NCC(C)(CO)NC(=O)CC1(O)CCOCC1 c1(C(=O)NCCCN(CCO)C(C2C3CCCOC23)=O)cn2ccnc2cn1 C1(CN(C(=O)C(C2CC=CCC2)NC(=O)CSCC(F)F)C)CCCC1O c1(CN2C(CC(C)C)C=CC2)cc(C(C)(C)C)cc2c1CCC2(C)C N=c1cc(C(N2CCC(NC(=O)C(Cl)=CCl)C23CC3)=O)c(Br)c[nH]1 C(=O)(C(C)(C)CC(F)F)N(CCCCN(C(C1CCC(C)C1)=O)C)C CC1CC(N=c2ccc3c([nH]2)CCCC3=O)CCN1C(=O)CSCc1cccs1 C1(C(N)=O)CCC(NC(C2CCCCC2c2ccccc2)=O)CC1 Cc1[nH]nc2ncc(-c3nn[nH]n3)cc12.N12CC(CS1(=O)=O)C2=O C1(C(=O)NCC(C)NC(=O)C(c2ncccc2Br)(F)F)CC(C2CC2)=NO1 C1(NC(c2c(C(C)C)cccc2)=O)CCC(S(C)(=O)=O)CC1 c1(NC)ccc(C(=O)NCCN2CC(CC3CCC(C(=O)NC)CC3)C2)c(N)c1 N1(C(C(C)n2ccnc2)=O)CCC2C1CCCN2C(c1cc(Cl)cc(F)c1Cl)=O c1(C(=O)NC2C3(CC(NC(COCC=C)=O)C3)C2)ccc(N)cc1C Cn1ccc(=O)c(C(=O)OCc2nc(-c3cnccn3)no2)c1 CCCC(C)(CCC)C(=O)N1CC2CCC2(CCNC(=O)CC2=CCCC2)C1 C1(C(=O)Nc2cncc(OC)c2)CN(C(c2cnccc2C#N)=O)CC12CCC2 CC1CN(C(c2c(F)cccc2Cl)=O)CCCN1C(C1CCCC1(F)F)=O CCCCCC(C)(C)C(=O)N1CCC(N(C(=O)CCCN(C)C)C)C1 c1(NC(C(C2CCOCC2)OC)=O)cccc(CNC(=O)C(C)c2ccsc2)c1 C1(CNC(c2nc(C(C)=O)sc2)=O)CC(C)(C)CCC1NC(c1ccc(C)s1)=O C12(C(=O)NC(C3CCCN(C(=O)CN(C)C4CC4)C3)C)CCC(CC1)CC2 C(C(=O)NOC(CC(C)C)C(=O)N(c1ccccc1)C)(C(C)C)SCC N1(C(C(CCC)NC(=O)CC2CC2C2CC2)=O)CC(C)OCC1C N=c1ccc(C(N2C(C(=O)NCC(O)CF)CCC2C2CC2)=O)n[nH]1 C12(CNC(=O)CC3OCCO3)CCC1CCN2C(=O)COc1cc(F)cc(Cl)c1 C(=O)(C(C)(CC)C(=O)NCCC1(O)CN(C(c2ncc(F)cn2)=O)C1)OCC c1(CC(CCO)NC(=O)CNC2CCOCC2)ccc(F)cc1F CC1(C)CCCCC1C(N1CCC(=CC(N2CC3CC2CO3)=O)CC1)=O c1(NCC(=O)NCCC(C)N(C(=O)CCC2CCOC2)C)ccccc1Cl n1(CC)nc(C(=O)NCC2(CNC(=O)CCc3cnn(C)c3C)CC2)cc1C C1(C(=O)OC)CCC(C2CC2)N1C(C1CN(C(=O)N(CC)CC(C)C)C1)=O c1(C(N2Cc3c(C(=O)NC4CC4)ncn3CC2)=O)cc(F)cc2cc[nH]c12 N1(C(c2cccc(OC)n2)=O)CCN(C(C2(C)CCCCC2C)=O)CC(C)(C)C1 C(=O)(CCCCCS(N)(=O)=O)N(CC(CN(C(=O)CCn1cnnn1)C)O)C Cc1cccc2c1OC(C(=O)NCCCN(C)C(C1C(C)(C)OC1(C)C)=O)C2 c1(CCC=C)ccccc1C(N1CC(CNC(=O)CC2CCCOC2)C(C)C1)=O Cc1nc(O)ccc1C(N1CCCC(C(=O)NCC2CCC(CO)CC2)C1)=O c1(C2(C(=O)NC3(C(=O)O)CCN(C(=O)OC(C)(C)C)C3)CC2)cccc(Cl)c1F CC1CC(C(=O)NCC2CN(C(c3snc(O)c3Cl)=O)C2)Cc2nn[nH]c21 N1(C(CCN(C)CC)=O)CCC(C)(CNC(c2ccc(C)cc2N)=O)CC1 N1(C(CC(=C=C)C)=O)CC(NC(=O)C=Cc2nccs2)CC2(CC2)C1 Cc1c(Cl)ccnc1C(=O)NCC1(CNC(=O)CC2CCC(O)C2)CCCC1 C(=O)(CCC[N+](=O)[O-])N(CC(C)CNC(c1ccn(C)c1)=O)C C1(NC(Cn2cc(C3(COC)CCC3)nn2)=O)CCCCCC1OC C1(N=c2[nH]c(=N)[nH]c(=NC(C)COCC3CCC3)[nH]2)(CC)COC1 N1(C(c2cncc(C)n2)=O)CCC2CN(C(C3CCC34CCC4)=O)C2C1 C1(S(N)(=O)=O)(C(=O)NC2C(CNC(Cc3cnc(C)s3)=O)CCCC2)CCC1 CN1CCN(C(=O)C(O)C2CN(C(C3(C)CCC4CC4C3)=O)C2)C(CO)C1 c1(C(=O)NCC2CCCN2C(=O)CCc2cccc(CO)c2)ccc([N+](=O)[O-])o1 C12(NC(C(CCC)NC(C)=O)=O)CC3CCC(C1C2)N3C(=O)C(=O)NCC(F)F N1(CC(=O)NC(CC)CN(C)C(C2CCCC2C)=O)CCC(OCC(F)F)CC1 c1(C(=O)NC(C)C)cncc(=NC(c2ccc(F)c(F)c2)c2ccccc2)[nH]1 c1(CC)ncc(C(=O)NC2CCC(C(=O)NCCN3CCCCC3C)C2)cn1 c1(C(N2C(C)C(C)N(C(c3cscn3)=O)CC2)=O)cnn2c1OCC(C)(C)C2 S(=O)(=O)(c1ccc(NCCOCC2CC2)nc1)NC1CC(C)SCC1 C1(C(C)NC(=O)CC2CC(C(F)F)C2)CN(C(c2nccnc2N)=O)CCO1 C(=O)(C(C)C(O)CC(C)C)N(CC(C)NC(=O)CSCC(N1CCCC1)=O)CC C(CC(CNC(=O)C(C)NC(c1cnoc1C)=O)NC(=O)Cc1cnc[nH]1)OC C1(CC)CCN(C(C2CNC(=O)N2)=O)C1C(=O)NC(C(C)C)c1ncc[nH]1 c1(N(CCNC(C2CC(=O)N(CC(C)C)C2)=O)CC)cncc(C#N)n1 C=C1CC2CC1CN2C(c1ccc(C(F)F)o1)C(=O)NCCCF C(C)(C)(C(C)NC(=O)CSCc1cscn1)NC(C(C)c1cccs1)=O Cc1cccc2sc(-c3nc(C4CC=CCC4)nn3CC(C)(C)CO)c(Cl)c12 c1(CC(=O)NC(CN(C)C(C2CCCC(C)(C)C2)=O)(C)C)cc(F)c(F)cc1F Cc1c(C(=O)N(C(C)(C)CC(=O)NCCC2CCC(C)O2)C)cncc1F N1(C(C2N(C(C)=O)CC(O)C2)=O)CCN(C(C2CCCCC2)=O)C(C)C1 Cc1nn(C)c2c(NCCC3CC3(Cl)Cl)nc(=NCC34CC(C)(CCO3)C4)[nH]c12 N1(C(c2ccc(C)c(C)c2O)=O)CC2CCCC(C1)N2C(=O)C(C)(C)S(C)(=O)=O n1(CC(=O)NCC2(C)CC(NC(c3c(C)noc3)=O)C2)ccc(=O)c([N+](=O)[O-])c1 Cc1cc(C(=O)NCc2c[nH]nc2C(=O)NC2CCOC2(C)C)ccc1C#N C(=O)(CC(CC)c1ccccc1)N1CCC(N(C(=O)Cc2ccno2)CC#C)C1 c1(CC)ncncc1C(N1CC(O)(CNC(=O)CC2CC2(C)C)C1)=O C1(CCN(C(C(C)OCCN(C)C)=O)C)CCN(C(=O)CCS(C)=O)CC1 c1(CN(C(=O)CCCc2nc(-c3cnccn3)no2)CC=C)cncc(F)c1 c1(C(N(CC(C)NC(Cc2c(CC)con2)=O)CC)=O)cccc(OC)c1F c1(CC(=O)NC23CCN(C(c4nocc4C4CC4)=O)CC2C3)ccc(Cl)cc1F C1(CC)(NC(c2ccc(O)c(N)n2)=O)CCN(C(c2ncccc2Br)=O)CC1 Cc1ncc(C)c(=NCCC2CCN(C(c3cnn(CC(F)(F)F)c3)=O)C2)[nH]1 C1(CCNC(CC2CC(C)(C)C2)=O)CCCN(C(c2cccc(Cl)c2N)=O)CC1 c1(C(N2CC(NCc3ncn(C)c3)C2)=O)ccccc1S(=O)(=O)N1CCCCC1 c1(CCCc2ccc(C)s2)nc(-c2cncnc2)nn1C1CCOC1C Cc1cc(O)cc(O)c1CNC1CCC(C(N2C3CCCC2COC3)=O)C1 c1(CCCC(=O)N2CC(N(C)C(c3coc(O)n3)=O)C2)ccc(Br)cc1 C(=O)(C(C)(CCC)CCC)N1CC2C(C(N(C(=O)C(F)(F)F)CCCC)=O)(C2)C1 C1(C(=O)NCC2(NC(CCOCCC)=O)CCC2)CC(O)C(F)C1 C1(C(N2C(C3CCN(C(CNC(N)=O)=O)CC3)CCC2)=O)Cc2cccnc2C1 N1(C(C2(CC)COC2)=O)CC2CN(C(C3CC4CCCCCC34)=O)CC2C1 C(=O)(C(F)(F)C(C)(C)O)N1C(C2CCN(C(c3cc(SC)oc3C)=O)C2)CCC1 C1(NC(CCCCCCCC)=O)CCOC12CCN(C(C1(OC)CC1)=O)CC2 C1(NC(c2c(C)ccnc2)=O)CCCC(NC(c2ccc(C#N)s2)=O)CC1 C1(CC)(NC(=O)Cn2cc(CN3CCC(O)CC3)nn2)CCSCC1 c1(C(=O)NC2(c3ccccc3)CCN(C(C)=O)C2)ccc2c(c1)B(O)OC2 C1(CCNC(=O)CC2CCC(=O)O2)CCCCN1C(c1cc(C2CCC2)no1)=O C=CCC(C)(C)CC(=O)NC1CN(C(c2cncc3n[nH]cc23)=O)CC1C(F)F N1(C(C(COCC=C)c2ccccc2)=O)CCC(c2ccc(C)cc2)CC1C c1(C2(F)CN(C(C3CCC(n4cc(COC)nn4)C3)=O)C2)ncccc1C c1(C(=O)OC)c[nH]c(=NCC2CCCN2C(=O)C(C2CC2)SC)s1 C(C(C)(C)CNC(=O)CC1(O)CCOC1)N(C(=O)CC1CC2(CC2)C1)C N1(C(Cn2c(C)nnn2)=O)CC(C(N2CCN3CCCC3C2)=O)C2(CCC2)C1 Cc1ccc(CC(N2CC(F)(C(=O)NC3CSC3)C2)=O)cc1 N1(C(CCOC)=O)CCN(C(c2nc(C)sc2-c2cccs2)=O)CC1CCO CC(C(=O)N1CCC(NC(c2cnn(CC3CC3)c2)=O)C12CC2)S(N)(=O)=O CC(C)(C(=O)N1CCC(C)(NC(c2ccc(N)cc2Cl)=O)C1)C1=CCSCC1 c1(C(=O)NC2CC(C)N(C(C3CC(=O)N3)=O)CC2)cn2cccnc2n1 c1(OCC)ccc(C)c(F)c1-c1ccc(C(=O)NCC2(O)COC2)nn1 N1(C(C2CCC(C)O2)=O)CCCC12CCN(C(c1cc(C3(C)CC3)on1)=O)C2 c1(CCC(=O)NCC(O)CNC(=O)C(=O)Nc2ncc[nH]2)ccncn1 c1(OC)c(C(=O)NC2COCCN(C(=O)Cn3nnc(=O)[nH]3)C2)c(C)nn1C CCC(C)(C)C(O)C(=O)NC1C(NC(=O)C(C)(C)CN2CCOCC2)COC1 C(=O)(C(CCF)NC(=O)CCCn1cncn1)N(CC(=O)NC(C)C)C C1(NC(c2cccc(NC(C)=O)n2)=O)CCN(C(=O)Cn2cccc2)CC12CC2 c1(C(N2CCC2C(N2CCC(c3ccc(Cl)cc3)C2)=O)=O)n[nH]c2cccc(F)c12 C(C(C)(CC(C)C)NC(=O)C#CC1CC1)NC(c1c(CC)nco1)=O c1(OC(C(=O)NCCC)C)cccc(NC(=O)C(c2ccccc2F)OCC)c1 C(=O)(C1=NOC(c2ccccc2)C1)N1CCC(Cc2c(C)ccs2)C1 CC1CN(C(C2(C)CC(C)(C)C2)=O)CC1CNC(c1cc(Cl)sc1Cl)=O C1(CCC(=O)NC(C)C(CO)NC(c2cnc(S)n2C)=O)CCC(=O)NC1 CC(C)CCN=C(NCc1ccc(C(C)C)cc1)N1CCC(OC(F)F)C1 c1(C(=O)NCC(CC)NC(C2(F)CCCC2)=O)ccccc1Cn1ccnn1 CCCCC(CNC(c1ccc(C(C)C)nc1)=O)NC(C1CCCOC1)=O c1(C(N2CCN(C(C(CC)C(C)C)=O)CC2C)=O)c(C)nc(C)nc1C Cc1cc(C)c(NC(C2(F)CCCN(C(C3CCN(C)C3)=O)C2)=O)cc1O C12(CC(=O)NCC(=O)NC34CCC(COC)(C3)CO4)CC3CC(CC(C3)C1)C2 C#CCC(C)C(=O)NCC1CCC1NC(C1CCCC1C(C)C)=O c1(OCC(=O)NCC(CC)NC(C2(C#N)CC=CC2)=O)c(C)cc(Cl)cc1Cl N#Cc1ccc(S(=O)(=O)N2CCCc3n[nH]cc3C2)cc1F C1(CNC(C(C)=C(C)C)=O)CN(C(c2nc(C3CC3)cs2)=O)CC1(F)F C(=O)(C(C)(C)C(=O)N1CC2(C1)CN(C(C1CC1c1ccc(O)cc1)=O)C2)OCC C1(CNC(c2nc(C(=O)OC)sc2)=O)CN(C(c2cc(CO)[nH]n2)=O)CC12CC2 CCC(C)(C)C(O)C(=O)NC(C)CCCNC(=O)Cc1ccsc1 c1(C(=O)NC(C(C)C)C(=O)NCC2CC2c2ccco2)cc2n(n1)CCC2 C1(C(=O)NC2CC(C(N(CC(C)C)C(C)C)=O)C2)CCCCCN1C N1(C(c2cnc(S(C)(=O)=O)s2)=O)CCCC12CCN(C(=O)Cc1cscn1)CC2 Cc1cccc(C(N2CCCCCC2CNC(c2ccnn2C)=O)=O)c1N C(=O)(CCCC(F)(F)F)NCC12C(CN(C(c3c(OC)ncc(Cl)c3)=O)C1)C2 N1(C(c2cc(C)cc(O)c2)=O)CCC2CCN(C(=O)CC3=CCOCC3)CC12 N1(C(c2nc(CC)on2)C)CCC(CCNC(c2nc(CC)cs2)=O)CC1 c1(OCCC)ccc(C(=O)NC(C)CCNC(c2cc(C3CCC3)no2)=O)cc1 c1(CC)nn(C)c(CC(=O)NC2CC(CNC(=O)C(O)C(C)SC)C2)c1Br C1(NC(C(CCC)=CCC)=O)CCN(C(c2ccc(CC)c(N)c2)=O)CC1F c1(C(=O)NC2CCCN(C(=O)CCN3CCCC3)CC2)cnc2cc(Cl)ccn12 C(CC(=O)NC1CCN(C(c2cocn2)=O)CC1O)(C(N)=O)NC(C)=O N#Cc1cccc(CN2CCOCC(NC(C3CC3C3CC3)=O)C2)n1 C(CCCCCC(=O)N1CC(C2CC2)(CC)C1)NC(c1nc(CC)sc1)=O N1(C(C2C(C)N(C)CC2)=O)CC2CN(C(c3ccccc3Cl)=O)CC2(C)C1 c1(C(N2CC(C)(C)C2COC)C(=O)NCCCCCC)nc(C)n(C)n1 C#CCC(C(=O)Nc1cnc(SC)nc1)NC(C1CC1Cl)=O CCCC(CC)C(=O)NC1CCCCC1CNC(=O)Cc1c(C)noc1Cl N1(C(Cn2c(C)ccn2)=O)CCN(C(=O)C=C(Cl)Cl)C(C(C)(C)C)C1 C1(NC(C2C(=C)CC2)=O)(CNC(c2cc(Br)no2)=O)CCCC1 c1(OC)cc[n+]([O-])c(C(=O)NCCC2CC(NC(c3cc(Cl)c(C)cn3)=O)C2)c1 c1(C(=O)NCCN(c2cnc(OC(C)C)cn2)CCC)nc(C)c(C)s1 C1(CNC(CSCC)=O)CCC2CN(C(c3c(C)ccc(Cl)c3F)=O)CC12 C#Cc1cnn(C)c1C(=O)NCC1CCCCN1C(=O)C(COC)N(C)C c1(CC(=O)N(CC2CCN(C(CC3C(CC)C3)=O)CC2)CC)ccc(F)c(Cl)c1 c1(C(N(C(C)C)NC)=O)ccc(CNC2(N3CCCC3)CCOC2)o1 c1(OC)c(C)cc(C(=O)N(C2CC(C(=O)NCc3ccccc3F)C2)C)cc1C C1(CNC(CCc2cncc(OC)c2)=O)CC(NC(=O)C(=O)N(C)C)C12CCC2 CCCC(C#N)C(=O)N1CC(C)(OCC(=O)N(C)C(C)C2CC2)C1 CC1(C)CCCC1CNC(=O)C=CCNC(=O)CNC(=O)C1CC1 N1(C(C(C)n2cccn2)=O)CCC(CCNC(C23CCC2C3)=O)CC1 CC(C)CCC(C(=O)NCC(C)CC1CCCC1)NC(C12CCC(C1)C2(C)C)=O c1(NC(COC(CNC(COC(CC)(C)C)=O)(C)C)=O)cc(Cl)c(Cl)n1C C=CC(C(F)(F)F)NC(C1CCCN(C(=O)C(C)C(=O)OC)C1)=O C(=O)(CCS(=O)(=O)C1CCCC1)NCC1CC(OC)CN1C(C1CCCN1C)=O c1(C(=O)NCCC(C)N(c2ncnc(CO)n2)C)ccc(O)nc1 C(C(C(C)C(C)C)NC(c1cn(CCO)nn1)=O)NC(CCOCC(C)C)=O C1(O)(C(C)NC(c2n(CC=C)ccn2)=O)CCN(C(=O)CC2CC3CCC2C3)C1 C1(C(=O)NCC2(C)CC2)CCN(C(=O)C2C3CC(=O)CC23)O1 C(CCN=c1cc[nH]c(=NCCCCC2CCCC2)[nH]1)N1CCNCC1 C1(NC(c2c(C)n(C3CC3)cc2)=O)CCN(C(=O)C=CC(C)(C)C)CC1CO C1(NC(CSCCCC)=O)(CNC(c2ccccc2SC)=O)CC2CCC1CC2 C(=O)(C(C)(C)C1=CCSCC1)NC1CCN(C(CCC(CCC)CC)=O)CC1F N1(C(C2(F)CCCN(C)C2)=O)CC2CC1CCN2C(c1ncccc1Cl)=O C1(C)(CNC(C(CC)COC)=O)COCCN(C(=O)C(F)(F)c2ccccn2)C1 N1(C(c2cc(C)cc(Cl)c2)=O)CC2CCCC2(NC(c2ccn(C)c2C)=O)C1 N1(C(C(C)N(C(C)=O)CC)=O)CCC(n2[nH]c(-c3ccccn3)nc2=S)CC1 c1(C(=O)NC2(COC)CN(C(CC3CC(CC)C3)=O)C2)cnc2ccncc2c1 C(=O)(C1c2c[nH]nc2CN1C(=O)C1=C(Cl)CCCC1)Nc1cncc(OC)c1 CC1(C)OCCOC1CC(N1CC2CC1C2NC(C1CC12CCCCC2)=O)=O C1(CNC(C2CCCN(C(C(CC)CC)=O)C2)=O)CC(=O)NC(C)C1 c1(C(=O)NCCCOCCNC(C2C(C)C2)=O)cc(C2CCC2)on1 c1(CN(C)C(=O)NCCS(=O)Cc2ccccc2)cccc(C(C)(C)C)c1 c1(CC(N2CCC(C(F)F)C2)=O)csc(C2CC2)n1 C(CCC(C(=O)NCc1ccccc1OC)N(C(C)COC)C)OCC=C c1(C(=O)NCC(=O)N(CC(=O)NCCSC)CC)cc2c(nn1)CCC2 N1(C(C(C)(C)NC(=O)C(F)(F)F)=O)CC2CC2(C(C2CC2)NC(=O)CC=C(Cl)Cl)C1 Nc1ccc(Cl)cc1C(=O)NC1COCC1CNC(C1CC1c1cn[nH]c1)=O C1(C(=O)NCCC(C)(C)NC(c2c(CCC)n(C)nn2)=O)C2CCC(F)(F)C12 c1(C(=O)NC2C(CC)N(C(=O)C(C)=C3CCCC3)CC2)[nH]c2ccccc2c1Cl C(CCCCCCCO)=CC(=O)NC(C(C)NC(=O)C(O)Cc1cnc[nH]1)(C)C C(=O)(C(CCC1OCCO1)NC(=O)C(C#N)C=Cc1ccccc1)OCC C1(NC(C(C)n2cncn2)=O)CC2(C1)CN(C(=O)C(C1CCOCC1)O)C2 Cn1nc2cc(Br)ccc2c1CN1CCC(NS(=O)(=O)c2cccc(F)c2)CC1 c1(NC(=O)NC(Cc2ccoc2)CO)csc2c1CCCC2 Cc1ccc2c(ccn2CCC(=O)N(CC(C)NC(=O)C=CC(F)(F)F)C)c1 Cc1cc(CCC(=O)NCCC2(NC(=O)C(C)CF)CCC2)cc(C)c1 C(=O)(CC(C(C)CC)NC(=O)C(C)SCCCC)NC(CCC=C)C(=O)OC c1(CC)nocc1CN(C)CC1CCC(=O)N1 c1(C(N2CCC(NC(CC(C)F)=O)C2)=O)ccc(NCCON)cc1 C=CC(C)(C)C(=O)NC1CCCN(C(C)C(=O)NC(c2ccc(O)cc2)C)C1 O=C(C1COc2ccccc21)NC1(C2CCN(C(C3CC4CC4C3)=O)CC2)CC1 c1(C(N(CCC)CCNC(C2CCC(C)(C)CO2)=O)=O)ccnc(S(N)(=O)=O)c1 c1(N(CCCC)C)nnc(-c2ccco2)n1CCCn1cccn1 CC1CC(CNC(=O)CC=CCNC(C2(CO)CCOCC2)=O)CCO1 C1(CCOC)CN(C(=O)C(C)NC(N)=O)CCN1C(=O)C(=O)NCCC(N)=O C1(CNC(c2c(C)cns2)=O)CN(C(=O)C(c2ccccn2)O)CCC1C n1(CC(=O)NC2C(NC(CCCC(CC)C)=O)COC2)cc(C)c2ccccc12 N1(C(C(C)NS(CC)(=O)=O)=O)CC2CC(CNC(=O)CC3OCCCO3)C2C1 c1(C(=O)NCC2CN(C(C3CCC(C)(CC)O3)=O)C2)cc(N)c(C)c(N)c1 N1(C(CC(=C)C)=O)CCC(CCNC(c2scc3c2CCCC3)=O)C(F)(F)CC1 C(=O)(C1SCCc2sccc21)N1CC(N(C(=O)CCc2cnoc2)C)C1 C1(Cn2cc(CCCCC)nn2)CCN(C(=O)C(C)C2CC2)CC1(F)F C1(C(=O)NC2C(NC(c3c(N)c(Cl)ccc3)=O)CC2)CCOCC12CCC2 c1(C(N2C3CN(C(c4ccc(C(N)=O)cc4)=O)CC32)=O)cc(O)cc([N+](=O)[O-])c1 C1(C(=O)NCCN(C2CC2)CC)C(C)OCCN1C(=O)CC1CCC(C)CO1 N1(C(c2c(CC)[nH]nc2Cl)=O)CCN(C(=O)CN2CC(=O)NC2=O)C2CC12 Cc1ccc(C(C)(C)C(N2CCC(CO)(NC(c3ccsn3)=O)C2)=O)cc1 Clc1ccc(C2(C(=O)NOCc3cn(-c4cccc(Br)c4)nn3)CCCCC2)cc1Cl c1(N2CCC(CNC(CSCCCC)=O)C(C)C2)nc2cc(C)ccc2o1 CCC(CC(=O)NC1CN(C(=O)Cc2nc(=N)[nH][nH]2)C1)C(F)F CC(N=c1cc[nH]cc1S(=O)(=O)NC1(C)CCCC(C)(C)C1)C1(N(C)C)CCC1 N1(CCOC)CCC(NC(c2cc(=O)n(C)cn2)=O)C(O)C1 C(=O)(C1=CCCCCC1)NCC1CN(C(=O)CC2COCC2O)CCC1CO Cc1ccccc1-n1cc(C(N2CCN(C(N)=O)CC2)C2(N(C)C)CC2)nn1 C1(C(N(C)Cc2cn(CCCOCC(C)C)nn2)=O)CC(c2ccccc2)=NO1 C1(CC(N2CCCC(C)C2)=O)N(C(c2ccn(C3CC3)n2)=O)CCC1(C)C C(Cc1ccoc1)(C(=O)NOCCCC1CC1)NC(c1cc(C(C)C)on1)=O C(C(=O)NC1C=CC(C(N2CC(OC(F)F)C2)=O)C1)(C(C)C)SC C(=O)(C1CCCc2nnn(C)c21)NC1CN(C(c2c(CC)n[nH]c2)=O)CC(F)C1 C1(C(N2C(CC)C(CO)CC2)=O)Cc2c(C)cccc2O1 c1(C(=O)NC(CNC(C(C#N)C2CC2)=O)C2CC2)ccc(-n2cccn2)cc1 Cc1c(Cl)ccnc1C(=O)NC(C1CCCCN1C(=O)CCCSC(C)(C)C)C N1(C(c2cc(C3CC3)c(CC)o2)=O)CCN(C(=O)C(C2CC2)OC)CC1CC.CC C(=O)(C1=Cc2ccccc2C1O)NCCN(C)C(c1cccc2nc(O)oc12)=O C=CC1(CO)CCN(C(C2C=CCCN2C(c2cc(Cl)ns2)=O)=O)CC1 N1(C(C(C(C)C)N(CC)CC)=O)CCC2(C1)CN(C(=O)CN1CC=CC1)C2 Cc1nc(C(C)C)ncc1C(=O)NCC(C1CCC1)NC(=O)C(Cl)=CCl c1(COC)cccc(C(=O)NC2(CNC(=O)CN3CCOC3=O)CCCCC2)c1 N1(C(C=C(C)C(F)F)=O)CC2C(CN(C(=O)CC(C)N(C)C)C)C2C1 C1(C(=O)NCC(C)(Cn2cccn2)NC(C=C(C)Cl)=O)CCN(C)S1(=O)=O C(CCCCF)NC(=O)Cn1cc(COCCCCO)nn1 N1(C(CONC(c2c(C#C)ccs2)=O)=O)CC2CC(C)C2C1 C1(NC(CC=CC=C)=O)CN(C(C2(N(C)C)CCCSC2)=O)CCC1C(F)(F)F Cc1n[nH]c(=NC(=O)c2ncn3cc(C(N)=O)sc23)n1C C1(CNC(C(C)OCCCC)=O)CCN(C(c2ccnnc2)=O)C12CC2 CCN=C(NCCC1CCC1)NCc1cccn1CC1OCCC1C CC1OC2(CNC(N3CCOC(c4cccc(F)c4)C3)=O)CCC1C2 c1(C(N2CCCC(N(C(C=COCC)=O)CC)C2)=O)cn2ccn(C)c(=O)c2n1 N1(C(=O)NCc2cccc(CN(C)CC)c2)C2C=CCC1CCC2 c1(C(=O)NCCCCC(C)NC(C2CCS(=O)(=O)C2)=O)c(N)nn2ccccc12 CN=c1ccc(C(N2CCCC2C(C)(C)C(N2CCSCC2C)=O)=O)c[nH]1 C1(NC(C2(C)CC3CC3C2)=O)CN(C(c2ccsc2)=O)C2(CCCC2)C1 c1(OCC)cncc(C(=O)NCc2cc(C(N3CCC(C)C3C)=O)n(C)n2)c1 C1(O)(CNC(C=CC=CCCCCC)=O)CCN(C(=O)CC2CNC(=O)C2)C1 C1(NC(c2ccc(C)nc2)=O)CC2CN(C(C3(C4CCC4)CC3)=O)CC12 C1(C(C)OC)CCN(C(=O)C=CC2CCCN2C(c2n[nH]c(=N)[nH]2)=O)CC1 N1(C(COCC#C)=O)CCC(F)(C(=O)NC2CCC2OC(N2CCCC2)=O)CC1 C1(NC(=O)OC(C)(C)C)(NC(C2C3CC4C(C3=O)C24)=O)CCS(=O)(=O)CC1 C(=O)(CS(=O)(=O)C1CC1)NC1CC(NC(c2c(COC)nn[nH]2)=O)C1 N1(C(C2CCCOC2)=O)CCC(C(F)(F)F)C(N=c2cc(Cl)c(O)n[nH]2)C1 C1(CNC(c2c(CC)non2)=O)CCN(Cc2ccnn2C(C)(C)C)CC1 C=C1CC(C(F)(F)F)(C(N2CC(O)(CNC(C3CCCCS3)=O)C2)=O)C1 C1(O)(C(N2CCCC(NC(c3occ4c3CCC4)=O)C2)=O)CC2(CCOCC2)C1 c1(CN(C(C2(CC)CN(C(c3ccsc3C)=O)C2)=O)C)cccc(C)c1 c1(C(=O)NCCOCC(=O)NC(c2nccs2)CC)cnccc1OC Cc1ccccc1C(=O)NC1(CCNC(=O)CC2CCC(=O)N2C)CC1 N1(C(CC=CC)=O)CCC(c2ccccc2)(NC(=O)C(CC)OCC)C1 C1(CCCNC(c2c(SC)csc2)=O)CCN(C(=O)C(CCO)N(C)C)CC1 c1(C(N(C(CCNC(COC(CC)C)=O)C)C)=O)c(F)ccnc1Cl Cc1nn(C)c(C)c1C(=O)NC1CCCCC1C(N1CCCC(CCCO)C1)=O C(=O)(C(F)CCC(C)C)NCC(C1CCN(C(C2CC(CC)OCC2)=O)CC1)O O=C1CC(C(=O)N2CCN(C(C3CC4CCCC34)=O)CC2)=NN1.C12(CC1)C(=O)N2 Cc1nc(N2CCC(NC(c3sccc3C(C)C)=O)C2)ccc1C#N Cc1ccc2c(CCC(N3CC(F)(CNC(C4CC4(C)CF)=O)C3)=O)c[nH]c2c1 CC(O)C(C)CNC(=O)C(CC1CCC1)NC(=O)CC(C1CC1)C1CC1 CC#CCC(C(=O)NCC1CC2CCCC2C1)NC(c1cccc(C)c1)=O C1(C(C)(C)C)CC(CNC(C2(F)CCOCC2)=O)CN(C(C2CCCOC2)=O)C1 C(=O)(CCC1=CCCCC1)N(C(CC(=O)NCC1(C)ON=C(C)C1)C)C C1(NC(C(CO)OC)=O)COC2CN(C(=O)CC3CCSC3)CC12 C1(CNC(c2cncc(CC)c2)=O)CCCCCN1C(c1cn(CC)nc1C)=O N1(CC(COCC(C)C)O)CCC(C)(NC(c2cnc(Cl)c(Cl)c2)=O)CC1 C1(C(=O)NCCCC2(NC(C(=O)NCCOC)=O)CC2)CS(=O)(=O)CC12CC2 CC(N=c1[nH]c2cc(Cl)ccc2o1)C12COC(CCO1)C2 Cc1ccc(C(=O)NCCOCCC(N2CC(=O)NC(C)C2)=O)c(C)c1 CC1=C(C(=O)NCC2CC3(CC(NC(c4cnc(S)nc4)=O)C3)C2)CCC1 CCC(F)(F)CC(=O)N1CCCCC1C(C)NC(c1cc(C2CC2)[nH]n1)=O CC1CCC(OC(c2c(O)ncc(Br)c2C)=O)C=C1C(N)=O Cc1ccc(C)c(C(N2CCC(NC(=O)C(C)(C)n3ccc(C4CC4)n3)C2)=O)c1C N1(C(CC=CC)=O)CCN(C(c2ccnc(C3CCC3)c2)=O)C(C(F)F)C1 C1(O)(CNC(C2CC(C)(CNC(CSC)=O)C2)=O)CC(C)(C)C1 c1(C(C)NC(c2c(C)n(CC(F)(F)F)nc2)=O)ccc2c(c1)CC(=O)N2C c1(CC)ncc(C(N2CC(NC(C3CC34CCOCC4)=O)CC(F)C2)=O)c(O)n1 c1(C(N2C(c3ncc(C)s3)CCCC2)=O)cc(O)c(Br)c(O)c1 CC1CN(C(=O)C(F)CC2CCOC2)CC1NC(C1CCNC(=O)C1)=O Cc1nc(C=CC(N2CCCC2(C)CNC(c2ccncc2)=O)=O)cs1 C(=O)(CC(C(F)F)n1ccnc1)N(CCCN(C(c1nn(CC)c(C)c1)=O)C)C c1(C(=O)NCC2OCCCN(C(C3C(C)CCO3)=O)C2)cccn2[nH]c(=N)nc12 c1(NC(c2ccc(CC)[nH]2)=O)cc2cccc(Br)c2nc1C C1(C(C)(F)F)(C(=O)NC2(C)CN(C(C(C)NC(N)=O)=O)C2)CCOCC1 C=C(C)CCCC(=O)NCC1CC1CNC(=O)C(C)(C1CCOCC1)OC Cc1cnc(NC(Cc2cccc(Cl)c2)CO)c(S(=O)(=O)N2CCC(CF)C2)c1 c1(C(N(C2CCN(C(C3(C(=O)OC)C=CCC3)=O)C2)C)=O)cccc2ncsc12 C(=O)(C(F)(F)CC(C)C)N1CC2C(NC(Cc3c(CC)cccc3)=O)(C2)C1 N1(C(C2C(C)=C2)=O)CCC2(CC1)CCN(C(C1(CCF)CC1)=O)CC2 N1(C(c2c(C)snc2)=O)CCc2cc(-c3cn(C4CCOC4)nn3)ccc21 c1(C(=O)NC(C(CO)NC(C(C(C)C)c2ccn(C)n2)=O)C)n[nH]c2c1CCC2 C(CCC(C(=O)NCCc1[nH]cnc1C)NC(c1ccsc1OC)=O)OC C1(NC(C2CCCCN2CC(F)F)=O)CCN(C(C2CC(F)C2)=O)CC1F C1(NC(C2CCN(CC#C)CC2)=O)COCCN(C(C2CC3CCC2O3)=O)C1 c1(OC)ccc(C(=O)NCC2(F)CC(NC(C3CCCS3(=O)=O)=O)C2)nc1Cl c1(CC2(C(C)NC(C3CCC(CC(C)C)C3)=O)CC2)noc(C(N)=O)n1 C(=O)(CC1NC(=O)c2ccccc21)N1CCC(NC(CNS(NC)(=O)=O)=O)CC1 c1(C(=O)NCCCn2cc(CCS(C)(=O)=O)nn2)ccc2ncccn12 Nc1ccc(C(=O)NC2CCCC(NC(=O)CN3CCCC3=O)C2)cc1O N1(C(C(CCC=C)NC(=O)CCSCC)=O)CC2CC(C1)N(C)C2 c1(C(N2C(C(C)NC(=O)CC3CCC34CCC4)CCC2)=O)cnn2ncccc12 CC1Cc2c(Cl)cccc2C1NS(=O)(=O)c1ccc(NC2CC2)cc1F N1(CC)CCC(NC(c2ncoc2CNC(=O)C(C)(O)C2CCC2)=O)C1 N1(C(C2CN(C(=O)C=CCO)CCO2)=O)CC(F)(F)CC1CO CCC(C)C(O)C(=O)NC1CCC(C(N2CCOC(CC)C2)=O)CC1 CCC(C)(C)CC(=O)NC1CCCC1NC(=O)C(C)CCCC CCC(C)C(C(=O)NC1CCC(CNC(C2(CC(C)C)CCCC2)=O)CC1)OC c1(OC)cc(C(=O)N(CC(O)CN(C(=O)C2=CSCS2)C)C)n(C)n1 C1(C(N2CCCC2CO)=O)CN(C(c2cnccc2-c2ccccc2)=O)CCO1 C(C)(C(C)(C)C(=O)N1CCCC(OC)C1C)NC(c1n(CC)nnc1)=O c12cc(Br)ccc1SOc1scc(n1)N(C(C)=O)C2=O.C(C(=O)OCC(N)=O)OC N1(C(COC(C)=O)=O)CCC(NC(c2cc3c(cn2)CCCC3)=O)C12CCCC2 C1(O)(CC(=O)NCC2(OC)CN(C(c3cn(CCO)nn3)=O)C2)COC(C)(C)C1 Cn1nc(C(=O)NCC2CCCN2C(=O)CC2(C)CC2(F)F)cc1CO c1(C(=O)NC2CCC(N(C(C=CC)=O)C)C2)ccc(Cl)c(F)c1O c1(C(=O)NCC(C2(O)CCN(C(c3nn(C)cc3N)=O)C2)C)ccc[n+]([O-])c1 C1(C(N(C)Cc2nnc(C)s2)=O)CN(C(c2[nH]ccc(=O)c2C)=O)CC1C1CC1 C(CO)(C(=O)N(CCCN(C)C)CCNC(C1CCC1(C)C)=O)OC C=CC(C)(C)CC(=O)N1CCC(NC(C2CC23CCSCC3)=O)CC1C N#Cc1ccc(CNC2CCCCC2NC(=O)CCC2CCOCC2)nc1 C(=O)(CC(C)(C)CC(F)F)N(c1n[nH]c(C)c1C)N1CC(C2CCCO2)C1 c1(C(N2CC(O)(CNC(C3(OC)CCC3)=O)C2)=O)cccc(C(F)(F)F)c1N Cc1nc2cccc(C(=O)N(CC(C)NC(=O)C=Cc3cncnc3O)C)c2s1 n1(CC(=O)N(C2CC2)CC23CCC(C2)C3)cc(C2CC23CC3)nn1 C1(C(N2CC(=C(CNC(c3cc(C4CCC4)no3)=O)F)C2)=O)C(F)(F)C12CC2 C1(OCCC)CCCN(C(C2CN(C(=O)C(C(C)C)N(C)C)CC2C)=O)C1 Cc1c(C=CC(=O)NC2(CCCNC(C3COC(C)C3)=O)CC2)cnn1C C1(SC(C)C(=O)NC(=O)CC2CCCC2)CCN(C(=O)CS(C)(=O)=O)C1(C)C c1(C(N(CCCN(C)C(C2CC2Cl)=O)C)=O)cc2c(nc1O)CCC(C)(C)C2 CCC(C)CCC(=O)NC(Cn1cccn1)C(=O)NCC1(C)CCOCC1 N1(C(c2cnc(O)[nH]2)=O)CCc2ccc(-c3ccc4c(O)ncnc4c3)cc2C1 C#CC1CCCN(C(C2CCC=CC2NC(C2CC(C)(C)C2)=O)=O)CC1 C(CCF)(C(=O)NCCCNC(=O)OC)NC(C(CC)=CCCC)=O N1(C(C(C)NC(=O)OC)=O)CC2(C1)CN(S(=O)(=O)C(F)(F)F)C2 C1(C2CC2)(CNC(C(C=C)O)=O)CCN(C(c2cc(CC)nnc2C)=O)C1 C(=O)(C(C(C)C)C(C)C)NC12CC(CNC(CCCCOCC)=O)(OC1)C2 CC(C(=O)N1CCC(N(C)C(c2cnc(N(C)C)nc2)=O)CC1)P(C)(C)=O C1(NC(CC(C=C)(C)C)=O)CN(C(=O)C2=CCCOC2)C2CCCCC12 C1(C(N(C2CCN(C(=O)C3=CCCCC3)CC2)C)=O)CC2CCCC2C1 N1(C(c2cnc(OC)nc2C)=O)CC(NC(=O)CCCCCF)C(C2CC2)C1 c1(CCC)cc(C(N2CCCC(N(C)C(C3CC4CC4C3)=O)C2)=O)cc(O)n1 c1(C(=O)NC(CC)CNC(C2CCCC3(CC3)C2)=O)cc2c(Br)cccc2[nH]1 C1(N(C(=O)CC2C=NN(C)C2=O)C)CCCN(C(C2(c3cc[nH]n3)CCC2)=O)CC1 C1(C(N2C(CN(C(CNC(CC)=O)=O)C)CCC2)=O)CCCN1N=O c1(CC(C)(C)C)noc2ncc(C(N3CCN(C(=O)C(F)F)C(CF)C3)=O)cc12 C1(C(N2CCC3(CCC3)C2)=O)CCN(C(=O)c2cccc(CO)c2)O1 C1(C(N2CCC(N(C)CC)C2)=O)CC(NC(C2CCCC2O)=O)C(O)C1 c1(OC)cccc(C(N2CCC3(CC3C(=O)NCC3(C)OCCO3)C2)=O)c1OC c1(C(N(CCC(C)NC(c2cn(CCC)nc2)=O)C)=O)sc2ccsc2c1C CC(C)(CN=c1[nH]nc(C#N)s1)NC(c1csc([N+](=O)[O-])c1)=O N1(C(C2(C)CC(F)C2)=O)CCCCC(CNC(c2ccc(SC(F)(F)F)o2)=O)C1 N1(C(CCC#CC)=O)CCC(C)(C(=O)NCC(C)COCC)CC1 C(=O)(CC(C)(O)C(F)(F)F)N1CC(C)(CNC(C2C(C)C2)=O)OCC1 C1(C(N2C(CNC(CC=C)=O)CCC2)=O)CCC(C(F)(F)F)CC1 C1(CC)CCC(n2nc(-c3ccoc3C)nc2C2CC=CCO2)CC1 C1(NC(CC)=O)CC(O)CN(C(C2(NC(=O)OC(C)(C)C)CC2C)=O)C1 c1(OC(C)(C)C)ccnc(CNCC23CC(CCO2)C3)c1 c1(C(=O)Nc2ccc(-n3ccnn3)cc2)ccc2c(c1)CNCCN2 C1(CC)CCCCC1C(=O)N(C1CCN(C(c2ccncc2)=O)CC1)CCO C(=O)(CCC(F)(F)C(F)F)N1CCCC(O)(CNC(CC(=C=C)C)=O)CC1 C(CC(C)C(=O)NC(CNC(C1(c2ccn(C)n2)CC1)=O)CC)=CC N1(C(C(C)C#N)=O)CC(O)(C2CCN(C(=O)COc3c(F)cccc3F)CC2)C1 c1(C(=O)OCCCOCCC(=O)N(C)CCNC)ncccc1O C1(C(N2CCN(CCn3cc(COC(=N)O)nn3)CC2)=O)CC2COCC(C1)C2 CC1CCN(C(=O)CCNC(N)=O)C1C(=O)NC1CCCC1(C)CO c1(OC)ccc(S(=O)(=O)N2CCC3(CC2)CC3(C)C(=O)O)c([N+](=O)[O-])c1.C1CN1 C=CC(C)CC(=O)N1CC(N(C)C)C(CNC(C2(C(C)(F)F)CC2)=O)C1 N1(C(=O)CC2CCCCO2)CC2CCC1CN2C(c1cocn1)=O CC(C(=O)NC1CC(O)CN(C(c2ccncc2-n2cccn2)=O)C1)S(N)(=O)=O c1(NCc2c(CC)nco2)cccc2nc(COc3cccc(OC)c3)[nH]c12 S(=O)(=O)(c1ccccc1C#N)N(C)Cc1nc(Br)cs1 C1(C(=O)OCC)CCN(C(=O)C(Cc2ccc(C)cc2)NC(C)=O)C1C N#Cc1cnn2cc(C(=O)NC3CCCN(C(c4ccccn4)=O)C3)cnc12 C1(C)(CNC(C(CC)SC)=O)CCC(NC(c2cc(C(C)C)[nH]n2)=O)CC1 c1(C(=O)NC2CN(C(C34OC(C)(C)C(C3)C4)=O)C2)cnn2ncccc12 N1(C(c2c(OC)nccc2)=O)CCOC2(C1)CN(CCN=c1cc(C)nc[nH]1)C2 CC(C)CC(CNC(c1ccn(CCNC(C2(C3CCCO3)CC2)=O)c1)=O)CO C(=O)(CCCCC(C)=O)N1CC(C)(COC)C1 C1(NC(CC(C=C)C)=O)CN(C(=O)C=CC=C(Cl)Cl)CCC12CCOCC2 CC(O)(CC(=O)NC1(C)CC(NC(c2cccc(N)c2)=O)C1)c1ccccc1 c1(NC(N(C)C)=O)ccnc2ccc(C(N3CCCCC3CS(C)(=O)=O)=O)cc12 c1(C(=O)NCCC2N(C(CC=CC)=O)CCC2)c(O)cc(=O)n2c1CCCC2 C=CCC(CNC(c1ccoc1CNC(C1(C)CC=CCC1)=O)=O)CC(C)C CC(C)C(CCC(=O)NC1CCC(=O)N(C)C1=O)NC(=O)C=CC1CCOCC1 CC(C)(CCC(=O)NCC1CC2CCCC2N1C(=O)C=Cc1cc[nH]n1)[N+](=O)[O-] c1(C(C(=O)NC2CC(NC(c3ccc(OC)nn3)=O)C2)O)cc(F)c(F)c(F)c1 CC1(C)CN(C(c2ccccc2Br)=O)CC(C)(C)C1NC(=O)C1=NOCC1 c1(OCCC(=O)N(C)CC2CCCN(C(C(CC#C)C)=O)C2)ccc(F)cc1Cl C(=O)(C1OCCc2ccccc21)N1CCCCC(NC(c2ccco2)=O)C1 C1(O)(CCNC(C=CCN(C)CC)=O)CCCN(C(=O)C(C)C2(O)CCC2)C1 C1(C(N(CCCC(=O)OC)C)=O)CCC(C)N(C(=O)CCC2CC2)C1 C=CCCCCCCC(=O)NC(C)(C)CNC(c1ccnc(NC2CCC2)c1)=O CC1(C)CC(C(=O)NCCNC(C2CCCN(C(=O)CC(F)(F)Cl)C2)=O)CCO1 C(C(C)(C)C(=O)NC1CN(C(=O)Cc2cccc(F)c2)C2CC12)OC CCC(C)CCC(=O)N1CCC(OCCNC(=O)CCCn2c(C)csc2=O)C1 N1(C(CC(=O)NCC#C)=O)CCC(C2CCCN2C(=O)C(F)C2CCC2)CC1 N1(C(COCC)=O)CCC2(CCCC2C(N2CCC(C)(C)C2)=O)C1 C1(CNC(CCc2ccc(N(C)C)cc2)=O)CCOC2(CCCC2)C1 C1(Cc2cn(CC(=O)NCCCS(C)=O)nn2)CCC(C)(C)CC1 c1(C(N(C2CCCCC2NC(=O)Cn2cc(Br)cn2)C)=O)cnncc1O N1(C(C)=O)CCCC1C(=O)NC1CC(N(C(=O)C(C)C2CCOC2)C)C1 N1(CCC)C(=S)NC(c2c(Br)n[nH]c2Br)C(C(=O)OC)=C1c1cnn(C)c1 C(=O)(C(C(C)NC(C1CC2C=CC1O2)=O)C(C)C)NCc1c(C)nn[nH]1 C1(NC(CCCCC(CC)C)=O)CCOC12CCN(C(=O)CC(C)C(F)F)CC2 C(=O)(CS(=O)(=O)C1CCCC1)NC1CC(NC(c2ccc(C#C)c(C)c2)=O)C1 C1(C)(CNC(c2cc(OC)ncc2)=O)CCCN(C(C2CC(=O)C2(C)C)=O)C1 N1(C(C2N(C(c3ccnc(C)c3N)=O)CCC2(C)C)=O)CCOC2COCC2C1 N1(C(c2ccc(C)n2C)=O)CCC(NC(=O)CC2CCOC2)C(F)(F)CC1 N1(C(C(C)(c2ccccc2)OC)=O)CC2CCCC(CNc3nccc(C)n3)C2C1 N1(C(C2(C)CCSCC2)=O)CCCC(CO)(NC(=O)C=Cc2ccncc2)C1 C(=O)(CCCCCNC(=O)CC(C)(C)C)N(C)CC1CC1c1ccco1 CC(C)CC(C(=O)N1CCC(n2cc(C(c3nn(C)cc3Br)=O)nn2)CC1)N(C)C C1(NC(COC(CC)C)=O)CCCCN(CC(c2ccccc2)O)C1 N1(C(C2C(C)C2)=O)CC(O)(C(C)NC(c2csc(-c3cnc[nH]3)n2)=O)C1 Cc1c(C(=O)NCC(C2CCCN2C(=O)CCOC(C)C)(C)C)ccn1CCO Cc1nn(C)c2c(NCC3CC3(C)C)nc(N(C)Cc3cc(Cl)ccc3Cl)nc12 N1(C(c2n(CCC)ncc2)=O)C2CCC1CN(C(C1CCOCC1)=O)CC2 C(=O)(C(CNC(=O)C(O)C=CC)(CC)CC)NCC#CC N1(C(c2ncn(CC)n2)=O)C2CCC1C(F)C(NC(c1coc(Cl)n1)=O)C2 Cc1ncc2ccccc2c1C(N1CC(NC(=O)C(C)C2CC2)C2(CCC2)C1)=O C(C(C)(C(=O)N1CC2C(CC(=O)NCC3CC(OC)C3)C2C1)OC)OC c1(C(N(C)CCNC(C2C3CCC4C(C3)CC24)=O)=O)cccc2c1CCCC2=O Cc1cccc2c1CCC2NC(c1ccc(OC(F)(F)F)cc1Cl)=O c1(CN2CCN(C(c3cc(F)ccc3Br)=O)C(CO)C2)c[nH]c2c(F)cccc12 N1(C(C2CC(OC)C2)=O)CCC(NC(=O)C(C)Cc2cccnc2)C(O)C1 C1(C(N2CCC(NC(C3CC3C(F)F)=O)C2)=O)CCN(Cc2ccccc2)CC1 c1(C(=O)NCC(C2CC2)NC(c2nc(COCC)sc2)=O)sc(CC)nc1C C1(C)(CC(=O)NC(C(C)C)CNC(C2CCOC2)=O)CC(F)(F)C1 Cc1cc(N(C)Cc2ncoc2C(F)F)nc(N(CC(C)(C)C)C)n1 C(CCC(=O)NC1CCCC1NC(C1CCN(CC(F)(F)F)C1)=O)=CCC=C c1(C(N(CCN(C(C(C)Sc2ncccn2)=O)C)C)=O)cccc([N+](=O)[O-])c1Cl C1(CNC(=O)C(F)n2ccnc2)C2CC1N(C(c1cccc(C(F)(F)F)c1)=O)C2 c1(N2C3CC(CC(NC(c4c(CCC)n[nH]c4)=O)C3)C2)c(C)cncc1[N+](=O)[O-] c1(C(=O)NC2CCC(NC(c3cc(Br)ccc3Br)=O)CC2)cc(Cl)cc(Cl)c1Cl c1(CCC(=O)N(C(C)CO)Cc2cccnc2)ccc(Br)c(Cl)c1 c1(C(CC)C)nccc(N2CC(C)(NC(=O)Cc3ccnn3C)C2)n1 c1(N2CCCC(CNC(c3cn4c(n3)CCC4)=O)CC2)nc2ccccc2s1 Cc1cc(C(=O)Nc2ccc(N3CCCC3)cc2C(N)=O)n2nc(C)cc2n1 c1(C(=O)NCC(CC)NC(c2cc(C)ncc2C)=O)ccn2c1CSCC2 N1(C(C(C#N)=CC(C)C)=O)CCC2(NC(=O)C(Cl)=CCl)CCCC12 C1(C)(C(=O)NCCCCN(C)C(c2ccc(N3CCCC3)cc2)=O)CCCOC1 N1(C(c2cc(Cl)cc(C)c2N)=O)CCN(C(c2nccnc2C)=O)CC(C)(C)C1 C12CCC(CC1)NC2=O.c1(C(CC)OC)cn(CC)nn1.c1(CC(=O)N)cnnn1C c1(C(=O)NC(C2CCN(C(c3cncc(SC)c3)=O)C2)(C)C)cnc(C)cc1C Nc1cccc(C2CCN(c3cc(NC4CC(=C5CC5)C4)ncn3)CC2)c1N CCCCCCCCCC(=O)NC1C2CCN(C(=O)C(=O)C(C)(C)C)C12 C1(NC(c2cnc(Cl)s2)=O)CC2CC1N(C(c1ccc(-c3ccco3)s1)=O)C2 C1(CNC(COCCCN=[N+]=[N-])=O)CCC(NC(=O)C2=CCCS2)CC1 C1(CNC(=O)CCOc2cccc(Cl)c2)CN(C(=O)C=Cc2ccoc2)CCCO1 c1(COC)nc(Cl)cc(=NC2CCN(C(c3cn(C)c(=O)n3C)=O)C2)[nH]1 O=C(C1=CCCN(C(=O)COC2CC=CC2)C1)Nc1cccc(C2CC2)c1 N#Cc1cc(S(=O)(=O)NC2CCOCC23CCC3)ccc1N1CC(O)C(F)C1 Cc1[nH]c(=N)nc(O)c1CC(=O)NCC1(CNC(=O)C(C)N2CC(C)C2)CCC1 C1(C(C(=O)N(C(COC)C)CC)C)CCN(C(c2n[nH]cc2Cl)=O)CC1 c1(CSC)ccc(C)cc1OCCc1cccc(NC(=O)NCC(=O)N(C)C)c1 c1(C(=O)NC2C(C=C)CN(C(C3(C)CCCCO3)=O)C2)nccn2cc(C)nc12 C1(C(=O)NC(CCC)C2CCC2)CCN(C(=O)C(C)CC#N)C(C)(C)C1 CCCC(CC)CC(=O)N1CCCC(C)(CNC(c2cccc3scnc23)=O)C1 C#CCC(C)(C(=O)NCCc1ccc(O)cc1)NC(=O)C(C(C)C)SC c1(N2CC(C(=O)NC3CC3)C(OC)C2)ncnc(N(CC)CC)c1N c1(C(=O)NCC2C3CN(C(Cc4c(C)noc4)=O)CC32)cccc(F)c1F c1(C(N2CCN(C(=O)CCCn3ccnn3)C3C2C3)=O)cncc2nc[nH]c12 c1(C(N(CC)CC2CCCN2C(=O)C(C2CCCOC2)OC)=O)cc(C)nn1C c1(CNC(c2c(C)scn2)c2nnnn2-c2ccccc2)cccc(C(N)=O)c1 C1(OC)CC(NC(C2(c3cccs3)CC2)=O)CN(C(=O)Cc2cc(C)[nH]n2)C1 N1(C(=O)C=C2CCC2)CCOC(CCNC(C2(F)CC=CCC2)=O)C1 C1(CNC(=O)NCC2CCC(C)(C)O2)CCCC(F)(F)C(=O)N1 c1(C(=O)Nc2scc(-c3c(C)cc(O)cc3)n2)cc(F)c(F)c(Br)c1F C(C)(CCC(=O)N1CCOC(CCNC(c2cnn(C3CCC3)c2)=O)C1)SC c1(C(=O)NCCOCCCNC(C(C)c2cccs2)=O)ccc2c(n1)OCCO2 c1(N(C)CC2CCC2)cc(NCC2CC2C2CCC2)ncn1.c1(O)cccc(Cl)c1 N1(C(C2(CC)CC2)=O)CCCC(CNC(C2CC(=O)N(c3cnn(C)c3)C2)=O)C1 c1(COC)ccc(C(=O)NC(C)C(C)(C)NC(c2cnsc2)=O)[nH]1 N1(C(CC=C)=O)C2CCC1C(CNC(=O)CN(C(=O)C(c1ccccc1)F)C)C2 C1(CC(=O)NC(C=CC(=O)NCc2occ(C)n2)C)COCC(C)O1 N1(C(c2cc(C(N)=O)co2)C(=O)NC)CCCN(CC#N)CC1 C(=O)(C(CC(C)C)NC(=O)C=Cc1ccco1)NC(c1ccc(C)cc1)C CC1(CNC(=O)C=CBr)CN(C(c2ncc(F)cc2N)=O)CCO1 Cc1cc(=NC(CCO)C2CCC2)[nH]c(C)n1 CCC(C)C(=O)NC(c1ccccc1)C(=O)NCCC1(C)CCOC1 c1(N2CC(CC=C)(NC(C3CCCCC3O)=O)C2)nc2c(cc1C#N)CCC2 C#CCCCCC(=O)N(C1C2CN(C(c3ccc(CSCCC)o3)=O)CC12)C C=C(C)C1CN(C(C2CC3(CCN(C(C4CN(C)C(=O)N4)=O)C3)C2)=O)CCO1 C1(C)(C(=O)OC)CN(C(=O)CC2(NC(=O)CC3(C)CCOC3)CCC2)C1 N1(C(=O)CC2(O)CCC2)CC2(CC2C(N2CCC(n3ccnn3)C2)=O)C1 Cc1ccc(C)c(NC(C2(NC(c3cc(C)c(C)[nH]3)=O)CC(CO)C2)=O)c1 C(=O)(NNc1cc(C)nc(F)c1)N1CCC2(CCC(CC(=O)OC)C2)C1 C1(OCC=C)CCN(C(C2CC(CNC(=O)CCC=C(C)C)C2)=O)C1 N1(C(C(=C(C)C2CC2)F)=O)CCCCC1CCNC(C1CC(C)CCO1)=O C12(CNC(=O)CSC(F)F)CCC(CC1)N2C(=O)C(=O)Nc1ccc(Cl)cc1 C1(C)(CC(=O)NC(C(C)(C)C)CNC(=O)Cc2csc(=N)[nH]2)CCS(=O)(=O)N1 C=C(C)CCC(=O)N(C1CCCN(C(=O)C(O)CSC)C1)C C1(C(=O)NC2CC(CCNC(CCOCC(C)C)=O)C2)CCc2nncn2C1 N1(C(C(C2CC(F)(F)C2)OC)=O)CCCN(C(c2c(C)noc2C(F)F)=O)CC1C Cc1cn(CC(N2CCC2(C)C(N2CCOC3CC23)=O)=O)c(=O)nc1O Cc1nc(C(=O)N(C2C3CN(C(c4cc(C)c(Cl)s4)=O)CC23)C)c(C)o1 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CC(CNC(C(CC)CC)=O)C(O)C1 CN1C(=O)Cc2cc(S(=O)(=O)N3CCCC3C(F)F)ccc21 CCC(C)CC(=O)NCc1cc(C(=O)NC(C)Cc2cn[nH]c2)co1 c1(CNC2CC(C)(C)OC2)cccc2c1CNCCO2 c1(NC)nc(C)ccc1C(=O)NC(C1CCCN(C(=O)CCOCC(F)F)C1)C C1(C(N(C(CC(=O)OC)C)C)=O)CCN(C(C23CCC(C2)C3)=O)C12CC2 c1(C(=O)NC(CNC(C2(C#C)CCCC2)=O)(C)CO)cncc2[nH]ccc12 N1(C(C(C)(C)C)=O)CC2CCCC2(CNC(C2CC(=O)N(C(C)(C)C)C2)=O)C1 c1(C(=O)NCCN2CCCCC2)[nH]nc2ncc(-c3ccc(O)c(F)c3)cc12 C1(C(=O)Nc2cc(C)nn2C(C)C)C2CC(CC2F)N1C(=O)C(Cl)Cl C1(C(=O)NCCCC2(NC(c3cn(C)nc3)=O)CC2)CCC(C)(C)OC1 N1(C(C(C)=C2CCCC2)=O)CC2N(C(c3cccc(Cl)c3)=O)CCC2(C)C1 Cc1cccc(C(N2CCC(NC(=O)CC3CC(C(F)F)C3)C(O)C2)=O)c1Cl c1(SCC(N2CCCC(NC(C3CC4CC4C3)=O)C2)=O)ccc(F)cc1 C(CC)(CCCC(=O)Nc1ccc(F)nc1C)NC(C=CCCC)=O N1(C(C2(SCC)CC2)=O)CCC2(COCC(CNC(=O)C#CC3CCC3)O2)C1 Cc1cc2c(C(N3CCCN(C(C4(O)CCC4)=O)CC3C)=O)nccn2n1 c1(C(=O)NCCCN(C(C2CC(n3cnnc3)C2)=O)C2CC2)coc(C2CC2)n1 N1(C(=O)C2COc3ccccc32)Cc2ccccc2Sc2ccccc21 N1(C(C(CCC)OCC)=O)C2CCCC1CC(NC(C1CCC3CC3CC1)=O)C2 S(=O)(=O)(c1c(N2CCC(C)(C)C2C)cccc1[N+](=O)[O-])NC c1(CC(=O)NC2C3CN(C(C4(C#N)CCCC4)=O)C(C3)C2)ccc2c[nH]nc2c1 C(=O)(CCCC(=O)OC)N(CCCNC(CC(C)NC(C1CCCCC1)=O)=O)C c1(OC(N2CC(NC(C(c3cccs3)N(C(=O)OC)C)=O)C2)=O)ccccn1 C1(O)(CNC(CN(C(=O)CC2CCOCC2)CCOC)=O)CCOC1C c1(C(c2nnnn2CC(F)F)NC(c2ccn(C)c2)C)cc(Br)ccc1Cl c1(OC(C(=O)Nc2ccnn2CC=Cc2ccccc2)(F)F)ccccc1F c1(C(N(C2CCN(C(C3CC3F)=O)CC2)CC(C)C)=O)nnn2c1CSCC2 c1(C(N2CC(C)C(NC(c3nc(O)nc(O)c3F)=O)C2)=O)cc(Cl)cc(Cl)c1O C1(OC(=O)OC(C)(C)C)CC12CC(C(=O)NCCNC(S(=O)(=O)C(F)F)C)C2 N1(C(c2c(C)ncc(Br)c2)=O)CCCN(C(=O)C(C)CO)C(C)C1 CC(F)CC(=O)NCC1CC1.C1(C)CCNC(=O)C2(CCC2)C(=O)N1 c1(OC)ccc(Cl)cc1CN1CCCOC(CNC(c2ccc(Cl)nc2O)=O)C1 C1(NC(C2CCC2)=O)CCCC12CN(c1cc(Cl)nc(C(F)(F)F)n1)C2 c1(C(N2C(CCNC(=O)CC3CSCCS3)CCC2)=O)cc([N+](=O)[O-])n[nH]1 Cc1cc([N+](=O)[O-])cnc1N(C1CCCN(C(c2cncn(C)c2=O)=O)C1)CCO C1(N(C(Cc2nc(NC(C)=O)sc2)=O)C)CCCC(NC(C2CC(N(C)C)C2)=O)C1 c1(OCC(CNS(C)(=O)=O)O)ccccc1OC.C1(C)CCCCN1CC CCCC(CC)C(=O)NCC(C)(CC(C)C)NC(c1ccc(C2CC2)c(F)c1)=O c1(C(=O)NC(CC=C)CNC(c2scnc2CC)=O)ccnc(-n2cccn2)c1 c1(C(C(=O)NCC(CN(C(C=CC)=O)C)O)C)ccc(C(F)F)cc1 c1(C(=O)NCCCOCCOCCNC(c2ccccc2)=O)ncncc1Cl c1(OCCNC(=O)OC)cc(Nc2c(Cl)cccc2Cl)ccc1Br N1(C(c2cnc(CC)s2)=O)CCOCC1CN(C(=O)C(C1CCOCC1)F)C C1(C(=O)NCC(c2cn(C)nc2)O)CCC2(CC2)N1C(c1cncc(O)c1)=O C(c1c(F)cccc1F)=CC(=O)NCC(CN(C(=O)CC1CCOC1)C)O N1(C(CN2CCC(C)CC2)=O)C2CC=C(C(=O)NCC3(O)CCN(C)C3)C1CC2 CC1CON(C(=O)C23COC(CN4CCSCC4)(C2)C3)C1 C1(COC)(CNC(=O)C(C)NC(=O)C(C)(C)OC(C)=O)CCCO1 Cc1ccc(C(C)(C)C(=O)NCC2(NC(C3CCC4CCC34)=O)CC2)cc1 C12(C(=O)NCCC(C)NC(C3CCCN3C3CC3)=O)CCC(N=[N+]=[N-])(CC1)C2 Cn1c(C(=O)NC(C)(C)CNC(=O)CCC2CCCC(O)C2)cc2sccc12 c1(C(=O)NCC(CO)NC(C(=O)NCCOC)=O)cnc(O)n1C N1(C(c2oc(C3CC3)nc2C(F)(F)F)=O)CC2(CNC(C3(O)CC3)=O)CCC1C2 N1(C(C2N(CCC)CCC2)=O)CCCC12CCN(C(=O)C(O)CC)C2 CC(N=c1[nH]c2ccc(Br)cc2o1)C1CCCCN1C(c1ccc(F)c(Cl)c1)=O C#CCC(CC(=O)Nc1cc(CO)cc(F)c1)NC(c1ncoc1CC)=O C(=O)(CCCC(C)(C)C)N1CC(O)(CCNC(c2ccc(CC)[nH]2)=O)C1 C(=O)(C(CNC(=O)Cc1cc(C)on1)CC1CCCC1)NCC(CC)C c1(C(N(CCNC(=O)CC2CCCC2(F)F)CC)=O)cc(C)nnc1O C(CC(=O)N1CCC(CO)(OC)C1)(C(C)(C)C)NC(C(CC1CC1)OC)=O C=CCC(C(=O)N1CC(=C)CO1)NC(=O)C=C(C)C(C)C c1(C(=O)NCC(CNC(C23CCCC2C3(F)F)=O)OC)ccc(C)c(Cl)c1 N1(C(CN(C)CC)=O)CCC(CO)(NC(C2CCCS2)=O)C1 Nc1cc(Cl)nc(C(N2CCS(=O)(=O)C(CCNC(C3CC3F)=O)C2)=O)c1Cl N1(C(CC=C(C)C)=O)CC(NC(=O)Cc2csc(S)n2)CC(C)C1 CC(CCNC(=O)CC1CCCOC1)CCNC(c1cc(=O)n(C)o1)=O c1(C(=O)NC2C(NC(C3=CCCC3(C)C)=O)C2)ccc2c(Br)cccc2c1 c1c(F)ccnc1F.O=C1CCCN1Cc1cn(CC2CCCO2)nn1 Cc1nn(C)c(C)c1CC(C)C(=O)NC(C)CC(C)NC(C1(C)C=CCCC1)=O Cc1nc(C)c(C(C)NC(=O)COC2CC(NC(=O)CCC3CCC(C)O3)C2)[nH]1 C(=O)(N=c1[nH]nc(-c2ccc(C)cc2)s1)N(CCNC(C)=O)C(C)C N1(C(c2ccc(OC)s2)=O)CCC(O)(CCNC(c2sc(C)cc2Cl)=O)CC1 c1(C(N2C(CNC(CCC(=O)N(C)C)=O)CC2)=O)cc2c(F)cc(F)cc2[nH]1 C1(CNC(C2(COC)CCC2)=O)CCC(C)N(C(=O)CCc2cscn2)C1 c1(C(N2CCC(NC(C(C#C)(C)C)=O)C(C)(C)C2)=O)cccc([N+](=O)[O-])c1NC N1(C(C(NOC)=O)=O)CCN(C(C23COCC2C3)=O)CC(C)C1 C1(CN(C(=O)C=Cc2sccc2C)CC)CCCN(C(=O)C(C#N)C2CC2)C1 CCCC(C)(O)CC(=O)N1CCC(CNC(C2CN3CCN2CC3)=O)C(O)C1 Cc1cccc([N+](=O)[O-])c1N1CCC(N(CCO)CC)C1.C1(CC=O)CC2(CC2)CO1 c1(OC)nc(N2CC3CC3(CNc3cn(C(C)(C)C)nn3)C2)ncc1F C1(CCC(=O)NCC(c2ccccc2)NC(=O)CC2(O)CCC2)CCCC(=O)N1 c12cc(ccn1)CNCCCCCNc1ccc-2o1.N1(S(C)(=O)=O)CCCC1 c1(C(=O)NC2CC2NC(=O)C(O)Cc2ccc(F)cc2)cccc2ncccc12 c1(N(CCNC(=O)C=Cc2cc[nH]n2)CC)nc(C)cc(C)c1C(=O)OC C(CC(C)N=c1nc(N2CCC3(CC2)CC3C#CC(C)CC(=O)NC)c2ncccc2[nH]1)SC C1(C)(CNC(C2C(C=C)OCC2)=O)CCN(C(c2nocc2CC)=O)CC1 CN1CC(NC(C2CCC2CNC(=O)CN2C(=O)CCC2=O)=O)CCC1=O C1(c2n(CC)cnn2)CCCN(CC2(C(C)N)CC2)C1 C(=O)(C1CCCc2nncn21)NCC(CC)NC(c1csc2cc(Cl)cnc12)=O C#Cc1ccc(CC(=O)NC2CC(O)CN(C(=O)CCC3CCCC3)C2)cc1 c1(CC(=O)NCC(C)NC(CC2C(C)CCC2)=O)cccc(F)c1F C1(NC(=O)CCN2CCCCC2)COC2(CCN(C(=O)CNC(N)=O)C2)C1 c1(C(N2CCC(CNC(c3ccc(F)cc3)=O)C23CC3)=O)ccc2c(n1)CCO2 c1(SCC2CC(C)(C)C2)cc(C(=O)NCCC(O)CNC(=O)CCF)ccc1O C1(CC(=O)NC(C)C(CO)NC(N)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 Cc1cc(C(=O)NC2CCN(C(=O)C(=O)NC3CC3)CC2C)c2c(O)n[nH]c2n1 N1(CC)CC(C(N2CCC(C(C)NC(C3CC(=O)CO3)=O)C2)=O)CCC1=O Cc1nsc(C)c1C(=O)NCC1CC(F)(CNC(=O)CC2CCCO2)C1 C1(CNC(CC(CC)N(C(=O)CC2CCCCO2)C)=O)CCC2(CC2)CO1 C=CCC(C(=O)N(C1CCN(C(=O)CC2NC(=O)NC2=O)C1)CC)C(C)C N1(C(c2ccc(NC(C)=O)cc2)=O)CCCOC(CNC(=O)Cc2cnoc2)C1 c1(CNC(C2CCC(NC(c3csc(C)c3C)=O)C2)=O)nnc2n1CCC2 C(=O)(C(F)C(C)(F)F)NCCN(C(C)C)C(C1CC12CCSCC2)=O N1(C(=O)C(c2cccc(Cl)c2)O)CCC2(CCN(C(C3(CC4CC4)CC3)=O)C2)C1 [N-]=[N+]=Nc1ccnc(NCC2CCN2)c1 c1(CN(C)C(=O)NC2CNCC2O)ccccc1Cl C1(C(=O)NCC(C2CCC2)NC(c2cncc(C)n2)=O)CCC(F)(F)CC1 N1(C(C(c2ccc(C)cc2)C2CCCC2)=O)CC2CC1CN2C(C1CCOC1)=O C1(CNC(c2c(C(=O)OC)scc2)=O)CCN(C(=O)CC(C)F)CC1C C1(C(N2CCC(C(=O)OC)C2)=O)CC(C)(C)CCN1C(=O)C(C1CCOCC1)F Cc1cc(C(C)C)ccc1C(=O)OCC1CCN1C(=O)OC(C)(C)C C(CCCN=c1[nH]c2ncc(Cl)cc2s1)NC(c1cncc(CC)c1)=O c1(CC)ccc(C(=O)NCCCCCCNC(C2CCNC2=O)=O)cc1Br Cc1cc(C)c(OCC(=O)NC2CCC2NC(C2(C)CCNC2=O)=O)c(C)c1 C1(COC)CC(C(=O)O)N(C(c2coc(OCc3scnc3C)n2)=O)C1 Cc1csnc1C(=O)NC(c1ccnn1C)C(=O)N(CC(O)CN(C)C)C C1(C(=O)NC(C=C)C2CCC2)CC=CCN1C(=O)C(C(C)OC)N(C)C C1(NC(Cn2ncc(C#C)c2)=O)CN(C(=O)CSC)C2(CCCOC2)C1 C(C(C)C)(C(O)C(=O)NCC(C)(C)CNC(c1cc(Cl)ccc1O)=O)OC c1(C(=O)NC2CC(CNC(c3cc(CCC)on3)=O)CC2O)ncc(N)cc1Cl c1(C(=O)NC2(CF)CCN(C(=O)CCNc3cncnc3)C2)cnc(Cl)c(Cl)c1 N1(C(C2N(C(c3c(C)n(C)nc3)=O)CC(=O)C2)=O)CC2CC1CS2=O C1(F)(C(=O)NC(C(CC)C)CO)CCN(C(c2cccc(C#N)c2)=O)CC1 C1(CC(=O)Nc2[nH]nc(C3CCN(C(CCC#C)=O)CC3)n2)CCOCC1(C)C O=C(C1CCCc2nccn21)NCC1(F)COCCN(C(c2cncnc2)=O)C1 c1(C(=O)NCCCCC(C)NC(=O)CC2COCCOC2)ccc(Cl)c(Cl)c1N c1(OC)ccc(CCCC(=O)N(C(C)CN(C(=O)C(O)C(C)C)C)C)cc1OC c1(CNc2ccc(OCc3nc(C)sc3)cc2)cnc2cc(F)nn2c1 Cc1csc(=NCC(=O)NCC(C)(C)CNC(c2cc[nH]n2)=O)[nH]1 C(C1=NOC2COCC12)CNC(CCOC1CN(C(C(CCCC)O)=O)C1)=O C1(C(=O)NCC2N(C(=O)CCSC(F)(F)F)CC=C2)CCCCC12CCC2 c1(CC)ccc(F)cc1C(=O)NC1CN(C(=O)C(O)CC(N)=O)CC1C(F)F C(=O)(C1CCCCc2ccccc21)NCC1(O)CN(C(Cc2cc(C)no2)=O)C1 c1(C(=O)NCC2CCN(C(C(c3ccc(F)cc3)CC)=O)C2)cccc(N)c1C C1(C(=O)NCCNC(c2cc[nH]n2)=O)CN2CCCC1C2 N1(C(C2C(=C)CC2)=O)CC2CC2(CNC(c2cncc(C(F)F)c2)=O)C1 c1(OC)ccc(CNC2CC2C(=O)NCc2cc(Br)ccc2F)c(F)c1 Cc1cc2ccc(C(=O)NC(CO)CCCCNC(=O)CCC3CC3C)cn2c1 c1(CC)oc(C(=O)NC2CC(CCNC(=O)C(c3ccccc3)C)C2)cc1C c1(C(NOCC(=O)N(C2CCNC2)CC)=O)cc(O)ncn1 C(CCCCC(=O)NC(C)CS(C)=O)N(C(c1cc(CC)oc1C)=O)C c1(OC)cc(C(N2CCC(NC(c3nc(C)cs3)=O)C(C)C2)=O)cc(Cl)n1 C(C(CNC(C1(NC(=O)Cc2ccccn2)CC1(C)C)=O)C(C)C)OC c1(C(=O)NCC(C#C)CC(C)(C)C)cccc2ccc(O)nc12 C1(NC(COC(CC)C)=O)CCC(CNC(c2nc(C(C)(F)F)cs2)=O)C1 C(CCC(=O)NC(C)CNC(C1CC(F)(F)C1)=O)NC(=O)OCC N1(C(CNS(CC)(=O)=O)=O)CCC(C2(CNC(=O)CC(C)O)CCOCC2)CC1 N(C(=NCCC(C)=O)NCc1cc(F)c(Cl)cc1F)C1CC(CCC)OCC1 C1(NC(C(C)n2cnnn2)=O)CCC(O)CN(C(=O)C=CC(F)(F)F)C1 N1(C(c2cc(C)nc(O)n2)=O)CC2CC1CCC2NC(c1n[nH]cc1Br)=O CC(C)C(C(=O)NCC(C)(C)CN(C(=O)C(O)C1CCC1)C)N(C)C c1(C(C)(C)C)cncc(C(=O)NC2COCC2NC(c2c[nH]c(=N)o2)=O)c1 N1(C(C(C)OC2CCOC2)=O)CCC(NC(=O)C2=CC(C)(C)C2)C2(CCC2)C1 C(=O)(CN(Cc1ccc(OC)c(OC)c1)N(C)Cc1cc(Cl)cs1)OCC N1(C(C(n2ncc(C)c2)C)=O)CC2CC(O)C1C2NC(c1cccc(Cl)c1O)=O c1(C(N2C(CNC(C(CC=C)NC(C)=O)=O)C(C)CC2)=O)n[nH]c2ccccc12 N1(C(C2C3COCC23)=O)Cc2ccc(F)cc2C1.CC12CCCN(C1)C2=O c1(C(=O)NC2C(CNC(c3c(OC)scc3)=O)CCC2)ccccc1C(N)=O c1(C(=O)NCC(CC)NC(C2CCCCC2O)=O)cc(Br)c2occc2c1 c1(C(N2CCC(C3N(C(CSCC#C)=O)CCC3)CC2)=O)cc(N)c(Cl)cn1 n1(C(C)C(=O)N(C2CCOCC2)C)cnc2ccccc12 N1(C(C(CC(C)C)OC)=O)C2CCC1CC(CNC(c1cc(C(F)F)no1)=O)C2 C(=O)(C(CCOCCO)NC(=O)CNC(N)=O)NCC(CC)(C)Cl CC1CN(C(C2CC(F)(F)C2)=O)CCN1C(=O)C(F)(F)C1CCOCC1 N1(C(C(CN(C(Cc2c(C)occ2)=O)C)C)=O)CCC(CO)C1(C)C CC(C)C1=NOC(C(=O)NCCCCC2CN(C(C3CC4C=CC3C4)=O)C2)C1 c1(OCC(=O)N(c2c(OC)ccc(F)c2)C)ccc2c(c1)CCC2 C1(CCCNC(c2cccc(Cl)n2)=O)CCN(C(C2CC(O)C2)=O)CC1 C1(CNC(C(C(C)C)F)=O)CN(C(C2C3(CC3)C23CC3)=O)CCC1(C)C CC(C)CC(C)CC(=O)NCC(C)(C)CCNC(=O)C=CC(F)(F)F C1(C(N(C(CCNC(c2cnn(CCOC)c2C)=O)C)C)=O)CCC(C)(C)CO1 CC(C(=O)NCC1COCC1NC(=O)COc1ccccc1F)P(C)(C)=O C1(NC(c2ccc(C)cc2O)=O)CC2CC1CN(C(=O)CS(=O)(=O)C(C)C)C2 CCC(CC(=O)NCC1CN(C(c2ccsn2)=O)C(C)(C)C1)C(F)F C12(CC(N3C(CNC(c4coc(C5CC5)n4)=O)CC(O)C3)=O)CCC(CC1)CC2 C(c1cccc2ccccc12)=CC(=O)NC1CN(C(c2n(C)ccc2)=O)C2C1C2 c1(C(=O)NCC2(NC(=O)Cn3cncn3)CCC2)ccc(Cl)nc1 N1(C(C(CCC)OC)=O)CCCC(NC(c2cnn(CCN(C)C)c2C)=O)C1C C1(C(=O)NCCc2nccs2)CCC2CNCCN12 S(=O)(=O)(CCC(=O)NCCNC(=O)CN1CC=CC1)NC CS(=O)(=O)CC(=O)N(CCC(=O)NCC1CCCC12CC2)CCO Cc1nnc2n1CCC(C(=O)N(CCCNC(c1cc[nH]n1)=O)C1CC1)C2 n1(CC)ccc(S(=O)(=O)Nc2ccc(N3CCCC4CCC34)nc2)n1 c1(CN2C(C)(C(=O)NC(C)(C)CO)CC2)ccnc(Br)c1F C1(NC(C(c2ccc(Cl)s2)C)=O)CCC(C)(CNC(=O)C=Cc2ccoc2)C1 CCC(C(=O)N1CC(O)(C2CCCN2C(=O)C(C)OCCN(C)C)C1)N(C)C c1(OC)cc(C#N)ccc1-c1noc(-c2cc3scnc3[nH]2)n1 C1(C(N)=O)CCC(CNC(C2OCCC2CNC(C2(CCO)CC2)=O)=O)O1 C(C)(C)(CC(=O)NC1(C2CCCN2C(=O)CCN2CCCC2=O)CC1)OC N1(C(c2n(CCC)nc(C)c2)=O)CCC2(CCC(NC(=O)CN(C)C)CC2)C1 N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCN(C(c2nn(C)cc2N)=O)C(C)C1 CC(C)C(CCNC(=O)C(C1CC1)N(C)C)NC(=O)CN1CC=CC1 C=Cc1ccc(NC(C2CCN(C(c3ccns3)=O)C2c2cccnc2)=O)cc1 C(C(C)(C)C(=O)NCCC1CCCN1C(c1cnn(C(F)F)c1)=O)OCC CCCCC(CNC(=O)Cc1cccnc1C)NC(C1CCCC(F)C1)=O CC(CC(=O)NC1C2CCCCC12)C(C)(C)NC(c1cccc2ccnn12)=O c1(-n2ccc(CC(=O)NC(C)C(CO)N(C)C)n2)ccc(F)c(F)c1 C1(O)(CC(=O)N(C(CNC(c2cncc(C)n2)=O)C)C)CCCN(C)C1 c1(CN)cc(F)ccc1N1CCCC1.c1(N2C3CCC(C3)C2=O)ccc(Cl)nc1 C1(C#CC(=O)N2CCC(N(C(=O)CC(C)(F)F)CCO)CC2)(CC)CC1 c1(CN2CCC(N(C(C3CCC(C(C)C)CC3)=O)C)C2)ccccc1[N+](=O)[O-] Cc1ccc(C=CC(N2CCN(C)CC2CNC(=O)Cn2cc(Cl)cn2)=O)cn1 c1(OCCC)ccc(CNC(C(=O)O)C(C)OC)cn1 c1(CC(N2CCN(CCNC(C(CC)COC)=O)CC2)=O)ccc(Cl)c(C)c1 C(=O)(C(=O)N=c1ccn(-c2ccc(Cl)cc2Cl)[nH]1)NCC(C(C)N)(C)C C(CN=c1ncc(C(F)F)c[nH]1)C1CCN(C(=O)CC2C=CCC2)C1 c1(NCC(C)Nc2ccccc2)[nH]c(=NC2CCCCCCC2)nc2scnc12 c1(C(N2C(CNC(COCCCCC)=O)CC2)=O)cc(C(F)(F)F)cnc1C N1(C(C=CCNC(c2c(CC)oc(C)c2)=O)=O)CCC(OC)C(C)(C)C1 c1(C(=O)NC(CNC(C2CCCN2C2CC2)=O)CO)cc(F)cc2ccncc12 C(C)(C)(C(C)CC(=O)NCCC(CO)C(C)C)NC(c1cncc(C)n1)=O n1(CC(=O)NC(C)CCCNC(c2ccon2)=O)cc(C#N)c(O)nc1=O C(CC1=CCN(C(C2CC23CC(F)(F)C3)=O)CC1)NC(C1(CC#C)CCCO1)=O C1(OC)CC2CC(NC(=O)C(C)N(C(=O)CCn3cccc3)C)CC12 C1(CCN(C(C(F)=CCC)=O)C)CCCCN1C(=O)CC1CCC(=O)N1C c1(C(N2CC(NC(C3(C(F)(F)F)CCCCC3)=O)C(F)C2)=O)cc[n+]([O-])cc1 C1(NC(CC2CC(C)(C)N(C(C3C4CC(=O)CC34)=O)C2)=O)CCCCC12CCC2 c1(C(=O)NC2(C)CC(NC(CC3CC(=C)C3)=O)C2)noc2c1CCCC2 C1(NC(CC2CC(NC(C(C)SC)=O)C2)=O)CCc2n[nH]cc2C1 C1(CC(=O)NC(C)=O)CCCCN1CC(CC)(C)CNC(c1cc(CF)on1)=O C1(C(=O)NC(C(N)=O)CO)(NC(c2ncncc2Cl)=O)CC(F)(F)C1 CCCCS(=O)(=O)CC(=O)N1CC2CC1CN2C(c1[nH]nc([N+](=O)[O-])c1Cl)=O Cc1ccccc1-c1nc(-c2cc(CC(C)C)on2)n(CCOC(C)C)n1 c1(CCC(=O)NCC(CC)NC(COC(CC)CC)=O)nc(C)c(C)[nH]1 N1(C(C(=O)NC(C(=O)OC)C)C)CCN(C(c2ccc(C)cc2F)=O)C(C)C1 c1(CC(=O)NCC2N(C(C3CC(C)OC(C)C3)=O)CC2)ncn2c1COCC2 C1(C2CCOCC2)(C(=O)NC2CN(C(Cc3c(C)nc[nH]3)=O)C2)CC1(F)F C(=O)(C1CCc2ccccc21)N1C(C=CC(NOCC2(C)CC2)=O)CCC1 C1(C#N)(C(=O)NC(C2CCN(C(=O)C=Cc3cscn3)CC2)C)CC=CC1 c1(CCC(=O)NC(CC=C)CNC(=O)C(C)O)cc(OC)ccc1OC Cn1nc([N+](=O)[O-])cc1C(=O)NC1CC1CNC(c1cncc(C2CC2)c1)=O c1(C(N2CCCC(C(=O)NC(C(=O)OCC)C)C2)=O)c(C)nc2ccc(F)cn12 CC1CCC(C)(C(N2CC(CN(C(=O)CCCC#N)C)C2)=O)C1 C1(C)(CC)CN(C(C(=O)Nc2ccccc2OC)C2CCOC2)CCO1 c1(C(C)C)ncc(C(=O)NC23CC(C(N4CCC4C4CCCC4)=O)(C2)C3)cn1 N1(C(c2cc(CC)c(C)s2)=O)CC(N(C)C(C2CC=CCO2)=O)C(C)(C)C1 N1(C(C(CC=C)OC)=O)CCC2(CC1)CC2NC(=O)CC1(N(C)C)COC1 CC(C)C(F)C(=O)NCCC1CC(NC(c2csc(Br)c2Cl)=O)C1 N1(C(Cc2c(C)non2)=O)CCN2CCN(C(=O)CCc3cscn3)CC2C1 C1(CNC(CCSC)=O)(CNC(=O)CN2CCCCC2C)CCCCC1 c1(C(N(C2CCN(C(C3C(C)C3C)=O)C2)CC)=O)cc(F)c(C)cc1Cl N1(C(c2ccc(OC)o2)=O)CC(NC(=O)CCc2ccc(C)nc2)CCC1C C1(C(N(C2CN(C(CC3(OC)CCC3)=O)C2)C)=O)CC(=O)CO1 c1(OC(C)C)nc(C(N2CC(CCNC(=O)COCP(C)(C)=O)C2)=O)cc(O)n1 c1(C(=O)NC2CN(C(Cc3c(C)con3)=O)CC2C)csc2c(F)cccc12 C1(C#CC(=O)NC2CC(O)(CNC(=O)C3=CCCCC3)C2)(CC)CC1 N1(C(C2(CC#C)CC2)=O)CC2CCC(NC(=O)C=C(C)C(C)(C)C)(C2)C1 c1(C(N2CCN(C(c3ccccc3)=O)C(CO)C2)=O)cc(Cl)c(F)cc1F N1(C(=O)CC2C=CCC2)CCC2CN(C(c3cc4c(nn3)CCC4)=O)C2C1 c1(NS(C)(=O)=O)ccc(CCNC2CCCC(N3CCCC3)C2)cc1 N1(C(c2nc(COCC)sc2)=O)CC(C)CN(C(=O)C2=CCOC2)CC1C C(=O)(C(CC)C(=O)NCCC(C)NC(=O)C(C)(C)c1cscc1Cl)OCC C=C1CC(C(=O)NC(C)(C)C)(CO)C1.C1(OC(=O)NCCO)CN(C(C2(Cl)CCC2)=O)C1 C1(C(=O)NCC2(C(F)F)CCN(C(CN(CCC)C)=O)C2)CC2CCC(C1)O2 Cc1cnc(C(=O)NCC(C2CC2)NC(c2ccc[n+]([O-])c2)=O)c(Br)c1 c1(C(N2C(C(=O)NCC(=O)N(C)C)CC(OC)C2)=O)ccc(C)c(C)c1I n1(CCN2CCC(N(C)C)CC2)ccc2cc(C(=O)OCCCO)ccc12 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CCC(NC(C2CC3(CCC3)C2)=O)C(O)C1 Cc1cccc(-c2cc(C(=O)NCC(C)(C)CNC(=O)C(C3CC3)N(C)C)on2)c1 C12(C(=O)NCCCCCNC(C(C)O)=O)CC3(F)CC(F)(C1)CC(F)(C2)C3 c1(CC(N2CCC(C)C2CNC(=O)CNC=O)=O)csc2ccc(Cl)cc12 CC1(C)OCCOC1C(c1nnnn1C1CC1)NCC1CC2CCC(C1)O2 C1(NC(C(C)=C2CCCC2)=O)C=CCN(C(C2CC(=O)N(C(C)(C)C)C2)=O)C1 c1(CC(=O)N2C3CN(C3)C(=O)C3C2C3)c[nH]ccc1=O.CC(C)(C)OCCF N1(C(CCCCC)=O)CCOC2CN(C(c3cnn(C4CCCC4)c3)=O)CC12 C(C(C)CC(=O)NNC(=O)C(C)(C)CCCCNC(c1cc(C)n(C)n1)=O)OC c1(C(=O)NC2C(CNC(=O)CCCc3ccsc3)C2)ccc2n[nH]cc2c1Cl c1(OC)ccccc1NC(=O)C(C)N(C1CCN(CC2CC(O)C2)CC1)C C1(CC(=O)NCCN(C(c2cnn(CCF)c2)=O)CC)CN2CCN1CC2 N1(C(c2cc(C)n(C)c2)=O)CCC(C(=O)NCCC2CCOC2)C(C)C1 C(C)(C(CCc1ccccc1)NC(=O)C(C)(C)c1ccno1)NC(CC=C=C)=O C1(C(N2CC(CCNC(=O)C(C)n3ccnc3)(OC)C2)=O)(CO)CCCCO1 C1(NC(c2c(COC)ncs2)=O)CC(CO)N(C(c2scnc2Cl)=O)C1 c1(OCC)ccccc1CCC(=O)NCC1CC(NC(C2CC(F)C2)=O)CC1O Cc1c(CNC(C2C3CC3CN2C(=O)CCN(C)C)=O)nnn1C N1(C(c2c[nH]c(=NC)o2)=O)CCC(NC(=O)C(C)OC2CCCCC2)CC(O)C1 C1(C(=O)OC)CCOC1C(=O)NC12CC(NC(=O)CCSc3ccccn3)(C1)C2 c1(NCC(CC)N(C)C)cc(N(C)Cc2ccc(=N)[nH]c2)ncn1 CC1CCCCC1CC(=O)N(CC(O)CN(C(=O)CN(C1CCSC1)C)C)C CC1CCN(C(=O)C(=O)N(C)C)CCN1C(c1cncc(O)c1Cl)=O c1(C(N(C2CCN(C(C=CCCC)=O)C2)CCC)=O)ccc(=O)n(C)n1 N1(C(CCC#C)=O)CCC2(CC2NC(=O)CCNC(c2ccccc2)=O)C1 N1(C(C(c2n(C)ncc2)O)=O)CC2=C(C1)CN(C(c1ncc3ccccn13)=O)C2 C1(CC#C)(C(=O)NC(C2CN(C(=O)C(C)(C)N3CCCC3)C2)C)CCCO1 C1(CNC(c2n(CC)ncc2)=O)CN(C(C2(OC)CCC(C)(C)C2)=O)CCCO1 c1(OC)c(Cl)cc(C(=O)NC2CCCN(C(=O)CN3CC=CC3)C2)nc1Cl C1(NC(C(C)OCC)=O)(CF)CN(C(=O)COCC2CCC2)C1 c1(C(=O)NC2C(NC(C3(C)CC=CCC3)=O)CCC2)ccc([N+](=O)[O-])cc1Cl C1(CNC(CSCC)=O)C(C2CC2)CCN1C(c1c[nH]c(C(F)(F)F)c1)=O c1(C(N2CCC(N(C(CC=C=C)=O)CCO)C2)=O)cccc(N2CCOCC2)n1 C#CCCCC(C(=O)NC(C)(C)CC)N1CCC(OCCN(C)C)C1 c1(CN(C)Cc2c[nH]nc2-c2ccc(Br)cc2)ccc2c(c1)CCCN2C N1(C(c2cc(CCC)on2)=O)CCOC(CNC(=O)CCCCN2CCCC2)C1 Cc1nc(NC2CCCc3n[nH]cc32)c(Cl)cc1C#N.C(=O)(C(F)(F)F)N1CCC1=O N(C1CCc2cccnc21)C(C(CC(C)(C)C)NC(=O)CC1CC(F)C1)=O C1(NC(=O)CN2C(=O)CCC2=O)CCCCN(C(c2cocn2)=O)C1 c1(C(N2CCC(NC(=O)NC(C3CCOCC3)COC)C2)C2CC2)ccccc1C C1(O)(C(=O)NCCOCCNC(Cc2nc(C)oc2)=O)CCC(C)CC1 N1(C(c2cc(C)sc2C)=O)CC(C2CC2)(C(=O)NCCc2ccncc2)C1 C(=O)(CC(F)(F)C(F)(F)F)NCC1N(C)CCN(C(C(COC)C)=O)C1 c1(CNC(C2CNCCN2Cc2c(F)cccc2F)=O)c(F)c(F)cc(F)c1F C(=O)(C(CCC1CC=CCC1)N1CCN(c2ccc(OC)nn2)CC1)NCC=C C1(N(C(=O)CC2CC2(C)C)CC#C)CCN(C(=O)C(n2ccnc2C)C)CC1 c1(CC(N2C(CNC(CCN(CC)CC)=O)CC2)=O)c[nH]c2ccc(F)cc12 C=CC(CC)CC(=O)N1CCCC(CC(N2CC(OC(=O)NC)C2)=O)CC1 C1(NC(c2c(COC)cco2)=O)COCCN(C(C2C(Cl)(Cl)C23CC3)=O)C1 C1(CNC(=O)CCc2ccccc2)CC2CC(C1)N(C(c1cc(O)cs1)=O)C2 c1(C(=O)NC2CN(C(C=CC(=O)OCC)=O)CC2O)cc2scc(Cl)c2[nH]1 c1(C(C(=O)NCC(CO)NC(c2c(CC)con2)=O)O)ccc(F)c(Cl)c1F C1(C(=O)Sc2n(C)nnn2)CCC2(C1)CC2(F)F.c12ccc(cc1NC1CC1)[nH]2 c1(C2N(c3nnc(CCC)n3CC)CCC2)cccc(F)c1 C1(NC(C2(OC)CCSCC2)=O)CCN(C(C2CCC3CC23)=O)CC1(C)C CC(C)S(=O)(=O)CC(=O)NC1CC(NC(=O)COc2cnccc2C(F)(F)F)C1 CN(C1CCc2c(F)cccc21)C(C1CCC(OC(F)F)CC1)=O C1(CNC(CNC(CC)=O)=O)CC(C)(C)CCC1NC(=O)CN(CC)CC C=C(C)CC(C(=O)NCC1(NC(=O)C(C)OCCN(C)C)CCOCC1)OC CC(C)C(F)(CNC(C1C2CC(=O)CC12)=O)C(=O)NCc1cccnc1O c1(C(N2CC(C)(C)C(NC(C3CCOC3)=O)C2)=O)cc2cc(Br)cn2cn1 C1(NC(C(C)SC)=O)CN(C(c2c(C)nc(C)n2O)=O)CC2(CCC2)C1 C1(C(=O)NC(C)CCCNC(C2(c3cc[nH]c3)CC2)=O)CCCN(CC(F)F)C1 C(=O)(C1=CCSC1)NCCN(C(C1(C)CC(CNC(C)=O)C1)=O)C.C1CN1.C1CN1 N1(C(c2cnc(-c3c(F)cccc3F)cn2)=O)CCc2cc(O)ccc2C1 C1(O)(CCNC(c2cc(C)oc2)=O)CCCN(C(c2cncc(O)c2)=O)C1 CCC(CCOC)NC(=O)C(CO)NC(C12COCC1C2)=O C1(C(=O)OC)CCC(n2nnnc2C(C)(C2CC2)NC2(CCF)CC2)C1.C1(C)CC1 C1(NC(CNC(C(C)C2CC2)=O)=O)CCC(C)(N(C)C)CC1 CCCC(CCC)CC(=O)N1CCC(NC(=O)CN2CSCCSC2)C1 c1(OC)cc(C(=O)Nc2cnc(Cl)nc2)c(-c2c(SC)n[nH]c2C)cn1 N1(C(c2cnn(CC)c2Cl)=O)CC(NC(C2CC(C(N)=O)C2)=O)CC(F)C1 C1(C(N(C2(C(=O)NCCS(C)(=N)=O)CC2)C)=O)CCCC1C1CC1 N#Cc1ccc(F)c(NC(C2CCCC2NC(=O)CCc2ncc[nH]2)=O)c1 N1(C(C(COC(C)C)NC(C(CSC)(C)C)=O)=O)CCCN(C)CC1C c1(C(N2CC(CC(C)C)(C(=O)NC(C)CN3CCCC3)C2)=O)nnn(C)c1N C1(CNC(C(C)SC)=O)CCCN(C(=O)C=Cc2ccsc2C(F)(F)F)C1 C(=O)(CCCC(O)c1nn[nH]n1)NC(C)C(=O)NC1CCOC(C(C)(C)C)C1 C(=O)(CC(C)(C)C(F)F)NC1C(=O)NCC1(C)C.C12CC(C1)C(=O)N2C C(C(C)CC(=O)NCCNC(C1CCCN(C(c2cscc2F)=O)C1)=O)OC c1(C(N2CC(C)N(C(c3cc(O)cc(F)c3F)=O)CC2)=O)cc(C#N)ccc1F c1(CCC=C)ccc(C(=O)NCC=CCNC(C2CN(C)CC2C)=O)cc1 c1(C(=O)NCc2c(C(=O)NCc3ccc(C)cn3)n[nH]c2)ccc(C)c(C#N)c1 C(=O)(C1CCCc2nn(C)cc21)N1CC(NC(c2nn(CC)c(O)c2)=O)(CO)C1 CC12CN(C(=O)CN3CCOC3=O)C(C(=O)NC3(C(=O)C4CC4)CC3)(C1)C2 c1(C(=O)NC(C)CC(=O)NCCC2CCCC2)cc([N+](=O)[O-])c[nH]1 N1(C(CCNC(=O)OC)=O)CCC(N(C)C(C2CC(SC)C2)=O)C2(CC2)C1 N1(C(C(CSC)O)=O)CCCCC1C1(NC(c2cccc(F)n2)=O)CC1 Cc1ccc(Br)c(CC(=O)NCC(C)(CO)NC(=O)COCCC(C)C)c1 N1(C(C(COC)C)=O)CCCC(C2CCN(C(c3cncc(Cl)c3C)=O)C2)C1 C1(NC(c2csnc2C2CC2)=O)CN(C(=O)CC2=CCCCC2)CC2(CC2)C1 C(=O)(C(C)(C)C(C)(F)F)NCCOCC(=O)NC(COCC)C(C)C C1(NC(c2cc(C)c(Br)o2)=O)C2CC1CN(C(C1CCSCC1)=O)C2 c1(C(=O)OC)csc(C(N2CC(C)C(F)C2)C(=O)NCCSC)c1Cl Cc1ccccc1CC(C)C(=O)NCC#CCNC(C1(C(=O)NC2CC2)CC1)=O C1(NC(C(C(C)C)NC(C)=O)=O)CCN(C(=O)Cc2cc(C)cc(C)c2)C(C)C1 C1(NC(c2nc(COC)sc2)=O)CC2CN(C(=O)C(F)(F)C3(O)CCC3)CC12 CCCC(CNC(=O)CCc1csnn1)NC(C1CCN1C)=O C(=O)(CCCCCCSc1ccccc1)N1CCN(C)CC1Cn1cc(-c2ccccc2)cn1 Cc1ncc(CNC(=O)C(C)CN(C(=O)C(=C2CCCCC2)F)C)o1 c1(OC)cc(NCC2CCCCC2NC(=O)C(F)CC2CCCCC2)ncn1 N1(C(C2CCCC(NC(C3CC4CC4C3)=O)C2)=O)CCCC2(CCC2)C1 C1(C(=O)NCC(c2ccccc2F)NC(=O)CCC2CC2)CCCCCC1 C1(NC(c2ccc(OC)s2)=O)CC(NC(=O)C=CSc2nc[nH]n2)C12CCC2 Nc1c(C(N2CCC(NC(=O)Cn3cnc4ccccc34)C2)=O)cc(F)cc1Cl C12(NC(c3ccccc3)C3(NC(C4C(C)(C(C)C)C4)=O)CC3)CC(F)(C1)C2 c1(C(N2CC(CCC)N(C(c3nnn(C)n3)=O)CC2)=O)ccc2snnc2c1 CCC(C)CCCCC(=O)NCC1CCC2(CN(C(c3c(Cl)cnn3C)=O)C2)O1 C=CC1CCN(C(C2CC(F)CN2C(C2COCCC2C)=O)=O)CC1 C=CCCCCC(=O)N(CC(CC)NC(=O)COc1ccccc1C(C)C)C C1(C(N2CC(N(C(CC(=O)NCC)=O)C)C(C)(C)C2)=O)CSc2ccccc2O1 C1(C(=O)NC2CC(NC(c3ccc(=N)[nH]n3)=O)C2)CS(=O)(=O)CC(=O)N1 C1(C(N(C2CN(C(c3cccc(OCC(F)(F)F)c3)=O)C2)C)=O)CCC(C)(C)C1 CC(C)CC(C(=O)N(C(C)C(=O)NOC1CCCCC1)C1CC1)C(N)=O n1(C(C)C)ncc(Br)c1Cn1nnn(-c2cccc(C(F)(F)F)c2)c1=O C#Cc1ccc(Br)c(C(=O)NCC(C)NC(C2CCN(C)S2(=O)=O)=O)c1 C1(CC=C)(NC(=O)CCS(C)=O)CCCN(C(C2CC2(c2ccccc2)C)=O)C1 C(=O)(N=c1cc[nH]cc1F)C1CCCC(NC(c2cccc(O)c2O)=O)C1 N1(C(CC(C)C(F)F)=O)CC(CNC(c2cn3c(n2)CCC3)=O)CC12CCC2 N1(C(C(C)=C(C)C)=O)CC2CCOCC2(NC(=O)CCCc2ccsc2)C1 CCCC(C)(O)CNC(C1(CCNC(=O)Cc2coc(C)n2)CCC1)=O c1(N(CCCOC(CC2CC(OC)C2(C)C)=O)C2CC2)ncc(C#N)cc1Cl c1(C(=O)NCCC2CN(C(C3C(Cl)(Cl)C34CC4)=O)CCO2)ccc2nc[nH]c2n1 N1(C(CC2CC(C)(C)C2)=O)CCCC(C)(CNC(C2CC23CCCC3)=O)C1 c1(C(=O)NC(C(C)C)CNC(=O)C(F)(F)C2CC2)ccc2occc2c1 c1(C(N2CCCC(NC(C(C)OCCOC)=O)C2)=O)c(N)sc2c1CCC2 NC(=O)CCCCC(=O)NC1CCC(C(=O)NCCCNC(=O)C2CC2)CC1 N1(C(C2CCc3cncn3C2)=O)CCC2CCC(C1)N2CCCc1ccccc1 S(=O)(=O)(c1c[nH]ccc1=NCCC1CC=CCC1)NCCN=S(C)(C)=O Cc1cnc(C(N2CC(C(=O)NCC(F)Cl)C(C)C2)=O)c[n+]1[O-] c1(C(=O)NCCC2(CNC(C3C(C)COCC3)=O)CC2)cnc2c(c1)CCCC2 C(=O)(C#CC1CCOC1)Nc1c(C)cc(NC(C2C3CC4C(C3=O)C24)=O)cc1 C1(C)(C(N2CC(O)(CCNC(CC(C)c3ccco3)=O)C2)=O)CCSCC1 CN1CCCC12CCN(C(C1C=CCN1C(=O)C1=C(Cl)CCCC1)=O)C2 C(=O)(C1=NOC(C)(C)C1)NCC1CC(C)N(C(c2ccsc2Cl)=O)C1 n1(CC(=O)NC2C(NC(C3(C)CCC3)=O)CCC2)cc([N+](=O)[O-])cn1 N1(C(c2cn(C)nc2)=O)CCC(NC(=O)CCc2cc(Cl)cs2)C12CCCC2 c1(C(N2CCC(O)(CN(C(CSC)=O)C)C2)=O)ccc2cnccc2n1 C(=O)(CCCCCS(N)(=O)=O)N1CCC(C)(CNC(c2c(N)c(C)n(C)n2)=O)C1 CC(C)CCCCCN=c1[nH]c(=NCCn2cc(Br)cn2)[nH]c2ccccc12 C=C(F)C1(CC(=O)N(CCNC(=O)C(C2CCC(C)CC2)CC)C2CC2)CCC1 CC(c1cnn(C)c1)=CC(=O)NCC1CC2(CC2)CN1C(C1CCCS1(=O)=O)=O N1(C(C(CC)OC2CCCC2)=O)CCCC2C1CCN2C(=O)C1=CC(C)(C)C1 C1(C(N(CCCNC(=O)CCc2ccco2)C)=O)CCCN(S(C)(=O)=O)C1 C1(NC(C2CCC(C)O2)=O)COC2(C1)CN(C(c1cc(Cl)on1)=O)C2 C(=O)(C(O)C(F)(F)F)N1CC2C(C(=O)NCC3(C#N)CCCC3)(C2)C1 c1(C(N2CCCC(NC(CNC(C)=O)=O)(CO)C2)=O)cncc2cccnc12 CC(C)(C)CC(O)C(=O)NCC1(F)CC(NC(=O)CC2CCCC2(F)F)C1 C1(=O)C(CC(C)C)n2cc(nn2)C2CN1CCO2.c1(CC)onc(C)c1CO CC1CN(C(=O)CSCC(N)=O)CC(C)C1NC(c1cc2sccc2s1)=O Nc1ccc(-c2noc(-c3cnc(-c4cccs4)s3)n2)c(Br)c1F c1(C(=O)NCC(CNC(CCn2c(C)nc(C)n2)=O)O)cnn2c1OCC(C)C2 CCC(C)(C)CCNC(C1(CO)CCN(C(=O)CC2C=CCCC2)C1)=O N1(C(CCNC(c2ccc(F)cc2)=O)=O)CC2CC(O)CC(C2)C1 C(CCC(C)CC(=O)NCCC1CSCCN1C(=O)CCS(C)(=O)=O)=C(C)C C(=O)(CCC(CF)CF)N1CCCCC(NC(c2n(CCOC)ncc2)=O)C1 c1(C(N2CCC(O)C(CC(C)C)C2)C(=O)NCCCC)ccc2cccnc2c1 C1(OCC(N2CC(CC=C)(NC(=O)COC)C2)=O)CCC(=O)NC1=O C(N(C)N1CCN(S(C)(=O)=O)C2(CCCC2)C1)c1ccc(SC)cc1 C(CC(C)C)(C(=O)NCc1ccncc1)ONC(C=CCCC)=O CCCC(C(O)C(=O)NCCN(C(C)C)C(C)C)NC(=O)C(F)OC(F)(F)F C=CCC(C)(C)C(=O)NC(C1CCCN(C(c2conc2C)=O)C1)C c1(C(=O)OC)ccc(NC(C2CCC(NCc3cncc(O)c3)C2)=O)cc1OC c1(C(N2CC(CC(C)NC(c3c(C)nsc3)=O)C2)=O)csc2cc(Cl)cnc12 C1(N(c2cnn(C)c2)CC)CCCN(C(=O)C(N)=O)CC1 c1(C(N2C(CNC(=O)Cc3ccc(F)cc3C(F)F)CC2)=O)n[nH]c2c1COCC2 C1(C(=O)OC)CC2(CCCC2)CN1C(c1cc(Cl)cc([N+](=O)[O-])c1)=O C12(CNC(c3ccc[nH]3)=O)CC(C1)C(NC(C1CCCC(F)(F)C1)=O)CO2 CCC(N=c1cc(C)c(C#N)c(C)[nH]1)c1nnnn1CC.c1ccccc1 CN1CCC(=CC(=O)NCCC(O)CNC(c2ccccc2CO)=O)CC1 c1(C(=O)NCC2N(C(C3CC(SC)C3)=O)CC(F)(F)C2)ccc2sncc2c1 N1(C(CN(C(COC)=O)C)=O)CC(NC(c2scnc2C(C)(C)C)=O)CC(O)C1 c1(CC2NCCN(c3nc(=N)s[nH]3)C2)ccc(F)cc1[N+](=O)[O-] c1(C(N2CC(CNC(C=C(C)c3cccs3)=O)C(C)C2)=O)c(C)ccc(C)c1O CC1=NS(=O)(=O)NC=C1C(=O)N(C(C)CNC(c1c(C)cc(F)cc1C)=O)C CCC(C(=O)N(CCNC(c1c[nH]nc1C(F)F)=O)C(C)C)OC C1(CNC(CC=CCC)=O)CC(C(=O)NCc2cnc(C)s2)=NO1 C(CC(C)C)(C(=O)NC(C)C(=O)NCC(C)(C)C(N)=O)OC C1(C(N2C(CNC(c3ccc(C(F)(F)F)o3)=O)CC2)=O)Cc2ccccc2O1 c1(N2CCCC(NC(c3cscc3Cl)=O)CC2)ncnc2cccc(F)c12 N#Cc1ccc(C(=O)N(C2CCN(C(=O)C(O)C3CCC3)CC2)CCO)c(F)c1 c1(N2CC(CN(C(C=C(C)c3cccs3)=O)C)OCC2)cc(C)nc(C(C)C)n1 CC(=O)n1cc(CN2CCSC(C(=O)Nc3nnc(C)o3)C2)c2cccnc12 n1(CCCC)nc(C(=O)NC2CC2CSc2ccccc2)c2ccccc2c1=O N1(C(CN2CCC(OC)C2)=O)CCOC(C)(CNC(c2ncc(C)cc2F)=O)C1 c1(NC(C2CCCN2C(=O)NC(C(=O)OC)CO)(C)C)cncc(F)c1SC CC1(C)C(CNC(C23CCC(C2)C3)=O)CCN1C(c1cc(O)cc(F)c1)=O C(=O)(C(C)(C)CC(=O)N1CCOCC1CC(=O)NCCCCCCO)OC C1(C(=O)NC2(CC(=O)NC3C(CC)COC3)CCC2)C2(CC2)C12CC2 Cc1ncnc(O)c1C(=O)NCC1CC(C)(C)CN1C(c1ccoc1)=O C1(C(=O)NCC2(CO)N(C(c3cc(CC)no3)=O)CC2)CC(=O)N(C(C)C)C1 N1(C(C2C=CC2C=O)=O)CC(C)(OCC(=O)NOC2COCC2O)C1.CO N1(C(C=CC(CC)=CC)=O)CCCC2(CCCCC2NC(=O)CC(C)C)C1 C1(C(=O)NC2CC2c2ccsc2)CCc2ccccc2C1=O O=C(C1=C(Cl)CCCC1)NCC1(CNC(=O)C2CC2)CCCCC1 CCC(CC)CC(=O)NCCCOCCNC(=O)C(C)C(C)c1ccc(Cl)cc1 C(=O)(CC(F)(F)CC)N1C(C(=O)NCCOCC=C)CSCC1 N1(C(C2CCN(C(C)=O)C2)=O)CC2CC1CCC2NC(C12CC3CC1C2C3O)=O CC(CCC(=O)NC(C(N1CC(CO)(CF)C1)=O)c1ccco1)N(C)C CC(CS(C)=O)C(=O)N(C)CCNC(C1(CCF)CCOCC1)=O Cc1cc(C(=O)NCC2CC2CNC(c2cc(CO)c(C)o2)=O)c(O)cc1F N1(C(CCCOCCOC)=O)CC=C(C(C)(C)C(=O)N2CC(OC)CC2CO)C1 CC12CCC(n3cc(CCC4CCCN4C(=O)C(N)=O)nn3)(CO1)C2 C(CN=c1cc(Cl)nc(CS(C)(=O)=O)[nH]1)(N(C(C1C(C)OCC1)=O)C)C1CC1 N1(C(C2CCN(C(C)=O)C2)=O)CC2CC(C1)C2NC(=O)C(C(C)C)n1cnnn1 c1(C(=O)NC(C)C(C)(C)NC(=O)C(C)C(C)(F)F)ccc([N+](=O)[O-])c(Cl)c1 c1(OC)cc(C(=O)NC(C)CCNC(=O)C(C2CCCCC2)O)cc(N)c1O N1(C(c2scc(COC)c2)=O)CCC(NC(=O)CCCSC)C(F)(F)CC1 N1(C(CC2C(C)C2(F)F)=O)C2CCC1CC(CNC(c1nnc(S)n1C)=O)C2 C1(C(N2CCC(COCC)C2)=O)CN(C(=O)CN2CC(=O)NC2=O)CC1F C1(C(CC)NC(=O)C(O)Cc2[nH]cnc2C)CCN(C(c2conc2C)=O)CC1 C1(NC(CSC)=O)CCCC1(C)NC(=O)CCCn1nc(C)nc1C c1(-c2nnc(C(C)NC(=O)NC(c3nc[nH]n3)CC)s2)ccccc1F n1(C(C)C)cc(CNC(=O)CC2CC(NC(=O)C(=O)C3CCCC3)C2)cn1 C1(NC(CSCCC)=O)C(C)(C)CN(C(c2cn3ccccc3n2)=O)CC1(C)C C1(N(C(C2(n3cccn3)CC2)=O)CC)CC(NC(=O)CC(F)(F)F)CCO1 N1(C(C=Cc2ccc(C)s2)=O)CC2CCN(C(C3CC3c3ccnn3C)=O)CC12 N1(C(c2cc(C)n(CCO)n2)=O)CCN(C(c2ccsc2)=O)CC1CS(C)(=O)=O C1(F)(C(N2CC(c3ncc(SCCO)[nH]3)C2)=O)CCCOC1.CC1(C)CNC(=O)N1 Cc1nn(C)cc1CCC(=O)NCC1C2CN(C(C3CCCN3C(C)C)=O)CC12 N1(C(CN(C(COC)=O)C)=O)CC(C)C(C)(CNC(=O)CC2CCOC2)C1 CCCCC(C)C(=O)N1CCOCC(C(=O)NC(c2c(C)n[nH]c2C)C)C1 N12CCC(CC1)C2=O.C1(N(C)C(C2(OC(C)=O)CC2)=O)CCN(C2CC2)C1 CC1CN(C(=O)C(O)C(C)(C)C)CCCN1C(C1CCN(C(=O)C2CC2)CC1)=O Cn1cc(NC(C2CCC2CNC(c2cccc3c2CCC3)=O)=O)c(O)nc1=O C(=O)(C(CCC(C)C)NC(=O)C(F)C1CCC1)NCc1cccc(CC)c1 C1(O)(CNC(=O)COc2ccccc2)CCCN(C(c2cccc(=O)o2)=O)CC1 N1(C(C2(CC(C)=O)CCCC2)=O)CCCC(C(C)NC(c2cc(C(F)F)cs2)=O)C1 C1(C)(CN(C2(C3CCCO3)CCC2)C(C)=O)COCCN(C(C2CCOCC2)=O)C1 C1(CNC(C=CSC)=O)CCCC2(CN(C(c3n[nH]c4c(C)cccc34)=O)C2)O1 N1(C(c2cnc(C)[nH]2)=O)CCC2(CCC2NC(=O)C(N)CCC(N)=O)CC1 c1(C(N2C3C(NC(c4ccc(-c5c(C)ccs5)s4)=O)C(C3)C2)=O)cc(C)c(N)cn1 CC1(CNC(c2cccc(C3CCC3)c2)=O)CCCN1C(=O)Cc1ccsc1 c1(NC(C2N(C(c3c(CC)ncs3)=O)CCC2O)=O)ccc(Br)cc1I c1(C(N(CCCNC(CN(C(C)C)C)=O)C)=O)cc([N+](=O)[O-])ccc1OC(F)F N1(C(C(C)Cc2ccnn2C)=O)CCCCC(NC(c2c(O)cccc2Cl)=O)C1 c1(C(=O)NC(C2CC(C)(C)C2)C(=O)OC)cc(-c2cccc(F)c2)n(C)n1 CCC(C)(CC)C(=O)N(CC(C)NC(=O)C(C)(C)Oc1ccc(Cl)cc1)C N1(C(C(C)N(CCC)C(c2ccc(OCC)cc2)=O)=O)CCCC2OCCC12 C1(C)(CC)C=CCN1CC(=O)Nc1ccc(F)cc1 c1(CNC(=O)C=CC2CC2)ccc2c(c1)CCC2NC(=O)C1CCc2c[nH]nc21 c1(OC)ccccc1-c1ncsc1C(C(=O)Nc1nc(C(F)(F)F)nn1C)OC C(CCCCCNC(C1(CF)COC1)=O)N(C)C(C1(N(C)C)CCC1)=O N1(C(CCC(C)OC)=O)CCC(C)(C)C(C(=O)NC(C)(CO)CO)C1 c1(C(=O)NC2CC(NC(CC(c3ccc(C#N)cc3)C)=O)C2)ncnc(O)c1F c1(C(=O)NC)cccc(C(N2CC=CC(NC(=O)C3=COCC3)C2)=O)c1 C1(CC(=O)NC2C(C)CN(C(=O)CSCCC#N)C2)CCC2(CC1)CC2 N1(C(C(CCC)C)=O)CCC(C(=O)NC2CC2CCOC)C12CCC2 [N-]=[N+]=NCCCCCCC(=O)NC1CC2CN(C(=O)CN3CCCS3(=O)=O)CC12 CC(C)C(F)C(=O)N1CCOCC1CC(=O)NCCCC(C)(F)F Cc1cc(Br)cc2cc(CN3CCC(C)(C(=O)O)C3C)[nH]c12 C1(C(=O)NCCN(C(=O)CCC2CCCN2C)CC)(COC)CC2(CCC2)C1 Cc1ncn(C)c(=O)c1C(=O)NCCC(C)CCNC(c1cc(O)cs1)=O N1(C(c2c(C)scn2)=O)CCC(O)(CCNC(=O)CCC2CCCN(C)C2)C1 C1(CN(C(COCC(=C)C)=O)C)CCCN(C(=O)COC2CCN(C)CC2)C1 N1(C(Cc2cnc(C)s2)=O)CC2CCN(C(C3CCCS(=O)(=O)N3)=O)CC2C1 c1(-c2scc(CC(=O)NC(C3CN(C(C=CSC)=O)C3)C)n2)ccc(F)c(F)c1 Cc1ccncc1C(=O)NCC(N1CCN(C(=O)C(O)Cc2cnc[nH]2)CC1)=O C1(CNC(CCC(=O)NCCC)=O)CCC(C)N(C(c2nccnc2C)=O)C1 n1(C(=O)NC2CC3CCC2(CNC(=O)CCCCC2CC2)C3)cc(F)ccc1=O N1(C(c2cc(CCO)on2)C(=O)NC2(C)CC2)CCN(C)C(c2ccccc2)C1 C1(N(C(=O)C=C(Cl)Cl)C)CCCN(C(c2cc(COc3ccccc3)on2)=O)CC1 c1(N(C)C)ncccc1CNC(N1CCCC1c1ccc(Cl)cc1)=O CC(C)CC(Cc1ccccc1)C(=O)NCC1CC(NC(=O)C(C)C(C)(F)F)C1 c1(C(N2C(CCC(=O)NCc3cccc(F)c3)CCC2)=O)ccnc(CO)c1 C12(CNC(C3CC34CC4)=O)CC(CO1)N(C(c1cncc(Cl)n1)=O)C2 C1(NC(c2cnn(C)c2-n2cccc2)=O)CC2(C1)CN(C(C1CCC(O)C1)=O)C2 C1(O)(CC(=O)N(CC(CC)NC(=O)CN(CC)CC)CC)CCCN(C)C1 CCCCC(C(=O)NC1CCCC(O)C1)NC(=O)COCC C1(C(N(C2CC(NC(C3(CO)COC3)=O)C2)C)=O)CN(S(=O)(=O)N(C)C)CCO1 C1(CNC(c2cncc(C(F)F)c2)=O)C2CN(C(=O)COC3CCCOC3)CC12 C(=O)(CC(C)(C)CC)NC1C(CC(=O)Nc2ccc(CC=C)nc2)CCOC1 N1(C(c2c(CC)non2)=O)CC(C)CCC1CNC(C1(C2CC2)CCC1)=O CCCC(C)(C)C(=O)NC1CN(C(=O)Cc2cccc(OCC3CC3)c2)CC1C C12CCCC1NC1(C(F)(F)C(=O)N2CC(=O)NC)CCC1.C(c1ccc[nH]1)=CC CCCC(F)C(=O)N(CC(C)C(=O)N(C)CCN(C)C)C C(C)(CNC(C1CCOC1C1CC1)=O)(CC(C)C)NC(c1c(SC)csc1)=O C(CCNC(c1cccc(=O)o1)=O)(C(=O)NCC1COCCO1)OC c1(C(=O)NCC(CNC(c2ccc(CC)s2)=O)F)cc(C)nc2c1CCCC2 C=CCCC(C)(C)C(=O)NCc1nc(C(=O)NC(CN2CCCC2)CC)co1 C(=O)(C(F)C(=O)NCCC1CCCCN1C(c1c[nH]nc1CC)=O)OCC C1(C(C)C)(C(C)C)C(=O)N1.C(=O)(CCn1ccnn1)N(C)CC1(NC(C)=O)CC1 c1(C(N(CCNC(C(COC)O)=O)C(C)C)=O)cnn(-c2ccc(F)cc2)c1C c1(C(N2CCN(C(c3cc(C)c(C)[nH]3)=O)C(C)C2)=O)nn2cccnc2c1Cl c1(C(C(=O)NC2(CN(C)C(C3CC34CC4)=O)CC2)C)ccc(Cl)c(Cl)c1 c1(N2CCCC(CCNC(c3cc(F)cc(F)c3)=O)CC2)ncnc2c1COC2 N(C1CCCn2ccnc21)C(C(CC=C)CNC(=O)C(C(C)C)NC(C)=O)=O N1(c2c(C(N3CCC(c4ccc(F)cn4)CC3)=O)nsc2)CCCS1(=O)=O c1(C(=O)NCC(CC)(CC)NC(=O)CC2CC2(Cl)Cl)ccc(NC)c(F)c1 CC(C(=O)NC(CC1CC1)C(=O)N(CC(C)(C)C)C)S(C)(=O)=O Cc1c(C(=O)NCC(C2CC2)NC(=O)CCC2CC2(F)F)ccc(Br)c1F C(C(=O)N1CC(NC(=O)CCCN(C)C(=O)OC)C1)(C(C)C)OC c1(CCNC(C(CSCC)NC(c2cnccn2)=O)=O)ccc(F)cc1 CCCCC(C(=O)NC(C)C(=O)N1CC(n2cc(C)cn2)C1)C(C)C.C(C)C c1(C(=O)NC(C)CCNC(=O)Cc2cncc(F)c2)ccc(S(N)(=O)=O)cc1 c1(NC(C2C(NCc3c(OC)ccc(Br)c3)C2)=O)ccc2c(c1)COC2=O c1(OCC)ccc(C=CCNC(=O)COCCCSC2CC2)cc1.C1C(C)N1 c1(N2CC(OC)CC(CC)C2)nc2cccnc2c(=NC2CC(=O)N(C)C2)[nH]1 c1(NC(c2n(C)cc(NS(CC(=O)OC)(=O)=O)n2)=O)cc(Cl)c(Cl)c(Cl)c1 N1(C(C=COCC)=O)CCN(C(C2CN(C3(C(=O)O)CCOCC3)C2)=O)CC1 CC1(C)CC(N=c2nc(N3CCCCCCC3)c3cc(F)cc(F)c3[nH]2)CCO1 c1(OC(C)C(=O)N2CC(NC(C3SCCS3)=O)C2)ccccc1Cl N1(C(CC2(COC)CC2)=O)CCC2(CC1)CN(C(c1sc(COC)nc1C)=O)C2 C(CC(=O)NC1(C)CCOC1)(C(F)(F)F)NC(c1c(OC)nsc1)=O c1(C(=O)NC23CC(NC(c4cccc(NC(C)=O)n4)=O)(C2)C3)ccc(F)c(C)c1 c1(N2C(C(N(C3CCCC4CC34)C(C)=O)=O)CCC2)ncc([N+](=O)[O-])c(C)n1 C=CC(C)(O)CC(=O)NCC1CCC(NC(C23C=CC(CC2)C3)=O)CC1 C1(C(N(C(C)CN(C(=O)Cc2ccc(C(N)=O)cc2)C)C)=O)CC(C2CC2)=NO1 c1(NC(C)=O)ccc(S(=O)(=O)NC(=O)NCCCc2ccc(F)c(F)c2)cc1 C(CCC)(CCCC)NC(CC1(C=C)CN(C(=O)C(F)(F)CCC)C1)=O C12(NC(C=COCC)=O)CCCCCC1N(C(c1cccc(F)c1C)=O)CC2 C1(C(=O)NC2CN(C(C(N3CCNC3=O)C)=O)C2)CCc2nc[nH]c2C1 N1(C(C(C)=C2CCC2)=O)CC2(C1)CN(C(=O)CC1CSC1)CC2CO N1(Cc2ccc(C3(C)C(C)(C)C3)cc2)C(=O)CN(CC(N)=O)C1=O N1(C(C2C(C#C)C2(C)C)=O)CCN(C(=O)C=C(C2CC2)C2CC2)C(COC)C1 c1(C(=O)NC2CC3CC2CN(C(c2cncnc2)=O)C3)cnn2cccc(Cl)c12 c1(-c2cn(CCN(C(c3ccoc3C)=O)CC)nn2)cc(F)cc(F)c1 N1(C(CCN(C(=O)C(C2CC2)OC)CC)=O)CCC(O)CC1 C1(CC(=O)NC2CCOC2C2CC2)COCCN1C(=O)COc1ccsc1 C(=O)(C(C)(C)C(O)C(C)C)N(CCCCCC(=O)NCCCC(C)C)C Cc1cc(C(=O)NC(C(=O)NCCC(F)F)C2CCCO2)oc1C Cc1cc(C(N2CCC(O)C(NC(C3(C(F)(F)F)CC3)=O)C2)=O)cc(C)n1 CN(C)S(=N)(=O)N1CCCC1C(=O)NC1CC(NC(c2ccc(C(N)=O)o2)=O)C1 C1(NC(C=C(CNC(C(COC)(C)OC)=O)C)=O)CC2(C1)CC21CC1 c1(C(N2CCOCC(CNC(C3(C4CC4)CCCO3)=O)C2)=O)cnc(O)cc1O c1(C(N2C3CCC2COC3)=O)ccc(=NCc2cccc([N+](=O)[O-])c2)[nH]c1 c1(C(C2CCN(C(c3ccccn3)C)CC2)=O)cccc2cnccc12 c1(OC)ccccc1OCCC(=O)NC1(CN(C(=O)CCN(C)CCO)C)CC1 C(CCN=c1nc(N2CCS(=O)(=O)CC2)c2c([nH]1)CCCCCC2)OC.C1CO1 COn1cnc(C)c1C(=O)NC1CN(C(=O)CNc2ccccc2Cl)CC1F N1(C(CCN(C)C(c2c[nH]nc2C(F)F)=O)=O)CCC2(CCOC2=O)C1 C1(C(N2C(CC(=O)N(C)Cc3nccn3C)CC(F)C2)=O)CCCC2(CC2)C1 c1(CC(=O)N(CC=C)CCSc2ccccc2)ccc2nc(Cl)sc2c1 C(CCN=C(NCCOc1ccc(C#N)cc1)NC1CC2CCC1O2)NC(C)=O C1(NC(C2C(C)(C)C2)=O)CC2(NC(=O)C=C3CCSCC3)COC1C2 CC1CN(C(=O)CC2CCOC2)CC1CNC(c1ccc(-c2ccncc2)o1)=O c1(C(N2CCC(CNC(C3(C)CCOC3)=O)C2)=O)c2c(cc3c1CCC3)CCC2 c1(C(N2CCC(C3CCCO3)CC2)=O)ccc(-n2cccn2)cc1 C1(CC)(NC(=O)C(C)SC)CCN(C(C2CC(C)(C(C)(C)C)C2)=O)CC1 N1(C(C=Cc2ccc(C)o2)=O)CCC(C)N(C(=O)CCc2ccn(C)n2)CC1 Cc1cc(C(=O)NCCNC(=O)C(C)NC(=O)CC(F)(F)F)n(CC(F)(F)F)n1 C1(C(=O)NCC2OCCN(C(C)=O)C2)CC2CC(CN2)O1 C(=O)(C#CC1CCCCO1)N1CCN(C(Cn2ccc(C)cc2=O)=O)CC1C c1(C(CC(=O)NCC(C)CNC(c2cc(Cl)no2)=O)C)c[nH]c2ccccc12 N1(C(c2cc(C)sn2)=O)CCC(CC(C)NC(C2(O)CCOC2)=O)CC1 Cc1cc(O)ncc1C(N1C2CC1CN(C(=O)Cn1cnc(=N)[nH]1)C2)=O C1(C(=O)OC)CC2(CC(NC(C3(F)CCN(Cc4ccc(F)c(O)c4)C3)=O)C2)C1 c1(C(=O)OCC#CC(C)C)ccccc1OCc1cccnc1 CCC(CC)CC(=O)NC12CCCC(NC(C3CC4OC3C3CC43)=O)(C1)C2 C1(NC(=O)C2=CCCS2)CCN(C(c2cnc(O)c(Cl)c2)=O)CC1F c1(C(=O)N)cc(Cl)c2ccncc2n1.N1(C(C=C(C)Cl)=O)CC(CCC#N)C1 N1(C(C(C(C)C)OCC)=O)CC2(CCNC(=O)Cn3nc(C)nc3C)CCC1C2 Cc1cn(C)nc1C(=O)NCC1CC1NC(=O)C(C)CN(C)C C1(S(N)(=O)=O)(C(N(CCC)CCNC(=O)CCOc2ccccc2O)=O)CCC1 C1(C(=O)NC2(c3ccc(F)cc3)CC2)CC2CC2N1C(c1cc(Br)cs1)=O c1(C(N2CC(O)CC(NC(COCCC#C)=O)C2)=O)cnc2ccccc2n1 Cn1nnnc1C(C)(CCC1CCCC1)NCCCOc1nncs1 C(=O)(C1c2c[nH]nc2CN1C(c1nc(Cl)cs1)=O)NC(c1cccnc1)CC CC(C)(C)C(CC(=O)N1CCC(CCCNC(c2cc(Cl)n[nH]2)=O)CC1)C(F)F c1(C(N(CC(CC)NC(C(C)OCC=C)=O)CC)=O)cncc2nc(C)[nH]c12 N1(CC)CCCC(c2nc(-c3ccncc3)nn2-c2ccn(CC(C)C)n2)C1 Fc1ccc(-c2nc(C3CCCS3)nn2C2(c3ccccc3)CC2)c(F)c1 N1(C(c2cc(C(C)=O)sc2)=O)CCC(NC(=O)CC2CCN(C)C2)C(F)C1 N1(C(c2ccn(CC)n2)=O)CC(OC)CC(NC(c2cnn(CC(C)C)c2)=O)C1 c1(CCC(=O)NC(CNC(c2cn(C)nc2)=O)C2CCC2)ccc(N(C)C)cc1 C(=O)(CC(F)(F)F)N(CC(C)NC(=O)C(c1ccccc1)O)C C=C=CCC(=O)NCCN(CCCN(C)C)C(c1cc(-c2ccn(C)n2)on1)=O C#CCC(CC#C)C(=O)NCC1CC(NC(c2cc(N)cc(F)c2)=O)C1 c1(CC(C)(C)N(C(=O)C(c2ccc(Cl)cc2)(F)F)CCO)ccc(-c2ccco2)cn1 CN1Cc2ccc(C(N3CCOCC(CNC(=O)Cc4cccs4)C3)=O)cc2C1 CC(CCNC(C1(CF)CCC1)=O)CCNC(C1(F)CC1c1ccccc1)=O c1(OC)c(C(=O)NC2CN(C(C3CCCC(C)C3)=O)C2)cc(Cl)cc1Cl N1(C(C(=O)N(C)CC2CC(F)C(C#N)C2)=O)CCC2(CCCO2)CC1 n1(C(C(=O)NC(CNC(C=C(CC)C2CC2)=O)CC)C)ccnc1C CC(CS(C)=O)C(=O)N(CCNC(c1cccc(NC(N)=O)c1)=O)C1CC1 C12CCCC1NC(=O)C2.c12sccc1OC2=O.C1(CN(CC)CC)CCC1 N1(C(C(CCC)O)=O)CCN(C(c2[nH]ccc2C)=O)C2CCCC12 Nc1ccc(C(=O)NCC2CCCN2C(c2coc(C(F)(F)F)n2)=O)nc1N c1(CNC23CC(CC(=O)NCC4OCCN(C)C4)(C2)C3)ccc([N+](=O)[O-])cc1 C(=O)(C1=CCCOC1)N1CC(C)C(CNC(=O)CCc2cccc(Cl)c2)C1 C=CCCC(F)(F)C(=O)N(C)CCN(CC(=O)O)C CC(C)CC(C)(C)C(=O)NC(C)C(C)NC(C1(CCN(C)C)CC1)=O C(=O)(CCC(=O)Nc1nccs1)NCC(C1CCC1)NC(c1ccc(CC)s1)=O CS(=O)(=O)c1ccc(CNC2CC(C(=O)Nc3cc(Br)ccc3C(N)=O)C2)cc1 N1(C(C)=O)CSCC1C(=O)NCCC1(NC(=O)Cc2ncc(C)s2)CC1 N1(C(c2ccc(SC)s2)=O)CC(N(C)C(c2cc(C)cc(F)c2)=O)C(C)(C)C1 CC1CC(CNC(c2cc(=N)[nH]n2C)=O)CN1C(c1cnn(C2CC2)c1)=O C1(F)(CNC(COC(C)=O)=O)CCN(C(c2cnncc2C)=O)CC1 C1(COC)(NC(=O)Cc2nnc(C)o2)CCN(C(=O)CC2CCN(C)C2)C1 N1(CCC(=O)NCC(C2N(C(C=CC=CC)=O)CCC2)(C)C)CCN(C)CC1 c1(OC)ncc(Cl)c(=NC2CCC(N(C)C(C3CCCC(C)CC3)=O)CC2)[nH]1 N1(C(COCc2cc(C)on2)=O)CCCC(N(C(=O)C(C)C(C)C)CCF)C1 CCC(CC)(CC)C(=O)NCC(C(=O)NC(c1csnn1)C)N(C)C C1(CCCC)CCCN1C(=O)CCC1CC(NC(=O)CC2CC2(C)C)C1 Cc1cccc(CNC(=O)C(Cc2cn[nH]c2)NC(c2c(C)nsc2C)=O)c1 CCC(F)(F)CC(=O)N(CCNC(=O)Cn1ccc(=O)cc1C)CCOC c1(C)c(F)cccc1F.c1(NC(C2(C)C(C)(C)C2)=O)cccnc1C(=O)OC CC(C)CC(C)CC(=O)NCC1(F)CCN(C(C2(C)CCNC2=O)=O)C1 O=C1CCCC2C(CCCN2C(C2(C3CCCCO3)CCOCC2)=O)N1 C1(C(=O)NCCC(C)NC(c2c[nH]c(C#N)c2)=O)CCCC1P(C)(C)=O C1(NC(c2csc(C3CC3)n2)=O)C2CN(C(c3cncnc3C3CC3)=O)CC12 c12cc(ncn1)C(=O)N2CCN1CCC(O)CC1.C1(F)(NC(C)=O)CCNCC1 Cc1ncc2n1CCN(C(=O)CC=CCNC(C1CC(=O)CCO1)=O)C2 C1(C(N2CCCC(NC(=O)CCc3ncc[nH]3)CC2)=O)CCc2nc(O)[nH]c2C1 CCCC(F)C(=O)N1CCCC1CNC(C1(OCC)CCCCC1)=O N1(C(C(C=C)(C)CC)=O)CCC2C(C1)NC(=O)CN2C(=O)C1=CCCOC1 N1(C(C(CC)COC)=O)CCC(CNC(=O)CCCC2CCC2)C(F)(F)C1 CC(C)(CCCNC(C1CC12CC2)=O)C(=O)NCc1cc(O)ns1 N1(C(C(CCC)C)=O)CC(CNC(c2cccc[n+]2[O-])=O)OC2CCCC12 c1(N2CC3CCN(Cc4ccn(CC)n4)C3CC2)ncnc2ccc(OC)cc12 C1(NC(c2c(OC)nccc2)=O)CC2CCC1N2C(=O)Cc1csc(C)n1 N1(C(C(CSC)(C)C)=O)CC2CC(NC(c3cc(C4CC4)ccc3Cl)=O)C1C2 C1CCN=C2C=CN=C(N2)N1.N1(CC(=O)NCCSCCC(F)(F)F)CCOCC1 C1(CNC(C(C)SC(C)C)=O)CCC(C)(C)CN1C(C1CCN(C(C)C)CC1)=O Cc1cc(Br)cc(CNC2CCC(C(C)(C)C)C2)c1OC(F)F c1(C2(N(C(N3CCC(CC(O)CO)CC3)=O)C3CC3)C(CC)C2)cccc(F)c1 N1(C(C(C2CC2)OCC)=O)CCC2(C1)CN(C(=O)C#CC1(C)COC1)CCO2 C1(C(N(C(C(=O)N(CCF)CC)C)CC)=O)CC(C)CC(=O)N1 Cc1nc2ccccc2c(C)c1C(N1CC(NC(=O)CC2CCC2)CC1C)=O c1(C(=O)NCC(CC(C)C)(C)NC(=O)COCCCF)occ2c1CCOC2 CC1CC(C(=O)NCC2=CCN(C(=O)COCC3CCOCC3)CC2)CC(C)C1 C1(O)(C(=O)NCC2C(CNC(c3c[nH]c(=N)s3)=O)C2)CCSCC1 C1(C(N2CC(NC(C3(C)CN(C)C(=O)C3)=O)C2)=O)CCC(C2CCCO2)O1 c1(CC)conc1CC(=O)NC(c1nocc1C(=O)NC(c1cscn1)C)C c1(C(=O)OC)cc(=NC(=O)C2(F)CCN(C(c3cc(Cl)c(Cl)nc3Cl)=O)C2)[nH][nH]1 N1(C(c2cc(CC)[nH]n2)=O)CCN(C(c2c(C)cccc2F)=O)CC1C#N CN1CCC(O)(CNC(=O)CC2(F)CCN(C(=O)C(C)(C)N(C)C)C2)C1 CC(C)(C)C(CO)C(=O)NC1CCCC1NC(c1c(Br)cnn1C1CC1)=O c1(C(N2CC3C(NC(C4CC(O)(CC#C)C4)=O)C(C3)C2)=O)cc2c[nH]cnc-2n1 C1(CC)CCN(C(=O)OC(C)(C)C)C1C.C12(CSC1)NC2 CC12CC(CCNc3nccc(N4CCC(SC(F)F)C4)n3)(CO1)C2 c1(OC)cc(C(=O)NCC2CCCC2NC(c2cc(C)ns2)=O)sn1 C1(NC(CC2N(C(C)=O)CCC2)=O)CC(F)CN(C(c2cnn[nH]2)=O)C1 C1(C(=O)NC(CC#C)C(=O)NCC2CCCC2N(C)C)CC2C=CC1CC2 CCCC(CCC)C(=O)NCCC(C)N(C(=O)CN(C)Cc1ccc(C)cc1)C C=C1CCC(C(=O)NC(C(=O)NCc2cccc(Cl)c2)C2CC2)CC1 c1(C(N2CC(C(N)=O)(CNC(CCC3CCC(C)O3)=O)C2)=O)ncncc1N C(=O)(CCC1=NNC(=O)CC1)N1CC(CN(C(C(CC)CC(F)F)=O)C)OCC1 C(=O)(C(O)(C(F)(F)F)C1CC1)N1CCC(CCNC(C=CCCC)=O)CC1 CCC(CC)CCCN(C)C(C1(NC(=O)COCCN(C)C)CSC1)=O N1(C(=O)OC(C)(C)C)CCCC1C=CC(N1CCOCC1C(C)(C)C)=O c1(OC)cc(C(N2CC3CN(C(=O)CCS(C)(=O)=O)CC23)=O)ccc1O C1(C(=O)NC(CC)CNC(=O)Cc2cnn(C(C)C)c2)CN2CCCCC2CO1 c1(C(=O)NC2C(CNC(c3c(C)n(C)nc3)=O)C2)cc2c(C)c(Cl)ccc2[nH]1 c1(C(C)NCC2CCN(c3ccc(OC)cc3)CC2)ccc(F)cc1Br C1(C(=O)NC(C(C)NC(c2ccccc2)=O)(C)C)CCCOC1C c1(C(N2C(CNC(C3CC(=C)C3)=O)(CO)CCC2)=O)ccc(OC)c(Cl)c1F c1(CC)nc(=N)[nH]cc1C(=O)NCC=CCNC(=O)CCC1CC1(Cl)Cl C(C)(CCNC(=O)Cc1cnoc1)NC(C1C(=C)C1)=O c1(C(C(N2C(CNC(c3cnc(CC)[nH]3)=O)CCC2)=O)OC)ccc(Br)cc1 Cc1cnc(C(=O)NCCC(C)NC(=O)C(C)OCCN(C)C)cc1Cl Cc1ccc(C(CN2CCCCC2)Nc2ccc(-n3cnnn3)cc2)cc1 Cc1cc(CCC(N2CC(NC(c3cnc(N(C)C)o3)=O)C(F)C2)=O)ccn1 O(S(=O)(=O)c1ccccc1S(=O)(=O)N1CCCC1)C1CN(C(C)COC(F)F)C1 c1(OC)cc(CN=c2[nH]cc(CCNC(=O)CCN(C)C)s2)cc(O)c1O C1(C(N(CC)Cc2cccnc2O)=O)CCc2nc(C)nc(C(F)(F)F)c2C1 N1(C(CC2C(C)(C)C2)=O)CCC(CO)(CNC(c2csc([N+](=O)[O-])c2)=O)CC1 c1(NC(C2CC(CC(=O)NCC3(OCCO)CCC3)C2)=O)ccc(Br)nc1 C(=O)(C(C)(C)C1CCCCC1)N(CCNC(=O)CC1CCCO1)CC c1(C(N(CCOC)CCNC(=O)C2=NOC(C)C2)=O)cc2c(s1)CCCCC2 c1(C(=O)NC(CCNC(c2nc(OCC)sn2)=O)C(C)C)ccc(S(N)(=O)=O)o1 CC1(C)CN(Cc2nn[nH]c2Cl)CC1NC(C1CCN(c2nncs2)CC1)=O C1(NC(CN(CCC#C)C)=O)CC2(CCCN(C(=O)CCCc3ncco3)C2)C1 c1(C(=O)NC2CC(C)(NC(C(CCCCC)O)=O)C2)cccc2nc(C)[nH]c12 c1(OC)ccc(C(=O)CNC(c2ccc(Cl)cc2Br)=O)cc1F C=CCCCCC(=O)N1C2CCC1C(CNC(=O)CS(=O)(=O)N1CCCCC1)C2 c1(C(=O)NC(CNC(C2CS(=O)(=O)C2)=O)CO)c(C(F)(F)F)cccc1Cl CC1(C)CCCN(C(c2cccnc2N)=O)C1CNC(C1CCC2CC12)=O N(C(=NCCCN(C)C(C)C)NCc1c(F)cccc1F)C(CC)C c1(C(N2CCC(O)(CN(C(=O)C=C3CCC3)C)C2)=O)cnn2ccc(O)nc12 C1(CC)C(C(=O)N(C2CCOC2)C)CCCN1C(=O)CCCCNC(N)=O CC1(CNC(C2(CC(F)(F)F)CC2)=O)CCN(C(=O)C=CC=C(Cl)Cl)C1 CC1CN(C(=O)CNC2CC2)CC(C(=O)NC(c2cn[nH]c2)C)O1 Cc1ccc(C=CC(=O)NC2(C3CCCCN3C(C3CCC3(C)C)=O)CC2)o1 Cc1cc(O)c(F)cc1NC(C1COCCN1C(c1ccc2cc[nH]c2c1)=O)=O C(=O)(C(C#N)C(C)C)NC(C(=O)N(C1CC(OCC)C1)C)CCF N1(C(c2c(CC)[nH]nc2Cl)=O)CCC(C)(C)C(CNC(C2CCN(C)CC2)=O)C1 c1(C(N2C(CCC(=O)N(C)CC3CC3)CCC2)=O)ccnc(Br)c1F CCC(CC)C(c1nnnn1-c1ccccc1OCCCOC)NC(CCO)C1CC1 N#Cc1cc(CNC(C2CC3(C2)CN(Cc2cc([N+](=O)[O-])cs2)C3)=O)ccc1F N1(C(COCCNC(C2C(=C)C2)=O)=O)CCC(c2ncco2)C1 Cc1cc(Br)c(NC(C2CN(Cc3ccc(O)c(F)c3F)CCC2O)=O)nc1C C(C(C)(C)C(=O)N(C1CCOC1)C)NC(C(CC)SC)=O c1(C(=O)NCC(C2CC2)NC(C=Cc2c(C)cccc2)=O)ncc(C#N)cc1Cl C(=O)(CC1OC(=O)c2ccccc21)N(CCC(C)NC(c1scnc1Cl)=O)C N1(C(c2cnsc2)=O)CCC2(CCCC2NC(=O)C(O)(C2CC2)C2CC2)CC1 CC(C)C(C)(C)C(=O)NCCCN(C(=O)C(=O)NC(C)C)CC1CC1 N1(C(C(CCC)OC)=O)CCCN(C(C2CC3CCC(C2)C3=O)=O)CC1C c1(C(=O)NCCCC(CCC)NC(c2ccco2)=O)cnn2ccc(OC)cc12 CCC(C)CCCC(=O)NCCCN(C(=O)C(C(C)C)N(C)C)CC c1(C(=O)NC2CC(C)(CNC(C3N(CC)CCCC3)=O)C2)ccc(C#N)c(C)c1 c1(C(=O)OC)ccccc1NC(C12CC(C1)C(C(F)F)N2)=O c1(NC(C(CCC)N(C)C)=O)ccc2c(n1)CCC2=O C#Cc1ccc(F)cc1C(=O)NC1(C)CC(NC(=O)C(c2cccn2C)=O)C1 c1(NC(c2c[nH]n3c2nc(=O)c2ccccc32)=O)nc2ccc(Cl)c(Cl)c2s1 c12ccc(cc1)CSCC(C)(CC)NC2=O.CCC(O)C=O c1(C(=O)NC(CO)C2CCC2)ccc(F)c(O)c1 N1(C2CCCN(C(C3C(C(N)=O)C3)=O)C2)CCN(C(=O)C(O)C2CCC2)CC1=O c1(N2CCC(CC=C)(NC(=O)C(c3ccccc3Cl)C)C2)ccncc1[N+](=O)[O-] Cc1nn(-c2ccc(F)cc2)cc1C(=O)NCCNC(c1n[nH]cc1C(C)C)=O CCCC(O)C(=O)NCC(Cc1ccccc1)NC(=O)C=CC(C)(C)SC CC1(C)CC(CNC(C2NC(=O)OC2(C)C)=O)N(C(C2C(C)(C)C2(C)C)=O)C1 c1(C(N(C)CC2CCN(C(c3ncoc3C3CC3)=O)C2)=O)cnc2ccoc2c1 CC(C)CC(C(=O)NCC1CC(C)C1)ONC(c1cc(Cl)cn1C)=O N1(C(C)C)CCOC(C(=O)NC(C2CCN(C(=O)COc3ccsc3)CC2)C)C1 c1(OC)ccc(Br)c(CC(=O)NC2CCCC2NC(C2CCOC2)=O)c1 C1(C=C)(C(=O)NC(CC=C)CNC(c2nc(C)sc2C)=O)CCOCC1 c1(OC)ccc(CO)cc1C(=O)NCCC1CCN(C(=O)Cc2ccsc2C)C1 Cc1ncc(C(N2CC(CC(N3CC(CO)C(O)C3)=O)C3(CC3)C2)=O)c(=N)[nH]1 C12(C(N3C(CNC(C4N(CCC)CCC4)=O)CC3)=O)CC3CC(C1)CC(O)(C3)C2 CC1CC(C(=O)NC2(C)CC(C(=O)NCCc3cccnc3F)C2)CCS1 N1(c2c(C)cn(C(C)C)c2)CC2CN(N(C(=O)OCc3ccccc3)C)CCC12 c1(CC(N2CC(SC)C(NC(C3(CC(F)F)CC3)=O)C2)=O)ccc(O)c(F)c1 c1(C(N2CC(C3CCCCCN3C(C3CC=CC3)=O)C2)=O)cccc2[nH]ccc12 C1(NC(c2noc(CC)c2C)=O)CN(C(c2cccc(Br)c2F)=O)CC2CC12 N1(C(CCCCSC)=O)CCN(C(=O)CSC2CC2)CC1CO C1(C(N(CC#C)CC2(CF)CCC2)=O)CCN(C(C2CC2)=O)CC1 C1(N(C(=O)Cc2csc(S)n2)C)CCCN(C(c2cc(Cl)n[nH]2)=O)CC1 c1(C(=O)NC(C=CC(=O)NCC2(SC)CCC2)C)cc2ccccc2[nH]1 N1(C(=O)CCOCC(F)(F)C(F)F)CCN(C(c2cc(CCO)on2)=O)C2CC12 CCC(C(O)C(C)C)NC(C1(CC)CCN(C(=O)CCCC(C)=O)CC1)=O C=CCC(C(=O)NCC1CCCN(C(=O)C(=O)NC(C)C)C1)c1ccccc1 C1(C(=O)OC)CC(OC)CN(C(c2nc[nH]c2CNC(C)=O)=O)C1 N1(C(C(CCC#C)O)=O)CC2CC(NC(=O)CCCCCOC)CC1C2 O(C=C(C#N)C(=O)NCC1CCN(C(=O)C2=COCCO2)CC1C)CC C#CC1CCCC(N=c2[nH]nc(-c3ccc(Br)cc3)n2C2CC2C)C1 C(=O)(C(F)CC(C)(C)C)NC1CC=C(C(=O)NCC(c2ncn(C)c2)O)C1 Cc1ccn2cnc(C(=O)NC(C)CC(C)NC(c3cccc(O)c3)=O)c2c1 C(=O)(CCCCCN(C)C)NCC(CC(C)C)NC(c1cc(C(C)C)n(C)n1)=O CC(C)CCC(C(=O)NCC(F)C(C)(C)O)NC(=O)C(C)C1CC1 C1(C(=O)NC(C(=O)N(C)CC2CC(=C)C2)CCOCC)CC2(C1)CC(C)C2 c1(C(=O)NC2CC(CCNC(CC(C=C)(C)C)=O)C2)c[nH]c2cc(Cl)ccc12 C(=O)(CCS(C)(=O)=O)NCCNC(c1nc(COCC)sc1)=O C1(C(N(CC(C)N(C(c2c(OC)nsc2)=O)C)C)=O)CC(C)OC(C)C1 C1(CNC(c2cccc(NC(C)=O)n2)=O)CC2(CO1)CN(C(c1cnoc1)=O)C2 CC1CC(N(C(=O)C(=O)N(C)C)C)CCN1C(c1ccc(Br)cc1CC#N)=O Cc1cnc(C(=O)N(C2CCN(C(=O)COc3cccnc3Cl)C2)C)cn1 c1(C(N2C(CCNC(c3n(C)nnc3)=O)CCCC2)=O)ccc2c(c1)NCC2 c1(N2CCC(C)C(NC(C3CCCCN3N=O)=O)C2)ncnc(Cl)c1[N+](=O)[O-] C1(C(N2C(C(N(CCCC)CC)=O)CC(O)C2)=O)COCCC1(F)F.C=CC N1(C(c2ncc(OC)cn2)=O)CC(NC(C2CCCCO2)=O)C(C)(C)C1 N1(C(c2ccc(C)[nH]2)=O)CCCC12CCN(C(=O)C(F)(F)C1CC1)C2 C(C(C)(C)CC(=O)NC(CO)CC(C)(C)C)NC(c1cn(CC=C)nn1)=O N1(C(c2n(C)ncc2)=O)CC2(C)CN(C(c3cccnc3)=O)CC2(C)C1 C1(C(=O)NC2(C)C(NC(c3cc(C)on3)=O)CCC2)CCCC12CCC2 Cc1nn2c(C(=O)NC(C)CN(C)C(c3ccc(C)n(C)c3=O)=O)c(C)nc2s1 CCC(COC(=O)CC1(C(=O)O)CCCC1)C(=O)Nc1ccc(C)cc1 N1(C(C2(CC(=O)OC)CCNCC2)=O)CC(=O)N(C)C1C(C)C C1(C(C)NC(c2cnc(C(C)C)[nH]2)=O)CCCN(C(=O)C(=O)NCC(F)F)C1 N1(C(Cc2cc(C)n(C)n2)=O)CC2(CCC2)CC1C(=O)NC1CN(C)CC1C C1(N(C(CCCC#C)=O)C)CCN(C(=O)CCCC(C)C)CC12CC2 C1(NC(C(COC)CC(C)C)=O)CCN(C(c2n[nH]cc2Cl)=O)CCC1(F)F Cc1c(C(=O)NC(CNC(=O)C(C)(C)C2CCCO2)C2CCC2)cnn1CCO N1(C(CCCC(CC)CC)=O)CCC2(C=C(C(=O)NC(C)Cn3cnnc3)C2)C1 N1(C(c2c(CC)oc(C)c2)=O)CCOC(C(N2CCN(CC)CC2C)=O)CC1 c1(C(=O)NCCC2N(C(CC(C)C(F)F)=O)CCSC2)cccc2nn[nH]c12 N1(C(c2ccnc3cc[nH]c23)=O)CCC2CN(C(C3CC3C3CC3)=O)CC2CC1 C12CN(CC13CC3)C(=O)CCC(C)(C)NC(=O)N2.C1(C(=O)OC)(CO)CCCC1 c1(OC)cccc(CCC(=O)NC(C)CN(C(=O)COc2cccc(C)c2)C)c1 Cc1ccc(Br)c(C(N2CC(CNC(c3nnn(C)c3N)=O)C(C)(C)C2)=O)c1 S(=O)(=O)(c1ccc(N2CCC(NC3CCCCC3)CC2)nc1)N(CC(C)CO)C C(c1ccc(O)cc1)=CC(N1C(CCNC(c2c(C)scc2)=O)CCCC1)=O c1(C(=O)NC2C=CCN(C(CC(C)SC)=O)C2)ccc2ncsc2c1 c1(OC)ncc(C)c(C(=O)NCC(C)(C2CCC2)NC(=O)Cn2cccc2)c1Cl c1(C(=O)NC2CC3(C2)CC3C(=O)NCC2CC(F)(F)CO2)occ2c1CCC2 c1(C(N2CCN(C(C(C=CC)O)=O)CC(O)C2)=O)ccc2nc(C)[nH]c2c1 C1(CNC(CCC#C)=O)C(C)CCN1c1cc(CC(C)C)ncn1 CC(C#N)CCC(=O)N1CCOC(C)(CNC(c2ncc[nH]c2=O)=O)C1 CCCCC(O)C(=O)N1C(CC(N2CCC(OC)C2C)=O)C2CCCC12 CN1C(=O)CN(CC(=O)NCC2CCN2C(=O)CC2NC(=O)CNC2=O)C1=O C=CCC(CC)C(=O)N(CCC(C(C)C)NC(C1(OC)CCC1)=O)C c1(C(N(CC(C)NC(C=CC(C)(C)SC)=O)C)=O)cnn2c1CN(C)CC2 C1(N(C)Cc2ccc(C(=O)OC)[nH]2)Cc2ccccc2C1OC C1(CCNC(=O)C(F)CC2CC2)CCN(C(C2(Cl)CCC2)=O)CC1 C=CCCC(F)(F)C(=O)N1CC2CC1C2NC(C1CN(C(=O)N(C)C)C1)=O C(CC(O)C(=O)N(CCNC(C1CC12CC(O)C2)=O)Cc1ccccc1)SC C1(C)(COC)CCCN(C(C2CN(C(C3(N(C)C)CCCC3)=O)CC2CO)=O)C1 C1(N2C(=O)C2)CCS(=O)(=O)C1.c1(C2CN(C(=O)CC(C)F)C2)cn(C)nn1.CO C12(C(=O)NCCc3c(C)n[nH]c3)CCN(C(c3[nH]ccc(=O)c3C)=O)CCC1C2 O=C1Nc2ccc(Br)cc2CCC1Sc1ccc(Cl)cc1 c1(C(N2CCC(O)(c3cn(CCOC(C)=O)nn3)C2)=O)cc(F)cc2c1CCC2 C(C)(CCC(C)(C)C)NC(CSCCNC(CCCCOC)=O)=O Cc1nc(NCC2CN(C(=O)CCNC(c3ccco3)=O)C2)c(C)c(O)n1 c1(NC(c2c(-n3ccc(C)n3)cccc2)=O)nc(C)ccc1F C1(CC2CCC(C(=O)NCC(=O)NCC3CCN(C4CC4)C3)C2)NC(=O)NC1=O C1(N(C(CSCCC)=O)C2CC2)CC(C(=O)N(CC(C)C)CCO)C1 C(CN(C)C)(C(=O)N1CCCC1c1ncc[nH]1)NC(C(C)OC(C)=O)=O c1(C(=O)NCC2CC(F)(F)CN2C(=O)C2CC2)ccc(F)c(Cl)c1F C=CC(CC)CC(=O)N1CCC(N=[N+]=[N-])(C(=O)N(C)CCNC(C)=O)C1 N1(C(CCCC#N)=O)CCCC(CC(=O)NCC2(c3ccccc3F)CC2)CC1 c1(OC)csc(C(N2CCN(C(=O)CC3CCCC3)CC2)=O)c1OC C(=O)(C(C)CC(C)CC)NCC(CC(C)C)NC(c1ccc(OC)cc1C)=O c1(C(=O)NC2CC(F)(CNC(C3(F)C(C)(C)C3(C)C)=O)C2)ccc2cccnn12 c1(OC)cc(C#N)ccc1NC(=O)Cc1cc(F)c(C)cc1F C1(NC(c2cc3scnc3[nH]2)=O)CC2CCC1N(C(C1CCOC1)=O)C2 c1(C(N2CC(C)(NC(Cc3nc(C)sc3)=O)C2)=O)cc([N+](=O)[O-])cnc1C c1(C(=O)OCC)nc(=NCC2(OC)CCSC2)cc(CCNC(C)=O)[nH]1 Cc1oc(Cl)nc1C(=O)N(CC(N1CCCC(C)C1)=O)CC(C)C N(C1CCOc2ccccc21)CC(=O)NCCc1cccnn1 c1(C(N2CC(O)(C(C)NC(=O)CCCC(N)=O)C2)=O)ncc(C#N)cc1Cl Cc1ccc(-n2nnnc2C(CCc2ccccc2)Nc2nc(C)c(C)[nH]2)cc1 C1(NC(C(C)Sc2ccccc2)=O)CC2CC(C1)N(Cc1csnn1)C2 C(=O)(C(C)S(=O)(=O)C1CCOCC1)N(CC(C)N(C(CCCCCOC)=O)C)C C(c1ccc(OC)cc1)=CC(=O)NC(CNC(C1(COC)CCC1)=O)CO C1(NC(C(C)(C)C)=O)CC(F)CN(C(C2CC3C=CC2C3)=O)C1 c1(C(N2CCCC(CN(C(C(CC(=C)C)C)=O)C)C2)=O)cc2c(nn1)CCOC2 c1(CC(=O)N(CC(CC)NC(c2cc(Br)co2)=O)C)cnn(C(F)F)c1 N1(C(=O)NC2CCN(c3ccc(OC)cc3)C2)CC2C=C(Br)C2C1 c1(OC)ccc(NC(=O)C(C2CCCCC2)NC(c2ccco2)=O)nc1 Cc1cc(C(=O)NCC2CCCN(C(C34CCC3C4)=O)C2)nn1-c1ccccc1 C(=O)(C1CNC(=O)c2ccnn21)NC1(C)CN(C(c2c(OC)ccc(C)n2)=O)C1 c1(CC)c(C(=O)NC(CNC(=O)CCC2CC2C)CCOC)[nH]c(C)c1C(N)=O C1(CNC(NC(COC)C)=NCCC2(O)CCOCC2)COc2ccccc2C1 Cc1c(C=CC(N2CCC(CNC(c3sccc3F)=O)C2(C)C)=O)cnn1C C1(C(=O)NCCNC(C2CCN(CC)C2)=O)CCC(Cc2n[nH]c(C)n2)CC1 C12(NC(C(C)SC(C)C)=O)CCC(C1)N(C(c1cc(CN(C)C)on1)=O)C2 c1(C(=O)NC2CC(CNC(C3CC3C3CC3)=O)C2)cc2sccc2s1 CC1=NOC(C)(C(=O)NCC2(C(N)=O)CN(C(C3(C(F)F)CCCO3)=O)C2)C1 C1(F)(CNC(C2CC2Cl)=O)CCCN(C(c2cnn3c2OCC3)=O)CC1 Cc1cccc(C(F)C(N2CCSCC2CCNC(=O)C=CBr)=O)c1 Cc1[nH]nc(C(C)C)c1C(N1CCC(N(C)C(C2CCC(C(N)=O)O2)=O)C1)=O OCCC(N=c1ccnc(NC2CCNC(=O)CC2)[nH]1)C1CC1 Nc1ccc(Br)cc1C(=O)NCC1CCCC(NC(=O)Cc2cccnc2)C1 c1(C(N(C)CCOCCC(=O)Nc2cnn(CCF)c2)=O)ncccc1O N1(C(CC(COC)C)=O)CCOCC(NC(c2ccc(OC(C)C)cc2)=O)C1 N1(C(C(CCC2CC2)NC(=O)C(F)CC2CCOC2)=O)CC(F)(F)C(F)(F)C1 C1(NC(CCN(C)CCO)=O)CN(C(=O)C2=CCCCO2)CCC12CCC2 N(C(=NCCC)NCCc1ccc(C(C)SCC#C)cc1)Cc1ccc(Cl)cc1 CC1(CNC(=O)CSC2CC2)CCCN1C(=O)CN1CCCOC1=O C1(NC(=O)CCCN2CCCC2)CC2(CCCCN2C(c2ccc(Cl)nc2)=O)C1 CCC(O)C(C)C(=O)N1CCC(C)(CNC(C23CC2C3)=O)CC1 CC(C)C(C(=O)NCC1CCCCC1NC(=O)Cn1nccn1)C(C)C CC(C)C(C)(O)C(=O)NCc1nc(C(=O)NCC(C)(C)n2ccnc2)co1 Cc1cc(COC(=O)C(C2(O)CCOCC2)(C)C)ccc1C#N C(=O)(CS(=O)(=O)CC(C)C)NCC(CC=C)NC(C1(CCOC)CC1)=O N1(C(C=CCOCCOC)=O)CC(F)CC1C(=O)NCC(C)(C)CCC C12(CC)CN(C(c3c(C)ccn3C)=O)C(CNC(=O)C#CC(C)C)(C1)C2 c1(CSCC(=O)NCC(CNC(C2(CC)CCCC2)=O)O)cccc(C)c1 CN1C(=O)CCC1C(=O)NCC(O)CNC(=O)Cc1cccc(C(F)F)c1 Cc1ccc(O)cc1NC(C1(CNC(=O)C=CC(F)(F)F)CCCC1)=O c1(C(N2CCC(C3CCN(c4nnc(C)s4)C3)CC2)=O)ccc2cncn2c1C Cc1ccc(C)n1CCC(=O)NCCC1CCN(C(C2CCCCCC2)=O)CC1 C(=O)(C(F)(F)CCc1ccccc1)N(CCC)CCNC(c1scc(C)c1C)=O C(=O)(C1=NOC(C)C1C)NC(C(=O)N(C(CC)CC)CC(C)C)CCOCCO C12(CCCCC1)c1nc(sc1)N1CCC(C1)O2.C(CCC(=O)NC)SC.C(F)(F)F C1(C(N2C3C(NC(c4cc(C5(C)CC5)n[nH]4)=O)C(C3)C2)=O)CC2(C1)CC1(CC1)C2 c1(C2(C(N(CCNC(CSCCC)=O)C3CC3)=O)CCC2)ccc(Cl)cc1 CCC(C)C(O)C(C)C(=O)N1CCOC(C)C1C(=O)NCc1nc(C)ccc1O N1(C(C(C2CC2)OC)=O)CC=CC1CNC(=O)C(C)(C)c1ccn(C)n1 C(C(=O)NC1CCCCC1)(C1=CCCCCC1)N1CC(C)OC2(C1)CCC2 c1(CC(C)N(C(C)(C)C)C(C2C(O)C(O)CN2C(C)=O)=O)cc(Br)ccc1F C1(C(=O)NCC2CN(C(C3CC3(Cl)Cl)=O)C2)CC2CC1CO2 CN1CC(C(=O)NCC(C2CCC2)NC(c2cc(O)cc(O)n2)=O)CCC1=O CCCCCC(O)C(=O)NC(C)(C)C(=O)NC1CCN(CC)C1 CCC(CC)(C(=O)N1CC2CCC(C(=O)NC3CCSC3)(C2)C1)C(C)C C(=O)(C1=CCCOC1)NC1C(CNC(Cc2ccc(OC)nc2)=O)CC1 C1(C(N(CC(CNC(CC(CC)SC)=O)(C)C)C)=O)CCC(F)(F)CO1 N1(C(=O)OC(C)(C)C)CCC(CC(=O)Nc2ccc(F)c(F)c2)C(F)(F)CC1 c1(C(=O)NC(C#C)(CO)CO)n[nH]c2c1CN(C(=O)CN(CC)CC)C2 CC(C)C(C)(O)C(=O)NC1CCN(C(C2CCCN2C2CCOCC2)=O)CC1 CCCCC(F)C(=O)N1CCN(C(=O)CC(C)(F)F)CC1CC CCC(CC(=O)N1CC2(CCN(C(C3C(F)(F)C34CCC4)=O)C2)C1)C(C)C C1(O)(C(C(=O)NCCOCCNC(=O)C)F)CCCC1.n1(C)cc(C2CC2)cn1 C(=O)(C1CCc2c(Cl)cccc21)NC1CN(C(C(C)NS(C)(=O)=O)=O)C(C)C1 N1(C(c2cnn(-c3cccc(Cl)c3)c2)C(=O)NCC(=C)C)CCS(=O)C(C)C1C C12(C(N3CC(=C)C3)=O)CC(CN(C(C3CCCSC3C)=O)C1)C2 N1(C(C23CC(C)C2C3)=O)C2CCC1CN(C(=O)Cc1sccc1Cl)CC2 C(=O)(C(C)(C)CN(C)C)N1CCC(NC(c2cc(OCCOC)no2)=O)C1 C(=O)(C(CC)CCCC)N1CCC(CNC(CC=CC)=O)(CO)CC1 N#Cc1ccc2c(c1)CCCC2Nc1cc(C(F)(F)F)ncc1Cl C(=O)(C(C)S(N)(=O)=O)NCC1N(C(CN(C(C)C)C)=O)CCCC1 CN1CCN(CC(=O)NCC2CCC(NC(=O)C=CCN3CCCCC3)C2)CC1 Cc1nc2c(N3CCCC4(NC(C5CC5(Cl)Cl)=O)CC4C3)ncnc2s1 C(=O)(CCCC(F)(F)CO)N1CC(O)(CNC(COC(CC)(C)C)=O)C1 C1(NC(C(C)Sc2ccccc2)=O)CCC(NC(c2cnn(C)c2)=O)CC1 c1(OC)csc(C(=O)N(CCCCNC(c2cc(-c3ccco3)c[nH]2)=O)C)c1 c1(OC)cc(Cl)c(C(N2CCC(C(C)NC(c3csnn3)=O)CC2)=O)cn1 CC(C)C#CC(=O)NC1(C)CCN(C(=O)C(c2ccc(Cl)cc2)(F)F)C1 S(=O)(=O)(c1c(Cl)cccc1Cl)N1CC(NC(c2ccc(F)c3occc23)=O)C1 c1(OC)cccc(COC(C)C(=O)N(CC(C)NC(c2cnccc2Cl)=O)C)c1 c1(C(CC)C)ccc(C(=O)NC2CN(C(C3CC3C)=O)CC2F)cc1 C1(C(=O)NC2CCC(N(C(=O)CSC3CC3)C)CC2)OCC2COCCC12 C#CCC(CC(=O)NC1CCOC(C)(C)C1)NC(c1cnn(C=C)c1N)=O N1(C(C2CN(CCC)C(=O)C2)=O)CCCC(C)(CNC(c2cnc(C)[nH]2)=O)C1 C1(C(N(C2CCN(C(c3c(C)cc(Br)o3)=O)C2)C)=O)CC2C=CC1C21CC1 c1(C(N2CC(NC(C(n3cnc(C#N)n3)C)=O)C2)=O)ccc(F)c(C(C)(C)F)c1 N1(CC(C2CCCNC2)(C)C)CCC(O)(Cc2ccccc2)CC1 C(=O)(C(CC(C)C)N(C)C(c1cc(C(N)=O)co1)=O)NCC(C#C)C(C)C Cc1ccn(CC(=O)NCCC2CCN(C(c3cnn(C4CC4)c3)=O)C2)c(=O)c1 N1(c2n(C(C)CC3CCC3)c(-c3ccsc3)nn2)CCC2(CC(=O)NC2=O)C1 C(=O)(CCCC(C)=O)NC1CCC(CCNC(C=CSC)=O)C1 Cc1nc(C=Cc2cccs2)nc2c1[nH]c(=NC1(CCC(N)=O)c3ccsc31)n2C N1(C(COC(C)C)=O)CCCC(C)(CC(=O)NC(C)Cn2ccnc2)C1 C1(NC(C2(COC)CCOCC2)=O)COCCN(C(C2(C)CCOC(C)C2)=O)C1 N#Cc1ccc(=NCC(=O)NC(CNC(=O)CCC(F)(F)F)CO)[nH]c1 C=CCCCCCCNC(=O)C(Cc1cnc[nH]1)NC(C1CCCC(CF)C1)=O C12(CCC1)C(=O)NCC(=O)N2.c1(C(=O)NC(CNCCCC)C2CC2)ccco1 c1(N2C(C)CC(CNC(C3(CCOCC)CCC3)=O)C2)ncnc(Cl)c1[N+](=O)[O-] C(C1(C)CCOCC1)=CC(=O)NCC(CC)N(C)C(c1ccnc(O)c1)=O N1(C(CNC(C(CC)C)=O)=O)CC(C)(C)CC1CNC(c1cn(C)nc1SC)=O c1(C(N2CCCC(C)(C(C3CC3)Nc3cc(Cl)ncn3)C2)=O)ccnc2[nH]cnc12 Cc1ccc(C(=O)NC2CC3CN(C(C4COCCO4)=O)CC3C2)c(F)c1F CC1CN(C(=O)CC2CCCC2O)CC1CC(=O)N(C)Cc1cn[nH]c1 c1(NC(C2CCN(C(=O)C=CC3CCOC3)C2)=O)cnccc1CO C1(C2CN(C(c3cccc(C)c3N)=O)C2)(NC(C2CC(CC)C2)=O)CC1 C(CCCCC(=O)N1CC2CC(NC(c3cnn(C4CC4)c3Cl)=O)C1C2)OC CC1=C(C)CC(C(N2CCC(CO)(NC(C3CS(=O)(=O)C3)=O)C2)=O)CC1 C1(CC)CC(C(=O)OCCOc2cccc(N3CCOCC3)c2)CCN1 C1(OC)CCCN(C(=O)C(=O)Nc2cccc(Cc3nc(C)cs3)c2)C1C C(=O)(C1=C(Cl)CCC(C)C1)NCC1N(C(C=C(CC)C)=O)CC(C)(C)CC1 C1(C(=O)OCc2cn(C)nc2)CC2CC1(c1ccnn1C(F)F)C2 c1(C(N2CCC(C)(NC(c3c(C)coc3C)=O)C2)=O)cc2c(Cl)cccc2s1 C1(NC(C2(C#N)CCCC2)=O)CN(C(c2ccnnc2)=O)CC2(CCC2)C1 C#CCC(C)(C(=O)NCC1(CC)CCOC1)NC(C)=O Cc1ccc(F)c(C(=O)NC2CCC(NCc3ccc(C)nc3Br)C2)c1 c1(OC)cc(C(N2CCCN(C(c3cc(Br)oc3C)=O)CC2)=O)cc(C)n1 N1(C(c2c[nH]c(Br)c2)=O)CCN(C(c2ccnnc2)=O)C2CCCCC2C1 C(=O)(CCCC(=O)NC(C)CCCNC(C1CCN1C1CCCC1)=O)OC Cc1cc(N2CCCC2CN(C(=O)C(C)Oc2ccccc2)C)nc(C)n1 c1(OC)nccnc1C(N1CC(O)CC1C(=O)Nc1ccno1)=O N1(CC#C)CCCC1C(N1CC(C(C)NC(=O)C(c2cscn2)N(C)C)C1)=O C1(NC(C=CC)=O)(CC)CCCN(C(=O)C(C)N(C)C)C1 C(CC(=O)N1CCC(NC(c2cc(C)n(C(C)C)c2C)=O)C1)(C(N)=O)NC(C)=O C(CC(=O)NC1CC(NC(=O)CC2C=CCC2)C1)N(C)CC N1(C(C2C(C)CN(C(c3cccc(CC#N)c3)=O)C2)=O)CCOCC(C)(C)C1 CCN=c1cc(C(=O)NC2CN(C(c3coc(C(N)=O)c3)=O)CC23CC3)cc[nH]1 c1(NCC(=O)NC2CC(NC(C(c3cccc(F)c3)C)=O)C2)ccc(C(N)=O)cn1 C1(C(N2CCCC(COc3ncccn3)C2)=O)CCC2(CC2)C1 N1(C(C2N(C(C)C)CCCC2)=O)CCOCC(F)(CNC(=O)C(C)(F)F)C1 N1(C(c2c(C)ccnc2)=O)CC(CC(=O)NCC(C)C(C)(F)F)CC1(C)C c1(CCCCC)nc(C(=O)NCCCC2CCCN2C(C2CCC(=O)O2)=O)cs1 N1(C(c2cc(Cl)ncc2Br)C(=O)NC(C(=O)OC)C)CC(C)S(=O)C(C)C1 C1(c2nnnn2-c2ccccc2)(Nc2cccc(C(C)C)c2)CCN2CCCC2C1 N1(C(CC2(C(=C)F)CCC2)=O)CCCN(C(C2CCS(=O)(=O)CC2)=O)C(C)C1 C(=O)(CC(C)P(C)(C)=O)NCCC1(O)CCN(C(c2c(NC)cnc(Cl)c2)=O)C1 CS(=O)(=O)C1CN(C(=O)C(O)C2CC2)CC1NC(c1cc(-c2ccco2)no1)=O N1(C(c2c(C)ccc(C)n2)=O)CC(NC(=O)CC2CCC2(C)C)C2(CCC2)C1 C1(NC(=O)CCC2CCCC2)CC2CC1N(C(=O)Cc1cnns1)C2 N1(C(C(CC=C)N)=O)CC=C(c2cccc(Cl)c2)CC1 Cc1ccc(CC(=O)NC(C)C(C)NC(c2ccc(C(C)C)c(F)c2)=O)cc1Cl N1(C(C=CSC)=O)C2CCCC1CC(NC(C1CCCC3(CC3)C1)=O)C2 C1(NC(C(C2CCC2)OCC)=O)(CF)CCN(C(=O)CCCc2ncco2)C1 C1(C)(C(=O)NC2CN(C(C(CCC)(C)O)=O)CC2C)Cc2ccccc2C1 Cc1cc(C(=O)NCC2(C)CCC(NC(=O)C(C)C(C)(F)F)CC2)cc(C)c1C c1(C(N2CCC(O)(CCNC(C3CCC3)=O)C2)=O)nnn2ccccc12 C1(C(=O)NCCC2(NC(=O)C3=CCCCO3)CCC2)CCn2c(O)nnc2C1 C#CC1(C(=O)NC2CC(C)CC(C)(C)C2)CCN(C(=O)CC2CCC(C)C2)CC1 c1(CCC(=O)N(C2CCN(C(c3ccco3)=O)C2)CCO)ccc2c(c1)CCO2 N1(C(CSc2cn(C)nc2)=O)CC2(NC(c3cn(C(C)(C)C)cn3)=O)CCC1C2 C1(C(=O)NCC(C)=CC(=O)NCC2COCCO2)(CO)CC(C)(C)C1 c1(C(=O)NC2(C(=O)NCC)CC2)cnn2c(C)cc(C)nc12 N1(C(C(CCO)N(C)C)=O)CCCC(CCNC(c2ccoc2)=O)CC1 CC1(C(N2CCC2C(=O)O)=O)CC12CCN(C(=O)C=Cc1cccc(F)c1)CC2 C(=O)(C(CCC(C)C)NC(=O)Cn1cc(CO)nn1)NCC1(OCC)CCCC1 c1(OC)cccc(C2(C(=O)NCC(C)(C(C)C)NC(C3CC3OC)=O)CC2)c1 c1(OC)cccc(C(=O)NCCC2CC(OC)CN2C(=O)COC(F)F)c1C c1(C(=O)NCCN(C(CC(=C=C)C)=O)C)ncc(F)c2ccccc12 c1(CN(C)C)cc(C(=O)NC2CCN(C(=O)CCc3nncs3)C2)no1 Cc1onc(C2CCCC2)c1C(=O)NC1CCCCC1NC(=O)C=CCO C1(NC(=O)NCCc2nc(CC)sc2)CCCC1(C)O C1(n2cc(CCCNC(c3cn(C)nn3)=O)nn2)CCCC1(C)O N1(C(=O)Cn2cnnn2)CCC(F)(C(=O)NCCCOC2CC2)CC1 C(=O)(C1CCc2scnc21)N1CCC(OCCNC(C(C=C)O)=O)C1 CCC(C)CC(C)C(=O)N(C(C)CNC(c1ccc([N+](=O)[O-])cc1)=O)C N1(C(COCC(C)(C)C)=O)CC(=O)NCC1C(N1CCSC2(CC2)C1)=O C1(CNC(CC2C(C)C2(F)F)=O)CN(C(=O)C(C2(O)CCCCC2)(F)F)CC1O c1(CC(=O)NC(CCN(C(C(CSC)OC)=O)C)C)c(C)nc(C)nc1O c1(C(N(C)CC2OCCN(C(C(CCOC)C)=O)C2)=O)cccc(C#CCO)c1 N1(C(c2cn(C(C)C)nc2)=O)CCC2(CNC(c3ccoc3)=O)CCCCC12 c1(C(N2CCC(C)C2C(=O)NC2CCCC2)=O)cc(=O)n(C)cn1 CCC(O)C(C)(C)C(=O)N1CC2(CC(NC(=O)CC(C)(C)CN(C)C)C2)C1 Cc1cc(C(=O)NC2CC2CNC(C2(CO)CCOCC2)=O)cnc1C(F)(F)F C1(F)(CNC(C2(C(=O)NC)CC2)=O)CCCN(C(=O)CCCCCC#N)CC1 C(=O)(C#CC1CCCC1)N1CC(C=C)(CC(=O)N(CC(F)Cl)C)C1 C1(C(=O)NC2C(CNC(C(C(=C)C)(C)C)=O)CCC2)CC2(CCOCC2)C1 c1(C(=O)OC)ccc(C(N2CCC(N)CC2C)=O)c(F)c1 C1(CC=C)(NC(=O)CC2CC3CCC2O3)CCN(NC(=O)CCC(C)(F)F)CC1 c1(C(=O)NCC2OCCCN(C(C(CC(=C)C)C)=O)C2)cc(C#N)ccc1O CC(C)(C)CC(O)CC(=O)NCC(C)(C)NC(=O)CCc1ccc([N+](=O)[O-])cc1 FCC(N=c1[nH]c(=NC2CCC(CO)CC2)[nH]c2c1COC2)c1ccc(F)cc1 Cc1cn(CC(=O)NCC2CC(O)(CNC(=O)C(Cl)=CCl)C2)c2ccccc12 S(=O)(=O)(c1ccc(NC2CC(CO)C2)c(Br)c1)N1CC(CC)OCC1C N1(C(CC(C)NC(C2CC(O)C2)=O)=O)CC2(C)CC1CCO2 c1(CCC(C)NC(=O)NC2(C(=O)O)C(C#C)C2)cc(OC)cc(OC)c1 C(=O)(C1=CCCOC1)N1C(C(=O)NCCN(CCC)C(C)C)CC(C)C1 N1(C(c2ccc(OCC)cc2)=O)CC(NC(c2coc(N(C)C)n2)=O)CC1(C)C CC(O)(CNC(c1cn(CCO)nn1)=O)CNC(c1cn(C2CC2)cn1)=O C1(C)(NC(CN2CCN(C)CC2)=O)CCN(C(C2COCC2(C)C)=O)CC1 n1(CC(=O)NCC2CN(C(C(C)=CC)=O)CC23CC3)nc2c(n1)CCCC2 CC1(C)CC(NC(c2ccnn2C(F)F)=O)CN(C(=O)COc2cccnc2)C1 c1(-c2cn(C(C)CNC(=O)CO)nn2)ccc(C(C)(C)C)cc1 C1(C(=O)Nc2ccc(C)cc2O)C2C(CN1C(c1cc(O)cc(O)c1)=O)C2(C)C c1(N)ccc([N+](=O)[O-])cc1C#N.C(C(F)(F)F)SCC.C12CC(C1)NCC(=O)N2 CC1CCCC1(C(N1CCC1(C)C)=O)NC(c1ccsc1C#N)=O C(C(C)(C(C)C)NC(=O)CNC(c1ccncc1)=O)NC(c1c(C)nns1)=O c1(SCC(=O)NCCC2(CNC(C(F)OC)=O)CC2)nnc(S)s1 CCC(CC)CCCC(=O)NC12CC(C(=O)NC(C)C(C)(C)CN(C)C)(C1)C2 c1(C(=O)NCC(CNC(C2CC2CC(C)C)=O)OC)ccc2nc(C)n(C)c2c1 c1(CC(=O)N(CCOC)Cc2cc(C)ccc2O)cc(OC)cc(Br)c1 N1(C(CC(CC)C(C)C)=O)CCCCC2(CCN(C(C3(C#N)CC3(C)C)=O)C2)C1 CC1(C)CCN(C(C2(C)CC3CC3C2)=O)CC1NC(C1CCC(F)CC1)=O c1(C(N2CCN(C(C(CCC)C)=O)C(CC)C2)=O)cc(O)c(O)c(O)c1 Cc1ccc(CC(=O)NC(C2CCCN(C(c3cnsc3)=O)C2)C)cc1 c1(C(=O)NC2CC(F)(CNC(C(C)(C)CO)=O)C2)cc2cccc(Cl)c2s1 C=C(Cl)CCC(=O)NC(CNC(c1cc(Cl)cnn1)=O)CC(C)C c1(C(=O)NC2CCN(C(C3(C)COCCO3)=O)CC2O)ccc([N+](=O)[O-])cc1Cl C1(NC(CCN(CCC)C)=O)CN(C(C2CCC(N=[N+]=[N-])C2)=O)CC2(CC2)C1 C1(C)(CC)CCC(C(N2CC(C(=O)NC3COCC3N(C)C)C2)=O)O1 c1(C(N2C(C)(CNC(C(CSC)C)=O)CCC2)=O)ccc2c(c1)CCN(C)C2 C1(C(=O)NCC2C3CN(C(c4sccc4F)=O)CC23)CCOCC12CCC2 N1(C(CC(C=C)C)=O)CCCC(N(C)C(c2ccc(CCO)cc2)=O)CC1 c1(NC(CC(=O)NC2(COC)CN(C(C=CCC)=O)C2)=O)ccc(C)c(C)c1 N1(C(C=Cc2nnc(C(C)C)o2)=O)CC2CCN(C(C3OCCC3C)=O)C2C1 C(CCN=c1[nH]c(=NC(C)C(C)C)[nH]c2cccc(F)c12)c1c(C)n[nH]c1 C(C1CCCCC1)=CC(=O)N(C)CC1(CNC(=O)Cc2coc(C(F)F)n2)CC1 N1(C(C(CC(C)C)C)=O)CC23CCCC2(C1)CN(C(c1occc1C1CC1)=O)C3 C1(NC(C2CCC(=O)NC2)=O)CN(C(=O)CN2CCNC2=O)C2CCCC12 N1(C(C(C)O)=O)CC2CCN(C(c3csc(C(C)N(C)C)n3)=O)CC12 c1(C(N2CCC(NC(C3(CCC)CC3)=O)C(C)C2)=O)n[nH]c2c1CCSC2 C(=O)(C=CS(=O)(=O)CC)NC(CC)CNC(=O)CC1CCCCN1C N1(C(c2ccc(C(C)NC(C3(CO)CCCO3)=O)o2)=O)CCOC(CC(N)=O)C1 Cn1cc(CC(=O)NCC2CCCC2NC(=O)Cn2cncn2)cn1 N1(C(CCCNC(=O)C2CC2)=O)CC2CCN(C(=O)CC34CCCC3C4)C(C2)C1 CC1ON=C(C(=O)N2CC(CNC(c3c(F)ccc(O)c3F)=O)C(O)C2)C1C CCCC(CCC)C(=O)NCC1(O)CCCN(C(C2CNC(=O)O2)=O)CC1 N1(C(Cc2c(C)con2)=O)CCC2CCN(C(=O)C3=CCSC3)C2C1 c1(CCc2ccc(C)o2)nc(-c2ccc(Cl)cn2)nn1-c1nc(Br)nn1C N1(C(c2cc(C(=O)OC)on2)=O)CC2CC(NC(C3CCOC(C)C3)=O)CC1C2 Cc1ccc(Cl)c(C(N2CCC(C(C)(C)CNC(C3COC(C)C3)=O)CC2)=O)c1 N1(C(c2n(CCC)ccc2)=O)CC(N(C)C(C2CCCCCS2=O)=O)C2(CC2)C1 Cc1cccc2c1CN(C(=O)Cc1ccccc1NCc1c(F)cccc1Br)C2 c1(CNC2CC(NC(=O)CN3CCc4ccccc43)C2)n[nH]c2ccc(F)cc12 c1(C(=O)NCC2N(C(CC=C(C)C)=O)CCCC2C)cc2ncccc2[nH]1 N1(C(C2(C(=O)NC)CCC2)=O)CCOCCC1C(=O)NC1CCC=CCC1 N1(C(CSC)=O)CCCC(C2(NC(C3CC34CCC4)=O)CC2)C1 c1(OC)cccc(C(N2CCN(C(c3ccc(C)c(F)c3)=O)CC2CO)=O)c1N Cc1ccc(F)c(C(=O)NCC#CCNC(=O)CC2=CCCC2)c1O c1(C(N2CC(C#N)C(NC(C3CCCO3)=O)C2)=O)cccc2nc[nH]c12 c1(C(N2CCC(NC(=O)CC3CCCC(O)C3)(CO)C2)=O)ccn2nccc2c1 c12c(C)nc(nc1O)SC(=O)CC2.c1(CC(CCSC)CO)ccc(F)c(F)c1 C1(NC(c2cnn(C)c2Cl)=O)CC2CCC1(N=c1[nH]nc(-c3ccccc3)o1)C2 C1(CC(=O)N(C)Cc2cccs2)CCN(C(C2CCC(=O)O2)=O)C1(C)C C1(NC(C(CCC)C)=O)CC(O)CN(C(=O)CCc2cccnc2F)C1 C1(NC(c2cn(CC)nc2C)=O)CCN(C(=O)Cc2cccc(F)c2F)CC1F C(C)(N=c1[nH]c2cc(C)cnc2s1)c1cc(OC)cc(OC)c1.N1(CC)CCNCC1 C1(CCCCNC(CSCC=C)=O)CCN(C(=O)C(C)(C)C#N)CC1 C(=O)(C(O)C(C)(C)CC)N1C(C(=O)NC2(C=C)CCCC2)(C(C)C)CCC1 C1(C(N(C)CC2CCN(C(c3n(C(C)C)ccc3)=O)C2)=O)CCS(=O)(=O)C1(C)C CC1C(NC(=O)Cn2nccn2)CC2CCC1N2C(=O)CN1CC(=O)N(C)C1=O CC1(C)CCCC(C(=O)NC2CC(C)(NC(=O)CNS(=O)(=O)C3CC3)C2)O1 C1(CCCNC(C2CC(=C)C2)=O)CCN(C(c2sc(C)cc2Cl)=O)CC1 c1(NC(C2CCN(C(=O)NC(c3ccccc3)C)CC2)=O)cc2ncsc2[nH]1 N1(C(C(=O)NCC)=O)CCN(C(c2ccn(CCO)c(=O)c2)=O)CC1COC CCC1(CNC(=NCC(C)CC)NCc2nnc(C)s2)OCCc2ccccc21 Cc1ccc(NC2(NCCN(C)C(=O)OC(C)(C)C)CCCCC2)c(I)c1F C1(CC(=O)NC(C(C)C)CCN(C(=O)CO)C(C2CCOC2)=O)CCC(C)(C)CO1 Cc1cc(=NCC2CCOC(C)(C)C2)[nH]c(N(C)CC2CCN(C)CC2)n1 Cc1cccc2cc(C(=O)NCC3CCCCC3NC(c3ccns3)=O)[nH]c12 CCCCCCCCCCC(=O)N(C)CCN(C)C(C1(OC)CC1)=O C(C(=O)NCc1ccsc1C(=O)NC(c1nn[nH]n1)C1CC1)(C(C)C)SC N1(C(C(C(CC)O)C)=O)CCC2CN(C(c3cc4nc(C)sc4[nH]3)=O)CC2CC1 c1(C(N2CCC(OCCNC(=O)C3CC3)C2)=O)cc2ccccc2cn1 CCC(CCCC(=O)Nc1cnccc1C)NC(C1(C)CCCCC1)=O CCC(CC(F)(F)F)C(=O)N1CCCCC1CNC(c1c[nH]nc1C1CCC1)=O C(=O)(C(CNC(C1(C(C)(C)O)CCC1)=O)C(C)(C)C)NC(c1ccccc1)C c1(C2CN(C(C3(Cl)CC3)=O)C2)cn(CCCOC2CCCC2)nn1 c1(OC)ccc(F)c(CN2CC3CN(Cc4c(C)noc4C)CC3C2)c1OC N1(C(c2c(OC)ccnc2)=O)CCC(CC(=O)NCC(O)C(N)=O)C1(C)C c1(CC(N2CC(O)(CCc3cn(CCC(C)C)nn3)C2)=O)ccc(Cl)nc1 Cc1cnc(F)c(NC(=O)N(CC(C2CCOC2)O)C)c1 CCC(C)C(C(=O)NC12CC(C)(C1)C2)N(C(=O)CC1CC2C=CC1C2)C CCCCCC(CC)C(=O)N1CCC(C)(NC(c2ccc(OC)nc2F)=O)C1 N1(CC)CC2(CN(C(=O)C(C)(C)C3CCCN3C(=O)CCc3ccccc3)C2)C1 C(=O)(C(F)C(C)C)NCC1(C(N)=O)CN(C(c2n(COC)ncc2)=O)C1 C(=O)(C1CCCn2cnnc21)NC1C(C(C)C)N(C(=O)Cn2nnc(=N)[nH]2)CC1 C(CCCCCC(=O)N1CC2(COC(=O)C2)C1)SCC C(=O)(C(=O)C(C)(C)C)NCC(N1C(CN(C(C)=O)CC)CCCC1)=O C12(C(=O)NCC3CC(NC(CN(c4ccccc4)CC)=O)C3)CC=CC(C1)OC2 C1(C(=O)OC)OC(C(=O)NC2(C)CC(NC(c3cnnc(O)c3)=O)C2)CC1C C12(NC(CCC(=O)NC)=O)CN(C(=O)CCCn3cncn3)CC1CS(=O)(=O)C2 N1(C(c2c(CC)n[nH]c2)=O)CC2CC2(CNC(=O)CCc2ccc(CO)cc2)C1 C(C)(c1ccccc1C)=CC(N1C(CNC(C2CCCSC2)=O)CC(OC)C1)=O C1(NC(C2CCC(CNC(c3c(C)nns3)=O)O2)=O)CC(=O)N(C(C)C)C1 c1(CCNC(=O)Cn2cc(-c3cnn(CC4CCC4)c3)nn2)ccc(F)cc1F CCCCCCC(C)C(=O)NCC1=CCCN(C(=O)CCC(C)(C)N(C)C)C1 Cc1cnn(CCC(=O)NC2CC2NC(=O)C=C(Cl)Cl)c1 c1(NC(C2(O)CCN(C(C(C=CC)O)=O)C2)=O)cc(OC)ccc1C C1(C(N2CC(C)N(C(=O)CC3NC(=O)NC3=O)CC2)=O)CCc2nc(O)[nH]c2C1 N1(C(c2cnc(COC)s2)=O)CC2CC1CN2C(=O)C=Cc1cc(F)c[nH]1 N1(C(C2(SCC)CC2)=O)CCCOC(CCNC(=O)CC2CCCCC2(F)F)C1 C1(CC(=O)N(C2CN(C(=O)Cn3cc(Br)cn3)C2)C)C=CCCC1 N1(C(Cc2cc(COC)on2)=O)CC(NC(c2csc(O)n2)=O)C(C(F)F)C1 c1(SCC)cccc(CC(N2CCN(C(=O)C(C)C(=O)OC(C)(C)C)CC2)=O)c1 CP(C)(=O)c1ccc(C(=O)NC2CCN(C(C3OCCCO3)=O)C2)cc1 C(Cc1cn[nH]c1)(C(=O)NOCCCN(C)C)NC(CNC(CC)C)=O CC(C)(C)S(=O)CCCN=C(NCCOc1ccccc1)NCCc1ccoc1 c1(OC)c(C(=O)NC23CC(C2)N(C(=O)CC2(CO)CC2)C3)cccc1F N1(C(CC(C=C)c2ccccc2)=O)CC2(CCN(C(C3(C#N)CC(C)C3)=O)C2)C1 C(CCC(C)C)(C(=O)NCC1C(=O)NCCC1C)NC(C)=O C1(CNC(C2CC3(C(NC(C(NOC)=O)=O)C3)C2)=O)Cc2nccn2C1 C(CC(CC)C(=O)N1CC(O)(CNC(=O)COc2cn[nH]c2)C1)=CC c1(OC)cc(CC(=O)NCC(C)(C2CC2)NC(c2occc2C)=O)c(F)cc1O Cc1cc(C)c(C(N2CCCN(C(=O)C=Cc3ccc[nH]3)C(CO)C2)=O)c(S)n1 C=CCCCCC(=O)NC12CCN(C(=O)CCCCC=C)CC1C2 c1(C(C(=O)NC2CCCC2)N(CCC)CC)ccc(OC(F)F)c(C)n1 N1(C(C(CC)SC)=O)CCCC(F)(CNC(=O)C=C(Cl)Cl)C1 N1(C(CC2CC(C)C2)=O)CC2CC1(C(=O)NC1CCOC1(C)C)C2 c1(C(=O)OC)cncc(C(=O)NCC(C)CNC(C2CCC2C)=O)c1C C1(C(=O)NCC2CCN(C(Cc3nnc(C)o3)=O)CC2)CCCNS1(=O)=O C(=O)(C(C)(F)C(C)(C)F)NC(CCC(=O)NC(c1nncs1)C)C C1(CC(N2C(CNC(C(C)NC(C)=O)=O)CCC2)=O)CC(=O)NC1=O C1(N(C(COCCCC)=O)C)CCC(NC(=O)CN2CC(C)(OC)C2)CC1 Cc1nccnc1C(=O)N(C1CCCN1CC(=O)NC1CCCC1)C(C)C C12(CCNC(C3(CC)COC3)=O)CCC(C1)N(C(=O)Cc1ccc(F)c(F)c1)C2 c1(N2CCCC(CCNC(c3c(C)ocn3)=O)C2)nc(Cl)nc2c1SCC2 CC1(C)OCC2CC12C(=O)NC1COCCC1NC(c1csnc1Br)=O CC(CCC(C)(C)C)C(=O)N1C(C(=O)N(C2(C3CC3)CC2)C)CCC12CC2 C1(CNC(CCNC(N)=O)=O)CN(C(c2ncc(Cl)cc2O)=O)CC1(F)F C(=O)(C1=NN(C2CC2)C(=O)CC1)NC1C(C)CN(C(C2CCC2)=O)CC1 Cc1c(C(N2CCC(OCCNC(C3CCCN3C(C)C)=O)C2)=O)ccn1C Cc1cnc2n1CCCC2C(=O)NCC(O)CNC(c1cc(Cl)cc(F)c1F)=O CCC(CC(F)F)C(=O)N1CCC(N2CCN(C(c3ccc(N)cn3)=O)CC2)C1 C(=O)(C(C)(C)C(C)(C)O)NC1CC(CCNC(C(C)OCC)=O)C1 c1(C(=O)NC2(CNC(C3N(CC)C(=O)CC3)=O)CCC2)ccnc(Cl)c1N c1(OC(C)C(N2CCCC2C(C)(C)CNC(=O)CCF)=O)ccccc1C#N c1(SC)cccc(OCc2n[nH]c(C)n2)c1 C(C)(C)(CC(=O)OCC)NC(C=CC=CC)=O.c1(C2C(=O)N2)ccccc1 C(=O)(N=c1cc[nH]cc1C1CCCCC1)SCCNC(=O)OC(C)(C)C C=CC(C)(CC)C(=O)NC1CCC1NC(=O)Cc1ccc(Cl)cn1 c1(C(C(=O)OCC)OC(c2c[nH]nc2CC)=O)ccccc1Cl C(=O)(C1=C(Cl)CCC(C)C1)NC1COCCN(C(c2c(OC)c[nH]n2)=O)C1 c1(NC2(C(=O)OCC)CC3(CCCCC3)C2)nccc2oc(I)cc12 c1(CNC(C2(C=C)CCC2)=O)cnn(C)c1NC(C1CCN(CC)C1)=O C1(C(=O)NCC(CNC(C(C)c2ccsc2)=O)(C)F)CCCC2(CCC2)O1 c1(CC(=O)N(CCCNC(=O)Cc2cc(Cl)ccc2O)C)nc2ncccn2n1 CCC(CC)C(C)C(=O)NCC1(CN(C)C(c2ccnn2C2CC2)=O)CC1 N1(C(C(C)C(C)O)=O)CCC(C2(NC(=O)COCC3CCCO3)CC2)CC1 c1(C(=O)NCC(CNC(c2cc3sccc3[nH]2)=O)OC)cccc2c1OC(C)C2 S(=O)(=O)(c1cc(C)cnc1NCC1CCC(F)C1)N(C1(COC)CCC1)C N1(c2c(OC)c(Cl)ncn2)CCC(NC(=O)Cc2c(Cl)cnn2C)CC(C)(C)C1 C1(OC)CN(C)C(C)(C(=O)NC2CN(C(=O)CCc3cncs3)C2)C1 CCCC(C)(O)CC(=O)NC1CCN(C(=O)C(=O)NC2CC2)C1 C(=O)(C1CCCc2nnn(C)c21)N(CC(C)NC(c1onc(C)c1C)=O)C C=CCC(CC(C)C)C(=O)Nc1cccc(NC(=O)CC2CCCNC2=O)c1 Cc1cc(OCC(N2CCC(CN(C)C(c3cc(C(C)(C)C)no3)=O)C2)=O)no1 C(=O)(C(O)C(F)(F)F)N(C1CCCCC1)CCNC(C(C)NC(C)(C)C)=O N1(C(C(CC(CC)C)NC(c2ccc(C(C)C)o2)=O)=O)CCCC(C2(C)CC2)C1 N#Cc1cc(C(N2CC3(CC3C(N3CCN(C4CC4)CC3)=O)C2)=O)ccc1Br C1(C(N(CC(F)Cl)C)=O)CN(C(=O)C(C)(C)C2CCOC2)CC12CC2 C(CCC(F)(F)F)N(C(=O)CCCN(C)C(C1CCCOC1)=O)C C1(CNC(N2CCC3CC2CO3)=O)CCC2(CCOC2)O1 C1(OC)CC(NC(C2CC(=O)NC(C)C2)=O)CN(C(c2ncncc2Cl)=O)C1 c1(NC(=O)NCC2CCN(c3cccc(OC)c3)C2)cccc2c1C(=O)OC2 C1(NC(CC2N(C(CC3N(C)CCC3)=O)CCC2)=O)CCC2CCC12 CC1CCCn2ncc(C(=O)NCC3CC(NC(c4cncs4)=O)CC3O)c21 CC1Oc2cc(NC(=O)NCC(O)Cc3ccccc3)ccc2NC1=O n1(CC(C)O)cc(C(=O)NC2C=CCN(C(c3ncc[nH]3)=O)C2)ccc1=O C1(CNC(Cc2c(C)occ2)=O)CN(C(=O)Cn2cnc(=N)[nH]2)CC1C C1(CC=C)(NC(C2CC23CCCC3)=O)CCN(C(=O)CS(=O)(=O)NC)CC1 C1(C(N2CCN(C(C)=O)CC2)=O)CN(C(=O)Cc2ccc(C)s2)C2(CCC2)C1 C1(NC(C2(CC)CCN(C(=O)Cn3ncccc3=O)C2)=O)CCOC12CCCC2 c1(CC)ccc(C(=O)OC2CCCN(C(=O)NC)C2)c(F)c1 C1(C)(C(=O)NCCC2CC(NC(c3ccn(CC)n3)=O)C2)CC2CC2C1 c1(CS(N)(=O)=O)ccc(OCC(N2CCC(Nc3ccc(Br)cc3)C2)=O)cc1 C1(NC(c2cc(F)n[nH]2)=O)CC(C2CCN(C(=O)CC3CC=CC3)C2)C1 CC(C)CCCCC(=O)NCCCN(C(C1CNC(=O)N1)=O)C1CC1 C1(CNC(=O)CSc2cncs2)COCCN1C(=O)C(F)=C1CCCC1 N1(C(C(CSC)O)=O)CCCCC1CCC(N1CC(F)(F)C1C1CC1)=O CC1CCN(C(=O)Nc2nc(-c3ccc(Cl)cc3)ns2)CC1C(F)(F)F C(=O)(CC1NC(=O)c2ccccc21)N1CC(CCNC(c2c(N)nccc2)=O)C1 CCC(CC(=O)NCCCN(CCCNC(=O)C(C1CC(F)(F)C1)O)C)C1CC1 c1(CC2(CN(CCOCC)CC)CC2)[nH]c2ccc(C)cc2c1CC(=O)O c1(C(=O)NC2C(CNC(C3(C)CC(=C)C3)=O)CC2)cncnc1CC C1(C(N(C(C)CNC(c2cnc(SC)s2)=O)CC)=O)CC(C)=NO1 c1(-c2n(C(COC)C)nc(C3CSC3)n2)cc(Br)c2cccnn12 CC(C(=O)NCC1CC1C(=O)NCCN1CCC1)C(C)(C)C CC1CN(C(C2CC3(CCO2)CC3)=O)CCC1NC(c1cnc[nH]1)=O c1(CN2CCN(C(=O)Cc3ccccc3Cl)C(CCO)C2)ccc2c(c1)COC2 N1(CCN(C(CCN(CC#C)C(C2CC2Cl)=O)=O)C)CCCC1=O C1(NC(c2ccc(C)nc2)=O)C2CCC(C2)C1C(=O)Nc1ccc(N(C)C)nc1 N1(C(C2(C)CCOC2)=O)CC2(CCN(C(=O)C(N3CCCC3)C3CC3)CC2)C1 CC(C)(C)CC(C(=O)NC1(C2CCCCO2)CC1)NC(c1cccn2ccnc12)=O c1(C(C(=O)NCC(C)C)N(C2CCOC2C)CCOC)cc(F)ccc1C c1(C(N2C(C(C)NC(=O)C(=O)NCC(F)F)CCCC2)=O)nnc(O)nc1O C1(C(N(CCCO)C)=O)CC2CC2N1C(c1cc(C2CC2)on1)=O Cc1ncccc1CCC(=O)NCC1(F)CC(NC(C2CCCN2N=O)=O)C1 C(CN=c1[nH]c(N2CCc3cncnc3C2)nc2cccc(F)c12)SCCCO CC1CN(C(c2cn(CCNC(=O)Cc3ccoc3)nn2)=O)CC(C)O1 CCCCCC(C)CC(=O)N1CC2(CCC2CNC(=O)CNS(=O)(=O)C2CC2)C1 C=CCCCC(=O)N1CCCCC1CCCNC(c1cc(CC)oc1C)=O C1(C(N)=O)(NC(C2C(NC(CC(C)O)=O)COC2)=O)CCCCC1 C(=O)(C(C)C(CC)CC)N1C(C(N2C(CC=CC)CCCC2)=O)CCCCC1 C(C(C)(C)CC(=O)NCCC1CCCN(C(=O)CCC(C)(C)C)CC1)OC C1(N(C(c2c(CC)ocn2)=O)C)CCCN(C(C2(C)CC(F)(F)C2)=O)CC1 N1(C(CCC=C)=O)CC2(CC(NC(=O)COc3cnn(C)c3)CO2)C1 N1(C(c2ccc(SC)o2)=O)CC(O)CC1(C)C(=O)NCc1ccc(C(N)=O)o1 c1(CC(=O)NC2C3CN(C(C(C(C)C)SC)=O)C2C3)cc(C)cc(C)c1 c1(SCCC(=O)NCC(C)(CO)NC(C(C)N2CCC2)=O)ccc(Cl)cc1 C1(NC(C2CCCC(C)(C)C2)=O)CN(C(=O)CC2CC(=O)C2)Cc2ccnn2C1 N1(CCNC(c2n(CCC)ccn2)c2nnnn2CCSC)CCC(F)(F)CC1 c1(NC(C(C)C2CCOC2)=O)cnc(O)c(F)c1 N1(C(Cc2nc(C)[nH]n2)=O)CCC(O)(CNC(c2ccc(-c3cc[nH]n3)s2)=O)C1 c1(C(=O)NC(CCC)CC(=O)NCc2n[nH]c3c2CCC3)ccc2cnoc2c1 CON1CCC(C(=O)NC(C2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CCO2)C)CC1 N1(C(C(COC(C)C)(C)C)=O)CC2CC(NC(c3ccc(C(N)=O)nc3)=O)C1C2 N1(C(CCSCC(C)C)=O)CCC(CNC(C2(N(C)C)CCCCC2)=O)CC1C C1(CC(=O)NC2CC(CNC(C(N3CC(C)C3)C)=O)C2)CCC(=O)C1 c1(C(=O)NCC23C(CN(C(c4scc(COC)c4)=O)C2)C3)cnc(Cl)c(N)c1 c1(C(=O)NCCN(CCC)C(c2cncc(OC)n2)=O)cc(OC)nc(C)c1 C(=O)(C1=C(Cl)CCCC1)NCC(CCC)NC(c1ccn(CC)c(=O)c1)=O c1(OC)cc(C(N2CC(C)CC(C)C2)=O)c2ccccc2c1 N1(C(C2(NC(C(C)O)=O)CCC2)=O)CC2CC1CO2 N1(C(c2nccc(C)c2N)=O)CC2CCC(C1)N2C(=O)C=C1CCCCC1 C1(CC)CCC(C(=O)NCC(C)(C)NC(c2cc(C)ns2)=O)C1 C(CCCCNC(C1CC1Cc1ccccc1)=O)NC(c1cncs1)=O C(CN=c1[nH]c2c(c(=NCC3CCC=CCCC3)[nH]1)CCCC2)c1c(C)ncs1 c1(C(=O)OC)cc(N2CCC(C)(NC(c3ccc(Cl)s3)=O)C2)nc(C)n1 c1(C(=O)NC(C(=O)N(CC(C)NC(C)=O)CC)C)cc2n(n1)CCCCO2 CC1CC(C(=O)N(CC(=O)N(C)C)C)N1C(=O)COc1cn[nH]c1 c1(N2CCC(C)(NC(c3nccc(SC)n3)=O)C2)ncnc(Cl)c1C(C)C N1(C(c2n(C)cnc2)=O)CCN(C(c2ccc(C(C)(C)C)s2)=O)C2CCC12 C1(C(N(C)Cc2n(CC)cnn2)=O)C=CCCN1C(=O)CC=CC(C)(C)C N1(C(CC=C=C)=O)CCC2(CCOCC2)C(NC(=O)C(C)CCCOC)C1 c1(C(=O)OC)ccc(C(C(=O)NC2CCOC2)N(C)CC2CC(O)C2)o1 C1(F)(CNC(c2ncc(C)nc2)=O)COCCN(C(=O)CCC2CC(F)(F)C2)C1 C1(NC(C2(C(C)C)CCN(C(c3c(C)ocn3)=O)C2)=O)CCCCC1N=[N+]=[N-] N1(C(c2ccc(OCOC)cc2)=O)CCCC12CCS(=N)(=O)CC2 c1(C(=O)NC(CNC(C(C)(C)SC)=O)CO)cnc(C(F)F)nc1 Cc1nn(C)c(C)c1C(N1CCCC(CNC(=O)CN2CCC(C)(C)C2)C1)=O N1(CCCCC)CCOC2(CCN(C(=O)Cn3nc(C)c(C)c3C)CC2)C1 N1(C(C2(C)CCC(C)C2)=O)CC2CC(NC(C34CCCC(C3)OC4)=O)CC1C2 C(=O)(C1=CCC(C)(C)CC1)N1CCCC(N(C(C2OCCN(C)C2)=O)CCF)C1 C1(C(N(CCCC)CC(N)=O)=O)CC(=O)CN1C(c1cc(CC)sn1)=O C1(C(=O)NC2C(CNC(C3CCC(=C)CC3)=O)C2)CCOC2(CCOCC2)C1 c1(C(=O)NC2CN(Cc3c(F)cccc3F)CC2O)c(F)cc(F)cc1Cl Cc1nnc(O)c(C(N2CC(C3CN(C(=O)CCC4(C)CC4)CCO3)C2)=O)c1C N=c1[nH]cnc2c(C(=O)NCC3CCCCC3NC(=O)CS(N)(=O)=O)cnn12 C1(O)(C(N(C)CC2CCCN2C(C2CC3CCC2C3)=O)=O)CCCCCC1 S(=O)(=O)(c1c[nH]ccc1=NCC(CO)C1CCC1)N(CCC(O)C(C)(C)C)C C#CC1(C)CCCN(C(c2csc(C(=O)OC)c2)C(=O)Nc2ccccc2Cl)C1 CC1(C#N)CN(C(=O)C(CO)NC(c2ccc(Cl)o2)=O)C1 Nc1[nH]c(=O)c(Cl)nc1C(=O)NCC1CCCCC1NC(c1cnns1)=O c1(C(=O)NCCCOCCNC(C2(C(=O)NC)CCC2)=O)c(Cl)ccc(C)c1O N1(C(N=c2cc(C)n(CCO)[nH]2)=O)CCc2cc(F)cc(F)c2C1 n1(C(C)(C)C(=O)NCC2(NC(C3CC(C#N)C3)=O)CCOC2)cc([N+](=O)[O-])cn1 C(C)(CC(C)NC(=O)C(F)(F)C1CCCCC1)NC(C1CN(S(CC)(=O)=O)C1)=O C1(C(=O)NC)C2CCC(=O)C12.O=C1C(=O)CC(=O)N(C2CCCC2)CCN1 N1(C(CC(C=C)c2ccccc2)=O)CC2(CNC(=O)C(C)CO)CC1CO2 c1(C(=O)NC2C(NC(C3N(C)CCOC3)=O)COCC2)cccc(C(F)F)c1Cl c1(CNCC2(C(=O)Nc3ccc(Cl)c(Cl)n3)CC2)cc(F)ccc1Cl C1(NC(c2ncc(Cl)cc2Br)c2n(CC)nnn2)CCOC2(CCCC2)C1 C1(NC(CCNC(C)=O)=O)CCCN(C(=O)Cc2ccccc2C)CC1F c1(C(=O)NC(c2cnn(C)c2)C(=O)NC(CCSCC)C)ncc(F)cc1F C1(C(=O)NCC(C2CCCCC2)NC(C2(CCCC)CC2)=O)CC2CC2CC1C C(=O)(CC(C(N)=O)NC(=O)OCCC(C)C)OC c1(OC)cc(N)ccc1C(=O)N(C)CCNC(=O)C(C(C)C)N1CCN(C)CC1 N(C1CCc2c(OC)cc(F)cc21)c1nc2ccc(OC)cc2cc1 C=CC(C)CC(=O)NCCC(C)N(C)C(C1C(C(=O)OC)C1(C)C)=O C1(O)(CNC(c2n(C)c(S)nc2)=O)CCCN(C(C2CN3CCN2CC3)=O)C1 C1(O)(C(C(=O)N(C)CC2(CN(C)C)CC2)F)CN(C(c2cnsc2)=O)C1 C1CCC(=O)N2CCC(O2)O1.C1(NC(C)=O)CCC1.C1(C)CO1 N1(C(CC)=O)CCCCC1C(N1CC(CO)(NC(=O)CN2CCC2C)C1)=O C(=O)(C(C)CC(F)(F)F)NC1CN(C(C2CC(C(C)C)C2)=O)C(CO)C1 c1(C(=O)NCC(CO)NC(=O)CCc2ccc(Cl)s2)ccnnc1S CC(C)(C#N)CC(=O)N1CCC(O)(CCNC(=O)CCOc2cccnc2)C1 C1(N(C(CONC(C2(C(C)=O)CCC2)=O)=O)C)CCCC1C n1(CC)c(C(=O)NCC(C)(CO)NC(=O)CCCn2cccn2)cnc1O c1(CC(=O)N(C2CCN(C(C3(O)CCOC3)=O)CC2)C)ccc2c(c1)CCC2 C12(C(=O)OC)CCC(C(=O)NCCC3(O)CN(C(C4CCCO4)=O)C3)(C1)C2 c1(CCC(N2CCC(N(C(=O)CC3CC3)CCO)C2)=O)ccc(Br)c(F)c1 c1(C(=O)NCCC2CN(C(C3COCC(C)O3)=O)C2)ccc(F)c(Cl)c1F C(=O)(CS(=O)(=O)CCC(F)(F)F)NC1CC(C)N(C(=O)C=CS(C)=O)CC1 Cc1cc(CNC(=O)OC(C)(C)C)nc(Br)c1.C12CC(F)(C1)CNC2=O N1(C(CC2(OCC)CCC2)=O)CCC(C)CC1C(=O)Nc1cccc(C(C)C)c1 N1(C(CNc2n(C)cc(-c3ccc(C(F)F)cc3)n2)=O)Cc2ccc(F)cc2C1 c1(OC)cccc(CCC(=O)NCCC(C)(C)NC(=O)CC(C)n2ccnc2)n1 C1(NC(CCCOC(C)C)=O)CN(C(C2CCC(C)(C)O2)=O)CC2CCCC12 N1(C(c2c(OC)nsc2)=O)CC(C(=O)NCc2cncc(C#N)c2)C2(CCC2)C1 N1(CC)CCCc2cc(NC(=O)Cc3ccc(C(c4ccccc4)=O)s3)ccc21 c1(OC(C)C)ccc(F)cc1COC(N1CCCC(c2nc(C)nn2C)C1)=O C#Cc1ccccc1CC(=O)NCCOCCN(C)C(C1(C)CCNC(=O)C1)=O N1(C(C(=O)N(C)C)=O)CC(NC(=O)CCCOc2cccc(F)c2)C(C(F)F)C1 c1(C(N(CCN(CC)CC)C)=O)ccc(NCc2ccc(C)cc2F)cc1C c1(C(N(CC(CNC(C(CSC)OC)=O)O)C)=O)cc(O)nc(N(C)C)n1 Cc1c(CCC(N2CCC(C)(NC(=O)C(C)Cn3cccn3)C2)=O)cnn1C CC1CN(C(C2(C(N)=O)CCC2)=O)CC1(C)CNC(c1cc(Br)sn1)=O N1(C(CC2CC(CC)C2)=O)CC(N(C(=O)COc2cccc(C)c2)C)C(C)(C)C1 C#Cc1cc(F)c(C(=O)NC2CCN(C(=O)CN(C)C3CC3)CC2C)cc1F N(C(=NCCCCCCSC)NCc1nc(Cl)cs1)CC1C(OC)CCC1 C(=O)(CCCCCC(C)O)NC1C(CNC(c2c(CC)[nH]c(=N)s2)=O)CCC1 C1(N(C)C)CN(C(=O)Nc2cccc(-c3ccsc3)c2)CCC1C(=O)O N1(C(C2(COC)C=CCN2C(=O)Cc2ccsc2C)=O)CC=C(CO)CC1 CC(C)CC(CNC(=O)C(CC1CCCC1)NC(c1ccoc1)=O)CO C1(C(N(CC)CC2CCCCO2)=O)CCC(NC(=O)Cn2cnnn2)CC1 C(N=C(NCCN(C1CCCCC1)C)NC1CC1)C1C(C#C)C1 n1(C(C)C)cnc(C(=O)NC2(CC(=O)NC3CC3c3ccnn3C)CC2)n1 C=CCC(CC)C(=O)NCC1CC(OC)CN1C(=O)Cc1nc(C)sc1Cl c1(-c2cn(C3CCC(C(=O)Nc4n(C)nnc4)CC3)nn2)ccc(Cl)c(F)c1 CC1CC(NC(C2(C(F)(F)F)CCC2)=O)CCN1C(=O)CCC1CC1 C(=O)(C(CC(=C)Cl)NC(C1CCC(F)CC1)=O)N(CCCC=C)C O=C1OC2CC(C(N3CCCN(C(C4CC(CCO)C4)=O)CC3)=O)CC2O1 c1(OC)ccnc(F)c1C(N1CCCC(CNC(c2ccn(COC)n2)=O)C1)=O CN1CC(O)CC1(C)C(=O)NCc1cc(C(=O)NCC2=CCCC2)on1 C1(C(=O)NC(C)CC(C)NC(=O)CSC(F)F)C2CN(CC(F)(F)F)CC12 N1(C(CC2CCN(C(c3cc(C)cc(Cl)n3)=O)C2)=O)CCCC2(CCO2)C1 C1(C(=O)NC2C(CNC(c3c(C)nn(C(C)C)c3)=O)COC2)CC(C)(C)CN1C c1(C(N(CC(CNC(C(c2ccnn2C)C)=O)O)C)=O)cc2c(nn1)CCCC2 C1(C(=O)NC(CCCC=C)C2CC2)CC12CCN(C(=O)C1=CCSC1)C2 C1(C(=O)NCCCNC(C(C2CCCCC2)N(C)C)=O)C(C#N)C1(C)C c1(CNC(C(N2CCCC(C(=O)NC(CCC)C)C2)=O)=O)cnn2ncccc12 CC1CN(C)C(C)CC1NC(C1C(CNC(C2(C)C=CCCC2)=O)C1(C)C)=O Cc1ccc(Br)cc1CC(=O)NC12CC1CN(C(=O)C(C)Cc1ccco1)C2 N1(C(CC2(OCC)CC2)=O)CC(NC(c2ccn(C)c2)=O)CC(O)C1 C=CCCC(CC(C)C)C(=O)N1CC(NC(c2n[nH]c3c2CCSC3)=O)C(O)C1 c1(CC(=O)NCC(CC)NC(=O)CCc2nc(CSC)no2)cccc(C)c1C C1(C(NOCC)=O)CCOC1CN.C(=O)(CC1CCC1)CC#C c1(C(C)C)nnc2cc(N3CC(NC(c4ccc(F)nc4)=O)CC3C)ncn12 N1(C(C(CCC)OC)=O)CCN(C(C2CCCC2OC)=O)CC1C1CCCC1 C=Cc1ccc(C(=O)NCC2COCC2NC(=O)C(CCOC)OC)cc1 CC(C(=O)NCC1CCC2(CN(C(C3(C(C)(F)F)CC3)=O)C2)O1)C(F)(F)C(F)F c1(NCC2CN(C(CNC(CCC(C)C)=O)=O)C2)ncnc2sc([N+](=O)[O-])cc12 C1(C2CC2)(C(=O)NC2C(C(=O)OC)CC2)CN(C(=O)C(C)N=[N+]=[N-])C1 CCCCS(=O)(=O)NCC(=O)NC(CN(C(=O)Cc1csc(CC)n1)CC)CC c1(C(N(CC(CC)NC(=O)C(C)(C)CO)C)=O)cnc2ccc(C)cc2c1 C(c1ccccc1C)=CCN(CC(N1CCN(CC)CC1)=O)CC(C)C N#Cc1cc([N+](=O)[O-])ccc1CNC(=O)NCC1CC1c1cccs1 c1(NC(N2CC3C(C)C3C2)=O)cc2c(cc1Br)OCCO2 c1(OC(C)C)nc2ccccc2cc1C(N1CC2CC1C2NC(=O)CNC=O)=O C1(NC(C(C)OCCCC)=O)C2CN(C(c3cnoc3COC)=O)CC12 Cc1ccc2c(C(=O)NCC3CCN(C(C4(F)C(C)(C)C4(C)C)=O)C3)onc2c1 c1(N(C(COC(c2c(CC(=O)OC)occ2)=O)=O)C)ccc(Br)cn1 CC1CN(C(=O)COCCCF)CC1C(N1CCC(C(C)(C)C)CC1)=O N1(C(C(C)=C2CCC2)=O)CCC(N(C(=O)CC2CCC(C(F)(F)F)O2)CCO)C1 c1(C(=O)NCCc2cn(-c3cc(Cl)cc(Cl)c3F)nn2)[nH]cc2c1CCCC2 C(=O)(C1=CC2(CCOC2)C1)N(CCNC(c1ccc(CC(C)C)nc1)=O)C C1(NC(C2CC(NC(Cc3cccc(C)c3)=O)C2)=O)CCc2[nH]c(=N)sc2C1 c1(C(=O)NC2C(NC(c3c(CC)n(C)nc3)=O)COCC2)cccc2ncnn12 CCCCC(C)C(=O)NCC1CC(O)(CNC(c2cnc(C(C)C)nc2C)=O)C1 N1(C(CCc2cnc(C)o2)=O)CC(C(=O)NCCOCC(C)(C)O)C2(CC2)C1 c1(C(=O)NCC2C(NC(C(C)OC)=O)CC2)ccc(O)cc1C(F)F CCCC(CNC(=O)COc1ccsc1)C(=O)NCCC1(C)CCCO1 C1(NC(C2CC=C(C)CC2)C)CCCN(S(N)(=O)=O)C1 C(CC1CC1)(C(=O)NC1CCSC1)NC(=O)CCC1CC1 C1(CC(=O)O)CN(C(=O)NCCNC(=O)Cc2ccsc2)C1 N1(C(c2c(C)cc(N)cc2)=O)CCCN(C(=O)C(C)NC(=O)C(C)(C)C)CCC1 C1(C(=O)NC(C(C)C)CNC(=O)Cc2csc(Cl)n2)CC(C)(C)OC1(C)C C(CC(CNC(=O)CC)NC(=O)C(C)C1CC1)OC.C1C(=O)N1 C(CCCOC)(C(=O)N(CCO)CCOC)NC(C(C=C)CC)=O C12(C(=O)OC)CCC(CC1)N(CCC(=O)Nc1cc(Cl)ccc1Cl)C2 Cc1c(C(=O)NCCC(C)NC(c2sccc2F)=O)nn2c1CCCC2 C(CC(C(=O)NC(c1cccc(C)n1)C)NC(C1CC2(CSC2)C1)=O)OC c1(C(=O)NC(C2CCN(C(=O)CC34CCC(CC3)C4)C2)C)ccc(O)nn1 CC(C)CC(C)(CNC(C1CCC(C(C)C)CC1)=O)NC(=O)C(O)CC(N)=O N1(C(c2csc(C(F)(F)F)c2)C)C(=O)CCN(CC23CCCC2C3)C1=O C1(CC(=O)NC(CC)C(N)=O)CCCN(C(C2CCN(C)C2C)=O)CC1 N1(C(C(CC)n2cncn2)=O)CC=CC(C(=O)N(C)Cc2ncnn2C)C1 C=CCCC(=O)NC(CNC(c1csc(CCCOC2CCC2)n1)=O)CCOC C=CCCC(O)CN(C)C(C1(NC(C2(OC(C)C)CCC2)=O)CC1)=O c1(C(=O)OC)c(NC(C2CC3CC3N2Cc2cncc(Cl)c2)=O)cccc1Br Cc1ccc(CCC(=O)NC2CCC2C)o1.C12(CCCC1)C(=O)NCC2 CC1(C)CC(O)(CC(N2CCC(O)(CNC(C3(C)CC=CCC3)=O)C2)=O)CO1 C1(OC(C)C2CC2)CCCC1N.C1(C(C)C#N)CCCCC1 c1(C(c2n(CC)nnn2)NCCCCF)cccc([N+](=O)[O-])c1C c1(C(=O)NC2C(NC(c3cn(CC=C)nc3)=O)CCC2)cc[n+]([O-])cc1 C1(NC(C(CC#C)O)=O)CCCCN(C(=O)CC2CSCCO2)C1 C1(CNC(CNC(=O)NC)=O)CCN(C(=O)CC2CCCC(F)(F)C2)C1(C)C C(=O)(CC(C(F)F)NC(c1ccnnc1O)=O)N1C(CC)CC(C)C1 C1(O)(CC(=O)NC2C3CN(C(C4CCC(N(C)C)CC4)=O)CC32)COC(C)(C)C1 CC1CN(C(=O)CCCC2CCC2)CC(C)N(C(c2cc(N)cc(F)c2)=O)C1 N1(C(C(C2CCOC2)OC)=O)CC2(CCN(CC3CCCCCC3)CC2)C1 c1(C(=O)NCC(C(=O)NCC2CCC(C3CC3)O2)OC)cc(CO)oc1C C1(CC)CCN(C(=O)CC(C)(C)N(C(=O)CCOCC(F)F)C)CCO1 C(C)(C)(CC(=O)N1CCOC(C(=O)NC2CC(CSC)C2)C1)OC C(=O)(C(C)(C)C1=CCS(=O)(=O)CC1)NCC1C(NC(COC(C)=O)=O)CCCC1 C(=O)(CCC(F)(F)C(F)F)N1CC(NC(C(C(=O)OC)(C)F)=O)C1 N1(C(C(CCC)OC)=O)CC2CCC(C(=O)NCC3(O)CCCOC3)(C2)C1 C1(C(=O)NCC(CN(C)C(c2cnccc2Br)=O)O)C(F)(F)C12CC2 C#Cc1cc(NCc2nc(C(C)C)n(C)n2)ccc1Cl C1(NC(C(C)OCC)=O)CC2CC(NC(=O)CCc3ccccc3)CC12 CN1CCN(C(=O)C2=CCSC2)CC1C(=O)NCC12CCC(CC1)CC2 C(=O)(C1=NOC2(CCOC2)C1)NCC12C(CN(C(CNC=O)=O)C1)C2 C1(N(C(C(F)OC)=O)C)C2CN(C(C3(F)CCCC3)=O)CC12 CCC(C)(CC)C(=O)NCC1CC(NC(C2(C3CC3)CC2)=O)C(O)C1 CCC(CC)C(C)C(=O)N(C)CC1C2CN(C(c3ccc(C(F)(F)F)s3)=O)CC12 N1(C(c2sccc2Br)C(=O)Nc2ccc(OC)cc2)CC2CCC1C(O)C2O N1(C(CCC(C)SC)=O)CC(C)CN(C(c2c[nH]c(=N)nc2O)=O)CC1C C1(NC(CC(C)N(C(c2cnn(CC)c2C)=O)C)=O)CCC2(CCC2)C1 N1(C(CCCOCCC)=O)CCC2(CC1)CCN(C(C1CCCN1C)=O)CC2 C1(C)(CC(=O)NCCOCCN(C(=O)C(C2CC2)C2CC2)C)CCCO1 CCCCC(C)(F)C(=O)N1CCC(CNC(=O)CC2CCCCC2O)C(C)C1 CCC(C(=O)N1CCN(C(=O)C(c2csc(C)n2)=O)C(CCO)C1)C(C)(F)F N1(C(CCN(CCC)C)=O)CCC(NC(c2oc(C(C)C)nc2C)=O)C1C c1(C(N2C3C(NC(C(C4CC4)OC)=O)CC(CC3)C2)=O)nn2cccnc2c1Cl c1(N(C(CNC(=O)OC)C2CCC2)CC)ccccc1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)NC(C)C(=O)NCCc1ccccc1F C1(C)(NC(c2c(C)cco2)=O)CCCN(C(=O)CC2NC(=O)NC2=O)C1 C12(CNC(c3cccc(CC)c3)=O)CCCOC1CCN(C(=O)C(S)C(C)C)C2 N(C(=NCCF)N1CCC(SC)C1)C(c1nc(C(=O)OCC)sc1C)C Cc1cc(C(=O)NCC(C)(C2CCC2)NC(c2nocc2C)=O)c(Br)c(C)c1 c1(NC)cc(C(=O)NC(CNC(c2occc(=O)c2OC)=O)CO)cc(Cl)n1 C1(NC(CNCC2(O)C(C)(C)OCC2)=O)CCc2c[nH]nc2C1 c1(C(C(=O)NC2COC2)N(C(c2ccncc2)C)C)cc(F)nc(F)c1F c1(C(=O)NC2CCC(OC)(OC)CC2)c(C)oc(C)c1S(N)(=O)=O c1(C(=O)NCCC(C)(C)NC(Cc2c(C)ncs2)=O)[nH]cc2c1CCCC2 N1(C(c2cc(C(C)C)on2)=O)CCC2CN(C(=O)CN3CCC(O)CC3)CCC12 c1(C(C)NC(C(c2ccnn2C)N(CC(=O)OC)CCC)=O)ccccc1 Cn1ccc2cc(C(=O)NCC3CN(C(C4CC4CN(C)C)=O)C3)cnc12 c1(C(=O)NC2CC(N(C(C(C3CCOCC3)C)=O)C)C2)cccn1C C1(NC(C2C(C)C2)=O)CC2CC1N(C(C1(c3ccc(F)cc3)CCCCC1)=O)C2 c1(CC(=O)OCC(=O)N(CCC#N)CC)ccc(F)cc1C(F)F c1(NC(C2(CN(C(CC(C=C)c3ccccc3)=O)C)CC2)=O)ccc(N)c(O)c1 c1(C(=O)NC(C(C)NC(C2CCCN2C(N)=O)=O)CO)cc2n(c1)CCSC2 N1(C(C(C(CCC)NC(=O)C(C)SC(C)C)O)=O)Cc2cccc(F)c2C1 CC1(CNC(=O)Cc2ccc(CO)cc2)CCCN1C(c1ccsc1Cl)=O Cc1cc(C(=O)NCC(CNC(=O)CC(C)(C)C#N)CO)cc(C)c1F C1(C(=O)NC2(c3ccc(F)cc3)COC2)CC2CC1C1CC21 c1(C(N2CCC(NC(C3CSCCS3)=O)C(O)C2)=O)cc(F)cc2ccoc12 C1(CC(=O)NCC(=O)N(CC)Cc2cccnc2)CCC(C)C1 C1(NC(=O)NCCSC)COCCC12CN(C(=O)OC(C)(C)C)C2 N1(C(CCC=CC(C)C)=O)CCC(C(=O)NCCc2ocnc2CO)C1C CC(C)(C)CCCCC(=O)N1CC=C(CCNC(C2(n3cccn3)CC2)=O)CC1 C1(C(=O)NCCCCCN(C(c2cnc(C(C)OC)s2)=O)C)CCCC12CC2 c1(C(N2CC(C(C(=O)NCC#CCCO)OC)C2)=O)ccc(C#N)n1C c1(CC)ncncc1N1CCC(C(O)C(F)F)C1 c1(OC)cccc2sc(NC(CN(C)C)CC(C)C)nc12 C1(C(=O)OC)CCN(Cc2cc(O)nc(SC)n2)C12CCSCC2 C(=O)(C(C)S(N)(=O)=O)N(CC(C)C(=O)NC(C12CCC(CO1)C2)C)C c1(C(=O)NCCC(C)(CC)NC(C(CC)OC)=O)cnc(OC)nc1C(F)(F)F c1(OC)ccc(-c2cnc(C3CCCN3C(=O)C(O)O)[nH]2)c2cn[nH]c12 N1(C(Cc2ccc(C(=O)OC)cc2)C(=O)OC)CCCN(c2ccccc2C)CC1 Cc1[nH]nc(C(=O)NC2CCC2CNC(c2ccc(CO)c(Cl)c2)=O)c1[N+](=O)[O-] C1(CC(=O)Nc2c(OC)nn(C)c2)CC2(C1)CN(C(c1ccsc1Cl)=O)C2 CCCCCCCCC(=O)N1CCN(C(c2cnc(C3CCC3)o2)=O)CC(C)C1 c1(OC)n[nH]cc1C(=O)N(CCCNC(C1CCC1C(C)(C)C)=O)C N1(C(c2cnc(OC)s2)=O)CC2CC2(CNC(C2CCOC2)=O)C1 N1(CC(CCC(=O)OC)C(=O)OC)CCn2c(C(C)(C)O)nnc2C1 n1(CC(=O)NCCC(F)Cl)cc(CO)nn1.N12CCC(C1)C2=O CS(C)(=O)=Nc1ccccc1C(=O)NC1COCCC1NC(C12CCC(C1)C2)=O c1(CC(=O)N(CC(C)NC(c2ccnc(F)c2F)=O)C)cc(F)cc(F)c1 S(=O)(=O)(c1nc(NC2CCc3c(cnn3CC)C2)ccc1Br)N(CC(CC)C)C C1(CNC(c2c(CC)n[nH]c2)=O)CCCN(C(C2(C3CCCCO3)CC2)=O)C1 c1(C(=O)NC2C(C)(C)C(CNC(=O)CSC(F)F)C2)cc2sccc2[nH]1 c1(C(=O)NCC(CCNC(Cc2cc(C)sc2)=O)O)cc2c(Cl)cccn2n1 C(=O)(CCCCCC(C)C)NCC1N(C(Cc2ccc(OC)nc2)=O)CC1 C1(O)(CCNC(C2COCCO2)=O)CN(C(C2CC2c2ccc(Cl)s2)=O)C1 CC(C)CC(O)C(=O)NCC1CC2CC2N1C(c1cc(C(C)C)nn1C)=O N1(C(C(COC)NC(C)=O)=O)CCCCC(NC(C2CCN(OC)CC2)=O)CC1 C1(CC)CN(C(C2CN3CCC2CC3)=O)CCN1C(=O)C(c1ccc(C)s1)C C(CNC(c1cc(Cl)nnc1O)=O)(CC(F)(F)F)NC(C1(CC#C)CC1)=O C1(C(C(=O)NC)F)CCN(C(c2cnn(C(F)F)c2)=O)C1 C(=O)(C(F)(F)C(C)(C)O)N1CC(CCC)N(C(=O)CSCc2cccnc2)CC1 C1(C(=O)NC(C)C(C)(C)C#N)CCCCCN1C(=O)CCCN(C)C C1(C(=O)OC)COC(C(F)(F)F)CN1CC(O)C(C)(F)F c1(C(=O)NCC2N(C(C(n3ccc(C)n3)C)=O)CC2)cccnc1OCCO N1(CCN(C(c2ccc(CC)o2)=O)C)CCN(C(=O)C(c2cnn(C)c2)=O)CC1 C1(OC)COc2c(C(=O)NCc3ccc(C)c(C4CC4)c3)cnn2C1 N1(C(c2c(C)nc(C3CC3)o2)=O)CCCC(C2CC2NC(=O)CNS(N)(=O)=O)C1 Cc1c[nH]c(C(=O)NCCn2cc(C(=O)NCC(C)(O)C(F)F)cn2)c1C C(=O)(C1=CC(O)C(NC(=O)CC2CC(C)(C)CO2)C1)N(C(C)CO)CC C1(C(=O)NC2CCCC2CNC(c2cnc(Cl)s2)=O)(COC)CC1(F)F c1(N2CCCC(CC=C)C2)nc(=N)[nH]c(=NC(C)CCO)[nH]1 C1(CC=C)(NC(C2CCCN(C)C2)=O)CCN(c2nnc(CCC)s2)C1 Cc1nc2n(n1)CCC(C(N1CC3CC1(c1cn(C4CCCC4)nn1)CO3)=O)C2 Cc1cc(C(=O)NCC2CC3CCC2N3C(c2ccc[nH]2)=O)c2c(C)noc2n1 N1(C(c2n[nH]c(C)c2Cl)=O)CC(N=c2[nH]cnc3cnn(C)c23)CC2(CCC2)C1 C(=O)(CC(C(C)=O)N1CCC(n2ncc(N)c2C(F)F)CC1)OCC C1(C(N(CC(CC)C)C)=O)(CCOC)CCN(C(c2ncc(C)cc2C)=O)CC1 C1(NC(C(C)Cc2ccccn2)=O)CCCCC1NC(c1cnco1)=O c1(C(=O)NCCCN(C(C(CC)OCC)=O)C)cc(Cl)c2cc(Cl)ccc2n1 CCC(C)(COC)C(=O)N1CCC(C(C)C(N2CCCC2(C)C)=O)CC1 C(CC1CCCC1)(C(=O)N=c1ccn(CCO)[nH]1)NC(c1cc(CC2CC2)on1)=O C1(NC(c2c(C)nc(C)[nH]2)=O)CCCC(NC(C2(CS(N)(=O)=O)COC2)=O)CC1 C1(C(=O)NC(C(C)C)C(C)NC(=O)C=Cc2ccnn2C)CCC2(CC1)CC2 c1(CC(=O)N(CCNC(C(COCC)C)=O)CC)c(C)cccc1F CCN=c1[nH]c(C(=O)NCC2(CNC(=O)CC3C=CS(=O)(=O)C3)CCCC2)cs1 N1(C(C(CC)CC)=O)CCC2C(CCCN2C(c2c[nH]c3cc(Cl)ccc23)=O)C1 C1(=O)CCC(N)CC2(CCC2)N1.C(=O)(C(C)C)OC Cn1ncc2ncc(C(N3CCC(CO)C(NC(=O)CCC4(C)CC4)C3)=O)cc12 C(=O)(C(C)(C)CC(C)C)N(C(C(=O)NCCC(C(C)C)OC)C)C1CC1 C(c1ccc(CC(C)C)cc1)=CC(=O)NCCCCN(C(CCCCOC)=O)C C1(C(=O)NCC2CCN(C(c3cn(C(C)(C)C)nn3)=O)CC2)CCC2(CCC2)C1 CC1(C)CCCCCC1NC(c1ccc(C(F)(F)C(F)(F)F)s1)C1CC1 c1(C(C(=O)NC(C(=O)NCC(=C)CC)c2ccoc2)C)cncnc1 C1(C(=O)NCc2c(CC)nco2)CN(C(=O)CC2CN(C(C)=O)C2)CCC1(C)C CCCCC(C)CCC(=O)Nc1cnc(Cl)cc1C(N1CCC2(CCOC2)C1)=O C1(C(=O)NC(C2(O)CCN(C(c3cc(Cl)c(Cl)[nH]3)=O)C2)C)CCC2(CCC2)CO1 C(=O)(C(CCc1cn[nH]c1)NC(c1c[nH]cc1C(F)(F)F)=O)OC c1(C(=O)NCC2(OCC)CN(C(c3c(C)ncn3OC)=O)C2)cc(C)nc(O)n1 C1(CNC(c2cc(C)no2)=O)CCN(C(=O)C(C)NS(C)(=O)=O)CC1C c1(C(=O)NCC23C(CN(C(CCCCC#C)=O)C2)C3)sc2[nH]cnc(=O)c2c1C Oc1ncnc2c1CCN(N1CCCC(c3n[nH]c(=O)[nH]3)C1)CC2 N1(C(CCC(C)C)=O)CCN(C(C2CC3(C2)CC3F)=O)CC2(CC2)C1 Cc1cc(CC(=O)N(CCCNC(=O)COc2ccccc2C(C)C)C)ccn1 c1(C(N(C2CCCN(C(=O)CC3(O)CCC3)C2)CC)=O)cnn2c(C)cccc12 n1(CC(=O)OC(C)(C)C)ncc(Cl)c1C(=O)NC1CCC(NS(C)(=O)=O)CC1 C(=O)(C(CC)C(=O)NC1CCCN(C(=O)CSCc2cccs2)C1)OCC C(C(C)(C)C(=O)N1CCC(CCC(=O)N2CC(CF)C2)C1)OCC CCCC(CC)C(=O)NC1(C(=O)N(C)CC2(F)CCCC2)CC(CO)C1 C#CCC(C(=O)NCCC1CCCN(C(c2nnccc2C)=O)C1)C1CC1 C1(C(=O)NC(CC#C)C(=O)NC)C2CC3C(C2NC(C2CC(C)=NO2)=O)C13 N1(C(C(=O)NCCCC)C2CC2Cl)CCOc2c(C(=O)OC)cccc2C1 N1(C(C2N(C(C)=O)CCC2)=O)CCC(NC(c2nnccc2C)=O)C2(CCC2)C1 N1(C(CNC(CC(C)(C)C)=O)=O)CCCC2CN(C(c3sccc3F)=O)CCC12 c1(NC(C(CC)N(CSC)CC)=O)ccc(N=S(C)(C)=O)s1.C12(CCC1)C(=O)N2 c1(CNC(C(N2CCCC(C(=O)OCC)C2)=O)=O)oc2ccccc2c1Cl CCCCC(CC(=O)NC(C1(O)CCCC1)(C)C)NC(c1cc(Cl)no1)=O c1(NC(C(=O)N(C2CCOCC2)CC(=O)NCC2C(C)C2C)=O)cccnc1 C1(CC(=O)NC2CCN(C(c3c(CCC)n[nH]c3)=O)C2)(OC)CCCCC1 c1(CCN(C)C)cccc(C(=O)NCCCN(C(=O)CCC2CCCC2)C2CC2)c1 C1C(CCCC)N1C(C(F)=CC)=O.C1(C(C(=O)OCC)C2CCCC2)CCOCC1 C12(OC)CCC(C(N3CCC(CCNC(=O)CC4CC(=O)NC4=O)C3)=O)(CC1)C2 c1(NC(C2C=CC(Nc3cc(N4CCCC4)ncn3)C2)=O)cc(Cl)ccc1Br C1(C(=O)NCCn2nnnc2-c2ccccc2Br)C2Cc3ccc(Br)cc3C12 N1(C(c2cn(CCOC)nn2)=O)CCCC(CO)(NC(C2CCC2(F)F)=O)C1 C(=O)(C(O)CC(C)(C)C)NC1(CC=C)CCN(C(=O)CC(C)(C)O)C1 N1(C(=O)CC2CCC2)CC(C2CN(C(C3CC34CC(F)(F)C4)=O)C2)C1 N1(CC(=O)NC(CC)CN(C(C2CCS2(=O)=O)=O)CC)CCC(=O)NC1=O C1(C)CN(C(c2cnc(C)cn2)=O)CCO1.n1(CCCCC)cc(C)nn1 N1(C(CCCN(C(C)=O)C)=O)CCCCC1CN(C(C1CC1(C)C(F)F)=O)CC N1(C(C2(C#N)CCC2)=O)CC2COCC(C1)C2NC(=O)C=CSCc1ccco1 C(=O)(C(CCC)CC(C)C)NC(CCCC)CNC(c1cnccn1)=O c1(C(N(C2CCN(C(C(CC(C)C)F)=O)C2)C)=O)ccc2c(c1)C(=O)C(=O)N2 c1(C(=O)NCCN(C(c2cccc(O)c2)=O)CC)csc(N=S(C)(C)=O)n1 N1(C(C(C)O)=O)CCCC(CNC(=O)CCc2cnn(C)c2)CC1 C1(NC(c2c(C)ocn2)=O)CS(=O)(=O)CC1NC(=O)C=CC(c1ccccc1)=O CC1CCCN(C(=O)CC2CN(C(C3CCO3)=O)C(C)(C)C2)CC1 Cc1nc2c(o1)CCCC2CC(=O)N1CC2(NC(c3snnc3C)=O)CCC1C2 CCC(O)C(F)(F)C(=O)NC1CN(C(c2cnc(C3CCCO3)s2)=O)C1 C1(C(=O)NC(C)CC2CN(C(c3cnn(C(F)F)c3)=O)C2)OCC2COCCC12 c1(C(=O)NCCC(=C)CNC(C2CC2CC(C)C)=O)ccc2nonc2c1 c1(C(N(CC(C)CNC(=O)C(=O)NCC2CC2)C)=O)cn2c(n1)CCC2 c1(C(=O)NC2CC(C(C)NC(Cn3ncc(CC)c3)=O)C2)n[nH]cc1[N+](=O)[O-] c1(C(=O)NC(C)CNC(c2ccc(N)cc2)=O)cccn2nnnc12 C1(CNC(C2(C)CCCOC2)=O)CN(C(=O)CCOC2CC2)C2(CCC2)C1 c1(C(N(C(CNC(C2C3CC4C(C3=O)C24)=O)C2CC2)C)=O)ccc2cnnn2c1 N1(C(=O)C=CCc2ccccc2)CC2(C1)CN(C(C1(c3cccc(F)c3)CC1)=O)C2 c1(C(C(N2C3C(NC(C=CC(=O)OCC)=O)C(C3)C2)=O)C)cc(F)cc(F)c1 Cc1nn(C)cc1-c1ccc(NC(c2cc(Cl)sc2Cl)=O)cn1 Cc1cc(C)c(C(=O)NC2CC(CNC(=O)CCn3ncn(C)c3=O)C2)cc1C C1(CNC(N(c2ccn(C3CCCC3)n2)C)=O)CC12CN(C(=O)OC(C)(C)C)C2 N1(C(CCN(CCCCC)C)=O)CCC(C2(NC(=O)CCCNC(C)=O)CC2)C1 Cc1cc(C(=O)NCC2CCC2NC(c2ccnn2CCF)=O)ncc1N C1(CCCC)CN(C(C2CC2C2CC2)=O)CCN1C(=O)Cc1csc(Cl)n1 C1(C(=O)NC(C(CO)NC(c2nc(C)sc2)=O)C)CCC(C)(C)OC1 c1(C(N2CCCC2c2cc(C)nn2C)C(=O)NCCC)sc2ccccc2c1C N1(C(CN(C(=O)CN2CCC(OC)C2)CC#C)=O)CCC2(CCOC2)CC1 Cn1ncc2c1CC(C(=O)NCC(C1CCC1)NC(C1C3COCC13)=O)CC2 N1(C(CCc2c(C)n(C)nc2)=O)CCN(C(c2cncc(C(N)=O)c2)=O)C(C)C1 c1(C(=O)NC(C(C)NC(c2ccc(CC)[nH]2)=O)C)ccccc1CC#N c1(C(=O)NCC2(CCNC(Cc3cc(C)[nH]n3)=O)CC2)cc(O)cc(=O)o1 Cc1ccc(C=CC(=O)NC2CC2NC(C2CCC(OC(C)C)CC2)=O)c(C)c1 CC1(C)CC(CNC(c2scnc2Br)=O)N(C(=O)CN2CCCC2=O)C1 CCC(CNC(=O)Cc1ncn(C)c1C)(CC)C(=O)N(C1CCN(C)CC1)C N1(C(C)=O)CCN(C(c2cc3c(s2)CCC3)=O)C(CS(C)(=O)=O)C1 Cc1nc2ccccn2c1C(N1CCNC(C(F)F)C1)=O N1(C(c2cnn(C)c2F)=O)CCN(C(C2CCN(CCF)CC2)=O)C2CC12 N1(C(C(CC=C)C(C)C)=O)CC=C(C(C)(C)C(=O)N2CC3CCCC23)C1 N1(C(Cn2c(C(C)C)ncc2)=O)CCCN(C(=O)Cn2cncn2)CC1 c1(CNC(C2CCC(n3cc(CC4CCC(=O)C4)nn3)C2)=O)cc(F)ccc1Cl C(=O)(CC(C(C)C)NC(C1(CCC)CC1)=O)NC(C=C)C(F)(F)F CCC(CCC(=O)NCC1CC(NC(=O)Cc2cccc(O)c2F)C1)OC c1(C(=O)NCC2CC(F)(CNC(C3CCN(C)C3=O)=O)C2)cccc2sncc12 C1(CC(=O)NCCCn2cc(CC(C(C)(C)C)O)nn2)CC2OCCC2O1 N1(C(CCC(CC)NC(=O)CC2CCOC2C)=O)CCCC2CC1C2(C)C CCCC(O)C(=O)N(C)CC1CCN(C(C2(C)CCSCC2)=O)C1 c1(C(=O)OC)nc(=NCC2(C)CCCN(C(=O)C(O)C3CC3)C2)c2c([nH]1)CCC2 C12(CCNC(CCCNC(C)=O)=O)CCC1CN(C(c1c[nH]c(=N)nc1C)=O)C2 N1(C(CC2CCC(C)C2)=O)CCC2(CC1)C(NC(=O)CC1CN(C)C1)CS2(=O)=O Cn1c(CC(=O)NC(Cn2ccnn2)C(=O)NCc2nccs2)nnc1S c1(SC)cn(C)nc1C(=O)NC1CN(C(=O)C=Cc2cocn2)C1 C1(COC)CCN(S(=O)(=O)N2CCC(C)(C(=O)NC)CC2)C1 c1(C(=O)NCC2CC(NC(CC3C(C)OCC3)=O)C2)ccc2oncc2c1 C(=O)(CCN(C(C1CN(C2COC2)C1)=O)C1CC1)N(CCCO)CC#C c1(C(=O)NCC2C(NC(CN(CC)CC)=O)C2)c(O)ccc(Br)c1Cl C1(CNC(CCc2cc(C)[nH]n2)=O)CC(NC(=O)C=Cc2scnc2C)C1(C)C c1(OCC)ccccc1C(=O)NC(C)(C)CCCNC(=O)CC(CC)OC c1(CN(C(CCCn2cc(C(CC)O)nn2)=O)CC)ccc(F)c(Br)c1 c1(C(=O)NCC2CC3CN(C(C=CCCC)=O)CC32)ccc([N+](=O)[O-])n1C C1(CC(=O)N(C2CC(CNC(C3CC4CC4C3)=O)C2)CCO)CCC(C(F)(F)F)O1 N1(C(C2C(CC(C)(C)C)C2)=O)CCCCCC(NC(=O)CC2CCC(=O)O2)C1 C#CCC(CC#C)C(=O)NC1CN(C(C2(N3CCCC3)CCC2)=O)CC1OC C(C(COC)CC(=O)NC1CC(O)CN(C(=O)CCCc2cnccn2)C1)OC c1(C(=O)NC(CC=C)CNC(=O)C(CCC)OCC)ccnc2c1cnn2C c1(CN(CCC(C)(C)C#N)C2CC3(CNC3)C2)c(Cl)c[nH]c2nccc1-2 C(=O)(C1=C(Cl)CCOC1)NCC12N(C(CCOCCN(C)C)=O)C(CC1)CC2 N1(CC)CCC(N(C(=O)CCCn2nnc(-c3ccccc3)n2)C)C(C)C1 c1(C(N2CCN(C(CN(C(CC(C)F)=O)C)=O)CC2)=O)cc2[nH]ccc2s1 C(=O)(C(F)(F)CC1CC1)NC(C1CCN(C(=O)CC2C=NN(C)C2=O)CC1)C C#CCCCCC(=O)NC(C)CNC(C1(OC)CS(=O)(=O)C1)=O C1(CNC(CC2CCC(NC(C3(C(C)C)CC3)=O)C2)=O)CCC(C)(C)CO1 c1(C(=O)C2CC2)ccc(F)c(N2CCOCC2)c1.C12OCCC1NC(=O)NC2 C1(CNC(C=CCOC)=O)(NC(=O)C(c2ccccc2F)C)CCCCC1C CC1CN(C(C2(C)CCCN2C)=O)CC(C)N1C(C1CCCCCCC1)=O S(=O)(=O)(c1cnc(NCCc2ccccc2F)c(Cl)c1)NCC1CCCC(C)O1 N1(C(CN(C(C)C)C)=O)CCOCC(CNC(=O)CCc2ccc(Cl)c(F)c2)C1 Cc1ccc(CCC(=O)OCc2cccc(N3CCCC3=O)c2)c(C)c1 C12(C(=O)NC3CC(C)(NC(CSCC=C)=O)C3)CCC(OC)C1C2 c1(CC(=O)N(CCN(C(=O)Cc2ccco2)CC)C)cccnc1Br.C(C)(=O)O Cc1oc(C2CC2)nc1C(N1CC2C(CNC(c3ncc[nH]c3=O)=O)C2C1)=O N1(C(c2n(CC)cnn2)=O)CC(CCNC(=O)Cn2cccnc2=O)C(C)C1 CC1(C)CC(NC(=O)Cc2ccco2)CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)C1 C1(CC(=O)N(CC(O)C2CCC2)C)CCCN(C(C2(C)CCN(C)C2)=O)C1 c1(C(=O)NC(CN(C(C(CC)N(C)C)=O)CC)C)sc(C)nc1C(F)(F)F Cn1cncc1C(=O)NCc1csc(C(=O)NCCN2CCOCC2)n1 Cc1noc(C)c1-c1cn(CC2COCCN2C(C2(C)CCCCC2)=O)nn1 Cn1ncc(C(=O)NC2CN(C(C3(O)CCC3)=O)CC3(CC3)C2)c1S(C)(=O)=O c1(C(N2CCCC(NC(C(C)OCCN(C)C)=O)C2C)=O)ccn2nccc2n1 C1(NC(c2c(C)ocn2)=O)C(C)(C)C(NC(=O)C(O)CC2CCOCC2)C1(C)C c1(OCCCOC)ccc(C(=O)NC(C)CCNC(=O)CCC=C(C)C)cn1 C(C1=CCN(C(=O)CCc2nc(C)c(C)o2)CC1)NC(c1c(SC)cccc1)=O C1(NC(C(CCC)O)=O)COC2C(NC(=O)C(C(C)C)n3cccc3)COC12 C(c1ccccc1C(F)(F)F)=CC(=O)NC(CSC)C(=O)N(C)CCO C1(NC(C(CC#C)NC(c2nn(C)cc2C)=O)=O)CC(C)N(C)CC1C C(=O)(C1Cc2ccccc21)N(CCCNC(c1ccn2c1CCCC2)=O)C(C)C C#CCCCCCNC(C1(C(C)C)CCCN1C(C1CCC1C(C)(C)C)=O)=O Cc1cc(C(=O)NCC(CNC(=O)CCc2ccccn2)CO)nc(O)n1 C1(NC(C(C)OCC2CC2)=O)CN(C(c2cc(F)cc(F)c2O)=O)CC(F)(F)C1 CC1(C)CCCC(CNC(=O)NCC(N2CCCCC2)C2CCCCC2)C1 C1(NC(C(C)C2CC2)=O)Cc2ccccc2C1NC(c1cnsn1)=O C(=O)(CCC(C(=O)OC)NC(=O)CSC(C)Cn1cc(C)cn1)OCC c1(NC(C(CC)OC)=O)cccc(CNC(c2cnc(O)n2CC)=O)c1 n1(C(C)C)cnc(C(=O)NC2CC(C(F)C(=O)NC(CN3CCCC3)CO)C2)n1 c1(OC)cc(CNc2ncccc2-c2cncc(F)c2)ccc1F C1(CNC(=O)C(F)(F)c2cscc2Br)(CC2CC2)CCCCC1 C(=O)(CC1=NNC(=O)C1)NCC1CN(C(c2nc(CC)oc2)=O)C(C)CC1 C=CC1(CC(=O)NCC2CCN2C(c2cscn2)=O)CCC1 c1(C(=O)NC2C(CNC(c3ccc(C(N)=O)[nH]3)=O)CC2)[nH]cc2c1CCCC2 c1(OCC)ccc2oc(C(=O)OCCC3CC34CCOC4)cc2c1 N1(C(C(CCC)NC(N)=O)=O)CCC=C(C(=O)NCC2CC(N(C)C)C2)C1 CC(C)(C)CC(O)CC(=O)NCCCN(C(=O)CC(F)(F)F)Cc1ccccc1 C1(C(N(C(C)CNC(=O)CSC(F)(F)F)C)=O)CN2CCCCC2CO1 C1(C(=O)NC2C(C)C2C)C2CCC(C2)N1C(=O)CC(O)C1CCCC1 c1(C(N(C2CN(C(C(=Cc3cccs3)C)=O)C2)C)=O)ccc(S(=O)CC#N)cc1 C(=O)(C#CC1CCOC1)N1CCCCC(NC(COCc2onc(CC)n2)=O)C1 C1(CC(=O)NC23CC(NC(Cn4nnc(C(C)(C)C)n4)=O)(C2)C3)CC2CCC1C2 C12(NC(=O)CSCc3ccccc3)CCN(C(c3ccc([N+](=O)[O-])o3)=O)CC1C2 N1(C(c2c(OC)cccc2Cl)=O)CCC(C2CCN(C(=O)COCC(C)C)C2)C1 N(C1CCCc2cc(F)ccc21)C(c1ccc(Cl)cc1)CO CC(O)CCCC(=O)NC(C)CCNC(=O)C1=NNC(=O)C1 C(=O)(CCCCCN=[N+]=[N-])N1C(C)(C(=O)NCCC=CCCC)CC(O)C1 Cn1cc(C(C(=O)NCCC2CCSC2)NC(=O)CC2(C)CCN2C(N)=O)nn1 Cc1cc(NC2(CO)CCCN(C(=O)CC(C)C(F)(F)F)C2)ccc1[N+](=O)[O-] c1(NC(C2CCN2C(=O)CSc2ccc(Br)cn2)=O)nc2ccccc2s1 C=C(Cl)CC(C(=O)N1CC(C#N)(SC)C1)NC(=O)CC1CCCOCC1 c1(OCC)ncc(NC(C2CC(OC)CN2C(c2c[nH]c(=N)s2)=O)=O)cc1C Cn1ncc2c(N3CC4(CC4)CC3CNC(C3(C(F)F)CC3)=O)ncnc12 c1(CCC(=O)NCC2N(C(C=CCCC)=O)CCC2C)cc(OC)cc(OC)c1 c1(C(=O)NCc2cccc(NC(C3C(C)COCC3)=O)c2)ccc(F)c(N)c1 c1(CN(CCNC(C2CC2c2ccccc2)=O)CC)nc2cnccc2s1 N1(C(C(C)N(C)C)=O)CCC(N(C(=O)C=CC(C)(C)C)Cc2ccccc2Cl)CC1 N1(C(CC2N(CC)CCOC2)=O)CC(O)(C2(CNC(=O)CNC(C)=O)CC2)C1 C1(NC(C(COC)COC)=O)CN(C(=O)COc2ccccc2)C(C)(COC)C1 N1(c2nc(CCN(C)C)c3c(n2)ncn3C)CCS(=O)(=O)C2(CCCCC2)C1 O=C(C1CCOc2ccc(F)cc21)NCC1CCN1C(=O)C=CCO n1(C(CC)CC)nc(C(=O)OCC(C)(C)C)cc1C.c12ccccc1OC2 CC1CN(C(C2CCC2C)=O)CCCN1C(c1ccc(-n2ccnn2)cc1)=O O=C(CC1=CCOCC1)NCC1CN(C(=O)CCc2ccncc2)CCO1 CC1CCCn2ncc(C(=O)NC3CCCCN(C(=O)CCc4ccco4)C3)c21 N1(C(CCc2c(C)cccc2)=O)CCC2(CC(C(=O)NC(C)CCO)=NO2)C1 C(=O)(C(C)(C)CNC(C1CC1C(C)C)=O)NCc1cnc(C(C)C)[nH]1 N1(C(Cc2ncn(C)c2)=O)CCCCC1CCNC(=O)CCC1CCCOC1 C(c1cccc(F)c1F)=CC(N1CCCC(C)(NC(C2C(C)(C)COC2)=O)C1)=O Cc1ccc(CC(=O)N(c2ncccn2)C)c(Br)c1 c1(C(=O)OC)cccc(F)c1CNC1(CCCCSc2ccccc2)CCC1 N1(C(C(C)OCC=C)=O)CCC(N(C(c2cc(C(=O)OC)c(C)o2)=O)CC)CC1 C1(C(N2CCC(=C)CC2)=O)CC2OCCC2N(C(C2CCC(F)(F)C2)=O)C1 Cc1ccc(C(=O)NC(C)CCCNC(C2CC(c3ccccc3)C2)=O)c(N)c1 Cc1cc(CC(N2CC(F)CC2CNC(=O)C(C)CC2CC2)=O)cc(F)c1 C1(N(C(C(C)OCCC=C)=O)CC)CCCN(C(c2ccnn(C)c2=O)=O)CC1 N1(C(C2C(C)(NC(C(C=C)CC)=O)CCCC2)=O)CCc2nnnn2CC1 C(CC(=O)NC(C(=O)N(CC(O)COC)C)c1cccs1)OCC C(CC(F)F)(C(=O)N1CCC2(CCO2)C1)NC(C1CC(CC2CC2)C1)=O C1(C(=O)NC(CN(C(c2cnn(C3CCC3)c2)=O)CC)C)CCCN1C c1(CCC(=O)NC(C(C)C)(C)CNC(=O)C(C)CN(C)C)cc2ccccc2o1 O(NC(=O)CS(=O)CC)CC(=O)NC1CN(CC)CC1C c1(C(=O)NCc2c(C(=O)NC34C(C)OC(CC3)C4)n[nH]c2)ccn2cncc2c1 c1(C(N2CCC(C(N3CCCC3CO)=O)C(O)C2)=O)cc(O)ccc1[N+](=O)[O-] n1(CC)cnc(C(=O)NCC(C(=O)N(CC(C)SC)C)N(C)C)c1 C1(O)(CC(=O)OCC)CCN(C(=O)NC(c2ccc(OC(F)F)cc2Cl)C)CC1 c1(NC(=O)CNC(C2CCC2(F)F)=O)cccn(C2CC2)c1=O N1(CC2CN(C(C)C)C2)CC2CC(N3CCCC(C)CC3)C1C2 c1(OC)ccc(C2CC(NC(c3cc(Br)c(Br)o3)=O)C2)cn1 c1(NC(=O)NC2CCN(C(C)=O)C2)ccc(OCC2CC2)c(C#N)c1 CCCCCC(O)C(=O)N1CC2CC1(C(N1CCC1C(N)=O)=O)C2 C1(C(=O)NC2CC3CN(C(C(COC)(F)F)=O)C2C3)Cc2cc(F)cc(F)c2O1 C1(NC(c2c(OC)scc2)=O)C2CCN(C(=O)C=Cc3nc(C)cs3)CC12 C1(C(=O)NCC(C)(O)CNC(C2COC2)=O)CCOC2(CCCC2)C1 c1(-c2cc(NC(c3cnc(OC)c(C)c3)=O)ncc2)cccc(C#N)c1F c1(C(=O)NCC2N(C(CS(N)(=O)=O)=O)CCC2)cc([N+](=O)[O-])ccc1N(C)C C1(C2CCC2)(C(=O)NC2CN(C(C(c3cn(CC)nc3)=O)=O)C(C)C2)CC1(F)F c1(C(=O)NC(C)CC2CN(C(c3c[nH]c(C(C)(C)C)n3)=O)C2)ccc(Cl)nn1 C1(NC(=O)C(c2cc(Br)c(Cl)s2)N2CCCC2Cc2cccs2)CCC(F)(F)CC1 N1(C(CSCCCC)=O)CC(C(=O)N(CC2=CCCOC2)C)C(CC)C1 c1(NCCC2CCN(C(c3c(C)scn3)=O)C2)nc2c(cc1C#N)CCCC2 CC1CCN(C(=O)CNS(N)(=O)=O)C1CNC(=O)CCC=CBr Cc1nnc2n1CC(C(=O)NC(C1CCN(C(=O)C3=NNC(=O)CC3)C1)C)CC2 C1(C(N(CCC(N2CCC(C)(N(C)CC)C2)=O)C(C)C)=O)CC2(CCO1)CC2 Cc1ccc(C(=O)NCC2CCCC(NC(c3coc(C4CC4)n3)=O)C2)nc1 C1(C(=O)NC(CC)CN2CCCC2)CN(C(C2(CC)CCCCO2)=O)CC1(F)F C1(CC(=O)N(CCCOC)C)CN(C(C2CCC2)=O)C(C)(C)C1 C(CC(=O)NC1C(C)(C)C(NC(C2(C)COC2)=O)C1(C)C)(C(F)(F)F)OC C1(C(=O)NCC(CNC(c2cc(CC)[nH]n2)=O)C)(Cn2cncn2)CCOCC1 c1(NC(C2C(CC)CCN2C(=O)C(C)OCCOC)=O)ccc(O)c(Cl)c1 C(=O)(C(C)C1=CCCC1)N(c1c[nH]nc1OCC(F)F)C1CC(N(C(C)=O)C)C1 c1(C(N2CCC(C(=O)NCCCc3ccccc3Cl)C2)=O)n[nH]c2c1CCC2 C(CCC(=O)NCC1CC1CNC(=O)CCc1cnn[nH]1)SC c1(OC)cc(C=CC(=O)NCC#CCNC(c2cncc(SC)c2)=O)ccc1O c1(C(N(C(C)CNC(=O)Cc2cc(OC(F)F)no2)C)=O)ncc(Br)cn1 N1(C(C(CC)(C)Cl)=O)CC2CCCC2(CNC(c2ccn(C)n2)=O)C1 CC1CCCCC1(CO)NC(C12CC(CN1C(=O)CN1CCC(F)CC1)C2)=O Cc1nc2ncccn2c1C(=O)NC1CC(NC(c2ccc(Br)c(C#N)c2)=O)C1 n1(CC)ncc2c(C(=O)OCCCn3ccnn3)cc(C3CC3)nc12 C1(CNC(c2cccc(C(N)=O)c2)=O)CN(Cc2ccc(F)cn2)CCCO1 c1(CC)cc(-c2nccn2C(C)C(=O)O)ccc1OC.c12nn(C)cc1NC2=O c1(C(=O)NCC2C(NC(c3cc(C)sc3)=O)C2)ccc(N2CCCC2=O)cc1 C(=O)(CS(=O)(=O)C1CCCC1)N1C(CNC(C(CC)CC2CCCC2)=O)CC1 C(=O)(C1CCc2nccn21)N1CC(NC(c2c(S(C)(=O)=O)scc2)=O)C1 C#Cc1cccc(C(=O)NC2(CNC(c3ccsn3)=O)CCC(C)(C)CC2)c1F C1(=O)C(CC(C)C)CCN1.CCC1CNC(=O)OCC(=O)N1.C(C)(C)(C)O c1(C(N2CC(C)(NC(=O)C=Cc3cc[nH]c3)C2)=O)cc2sccc2cn1 CC(F)(C(=O)NCCC1CCCCN1C(=O)CN1C(=O)CCCC1=O)C(F)(F)F N1(C(c2cc(OCC)no2)=O)CC(NC(C2CC2F)=O)C(CC)C1 C(=O)(C(C#N)C(C)(C)C)NCc1occ(C(N2CCC(SC)C2)=O)c1 Cc1cccc(C(=O)NC2CCCN(C(=O)COc3ccc(F)c(Cl)c3)C2)c1F C=CC1CN2CC1NC(=O)CCC(C)OCC2=O.C1(NC(=O)COC)CCCC1 C1(OC)(CNC(=O)CSC2CC2)CCN(C(=O)C(C(C)C)n2ccnc2)C1 N#CCCCC(=O)N1CCOCC1CCNC(C1(c2ccncc2Cl)CC1)=O c1(C(=O)OC)ccc(NCC2CCCN2c2ncnc3[nH]ccc23)c(C#N)n1 C#CC1CC(NC(=O)C(C)(C2CCC2)NC(=O)CSCC=C)C1 Cc1ccc(C#N)cc1C(=O)N(CC(C)C(=O)NC1CCC(C(=O)OC)C1)C C(=O)(CN=c1ccc(Cl)n[nH]1)NC1(C2N(C(C(CC=C)C)=O)CCC2)CC1 C1(NC(=O)CC2OCCO2)C2CCC(C2)C1C(=O)NCC12CCC(CO1)C2 CCC(CC)(CC)C(C(=O)N1CSCC1C(=O)OC(C)=O)NC(N)=O c1(CCCc2ccc(C(=O)OC)[nH]2)cccc(CO)c1.C1C(C)NC(=O)N1 N1(C(COC)=O)CCC(C(=O)Nc2cc(C)ccc2OC)C(C)(C)C1 N1(C(C2(C)CCOC2)=O)CCOC2(CCC(NC(=O)Cc3cn[nH]c3)CC2)C1 N1(C(CSCCC)=O)CCSCC1CCNC(C1CCCCC1C)=O Cc1ccc(-c2nc(CNCc3ccsc3I)cs2)s1 Cc1cnc(N2CC(CNC(c3sccc3C3CC3)=O)CC2C)nc1C C(=O)(C1CCCc2ccccc21)N1C(CC)CN(C(=O)CCC(F)F)CC1 c1(C(=O)OC)ncc[nH]c1=NC1CC(O)(CNC(c2nc(O)c(C)s2)=O)C1 c1(C(N(C(CNC(C(CC=C)C)=O)C)C)=O)c(F)cccc1[N+](=O)[O-] C(=O)(CC(C(C)OC)NC(c1c[nH]c(=O)cn1)=O)N1CCN(C(CC)C)CC1 c1(C(N2CCC(C)(c3cn(C4CCNC(=O)C4)nn3)C2)=O)nccc2cc[nH]c12 CC1CC2(CCN(C(C3CCCN3C)=O)CC2)CN1C(c1coc(N(C)C)n1)=O CC1(C)CC(NC(C2CCC(=C(F)F)CC2)=O)CN(C(C2CCCC23CC3)=O)C1 N1(C(c2c(C)nsc2)=O)CCCCC1CNC(c1ccc(Cn2cccn2)cc1)=O c1(CO)ccc(-c2nc(COc3ncccn3)nn2Cc2ccccc2F)cc1 C1(C(=O)Nc2nccc(OC)c2C)CCOC2(CCSC2)C1 C1(C(=O)NC2(CF)CCN(C(C(C(C)C)F)=O)C2)CC2CCCC(C1)C2 C1(C(=O)Nc2c(C)c(N3CCCCC3)ccc2)CC2C=CC1CCC2 CC12CCC(=O)N1CCCN2C(=O)C(c1cccnc1)O C(C(CO)C(C)(C)C)NC(c1c(C)cc(CNC(c2ccnc(CO)c2)=O)o1)=O c1(CN=C(NCC(COC)(C)C)NC(C)C)ccc(C#N)c(F)c1 C1(C(=O)NC2(CCC(=O)NCc3c(C)noc3)CCC2)CC(C)(C)CO1 N1(C(C2CC(=C)C2)=O)CC2CCCC2(CNC(c2cc(CC3CCC3)c[nH]2)=O)C1 C1(NC(c2c(C)cccc2C)=O)CN(C(c2cn(CCO)nn2)=O)CC(F)(F)C1 c1(CNCC2N(C(C3CC(=C)C3)=O)CCCC2)c(OC)cccc1OC Cc1cc([N+](=O)[O-])nn1CC(=O)NCC#CCNC(C1CCN(C)C1C)=O c1(CN(C(C2CCN(CCC)C2)=O)C)nn(C)cc1Br C#CCCCCCC(=O)N(C)CC1(C)CCCC1NC(c1ccccc1OC)=O C1(CCOC)CN(C(=O)C(c2ccccc2)OC)CCN1C(=O)CNC(C)=O C(CNC(C1CC1C1CCCC1)=O)(CC(=O)NOC1CCOCC1)OC C1(CNC(=O)CC2CC=CC2)CCCCC1C(c1ccc(CC(=O)NO)cn1)=O c1(OCCC(=O)NCC2(C(=O)OC)CC2)ccccc1OCC c1(OC)cc(NC(C2C(O)CCN2C(c2sccc2Br)=O)=O)nc(Cl)c1 c1(CNC(C(N2CC(COCC)OCC2)=O)=O)cc(Br)ccc1I c1(CC(C)C)ccc(C(C)C(=O)NCC(c2ccccc2)O)cc1 N1(C(COCCC#C)=O)CC(F)(F)CC1CNC(c1onc(C)c1C)=O CC(CCC(C)(C)C)NC(=NCC1CC1)NCc1c[nH]nc1C(F)F c1(C(=O)NC2C(NC(C3(CC#C)CCC3)=O)CCC2)n[nH]c2c1CCCC2 C12(C(=O)NC(CCOCC)C)CCCC1N(C(c1cc[n+]([O-])cc1)=O)CC2 N1(C(=O)Nc2cc(C)sc2)CCS(=O)(=O)CC1C1CCC1 CC(O)(CC(=O)NCC1(O)CN(C(C2CC3(CCC3)C2)=O)C1)C1CC1 CC1CC(NC(c2ccc(Sc3ccccn3)cc2)=O)CN1C(=O)COC1CC1 N1(C(c2cc(OCCN(C)C)ncc2)=O)CCC(NC(c2cscc2F)=O)C(O)C1 c1(C(N(CCC(=O)NCC2CCN(CC)C2)C(C)C)=O)ccc(C)cc1 c1(C(N2CCCC(NC(CCC(=C)C)=O)C2C)=O)cc2cccnc2nc1C C(C(CC(C)C)NC(=O)C(O)CC1CCCC1)NC(CC1(CC(=O)OC)CC1)=O c1(CC(=O)NC2CCN(C(C3CC3c3nc[nH]n3)=O)C2)ccc2oc(O)nc2c1 N1(C(C(c2cccc(OC)c2)O)=O)CC(NC(c2csc(C)c2N)=O)C2(CC2)C1 C1(CC)CCCN(C(=O)CC(COC)NC(=O)Cc2cccnc2O)C1 N1(C(CN(CC)CC)=O)CC2C3CCC(C2C1)N(C(c1cccc(CO)c1)=O)C3 c1(CN2CC(CNC(c3ccc(C)s3)=O)OCC2)c[nH]c2cnccc12 c1(C(=O)NC(C(C)=O)(C)c2ccccc2)ccn2ncc(Cl)c2n1 CCCCC(=O)C(=O)N(CC(C)(C)CNC(C1CCOC(CCC)C1)=O)C N1(C(c2cn(CC)nn2)=O)CCC2(CCCCN(C(=O)Cc3nnc(C)o3)C2)C1 C1(NC(C2(CC#C)CCCO2)=O)CN(c2nncs2)C2(CCOCC2)C1 c1(OC)cc(-n2nc(C3CC=CCC3)nc2Cn2c(C)csc2=O)ccc1Cl Cc1cccc(F)c1C(N1CCC(=CCNC(c2cc(Br)c[nH]2)=O)CC1)=O c1(COC)nc(NCc2cc(Br)ccc2C)cc(=NCCC2CCCN(C)C2)[nH]1 c1(C(=O)NC(CN(C(c2ccc(OC(C)C)cc2)=O)C)C)cccc(S(C)=O)c1 N1(C(C(C=C)C)=O)CCN(C)C(Cn2cc(-c3ccc(C(=O)O)nc3)nn2)C1 N1(C(C=C(CC)CC)=O)CC2CC(CNC(c3ccc4occc4c3)=O)CC1C2 N1(C(Cc2c(C)cnn2C)=O)CC(C)(C)CCC1CNC(c1cnsc1)=O S(=O)(=O)(c1cccc(C(=O)O)n1)NC1C(OC)C2(C1)CCC2 Cc1ccc2[nH]c(C(=O)NCC(C)CNC(C34COC(CCO3)C4)=O)cc2c1 c1(C(C(C)C)O)cn(CC2CCC(NC(=O)C(F)F)C2)nn1 N1(C(=O)OC(CC)C)CC(Nc2[nH]c(C)nc2C#N)C2(CC2)C1 C1(CCC(=O)NC(c2nccs2)CC)CCCN(C(c2cc(O)n(CC)n2)=O)C1 C12(C(=O)Nc3cc(C)c(NC(=O)C(O)C(C)C)cc3)CCC(CC1)C2(C)C CC(C)CC(=O)NC(C)CC(C)NC(c1csc(C(F)(F)F)c1)=O c1(C(C(=O)NC(C2CN(CC=CC#N)CCO2)C)(C)O)ccc(F)cc1 C1(CNC(C(COCC)C)=O)CC2(CO1)CN(C(=O)CCCCNC(N)=O)C2 N1(C(C2C(C)OCCO2)=O)CCCC12CCCN(C(C1(C)CCN(C)CC1)=O)C2 C1(C(=O)NCC2CCCN(C(c3ccccc3)CCOC)C2)CC1C1CCCC1 CC1COC2(C1)CN(C(=O)C(CCN(C)C)NC(=O)CN1CCCNC1=O)C2 n1(CC2CCN(C(C)=O)C2)nnn(-c2cccs2)c1=O.C1CS1 N1(C(CCNC(C(=CC2CCCC2)C)=O)=O)CCCC(C)C1C(N)=O C1(NC(C(C2CC2)OCC)=O)CN(C(=O)CSCCC#N)CCC1F C12(C(=O)NCCCCC(OC)OC)C(NC(=O)C(C)C#N)C3CC1C2C3 N1(C(C(=O)NC2CC2)CC2CCC2)CCC(C2OCCO2)CC1C(F)F C1(N(c2nnc(CC)o2)CCO)CCCN(C(=O)C(C)NC(C)=O)C1 C1(C(N2CC(n3cc(-c4ccc(F)c(Br)c4)nn3)C2)=O)CCCC(C(F)F)CC1 N(C(=NCCNc1ccc(F)cc1)NC1Cc2ccccc21)CC(=O)OC(C)C C(CCCCC(=O)NC1COCC1C)NC(c1cccc(NC)n1)=O c1(CC)nc(C(=O)NC(C)(CNC(=O)C(C)c2cncs2)C2CC2)co1 C12(C(N(CC(C)CO)C)=O)CC1CN(C(c1ccc(F)cc1)=O)C2 c1(-n2ccc(C(=O)NCCC(C)NC(c3cnnn3C)=O)n2)ccc(Cl)c(F)c1 Cc1cnc(Cl)c(NC(C2CSCCN2C(c2noc(C)c2C)=O)=O)c1 CC1C(NC(=O)CC2CCC(=O)NC2)CCCN1C(c1ccc(C(N)=O)cn1)=O c1(CC)ccc([N+](=O)[O-])cc1C(=O)NC1CCCC1NC(C1CC(C)(F)C1)=O C1(NC(CNC(C2C(C)C2)=O)=O)CCOCC1C(N1CCC(C(C)C)(CO)C1)=O C(=O)(C(C(C)C)C1CCC1)NC(C(=O)NC1C(C(=O)NC)CCC1)C1CCCC1 CCCC(O)CC(=O)N1CC(=C(F)CNC(c2nncn2C)=O)C1 c1(NC(C2CC(CCNC(C(C3CCCCC3)C)=O)C2)=O)cn(C)nc1C(N)=O C(=O)(CCCCCCC(=O)N1CCC1CNC(c1c(C)nc2sccn12)=O)OC Nc1cc(C(N2CCC(NC(C3CC=CCO3)=O)C2)=O)ccc1-n1cnnc1 C1(NC(C(CSC)OC)=O)(CNC(c2csc(C)c2)=O)CC2CCC1CC2 CCC(CC)C(O)CNC(=O)CC1(OC)CN(C(=O)C(C)C(C)(C)C)C1 N1(C(CC(C)O)=O)CC23CCCC2(C1)CN(C(=O)C=Cc1ccncn1)C3 c1(OC)ncc(Cl)cc1C(N1CCC(NC(c2cn(C3CCOC3)cn2)=O)C1)=O Cc1cc(C(=O)NC(CNC(=O)C(C(C)O)N(C)C)C(C)C)c(O)c(C)n1 N1(C(C=CCCC)=O)CCC2(C=C(C(=O)NCC3CCCC34CCC4)C2)C1 Nc1ccc(-c2cn(CC3CCCCN3C(=O)C(O)C3CC3)nn2)cc1[N+](=O)[O-] C1(C(N(C2CCCC2)CCNC(C2(C)CC2(Cl)Cl)=O)=O)CCn2cncc2C1 S(=O)(=O)(c1ccccn1)N(c1nc(OC)c(Br)cn1)C1CCCNCC1 c1(NC(C23C(CN(C(c4ccc(Br)s4)=O)C2)C3)=O)cccc2cccnc12 c1(OC)ccc(Cl)c(CC(=O)NCC2CC(F)CN(Cc3ccsc3Br)C2)c1F N1(C(c2c(OC)ccs2)=O)CCC2(CNC(C)=O)CC12 c1(CC(=O)NCC2(OC)CN(C(C34CCCC3C4)=O)C2)ccc2ccccc2c1 C#CC1CCN(C(=O)C(CC2CC2)NC(=O)C=Cc2cncs2)C1 C(=O)(CCCC(F)(F)CO)N1C(CNC(C23OC(C)C(CC2)CC3)=O)CCCC1 C(=O)(CC1COc2ccccc21)NC1CC(CNC(Cc2cn(C)nc2)=O)C1 C12(C(N3C4CC(C(=O)NC(CC(C)C)CO)C3CC4)=O)CC3CC(CC(C3)C1)C2 N1(C(C(C)c2cccs2)=O)CC2CCC1CC2NC(=O)CCC(N)=O C1(CNC(C2C3CC4C(C3)C24)=O)C2CCCC1N(C(c1cn[nH]c1)=O)C2 S(=O)(=O)(c1ccc(Cl)cc1F)C=O.C(=O)(C1=NOC(CNC2(CO)CCC2)C1)NC C12(NC(CCCN(C)C)=O)CN(C(C3CSCCS3)=O)CC1CS(=O)(=O)C2 c1(C(c2n(CCCC)nnn2)NCc2ccoc2C)cnc(SC)nc1 CC1CN(C(c2ccn(C)c(=O)c2)=O)CC1(C)C(N1CCC2(CCC2)C1)=O CN(S(=O)(=O)N1CCCCC(CO)C1)c1ccc(N(C)C)c(C(N)=O)c1 C(C1CCCc2nc[nH]c21)NC(=O)C(c1ccc(Cl)cc1F)O C(=O)(C1CCc2nccn21)NC(C)(CNC(c1cnn[nH]1)=O)C1CCC1 Cc1cccn(CC(N2CC3(CCC3NC(C3CC=CCO3)=O)C2)=O)c1=O CS(=O)(=O)c1cc(C(=O)NCC2CCC2NC(=O)Cc2ccccc2)ccc1F C1(OC)CN(C(=O)Cn2cc(C(OC)OCC3CC3)nn2)C(C)(CSC)C1 N1(C(C(CC)OC)=O)CCC2(CC1)CCN(c1cc(-n3cncn3)ncn1)CC2 C12(CNC(c3nc(CC(C)C)sc3)=O)CC1CN(C(=O)CCCc1ccsc1)C2 C1(C(=O)OC)CCCN(C(=O)COC(c2cnccc2-n2cc(C)cn2)=O)C1 Cc1cccc(Cn2nc(CO)nc2-c2cnc(-n3nnnc3O)s2)n1 CCCCCCN(C(=O)CSCCNC(=O)C(C1CCC1)OC)C C(C(C(=O)N(CC(O)CNC(c1ccc(Cl)cn1)=O)C)C(C)(C)C)OCC=C C1(C(N2C3CN(C(c4c(CC)non4)=O)C(CC3)C2)=O)COc2ccccc2C1 C1(C(=O)NCC(CO)NC(CCC)=O)(COC)CCCCCC1 CC(CN(C)N1CCOCC2(CCOCC2)C1)OCC(F)(F)F C1(COC)(CNC(=O)CNC(C2OCCC2NC(=O)OC)=O)CC=CC1 c1(C2(C(=O)NCC#CCNC(c3cn(C)nc3)=O)CC2)ccc(Cl)cc1Cl C(=O)(C(C)CC(F)(F)F)N(C1C(O)CCN(C(CCc2scc(C)c2)=O)C1)C N#Cc1ccc(OCC(=O)Nc2cc(N3CCCC3)nc(Cl)c2)nc1 C1(c2n(C)ncc2)CCCCC1NCc1ccc(O)nn1 C1(CC(=O)NC2CCCCC2CCNC(c2ccnc(F)c2)=O)CCCC12CC2 N1(C(c2c(C)c(N)ccc2)=O)CCC2CC(NC(c3ccncc3)=O)CCC2C1 c1(C(=O)NCC(CNC(C(C)Cn2ccnc2)=O)O)ccc(F)c(Cl)c1F C(=O)(C1=C(Cl)CCC1)NCCC(C)NC(c1c(C)coc1C1CC1)=O c1(C(N2C(C)(c3cn(CCO)nn3)COCC2)=O)cc2ccncc2cc1F N1(C(C=CCN(C)C)=O)CC(NC(=O)CC2CCC(C)(C)O2)C(C(F)F)C1 C1(C(CNC(C(C=C)C)=O)C)CCN(C(C2(C)CC2(Cl)Cl)=O)CC1 C1(NC(c2ccccc2)=O)CCC12CCN(C(=O)CCN1CCCCC1)CC2 c1(C(N2C(CCNC(c3cc(C4CC4)no3)=O)COCC2)=O)cc(F)ccc1O c1(C(=O)NC(C2CCN(C(c3cncc(O)c3)=O)C2)C)ncc2cc(Cl)ccn12 C1(C(N2CC(NC(c3ccc(C)c(Cl)c3)=O)C(F)C2)=O)CCC2C(C1)C2(F)F N1(C(CC2CCCC(=O)N2)=O)CC(=O)NCC1C(=O)NCC=CC=C(Cl)Cl CCCC(C(O)C(=O)N(CC(F)Cl)C)NC(C1OCCCC1(C)C)=O C1(O)(C(=O)NC(c2ccccc2-c2ccccc2F)C)CC2(CCNC2)C1 c1(C(=O)NCCCCC(C)NC(=O)C=CS(C)=O)cc(Cl)cc2cccnc12 c1(C(N(CCNC(c2c(CC)scn2)=O)C2CC2)=O)ccc(C2CCOC2)cc1 C(=O)(CCC(=O)c1ccc(Br)cc1)NC(C1CCCCC1)(C)CO C1(C(N(CCCNC(c2ccc(OC)o2)=O)CCO)=O)CCCNS1(=O)=O C12CC(C1(C)C)NC(=O)N2.C(CS(=O)(=O)N1CCCC1)OC(C)C C(C(O)CC(F)(F)F)NC(CC1N(C(C2(C)CCN(C)C2)=O)CCCC1)=O N1(C(CCC=CC(C)C)=O)CC(C(=O)NCCn2ccc(=O)cc2)C2CCCC12 c1(OCCC(=O)NC2CN(C(c3ns[nH]c3=O)=O)C2)ccc(Cl)cc1 N1(C(CC(CN(C)C)O)=O)CCC(NC(c2ccnc(C(C)C)n2)=O)C12CCC2 Cc1cc(F)ccc1NC(C12CC(CN1C(=O)CC1(O)CCOC1)C2)=O c1(C(N2CCC(C)(NC(C3CC4(F)CC3C4)=O)C2)=O)cccc2occc12 CC1CCc2ncc(C(N3CC4C(CNC(c5ccc(Br)o5)=O)C4C3)=O)n2C1 C(CC(C)C(=O)NC1(C)CN(C(C2(C)CC2(Br)Br)=O)C1)OC CCC(O)CC(=O)N1CC(O)CC1c1cn(-c2ccc(Br)nc2)nn1 N1(C(CCCC#C)=O)CC(=O)NCC1C(=O)NCC(C)(C)CC(C)C N1(C(C=C)=O)CCCC(CN(C(=O)C(CC)c2ccccc2)CC)C1 N1(C(C(c2cccs2)SC)=O)CCC(C2CC2)(NC(c2cc(C)cs2)=O)C1 C(CC(O)CC(=O)NCC1CN(C(=O)CN2CCCC(N(C)C)C2)C1)SC c1(C(N=c2[nH]n(C)c(OC[O-])c2)=O)ccc2ncccc2c1Cl Cc1cc([N+](=O)[O-])ccc1NCC1CCC(NC(C2CC(C)CO2)=O)C1 c1(CN(CCC)CCC)ccc(C(=O)NC(C2(CO)CC2)C)s1 C1(C(=O)NCc2ccnc(Cl)c2)CN(C(c2ccc(O)cn2)=O)CCC1O c1(CC(N2C(C)(CC)CC(NC(C3CSC3)=O)C2)=O)c[nH]c2c(C)cccc12 C=CC1(C(=O)NCC(c2cnn(C)c2)C)CCN(C(=O)C(O)CC(C)C)C1 C12(C(=O)NCCN(C(C34CCC(C3)C4)=O)C3CC3)CC3CC1C2C3 C1(S(C)(=O)=O)(C(=O)NC2CN(C(CC(C(C)C)C)=O)CC2F)CCCC1 C=C=CCCC(=O)NC(c1nocc1C(=O)N(C1CCOC1)CC)C C12(C(N3CCC(C)(NC(c4c[nH]cc(F)c4=O)=O)CC3)=O)CCCCC1C2(F)F C#CC1(N(C)C)CN(C(C2CCN2C(c2ccc(NC)cc2)=O)=O)C1 C1(CN(c2c(C)cnn2C)C(C)=O)CC(O)C(O)CC1C(=O)NOCC(O)CO C1(C(N2CCCC(CCNC(CC(=C)C)=O)CC2)=O)CC2(CCC2)CCO1 c1(C(N2C(C(=O)NC(N3CCCCC3)CC)CC2)=O)cc(C)nc(C)n1 Cc1ccc(C=CC(N2CCCC(CCNC(c3nn[nH]c3Cl)=O)C2)=O)cn1 c1(OC)ccc2c(n1)N(C)CCN2C(=O)CN1CCC(C(=O)O)CC1 S(=O)(=O)(c1cccnc1NC(CCO)C1CC1)NCc1n(CC)c(C)nc1 C=CCC(C(=O)NCC1(CNC(=O)C=Cc2cnn(C)c2)CC12CCC2)C(C)C C(=O)(C1CCCc2nncn21)NCCNC(=O)C1=CC(O)CCC1 N1(C(C(C)NC(=O)NC)=O)CCC(ON(C(=O)CN(C)C(=O)C2CC2)C)CC1 N1(C(C2(CCC)CC2)=O)CC(CNC(c2cc(COC)cs2)=O)CC(C)(C)C1 CCCC(CNC(c1cc(CNC(c2cnn(C)n2)=O)ccn1)=O)CCO CCCCC(CC)C(=O)N1CCC(COC)(NC(C2CN3CCN2CC3C)=O)C1 N1(C(c2cn(C)nc2C(F)F)=O)CC(NC(c2ncn(C)n2)=O)CC2(CCC2)C1 c1(OC)ccc(Cl)c(Cl)c1C(N1CC2CCC1C(NC(=O)C=C(C)C)C2)=O CCCCCCCC(=O)N1CC2CCN(C(c3cc(C(N)=O)co3)=O)CC12 N1(C(C(CNC(CC(CC)C2CCC2)=O)C(C)(C)C)=O)CC(C)(C)OC(C)(C)C1 n1(CCNC(C2C(C)C2)=O)cc(C(=O)NC(C2CCCCC2)(C)C)cn1 C(=O)(C1=CCC2(COC2)OC1)N1CCC(NC(C(C)Cc2cccc(F)c2)=O)C1 N1(C(C2CCC(=O)OCC2)=O)CCC(CNC(C2CC3(CC3)CO2)=O)C(F)(F)C1 C1(CNC(C(=O)NCCC2(C)CCCO2)=O)CCCCN1Cc1cccc(F)c1 Cc1ccnc(C)c1C(=O)NC1CCOCC1C(=O)NCc1ncsc1C c1(C(N2C3C(NC(COCCCC#C)=O)CC(C3)C2)=O)ccc(OC)c(C#C)c1 C1(C(=O)NCC(C(C)C)NC(=O)COc2ccon2)Cc2c[nH]cc2S1(=O)=O Cc1nc(NC(c2nc(C(=O)NCCc3cccnc3)cs2)=O)nc(Cl)c1Br Cc1cc(C(F)(F)F)nn1CC(=O)NCCCN(C(=O)C=C1CCC1)C(C)C c1(OC)ccc(C(=O)NC2CCN2C(c2ccncc2Br)=O)c(OC)c1 S(=O)(=O)(c1cccc(N2Cc3cnc(Cl)cc3C2)n1)N1C(C)C(O)CCC1 C(=O)(C1=CCC(C)(C)CC1)NC(CNC(C1CN(C(=O)NC)C1)=O)(C)C1CC1 C#CC1CCC(C(N2CCC(C(C)NC(=O)COc3ccccc3C)C2)=O)CC1 c1(N2C(CNC(CCCCC)=O)CCC2)cc(Cl)nc(C)n1.C1C(=O)O1 C1(CC=C)(C(=O)NCC(F)C(C)(C)O)CCCN1C(=O)C(CN(C)C)CC CC1(C)CC(=O)NCC1C(=O)NC1CCN(C(c2ccsc2C#N)=O)CC1 Cc1ccc(C(=O)CN(C(C)(C)C)CC2COC2)s1 CC(C)(C)CC(C)(C)C(=O)NCC1(C)CN(C(C2(F)CC=CCC2)=O)CCO1 c1(N(C)C2CC2)ccccc1.C1(C2CCC2)C(=O)NCCSC2C(CC2)N1CC.C(C)O C(C(CC(C)C)C(=O)NC1(CNC(c2nn(C)c(Br)c2C)=O)CCC1)OC C1(C(N2CCN(CCCNC(C3N(C)CC(O)C3)=O)CC2)=O)CC12CCOCC2 C(=O)(CCC1=CCCCC1)N1C(C(N2C(CO)CC(OC)C2)=O)CN(C)CC1 Cc1nc(O)[nH]c1C(=O)NC1CC1CNC(C1(c2ncco2)CCC1)=O C(CCCC(=O)N1CCC(C)(CCC)C1)N(C(C(C)=CC=C)=O)C C#Cc1cccc(CC(=O)N(CCNC(c2ccc(COC)c(C)c2)=O)CC)c1 c1(C(N2CCC(C)(C(=O)NCCc3ccsc3)C2)=O)ccc2cc(O)ccc2n1 N1(C(C=C2C(C)(C)CCCC2)=O)CC2CC(NC(c3cncc(F)c3)=O)CC2C1 N1(C(c2c(C)con2)=O)CCC(CO)(CNC(C2(CF)CC2)=O)C1 C1(CCC)CCCCN(Cc2ccc(N(C)C3CC3)cn2)C1.c12ncccc1S2 CC1=C(C(=O)NC2CN(C(c3snc(Cl)c3Cl)=O)CC2F)SCCO1 c1(NC(C(C)C)CCO)ncccc1S(=O)(=O)NCC(c1ccccc1F)NC c1(NC(c2n(CCSC)nnn2)(C)C(C2CCOC2)C)ccc(-n2cncn2)cc1 C1(OC)(OC)CCC1C(=O)NC(C(=O)N(C(C)C(F)F)C)C1CCCO1 C1(NC(c2cnn[nH]2)=O)CCC2CCN(C(c3csnn3)=O)C12 N1(C(c2cn(CCOCC)nc2)=O)CC(NC(=O)C(C)C(F)F)CCC1C C(=O)(C1=CCCCCC1)NCC(C(=O)NCC(CCC=C)O)C(C)C C1(NC(c2cc(C)nn2C(C)(C)C)=O)CN(C(=O)Cn2cnnn2)CC2CC12 C1(C(=O)NCCC(CNC(C(COCC)C)=O)(C)C)CC2C=CCC(C1)C2 N1(C(C2CC(N(C)C)C2)=O)CCCC2(C1)CN(C(=O)COC1(C)CCC1)C2 Cc1cccc(C(CNC(=O)CCC2CCOC2)NC(c2cc(C#N)c[nH]2)=O)c1 C1(OC)CC(CCNC(c2cc[nH]c2)=O)N(C(=O)CCCOc2ccccc2)C1 CC1CCN(CCC(=O)NCC2(C(N)=O)CN(C(=O)CC(F)(F)F)C2)CC1 N1(C(CCn2ncc(C)c2)=O)CCC(CNC(c2nnc(O)cc2C)=O)C(C)C1 Cc1nc(CNC(=O)C(C)CN(C(=O)CCC2CCCN2C)C)[nH]c1C CCCCCCCC(=O)N1CC2CCC2(C(=O)Nc2nccc(Cl)c2I)C1 c1(C(=O)NC(CC(C)C)CO)c[nH]c2cc(-c3scc4c3OCCO4)cnc12 N1(C(CCCOCCC)=O)CC(O)CCC1C(=O)Nc1cccc(OCF)c1 c1(C(=O)NCC(CO)NC(C(C)CC2CC2)=O)ccccc1OCC(N)=O C(=O)(CC(O)C(Cl)(Cl)Cl)NC1CCCC(NC(C2(C)CCCCCC2)=O)C1 C(C(COC)CC(=O)NC1CC(O)CN(C(=O)CCOCCCOC)C1)OC N1(C(c2ccn(CC)n2)=O)CC(OC)CC(NC(c2ccc(I)c(C)c2)=O)C1 C#Cc1cc(NC2CCN(C(=O)NC3(c4ccccc4)CCCO3)C2)ccc1C CC1CC(=O)NC(C(=O)NCC2C=CC(NC(=O)C=Cc3cnc[nH]3)C2)C1 C(C(C)(C)CC(=O)N1CCCC(C(C)(C)C)C1)N(C)CC1(C(=O)OC)CCC1 C=C(F)C1(CC(N2CC3(CCC3NC(=O)C3CC3)C2)=O)CCOCC1 Cc1ccnc(C(=O)NCC(C)N(C(=O)C(F)CC2CCCCC2)C)n1 N1(C(C=C(CC)C)=O)CCC(N(C)C(c2cc(C3CC3)[nH]n2)=O)C1 C1(C(N2CCCC(C)(NC(c3cc(Cl)no3)=O)C2)=O)CCCC2(CCC2)O1 c1(C(=O)NC(C)C(CO)NC(C2CC(C)(F)C2)=O)cccc(N2CCCCC2)c1 C=C(C)CCCC(=O)NC1CC(O)(CNC(=O)CCSc2cc(F)ccc2F)C1 C1(CNC(C(n2cc(C)nc2)(C)C)=O)CC2CCC(C1)N2C(C12CCC(C1)C2)=O Cc1cc(=NCC2CCOC2)[nH]cc1S(=O)(=O)N1CC2CS(=O)(=O)CC2(C)C1 n1(CC(=O)N(CC(O)CN(C)C(=O)C2CC2)C)nc2n(c1=O)CCCCC2 C(C(=O)N(C)Cc1cocn1)(C1CC1)NC(C1C(CCOC)C1)=O C(CN=c1[nH]c(=NC)[nH]c(=NC2CCC(OCC)CC2)[nH]1)NC1CCCN1CC Cc1nc2c([nH]1)CC(C(=O)NC1CC1CNC(=O)C(C)(C)C(=O)N(C)C)CC2 c1(N2CCCC(O)(CNC(CNC(C)=O)=O)C2)nc2c(C)c(C)ccc2s1 c1(OC)ccc(CC(=O)NCC2(NC(=O)Cc3cncnc3)CC2)nn1 Cc1c(C(=O)NC(C(=O)NCC(C)(C)O)C2CCCO2)ccn1C c1(C(N2CC(C(C)NC(C(C)NC(=O)NC3CCCC3)=O)C2)=O)cnc(Cl)s1 c1(C(N(C2CCCN(C(C(CC)O)=O)C2)CCF)=O)cc2ccccc2nc1O N1(C(C(C2CCCOC2)OC)=O)CCN(C(=O)Cn2cc(C#N)cn2)CC1C N1(C(C(=O)NCC(C(F)OC)C)=O)Cc2cccc(C)c2C1c1ccc(F)cc1 CCS(=O)CC(=O)N1CCC(NC(=O)C=Cc2ccc(C3CC3C)o2)C1 C#CCC(CC(=O)NCC(F)CNC(c1cc(OC)cnn1)=O)c1ccccc1 N1(C(Cn2c(C)c(Cl)cn2)=O)CC2CC(NC(=O)CC3CCCC3O)C1C2 n1(CC)c(C(=O)NCC2(C)CC(NC(=O)C3=NOC(C)C3)C2)cc2ccccc12 C(=O)(C(C)P(C)(C)=O)NC1(C)CCN(C(C(CCC)c2cccc(Br)c2)=O)C1 Cc1cc(C(=O)NCCC2CCN(C(=O)C(C)C3CCC3)C2)c(Br)c(C)c1 C(=O)(C(CNC(=O)CCCOC)C(C)(C)C)N1CC(C(=O)NCC)C1 c1(C(=O)NCCCN(C(C(C2CC2)SC)=O)C)ccc(C(O)CF)cc1 N1(C(C(C)C2CC2)C(=O)NCCC2CC2)CC(=O)N(C)C(C)C1 C(C)(CNC(=O)C=CC(C)(C)C)(CO)NC(C1C(C(=O)OC)CC1)=O c1(OC)cc(NC(=O)C(=O)C(C)(C)C)ccc1CN(C)CCOC(C)=O n1(CC(=O)NC2CCC(NC(c3csnn3)=O)C2)cc(Br)ccc1=O C1(NC(C(C2CCOC2)NC(C)=O)=O)CCCCN(Cc2nccs2)C1 N1(C(c2c(CC)ncs2)=O)CCC2(C1)CN(C(c1cc(C(C)=O)on1)=O)CCO2 Cc1cc(OCCC(=O)N(C)CC2CCN(C(=O)C(C)CC(C)C)C2)cc(C)c1 C=CC(C)CC(=O)N1CC(C)(NC(CCC(O)C2CCCC2)=O)C1 c1(C(N2CC(C)C(CNC(C3SCCS3)=O)CC2)=O)ccc(F)c(S(N)(=O)=O)c1 C(=O)(C(C1=NOCC1)N(C)Cc1ccncc1)NCCCC Cc1cccc(CC(=O)NCCC2(NC(C3CCCOC3)=O)CCC2)c1Cl c1(NC(C2CC2C(=O)Nc2cccc(Br)c2[N+](=O)[O-])=O)cc(Br)ncc1[N+](=O)[O-] C(=O)(C(C)CCCC(C)C)N(CCNC(c1nc(C(C)OC)oc1)=O)C(C)C S(=O)(=O)(c1cccc(Cl)c1F)N.N1(C(=O)CCCCCl)CCc2c(cccc2F)C1 c1(CNC2CC(O)C(O)CC2)c[nH]c2c(OC(F)(F)F)cc(Cl)cc12 C1(CC(=O)NC2CC(CCNC(=O)CC3CCC=CCC3)C2)CC(O)C12CCC2 N1(C(C2(COC)CCCC2)=O)CCCCC(NC(=O)C(c2ccc(Cl)cc2)O)C1 C1(C)(C(=O)NC(c2cc[nH]n2)COC)CCN(Cc2ccccc2)C1 n1(CC(=O)OC)cc(-c2ccc(C(N3CCC(N(C)C)C3)=O)o2)nn1 N1(C(c2c(C)nsc2Br)=O)CCC(CNC(c2c[nH]c(=N)o2)=O)C(C)C1 c1(SC)nc(NC2C3CC2CN(C(=O)CC2CCCCO2)C3)cc(Cl)n1 c1(OC)ccc(C(N2CCC(NC(c3ccc(C(N)=O)[nH]3)=O)C2C)=O)c(OC)c1 c1(CC)cccc(C)c1C(N1CCC(CNCCCN(C)CCOC)C1)=O c1(CCC(=O)N(CC(C)NC(C2(C)ON=C(C)C2)=O)C)cccc([N+](=O)[O-])c1 N1(C(=O)Nc2ccc(Oc3cc(C)cc(C)c3)cc2)CCC2(CC1)CNC(=O)O2 C1(O)(CN(C)C(C2CC(N(C)C)C2)=O)CCN(C(=O)Cc2cn[nH]c2)C1 n1(CC(=O)NCCC(C)N(C)C(C2C(F)(F)C23CC3)=O)nc(Cl)ccc1=O N1(C(C(CC)CC)=O)CCCC2(CCN(C(=O)C(C)n3ccnn3)C2)C1 C1(F)(CNC(c2cncc(C)n2)=O)CCCN(C(=O)C2=CCCCC2)C1 C1(C(N2CC(NC(CCC(C)C)=O)C(F)C2)=O)CCOC2(CCCCC2)C1 C1(NC(c2nn(C)c(O)c2)=O)CC2CCC(C1)N2C(c1cncc(CO)c1)=O C1(CN(C(C(C2CC2)OCC)=O)C)CCCCN1C(=O)CCc1ccncn1 C(=O)(C(F)Cc1ccccc1)N1CC(CC(=O)NC2CCN2C2CCCC2)C1 C(=O)(C1=COCCC1)NC(c1cc(C(C)(C)C)ccn1)C c1(OC)c[nH]nc1C(=O)NC(C1(O)CN(C(=O)CN(C(=O)C(C)C)C)C1)C C12(NC(c3nc(C)n(C)c3)=O)CCCC1N(C(=O)CCCOC(C)(C)C)CC2 N1(C(c2cc(C)[nH]c2C)=O)CCC(CNC(C2(C)CCN(C)C2)=O)CC1C N1(C(CCN(CC(C(C)C)C)C)=O)CC(NC(c2nsnc2O)=O)C(N=[N+]=[N-])C1 C=CC(C)CC(=O)NC(C)(CNC(=O)CCCOc1ccc(F)cc1)C1CC1 C1(C(N2CC(CC)N(C(=O)CCc3nccn3C)CC2)=O)OCCOC12CCC2 n1(C2(C(=O)NCC3C(CNC(CCCSC)=O)C3)CC2)cnc2ccccc12 C1(CNC(COCC(=O)NC)=O)CCN(C(=O)CC2CCCCC2(F)F)C12CC2 C(CN=C(NCc1cnc(-c2ccccc2)o1)NC1(CF)CC1)OCC=C c1(C(N2CC(C)(CNC(C34CC(C)C3C4)=O)OCC2)=O)ccc(C#N)c(C)n1 N1(CC)CCC(NC(=O)CN(c2ccccc2)C(C2CC(C)(F)C2)=O)CC1 Cc1nccnc1C(=O)NC1CC(NC(c2ccnc(OC3CCOC3)c2)=O)C1 CC(CC(=O)NCCC1CC(NC(=O)Cn2cnc([N+](=O)[O-])n2)C1)C(F)F N1(C(c2ccc(OC)s2)=O)CCCC(C(=O)Nc2ccnc(Cl)c2)C1 c1(CC(N2CCC3CC2CN3C(c2ccsc2)=O)=O)ccc2nonc2c1 c1(C(N2CC(SC)C(NC(=O)C3=C(Cl)CCC3)C2)=O)ccc2c(c1)S(=O)(=O)NC2 C1(NC(c2nn(CC)c(C)c2)=O)CCCC(C(N2CCOC(CCO)C2)=O)CC1 N1(CC(=O)NCC=C)CCN(C(=O)CN2CCCC2)CC1.C123CC(C1)(C2)NC3=O c1(C(N2CC(C)C(NC(=O)CSCC(N)=O)C2)=O)cnc2cccnc2c1 N1(C(c2cncc(N)c2)=O)CCCC(CNC(=O)C(F)OC(F)(F)F)CC1 CC(CCCc1ccccc1)C(=O)NC1(c2nc[nH]n2)CCCC1 C1(C(N2C(C)(CC(=O)NCCCC#C)CC2)=O)(C(N)=O)CCCCC1 N1(C(c2c(OC)ccnc2)=O)CCOCC(NC(=O)C(C(C)C)C2CCC2)C1 C(CC(C(C)(C)C)NC(c1ccc(C#N)o1)=O)N(C)C(c1cccc(F)c1Cl)=O N1(C(c2n(CC)ccn2)=O)CCCC2CN(C(=O)CSCc3cscn3)CCC12 N1(C(=O)CSCCNc2nccc(COC)n2)CCC(Cc2ccccc2)CC1 CC1COCCN(C(C23COC(C2)C(NC(C2CC2Cl)=O)C3)=O)C1 Cc1ccc(C(CNC(C2CC=CCC2)=O)NC(c2cncc(Cl)c2)=O)cc1 c1(NC(C2CC(NCc3cc(Cl)ccc3Cl)C2)=O)cc(F)c(Cl)cc1F N1(c2c(C)cncn2)CC2CCC(NC(C3CC3c3c(C)nn(C)c3C)=O)CC2C1 CC(C(=O)N(C(C)CNC(=O)CCC1CCC(O)CC1)C)C(C)(C)C C1(CNC(=O)CCCC2(NC(=O)C(C3CCCCC3)O)CCC2)C2CCCCC12 c1(C(C)=O)cccc(C(=O)NCC2(CCNC(c3cnsn3)=O)CC2)c1C(C)C Cc1cnc(C(=O)NC(C)(CO)C(=O)N(CCC(C)(C)O)C)c(F)c1 CCCCC(C)(F)C(=O)NCc1ccc(C(=O)NCC2CC23CC3(F)F)nc1 Cc1cc(Cl)cnc1-c1cn(CC2CCCN2C(c2ccns2)=O)nn1 CCC(CO)(C(=O)NC1(CCCC(=O)NC2CC2CN(C)C)CCC1)OC C1(C(N2CCC(CCC(=O)NC(C)Cc3nc[nH]n3)C2)=O)CC(=O)C1(C)C c1(C(N(CCCNC(C(=Cc2ccccc2)CC)=O)CC)=O)cc2cscc2s1 CC1CN(C(c2cnc3cccnc3c2)=O)CC(C)N(C(c2ccncn2)=O)C1 N1(C(c2cc(C)n(C)c2)=O)CC2CCC1CN2C(c1ccc2snnc2c1)=O C12(CC(=O)NOCCC(F)(F)F)CCCC1CN(C(c1ccccc1)=O)C2 CCC(C)CC(=O)N1CC(NC(c2ccc(C3CCCCC3)s2)=O)C(CC)C1 Cc1cc(C(=O)NCCC2CC(NC(c3csc(C#N)c3)=O)C2)c(C)cn1 N1(C(C(C)OCC)=O)CC(NC(c2nc3cccnc3s2)=O)C2(CCC2)C1 C1(C(N2CCCC(NC(c3cccc(CO)n3)=O)C2)=O)CCCC2(CCC2)C1 Cc1cc(C)nc(-c2cn(C(C)CNC(C3(c4ccon4)CCC3)=O)nn2)n1 N1(C(C2(C3N(C(c4cccc(CC)n4)=O)CCC3)CC2)=O)CCC(C)(CC)CC1 N1(C(c2cc[nH]c2)=O)CCN(C(=O)C(O)Cc2cccc(Cl)c2)C2CCC12 c1(CCC)ccc(C(N2CC3CC2C3NC(C2(C3CC3)CC2)=O)=O)cc1N C=C(Cl)CC(C(=O)N(C)Cc1ncco1)NC(=O)C(C)c1ccco1 C1(CNC(c2c(C)ncnc2O)=O)C2CCCC1N(C(C1CC(C(C)C)C1)=O)C2 C(=O)(CC(CC)C(C)(C)C)NC1(CCC(=O)N(C(CCC)C2CC2)CC)CCCC1 C1(n2c(-c3cnn(CCO)c3)nc(C(C)C)n2)CCC(F)(F)CC1 C1(C)(C(=O)NCC2(CC)CC2)CCCN(C(c2ccc(I)cc2)=O)C1 C1(F)(C(=O)NC2CC(C)(NC(=O)CCN3CCOC3=O)C2)C2CCCCC12 c1(C(N2CC3C(NC(C(CCCC)C)=O)(C3)C2)=O)cc(O)cc([N+](=O)[O-])c1 c1(NC(CN(C)CCC2CCN(C(=O)CC(F)F)C2)=O)ccccc1 c1(C(=O)NCCCc2cn[nH]c2)ccc(CNC(c2ccccn2)=O)cc1 C1(C2CC2)(CNC(c2cc(CC(C)C)on2)=O)CCN(C(C2CNC(=O)C2)=O)C1 c1(C(=O)OC)cc(C(N2CCC2)=O)cc(F)c1.C12CCCCC1n1cc(nn1)C2 Cc1cc(Cl)cc(Cl)c1CN1CCN(C(=O)C(CN)N(C)C)CC1 C1(N(C)C)(CC)CCN(C(C2C3CC2N(C(=O)C(C)=C2CCCC2)C3)=O)C1 CC1(C)CCCC(O)(C(=O)NC2CCC2NC(c2cccc3nccn23)=O)CC1 c1(CC)ccc(CNC2CC(C(=O)Oc3cc(C(F)(F)F)ccc3Br)C2)cc1F c1(C(N2CCC(CNC(C3(N(C)C)CCC3)=O)C23CC3)=O)cc2occc2n1C c1(C(=O)NC2CC(CCNC(C(C)(C)SC)=O)C2)n[nH]c(C)c1Br C1(NC(c2c(C)csc2)=O)CCN(C(c2cc(Cl)ns2)=O)CCC1CO C(C(=O)NCC1C=CCN1C(c1cn(CC(F)(F)F)cn1)=O)(C(C)(C)C)SC c1(OC)ccc2c(c1)CC(C(=O)NC(C1CCCCC1)CNC(=O)CC1CC1)O2 c1(C(=O)NCC(=C)CCNC(c2ccoc2C)=O)coc2ccc(C(C)C)cc12 c1(CNC2(CCCC(N3CCC(c4c(N)c[nH]n4)C3)=O)CCC2)ccc(F)cc1 Cc1noc(C)c1CCN(C(=O)CCN(C)C)C1CC1.C12CN(C1)C(=O)O2 N1(C(Cc2ncc(C)s2)=O)CC2C3CCC(C2C1)N(CC1CCOC(C)C1)C3 Cc1ccc(C(=O)NCCNC(=O)CC(=O)OC(C)(C)C)c2cccnc12 c1(C(N2CC(CNC(C3(OC)CCC3)=O)(OC)C2)=O)cn(C(C)(C)C)nc1C Nc1ccc(C(N2CC3CC2C3NC(c2cnn(CCF)c2)=O)=O)c(Cl)c1 N1(c2nc(=N)nc(N(C)Cc3cccnc3)[nH]2)CCC(C2CCN(C)C2)CC1 C1(CC(=O)NC(C#C)C2CCC2)CCN(C(=O)C(O)C=CCCC)CC1 C12(CNC(c3n(C(C)C)ccc3)=O)CC(NC(C34CC(C)C3C4)=O)(CO1)C2 Cc1cc(=O)ccn1CC(=O)N(C)CC1(O)CCN(C(=O)Cn2ccnn2)C1 c1(N2CCC(NC(C(C)NS(CC)(=O)=O)=O)C23CCC3)ncnc2c1nnn2C C1(CC)CCCN(C(=O)C2=C(Cl)CCC2)C1C(=O)NCCc1ccnn1C N1(C(C=CC(C)NC(c2ccc(C(C)C)o2)=O)=O)CCN2C(=O)OCC2C1 C(C(C)(C)CC(=O)NCC(c1ccncc1)C)NC(CC1C(C)OCC1)=O C1(NC(c2ccc(C)nc2O)=O)CN(C(=O)C(C)(C)CF)Cc2nccn2C1 NC(=O)C(F)CC(N)C(=O)NC(c1ccc(Br)cc1)c1cccnc1 N1(C(c2cc(C)[nH]n2)=O)CC(C)(C)CC1CC(=O)NOCc1ccccc1 c1(C(=O)NCCNC(C(C)NSS(C)(=O)=O)=O)ccc(C2(C(F)(F)F)N=N2)cc1 N1(C(c2c(CC)nn[nH]2)=O)CC(NC(=O)C(c2ccccc2)C)C(SC)C1 c1(NC23CCC(CNC(=O)OC(C)(C)C)(OC2)C3)c[nH]c2ccc(Br)cc12 N1(C(CC(C)N(C(=O)C(Cl)=CCl)CC)=O)CCN(C(=O)Cn2cnnc2O)CC1 Cc1ccnc(N(CC(C)C)C(c2ccc(C(F)C(F)F)cc2)=O)c1 c1(CC)ccc(CNC(=O)C(C2(O)CN(C(=O)CCOCC(C)(C)C)C2)F)o1 c1(C(c2cn(C3CCN(Cc4conc4C4CC4)C3)nn2)O)cccc(Cl)c1 C[S+](C)CCC(O)C(=O)NCC1(C)CCN(C(=O)CC23CCCC2C3)CC1 C1(C(N2CC(NC(c3c(C(=O)OC)cccn3)=O)C2)=O)CCC2C1C2(F)F n1(CC)cc(CC(=O)NCC2CC(NC(c3cnoc3C3CC3)=O)C2)cn1 C=CC1OCCC1CNCc1nc(C)cs1 CC(C)CC(O)C(=O)NCCCCC1CN(C(=O)C(C(C)C)c2cccnc2)C1 c1(C(=O)NC2C(C(N(C(CC)C)C)=O)OCC2)ncccc1Cl CCCC(C#N)C(=O)N1CC(CNC(c2cnc(C3CC3)nc2)=O)C(O)C1 CCC(CC)C(C)C(=O)N(C(C)C(=O)N(C)CC1CCCCC1O)C CC1(C)CCCOC1C(=O)NCc1csc(CNC(C23CCC(CC2)C3)=O)n1 CC1(C#N)CCCN(C(=O)C(C)(C2CCC2)NC(c2ns[nH]c2=O)=O)C1 c1(C(=O)NCC(C(=O)OCC)CC)cc2cc(C)cc(C)c2[nH]1 CC1CC=C(C(=O)NCC(O)CCNC(=O)C=CC(F)(F)F)CC1 C1(C2CCC2)(CNC(CN2C(C)CC2)=O)CCN(C(=O)Cc2nc[nH]n2)CC1 N1(C(CCC)=O)CCCC(C(N2CCC(N(C)C(c3cc(Cl)n(C)n3)=O)C2)=O)C1 CC(C)C(CNC(c1csc(O)n1)=O)NC(=O)C=CCn1cncn1 N1(C(c2ccc(C(F)(F)C(F)F)cn2)=O)CC2CC1CN2Cc1ccccc1 c1(CNC2C(C(N(C(C)C)CCO)=O)C2)cc2ccccc2nc1O N1(C(CC(C)N(C(CSCC)=O)C)=O)CC(C)C(C)C1C Cc1cc2c(C(=O)NCC(C)N(C)C(C3CCC4(CCC4)C3)=O)cccc2o1 c1(C(=O)NCCC(C)NC(=O)C(C)Cc2ccco2)ccc(F)c2cnccc12 c1(C(=O)NCC2CN(C(c3c(C)onc3)=O)C2)cccnc1CC(C)C c1(CC#N)cccc(S(=O)(=O)N2CCCC3(CCO3)C2)c1 C1(F)(CNC(c2cccc(F)c2F)=O)CCCN(C(=O)C(C2CCOCC2)O)C1 C(=O)(CCCCC(C)(C)C)NC1CN(C(CC(C)CF)=O)CC1c1ccccc1 C12(NC(CC3(C)CC3(Cl)Cl)=O)CCC(C1)N(C(c1ccc(O)cc1)=O)C2 c1(C(CC)(C)C)ccc(CNC23CC4CC2C3C4)cc1 C1(NC(C2CCC(C(=O)O)C2)=O)CCC(NC(C2CC(n3ccnn3)C2)=O)CC1 c1(C(N2CC(O)CCC(NC(C(C)(C)C(F)F)=O)C2)=O)cn2cccc(Cl)c2n1 C1(NC(C2CCSC2)=O)CN(C(C2CS(=O)(=O)C2)=O)CC2(CC2)C1 C1(C)(C(=O)NC(CCC)CCCNC(c2ccc(C)o2)=O)CCS(=O)(=O)CC1 C1(CNC(C(C)CF)=O)CC2(C1)CN(C(c1cccnc1)=O)C2 c1(C(N2C3CN(C(=O)CC4CCCO4)CC2CC3)=O)ccc2c(c1)OC(F)(F)O2 CCC(CCNC(=O)CCCn1cc(C2CC2COC)nn1)C1CCC1 C1(C(=O)NC2C(NC(Cn3nnc(C)n3)=O)C2)CCc2ccccc2O1 N1(C(C(CC2CC2)OC)=O)CC(NC(=O)COc2cc(C)ccc2F)CC(C)C1 c1(C(=O)NC2CCC(N3CCCCC3)C2)cc(F)c(Br)cc1C(F)(F)F c1(CNCc2c(C(=O)OC)[nH]cc2Br)c(C)ccnc1C C(=O)(C1CCCc2n[nH]cc21)NCC1C(C)CCN1C(=O)CCc1cnoc1 c1(C(=O)NCC2(CNC(=O)C=CC3CCOCC3)CC2)cc2cc(O)ccc2[nH]1 c1(C(=O)NC(CNC(C2CCC(=O)N2C2CC2)=O)C2CC2)cc2cnccc2o1 CC1(C#CC(=O)N2CCOC3CN(C(=O)COCCF)CC23)CCCO1 CC1CC2CCC(C(=O)NC(C)CCCCNC(=O)CC3(O)CCOC3)CN2C1 c1(C(N2C(CC(=O)NCC(O)CO)CCC2)=O)ccc(O)nc1 c1(CN2CC(CC(N3C4CCC3COC4)=O)C2)c(Br)ccc(F)c1F c1(N(CC(=O)NC2CCN(C(C3CCSC3)=O)CC2O)C)ncnc2[nH]cnc12 N1(C(c2c(C)onc2)=O)C2CCC1C(CNC(=O)Cc1csc(Cl)c1)C2 Nc1cc(C(=O)NCC(CNC(=O)C(O)C2CCCC2)S(C)(=O)=O)cnc1Cl CCCCCCC(C)C(=O)NC1COCC1CNC(=O)CC1(SC)CCC1 c1(C(=O)NCCC(Cc2ccccc2)NC(COC)=O)cn2cccc(C)c2n1 c1(-c2n(-c3c(CC)cccc3)nc(CC(C)C)n2)ncc(F)cc1N c1(OC)cccc(C(=O)N(C)CCN(C(=O)C(C2CCCCC2)O)C)c1[N+](=O)[O-] CC1CCC(CNC(=O)CCSc2ccc(F)cc2)N(C(=O)C(F)=C2CCC2)C1 C1(CC(C)(C)C)CN(C(C2NC(=O)C3CCC23)=O)CCN1C(=O)CS(N)(=O)=O CCCC(CC)CC(=O)N1CCC(OC2CN(C(c3cnn(C)c3N)=O)C2)CC1 c1(SCCOC(C)(C)C)ccccc1OC(C1(OC(F)F)CC(F)C1)=O c1(C(C)C)cc(C(=O)NC(C2CN(CCOC3(CN(C)C)CC3)C2)=O)no1 c1(CNC(c2n(CCOCC)nnn2)(c2ccncc2)C)ncc(F)cc1F C1(NC(COc2ccn(C)n2)=O)CCCCC1C(=O)NCC(C)(C)C1CC1 Cc1cnccc1C(C)C(=O)NC1CCCCC1N(C)C(c1cccs1)=O C1(C(N2CCN(c3ncc(C)c(C)n3)C(C(C)C)C2)=O)CCOC2(CCCC2)C1 c12cc(cnc1C)NC2=O.c1(CC)ccc(Oc2ccc(C)nn2)cc1 n1(CCC(=O)NC(CC=C)CNC(c2c[nH]nc2C(C)C)=O)cnc(C)cc1=O C(=O)(CCCC(F)(F)C(F)(F)F)N1CC(NC(=O)CC(C)(C)CN(C)C)CC(C)C1 C12(NC(C3C(C)CCC3)=O)CC(CNC(c3cc(Br)c[nH]3)=O)(C1)OC2(C)C C12(C(=O)NC(C(=O)OCC)CCc3ccccc3)CCC(CC)(C1)OC2 Cc1cc(C#N)nc(NC23CCCC2CN(C(c2cn(C4CCC4)nn2)=O)C3)n1 c1(SC)ccc(S(=O)(=O)NC(C)(C)C(=O)NC2CN(C(=O)C(C)C)CC2(C)C)o1 c1(CC(OCC)OCC)cn(CCNC(=O)CCn2ccnn2)nn1 c1(C(=O)NCC2CCC2=O)cncc(-n2cc(-c3cc[nH]n3)nn2)c1 c1(C(=O)OC)ccc(N2CC(CCCCNC(c3cnc[nH]3)=O)C2)nc1 c1(OC)ccc2c(c1)C(CCNC(C1CCCO1)Cc1cccc(C)c1)=CC2 N1(C(CN(c2ccccn2)C)=O)CCC(O)(CCNC(=O)C(C)(C)N(C)C)C1 CCCN=C(NCC1CCCCN1COC)N1CCC(F)(c2ccccc2)CC1 c1(NC(c2n(C(CC)C)nnn2)c2ccc(C(F)F)o2)ccc2nncn2c1 C#CCC(O)C(=O)NC1CC(NC(=O)C(F)(F)c2ccsc2Cl)C1 N1(C(c2cc(OC)n(C)n2)=O)CCOCCC1C(=O)NC1C(C)C1C C(=O)(C#CC1CCC1)NC1C(CNC(c2c(COC)cccc2)=O)CCCC1 C1(C(N2CC3C(NC(C=C(COC)C)=O)(C3)C2)=O)CC2(CC(C)=NO2)C1 N1(CC(F)(F)F)CC2CCC1CN(c1ncc3cn[nH]c3n1)C2.c1ccncn1 O=C(C(C1=CCCCCC1)N1CCSCC1C1CC1)NCCO N1(CC(=O)N(CC(C)NC(=O)CSC(F)F)CC)C(=O)c2ccccc2S1(=O)=O c1(OC)c(C(N2CC=CC(NC(=O)CC(C)N(C)C)C2)=O)[nH]c2ccccc12 [N-]=[N+]=NC1CN(C(C2(CO)COC2)=O)CC1NC(C1CN2CCCC2CO1)=O c1(C(N2CC(NC(c3ccc(OC(C)C)cn3)=O)C2)=O)cc2ccsc2n1C c1(C(N=c2nc(C)[nH]o2)=O)cc(Br)c2c(c1)CCO2.c12ccc(cc1)CNC2=O c1(OC)ccc(CN2CCNCC2C(=O)NCc2ccc(Br)cc2)c(Br)n1 N1(C(CC=CCC)=O)CC2CCC(C1)N2C(=O)Cc1nnc(S)n1C c1(COC)c(C(N2CC(CC(C)NC(C)=O)C2)=O)oc2ccccc12 N1(C(C2(SC)CC2)=O)CCCN(C(C2CC(C)N(C(=O)OC(C)(C)C)C2)=O)CC1 N(C(=NCCC1CCN(CC)CC1)NC(c1ccccc1)C)CC1(SC)CC1 C12(CNC(CC(=O)OCC)=O)CCC(C1)N(C(=O)C(C)OC1CCCCCC1)C2 C1(NC(C2CC(N(C)C)C2)=O)C2CC(O)C1N(C(=O)C=CCN1CCOCC1)C2 c1(OCCCC(=O)N(CCNC(C2C(CCOC)C2)=O)CC)cccc(C)c1C c1(NC(c2ccnc(C)n2)=O)ccc(NC(c2scnc2C)=O)c(F)c1 c1(SC)cc(NC(c2cc(-c3ccn(C(C)C)n3)ccn2)=O)ccn1 C(CC(C(C)(C)C)NC(=O)C1=C(Cl)CC1)N(C(CCCN(C(C)C)C)=O)C C1(NC(COC(CC)(C)C)=O)CN(C(=O)C2=CC(C)(C)C2)CCC1C(F)(F)F C1(C(C)(F)F)(C(N(C)CCNC(C2CCCS2)=O)=O)CCOCC1 C1(C)(CNC(C2(C=C)CCC2)=O)CCN(C(=O)CN(CC)CC)C1 N1(C(C=CC=CC)=O)CCCCC1C1CCN(C(=O)C(C)n2cnnn2)CC1 N1(C(CN(C)C)=O)CCN(C(=O)C=CSCc2ccco2)CC(C)(F)C1 C#CC1(CNC(=O)C(CC(C)C)NC(=O)CCCSCCC)CCOCC1 c1(C(=O)NCC2(C(=O)O)C(C)(C)C2)cc2occc2[nH]1 C1(NC(C(C)N(C(CC)=O)CCC2CN(C)C2)=O)CN(C(=O)C(C)(C)C)CCO1 C1(CC)CCCCC1C(=O)NC(C)(C)CNC(=O)COC(F)(F)C(F)(F)F Cc1cc(C(N2CC3(NC(c4cc(C(C)C)[nH]n4)=O)CCC2C3)=O)cc(C)c1N C1(CNC(c2c(CC)ccs2)=O)CCC2(CN(C(c3[nH]ncc3C#N)=O)C2)O1 C1(NC(C=CC(=O)N(C)C)=O)(CF)CCN(C(C2COC(=O)O2)=O)C1 CN1CC(O)CCC1C(=O)NCC1CC(n2cc(COc3ccccc3)nn2)C1 N1(C(c2c(C)nn[nH]2)=O)CCCCC1CNC(c1ccc(Br)nc1)=O N1(C(c2cc(C)sc2)=O)CCC(F)C(NC(c2nc(C)oc2C)=O)C1 c1(C(CNC(=O)C(C)(O)C2CCC2)NC(C2(C)CC2(F)F)=O)ccccc1F c1(C(=O)NC(CC(=O)NCC(=O)NCC)C)nnn(C)c1N Cc1ccc(C(=O)NCCCC2CCCN2C(C23COCC2C3(F)F)=O)nc1C C(=O)(CCCN(C(=O)CC1CC1CNC(=O)Cc1cscn1)C)OC C(=O)(C1COc2ccccc21)NC(C(C)NC(c1cc(OC)c(O)nc1)=O)CO C=CCCC(C(=O)NC(C)(C)C)N1CCC(CO)C(C)C1 CCC(S(=O)(=O)NC(C1CCC(N)CC1)=O)c1ccccc1 C1(C(=O)NC(COC)C)CN(C(C2CCCCC2C(C)(C)C)=O)CC1(F)F C(=O)(C1=C(C)CCCC1)N(C1CCN(C(c2cc(C(N)=O)[nH]n2)=O)C1)CC C12(CC1(F)F)C(=O)N2.C1(C(=O)NCCC2CN(C(C)=O)C2)(OC(C)C)CCC1 N1(C(c2n(CC)ccn2)=O)C2CCCC1CC(N=c1[nH]c(Cl)ncc1C1CC1)C2 N1(C(C=Cc2cn(C)nc2)=O)CC2CCCN(C(C34COC(CCO3)C4)=O)C2C1 N1(Cc2ncc(C3CC3)s2)CCOC2(CCCNC2)C1 c1(CSCC(=O)N(CC)CC)ccc(O)c(C(N2CCOC(CC(N)=O)C2)=O)c1 c1(-c2cn(CC3CCC(NC(c4n(CC)ncc4)=O)C3)nn2)cc(C)cc(F)c1 c1(C(=O)NCCC2CCN(C(C3CCNC3=O)=O)C2)cccc2c(O)nncc12 c1(CC(N2C(CNCc3cc(OC)ncc3)CCC2)=O)cccc(OC)c1OC N1(C(C2=CCN(C)C2)=O)CCC2(CCN(C(=O)Cc3ccc(F)cc3)C2)C1 CC(CC(=O)NC1(CNC(c2ccccc2C2CC2)=O)CC1)C(F)F C1(CN(C)C(=O)C2CC2)CCN(C(C2CC(N(C)C)C2)=O)CC1 C(C)(CC(C)NC(c1csc(-c2ccncc2)n1)=O)NC(C(C)SC)=O N1(c2nc(COC)nc(C)c2)CC2CCC1C1CN(C(C3CC3(C)Br)=O)CC21 C1(C)(CNC(C2CCN(C)C2)=O)CCCN(C(=O)CCCNC(=O)C(C)(C)C)C1 N1(C(c2c(C)oc(Cl)n2)=O)CCC(C)(C)C(CNC(C2CCCN2C)=O)C1 C1(NC(C=CC(CC)C)=O)CCN(C(=O)Cn2nc(C(F)(F)F)cc2C)CC1O CC(C)(CCNC(=O)CSc1nc[nH]n1)C(=O)NCC1CCC(CO)O1 C12(NC(C(CCSC)O)=O)CCCC(NC(=O)CCc3ccc(N)cn3)(C1)C2 c1(C(N2C(C)CC(CNC(CN(C)CC)=O)C2)=O)cc(Br)cc2c1OCO2 C(=O)(C1=CCCCC1C)N(CCOC)CCNC(=O)Cc1ccc(OC)cc1 C(CCCl)(CCCl)(N(C1CCSCC1)C)Cc1ccccc1 N1(C(COCC=C)=O)CCC(C)C(CNC(=O)Cn2cccn2)C1 CC(C)CC(c1ccccc1)NC(=O)N(C(C1CCCO1)=O)CC1CCCO1 C(=O)(C(CC1CCCC1)NC(=O)CC1CCCC1)NCC(=O)NC1CCCCC1 CC1(C)C(=O)CC1(P(C)(C)=O)CCNC(C1CCC2CNCC2O1)=O C(=O)(C#CC1CCOC1)N(CC)CC1CCCCN1C(c1ccsc1)=O c1(OCC)ccc(=NC(=O)CC2CCCN2Cc2cccc(Br)n2)[nH]n1 N1(c2nc(=N)nc(N3CCCCC(C(C)C)C3)[nH]2)CCOC2COCC2C1 c1(C(=O)NC2C(OC)CN(C(C3N(CC)C(=O)CC3)=O)C2)cnc2[nH]ccc2n1 C=C(C)CC(C)C(=O)NCC(CC(C)C)NC(c1ccc(OC)c(N)c1)=O CCS(=O)(=O)c1ccc(CN2CCCC(CO)(NC(=O)CCC3CC3)C2)cc1 N1(C(Cc2nc(NC=O)sc2)=O)CCN(C(=O)Cn2nnc(=O)[nH]2)C2CC12 c1(C(=O)NCCC2CCCCN2C(=O)CN2CC=CC2)csc2ccncc12 c1(C(=O)NCC2(CNC(CCC=CC)=O)CCCC2)ccc2ncccc2c1F Cc1nccn1CC(=O)NCC(C)(C)OCC(=O)NCC(c1cnn(C)c1)C C(C(C)CC(=O)N1CCCCC1C(=O)N(CCS(C)(=O)=O)C)OC N1(C(C(CC)CN(C)C)=O)CCC(NC(c2cc(C(N)=O)[nH]n2)=O)CC(C)(C)C1 S(=O)(=O)(c1ccc(C(=O)NCC2CCCN(C(=O)CC3C=CCC3)CC2)o1)NC C1(N(C(C2C(=C)C2)=O)CC)CCCN(C(c2cc(OC)cc(C)c2)=O)CC1 CC(C)(CCN=c1ncc2ccccc2[nH]1)NC(C1(c2ccc(F)cc2)CC1)=O CCC1=C(C(=O)NCCCOCCNC(c2c(C)ncn2O)=O)CCCO1 N1(C(CCCC(=O)NCC)=O)C2CCC1CN(C(=O)C(C)C(O)CC)C2 C1(C(=O)NC(c2ncc(C)o2)C)C(C)OCCN1C(=O)C(C)N=[N+]=[N-] N1(CC)OCC(NC(=O)CC2(C)CCN(C(C3CCC3C#N)=O)C2)C1=O CC1COCC(CC(=O)NC(C(=O)NCCC2CC=CC2)C(C)O)O1 N1(C(CCC(=O)N(CCC)CCC)=O)CCC(C)C(NC(=O)CC(C)(C)SC)C1 c1(C(=O)NC2C(CNC(=O)CNC(=O)C3CC3)COC2)cccc(O)c1 c1(C(N(C2CN(C(C(C)OCC#C)=O)CC2(C)C)C)=O)cccc2nn(C)nc12 N1(CC(CC(C)C)N(C)C)CCC23CCC(CC12)C3(C)C c1(C(=O)NCC2(C)N(C(C(C=C)O)=O)CC(F)(F)C2)ccc2cnc(C)n2c1 c1(CC)onc(C(=O)NCC(C)C(=O)NC(C)C(C)(C)C#N)c1C C1(NC(CC(CCC)C)=O)CN(C(=O)CCc2cc(C)[nH]n2)Cc2ccnn2C1 C(=O)(C(C)(C)CC(=O)NC(C)(C)CNC(=O)CCN1CCC(F)C1)OC N1(C(CN(C(=O)OC)C)=O)CCC(NC(=O)C(C)CC(F)(F)F)C12CCC2 C=CC(C)CC(=O)NCCC1(F)CC(NC(=O)CCCNc2cccnc2)C1 S(=O)(=O)(c1cnc(Cl)nc1)N1C(C(N2CC3CCC2C3)=O)CC2CC21 C1(CNC(c2ccc(F)c(CO)c2)=O)CCCN(C(C2CC2C(F)F)=O)CC1 c1(C(=O)NCC(C)(C)OCCN(C)C)cncc2c1CCC2.N12CC(C1)C2=O c1(C(N2CC(CNC(c3cc(CCC)nn3C)=O)(OC)C2)=O)cc(C)c(O)nn1 C1(O)(CN(C(C=Cc2ccc(C)s2)=O)C)CCCN(C(C2(C)C=CCCC2)=O)C1 c1(C(=O)NC(CNC(c2cc(C)no2)=O)(C)C)ccc2cc(F)ccc2n1 C1(C(=O)NC2CC(C#C)C2)CCCCC1C1CC1 Cc1ccc2c(c1)CCC(C(=O)OCc1cn(C(c3ccccc3)(C)C)nn1)O2 N1(C(c2ccc(C#C)c(Cl)c2)=O)CCOC2(C1)CN(C(c1cc(O)n(C)n1)=O)C2 N1(C(C23CC(OC)C2C3)=O)CCC(N(C)C(c2cc(C(C)(C)C)n[nH]2)=O)CC1 CCC(C)CC(=O)NCC1(c2ccccc2)CC(NC(=O)CCN2CCC2)C1 C(=O)(C1Cc2ccccc21)NCC1CN(C(c2ccnc(C)n2)=O)CC1O c1(C(=O)NCCCC(C)NC(c2ccncc2)=O)cccc(C2(F)CC2(F)F)c1 c1(OC)cc(C(N2CCC(O)C(NC(C3CCCN3C=O)=O)C2)=O)ccc1C Nc1cc(Br)ccc1C(=O)NCC1CN(C(=O)C(O)C(F)F)C1 C1(NC(c2ccc(Br)cc2)=O)CN(C(=O)Cc2cnccn2)CCC12CCC2 N1(C(CC(=C)Br)=O)CC(CNC(c2ccc(OC)nn2)=O)CC12CCC2 C(CN=c1nc(N(C)CCF)c2c([nH]1)CSC2)c1ccc(C)c(F)c1 C1(CC(C)NC(c2cccnc2)=O)CCN(c2ccnc(C3CCC3)n2)CC1 C1(C2C(NC(C3CC(=C)C3)=O)CCO2)CCN(C(c2cc(O)cs2)=O)CC1 C(=O)(C1SCc2cccnc21)N1CC(C(=O)NCC2(CO)CCC2)C1 c1(OC)cc(C(=O)NC(C(C)NC(C2CC3CC2C3)=O)C(C)C)ccc1Cl N1(CCC)CCCCC1C(N1CCC(F)(CNC(c2coc(C)n2)=O)C1)=O C(=O)(CCC(=O)NC)N(C1CCCN(C(=O)C=CCN2CCCC2)C1)CC c1(C(C(=O)NC2(CF)CC2)NC(CS(CC)=O)=O)c(C)cccc1Br C12(C(N(CC(CC)(O)CC)C)=O)COCC1CN(C(C1CCCC(C#N)C1)=O)C2 C(=O)(C(C(C)CC)NC(C12CCCC1CCC2)=O)NC N1(C(COCCOC)=O)CCN(C(CNC(=O)NC2(C#N)CC2(C)C)C(F)F)CC1 C1(C(C)NC(C(CC)OC)=O)CCN(C(=O)C(C)(C)COc2ccccc2)CC1 Cc1cc(Cl)ccc1C(=O)Nc1cc(-c2ccccc2NS(C)(=O)=O)ccn1 c1(C(=O)NCC(C)(C2CC2)NC(=O)Cn2nccn2)cc(F)ccc1Cl C(=O)(C(F)C(C)(C)O)N(C)CC1CCN(C(CC(=C)Br)=O)CC1 C1(C(C)(C)C)(CNC(C2(CC=C)CCC2)=O)CCN(C(c2ccc(F)cn2)=O)C1 c1(NC(C2CCC(C(C)C)N2C(=O)C=CCF)=O)cc(F)c(O)cc1C n1(CC(=O)NC2C(NC(CC3(C)CC(F)(F)C3)=O)C2)ccc(O)nc1=O Fc1ccc2c(c1)C(c1nc(-c3cccc(Cl)c3)nn1CCCn1ccnc1)C2 n1(C2(C(N(CCCNC(C3CC(O)C3)=O)C3CC3)=O)CC2)cc(Br)cn1 c1(C(=O)NC(C(=O)N(C)CCc2ncon2)C2CCCO2)ncccc1O C(=O)(C(C(C)(C)C)NC(N)=O)NCC(C)NC(C(C)CC1CCCC1)=O C(=O)(C1CCCc2cncn21)N1CCCC2(CN(C(C3C(=C)C3)=O)C2)C1 N1(C(C2(C=C)CCOCC2)=O)CC(NC(C2OCCC2C)=O)C(C2CC2)C1 c1(C(N2CCCN(C(C3CCCN3C3CC3)=O)CCC2)=O)ncc2ccccn12 O=C1CCN(CCC2OCCO2)C(=O)N1CC1CC1c1ccco1 c1(OC)ccc(NC(=O)C(C2CCN(Cc3ccc[nH]3)CC2)C)c(C)c1 c1(C(=O)NC2C(NC(c3cc(C)c(O)cc3)=O)CC2)cc(P(C)(C)=O)cs1 C1(C(C(=O)NC2(CC(N)=O)CCC2)NC(c2cn[nH]c2)=O)CCCCC1 c1(C(=O)OCC(c2n(C(C)C)cnn2)=O)ccccc1N(S(C)(=O)=O)C c1(OC)ccccc1OCC(=O)NC1C=CCN(C(C2C=C2C)=O)C1 O=C(CCCCCF)NCC1C2CCC(C2)N1C(C1CCCOCC1)=O N1(C(C2CSCN2C(C2CC2C(F)F)=O)=O)CCCC2(CC(O)C2)C1 c1(CNCC2C(C(C)(C)C)OCC2)nc(F)ccc1F Cc1cccc2c(CC(=O)NC3CN(C(=O)CC(C)(C)C)CC3N=[N+]=[N-])c[nH]c12 c1(C(=O)NCCN(C(c2ccc(F)cn2)=O)CC)cccc(C)c1[N+](=O)[O-] c1(CN(C(=O)CNC(=O)CC2CC2)CC)cccnc1 C1(NC(C(C)NC(C2(OC)CCCC2)=O)=O)CCN2CCC1C2 Cc1c[nH]c2ncc(C(N3CC(NC(c4cc(C#N)c[nH]4)=O)C(C)(C)C3)=O)cc12 C1(NC(c2cnc(OC)c(Cl)c2)=O)CCN(C(c2sncc2C)=O)CC(C)(C)C1 Cc1ccc(OCCC(=O)NC2CCC2NC(=O)C(C)n2cncn2)c(C)c1 C#CCCCC(=O)NC(c1ccccc1Br)CNC(C1CC1C(C)(C)C)=O C1(CCO)CCC(N=c2nc(N3CCC4(CCNC4=O)CC3)c3sccc3[nH]2)C1 C1(NC(COC(C)=O)=O)CCC(N(C)C(c2sc(Cl)cc2Cl)=O)CC1 c1(OC)cc(CN2CC3C(C2)N3C(c2cccc(F)c2Br)=O)c(Cl)cn1 Cc1cccc2c(C(=O)N(CCNC(C3CC(n4ccnn4)C3)=O)C(C)C)coc12 Cc1ccc(Cl)c(C(=O)NCC2(O)CCN(C(=O)C(C)C3CCCC3)C2)c1 c1(C(=O)NC)cc([N+](=O)[O-])ccc1N1CC2(CN(C(=O)CC(C)SC)C2)C1 C1(CNC(CNC(C)=O)=O)CC(CNC(c2ccc(CNC(C)=O)o2)=O)CO1 N1(C(COCCCCC)=O)CCC(NC(c2cnc(C)cc2C)=O)CC1C1CC1 N1(c2n(CCC#C)c(-c3ccc(Br)c(C)c3)nn2)CCc2c(I)n[nH]c2C1 C1(C(=O)NC2CC(NC(CC3CC(CC)C3)=O)C2)C2CCC(C2)C1CO C1(CC#C)(C(N2CC(OCCNC(=O)CCc3cccnc3)C2)=O)CCCCO1 c1(N(C(=O)NCCN2CCCCC2)CCc2ccccn2)nsc2ccccc12 C(=O)(C#CC1CCOC1)N1CCC(C)(NC(c2c(C)ccc(CC)c2)=O)CC1 c1(C(N(CC(C)CNC(C2(c3ncco3)CCC2)=O)C)=O)nc2ccccc2[nH]1 C1(O)(C(C)NC(=O)Cn2cnnc2O)CCN(C(=O)CNC(=O)C(F)(F)F)C1 CCCC(CC(=O)NC(C)C(N)=O)NC(C1C=CCC1)=O N1(C(c2cc(C)[nH]n2)=O)CCC(C)(C)C1CNC(=O)CCN1CCCC1 Cc1cc(Br)ccc1CC(=O)Nc1c[nH]nc1C(=O)NCc1ccc[nH]1 CC1=CC(C)CN(C(=O)NCc2cccnc2N(C)C)C1 c1(OC)cc(C(N2CCOCC(CNC(c3nnc(S)n3C)=O)C2)=O)cc(F)c1 Cc1cccc2c1OCC2C(=O)NC(C)CNC(C1(CO)CC1)=O N1(C(C=COCC)=O)CCN(C2CCN(C(C34CCC3CC4)=O)CC2)CC1 C(=O)(C(C)(C)C(=C)C)C(C(COCC=C)N)=O.C1(N)CCCC(O)C1 C1(C(=O)NC2(CC(=O)OC)CC2)CCC(C)CN1C(=O)CC(C)F N1(C(CC=C)=O)C2CCC1CN(C(=O)C(O)C1CC1)C2 C1(C(N2C(CCCC)CCC2)=O)CC(C)(C)CCN1C(c1cc([N+](=O)[O-])c[nH]1)=O CC1CCCCC1(C)C(N1CCC(C(=O)Nc2ccccc2)C(C)C1)=O C1(C(=O)NC(CNC(Cc2cn(C)nc2)=O)(C)C2CC2)Cc2cc(Cl)ccc2O1 c1(C(N(C)CC2CN(C(C3CN4CCN3CC4)=O)C2)=O)ccc2c(c1)ncn2C C(=O)(CCCCC#N)NC(CCCNC(C1(F)C(C)OCC1)=O)C c1(CC)nc(N2CCCC(C(C)NC(c3cnc(O)cc3C)=O)C2)[nH]c(=N)n1 C12(NC(C3C(NC(c4cccc(C)c4F)=O)CCOC3)=O)CC3CC(CC1C3)C2 C1(C(N2CC(C(N)=O)(CNC(CCC3CC(C)C3)=O)C2)=O)CC(=O)CCO1 C(=O)(N=c1cnn(C2CCOC2)[nH]1)N(CCC#N)CC C(=O)(C(O)CC[S+](C)C)NCC(CC1CN(C(CC(C(C)C)O)=O)C1)(C)C c1(CNC(C2C(CNC(C3C(C(=O)OCC)C3)=O)CCC2)=O)ccc(O)c(C)c1 C1(C(=O)NCC(C(=O)OCC)C)CCN(C(=O)C(CO)C(C)(C)C)O1 Cc1nccc(C(=O)NCC2CCC(NC(c3ccnnc3Cl)=O)C2)n1 N1(C(c2cccnc2)=O)CC2CCC(C1)C2CNC(C12COCC1C2)=O C(CCCCC(=O)NCc1cccc(O)c1)N(C(=O)CC1CCC(=O)C1)C c1(C(=O)NC(C)C(C)(C)NC(=O)CC2C=CS(=O)(=O)C2)ccc2nn[nH]c2c1 c1(C(=O)NC(CNC(C(C(C)C)F)=O)C2CCC2)cc(F)cc(Cl)c1N CC(C)CC(CNC(=O)C(C)O)C(=O)NC(CN(C)C)CCO C1(C(N2CC(NC(=O)CC(=O)N(C)C)CC(C)(C)C2)=O)CC2OC(C)(C)OC2C1 c1(C(c2n(C(C)C)nnn2)NCCCn2ccnn2)cnc(N(C)C)cn1 C1(NC(CC2CC(C)N(C(=O)CC3CC4(CC4)CO3)C2)=O)CCOC2(CCC2)C1 N1(C(C(CC)(C)CNC(=O)CCc2cnccn2)=O)CCC(=C(F)F)CC1 Cc1c(C(N2CC(CNC(c3cncc(CO)c3)=O)C(C)C2)=O)ccn1CCO c1(C(N(CCCNC(C(C)C(F)F)=O)C2CC2)=O)n[nH]c2c1CC(F)(F)CC2 N1(C(C(CC#C)NC(=O)CCC(C)OCC)=O)CC2CC(O)CC1C2 c1(C(=O)NC2CCC(CNC(Cc3cc(C)ns3)=O)C2)ccc([N+](=O)[O-])[nH]1 N1(C(c2c(C)occ2)=O)CCCN(C(C2CCN(CCO)C(=O)C2)=O)CC1CO C1(C(=O)NCC(CC)NC(=O)CCCCOC)CCCN1S(=N)(=O)N(C)C c1(C(N2CCC(C)C2CNC(C23CCC(C2)C3)=O)=O)cc2n(n1)CCCO2 C1(NC(C(CO)OC)=O)CN(C(=O)C(c2ccccc2F)C)C2CCCC12 CCC(CNCC1(c2cccc(F)c2F)CCCC1)(CC)C(F)(F)F Cc1ccc(C)c(CC(=O)NCCNC(=O)C(c2cccc(Br)c2)C)c1 C12(C(=O)NCC3CCN(C(C(C)(C)C(F)(F)F)=O)C3)CCC(CC1)C(C)(C)O2 C1(C)(CNC(C2N(C(C)C)C(=O)CC2)=O)CCN(C(C2(CCO)CC2)=O)CC1 C(=O)(C1=C(C)C(C)(C)OC1=O)NC(CN(C(=O)Cc1cccc(OC)n1)CC)C N1(C(C(CC)NC(C)=O)=O)CC2CCC(NC(=O)C(C)Cc3ccco3)CC2C1 n1(CC)nc(C)c(C(=O)NC2CC(CC(N3CCCC(C)CC3)=O)C2)c1C C(=O)(CCCCC(=O)NCC1CC(O)CN1C(C1CCN(C)C1)=O)OC C12(C(N3CCC(C)(NC(C4CCCCC4)=O)C3)=O)CCC(CC1(F)F)C2 c1(CNC(C2(NC(Cc3ncn(C)c3)=O)CCC2)=O)cc(F)ccc1O CCCC(C(=O)NCCCOCCCNC(c1ccoc1Cl)=O)c1ccccc1 CC1OC2(C)CC1(C(=O)NCCC1CCN(C(=O)COc3ccccc3)C1)C2 C=C(C)c1cncc(C(c2nnnn2CCOC)Nc2cccc(Br)c2)c1.C1CC1 c1(C(=O)NC(C)CCNC(=O)Cn2ncc(Br)n2)cc2c(Cl)cccn2n1 c1(C(N2CCC(CCNC(C3CCC(F)(F)CO3)=O)C2)=O)ccn2ccccc12 N1(C(C2(OC)CCSC2)=O)CC2(CCCC(CNC(=O)CCOCC(C)C)O2)C1 N1(C(c2scc(OC)c2)=O)CC(C)(C)CC1CNC(c1cc(C)sc1C)=O c1(C(N2CCN(C(C(CCC)C(C)C)=O)C(C)CC2)=O)cccc2c1C(=O)CC2 N1(CCc2ccnc(N3C(c4n(C)ccn4)CNCC3)n2)CCN(C)C(C)(C)C1 CC1(C)CC(=O)NC1CN=C(NCc1cccs1)NCC(C)(O)C1CC1 CC(C)CC(O)C(C)C(=O)NCCOCCNC(c1ccc2cncnc2c1)=O C1(CCNC(C2CC2F)=O)CC(F)(F)CN1C(c1ccc(F)s1)=O N1(C(CC(C)C)=O)CCN(C(C2CCC(C(C)C)CC2)=O)CC(C)(C)C1 C(=O)(C#CC1CCOCC1)NC(CC)CN(C)C(c1cccc(SC)c1)=O c1(C(N2C(C(=O)NC3CCCN(C)CC3)CC3CC32)=O)ncc2ccccn12 C1(CC)CCC(C(N2CCC2C(=O)NC2(COC)CCCCC2)=O)CC1 c1(-n2cc(C(=O)NCCSCCC3CCC3)nn2)cccc(C(C)(C)OC)c1 N1(C(c2cc(C)c(C)nc2O)=O)CCC2CCC(C1)N2C(C12CC(C)(CO1)C2)=O N1(CC(=O)NC(C2(CNC(=O)CSCC3CCCO3)CC2)C)CCNC1=O C1(NC(c2n(CC)ncc2)=O)CC2CCC(C1C)N2C(=O)CC(C)n1ccnc1 c1(C(CC)N(C2CCN(C(=O)C(c3ccc(Cl)cc3)OC)C2)C)ccc(F)cc1 C(C(=O)N1CCCC1CNC(N)=O)(C(C)O)NC(c1cnc(OC)s1)=O c1(CN(C(C(C)NC(=O)Cc2ccccc2)=O)C)cnn2c1CNCC2 C(=O)(C1CCCc2nn[nH]c21)N(C1(CNC(=O)CN2CC3CC3C2)CCCC1)C Cc1scc(C(=O)NCCCOCCNC(C2(C#N)CC2C)=O)c1C C1(C(NOCCCC#C)=O)CN(C(C2CCC(=O)NC2)=O)CC1C(C)C C1(N(C(C2(C3CCC3)CC2)=O)NC(=O)NCCC)CC(OCc2cccnc2)CCO1 C(=O)(CS(=O)(=O)CC(=O)N(C)CC1CCN(C(c2ocnc2C(F)F)=O)C1)OC CC(C)CCCC(C)C(=O)N1CCCC(C)C1CNC(=O)CSS(C)(=O)=O C1(C(C)NC(c2nc(C(F)(F)F)cs2)=O)CN(C(c2cnoc2)=O)CCO1 C1(C)(NC(c2c(C)occ2)=O)CCCN(C(=O)CC2CCCOC2)C1 C(CN=c1cccc(S(=O)(=O)NCCn2ccnn2)[nH]1)OCCCOC Cc1nc(C(=O)N(CCCCCNC(C2(C)COC2)=O)C)nn1C(C)(C)C CC(CNC(c1ccc(N(C)C)cn1)=O)CN=c1[nH]cc(C#N)c2ccsc12 C(=O)(CC(O)C(Cl)(Cl)Cl)N(C1CCCCN(C(CCCCN(C)C)=O)C1)C N1(C(COCCCC#C)=O)CCCC(CCCCNC(C2CCN(C)C2)=O)C1 CCCCC(CC)CCC(=O)NCCC(C)(C)NC(C1CC(=O)NC(=O)N1)=O N1(Cc2ccsc2NC(CCc2cn(CCC=C)nn2)=O)CC(CO)CC1CO c1(C(=O)NC2CN(C(C(C3CCCCCC3)C)=O)CC2F)cc([N+](=O)[O-])ccc1Cl C(N=c1[nH]cnc(Cl)c1F)C12CCC(CNC(=O)C=Cc3cocn3)(CC1)OC2 C1(C(N2CCOCC2)C(=O)N(C(c2cn(C(C)C(=O)O)nn2)C)C)CC(F)(F)C1 C1(NC(C(C)(C)NC(=O)OC)=O)CC(OC)CN(C(=O)C=Cc2ccccn2)C1 C1(C(N(CCN(C)C(c2ncc(F)cc2F)=O)C)=O)CC(C)(C)CCO1 N1(CC)CCC(CNC(=O)CN(C(=O)COC2CCCOC2)CC)C1 Cc1cn2ccc(C(=O)NC3COCC3NC(=O)C(C#N)C(C)C)cc2n1 C(=O)(CCCC(=O)NCCC1(OC)CCN(C(C2CCC2COC)=O)C1)NCC c1(C(=O)NC(CN(C(C)=O)CC)C)nc2ccc(C)cn2c1N Cc1nccc(C(=O)NCC(C)(CO)NC(=O)CCc2nc(C3CC3)no2)c1C C1(C(C(C)NC(=O)CC2(C#N)CC2)NC(COCC(=C)C)=O)CCCCC1 C(C(=O)NCC(C)CNC(c1ncn(C)n1)=O)(C(C)C)NC(=O)OCC C1(C(=O)NCC(C)NC(c2c(C(F)(F)F)cnn2C)=O)CC12CC(C)(C)C2 C=CCC(CC)C(=O)NCC1CN(C)CCN1C(c1cnc(C2CC2)s1)=O C=CC(C)(CC)C(=O)NCCC1(O)CCN(C(c2ccccc2CC)=O)C1 C(=O)(C(CN(C(=O)Cn1ccnc1)C1CC1)C(C)C)N(CC(C)C)CCC C1(CC(=O)NC(c2cccc(C)c2)C)COCC(C)(C)O1 CN1C(=O)CCCC1C(N1CCCC(N(C(=O)CCCNS(C)(=O)=O)C)C1)=O N1(C(CC(C)C2CC2)=O)C(C)CC2CN(C(C3CCN(c4ncco4)C3)=O)CC12 C=CCC(CNC(=O)CN1CC2CCC1C2)C(=O)NCCCOCC(C)C c1(C(N(CC(=O)NCCCCSc2nc[nH]n2)C2CC2)=O)cscc1F c1(C(=O)NC(CNC(C2(CC)CCC2)=O)C2CC2)cccc(C2CC2)n1 c1(NC(c2cncc(NC(c3ccc(C)nc3)=O)c2)=O)cnc(Cl)c(C)c1 N1(C(C2C(=C)C2)=O)CCOC2(CCN(C(=O)Cc3cccc(OCC)c3)C2)C1 Cc1cc(CC(=O)NCC(C2CC2)N(C(=O)CCc2cc[nH]n2)C)c(C)s1 Cc1cc(C(=O)NCCC(C)(C)NC(=O)Cn2cccnc2=O)cc(=O)n1C CC1(C)CN(C(c2ccnn2C(F)F)=O)CC1NC(=O)CCn1cnccc1=O c1(C(N2CC3C(NC(CC(c4c(C)noc4C)C)=O)(C3)C2)=O)cc2n(c1)CCC2 N1(C(c2c(C(C)C)ncs2)=O)CC(NC(c2cc3scnc3[nH]2)=O)CC2(CC2)C1 C(=O)(CC(C(F)(F)F)N(C)C)N(CC1(F)CC(C)C(N(CC)CC)C(=O)NC1)C N1(C(c2ccc(C)o2)=O)CC2C3CCC(C2C1)N(CCC1CCCO1)C3 c1(NCC)cc(Cl)ccc1C(N1CCC(CNC(=O)C(CC)OC)C12CC2)=O C=CC(CC)CC(=O)NC(C)(CNC(c1cc([N+](=O)[O-])c[nH]1)=O)C1C(CC)C1 Cc1nc(Br)cnc1NC(=O)CC1CCN(Cc2cc(CO)ccc2O)CC1 C1(NC(CCN(C)CC)=O)CN(C(c2cc(Cl)cnn2)=O)C2(CCCOC2)C1 C1(CC(=O)OCC)CCN(C(=O)NCC2CC(C)(C)CO2)C2(CC2)C1 c1(C(=O)NCC(CCNC(C=C(C)C)=O)O)cc(Cl)ccc1OC(F)(F)F c1(SC)cc(C)c(C(=O)NC(C2CCN(C(=O)Cc3cn[nH]c3)C2)C)o1 c1(C(=O)NCC2(CCNC(C(C)SCCCC)=O)CC2)ncc(F)cc1C N1(C(C(F)=C(C)C)=O)CC(F)(F)CC1CNC(c1ncoc1C(C)C)=O Cc1ccc(OCC(O)CSc2ccn(C(C)C)c2)c(F)c1 C1(O)(CNC(C2(C(N(C)C)=O)CC2)=O)CCCN(C(=O)CCn2cc(Cl)cn2)C1 Cc1nc(C(=O)NC2CC(F)CN(C(C3CCC(O)CC3)=O)C2)c2n1CCCC2 C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(OC)C(NC(c2cc(Cl)n(C)n2)=O)C1 c1(OC)cccc(F)c1-c1cccc(C(CC2SC(=N)NC2=O)OC)c1 c1(NC(=O)CC2CCC(NC(c3c(O)cccc3F)=O)CC2)cc(Cl)c(Br)cc1Cl N1(C(=O)NCc2nccs2)CCC(Cc2cnccn2)C1 C#CC1(NC(C2(CNC(=O)C(O)CCSC)CC3(CC3)C2)=O)CCC(C)CC1 N1(C(CN(C)C)=O)CCOCC1CC(=O)NCc1cccc(F)c1 c1(C(=O)NCCN(c2nnc(CO)s2)CC)c(C)oc(C)c1C C1(C(N2CC(CC(=O)NC3CCN(Cc4ccccc4)C3)C2)=O)CC2CCCC2C1 c1(C(N(C(CN(C(CC(=C)C)=O)C)C)C)=O)nc(C(F)(F)F)oc1Br c1(C(=O)NCC(C(C)C)NC(=O)CCC2CC2)cccc2occ(Br)c12 C1(CCC(=O)NC2CC(C)(NC(=O)CC#N)C2)NC(=O)NC1=O C1(CC(=O)NCC(CN(C)C(c2cocc2C(N)=O)=O)O)CCCCC1O N1(C(C(c2c(C)noc2C)C)=O)CC2CC(NC(c3cn[nH]c3)=O)C1C2 Cc1ccccc1C=CC(=O)NC1CCOC1C(=O)Nc1cncnc1O CC1CC(CNC(C2(P(C)(C)=O)CC2)=O)CN1C(c1coc(C2CC2)n1)=O n1(CCC(=O)NCC(CNC(=O)C(O)CSC)OC)ncn(C)c1=O C1(C)(C(N(CC(CN(C(=O)CNc2ccccn2)C)O)C)=O)CC1(F)F C1(CNC(C2(OC)CCSC2)=O)COC(C)(C)CN1C(=O)COCC1CCC1 c1(OC)nccnc1C(=O)NCC(C1CC1)NC(c1cccc(OC(C)C)n1)=O Cc1ncc(C=CC(=O)NCCC2(C)CCN(C(C3CC(N(C)C)C3)=O)C2)s1 N1(C(C(=O)NCCCSCC)c2ccns2)CCCCC1c1cccc(O)c1 CC(C)CS(=O)(=O)NC1CCC(c2ccccc2)C1 C1(CC(N2CCC(C(C)(C)NC(=O)Cc3cnco3)C2)=O)CCCC(F)(F)C1 Cn1cnc(C=CC(N2CCC(C(F)CNC(c3cc(F)c[nH]3)=O)CC2)=O)c1 Cn1nc(CN2CCC(C)(C)C2)cc1CC1CCCCO1.C1(=O)CO1 C=C(C)CC(C(=O)NC1CC2CN(C(=O)C=Cc3ccccn3)CC12)NC(C)=O N1(C(C(n2cnc(C#N)n2)CC)=O)CC2(C1)CC(C)(O)C2 C1(C(N2CCC(C(=O)N(C)C)C2)C(=O)NCCC)CCC2COCCC2C1 C1(CC(C)C)COCCN1C(=O)NC(C)CCc1cn(C)nn1 C(CNC(c1ccc(C(F)F)c(Cl)c1)=O)(CCS(C)(=O)=O)OC CC1CN(C(c2ccnc(C(C)(F)F)c2)=O)CCC1NC(=O)CCN(C)CCO C1(OC)CC2(C1)CC(C(=O)NC(C)CCNC(=O)CC(CC)OC)C2 C1(F)(CNC(C(c2cccs2)SC)=O)CC(NC(c2cnccn2)=O)C1 C1(C(C)C)CN(C(C2CCCCS2)=O)CCN1C(=O)CC1CCC(C)CC1 c1(CC(=O)NCCCOCCN(C)C(c2csnc2Cl)=O)ccc(Cl)cc1 C1(Nc2cc(OCC)ncn2)CC2(CCN(C(c3cc(Cl)ccc3C)=O)C2)C1 c1(COC)ccccc1-n1cc(C(C(=O)NC)N(C(CC)CC)C)nn1 c1(C(=O)NC2C(NC(c3c[nH]c(=N)o3)=O)CCC2)nc(Cl)sc1Cl C=C(Cl)C(C)(C)C(=O)NCC(CCOC)NC(=O)COC(c1nccn1C)C C1(O)(C(=O)NC2CCN(C(C34CC(CC)(OC3)C4)=O)C(C)C2)CCC(C)(C)CC1 CN1CCCC(C(N2CCCC2CCC(=O)NC(C2CCCO2)(C)C)=O)C1 C1(NC(=O)CC(F)(F)F)CN(C(=O)C=Cc2cncnc2O)CC2CCCC12 c1(SCC)ccc(C(N2CC(OC)CC2CNC(C2CCC(C)O2)=O)=O)cn1 c1(CCC)n[nH]cc1C(=O)NCC(CC)NC(=O)CC(C)N(C)C C1(C(=O)NCC(C)(C)NC(=O)C(F)=C2CCC2)CCCN1C=O C(CS(=O)(=O)C(C)(C)C)NCCNC(c1ccc(C(CC)C)cc1)=O C1(CC(=O)NCC(=C2CN(C(C(C)OC3CCCC3)=O)C2)F)CCn2cncc2C1 C1(C)(C(NOC(c2ccncc2)C)=O)C=CCN1C(=O)CC#N c1(C(=O)NCC(CNC(COCCC(C)C)=O)O)n[nH]c2ccc(Cl)cc12 C(=O)(C(CC(F)F)NC(C1CC(C)(C)C1)=O)NC1(C)CC(C)(C)C1 Cc1ccc2c(c1)ncn2CC(N1CC(NC(=O)CO)C(C2CC2)C1)=O C1(CNC(C(=O)NCC)=O)CC2CC1CN2C(c1cc(C)nn1CC)=O C1(OCC)CCCN(C(=O)C(CNC(=O)CC2CCCCO2)CC2CCCC2)C1 C1(C(N2CCC(=C)CC2)=O)CN(C(=O)C(C)NC=O)CC(C)(C)C1 N1(C(CC(=C)Br)=O)CC(CNC(=O)COC2CCOC2)C2(CCC2)C1 c1(C(=O)OC)cnccc1N1CC2C(CNC(c3nccnc3C)=O)C2C1 N1(C(=O)CCOCC(F)F)CC2CC1CN2C(c1nccc(Br)c1O)=O N1(C(NNC(c2c3cccc(C)c3oc2)=O)=O)CCCC2NC(=O)C(C)(C)C12 c1(CC(=O)N(C(C)CN(C(=O)CNC(c2cnn(C)c2)=O)C)C)ccc(Cl)nc1 N1(C(C(C(C)C)(C)O)=O)CC2C3CCC(C2C1)N(C(c1sccc1C(F)F)=O)C3 C1(CCNC(C2C(C)C2C)=O)CN(C(c2n[nH]cc2Cl)=O)CCS1(=O)=O C(c1ccc(C(N)=O)o1)=CC(=O)NC(CNC(C(C)CN(C)C)=O)(C)CO C1(CC(=O)N(CC)CC2CCCO2)CC(F)CN1C(c1cc(COC)c(C)o1)=O CCC(C)(C)CC(=O)NC(C)C(C)NC(c1ncoc1-c1cnn(C)c1)=O C1(N(C(C=CC=CCC)=O)C)CCCCN(C(c2ccc(COC)cc2F)=O)C1 N1(C(c2ccc(C(C)=O)o2)=O)CCCC(C(=O)NC(C)C(F)F)CC1 c1(C(=O)NCC2(C)CCCN2C(=O)CC2CC3CC3C2)cc2c(cn1)CCCC2 N1(C(CCc2c(C)ncs2)=O)CCOC(CNC(=O)C=CCOC(C)(C)C)C1 C1(NC(CN(CC)CC)=O)CCCN(C(=O)CCCOC(C)(C)C)C1C N1(C(=O)Cn2nnc(C3CC3)n2)CC(NC(C23CC(CO2)C3)=O)CC(O)C1 N1(C(CC(=C)C)=O)CCC2(CCN(C(=O)C(C)C(F)F)CC2)C1 C#CC1CCN(C(=O)OCC)C1.c12nc(C)c(s1)C(C)N2C N1(C(C=C(C)C)=O)CC2(C1)SCCC2NC(=O)CC(c1c(C)noc1C)C Cc1ccc(O)c(CN2CCCCC2c2n[nH]cc2N)n1 c1(C(=O)NC(C2CCN(C(C(C)=C3CC3)=O)C2)(C)C)ccc(C(C)=O)cn1 Cc1oc2ccccc2c1CO.C12(S(=O)(=O)C(=O)N(C)CCn3cc1nn3)CC2 N1(C(C2CC=C(C)CC2)=O)CCC(C2CC2)(CNC(=O)Cc2ccnc(C)c2)C1 c1(C(=O)NCCn2cc(CCC3CCOCC3)nn2)ncc2ccccn12 C1(C(=O)NC2CC(CNC(=O)C3=CCCOC3)C2)CCn2c(O)nnc2C1 N1(C(C2(C)N(C(c3nc(C)sc3C)=O)CC=C2)=O)CCC2(CC(CO)C2)C1 c1(OC)ccc(-c2cnc(CNC(c3ccn(C(C)(C)C)n3)=O)nc2)c(C)n1 N1(C(C2C(C)(C(F)F)C2)=O)CC(CNC(c2cnoc2C2CC2)=O)C2(CCC2)C1 O=S(=O)(c1cc2cc(F)ccc2s1)NCc1nc2ncccn2n1 N1(C(c2c(CC)ccs2)C(=O)NC2CCC2)CCC(C2(O)CCC2)CC1 c1(C(=O)Nc2cc(F)cc(C(=O)OC)c2N)cc([N+](=O)[O-])ccc1Br Cc1ccc(COC(C)C(=O)N(C(C)CCNC(C2(C(F)(F)F)CC2)=O)C)cc1 c1(N(CCOC)CCNC(C2CCN2S(C)(=O)=O)=O)c(F)cccc1[N+](=O)[O-] C1(NC(COCCOCC#C)=O)C(C)CN(C(c2snc(O)c2Cl)=O)CC1C C1(C(N(C2CCN(C(CC(=C)Br)=O)C2)C)=O)CC2OC(=O)OC2C1 CCCCCC(=O)NC(C)(C)C(C)NC(=O)C(C)(CC1CCC1)OC c1(N2C3CC(=C)CC2CCC3)nc(=NCC2(NS(C)(=O)=O)CC2)[nH]c2c(F)cccc12 CC1COC(C)(C)CN1C(CSc1ccccc1)C(=O)NCCC#N Cn1ccc(C(N2CC(OCCC(=O)NCC3CC3(Cl)Cl)C2)=O)c1 c1(C(=O)NCCNC(C2CCN(C(=O)C(O)C(F)(F)F)CC2)=O)ccc(F)c(Cl)c1 Cc1[nH][nH]c(=NC(=O)C2CN(C(c3ccc(Br)c(O)c3)=O)CCC2O)c1Br C1(CNC(Cc2cccc(SC)c2)=O)C(C)CCCN1C(=O)CCc1cnoc1 N1(CC)CCC(C(=O)NCCC2CC2)CC1.C12(CC1)C(=O)NCCO2 C1(C(NOCCC(C)C)=O)CN(C(=O)CCc2cccnc2)CCC1(C)C C1(CCOC)(C(=O)NCC2CC2Cl)CCN(C(C2CCCCN2C)=O)CC1 S(=O)(=O)(c1ccc(NC2CC(CF)C2)cc1Br)NC(CC#CC)C C1(NC(C(C(C)O)(F)F)=O)CC2(CCCCN2C(c2cnncc2O)=O)C1 c1(OC)ncccc1CC(=O)Nc1cccc(CNC(=O)CC2CS(=O)(=O)C2)c1 c1(NCCCN(C(C2OCCC2c2cnn(C)c2)=O)CC)ccccc1Cl c1(CC(N2C(CNC(c3ncc(N(C)C)nc3)=O)CC2)=O)ccc(S(C)=O)cc1 Cc1nccc(C(=O)NCC23CC(NC(c4cc(CO)oc4C)=O)(C2)C3)c1C N1(C(C2N(C(C)=O)CSC2)=O)CCCCC1CNC(=O)CC1C=CCC1 C1(CCC)CN(C(c2cccc(COC)c2)=O)CCN1C(=O)C(C)C(F)F c1(N(C(=O)C(CC)C2CCOCC2)CCC)cccc(C(N)=O)c1 c1(CN(C(c2cccs2)COC)C)ccc(OC)c(-c2ccnc(C)c2C)c1 C(=O)(CCSCCN(CC(F)F)CCOC)OCC(F)F N1(C(C(N2CCOCC2)C)=O)C2CCC1C(NC(=O)COC1CCC1)C2 C(=O)(C1=CCCNCCC1)NC(c1ccc(Cl)cc1)C(N)=O C(C)(C)(CCCCC(=O)N1CC2CC(C(N3CC4(C=CCO4)C3)=O)CC2C1)OC c1(C(=O)NC2CC(C)N(c3cc(C4CC4)ncn3)CC2)occ2c1CCOC2 N1(C(C2CCCC(=O)N2)=O)CC2(CCC2NC(=O)C(=C2CCCCC2)F)C1 N1(C(CC(CC)(F)F)=O)CCOCC12COCCN(C(=O)CCC(C)O)C2 C1(NC(C(CC)C#N)=O)CCN(C(C2CN(CP(C)(C)=O)C2)=O)CCC1(F)F c1(C(=O)NCC(C)NC(c2nnn(COCC)c2N)=O)ccc2c(c1)CN(C)C2 CN1C(=O)CCC1(C)CNC(C1C=CCN(C(c2ncncc2N)=O)C1)=O N1(C(CCCC#CC)=O)CCC2(CC1)CC2CNC(C1(COCC)CC1)=O O=C(N1OC2C=CC1CC2)C1CSCN1C(C1(F)CC=CCC1)=O N1(C(C(N2CCOCC2)C)=O)CCC(NC(=O)COC(F)(F)F)C1C1CC1 Cc1ncc(Cl)cc1CC(N1CCC(NC(=O)CC2CNC(=O)C2)C(O)C1)=O c1(NC(C(CN(C)C)NC(c2n(CC)c(O)nc2)=O)=O)c(C)cc(C)cc1C c1(CC(N2CC(CCNC(=O)C=Cc3cn[nH]c3)OCC2)=O)cc(F)ccc1O c1(C(=O)NC2CCC(C(=O)NC(C3CCOC3)C)C2)cnc2c(Br)cccc2c1 Cc1cc(C(=O)NCCC2(NC(=O)CCC3CCC(=O)N3)CCC2)c(C)cc1Cl c1(C(=O)NC2C(CNC(C(C)n3ccnc3)=O)COC2)ccc(P(C)(C)=O)o1 C1(C(=O)NCCC(C)(C)NC(=O)CSCCc2ccccc2)CCCS1(=O)=O CC1(C(=O)NCC2(CCNC(c3cncnc3)=O)CC2)CCC(=O)NC1 C1(C(=O)NC2CCCC2NC(=O)CCS(C)=O)(NC(C)=O)CCCCC1 C(=O)(C1=CCCOCC1)N1CCC(CC)C1CNC(c1c[nH]c2nccc-2c1)=O N1(c2cc(C(=O)OC)ncn2)CCCN(C(C2CC(O)C2)=O)CC1 CC1CC(N=c2ccnc(NCc3ccc(N)cc3Cl)[nH]2)CCO1 c1(NC(CN2C3CC(C(N)=O)C2CC3)=O)ccc(S(=O)(=O)c2ccccc2)cc1 Cc1ccc2c(c1CO)CCCN2CC(c1cccc(C#N)c1)O c1(N2CCC(NC(C3C(C(=O)OC)C3)=O)C23CCC3)nc2ccc(N)cc2s1 c1(C(=O)NCCCNC(c2cc(-c3cccnc3)on2)=O)sccc1Br C1(C(=O)NCCOCCOC)CC2CC1CC2NC(c1ncncc1C)=O c1(CC)nccnc1C(=O)NCC(C1CCCC1)NC(C1(C(F)F)CCCO1)=O c1(C(=O)NCCN(C(=O)CS(C)(=O)=O)CCC)ccc(Cc2nc[nH]n2)cc1 N1(C(CC(C)N2CCCC2=O)=O)CCN(C(=O)CSCC(F)(F)F)CC12CC2 c1(C(=O)NCCN(C)C(C2CCS(=O)(=O)C2)=O)ccc2nn[nH]c2c1 c1(-n2c(-c3nccc(CSCC)c3)nc(CC3CCC3)n2)cnc(Cl)c(F)c1 N1(C(C(C)(C)c2ccsc2)=O)CC2CS(=O)(=O)CC2(CNC(=O)CCF)C1 C1(CC)CCC(n2nc(-c3nc(C(=O)CC)cs3)nc2-c2cc(SC)oc2C)CC1 c1(CCNC(CCOC2CN(C(c3cnc(C(C)C)o3)=O)C2)=O)ccc(F)nc1 N1(C(CC(CC)SC)=O)C2COCC1CC(NC(C1C=C(C)CS1)=O)C2 O=S(=O)(c1cc(C(F)(F)F)ccc1O)NCC1(CO)CCOC1 CC1CCCCCC1NC(C1(O)CC(CNC(=O)OC(C)(C)C)C1)=O C1(CC)CN(C(c2cc(O)nc(C)n2)=O)CCN1C(C1CN(C2CCOC2)C1)=O c1(C(=O)OCC)n[nH]c(=NCC2CCCC(NC(C3CCC(=O)N3C)=O)C2)s1 C1(C(=O)NCC=C(C(=O)N(C(CC)C)CC)C)CC=CCC1C C1(C(=O)NCCCNC(c2cc(CC)c(O)cc2)=O)COC2(CCC2)CO1 c1(C(N(CC(CNC(CC(CC)SC)=O)(C)C)C)=O)cc(C)ccc1N N1(C(C2(C)C(C)C2)=O)CC2CN(C(=O)C(C)(C)C(F)(F)F)CC2C1 N1(C(c2c(C)cncc2F)=O)CCC(C)C(C)(C)C1 N1(C(C(CC)C)=O)CCN(C(=O)CCc2nc(CSC)no2)C(CCO)C1 C(=O)(C1=NOC2(CCC2)C1)N(CCCCNC(=O)Cc1cc(F)ccc1F)C C1(c2n(CCCF)nnn2)(NCc2ccc3c(Br)c[nH]c3c2)CCN2CCC1C2 Cc1cc(=O)ccn1CC(=O)NCCC1CN(C(=O)CC2(O)CCC2)CCO1 O=C(CCCCC1CCC1)NCC1(F)CN(C(c2c[nH]nc2F)=O)C1 N1(C(C(C)C)=O)CCC(NC(=O)CC2=CCOCC2)CC(C)(C)C1 C1(CC(N2CC(CC(C)NC(C3(CC)CC(C)(C)C3)=O)C2)=O)CCCCC1(F)F C1(C(=O)NC(C)CNC(c2ccc(F)c(Br)c2)=O)CC12CCC(F)(F)CC2 CCCC(C(=O)N(C)CC1CC1(C)C)NC(=O)C(C)OC(C)=O C(C1=CCN(C(=O)C(C2CCCN(C)C2)(C)C)CC1)NC(Cc1c(C)noc1Cl)=O c1(C(=O)NC2(C)CC(NC(C3COCCC3(F)F)=O)C2)ccc(=N)[nH]c1Cl N#Cc1ccc(C(=O)NCC#CCNC(c2cc3c(s2)CCC3)=O)c(F)c1 C(=O)(CCS(C)(=O)=O)N1CC(CNC(C(CCC)C)=O)OCC1.C1(=O)CCCN1 C1(C(C)NC2CC3(C2)CC3F)CCCC(C)(C)CC1 C1(CNC(CC(=C)Br)=O)CCN(C(c2nocc2C(=O)OC)=O)CC1C N1(C(c2ccc(OC)cc2I)=O)CC(C(=O)O)C2(C1)CN(C(=O)C(=O)C1CC1)C2 N1(C(C2C(CCC)C2)=O)CC2(C)CC1(C(=O)N(C(CC)CC)C1CC1)C2 Cc1oc(CO)cc1C(=O)NC1(CC(=O)NC2CCN(CCCO)C2)CC1 N1(C(C)=O)CCCCC(NC(c2cc(Cl)c(Cl)cc2Br)=O)CC1 C1(CNC(N2C(C)CC(C(=O)OC)C2)=O)CCCCCC1C1CC1 c1(Cn2cc(C(CCC)NC(=O)CCn3cccn3)nn2)cc(Cl)ccc1C c1(CN2C(C(N3CCn4cnnc4C3)=O)CNCC2)ccc2ccccc2c1Br N1(C(C(CCSC)O)=O)C2CCC1C(CNC(c1oc(CC(C)C)nc1C)=O)C2 c1(OC)cncc(C(=O)NC2COCC2NC(=O)CSc2c(C)n[nH]c2C)c1C C1(CC(=O)NCC2CCC=CCC2)C2CCCC2N1C(=O)C(O)c1ccsc1 C1(NC(COCC(=C)C)=O)CC2CC(NC(=O)CNC(=O)CN(C)C)CC12 c1(C(=O)NCC2C3CN(C(C4CC(C)OC4)=O)CC32)c(Cl)nc2ccccn12 CCC(C(=O)NC1CCCC(NC(=O)Cc2ccc(F)c(F)c2)C1)C(C)(C)CC C1(C2CCCN(C(c3ccno3)=O)C2)(NC(c2cc(C)nnc2O)=O)CC1 Cc1cc(NC(c2nn(C)c(C)c2Cl)=O)ccc1NC(c1[nH]nnc1C)=O C1(CNC(c2c(SC)snn2)=O)CC12CCN(C(=O)C=CCCC(C)C)CC2 N1(C(c2ccc(OC)c(Cl)n2)=O)CCC2(C1)CN(C(c1ocnc1C)=O)C2 C1(C(=O)NCCOC2CCN(C(CCSCCCC)=O)C2)(N(C)C)CCCSC1 n1(CC(=O)NCC(CN(C(CC(COC)(C)O)=O)C)C)ccc2ccc(F)cc12 C1(NC(C(C)NC(=O)C(N2CCOCC2)C)=O)C2CCCC1COC2 C(CC(C)CC(C)(C)C)NC(c1c(CNC(c2ccc(C)c(C)c2)=O)n[nH]c1)=O c1(CC)nc(C)c(CC(N2CCCN(C(c3cncs3)=O)CC2CO)=O)c(C)n1 c1(C(=O)NC2CN(C(c3n(C)ncc3)=O)CC2F)nccn2ccnc12 N1(C(C2CC(CCC)C2)=O)CCCC2(C1)CN(C(=O)Cc1ccsc1)CCO2 C=C(C)C(C)(C)C(=O)NC1C2CC(NC(C3CCC(F)C3)=O)CC12 c1(CC)cc(C(N2CCCCC2CN(C)C(C2(F)CCOC2)=O)=O)c(C)nn1 CCC(C(=O)NC12CC(NC(=O)CCc3cc(C)no3)(C1)C2)C(C)(F)F c1(C(N2CC(CNC(c3ccc(-c4cn[nH]c4)cc3)=O)C2)=O)cc(Br)cnc1O N1(CCC2CC(C)OCC2)C(=O)CN(Cc2ncc(Br)s2)C1=O c1(C(=O)NC(CN(C(CNC(=O)NC)=O)CC)C)cncc2ccccc12 CC(C)CC(C)C(=O)N(CC(C)(C)C(=O)N(C(C)C(C)C)C1CC1)C c1(CN(C(CN(C(=O)C=Cc2ccncn2)CCOC)=O)C)c(C)cnn1C c1(OC)cc(C(=O)NCC2CC2NC(C23CC2COC3(C)C)=O)cc(C)n1 c1(N(CC(C)NC(C2CS(=O)(=O)CC(=O)N2)=O)C)ncc([N+](=O)[O-])cc1Cl C1(C=O)CCCN(CC(F)F)C1.c1(C(C)C)nnnn1CC(=O)NC1CC(CF)C1 c1(C(N2CC(SC)CC(OCC)C2)C(=O)NC(C)C)cc([N+](=O)[O-])c(O)cc1F Cc1cc(F)cc(C(=O)NCC2CCCC2NC(=O)CC2CC3(CCC3)C2)c1O C1(F)(C(=O)NC(C2CCCN2C(c2cnn(C3CCCC3)c2)=O)C)CCCCC1 CC(F)(F)CCC(=O)NCC1CCCC1NC(=O)C(O)CC1CCCCC1 C(CCC(C)C(=O)NCC=CC(N1CC(=O)NCC1C)=O)OC c1(C(=O)NCC(CCCC)NC(C2CCC(C)(C)C2)=O)ccc(C2CC2)c(F)c1 CCC(CC)C(C(=O)NC1CC(O)(CNC(=O)CC2C(C)(C)C2(C)C)C1)OC CC1=C(C(=O)NC2CCN(C(=O)C=CC3CCCO3)C2(C)C)CCC1 c1(C(C)C(=O)NCCC2CCN(C(C3CN(C)C3)=O)CC2)noc2ccccc12 Cc1cn(CC(=O)NC2CC2CNC(c2nnsc2C(F)F)=O)c2ccccc12 C1(NC(CCCOCCC)=O)CCCN(C(c2ccc(C)c(C)c2)=O)C1C c1(CC)oc(C)cc1C(=O)N(C(CNC(c1cnc(O)n1C)=O)C1CC1)C CC1SCCN(C(=O)CC2(NC(c3cc(C4CC4)nn3C)=O)CCC2)C1C C1(NC(C(CC)C)=O)CC1C1CCN(C(c2cc(NC(C)=O)ccc2F)=O)CC1 C(=O)(C(C)(C)CN(C)C)NCC(CCNC(C1(C)CCCC1)=O)OC Cc1nccc(C(N2CCN(C(=O)CC3CC(=O)NC3=O)C(C(C)C)C2)=O)c1O O=C(CCCCO)NC1CC(CNc2ccnc(C3CCCC3)n2)C1 C1(C)(C(=O)Nc2cc(C(C)C)on2)CCN(C(=O)NC2CCOCC2)C1 C(=O)(C(C)CC(C)CC)N(c1cccc(C(NOCCOCC)=O)c1)CC C(CC(C)C)(C(=O)NCc1ncccc1C(=O)N(C)CC1(O)CCC1)OC C=CCC(CNC(=O)CC1COCCO1)C(=O)N(C)C(C)C c1(C(c2nn[nH]n2)NC(c2cccc(OC(CC)C)c2)=O)ccc2cc[nH]c2c1 C(C(=O)N(CC(=O)OC)C(C)C)(C(C)C(C)(C)C)N1CCC(C)(CCC)C1 N1(C(Cc2c(C)n[nH]c2C)=O)CC(N=[N+]=[N-])CC1C(=O)NC(C1CCCC1)CO c1(C(=O)OC)ccc(CNC(C2(c3ccc(C)cc3Br)CC2(F)F)=O)cc1O C(=O)(C1=C(Cl)CCC1)N1C(C(=O)NCc2ncn(C3CC3)n2)(COC)C=CC1 C1(CNC(=O)C=Cc2nccs2)CN(C(c2ccn(CCF)n2)=O)CCCO1 c1(C(N2CCN(C(C(CC(C)C)F)=O)CC2)=O)ccc2c(c1)N(C)CCO2 CC(C)CC(C(=O)NCC(C)CNC(C1CC(C(F)(F)F)C1)=O)N1CCCC1=O N1(C(C(CCC)=CCC)=O)CCN(C(=O)CC(O)CC(C)C)CC(O)C1 c1(CCNC(c2scc(C(N3CCC(C)(C)C3)=O)n2)=O)ccc2ccccc2c1 Cc1cccc(Cl)c1C(=O)NCCOCCN(C)C(c1nscc1N)=O Cc1[nH]nc(CNC(=O)C=CCNC(=O)CC2CCCCO2)c1C N1(C(C2(COC)CCCO2)=O)CCCC(N(C(=O)C=CC=C(Cl)Cl)C)C1 c1(C(=O)NCC2CN(C(c3cc(SC)c(C)o3)=O)C(C)C2)cnn2c1N(C)CC2 C(CN=c1[nH]nc(-c2ccon2)s1)NC(C(N1CC(C)OC(C)C1)(C)C)=O C1(C(=O)OC)CN(C(=O)CNC(=O)CC(C)C)CC1C N1(C(c2n(CC=C)ccc2)=O)CCCN(C(c2cc(OC)nc(F)c2)=O)CC1C C1(CNC(C=C(C)C2CCCCC2)=O)CCN(C(=O)C(O)C2CC2)CCC1(F)F C1(CC(=O)NCC(CNC(c2ccn(C3CC3)n2)=O)OC)CCC(C)(C)C1 CC1c2c[nH]nc2CCC1C(N1CC(CNC(c2ccc(C#N)nc2O)=O)C1)=O Cc1cccc2nc(C(=O)N(C)CCNC(=O)CCCn3ccccc3=O)cn12 Cc1noc(C(=O)NCCCCCNC(=O)C(F)(F)c2csc(C)c2)n1 C(=O)(C#CC1(CC)COC1)NC1CC(C(C(=O)NC(CCC)C2CC2)F)C1 C=CCC(CNC(C1CC(C)N(C)C1)=O)C(=O)N1CCC(C)(CO)C1 C1(OC)CC(C(=O)NC(C)(CNC(=O)CC(C)n2ccnc2)CO)CC1OC C1(C(N(CCN(C(c2cncc(O)c2)=O)CC)CC)=O)CCC(N=[N+]=[N-])C1 C1(NC(c2ccn(COC)n2)=O)CN(C(c2ccc[nH]2)=O)CC1n1ccnn1 C(C(C)(O)CC1CCC1)NCC(CC)NC(=O)OC(C)(C)C CC1CCN(C(=O)NCCS(C)(=N)=O)C1c1cn(Cc2nc(C(=O)O)cs2)nn1 c1(CC(=O)NCC(=O)NCC(COC)C)ccn(C)c1 C1(F)(CNC(C2CCCO2)=O)CCN(C(c2cccc(-c3ccoc3)c2)=O)C1 C1(CN(C(=O)CCS(C)=O)C)CCCCN1C(c1ccc(CS(C)(=O)=O)cc1)=O C1(CN(C(CC2N(C(C)C)CCC2)=O)C)CCN(C(C2(CF)CCC2)=O)CC1 CC1=NNC(=O)C1CCC(N1CCOC(CN(C)C(C23CSCC2C3)=O)C1)=O Cc1cc(Cl)c(C(N2CCS(=O)(=O)C(CCNC(=O)CC=CCCO)C2)=O)cc1C CN1CCOC(C(=O)NCCCOCCCNC(c2cnn(C)c(=O)c2)=O)C1=O C(C(=O)N1CCC1(CO)CO)(C(C)(C)C)NC(c1c(CC)noc1)=O c1(C(N2CC3(CN(C(CC(C)OC)=O)C3)C2)=O)cc(Br)cc2c1CCN2 CC(C)CCCCCC(=O)N1CC2CCC2(CC(=O)NCc2ncc(Cl)cn2)C1 N1(C(CCOCCOCC)=O)CCCC1(C)CN(C(=O)Cc1ccc(C)s1)CC c1(C(CNC(C2CC2C(F)F)=O)NC(CC=CC)=O)ccccc1Br C1(NC(c2ccc(CC)nc2)=O)CCC2(C1)CN(C(C1(C)CC1C)=O)C2 c1(CC)cccc(C(c2nnnn2C(C)C)NCC2(OC)COC2)c1F c1(CC(=O)NCC(CNC(=O)CN2CC=C(C)CC2)OC)ccnc(F)c1F C=CCC(F)(F)C(=O)N1CC(C(C)(C)O)(CNC(C2(CC)CCC2)=O)C1 C(=O)(C(C)(F)C(C)(C)F)N1CCN(CC(C)NC(CSCCC(C)C)=O)CC1 N1(C(c2scc(C)c2)=O)CC2CCOC2(CNC(=O)C(O)C2CC2)C1 S(=O)(=O)(c1ccc(NCC2CCC2N(C)C)c(Cl)c1)NCc1c(C)scc1 CCC(CC(=O)NC1CCN(CCF)C1)C(C)C.c12ccsc1C(=O)NC2 CC1CN(C(c2nc(Cl)cc(N)c2Cl)=O)CCCN1C(=O)COc1cnn(C)c1 C(CCCNC(C1CC1C(N1CCCC1)=O)=O)C1C(C)C1.C1(C)(C)CNC(=O)N1 C1(N(C(c2c(C)cno2)=O)C)CC2CCC(C1)N2C(=O)CCS(C)=O Cc1[nH]c2ccc(C(N3CC(NC(c4ccc[nH]4)=O)C4CC4C3)=O)cc2c1C C1(NC(=O)COC2CCCC2)CCCC12CN(C(=O)CC(O)C1CCCC1)C2 C1(c2ccc(OC)cn2)NC(=S)N(CC(C)C)C2=C1C(=O)NC(C)(C)C2 C(=O)(C1=Cc2ccccc2C1)NC(CNC(c1c(OC)noc1C)=O)(C)C1CC1 c1(OC)ccc(OCC(C)(C)CC(=O)NCCc2nn[nH]n2)cc1 C(=O)(CCCCSC)N1CC(C(=O)NCC2(C(N)=O)CCCC2)(CC)C1 N1(C(C2(C(C)C)CCN(C(C=C(C)C(C)C)=O)C2)=O)CC2CC(O)CC1C2 c1(C(=O)NC2CC(=O)N(C3CN(C(=O)C4CC4)C3)C2)c[nH]c(=O)c2ccnn12 c1(C(=O)NCCC2(CNC(C(COC)C)=O)CC2)cn(C)c(=O)cn1 Nc1ccc(F)c(C(N2CCN(C(=O)CN3CCS(=O)(=O)CC3)C3CC23)=O)c1 C(=O)(CCC(C)(C)NC(=O)CC1CCCOCC1)NC(C1(O)CCC1)C C1(C)(CNC(C2N(C)CCCCC2)=O)CN(C(=O)CC2CC=CC2)C(C)(C)C1 c1(OC)cc(-c2nc(CCCO)no2)cc(OC)c1OC Cc1cc(C(=O)NC(C)CNC(c2csc(Cc3ccccc3)c2)=O)nc(O)c1 c1(OC)cc(OC)nc(C(=O)NCC2(C)CCN(C(C3NC(=O)CC3C)=O)C2)n1 Cc1ccc(Cl)c(OC(C)C(N2CCC(CNC(c3cc(C#N)cs3)=O)C2)=O)c1 c1(C(=O)NCCC2(O)CCCN(C(=O)CC(F)(F)F)C2)cnnc2ccccc12 c1(C(=O)NCC2N(C(c3c(C)nc(Br)o3)=O)CC2)ccc2c(c1)C=CCC2 c1(C(=O)NCC2CCN(C(c3scnc3C3CC3)=O)C2)cc(Cl)cc(Cl)c1O c12ncc(Cl)c(n1)C(=O)NC2C1CC1.C(=O)(C1=CC(C)(CC)C1)N1C(CC)CCC1 N1(C(=O)C(F)F)CCOC2(CCCN(c3ncc4c(Br)cccc4n3)C2)C1 c1(C(=O)NC(C(=O)NC2CCC(=O)NC2=O)CC2CCC2)ccn2ccnc2c1 C1(CNC(C=CCCC(C)C)=O)CN(C(C2(F)CCC2)=O)CCC1C(F)(F)F CC1(C)CC(NC(=O)CCCCc2ccccc2)CN1C(=O)C1=CCCOC1 C(=O)(C(CC)CCc1ccccc1)NCC(CC(C)C)NC(C1(OC)CCC1)=O N1(C(C(c2ccc(F)cc2)OC)=O)CC(NC(c2sccc2C(C)C)=O)C(C)C1 N1(C(C(C)SCC)=O)CC(C(N2CCCC(F)(F)C2)=O)C2(CC2)C1 C(CC(=O)Nc1cncc(C)c1)(CC(C)C)NC(C12CCC(OC)C1C2)=O C(c1cccc2ccccc12)=CC(N1CCCCC(NC(=O)C=CC2CC2)C1)=O N1(CCC2CCCC2n2cc(C(N(C3(C4CC4)CC3)C)=O)nn2)CCNC(=O)C1 CC(C)C1=NOC(C)(C(N2CC3(C2)CN(C(C2CN4CCC2CC4)=O)C3)=O)C1 O=C1CCC(CC(=O)NCC2CC(NC(=O)CC3(O)CCC3)C2)C1 N1(C(CCCC(=O)OC)=O)CCC2(CCN(C(C3CC3F)=O)CC2)C1 c1(C(N2C(C(N3CCC(C(=O)OCC)C3)=O)COCC2)=O)cc(Cl)cnc1F O=C1NC2(C(=O)NC3CC(NC(C4(n5ccnn5)CC4)=O)C3)CC3CC1C2C3 C(=O)(C1(C)CCOc2ccccc21)N(CCCNC(C1CC2C=CC1O2)=O)C c1(CC)nn(C)c(CC)c1C(=O)NCC(C)(C)CN(C(=O)CCCC#N)C C(=O)(CCCCNC(C1(F)CCCCC1)=O)NCCC1C(C(=O)OC)C1 CCC(CC(=O)N1CCC(NC(=O)CN(C(=O)C(C)C)C)C(C)(C)C1)C(F)F C12(C(N(CC(C)(C)CO)C)=O)CC(C)(CN1C(C1CCC(=O)C1)=O)C2 c1(SC)ccnc(NC2CCN(C(=O)C=C3CCSCC3)C2)n1 Cc1ccc2c(-c3nc(C(=O)Nc4ccc(I)nc4)cs3)c[nH]c2c1 C1(=O)C(CC(C)C)CN1.C1(=O)C(C(C)O)N1.C1(=O)CCCN1C.CN N1(C(C2CC(O)(CC#C)C2)=O)CCC(NC(c2ccsc2Cl)=O)C(C)(C)C1 C1(C(N(C2CN(C(C(C(CC)O)C)=O)C2)C)=O)(CC)CCC(F)(F)CC1 C(CC(C(=O)NCC1CCN(C(=O)C(C)N(C)C)C1)NC(C)=O)SC N1(C(C(CSC)C)=O)CC(N(C)C(c2cncc(C#N)c2)=O)C2(CC2)C1 c1(C(N(C(CN(C(C(CC(C)C)O)=O)C)C)C)=O)cc2ccsc2n1C Cc1cc(C(=O)N(CC(C)(C)NC(c2csc(Br)c2Cl)=O)C)[nH]c1C N1(C(C=C(C)C)=O)CC2OCCN(C(=O)CC3CC4C=CC3CC4)C2C1 CC(CCO)CCN=c1nc(N2CCCC3(CCCO3)CC2)cc[nH]1 C(=O)(C(O)C(C)(C)SCC)NCCN(C(C(C)(C)NC(=O)OCCC)=O)CC CC1CCCN(CC(N2CCCC(CNC(c3ccn(C(F)F)n3)=O)C2)C)C1 Cc1cc(F)c(C(=O)NC2CCN(C(c3cccc(F)c3Br)=O)CC2O)cc1F c1(C(=O)NCCN(C(C2CC2Cl)=O)CC2CC2)cc(-c2ccccc2)ccc1Cl C1(C(C)C)CCC(C(=O)NC2CCCC2NC(C2(c3ccno3)CCC2)=O)CC1 N1(C(C(CC)(C)C#N)=O)CCC2(C1)CN(C(=O)CC1COC(C)(C)C1)CC(C)O2 C(=O)(C(CCCCO)NC(=O)CC1CC=CCN1C)NCC1CC(COC)C1 c1(CC)ccc(C(=O)NCC2(C(N)=O)CN(C(c3occc3C)=O)C2)c(OC)c1 C=CCC(CC(F)F)C(=O)NCC(c1cccc(C)c1)NC(=O)C(C)S(C)(=O)=O c1(C(C(=O)NCCC)N(C)Cc2cc(C3CC3)on2)cnn(CC(F)F)c1 C(CC(=O)N1CCN(C)C2(CC2)C1)(C(C)(C)C)NC(C(C)=C1CC1)=O N1(C(c2nc(C)c(Br)cc2)=O)C2CCCC1CC(n1ccnn1)C2 c1(C(C)=O)ccccc1C(=O)NCCC(O)CNC(=O)C=CC1CCCC1 N1(C(CC2ON=C(C)C2)=O)C(C(=O)NC(C)Cn2cc(C)cn2)CCC1C1CC1 C#CCCCCS(C)(=O)=NC(=O)C(c1ccccc1C)N1CCCCC1 c1(C(=O)NC2CC2C(=O)Nc2ncccc2C(F)(F)F)cnc(O)nc1O C1(NC(c2scc(C)c2)=O)C2CCN(C(=O)CCn3cnnn3)CCC12 c1(C(=O)NC(CC)(CC)CCNC(C2CC2Cl)=O)ccc2ccccc2c1 C1(NC(=O)NCC(c2c(OC)ccc(Cl)c2)O)CCC12CCCCC2 c1(C(=O)NCCNC(C23CCCCC2C3Br)=O)sc([N+](=O)[O-])cc1Cl C1N=C2Nc3cccc(c3S2)Oc2ccc1cc2.C(CC(C)C)(OCC)OC c1(C(N2CC(NC(c3cc(C)sc3C)=O)C2)=O)ccnc2ccc(F)nc12 C12(C(=O)OC)C3C4C1C1C2C3C41Oc1ccccc1.C12CCCC1C(=O)N2 C(=O)(C(Cc1cn(-c2ccncc2)nn1)NC(C1CCN1S(C)(=O)=O)=O)OC C1(C(N2CCCC(CCC)(NC(c3csnn3)=O)C2)=O)Cc2cc(F)ccc2O1 c1(C(N(CC(CC)NC(=O)CC2CCC(=O)O2)C)=O)cc([N+](=O)[O-])ccc1C NS(=O)(=O)c1ccc([N+](=O)[O-])c(NCCc2ncc[nH]2)c1 N#Cc1ccc(Br)c(F)c1NC(C1CC2CC2N1C(=O)CCN1CCOCC1)=O C1(NC(C(CSC)O)=O)(CO)CCCN(C(c2cccc(C)n2)=O)C1 CCCCC(C)C(C(=O)NC1CC1)N1CCc2cc(C(C)(C)C)ccc21 N1(C(c2nc(-c3cccc(OC)c3)oc2C)=O)CCN(C2CC2)C2(CCOC2)C1 C1(CCNC(CN(CC)CC)=O)CCCN(C(c2c(C)oc(C)c2C)=O)CC1 c1(OCCC)ccc(C(=O)NCCN(C(=O)Cc2csc(S)n2)C(C)C)cc1N N1(N(c2csc(Cc3ncc(C#N)cc3Br)n2)C(C)=O)CCc2sc(Br)cc2C1 Cc1ccc(C(=O)NCC(=O)NCCNC(=O)CC(C)N2CCCC2=O)s1 C12(CNC(=O)C(F)CC3CCC3)CCC(C1)N(C(c1coc(CO)c1)=O)C2 N1(C(C2(OCC)CCC2)=O)CCC2(CC1)CCN(C(=O)C(C#N)CC)C2 C1(NC(c2cccs2)=O)CC2CC1N(C(c1cc(Br)c[nH]1)=O)C2 N1(C(CC=CCC)=O)CCC(OCC(=O)OCC)C1 Cc1cc(C)c(C(N2CCC(N(C)C(C3CC(C(F)F)C3)=O)C2)=O)cc1C CCC(CC)C(F)C(=O)N1CC(C)CCC1CNC(c1cc2n(n1)CCCN2)=O N1(CC(=O)NCC(n2cc(-c3cnc(CC)o3)nn2)C)CCOCC1=O C1(C(=O)NC(C(C)C)(C)CO)CN(C(c2cncc(F)c2)=O)CC1(F)F C1(C(=O)Nc2nc(C)c(C)s2)C2CCC(C2)C1NC(c1cnnc(Cl)c1)=O CCCC(C(=O)N(C(C)CN(C(=O)CCc1cc(Cl)no1)C)C)c1ccccc1 c1(SCC(=O)NCC(C)(CC)NC(CCC=C=C)=O)cc(=O)n2ccsc2n1 C1(C(N(CCSC)C)=O)CC(F)CN1C(=O)CC1CCCC1O C(C)(C(=O)NCCC1(O)CN(C(=O)C(C)N(C)C)C1)(c1ccccc1)OC C(=O)(C(O)CC(F)(F)F)NC(CC)CNC(c1ccc(N2CCCCC2)nc1)=O N1(C(c2cc(C(=O)OC)on2)=O)CCN(C)CC1CNC(=O)C(C)(CO)OC c1(C(C(=O)N(C2(CNC(C3CCC4CC34)=O)CC2)C2CC2)(F)F)ccc(Cl)cc1 Cc1cccc(O)c1C(N1CC2CN(C(c3ccc(I)cc3)=O)C2C1)=O CCCC(C)(C)C(=O)NCC(O)CCNC(=O)CC1CC(OC)C1 c1(C(=O)NC(C)(C)CCNC(C2CC23CC3(F)F)=O)nccc2cccnc12 C(=O)(CC(C)C(=O)N1CC(OCCNC(=O)CC2CC(C)OC2C)C1)OC N1(C(C(C)(C)NC(=O)OC)=O)C2CCC1C(F)C(NC(=O)CC(F)(F)C(F)F)C2 c1(CN(C(c2cc(C(C)C)on2)C(=O)NC2COC2)CCC)ccccc1F N1(C(C(CC)NC(C)=O)=O)CCC(O)C(C(N2CCCC(CCOC)C2)=O)C1 CS(=O)(=O)c1ccnc(NC2CN(C(c3cncs3)=O)CC3(CCC3)C2)n1 Cn1cc(C(N2CCC(NC(=O)C=CSc3nc[nH]n3)C2)=O)cn1 c1(OCC)cc(C#N)ccc1OC(C(=O)OC)C(C)C C1(CC(=O)NC(CSCC)C(=O)NC(C)C(C)F)OCCC1(C)C C1(C)(CNC(C(CCC)N(C)C)=O)CCCN(C(=O)Cc2cc(C)cs2)C1 CC(C)CCCC(=O)N1CCCCC1C1(NC(=O)COCCF)CC1 C1(N(C)C)CCC(C(N2CCC(SC3CCOC3)C2)=O)CC1 C1(CC(=O)N2CCN(CCO)CC2)OCCOC1(C)C.C(=O)(C1CC1)OC c1(C(N2CC(C)(C(=O)NC(CCC)c3ccco3)C2)=O)[nH]cc(C)c1C Cc1cc(C=CC(=O)NCC2CCN2C(=O)C(c2cnn(C)c2)C)ccc1F c1(C(=O)NCC2CCN(Cc3n(C)ncc3Br)CC2)cc2ccccc2cn1 NS(=O)(=O)CCCC(=O)N1CC(O)C(O)C1CNC(C1CC2CC2C1)=O c1(COC(C2CC2c2cc(Br)cc(Br)c2)=O)noc2c1CCCCC2 C1(C(=O)NC2CC2CNC(=O)C(C)Nc2nc(C)cs2)(OCC)CCOCC1 c1(C(=O)NC2CC(NC(C3(C)COCCO3)=O)C2)ccc(S(N)(=O)=O)nc1 N1(C(CNC(=O)NC)=O)CCC2(CC1)CC2(CO)CNC(c1ncccc1C)=O C1(CCC(=O)NCCC(C)NC(Cc2ccc(SC)o2)=O)COC(C)(C)O1 C#CCCCCCCCNC(=O)C=CC1CCCN1C(c1ccc(C)nc1O)=O c1(C(=O)NC2(C(=O)OC3CCN(C(=O)OC)C3)CCSC2)cnc(N)cn1 C1(CNC(C(C)SCC)=O)(OC)CCCN(C(=O)CCSCC(C)C)C1 C1(C(=O)NCC2(C#N)CCC2)(COC)CN(C(c2ccc(C)o2)=O)C1 CCC(C)(C)CCCC(=O)NC(C)(C)CNC(c1cc([N+](=O)[O-])ccc1OC)=O c1(OCC)nc(C)ccc1C(=O)NC1CCC1NC(=O)C=Cc1cscn1 Cc1ccc2scc(C(N3CCC(C)C(NC(=O)Cc4cscn4)C3C)=O)c2c1 c1(CC(N2CCC(CNC(C(C)NC(C)(C)C)=O)CC2)=O)ccc(Cl)c(Cl)c1 Cc1cc(F)cc(C)c1C(=O)NCC#CCNC(C1(C(C)C)CCC1)=O C1(NC(c2cc(C)sc2)=O)CC2CCC(C1)N2C(C1(CN2CCCCC2)CC1)=O C#CC1CN(C(=O)CC2C(=O)N(C)N=C2C)CCN1C(=O)COc1cc(C)on1 CC1CCCC=C1C(=O)NCCCCCNC(=O)Cn1ccc([N+](=O)[O-])n1 Cc1ccc(C#N)cc1S(=O)(=O)N1CCC2C(CCN2C(c2cc(C)[nH]n2)=O)C1 C12(C(N(CC(C)O)CCNC(C(CC)CC(F)F)=O)=O)CC3CC(C1)CC(O)(C3)C2 c1(-c2cccc(C)c2)nnc2ccc(=NC3CSC(NC(=O)C(C)C)C3)[nH]n12 C1(CNC(C(C)N(C(C(C#C)(C)C)=O)C2CC2)=O)CCC2(CCC2)O1 C#CC1(O)CC(C(N2CC(NC(c3nccn3CC=C)=O)C(CCC)C2)=O)C1 CCCCC(C)(F)C(=O)NCCOC1CCN(C(c2cncc(F)c2Cl)=O)C1 C1(CCC)CN(C(=O)CCC(C)(C)N(C)C)CCN1C(=O)CNc1ccncc1 S(=O)(=O)(c1ccc2[nH]c(=NCC(CO)OC)ccc2c1)NC(COC)CO N1(C(c2ccc(CC3CCCC3)o2)=O)CCOC(C(=O)NOC2CC2)CC1 C1(C(N2C(C(C)C)CN(C(C3CCN(C)C3=O)=O)CC2)=O)CCc2ccnn2C1 c1(C(=O)NC2C(NC(CC3(OCC)CCC3)=O)COC2)ccc(CC)c(F)c1 CCC(CCC(=O)N1CCC(NC(c2ccc(Cl)cc2OC)=O)C1(C)C)OC CCC(C)C(C(=O)NC(c1ncc(C)cn1)C)N(C(=O)C=C(C)C(C)C)C C#CC1(NC(C2C=CCN(C(=O)CCCOC(C)=O)C2)=O)CCC(C)(C)C1 c1(CC(N2C(C(=O)NC(C)CCc3cn[nH]c3)C=CC2)=O)ccc(O)cn1 C1(NC(C2(CCCC)CC2)=O)CC2CC1N(C(c1csc(CC)n1)=O)C2 c12noc(n1)CN(C)C2.C1(C(=O)NC)CCN(c2ccccc2)C1 C1(NC(C(c2ccc(Cl)s2)C)=O)COCCN(C(C2(S(C)(=O)=O)CC2)=O)C1 n1(C(C(=O)NCC2(F)CC(NC(C3(C#C)CC3)=O)C2)C)nc(C)c([N+](=O)[O-])c1C N1(CCC(N2CCN(c3ccc(Cl)cc3)CC2)=O)CCC(F)C(O)C1 C1(NC(c2c(OC)ccs2)=O)C2CC1N(C(C1CCCN1C(N)=O)=O)C2 Cc1ncc(C(N2CC3C(CC(=O)NC4(CO)CCC(C)C4)C3C2)=O)n1C c1(NC(C2(c3ccccc3)C(C)C2)=O)ccc2c(c1)CN(C)C2 CC(CCN=c1[nH]c2c(cc1C#N)CN(C)CC2)NC(C1(C)CC1(F)Cl)=O Cc1ncccc1NC(C1CCC1NC(=O)CC1COCC1O)=O c1(C(=O)NCC2(CCNC(C34CCC(C3)C4)=O)CC2)coc2cc(F)ccc12 c1(C(=O)NCC(C)NC(C(c2cccc(C)c2F)O)=O)cc2n(c1)CCSC2 c1(SC)cc(C(=O)NC(C)CCN(C(=O)C=Cc2cccs2)C)cc(Cl)c1 n1(CCC(=O)NCC2(OC)CN(C(c3cc(C)c(C)o3)=O)C2)cc[nH]c(=O)c1=O c1(OC)cc(CO)ccc1C(=O)NC1CCN(C(=O)Cc2cccnc2)C(C)C1 N1(C(c2nc(C)sc2)=O)C2CCCC1CN(C(c1nc(C3CC3)ncc1Cl)=O)C2 C(=O)(CCCCCC(C)O)NCCCN(C(C(CC)c1cccnc1)=O)CC c1(NC(C2CN(C(=O)CCc3ccc[nH]3)CCC2O)=O)ncc(I)cc1[N+](=O)[O-] C(=O)(CC(C)C(C)(C)C)NC1C(CC(=O)NC(C)CN2CCCC2)C(O)C1 N1(C(c2c(C)c[nH]n2)=O)CCC2(CC1)CN(C(C1C3CCC(=O)C13)=O)C2 c1(CSC)cc(C(N2CC3(C2)CN(C(C2(C)CCC2)=O)C3)=O)ccc1F N1(C(c2c(C)nn3c2CCCC3)=O)CCc2cc(Br)cc(F)c21 c1(NC(N2C(COC)(CO)CCC2)=O)cc2[nH]ccc2cc1C#N CCCC(C(=O)N1CCCC1C(C)NC(c1oc(CO)cc1C)=O)NC(N)=O N1(C(CC(C(C)C)C)=O)C(CNC(c2nc3ccccc3[nH]2)=O)CC2COCC12 Cc1cnc(C(N2CC(CNC(=O)CCn3cc(C)cn3)C2)=O)c(F)c1 N1(c2cc(NCCc3ccc(C)c(F)c3)ncn2)CC(=O)Nc2ccccc2C1 N1(C(C=COCC)=O)Cc2occ(C(N3CCC(O)C(C)(CO)C3)=O)c2C1 C(=O)(C(C)(C)C(N)=O)NCCCOCCOCCNC(CC(C)F)=O C=CCC(CNC(C1CC1c1ccccc1)=O)NC(=O)C(C)=C(C)CC O=C(C1CCCc2cccnc21)N1CCN(C(=O)C2=COCC2)C(CF)C1 N1(C(C(N2CCCCC2)C)=O)CC(C2CC2C(N2CC(S(C)(=N)=O)C2)=O)C1 c1(OC)ccccc1NC(N1CC(F)CC1C(N1CCC(F)(CO)C1)=O)=O N1(C(c2c(C)snn2)=O)CCCC(CCNC(=O)C(N2CCN(C)CC2)C)C1 c1(C(=O)NC2(C)CCN(C(c3c(C)cnn3C)=O)CC2)cnc2c(c1)NCC2 C1(c2nnnn2CCC2CC2)(NCC(=C)Br)CN(C2CC2)CC1C C(C(=O)NCC12CCCC1OCC2)(C(C)(C)C)NC(c1n(CC)nc(C)c1)=O C1(O)(C(N(C(C)CO)C(C2(N(C)C)CCCC2)=O)=O)CCN(CC)CC1 C1(NC(C2(CSC)CCC2)=O)CC2CCC1N(C(=O)CNC(=O)OC(C)(C)C)C2 CC(C)CCCC(C)C(=O)NC(C1(O)CCN(C(C2CCCC2(C)C)=O)CC1)C Cc1nc2ccc(NC(=O)NCCc3cncn3C)cc2nc1C N1(C(CSCCOC)=O)CCOCC1C(=O)NC(Cn1cncn1)CC c1(C(=O)NC2C(NC(CCC=C)=O)CCC2)ccc2nccc(Br)c2c1 S(=O)(=O)(c1cccc(=NC(C)CCCO)[nH]1)NCC1(SC)CCC1 C1(C(=O)NCC(C)(C)NC(=O)CSc2nc[nH]n2)CCCCC1C1CC1 C(=O)(CCCS(N)(=O)=O)N1CCC(N(CCC)C(c2cc(F)cc(F)c2)=O)CC1 C12(C(N3C(C=C)CC3)=O)CC(CO)(CN1C(=O)C(CCC)N(C)C)C2 N1(c2nccc(OC)n2)CC2C3CCC(C2C1)N(C(=O)CN1CCCNC1=O)C3 N1(C(C(c2ccc(C)s2)C)=O)CCOC(CNC(=O)Cc2cncn2C2CC2)C1 N1(C(c2c(CC)nnc(C)c2)=O)CC2CCC1C(CO)C2 C12(NC(C(C)C3CCC3)=O)CC(C1)N(C(=O)COCc1cccnc1)C2 Cc1cc(F)cc(C)c1C(N1CC2(C1)SCCC2NC(=O)CC(=O)NC1CC1)=O C(CC1=CCN(C(=O)CC2CCC2OC)CC1)NC(CC1(OC)CCOCC1)=O N1(C(CC2CC(=C)C2)=O)CC(C2CN(C(c3cncc(F)c3)=O)C2)C1 C1(F)(C(=O)NCC(C)N(C)C)CCN(C(C2CCC(C)(C)C2)=O)CC1 C(=O)(C(C)CCOC)NCC(=O)NCC(=O)NC(CC)C1CC1 C1(C(=O)NC2(CC=C)CN(C(=O)Cc3cncn3C3CC3)C2)OCC2CCCC12 C(=O)(C(=O)CC(C)C)NCC(C1CCCC1)NC(c1cc(C)no1)=O N1(C(c2cc(SC)nn2C)=O)C(CNC(c2scnc2C)=O)CC2CCCC12 C(c1ccc(C(N)=O)cc1)=CC(=O)NC1CC(CCNC(c2nc(C)sc2)=O)C1 N1(C(C(CCC)F)=O)CCC(C)C(CC(=O)Nc2cn(C)nc2C2CC2)C1 N1(C(C2CN(C)C(=O)CC2)=O)CC2CCC1C(NC(C1CN(C)C1)=O)C2 c1(OCC)cc(CNC(Cc2ccncc2Br)C(=O)O)cc(F)c1 n1(CC)cnc(C(=O)NCC2(C(C)(C)O)CN(C(=O)CCn3cc(Cl)cn3)C2)n1 C#CCC(C)(C(=O)NCCC(O)C(F)(F)F)NC(c1cnsc1)=O C(C(CC(C)C)C(=O)N1CC(C)C(C)(CNC(=O)CSC(F)(F)F)C1)OC Cc1cc(C(=O)NC2CC(CNC(=O)C(C)C3CC3)C2)c(Br)cc1F C1(NC(=O)C2=NOCC2)CS(=O)(=O)CC1NC(=O)CSc1ccccn1 Cc1cccc2[nH]c(C(N3CCN(C(c4ccc(F)cc4N)=O)C4CC34)=O)cc12 CC(O)(CNC(c1csc(C2CC2)n1)=O)CNC(=O)C=CSc1nc[nH]n1 C1(NC(CC(C)SC)=O)CCC2CN(C(=O)C=Cc3ncc[nH]3)CC2C1 c1(C(=O)NC2C(CNC(C3CNC(=O)N3)=O)CCC2)cnc2n1CCOC2 C1(C(=O)NCC(C(C)C)NC(C2(C)COC2)=O)CCc2cnnn2C1 c1(C(=O)NC2CC(NC(c3ccc4nccnc4c3)=O)C2)ccc(F)c2occc12 c1(C(C(=O)N(CC(C)NC(c2c(CC)scc2)=O)C)(F)F)nc2ccccc2s1 c1(C(CCC(=O)N(C(CCNC(C(C(C)C)O)=O)C)C)=O)ccc2c(c1)CCC2 C1(NC(=O)Cc2ccsc2)CN(C(c2occ3c2CCCC3)=O)CC(F)(F)C1 N1(C(=O)Cc2cccs2)CC2CN(C(c3cc4scnc4[nH]3)=O)CCC2(CO)C1 CC1(C)CCCN(c2nnc(C(F)F)o2)C1CNC(=O)CCc1nc[nH]n1 Cc1[nH]c(=NC2CCCN(C(=O)CC(C)(O)C(F)(F)F)C2)ccc1C#N C1(C(=O)NC2C(NC(c3cc(OC)ncn3)=O)C2)CCN(C)C(=O)C1 Cc1ccc(CC(C(=O)O)NC(=O)Cc2conc2C)cc1F c1(OCC)nc(NC(c2ccccc2)CCC2CCCCN2)ncc1C c1(C(=O)Nc2cc(C(=O)OC)sc2)ccc2ncc(-c3cc(O)ccc3F)n2c1 C1(CNC(C23CC(NC(CC(CC)SC)=O)(C2)C3)=O)COCC(=O)N1C c1(C(=O)NCCn2cc(CCC(=O)O)nn2)cc(F)c(F)cc1Cl N1(C(Cn2c(C)cc(C)n2)=O)CC(C)CCC1CNC(C1(CO)CCOCC1)=O c1(C(N(C)CCN(C)C(c2ccc(C(C)(C)C)s2)=O)=O)cc(N)cc(O)c1 N1(C(c2c(C)cno2)=O)CC(C)(C)OCC1CNC(=O)COC1(C)CCOCC1 N1(C(=O)Cc2csnn2)CCOC2(C1)CN(C(c1cc3ncccc3s1)=O)C2 c1(CNC(CN(C)CC)=O)cc(C(=O)N(CC(C)C(C)C)C)on1 c1(C(=O)NCC2C3CN(C(C(CC)O)=O)C(C3)C2)nc2ccccc2o1 CN=c1[nH]c(C(=O)NC2CCCN(C(c3cccc(Cl)c3)=O)C2)cs1 N1(C(C(COC)N(C)C)=O)CCC(C2(NC(=O)CNC(c3cccs3)=O)CC2)C1 C(CCN=c1nc(N2CCC(CC3CC3)CC2)c2sccc2[nH]1)c1cc(C)no1 CC1OC(C)CC1CC(=O)NCCOCCN(C)C(C1(CO)CC(F)(F)C1)=O N(C1CCCc2occc21)C(C(N(C(C1CCCC1)=O)C1CC1)C1CC1)=O CCC(CCCC(=O)NC1CCN(C)CC1C)NC(C1(n2cccn2)CC1)=O C(CNC(=O)CCc1cscn1)(C(C)(C)C)NC(CCOCCCOC)=O c1(C(=O)NC2(C)CCN(C(CC(C=C)C)=O)C2)cc(OC(F)F)cc(Br)c1 C1(NC(c2ccn(CC(F)F)n2)=O)CCC2CN(C(C3OCCCO3)=O)CC2C1 C(=O)(C1=CS(=O)CCC1)N1CCC(=CCNC(C2ON=C(C)C2)=O)CC1 N1(C(Cn2c(C)ccn2)=O)CC2(NC(C3CC4(CCC4)CO3)=O)CCC1CC2 c1(C(=O)NC2CCCN(C(C(CCC)CC)=O)C2C)cc(C)c(F)cc1N C(CC(=O)NC(C(CC)C#N)=O)(C(C)OC)C1N(C(C2C3CCCOC23)=O)CCC1 C1(C(=O)NCc2nnc(CC)s2)CCN(C(c2ccc(O)nn2)=O)CC1O C(=O)(CC(C)(C)C)NC(C)C(N1CCOCC1CNC(c1sncc1Br)=O)=O CCCCC(C(=O)NCCC(O)C(C)C)NC(=O)CN1CCCCC1C c1(C(N2C(C(C)NC(c3c(C)cno3)=O)CCC2)=O)ccc(Cl)cc1F N1(C(CC(=O)OCC)=O)CC2CCCN(C(C3CC(F)(F)C3(F)F)=O)C2C1 c1(CNC(C2(C)CC(C)OCC2)=O)nc2c(s1)CN(C(=O)C(C)(F)F)CC2 n1(CC)c(C(N2CCN(C(=O)C(F)OC)CC2C)=O)cc2ccccc12 CC(C)(F)CCC(=O)NC12CCOC(CNC(C3CS(=O)(=O)C3)=O)(C1)C2 CC(CC(=O)NCCN(C(=O)CSC(C)(C)C)CC1CC1)n1ccnc1 CC1=C(C(=O)Nc2nccc3cc[nH]c23)C(C)(C)CCC1 Cc1nn(C)c2ccc(C(=O)NC3CC(NC(C4CCC(F)(F)C4)=O)C3)cc12 C1(C(N(C(CC)CSC)C)=O)C(C)OCCN1C(=O)C(C)NC(=O)C1CC1 N1(C(c2ccc(SCC)nc2)=O)CC(NC(C2CCC(=O)C2C)=O)CC12CCC2 C1(C(N2CC(C(N)=O)C(O)C2)=O)CCN(C(=O)C2=CCCC2)C12CCC2 C1(CNC(C(c2ccnn2C)C)=O)CCC(NC(C2C=CCC2)=O)CC1 C1(C(N2C(C#C)CC2)=O)(NC(c2nc(C)c(C)s2)=O)CCN(C)C1 c1(C(=O)NCC(CNC(c2n(CC=C)ccc2)=O)C)c2c(nn1CC)CCCC2 n1(CC(=O)NC(CC)(C)CNC(=O)C2=C(Cl)CC2)cc([N+](=O)[O-])cn1 C1(C(N2CCC(O)(Cn3cc(CCCC=C)nn3)C2)=O)CC12CCOC(C)C2 N1(C(C(CC(=C)C)C)=O)CCCC2(C1)CN(C(c1ccc(C)c(C)c1Cl)=O)C2 C(=O)(CCCCC(C)=O)NCCCNC(c1c(OC)cncc1)=O C1(NC(CCSCCCC)=O)CCCC12CN(C(c1cc[nH]c3nccc1-3)=O)C2 C(CN=c1nc2ncn(C)c2c(Nc2ccsc2)[nH]1)NC(CN(C(C)C)CC)=O Cn1nnc2c1CCN(c1cc(NC3CCc4n[nH]cc43)ncn1)C2 Cc1ccc(C(=O)NCC2CC(NC(C3(C)C=CCC3)=O)C2)cc1F N1(C(C)=O)CCC(C(N2CCCC(N(N3CCCCC3)CC3CC3C)C2)=O)CC1 c1(C(C)C)cc(C(=O)NC2CCC(NC(C3CC34CCCC4)=O)C2)nn1C c1(C(=O)NC(CN(C(CCC)=O)CC)C)ccc(Oc2ccccc2)cn1 C(=O)(CC(CC1CC1)NC(=O)COCCCN=[N+]=[N-])N(C(CO)CO)C C12(C(=O)NCC3(NC(c4cn(C)[nH]c4=N)=O)CCOC3)CCN(CC1)CC2 C(C)(CCC(=O)N1CC(C)CC1C(N1CCC=CC1CC)=O)OCC c1(NC(=O)CCC2CCOC2)cc(CC(=O)NCCc2ccsc2)no1 N1(C(c2c(C)sc(-c3nc[nH]n3)n2)=O)CCCN(C(C2CCCO2)=O)C(CO)C1 CCCC1CNC1=O.C1(NC(=O)OC(C)(C)C)(CC)CCCSC1 C12(CNC(C(C)(N(C(C3C(C)CCO3)=O)C)C3CC3)=O)CCC(CO1)C2 C1(CNC(CN(C2CC2)CC)=O)CN(C(c2cc(CC3CCC3)c[nH]2)=O)CCO1 C1(CC(C)C)CCN(C(=O)CSCCNC(=O)Cc2ccc[nH]2)C1 Cc1c(C(=O)NCC(O)CN(C)C(c2sc(F)cc2Cl)=O)ccn1CCO CC(C)C(CCN(C)C(C12CC3CC1C2C3)=O)NC(C1CC1C)=O C1(C(=O)OCCC2(CC)OCCO2)CCC2CNCCC2C1 C1(CC)(NC(=O)CC2COC(C)(C)C2)CCS(=O)(=O)CC1 C1(C(=O)NC(C(C)C)C(C)(C)O)CN(C(=O)CCc2ccccn2)CC(C)(C)C1 Cn1cc(C(N2C3CCC2C(CNC(=O)CSc2ccccn2)C3)=O)ncc1=O CC(C)C(C)C(C)CC(=O)NCCCCN(C(=O)C(C)(C)c1ccnn1C)C c1(C(=O)NCC2(CNC(C(C)(C)OC)=O)CCOCC2)cc2n(n1)CCCC2=O c1(C2C(NC(=O)NC3CC(CNC(=O)OC(C)(C)C)C3)C2)cc(F)cc(Br)c1 C1(C)(C(=O)NCc2c(C(N(C(CCSC)C)C)=O)c[nH]n2)COC(=O)N1 N1(C(C2(O)CCC2)=O)CCCC(F)(C(N2C3CSCC2C3)=O)C1 C(=O)(CCCc1nc(C2CC2)no1)N(C(C)CNC(=O)COC)CC CN1CC(C)(C)CC1C(N1CCC(F)CC1C(=O)NC1(n2cccn2)CC1)=O Cc1nc(=NCC2CCCC(NC(C3(C(=O)N(C)C)CC3)=O)C2)[nH]cc1[N+](=O)[O-] CC1=C(C(=O)N2CC(C)N(C(=O)CCCc3cnn[nH]3)CC2C)CCCC1 c1(C(=O)NC(CC(C)Nc2cc(SC)nc(SC)n2)C)nccc2ccccc12 C12(C(N(C)CCN(C)C(C3(Cl)CC3(F)F)=O)=O)CCC(C1)S(=O)(=O)CC2 c1([SH](C2ON=C(CC)C2)(Cc2ccnnc2)=O)ccc2oc(O)nc2c1 N1(C(C2CC(=O)CC23CCC3)=O)CCSC2COCCC12 c1(C(=O)NC2(CC=C)CN(C(c3snc(C)c3N)=O)C2)cc(F)c(F)c(Cl)c1F N1(C(c2c(CCC)nns2)=O)CCCN(C(=O)CNS(N)(=O)=O)C(CO)C1 N1(C(COCCC=C)=O)CCC2(C=C(C(=O)NCC3(C)CCCS3)C2)C1 C12(CNC(C=C(C)c3cccs3)=O)CN(C(c3occc3C)=O)CC1CCO2 N1(CC(=O)NCC2N(C(C(CCC#C)O)=O)CCC2)C(=O)c2cccnc2C1=O C1(NC(CSCCC)=O)CCCC1C(=O)OC(C)(C)C.c12cc(no1)NC(=O)C2 c1(CC)ocnc1C(=O)NCC1(F)CC(NC(=O)C(CN(C)C)N(C)C)C1 c1(OC)ncc(Cl)c(=NC2CC3CC(C2)N(C(c2cccc4cc[nH]c24)=O)C3)[nH]1 N1(C(c2n(C)c(C(F)(F)F)cc2)=O)CCC=C(C(=O)Nc2cc(F)c(F)c(F)c2)C1 N1(C(C2CC(=O)OC2)=O)CCCC(C(N2CCC(OC3CCC3)CC2)=O)C1 CCC(CCCC(=O)N(C1CCC(C)(C)CC1)C)NC(=O)CC1OCCCO1 C(=O)(C(C#N)(CC)CC)N1CC2(CN(C(c3c(C(C)=O)cc(Cl)s3)=O)C2)C1 C1(NC(=O)CCc2ncc[nH]2)CN(C(c2ccon2)=O)CCC1C(F)(F)F C1(C(=O)NCC(C=C)O)(CC=C)CN(C(C2CCCO2)=O)C1 N1(C(C(CC)=CC)=O)CCCCC1CCCNC(C1(CC)CCCO1)=O C1(CC(=O)OCC)CN(c2ncccc2C(F)(F)F)CC(C)O1 c1(C(=O)NCCC(C)NC(c2nnc(O)nc2O)=O)ccc(C(F)F)c(F)c1 C1(CC(=O)NCc2cc(CO)[nH]n2)CCCC(NC(c2nncn2C2CC2)=O)C1 CCC(CC)C(=O)NC1CCCCC1CNC(c1ccccc1)=O C12(COC)CN(C(c3cnc(C(C)C)nc3)=O)C(CNC(=O)CC(C)SC)(C1)C2 CC(C)C(CO)C(=O)N1CCCC1C.C1(C)(C(=O)OC(C)(C)C)CCCN(C)C1 CCCC(O)CC(=O)NC(Cc1ccccc1)CCNC(=O)CCC1CCOC1 C1(CC(=O)NC(C)CNC(=O)CC2CC(=O)NC(=O)C2)C2CC3CC(C2)CC1C3 C(=O)(C1CCCc2n[nH]cc21)NC(CNC(c1cc(C)nc(C)c1O)=O)(C)C c1(C(CCNC(c2n(CCOC)nnn2)C2(C)COC2)O)ccc(Br)cc1 C=C1CCC(C(N2CC(OC)CC2CNC(=O)CNC(=O)CC)=O)CC1 c1(C(N2CCC(CCNC(C=CC(C)=O)=O)C2)=O)ccc2nc(O)n(C)c2c1 c1(SCCCC(=O)OCCC)ccc(NC2CCN(OC)CC2)cc1C c1(C(=O)NC(C)CN(C(=O)C=CCN(C)C)C)cn(CCO)nn1 C=CC1CC(N=c2[nH]c(=NC(C)c3ccc(Br)s3)[nH]c3ccsc23)C1 C1(C(N2CCCC(NC(CCCC#CC)=O)(CC)C2)=O)CCC2(CC1)CC2(F)F C1(CC(N2CC(CN(C(=O)CCC(F)F)C)OCC2)=O)CCCCC1(C)C C1(C2CCN(C(=O)CC(c3cccs3)N(C)C)C2)(NC(CCC(=C)C)=O)CC1 C=CC(C)(C)CC(=O)NC(C)(C)C=CC(=O)NC1CCN(C)CC1C N1(C(C#CC(=O)O)=O)CCC2CCC(C1)N2C(=O)COC1CCCCCCN1 C1(C(=O)Nc2cc(C(=O)OC)c(C)nc2)CCc2n[nH]c(C)c2C1 N1(C(c2cc(C(N)=O)oc2)=O)CC(CNC(=O)C(F)=CC2CC2)OC2CCCC12 Cc1cccc(C(CNC(C2CC2(C)C)=O)NC(c2ccc(-c3cccs3)[nH]2)=O)c1 C(=O)(CCCCC(F)(F)F)NC1(C)CCCN(C(CC2CCC(C)(C)CO2)=O)C1 Cc1cccc2c1CC(C(=O)NC1(CNC(c3cc(C)n(C)n3)=O)CCOC1)O2 C(=O)(C(F)(CNC(C1CC(=O)NC1(C)C)=O)C(C)C)NC(C(=O)NCC)CC c1(CC)ccc(C=CC(=O)NC2CN(C(=O)CCn3ccccc3=O)C3CC23)o1 C1(N(C(=O)CN2CCSCC2)C)CC2CC1N(C(=O)C=Cc1cn(C)nn1)C2 C12CCN(C1)C(=O)C(C)O2.C(CC(=O)NCCO)OC.C(C)(C)(C)O.C1CNC(=O)N1 N1(C(c2cc(C)nn2C)=O)CCC(CNC(=O)CN2CCOCC2=O)C(C)C1 CC(C)C(C)C(=O)NCC(C)(C)CNC(c1ccc(OCCN(C)C)nc1)=O N1(C(CCC2CC(OC)C2)=O)CC(NC(c2conc2C)=O)C2CCCC2C1 N1(C(C(C)O)=O)CC2CC1CCN2C(=O)CCc1cc(Cl)no1 C(CC(=O)NCC1(C)CCOCC1)(C(F)(F)F)NC(Cc1c(C)cnn1C)=O c1(C(N2CCCC(C3N(C(C=CC=CC)=O)CCCC3)C2)=O)cc(F)c(Cl)cc1Cl N1(C(C(Cc2ccco2)NC(c2cc(CC)[nH]n2)=O)=O)C2CCCC1COC2 c1(C(N2CC(NC(CCCOCC)=O)C(C)(C)C2)=O)c[nH]c2cccc(C#N)c12 c1(SC)nccc(=NC(=O)CN2CCN(c3ccc(C(F)(F)F)cn3)CC2)[nH]1 Cc1cc(O)c(Cl)cc1C(=O)NCC1CCN1C(C12CC1COC2(C)C)=O C1(C(=O)OC)CCC(C2CCCCC2)CN1C(C1CC1c1ccco1)=O C1(C(C)NC(C(C)OCC(C)C)=O)CCCCN(c2cc(OC)ncn2)C1 N1(C(c2c(C)ccc(F)c2)=O)CC2(CC(C(=O)NCC3CC=CC3)CO2)C1 N1(C(c2c(Br)ccc(C)c2)=O)CCC2(CCN(C(c3cnc(O)s3)=O)C2)C1 N1(C(c2scc(C(=O)OC)c2)=O)CC(C2CN(C(=O)C(C)CC(N)=O)C2)C1 C#Cc1ccc(CCCC(=O)Nc2cnn(CCN3CCNC3=O)c2)cc1 C#CC1CCCCN1C(c1ccc(CNC(=O)C(O)C=C)nc1)=O Clc1cc(Cn2cc(C3CCOCC3)nn2)on1 C(=O)(C(O)CCC(C)C)N1CC(NC(c2cc(OCC)ncc2)=O)C(OC)C1 C1(NC(c2c(C)nco2)=O)CCCC12CCN(C(=O)C=C1CCN(C)C1)C2 C(=O)(CCS(N)(=O)=O)N1CC(SC)C(NC(=O)C(c2cnn(C)c2)N(C)C)C1 c1(C(=O)NCC(C)N(C(c2cnnc(O)c2)=O)CC)cc2cccnc2cc1F n1(CC)nc(C(=O)NCCC(C)NC(=O)C(C)CN2CCCCC2)ccc1=O CCCC(C(=O)N(C)CCC1CCN(C(=O)C(C)(O)C(C)C)CC1)S(N)(=O)=O C(CCN=c1[nH]c(=NCCC(OC)OC)[nH]c2c1COC2)CC Cc1ccc(NC(=O)CC2COCCN2C(c2cc(F)ccc2I)=O)c(CO)c1 c1(CC)cc(C(N2CCCC2CC(N2C(CO)CCC2CO)=O)=O)c(C)o1 c12ccc(cc1)CCO2.C12CCCN1C(=O)CCN2.C(CC(C)C)OC CN1CCN(C(=O)CCCNC(C23CCCN2CCC3)=O)CC1(C)C C(=O)(CC(C)C(C)(C)C)NCC(C1CCC1)NC(Cc1nc(CC)sc1)=O Cc1cccc(CCC(=O)N(C(C)CCNC(C2CCC2)=O)C)c1Cl c1(CNC(N(C(C)C)Cc2cccs2)=O)nnc2n1CCCC2C(F)(F)F C1(CN(C(C(CC)O)=O)C)CN(C(=O)CCn2ccnn2)CC12CC2 N1(C(CC(C)(C)OC)=O)CCC2(CC(NC(=O)C(F)=CC3CC3)CO2)C1 C=CC1(C(=O)NC2CN(C(c3ccnnc3O)=O)CCC2CO)CCCCC1 C1(NC(=O)CC2CCCOC2)CC2CN(C(c3ccc4cncn4c3)=O)CC2C1 N1(C(c2nc(C)n(C)c2)=O)CCC(O)(CNC(c2cc(Cl)cnc2O)=O)CC1 C#CC1(O)CC(C(=O)NCCN(C(c2cc(Cl)cnn2)=O)Cc2ccccc2)C1 N1(C(C2ON=C(CC)C2)=O)CCN(C(=O)CCCCCC(C)O)C2CCCC12 CCC(C)CCC(=O)N1CCN(C(C2COCCOC2)=O)C(CO)C1 N#Cc1ccc(C(=O)NC2C3CN(C(c4coc(Cl)n4)=O)CC23)c(O)n1 Cc1cc(O)n2ncc(C(N3CCCC3CN(C(=O)Cc3cnsc3)C)=O)c2n1 c1(C(N2C3C(NC(c4ccccn4)=O)CC(C3)C2)=O)cc2cn[nH]c2cn1 C1(C(=O)NC2(CNC(CCC3CCC(C)O3)=O)CCCCC2)COCCN1C=O N1(C(C2N(C)C(=O)NC2)=O)CCC(C2CCN(C(=O)C(C)(C)CCC#N)CC2)C1 c1(C(=O)NC2(C3CN(C(Cc4ncc(C)s4)=O)C3)CC2)noc2c(F)cccc12 C1(C(=O)NCCc2nc(C)sc2)CN(C(=O)C=CC(C)C)C2(CCC2)C1 c1(C(=O)NCC2(CNC(c3nnn(CC)c3C)=O)CC2)ccc(Br)cc1N c1(C(N(CCNC(CCOC)=O)C(C)C)=O)ccc2n[nH]c(C)c2c1 C=CCC(F)(F)C(=O)N1CCSCC1c1cccc(OC(F)(F)F)c1 CCCCCS(=O)(=O)CC(=O)NCC12CC(CN1c1ccc(S(C)(=O)=O)cn1)C2 c1(CC)ccc(Cl)c(C(N2CC(NC(C3(CSC)CCC3)=O)C(O)C2)=O)c1 C1(CC(=O)NCC2(C)CCC(=O)N2)C2CCCC2N1C(=O)C(=O)NCC(F)F Cc1onc(Cl)c1C(=O)NC(C)CCCNC(=O)CCCOc1ccc(F)cc1 C(CCC(=O)NC(C1CC=CCC1)C(=O)NCCSC(C)C)OCC C1(C(=O)NCC(N(C(CCc2onc(CC)n2)=O)C)C2CC2)CCCCC1(F)F C12(CNC(C(=O)OCC)C(O)c3ccc(OC)cc3)CCCC(C1)OC2 C(C(=O)NOCc1nc[nH]n1)=CCCN(C(=O)COCC1CC1)C C1(C(=O)NCCC2CN(C(Cn3ncn(C)c3=O)=O)C2)CCCN2CCCC12 C=C(CNC(C1CCC(C)S1)=O)CCNC(c1cn(CC(N)=O)nn1)=O c1(OCC(=O)NC2C(C(=O)NC3C(CC)C3)C2)ccc(CO)c(C)c1 c1(NC(c2ccc(Cl)nc2F)=O)ccc(NC(C2COCCO2)=O)cc1F c1(C(=O)NCC2(F)CC(NC(C3(OC)CCOC3)=O)C2)cc2sccc2s1 C1(CC)C(C(=O)N(CC(O)CN(C)C(c2cc(Br)ccn2)=O)C)CCN1C C(=O)(CC1OCc2cc(Cl)ccc21)NC1CN(C(CNS(C)(=O)=O)=O)C(CO)C1 c1(C(=O)NCC2(F)CC(NC(C(C)O)=O)C2)c(Cl)cc(Cl)nc1N C(N=c1[nH]c2ccc(Cl)cc2s1)C1C(NC(C2CCCC(C(N)=O)C2)=O)CCC1 c1(C(=O)NC(CNC(C(CC)OC)=O)CO)ccc(OCC(N)=O)cc1 C1(CC(=O)N(C2CCCC2)CC#C)C2CCCC2N1C(C1CC(CC2CC2)C1)=O N1(C(CC(C)(C)C(F)(F)F)=O)CCC2CC(NC(=O)CS(N)(=O)=O)CCC2C1 C(CC1=CCN(C(=O)C=CC(C)O)CC1)NC(CC=C)=O c1(CCC)nc(=NCCCc2ccccc2Br)s[nH]1 Cc1cccc(C)c1C(=O)NC(C)CNC(c1cc(Br)n[nH]1)=O C1(CNC(CN(C2CC2)CC)=O)(CO)CCCN(C(C2(C(N)=O)CCC2)=O)C1 c1(NCC)ccc(C(N2CCC(C)(CNC(=O)CCCOC)C2)=O)cc1[N+](=O)[O-] C1(CNC(C(C)CO)=O)CCCC2CN(C(=O)CN3CCNC3=O)CC12 CCCCCC(C(=O)N(C)CCOCCCNC(C1COCCO1)=O)C(C)C C12(CNC(C(CC#C)C)=O)CCC1CN(C(c1ccc(Br)cc1O)=O)C2 C1(C(=O)NC2C(NC(Cc3cccc(CC)c3)=O)CC2)C2CCC1(C)C2(C)C c12nnc3ccc(nn13)OCCS2.c1(Oc2c(C)cccc2)cc(F)cc(F)c1 c1(C(N(C2CC(C#N)C2)CC(=O)NC(CCC)C(=O)NC)=O)cc(F)ccc1C C1(NC(=O)NCc2cc(C(=O)OC)cc(F)c2)CCC2=NN=NN(C2)C1 C1(CNC(C2C(=C)CC2)=O)CCC2(CO1)CC(NC(c1csc(Cl)n1)=O)C2 c1(CC(N2CCN(C(c3ccccc3)CN3CCCC3)CC2)CO)ccc(O)cc1 C1(c2nnnn2C(C)(C)C)(NC(c2cncc(NC)c2)=O)CCN(C)C(C)C1 N1(C(c2c(CC)nns2)=O)CCCCC(CNC(c2cc3n(n2)CCO3)=O)C1 CCC1C(=O)Nc2ccc(C(=O)NCCC(C)(C)NC(=O)COC3CCC3)cc21 CS(=O)(=O)C1(C(N2CCC2CNC(C23CCC2C3)=O)=O)CCCC1 c1(CC)sc(N2CCC(C)(NC(=O)C(C)NC(C3CCCCC3)=O)C2)nc1Cl N1(C(C=C(C)c2ccsc2)=O)CCC(CNC(c2cc(Cl)n(C)n2)=O)C12CC2 C1(NC(C=CCC)=O)CCC(CC(=O)NCCC(C)(C)CO)CC1 CCCCCCCC(F)C(=O)NCCCN(C(=O)C(CC1CC1)OC)C Cc1ccc(O)c(CC(N2CC(NC(C3(C)CCCCCC3)=O)CC2(C)C)=O)c1 Cc1cc(C(=O)NC23CC(CNC(c4cc(C)nn4C(F)F)=O)(C2)C3)nc(O)n1 c1(OC)ccc(C(=O)N(CC(C)(C)CNC(=O)C(=Cc2cnn(C)c2)C)C)nc1 C12(C(NOCCOC)=O)CC(CO1)N(C(=O)CCCCCOC)C2 c1(NC2CC(CNC(c3c(C)nc(CCC)o3)=O)C2)cc2c(cn1)C(=O)CCC2 c1(CN2CC(C(N3CCC(C(=O)OC)CC3)=O)C(O)CC2)ccccc1[N+](=O)[O-] C(=O)(C1SCc2cccnc21)N(C)CC1CN(C(C2CC(O)C2)=O)CCO1 C1(CC(=O)N(CCC(=O)N(CC(C)C#N)CC)CC)COCC(C)O1 C(=O)(CC(F)(F)Br)N(C)CC1N(C(c2cc(C)ns2)=O)CCC1 c1(C(=O)OC)ccc(C(N2CCCC(C(=O)NCCOC(C)C)C2)=O)c(F)c1 CC1CN(C(C2CNC(=O)CN2C(C2CCC3(CCC3)C2)=O)=O)CC(C)(C)O1 C1(N(C(CNC(C(CC)C)=O)=O)C)C2CN(C(c3csc(COC)c3)=O)CC12 C(=O)(C(C)C(O)CC(C)C)N1CCC(CCOC)(C(=O)NC2CC(OC)C2)CC1 CC(C)CC(C)CC(=O)N1CC2CCCC2(NC(C2CCS(=O)(=O)CC2)=O)C1 c1(CN2CCCC(n3cc(C(=O)O)nn3)C2)ccc2sccc2c1 N1(C(C#CCNC(Cn2c(C)nnn2)=O)=O)CC(C#N)(N(C)C)C1 C(=O)(CCCC(CC)NC(C1Cc2nccn2C1)=O)Nc1ccc(CC)nc1 C(CCN=c1nc2scnc2c(N2CCC(S(C)(=O)=O)C2)[nH]1)C1(C)CC1 N1(C(C(C(C)NC(c2c(C)non2)=O)C)=O)CC2OC(=O)N(C)C2C1 N1(C(c2c(CC)nccc2)=O)CC2(CC(CNC(=O)COC3CC=CC3)C2)C1 c1(C(=O)Nc2csc(C3CCCO3)n2)ccc(F)c(SCC(O)C(F)(F)F)c1F Cn1ncc(C(F)(F)F)c1C(=O)NC1CCCCC1NC(C1(C)CC1(F)F)=O C1(NC(c2n(C(C)(C)C)nnn2)CCC2CC2)CCOC(c2cccc(Cl)c2)C1 CC1(C)OC(C)(C)C1(O)C(=O)NCCOCC1CCOC1 C(=O)(C1=NOC2(CCC2)C1)N1C(C)C(NC(=O)C(=O)NCC(F)F)CC1 C1(n2c(C(c3csc(CC)c3)NCc3ncc(CC)s3)nnn2)CCCCCC1 CCCC(C)(O)CC(=O)N(CC(=O)N(CC(N1CCCC1)=O)C)C C(=O)(C(C)(C)CCC(=O)NCC1CCCC2(CN(C(=O)C(C)(C)F)C2)O1)OC N1(C(c2cn(CC(C)C)nc2)=O)CCN(C(=O)C(C)C2(O)CCC2)CC1C(C)C C(=O)(C(C(C)(C)C)c1cc[nH]n1)N1CC(OC)C(NC(=O)C(C)(C)C(F)F)C1 N1(C(C2(C#N)C(C)(C)C2)=O)CC2(C1)CN(C(C1C3CC4C(C3=O)C14)=O)C2 C(N=c1[nH]cnc(Cl)c1CO)CCCN1CC(CC(=O)NCCOC(F)(F)F)C1 c1(C(N(C2CCCN(C(=O)C(C)CO)C2)CC)=O)cc(C(F)(F)F)cc(F)c1 N1(C(c2onc(CC)n2)C)CCC2C(CCCN2C(C2C3CCCC23)=O)C1 N1(C(CCC2CCN(C(C(C=C)O)=O)C2)=O)C2CCCC1CC(=C)C2 C(=O)(CC(C)C(=O)OC)NC1CCN(CCNC(C=COCC)=O)CC1 c1(C(=O)NCC(C)NC(C2N(C(C)C)CCC2)=O)ccc2nn[nH]c2c1O N1(C(C2CSCCN2Cc2nn[nH]n2)=O)CC(CO)C2(COC2)C1 c1(C(=O)NC(C2CCCC2)CNC(C2(C)C(C)C2)=O)cc2n(n1)CCCO2 N1(C(c2ncc(OCC)nc2)=O)CCC(F)C(NC(=O)Cc2cnnn2C)C1 c1(-n2c(C(CCCC3CC3)NC(CCC=C)(C)C)nnn2)ccc2c(c1)CCC2 CN1C(=O)NCC1C(=O)NC1CC(CNC(=O)CC2(O)CCCCC2)C(O)C1 C1(n2c(=O)c2=O)CCOCC1.c1(C2N(C(C)C)CC2)ccccc1 N1(C(c2occ(C)c2C)=O)CC2CC(C1)CN(C(c1cc3ccnn3cn1)=O)C2 N1(C(C23C(C)OC(C)(C2)C3)=O)CCC(C2CC2)(CNC(=O)C=C2CCSCC2)C1 N1(C(c2ccc(SC)cc2)=O)CCC2(CCN(C(=O)Cn3cncc3C)C2)C1 N1(C(CC(CC)C)=O)CC2C3CCC(C2C1)N(C(C1CCC2(CCOC2)O1)=O)C3 C1(C(N2C(CNC(=O)CCc3ccccc3F)CC(O)C2)=O)CC12CCSCC2 S(=O)(=O)(c1ccc(Br)c(F)c1)N1CCC2(C(C(=O)Nc3ccc(Cl)nc3)C2)CC1 N1(C(CC=CCC)=O)CCOC(CCNC(C2(C#N)CCOC2)=O)C1 C12(C(=O)NC3CCC(N(C(=O)CS(=O)(=O)NC(C)(C)C)C)CC3)COCC(C1)OC2 c1(C(=O)NCC(C)NC(=O)C(c2ncc(Cl)n2C)(F)F)cc2cc(Cl)ccc2o1 N1(C(CC2C(NC(CNC(=O)OCC=C)=O)CCC2)=O)CCCC(N=[N+]=[N-])C1 c1(C(N(CC(CC)NC(=O)CN2CCOCC2)CC)=O)cc2n(n1)CC(O)CO2 C1(N(C)Cc2occc2CSc2ccccc2)CCS(=O)(=O)C1 c1(OC)cc2nc(n1)COC1CCN2CC1.c1(NC(C2CCC2)=O)cnccn1 c1(C(N(CCCNC(CC(C)OC)=O)C(C)C)=O)cc(C2CC2)cc(F)c1 C12(CNC(c3c(C)nc(O)[nH]3)=O)CCCC1N(C(=O)CCC1CC1(C)C)CCC2 C1(C(=O)NCCCCNC(CC)=O)CCC(=O)N(CC)C1 c1(CCC)n[nH]cc1C(=O)NCCOCCC(=O)N1CCC1CC(C)C CCCC(C)CC(=O)N(CC(CO)(CO)NC(c1cc(C2CCC2)no1)=O)C N1(C(C2(NC(c3cnc(O)o3)=O)C(C)C2)=O)Cc2ncsc2C1 N1(C(C2(C)CCC2)=O)CCc2ccccc2C(NC(=O)CSC2CCCC2)C1 c1(CNC(=O)CC2C=CCCC2)ccc(CNC(C2CC23CCOC3)=O)cc1 C=CCCCC(C(=O)NC(c1ccn(C)c1)C)NC(c1ccc(C#N)cc1)=O N1(C(C(COC)O)=O)CC2CN(C(c3ccnc(OCCO)c3)=O)CC2C1 C1(F)(C(N2CC3C(CNC(COCCCC#C)=O)C3C2)=O)C(C)(C)C1(C)C C1(NC(CCC2CC(OC)C2)=O)CN(C(C2(C#N)CC3(CC3)C2)=O)CCC1CO c1(Cc2n(CC)c(CN(C3CCC(C)C3)C)nn2)c(F)cccc1F c1(C(=O)NC2C(C(C)C)CN(C(c3ccc[nH]3)=O)CC2)noc2cc(F)ccc12 C1(NC(CCC(=O)OCC)=O)(CNC(=O)C(C2CCOCC2)C)CCCCC1C N1(C2CCCN(C(C3C(C)(C)CCC3)=O)C2)CCN(C(=O)C=CCO)CC1=O Cc1cc(C(F)(F)F)nc(N2CC(NC(c3cnc(C(C)C)[nH]3)=O)C(C)C2)n1 c1(OC)ccc(-c2ccc(NC(=O)CCOC3CCNC3)c(F)c2)cc1F c1(C(N2CCC(CNC(C(C)(C)C3CCC3)=O)C2)=O)ccc(O)c(F)c1 C1(NC(c2c(C(C)=O)ccs2)=O)CCOCC1NC(c1ccc(C(F)F)cn1)=O c1(OC)ncc(C)cc1C(N1CC2CC1C2NC(C1CC1[N+](=O)[O-])=O)=O CC1OC(C)C(C(=O)NCCC(C)N(C(=O)C=CC(C)(C)C)C)C1C c1(C(=O)NCC2CC(C)N(C(C3CCCCO3)=O)C2)cnc2[nH]nnc2c1 c1(C(N2CCC(CCCNC(CC3C(C)C3)=O)CC2)=O)ccnc(Cl)c1N c1(-c2nnc(N(C3CCSC3)C)n2C2CC2)ccc(S(N)(=O)=O)cc1 c1(OC)ccnc(O)c1C(N1CC=CC(NC(c2nccc(C)n2)=O)C1)=O C1(C(N(CC(=C)C)CC)=O)CCCN(C(=O)Cn2[nH]cnc2=N)C1 N1(C(c2c(C)nns2)=O)CCC(C)(CCNC(c2cn(CCCC#N)nn2)=O)C1 c1(CN(CCCN(C(=O)C(C2CCOCC2)=O)C)C)ccc(C(F)(F)F)nc1 c1(C(=O)NC(CC(C)NC(C2CC2c2cccs2)=O)C)cc2occc2[nH]1 N1(C(C2CCCC2(F)F)=O)CC2CCCC(C1)N2C(c1c(F)ccc(F)c1O)=O C1(CNC(C2C(CC)CCC2)=O)CCCC12CCN(C(C1C=C1C)=O)CC2 c1(C(=O)OC)nccnc1C(=O)NC(C)CC(C)NC(=O)Cc1cnn(C)c1 c1(N(C)Cc2ccc(F)cc2)ccc2c(c1)CN(Cc1ccc(N)cc1Br)CC2 Cc1ncnc(N2CCCC(CO)(NC(=O)CCC3CCCC(=O)N3)C2)c1C#N N1(C(c2n(CC)ccn2)=O)CCN(c2ncnc(Cl)c2Br)C(C)C1 C1(C(C)C(=O)NCC=CBr)CCN(C(=O)CCc2cccn2C)C1 c1(C(c2nnnn2CCCF)NC(c2ccc(C)o2)CC)ccc(OC)nc1 c1(C(=O)NC2(CO)CCN(C(CSCCCC)=O)C2)cc2ccc(OC)nc2[nH]1 c1(C(=O)NC2(CNC(c3csnc3Cl)=O)CC(OC)C2)c[nH]c2ncccc12 C1(=CCNC(C(CC)O)=O)CCN(C(=O)Cc2ccc(-n3cccc3)cc2)CC1 c1(CC)cc(C(N2CCCCC2c2cn(-c3ccc(NC)cc3)nn2)=O)c(C)o1 CC1COC2(C1)CN(C(=O)C#CCNC(c1ccncn1)=O)C2 C1(C(=O)NCCCN(C(=O)CC2CC=CC2)C)CSCN1C(=O)OC(C)(C)C CC1(c2ccccc2)CCN(n2cc(CC3CC4CC(CO)C3C4)nn2)CC1 NS(=O)(=O)C1CCC(C(=O)NCCNC(c2ccc([N+](=O)[O-])cc2O)=O)CC1 CCCCC(C(=O)NCc1cc(C)cc(C)c1)NC(c1cc(C(C)=O)[nH]n1)=O N1(C(c2n(C(C)C)ncc2)=O)CC2ON=C(CNC(c3ccsc3)=O)C2C1 c1(CC)cc(C(N2CC(CC(C)NC(=O)C=CBr)C2)=O)ccc1F c1(CNC2C(NC(=O)CC3CCOCC3)COC2)cc(C(N2CCCC2)=O)no1 c1(C(=O)NCC(C(C)C)NC(C(CNC(C)=O)(C)C)=O)nc2ccccc2[nH]1 C1(CN(C(=O)CC2CC2)CC)CCN(C(=O)CC2CC3CCC2O3)CC1 C(=O)(C(C)CCCC(C)C)NC1CC2CN(C(c3ncc(C)nc3)=O)C(C1)C2 CC1CN(C(c2c(O)cccc2F)=O)CCC1CNC(C1(CO)COC1)=O N1(C(c2c(OC)c(C)cs2)=O)CC(NC(=O)C(C)=C2CCCC2)C(C)(C)C1 C(=O)(C1=CCCCO1)NC1CCC(CCNC(=O)Cc2nc[nH]n2)C1 C1(CC(=O)NCC(N(OC)C)=O)CCN(C(=O)C(C)CC#N)C1(C)C c1(CN2CC(CNC(C3CCCCO3)=O)OCC2)ccc2occc2c1 c1(C(=O)NCCN(C(CC)C)C)n[nH]c2c1CN(C(=O)C1=CCCCCC1)C2 Cc1cc(P(C)(C)=O)oc1C(N1CC(O)(CCNC(=O)CC(C)C2CC2)C1)=O Cc1cncc(C)c1C(=O)NCCCCC(=O)NC(c1ccccc1O)C C1(CC(N2CC(C)(OCC(=O)N(CCCOC)CCO)C2)=O)CCCC(C)O1 C1(C(=O)NCc2c(C)noc2)(CNC(=O)CC2CCCCO2)CC12CCC2 c1(OC)cccc(C(C)CC(=O)N2CCCC2C(C)(C)NCCO)c1 C(=O)(C1CCCc2nn[nH]c21)N(CCOCCCNC(C1C(C)C1C)=O)C N1(C(c2c(CC)cc(Cl)cc2)=O)CC2(CC(NC(=O)C(C)(O)CC)CO2)C1 N(C(=NCCc1ccc(CO)cc1)NC1CCCC1)CC1CCCC(C)O1 C1(C(=O)NCC(C)(C)NC(c2ccc3sncc3c2)=O)CCCCC1P(C)(C)=O C(CCCCC(=O)N1CC(O)CC1(C)C)N(C(C1C(CC)CCO1)=O)C c1(OC)ccc(C(=O)NC2CCC(NC(=O)C(Br)=C(C)C)C2)c2[nH]ncc12 C(=O)(C(C)(C)C(=O)N1CCCC(C)(NC(=O)Cc2ccc(C(F)F)cc2)C1)OC N1(C(C(C)OCC2CC2)=O)CC(O)C(O)C1CNC(=O)CC1OC(C)(C)OC1=O c1(C(N2CCC(C(=O)Nc3cccc(O)n3)C(O)C2)=O)cc(Cl)ccc1[N+](=O)[O-] S(=O)(=O)(c1ccccc1Br)C1CC1.CC(C)(C)CN C(CCF)(C(=O)Nc1ccc(CO)nc1)NC(C1CC=CC(O)C1)=O C1(NC(C2CC(NC(C(C)C3CC3)=O)C2)=O)(CO)CCSC1 C1(C(=O)OC)Cc2ccsc2CN1C(=O)C(=O)NCCc1ccc(C)cc1[N+](=O)[O-] C1(NC(COCC(=C)C)=O)CCN(C(C23CCCC2C3(F)F)=O)C12CCC2 c1(CNC(C2C(NC(c3cnn(C)c3C(F)(F)F)=O)C2)=O)c(F)cc(F)cc1F c1(C(=O)OC)ccc(O)nc1NC1CC(NC(c2sncc2C)=O)C1 c1(C2(C(=O)NC3CC(CCNC(=O)Cn4ccnn4)C3)CC2)ccc(Cl)c(F)c1 N1(C(C(C=C)OC)=O)CC(C(=O)NCC2(N(C)C)CCC2)C(C2CC2)C1 N1(C(C(C(C)C)NC(N)=O)=O)CCCOC(CNC(C2COCCO2)=O)C1 CC1CCCC=C1C(=O)N1CCOC(CNC(=O)Cc2c(F)cc(F)cc2F)C1 CCC(C)C(C(=O)N1CC2CC2(C(=O)NC2CCN(C)C(=O)C2)C1)N(C)C N1(C(C(C)=C(CC)C)=O)CC2CCCC(CNC(=O)CCC(F)(F)C(F)F)C2C1 C1(CC)C(=O)NCCN1C(c1n[nH]c(SCc2ccccc2)c1Br)=O N1(C(C(CC)=CC)=O)CC(CNC(c2cc(-c3ccccc3)ns2)=O)CC1C C=CCC(C(=O)N(CC(C)NC(C1(N(C)C)CCC1)=O)C)C(C)C N1(C(C#CC)=O)CCC2(C1)CN(C(c1ccc(-c3cccc(OC)n3)cc1)=O)C2 N1(C(CN(CC(=O)NC(C)C)C)=O)CCN(C(C2(C)C=CCC2)=O)CC(C)(F)C1 CC#CCC(CO)NC(C1(NC(c2ccsc2Cl)=O)CCCC1)=O C1(NC(c2ccc(CC)nc2)=O)CCC12CN(C(=O)C=CC(=O)NC1CC1)C2 c1(N(C)C(C(CNC2CC2)N(C(=O)OC)C2CC2)=O)cccc(C2(C)CC2)c1 c1(C(=O)NC2CC(NC(=O)COCc3nc[nH]n3)C2)cc(C2CC2)cc(F)c1 c1(CCNc2cc(N(C)Cc3cnccn3)ncn2)cccc(Cl)c1Cl C(CCCC(C)NC(C(OCC)OCC)=O)NC(=O)CC(C)n1ccnc1CC C1(C(N2CCCN(CC(N3CCOCC3)=O)CC2)=O)CC2(CCC2)CCO1 O=C(N=c1c(Br)c[nH]cc1I)C1CCN(S(=O)(=O)C2CCCCC2)C1 c1(C(=O)NC2CCC3CC2CN3C(C2CC(Cl)(Cl)C2)=O)coc2ccc(F)cc12 C1(NC(C2(C)CC2)=O)CN(C(=O)C(c2cccc(Br)n2)(F)F)C(C)(C)C1 c1(NC(CN(C)C)=O)cccc(S(=O)(=O)NC2CCC2C(=O)O)c1 C12(CNC(CN(C3CC3)CC)=O)CC1CN(C(=O)COCc1nc(C)no1)C2 N1(C(C(C)OCCOCC)=O)CC2CN(C(C)=O)CC2C1.C1(CC)C(=O)N1C Cc1nc(C(C)C)sc1C(C)N(C)C(=O)NCC1CCCC1C Cc1ccc(F)c(C(=O)NOC(CC(C)C)C(=O)NC2CCN(CC3CC3)C2)c1 C=C(C)CC(C(=O)NCCc1cnn(C)c1C)NC(=O)CNc1ccccn1 S(=O)(=O)(c1c(C)cc(C)cc1C)NCCC(=O)NC(CC#C)C(N)=O c1(C(=O)NCC(CNC(CCC#C)=O)F)cc(F)ccc1-n1ccnc1 c1(C(N(CC(CNC(C(CC)(C)F)=O)C)C)=O)ccc(C)c(N)c1 CC1(C)CCCCC1NC(=O)CCC1CCCN1C(C1CN2CCC1CC2)=O C(CCCC(=O)N1CCC(F)(CNC(C2(Cl)CC2(C)C)=O)C1)N(C(C)=O)C N1(C(CC(=O)OCC)=O)CC2(CC(CC(=O)NC3(CC)CCOC3)C2)C1 CC1(C)CC(=O)NCC1C(=O)NCC=C1CCN(C(=O)CCP(C)(C)=O)CC1 CC(O)C(F)(F)C(=O)NC1CCC(CNC(C2COC(C)(C)C2)=O)CC1 N1(C(C2CC(C)C2)=O)CCC(C)(CC(=O)NCC(C)CN2CCCC2)C1 C1(NC(C)=O)CCCN(Cc2cnn(C)c2CCO)C1 c1(C(N2CC(NC(C3CCCC3)=O)CC(C)(C)C2)=O)cc(F)c(C#N)c(F)c1 C1(C(=O)OC)N(C(C2CCCOC2)C(=O)NCc2cccs2)CCOC1(C)C C#Cc1cc(C(=O)NC2CCCCC2NC(C2CCC(C)(C)C2)=O)ccc1C Cc1ccc(C(N2CCC(C(F)(F)F)C2C)=O)cc1S(=O)(=O)N(C)C C12(NC(C(CCN(C)C)O)=O)CCCC1CN(C(=O)C=Cc1ccccc1F)C2 c1(OC)cc(C(n2cc(CC3C=CCCC3)nn2)C)ccc1OC1CCCC1 N1(CC(=O)NC(C(=O)NCC)Cc2ccncc2)CCC(NC(=O)OC)CC1 CC(C)C(C(=O)NC1CCN(C(C2(C)CCC2)=O)CC1F)C(C)C C(=O)(C1COc2ccccc21)N1CC2CCN(C(c3n(C=C)ncc3)=O)C2CC1 C1(CNC(CC(C=C)CC)=O)CN(C(C2CC(C(F)(F)F)C2)=O)CCC12CCC2 N1(CC)CCCC(C(=O)NC2CC(O)(CNC(c3csc(C(F)(F)F)n3)=O)C2)C1 C(=O)(C1CC(=O)c2ccccc21)N1CCC(F)(C(=O)OC(C)(C)C)C1 N1(C(CSCC#C)=O)CCC(C(CNC(=O)CCc2ccon2)OC)CC1 CS(=O)(=NC(=O)CCC1CS(=O)(=O)C1)c1cc(F)ccc1F CC1CC(NC(=O)C(=O)NCc2ccnc(-c3ccccc3)c2)CC(C)O1 c1(C(=O)NCc2ccc(-c3cc[nH]c3)nc2)ccc(O)cc1Cl CC1COCC(CC(=O)NC2CC(F)(CNC(=O)CCc3cnc(O)[nH]3)C2)O1 C1(C(C)(C)C)CCN(C(C2CCCOCC2)=O)C(CNC(c2cc[nH]n2)=O)C1 N1(C(C(CCO)N(C)C)=O)CC2CS(=O)(=O)CC2(CNC(c2cnco2)=O)C1 Nc1ncc(C(=O)NCCOC2CCN(C(=O)C=Cc3cnc[nH]3)C2)cc1Br c1(OC)cnccc1C(N1CCOCC1C(=O)NCCOCC1CCOC1)=O CC(Cc1cnn(C)c1)C(=O)NC1CN(C(=O)COc2ccsn2)C1 N1(C(CNC(C(C)(C)OC(C)C)=O)=O)CCC(O)C(C)(C)C1 C1(O)(C(=O)NC2CC3(CC(NC(c4scc(C)c4C)=O)C3)C2)CCCC(C)(C)C1 N1(CC(=O)NCc2c(Cn3cc(CC(C(=O)OC)C)nn3)nco2)CCCS1(=O)=O C1(CCNC(c2ncn(CC)c2)=O)C(C)CCCN1C(=O)C1=COCCC1 c12ccccc1NC(=O)C1(CCC1)C(=O)N2.C1(Sc2ccccn2)CCOCC1 c1(C(=O)NC2C3CN(C(C4C(C(C)(F)F)C4)=O)C2C3)cnc2c(c1)COC2 c1(C(N2CCCC3(C2)CN(C(C2CC=CC2)=O)C3)=O)ccc2cc[nH]c2c1F c1(N2CCN(CC(C)(C)NC(=O)C(N)=O)CC2)nc(Cl)nc2c1CCOC2 C1(NC(C(CC=C)CC=C)=O)CN(C(c2nc(=N)cc[nH]2)=O)CCC12CCC2 N(C1CCc2c(Br)cc(F)cc21)C(=O)NCC(=C1CCCC1)F C(=O)(CC(F)(F)C(F)F)N1CC(CC=C)(NC(c2nonc2CC)=O)C1 C1(CN(C(CCCOCC=C)=O)CCN(C)C)COCC(C)O1 Cc1cc(C2(CNC(=O)C(F)CC3CCCCC3)CC2)on1 C1(NC(CN(CC)CC)=O)CCC(CN(C(=O)CNS(N)(=O)=O)C)CC1 O(N=C1CCCCCC1)CC(N1C2C(NC(CC=C)=O)CC(C2)C1)=O C1(C(N2C(C(N(C)Cc3cnc[nH]3)=O)CC(O)C2)=O)CCCC2(CC2)C1 C1(C(=O)OC)CN(C(=O)C(=O)NCc2c(Cl)cnn2C)CCN1C N1(C(C(C)Oc2ccccn2)=O)CCc2[nH]nc(CNC(c3cnco3)=O)c2C1 N1(C(c2c(C)c[nH]n2)=O)CC(NC(=O)Cn2nnc(=N)[nH]2)C2(CCC2)C1 N1(C(C=Cc2ncn(C)c2)=O)CC2CC(C1)N2C(=O)CC1CC(C)(C)CO1 N1(C(C2CCC(C)O2)=O)CCCCC1CN(c1ncncc1I)C C(=O)(C(F)C(F)(F)F)NC1(CNC(C(SC)SC)=O)CCCCC1 c1(NC(C2(NC(C(C)CCN(C)C)=O)CC(F)C2)=O)cnc2[nH]ncc2c1 C12(NC(C(c3ccc(CC)s3)=O)=O)CC1CN(C(C1CCC(C)CC1)=O)C2 C1(NC(C2(F)CC2)=O)COCC1NC(C1CN(C2CCOC2)C1)=O Cc1nc2ccc(C(=O)NC3CC4CC3N(C(=O)CC35CCCC3C5)C4)cc2o1 c1(NCc2ccc(CC)[nH]2)nc(OCC(F)(F)F)ccc1Cl N1(C(C(CC)N2CCCC2=O)=O)CCC(C#N)(CC)CC1 N1(C(C(n2cc(-c3cnc(O)nc3O)nn2)C)=O)CC(=O)N2CCCCC2C1 c1(C(N(C(CN(C(C(C)SCC)=O)C)C)C)=O)cc2c(cn1)OCCO2 Cc1c(C(=O)CNC(=O)C(c2ccc(Cl)cc2)C2CC2)sc2ccccc12 N1(C(c2c(C)ccn2C)=O)CCN(C)C(C(=O)N(C)CCN(C)C)C1 c1(NC(N2CCC(N(c3ccccc3)C)C2)=O)ncnc2c1ncn2C c1(C(=O)NC(CCOC)CNC(=O)CC(F)(F)Cl)ccc(N=[N+]=[N-])cn1 CC(CS(=O)(=O)N1CCC(O)C(c2ccccc2OC(F)(F)F)C1)C(C)(F)F Cc1ccc(C(=O)NCC2(C(=O)NCC3NC(=O)NC3=O)CCCC2)nc1 Cc1nncc(C(=O)NC2CC(F)(F)CC2NC(C2CCSC2)=O)c1C N1(C(C(=O)NCCSc2ccccc2)=O)CCn2c(cc3c(Cl)cccc23)C1 c1(C(=O)NCC(c2cccc(C)c2)NC(C(CC)F)=O)cccc2nn[nH]c12 C1(C(N2CC(NC(C3C(COC)CC3)=O)(COC)C2)=O)CC12CCCC2 c1(C(N2CC(n3cc(C(=O)OC)nn3)C2)=O)cccc(OC2CCC(C#N)C2)c1 Cc1nc(NC(=O)CCNC(C2C3CCCCCC23)=O)ccc1C(F)(F)F c1(C(C(=O)NCCC(=C)CNC(C23CC(C)C2C3)=O)(F)F)ccc(C)cc1 N1(C(=O)NC(c2cc[nH]n2)C2CC2)CCS(=O)(=O)CC1C1CC1 C1(C(=O)NCC(CN(C(c2ccc(CC)s2)=O)C)C)CCCC2(C1)CC2(F)F c1(OCC)cccc(NCCC(C(C)C)NC(c2cnc[nH]2)=O)c1[N+](=O)[O-] N1(C(C(C)(C)C#N)=O)CC2CC1CC2CNC(=O)CCC1CC(C)(C)CO1 c1(C(=O)NC2C(NC(c3c(Cl)cn(C)n3)=O)CC2)cc(O)ccc1OC(F)F C(C(F)(F)C(C)(C)O)NC(C1(CNC(CCC2N(C)CCC2)=O)CC12CCC2)=O c1(C(=O)NC2(C)CCN(C(c3nnn(C)n3)=O)C2)cccc(F)c1Br C1(CC(=O)NC2CCN(C(=O)Cc3ccno3)CC2O)CCCCC12CC2 N1(C(c2sccc2Cl)=O)CC(CO)C2(C1)CN(C(c1csc(O)n1)=O)C2 C(=O)(C(CCC)C(C)C)NCC1(F)CCN(C(COCC(=C)C)=O)C1 Cc1ccccc1NC(N1CCN(C(=O)NC23CCC(CO2)C3)CC1)=O CC1CN(C(c2cnc(Cl)c(Cl)c2)=O)CCC1NC(c1cc(O)no1)=O Cc1csc2ncc(C(=O)NCC3CCCN3C(=O)Cc3cccc(Cl)c3F)n12 C12(C(N3CC(COC)C3)=O)COCC1CN(C(=O)CCCn1ccnc1)C2 c1(C(C(=O)NCC(C2CC2)NC(CC(=O)NCC#C)=O)C)cc2ccccc2o1 N1(C2CC2)CC(CNC(c2cn(CCC)nn2)=O)CC1C.C12(CC1)C(=O)NC2=O c1(C(N2CCCN(C(C(C)C3CC3)=O)C(C)C2)=O)cc2c(n1C)CCOC2 C1(CNC(C(CC)F)=O)CCCCCN1C(=O)CNc1ccc(OC)cc1 C(=O)(C1=C(C#N)CCC1)NC(C(=O)N(C)Cc1ccoc1)CCF N1(C(C2(CC)CCCC2)=O)C2CCC1CN(C(=O)C(C)SC)C2 N#CC1(C(N2CCC(F)(CNC(c3cncn3C3CC3)=O)C2)=O)CC2(CC2)C1 Cc1cc(NC(=O)CCC2CCN(C(C3(Cl)CCC3)=O)C2)cc(C)c1C Nc1ccnc(C(N2C3CCC2C(NC(=O)Cn2cc([N+](=O)[O-])cn2)C3)=O)c1Cl Cc1nc2c(C(=O)NC3CC3CNC(c3ccc(C)c(C#N)c3)=O)ccnc2[nH]1 CC1=NOC(=O)C1CC(N1CCOC(CNC(c2cn(C)cn2)=O)C1)=O c1(NC(C)=O)cc(Cl)ccc1C(=O)NCCC(C)NC(=O)CN1CCC1C N1(C(C(CO)N(C)C)=O)CC23CCCCC2(C1)CN(C(c1ccc(Cl)o1)=O)C3 CC(C)C(O)C(=O)NCC12CC1CN(C(c1ccc(CO)cn1)=O)C2 C1(C(=O)NCC2CCCN(C(=O)Cn3cncn3)CC2)Cc2cccc(F)c2O1 C1(CCNC(CC=CCC)=O)CC(F)(F)CN1C(C1CC2OC1C1CC21)=O CC(C(O)C(F)F)NC(C1(NC(=O)C#CC2CC2)CC(F)C1)=O N1(C(CN(C2CCC2)C)=O)CCCCCCC1C(N1CC=CC1CF)=O c1(C(N2CC(NC(C(CC)(C)CO)=O)C(O)CC2)=O)c[nH]c2cc(F)c(F)cc12 C12(CNC(CN(C(C(n3ncc(C)c3)C)=O)CC3CC3)=O)CCCC(CO1)C2 Cc1ccn(CC(=O)NC2(CCCCNC3CCOC3C(=O)OC)CC2)n1.C CCC(CC(=O)NCC1CCCN(CC(=O)NCCCCl)C1)C(C)(C)C c1(C(=O)NCC(CC)NC(C(C2CCC2)OCC)=O)oc(Br)cc1C CC1(C(N)=O)CCCN(C(C23C(=O)C4CC2C3C4)=O)C1.C1CCC(=O)N1CCO C1(O)(C(=O)NCC2(C)CCN(C(CC3(C(=C)F)CCC3)=O)C2)CN2CCC1CC2 c1(NC(=O)CNC(c2cc(C3(O)COC3)on2)=O)cccc(Br)c1 c1(OCC(=O)NC2CCC(CNC(CCSCCC)=O)C2)ccc(F)nc1 C(C)(C)(CC(=O)NCC(C)(O)CN(C)C)NC(C(CC)SC)=O C1(NC(c2ncc(CC)s2)=O)CCC(C)N(C(=O)CN2CCCS2(=O)=O)C1 C1(CNC(=O)Cc2nc[nH]n2)CC2(CN1C(=O)C=Cc1cccnc1)CC2(F)F C1(CNC(C(Cc2cc[nH]n2)NC(=O)C=CC(F)(F)F)=O)C2CCCCC12 c1(N2CCC(NCC(C(C)C)NC(=O)C3=CCOC3)C2)ncccc1C(F)(F)F N1(C(COCCCOC)=O)CCCC12CCCN(C(c1cc(C)oc1C)=O)C2 c1(OC)ccc(CNC(=O)COc2c(F)c(F)c(F)c(F)c2F)cc1S(N)(=O)=O N1(C(C2(COCC)CC(=C)C2)=O)CCCCC1c1nn[nH]n1 c1(C(=O)NCCOC2CCN(C(CC=CC)=O)C2)cc2ncccc2cc1Cl N1(C(C(c2ccoc2)NC(CCC2(C#N)CCC2)=O)=O)CCC2CCCC12 Cn1cc(C(O)C(=O)N2CC(NC(=O)C=Cc3ncc[nH]3)C2)cn1 C#CCC(CC#C)C(=O)NC1CN(C(=O)C(n2ccc(C)n2)C)CC1C1CC1 C1(C(=O)NCC(C)NC(c2c(C)noc2C(C)C)=O)CC(c2ccncc2)=NO1 c1(C(=O)NC(CN(C(c2c(C)scc2)=O)C)C)c[nH]c(=O)cn1 C1(CC(=O)NCCCCn2cc(CCCC(C)=O)nn2)CCC(F)(F)CO1 Cc1cc(N)c(C(N2CCN(C(=O)Cn3cnnc3O)CC2C(F)F)=O)cc1C C1(NC(c2ccc(CC)o2)=O)CC(F)CN(C(C2CC2(Cl)Cl)=O)C1 C1(CN(C(CC2C(N(C(CCC#C)=O)CCC)C2)=O)CC)CC(=O)N(C)C1=O C(CC1CCC1)(C(=O)NC1CCC2CC12)NC(C(C)=C1CCC1)=O c12ccc(cc1)C(C1CC1)NC(=O)N2.N1(C(CC)C)CCN(C2CC2)CC1 n1(CC)ccnc1C(=O)N(CCC(=O)NCC(Cl)C(C)O)C1CC1 C1(C(CC)NCc2cncn2C(C)C)Cc2ccccc2C1 C1(NC(c2c(C)cc(F)c(Cl)c2)=O)CC1C1CCN(C(=O)Cc2cnc[nH]2)CC1 C(=O)(C#CC1CCCOC1)NC1(CO)CCN(C(c2nn(C)c(Cl)c2)=O)CC1 N1(C(CC2CC(OC)C2)=O)CCN(C(=O)C(C)C(=O)N2CCCC2)C(C)C1 N1(C(C(Br)=C(C)C)=O)CC2CCN(C(C3COC4(CO)CC3C4)=O)C2C1 C1(C(=O)NCC(CC)O)C2CCCC2CN1C(C1CCC1C)=O CC(C)C(C)(O)C(=O)NC(C)C(CO)NC(C1(F)CCCC1)=O C1(C(=O)NCCCNC(C2(OC)CCC(C)(C)C2)=O)CCOC2(CCCC2)C1 C1(C(N2C(CC#C)CCCC2)=O)CN(C(=O)CC2CCOC2(C)C)CCC1(C)C N1(C(c2oc(C)c(CO)c2)=O)CCN(C(C2OCCC2C(F)(F)F)=O)CC1C CCC(CC(=O)N1CC(C2CN(C(c3c(CC)nc(C)n3C)=O)C2)C1)C(C)C c1(C(N(CCCCNC(Cn2c(C)cc(C(F)F)n2)=O)C)=O)ccc(Cl)cc1N Cc1cc(C(C)C)nc(=NCC(CC(C)C)NC(=O)CN2CCCCCC2)[nH]1 c1(OC)ccccc1OCC(=O)NC(C1CCN(C(c2ccnnc2Cl)=O)C1)C c1(CONC(c2ccc(C(F)(F)F)cc2)=O)nc2cnccc2[nH]1 N1(CC2CCCO2)CCCC(N(CC(CC=C)(F)F)C(c2cn(CC)nn2)=O)C1=O C1(CNC(c2ccc(CNC(C3C(C)=CCS3)=O)s2)=O)CC12CCOCC2 Cn1cc(CNC(c2cc(CCNC(=O)CC3CC(F)(F)C3)on2)=O)cn1 N1(C(C(C)NC=O)=O)CCOC2CN(C(=O)Cc3ccccn3)CC12 C1(NC(C2CCC2c2nc(S)n[nH]2)=O)COC2(C1)CN(C(=O)C1=C(Cl)CCCC1)C2 CCCC(C)C(=O)NC1(C)CN(C(C23CCC2C3)=O)C1 N1(C(C(COC)OC)=O)CCC=CC1C(N1CC(C#N)(CCF)C1)=O N1(C(c2c(Cl)cn(CC)n2)=O)CCC2(CC1)CC(C)N(C(=O)C(C)CO)C2 Cc1cccnc1C(=O)NCCC(C(C)C)NC(c1ncnn1C)=O CC1CC(C)N(C(c2cnc(O)n(C)c2=O)=O)CCN1C(c1c[nH]c(=O)cn1)=O C(CC(C)C)(C(=O)N(OC)C(C)C)NC(CSCC=C)=O CCCCCCC(F)C(=O)N(C(C)CNC(c1cc(C(F)F)nn1C)=O)C c1(OC)ccc(C(N2CC(N(C(=O)CCC3CCCO3)C)C2)=O)c(F)c1 N1(C(C=CC(CC)C)=O)CC2(NC(C3CC(C(F)(F)F)C3)=O)CCC1CC2 c1(CC(=O)OC)cccc(CN2CCOC(c3nc(C(=O)OC)cs3)C2)c1 c1(CC(N2CCC(C)(NC(C(CCCCC)O)=O)C2)=O)cnc2ccccc2c1 N1(C(CN(C)C)=O)CC(CO)C2(C1)CN(C(c1ccccc1C1CC1(F)F)=O)C2 C1(CN(C(=O)CSCC(F)F)CC)CCCN(C(c2sc(F)cc2C)=O)C1 Cc1cnn(CC(=O)N(C)CC2CN(C(c3cnc(C(F)(F)F)s3)=O)C2)c1 c1(C(N2C(CN(C(=O)Cc3ccoc3)C)CCC2)=O)cnccc1Br C1(CCC(=O)NCC2(C)C(C)(C)C2)CCCCN(C(c2cccs2)=O)C1 N1(C(C=NOC)=O)CCC(C)(C)C(NC(=O)COc2ccc(Br)cc2)C1 N1(C(CC2(OCC)CC2)=O)CCC(C2CCCN(C(c3sccc3C)=O)C2)C1 C1(NC(CC(C)(C)SC)=O)CCN(C(=O)CCOC2CC2)CC1c1ccccc1 c1(CC(=O)NCC2(F)CCCN(C(c3c(C)c[nH]c3)=O)C2)ccc2ncsc2c1 n1(CCCC)nnnc1C(CCCC1CC1)NCCCNC1CC=CCC1 CN1N=C(CC(=O)N2CCCC(NC(C3(n4cncn4)CC3)=O)C(F)C2)CC1=O C1(CC(=O)NC(C(=O)OC)C2CCC2)CN(C(=O)CC2CCCN2C)CCO1 c1(OC)ccc(CN=C(NCC2(C)COC(=O)N2)NC2CC(C)(CC)C2)cc1 N1(C(C2N=C(C)SC2)=O)CCC2(CCCN(C(c3c[nH]nc3[N+](=O)[O-])=O)C2)C1 C(=O)(CC(=O)NC1(C)CC(NC(c2cc(COC)on2)=O)C1)NCC#C Cc1ccc(C(N2CCCCC2CC(=O)NC2CCSC2)=O)nc1 c1(C(=O)NCCC(C)NC(c2cc(Cl)cs2)=O)ccc(OC2CC2)cc1 c1(C(=O)NCC2N(C(C(F)=CCC)=O)CCN(C)C2)cc(F)cc2cnccc12 N1(C(Cc2c(C)ocn2)=O)CCC(C2CCN(C(=O)CC3=NNC(=O)C3)CC2)C1 CCC(CC)C(F)C(=O)NCC1CC(COC)CN1C(=O)Cc1cccnc1O C(CC1=CCN(C(C)(C)C)CC1)NC(=O)NCC(CC(=C)Br)(C)C CC1C(NC(c2cn(C(F)F)cn2)=O)CCN1C(C1CC1C#N)=O N1(C(C=C(CC)CC)=O)CCC2(CC1)CN(C(C1CCCC(C(N)=O)CC1)=O)C2 c1(C(N(C(CC(=O)NCCCSCC)CC)C)=O)c[nH]c2cnccc12 S(=O)(=O)(CC(C)CC)N1CCN(c2ccn(CC)n2)CC1 C1(O)(CC(N2CC=CC2CN(C(=O)C(F)(F)Sc2cnn(C)c2)C)=O)CCCC1 Nc1c(C(N2CCOC3CN(C(=O)C4=CCOCC4)CC23)=O)sc2ncccc12 C1(C(N(CC(CC)NC(=O)Cc2c(C)cnn2C)C)=O)CC(C)CC(=O)N1 C1(C(N(CCCN(C)C(c2ccn(C)n2)=O)C)=O)CCCCC1n1cccc1 c1(C(=O)NC(C(=O)NC2CC(OC)C2)Cc2ccccc2)cc(F)ccc1O N1(C(C23N(C(C(C)N=[N+]=[N-])=O)CCC2C3)=O)CCn2ncnc2C1 c1(C(c2nnnn2C2CC2)NC(c2nc(C)cs2)CC)cc(-c2ccccc2)cs1 O=C1CCC(C(=O)NCC2(O)CCN(C(=O)CSCc3ccccc3)C2)CN1 N1(c2nnc(-c3ncc(C)o3)s2)CC2CCCC(NC(=O)C(CC)NC(N)=O)C2C1 c1(C(C)(C)C)cccc(C(=O)Nc2ccnc(NC(CO)C(F)(F)F)n2)n1 C1(NC(=O)CCSC(F)(F)F)CC12CC(NC(c1c[nH]nc1F)=O)C2 N1(C(c2ccn(C)n2)=O)CC2C3CCC(C2C1)N(C(c1ccc(S)cc1)=O)C3 C1(C(=O)NCC2C(NC(C(OCC)OCC)=O)C2)(COC)CC(F)(F)C1 [N-]=[N+]=Nc1cc(NC(c2cc(Br)nn2C2CCCCO2)=O)ccn1 N1(C(COCCOCC#C)=O)CCN(C(=O)C(c2cnn(C)c2)=O)C(C(C)C)C1 C1(CC(=O)NCC(C)(C)NC(=O)CCc2nc(=N)[nH][nH]2)CCCCC1F c1(C(N2CCCC(C)(NC(c3cc(C)ncc3)=O)C2)=O)ccc2ccccc2c1 C(=O)(CCCS(C)(=O)=O)NCC(C)(CNC(C1CCCCS1)=O)OC O=C1CCc2cc(C(N3CCCC(NC(C4C=CCC4)=O)CC3)=O)ccc2N1 C(C(C)C(=O)NCC1CCCCS1)N(C(C1(CC(=O)OC)CC1)=O)C C=CCCC(CC(C)C)C(=O)NC1(CNC(C2CCN(CC(C)C)C2)=O)CC1 C12(CNC(=O)NCCCOCC#C)CCCC1NCC2 C(=O)(C1CNC(=O)c2ccnn21)N1CC2(CN(C(CCC(=C)Cl)=O)C2)C(CO)C1 Cc1ncc(Cl)cc1C(=O)NCC#CCNC(c1cnn(-c2ccncc2)c1)=O N1(CCNC(C(n2ccc(C)n2)C)=O)CCN(C(C2(n3cncn3)CC2)=O)CC1 c1(C(N2CC(O)(CNC(C(CC)(C)O)=O)C2)=O)cnc2c(c1)c(C)nn2C C1(C(N2C(CC)CC2)=O)CC2CCC(C1)N2C(c1[nH]nnc1C)=O c1(OC)cccc(SCC(N2CCOCC2CN(C)C(C2CCCOC2)=O)=O)c1 c1(C(=O)NC2(COC)CCN(C(=O)CCOC(C)C)C2)cccc([N+](=O)[O-])c1 c1(C(=O)NC2(C)CCN(C(CC=CC=C)=O)C2)cc2c(Br)cccn2n1 c1(CN(C(=O)Cn2cc(CCSc3cccc(Cl)c3)nn2)C)cccc(I)c1 c1(OC(C(=O)N(CCN(C(C=CC(CC)=CC)=O)C)C)C)ccc(Cl)c(C)c1 CCC(CC)(CC)C(=O)NC1CCC(F)(CNC(c2ccc(C)cc2N)=O)C1 N1(C(=O)Cc2ccoc2)CC(NC(C2(C(F)(F)F)CCCC2)=O)C2CCCCC12 CC1=C(C(=O)NC2C(NC(C3(CC(=O)N(C)C)CCCC3)=O)C2)C(C)(C)CCC1 C1(C(N2CCC(N(C(=O)Cc3nnc(C)o3)CC)C2)=O)OCCOC1(C)C CCCC(C)CC(=O)N1CC2CC2C1CNC(=O)CN(C)CCc1ccccc1 c1(C(=O)NC(CCCC)CNC(=O)C#CC2CC2)cnc(OCC(F)F)c(Cl)c1 c1(NCC2(C)CCN(C)CC2)nc(Br)cn2ccnc12 N1(c2n(C)nnn2)CCc2ccccc2C(NC(=O)C(C)(C)CS(N)(=O)=O)C1 Nc1[nH]c(=NCCn2ccnc2-c2ccccc2)[nH]c2ncnc1-2 C1(C(=O)NC(c2ccc(F)c(F)c2)C)CC2(CNC2)CO1 C1(CNC(C2CC(SC)C2)=O)CC2CCCCC2N1C(C1CNC(=O)C1)=O C(CN=c1nc(C)c([N+](=O)[O-])c[nH]1)NC(C1(C)C(CC)CCC1)=O c1(C(N2C(C)(C)CC(N)C2)=O)cn2c(n1)CCC(C(F)(F)F)C2 c1(C(=O)NCCCCNC(CC(C)F)=O)cncc(-c2ccc(F)cc2)c1 c1(OC)cc(C(=O)NCC(CO)NC(C2(C)CCCNC2=O)=O)cc(Cl)c1 CN1CCN(C(c2cccnc2N)=O)CC1CNC(=O)C#CC1(C)CC1 CCCC(C)(C)C(=O)N1CCCCC(CNC(=O)CC2CCCN2C)C1 c1(OC)nc(N2CCOC(CN(C)C(c3ccn(CCF)n3)=O)C2)cc(C)n1 CCCC(CCCO)C(=O)N1CCC2(CNC(=O)C(F)(F)C3CC3)CCCCC12 n1(CC(=O)N(CC(C)C)CC(=O)N(C)CCN(C)C)ncnn1 c1(CC(=O)NCC(C)(CC)NC(CN(CCC#C)C)=O)c[nH]c2c(F)cccc12 c1(OC(N2CCCC(N(C)C)C2)=O)ccc(NS(N)(=O)=O)cc1 N1(C(c2cnc(Cl)s2)=O)CC2CC(C1)N2C(c1cnn2ccsc12)=O c1(C(=O)NCCC2CCC(NC(C(CSC)(C)C)=O)C2)n[nH]c2c(C)cccc12 C1(C(N(C2CCSC2)C)=O)CC(C)(C)CCN1C(=O)C=C1CCC1 N1(C(C2CN(C)C(=O)N2)=O)CCC2(CCN(C(C3CC(Cl)(Cl)C3)=O)C2)C1 C1(C(=O)NC2C(NC(COCCC(C)C)=O)CCC2)CCCCN(C)C1=O CN1CCC(C)(C(=O)N(C)CC2CN(C(=O)C(F)(F)C(O)C3CC3)CCO2)C1=O N1(C(C2CC(C)(NC(C3CC4C=CC3O4)=O)C2)=O)CCCN2CCCC2C1 C(CCc1ccc(Br)cc1)(C(=O)NC(C)C)N(C)Cc1ccc(CC)s1 Cc1ccc(S(=O)(=O)NC(C)(C)C(c2ccc(O)cc2)=O)cc1C Cc1[nH]c(C#N)cc1C(=O)NC(C(=O)NC1C=CCCCC1)C(C)(C)O CCC(C)CC(=O)NCCCCN(C)C(C1CC(C)C(C(=O)OC)O1)=O N1(C(C=CC(CC)C)=O)CCCC(O)(CNC(c2ccsc2)=O)CC1 c1(C(N2CCC(F)(CNC(C3CCCO3)=O)CC2)=O)cc(Cl)c(F)c(Cl)c1 C(=O)(CCS(=O)(=O)c1ccccc1)NC1(CNC(C2(C)CC(C#N)C2)=O)CCC1 C=C(C)C1OCCCC1C(=O)NCC1CN(C(C2(O)COC2)=O)CCC1(C)C Cc1oncc1C(=O)NCC(=O)NC1CC1CNC(C1CCNC1=O)=O c1(C(C)C(=O)NC(C)C=CC(=O)NC(C)(C)Cn2cccn2)ccn(C)c1 C1(CNC(c2ccsc2Cl)=O)CCCN1C(C1(CC(F)(F)F)CC1)=O c1(C(N2CCC(N(C)C)(CC)C2)C(=O)NC(CC)C)cc(Cl)ncc1Cl c1(CN(C(=O)CCn2cc(-c3ccsc3)nn2)C)cccnc1Cl Cc1cc(Br)cc2cc(C(N3CCC(N(C)C(c4ccco4)=O)C3)=O)oc12 CCN=c1[nH]cc(C(=O)N(C)CC2CCN(C(C3CC3F)=O)C2)s1 Cc1coc(C)c1C(N1CCN(C(N2CCN(C(=O)C(C)N(C)C)CC2)=O)CC1)=O C(C(C)(O)CNC(c1csnc1C(F)F)=O)NC(C(c1ccccc1)C)=O CCC(F)(F)CC(=O)NCCCNC(C1COCC1C(F)(F)F)=O C1(C(N(CCn2cc(C(N3CCOC3=O)C)nn2)CC)=O)CCC2(CCC2)C1 N1(C(CC2N(C(=O)CCC3CCCC3)C3C2CCC3)=O)CCC(F)(F)CC1 Cc1cc(Cl)c(C(N2CC(NC(c3coc(C(C)(C)C)n3)=O)CC2C)=O)cn1 N1(C(C(C)NC(CC)=O)=O)CCC2C(COC2CC(=O)NCc2cscn2)C1 c1(CC(=O)NCC(C(C)C)NC(c2cc(N)ccc2Cl)=O)ccc2nsnc2c1 C1(CNC(c2n[nH]c(C)c2O)=O)CC2(C1)CN(C(=O)CCCc1ccccn1)C2 C1(CNC(COCC(N2CCCC2)C)=O)CC2(CO1)CN(C(C1CS(=O)(=O)C1)=O)C2 c1(C(=O)NCC2C(C(NOCC(C)O)=O)C2)nccc2[nH]ccc12 OCCC(N=c1nc2scnc2c(N2CC3CCC3C2)[nH]1)c1ccco1 c1(OC)ccc(C(N2CCC(C)C(NC(C3(C)CCC(F)(F)C3)=O)C2)=O)c(Cl)n1 Cc1nn(CC(=O)NC2CC3(C2)CC3NC(=O)C(C)OCC2CC2)c(=O)o1 C1(NC(CCC(=C)C)=O)CC2CC1CN(C(c1ccc(F)cc1C(F)F)=O)C2 C#CCC(C)(C(=O)N1CCC(CC(C)O)CC1)NC(c1cc(CC)[nH]n1)=O N1(C(c2c(C)ocn2)=O)CC2CCC2(NC(=O)Cc2ccc(OCC#N)cc2)C1 CC1NC(=O)CCC1CNC(=O)C(N1CCC(Cc2nccs2)C1)=O c1(C(=O)NCCC(C)NC(c2c(Br)cnn2C)=O)ncn2c1CCCC2 c1(CC(N2CCC(C)(NC(C(C)CC3CCC3)=O)C2)=O)cccc2cnccc12 N1(C(c2c(S(C)(=O)=O)csc2)=O)CCC2(CCN(C(=O)Cc3ccco3)CC2)C1 C1(C(=O)NC2C(NC(c3csc(-c4ccccc4)n3)=O)C2)CC=CCO1 C(CCCCCNC(=O)C=CCCC(C)C)NC(Cc1c(C)ocn1)=O CC1COCC(C)N1CC(=O)NC(c1ccc(F)cc1)=O c1(N(CCNC(=O)C2CC2)CC)cc(Cl)nc(C(C)(C)C)n1 c1(C(C(=O)NCCC(C)N(C(c2ccc(C)s2)=O)C)C)c(C)noc1C Cc1n[nH]c2cccc(C(=O)NC3(c4ccc(F)cc4F)CC3)c12 N1(C(c2n(C(C)C)ccc2)=O)CCC(C)(NC(c2cc(-c3cccs3)on2)=O)C1 c1(C(=O)NC(CCOC)CNC(C23CC(C#N)(C2)C3)=O)ccc(F)c(O)c1 C1(NC(C(C)NC(=O)NC)=O)CC2CC1N(C(=O)CCC1CCC(=O)N1)C2 N1(C(=O)NC2(C)CC2C(F)(F)F)CCn2ncc(S(C)(=O)=O)c2C1 C1(CC)CCCCC1C(N1CCCC1CC1CCOC1)C(=O)NCC1CC1 c1(NC)ccc(-c2cn(CC3CCCN3C(=O)CN3CCCCCC3)nn2)cc1 C1(CC(=O)NCc2ncc(C)[nH]2)CN(C(c2cc(C3CC3)[nH]n2)=O)CC12CC2 C1(NC(C2(CC)CCCC2)=O)CN(C(=O)CCCCC#N)C2CCCCC12 N1(C(c2cccc(-n3cccn3)n2)=O)CC2CCC1CN2C(C1CSC1)=O CC1OC2(CO)CC1(C(=O)NC(C)(C)CN(C(=O)C=C1CCN(C)CC1)C)C2.O C(=O)(C(C(C)C)C(C)C)N1CCC(C(C)NC(CCc2cc(C)nn2C)=O)CC1 N1(C(c2cc(OC)ns2)=O)CCCC(NC(=O)CCC(=O)NC2CCCC2)C1C c1(CNCC(CC=C)NC(c2ccccc2)=O)ccc(S(=O)(=O)CC)cc1 c1(C(=O)OCC)cc(Br)c(C)cc1OCC(O)CNc1ccccc1OC C1(NC(C(C)NS(CCC)(=O)=O)=O)CN(C(C2(C#N)CC2)=O)CC(F)(F)C1 C1(CNC(C(C)OCC)=O)CCCC2(CN(C(=O)CCc3cncs3)C2)O1 C1(CNC(=O)C(F)C2CCOC2)CN(C(=O)C(O)C2CC2)CCC12CCOCC2 C1(NC(C2(C(=O)NC)CC2)=O)CN(C(C2COC3CC2C3)=O)CC1C c1(CC(=O)NCC(CN(C(=O)C2=C(C)CCC2)CC)(C)C)cnn2c1CCCC2 S(=O)(=O)(c1cc(C(=O)NCC2CCN2C(C2(C)CC=CC2)=O)ccc1OC)NC Cc1cnc2c(C(N3CCN(C(c4cc(Cl)on4)=O)CC(C)(F)C3)=O)cnn2c1 Cc1nc2cc(C(N3CCN(C(=O)CC(C)(F)F)C(CC(F)F)C3)=O)cnc2[nH]1 CC1(C)C2CCC1(C(=O)O)C(NC(c1c[nH]nc1Cl)=O)C2 c1(SCC(C)O)ccc2ccccc2c1.N1(C2CN(CC)C2)CCN1 CC1CCOC(C(=O)NCC=CC(=O)NC2(c3nc[nH]n3)CC2)C1 C1(NC(Cc2ccc(C)c(F)c2)=O)CC12CCN(C(C1CC=CC(O)C1)=O)CC2 CC(C(=O)NCCC1CN(C(c2cccc(CS(C)(=O)=O)c2)=O)C1)C(C)O c1(C(=O)OCC)ccc(F)cc1.C12CCN(C1)C(=O)CCNC2 Cc1ncccc1C(C)NC(C1CCCN1C(=O)C(C)C1(O)CCC1)=O C1(NC(C=CC=CC)=O)CN(C(c2ccc(Br)c(F)c2)=O)C2(CCOC2)C1 C=CC1(CC(=O)NCC(C)(CC)OC)CN(C(=O)C=CC2CCOC2)C1 O=C(C1=NOC2(CCN(Cc3cc(Br)c(F)cc3[N+](=O)[O-])C2)C1)N1CC2CC2C1 n1(CC)nnc(C)c1CNC(=O)C(c1ccoc1)NC(=O)CCc1nc[nH]n1 Cc1noc(C)c1S(=O)(=O)NC(C1CC2CN(C(=O)CCC(F)(F)F)CC2C1)=O C(=O)(C#CC1(CC)COC1)N1CCC(NC(c2c(Cl)cn(CCC)n2)=O)C1 c1(C(N2CC(NC(C=CC(=O)OCC)=O)C3C(C2)C3)=O)csc(S(N)(=O)=O)c1 Cc1csc(C(N2CCC(OCCNC(=O)C(=O)N(C)C)CC2)=O)c1Cl Fc1ccc(OCC(F)(F)F)cc1NC(=S)Nc1ccc(Cl)c(Cl)c1 N1(C(C(F)OC)=O)CC2(C1)CN(C(c1c[nH]nc1Br)=O)CC2CO Cc1ccc(CCC(=O)NC2CCC2NC(=O)CSC2CC2)o1 C1(C(N(c2ccccc2F)C(=O)CC2CCOCC2)=O)COC2(CCNCC2)C1 c1(CNC(C2(c3n(C)cnn3)CCC2)=O)cccc(CNC(C2(O)CC2)=O)c1 N1(C(c2c(OCC)ccc(C)n2)=O)CCC2CC2(NC(=O)Cn2cccn2)CC1 C1(CNC(c2ncn(C(C)C)c2)=O)CCN(C(C2(C)CNC(=O)C2)=O)CC1C C1(CC)(NC(=O)CC2(C)CC2(F)Cl)CCN(C(=O)Cc2cncs2)CC1 c1(OC)ccc(CCC(N2CCOC(CNC(=O)C(C)OC(C)(C)C)C2)=O)cc1 c1(C(=O)NCCC(C(=O)N(CC(O)CO)C)OC)ccc(O)c(F)c1 C(C(C)C)(C(O)C(=O)N1CCC(C(C)C(=O)NOCCN(C)C)CC1)OC c1(-c2scc(C(C)NC(=O)NC3CCC(C4CCNCC4)N3)n2)ccc(Cl)cc1 CCCCC(C(=O)N1CCC1C(C)O)NC(c1cccc(F)c1O)=O C(=O)(C(C)(O)CCC)N(C1CCN(C(C(C(=O)OCC)F)=O)CC1)C Cc1c(C(N2CCC(C)(NC(=O)CC(O)C(C)C)CC2)=O)sc2cncn12 C(C1CCOCC1)=CC(=O)NCCC(=O)NOCCCF c1(C(C)(C)CNC(=NCC2(CO)CC2)NCc2ccc(F)cc2)cccc(F)c1 CN1CCN(C(=O)CCc2cscn2)C(C(=O)NC2CN3CCCC2C3)C1 C(=O)(C(O)C(C)CC)NC(CC1CCN(C(c2c(OCC)nccc2)=O)CC1)C Cn1cncc1C(=O)NCC1(CC(=O)NCc2nc[nH]n2)CC1 c1(OC)cncc(C=CC(=O)Nc2ccccc2CN=c2ccnc[nH]2)c1 CC1(CNC(C2CCOCC2)=O)CCN(C(C2SC3C=CC2CC3)=O)CC1 Nc1c(F)ccc(Cl)c1C(=O)NC1CCN(C(=O)Cn2cnnc2O)C1 CCCC(C(=O)NCC1(CO)CC12CCC2)NC(c1cc(C)ccn1)=O c1(COC)cccnc1C(N1CCCC1CN(C)C(c1cn(C2CC2)nn1)=O)=O C1(NC(c2c(COC)cc[nH]2)=O)CN(C(c2cc(C)c(C)nn2)=O)C(C)(C)C1 N1(C(c2c(C)cccc2Br)=O)CCN(C(C2CC(C)C2)=O)C2(CCC2)C1 C1(CC=C)(NC(=O)Cc2cc(C)no2)CCN(C(C2CNC(=O)N2C)=O)CC1 c1(C(=O)NC2(C)CCN(C(=O)COCC3CCCO3)CC2)ccc([N+](=O)[O-])cn1 CC1CC(NC(=O)C=Cc2ccsc2)CN1C(c1cnn(C(C)(C)C)c1N)=O c1(C(N2CC3CC3C2C#N)=O)cc2ncc(-c3cnn(CCCO)c3)cc2[nH]1 C1(NC(Cc2n(C)ccc2)=O)CCC2(CCN(C(C3(C)C=CCCC3)=O)C2)C1 c1(OC)nc(Cl)ccc1S(=O)(=O)NC1CCCc2c1cnn2C(C)(C)C c1(-c2ccc(NC(CNC(CC)COC(F)(F)F)=O)cc2)ccc(Br)c(C)c1 C=CC1(COC(C2CC(=O)N(C3CCOCC3)C2)=O)CCOCC1 C(=O)(C(C)(C)NS(C)(=O)=O)NCCCC1(NC(CSC)=O)CC1 C(=O)(C(C)CC(N)=O)N1C(C(C)NC(c2c(C)oc(-c3cccs3)n2)=O)CCC1 CC1CCOC1C(=O)NCC1CC(C(N2CC(O)(c3nn[nH]n3)C2)=O)C1 c1(-c2cccc(OC)c2C)cccc2c(C(=O)NCc3noc(CO)n3)n[nH]c12 C(=O)(C1=CS(=O)(=O)CCC1)N1CCN(C(CSC(C)C)=O)C(CO)C1 C#Cc1cccc(CC(=O)N(C(CC)CC(=O)NC(C)C(C)C)CC=C(C)C)c1 c1(OCC)cc(CNC(C)CCCN=[N+]=[N-])c(OC)cc1C c1(C(C)C)ccc(C(=O)NC(CNC(c2n[nH]cc2C2CC2)=O)C2CC2)c(F)c1 c1(C(N2CCC(N(C(CN(CCC#C)C)=O)CC)C2)=O)cccc2c1CCC2 N1(C(Cc2n(C)nnc2)=O)CCC(C)(C)CC1C(N1CC(CC(N)=O)C1)=O CC(C)(O)C(F)C(=O)NCC1(F)CC(NC(C2CC3CCC(C2)O3)=O)C1 C(=O)(C(C#N)C1CC1)NC(C1CCCN1C(=O)CSS(C)(=O)=O)C C#Cc1cc(C(=O)NC(C)(CNC(c2cc(CCOC)on2)=O)CC)cc(F)c1 C1(C(=O)OC)CCCCN(C(=O)CC2(C)CCN(Cc3ccc(CC)cc3)C2)C1 N1(C(C(CCOC)(C)C)=O)CCC2(CC1)COC(CNC(=O)C(F)(F)COC)C2 Cc1nc(C(C)C)sc1C(=O)N(C)CCN(C(=O)CNC(=O)CCC(C)C)C c1(C(N2CC(CCCNC(C=CC)=O)OCC2)=O)ccc2oc(C)nc2c1 c1(C(=O)NC(c2ccncc2Cl)C)ncccc1N1CCOCC1 C1(CCNC(CCCOCCC)=O)CCCN(C(=O)CC2CCCC2C)CC1 C1(NC(c2c(C)snc2)=O)CCC2(CC1)CN(C(c1ccc(CO)cc1)=O)C2 N1(C(c2cc(C(=O)OCC)on2)C(=O)NCCCSC)CC(C)OC(C)(C)C1C CC(c1cccnc1)=CC(N1CCC(NC(C2CC(C)CCO2)=O)CC1)=O Cn1nc(C(N2CCCC2CN(C(=O)CC23CC(C2)C3)C2CC2)=O)cc1Cl C1(C(C)NC(c2cc(CN(CCC)C)on2)=O)CN(C(=O)C=C(C)C)CCO1 C1(O)(CN(C(c2c(C(C)C)ocn2)=O)C)CCN(C(=O)C=CC2(C)COC2)CC1 C(C(C)(C(=O)NC1C=CCN(C(=O)Cn2cc(Br)c(C)n2)C1)OC)OC C(CN(C)C)(CC(C)C)NC(C(c1cnn(C)c1)NC(C1C(OC)CCC1)=O)=O c1(C(=O)NC(C)(C)C(N2CC3(CCNC3=O)C2)=O)cc2ccccn2c1 c1(OCC)oc(C)nc1C(=O)NC1CCCC1NC(c1ccon1)=O c1(OC)cc(C)c(CNC(c2conc2C2CC2)c2nnnn2C(C)C)cn1 N1(C(CC(COC)C)=O)CC2(C(=O)NC(CCO)C3CCCC3)CC1CCO2 C(=O)(C1CCOc2ccccc21)NCC1(F)CC(NC(c2cc(C)c(C)s2)=O)C1 c1(OC)cncnc1C(=O)NCCC(=O)NCc1cn[nH]c1 C(=O)(CC(O)(C(F)(F)F)c1ccccc1)OC.C1(C(=O)OC)SCC(C(C)(C)C)N1C Cc1ccc2c(C(=O)NCC=CCNC(=O)C(C3CCOCC3)O)n[nH]c2c1 N(C1c2ccccc2CCC1C)C(=O)Nc1c(C)n(C(F)(F)F)nc1 C1(C)(NC(c2ccc(C(C)C)cc2)=O)CCCN(C(=O)C2=COCCC2)C1 Cn1nc2ccccc2c1-c1nc(-c2ccccc2Br)no1 CCC(C)(C)C(C(=O)N1CCCC(N(C)C(c2cc(C)oc2C)=O)CC1)OC C(CC(=O)N(CCC(=O)NC(C1CCCC1)C)CCC1CC1)SCCC c1(CN2C(C(N(C)CC#N)=O)CSCC2)cc(Cl)cnc1Br C1(C)(C(N2CC(CCNC(C(C)C3CC3)=O)C2)=O)CC=CCO1 CCC(CC(=O)N1CC(C)(C)CC1CNC(C1(C)CC1)=O)C(C)(C)C C1(C(=O)OC)CCC(C)(C)N(C(=O)CCc2cn(C(C)CO)nn2)C1 O=C(C1=CCCN(C(C2CCCS2)=O)C1)NC1CC2CC3C(C2)C13 N1(C(CC(CCC)C)=O)CC(NC(=O)Cc2c(Cl)c(CC)nn2C)CC2(CC2)C1 Cc1ncc(CNCC23CC2CN(C(=O)CCc2cnc[nH]2)C3)cn1 c1(CNC(=O)C(=O)NCc2ncco2)ccc(C2CCOCC2)cc1 CN1CCC(CN(C(=O)C(CC2CCOCC2)NC(=O)CCC2CCOC2)C)C1 c1(CNC(CC(COC)NC(=O)Cc2cnnn2C)=O)ccc(F)nc1F C(=O)(C1=NN(c2ccc(C)cc2C)C(=O)C1)NCC1C2CN(C(CC)=O)C1C2 c1(C(c2nnnn2C)NCc2occ(C)c2)cccc(C(C)C)c1 N1(CCC)CCN(C(=O)CCC2CCCN(C(C3CCCS3)=O)C2)CC1 c1(C(=O)NC(CN(C(C(C)=CC)=O)CC)C)c[nH]c2cc([N+](=O)[O-])ccc12 c12ccc3c(c1)CN(C3)C2=O.C1(N(C(C)(C)C)C)CCN(Cc2cccnc2)C1 C(=O)(C(CCC1CCC1)SC1CC1)N(CC(F)F)CCNC(C1C=CCC1)=O c1(CN(C(C)C)C)cn(C(C)C(=O)NC2CC(CC#N)C2)nn1 c1(NCC(C)NC(c2csnn2)=O)ncn(C)c(=O)c1Br N1(C(c2ccc(CC)nc2)=O)CC(C(=O)NCC=CBr)C(C)(C)C1 C1(N(C(C(C)C2CC2)=O)C)CCN(C(=O)Cc2ccco2)CC12CC2 N1(C(c2cnc(O)c(F)c2)=O)CC(NC(C2CC(F)C2)=O)CC2(CC2)C1 C(=O)(CS(=O)CCC(F)(F)F)NC1(C2CCN(C(c3ccn(CC)n3)=O)C2)CC1 N1(C(c2c(SC)nn(C)c2)=O)C(CNC(C2CC2[N+](=O)[O-])=O)CC2CCCC12 N1(C(C(CSC)C)=O)CC(=O)CC1C(=O)NCC1(C)CCOCC1 C#CCCCCCC(=O)NCC1CCN1C(c1c(C)ncnc1C)=O C(=O)(C(F)(F)C(O)C(C)C)NC1CN(C(c2ccc(S(=O)(=O)NC)o2)=O)CC1O Cc1c[nH]nc1C(=O)NCC=CC(=O)NC1(CO)CCSC1 CCC(CNC(c1ccc2cc[nH]c2c1)=O)(CC)C(=O)NCCC(C)CCO c1(NC(C2N(C(c3n(CC)nnc3)=O)CCC2(C)C)=O)ccc2occc2c1 c1(OC)cccc(C(C)(C)C(=O)N2CCC(N(C(c3nccs3)=O)CC3CC3)C2)c1 c1(NC(=O)NC)ccc(C(=O)NC(CO)C(C)NC(=O)C(C)c2cccs2)cc1 CC1(O)CCC(C(=O)NC(Cc2cc[nH]n2)C(=O)NCC2(N(C)C)CC2)CC1 c1(C(N2C(C)CN(C(c3coc(C(F)F)n3)=O)CC2)=O)cnc2c(c1)CCCO2 C1(NC(CSCC#C)=O)CC1C1CCN(C(=O)C(c2cc(F)cc(F)c2)C)CC1 N1(C(CCc2c(C)noc2)=O)CCCCC(C(=O)NCCCCN=[N+]=[N-])C1 Cn1ncc2nc(Cl)nc(NC(CNC(c3ccc4nc[nH]c4c3F)=O)CO)c12 N1(C(C2(CC=C)CC=CC2)=O)CCCCC(C(N2CCCC(N(C)CC)C2)=O)C1 C(=O)(C1=COCCC1)N(C(C)(C)CC(=O)N(C1CCNC1=O)C)C C(=O)(C(CO)C(C)(C)C)NCCCNC(CC(c1cccs1)NC(C)=O)=O N1(C(c2cc(C)c(Cl)cc2)=O)CCCC2CN(C(=O)C#CC3CC3)CC12 c1(C(=O)O)ccc(C(N2CC(C(=O)O)CCC2C(=O)O)=O)c(Cl)c1 C1(NC(C2C(C)CCC2)=O)CCCOC12CCN(c1cnc(C#N)cn1)CC2 N1(C(C(C)OCCC=C)=O)C(C(=O)NOCCn2cc(CO)nn2)CC1C c1(C(N2C(C)CCC(NC(c3cc(C)ns3)=O)C2)=O)cccc(S(=O)(=O)CF)c1 c1(C(=O)NC(CC)CNC(=O)CCc2ccc(OC)cc2)ncc2n1CCCC2 CC1(NC(N2CC(CS(=O)(=O)CCCc3nn[nH]n3)C2)=O)COC(=O)OC1 N1(C(C2C(=C)C2)=O)CCOC2(CCCN(C(=O)C3=C(CC)OCCC3)C2)C1 C=C1CCN(c2nnc(-c3cccnc3)n2CCCSC)C(CO)C1 C#Cc1cc(C(=O)NC(C)(C)C(C)NC(=O)Cc2ccc(Cl)cc2C)cc(F)c1 C1(C(=O)NC2CC(=O)N(O)C2)CN(C(=O)CCOCC2CCC2)CC1(F)F C1(C)(C(N2CCCC(N(C(COCCCC#C)=O)CC)C2)=O)CCCCC1(F)F c1(C(=O)NC2C=CC(CNC(C3CCOC3)=O)C2)ccc2c[nH]nc2c1 C1(N(c2cccnc2)C(N2CC(Cc3cn(CCCF)nn3)C2)=O)CCCCO1 N1(C(C(C)CF)=O)CCOC2(CCN(C(C3(C)CCC(F)(F)C3)=O)CC2)C1 N1(C(C2CC2c2ccc3ccccc3c2)=O)CCCc2c(F)ccc(Br)c21 Cc1ccc(C(=O)NC2CC(CNC(=O)C(C)C3CCC3)C2)c([N+](=O)[O-])c1 c1(OC(C2N(C)C(NC(=O)OC(C)(C)C)CC2)=O)cc2oc(O)nc2cc1F C(N=c1[nH]c2c(c(=NC3CC(C(N)=O)C3)[nH]1)SCC2)c1nc(CC)sc1 N1(C(CCNC(C(C2CCC(=O)N2)C)=O)=O)CCC12CCCC2 c1(C(C)=O)cnc2n1CCN(C(c1ccn(CC3CC3)c1C)=O)C2 N1(C(C(C)OC(=O)OCC)=O)CCC2(CC2NC(c2cccnc2C2CC2)=O)C1 c1(C(N2CC(C)C(CNC(c3ccncc3F)=O)CC2)=O)ncc([N+](=O)[O-])n1C Cc1cc(C(N2CCC(C(c3ccccc3F)F)CC2)=O)c(N)s1 c1(CN2CC(NC(c3cnc(C)[nH]3)=O)C(F)C2)cc(Cl)c(C)cc1O N1(C(C2CC(C)SCC2)=O)CCC2(CNC(c3nsnc3O)=O)CCCCC12 c1(C(=O)NC2C(NC(CC(C(=O)OC)(C)C)=O)CC2)nccc2ncccc12 N1(C(c2ccc(CC)[nH]2)=O)CCC(O)(C(C)CNC(=O)CCn2cc(C)cn2)C1 c1(CC(C)C(=O)NCC(F)CNC(=O)C2=CCSC2)ccccc1Br c1(C(=O)NCC2N(C(c3cc(SC)oc3)=O)CC2)cc(O)c(O)c(O)c1 c1(C(=O)NC(C)CN(C)C(C2C(C)(C)C2(F)F)=O)ccc2nc(O)nc(O)c2c1 C1(CNC(C2(CCCC)CCCC2)=O)CCN(C(=O)Cn2cnnc2)C12CC2 Cc1coc(C)c1C=CC(=O)NC1CC1NC(=O)Cn1cnc([N+](=O)[O-])c1 C1(NC(c2c(C)[nH]nc2Br)=O)CCCN(C(c2cnsc2C)=O)CC1F N1(C(Cn2c(C)cc(C(F)F)n2)=O)CCCC2(C1)CN(c1nnnn1C)CCO2 Cc1coc(C(N2CCCC2CCNC(=O)CCc2c(C)noc2Cl)=O)c1C c1(C(N2CCC3(C(N(C(C)C)C)C3)C2)=O)cc2cc(F)ccc2s1 N1(C(c2cnn(CC)c2Cl)=O)CC(NC(=O)CNS(=O)(=O)CC)C2(CCC2)C1 C(=O)(CS(=O)(=O)CC(C)C)NCC1N(C(C2C(OCC)C2C)=O)CCC1C N1(C(CO[Si](C)(C)C)=O)CC2CC(C1)N(C(c1ccc(C(F)F)cc1)=O)C2 CN=c1nc(C(=O)NC2CC(CNC(=O)C(C)(F)F)C23CCC3)cc(C)[nH]1 N1(C(C(Cc2ccco2)NC(c2c(C)c(O)ccc2)=O)=O)CCC(F)(F)C(O)C1 c1(CCC(=O)O)ccc(CNC2CCCCC2n2ccnc2)nc1 C1(CCNC(C2CCCC2O)=O)CC2CCC(C1)N2C(c1cc(CCO)on1)=O c1(C(=O)NC(CNC(Cn2cc(C(=O)NC)nn2)=O)(C)C)cc(C)c(C)s1 c1(C(N(CCN(C(c2ccc(CC)s2)=O)C)C)=O)[nH]ncc1C#N N1(C(CCCOCCOC)=O)CC(C(N2CC3CCC3(C)C2)=O)CC(C)C1 N1(C(CC(C)n2cccc2)=O)CC(=O)NCC1C(=O)NOCC(O)C(C)(C)C C1(SC(c2ccc(OC)cc2)CCC)CCC(C)N1C(=O)CC(=O)OC C(CC1=CCN(C(C2CCN(C)C(=O)C2)=O)CC1)NC(C1(CC)CCNC1=O)=O N1(C(CN(C)C(N)=O)=O)CCC(F)(CNC(c2ncccc2N(C)C)=O)CC1 c1(C(N2CC(CN(C(c3c(C)c[nH]n3)=O)C)OCC2)=O)cc(C)c(C#N)c(C)c1 C(C)(CCC(C)C)NC(C1(NC(C=CC(CC)C)=O)CC1)=O C1(CN(C(c2c(C)onc2)=O)C)CCCN(C(c2cccnc2C(F)F)=O)C1 C1(CN(C(C(C=CCCC)O)=O)C)CCCN(C(=O)C=Cc2cncn2C)C1 N1(C(C(=O)NC2COC2)CCc2ccccc2F)CCC2(CCCOC2)C1 N1(C(Cc2cccc(C)n2)=O)CCC2(CC1)CCN2C(C1C=CCN1)=O Cc1cnn(C)c1C(=O)NC(C)(C)CCCNC(C1CCN(C2CC2)CC1)=O C1(NC(c2c(C)cc(C(F)F)nc2)=O)CCc2n[nH]cc2C1C N1(C(C2C=C(C)CS2)=O)CC2OCC(NC(c3cccc(F)c3)=O)C2C1 CC1C(C(=O)N2CCC3(CCCN3C(=O)C#CC3(C)CC3)C2)=Cc2ccccc21 N1(C(CC(C=C)CC)=O)CCCC2(CCN(C(=O)CCOC)CC2)C1 CC(=O)CCCC(=O)N1CCCC(N(C(=O)CCS(N)(=O)=O)CCO)C1 c1(C(=O)NCCN(C2CCCC2)C(C=CCC)=O)oc2ccc(Cl)cc2c1C N1(C(=O)OC(C)(C)C)CC2CC(C1)N2C(C1CCCCC1(C)C)=O O=C(CC(F)(F)C(F)F)NC1CCCCCN(C(=O)CC2CCOCC2)C1 c1(C(=O)NC(C(N2C(CC)CC(O)C2)=O)C2CCCO2)ncn2c1CCC2 CC(C)(CCC#N)C(=O)NC1CC1NC(c1ccc(C2CCOC2)s1)=O c1(C(N(CC(CC)NC(c2ncccc2N)=O)C)=O)cnc(OC(C)C)c(Cl)c1 CON(C)C1CCN(S(=O)(=O)Cc2ccc(C#N)cc2)CC1 c1(C(N2CCC(CNC(c3cnoc3-c3ccco3)=O)C2)=O)csc2cncn12 C1(CNC(C=CCC)=O)CCN(C(=O)CCc2cncn2C)C12CC2 C1(NC(c2c(CC)n(C)nc2)=O)CN(C(c2cccc(N)c2F)=O)CC(C)(C)C1 c1(CNC(COC(C)(C)C)(CF)c2nnnn2CCSC)ccc(S(N)(=O)=O)cc1 N1(C(C=CC(C)(C)NC(C2CC23CCCC3)=O)=O)CCC2(CCCCO2)C1 CC(C)CC(C)CC(=O)NC1(C(=O)NC2CC3CCCC3C2)CCCC1 Cc1ccc(OCCCC(=O)N2CC(NC(C3CCCC3)=O)C2)c(Cl)c1 C1(COC)CCN(C(C2CC(NC(C3(C)CC3)=O)C2)=O)C1(C)C C1(C(C)C)CN(C(=O)CCCOc2csc(Cl)c2)CC1C(=O)OC(C)(C)C CCCC(C(=O)NCc1c[nH]nc1C(=O)NC1CNC(=O)C1)OCC C1(CN(C(C(C)NC(C)(C)C)=O)C)CCN(C(=O)CCN2C(=O)CCC2=O)CC1 N1(C(C(C)(C)OC)=O)CCCCC2(CCN(C(=O)CNC(=O)CCCCO)C2)C1 C#CCCCCCC(=O)NCC(COC)NC(C1CCN(C(=O)OC)C1)=O C1(NC(=O)Cc2ccccc2O)CN(C(c2[nH]ccc2C2CC2)=O)C2(CCC2)C1 n1(CC(=O)NCCn2cc(C3CC3)nn2)nnc(C2CC2)n1 Cc1cc(C(N2CCC(C)(C)C2CC(=O)NCC(C)(C)O)=O)cc(C)c1 c1(OC)ccn2cc(C(=O)NCCCN(C(c3csc(C)c3)=O)C(C)C)nc2c1 c1(C(=O)NC2CN(C(c3c(COC)cco3)=O)C2)ccc(C(C)(C)OC)cc1 CC1(C#N)CCCN(C(=O)C(=O)NCc2ccc3c(c2)OCC3)C1 c1(SCCc2nc(CC)nn2-c2ccccc2OC)cc(C)ccc1Br N1(C(CC2CCCC(C)O2)=O)CC2(CCN(C(=O)CN(S(C)(=O)=O)C)CC2)C1 C(=O)(C(C(C)C)NC(c1ncc(F)cn1)=O)NC(C(=O)OCC)C C=CCC(C)(CC=C)NC(=O)C1=CCC(NC(=O)CC(CC)C2CCC2)C1 CC(C)C(CCN(C)C(c1cn(C(C)(C)C)nn1)=O)NC(c1ccno1)=O N1(C(C(CC)N(C)C)=O)CCOC(CN(CC=CCl)C)C1 c1(C(N2CCC(NC(C3C(C(=O)OC)C3)=O)C(C)C2)=O)cnn2c1NCCC2 c1(C(CC)NCC2CC(C)=NO2)ccc(N2CCOCC2)cc1Cl C=CCCCC(=O)N1CCC1(C)CC(N1CCCC1C1CCOC1)=O C1(C(N(CC#CC)CC#C)=O)CCCCCCN1C(=O)C(C)OCC=C N1(C(c2scc(C)c2)=O)CCCCC(C(=O)NCC2OC(=O)CC2(C)C)C1 c1(C(=O)NCCN(C(=O)CC2CCC2)C)ccc(N2CCCCCC2)cc1 C(=O)(C(C(=O)N1CC(CNC(C2(C)CCN(C)CC2)=O)(OC)C1)C(C)C)OCC C(CCC(C(=O)NC1CCCC12CC2)NC(=O)C(C)CC#N)OC c1(N2CCCCC(NC(c3c(C(C)C)nn(C)c3)=O)C2)ccncc1[N+](=O)[O-] c1(C(=O)NCC2C(C)CCN2C(=O)COC(F)(F)F)cnc2c(cnn2C)c1 c1(CCCOC)nc(CC2CC2(Cl)Cl)n(-c2cccc(C(F)(F)F)c2)n1 CCCCCC(=O)N(C1CCN(C(=O)CCC2CCCN(C)C2)C1)CC1CC1 c1(C(=O)NC(CNC(c2c(O)cccc2Cl)=O)C2CC2)c(F)ccc2c1OCC2 C#CCC(C)(CC)C(=O)NC1CN(C(C2CC3(CC3)C2)=O)CC1C(F)(F)F n1(CC(=O)NC2C(CNC(CCCCC#C)=O)C2)c(=O)c(=O)[nH]c2ccccc12 c1(NC(C2CCN(C(C3=NOC(C)C3)=O)C2C2CC2)=O)ccc2ccncc2c1 c1(C(N2CCC(OC3CCCCC3)CC2)C(=O)NCC(=C)C)cc(Cl)sc1C N1(C(c2cccc(N(C)C)n2)=O)CCCC(B2OC(C)(C)C(C)(C)O2)C1 CC1=C(C)C(NC(=O)C(=O)NCCSc2ccccc2F)CCC1 c1(OC(N2CCC(OCC(=O)OC)C2)=O)cc(OC(C)(C)C)cc(Cl)c1 C1(NC(C(C)c2ccco2)=O)CCC(NC(c2cnc(Br)s2)=O)C1 C(C)(C(=O)N1CC(O)CO1)N(C(C(C)(C1CC1)OC)=O)CC N1(C(C)=O)CCCC(NC(=O)CC(C2CC2)NC(=O)C=Cc2cc[nH]n2)C1 c1(CC(=O)NCCCC2N(C(c3nc(SC)sc3)=O)CCC2)cncc(C)c1 N1(CC)C(=O)CCC1C(N1CC(COC)(NC(c2ncoc2)=O)C1)=O.C1(COC)CC1 O=C(CCCCC(F)(F)F)NC12CCC(C1)N(C(c1ccc3n[nH]cc3c1)=O)C2 N1(C(=O)NC2CCCC(C(N)=O)C2)CC2CCC1C(O)C2O Cc1nc2ccc3nc(NC(C4CC5CCC4N(C)C5)=O)sc3c2s1 c1(NC(C)=O)cc(F)ccc1C(=O)NCCN(C(=O)CC1CCCN(C)C1)C c1(OCC)cccnc1C(=O)NCCCCC(C)NC(c1c[nH]nc1Br)=O Cc1nc(C(=O)NCCC(C)NC(c2nc(=N)cc[nH]2)=O)ccc1Br c1(C(=O)NC2C=CCN(C(=O)Cc3ccccc3CO)C2)cn2cnnc2cn1 CCCCC(C(=O)N1CCC(NC(c2ccc(C(C)=O)cc2)=O)C1)N(C)C N(C(=NCc1ccc(F)cc1)N(C)CC1CN(S(C)(=O)=O)C1)C1CCC(CC)CC1 C1(CNC(C2CCN(CCCC)C2)=O)(CNC(=O)C(C)(C)SCC)CC12CCC2 c1(C(N(CCCN(C(C(C(C)C)O)=O)C)C)=O)cc(C(F)(F)F)cnc1N Cn1cc(C(N2CC3CC3(CNC(C3(CO)CCCO3)=O)C2)=O)c(C(F)F)n1 N#CC1(C(=O)NC2CC(NC(=O)CC3CC=CC3)C23CCC3)CC2CCC1CC2 c1(OC)ccc(C(N2CC(CC(=O)Nc3ccccc3N(C)C)C2)=O)c(F)c1 N1(C(Cc2c(C)cccc2)=O)CC(NC(c2cc(Cl)ns2)=O)C2CCCC12 c1(C(=O)NCC2N(C(C3CC(C)N(C)C3)=O)CCC2)cc(Br)cn2ccnc12 C(=O)(CCCC(=O)C(C)OC(C1(C)C=CCC1)=O)OC c1(CC)nc(C)c(-c2ccc(CNC(=O)NC3(C)CCCC3C)o2)s1 c1(SC)cc(F)ccc1C(N1CCCC(O)C1c1ccccc1)=O CC1(C)CCOC(C(=O)NCC#CC(=O)NC(c2ccccc2)(C)C)C1 C1(C(=O)NCC2CCN(C(=O)Cn3cnc(Br)c3)C2)CCCS(=O)(=O)C1 c1(C(=O)NCC2(NC(C=CCC)=O)CC2)cccn2ncnc12 c1(SCC)ccccc1CCNC(=O)Cn1cc(CC2CCCC(CF)C2)nn1 c1(C(=O)NCC2(NC(c3nc(CCC)sc3)=O)CCC2)nc(OC)ccc1Cl C#Cc1ccc(F)c(C(=O)NCC2CC2NC(C2(Cl)CC2(C)C)=O)c1 c1(C(N2CC(CNC(c3c(C)noc3C)=O)N(C)CC2)=O)cc(F)c(F)cc1O C1(CNC(c2ccn(CC)n2)=O)CC2COCC2N1C(=O)CSc1nncs1 C1(COC)CCOCCN1C(C1CCCN(CCOc2ccc(Cl)cc2)C1)=O C1(CNC(=O)NC2(C(=O)NC)CC(O)C2)CC(OC)(OC)CO1 CC1C(NC(=O)Cc2cc(Cl)ccc2Cl)CCCN1C(=O)Cn1cccnc1=O Cc1ccc2c(c1)CCC2Nc1conc1C1CCNCC1 C1(CNC(C(COC)(C)O)=O)C(C2CC2)CCN1C(=O)C(C1CCOC1)OC.OC C(=O)(N=S(C)(=O)C1CCNCC1)C1(NC(c2ccccc2)=O)C(C)(C)NC1 C12CCN(C1C)C(=O)C(CO)COC2=O.CC(C)C=CC(=O)OC(C)(C)C C(C(=O)NC1CC(CCNC(=O)C=Cc2ccccc2)C1)(C(C)C)OCC CCS(=O)(=O)C=CC(=O)N1CCC(C)C(CNC(=O)C2=C(C)OCC2)C1 c1(OCC)cncc(C(N)=O)c1.c12ccc(cc1)N(C)C2.C12CC(C1)COC2=O N1(C(C2C3CN(C(C(C(C)C)C4CCC4)=O)C2C3)=O)CCCC(O)(C2CC2)C1 c1(OC)cc(C(C(=O)NCCC2CC2)N(CCC(=O)NC(C)C)C)ccc1C c1(COC)ccoc1C(=O)NCc1cc(C(=O)NC2COC(C(C)C)C2)on1 CC(N=c1[nH]c2c(c(=NCC(O)c3cccc(C(F)(F)F)c3)[nH]1)SCC2)C(F)F S(=O)(=O)(c1ccnc(NC(c2ccc3c(c2)CN(C(C)=O)C3)=O)c1)NC N1(C(CC=CC)=O)CC2C(C(=O)NCCCn3cc(-c4ccccc4)nn3)C2C1 C1(NC(c2cc(C)ncn2)=O)CCSC12CN(C(c1cccnc1C1CC1)=O)C2 C1(CCC)(NC(C)=O)CCCN(C(c2cnn(C3CCOCC3)c2)=O)C1 N1(C(CC2CCN(C(c3cc(=N)[nH][nH]3)=O)CC2)=O)CCC(O)C12CCCC2 C(C(C)C(=O)N1CCC2CC12)NC(COCC#C)=O N1(C(c2cccc(C)n2)=O)CCN(C(c2sc(C)cc2Cl)=O)C2CCCCC2C1 N1(C(C=CC(=O)OCC)=O)CCC(C)(CNC(C2CC(CN(C)C)C2)=O)C1 c12nc(C)c(s1)C(=O)NC1(CC)CN(C1)C2=O.C1(C(N)=O)C2CC3C(C2)C13 c1(C(=O)NC2CC(NC(C3(Cl)C(C)(C)C3)=O)C2)cc([N+](=O)[O-])cc(Cl)c1Cl c1(CNC(C2(C)CN(Cc3cccnc3-n3cncn3)C2)=O)cccnc1Cl N1(C(C2CCN(C)CC2)=O)CCCCC2(CCN(C(C3CC4CC34)=O)C2)C1 c1(-n2c(C(=O)OC(c3nc(-c4ccccc4)no3)C)cnn2)c(Cl)cccc1Cl C(=O)(CCN=c1ccc(C)c[nH]1)N1CCN(C(C(CC)(C)CO)=O)CC1 CCCCCCC(=O)NC(CC(N)=O)C(=O)N1CC(CO)C1 c1(SC)ccc(C=CC(=O)N(CCCNC(C2C(C)C2(F)F)=O)C(C)C)cc1 N1(C(c2cncc(OC)c2)=O)CC2CC(NC(c3c(C)nn(C)c3Cl)=O)CC1C2 C1(CCOC)(NC(=O)CC(C)O)CCN(C(=O)CCSc2ccccc2)CC1 C=CC(C)CC(=O)NC(C(=O)NCCC(C)(C)F)C1(O)CCC1 c1(CNC2C(C(=O)Nc3ncc(C)s3)C2)cc(C)c(Br)cc1C N1(C(COC(C)C)=O)CCN(CCCCCNC(c2scnc2C2CC2)=O)CC1 N1(C(c2c(C)c(Br)cs2)=O)CC(C)(C)CC1CNC(=O)C(C)CO c1(C(C(=O)CN)=O)csc2cnccc12.c1(C(=O)NCC=CCSS)ccc(Cl)s1 CC1(C(=O)N(CCCN(C(=O)C=C2CCCC2)CC)Cc2cccnc2)CCCO1 N1(C(C2C(C)=CCC=C2)=O)CCN(C(c2ccc(Cl)cc2)=O)C(C(F)(F)F)C1 C1(NC(C2(COC)CC=CC2)=O)COC2C(NC(=O)C(C)(C)OC(C)=O)COC12 c1(C(C)C)ccsc1C(N1CCC(c2cn(CCNS(C)(=O)=O)nn2)C1)=O C12(CNC(N3CCC(c4cccc(CC)c4)C3)=O)CC3CC(CC(C3)C1N)C2 C12(C(N(C)CC3CN(C)C(=O)C3)=O)CCC(C(=O)Cc3cccnc3)(CC1)C2 N1(CC)CCN(C(=O)C(C)N(C(c2cn3c(n2)CCC3)=O)CC)CC1C N1(C(C2C(OC)CCC2)=O)CCOC2(CCCN(C(=O)CNS(N)(=O)=O)C2)C1 c1(OC)ncncc1NC(=O)C(CC1CCCC1)NC(=O)C=Cc1ccncn1 c1(C(=O)Nc2ccc(SC(F)(F)F)nc2)cccc2c1S(=O)(=O)CC2 N1(C(c2cc(C(=O)OC)oc2)=O)CCC2(CC1)CN(C(=O)C=CCO)CC(C)O2 Cc1cccnc1CNC(=O)C(C)N(C(c1c[nH]c(C)c1)=O)C1CC1 CC(CC(F)(F)F)C(=O)NCC(C)N(C)C(C1CC2(CCCC2)C1)=O CC1CCCC=C1C(=O)N(CCCNC(=O)CCc1ncc(F)cn1)CCO CS(=O)(=O)c1cncc(-c2ccc(C(=O)N(CC(F)(F)F)CCN)nc2C)c1 c1(OC)ccc(C)c(C(=O)NCCC23CCC(C2)N(C(C2(OC)CCC2)=O)C3)c1 c1(C(=O)NCC(C)(C2CC2)NC(CCOCC)=O)cc2cc(C)ccc2o1 C1(C(=O)NCC(F)Br)CC(O)CCN1C(C1CCC2CC1CO2)=O Nc1ccc(C(=O)NCC2CCCCC2NC(C2(F)CCOCC2)=O)cc1 C1(N(C)C(c2cncs2)=O)CC2CC1N(C(=O)C(c1ccccc1F)(C)F)C2 CC(C)(C(=O)NC1CCC(CNC(C2CC3CC3C2)=O)C1)c1cccs1 N1(C(CC2(C#N)CCC2)=O)CCOC2(CCN(C(=O)CC3CC3(Cl)Cl)CC2)C1 c1(C(N2CCCCC(CCC(N3C(C#C)CC3)=O)C2)=O)cccc2ccoc12 N1(C(c2cn(C)nc2)=O)CCC2CCN(C(=O)C3=NN4CCCN=C4N3)CC2C1 N1(C(=O)NCC(C)NC(C2CC=CCC2)=O)CCC(CO)CC1 c1(OC(C(=O)NC(CCCNC(C(COC)(C)C)=O)C)C)cc(C)ccc1Cl C1(CNC(COC2CCN(C)CC2)=O)CCN(C(=O)CC2CCCC2(F)F)CC1O CN=c1nc(C(=O)NC2CN(C(C3CCCN3C=O)=O)CC2C2CC2)cc(C)[nH]1 N1(C(n2cc(-c3cc(F)c(Cl)cc3Cl)nn2)=O)CCCC(O)(c2ccccc2)CC1 C1(CCC(=O)Nc2cn(CC)nc2)CCCCN1C(=O)C(C)N1CC(C)C1 C1(NC(c2cc(C(C)C)[nH]n2)=O)CCC(F)(CNC(C2CC2C(F)F)=O)C1 c1(OC)cccc2c(N3CCOC(CNC(=O)CCn4cnnn4)C3)ncnc12 N1(C(Cc2n(C)cnn2)=O)CCCCC(NC(=O)CCn2ncn(C)c2=O)C1 C(=O)(C1=CNC2=NCCC2=C1)N1C(C)C(NC(=O)CC2CC2(Cl)Cl)CCC1 CC(N=c1[nH]c(=NCc2nnc(O)o2)c2c(F)cccc2[nH]1)c1cc(Br)ccn1 N1(C(c2c(CC)ncs2)=O)Cc2n[nH]cc2C1C(=O)N1CCC(CCN(C)C)C1 C(C(C)(C)C(=O)NCCC(C)N(C(=O)Cn1cnnn1)C)OCC CC1(C)CN(C(c2cnc[nH]2)=O)CCN(C(c2ncoc2Br)=O)C1 c1(C(N2C(CNC(CC(C)F)=O)CC(O)C2)=O)ccc2cccnc2n1 c1(C(N2CC(COC)(NC(=O)C(C3CCC(=O)N3)C)C2)=O)ccc(F)cc1O c1(C(=O)NCCC(C)NC(C2CCCC2(F)F)=O)ccc(-c2ncc[nH]2)nc1 C(CCN=C(NCC1=NOC2CCCCC12)N1CCCC(CSC)C1)OC N1(C(C2C3CC2N(C(c2cnon2)=O)C3)=O)CCc2ncccc2C1 C1(NC(c2n(CCCC)ncc2)=O)CCCCN(C(=O)CC2COC(C)(C)C2)C1 Cn1cc(C(N2CCC(CCNC(c3ccc(O)cn3)=O)CC2)=O)c(O)nc1=O N1(C(C(CCC)OC)C(=O)NC(C)(C)C)CC2C(C1)C2(F)F C1(NC(c2scc(COC)c2)=O)CCN(C(c2cn(CCO)nc2C)=O)C1(C)C c1(COC)cccc(C(N2CC=CC2C(N2CC[Si](C)(C)C2)=O)=O)c1 c1(CC(=O)NCCCCC(C)NC(=O)C2=NOC(C)C2)ccc(C#N)cc1F CC1CCC(Cl)=C(C(=O)NCC(O)CCNC(=O)COc2cccc(F)c2)C1 CCC(C(=O)OC)C(=O)NCC1CCCCN1C(c1cc(Cl)ccc1F)=O CC1C(NC(C2CCCN2N=O)=O)CC2CCC1N2C(c1ccnc(C#N)c1)=O N1(C(C2(C)CC(C)C2)=O)CC2C(NC(=O)COC(F)F)CS(=O)(=O)C2C1 c1(CNC(C(=O)N(C)Cc2nnc(C(=O)OCC)s2)=O)ccc(C)cc1F c1(CC(=O)NCC(C)CNC(C2(C3CC3)CCOCC2)=O)cccc2sccc12 Cc1noc(C)c1C(C(=O)NC1COC1)N(c1ccccc1)C1CC1 Cc1ccsc1CNCC1(c2ncccn2)CCOC1 C#Cc1ccc(C(=O)NCC2CN(C(=O)Cc3ccnc(Br)c3)C2)cc1Cl c1(CN(CC)CC)ccc(-c2ccc(Nc3cccc(O)c3)nc2)cc1 c1(C(=O)NCC(CC)NC(=O)CC2CC(C)=NO2)c(C)nn(C)c1N C1(CNC(C(C)(F)F)=O)COC(C(F)(F)F)CN1C(C1CCCC1)=O c1(CN(C2CCCC2)C#N)ccc2c(c1)CC(C)O2.C12(CC1)C(C)NC2 N1(c2nnc(Cc3n(C)ccn3)n2CC2CCOC2)CCOC2(CCCC2)C1 c1(C(N(C2CCN(C(c3cccc(NC(C)=O)c3)=O)C2)C)=O)nc(C)ccc1C c1(C(=O)NC2C(NC(C3CN(C)C(=O)N3)=O)CC2)cc(Cl)ccc1F C(CCN=C(NCC1CCCC1(F)F)NC1CCCSC1)OC(C)C N1(C(C2(SC)CCC2)=O)CC2(CC(CNC(C3(CF)CCOCC3)=O)C2)C1 Cn1c(C(N2CCCCC2CCNC(C2CC(=O)NC2(C)C)=O)=O)cccc1=O C1(NC(C2(C)C(C)CCC2)=O)CCC2CN(Cc3ccncc3Cl)CC2C1 C1(C(N2CCCC(CNC(CCCOC(C)=O)=O)C2)=O)Cc2nn(C)cc2C(=O)N1 Cc1cccn2ncc(C(N3CCC4C(CCN4C(=O)COC4CCC4)C3)=O)c12 c1(C(=O)OC(C2(O)CN(C(=O)OC(C)(C)C)C2)C)cc(C(C)(F)F)ccc1C C(=O)(C(COCc1ccccc1)OC)N(CCCC)CCNC(C)=O C1(c2ccccc2)(C(=O)NC(CN(C(COCC)=O)CC)C)CCOC1 C(=O)(CCCCCSC)N1CCC(CC)C1CNC(C1CC12CCCC2)=O N1(C(c2cn(CC)nc2C)=O)CC2CC1CN2C(=O)CCC1CCOC1 C(=O)(C(C)(C)C(F)F)N(CC(CNC(c1cc(OC)no1)=O)O)C C(CCCN=c1ccnc(N2CCOC(c3ccc(Cl)cc3)C2)[nH]1)OC C1(CNC(=O)CC2(CO)CCC2)CCCCN(C(C2C=CC=CC=C2)=O)C1 c1(C(=O)NCCC2CCCN(C(CNC(C=CSC)=O)=O)C2)cc(C)ccc1O CC1=CC(C)=NS(=O)(=O)N1CC(=O)NC1CCN(C(=O)Cn2cccc2)CC1C C1(CCOC)(C(=O)NC2CCC2N(C)C)CCN(C(=O)CCc2csnn2)CC1 C1(CCC)CCCC1C(=O)NCCC1(CNC(=O)Cc2csc(=N)[nH]2)CC1 c1(OC)cc(OC)nc(C(N2CCC(C(C)NC(=O)CCCC3CC3)CC2)=O)n1 c1(C(=O)NCCOCCCNC(COC(C)C)=O)csc(NC(C)=O)n1 c1(NC(c2cc(C)[nH]n2)=O)cc(C(N2CCOCC2)=O)ccc1C C1(C(=O)NCCNc2c(C)ccnc2)CCC(C)C(C)C1 C12(C(=O)NCC(CC)(C)C)CCC(CC1)N(C(=O)C(C)C1CCC1)C2 C1(NC(CC2CCCN(C)C2)=O)CCS(=O)(=O)C12CN(C(C1(CO)CC1)=O)C2 Cc1nn(C)c(Cl)c1CC1CCCCC1C(C(=O)N)N(C)C(C1(C)CC1)C c1(OC)cc(C(N2C(C)CN(C(=O)C(O)CSC)CC2C)=O)c2occc2c1 C12(CNC(C3CCS3(=O)=O)=O)CCCC1N(C(=O)CSCCC(F)(F)F)CCC2 c1(C(=O)OCC)nccc(C)c1NC(C1(C)CC1(Cl)Cl)=O C1(CN(C(=O)C(C#N)C2CC2)C)C2CN(C(c3ncncc3Br)=O)CC12 Cc1cc(N2CCC(C(F)(F)F)(CO)C2)nc(=NCC(C)CC2CCC2)[nH]1 N1(C(c2cnoc2C2CC2)=O)CCN(C(=O)CCc2cocn2)C(C2CC2)C1 N1(C(c2cc(OC)no2)=O)CCN(C(C2CCN2C)=O)CCC1C c1(N(C(C)=O)C)ccc(-c2nc(-c3cc(Cl)ccn3)nn2C(C)C(C)(C)C)cc1 c1(C(=O)NCC(C(=O)N(C(C)C(N)=O)C)CC2CC2)cc2n(n1)CCO2 c1(C(N(CC(CC)NC(C2(C(C)C)CC2)=O)C)=O)ccccc1CC#N C(=O)(CC(C)C(C)(C)NC(c1ncoc1CC)=O)NC(C=C)C1CCC1 c1(CCC)nc(CNC2CC2C(=O)Nc2cnc(C)cn2)c(Cl)[nH]1 Cc1nc2cncc(C(=O)NCC(C(C)C)NC(=O)C(F)OC(F)(F)F)c2[nH]1 c1(C(N2CCC(CN(C(C(C)S(C)(=O)=O)=O)C)C2)=O)c2ccccc2nn1C c1(C(=O)NC2(CC=C)CN(C(=O)CSCC3CCCCO3)C2)cc(C)sc1C O=C1CCC(C(=O)N2C3CCC2CC(NC(C2CNC(=O)N2)=O)C3)=NN1 C12(C(N3CC(NC(C45CCCCC4C5(F)F)=O)C3)=O)CCCN(CCC1)C2 C1(CNC(N(C(CC#C)C)C)=O)CC(O)(C(F)(F)F)C1 C(CCCCC(=O)N1CCCC1C(C)(C)CN(C(=O)C(F)OC(F)(F)F)CC)ON=[N+]=[N-] c1(CNCC23C(CN(C(C(n4ncc(C)c4)C)=O)C2)C3)cc(O)ccc1Cl c1(C(C(=O)NCC=C)N(C(C)C(=O)OC)CC(C)C)nn(CC)cc1Br Cn1nccc1C(F)=CC(N1CCC(C)(CNC(C2CC3CCC2O3)=O)CC1)=O N1(C(c2cc(C)ncn2)=O)CCC(NC(=O)CC2CCC(C3CC3)O2)C12CCCC2 C(C(O)C(=O)NC(CNC(=O)CSc1ccc(Cl)s1)C(C)C)=CCCC C1(C(=O)OCC)CN(CCCC(=O)NC(=O)NC(C)(C)C)CC12CCC2 C(=O)(CCCC(C)(C)C)NCCC1CN(C(C2(CC)CC(C)(C)C2)=O)C1 c1(COCC(=O)N(C2CCN(C(=O)C(F)=CC3CC3)C2)C)cccc(C(N)=O)c1 Cn1ncc(CNC(=O)CC2NC(=O)NC2=O)c1C(=O)NCc1ccco1 C1(NC(Cn2ncc(C)c2)=O)CCCC(Nc2ncnc(=N)[nH]2)C1 C(c1ccc(Cl)cc1)=CC(=O)NCC(C1CC1)NC(CCNC(C1C(C)C1)=O)=O C12(NC(C(=O)NCCN(C(=O)CCc3ccccc3)CC)C)COC(C)(C1)C2 C1(C(=O)NC(CNC(=O)C=Cc2ncc[nH]2)C2CCC2)CCc2nnnn2C1 C1(CC(=O)N(CC(CC)NC(c2cc(OCC)n[nH]2)=O)C)CCCNC1=O C(=O)(C(C)(C)CSC(c1ccccc1)C)OCC(=O)N(c1ccccc1)C(C)C N1(C(C2(CC#C)CC2)=O)CC2CC(C1)N(C(=O)C(C)CC(C)(C)C)C2 C(=O)(CCC(C)C)N(CC(=O)N(C)CCC1CCCN1C)CCOC C1(CN(C(CNS(CC)(=O)=O)=O)C)CCCN(C(c2cnn(C3CC3)c2Cl)=O)C1 N1(C(CN(CCOC)C)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)CCC1C C1(CC(N2CC(CC=C)(NC(=O)Cc3cc(C)cs3)C2)=O)CCN(OC)CC1 CCC(CC)C(C)C(=O)NCC1(C2CC2)CCN(C(C2CCOC2)=O)C1 c1(CCNC(CCC#C)(C)c2nnnn2C(C)CC)nc2cnccc2[nH]1 C(C(C)(C)C#CC(=O)N1CCC(CO)C(O)C1)NC(COC(CC)(C)C)=O C(=O)(C1=CCCCCC1)N1CCCC(NC(=O)CCn2cnnn2)C1 c1(CC)nc2c(C(=O)Nc3cc4c(cc3Br)CCC4)ccnc2[nH]1 C1(CC)C(NC(=O)C(O)COC)CCCN1C(c1ccc(C(N)=O)cc1)=O C(=O)(CCCCCCCCCO)NC1CC(F)(CNC(=O)C=CC2CCCC2)C1 C1(C(N2CC(O)(c3cnn[nH]3)C2)=O)(CC)CCCN1C(=O)C=C1CCOCC1 N1(C(C(C2CCC2)OCC)=O)CC2(C1)CN(C(C1(CO)CCOCC1)=O)CCO2 N1(C(c2cnc(C(C)O)s2)=O)CC2(C1)CN(C(C1(CC3CCC3)CC1)=O)C2 N(C(=NCC(C)C)NC1CCCn2nc(C)nc21)CC(CC=C)(C)C C1(C2CC2)(CNC(c2ccnc(CO)c2)=O)CCN(C(=O)C(=O)C(F)(F)F)C1 N1(C(C2C(NC(CCC(=O)NCC)=O)CC2)=O)CCOC(C)(C)CC1 c1(OC)cccc(O)c1C(=O)NC1CCC(CCNC(=O)C(O)CCSC)C1 C(=O)(CCC(C(C)C)NC(=O)C(C)CC(N)=O)Nc1c(OC)ccnc1 C#CCC(C)(C)C(=O)NCC1C2CCC(C2)N1C(=O)COCCN(C)C CC1(NC(=O)C2CC2)CCN(C(C23CCC(CO2)C3)=O)CC1 C1(CCC(=O)Nc2cnn(CCF)c2)CCC(C(=O)NCC2CCCSC2)C1 c1(C(N2CCC(CF)C2)C(=O)NCCC(=O)OCC)nc(Cl)cc(Cl)c1C c1(C(N2CCC(O)(C(C)CNC(=O)COCCF)C2)=O)cccc2sncc12 C1(N(CC(=O)N(C2CCCC2)C(C2CCCCN2)=O)C(C)=O)CCS(=O)(=O)C1 CCC(O)(CC)CCNC(C1CC(NC(c2sccc2C#N)=O)C12CCC2)=O C1(C2CCOCC2)(NC(C(COC)C)=O)CC1.c1(C2C(=O)N2)cnn(C)c1 c1(C(=O)NC2CCC(NC(C3CS(=O)(=O)CCO3)=O)C2)ccc2sccc2c1 CCC(CNC(=O)CC=CCNC(c1cc(C(C)C)n(C)n1)=O)(CC)OC C(C(C(C)(C)C)NC(c1cnn(-c2ccc(Cl)cc2)n1)=O)NC(CC(C)OC)=O C1(NC(c2nnnn2C(C)(C)C)C2(SC)CCC2)C2CCCOC12 C1(NC(C2CCC(=C)CC2)=O)CN(C(c2ccsc2C#N)=O)CC1N=[N+]=[N-] C(=O)(CCC(F)(F)C(=O)N1CCC(C)C(NC(=O)CC2(O)CCCC2)C1)OCC n1(CC(=O)NC(c2cc(C(=O)NCC(C)Cc3cn[nH]c3)no2)C)cnc(=N)[nH]1 c1(C(N2CC3(CN(C(C(C)=C4CC4)=O)C3)C2)=O)cc(C)c(C)c2ncccc12 C1(C(C)C)(CO)CCCN(N2CC(NC(=O)OC(C)(C)C)C3(CC3)C2)C1 N12CCC(C(C)(C)C1)C2=O.c1(C(=O)OC)cc(C)sc1NC(=O)CCC(=O)N(C)C C#CCC(C(=O)NCc1cncn1C(C)C)NC(=O)Cc1ccc(C)o1 C#CC1(O)CC(C(=O)NC(C)C(C)(C)NC(=O)C(C)OCc2ccncc2)C1 c1(C(=O)NC(C(C(C)C)NC(COCCC)=O)C)ccn2ncnc2c1 c1(C(=O)NCC(CNC(COC)=O)C)c(C(F)(F)Cl)n[nH]c1C C1(NC(C(C2CC2)SC)=O)C2CC1N(C(=O)CCCc1nc(C)no1)C2C c1(C(=O)NC(CC)CNC(C2CNC(=O)N2)=O)cc(Br)c2[nH]c(C)nc2c1 C1(C(C)NC(COCCCC#C)=O)CCN(C(C2(COC(CC)CC)CC2)=O)C1 C1(CNC(c2cnoc2)=O)CC2(CCOCC2)CN1C(c1cc(F)ccc1Cl)=O C12(C(=O)NC3CCN(S(C)(=O)=O)C3)CCCC1CCN2 n1(CC)cc(CC(=O)NCc2ocnc2C(=O)NCC(F)Cl)nn1 Cn1cc(C=CC(=O)NC(Cn2cncn2)C(=O)NCCc2nccn2C)nn1 C1(CNC(c2c(C)sc(O)n2)=O)(NC(=O)Cc2nc[nH]n2)CC2CCC1CC2 c1(C(N2CCC(CC=C)(C(=O)NCC(C)(C)CN(C)C)C2)=O)occ2c1CCC2 CC1NC(=O)CCC1NC(=O)CC1(C)CCN1C(C1CC1c1ccco1)=O C(=O)(CC(C)(C)C(C)=O)N1CCC(C(N(CC(CC)C)C)=O)C(C)C1 N1(C(C2(C#C)CC2)=O)CC2(C1)CN(C(C1CCN(C)C1)=O)CC(C)(C)O2 C1(OC)CC(C(N2CCN(C3CC3)CC2)=O)N(C(=O)Cc2ccccc2F)C1 C1(=CC(=O)NCCC2(OC)CN(C(=O)C(O)CN(C)C)C2)CCN(C)CC1 C1(C(=O)NCCN(CCCc2ccccc2)C2CC2)(OC)CCSC1 C1(C(N2C(C)(CNC(=O)CCc3cnn[nH]3)CCC2)=O)CCC2(CCOCC2)C1 C1(NC(C2(C=C)CCC2)=O)CN(C(c2ccnc(SCC)c2)=O)CCC1CO Cc1ccc(NC(=O)CC2(C)CCN2C(c2ccc(O)cn2)=O)c(O)c1 C(CCCCCNC(=O)CSc1nccn1C)N(C(c1c(C(C)C)scn1)=O)C N1(C(C(CC)N(C)C)=O)CC2(CNC(=O)C=Cc3scnc3C)CCC1CC2 N1(C(c2cncc(-c3cncc(OC)c3)n2)=O)CCc2c(C)cc(Br)cc2C1 C(CC(C)(C)C(=O)NC1CCCN(C(c2ccc(F)c(O)c2)=O)CC1)OC C1(C(=O)OC)CC(C)N1C(C1CCC1Cc1ccccc1)=O Cc1cc(CC(=O)N(CCC(=O)NC2CCOCC2C)CC2CC2)n(C)n1 N1(C(C(CC)SC)=O)CCOC(CCNC(=O)CC2(O)CC2)C1 N1(CC(C)C)CCCC1C(=O)NCC1(CNC(=O)C=Cc2cscn2)CC1(F)F C12(CNC(C3CC(=C)C3)=O)CCCCC1N(C(=O)C(C)CCOC)CCC2 C(C)(N=c1[nH]c(Cl)ncc1C(F)(F)F)C1CCN(C(C2(C)C(CC)CCC2)=O)C1 C1(C)(C(=O)NC(C2CN(C(c3nnc(O)cc3O)=O)CCO2)C)C(C)(C)C1(C)C CC#CC1CN(C(C2CCN(C(=O)CCCN(C)C)C2C(C)C)=O)C1 C(c1cccc(Cl)c1Cl)=CC(=O)NCCCCNC(C1CC2CCC1O2)=O N1(C(=O)C=Cc2cccnc2)CCC2(CCN(Cc3cccc4nc[nH]c34)C2)C1 C12(NC(C3C4CCCCCCC34)=O)CCCC1N(c1ccc3cc[nH]c3n1)CC2 Cc1cnc(N2CCCN(C)CC2)c(S(=O)(=O)NCc2ncc(Br)cc2F)c1 c1(C(N(CC(O)CNC(C23CC(C)(C2)C3)=O)C)=O)cccc(C(N)=O)n1 c1(C(N2CC3CC(NC(=O)Cn4ncnn4)CC3C2)=O)cc2ccc(Cl)cc2o1 Cc1cccc2oc(N3CCC(CNC(=O)C4=COCC4)C(C)C3)nc12 C(Cc1ccccc1)(C(=O)N(CCNC(C1OCC1(C)C)=O)C(C)C)OC C(=O)(C(C)(C)C(F)(F)F)NC(CNC(c1cn(CC(CC)O)nn1)=O)CO C1(NC(CNC(=O)OCC=C)=O)C=CC(CNC(c2csc(C(C)C)n2)=O)C1 C1(NC(C(C)c2ccsn2)=O)CCC(O)CN(C(c2cn3ncccc3n2)=O)C1 N1(C(CC2(C)CCCC2)=O)CC(NC(C2CCCC(O)C2)=O)CC2(CC2)C1 c1(C2C(C(N3CCC(C)(CNC(CCCSC)=O)C3)=O)C2)c(F)cccc1Cl c1(C(=O)NCC2C(NC(C3CCC(=C)CC3)=O)C2)ccc(F)cc1C(F)(F)F N1(C(CN(CC(C)C)C(=O)CC2CC3CC3C2)=O)CCCC(CCF)C1 c1(C(N2CCC(NC(C3CCCC3)=O)C2)=O)cc(C(F)(F)F)ccn1 c1(N2C(CCCNC(c3cnn(CC4CCCC4)c3)=O)CCC2)ncc(I)cn1 N#Cc1cc(C(=O)NC2C3CC(O)C2N(C(c2csnn2)=O)C3)cc(O)c1 CC(C)(C#N)CC(=O)NCC1CCCC(NC(=O)C(C)(C)N2CCOCC2)C1 N1(C(C2(CC=C)CC2)=O)CCC2CCN(C(=O)C=C(C)c3ccccc3Cl)C2C1 Cc1nn(C2CCCC2)c(Cl)c1C(N1CCC(CO)(NC(=O)COC(C)C)C1)=O C(C1=CCN(C(C23CC(CN2C2CC2)C3)=O)CC1)NC(CC1C(=O)NC(=O)N1)=O C#Cc1cccc(C(=O)NC(CN2CCN(C(=O)CN(C)C(N)=O)CC2)C)c1 N1(C(C(CC)O)=O)CCn2nc(C)c(CNC(c3cc(=O)n(C)o3)=O)c2C1 C12(CNC(COCC)=O)CCC(CNC(c3cc(CC)ccc3Cl)=O)(CC1)CO2 N1(C(CCCC)=O)CCC2CCC(NC(c3cc4c(C)cccn4n3)=O)C1C2 CC(C)CC(C(=O)N(CCCNC(=O)Cc1cccs1)CCO)C(N)=O Cc1nc(NC2(c3ncc(C)o3)CC2)cc(=NCC2CCCCN2C)[nH]1 N1(C(CN(C(CNC(CCC)=O)=O)CCOC)=O)CC2(CCC2)OCC1C CC1CN(C(=O)C(O)C(C)c2ccccc2F)CCN1C(c1cc(CF)on1)=O Cc1cc(C(=O)C(N2CCC(C)(NC(C3CC4(C3)CC4F)=O)CC2)=O)ccc1F C1(NC(c2cnc(C)[nH]2)=O)CN(C(=O)CCc2cn(C)nn2)CCC1(C)C c1(C(=O)NC2(CC(=O)NC3CCN(CC)CC3)CCC2)cc2[nH]ccc2cc1Cl C1(NC(C(=O)NCC2CC2)=O)CCN(C(c2occ3c2CCC3)=O)CC1CO N1(C(CC2CC(CC)OCC2)=O)CC2CC(C1)N2C(=O)C(C)(C)CN(C)C Cc1cc(CNCC2CN(C)CCN2C)c2ccccc2n1 N1(C(COCCOCC#C)=O)CCC(CNC(C23COCC2C3)=O)C12CCC2 C=C1CC(C)(C(=O)NCCN(C(=O)CCCC2CCCCC2)CC(C)O)C1 C1(C2CCN(C(=O)C(F)CC3CCCC3)C2)(NC(=O)CCCC2CC2)CC1 c1(OC)ccc(C(N2CCC(C(F)C(N3CCNCC3)=O)CC2)=O)c(Br)c1 C(=O)(C1=CCCC1(C)C)N(C1CCC(NC(C2CN(CC)C(=O)CC2)=O)CC1)C Cc1scnc1C(=O)N(C(C)(C(=O)N1CCC1CC(C)(C)C)C1CC1)C c1(C(=O)NC2C(NC(c3c(C)n(C)nn3)=O)COC2)cc2nnn(C)c2s1 C1(CNC(c2cc(C(C)=O)[nH]n2)=O)CC(O)CN1C(c1ccc(C(N)=O)cc1)=O C(CC(C(=O)NC(C)CNC(=O)CCSc1cccc(Cl)c1)N(C)C)SC C1(c2cccc(OC)c2)CN(C(=O)C(F)C2CCC2)CCN1C(=O)CC(C)(F)F C1(C(N(C(CCNC(CN(C(C)C)C)=O)C)C)=O)CCc2cc(F)ccc2O1 N1(C(C(CNC(=O)CC(COC)COC)OC)=O)CCn2c(C)nnc2C1 O=C1CC(C(=O)NC2COCC2NC(C2(CO)CCC2)=O)c2ccccc2N1 C(C(CC(F)(F)F)NC(=O)C(F)F)NC(C1CN(C(CC)CC)C(=O)C1)=O O=C1NC(=O)C2(CC(C(N3CCN(C(C4CCCCC4O)=O)C(CF)C3)=O)C2)N1 C(CCC1CCC1)(C(=O)NCC(C)C(C)(C)C)NC(c1c(CC)csc1)=O CC1CN(C(C2C3CN(C(=O)CCc4cccc(O)c4)CC23)=O)CCC1=O N1(C(CNC(CC)=O)=O)CCC2(CC1)C(OC)CC2NC(c1ncn(C)c1C)=O Clc1ccccc1-c1ccc(-c2ccc(OCC3CC3)s2)cn1 Cc1ccc2occ(C(=O)NC(C)C(CO)NC(C3CN(S(N)(=O)=O)C3)=O)c2c1 C(CN=c1nc(C#N)[nH]cc1Cl)=CCNC(C(CC)C(C)O)=O c1(C(=O)NC(C2CN(C(C3CCCC3O)=O)CCO2)C)ccn2cccc2c1 c1(N2CC(COC)N(c3ncc(C(F)(F)F)cn3)CC2)ncnc2n[nH]c(Br)c12 N1(C(c2ccc(N(C)C)nc2)=O)CCC(CNC(=O)Cc2cnns2)C12CC2 N#Cc1ccccc1CCC(=O)NCC12CCCN(C(=O)CCCC3CC3)C1C2 c1(CCNC(c2n(CC)ccc2)=O)cccc(-c2cccc(F)c2)c1 C1(NC(C(CC=C)OC)=O)COC2C(NC(=O)CCC(C)CN(C)C)COC12 C(=O)(CCCCCSC)NCC(C1CC1)NC(C(COC)N(C)C)=O CCCCC(O)C(=O)N1CC(NC(=O)C(F)F)C(C(F)F)C1 C#CCC(C)(C(=O)Nc1ccc(F)c(CC)c1)NC(C1CCOC1(C)C)=O C1(C#N)(CC)CCN(C(C2(C)CCC(C)C2(C)C)=O)CC1 N1(C(C2C(CC)CN(C(=O)CC3(O)CCCC3)C2)=O)CCC(C2CCCC2)C1 Cc1ccc2cc(CNC(=O)C=C3CCN(C(=O)C(C)NC=O)CC3)ccc2n1 c1(CCC(N2C(C3(NC(=O)C(O)C4CC4)CC3)CCC2)=O)ccc2ncsc2c1 C(=O)(CCCC(=O)NCC1CCOC1C(F)(F)F)NCC1(OC(C)C)CC1 Cc1cc(C(C)NC(=O)C=CC(C)(C)NC(c2ccn(C3CC3)n2)=O)no1 Cc1cc2[nH]c(C(N3CCC(n4cc(-c5cc[nH]n5)nn4)C3)=O)cc2o1 c1(C(=O)NCCNC(CC(C)C2CCCO2)=O)cc(Cl)cc(Br)c1 C12CCCC1C(=O)NC(C)(C)C=CC(=O)N2.C1COCCO1.CCSC c1(C(N(C(c2cn(CCN3CCOCC3)nn2)C)C)=O)cnn2c1OCCCC2 C1(CNC(C(C)(C)OC(C)C)=O)CCCC(CNc2ccns2)C1 CCCC(C)(CCC)C(=O)NC(C)CNC(=O)C(C)(O)C(F)(F)F C=C(C)CCCC(=O)NC1CC(C(=O)NCC(CC(C)C)OC)CC1O C(=O)(C1=CC2(CCOCC2)C1)NC(C(C)NC(CCC1CC(OC)C1)=O)CO CCC(C)C(C)CNC(C1(C)CN(C(C2(n3cccn3)CC2)=O)C1)=O C1(O)(C(=O)NC2N(C(C(CC)CN(C)C)=O)CC2)CCCC1(C)C N1(C(c2c(C)nc(C)s2)=O)CC(=O)NCC1C(N1CC=CC(O)C1)=O C12(CNC(C=C(C)Cl)=O)CCC(CN(C(=O)CCN(C)C(=O)OC(C)(C)C)C1)C2 N1(C(c2cccc(SC)c2)=O)CCC(NC(C2(C(F)(F)F)CC(F)C2)=O)CC1C N1(C2CCN(CC)C2=O)CC(C(=O)OC)S(=O)(=O)C(C)(C)C1 C(=O)(C(F)C(C)CNC(c1sccc1F)=O)NCc1cc(OC)ncn1 N1(C(COCC#C)=O)CC(NC(=O)C(F)C(F)(F)F)CC12CCC2 CN1CCCCCC1C(=O)NC1(CC(=O)NC2C(O)C3CCOC23)CCC1 C1(CNC(C2CCN(C)C2=O)=O)CCN(c2nccc(C(C)(C)C)n2)C12CC2 c1(C(N2C(C(C(=O)OC)NC(=O)CC(C)C)CCC2)=O)ncc(C)cc1Br c1(C(N2CC(F)(C(=O)NCCOCCC#C)C2)=O)cc(N)cc(F)c1 N1(CCNC(=O)CC(C2CC2)C2CC2)C(=O)NC2(CCCCC2C)C1=O CC1CCOC1C(N1CCCC1CN(C(=O)CCc1nc[nH]n1)C)=O c1(CC(=O)NC2CC(NC(C(Br)=C(C)C)=O)C(O)C2)cccc(C)c1C C1(C(=O)NC(C#C)CC2CCC2)(CNC(=O)CCC2CCCO2)CC12CCC2 C1(N(C(=O)C=C(Cl)Cl)CCF)CCCN(C(c2ccc(-c3cnco3)cc2)=O)C1 C(=O)(C(C)(C)C(O)C(C)C)NCCCCC(=O)NC(COCC)CO N1(C(C2C(c3cc(C)sc3)C2)=O)CCCCC1C(C)(C)CNC(c1ccon1)=O c1(C(N2C(CNC(=O)COC3CCCOC3)CCC2)=O)ccnc2[nH]nnc12 C1(CN(C(C=COCC)=O)C)CCCN(C(=O)C(=CC2CCCC2)C)C1 N1(CC)CC(C(=O)NCc2cc(C(N3CC(CCO)C3)=O)cs2)CC1=O c1(CC)ncc(CNC(=O)C(C)N(C(=O)CC2CC(C)=NO2)C)[nH]1 CC1CCC(C(=O)NCCc2noc(=O)n2C)CN1C(c1ccc([N+](=O)[O-])o1)=O N1(C(C(c2ccccc2)C)=O)CCOC(C(C)NC(C2CCCN2C)=O)C1 C(N=c1[nH]cnc2c(OC)cccc12)C1CCN(C(C(COCC)N=[N+]=[N-])=O)C1 N1(C(C2CC(C#C)(O)C2)=O)CCCCC(CCC(=O)NCC(=O)OC(C)C)C1 C12(C(=O)NCC3N(C(c4c(Cl)cn(C)n4)=O)CC4(CC4)C3)CCCCC1OCC2 C1(C(=O)NC(CC)CNC(=O)CCCn2cc(C)cn2)CC12CCC(=O)CC2 C1(C)(COC)CC(NC(c2cn[nH]c2)=O)CN1C(C1CC(F)(CF)C1)=O N1(C(CCOCCOCCCC#C)=O)CCN(C)C(NC(=O)C(O)CC(N)=O)C1 C1(CNC(C(CC#C)C)=O)CCN(C(=O)CSCc2c(C)noc2C)CC1(F)F C12(NC(c3csc(-c4ccccc4)c3)=O)CC1CN(C(C1(CO)COC1)=O)C2 C1(NC(N2CCCC(CNC(C3CSC3)=O)C2)=O)(CO)COc2ccccc2C1 c1(C(=O)NC(C(=O)N2CC(NC(=O)NC)C2)C(C)O)ccc(C)c(C)n1 C(CCCC(=O)NCC=Cc1cccnc1)N(C)C(c1ccnnc1O)=O c1(C(=O)OC)ccccc1CC(=O)NCCCN(C(=O)CCC(F)F)CCO C1(C(N2C(C)(C(=O)OC)CC2)=O)C2CCCC2CN1C(=O)CC1C=CCCC1 C1(C(N2C(C(=O)NCC)CCC2)=O)(NC(=O)C2=C(Cl)CC2)CCCCC1 Cn1c(NCC2(C)CCCN(C(=O)CC3CCC(=O)N3)C2)cc(O)nc1=O c1(C(=O)NCC(CN(C(=O)C(C)(C)n2cncn2)C)O)n[nH]cc1C1CCC1 N1(C(C2C(CC(C)C)C2)=O)CCC(C)(C(=O)NCC2(C)CSC2)CC1 C(=O)(C1=CCOCC1)NCCC1CCC(NC(C=C2CCN(C)CC2)=O)C1 C1(C(N2C(C)(C(=O)NCC3C(C)OCC3)C=CC2)=O)CCCC1C1CC1 C1(C(N(C2CN(C(=O)CCCc3ccncc3)C2)C)=O)CCS(=O)(=O)N1 C(N=c1[nH]c(NCC(c2ccccc2)C)nc2c1CCCC2)c1ncc(C)cn1 N1(c2ncc(C(=O)OC)cc2Cl)CC2CC1CCC2NC(=O)C1=CCSC1 N1(C(c2c(OC)ccc(C)n2)=O)CC2CCCN(C(C3CC3C)=O)C2C1 CC1CCC(CC(N2CCCC2Cc2cn(Cc3cccc(O)c3)nn2)=O)CC1 C(C(C(=O)NCC1C2CCC(F)(F)C12)C(C)(C)C)NC(C(C)(C)OCC)=O CN=c1[nH]cc(C(=O)N(C(C)CNC(C2CC2(c2ccccc2)C)=O)CC)o1 C1(NC(=O)NCC2N(CC(=O)N(CC)CC)CCC2)CN(C)CCO1 C1(C(=O)Nc2cnc(Cl)c(Cl)c2)CCc2nc(-c3cccc(O)n3)sc2C1 C12(C(=O)NCC(CC(C)C)(C)NC(c3ccc(Cl)o3)=O)CCCC1CC(=O)C2 N1(C(C(CCC#C)NC(=O)C(C)CC=CC)=O)Cc2cccc(F)c2C1 C(C)(C)(CC(C)(C)C)NC(CC1CCC(NC(C2C(C(C)C)OCC2)=O)CC1)=O c1(C(=O)NCCC2CN(C(C3(CC)CC3)=O)CC2C)cc(=O)c2ccncc2o1 c1(C(C)=O)cccc(C)c1NC(c1cc(C)nc(C2CCC2)n1)=O C1(C(N2CCCC(C)(O)C2)=O)CN(Cc2cc3sccc3s2)CCC1(F)F C(CC1=CCN(C(C2CC2C)=O)CC1)NC(C1N(C(C)=O)CC(O)C1)=O C(C(O)C(=O)N(C(C)CN(C(=O)C(COC(C)=O)N)C)C)SC.N1(C(C)C)CCCC1 C(CC(CC)C(=O)NC1CC1CNC(=O)C(=O)N(c1ccccc1)CC)=CC C1(C(=O)Nc2nc(O)cc(C(=O)OC)n2)CCCC2CCCCC12 C(=O)(CCCC(=O)NC1CS(=O)(=O)CC1NC(=O)C(F)(F)c1ccccn1)OC C1(NC(c2ccc(C)c(C)c2)C)CCc2nnnn2CC1 CC1CCN(C(=O)Cc2cccc(Cl)c2)C1CNC(=O)Cc1cc(Cl)no1 O=C(C#CC1CCC1)NCC12CC1CN(C(=O)CCC1CCC(C(F)(F)F)O1)C2 N1(C(c2c(C)nco2)=O)CC2(CCNC(=O)C(c3cnn(C)c3)C)CCC1C2 C(N=c1[nH]c(=NC)[nH]c(=NCC(CSC)SC)[nH]1)c1ccc(OC)c(Cl)c1 C(=O)(C(N=[N+]=[N-])C(C)C)NC12C(CN(C(C(COC)OC)=O)C1)C2 C1(OCC)CC2(C1)CC2C(=O)NCC1CC(O)CN1C(=O)C(C1CCCCC1)C C1(NC(C=CCC)=O)(COC)CCN(C(=O)CS(=O)(=O)N(C)CCOC)C1 N1(C(CC(C)(C)C2CC2)=O)CCC2(CCCCN(C(C3(CO)CCCO3)=O)C2)C1 N1(C(C2C(C)CC(=O)N2)=O)CCC2CCC(NC(=O)C(N)=O)C1C2 C1(CNC(C=COCC)=O)CCCC(CNC(c2cnn(C3CCC3)c2)=O)C1 CC1(NC(C2CC3CC3C2)=O)CC(NC(c2ccsc2-n2cnnn2)=O)C1 Cc1nc2c(C)cc(C(N3CCOC(CN(C(=O)C(C)CO)C)C3)=O)cn2n1 N1(C(C2C(C(=O)OCC)CC2)=O)CCC(C2CC2)C1C(=O)NC.N12CCC(C1)C2 CC(C)S(=O)(=O)CC(=O)N(C)CC1(CNC(C2CCC(=O)O2)=O)CC1 CCCC(CCC)C(=O)NC1(C)CC(NC(=O)CC2CCS(=O)(=O)C2)C1 C(=O)(CC(C)C(F)F)NCCC(C)NC(=O)C(F)(F)CC1CC1 Cc1ccc(CC(=O)NCC2(CCCNC(=O)COC3CCC3)CC2)c(C)c1 c1(C(N(CCNC(C(CC=C)Cc2ccccc2)=O)CC)=O)ccc(N)c(Cl)c1O N1(C(C=Cc2ncn(C)c2)=O)CCN(C(c2n[nH]cc2Br)=O)C2CC12 C(=O)(C1=CCC(C)CC1)NCc1ccc(CNC(CC(C)C)=O)cc1F c1(C(N2CC3CC(C)N(C(C=CCC)=O)C3C2)=O)ccc(OC)c2ccncc12 C(=O)(C1=C(C)CCC1)N(C(C(=O)NCC1(CCOC)CCC1)C)C1CC1 CCC(=O)NNC(=O)C(C)NC(c1cnn(C)c1C1CNC1)=O C1(CC(=O)NC2CC(CNC(c3csnc3Cl)=O)C2)CCCOC1 c1(C(=O)NC2CCC(N(C(CS(=O)(=O)NC)=O)C)C2)ccn2c1CCCC2 Cc1nnn(CC(=O)NCCC(C)N(C)C(C2(CO)COC2)=O)n1 c1(CC(N2CCC(NC(C3C(=C)C3)=O)(COC)CC2)=O)sc2ccccc2c1C C1(CC(=O)NCC(CNC(=O)CC(F)(F)F)CO)NC(=O)CNC1=O c1(CC(N2CC3CCN(C(=O)CCOCC4CC4)C3C2)=O)c(F)cccc1F N1(C(CCOCCOC)=O)CC(NC(C2(NC(N)=O)CC2)=O)C(C)C1 S(=O)(=O)(c1ccc2oc(=O)ccc2c1)N1C2CC(C(N3CC(F)C3)=O)C1CC2 C1(C(C)NC(C2(SC)CCC2)=O)CCN(C(c2ccc(-c3cc[nH]n3)s2)=O)CC1 C1(NC(c2nc(C)nn2C)=O)CCC2(CC1)CN(C(C1CC1F)=O)CCO2 n1(CC)cc(C(=O)NC2C=CCN(C(c3cc(OC)c(Cl)s3)=O)C2)c(C)n1 Cc1cc(C)c(CC(=O)NCC(C(C)(C)C)NC(C2CCCC23CC3)=O)s1 C1(C(N(C(CC)CO)C2CC2)=O)CC2CN(C(=O)C(C)N3CCCC3)CC2C1 n1(CCCCC)nc(-c2ccccc2C(F)F)nc1CCS(C)=O N1(C(C(n2ccc(C)n2)C)=O)CCCC(NC(C2Cc3nccn3C2)=O)CCC1 N1(CC)CCN(C(=O)C(C)(CNC(C2CC2(C)C(F)F)=O)CC)CC1=O c1(C(N2CCCC(N(C(=O)COC3CCC3)CC)C2)=O)cc2ccncc2s1 c1(OC)ncc(C(=O)NCC2CN(C(=O)CN3CC(C)(C)C3)C3CC23)cn1 N1(C(c2ccc(Oc3ccncn3)cc2)=O)CCC(N2CC(F)(F)C2)CC1 C=C(C)c1cn(CC(C2CN(C(=O)CCNC(=O)NC3CC3)C2)F)nn1 CCCS(=O)(=O)C1CCCC1NC(=O)Nc1nnnn1C1CCC2(CC1)CNC(=O)C2 N1(c2nc(N3CCC(c4cccc(C)c4)C3)nc(C)c2)CCC2(CCCOC2)C1 c1(C(=O)NCC(C)N(C(c2c(C)cc(SC)o2)=O)C)cc(C)cc(C)c1 C1(NC(COCCC=C)=O)(CNC(=O)CC2CCCOC2)CCC(F)(F)CC1 CCC(F)(F)CC(=O)NC1(CNC(=O)Cc2cc(F)cc(Cl)c2)CC2CCC1C2 C(CCF)(C(=O)NC(C)CCO)NC(c1c(COC)cc[nH]1)=O N1(C(C(CSC)OC)=O)CC2COCC2(C(=O)NCc2cccc(F)n2)C1 c1(CC)c(N2CC3C(NC(=O)Cc4cccc(OC)c4)C3C2)nc(C)nc1Cl c1(OC)cc(C(N2CCC(NC(=O)C3=CCOCC3)C(O)C2)=O)c(Cl)cn1 N1(C(N2CC(c3ccc(OC)cc3)C2)=O)CC2(Cc3nnnn3C)CCC1C2 CC(CCN(C)C(C1CN(C)C1)=O)NC(=O)COCC1CC1 CC1(C)CN(CC(=O)NCCCC2CCCNCC2)CCS1 C(C(C(=O)NC1C(C(C)=O)C1(C)C)C(C)C)NC(C=CC(CC)C)=O N1(C(C)C)CCC(C(=O)NC(C2CCCN(C(=O)C(=O)NCC3CC3)C2)C)CC1 n1(CC(=O)N(C2CCN(C(c3cn(C4CC4)cn3)=O)C2)CC)cnc(Br)n1 c1(-n2c(-c3cc(CC)c(C)o3)nc(C3CCCC3)n2)cc(Cl)cc(Br)c1F C(=O)(C1(C)CCn2c(C)nnc21)NCC(CNC(Cc1c(C)cccn1)=O)(C)O C(C(CC(=O)N(CC(C)(C)C)CC1CC1)C1CCC1)NC(COCCSC)=O c1(C(N2C3(CNC(CCCOCCOC)=O)CC(C2)C3)=O)nccn2ccnc12 c1(C(=O)NCC(CN(C(=O)CC2COCCO2)CC)O)csc(CC(F)(F)F)n1 c1(OC)n[nH]c(=NC(C)(C)CCCO)c2ccc(C)cc12 c1(C(=O)OCC)cc(C(=O)NCC(C2CC2)N(C)C(C2CSCCS2)=O)nn1C N1(C(c2c(CNC(C3CCN(CC)C3)=O)ccs2)=O)C2CCCC1CN(C)C2 N1(C(c2c(OC)ccc(C)c2)=O)CC(C2CCCN(C(C3CCC(=O)N3)=O)C2)C1 C1(OC)CN(C(c2ccnc(CN(C)C)c2)=O)CC1NC(=O)Cc1cccs1 N1(CCC)CCC(C(=O)NC2(CNC(=O)C(=C3CCCCC3)F)CCOC2)CC1 CC1(CNC(=O)COCC(F)F)COCCN(C(C2(C)CC(C(F)(F)F)C2)=O)C1 N1(C(C2(CC)CCN(C(C(C)NC(CC)=O)=O)C2)=O)CCN(C)CC1CC c1(OC)ncc(F)cc1C(=O)NCC1CC1NC(=O)CCCc1ccc(C)cc1 N1(C(C(C2CCC2)OCC)=O)CCC(C)(CNC(c2c[nH]nc2C(F)(F)F)=O)C1 N1(C(c2c[nH]nc2Br)=O)CC23CCCC2(C1)CN(C(C1CCCC(F)C1)=O)C3 N1(CCC)CCCC(C(N2CCC(O)(CNC(c3ccoc3C(C)C)=O)C2)=O)C1 N1(C(C(C)(C)OCC)=O)CC(C(N2CCC(C)(F)C2)=O)CCC1(C)C C1(CCC)(NC(=O)CNC(=O)NC)CCCN(C(c2cc(OC)ccc2Cl)=O)C1 C12(C(=O)NCC(C)CNC(=O)CC3CC(C)(C)CO3)CCC(C)(CC1)OC2(C)C Cc1[nH]nc(C(=O)NCC(C2CCC2)NC(C2CCCC2C(C)C)=O)c1C CCC(C)CCC(=O)N1CC(NC(C2(C)CC2(C)C)=O)C(O)C1 C(CCC(C)C)(C(=O)NCC1CCOC1(C)C)NC(CC1(C(=C)F)CCC1)=O N1(C(CCC=CC)=O)CCC2(CC1)OCCC2NC(=O)C(C)NC(C1CCC1)=O CC1(C)CC(NC(c2c[nH]c(=S)cn2)=O)CN(C(=O)CNC=O)C1 C1(OCC)CCCN(C(=O)C(CCF)NC(=O)CC2CCSCC2)C1 Cc1ncc(C(=O)NC2CN(C(c3cn(C)nn3)=O)CC2C)n1-c1ccccc1 C1(C(N(CC(C)(C)NC(C=C(C)C(C)C)=O)C)=O)CCCCN1NC(N)=O C1(C(=O)NCC2CCC(NC(c3ncn(C(C)(C)C)n3)=O)C2)CC(S(N)(=O)=O)C1 N1(C(C(C=C=C)C)=O)CC2(CC2)CC1CC(=O)NCC(c1cccs1)C Cn1c(C(N2CCOCC2C(=O)Nc2c(C#N)cnn2C)=O)cccc1=O N1(C(C(C)OCCC=C)=O)CCC(C2CC2)(CNC(=O)COc2ccn(C)n2)C1 c1(C(=O)OC)sc(C(=O)NC(C)CCNC(c2nocc2C)=O)cc1C C(=O)(CCCC(=O)C(C)(C)C)NCC1CCN(C(C(C)CCC(C)(C)C)=O)CC1 C(C(C)(O)CC(=O)N1CCC(Cn2cc(-c3ccc(Cl)cc3)nn2)C1)SC C1(C)(CNC(CC=CC=C)=O)CCCC1NC(=O)Cc1cccnc1F C=CCCCCC(C(=O)NC(C)(C)C)N1CCCC1C1COCCC1(C)O CC1=CCC(C(=O)NCC2(C)CCCN2C(=O)C=Cc2cc(C)no2)CC1 c1(CC)nc(N2CCC(C(C)NC(=O)CC3(C)CCCC3)C2)c(C#N)cc1C N1(C(C=CC=CC)=O)CCC2(CC(C(N3CCCC(F)CC3)=O)C2)C1 c1(C(N(C(C(N2CCCC2C2CCCC2)=O)C2CC2)C)=O)nnc(O)nc1O C1(C(N(C(CNC(=O)C(C2CCCCC2)O)C2CC2)C)=O)CC(O)(C(F)(F)F)C1 C#Cc1ccnc(C(N2CCC(C(=O)NC3CC=C(C)CC3)C(O)C2)=O)c1 N1(C(c2nc(CC)oc2)=O)CC=C(CCNC(c2cc(Cl)ncc2OC)=O)CC1 N1(CCC)CCC(NC(=O)CC2(NC(C34CSCC3C4)=O)CC2)C1 C(C)(C)(CC(=O)N1CCC1(C)CCO)N(C(CCCC1C(C)C1)=O)C C1(NC(CN2CCC(C)CC2)=O)(CNC(=O)C(C)(C)N(C)C)CCCCC1C C#CCC(C)(CC)C(=O)NCCC1CCCN1C(=O)CCc1cc[nH]n1 C=CC(CC)CC(=O)NCC=C1CCN(C(=O)CC2CC(C)(C)CO2)CC1 CN(C)S(=N)(=O)c1ccc(-c2cccc(C=Cc3ccc(Cl)cc3)c2)cc1 c1(C(N2C(C)CC(NC(=O)C(C)(C)N(C)C)C2)=O)cc(O)c2sccc2c1 Cc1ccc(Cl)c(C(N2CC3(CNC(=O)CC4C=CCCC4)CCC2C3)=O)c1O C1(C(N2CCC(N(C(=O)CN(C)C(C)=O)CC#C)CC2)=O)OCCN(C)C1=O C1(C(=O)NC2(CO)CCCN(C(c3c[nH]c(=NC)o3)=O)C2)CCC([N+](=O)[O-])CC1 C1(C)(CC)CCCN(C(=O)CCC2CCCCN2C(C2C=CCCC2)=O)C1 N1(C(C(C2CCC2)NC(C2(c3cc[nH]n3)CC2)=O)=O)CCN(CCO)C(=O)C1 CC(C(=O)NCC1(CC(=O)NCCOC(=N)O)CC1)n1cncn1 CC(CC(=O)N1C(C(=O)NCCN(C)C)CCC1C1CC1)C(C)(C)C C1(C(N2CCC(CCC(=O)N(CC(O)C3CCC3)C)C2)=O)CCCCC(=O)C1 N1(C(C(CC)(F)F)=O)CCN(C(=O)CN2C(=O)CCC2=O)CC12CC2 c1(C(=O)NC2C(NC(c3ccc(Br)o3)=O)CCC2)nnc(O)nc1O c1(C(N2CC(CC(C)NC(c3cn(CC(F)F)cn3)=O)C2)=O)ccn(C)c1 c1(C(C(=O)N(CCCNC(=O)C(C)Cc2ccncc2)CC)C)ccc(C)cc1 C1(CNC(c2ccnc(C)n2)=O)CC2CCC(C1)N2C(=O)CC1CCS(=O)(=O)C1 Cc1ncc(CC(=O)NCCC2CN(C(c3ccns3)=O)CCO2)c(O)n1 C(C(O)CC(=O)N1CC(O)(CO)C1)NC(=O)Cc1ccsc1 C#Cc1cccc(C(=O)NC(C2(C(=O)NCCC3CCCC4CC34)CC2)C)c1C CC1(C)C(=O)CC1C(=O)NC(C)(C)C=CC(=O)NCC1(C)CCCS1 C1(NC(c2nnc(NC3CCC(F)(F)CC3)s2)C)C(=O)Nc2ccccc2S1(=O)=O CC(Cc1ccc(Cl)cc1)CC(=O)NCCCOCCNC(=O)C(F)CC1CC1 C1(NC(c2c(CC)non2)=O)CCOC(C(=O)N(CC)Cc2cn(C)nn2)C1 Cc1[nH]c(C)c(C(N2CC(CNC(C3CCCOC3c3cn[nH]c3)=O)C2)=O)c1C CN=S(C)(=O)c1cccc(C(=O)NCCN(C(=O)CC2OCCCC2(C)C)C)c1 c1(OC)ccc(CC(=O)NC2CCC2NC(c2cn(C)nc2C(C)C)=O)c(Cl)c1 N1(C(C2ON=C(C)C2)=O)CCCC(NC(C2(S(N)(=O)=O)CC2)=O)C1C C#Cc1cccc(C(=O)NCC2CC(C(=O)N(C3(CO)CC3)C)CO2)c1C CCCC(C)(CCC)C(=O)NC1CC2CCC1CC2NC(=O)C(F)(F)C(C)(C)O C1(C(=O)NC(C2CCOCC2)C)CC=CCN1C(c1cccnc1)=O C1(C(C)NC(c2c(C)snc2)=O)CCCN(C(=O)CC2CCN(C)CC2)C1 c1(C(=O)NC(C2CCCCO2)C(=O)OCC)cc(C)cc(C)c1O C1(CNC(C2(C(C)C)COC2)=O)CN(C(c2nc(=O)cc(N)[nH]2)=O)CCC1(F)F C1(C(=O)NC(C(=O)OC)C2CCC2)CCC2(CC2)N1C(=O)C(C)N1CC(C)C1 N#Cc1ncc(C(N2CCOC(CCCNC(=O)CCNC(=O)CO)C2)=O)s1 c1(CCC)cc(C(=O)NC(CN(C(c2nnn(C)c2C)=O)CC)CC)c(C)o1 C(=O)(C(O)C1=CCCCC1)NCCCC(C(=O)NCc1n(C)nnn1)(C)C c1(NC(CNC(C2COCCO2)=O)C2CC2)ccn2ccnc2n1 c1(CNC(=O)C(=O)NC2CNCC(c3ccccc3)C2)cc2ccc(Cl)cc2o1 C1(C(N(CCCNC(=O)C(c2ccccc2)C2CC2)CC)=O)COCC(C)(C)O1 C(C(C)(C)CC(=O)NCC(C1CC1)N(C)C(c1c[nH]nc1C(F)F)=O)OC c1(NC(C(CO)NC(=O)CCOC)C)ccc(C(N(CC)CC)=O)cc1 c1(CC)nc(C)c(C(N2CC(C(=O)Nn3cnnc3O)(CC)C2)=O)s1 CCC(O)C(C)(C)C(=O)NCC(C)CNC(C1CSC1)=O Cc1nc(NC(C(C)NC(C2CC3CCCCN3C2)=O)C(C)C)cc2nncn12 C1(C2CCCCC2)(C(=O)NC2CCC(NC(CCSCCC)=O)C2)CCCCC1 C1(OC)CN(C(=O)Cn2ncn(C)c2=O)CC1NC(c1ccc(Cl)o1)=O C1(n2cccn2)(NC(CCOCC)=O)CCN(C(=O)C(CCSC)OC)CC1 c1(CC)onc(C)c1C(N1CCCC1c1cccc(I)c1)C(=O)NC1CCCC1 C(C)(CCCCCO)NC(C1C(CNC(C(CC2CCC2)OC)=O)CC1)=O c1(SCC(=O)NCCC(CNC(=O)CC2CCOC2C)OC)ccc(C)cc1C N1(C(C(C)N2CCCC2)=O)CCC(C(O)CNC(=O)CCCNC(N)=O)CC1 C12(CC)CN(C(=O)NCc3ccc(C)c(O)c3)CC(CO)(C1)C2 c1(C(=O)NC(CCNC(CC(C)C)=O)C)cncc(-n2cccn2)n1 C(C)(C)(C(=O)N1CC(c2ocnc2NC(C2CC2C)=O)C1)CNC(=O)OC N1(C(c2c(C)cco2)=O)CCN(C(=O)C2CC2)C(c2cn[nH]c2)C1 C1(C(=O)NCc2n(CCC)ccn2)CCC2CCC1N2C(=O)CN1CSCC1=O c1(C(=O)NCC(CNC(C(C)OCC#C)=O)(C)C)cnc(S)n1C C1(C)(CNC(CSCCC)=O)CCCN(C(=O)C(C)NC(=O)C(C)(C)C)C1 C(C)(CN=c1[nH]cnc(Cl)c1Br)N(C(C(CCCC)ON=C(C)C)=O)C N1(C(C2C(CC)OCCC2)=O)CCN(C(=O)COc2cn[nH]c2)CC12CCC2 N1(C(C2(OC)CCC2)=O)CCC(CCNC(=O)C(F)=C(C)C2CC2)C1 C1(C(=O)NCc2n(C(C)C)ccn2)CCCC(NC(=O)C(C)c2ccco2)C1 c1(OC)cccc(C(=O)NC2CC(NC(=O)C(C)NC=O)C2)c1OC(C)C c1(C(N2CCC3(NC(c4coc5c4COC5)=O)C(C2)C3)=O)cnc2ccccn12 S(=O)(=O)(C1CCN(C(=O)C(=O)Nc2cc(C)c(Cl)cc2C(=O)OC)C1)NC C(C(CC(=O)N(CC(C)(C)O)C)NC(c1csc(F)c1)=O)OC c1(N2CCC(C)(OC)C2)nc(N2CCC(CN(C)CC)C2)c2ccc(C)cc2n1 Cc1sc(O)nc1C(=O)NC(C(=O)NCCc1nc[nH]n1)c1ccoc1 N1(C(C23CC(CN(C(C(CC4CC4)OC)=O)C2)C3)=O)CCC2(CCCCO2)C1 C(=O)(C1SCCc2ccccc21)N(CC(C)N(C(c1nccc(OC)c1)=O)C)C c1(OC)cc(F)ccc1N1CCN(C(=O)N(C(C)C)Cc2cccnc2)CC1 c1(OC)ncnc(C(=O)NCC(F)CNC(c2cn(CCO)nc2C)=O)c1F c1(C(=O)NCC(CC)NC(c2conc2C2CC2)=O)cnc2c(cnn2CC)c1 N1(C(COc2cccc(C)c2)=O)CCC(NC(C2(C)CCCS2)=O)CC(O)C1 C12(C(N3CC(C)(NC(C4(C)CCCN4C)=O)C3)=O)CCC(CF)(C1)OC2 C1(C)(CNC(C2CN(C(C)C)C2)=O)CCN(C(c2c[nH]nc2-n2cnnn2)=O)C1 Cc1ccc(C(=O)NCC2C(C(N3CCCCC3CF)=O)C2(C)C)c(F)c1 Cn1cc(S(=O)(=O)NCC2(F)CCCN(C(=O)Nc3ccc(Cl)cc3Cl)C2)cn1 C1(C(=O)NCC2(C)CN(C(c3ccc(F)s3)=O)CCO2)CN2CCCN1CC2 C(CCC)(CCCNC(=O)CSCC(N)=O)N(C(c1nc(CCC)sc1)=O)CC C12(CNC(c3c(C)nc[nH]3)=O)CN(C(C3(C)CCCCC3)=O)CC1CCO2 C(=O)(C(O)CC(F)(F)F)NCCc1c(C(=O)NCC2CCCOCC2)c[nH]n1 c1(OC)ccc(SCC(N2CC(CNC(=O)C=Cc3ncc[nH]3)C(C)C2)=O)cc1 c1(C(N2C(CNC(C3(CC4CC4)CC3)=O)CC(OC)C2)=O)ccc2c(c1)CCN2 Cc1ncc(NC(C2(C)CCN2Cc2ccnc(F)c2Cl)=O)cc1Br Cc1ccc(=N)[nH]c1C(N1CCC(C)(CNC(C2(C)CC=CCC2)=O)C1)=O c1(C(N2CCCCC2)CN(C(=O)NCC(C)(C)F)CCO)ccc(F)cc1F C=C(C)C(CC(=O)NC1CCC(N(C)C(C2CCC(F)(F)CC2)=O)CC1)OCC N1(C(CCCC(=C)C)=O)CCC2CN(C(=O)CSCc3ccncc3)CCC2C1 CC(C)(C)C(CNC(c1cn[nH]c1)=O)C(=O)NCCC1CCCC12CC2 C1(C(N2CC(N(C(C3CC(OCC)C3)=O)C)C2)=O)COCCO1 C1(c2cn(C)nc2)CN(C(c2ccc(Cl)cn2)=O)CCN1C(=O)C=CS(C)=O C1(C(N2CCC(CCNC(=O)Cn3cccnc3=O)CC2)=O)(OC)CCCOC1 Cn1c(CN2CCC(CO)C(O)C2)nc2cc(Br)ccc12 N1(Cc2c(C)cccc2)CCC2(CN(C(c3cc(Cl)ccc3F)=O)CC(C)O2)C1 n1(C(C)C)ncc(CNC(=O)OC(C)(C)C)c1F.C12CN(CC1C(C)(C)C)C2=O c1(C(N2CCC(C)(CNC(C3CC(=O)C3)=O)C2)=O)c(Cl)oc2ccccc12 CC1(NC(=O)CCc2nnc(C(F)F)o2)CCCN(C(C2CC2F)=O)C1 C1(OCC)CC(NC(=NCCCOC)NCC(F)=C(C)C)C12CCCCC2 N1(C(C2CCC(C)N2C(=O)CCC2CCCO2)=O)CC2CCCC2C1 N1(C(CNC(CC)=O)=O)CCn2ncc(CNC(c3csc(C)c3)=O)c2C1 N1(C(C(C)CC(F)F)=O)CC2=C(C1)CN(C(c1cccc(OCC(N)=O)c1)=O)C2 NS(=O)(=O)c1n[nH]cc1CN1CCC(CNC(C2(F)CCCCC2(F)F)=O)CC1 C=CC(CCC)CC(=O)NCC1(CNC(C2Cc3ccccc3O2)=O)CC1 c1(CC)conc1C(c1nnnn1C1CCCCC1)NCCSC(F)(F)F N1(C(C2C(CC)CCC2)=O)CCN(C(C23CC=CCN2CCC3)=O)CCC1C C1(O)(CNC(C2(C)CC2(F)F)=O)CCCN(C(c2cncn2C2CC2)=O)CC1 N1(C(C2N(C)CC2)=O)CCCC1C(N1CCC(c2ncc[nH]2)C1)=O C(=O)(C(=O)N=S(C)(C)=O)NCC(C)CN(C(=O)C(c1ccc(F)c(F)c1)(C)C)C C(C)(CC(=O)N1CCC1C)(C(F)F)N(C)C.c1(C(=O)OCC=O)cnc(S)n1C C1(OC)CC2(C1)CC(C(N1CCOCC(CNC(c3ccc(F)o3)=O)C1)=O)C2 C1(C2CCCCC2)(CNC(Cn2cc(-c3nccc(OC)n3)nn2)=O)CC1 c1(C(N2CC(OCC(=O)NCCC3C(C)C3)C2)=O)cc(C#N)cn1C c1(CCC(=O)N(CC(C)NC(C2CCC(C)(F)CC2)=O)C)ccc(F)cc1F c1(OC)ccc2[nH]cc(C(=O)NC3CN(C(c4coc(SC)c4)=O)C4CC34)c2c1 c1(OC)ccc(Br)cc1CCC(=O)NC1(CN(C(=O)C2=CC(C)(C)C2)C)CC1 c1(NC(C2CC2C(N2CCOC(O)C2)=O)=O)ccc(Br)nc1[N+](=O)[O-] N1(C(C(C(C)C)NC(COC)=O)=O)CCCCC2(C1)CN(C(c1cocc1C)=O)C2 S(=O)(=O)(c1nccs1)NCC1CCC(C(=O)NCc2ccc(Br)s2)CC1 N1(C(C(C)=C(C)C)=O)C(C(=O)NC2(CO)CCC2)CCC1C(C)C c1(C(=O)OC)ccc(NCC2CCC(OC)CC2)c(C#N)c1 CN1CCc2[nH]nc(C(N3CC(CNC(c4ccc[nH]4)=O)C4CC34)=O)c2C1 c1(C(=O)NC2CC3C(NC(c4ccccc4)=O)C3C2)ccc(F)c(F)c1 C(=O)(C(=O)C(C)(C)CC)N1CCC(N(CCCC)C(C2CC(N=[N+]=[N-])C2)=O)CC1 N1(CC(=O)NC(CNC(CC(CC)C)=O)C(C)C)C(C)=CC(C)=NS1(=O)=O N1(C(CC)=O)CC(C2CCCN(C(=O)C=CCN(C)C)C2)C1 N(C(=NCCCF)NCCC=CBr)C(c1cccc(Cl)c1)C c1(C(C)NC(=O)NCC2(c3ccccc3Cl)CC2)ccc2c(c1)CC(C)O2 C1(C(N(CC(=O)OCC)C)=O)CCN(C(=O)CCOCC(F)F)C(C)(C)C1 c1(CNC(C2(O)CCN(C(c3ccc(OC)nc3)=O)C2)=O)ccc(F)cc1Cl Cc1nccc(N2CC3CC2C3C(N2CCC2c2ccccc2)=O)n1 CC1(NC(C2CCCCO2)=O)CCCN(C(C23CC(CF)(CO2)C3)=O)C1 C1(NC(=O)CCOC2CC2)C2COCC1CN(C(C1CC3CC(=O)C1C3)=O)C2 N1(C(Cc2nc(C)oc2)=O)CC2(CCN(C(C3CCCCC3C(F)(F)F)=O)C2)C1 c1(OC)ccc2ccc(NC3CC4C5C=CC(O5)C34)cc2n1 C1(NC(c2cc(CC)c(C)o2)=O)CC2(CCC(C)(C)CC2)C1 C(=O)(C1CNC(=O)c2ccccc21)NCC1CCC(NC(C2C(=C)CC2)=O)CC1 CCC(CNC(=O)C(C(C)C)NC(=O)Cn1ccnn1)C(C)(F)F c1(OC)ccc(Cl)c(C)c1C(=O)NC1CC(C)(NC(C2CC(OC)C2)=O)C1 c1(C(=O)NCC2C(C)CN(C(c3cscn3)=O)CC2)ccc(C#CC2CC2)cc1 C1(NC(CC(=O)Nc2nccs2)=O)CCOC12CCN(C(=O)C(O)C1CC1)CC2 c1(C(=O)NC2CCC(C)(NC(C(CC)O)=O)CC2)cn2cccc(F)c2n1 C1(NC(C(CC)(F)F)=O)CCN(C(=O)C(C)C(=O)OC(C)(C)C)C12CC2 C1(SCCC(N2CCC(O)(C(N)=O)CC2)=O)CC1C1CCCCC1 N1(C(C(C)C(F)F)=O)CCCCC2(C1)CN(C(=O)Cc1sc(O)nc1O)C2 C1(NC(CC(=O)NCC#C)=O)CCCN(C(c2nc(CCC(C)C)no2)=O)C1C c1(NC(N2C(CN(C)C3CC3)C(C)(C)C2)=O)ccnc2c1ncn2C C1(C(=O)NCCc2c(C)[nH]nc2O)CCCCCN1C(C1CCCCC1)=O C1(NC(C2C=CCC2)=O)CCC2(CC1)CCN(C(=O)COCC(F)(F)F)C2 C(=O)(C1=CCC(C(F)(F)F)OC1)NCCN(C(c1n(CC#C)ccc1)=O)C1CC1 C(CCC(=O)N(CC(=O)N(c1cnn(CCOC)c1)C)CC)OCC c1(C(=O)NC2CCCC(CNC(CN(C)C)=O)C2)cncc2c1CCC2 Cc1c(C(=O)NC2CCN(C(c3cnn(C)c3Cl)=O)C(C3CC3)C2)cncc1Cl C1(CNC(=O)C(Cl)=CCl)CC2(CO1)CN(C(=O)CCCCc1ccc(Cl)cc1)C2 c1(CCC(=O)NC2CN(C(=O)CCn3cc(Cl)cn3)C2)ncccn1 c1(CC2(CO)CN(C(=O)C#CC3CC3)C2)cccc(Cl)c1.CC1C(=O)NCCO1 Cc1cc(C(C(=O)O)NC(=O)Cc2ccc(C3CCC3)cc2)cc(C)c1 C(CCCCCNC(C1C2CCCCC12)=O)N(C(C1OCC(C)C1)=O)C C1(C(=O)NC2(CNC(C3CC(C)(O)C3)=O)CC(OC)C2)CC2CCC1C2 C1(C(=O)Nc2ccc(F)cc2)CCC2CCC1N2C(=O)C(O)Cn1cncn1 CC(C)C(C(C)NC(C1CC(N(C)C)C1)=O)NC(c1cncc(O)c1)=O c1(C(=O)NCCN(C(=O)C(C)(F)C(=O)OC)CCC)c(F)ccc(C)c1Cl C#CC1CN(C(C2CCCN2C=O)=O)CCN1C(=O)C=CCOCCOC c1(C(N2CCN(C(C=C3CCC(C)(C)CC3)=O)CC2)=O)noc2c1CCCCC2 c1(C(=O)NCC2(O)CCN(C(C(CC)(F)F)=O)C2)cnc(CC2CCC2)nc1O C(=O)(C(CO)C(C)(C)C)NCC1C(NC(CC(=C=C)C)=O)CCC1 C1(CCCC)CCCC1N=c1[nH]c(=NCc2c(Cl)cccc2Br)[nH]c2c1CCC2 c1(C(N(CC(CC)NC(=O)C(C)CC(N)=O)C)=O)cc2ccccc2o1 N1(C(CC2(C=C)CCC2)=O)CCC(C2CN(C(c3ccccc3C(C)C)=O)C2)C1 C(CC(CNC(=O)COC)NC(c1cn(CC(N)=O)nn1)=O)OC c1(C(N2CC(F)(CNC(c3ccc(F)s3)=O)C2)=O)coc2c(F)cc(Cl)cc12 c1(OCC)cccc(C(N2CCN(Cc3csc(C)n3)CC2)C(=O)NC2CC2)c1 C12(NC(C(CC)OC3CCCCC3)=O)CC(CNC(C3CC3(F)F)=O)(C1)OC2C Cc1nc(S(=O)(=O)N2CCCC(NC(=O)Nc3cc(F)cc(F)c3)C2)cn1C S(=O)(=O)(c1cn[nH]c1)N1CC2(C(C(=O)NCCC(F)(F)F)C2)C1 c1(CCNC(C2(CCO)CC2)=O)ccccn1.C1CCCNC(=O)N1 c1(CCC(=O)NC(CC)CNC(=O)C=Cc2ncc[nH]2)ccc(Cl)nc1 N1CCN(NCc2ccccc2)C2CC12.Cc1csc(-c2ccc(C(=O)O)s2)c1 C12CCCN1NC(=O)C(=O)N2.CC1(C)CCCN(c2ccc(F)cc2OC(F)F)C1 N1(C(CC2(C(=O)OCC)CC2)=O)CC=C(C(C)(C)C(=O)OC)CC1 N1(C(C)C)CCCC1C(=O)NC(C)C(C)(C)NC(C1(OCc2ccccc2)CC1)=O c1(C(=O)NC(C)CCCNC(=O)C(O)CC(F)(F)F)ccc2ccccc2c1 c1(C(=O)NCCCCCN(C(=O)CC(C)(C)C(F)F)C)ccc2c(n1)CCO2 C(N=c1[nH]c2c(c(=NCC(C)CO)[nH]1)CCC2)c1c(C)nccc1 Cc1c(C(=O)NC2CC(N(C(=O)Cn3ccnn3)C)C2)cc(CC2CC2)n1C c1(C(=O)Nc2c(C)ccc(O)c2)ccc2c(c1)COC(=O)N2 CCC(CNC(=O)C(O)C(C)(C)C)(CC)C(=O)NC1CCC(C)(C)C1 N1(C(C(n2ccc(C)n2)C)=O)CCC(NC(=O)CSCc2cccnc2)C1C CC1CN(C)C(C)CN1C(c1ccc(NC(c2ccc(Br)cc2Cl)=O)cn1)=O c1(C(=O)NC(CNC(c2[nH]cc(C)c2)=O)C)ccc(C)c2c1NCCC2 C1(COCC#C)(NC(=O)Cc2n[nH]c(C)n2)CCCCC1.C12CCCN1C2=O N1(C(c2cn(CC)nn2)C(=O)NCCCC)CC(C2(O)CCC2)C12CCC2 CC1(C(N2CC(F)(C(=O)NCC(CO)C3CCC3)C2)=O)CCCS1 c1(OC)cnc(C(=O)NC2CN(C(=O)CCCn3cccc3)CCC2O)c(F)c1 N1(CC)CC(C(=O)NC2(CCNC(=O)CC3CCC(=O)N3)CCC2)CC1=O c1(N(C)CC2CC=C(C)CC2)ncc(C)cc1S(=O)(=O)N1CCC1 c1(C(=O)NC2CCN(C(CCCNC(=O)OC)=O)C23CC3)cnc2nccn2c1 c1(NCCc2c(C)ocn2)ncnc(NC(C2CC2c2ccccc2)=O)c1C C1(C(N2C(CC(C)C)CC2)=O)(NC(c2csnc2Cl)=O)CC1(C)C C1(NC(C(CNC(C)=O)(C)C)=O)CCCN(C(=O)CC2C=CCC2)CC1 n1(CC(=O)NC2CCN(C(C3(CC#C)CCOCC3)=O)C2)nnc2c1CCCC2 c1(C(=O)NC2CC(OC)CN(C(CCC(C)OC)=O)C2)ccc2c(c1)CCCO2 CCCCCCC(C)C(=O)N1CCC2CCC(C1)N2C(=O)C(C)(C)CCCF C1(C(C)NC(C=CC(CC)=CC)=O)CCCN1C(c1cc(C)[nH]n1)=O CC1CCSCCN1C(=O)CCN(C(=O)CCn1cnnn1)CC1CC1 N1(C(C2(CF)CCN(C(CCCCCC)=O)C2)=O)CCC2(COC(=O)N2)C1 C(=O)(C#CC(C)(C)C)N1CCC(c2c(CNC(C3(CCC)CC3)=O)c[nH]n2)C1 C1(NC(c2cc(C)c(C)s2)=O)CCN(C(=O)CC2OCCC2(C)C)C12CCCC2 CCC(C)CC(CO)NC(=O)CCC1(NC(=O)C(C)=C2CCCC2)CCCC1 Cc1cc(-c2ccccc2CN2CCNC(C)C2)ccc1-n1c(C)ccc1C c1(CC(N2CCC(OCCNC(CC(CC)SC)=O)C2)=O)ccc(F)cc1F c1(NC)ccc(C(=O)N(CCC(C)NC(=O)C(C)(C)COCC(F)F)C)cc1 N1(C(c2occ(C)c2)=O)CCC(F)(CNC(C2CCCCN2C(N)=O)=O)CC1 C(=O)(C(O)C(C)(C)C)N(CCNC(C(CC)C#N)=O)CC1CC1 c1(-c2n(CC3CCN(C)C3)ccn2)ccc(-c2cnn(C)c2CN)cc1F N1(C(C23CC(NC(CCC=C=C)=O)(C2)C3)=O)CCC(O)C(F)(F)C1 C12(CNC(c3cnc(COC)s3)=O)CN(C(=O)C(F)C(C)(C)O)CC1CCO2 C(=O)(CCC(CC)OC)N1CC(CCC)C(NC(C2(CCCCO)CC2)=O)C1 CC1(C)CCC=C(C(=O)NC23CC(CNC(=O)C#CC4(C)CCCO4)(C2)C3)C1 c1(C(=O)NC(CNC(CC2C(C)CCC2)=O)C)c(F)c(F)cc(F)c1F c1(NCC(C)S(N)(=O)=O)cc(S(=O)(=O)NCC2(N(C)C)CCC2)ccc1C#N C(c1cc(F)c(F)c(F)c1)=CC(=O)OCC(=O)Nc1ccc(NC(=O)C2CC2)cc1 c1(C(=O)OCC)ccc(C(=O)NCCCCC(C)NC(=O)CN(C)CC)nc1 C#CCCC(O)C(=O)NCCCN(C1CCCC1)C(C1CCCC(F)(F)C1)=O C#CC1(C(N2CCC(CN(C(=O)Cc3cn(C)nc3C)CC)CC2)=O)CCCC1 C(=O)(C(C)CC(C)C)N(C(C(NOCCOCC#C)=O)C)CC=C c1(C(=O)NCCCN(C(C2CC(=O)NC2)=O)C2CC2)cccc(-c2nccs2)c1 c1(N2CCC(C(C)NC(CCCOCCOC)=O)C2)ncc2c(ncn2C)n1 N1(C(C(C(C)(C)C)O)=O)C2CCC1CN(C(=O)CC1OCCCO1)CC2 C1(CNC(C(C2CCOC2)OCC)=O)CC2(CCC2)CN1C(C1COC(=O)C1)=O c1(C(N2CC3(CCN(C(C(CC)F)=O)C3)C2)=O)cc2c(cc1OC)CCC2 Cc1cnn(C(C)C(=O)NCCOCCNC(=O)CSc2cn[nH]c2)c1 N1(C(C2(C(C)C)CCC2)=O)CCC2CCN(C(=O)C=Cc3cnc[nH]3)CC2C1 C12(NC(CCC(=O)NCC)=O)CC(CNC(C3(C)CC3(Cl)Cl)=O)(C1)OC2C c1(C(N2CCC(CCNC(C(C)n3ccnc3)=O)CC2)=O)cc2n(n1)CCCN2 Cn1ncc2ncnc(N3CC(F)CC3C(=O)Nc3ccc(F)cc3[N+](=O)[O-])c12 CCCC(CCNC(=O)C(CC1CCCC1)NC(=O)C(C)N1CC(C)C1)CCC C1(CCCC(=O)NC(C)CC2CN(C(=O)C(C)N(C)C)C2)CCCC(=O)N1 C1(O)(C(=O)NC(C=CC(=O)N(C2(C#C)CC2)C)C)CCCC1 n1(CCC(=O)NC(CC)CNC(C2COC2)=O)sc2ccccc2c1=O C1(N(C(=O)CC2CC2C2CC2)CC)CCN(C(C2CC2COC)=O)CC1 c1(C(C)OC)nc(-c2cncc(-n3cnnn3)c2)n(-c2cccnc2)n1 N1(C(c2cc(C)n(C)c2)=O)CCCCCC1CNC(=O)Cc1cnnn1C c1(CC)cccc2sc(NC(=O)NCCc3ncc(-c4ccc(F)cc4)[nH]3)nc12 C1(NC(C(CSC)O)=O)CCN(C(c2cc(C)n(C(F)F)n2)=O)CC(O)C1 CC(C(F)(F)C(F)(F)F)=CC(=O)N(C(C)CNC(=O)COCCN(C)C)C C1(C(=O)NC2C(NC(CCOC)=O)C2)CCS(=O)(=O)N1C N1(C(C=CCC(C)(C)NC(C(C)OCC=C)=O)=O)CCN(C)CC1CCO N1(C(C(C2CCCCC2)OC)=O)CCN(C(C2CN(C)C2)=O)C(C(C)C)C1 N1(C(=O)COCC2CCCOC2)CCC2CCC(C1)N2C(=O)CCCOC1CC1 C1(CNC(c2cc(C(=O)OC)[nH]c2)=O)CC(C)N(C(c2cc(C(N)=O)no2)=O)C1 Cc1nc(N(C)C)sc1C(=O)NC1CCC1CNC(C1CC2(C1)CC2F)=O Cc1ccc(N)c(C(N2CCC(NC(=O)C(C)(C)CO)C2C(C)(C)C)=O)c1 c1(C(=O)NC2C(NC(CCC(N)=O)=O)CCOC2)cncc2cccnc12 N1(C(C2N(C)CC(O)CC2)=O)CC2CCC(C1)C(NC(c1ccc(F)s1)=O)C2 c1(NC(C2CCN(C(c3cnco3)=O)CC2)=O)ccc(C(F)(F)F)c(Cl)c1 c1(CC(=O)NCCCN(C(c2c(C)cnnc2O)=O)C)ccc2cnccc2c1 c1(C(=O)NCCCCNC(COc2ccc(C)cc2)=O)nn(C)c2c1CCC2 C=CC1(C(=O)NCC2CC(NC(=O)C(CC(C)C)OC)C2)CCCCC1 c1(CC)nc(C)[nH]c1C(N1CCC(C)(CNc2nccc(OCC#N)n2)C1)=O C=C(CCOC)C(=O)NOC1CC2CCC1C2 c1(OC)ncc(Cl)cc1C(=O)NCC1CCCN(C(=O)CC2(O)CCCCC2)C1 N1(C(C(c2nc(C)sc2)=O)=O)CCOCC(CNC(C2(C)CC3CC3C2)=O)C1 C1(C(=O)NCC(C)(CO)NC(=O)Cc2n[nH]c(C)n2)(CC)CNC(=O)C1 c1(OCC)cc(C(N2CCCN(C(=O)CN3CCS(=O)CC3)CC2)=O)oc(=O)c1 c1(C(N2CC(C)C(CNC(C3COC(=O)N3)=O)CC2)=O)n[nH]c2c1CCSC2 CCC(C(=O)OC)C(=O)NCCCN1CCN(C(C2CNC(=O)O2)=O)CC1 N1(C(C=CC=CC)=O)CCCC(NC(C2CCCC2(C)C)=O)C1C N1(C(C2CCN(CC)C2)=O)CCOC2CN(C(C3(C#N)CCCCCC3)=O)CC12 Cn1cnc2cncc(C(N3C4CCC3CC(NC(=O)CCC(F)(F)F)C4)=O)c12 C(=O)(CC(C)C(F)F)NCCN(CC(C)O)C(c1nc(C2CC2)ncc1Cl)=O S(=O)(=O)(c1ccc2nc(N3CCC(C#N)CC3)ccc2c1)NCc1c(C)scn1 C(CCC(C)(C)NC(c1cnc(OC)s1)=O)NC(CC=C)=O c12ccccc1S2.C(C(CNC(c1scnc1C(C)C)=O)CO)NC(CC=C)=O C1(C(=O)NCCCCn2cc(C3CC=CCC3)nn2)CC2CCC(C1)O2 C1(N(C(CCc2cc(OC)no2)=O)C)C2CN(C(c3ccc(O)cn3)=O)CC12 CCCCC(C(=O)NC)NC(C1COCCN1C(=O)C(c1ccn(C)c1)C)=O c1(C(N2C(CNC(c3ccc(C)cc3)=O)C3CC3C2)=O)cc2sccc2n1C c1(C(=O)NC(C(=O)NC2CC(=O)N(O)C2)C2(C)CC2)ccc([N+](=O)[O-])[nH]1 c1(C(=O)NCc2c(C(=O)NC(CCOC)C)c[nH]n2)ccc(C)nc1O c1(NC(C2(C)CCN2C(=O)CCCCCBr)=O)cccc2c1CC(=O)N2 C1(NC(c2cc(COC)oc2C)=O)CCN(C(C2CC(O)(C#N)C2)=O)C(C)C1 N1(Cc2cn(CC=C)nn2)CCCC(NC(C2CCC(=O)N2)=O)C1 CC1(C)CCC(CNC(c2cccnn2)=O)N(C(c2cnns2)=O)C1 c1(C(=O)NC(C2(O)CCN(C(C(C=C)C)=O)C2)C)ccc2cc[nH]c2n1 Cc1ccc(C(N2CCC(N(C(=O)C#CC(C)(C)C)CCO)C2)=O)c(=O)n1C C1(CNC(C2(C)CC2(Cl)Cl)=O)CC(NC(=O)C=CSc2nc[nH]n2)CC1O C1(CNC(C=CC(CC)=CC)=O)CN(C(c2cnc(C#N)s2)=O)C2CC12 C1(C)(C(=O)NCC(CCOC)NC(=O)Cc2ccc(C)cc2C)CC2CCC1O2 c1(COC)ncc2c(n1)CC1CCC2N1S(=O)(=O)C1CCN(CC(=O)O)C1 Cc1ccc(C(CNC(c2csc(O)n2)=O)NC(C2(F)CCCCC2)=O)cc1 Cc1nc(O)[nH]c1C(=O)NC1(C2CCCCN2C(=O)CC2C(C)(C)C2(C)C)CC1 Cc1ccc2c(C(=O)NCC3CCN(C(c4ccnc(C)c4N)=O)C3)c[nH]c2c1 C(=O)(C1=CCC2(COC2)OC1)N1CCC(C)(CNC(Cc2cccc(C)c2)=O)C1 CC1CCCCC1C(=O)N(C1CCN(C(=O)CC(=O)Nc2nccs2)CC1)CC N1(C(c2c(C)n[nH]c2)=O)CC(NC(c2cccc(C(F)(F)F)c2C)=O)C(C)(C)C1 c1(C(=O)NCC(CNC(C2CCSC2)=O)C(F)(F)F)cnnc2ccccc12 c1(C(Cn2cc(CC3CCN(C(C4(C=C)COC4)=O)C3)nn2)O)ccc(F)cc1 N1(C(c2cn(C)nc2)=O)CCN(Cc2conc2C(F)(F)F)CC1 c12cccc(c1)C2.CC1CCOC1C(=O)OCC(C)(C)C1CC1 c1(C(=O)NCCCNC(c2cnc(Cl)[nH]2)=O)cnnc(-c2ccccc2)c1 c1(C(=O)NC(c2ccccc2OC)C(=O)OCC)ccc(C(C)C)c([N+](=O)[O-])c1 C1(CC)(NC(=O)Cc2occc2C)CCN(C(C2(C(F)F)CCOCC2)=O)CC1 C=C(C)CCCNC(C1CCN(C(=O)CCC2CCC(OCC)C2)C1)=O N1(C(C2(OCC)CC2)=O)CCCC(C2CCN(c3c(C#N)cccc3[N+](=O)[O-])C2)C1 c12cccc(c1)NC(=O)NC2C.c1(C(C)OCC)cn(Cc2ccccc2)nn1 C1(NC(c2c(C)ccn2C)=O)CN(C(=O)C2=COCCO2)CC1N=[N+]=[N-] c1(-c2[nH]cc(C(N(CC(C)NC(c3ccoc3Cl)=O)C)=O)n2)cccc(Cl)c1 N1(c2n(CCOC)c(-c3cc4n(c3)CCCC4)nn2)CC2CC3CC(C2)CC1C3 c1(CC)onc(C(=O)NCCc2cn(CCCCC(=O)O)nn2)c1C N1(C(C(C)(C)C(F)(F)F)=O)CCCC(C2CC2NC(=O)C2=CCCCO2)C1 c1(C(=O)NCC2N(C(C=CC(CC)=CC)=O)CC2)nc2sc(C)cn2c1C Cc1cncc(C(=O)NC(c2cn(C)nn2)C(=O)NCC2CC2Cl)c1 c1(NC(c2scc(-c3cccc(C)n3)c2)=O)ccc2c(Br)nn(C)c2c1 Cc1ccc(N)c(C(=O)N(CCCCNC(c2cnn3ncccc23)=O)C)c1F N(C(=NCC1CC(C)(C)C1)NC1CCC1)CC1(CC)COC1 c1(C(=O)NC2CCC(CNc3nccc(C(=O)OC)n3)C2)ccc2ccnn2c1 C=CCC(CNC(=O)C=CCC(C)(C)NC(C1CC(C)=NO1)=O)CC(C)C C12(CNC(C(C)Oc3cccnc3)=O)CC(NC(C3CNC(=O)N3)=O)(C1)C2 c1(C(=O)NCC(CN(C(CC(CCC)O)=O)C)O)c(F)ccc(Br)c1C Cc1ccc(C(CNC(=O)C(C)O)NC(=O)C(C)(C)c2ccno2)cc1 CCC(C)C(CC(=O)NCc1ccnc(O)c1)NC(=O)CC1CC(=O)C1 c1(CC(=O)N(C(C(=O)N(C)CC)C)C2CC2)ccc(Br)c(OC)c1 c1(C(=O)NC2(CO)CCN(C(CC(CC)C)=O)C2)ncc(C#N)cc1Cl C1(C(=O)NC(CC)C)C=CCN(C(c2cc(Cl)cn2C)=O)C1 Cc1ccc2cc(C(=O)NC3CC4(CCN(C(=O)C(O)C(F)F)C4)C3)ccc2n1 N1(C(C(C)(O)C2CC2)=O)CCN(C(=O)Cc2cccc(F)c2F)CC1CF C(C(CC(C)C)C(=O)O)NC(=O)NCc1c(OC)cc(F)cc1 N1(C(c2nc(C)n(C)n2)=O)CCCCC12CN(C(C1CSCCS1)=O)C2 C(C)(C(C)(C)C(=O)NC1(C)CN(C(N)=O)C1)NC(Cn1nnc(C)n1)=O.CO C1(C(=O)NCCC2CN(C(c3cncc(C)n3)=O)C2)Cc2nccn2C1 C(CCCCCC(=O)NC(C)(C)CCF)NC(c1cc(C(C)C)[nH]n1)=O CC1(C(=O)NCCN(C(C2COCCN2C2CCCC2)=O)C2CC2)CS(=O)(=O)C1 c1(C(CN(C(C(CC)NC(C)=O)=O)CCO)NCc2nocc2Cl)ccccc1F C(=O)(C1=CC2(CN(C(C3CCCN(C)C3)=O)C2)OC1)N1CC(C(C)=O)OCC1 C1(O)(C(=O)NC2CCC(NC(C3(CO)CC3)=O)CC2)CCCCCC1 CN1CCC(C(=O)NCC(c2ccccc2)NC(c2cc(CCCO)on2)=O)C1 Cc1ncc(CC(=O)NCC2C(C)CCN2C(=O)CC2(C)CC(F)(F)C2)c(O)n1 C1(C#N)(C(=O)NCC=CC(=O)NCC(C)(C)F)CCCOC1 CC1CN(C(C2CCN(C)CC2)=O)CC1CNC(c1ccc(-c2cccs2)o1)=O N1(C(c2c(C)[nH][nH]c2=N)=O)CCC2(C1)CN(C(c1ncsc1C1CC1)=O)C2 N1(C(CCC(=C)Cl)=O)CCC2(CCC2NC(=O)CC2=CCCCC2)CC1 S(=O)(=O)(c1ccc(NCC(C)OC(C)(C)C)c(C#N)c1)N1CC(C)OC1 c1(CC(=O)NC(C2CCN(C(c3cncc(CC)c3)=O)C2)C)cc(C)ccc1C c1(C(=O)NC2CC(CNC(C3(C)CCCC3(F)F)=O)C2)ccc2c(c1)CNC2=O S(=O)(=O)(c1ccccn1)N1CC(CNC(c2cc(OC)c(O)cc2)=O)OCC1 Cc1cc(C)c(NC(=O)C(N2CCn3nncc3C2)c2cccc(Br)c2)c(C)c1 CCC(C)(C)OCCC(=O)NCCN1CCC1C c1(C(N2CC(SC)C(NC(=O)CC3=NNC(=O)C3)C2)=O)c(Cl)ccc(Cl)c1O C1(O)(CNC(C2CCN(CC)C2)=O)CCN(C(=O)C(F)=C2CCCC2)C1 c1(SC)ccc(NC(=O)C(c2ccco2)NC(C2CC3CC3C2)=O)cc1 c1(CC)cn2c(n1)CCC(C(=O)NC1(C3CN(C(c4ccncn4)=O)C3)CC1)C2 C1(C(N(C)CC2(O)CN(C(c3ccnn3C)=O)C2)=O)CCCC2(CCC2)O1 c1(NCCCNC(C2CC(OC)(OC)C2)=O)ccccc1SCC(=O)OC C1(NNC(CCF)C(=O)Nc2c(C(=O)C(C)=O)ncs2)CN(C)CCN(C)C1 CC#CCC(C(=O)NCC1CC[Si](C)(C)C1)NC(=O)C=Cc1cc[nH]n1 C1(C(N2CC(COC)C2)=O)C2CC3C(C2NC(C2(C(C)(F)F)CC2)=O)C13 C1(C(=O)NCc2cn(CC(=O)NCC(C(C)C)O)nn2)CCCOCC1 Cc1cc(Cl)c(C(=O)NCC(C)(C)CNC(C2(C(O)C(F)(F)F)CC2)=O)cc1F Cn1nc(C(=O)NCCC(O)CNC(C2(F)CCCOC2)=O)cc1Cl N=c1nc(O)cc(NC(=O)NC(COC(F)F)C2CC2)[nH]1 N1(C(c2occ(C)c2C)=O)C(CNC(c2coc(Cl)n2)=O)CC2CCCC12 N1(C(Cn2nc(C)oc2=O)=O)CC23CCCCC2(C1)CN(C(C1CC1(Cl)Cl)=O)C3 N#Cc1cccc(C(C(=O)Nc2ccccc2Cl)N2CCC2C2CCCC2)n1 c1(C(N2C(C)CC(NC(=O)CC3CC3)CC2)=O)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1 C1(C(=O)NCC2N(C(CC3CCC(OC)CC3)=O)CC2)Cc2cscc2C1 C1(NC(C(C)OCCC#C)=O)CC(C)(CNC(c2ccccn2)=O)C1 C1(CC)CN(C(=O)CC2CC(CF)C2)CCC1NC(=O)C(C(C)C)N(C)C CS(=O)(=O)c1coc(C(N2CC(NC(=O)CCCCC(N)=O)C(O)C2)=O)c1 C=CCCC(C(=O)N1CCN(C(C)=O)CC1)NC(C1(CC=C)CCCC1)=O C1(NC(c2nc(C)oc2)=O)COC2(C1)CN(C(=O)CN1CCC(F)(F)C1)C2 C1(CCC)CN(C(=O)CCC2CC2(F)F)CCN1C(=O)Cc1nnc(C)o1 CC(C(=O)NC(C1(C(N2CC(O)(CC3CC3)C2)=O)CCC1)=O)C(F)(F)C(F)F Cc1nn(C)c(Cl)c1C=CC(=O)NCC1CCN(C(c2ccccn2)=O)C1(C)C c1(C(=O)NCCCOCCNC(C(C)(C)C2CC2)=O)ccnc2ccccc12 N1(C(C2CCCCN2C(=O)C=Cc2cscn2)=O)CCOC2(CC2)C1 N1(C(C(C)NC(=O)NC)=O)CCCC(NC(=O)CC2CCOCC2)CC1 c1(NCc2ccc(C(=O)O)cc2F)cnc2cccnn12.N12CC3CC3(C1)C2=O N1(C(CC2CCN(C)CC2)=O)CCCC2(CCCCN2C(C2CCN(C)C2)=O)C1 C1(C(=O)OC)CCCCN1CCNC(C(C)(C)NC(=O)OC(C)(C)C)=O N1(C(COCCNC(C(CCC)OC)=O)=O)CCC(C)(COC)CC1 Cc1cccc(C)c1-n1cc(C2(F)CN(C(c3cccc(I)c3Cl)=O)C2)nn1 C1(c2n(C(c3ccc(C(C)(C)C)nc3)C)nnn2)(C(=O)O)CSCC1C c1(C(=O)OC)cc(C(N2CCN(C(CC(=O)OC(C)(C)C)C)CC2)=O)nn1C C1(C(=O)NC2C(C)CN(C(C3CCCC(C)C3)=O)CC2)CC(F)(F)CCC1(C)C CC(CN(C)C(c1coc(C2CC2)n1)=O)C(=O)N1CCC(CCN(C)C)C1 C=Cn1ncc(C(N2C(C(=O)NC3CC4CC4C3)CCC2C2CC2)=O)c1N Cc1ccc(C(=O)NC2CC2NC(=O)C(C(C)C)N2CCCC2=O)c(C)c1 c1(C(=O)NC(C)C)cc(-c2csc(NCC3CCSCC3)c2)ccc1F C1(S(C)(=O)=O)(C(=O)NC(CCCNC(CC(C)C)=O)C)CCCCC1 C12(NC(c3[nH]cc(C(C)=O)c3)=O)CCCC1CN(C(=O)CC1CNC(=O)O1)C2 C1(O)(C(C)NC(=O)CSc2n[nH]c(O)n2)CCN(C(=O)CC2COC(=O)C2)C1 C1(C(N2C(C(C)NC(c3c(OCC)scc3)=O)CCC2)=O)CCCC(F)(F)C1 C1(C(C)(C)C)CCN(C(=O)Cc2ccc(F)cc2)C(CNC(c2cnc[nH]2)=O)C1 c1(OC)ccc(C(N2CC(C(C)NC(=O)CC3(C)CC3)C2)=O)c(F)c1Cl N1(C(C(COC)(F)F)=O)CCC(CO)(CNC(=O)CCc2nncs2)CC1 c1(-n2c(C(F)Cc3ccccc3)nc(C(CC)O)n2)ccc(S(N)(=O)=O)cc1 c1(CC)cc(CC)nc(NCC2(NC(=O)C(C(C)C)SC)CCCCC2)n1 N#Cc1c[nH]c(C(=O)NC2CC2NC(C2(c3ccc(F)cc3)CCCC2)=O)c1 C1(OC)CN(C(c2cncs2)=O)C(C)(CNC(=O)CC#N)C1 CN1CCC2(CN(C(c3cnn(CC(F)F)c3)C(=O)NC3CC3)CCO2)C1 C1(O)(C(C)C)CCC(NC(c2cnn(C3CC3)c2Cl)=O)C1 C(C(=O)N1CCCC(CNC(=O)CSc2ccc(O)cc2)C1)(C(C)C)OC C(C(CC(C)C)C(=O)NC1(CO)CCCCC1C)NC(c1ccc(C)o1)=O C1(CC)CN(C(=O)Cc2c(Cl)cnn2C)CCN1C(=O)C(C)c1cncs1 N1(C(CC2OCC(C)(C)C2)=O)CCC(NC(c2ccnc(O)c2)=O)C(O)C1 C(C)(CNC(C1CC(N2CCCC2)C1)=O)(CC(C)C)NC(c1c(C)ocn1)=O C(C)(C(=O)N(CCC(=O)NC(C1CC1)C1CC1)CCO)OC C1(NC(C2CCN(CC#C)CC2)=O)CC(O)CN(C(=O)C(COC)NC(C)=O)C1 C1(C(=O)NC(C(=O)NC)(C)C)CN(C(=O)CN2CCC(C)CC2)CC1(F)F CCC(CC)C(C(=O)NC(C)(C)C)N(C)CC(N1CCOCC1)C1CCCO1 c1(CCC(=O)NCCCCCCNC(C(C)C2CCC2)=O)ccc2[nH]ccc2c1 C=CC1COCCN1C(C1CCCC1NC(C1CCCCS1)=O)=O CCC(C)C(O)C(=O)NCc1ccc(C(=O)N(C)CC2CCCN2C)o1 Cc1cc(C(N2CC(CNC(c3cncnc3)=O)C2)=O)c(Br)cc1F c1(OCCCC(=O)NC2C(CNC(CC3(C)CC3)=O)CCC2)ccccc1F Cc1cnc(C=CC(=O)NC2CCCC2NC(=O)COC2CCC2)[nH]1 N1(C(c2c(C)cns2)=O)CC(C(F)(F)F)C(CNC(C2CCCCC2)=O)C1 C1(C(N2CCC(Cc3ccsc3)C2)C(=O)NCCCSCC)CC2C=CC1C2 C(CCC(O)C(=O)NCC1C=CCOC1)NC(c1nc(CCC)oc1)=O CCC1CC(=O)NC(C23CCC(CC2)C3)CNC(=O)CN(C)C(=O)C1.NC.SC N1(C(c2cc(CC)no2)=O)CC(CNC(=O)CCc2cnc(O)[nH]2)C(C)C1 C(CNC(c1ccnc(OC)n1)=O)(CC(C)C)NC(C(CC)OC)=O CC(CCNC(=O)CC1(C)CCCO1)CCNC(c1coc(Br)n1)=O C1(C(N2CC(C(=O)NC(C(=O)OCC)CC)C2)=O)CCC2(CCC2)O1 N1(C(CSc2n(C)cnn2)=O)CCC(NC(c2csc(CO)n2)=O)C(F)C1 N1(C(=O)OC)CCC(C(=O)NCC2CCN2C(=O)C(C)NC(=O)CC)CC1 CCC(C)N=c1[nH]c2c(c(=NCC(C)(CCO)SC)[nH]1)CCCC2 c1(OCC)cc(C(=O)NC2CCC(CNC(c3cnc(N)s3)=O)C2)on1.C1CC1 C1(NC(CN2CCC(C)(C)CC2)=O)CCCN(C(C2(C)CCC2)=O)CC1F C1(NC(C(=O)NC(C)CCC2CCCO2)=O)(CO)CCOCC1 c1(C(=O)NCC2CCCC2NC(C2CCOCC2)=O)ccc2ncccc2c1F c1(C(N(CCNC(C2OCCC(C)C2)=O)C)=O)nn(C)c(Cl)c1Cl C1(NC(CC(C)N(C)C)=O)CCCCC1NC(=O)Cc1cnco1 C=C(Cl)CC(C(=O)NCC(C)(C)C1CCCC1)NC(=O)C(C)CO N1(C(CC(=C)C)=O)C2CCCC1CN(C(c1cccnc1NC(C)C)=O)C2 C1(N(C)C(c2cccnc2O)=O)CCCN(C(c2cnc(Cl)s2)=O)CC1 N=C1NC(=O)C(CC(=O)NCC(N2CCN(C(=O)CC3CC4(CC4)CO3)CC2)=O)S1 C1(N(C(Cc2cnc(C)o2)=O)C)CCCCN(C(C23CCCN2CCC3)=O)C1 c1(CNC(C2CC(NCc3ncc(Br)s3)C2)=O)nc2ccccc2[nH]1 N1(C(c2ccncn2)=O)CC2(CC(C(N3CCC4CC34)=O)CO2)C1 C1(C(=O)NC(C2CCN(C(C(CC=C)(F)F)=O)C2)(C)C)CCc2ncncc2C1 N1(C(C2C(CCOC)C2)=O)CCC2C(C(=O)N(C3CC3C)C)C2C1 C1(OC)CCn2cc(C(=O)NC(CNC(=O)C=Cc3nccs3)C(C)C)nc2C1 CC1CCCC(C)N1C(C1CCCN(C(c2cscc2Br)=O)C1)=O N1(C(c2cc(CC)on2)=O)CC2CC(C1)N2C(c1ccc(SC)s1)=O c1(C(C)(C)NC(=O)NCC2CC(N(C)C)C2)nnc(N)[nH]1 C(CCCCNC(=O)Cc1cnc[nH]1)N(C(=O)CSCc1ccccc1)C O=C(C1=CCOC1)N(C1CC1)Cc1cccs1.C12CCC13CC23 C1(NC(C)=O)CCC(C(=O)NCC2CN(C(=O)CC(C)(C)F)C2)CC1 N1(C(c2c(OC)cncc2)=O)C2CCC1C(CNC(c1cc(C)nc(O)n1)=O)C2 Cc1cc(C(=O)NC(Cn2cncn2)C(=O)NOCC(N)=O)nnc1O c1(OC)ccc2c(n1)NC(C(N1CCC(C(C)NC(c3nocc3C)=O)C1)=O)C2 C(CN=C(NCCSC)NC1CCC1)(c1ccc(F)cc1F)N(C1CCC1)C C1(C(=O)NC2CCC(N(C(=O)CCC#N)C)CC2)CCCCN1S(N)(=O)=O C(C(C)(C)CC(=O)N1CCCC1CNC(=O)C(C(C)C)NC(C)=O)OC C#Cc1ccc(C(N2CC(O)(C(C)NC(c3cnn(C(C)C)c3)=O)C2)=O)cc1F C1(C(N(C)CCN(C)C)=O)CN(C(C2CC(N(C)C)C2)=O)CCO1 C1(CNC(CC(=C)C)=O)CC2CCC1N(C(=O)C(c1ccccc1C)(C)C)C2 c1(CC)ccc(CC(=O)N(CC(O)CN(C(=O)C(C(C)OC)N(C)C)C)C)cc1 C1(C(=O)NC2CC(C)(NC(c3ccncc3C(F)F)=O)C2)CCc2nc[nH]c2C1 C(=O)(CCCC(C)(C)C)NC12CN(C(Cc3c(C)nc(S)s3)=O)C(C1)CO2 N1(C(C(CCC)C)=O)CCC2(CCOCC2)C(NC(=O)C(CC(C)C)OC)C1 N(C(=NCCC(=O)N(C)C)N1CCC(CS(C)(=O)=O)C1)CC(C)C c1(C(N2CC3CC3(CNCc3sccc3Cl)C2)=O)cc([N+](=O)[O-])c(Cl)cc1F C(=O)(C1=NOC(CNC(c2cccc[n+]2[O-])=O)C1)N(CC(C)(C)O)CC N1(C(C(C=C)OC)=O)CCC12CN(C(=O)CC1CCCN1C)C2 CCCS(=O)(=O)CC(=O)N1CC2CCOC2(CNC(C2CC2(C)C)=O)C1 n1(CCN(C(c2cc(-c3ccco3)[nH]n2)=O)CC)cc(CN(C)C)nn1 N1(C(C2CCN(C(C)=O)CC2)=O)CC(NC(C2CCC3(CC3)C2)=O)CC(C)(C)C1 C[Si](C)(C)c1cccc(C(=O)NOCC(F)(F)F)c1 c1(CC(=O)N(CC)CC2CCCN2C(=O)COC(C)C)ccc(F)c(Cl)c1F c1(C(=O)NC2CN(c3c(OC)c(Cl)ncn3)CC2C)cc2ccc(O)nc2s1 O=C(C1=CCCCCC1)N1CC2C(C1)N2C(C1CC12C(=O)Nc1ccccc12)=O c1(C(N(CCCNC(=O)CCc2ccoc2)C)=O)cc(F)cc([N+](=O)[O-])c1 c1(C(N2CCC(C)C2CNC(C2C3(CC3)C23CC3)=O)=O)nc2cc(O)ccc2[nH]1 c1(C(N(CCC(C)NC(c2cn(CC)nn2)=O)C)=O)cccc(N)n1 C1(NC(c2ccc(CC)cc2)=O)CCN(C(c2csc(CC)n2)=O)CC1O CCC(C(F)(F)F)NC(CC(C)c1ccccc1)c1nnnn1C c1(C(=O)NCC(CNC(CC(CC)C2CCC2)=O)OC)ccc(F)c(OC)c1 C(C1=CCCN(C(=O)C(=Cc2ccccc2)C)C1)NC(CN(C(C)=O)C)=O C1(CN(C(C2CN(C)C2)=O)C)CN(C(=O)CCC(=O)N(C)C)CCO1 c1(C(=O)NCC2N(C(C=CC(CC)=CC)=O)CCC2)cnc(OC)cn1 Cc1cnccc1CN(C)C(c1ccc(CNC(=O)CC2CC2C2CC2)nc1)=O C1(C(=O)NC2C(NC(CC(C)C)=O)CCC2)COc2ccc(F)cc2C1 c1(C(N2C3(CNC(C=CSC)=O)CCCC(C2)C3)=O)ccnc2ccccc12 C1(C(C)C)CCC(C)N(C(C23CC(CO)(C2)OC3C)=O)C1 C1(C(=O)NC(C=C)CO)CN(C(C2CC23CCOCC3)=O)CC12CCC2 c1(OC)ccc2cc(NC(=O)NC(C)Cc3cnccn3)ccc2c1 C=CC(C)(O)C(=O)NC1CCCC(NC(=O)C(F)(F)C2CC2)C1 C(c1cccc(O)c1)=CC(=O)NC1(CNC(=O)CC2(O)CCCOC2)CC1 C1(COC)(NC(=O)C(C)OCCN(C)C)CCN(C(=O)CCS(C)(=O)=O)CC1 C(=O)(C#CC1CCCO1)N1CCC(F)(CNC(=O)C=Cc2cnc[nH]2)C1 c1(C(N(C2CN(C(CNC(C)=O)=O)CC2(C)C)C)=O)ccc2cncn2c1 c1(CC)nocc1C(N1CC(O)(CN(C(=O)C(C)OCCN(C)C)C)C1)=O c1(C(N(C2CCCC2)CCNC(C=CCCC)=O)=O)cc(CN(C)C)on1 N#CC1=C(C(=O)NCC2CCC(NC(c3cnc(C4CC4)nc3)=O)C2)CCC1 C1(OC)CN(C(=O)CN(C)C(N)=O)CC1C(=O)NCC1(O)CC1 c1(C(=O)NCC2CC(C)N(C(=O)CC(C)(O)C3CC3)C2)ccc2cccnc2c1 C1(CC=C)(C(=O)NCC2(C(=O)NC3CC34CCC4)CCCC2)CCOC1 N1(CC(N2C(C)(C(=O)NC3COC(=O)C3)CCC2)=O)CCCCCC1=O CCC(CC(=O)N1CC=CC1(C)C(=O)NCC1(O)CC1)C(C)C n1(CCOC)nc(-c2ccc(F)cc2)nc1-c1ccc(CC(C)C)s1 C1(NC(c2c(OC)ccs2)=O)CC(NC(=O)CC23CC(C2)C3)CC1O N1(C(CCCC)=O)CC(CNC(=O)C(C)(O)CC)OC2(CCC2)C1 CCCN=C(NCc1cc(C)on1)NCC1CCCN1S(C)(=O)=O N1(C(C2C3N(C(CC4CC(SC)C4)=O)CC(C=C3)C2)=O)CC2(CCC(O)CC2)C1 Cc1cc(C(=O)N(C)CC2CN(C(C3CCCCS3)=O)CCO2)c(C)nc1C c1(C(=O)NCCC(C)N(C(=O)C(C)CC(F)F)C)cnc2sccn12 CCCCCCCC(=O)N1CC(O)CCC1C(=O)NCc1nnc(O)n1CC c1(CC)cc(C(=O)NC(Cc2cn[nH]c2)C(N2CCOC(C)C2)=O)nn1C C=CCCCC(=O)NC(C1CCCN1C(c1cc(-c2ccccn2)c[nH]1)=O)(C)C N1(C(C(C)NC(=O)OC)=O)CCOCC(C)(CNC(=O)CCc2cc(C)[nH]n2)C1 N1(C(C2C(=C)C2)=O)CCCC(CNC(c2ccc(CC(C)C)cc2)=O)C1 C1(CNC(=O)CONC(=O)C2CC(OC(F)F)C2)CC2CCCC2C1 N1(C(CCCC#C)=O)CCN(C(c2cc(C(C)=O)c[nH]2)=O)C(COC)C1 C(=O)(C1CCCc2ncnn21)N1CCC(NC(C2CCOC2)=O)C(O)C1 C1(C(C)C)(C(=O)NC(CCO)C(C)C)CCCN1C(c1csnn1)=O N1(C(C2C(=C)C2)=O)CC=C(CNC(=O)C(CN(C)C)c2ccccc2)CC1 c1(C(=O)NC(C2OCCN(C(c3scc(OC)c3)=O)C2)C)ccc(S(N)(=O)=O)o1 C1(NC(c2cn(C(F)F)cn2)=O)CC2(CCN(C(=O)C=C3CCSCC3)CC2)C1 CC(C)(CC1CCC1)C(=O)NCCC1(O)CCN(C(=O)C=Cc2cc[nH]n2)C1 C1(F)(C(=O)N(CC)CC)CCN(N2CCn3c(cnc3-c3ccccc3)C2)CC1 C12(COC)CN(C1)C2=O.c1(C)ccccc1.C(CC1CC1)(C(=O)O)NC(=O)OC c1(NCc2ccc(CNC(c3cc(CC)n(C)n3)=O)cc2)ncnc2scnc12 N1(C(c2cc(C)oc2C)=O)CCc2ccccc2C1CNC(c1cn[nH]c1)=O C(C)(C(=O)NCC1(NC(=O)CCc2ncccc2C)CCCCC1)(C(C)C)OC Cc1nn(C)c(Cl)c1CN(C)C(C1CC1(c1ccc(Br)cc1)F)=O CC1CCC(S(C)(=O)=O)CN1C(c1ccc(N2CCCC2=O)cc1)=O N1(C(c2c(C)nccc2)=O)CC2ON=C(CNC(C3(CC4CC4)CC3)=O)C2C1 C(c1cccc(Br)c1)=CC(=O)NC1(CNC(C(C2CCC(C)CC2)CC)=O)CC1 Cc1cc(C)c(C(=O)NC2(C(=O)NC(CO)CC(C)(C)C)CC(F)C2)cn1 c1(C(C2CC2)NC(C2N(C(C(CC)C)=O)CSC2)=O)ccccc1COC c1(C(=O)NCCN(C)C(c2cc[nH]c2)=O)n[nH]c(C2CC2)c1Cl Cc1ccc(C(=O)NCC(N2CC3CC3(NC(c3nc(Cl)cs3)=O)C2)=O)cc1 c1(CNC(Cn2c(C)cc(C)n2)=O)cc(O)nc(CNC(=O)C(C)NC(N)=O)n1 C1(CC(=O)NCC2(CO)C(C)(C)C2)CS(=O)(=O)CCO1.CCC(=O)O CC(C)CC(O)C(C)C(=O)N1CSCC1C(N1C2COCC1C2)=O c1(C(=O)NCCC(C)N(C(CC2CCC(CC)CC2)=O)C)cnc(CO)nc1C N1(C(C(CC)CCOC)=O)CC(C)CN(C(c2ccc3nc[nH]c3n2)=O)CC1C N1(C(CC(=O)OC)=O)CC2CC2(C(=O)N(C(C)CO)C2CC2)C1 c1(C(N2CCN(C(C(CC)=CC)=O)CC2COC)=O)cnc(O)c2ccccc12 CC1CN(C2CCC2)CC1(c1nnnn1C1CCCC1)Nc1c(Cl)nsc1Cl c1(C(=O)NCC=CCNC(C(CC)n2nccc2C)=O)cc(SC)ccc1C C(=O)(C(O)CCCC)N1C(C(N2C(CCC)COCC2)=O)CSC1 c1(C(=O)NC2CC3(C(C(N(C4CCCCC4)CCC)=O)C3)C2)ccc(C)nc1C C1(OC(c2ccc(SC)cc2)=O)CC2CC1CN(C(=O)COc1cccnc1)C2 N1(C(c2cnc(C(C)C)o2)=O)CCCCCCC1C(=O)NCCCOCCCO Cc1c(NC(C)CS(N)(=O)=O)ncnc1N1CCN2C(=O)CC12 CCC(CC)(CO)C(=O)NC1CC2C1CCN2C(=O)C(C(C)C)n1cnc(C)c1 C(=O)(C1=CCC2(COC2)OC1)N(CCCNC(c1ccnn1CC(F)F)=O)C c1(CNC(c2cc(CC)oc2C)=O)ccc(CNC(C2(C)CC2)=O)c(F)c1 CC#CCC(C)N=c1nc(N2CCC3(CC2)CC3(F)F)c2c([nH]1)CCC(C)C2 C12(CNC(C3(CCC)CCNC3=O)=O)CCC(C1)N(C(c1ccsn1)=O)C2 C(C)(CNC(=O)Cc1csc(C)c1)(CC(C)C)NC(C(CC)OCC)=O C1(CNC(=O)Cn2cccn2)CC2CCC1N(C(c1ccc(CO)o1)=O)C2 N1(C(c2cc(C(=O)OC)ncc2)=O)CCCC(CO)(NC(=O)CC(C)N(C)C)C1 C1(CC(=O)NC2(C)C(NC(Cn3nc(C)oc3=O)=O)CCC2)CCC(C)(C)CO1 C1(NC(C2CC2C2CC2)=O)CN(C(c2cc(I)ccc2F)=O)CCC1(F)F c1(N2C(CN(C(COC3C(C)CCCC3)=O)C)CCC2)ncnc(Cl)c1[N+](=O)[O-] n1(CC)ncc(C(=O)NC(C)C(CO)NC(=O)CC2CC(C)=NO2)c1Cl C(=O)(C(C)CC1CCCC1)N(C(=O)CNC(c1nccs1)C1CC1)CCF.CO C1(NC(c2c(CNC(=O)CCn3cnnn3)cc[nH]2)=O)CC2CC3C(C2)C13 C1(CC)CN(C(C2(C)CCCS2(=O)=O)=O)CC(C)N1 C1(C#N)(CC(=O)NC(CN(C(c2ccnc(C(C)C)n2)=O)C)C)CCOCC1 O=C1CCC(C(=O)NC2CCCC2CNC(C2CN(C(=O)CC(F)(F)F)C2)=O)CN1 C(CC1CCC1)(C(=O)N1CCCC1CF)NC(CC1CC(=C)C1)=O CC1CC(NC(=O)C=Cc2cn(C)nn2)CN(C(c2ccc(N)c(F)n2)=O)C1 Cc1ccc(O)c(C(N2C3CCC2C(C(=O)NC2(C)CCC(C)C2)C3)=O)c1 N1(C(C2CCC(C3CC3)CC2)=O)CCC2OCCN(C(=O)COCC3CC3)C2C1 n1(CCCC)ncc(C(=O)NCCN(CC(C)O)C(c2occ(C)c2C)=O)c1C N1(C(C)=O)CCCC(NC(=O)C(Cn2cncn2)NC(=O)Cc2cnn(CC)c2)C1 N1(C(c2cc(OCC)no2)=O)CC(CO)C2(C1)CN(C(=O)C(F)CCC(C)C)C2 CCCCC(CC(=O)N1CCC(C)(CC)CC1)NC(c1coc(C)n1)=O C(CC(C)(C)C(=O)Nc1ccccc1F)NC(C(C)n1cccn1)=O C1(C(N2CC(=C)C2)=O)CCN(Cc2ncsc2C)CC1O N1(C(C2CN(CC)C(=O)N2)=O)CC(CO)C2(C1)CN(C(C1(C(F)(F)F)CC1)=O)C2 C=CC1CCCN(C(c2cccn2CC)C(=O)Nc2ccccc2C)C1 C(=O)(C(C)CC(=O)OC)NC(CC(=O)NC(CCOC)C)CC1CC1 C#CC(CC(C)(C)C)NC(=O)CC(C(C)C)NC(=O)CC1(O)CCOC1 N1(C(C(C)S(N)(=O)=O)=O)CCC(CNC(=O)CCC(F)F)C(F)(F)CC1 Cc1cc(CC(=O)NC2CS(=O)(=O)CC2NC(c2cnc(S)n2C)=O)cc(F)c1 c1(C(=O)NCC=CCNC(C2C(CC)C2)=O)ccc([N+](=O)[O-])cc1C(F)(F)F c1(CC(=O)Nc2ccc(F)cc2Cl)cn2cc(-c3cccc(CO)c3)ccc2n1 C1(NC(CC(COC)C)=O)CC(N=c2[nH]nc(CO)s2)C12CCOCC2 N1(C(C(CC)CC)=O)CCN(C(=O)Cn2[nH]cnc2=N)CC2CCCCC12 CC(c1ccccc1)=CC(=O)NC(C)CCCNC(c1cocn1)=O c1(SCCC(=O)NC(C(C)NC(CCCC)=O)CO)ccc(F)cc1F Cn1ncc2cc(CN3CCC(NC(=O)C(=O)NCC(F)F)C3)cnc12 N1(C(C2CCN(C(C)C(=O)NC(=O)CC3CCC(=O)N3)C2)=O)Cc2ccccc2C1 c1(NC(C2COC(C)(C)O2)CO)ccc(S(=O)(=O)NCC2CCC2)cn1 N1(C(CCCOCC)=O)CCN(C(C2ON=C(C)C2C)=O)CC1c1cnn(C)c1 C1(C2CCN(C)CC2)(C(=O)NCCCN(C(=O)CCCC(C)(C)C)C)CC1 N1(C(C(CC=C)CC)=O)CCC(C)(C)C(C(N2CCC(OC)C2C2CC2)=O)C1 c1(CC)cc(C(=O)NCC(C)NC(C2CCC(C)OC2)=O)c2c(c1)CCO2 C(CCC(C)C)(C(=O)N1CC2(CCC2)CC1CNC(=O)C(F)(F)CO)NC(C)=O N1(C(c2cn(C3C(OCC)COC3)nn2)=O)CCN(CCC(Cl)Cl)CC1 CCC(CC(=O)NCC1(NC(C2(CO)CCCCC2)=O)CCC1)OC C(=O)(CC(=O)NC(C(=O)NCC(F)C1CCC1)c1cccs1)OC c1(C(N(C)CC2CCCN(C(CC(C)O)=O)C2)=O)ccc(C(C)(C)C)c(Cl)c1 C(CCC(=O)N1CCC(CCNC(=O)Cn2cc(Cl)cn2)C1)=C(C)C C1(C#CC(=O)NCC(C)(C(C)C)NC(c2cc(C#N)ccc2F)=O)(CC)COC1 c1(C(=O)NC(C2CCCN2C(=O)CCc2ccsc2)C)ccnc(C(F)(F)F)c1 c1(C(C(N2CCCC(c3cn(CC(=O)OC)nn3)C2)=O)C)ccc(F)c(OC)c1 c1(C(N)=O)cc(CCC(=O)NC(C(C)(C)C)c2nc(C3CC3)no2)c[nH]1 c1(C(=O)NC2C(NC(c3cccc(N(C)C)c3)=O)C2)ccc2c(n1)CCC2 Cn1nc(CC(=O)NC2(C)CC(NC(c3csc(C#N)c3)=O)C2)cc1Cl N1(C(CC2CC(=C)C2)=O)CCN(C(=O)C(C)OC2CCCC2)CC12CCC2 C(=O)(C(CC(C)CC)NC(C1C=C(C)CS1)=O)N1CC(C=C)(O)C1 C1(NC(c2scnc2Cl)=O)CC(F)CN(C(=O)CCc2cnc[nH]2)C1 C1(C(N(C)Cc2cnnn2C)=O)CC(C)(C)CCN1C(=O)CC1CCSC1 c1(C(=O)NCC2CN(C(=O)C=Cc3cc[nH]n3)CCO2)cc(F)cc2nn[nH]c12 CC1C(C(=O)NC2CCC(C(=O)NC3(C)CC(O)(CO)C3)C2)CCN1C C(=O)(C1=CC(C)CC1)NCCN(C(CCC)=O)CCc1ccccc1 c1(C(=O)NCC2CN(C(CCc3cnc(C)o3)=O)C2)cncnc1C1CC1 CC1(C)C(CO)CN1C(=O)CSCCNC(C1CC(F)C1)=O CC1CC(NC(=O)CCc2nncn2C)CN(C(=O)C(C)CN2CCOCC2)C1 CC(C(=O)NC1(CCC(=O)NC)CCC1)N(CCCCC1CC1C)CCO.N(C)C C1(NC(c2c(C)cns2)=O)CCN(C(C2CCSCC2)=O)C1(C)C N1(C(CS(CC)=O)=O)CCN(C(c2ccc(Cl)c(C)c2)=O)C(COC)C1 c1(C(=O)NC2CC(CCNC(C3CC(C)C3)=O)C2)c[nH]c2ccc(Br)cc12 N1(C(c2cncc(OC)n2)=O)CC2(C1)CN(C(C1CC1c1ccc(Cl)cc1)=O)C2 CCCC(C(=O)NC1C=CC(CNC(c2nccnc2C(F)(F)F)=O)C1)OC N1(C(CC(CCC)O)=O)C2CCCC1CN(C(c1c[nH]nc1C(F)F)=O)C2 C1(NC(CCN(CCC)C)=O)CC12CCN(C(c1ccc(C)nc1C)=O)C2 C1(C2CC2)(CNC(c2cc(OC)nn2C)=O)CCN(C(=O)CC(C)C2CC2)C1 c1(C(N2CCC(C)(NC(C(CC)SC)=O)C2)=O)cc(C)c2c(O)nc(O)nc2n1 C1(CCNC(=O)CC2CCOC2)CCCN(C(=O)C=Cc2ncc[nH]2)CC1 C1(NC(c2cc(CCC)on2)=O)CCCCC1NC(=O)CCc1ccccc1Cl C(=O)(CCC(=O)NCC(C)(F)CNC(c1nnc(S)n1C)=O)N(C)C N1(C(=O)OCc2ccccc2)CCN(C(C2C=CCCCC2)=O)CC(O)C1 Oc1nnc2n1CCN(c1nc(N3C4CCCC3CC4)nc3ccsc13)C2 C1(NC(c2ncc(C)nc2)=O)CCCN(Cc2nc(C)c(C)o2)CC1 N1(C(C2(CC#C)CCCCC2)=O)CCCC2(NC(c3cncc(C)c3)=O)CC2C1 c1(C(=O)NC(C)CN(C(=O)CCc2ccccc2O)C)c2c(nn1C)CCCC2 Cc1cc(C(=O)N(CC(=O)NCCOCC(N)=O)C(C)C)nn1C CC1CCC(C(=O)Nc2ccc(O)cc2Cl)N(C(=O)CCCN=[N+]=[N-])C1 Cc1ccc(CC(=O)N(C)CC2CCN(C(c3nscc3C)=O)CC2)c(F)c1 O=C1CC(CC(=O)NCC2CC3CCC2N3c2ncc(Br)c(O)n2)CCCN1 NC(=O)CCC(=O)N1CCC(NC(=O)C=CCOC2CCOCC2)C1 c1(C(N(C2CCCC(NC(c3ccc(CCC)s3)=O)C2)C)=O)cc(N)nc(Cl)c1 C(=O)(CCCCCC(=O)NC1C=CC(CNC(=O)C(C(C)(C)C)OC)C1)OCC C(C1CCOCC1)=CC(=O)N(CC(C(=O)NCC(C)(C1CC1)OC)C)C CC1CC(CC(=O)NCc2ccc(CO)cc2)CN1C(c1cccc(Cl)c1)=O S(=O)(=O)(c1c[nH]ccc1=NC1CCc2ccccc21)N1CCC(OCCSC)CC1 c1(OC)cc(Cl)c(C(N2C(C(N3CC4CCC3CC4)=O)CCC2C)=O)cc1OC N1(C(CC2CC(C)(C)C2)=O)CC(NC(=O)CC2CC(=O)NC(=O)C2)CC12CCC2 C1(C)(C(=O)NC2CCC(CNC(C(C)OC3CCCC3)=O)C2)CC(F)(F)C1 Cc1ncnc(C)c1CC(=O)NCC(=O)NCC1C=CCOC1 C1(O)(COC)CCN(C(c2n[nH]c(C)n2)C(=O)NCC2CCCO2)C1 c1(OC)ccc(OCC(=O)NC2(C3CCCN3C(=O)C(C)CN(C)C)CC2)cc1 CC1(CNC(C2(C)CC2Br)=O)CCCN(C(C2CC(=O)N2)=O)C1 c1(NC(=O)NC2CC(C(=O)Nc3cc(C)cc(Cl)c3)C2)c[nH]c2nccc-2c1 C1(NC(CCCCC)=O)CN(C(C2OCCC2C(=O)OC)=O)CC(C)(C)C1 N1(CC)CC(NC(c2conc2CNC(=O)CC2CCCC(=O)C2)=O)CCC1=O c1(OC)ccc([N+](=O)[O-])cc1C(C)NC(=O)C(c1ccccc1F)(F)F CC(O)CCCCCC(=O)N1CC=C(CNC(C2CC(C(C)C)=NO2)=O)CC1 c1(C(N(CC(CNC(c2c(C(C)C)cco2)=O)C)C)=O)ccc2c(c1)CCCO2 C1(CNC(=O)CCc2cnoc2)CCC(NC(c2ccnn2C2CCC2)=O)CC1 Cc1sc(Cl)nc1C(N1CC2CC2(NC(c2cc(Cl)ccn2)=O)C1)=O c1(C(N2CCC(NC(=O)CC3(CO)CC3)C2)=O)ccc(C(F)(F)F)nc1.C1CC1 C(C(C)(C)CNC(c1cnn(-c2ccccn2)c1)=O)NC(C(C)n1cccc1)=O N1(C(=O)NCCOC2CCSCC2)CCc2ccccc2C(O)C1 CC(C)CCC(=O)N1CC(CO)(NC(=O)C(N2CCCCC2=O)C)C1 c1(CC)[nH]c(Cl)nc(=NC(C)CNC(C2(C)CCOC(C)C2)=O)c1C#N C1(NC(CS(=O)(=O)NCC)=O)CN(C(=O)C=Cc2cc[nH]c2)CCC1O c1(NC(CC(=O)OCC)=O)cn(C)c(C(=O)NC(c2ccc(O)cc2)CO)n1 N1(C(c2c(SC)scc2)=O)CCOCC(NC(=O)CN2CCCC2C)C1 CCC(CC)CC(F)C(=O)N(C1CCN(C(=O)CCCCNC(N)=O)CC1)CC CC(CC(=O)N1CCN(C(=O)Cn2cccn2)C2COCC12)CC(F)(F)F c1(OCC)c(C(N2CC(CO)(NC(c3cc(C)cc(C)c3)=O)C2)=O)cccc1F c1(C(=O)Nc2ccc(NC(C(CN(C)C)(C)C)=O)cn2)cc2cnccc2[nH]1 N1(C(c2c(C)nsc2)=O)CCN(C(C2CS(=O)(=O)C2)=O)CC1C(F)F C1(N(C(CCOCC)=O)C)CCN(C(c2csc(COC)n2)=O)CC1C C(N=c1nc(N2CC3CC2CS3(=O)=O)c2ccccc2[nH]1)c1n(C)cnn1 N1(C(C2C(C)CC(C)O2)=O)CCN(C(=O)C(C)(C)c2ccccn2)CCC1C N1(C(C=C(C)c2ccco2)=O)CC2CCC(N(C(=O)C(C)n3cccn3)C)C2C1 C1(NC(C(CC)F)=O)CC2(C1)CN(C(C1CCCN(C(C)=O)C1)=O)C2 CC(CNC(c1cccnc1-c1ccncc1)=O)(C(F)(F)F)c1ccccc1 N#Cc1cn[nH]c1C(N1CC(OCCNC(=O)C(C2CCCCC2)F)C1)=O O=C(C1=COCCC1)NCC1C2CC1N(C(c1cn(C3CCC3)nn1)=O)C2 N(C(=NCCCSC1CCOC1=O)NCCF)C(C)C1CC1 Cc1nc(-c2nc[nH]n2)sc1C(=O)N(CCCCNC(C1CC12CCCC2)=O)C C1(C(=O)NCC(C)NC(=O)C(c2ccccc2F)C)(OC)CCCCC1 N1(C(CNC(c2cc[nH]c2)=O)=O)CC2CC2C2CC12 C#Cc1cncc(C(N2CC(O)(C(F)C(=O)NC(CC)(CC)CC)C2)=O)c1 N1(C(CCOCCC)=O)CCC(N(C(=O)CCc2cscn2)C)C2(CC2)C1 O(NC(=O)CCCCOC)c1c(OC)nsc1 c1(CNC(c2nnn(COc3ccc(F)cc3)c2-c2ccccc2)=O)cc(F)c(Cl)c(F)c1 CCC(C)C(C(=O)NC(C(=O)Nc1cccc(C(F)F)c1)C1CCCC1)N(C)C C(=O)(C(CC(F)F)N(C(=O)C1=COCCC1)C)NCP(OCC)(C)=O N1(C(C2CC(OC)CN2C(=O)CC(C)(C)OC)=O)CCC2(CCCCO2)C1 N1(C(C(CC)F)=O)CCN(C(c2cn(C)cn2)=O)CC1c1cccnc1 N1(C(c2nn(CC)nc2C)=O)CC(C(N2CCC2(C)CCO)=O)CC12CCC2 N1(C(c2cc(CC)[nH]n2)=O)CCN(C(C2CCOC2(C)C)=O)C(C(F)F)C1 CN1CCN(C(c2cc(CCNC(=O)CCc3cnco3)on2)=O)CCC1=O CC1CCCc2cc(C(N3CCC(CC(C)NC(=O)C4CC4)CC3)=O)nn21 C1(=O)CC(C)CC(=O)OC(CC)CN1.C(=O)(C(C)(C)CO)Nc1ccccc1 c1(OC)cc(NC(c2cccc(NCc3ccc(F)cn3)c2)=O)ccc1Br CCC(O)C(C)(C)C(=O)N1CCC1C(=O)NCCC(=O)OC(C)C c1(C(N2C(C(N3CCCC(C#N)C3)=O)CC3CC32)=O)cc2ncccc2[nH]1 Cc1cc(Cl)c(C(=O)NC2CC3CC2N(C(=O)CCc2cn[nH]c2)C3)cc1C Cc1cc(C(=O)NC2CC(C)CN(C(C3(S(C)(=O)=O)CCC3)=O)C2)ccc1F C1(NC(C2CC2F)=O)(CO)CCCN(C(=O)CCC2CCCCO2)C1 c1(C(N2CC(C(C)(C)O)(CNC(c3nc(C)c(C)s3)=O)C2)=O)ccc(Cl)nc1N N1(C(C2CCN(C)C(=O)C2)=O)C2CCCC1CC(NC(C1C=CCC1)=O)C2 c1(C(=O)NC2C(CCC)CN(C(C3C=CCC3)=O)C2)cnc(C)cc1C C12(CNC(=O)Cc3cnc[nH]3)CCC(C1)N(C(c1ccc(F)cc1Cl)=O)C2 C1(C)(C(=O)NC(CCCNC(c2c(CCC)n[nH]c2)=O)C)CCC(C)=C(C)C1 CC1CC(C(=O)NCC2CN(C(c3occc3-c3ccccc3)=O)C2)CO1 C1(CN(C(C2CC(C)(C(=O)OC)C2)=O)C)CN(C(=O)CC(O)C(C)C)CC12CC2 Cc1cc(OCC(=O)NCCCOCCNC(=O)Cc2csc(C)c2)no1 CC(C(C)C(=O)NCC1CCN(C(C2OCCO2)=O)CC1)C1CCCCC1 c1(C(N(C2CCC2)C(=O)OC(C)(C)C)=O)cc(=O)c(O)c[nH]1.C12(CCCC1)N(C)C2 c1(OC)cc(NC(=O)C(=O)NC2CCCC(C(F)(F)F)C2)c(F)cn1 Cc1oc2ccccc2c1CC(=O)NCCC(C)N(C(=O)CC(F)(F)C(F)F)C N1(C(CCCCC)=O)CCC(C2CCN(C(=O)C(c3cnn(C)c3)O)CC2)C1 Cc1cc2ncc(C(N3CCC4(CCCN4C(=O)Cc4cnc[nH]4)C3)=O)cn2n1 C1(NC(C(COCC)C)=O)CCCCN(C(c2cc(NC(C)=O)ccn2)=O)C1 c1(OC)ccc2[nH]cc(C(N3CC(N4CCN(C(=O)COC5CC5)CC4)C3)=O)c2c1 c1(C(=O)NC)ccc(CNC(=O)NC(C)(CO)C2CCC2)o1 C=CC(C)(C)C(=O)NCCC1(NC(c2cnn(CCC)c2C)=O)CC1 C(C(=O)N1CCCC1CN(C(=O)CCc1cc(C)no1)C)(C(C)C)SCC C1(C)(CNC(c2ncc(C)cn2)=O)CN(C(=O)CCCCCF)CCO1 C(=O)(CCS(C)=O)NCC1(CCNC(Cn2cc(C(C)O)nn2)=O)CC1 c1(C(=O)NC2C3(CNC(C=CCOC)=O)CCC(C2)C3)cccc2nc[nH]c12 CCCC(C(=O)NCCCc1cc(C)no1)NC(c1ccc(C#N)o1)=O c1(C(N2CCC(CNC(C(C=C=C)C)=O)C(C)C2)=O)c(F)cc(C#N)cc1F C1(NC(Cn2c(C)cnc2)=O)CC2CCC(C1C)N2C(c1ncsc1C(C)C)=O n1(C(C)(C)C)nnc(CC(=O)NCCCN(C(=O)COC2CCCCC2)C2CC2)n1 c1(C(=O)NCCCN(C(=O)CCN2CCCC2=O)C(C)C)cn(C(C)(C)C)cn1 C1(C)(OC)CN(CC(=O)NCC(C)(C)CN(C(=O)COCc2ccnn2C)C)C1 N1(c2nnc(C(C)C)o2)CCN(C2CCCN(C(C3CC=CCC3)=O)C2)C(=O)C1 C(CCC(C)C)(C(=O)NC(C1(O)CCC1)C)NC(c1ccc(C)[nH]1)=O c1(CC(N2CCC(NC(CN(S(=O)(=O)C3CC3)C)=O)CC2)=O)ccccc1S(C)=O CC1CN(C(C2CSC2)=O)CCC1NC(=O)C1=CSCS1 CC1(C(=O)NC2CC3C=CC2C3)CCCN1C(=O)CN1CCCC1=O CC1CN(C(C2(C)CC(=O)C2)=O)CC(C(=O)N(CC(O)CF)C)O1 N1(C(c2cnc(OCC)c(Cl)c2)=O)C2CCC1CN(C(c1cccs1)=O)CC2 N1(C(C(COCC)C)=O)CC(C(N2CC3CCC3(CO)C2)=O)C(F)(F)C1 C1(NC(C(C)OCC2CC2)=O)CCCOC12CCN(C(c1cnc[nH]1)=O)CC2 CC1(C)CCC(C(N2CCOC3CC23)=O)CN1C(C1C2CC3C(C2=O)C13)=O C1(C)(C(=O)NCC2OCCN(C(CCc3n(C)c(S)nn3)=O)C2)COC(=O)OC1 c1(C(c2n(CC=C)nnn2)NCc2ccco2)ccc(OCC)cc1 C1(CNC(C2(c3ccc(Cl)nc3)CC2)=O)COCCN1C(c1cc[nH]c1)=O C(=O)(C(CC)C(=O)N1CCC(C)(C(=O)NCC(O)C(F)F)CC1)OCC C1(C2CC2)(C(=O)NCC(CC)NC(c2cnn(C)c2F)=O)CC=CC1 C1(NC(c2cccc(OC)c2C)=O)CC2(CCN(c3ccn4ccnc4n3)C2)C1 N1(C(C(CSC)OC)=O)CCN(C(C2CCC(NC(C)=O)CC2)=O)C2(CCC2)C1 N1(C(c2cc(CCNC(=O)C(O)CC(F)(F)F)on2)=O)CC2CCCC2C12CC2 c1(C2(C(N(C3CCN(C(c4sncc4Br)=O)C3)CC)=O)CC2)ccccc1 C=CCC(C)(C)CC(=O)N1CCOC(C(N2CCC(F)(F)C(O)C2)=O)CC1 N1(C(CC(CC=C)NC(=O)CCCN(C)C)=O)CCC(O)CC12CC2 N1(C(C#CCNC(Cc2c(C)nccc2)=O)=O)CC(C)(C2CCC2)C1 C1(C(=O)NC2(CO)CC(O)C2)C2CC(O)C(C2)N1C(C1CC=CC1)=O N1(C(C(CC)OC)=O)CCCCC1CCNC(=O)CC1CC(C)OC1C C1(CNC(c2c(Cl)nc(OC)s2)=O)CCC(C)N(C(c2cc3occc3s2)=O)C1 C1(CNC(c2cc(CC)no2)=O)CC(F)(F)CN1C(C1CCCC(CF)C1)=O Cn1nc(C(N2CCC(O)(CNC(C3CCC(CCO)CC3)=O)C2)=O)cc1C#N O=C(C1=CC2(CN(C(c3ccnc(O)c3)=O)C2)OC1)NC1(CF)CCCC1 C1(CNC(c2cnc(OC)s2)=O)CC12CCN(C(c1cc[nH]c(=N)c1)=O)CC2 CC(O)CC(Cc1nc(C2CCC(N)C2)no1)c1ccccc1 Cc1cc(C(=O)NCC2COCC2NC(=O)CCC2CCOCC2)c(O)c(C)n1 c1(C(N(C)CC2CN(C(=O)CCF)CC23CC3)=O)ccc2ncc(=O)[nH]c2c1 CC(O)C(F)(F)C(=O)N1CCOC(CN(C)C(c2cncs2)=O)C1 c1(C(N2CCN(C(C#CC(C)(C)O)=O)C(CCN(C)C)C2)=O)ccn2cccc2c1 N1(C(C(c2ccc(F)cc2)(C)F)=O)CCCC(CNC(c2cnsn2)=O)C1 c1(C(=O)NCC2(CO)CCCNC2)cnn2c1NCCC2C(F)(F)F N1(C(C2OCCN(C(C(CC)N(C)C)=O)CC2)=O)CCN(CC)C(C)(C)C1 N(C(=NCCCC(F)F)NCc1cc(C)ccc1Br)CCOCC Cc1nc(Br)sc1C(N1CCC(C)(C(F)(F)F)C1)C(=O)NCCC1CC1 C(=O)(C1=CCCC1)N1CCC(N2CCC(N(C)C(c3ccncn3)=O)CC2)C1 C1(NC(CCSCCCC)=O)CC(CNC(=O)CCCc2cncs2)C12CCC2 c1(C(=O)NC2C(NC(C(C)OCC)=O)CCCC2)cccn(C2CCC2)c1=O C#Cc1cc(F)c(C(N2CCC3(C2)CN(C(=O)C(C)(CC)CC=C)C3)=O)cc1F Cc1oc(CO)cc1C(N1CCCCC1C1CCN(C(=O)Cc2cccs2)C1)=O c1(CC(=O)N(C(C)CN(C(=O)CC2CCOC2=O)C)C)ccc2nc[nH]c2c1 C(=O)(C1CCCc2nncn21)NCC(CC(C)C)NC(CN1CC(C)C1)=O CN1CCn2nc(C(=O)NCC3(C)CC(F)(F)CN3C(c3cc[nH]n3)=O)cc2C1 c1(C(=O)NC(CNC(c2cc(C)c(C)nc2)=O)(C)C)cc(F)cc2c1NCCC2 N1(C(C(C)c2ccsc2)=O)CCN(C(=O)C=CSc2ccccc2)CC1C(F)F N1(C(C=CC)=O)CCN(C(=O)C(CC(=O)OC)N2CCCCC2)CCC1C N1(C(CC(C)(C)CNC(c2ccoc2Cl)=O)=O)C2CCC1CC(F)C2 c1(C2CCN(C(C(OCC)OCC)SC(C)(C)C)C2)cnn2ccccc12 N1(C(CC2CC(=C)C2)=O)CC2(CC2)CC1C(=O)NCC1(CO)CCN(C)C1 C=CCCC(C)(C)C(=O)N1CCC=C(C(=O)NC(c2snnc2C)C)C1 C1(CCC(N2C(C(N)=O)CC2)=O)CCN(C(C2CCC(F)(F)C2)=O)CC1 N1(C(=O)NCC(N(OC)C)=O)CCCc2cccc(F)c21 N1(C(c2nc(C)oc2)=O)CCC2(C1)CN(C(c1cc3cn[nH]c3cn1)=O)CCO2 Brc1cc2ncnc(NCc3scnc3-c3ccc(C4(C(F)(F)F)N=N4)cc3)c2s1 c1(C(=O)NCC2CN(C(c3ccc(OC)s3)=O)C(C)C2)c(F)ccc(O)c1F N1(CC2(NC(c3c(C)onc3)=O)CC2)CCN(C(C2CCC(F)C2)=O)CC1 N1(C(=O)NCC)CCC(C(=O)NCC(C)NC(C2OCCC2C(F)(F)F)=O)CC1 c1(C(N2CC(CC(N3CCOC4CC34)=O)C2)=O)cc(Br)cc2[nH]ccc12 CN1CC=C(CC(=O)N2CC3CCCC(C2)N3C(=O)Cc2ccc(O)nc2)CC1 c1(OC)cccc(Br)c1C(N1CC(CNC(=O)CCc2cc(C)no2)C1)=O CC(C)(CNC(c1sccc1Cl)=O)CNC(c1c[nH]nc1-c1ccccn1)=O c1(OC)cc(C(=O)NC(C2CCCN2C(=O)CCC2CC2(C)C)C)n(C)n1 C1(C(=O)NC(C2CCOCC2)C)CC=CCC1NC(c1[nH]nnc1C1CC1)=O C(CC)(CC)(CCNC(=O)C(C)C(F)F)NC(c1cccc(SCCCC)c1)=O C1(O)(C(CC)C(=O)NC2CCC2CNC(C2(C(=O)NC)CC2)=O)CCCCC1 c1(C(=O)NC(C(C)C)CCN(C)C(c2cccnc2Cl)=O)cccc2c[nH]nc12 CC(=NO)C1CC(C(N2CCCC(CNC(=O)Cc3csnn3)CC2)=O)C1(C)C c1(C(=O)NC(C2CN(C(=O)Cc3cnccn3)CCO2)C)nccc2cc[nH]c12 C1(CC=C)(C(=O)NCc2ccc(C)nc2)CCN(C(=O)C(C)OCCOC)C1 C1(C(=O)NC2CC3CC(NC(c4cnc(CC)[nH]4)=O)CC32)CCOC2(CCC2)C1 C(=O)(C(C)(C)C(F)F)N1CCC(C(CNC(C(C=C)OC)=O)C)CC1 C(=O)(CC(C)(C)C(F)F)NC1C(OC)CN(C(Cc2cc(OC)c(O)cc2)=O)C1 C1(CNC(c2ncc(OC)nc2)=O)CN(C(=O)C(C(C)O)NC(C)=O)CCCO1 c1(C(N2C3CC(NC(CCC#N)=O)CC2CC3)=O)ccc(F)c2occc12 N1(c2cc(NCc3scc(C)c3)nc(C)n2)CC(C)CC(C)(C)C1 C#Cc1ccc(Cl)c(NC(N2CCS(=O)C(C)C2)=O)c1 Cn1nc(Br)nc1C(c1nnnn1CC(F)F)NCc1cc(Br)no1 C1(O)(CNC(C2CC(C3CCC3)C2)=O)CCN(C(=O)C(F)CC2CCOC2)CC1 c1(C(N2C(C(N(C)Cc3c(C)occ3)=O)CCCC2)=O)ccc2cc[nH]c2n1 c1(NC(c2cncc(NCc3c(N)cccc3F)c2)=O)ccc2c(c1)OCCO2 c1(C(=O)NCC2(F)CCN(C(CC(=O)NCC)=O)C2)ccc(C)cc1SC N1(C(C(CC)CC2CCCC2)=O)CCN(C(=O)CC(C)(F)F)C(C(C)C)C1 c1(C(=O)OCC(=O)NCC(C#N)COCCC(=O)OC(C)(C)C)ccnc(O)c1 N1(C(COCCCOC)=O)CC2C(NC(=O)COCc3ccncc3)C2C1 c1(N(C)CC2N(C(CNS(CC)(=O)=O)=O)CCC2)cc(Cl)ncn1 CC#CCC(C(=O)N(C1CC(C)CC(C)C1)C)NC(C1CCCCC(=O)C1)=O CCCCC(CC)CC(C(=O)NCC)N1CCOC(CC)(CC)C1 Cc1ccc(NCC(=O)N(C(C)CCNC(=O)CC2CC(C(F)F)C2)C)cc1 Cc1cc(C)c(CC(=O)NCC(C)N(C)C(c2cnc3[nH]cnc3c2)=O)c(O)n1 C(C)(CCCCNC(=O)CCC(C)c1ccccc1)NC(CN1CC(CC)C1)=O N1(C(CCNC(C)=O)=O)CC2CCOC2(CNC(=O)C(C)(C)CC(F)F)C1 N1(C(COCc2cccc(C)c2)=O)CC2CCC1C(NC(c1ccnnc1)=O)C2 c1(OC)cccc(C(=O)NC(C)C(C)(C)NC(=O)CC2CC(F)(F)C2)n1 c1(C(N2CC(O)(CN(C)C(C3CC3(F)Cl)=O)C2)=O)ccccc1-c1cncnc1 N1(C(c2c(C)snc2)=O)CC(C)C(NC(c2cc(O)cs2)=O)C(C)C1 c1(C(=O)NC2CCC(NC(CC(C)(C)SC)=O)C2)cccn2c(O)nnc12 Cc1cc(C(=O)N(C2CCC(NC(=O)CCN(S(C)(=O)=O)C)C2)C)nn1C1CC1 CC1(C)CN(C(c2cc(Cl)c(F)c(Cl)c2)=O)CC(C)(C)C1NC(=O)C1=CCCS1 Cc1cc(C(=O)Nc2c[nH]nc2C(=O)Nc2ncc(Br)nc2I)cc(O)c1 C=CCC(CNC(C1CCSCC1)=O)NC(c1cc(C(F)(F)F)ns1)=O Cc1nc(O)[nH]c1C(=O)N(C(CNC(c1cc(O)nn1C)=O)C1CC1)C c1(C(=O)NC2C(NC(CCn3ccc(C)n3)=O)CC2)ccc2c(c1)C(=O)CCC2 C1(C(CCC)(C)C)CCCN1C(=O)CNC(C1(C(=O)C(C)n2cccn2)CC1)=O C1(NCc2n(C=C)nnc2)CCN(Cc2ccccc2)CC1C c1(CC)cc(C(=O)NC(Cn2cccn2)C(=O)N(CC(C)(C)C#N)C)no1 CCCCC(C(=O)N(CCOC)CC)NC(=O)C(C)N(C(=O)COC)C C(C(C)(O)CNC(=O)C(Cc1cn[nH]c1)NC(=O)CCCNC(C)=O)OC C1(C(=O)NC2CN(C(CCCCSC)=O)C2)CC(C)(C)CCO1 C#Cc1ccc(C(=O)NC2CCC2C(=O)N(C(CO)CO)CC)cc1C C=C(C)C(C)(C)C(=O)N1CCC(C=CC(N2CCC2C(N)=O)=O)CC1 N1(C(C2(C=C)CC2)=O)CCCC(C2CCN(C(=O)C3=CCC3)C2)C1 C1(NC(=O)NCc2n(CC)cnc2)CCc2nc(NC(C)(C)C)ncc2C1 N1(CC(=O)NCC2(CN(C(=O)C(N3CCCC3)C3CC3)C)CC2)CC(=O)N(C)C1=O N1(C(c2c(OC)cccc2C(F)F)=O)CC2CCCC2(CNC(C2CC(O)C2)=O)C1 C(C1=NOC2CN(C(C3CCOCC3)=O)CC12)NC(c1cc(C(F)(F)F)c[nH]1)=O CON=CC(=O)NC(CNC(C1CC1(F)F)=O)C1CC1 Cn1ncc(C(=O)NC2CCC(NC3CCC3)CC2)c1C(F)(F)F c1(C(=O)NC2(CNC(=O)C(F)n3cccn3)CCOC2)cccc(OC(F)F)c1 C(CCN=C(NC(C)CC)N1CCC(F)(c2cc(C)cc(F)c2)C1)=CC Cc1ccoc1S(=O)(=O)NCCCc1cccnc1 C(=O)(C(C)(O)CNC(=O)C(c1cnn(C)c1)NC(c1nnsc1C)=O)OC C(=O)(C(CC(F)(F)F)c1ccccc1)N1CC2C(COC(C)(C)C)C2C1 c1(CC(=O)NC(CC)(C)CNC(c2nc(Cl)sc2C)=O)c(C)cc(C)cc1C C1(CCCC)CCCN1C(=O)CNC(=O)CC.C12(CC1(C)C)C(=O)N2 c1(OC)cc(C(=O)NC2CCCCN(C(c3ccsc3)=O)C2)c([N+](=O)[O-])cc1F CON=C(C(=O)N1CCOCC(NC(=O)C(c2ccccn2)C)C1)c1ccco1 C1(NC(c2ccc(CC)[nH]2)=O)CCC(N(C)C(c2ns[nH]c2=O)=O)CC1 N1(C(c2cc(C)sc2C)=O)CC=C(C(C)(C)C(=O)N2CC(C3=NOCC3)C2)C1 c1(N2C(c3c(OC)cccc3)CCC2)ncnc2[nH]cnc12 c1(C(=O)NCCC(=O)NC2CC3CCCC3C2)ccc2ccccc2c1 C12(C(N3C(C4(NC(CCC#C)=O)CC4)CCC3)=O)CCC(N(C)C)(CC1)CC2 C1(CC(=O)NCCNC(c2ccc(C(C)(C)C)cc2)=O)Cn2ccnc2NC1=O c1(CC(N2C(CCCNC(C3CC=CCO3)=O)CCC2)=O)ccc(O)c(F)c1 c1(C(=O)NCCCN(C(CC(CC)CN(C)C)=O)CCO)cc2scc(C)c2[nH]1 C1(NC(c2c(C(C)C)n[nH]c2)=O)CC(C)CN(C(c2cn(C)nc2Br)=O)C1 c1(C(=O)NCC2CC(C(=O)NCCCn3cnnn3)C2)c[nH]c2ccccc12 c1(CC(=O)N(C2CN(C(=O)Cc3ccccc3)CC2O)C)nc([N+](=O)[O-])n[nH]1 C(=O)(CC1=CCOCC1)NC(CCCC)C(=O)NC(c1nccnc1C)C C1(NC(C(c2cccs2)SC)=O)CC(C)CN(C(=O)Cc2[nH]cnc2C)C1 c1(C(=O)NC2CC(CNC(C(C=C=C)C)=O)OCC2)ccc(Cl)cc1C N1(C(c2cc(C)[nH]n2)=O)CCC(C(=O)NCC(C2CCCC2)C)(C(C)C)C1 c1(OCC)cc(F)ccc1C(N1CC2CC2(CNCc2cncc(Cl)c2)C1)=O C1(C)(CC)CC(NC(c2cc(-c3ccoc3)on2)=O)CN1C(c1cccn1C)=O C1(NC(CN2CC(C)(OC)C2)=O)CN(C(=O)CCCN=[N+]=[N-])C2(CCCC2)C1 C1(CNC(C#CC(C)C)=O)(NC(=O)CN(C)S(N)(=O)=O)CC2CCC1CC2 C1(CC)(NC(=O)CCCCCCN)CCCN(Cc2nc(-c3cccs3)n[nH]2)C1 C1(CC)CCC(NC(=O)CCOCCN(C)C(c2cnc(Cl)s2)=O)CC1 c1(COCCOC)ccc(C(=O)N(C(C)CNC(C2(F)CCOC2)=O)C2CC2)o1 C1(NC(c2ccc(COC)o2)=O)CC2(CCCN(C(=O)COC3(C)CCC3)C2)C1 C12(CCNC(=NCCC)NC3CC3COC)CC3CC(CC(C3)C1)C2 CC(CC(=O)NC12CC(CNC(=O)C(O)Cc3ccccc3)(C1)C2)CC(C)(C)C C(=O)(C(F)CC(C)(C)C)Nc1cccc(C(=O)NCCN(CCN(C)C)CC)c1 c1(C(=O)NCC(F)(F)Cl)ccc(F)c(Br)c1F C1(C(=O)NC(C)CNC(=O)CCCCc2ccccc2)Cc2cccc(F)c2O1 c1(SC)nc(Cl)cc(=NCCC2CCN(C(c3cc(C)nc4ncnn34)=O)C2)[nH]1 C=CC1(C(=O)NCC2(F)CC(NC(=O)CC(C)(C)C3CC3)C2)CCOCC1 c1(C(N2CCC(C)(CNC(=O)C3=CCCC3)C2)=O)c[nH]c2cc([N+](=O)[O-])ccc12 c1(C(N2CC3(C(C(=O)Nc4nnc(C)n4C)C3)C2)=O)ccc2cncn2c1 C1(CNC(C(CC)C)=O)CC2CCC(C1)N2C(C1CCS1(=O)=O)=O C1(C)(C(=O)N(CCC2CC(C(NOCC=CC)=O)C2)C2CC2)CC=CC1 c1(CC(C)NC(C(CSC)OC)=O)ccc(CNC(C2(S(C)(=O)=O)CC2)=O)cc1 CN1CCCCC1C(=O)NC(C1CCCC1)CNC(=O)C(C)(C)c1nncn1C C(c1nc(C)co1)=CC(=O)N(CCCCN(C(CCCn1ncc(C)c1)=O)C)C Cc1noc2cc(C(N3CC(NC(=O)C(F)(F)C(F)(F)F)C4CC4C3)=O)ccc12 C(=O)(C(O)CC(F)F)N1CCC(N2CCN(C(C3(C(=O)NC)CC3)=O)CC2)CC1 C1(CNC(COC(CC)C)=O)CN(C(C2CCN(C(C)=O)C2)=O)CC1N(C)C C=CC(C)(O)CC(=O)NC(CO)C(C)NC(C1CCOC1)=O N1(C(c2cnc(CCCC)s2)=O)CC2(C1)CN(C(=O)CCOCCOC)C2 Nc1cc(C(=O)NCC2CCN(C(=O)CNc3ncccn3)C2)ccc1Br CC(C)(C)C(CNC(c1cc(Br)sn1)=O)NC(=O)CCc1ccoc1 CCC(C)(C)C(C)CC(=O)NC1CCCC(NC(=O)CCCOC)C1 c1(-c2n(CC(=C)C)nc(C(C)O)n2)cn2cc(C)nc2s1 c1(C(CCC)NC(=O)C(C)NC(N)=O)ccc(Cl)cc1 CCC(O)C(C)C(=O)NCC(C1CCCC1)NC(c1n[nH]cc1Br)=O N1(C(c2c(C(C)C)occ2)=O)CCC(F)C(NC(=O)C=C2CCCCC2)C1 CC(CC(F)F)C(=O)NCC1CC(F)CN1C(c1coc(CO)c1)=O c1(C(N2CCC(NC(CCOCCC)=O)C2(C)C)=O)cc(Cl)cc2c1CCC2 N1(C(CCNC(=O)OCC)=O)CCCC(NC(=O)C(C)(COC)OC)C1 C1(NC(CCC=CCC=C)=O)(CF)CCN(C(c2snnc2C2CC2)=O)C1 C1(CNC(C(CC)N(C)C)=O)CC2CCC1N(C(c1ccc(C#N)c(Cl)c1)=O)C2 N1(C(C2C(OC)C2)=O)CCC(CNC(c2ccc(NC(C)=O)cc2Cl)=O)CC1C CCC(CC(=O)NC(C1CC(NC(=O)C(C)SC)C1)C)SC C(C(C)(C)CC(F)F)Sc1ccc(OCc2ccc(COC)cc2)cc1 C1(CNC(c2c(C)nc(Br)o2)=O)CN(C(=O)OC(C)(C)C)C2(CCC2)C1 c1(C(N2CCCN(C(c3c(C)n(C)nc3)=O)CC2)=O)csc2ccccc12 Cc1[nH]c(CNCc2ccc(Br)nc2F)c(C)c1-c1ccc(OCC2CC2)cc1 c1(C(=O)NCCNC(c2n(-c3cn(C)nc3)cnc2)=O)cnn2ccncc12 C12(C(=O)NCCCCNC(=O)CSCc3ccccn3)CCCN1CCC2 N1(C(CCN(CC)CC)=O)CC(N(C)C(c2ccc(C)cn2)=O)C(O)C1 c1(C(=O)NCCCN(C(C2CCN(C)CC2)=O)C)c(O)ccc(Cl)c1F c1(N2C(C(C)(C)NC(Cn3c(C)nnn3)=O)CCC2)ccc(C(F)(F)F)cn1 c1(NCC2(C)CC3(CCC3)C2)ncc(S(=O)(=O)NCC(C)(O)C(F)(F)F)cc1Cl c1(C(=O)NC(CC(C)NC(c2n(CCC)ncc2)=O)C)cc(F)cc(F)c1 N1(C(C2C(C(C)NC(C3CCCCCC3)=O)C2(C)C)=O)CCC(CO)C(O)C1 N1(C(c2c(C)coc2)=O)CCC(C(=O)NC2CCCSCC2)CC1 C1(C(C)C)CCN1C(C(=O)NC1COC1)c1cccs1 N1(C(C=C(C)C(F)F)=O)CC(C2CCCN(C(=O)CCn3cc(Cl)cn3)C2)C1 CC1(C)CN(C(c2ccnc3ncsc23)=O)CCC1NC(c1cccc(Cl)c1)=O c1(C(N2CCC(C(C(=O)N(C3CCCC(CF)C3)C)F)C2)=O)cc2occc2[nH]1 C#CCC(CC#C)C(=O)NC1CN(C(C2CC(CC)=NO2)=O)C1 C=CC1(CC(=O)NC2CCC(O)C2)CN(C(=O)Cc2ccc(C)nc2)C1 c1(C(=O)NC2C(OC)CN(C(=O)COC(F)(F)F)C2)nc(Cl)ccc1N c1(OCC#C)cccc(C(N2CCC2C2CCOC2)=O)c1 c1(C(N2CCCN(CCNC(=O)CCCCCF)CC2)=O)cc2n(c1)CCCC2 CN1CC(C)(C)CC1C(N1CCCC(O)(CNC(=O)CC2(N(C)C)CCC2)C1)=O C1(CC)CC(C)(C)C12CCC2.c12ccncc1NC2c1nnnn1CCCOC c1(C(=O)NCC2C(CNC(C(Cc3cn(C)nc3)O)=O)C2)cc(O)nc(Cl)c1 C1(C(=O)NCCN(C(C(C)(C2CC2)OC)=O)C)CCC(CCC(C)C)CC1 C(CC(=O)Nn1cccn1)C1CCN(C(c2c(CC)ccs2)=O)C1 C1(CNC(CSCCN(CC)CC)=O)C(C)CCN1C(=O)CCC(=O)NC C1(C(C(=O)NCCSC)N2CCC2CC2CC2)CCC(C(C)C)CC1 CC1C(NC(=O)CC2CCCCCCC2)CCCN1Cc1ccsc1 c1(C(=O)Nc2nc(CC(=O)OC)c(C)s2)sc(S(N)(=O)=O)cc1C N(C(=NCc1ccnn1C)NCCNCC1(C)CCCOC1)C(C=C)C.CCOC C1(NC(C2C(COC)C2)=O)CCCCC1n1cc(CCn2c(C)nnc2S)nn1 N1(C(=O)Nc2cnc(Cl)cn2)CCN(C2CCN(C3CCC3)C2=O)CC(O)C1 c1(C(N(C2CC(NC(C(C)C#N)=O)C2)C)=O)ccnc(SCC(F)(F)F)c1 C1(CCNC(c2c(C)nco2)=O)CCN(C(=O)CCOCCN(C)C)CC1(F)F C1(NC(C(N2CCCCC2)C)=O)COCC1C(=O)NCCn1cnnc1 C1(CNC(C(C=C)OC)=O)CN(C(=O)Cc2cnn(C)c2)CC1(F)CO CCCC(C(=O)NCC1CCCCN1C(c1oc(C)nc1CC)=O)OCC C1(CNC(c2c(CC)nn[nH]2)=O)CCC(C)(C)CN1C(=O)C(C)C(C)C c1(CC(N2CC3CCC3(O)C2)=O)cc(I)cc(I)c1 c1(N2CCC(NC(c3ccn(CC)n3)=O)C23CCC3)nc2ccc(OC)nc2s1 CC(CO)(CO)C(=O)NCC1(O)CCCN(C(c2ccc(-c3ccccc3)o2)=O)C1 C=Cn1nccc1C(N1CCCC(C2CCCN2C(c2cnc(O)o2)=O)C1)=O C(=O)(CCCCC(=O)NCC1CCC2(CN(C(c3c(C)n[nH]c3C)=O)C2)O1)NC C=CCN=C(NCC1CC2CC1C2)N(C)Cc1ccc(F)cc1 N1(C(CCCNC(C)=O)=O)CC(NC(c2nccnc2N)=O)CC(C)C1 N1(CC(=O)N(C(CNC(C(C(C)C)O)=O)C2CC2)C)CCP(C)(=O)CC1 C12(C(=O)NC(CC#C)C(=O)NC)CC(CO)(CN1C(C1(C3CC3)CC1)=O)C2 CC1(C)CN(C2CC(NCCn3cc(-c4cnccc4OC)nn3)C2)CC(C)(C)O1 c1(C(=O)NC2C(NC(c3n[nH]c(C)c3C)=O)CC2)ccc2nsnc2c1 N1(C(=O)CC2CCN2C(=O)CC2CCCC2)CCCC2(CCC2)C1 C1(C(=O)NC(C=C)(C)C)CCCN(C(C2Cc3nccn3C2)=O)CC1 c1(C(N2CC(C(N3CCC(CCCO)CC3)=O)C2)=O)ncc(Cl)cc1Cl c1(COCC)nc(C(=O)NCC(C)(C)NC(C2CCN(CC(F)(F)F)C2)=O)co1 C1(CC(=O)Nc2c(C)nsc2)CCCN(C(=O)CC(C)C)C1 c1(C(=O)NC2CC(C)(NC(C3=C(C)OCCC3)=O)C2)ccc2c(c1)C(=O)N(C)C2 c1(C(N(CC)Cc2cc(C)on2)=O)cn2c(n1)CCN(CC1(CO)COC1)CC2 C(=O)(CS(=O)CCC(F)(F)F)NCC1CN(C(C2C(OC)(OC)CC2)=O)C1 N1(C(c2c(CC)ocn2)=O)CCCC2CN(c3cnc(C#N)c(C#N)n3)CCC12 C1(NC(C2C(CCC)CCC2)=O)CCCC12CN(C(=O)C(C1CCCC1)OC)C2 c1(C(=O)OC)cc(COC(c2cc(-c3ccccc3F)no2)=O)ccn1 N1(C(C2N(C(c3c(C)nco3)=O)CCOC2)=O)CCCC(C)(O)C1 c1(C(=O)NC(CCCNC(CC=C=C)=O)C)c(OC)ncnc1C Cc1occc1C(=O)NCC1CCCC1C(=O)NCC1CC1Cl C1(NC(C2(N(C)C)CC2)=O)CN(C(=O)CCn2cccc2)CC2(CCC2)C1 c1(C(=O)NCC(C2CC2)NC(c2cc(SC)oc2)=O)cncc(Cl)c1Cl N1(C(CCn2c(C)csc2=O)=O)CC2COCCC2(N)C1 C1(CC(=O)NCC(CCOC)NC(C2(C(C)C)CCCO2)=O)CCN(OC)CC1 Cc1ccc2nonc2c1C(=O)NC1(CO)CCN(C(C2CCOC2)=O)C1 C1(C(C)C)CN(C(=O)Cc2c(Cl)cccc2Cl)CCC1NC(=O)Cn1ccnn1 c1(C(N2CC(C(C)NC(C3CC3(F)F)=O)C2)=O)ccc(=O)n(Cn2cccn2)n1 N1(C(c2c(C(C)C)ncs2)=O)CCC(C(F)(F)F)C(CNC(C2(F)CC2)=O)C1 Cc1cccc(-n2cc(CNCCC3CCC4CC34)cn2)c1 CC1CCCCN1CCC(=O)N(C1CCCC1)CCNC(c1ccsc1Cl)=O c1(C(=O)OC)ccc(Br)cc1S(=O)(=O)N1CC(c2cccc(F)c2)C1 c1(C(=O)NCC(CC)NC(=O)CCCCO)noc2ccccc12 CCCC(CCCNC(C1(N2CCOCC2)CCCC1)=O)NC(C1CSC1)=O C(CC(C(=O)NCCc1ccccc1O)NC(C1COCCN1C)=O)SC N1(C(c2nn(C)c(F)c2)=O)CC(C2CN(C(C3CC3c3ccnn3C)=O)C2)C1 c1(C(N2C(CNC(=O)Cn3cccc3)CCCC2)=O)ccc(OC(F)F)c(F)c1 c1(C(C)C)c(C(=O)NC2CN(C(=O)Cc3ccns3)CC2F)cnn1C N1(C(C(CCC)F)=O)CCC(CNC(=O)C2=C(C)CC2)C12CC2 C1(CC(=O)NCCCC(C)O)CCN(C(C2CC2C2(C)COC2)=O)C1(C)C c1(CCC(=O)NCC(COC)NC(C2CCC(F)C2)=O)nc(C)no1 c1(OC)ccc(F)cc1C1CCCN1CCCS(=O)(=O)Nc1ccccc1 c1(OC)cccnc1C(N1CCOCC1c1cn(CCNC(C)=O)nn1)=O C(C(C(=O)NCC(O)CN(C)C)C(C)(C)C)NC(C(OC)OC)=O Cc1cccn2ncc(C(N3CCCC3C(=O)N(CCC(N)=O)C)=O)c12 N1(C(C(=O)NC(c2ccc(Cl)s2)CN(C)C)=O)CCC(NC(=O)CO)CC1 c1(C(N(C2CN(C(CC(COC)C)=O)CC23CC3)C)=O)ccc([N+](=O)[O-])n1C N1(CC(=O)N(c2cccnc2)Cc2ccnc(Cl)c2Cl)CCOCC(C2CC2)C1 C(=O)(C#CC1CCOCC1)N(CCCCC(=O)NCC1(O)CCCOC1)C c1(CNC(C23CC(C)C2C3)=O)cnn2c1CN(C(=O)CSc1n[nH]c(O)n1)CC2 C1(N(C(Cn2c(CCC)ncc2)=O)C)CN(C(C23CSCC2C3)=O)CC1(C)C c1(C(N2C(CCNC(CC3CC(C)(C)C3)=O)CCC2)=O)ccc2c(c1)COC2 CC(C)CCC(F)C(=O)N1CC(C(N2CC(S(C)=O)C2)=O)C(C)C1 c1(C(=O)NCCCC(C)NC(C=C(C)c2ccsc2)=O)cccc2nsnc12 N1(C(C=C2CCN(C)CC2)=O)CCN(C(C2(CO)CCCCC2)=O)CC1CF c1(C(N2CC(CC(N3CCOCC3C3CC3)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 C1(NC(c2ccc(Cl)nn2)=O)CCN(C(C2CC23CC(O)C3)=O)C12CCCC2 n1(CC(N2CC(CNC(c3c(COC)noc3)=O)C2)=O)cnc2ccc(C)cc12 N1(CCCNCC(c2ccccc2C)NC)CCN(CC(=O)OC)CC1 c12ccc(c(F)c1)C(=O)N(C)C2.C1(CCn2cc(COC)nn2)CCCC2CC12 C#CCC(C)(CC)C(=O)NC1CC1NC(=O)CCCC#CC C1(C(=O)NC(CC)(C)C)C2CC(CC2F)N1C(c1cccn2nccc12)=O C=CCCCCC(=O)NCc1n[nH]cc1C(=O)NC(c1ncn(C)n1)C c1(N2CC3NC(=O)OC3C2)nc(N2CC3CC2C2CC32)c2ccsc2n1 C(CCN=C(NCc1cncn1C)NCC(COC)COC)OCC C1(NC(CC2(CC)CC2)=O)C(C)CCN(C(=O)C(CC)n2ccnc2)C1C C1(CCNC(CCOCC(C)C)=O)CCCN(C(C2CCC3CC23)=O)C1 Cc1ccnnc1C(=O)N(CC(CO)(CO)NC(C1CCSC(C)C1)=O)C C1(C(=O)Nc2cnoc2)CCN(C(c2cccc(F)c2O)=O)CC1F N1(C(Cc2c(C)noc2C)=O)CCOCC(C(=O)NC(C)CCO)C1 C1C(CCCC)C(C)(C)CC(=O)N1C(CC)C N1(C(C(C)CF)=O)CCC(C2CCCN(C(C3CCC4CC4CC3)=O)C2)CC1 c1(NC(c2csc(NC(c3ccc(Br)nc3)=O)n2)=O)cccc2ncsc12 c1(C(=O)NCC(CC(=O)N(CCN(C)C)C(C)C)OC)ccc(=O)n(C)n1 c1(CC)ccccc1C(N1CCC1CNC(=O)C(C)(F)c1ccccc1)=O C1(NC(CCc2nnc(C(C)C)o2)=O)CCN(C(=O)CCS(C)(=O)=O)CC1F C(=O)(C(CNC(=O)CC(C)C)CC1CCCC1)NC1(CC=C)CC1 C(=O)(CCCN=[N+]=[N-])N1CC2C(CNC(COCc3n(C)ccn3)=O)C2C1 c1(C(N2C3(CCN(C(C=CCOC)=O)C3)CCC2)=O)ccnc2cc(F)cnc12 N1(C(Cc2c(C)nc[nH]2)=O)CC2CCOC2(CNC(=O)Cc2ccsc2)C1 C1(C(N2C3CN(C(C4(O)CCCCC4)=O)C(CC3)C2)=O)COc2ccccc2O1 CC(CN(C)C)C(=O)NC1(CCNC(C2CCC(C)O2)=O)CCCC1 C1(C(=O)NC(CC)C2CCC2)CC1C1CN(C(C2(C#N)CCOCC2)=O)C1 C(=O)(CC1=Cc2ccccc2C1)N(C)CCN(C)C(C1CCCCC(F)(F)C1)=O C1(OC)CCC(NC(C2(NC(c3nccn3C)=O)CCSC2)=O)CC1 C1(CNC(C2CC(=C3CC3)C2)=O)CCCN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC1 c1(C(=O)NC)ccc2c(c1)CN(C(C1(C#N)CCC1)=O)CC2 C1(C2CN(C(C3Cc4cscc4C3)=O)C2)(NC(c2cc(C3CC3)ns2)=O)CC1 c1(C(=O)NC(CCOC)CO)c(CNC(C2CCCN2C=O)=O)nnn1C c1(C(N2C3CN(C(=O)CCCCBr)CC32)=O)cccc2c1CCC2 c1(C(=O)NC(C)CCNC(C2(O)CC2)=O)cnc2c(=O)[nH]ccc2c1 C(=O)(C1CSc2ccccc21)NCCC1(O)CCN(C(C#CC(C)(C)C)=O)CC1 n1(CC)nc(C(=O)N(CCO)CC2(F)COC2)cc1C(N1CC2C(NC)C2C1)=O N1(C(C2(COC)CC=CC2)=O)CC2(CC(C(=O)Nc3cncc(F)c3)CO2)C1 C=CCCCC(C(=O)NCCC(F)(F)CO)NC(c1csc(Cl)n1)=O C1(C(=O)NCCOCCOCCNC(C(COC)C)=O)CCC2(CCC2)O1 N1(C(C(C)SCC)=O)CCC(NC(=O)C(C)OCCC(C)C)C1C c1(CCCNC(C(C)N(C(=O)CCc2nc[nH]n2)C2CC2)=O)ccccc1 C(=O)(CC(C)C(F)(F)F)N1CC(C(=O)C(C)=O)(S)C1.C#CCCC(O)CCN C(=O)(C(C)C(C)NC(=O)CC1CCCCC1)NCc1cn(C(C)C)nc1 C(CCCCC(=O)NC(C(=O)N(C)CCc1cccnc1)C1CCOC1)N(C)C C1(CC=C)(NC(C2CC(n3ccnn3)C2)=O)CCN(C(=O)C(C)SCCCC)CC1 N1(C(C23N(C(c4n(CCC)ncc4)=O)CCC2C3)=O)CC2(CCNC(=O)O2)C1 C1(C(=O)NCc2c(C)cncc2)CCCCCCN1C(C1CC1C#N)=O C=CC(C(=O)N(C)CCOCCNC(c1n[nH]cc1F)=O)c1ccccc1 c1(C(N2CCC(C(=O)NC(CC#C)C(N)=O)CC2)=O)ccc(C=C)cc1 C1(NC(CC=CCC)=O)CN(C(=O)CC(C)F)C2(CCCCCC2)C1 N1(C(c2c(C)cco2)=O)CCC2CCN(C(=O)CCCc3cccnc3)CC2C1 OC1CC2(CCN(c3ncnc(N4CCOCC4)n3)CC2)C1 C12(CNC(C(C)NS(C)(=O)=O)=O)CN(C(c3ccc(N)cc3F)=O)CC1CCO2 c1(CC)cc(OCC(=O)NC2(C)CCN(C(=O)CC=C(C)C)C2)ccc1Cl CC1C(=O)CCC1CC(N1CCC(CN(C(=O)C(C2(O)CCCC2)F)C)CC1)=O Cc1ccc(CC(=O)NCC2CCN(C(=O)CN(c3ccccc3)C)CC2)cc1 Cc1nc(C)c(CC(=O)NCC2C=CC(NC(=O)Cc3cncc(F)c3)C2)s1 c1(C(N2CC(C)C(NC(c3cc(C4CCC4)on3)=O)C2)=O)cc2sccc2cn1 C(=O)(N1CC2COCC2O1)C1N(C(C(C(C)C)O)=O)CCCC1(C)C Cn1cc(NC(=O)CC2CNC(C)(C)C2)c(O)nc1=O C(=O)(N=c1ncn(Cc2cccc(F)c2)[nH]1)c1ccc(OCC)cc1 c1(C(N2C3C(C(=O)O)C(C3)C2)=O)ccc(S(N)(=O)=O)c(N)c1 C(=O)(CN=c1ccnc(NC(C)Cn2ccnc2)[nH]1)NCCC N1(C(CC(C)N(C(c2nc(CC)sc2)=O)C)=O)CC2CC(C1)C2(C)C c1(C(=O)NC(C2CCN(C(CC(n3c(CC)ncc3)C)=O)C2)C)cc(C)c(C)[nH]1 C1(C(=O)NC2(CF)CCN(C(c3cccc(Cl)c3F)=O)C2)C2CCC(F)(F)C12 c1(C(=O)NC2(C)CCN(C(=O)CN3CCCCCC3)C2)ccnc2c1CC(=O)N2 c1(C(N2CCC3CCN(C(CC(C)SC)=O)C3C2)=O)cc2ncccc2cc1Cl N1(C(c2c(OC)nn(C)c2)=O)C(C)C2CC1C2NC(=O)CCc1nc(C)c(C)[nH]1 C1(C(N2C(CN(C(=O)CS(C)(=O)=O)C)CCCC2)=O)CC(C)(C)CC(C)(C)C1 C1(CNC(CCC2(C)N(C(CSCCC(C)C)=O)CCC2)=O)CC2CC1CC2O N1(C(CCC=CC)=O)CCC(CCO)(CO)C1 C(C(C(=O)N(CCCO)C1CC1)C(C)(C)C)NC(C1C(C)(CC)C1)=O C(CN=c1[nH]c(=NC2COC(N(C)CC)C2)[nH]c2cccnc12)SC C1(CNC(C(CC)(C)C)=O)CCC2(CCC2)C1NC(c1ccc2occc2n1)=O C1(C(N(CC(F)(F)F)C)=O)CC2CCC1N(C(=O)CNC(=S)NCC(C)(C)C)C2 C1(CC(C(=O)NCCCSC)N(CC(C)C(=O)OC)C)CCCCN1C(C)=O c1(C(=O)NC2CN(C(c3cnn4ccsc34)=O)CCC2O)nc2cnccc2s1 c1(C(N(C(C)CNC(c2ncc[nH]2)=O)CC)=O)cc(C(N)=O)co1 CCC(CCC(=O)N1C(CO)CC1C)NC(c1ccncc1)=O C1(NC(C2CC2(Cl)Cl)=O)CC2CC1N(C(c1ccn(CCF)n1)=O)C2 c1(CC)c(C(=O)NC(CN(C)C(c2cnco2)=O)(CO)CO)cccc1C C(=O)(CCCC(CC)CC)N1CCC(C#C)(C(N2CC(CCO)C2)=O)CC1 C1(CNC(CCC#CC)=O)CCCCCN1C(=O)CNC(=O)Nc1ccccc1 C1(C(=O)NC(CSC)C)CC(C)(C)CN1C(C1CNC(=O)N1)=O C1(C(=O)NCC(CN(C(CCOCC)=O)C)C)CCCCC1C(C)(C)C C1(COC)CN(C(=O)C(SC)SC)CCN1C(c1nc(=N)cc[nH]1)=O C1(C(=O)NCc2cn(C3CN(C(c4ccns4)=O)C3)nn2)CC2CCC1O2 CC1(C)COCC1CC(=O)NCC1CC1NC(c1snc(O)c1Cl)=O C1(NC(CC2(COC)CC2)=O)CC2CC(OC)C2C1.N12CCC(CO)C(C1)C2=O c1(C(N)=O)cc(C(=O)NCC(CO)NC(c2cc(-c3ccco3)c[nH]2)=O)co1 N1(C(c2c(I)ccc(C)c2)=O)CCc2cc(-c3ccnc(C)c3)ccc2C1 c1(C(=O)NC2CC(CNC(CN3CC(C)C3)=O)C2)csc(C(F)(F)F)n1 N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)COCP(C)(C)=O)CC1CC(F)F c1(OC)ccc(-n2nnnc2C(c2occc2Br)NCC(C)CC2CC2)c(C)c1 N1(C(c2c(=N)[nH][nH]c2)=O)CCC2(CCC2)C(NC(C2CCCC(F)(F)C2)=O)C1 c1(C(=O)NCC2=CCN(C(c3c(C)nc(N)cn3)=O)CC2)cccc2nn[nH]c12 N1(C(CC=C=C)=O)CCCC2CN(C(C3(OCC)CCSCC3)=O)CCC12 Cc1cnnc(O)c1C(N1CC2(C(=O)N(C(C)C(C)C)C3CC3)CC1CO2)=O C1(COC)C=CCCN1C(C1(NC(=O)CN(C(=O)COC)C)CC(F)C1)=O S(=O)(=O)(c1cc(C(=O)N=c2ccn(C3CC3(F)F)[nH]2)ccc1Cl)NC(=O)C1CC1 CC(C(=O)NC(C1CC1C(=O)NC(c1ccccc1)(C)C)C)C(F)(F)F c1(CC)ccc(C(=O)NC2CC(C)N(C(=O)CCC(C)CN(C)C)C2)c(C)c1 NC(=O)CCCCC(=O)NC(Cc1cn[nH]c1)C(=O)NCC(O)CNC(N)=O CCC(C(=O)NC(C(=O)NC(C)CCN(C)C)C(C)(C)C)C(C)(C)CC CC(C)(C(=O)NCC(CNC(C1CC2C=CC1C2)=O)C(F)(F)F)C1=CCSCC1 N1(C(COCCCC#C)=O)CC(CNC(=O)C(C=C)c2ccccc2)CC1(C)C C1(O)(C(C)C)CCCN(C(=O)CC2COCCN2C(c2ccncc2N)=O)C1 CCC(CC(=O)NCCC(O)C(C)C)N(C(=O)C(c1ccn(C)c1)C)C c1(NC(=O)OCC)ccc(C(=O)N(C(C)CNC(=O)CSCCCCCC)C)s1 C(CC1c2ccccc2CCN1C(C1CCCCC1)=O)NC(=O)CO C1(NC(C(F)=CCC)=O)CCCC(N(C)C(c2ccc(CF)cc2)=O)C1 CC1(C)CCc2onc(C(=O)NCCC3CN(C(=O)C=Cc4ccsc4)C3)c2C1 Cc1sc(C(N2CCC(C)(NC(c3cc4occc4[nH]3)=O)C2)=O)c(C)c1C CN1CCCC1C(=O)NCCOCCNC(C1CC1[N+](=O)[O-])=O C1(N(C(=O)CSCC(=O)Nc2cccnc2)C)CCCN(C(C2CCCS2)=O)C1 C1(C(=O)NC2CC2)(CC)CCCN1C(c1cn(C)nc1C)=O C(C)(C)(CC(F)C(=O)N1CCN(C(C)C)CC1)NC(C(C(COC)C)C)=O C1(n2cc(COC3N(C(c4c(C)nns4)=O)CCC3)nn2)CCCNC1=O N1(C(c2ccc(C)c(O)n2)=O)CCC(C)(C)C(CNC(C2(Cl)CC2(F)F)=O)C1 N1(C(c2cccc(C#C)c2)=O)CC2CC(C1)CN(C(c1cnn3ccsc13)=O)C2 N1(C(c2ccn(C)c2)=O)CC2CCN(C(c3cc(F)cc(Cl)c3)=O)CC2C1 n1(CC(=O)NCC(CNC(C2(CC)CCC2)=O)(C)C)nnc2c1CCCC2 Cc1ccc(C(N2CC=CC2CNC(C2(C)CCC(=O)N(C)C2)=O)=O)c(N)c1C N1(C(C2CCC(C)(C)C2)=O)CCOC(C)(CNC(=O)Cc2csnn2)C1 C1(N(C(=O)CCCF)C)CC2CCC(C1)N2C(=O)CCc1nc(=N)[nH][nH]1 c1(C(N2CC(OC)(CNC(=O)CNC(=O)CN(C)C)C2)=O)ccc(Cl)cn1 N1(C(c2c(C)cn(C)c2)=O)CC2CCN(C(c3cnc4[nH]ccc4n3)=O)CC12 C1(C(=O)NCC=CCC(=O)N(C)Cc2c(C)cncc2)CCOC(=O)CC1 CCC(C)(COC)C(=O)N(CC(C)(C)NC(c1nccn1C)=O)C Cc1cc(C)c(C(=O)NC2CCN(C(c3ccc(F)c(N)c3)=O)CC2F)c(O)n1 N1(C(CCC=C)=O)CC(C)CCC1C(=O)Nc1cccc(C(C)=O)c1 c1(C(C(=O)NCC(=C)C)N(C2CCC2)CC)cnn2c1CCC2 c1(C(N2CCC(NC(C=CC)=O)C2c2ccccc2)=O)ccc(C2CC2)cc1F c1(C(N(CCOCCO)CC)=O)occc1CNC(=O)C(C)C1CCC1 Cc1cc(C(=O)NC2CC(O)CN(C(c3ccnc(C4CC4)n3)=O)C2)cc(C)n1 Cc1cc(C(=O)NC2CCN(C(C3CCC(=O)N3)=O)CC2CO)c(N)c(Cl)n1 N1(C(c2nc(COC)oc2)=O)CCC(C(=O)NC2(C(=O)OC)CC2)C1(C)C C(N=c1cc(NCc2nc(-c3ccc(Cl)cc3)n[nH]2)nc[nH]1)c1n(CC)cnc1 c1(CC(N2CC(NC(CCC3CC(OC)C3)=O)C(O)C2)=O)ccc(F)c(C)c1 C1(C(=O)NCCC2CC(NC(C3CCCSC3)=O)C2)CCn2cncc2C1 CC1=C(C(=O)NCC2CC(C)N(C(c3cnccn3)=O)C2)CCCC1 O=C1Cc2cc(C(=O)Nc3ccc(N4CCC(O)CC4)cc3)ccc2N1 C12(CNC(CC3(C)CC3)=O)CCC(CC1)N(C(c1cn(C3CCOC3)nn1)=O)C2 CC1=C(C)CC(C)(C(=O)NCC2CN(C(C3CCCCC(=O)N3)=O)CCO2)CC1 C1(NC(C(C)OCC(C)C)=O)(CO)CCCN(C(c2ncsc2C(F)(F)F)=O)C1 Cc1nn(C)c(N)c1C(=O)NC1C=CC(C(N2CCCC(C(N)=O)C2)=O)C1 C(=O)(CS(=O)(=O)CC(C)C)N(CC(C)NC(C1CCC(C)=C(C)C1)=O)CC N1(C(CCc2n[nH]c(=N)s2)=O)CCCCC(CNC(=O)C(c2ccccc2)O)C1 c1(CSC)noc(CCC(=O)N(CC(C)(C)NC(=O)CCc2csc(=N)[nH]2)C)n1 Cc1c(C(N2CC(O)(C(F)C(=O)N3CCC3CC3CC3)C2)=O)cccc1F C(=O)(C(O)C(C)(C)C)N(CCCNC(=O)CC1CCCOCC1)CCC N1(C(CC)=O)CC2CS(=O)(=O)CC2(CNC(C2CC2CN(C)C)=O)C1 c1(C(N2CC(NC(=O)C(O)c3ccco3)C3(C2)CC3)=O)cccc2nc(O)[nH]c12 C1(C(=O)NCC2N(C(C3CC(=C)C3)=O)CCC2)CCN(c2cnn(C)c2)C1=O C1(O)(CNC(C2C(CC(C)(C)C)C2)=O)CN(C(C2CC3CC3C2)=O)C1 C1(CNC(Cc2c(C)ocn2)=O)C(O)C(O)CN1C(c1cncc(Br)c1)=O n1(C(=O)NCCCN(C(C)C)CCC2CCC2)cc(Cl)cn1 c1(CC23CN(CC(=O)NCC4CC(F)(F)C4)C(CC2)CC3)cccc2[nH]ccc12 C(=O)(C1=CCC(C)(C)CC1)NCC1N(C(CCCCCSC)=O)C2(CC1)CC2 c1(NC(N2C(CC#C)CCC2)=O)cc(-c2ccsc2)nn1-c1ccc(C)cc1 Cc1c[nH]c2cc(C(=O)NC3CCN(Cc4c(F)cccc4I)CC3F)ccc12 C1(C(N(C2CCCN(C(C(F)=C(C)C)=O)C2)CCO)=O)CCc2c[nH]nc2C1 C1(O)(CN(C(CN2CC(C)C2)=O)C)CCN(C(C2C3COCC23)=O)C1 c1(C(=O)NCC2CCN(C(C(C(C)O)N(C)C)=O)C2)c[nH]nc1S(N)(=O)=O CCCCCCCCCC(=O)NC12CC1CN(C(C1CN=C3N=CNN3C1)=O)C2 C12(C(=O)NC3(CCC)CCC3)CC(CO1)N(C(C1CCCCN1CC)=O)C2 CC1CCC=C1C(=O)NCCCOCCOCCNC(c1cc(Cl)cnc1O)=O C1(NC(c2c(C)coc2C2CC2)=O)CN(C(C2CC23CC3)=O)C2(CCCCC2)C1 CC(C)(C(=O)N1CC2CC2(CNC(c2c[nH]c(C(F)(F)F)c2)=O)C1)C(N)=O C1(C)(NC(COCC#C)=O)CCN(C(C2CC2c2ccccc2)=O)C1 C=CC(CCC)CC(=O)NC(CNC(c1ccc(CC)[nH]1)=O)CC(C)C c1(C(N2CCCC(NC(C(CCC)O)=O)C2)=O)ccc2sc3ccccc3c2c1 c1(N(CC(C)C#N)C(N2CCC(c3ccc(C)cc3)(C)C2)=O)cccc(Cl)c1C c1(NCC(CC)(C)COC)ncnc(N2CCN(C3CN(C)C3)CC2)c1C C1(CCC(=O)NC(C(=O)NC(C)C)C)CCC(NC(=O)C(C)N(C)C)C1 c1(C(N2CC(C(C)NC(c3n(C=C)nnc3)=O)OCC2)=O)ncn2ccccc12 c1(OCC)ccc(C(=O)NC2CSCCN2C(=O)C(O)CC)cc1[N+](=O)[O-] Nc1c(C(N2CCNC(C(F)(F)F)C2)=O)ccc(F)c1Br Cc1ccc(C(=O)NCC2C3CN(C(c4nc(Cl)cs4)=O)CC23)c(F)c1F Cc1ccc(NC(=O)CCN2CCCC2c2ncc(-c3ccc(C)cc3)[nH]2)cc1 N1(C(c2cc(CC)on2)=O)CCCN(C(=O)C(N2CCCC2CC)=O)CCC1 C(=O)(CCC(C(N)=O)NC(N1CCCC(C)(CC#N)C1)=O)OC(C)(C)C C1(C(=O)NCCCNC(c2cc(CC)cc(F)c2)=O)C2CCC(C2)C1(C)C c1(NC(c2c(C3CC3)ccc(OC)c2)=O)cccc(S(C)=O)c1 C1(O)(C(=O)NC2C(NC(C3(C)CC4CCC3O4)=O)CCC2)CC2(CCOCC2)C1 C1(C(N2CCC(C(N)=O)(NC(c3ccc(C4CC4)o3)=O)C2)=O)CCCCC(=O)N1 c1(C(=O)NCCN(C(C(CC(N)=O)O)=O)CC2CC2)cnc2c(c1)NC(=O)CN2 C(=O)(CCCCCC(C)C)NC(CC#C)(C)C(=O)N(C)CC1CCN(C)C1 n1(CC(=O)NCC2CCC(NC(C3(C(C)C)CC3)=O)C2)ccc2cc(F)ccc12 C1(C(N(CC(CC)NC(c2cnn(CC)c2C)=O)C)=O)C=CC=CC=C1 C1(C)(CN2CC(C)N(c3ccccc3)CC2)Cc2ccccc2C1 c1(C(=O)OC)c(NC(C2CC(F)CN(Cc3ccc(=O)oc3)C2)=O)cccc1Cl C(=O)(CC1=CCCCC1)N1C(C2(NC(C(c3cccc(C)c3)C)=O)CC2)CCC1 c1(C(=O)NC(CC)CNC(=O)CN2CCOCC2=O)ccc(NC(C)=O)cc1Cl C12(CNC(c3c(SCC)cccn3)=O)CCC(CN1C(=O)CCn1ccnc1)C2 O=C1CCCCC(C(N2CC(O)CC2C(N2CCCC(O)C2)=O)=O)N1 c1(CC(N2CCC(F)(CNC(COC(C)C)=O)C2)=O)c(F)cc(F)cc1F Cc1ccc2c(C(N3CC4CN(C(=O)CC5CCN(C)C5)CCC34)=O)onc2c1 C1(NC(c2ccc(CSCC)cc2)=O)CCCN(C(c2conc2C)=O)CC1F N1(C(c2c(CC)occ2)=O)CC2CCN(C(c3ccc(C(F)F)cc3F)=O)CC12 CCCCCC(O)CC(=O)NC(C1(C(=O)OCC)CCCC1)C c1(OC)ccc(F)cc1-c1nc(C(=O)Nc2cc(C3CCCCC3)no2)cs1 C(=O)(CC(F)(F)CC(=O)OC)N1CCN(C(c2ccn(CC)n2)=O)CC1CCO C1(N(C(C=CC=CC)=O)C)CCCN(C(c2cncn2C(C)C)=O)C1 C(N=c1[nH]c(Cl)ncc1Cl)C1CCN(C(C2ON=C(C)C2)=O)CC1C c1(NC(C(C)N(C(CC#C)C(=O)OCC)C)=O)cccc2ccoc12 Cc1ccc2c(c1)CCC2(C)C(=O)Nc1cncnc1O C1(NC(=O)CCn2cc(CNC3CCC3)nn2)CC(O)C(O)CO1 c1(C(=O)NC2CCC2)cccnc1CNC(C1CCCCC1F)=O CCC(C)(C(=O)NC1CN(C(=O)COCC2CCCC2)C1)OC C1(CNC(C2(NC(C)C)CC2)=O)CC(NC(=O)C=CBr)C1(C)C c1(CC(=O)NC2CC(NC(c3cccc4nncn34)=O)C2)ccc2c(c1)COC2 c1(C(=O)NCC(C(C)(C)C)NC(C2=CC(C)(C)C2)=O)cc([N+](=O)[O-])c(F)cc1N c1(CNc2ccc(-c3c(C#N)nccc3)nc2)c(Cl)ccc(F)c1F C1(CNC(C(C)=CC2CC2)=O)CC2(CCC2)CN1C(c1ccc(F)c(N)c1F)=O C=Cc1ccc(C(=O)NC2CN(C(C3CC4(CC(=O)N4)C3)=O)CCC2C)cc1 CC1=CC(C)=NS(=O)(=O)N1CC(=O)NCC(O)CNC(=O)C(C#N)C(C)(C)C c1(C(=O)NC(CNC(c2cccc(NCC)c2)=O)C)cn2c(n1)CC(OC)CC2 n1(CCC(=O)NC2CCN(C(c3c(C)nns3)=O)C23CC3)ccc2ccccc12 c1(C(=O)NCC2CC(NC(COCC)=O)C2)ccc(F)cc1OC N1(C(c2c(C)cns2)=O)CCC(NC(=O)Cc2ccc(Cl)nc2)CC1C N1(C(C=C2CCN(C)C2)=O)CCOC2(C1)CN(C(=O)CCn1cnnn1)C2 N#Cc1c(N2CCC(CCNC(=O)CC3CCOCC3)C2)cccc1F N1(C(CNC(CCC)=O)=O)CCCC1CCNC(C1(N2CCCC2)CCC1)=O Cc1ccnc(C)c1C(=O)NCC1CCCC(NC(c2cnsc2)=O)C1 C(C(O)CC(F)(F)F)NC(CC1CCCC(NC(c2cn(C(C)C)nn2)=O)C1)=O N1(C(CC(CC)C)=O)CCCC2C1CCN2C(=O)CCCCCl C(=O)(N=c1[nH]n(C)cc1P(C)(C)=O)NC1C(CC)CN(S(=O)(=O)C(C)C)CC1 Cc1csc2c(C(=O)NC(C)CC(C)NC(C3(C#N)CCSCC3)=O)ncnc12 N1(C(C2C(CC)CN(C(=O)C=Cc3ccoc3)C2)=O)CCCSCC1C c1(C(=O)NCCC(CNC(c2csc(Cl)n2)=O)O)c[nH]c(=O)c2ccnn12 C1(CC)CN(C(=O)C(C)CC(C)C)CCC1CNC(c1cn(CC)nn1)=O C1(NC(C(C)c2cc[nH]n2)=O)CC2(C1)CC(C(=O)N(C1CC1)CC1CC1)C2 S(=O)(=O)(c1ccc(C)c(C)c1)N(CC(N1CCCC(C(N(CC)CC)=O)C1)=O)CC C(c1ccccc1)(C(F)(F)F)=CC(=O)NC(C1CCCC1)Cc1ccc(Cl)cc1 c1(OC)cnnc(C(N2CCC(CCC(=O)N(CCN=[N+]=[N-])C)CC2)=O)c1 C#CC1CN(C(C2CCC(NC(=O)CC(C)c3ccco3)C2)=O)CC1OC C(=O)(CCCC(=O)N1CCCC(C(=O)N2CCCCO2)CC1)OC C1(CNC(c2c(OC)csc2)=O)CC(NC(=O)C=C(C)Cl)C1(C)C Cc1ccc(C)c(C(N2CC(CNC(=O)Cc3csc(Cl)n3)CCC2C)=O)n1 c1(CC(=O)NC(CNC(C2C(C)CCC2)=O)C2CC2)ccc(Br)c(Cl)c1 C1(NC(CC(C)SC)=O)CC2(C1)CC(NC(=O)Cc1c(Cl)cccc1Cl)C2 c1(CN(C2CCN(C(c3c(C)nc(Br)s3)=O)C2)C)ccc(S(C)(=O)=O)cc1 c1(C(N2CC(O)(CNC(c3n[nH]cc3Cl)=O)C2)=O)ccc(Cc2nc[nH]n2)cc1 N1(C(c2ccc(C(CC)=O)cc2)=O)CCC2C(NC(c3ncn(C)n3)=O)C2CC1 c1(C(=O)NC(CC(=O)NCCCN(C(C)CCO)C)=O)cc(Cl)c(Cl)n1C N1(C(CN(C(CCC)=O)Cc2ncc(Br)s2)=O)CCCC1C(C)(C)CN1CCC1 N1(C(C)=O)CC(O)CC1C(N1CC2(NC(=O)CSc3ccccc3)CC1C2)=O C1(C(=O)NC2(CC)CC2)CNC(=O)CN1C(=O)CC1CC2CC2C1 Cc1nn(C)c(NC(C2CCCN2C(c2ccsc2C)=O)=O)c1C(N)=O N1(C(c2cc(OC)c(Br)s2)=O)CCC(C)(CCc2cn(C3CCOC3)nn2)CC1 c1(CN2CCCC2)cn(CC2(NC(=O)CNC(C3CCOCC3)=O)CC(O)C2)nn1 CC(Cc1ccccn1)C(=O)N1CCCC1CNCC(=O)OCC12CNCC1C2 N1(C(C(C=CCCC)O)=O)C2CCC1CN(C(c1cccc(CC#N)c1)=O)C2 C(CNC(c1cnn(C2CCC2)n1)=O)(C(C)(C)C)NC(CCC1C(C)C1)=O C1(C(N2CC(OC)C(NC(c3cc[nH]c3C3CC3)=O)C2)=O)CC(=O)NC(=O)N1 C(=O)(C1CCc2c(Cl)cccc21)N1CC(O)(CNC(C(C(C)(C)F)(C)F)=O)C1 c1(C2(C(=O)NC3CCC(CCNC(c4cc(Cl)no4)=O)C3)CC2)cccnc1Cl C1(F)(C(=O)NC2CCN(C(Cn3c(C)c(Cl)cn3)=O)C2)CCC2(CCC2)C1 C1(CNC(CC(C)SC)=O)CC(C)(C)CN1C(c1coc(N(C)C)n1)=O C1(N(C2(CN(C)C)CC2)C(C2(SC)CC2)=O)CCCOC1 C(C(=O)N1CC=CC(NC(=O)C(C)NC2(CO)CCCC2)C1)(C(C)(C)C)OC c1(CNC(=NCC(=C)C)NC(C)C)cc(OC)c(C(C)=O)cc1C N1(C(c2cc(OC)ns2)=O)CCC2CN(C(=O)CCCCCC(C)C)CCC12 N1(C(c2cc(C)c(C)o2)=O)CCCOC(CNC(=O)Cc2cc(F)cc(Cl)c2)C1 C1(C2N(C(CN(C(C)=O)C)=O)CCC2)CCCN(C(c2ccnn2C)=O)C1 C(=O)(C1CCc2snnc21)N1C(CNC(=O)C2=CCCOCC2)COCC1 c1(C(=O)OC)coc(C(=O)NCC(C)(C)NC(=O)C(C)c2ccon2)c1 C(=O)(C1=CC2CC=CCC12)NCCC1(NC(c2c(CCC)nco2)=O)CC1 c1(C(N2CC(N(C(=O)C=CC3CCOC3)C)C2)=O)cc(-c2cccnc2)n(C)n1 CC1CN(C(c2cc[nH]c2C2CCCC2)=O)CCC1NC(c1ccnc(Cl)c1Cl)=O N#CCCCCCC(=O)N1CC(F)CC1CNC(=O)C=Cc1cccc(Cl)c1 c1(C(=O)NC2C(NC(C3N(C(C)C)C(=O)CC3)=O)CCC2)ccccc1[N+](=O)[O-] C1(C(N2CC(CCC#C)C2)=O)COC(CNC(=O)C(C)CN(C)C)C1 C(=O)(CCCCC(F)F)N1C2CC(CNC(=O)C3=CCCCO3)(OC2)C1 Cc1ccc(NC(N2CC(NS(=O)(=O)Cc3cccc(Cl)c3O)C2)=O)cc1C N1(c2snc(SC)n2)CCOCC12COCCN(C(c1cc[nH]n1)=O)C2 CC(C)C(C#N)C(=O)N1CCC(NC(=O)COc2ccsn2)CC1C c1(C(=O)NC(CN(C(c2cc(C(C)C)ccc2F)=O)CC)C)cnc(N)c(N)c1 C=CC(CC)CC(=O)NC1CCN(C(c2ncsc2C)=O)CC1CC N1(C(COC)=O)CCC(O)(CCNC(=O)C(C)(C)C(N)=O)CC1 CC1COCCC1N(C(=O)CC1CCCC1NC(=O)CC1(O)CCC1)C C(=O)(C(C(=O)NCC1CN(C(c2ccc(C(F)F)s2)=O)CC1O)OC)OC N1(C(CCCn2c(C)ncc2)=O)CCN(C(=O)CC2(C(F)(F)F)CC2)C(C)C1C S(=O)(=O)(c1cccnc1NCC1(CO)CC1)N(CCCC=C)C CC(C(=O)NC(CCF)C(=O)NC(CCO)C1CCCC1)C(F)(F)F N1(C(C(=O)NCCOC)=O)CC2(CC1CNC(c1occ(C)c1C)=O)CC2(F)F C1(N(C(C2CC3(CC3)C2)=O)CCF)CCCN(C(c2csc(C(F)F)c2)=O)C1 N1(C(C2(CC)CCCC2)=O)CC2(CNC(=O)CCc3cncc(F)c3)CC1CO2 CC#CCCC(=O)N(CCNC(=O)Cc1cc(C)sc1C)Cc1ccccc1 N1(C(COc2cn(C)nc2)=O)CC2CC(NC(C3CC4COCC4C3)=O)C1C2 Cc1nn(C)cc1C1=NOC(C(=O)NC2CCN(C(=O)Cn3cccc3)CC2)C1 c1(C(=O)NC2C(NC(CN(C3CC3)CC)=O)COCC2)ccc2c(c1)CC(C)O2 Cc1oc(C(C)C)nc1C(=O)NCCC(N1CCC(CC(N)=O)C1)=O C=CC1CN(C(=O)CN(C)C(C)C)CC1NC(c1ccc(-n2cccc2)nc1)=O C1(CC(=O)NCC(=O)NC)(OC)CN(C(=O)C(CC)n2cncn2)C1 C1(CNC(C2CCC3(CCC3)O2)=O)CCN(C(c2csc3nnsc23)=O)C12CC2 CCC(C(=O)NC1(C(=O)N(C(CC)C2CC2)C)CCCC1)n1ccnc1 C(CC(F)F)(C(=O)NCCCCC)NC(C(C=C)C)=O C12(CNC(C(N)=O)=O)CN(C(c3ccc4cnoc4c3)=O)CC1CCO2 C1(NC(CC(n2ccc(C)n2)C)=O)CCN(c2snc(C)c2C#N)CC(C)(C)C1 C1(NC(CCCCN(C)C)=O)CCN(C(=O)Cn2cc(C3CC3)nn2)CC1F C1(NC(C(C)CSc2ccccc2)=O)CC2CC1CN(C(C1CC1F)=O)C2 c1(CCCC(=O)NC(CN(C)C(C2CC3CCC3C2)=O)(C)C)ccc(Cl)cc1 C1(NC(C2CCN(C(=O)NCC(F)(F)F)C2)=O)C2CCN1CC2 C(C(C(C)C)NC(=O)C(Cc1ccco1)NC(=O)COCCF)OC c1(NC)ccc(C(=O)NCC(C)(CNC(C2CC(n3cccn3)C2)=O)OC)nc1 CCCCCCCC(=O)N1CCCCC(NC(=O)CN2CCOCC2)CC1 c1(OCC)ccccc1OCC(=O)NCC1CCN(C(c2nn(C)cc2Cl)=O)C1 C1(NC(c2c(C)cc[nH]2)=O)CCCC(NC(C2(C)CCNC2=O)=O)C1 c1(C(=O)NC2CCN(C(c3cc(C)ncc3)=O)C(C)C2)c[nH]nc1S(N)(=O)=O c1(C(=O)NCC(C)(C2CC2)NC(C2N(CC)CCC2)=O)cc(N)c(F)cn1 N12CCN(C)CC1C(=O)OCC(O)C2.C(CN(C)C)OCC C(=O)(CC(C(F)(F)F)NC(=O)CCCCN(C)C)N1CCC(C(C)CC#N)CC1 c1(C(=O)NCC(CNC(C2N(C(C(C)C)=O)CCC2)=O)C)cnn2ncccc12 C(=O)(CS(=O)(=O)C(C)(C)C)N(CC(C)O)CCNC(=O)CN1CCCCS1(=O)=O C1(O)(c2cn(CCC=C)nn2)CCN(C(C2COC(C)(C)CO2)=O)CC1 c1(C(=O)NCC2CN(C(C(C)SC)=O)CC(C)(C)C2)ccc(S(C)(=O)=O)cc1Cl C1(NC(c2cc(OC)ncc2F)=O)COC2(C1)CN(C(c1ccc[nH]1)=O)C2 N1(C(CSC(C)=O)=O)CC2C(C(=O)NCc3ccc(OCC(F)(F)F)cc3)C2C1 c1(C(=O)NCC2C(NC(c3c(C)onc3)=O)CCC2)c(C)nc2ccnn2c1C C(=O)(CCC(C)(C)C(=O)N1CCC(C)C(CNC(C2(CF)CCC2)=O)C1)OC Cc1ccc(C(N2CC(N(C)C(C3CC34CCC4)=O)C2)=O)nc1 c1(OC)cccc(NC(=O)C(c2ccc(Cl)nc2)N(C2(C)CCC2)C)c1 C12(C(N(CCN(C(=O)CC3CC(C)(C)CO3)C(C)C)C)=O)CCC(CC1)C2 CCC(CNC(=O)C(C)CNC(C1OCCOC1C)=O)(CC)OC CC1CC(CCNC(c2cc(O)cc(Cl)c2)=O)CCN1C(=O)Cn1cnnn1 N1(C(c2onc(C)n2)C)CCC(NC(C2(C)CCCC2C)=O)C(C)(C)C1 C(=O)(CCCC(C)(F)F)NC1CC(CNC(C(CC)O)=O)C1 O=C1COc2cc(C(=O)NC3CCN(C(c4ccc(Cl)nc4O)=O)C3)ncc2N1 C=CCCC(C(=O)NCC(C)(C)CC(F)F)NC(C1CC(C)CC(=O)N1)=O C1(CN(C(C2CCCOCC2)=O)CC)CCN(C(=O)C#CC(=O)N(C)C)CC1 C1(NC(c2nc(COC)oc2)=O)CC2CC1CC2C(N1CCCC(C#N)C1)=O C1(C(=O)NCCN(C(=O)C(c2c(C)noc2C)CC)CCC)CCOC(C)(C)C1 Cc1nn2c(c1C(=O)OC(C)(C)C)CNCC2.C12(CCCOC1)C(=O)NC2 N1(C(C2OCCN(C)C2)=O)CCN(C(=O)CCC(N)=O)C2COCC12 C(=O)(C(c1cccs1)NC(=O)C(=O)NCCNCC1CC1)OC C12(CNC(c3cc(NC(C)=O)c(F)cc3)=O)CCC(CC1)CN2C(C1CC1F)=O N1(C(C(C)=C2CCC2)=O)CCCC1(C)CNC(c1ccnc(C(N)=O)c1)=O C(C(C)(C)CC(=O)NC1C=CCCC1C(=O)NC1CN(C)CC12CC2)OC N1(C(CCC#CC)=O)CC2CCCC2(NC(c2cc(OC)ns2)=O)C1 C1(NC(c2c(C)ccs2)=O)CC(O)CN(C(=O)CC2CCC2)C1 C(C1=CCCOC1)NC(C(C)(C)C1CCN(C(C2CC2C(N)=O)=O)C1)=O c1(CC)ccoc1C(=O)NC(c1cn(C)nn1)C(=O)NCCC1(C)CCCO1 c1(CC)cc(C(=O)NC(C(=O)NCCc2nccc(C)n2)C2(O)CCC2)c(C)o1 c1(CC)ccc(CSC(C)C)cc1.C1(CO)C(C)NC(=O)C2(CC2)C(=O)N1 N1(C(CCC)=O)CC(CNC(=O)C(C)Sc2ccccc2)CC(C)(C)C1 CC1C(C)N(C(=O)CN(C)S(=O)(=O)N(C)C)CCN1C(C1CC(O)C1)=O CCC(C)(C)C(=O)C(=O)NCC(C(=O)NCCN1CCNC1=O)N(C)C c1(C(=O)NC(CCCNC(c2cn(C)nc2Cl)=O)(C)C)coc2cc(O)ccc12 CC1CCCC(OCC(=O)NC2(NC(=O)CN3CCC(=O)CC3)CCCCC2)C1 N1(C(C=CC=CCC)=O)CCC2(CCCN2c2ncc([N+](=O)[O-])cc2F)C1 c1(OC)ccc(C(=O)O)c(C(F)(F)F)c1.c12ccc(cc1)CC(=O)N1CCC2C1 N1(C(C(C2CCC2)OCC)=O)CCC(C(C)(C)NC(=O)C(C)n2ccnc2)CC1 c1(OC(C)C)cc(C(N2CCC(CNC(C3CCC(C)S3)=O)CC2)=O)ccn1 CC(C)(C(F)(F)F)OCC(=O)NCC1CC1NC(=O)CCc1cccc(Cl)c1 c1(C(=O)NC2CCN(C(C)=O)CC(O)C2)cc(Br)c2nccnc2c1 CC(C)CC(CC(C)C)C(=O)NC1C2CCN(C(=O)C(C)N3CCC3)CC12 N1(C(CC2(OCC)CC2)=O)CCCCCC1C(=O)Nc1cc(C)cc(Cl)c1 Cc1cc(CNC(c2nnnn2CCCC2CC2)c2cn[nH]c2)cnc1O C1(C(=O)NC2CCCC(NC(C3(C)CCCS3)=O)C2)(OCC)CCCCCC1 c1(C(N2CC=CC(NC(C3C(C=C(C)C)C3(C)C)=O)C2)=O)ccccc1N=[N+]=[N-] c1(C(=O)NC2CN(C(C3CCCCO3)=O)CC2O)cc2ccccn2c1 c1(SC)cncc(C(=O)NC(CO)CCCNC(c2cnn(C)c2)=O)c1 Cc1ncc(CNC(=O)COCCNC(=O)COc2cnn(C)c2)n1C Cc1cccc(C)c1C(O)C(=O)NC1CN(C(=O)CCc2cnco2)CC1C C1(N(C(=O)C(CC2CC2)OC)CC#C)CCN(C(=O)Cc2ccc(O)nc2)CC1 C=CC(C(F)(F)F)NC(C1CC(O)CN1C(=O)CCC1CC1(F)F)=O N1(C(C=CC(CC)=CC)=O)CCN(C(c2cc(C)n(C)n2)=O)CC1CC(F)F c1(OC)cc(C)cc(CN2CC(CC(=O)Nc3ccnc(F)c3F)C2)c1O Cc1cc(O)ccc1N(C(=O)CC1CCN1C(=O)C(F)OC(F)(F)F)C1CC1 c1(C(N2CC(CNC(C(C(=O)OC)C)=O)C2)=O)csc2ccc(F)cc12 c1(NC(C2NCCN(C(c3c(C)ncnc3)=O)C2)=O)nn(C)c2ncc(I)cc12 c1(C(=O)NCC(CNC(C(C=C)O)=O)F)sc2cccc(F)c2c1COCC c1(C(N2CC(C)CC(NC(c3c(OC)csc3)=O)C2)=O)ccc2c[nH]nc2c1 c1(Oc2c(Cl)ccc(C)c2)ccc(C#N)cc1Cl C(=O)(C1CCCn2ncnc21)NC1CN(C(c2c(C)scc2)=O)C(C)CC1 Cc1ccn(C)c1C(N1CCC(NC(c2ccc(OC3CCOC3)cc2)=O)C1)=O CC#CCC(C(=O)N1CCCC(C(=O)OC)C1)NC(=O)C(C(=O)OC)OC N1(C(c2c(CC)n(C)nc2)=O)CCCC(N(C)C(c2occc2C)=O)CC1 C(=O)(CCN=c1ccc(C)c[nH]1)NCC(CC)NC(c1cccc(Cl)c1C)=O N1(C(c2cc(C)cc(C)c2N)=O)CCN(C(=O)CCOCC2CC2)CC2(CC2)C1 C1(NC(C(CSCC)NC(C2C(OCC)CC2)=O)=O)CC2C=CC1C2 C1(NC(COC(CC)C)=O)CCCCCC1NC(c1nc[nH]c1C(C)(C)C)=O c1(C(=O)NC(CC)(CNC(=O)CCCn2ccnc2)CC)ccc2ccnn2c1 c1(CC(=O)NCC(CC)NC(=O)CCc2ccccc2O)ccc(C)cc1Cl N12CCC(CC1)C2=O.c1(C(=O)NCC2(C(=O)NCCO)CC2)cc(Cl)ccn1 C1(NC(C(COCC)NC(c2n(C=C)nnc2)=O)=O)CCn2cnnc2C1 C(C(=O)NCCOC1CN(C(=O)C(c2ccccc2)O)C1)(C(C)C)NC(=O)OC CC1CN(C(=O)CC23COC(C)(C2)C3)CC(C)N(C(=O)CC(O)C(C)(C)C)C1 N1(C(CCN(C)CCO)=O)CCC2(CC1)CC2CNC(=O)C=CCO C1C(=O)N=C2C=C(N(C)N2)O1.C1(N(CCC)C=O)CCN(CC(C)C)C1.OCC c1(OCCC(=O)NC2CN(C(C(C)=C(CC)C)=O)CC2C)ccc(C)c(C)c1 C#Cc1cn(C)nc1C(=O)N(CCCCCNC(c1cn(C)nn1)=O)C(C)C CC1(O)CCN(CC(N2CC=CC(NC(=O)CCN3CCCS3(=O)=O)C2)=O)C1 N1(C(C(C)Oc2ccccc2)=O)CC(CN(C(=O)Cn2nccn2)CCl)C(F)(F)C1 CCN(Cc1ccc(OC)c(OC)c1)N1CC2CC2(C(=O)OC)C1 C1(CNC(C(C)(C)OCC)=O)CCC2CN(C(c3cc(C)ns3)=O)CC12 c1(C(N(C(CCNC(c2ccc(OC)cc2F)=O)C)C)=O)ccn2ccccc12 C1(CNC(C(CCCC)C)=O)CCN(C(=O)CCSCC(N)=O)CCC1(F)F C1(C(=O)NC(C2(O)CCN(C(=O)CN3CCOC3=O)C2)C)CC2(C1)CC2F c1(C(N2CCOCC2c2ccc(Cl)cc2)C(=O)NCCCC)cc(C)ccc1F CC(C)C(CO)ONC(=O)C1CC1C(C)NC(=O)C=CC1CCC1 c1(C(=O)OC)c(NC(=O)Cc2ccc(SCC(F)(F)F)cc2)oc2c1COCC2 C1(C(C)(C)F)CCN(C(c2cc(Br)sc2Cl)=O)CC1 N1(C(CCN(C(c2ncccc2N)=O)CC)=O)CCN(C)CC1C C1(C(N(CC(C)CNC(c2cn(C)c(C(F)F)n2)=O)C)=O)CC(C(C)(C)C)=NO1 CC1CN(C(C2CCSCC2)=O)CCC1CNC(c1ccccc1C(F)(F)F)=O Cc1cc(CNC(=O)CC2CCSCC2)oc1C S(=O)(=O)(CC(=O)NCCCN(C(=O)C(C)NS(C)(=O)=O)C)NC C1(C(=O)NCC2CC(NC(C=CC(C)C)=O)CC2O)Cc2c(F)cccc2O1 Cc1nc(CC(=O)NC2CC(NC(=O)CCS(C)=O)C2)c(C)s1 N1(C(C=C(C)C)=O)CCCC2CN(C(C3COc4ccccc4C3)=O)CC12 C(CC(=O)N1CC2(CC(N(C)C)C2)C1)(C(F)F)NC(C(CC#C)O)=O C1(C(=O)NC2CN(C(c3nc(Cl)c(Cl)s3)=O)CC2O)CC2COCC2C1 c1(C(C)C)cccc(CN2CCCC(OC3CCOCC3)C2)n1 Cn1nnc(=NS(=O)(=O)c2cccc(NC(=O)NCC(O)C(F)(F)F)c2)[nH]1 Cc1ncc(Cl)cc1NC(=O)NC1CCCCC1(C)C C1(CNC(C(C)(C)F)=O)C2CCC(C2)N1C(c1ccc(Cl)c(O)c1)=O C1(C(=O)NC2CCCC2c2ccc(C(F)(F)F)cc2)CCC(C=CCO)C1 C1(N(C(=O)CC2CC(=O)C2)CC)CCN(C(C2(SC)CC2)=O)C1 C1(NC(C)CCCCNC(=O)OC(C)(C)C)CCNC(=O)CC1 C1(C(=O)NCC(c2ccccc2)N(C(=O)CN2CC=CC2)C)CCCNC(=O)C1 c1(C(N2CC(CCCCNC(c3c(CC)ccs3)=O)C2)=O)cnc2scnc2c1 C1(OC)(CNC(C2CNC(=O)C2)=O)CCN(C(=O)Cn2ccnc2C)C1 C1(NC(Cc2c(C)noc2)=O)CCCN(C(=O)Cn2cnnc2)CC1 C#Cc1ccccc1CNC(=O)C(C)N(C(C1CN2CCN1CC2)=O)CC C1(NC(CCCC#C)=O)CN(C(C2CCCC(C)(C)O2)=O)CC2(CCOCC2)C1 CC(C)C(C(C)NC(c1cn(-c2ccccc2)nn1)=O)NC(=O)C(N)=O C1(NC(COCCOCC#C)=O)CCCC12CCN(C(C13CC(C)C1C3)=O)CC2 Cc1nc(CC(=O)NC2(CNC(c3cc(N4CCOCC4)ccn3)=O)CC2)c(C)s1 c1(C(=O)NC(CNC(CC(COC)C)=O)C2CCC2)cccc(N)c1O N1(C(CCSCC)=O)CCCC(O)(CNC(C2CC2C)=O)C1 CCCC(C(=O)N(C(C)CC(=O)OCC)C)NC(c1nc(O)sc1C)=O N1(C(C2N(C)CCOC2)=O)CC(NC(c2ncnc(O)c2Cl)=O)CC(C)(C)C1 c1(C(C)NC2CC(NC(C3(F)CC3C)=O)C2)nsc2cc(Br)ccc12 c1(OCCC)ccc(Cl)cc1CC(=O)OCc1nnnn1-c1cc(F)ncc1C C#Cc1cc(F)c(C(N2CCC(NC(c3ccsc3Cl)=O)C(C)C2)=O)cc1F c1(OCF)cccc(CNCc2ccsc2C(F)(F)F)c1 C12(NC(CC=C(C)C)=O)COCCC1CN(C(c1cn(C)nn1)=O)C2 N1(C(C(=O)NCCOCCCC)=O)CCC(C)(NC(=O)C2=COCC2)C1 c1(OC)ncnc(N2CCCC(CO)(NC(C3CCCC3O)=O)C2)c1OC N1(C(C2C(C=C(C)C)C2(C)C)=O)CCN(C(c2ccsc2C)=O)C2(CCC2)C1 N(C(=NCC1CCCN1Cc1cnccn1)NC1CCCC1)C1CCN(CC)C1 C1(NC(=O)C=C2CCCCC2)CCC2CC1CN2C(c1cnc(S)[nH]1)=O c1(C(=O)NCCCNC(=O)CCCCCc2cccs2)nnn2c1CSCC2 C#Cc1ccc(Cl)c(C(=O)NCCN(C(=O)C(O)CC(C)(C)C)CCOC)c1 c1(C(=O)NCC2C(NC(CCSc3nc(C)[nH]n3)=O)CCC2)n[nH]c(C)c1F Cc1ncnc2c1CC(C(N1CCN(C(=O)CP(C)(C)=O)C(CO)C1)=O)CC2 N1(Cc2c(OC)cco2)CCc2c(C(=O)Nc3ccc(C)s3)n[nH]c2C1 C(CCCCCNC(c1cnc(Br)s1)=O)NC(C1(CC#C)CCCO1)=O Cc1ccc(-c2n[nH]c(SCC(=O)NC(CCNC(=O)CC(C)(C)F)C)n2)cc1 c1(CN2C(CC(=O)Nc3cc(C)c(Br)cc3F)COCC2)ccc(O)c(C#N)c1 c1(C(=O)NC(CCC)CCCNC(=O)CS(N)(=O)=O)cc(F)c(C)cc1F C1(CNC(CC(CNC(c2nn(C)c(Cl)c2)=O)O)=O)CCCOC1(C)C CCCC(CCCNC(c1c[nH]nc1CC)=O)NC(C1ON=C(C)C1C)=O Cc1cccc(-c2cn(C3CC(C(=O)OCCCF)C3)nn2)c1N(C)C N1(C(C2N(C(C)C)C(=O)CC2)=O)CC2CCN(C(c3cc(Br)n[nH]3)=O)C2C1 CCCC(CC)C(=O)NC(C)(CNC(C1(CF)CC1)=O)CC(C)C N1(C(C(C)SCC)=O)CCCN(C(=O)COCc2ccc(C)cc2)CC1C(C)C N1(C(CC)=O)CCCC(C2CN(C(=O)CNc3ccc(C)cc3)C2)C1 C1(CCNC(C(C2CN(C(=O)CCc3nccn3C)C2)OC)=O)OCCC1(C)C c1(C(=O)NC2CC(CNC(CC3CCC(=O)C3)=O)C2)ccc2ncsc2c1 c1(C(=O)NCC(C2CCOC2)NC(c2n(CC#C)ccc2)=O)csc(C)c1C c1(C(N2CCC(C(C)(C)NC(C3CCCSC3)=O)C2)=O)cc2cccc(F)c2s1 c1(C(N2C(C(C)NC(=O)C=C3CCC3)CCC2)=O)cncc2[nH]ccc12 c1(C(=O)NCC2CC(NC(COCCOCC#C)=O)C2)ccc([N+](=O)[O-])c(O)c1 c1(C(N2CC3CC3(CNC(C34CCCC3OCC4)=O)C2)=O)n[nH]c2c1COC2 C1(C(N(C)CC2(O)CCN(C(CCC(CC)C)=O)CC2)=O)Cc2ccncc2N1 N1(C(c2c(C)n(C)cc2)=O)CCOC2(C1)CN(C(c1cccc3c1OCC3)=O)C2 CCCCC(CN=c1[nH]cc([N+](=O)[O-])cc1CO)NC(c1nc(C)c(C)s1)=O N1(C(C(COC)O)=O)CCC2CN(C(c3cncs3)=O)CC2C1 C(=O)(NNc1cc(C(=O)NC)ccc1Br)C1N(C(=O)OC(C)(C)C)CCC1 C(C(O)CN=C(NCC1(O)CCCC1)NC(C)C1CC1)c1cccc(C)n1 CC[Si]1(CC)CCN(C(c2cncn2-c2ccccc2C(F)(F)F)=O)CC1 c1(NCC2(CNC(CN(C(=O)CC(C)(C)C)C)=O)CC2)ccccc1OC(F)F C1(C(N2CCC(C(C)NC(C3CC3F)=O)C2)=O)CCC(=O)N1C1CC1 N(C(=NCc1ccnc(OCc2ccco2)c1)NC1CCC(=O)NC1)C(CC)C C1(NC(=O)COC2CN(C(c3n[nH]cc3C3CC3)=O)C2)CCCCCCC1 C1(NC(C(N2CC(C)C2)C)=O)CN(C(=O)CC2CC3(COC3)C2)CC1S(C)(=O)=O N1(C(C2=NOC(C)(C)C2)=O)CC(NC(c2cn(C3CC3)nn2)=O)CC12CCCC2 CC(C)(C)C1=NOC(C)(C(=O)NC2CC3CCC2(NC(=O)COC2CCC2)C3)C1 N1(C(c2c(F)ccc(C)c2)=O)CCOCC(C)(CNC(C2C3CCOCC23)=O)C1 CCC(CC)(C(=O)N1CCC(O)C(C(N2CCCCC2CO)=O)C1)C(=O)O n1(CC(=O)NCC(CNC(C=CC(=O)OCC)=O)CO)ncc(Cl)c1C c1(CC(=O)NC2(CF)CCN(C(c3cc(Cl)no3)=O)C2)ccc2c[nH]nc2c1 C1(NC(CCC#C)=O)CCN(C(c2ccc(OC)cc2OC)=O)C12CCC2 CN1CC(C)(C)CC1C(N1CC(O)CC1CNC(C1(CC2CC2)CC1)=O)=O N1(C(c2c(OC)noc2C2CC2)=O)CCc2sc(CNC(=O)COC)nc2C1 C1(NC(C(CC)N(C)C)=O)CCC2CN(C(c3cnc(C(C)C)[nH]3)=O)CCC2C1 CC(C)CS(=O)(=O)CC(=O)N(C1CCN(C(c2c[nH]c3cc(F)ccc23)=O)C1)C c1(C(=O)NCC2(NC(C3C(OC)C3)=O)CCCC2)[nH]c2ccc(F)cc2c1C n1(C(C)C)ncc(C(N2CCCC2C(C)NC(C2(C(F)(F)F)CCC2)=O)=O)c1N c1(CC(=O)NC23CC(NC(=O)CC4CCC5(CCC5)O4)(C2)C3)cc(F)cc(Cl)c1 c1(C(=O)NCC(C)(C)CNC(c2cc(N)c(F)cn2)=O)cc2ncccn2n1 c1(C(N(C2CCN(C(=O)CCn3ccnn3)C2)CC#C)=O)csc(CO)n1 C12(NC(CCOCCC)=O)CCN(C(c3cncc(N(C)C)c3)=O)CC1C2 c1(C(=O)NC(C(C)NC(c2ccc(F)cn2)=O)CO)cc(N)nc(Br)c1 C1(CCCC)CN(C(C2CC(C3CC3)=NO2)=O)CCN1C(c1sc(C)cc1Cl)=O c1cnc(-c2nc(Cc3cnc(-c4ccccc4)s3)no2)c(-n2cccn2)c1 C(=O)(CCS(N)(=O)=O)N(C)CC1(CNC(C2N(C(C)=O)CC(F)C2)=O)CC1 Cc1[nH]c(=N)[nH]c(=NCCC2CC(C)(C)NC2=O)c1C C(CC(=O)OC1CCC1C1CC1)(C(F)(F)F)OC C(=O)(C1=CCCOC1)NC1CCN(C(c2c(C(C)C)ncnc2)=O)C1 C1(C(=O)NCC=CCNC(c2cccc(CC)n2)=O)CCC=CCCC1 C(=O)(C1=NOC(C)C1)N(C(C)C)CCN(C(=O)CCN1C(=O)CCC1=O)C CC(C)CC(CNC(c1cn(CC(F)(F)F)nn1)=O)NC(=O)C(F)C(C)C c1(C(=O)NCC2CCN(C(C(CC)C)=O)CC2O)cc(F)c(F)cc1F C#Cc1cc(C(=O)NC2CCCCC2NC(c2cn(C)nc2C)=O)cc(Cl)c1 N#CCCCCCC(=O)N1CCC2(NC(c3[nH]cc4c3CCC4)=O)CC2C1 c1(C(=O)NC2CCN(C(Cc3cc(CC)no3)=O)C(C)C2)ccc2ccsc2c1 c1(C(N2CC(C(C)NC(C3C(C=C)C3)=O)C2)=O)cc(OC)cc(Br)c1N CC1CCN(C(c2cn(CCO)nn2)=O)C1CNC(c1ncoc1C(F)(F)F)=O CC1(C)OCCC1(O)C(N1CC(C(=O)NCCN2CC3CCC2C3)C(F)(F)C1)=O CC(C)CC(C)C(=O)N1CCCC(CCNC(=O)Cc2ccn(C)n2)C1 c1(C(=O)NCC(CCNC(c2cn3ccsc3n2)=O)O)ccnc2ccncc12 C(=O)(CC1=CCN(C)CC1)N1C(C)CCN(C(=O)CC2(C)CCOC2)CC1 c1(OC)cc(C(=O)N(C)CCNC(C2CSCN2C(=O)C(C)(C)C)=O)ccc1F C1(NC(c2ccc(C(C)=O)o2)=O)CN(C(c2c[nH]cc2C(C)(C)C)=O)CC1(C)C C(=O)(C(O)CC(N)=O)NCC1(O)CC(CNC(c2cnn(C)c2C(F)(F)F)=O)C1 C(=O)(C1CCc2cccc(F)c21)NC1(C)CCCN(C(c2c(C)csc2)=O)C1 c1(CC(C)C)nccc(C(=O)NCC2(C)CCN(C(C3(F)CCOC3C)=O)C2)n1 N1(S(CCNC(=O)CCc2ccc(F)cc2)(=O)=O)CCN(C(C)C)C(C)C1 N1(C(=O)CC2CCOCC2)CC2CCN(C(c3cn(CCCF)nn3)=O)CC2C1 c1(C(N2C(CCC(=O)Nc3c(C)nc(Cl)s3)CCC2)=O)c(Br)cc(Br)c(C)c1Br C(C(C)(C)CC(=O)NCCc1c[nH]nc1O)NC(C(C)c1cc[nH]n1)=O c1(C(=O)NCC2C(NC(CN(C)CC)=O)C2)ccc(F)c(OCC2CC2)c1F C1(OC2(CNC(C3(C(=O)OCC)CCC3)=O)CC2)COC(C(=O)ONC(C)=O)CO1 C1(C(=O)NC(CC=C)CO)CCC2(CN(Cc3c(F)cc(OC)cc3F)C2)O1 C1(O)(CNC(=O)CC2CC2)CC(C(=O)NC2CC(N(C)C)C2)C1 N1(C(C2N(C)C(=O)OC2)=O)CCOCC(C(=O)NCC2CCCS2)C1 c1(C(C)=O)ccc(OCC(N2CCN(c3cccc(O)n3)CC2)=O)c(Cl)c1 c1(CC(=O)Nc2c(C)nn(CC(=O)OC)c2C)ccc2c(cnn2C)c1 CCC(C)C(C)C(=O)NC1(C)CC(NC(=O)CCc2nc(-c3cccs3)no2)C1 c1(OCC)cnccc1C(N1CCC(NC(C2CC3CC3N2C(C)=O)=O)C1)=O Cc1cc(C)c(C(N2CC(NC(=O)CC3CCC(F)(F)C3)C(C)C2)=O)c(=O)o1 Cc1nnc2n1C(C(=O)NCCC1CCN(C(C3CCS(=O)(=O)N3)=O)CC1)CC2 c1(CCNC(C2C(NC(=O)Cc3cncn3C(F)(F)F)C2)=O)cccc(Cl)c1 C(C1CCN(C(C2CC3CC3C2)=O)CC1)=CC(=O)N(C1(C)CC1)C c1(SC(C)C)ccc(C=CC(=O)Nc2cc(C(F)(F)F)ccc2C)cc1 n1(CCCSC)nnnc1C(C1CCOCC1)NC(C1(n2cc(Br)cn2)CC1)C CC1CN(C(c2ccc(-c3cnccn3)cn2)=O)CC1NC(c1cncs1)=O N1(C(c2c(C)cns2)=O)CCC2CN(C(C3CCN(CC(C)C)C3)=O)CC12 c1(C(CCC(=O)NCC(O)CNC(=O)CC2C=CCC2)C2CCCC2)ccccc1 CCC(C)C(C(=O)NCc1cncc(OC)n1)NC(=O)CCC(C)(C)F Cc1cc(F)cnc1C(N1CCCCC1CCC(C)(C)NC(=O)C(C)O)=O C1(C(N(C(C#C)C)C)=O)(C(N2CCC2)=O)CN(Cc2ccccc2)C1 C1(CNC(C2(SCC)CC2)=O)CN(C(C2CCNC2=O)=O)C2CCCCC12 CN1C(=O)C(=O)N(CC(=O)NCC2C=CC(NC(C3(C)CCCC3)=O)C2)C1=O C(=O)(CCCCC(N)=O)N1CC(C(N2CCC(O)(CN(C)C)C2)=O)(CC)C1 c1(CN(c2ccc(F)cc2)CC2C(C)(O)CCCC2)cc(F)c(Cl)cc1F C1(C(N(C)CC2COCCN2C(c2ccnc(S)c2)=O)=O)CCCCC2(CC2)C1 Cc1nc2ccccn2c1CC(=O)NCC1C2CN(C(=O)CN(C)C(N)=O)CC12 CC1C(NC(c2ccnc(Cl)c2)=O)CC2CCC1N2C(c1nc(F)ccc1Cl)=O C1(CC)CC(C(=O)NC2CCC(CCC(=O)Nc3ccc(SC)cc3)C2)CCO1 C(C(O)CNC1C2CCCC12)(OCC)OCC N1(C(c2cc(-c3ccco3)no2)=O)CCC2CCN(C(=O)C3=CCCCO3)C2C1 C1(C(=O)NC(C(N2CCCC(CCF)C2)=O)C2CCOC2)CC2CC1CC2O c1(C(N2CCC(C)=C(C)C2)C(=O)NCc2cccc(OC)c2)ccn2nccc2c1 C1(CC(=O)NCCC(C)NC(c2cc(C3CCCN3C)[nH]n2)=O)COC(C)(C)C1 c1(CSCC(=O)NCCC(C)N(C)C(c2ccccc2)=O)csc(=N)[nH]1 C(=O)(CC(C)CC(C)C)NC1(CNC(C2CCCN(C(CC)=O)C2)=O)CCCC1 c1(C(=O)NC(CNC(c2ccc[n+]([O-])c2)=O)C2CC2)cccc2c1COCC2 C(CCS(C)(=O)=O)(C(=O)NCC1CCCCN1C(C1(SC)CCC1)=O)OC C=CCCCC(C(=O)NCC12CC(CN1C)C2)NC(=O)Cn1ccc(C)n1 C1(NC(COCCCC)=O)CCC2CN(C(C3CCCN3C(C)=O)=O)CC2C1 CC1CCN(CCC(=O)NCC(C)NC(=O)CC2CC(=O)NC2=O)CC1 C1(NC(C(F)OC)=O)CCN(C(c2cnc(C)nc2C)=O)C12CCCC2 C(C(=O)N(c1ccc2c(c1)OCO2)CC(F)F)(C1=NOCC1)N1C(CC)COCC1 N1(S(CC(C)C)(=O)=O)CC(NC(C2CCC(O)CC2)=O)CC2(CCOCC2)C1 N1(C(C2OCCN(C)C2)=O)CC2(CC2)CC1CNC(=O)C(F)(F)c1cnccn1 N1(C(C(CC)(F)F)=O)C(CC(=O)NCCS(C)(=O)=O)C2CCCC12 C1(O)(C(=O)NC(C2CN(C(C3CCc4nc[nH]c4C3)=O)C2)C)CCCC(C)(C)C1 O=S(=O)(c1cncc(Br)c1)NC1CN(CC23CC4CC(CC(C4)C2)C3)CCC1F c1(-c2cn(C(C(=O)NC(CC)(C)C(=O)O)C)nn2)cccc2sccc12 C1(NC(CSCC(=O)OC)=O)CCC(NC(=O)CC2CCC(C)CC2)CC1 c1(COC)cccnc1C(=O)NCC1(CNC(c2nocc2C)=O)CC1(F)F C1(CC(=O)NCC2(N(C(CC(=O)NCC#C)=O)CC)CCC2)OCCCC1(C)C N#Cc1cc(C(N2CC(NC(=O)COCC(F)(F)F)C(F)C2)=O)ccc1O N1(C(C(CC#C)C)=O)CCC2(CCCN2C(=O)CC2(COC)CC2)C1 C1(NC(c2ccc(OCCC#C)cc2)=O)CCN(C(C2(CC)COC2)=O)CC1O N1(C(C2(C)CC2)=O)CCC2(CC(NC(c3cncc(-n4cccn4)n3)=O)CO2)C1 c1(C(=O)OC)ccc(O)c(NC(C2CN(C(C3CCCO3)=O)CCC2O)=O)c1 CC1CCCC(CC(=O)OC(c2cccc(Cl)c2)CF)O1 CC(C)CC(C(=O)NCc1cn(C)nn1)NC(c1nnc(O)nc1O)=O C(=O)(C(C)(C)C(C)(F)F)NC1CC(NC(c2nc(C(C)C)oc2)=O)C12CCC2 C1(COC)(NC(=O)CCC2(C)CC2)CCN(C(=O)C#CC2(C)CC2)CC1 N1(CCNC(=O)CCn2cccn2)CCN(C(C2CCCC(O)C2)=O)CC1 c1(C(=O)NC(C)CCCNC(c2ccc(F)cc2)=O)ccc(OC(F)F)c(Cl)c1 N#Cc1ccc(C(=O)NCC2OCCC2C(=O)N(CC(O)CO)CCO)o1 C(=O)(CCCCCC(C)O)NCC(CN(C(C=CC(CC)C)=O)CC)(C)C C1(NC(C(CC)CC)=O)CC(CNC(=O)CC=CCc2ccccc2)C12CCC2 CC1CC(C(=O)N(CCCn2cc(COCC(N)=O)nn2)C)CO1 c1(C(=O)NCC2(F)CC(NC(C(CCOC)C)=O)C2)ccc2n[nH]cc2n1 c1(CC)ccnc(CNC(=O)NC(c2sccc2NC)C)n1 C(CC(=O)N1CC2CC1CN2c1nc(C2CC2)nc(=N)[nH]1)(C(F)(F)F)OC N1(C(C2C(C#C)C2)=O)CC(NC(C2(n3cncn3)CC2)=O)CC(F)C1 C1(C(N2CC(NC(c3c(Br)cn(C)n3)=O)C(O)C2)=O)SC2C=CC1CC2 C(CC(C(C)(C)C)NC(=O)C(c1cscn1)N(C)C)N(C(=O)C=CBr)C c1(OC)cc(C(N2CCC(C)C2CNC(c2csnn2)=O)=O)ccc1F c1(C(=O)NC2(CO)CCC(C)CC2)c(NC(c2cnc(O)[nH]2)=O)sc2c1CCC2 C1(C(N2CC(N(C(CN(C3CC3)CC)=O)C)C2)=O)CCOC1(C)C c1(CC(=O)NCC2C3CN(C(C=NOC)=O)C2C3)ccc(C)c(OC)c1 C1(NC(=O)OC(C)(C)C)CCN(c2cc(Cc3ccns3)ncn2)CC1 n1(CC)ccnc1C(=O)NC12CC(C(=O)Nc3cnsc3)(C1)C2 C1(C(=O)NCCNC(=O)OCC)CCC2(CC2)N1C(=O)C=C(CC)CC N(C(=NCC1(OC)CCCC1)N1CCC(C(=O)Oc2ccc(Cl)cc2)CC1)C(C)C NS(=O)(=O)CCC(=O)N1CCCC1CNC(=O)CC1CC(O)C12CCC2 CCC(C)CC(C(=O)NCC(C)C)NC(=O)CC1CCC1 C1(C2CC2)(NC(c2cccc(=O)o2)=O)CCN(C(c2onc3ccccc23)=O)C1 c1(CC)cnccc1C(=O)NC(CCF)C(=O)NCC(C1CCCC1)OC C(=O)(C#CC(C)(C)CNC(c1c[nH]ccc1=O)=O)NCc1cc(OC)ncn1 C1(C(C)C)CCC(C)CC1C(=O)NC1CC12CC(NC(C1(F)CCCCC1)=O)C2 c1(N(C)CCN(C)C(c2nnn3ccccc23)=O)nc2ccc(Br)cc2o1 N1(C(c2c(CC)n[nH]c2)=O)CCCC(C(=O)NC2CC(C(C)(C)O)C2)C1 n1(CC)nc(C(=O)NC(CCOCCO)C(=O)N2CCC(SC)C2)c(C)n1 C1(NC(C(C(C)NC(c2c(NC)nccc2)=O)(C)C)=O)CN(C)C(=O)C12CC2 CCCC#CC(C)(C)NC(=O)C(C)C(CC)NC(=O)C(C)NC(=O)CC C1(NC(c2cccc(Br)c2F)c2n(CCCCCC)nnn2)CCCCC12CC2 C(=O)(C1=NNC(C(F)(F)F)C1)N1CCC(NC(COC(C)(C)C)=O)C1 C1(C)(CNC(C(C)=C(C)C)=O)COCCN(C(c2cccc3ccsc23)=O)C1 n1(CC)ncc(C(=O)NC2CCCC2NC(c2c[nH]c(C(=O)OC)c2)=O)n1 C(=O)(C1Cc2ccccc21)NC(C(=O)NCc1cc(C)ncn1)C1CCC1 CCCC(C(O)C(=O)N(C(C)CC(=O)OC)C)NC(=O)CCN(C)C Cc1cc(CNC(Cc2cccs2)CC(=O)NC2CC2)cc(C)c1F O=C(C#CC1CCCCC1)N1CCCC(C(=O)NCc2ccc(Cl)cc2Cl)C1 CC(C)CS(=O)(=O)CC(=O)NC12CCOCC1CN(C(=O)C#CC(C)(C)C)C2 C(=O)(CCCCc1ccccc1)NCC(C)(C)CNC(C1(C)CC1(F)F)=O C1(NC(C2CCCC(=O)N2)=O)CCN(C(C23CCC(CC2)CC3)=O)CC1F c1(C(=O)NCC2(F)CCC(NC(C(CCC)(C)C)=O)C2)cnn2ccnc(N)c12 c1(C(=O)NCCCCC(=O)NC2C=CCN(C(=O)C3CC3)C2)ccnc2cc[nH]c12 C1(C(N(CCN(C(C)C)C(C2CCS(=O)(=O)C2)=O)C)=O)(C(F)F)CCCSC1 C1(C(N(C(CC(C)C)C)C)=O)CCN(C(c2ocnc2C2CC2)=O)C12CCC2 c1(OC)ccc(CCOCC(=O)NCCN(CC#C)CC2CC2)cc1 C(=O)(NN1CCCC1C(=O)NC(CO)C1(C)CC1)c1cc(C)on1 C1(NC(=O)COCF)CCC2(CC1)CCN(C(=O)C(F)(F)c1ccncc1)CC2 C(CC(=O)N1CCCc2nccn21)=CC1CN(C(C(CCCC)C(C)C)=O)C1 C1(CNC(CCc2cn(C)nn2)=O)CCN(c2cc(Cl)nc(C3CC3)n2)C1(C)C C(=O)(CCS(=O)(=O)Nc1cn(C2(C(=O)O)CC2)nn1)NCC1CCN(C)C1 c1(CN2CC(C(=O)Nc3ccc(NS(C)(=O)=O)cc3)C(O)C2)cc(Cl)ccc1Cl N1(C(c2c(CC)nco2)=O)CCCC(NC(C2CN(C(=O)N(C)C)C2)=O)C1CC N1(C(CCOCC#C)=O)CCOC(C(=O)N(CC(=O)NCC)C2CCC2)C1 CCCC(C)(O)CC(=O)N1CCCC(C)(CNC(C2CN(C)CC(C)O2)=O)C1 C(C(=O)NCC(C)NC(=O)CCc1cn[nH]c1)(C(C)C)NC(C)=O c1(C(c2cn(C)nn2)(c2ccccc2)NC(=O)CO)nc2cnccc2s1 c1(N2CCC(F)(CO)C2)nc(N2CCOC(CF)C2)c2c(F)cccc2n1 CC(C)C(CO)CCNC(C1(C)CCCN(C(C2CC=CCC2)=O)C1)=O C1(NC(C2C(c3c(C)cccc3)C2)=O)CCN(Cc2nccs2)CC1O c1(C(=O)NC(C2CC(NC(C(C(CC)C)C)=O)C2)C)cccn2ccnc12 N1(C(C2(C)CC=CC2)=O)CCC2CCN(C(=O)CCC(=O)NC3CCCC3)CC2C1 C(CC(F)(F)F)(c1ccc(F)cc1)NC(=NCC=C)NCC1CCN(C2CC2)C1 c1(NC(c2scc(C)c2)=O)ncc(F)c(=NCc2ccc(-c3cccc(Br)n3)cc2)[nH]1 Cc1cc(NC(=O)C(C)(C)C)sc1C(=O)NC1CC1CNC(=O)CC1CCCO1 Cc1ccnc2sc(C(=O)N(C)CC3(CNC(=O)C4=COCC4)CC3)c(C)c12 N1(C(C2C(CC)OCC2)=O)C2CCCC1CC(NC(c1cnn(C(F)F)c1)=O)C2 CCC(C)C(C(=O)NCC(C1CC(C)(C)C1)O)N(C)C(c1n[nH]c2c1COC2)=O c1(SC)c(C(=O)NC2CCOC(c3cccs3)C2)cccc1Cl c1(C(N2CC(O)(CNC(C(CCOC)C)=O)C2)=O)cc(OC)cc(C(F)(F)F)c1 Cc1ccncc1C=CC(N1CCC(NC(=O)C(C)CO)C12CC2)=O C1(CC)(CC)CC(C(N2CCC2(C)CC(=O)NCC2CCN2C(C)(C)C)=O)C1 C(=O)(C(CN(C)C)C(C)C)N1C(CC=C)(C(=O)NCc2cc(C)sc2C)CCC1 C(C(C)(O)C(=O)NCC=CCNC(=O)C(c1ccccc1)n1cccn1)OC N1(C(C(C(C)C)F)=O)CC2CC1CC2CNC(=O)Cc1c(Cl)cnn1C c1(C(=O)NC2CC(C)(NC(C3OCC(C)C3)=O)C2)ccc(F)cc1O CC(CC(=O)NC(C1CCCCCC1)CNC(c1nocc1C1CC1)=O)C(F)F C1(C(N2CC(N(C(c3cn(C(C)C)nn3)=O)C)C2)=O)C(C)(C)CCCC1(C)C N#Cc1cc(F)c(F)cc1NC(C1CC(F)CN1C(c1sc(Br)cc1Br)=O)=O CC(C)CC(CNC(=O)CN1C(=O)CNC1=O)NC(=O)CCn1ccnn1 Cc1cc(C(=O)NCC(O)CNC(C2CN(C)C(=O)N2)=O)cc2ccoc12 N1(C(C(C)C)=O)CC(C)CCC1C(=O)Nc1cccc(I)c1 c1(C(=O)N)ccccc1.C(C(F)CNC(COCC)=O)NC(C1(COC)CC1)=O C1(C2CC2)(NC(c2csc(C)c2C)=O)CCN(C(=O)Cc2cccc(F)c2)C1 C1(COC)(CNC(c2ccno2)=O)CCCN1C(=O)CCC1CCC(=O)C1 n1(CC(=O)NCC2CN(C(=O)C(O)Cn3cncn3)C2)c(O)nc2ccccc12 c1(N2CCCC(CCO)CC2)nc(NC2CC2C2CCCC2)nc2c1COC2 c1(CNC(C(CC)Cc2ccccc2C)=O)ccc2c(c1)CCCS2 c1(CNC(C2N(C(c3c(C)ncs3)=O)CCOC2)=O)cc2ccccc2[nH]1 c1(C(=O)NCCCN(C(C(CCC#C)O)=O)C)cccc2c1CCCN2 n1(C2(Oc3ccccc3)CC2)nc(CC2CC2)nc1-c1csc(CCOC)n1 c1(CC(=O)NC2CCC(OC(C)(C)C)CC2)ccc([Si](C)(C)C)cc1 C1(C(=O)NCCC2(C)CCN(C(CCCOC)=O)C2)CC2OC(=O)OC2C1 C(=O)(C(CNC(=O)CCC(N)=O)CCC)NC(CC=C)C1CC1 C12(C(=O)NCCCCN(C(C3N(CC)CCC3)=O)C)CCC(OC)C1CC2 C(=O)(CC(C)CC(C)C)NCC1(F)CCN(C(c2c(C)cc(O)nc2)=O)C1 c1(C(N2CCC(F)(C(=O)NCc3ccsc3)C2)=O)cc(Cl)c2cn[nH]c2c1 c1(C(N(CC#CC)C)=O)cnc(CNC(=O)C#CC2CC2)nc1 CCCN=C(NCc1cc(Cl)ccc1OC)NCc1nccn1CC(F)(F)F C1(CC(=O)NC(CCCC=C)C2CC2)CCN(C(=O)CC2CC(=O)C2)C1(C)C C1(CNC(C2CC(=C)C2)=O)CC2(CCN(C(c3cncc(C(F)F)c3)=O)CC2)C1 c1(N(C2CC3(CNC3)C2)C(C2(C3CC3)CC2)=O)ncnc2c(Br)c[nH]c12 n1(CC(=O)Nc2ccccc2C2CC2)c(=O)ccn(CC2CCCC2)c1=O C1(N(CC(=O)N(CCN(C)C)C2CC2)C(=O)COC2CCC2)CC2C=CC1C2 N12CCN(CC3(CC3)C1)CC(C)(C1CC1)C2=O.c1(SC)cc(N(C)C)n(C)n1 C1(C(N(CC(=O)OCC)C)=O)CN(C(=O)C(O)CCSC)CC(C)(C)C1 c1(OC)ccc(CCC(=O)NC2CN(Cc3nccnc3Cl)CC2O)cn1 Cc1nn(C)c2c(NCC3CCCN3C)nc(N3CCc4[nH][nH]c(=N)c4C3)nc12 N1(C(c2ccc(OC)s2)=O)CC(CO)C2(C1)CN(C(=O)C1=CC3(CCOC3)C1)C2 c1(CC)ccc(NNC(=O)NC2CCOCC2)c(CC2CCN2)c1 C1(NC(=O)NCC2CCC(C)CC2)CC2C(=O)N(C)CC(=O)N2C1 C12(NC(C(C)CN(C)C(C3CCCOC3)=O)=O)CCC(C1)OC2C c1(C(N(C2CN(C(=O)CCn3ccnc3)CC23CC3)C)=O)cc2ncccc2[nH]1 S(=O)(=O)(c1cc(C)cnc1N(C(CO)C1CC1)C)N(C)Cc1ccc(OC)cc1 N1(C(CC(C)CN(C)C)=O)CCCCC12CN(C(C1CC1C1CCC1)=O)C2 C1(C(=O)NC(C)C(=O)NCCSC2CCN2C(C)(C)C)CCCCC1 O=C1Cc2cc(C(N3CC(Oc4nccn5nccc45)C3)=O)ccc2CN1 CC(CC(=O)N1CCC(N(C(=O)COCCF)CCO)C1)P(C)(C)=O C(c1ccc(Cl)s1)=CC(=O)NCC1CC(F)(CNC(C=C(C)Cl)=O)C1 C=C1CC(C(F)(F)F)(C(=O)NCC2CCN2C(=O)CSc2cnn(C)c2)C1 CC1=C(C(=O)NC2(CN(C)C(c3nc(C)nn3C)=O)CC2)CCC(C)(C)C1 C1(CCNC(C(C)NC(CC)=O)=O)CCCCN1C(=O)CCc1ccc(C)s1 Cc1nc2ncc(C(=O)NC3CC3CNC(=O)Cc3nn(C)cc3Cl)c(=O)n2[nH]1 CC(C)(C#N)CCC(=O)NCC1CN(C(C2Cc3cccnc3C2)=O)C1 C1(C(=O)NCCCOC)(CC)CN(C(=O)C(C)=C(C)CC)C1 CCC(C)(C)CC(=O)NCCCN(C(c1oc(CO)nc1C)=O)C(C)C N1(C(c2c(C#C)c[nH]n2)=O)CCN(C(c2cnc(C3CC3)nc2)=O)CC1C(F)F c1(CC)nc(C)c(C(N2CC3C(NC(=O)C=CCOCC(F)(F)F)C3C2)=O)o1 C1(CC(=O)NC2CC(CCNC(=O)C=CC3CC3)C2)CCC2(CC1)CCC2O N1(C(=O)Cc2csc3ccccc23)CCN(C(C2CC=CCC2)=O)C2CCCC12 C1(C(=O)NCCC(CC)CO)C2CCCC2CN1C(=O)C(C(=O)OC)OC Cc1cnc(F)cc1C(=O)NCC1CCCC1NC(c1cn(C)nn1)=O N1(C(c2[nH]cc(CC(C)C)c2)=O)CC2CN(C(=O)C(N3CCOCC3)C)CC2C1 C1(CC(=O)NC2(CNC(C3(F)CCC3)=O)CCCC2)CCc2ncc(Br)n2C1 c1(COC)ccnc(C(=O)NCC23CC2CN(C(=O)C=CC2CCC2)C3)c1 C1(OC)CCCC(CC(N2CC(OCCNC(=O)CCC(C)C)C2)=O)C1 c1(C(=O)NC2CC(CNC(C3CC3CF)=O)C2)nccn2nccc12 c1(C(=O)NCCC(CNC(C=CC=CCC)=O)(C)C)ccc(S(N)(=O)=O)s1 c12cc(ncn1)N1CCOCC21.n1(CCCC#C)cc(C(=O)OCCOC)cn1 CCCCS(=O)(=O)CC(=O)NCC1CCN1C(=O)CCCCC#N c1(NC(C2CCN(C(c3cc(C)n(C)c3C)=O)CC2O)=O)ccc(C#N)cc1O N1(C(C2C(CC)C2)=O)CCC(C(=O)N(C)Cc2nc(C)ns2)C1C c1(C(N2CCC(C)(CNC(CC(CC)C3CCC3)=O)C2)=O)cnc(OC)c(C)n1 N1(C(CSC)=O)CCCCC(CNC(c2ccncc2Oc2ccccc2)=O)C1 N1(C(CC2(C)OCCO2)=O)CCCC(C)(NC(=O)C(F)CC2CCOC2)C1 c1(C(N2OCC(n3cc(C(C(C)C)O)nn3)C2)=O)cc(S(N)(=O)=O)cc(Cl)c1Cl N1(C(C(c2ccc(CC)s2)=O)=O)C2CCC1C(NC(=O)Cn1cc(C)cn1)C2 c1(OC)cccc(Br)c1NC(C1CCN(Cc2cnc(OC)nc2)CC1O)=O c1(C(=O)NCCCN(C(=O)C(c2cccnc2)O)C)cc(=O)c(Br)c[nH]1 C(C)(CCC(=O)N(CCCCCNC(c1ccnc(S)c1)=O)C)OC C12(NC(CC3CCCC(OC)C3)=O)CCCC1N(C(C1CCN(C)CC1)=O)CC2 C12(CNC(c3cc[nH]c3)=O)CCC(NC(C3CC3(Cl)Cl)=O)(CO1)C2 CC1(C(=O)NC2CC3CCC2(NC(=O)CCC(N)=O)C3)OCCc2ccccc21 N1(C(CC(=C=C)C)=O)CC2CCC1CN2C(c1ccc(Br)c(C)n1)=O C(CC1CCCCC1)(C(=O)NC(C)CCCNC(C1(CO)COC1)=O)OC N1(C(C2(C=C)CC2)=O)CCC(C2CCN(C(=O)C(C)SC(F)(F)F)CC2)C1 c1(C(=O)NC(C(C)NC(CNC(C)=O)=O)CO)cccc2cccc(Cl)c12 C1(CC=C)(NC(C2CCCC23CC3)=O)CCN(C(=O)CCCN2CCCCC2)C1 CC1CCC(NC(c2cc(CCO)on2)=O)CN1C(C12CC(F)(C1)C2)=O N1(C(c2nn(CC)c(O)c2)=O)CC2CC(NC(c3n[nH]c(C)c3O)=O)C2C1 c1(C2(C(N(CCCN(CC)CC)CC)=O)CCC2)cccc(C#N)c1 c1(CNC(=O)CC2OCCCO2)cccc(NC(c2ccc(F)o2)=O)c1 C1(C(=O)NCC2(OC)CC(C)C2)CC12CCN(C(=O)CC1CCSCC1)CC2 CC1(C)COCCC1CNC(=O)CC(C(F)F)NC(=O)CC1CCCCCC1 c1(C(N(CCC(C)NC(COC(C)C)=O)C)=O)cnc2c(c1)c(O)nc(=O)n2C Cc1ccc(C(=O)NC2CC(C(=O)Nc3ccc(Cl)c(Cl)c3Cl)C2)c(I)c1C C1(NC(c2ccc[n+]([O-])c2)=O)CCCCC1C(=O)NCc1cccnc1O Cc1cc(F)cnc1C1(CCCC(=O)N(C)C)CC1.C1(C)C(=O)N1 C(=O)(C1CCc2cc(F)ccc21)NCCN(C(COCCC=C)=O)CCCN(C)C c1(C(=O)NC2CCCN(C(c3nnc(CC)s3)=O)CC2)c(O)nnc(C)c1C C1(NC(C(CC)OC)=O)CC2C1CCN2C(=O)CCCc1ccc(Cl)cc1 S(=O)(=O)(c1ccc(Cl)cc1)NC(C(=O)NC(CC)(C(N)=O)C(C)C)C(C)C Cc1cc2c(C(=O)NCCC3CN(C(=O)CCc4cnn(C)c4)C3)nccn2n1 CCC(CC(=O)NCC1(O)CCN(C(c2c(Cl)noc2C)=O)CC1)C(F)F C#Cc1ccc(C(N2CCCC2C2(NC(=O)C(O)C=C)CC2)=O)cc1Cl N1(C(C)C(=O)NC(N)=O)CC2CC1CN2C(C1CC12CCCC2)=O C(=O)(C(CO)NC(=O)C1CC1)N(CC(CC)NC(=O)C(CC)C1CCOCC1)C N(C1c2ccccc2CC12CCCC2)c1cc(N2CC(CCF)OCC2)ncn1 c1(C(N(C2CN(C(=O)CCc3cc(Cl)cs3)CC2F)C)=O)ccc(F)cn1 C1(NC(c2nc(C(=O)NCC3(CC)CC3)sc2)=O)C=CC(=O)N=N1 C1(NC(C(C2CCC2)OCC)=O)COC2C(NC(c3nc(C)c(C)s3)=O)COC12 N1(C(c2c(C(=O)OC)scc2)=O)CCC(NC(c2cc(C(F)(F)F)n[nH]2)=O)C(F)C1 Cc1nonc1CC(=O)NC(C)(C)CCNC(=O)CC(C)NC(N)=O Cc1c(C(=O)NCC(O)CN(C)C(c2cccc(N(C)C)c2)=O)cccc1F c1(C(N(C(C)CCNC(C2(C)CCCOC2)=O)C)=O)c(O)cccc1Cl N1(C(C(C(C)CNC(=O)C(=C2CCCCC2)F)F)=O)CC2C3CCC(C3)C2C1 n1(CC(N2CC3C(CNC(C(F)OC)=O)(C3)C2)=O)ncc(C#N)c1N N1(C(CC=C)=O)CC2(CCC(C(N3CCCCC3CCO)=O)O2)C1 c1(OC)cccc(C(C)=CC(=O)NC2(CNC(=O)C3=CCCC3)CCC2)c1 C(=O)(CCCCCC#N)N(CCNC(C1(OC)CC(C)CC(C)C1)=O)C1CC1 CC1CN(C(=O)CC2COCCO2)CC1(C)CNC(=O)C=Cc1ccsc1 c1(COC(C2CCc3n[nH]cc3C2)=O)cnn2cc(Br)ccc12 c1(OC)ccc(-n2nc(C3CC3)nc2-c2cc(C3CCOCC3)on2)cn1 C=CC1(CC(=O)NOCC(C)(C)O)CN(C(=O)CC2CCCCN2C)C1 CN1CCC(CCC(=O)NCC(C)(CO)NC(c2ccc(F)s2)=O)C1 c1(CC)cc(CC)[nH]c(=NCC2CCCCN2C(c2ccc(Cl)c(Cl)c2)=O)n1 C1(C(N2CC(C(C)NC(=O)Cn3cccn3)C2)=O)CCCC1C1CC1 C(=O)(CCCC(F)(F)F)NC1(CF)CCN(C(C(C)C=Cc2ccccc2)=O)C1 CCCCC(CC)CC(=O)NC1CCC1CNC(c1ccc(Cl)c(N)c1Cl)=O C(CC(C(=O)Nc1nccs1)N1CCC(CO)CC1)C1CS(=O)(=O)C1 c1(CC)ccc(C=CC(N2CCC(CF)(NC(c3cc(OC)cs3)=O)C2)=O)o1 C1(CC(=O)NC)CN(C(=O)COc2csnn2)CCN1C(=O)C(C)C1CCCC1 c1(COCC(=O)NC(C2CCOCC2)C)n[nH]c(C(C)(C)C)n1 c1(C(=O)Nc2cnc(F)cc2C(=O)NCC(O)C(F)(F)F)ccc(O)c([N+](=O)[O-])c1 Cc1coc(C)c1C=CC(=O)NCCC1(C)CCN(C(=O)C(C)C2CC2)C1 c1(C(=O)NCC2N(C(C=CC(C)C)=O)CC(C)CC2)ccc2cnoc2c1 Cc1cc(CC(=O)NCCN(C(C2CCC(C(N)=O)C2)=O)C(C)C)sn1 c1(C(N2CC(C)(NC(C(n3ncc(C)c3)C)=O)C2)=O)ccc(C(C)=O)nc1O O=S(=O)(c1ccnc(C(F)(F)F)c1)NCCOc1ncccc1Br C#CC1(NC(=O)CC2(C)CCN2C(=O)CN(C2CC2)CC)CC2CCCC12 C#CCC(CC(F)F)C(=O)NCCC(C)(C)NC(=O)CC1CCCCC1 C12(C(N(C(C)C)CCO)=O)COC(C(=O)N(c3ccccc3C3(C)CC3)C)(C1)C2 c1(NC(CC2N(C(C=Cc3ccc(C)s3)=O)CCC2)=O)cc(F)ccc1O N1(C(CCC)=O)CCC2(CCN(C(=O)COc3cc(C)on3)C2)C1 c1(C(=O)NCC(C2CCOC2)NC(c2c(C#N)ccs2)=O)ncnc2sccc12 Cn1cc(CCC(=O)NCC(C)(CNC(C2(CCO)CC2)=O)OC)cn1 C(=O)(C(CNC(=O)C=C(C)COC)C(C)C)N(CCCC)C C1(C(N(C)CC2CCN(C(c3c(OC)csc3)=O)C2)=O)Cc2c(C)cccc2O1 C(C(C)(C(=O)NCCc1nc(C)no1)NC(=O)CCCn1cncn1)SC Cc1cc(F)ncc1NC(C1(CNC(=O)C(O)Cn2cncn2)CC12CCC2)=O N1(C(C(COC)OC)=O)CCC2CCN(C(c3cnc(OC)c(C)c3)=O)CC12 N1(C(C(N2CCSCC2)C)=O)CCN(C(=O)CCCc2cncs2)C(C2CC2)C1 S(=O)(=O)(CCCN=c1[nH]c(=N)[nH]c(=NCCCNC(N)=O)[nH]1)NC(=O)NC(C)(C)C c1(C(N2CC3C(NC(C(C)SCCCC)=O)(C3)C2)=O)cnn2c1CC(F)(F)C2 c1(C(=O)NC2C3(NC(C(C)OC)=O)CCC(C2)C3)nc2ccccc2cc1Cl N1(C(C2(CC)CCC2)=O)CCC2(CC1)CC2C(=O)Nc1cc(C)ccc1Br N1(C(c2c(=N)cc[nH]c2)=O)CC=C(CNC(C2(C3CC3)CCC2)=O)CC1 CCCC(C#N)C(=O)NCC(CC(=O)NC1C2CCC(F)(F)C12)C1CCC1 C1(NC(CC=C)=O)CCCC(NC(=O)OC(C)(C)C)C1.C123CC(C1)(C2)NC3=O c1(C(=O)NC(C2(O)CCN(C(=O)C(O)C(F)F)C2)C)cn(C)c2c(Cl)cccc12 CC1CC(CNC(C2CCN(C)C2)=O)CCN1C(c1ccc(O)cn1)=O c1(CNC(c2cc3c[nH]cnc-3n2)=O)cccc2c1CCN(c1ncns1)C2 C(C(C)CC(=O)NOCC1CCOCC1)NC(C1C(C)CC1)=O C1(CNC(CCCC(=C)C)=O)CN(C(=O)Cc2ccn(CC)n2)CCC12CCC2 N1(C(COC(CC)(C)C)=O)C2CCC1CN(C(=O)C(C)C(C)O)C2 c1(C(N(CCCN(C(C(C)OCCC#C)=O)C)C)=O)cc(C(C)(F)F)ccn1 c1(C(=O)NC2CCN(C(c3c(C)con3)=O)C(C)C2)scc2c1OCCO2 C1(NC(CC(C)NC(N)=O)=O)CC(CNC(c2cncnc2)=O)C(O)C1 C1(C(N2CCC(NC(C(C)(C)OC(C)C)=O)C(O)C2)=O)CCC2(CCC2)CC1 C1(CCC)(NC(=O)CC2(N(C(=O)CCc3cccnc3)C)CC2)CCNC1=O CC1(C)CCC2(CCN2C(C2(O)CC2)=O)CC1 CC(CSc1ccccc1)C(=O)NC1CC(C)(CNC(=O)C(C)(F)F)C1 C12(C(=O)NCCOCCCNC(c3n[nH]c4c3CCC4)=O)OCCCC1C2(F)F C1(C)(C(=O)NCCCn2c(C)nnc2)C=CCN1C(=O)CCC1CCCO1 c1(C(=O)NCCCC2(NC(C3C(C=C)C3)=O)CC2)cc(O)nc(C2CC2)n1 C1(CCC(=O)NC)CCCN(C(=O)N(c2cccc(Br)c2)CCN(C)C)C1 c1(CCC(=O)OCC)ccc(NC(=O)CCc2cncc(F)c2)cc1 c1(Cn2cc(CC)nn2)nn2c(c1C(=O)NC(C)C(C)C)CCC2 CC1(C)CCCC(C(=O)NCCC2CSCCN2C(c2cc[nH]c(=N)c2)=O)CC1 c1(OC(C(=O)NCC2C3CN(C(=O)CC4CCC4)CC32)F)ccc(Cl)c(F)c1 c1(C(=O)NCC2C(NC(CCS(C)(=O)=O)=O)C2)ccc(N)c2ccncc12 N1(C(C(C)(C)OC(C)C)=O)CCCC2(C1)CN(C(=O)CCn1ccnc1)CCO2 c1(CC(=O)NCC(C)NC(=O)C(C)NC(c2ccco2)=O)cncnc1.C(=O)(C1CC1)N CCC(CC)(CC)C(=O)N1CC2CC1C2NC(C1OCCC1C)=O CCC(CC(=O)NCC1(C(=O)NC2CC(OC)(OC)C2)CCCCC1)SC1CC1 N1(C(C=C(C)C(C)(C)C)=O)CCC2(NC(c3cccc[n+]3[O-])=O)CCCCCC12 N1(C(C2(CC)CCCO2)=O)CC(CCNC(c2cnc(O)n2C)=O)C(C)C1 c1(C(N2CC(CNC(C(C)(Cl)Cl)=O)OCC2)=O)cc(S(=O)(=O)NC2CC2)c[nH]1 C(CF)(C(=O)NCCSCc1ccncc1)OC(=O)NC(C)(C)C.C1C(=O)N1 c1(C(N2C(C(N(CCCO)C(C)C)=O)C=CC2)=O)c[nH]c2cc(Cl)ccc12 C1(C(=O)NCC2(n3ccnn3)CC2)CCC2CCC12 N1(C(C2(C#C)CCCC2)=O)CC(C)OC2(CCN(C(=O)COC(F)(F)F)C2)C1 C1(NC(C(=C)Cc2ccccc2)=O)COCCN(C(=O)CSC)C1 C1(C(C)NC(c2cscc2C(F)F)=O)CN(C(=O)CC2(N3CCCC3)CC2)CCO1 c1(C(=O)NCC2CC(CNC(c3c(C(C)C)csc3)=O)OC2)cn2ccnc2s1 c1(C(=O)Nc2cc(C)ns2)cccc2c1CN(Cc1ccncc1O)CC2 c1(C(N(CC(C)N(C(C(CCC)C)=O)C)C)=O)ccc2cc(C)ccc2n1 c1(C(C(=O)OC)NC(=O)Cc2csc(-c3ccco3)n2)ccc(F)c(Br)c1 NC1CCOCC1CNC(=O)NOCC(F)(F)C(F)F c1(CN2CC(CNC(C3(CC)CCOCC3)=O)OCC2)csc([N+](=O)[O-])c1 C(=O)(C(C)CC(F)F)N1C(C(C)C)CCC1C(=O)NCC1(C#N)CC1 Cc1ccc(C(=O)NC(C2CCCN(C(c3cc(O)cc(F)c3)=O)C2)C)c(F)c1 C1(C(=O)NC2(CNC(c3nc(C4CC4)cs3)=O)CC2)CC2C=CC1C2 N1(CC)CCN(C(C(=O)NCc2nnn(C)n2)C(C2CC2)OC)CC1C c1(OC)cccc(C2=NOC(C(=O)OCc3cnsc3)C2)c1 O=CN1CCCC1C(=O)NCCNC(C12CC(c3ccccc3)(CO1)C2)=O N1(C(C2CCN(C)C2)=O)CC2(CNC(c3cccc4nncn34)=O)CCC1CC2 N1(C(=O)CC2CCCCO2)CCC2CCN(C(c3nccc4occc34)=O)C2C1 N1(C(C(c2ccc(C)s2)C)=O)CCOC2(CCN(C(C3CCCC(=O)N3)=O)C2)C1 N1(C(CCCCC=C)=O)CC(C(N2CCOC(C(C)(C)C)C2)=O)C2(CCC2)C1 C12(C(N3CCC(NC(Cc4c(C)occ4)=O)C(CO)C3)=O)CC(C)(C1)OC2(C)C C1(C)(CC)CC(NC(c2c(F)cnn2C(C)C)=O)CN1C(=O)Cc1ccco1 C(=O)(C(O)C(F)(F)F)NCc1c(C(=O)OC)n[nH]c1.C12CCC1CNC2=O c1(CC(=O)NC(c2cnn(C)c2)C(=O)N(C(C=C)C2CC2)C)csnc1C C[Si](C)(C)C1CCCN(C(C2CCCN2C(=O)CC2CCOCC2)=O)C1 c1(CNC(C(N2CCCCCC2)C)=O)ccccc1C1CC1.C12CCC1NC2=O c1(C(N2CC3N(C(COCCC)=O)C(CC3)C2)=O)cc(C)nc(O)c1[N+](=O)[O-] N1(C(c2c(COC)cccc2)=O)CC2CC(C1)N(c1nnc(C)o1)C2 c1(OC)cnc(F)cc1C(N1CC2(C1)CN(C(c1ncc(C)cc1OC)=O)C2)=O N1(C(c2cccc(COC)n2)=O)CCC(NC(C2CC(OC)C2)=O)C12CCC2 NC1C=CC(CC(=O)N)C1.c1(CCC)nnnn1CCC1CC1 c1(C(N2CCN(C(C(N3CCC(C)C3)=O)=O)C(C)C2)=O)coc2cc(O)ccc12 C1(CC(=O)NCC(=C)CC)CC(C)(C)CN1C(=O)CC(C)(C)O CON(CCC(=O)NOCC1CCOC1)C(=O)c1ccc(C(N)=O)[nH]1 c1(C(=O)NCC(CC(C)C)NC(C2CC3CCC2CC3)=O)ccc(C#N)c(Cl)c1 N1(C(c2c(C)nsc2N)=O)CCC=C(CNC(=O)Cn2ncn(C)c2=O)C1 N1(C(=O)NCCCCN(CCCCC)C)CCCC1N(C(C)=O)CC.C(C)(C)(C)O N1(C(CC2(C)CCCC2)=O)CCC(O)(CNC(c2coc(C3CCC3)n2)=O)C1 N(C1CC(C)(C)Oc2ccc(F)cc21)C(c1c(OC)cncn1)=O CC(C)CCCCC(=O)N(C1CCC2CN(C(=O)CC3CCOC3C)CC12)C N1(C(C(C)C2CC2)=O)CC=C(C(=O)NCC2CCC(C)(C)CO2)CC1 C1(CC(=O)N(C2C(C)C2)C)CCCC(NC(=O)CCCOC(C)(C)C)C1 N1(C(C2CC(C)(C)C2C(F)(F)F)=O)CCC(CO)(NC(=O)Cc2cc[nH]n2)CC1 C(C)(CO)(CN=c1[nH]c(=NC(C)CN2CCCCCC2)[nH]c2cccnc12)OC Cc1cc(C(N2CCC(F)(C(=O)NCCC3CCN(C)C3)C2)=O)c(C)s1 C(N=c1[nH]c(NCCC#CBr)nc2c1CCC2)C1(CCC=C)CCCC1 N1(C(c2cc(OC)n(C)n2)=O)CCC(C)C(NC(c2cccnc2)=O)C1C C(=O)(CC(C)CC(C)(C)C)NCC(CC=C)C(=O)N1CCN(CC)CC1 c1(C(N2C(C(=O)NC(c3ccc(O)cc3)C)CC3CC32)=O)c[nH]c2nccc-2c1 C(N=c1[nH]c2ncnc-2c(C(F)(F)F)[nH]1)c1ccc(C2CC(=O)NC2)cc1 c1(C(c2n(CCOCC)nnn2)NC(c2scnc2C)C)cnc(Cl)n1C C1(NC(c2cc(C)no2)=O)CCN(C(=O)Cn2ccc(=O)n(C)c2=O)CC1(C)C c1(C(N(C(C)CCNC(C2CCC(C)O2)=O)C)=O)cccn(C2CCC2)c1=O CC1C(C(=O)NC2(C)CN(C(N)=O)C2)CCN1C(=O)CC1CCSCC1 N1(C(C(C2CCC2)OCC)=O)CCCC(N(C(=O)CC(C)SC)CCO)C1 c1(-c2ccn(C)c(=O)c2)nc(C(=O)Nc2cccc(C#N)c2Cl)n2ccccc12 N1(C(C=Cc2n(C)ncc2)=O)CCN(C(=O)CCc2cncs2)C(CO)C1 N1(C(CC2C(C)=NNC2=O)=O)CC2(C(=O)NCC3(C)CNC(=O)O3)CC1CCO2 CCC(CCCO)N=c1[nH]c(N2CCOCC2)nc(=NCc2cnn[nH]2)[nH]1 C1(NC(C2(CC=C)CCCC2)=O)CC=C(C(=O)NC(C=C)C2CC2)C1 N1(C(c2cccc(-c3cn[nH]c3)c2)C(=O)NCC(=C)C)CCC(O)C(F)(F)CC1 C(=O)(C1=NOC(C)C1C)NC1C(CC)CN(C(=O)CN2CC(=O)NC2=O)C1 c1(N(CCNC(C(C(C)C)NC(C)=O)=O)C2CC2)ncccc1C#N n1(CC(=O)NC(COC)CNC(=O)CC2(CO)CCC2)cc(Cl)c(C)n1 c1(Nc2cc(C(N3CCCC(C(=O)OCC)C3)=O)no2)cc(Cl)ccc1[N+](=O)[O-] c1(CC(=O)NC2CN(C(C(c3ccc(C)cc3)=O)=O)C(C)C2)cc(O)nc(O)n1 C(CC(C(=O)NCC1CCCO1)NC(=O)CCOCC(C)(C)C)=CC C(C(O)CC(F)(F)F)N(CCNC(c1ccccc1N1CCOCC1)=O)CC Cc1cccc2c1OCC(NC(c1oc3ccccc3c1SCC(N)=O)=O)C2 C#CCC(C(=O)NC)NC(C1CN(C(=O)CN(C)C(C)=O)CCS1)=O N#Cc1ccc(COC(c2c[nH]nc2COc2ccccc2)=O)cn1 c1(OC)ccc2[nH]cc(C(=O)NC3CCOCC3NC(C3CSCCS3)=O)c2c1 C1(C)(CC)CCC(CNC(=O)C(C)=CCNC(c2ccc[nH]2)=O)O1 c1(C(N(CCOC)CCNC(c2cc(C)sc2C)=O)=O)cncn(C)c1=O N=c1nc(Cl)cc(C(N2CCCC(CNC(=O)CCN3CCCCC3)CC2)=O)[nH]1 Cc1nn(C)c2sc(C(=O)NC34CCCC3CN(C(=O)C=C3CCC3)C4)cc12 CCC(CC)CC(=O)NCCOCCNC(=O)CCCOC(C)(C)C Cc1c(NC(=O)C(=O)N(C)CCc2cccc(Cl)c2)cccc1Cl C(=O)(C1=CCCO1)N1C(CN(C(CCSCC)=O)C2CC2)CCC1 CC1CCC2(CC1)CCN2C(c1ccc(F)c(Cl)c1F)C(=O)NCCCF C1(C2CCC2)(C(N(C)CC2(CNC(=O)CCCn3cncn3)CC2)=O)CC1 N1(C(C(C2CC2)OC)=O)CCCCC1C1CCN(C(=O)C(c2ccc(Cl)s2)=O)C1 C1(OC)CN(C(c2ncc(F)cn2)=O)CC1NC(=O)C(c1ccc(Cl)s1)=O c1(OC)cccc(C(=O)NC(C(C)NC(c2cc(C(C)C)no2)=O)C(C)C)c1F N1(C(C(C)Cn2cccn2)=O)CC2(COC(CNC(c3ccccc3F)=O)C2)C1 Clc1cscc1CNC(c1ccnn1C1CCC1)c1nnnn1CC1CCOC1 c1(C(=O)OC)ccc(O)c(C(=O)NCC2CC2NC(c2csc(Br)c2)=O)c1 Cc1cc(C(N2CC(C3(NC(=O)Cc4nccn4C)CC3)C2)=O)c(C)n1C(C)C Cc1cc(=NC(=O)CN(C(C)(C)CO)C(c2cccc(F)c2C)=O)[nH]o1 c1(CNC(C2CC3CC3N2C(c2ccc(O)nn2)=O)=O)c(F)cccc1F N1(C(COCCC(C)C)=O)CCC2(NC(=O)CCCn3c(O)nnc3O)CC2C1 C(=O)(C(C)(C)CC(F)F)N(C)CCOCCC(=O)NC1CCCCC1C(N)=O c1(C(=O)NCC2(C)OCCN(C(C=NOC)=O)C2)cccc2c1CCS2(=O)=O C1(CCNC(=O)CCc2ccc(C)o2)(OC)CN(C(c2ccoc2)=O)C1 CCS(=O)(=O)CC(=O)N1CCC(n2cc(-c3ccccc3O)nn2)C1 C1(CC)CCCN(C(c2cc(C3CC3)n(C)n2)C(=O)NCC2CCCO2)C1 C1(NC(C(c2ccoc2)NC(C(C)CO)=O)=O)CCCC(C2CC2)C1 c1(C(N2C(CCNC(c3c(C)cnnc3)=O)COCC2)=O)ccc(Br)c(F)c1 C1(C(=O)NC2(CC=C)CN(C(=O)Cc3[nH]cnc3C)C2)COCCN1C c1(NC(C2C3CN(C(C(CCC)CCC)=O)C2C3)=O)ccc2c(c1)OCCO2 c1(C(=O)NCC#CC(=O)NC(CO)C2CC2)c[nH]ccc1=O N#Cc1cc(C(N2CCCC(C(=O)Cc3ccccc3)C2)=O)sc1Br C1(NC(C2(NC(CCOC)=O)CCC2)=O)CCNC(=O)C1 c1(C(C(C)NC(=O)NCc2c(I)ccnc2F)OC)cc(Cl)cc(Cl)c1 C1(NC(c2ccc(SC)o2)=O)C(C)(C)C(NC(c2cc(Cl)ccc2F)=O)C1(C)C CCC(CC)CC(F)C(=O)NC(C)CC(=O)N(C)CC1CCCN(C)C1 c1(C2CN(C(C=C)C(=O)NCCOCC)C2)ccc(C2CCC2)cn1 c1(C(=O)NC2CC(N(C(C(CCOC)C)=O)C)C2)cc([N+](=O)[O-])c(C)s1 C1(CC)(NC(=O)CN2CCCOC2=O)CCCN(C(c2cc(Cl)nnc2O)=O)C1 CC(CF)C(=O)NCC(C)(C1CC1)NC(=O)CSS(C)(=O)=O C1(NC(c2ccc(Cl)s2)=O)CN(C(=O)Cc2ccc(Br)cn2)CC2CC12 c1(N(C)Cc2ccccc2Br)nc2ccc(Cl)cc2c(=NCC2CC23CCC3)[nH]1 C1(C(F)(F)F)(SC)CCCCC1.N12CCC(C1)N(CCO)CC2=O N1(C(CCC2CC(NC(=O)C3=NOCC3)C2)=O)CCC(CO)=C(F)C1 c1(C(=O)NC(CN(C(c2c(C(C)=O)cn(C)n2)=O)C)C)scc2c1CCCC2 C1(NC(C(C2(O)CN(C(C3(C)CCNC3=O)=O)C2)F)=O)C2CCC3C(C2)CC13 CC1CN(C(C2C3CCCC23)=O)CCC1N(C)C(c1cn(C)ccc1=O)=O CS(=O)(=O)c1cnn(CCNC(=O)C(=O)NC2CC2(F)F)c1 c1(C(N2CCC(CC(F)(F)F)C2)C(=O)NCCCSCC)cc(Br)nn1CC CCC(CC)CCC(=O)N1CCOCCC1C(=O)NC(C)CC(F)(F)F CC1CCCC=C1C(=O)N1CCC2CN(C(c3ncc(C#N)cc3Cl)=O)CC12 N1(CCNC(C(C)(C)C)=O)CCOC2(CCS(=O)(=NC(=O)NC3CCC3)CC2)C1 N1(C(CC)=O)CCCCC1C(=O)N(C)CC1CN(C(C2CN(C)C2)=O)C1 C1(C(=O)NC(CCNC(CCS(=O)(=O)NC)=O)C)Cc2ccncc2N1 C(=O)(C1=C(C#N)CCC1)N(C)CC1CCCC(NC(c2ccc(C)s2)=O)C1 CC(C)(CCNC(=O)C=C1CCCCC1)C(=O)NC1CCN(C2CC2)CC1 C(=O)(CC(C)C(C)C)N1CCC(C)(C(NOC(CC)CC)=O)C1 C1(NC(=O)C=CCO)COC2(CCN(C(c3cc4cccc(F)c4o3)=O)CC2)C1 C(=O)(C1CCc2nccn21)NCC1(C)CC(C(NOCCCC#C)=O)C1 Cc1nn(C)c(C(F)(F)F)c1C(=O)NCCSc1ccncc1 c1(C(=O)NCC2(C)CN(C(C34CCCN3CCC4)=O)C2)ccc(Cl)c(F)c1 c1(C(=O)NC2(CN(C(CCC(CC)OC)=O)C)CC2)cc2nccnc2cc1F CC1(C)C2CCC(C2)C1NC(C1COCC1NC(=O)C(=O)Nc1ccccc1)=O C1(C(N2CC3CCC2C3)=O)CCCCN1C(=O)Cc1ccc(Cl)cc1 C1(C(N2CCC(CC3(C)CC3)CC2)C(N2CCCC(C)C2)=O)CC2C(C1)C2(F)F c1(NC(N2CC(C(CC)C)C2)=O)ccn2nccc2n1 CC(C)C(F)(F)CC(=O)N1CCC1NC(=O)CNS(=O)(=O)C1CC1 N1(C(=O)NC2CN(C(C)=O)C3C2C3)CCCc2ccccc2C1 C(C(=O)NC(C)C(=O)OC)(C(C(C)C)C(C)C)N(CCc1ccco1)CC c1(NC(C(CC)OC)=O)ncccc1C(N1CCCCC1C(=O)OC(C)C)=O C(=O)(C(C)(C)C(C)(C)C)NCC(CC(C)C)NC(c1cc(C)c(C)o1)=O C(=O)(C1COc2ccccc21)NC1CCC(NC(C(CSC)(C)C)=O)CC1 CCC(CC)(CCC(=O)NC1CC(C)N(C(c2nocc2C(C)C)=O)C1)[N+](=O)[O-] C(=O)(C(CNC(c1cnc(S)nc1)=O)CC1CC1)NCCCN(CC)CC C(c1ccccc1F)=CC(N1CCC(C)(NC(=O)CCC2CC(F)(F)C2)C1)=O C1(OCC(=O)NCCC(=C)CNC(=O)C(F)=CCC)CCCCCC1 c1(C(N2CC(CNC(CC(CC)C)=O)N(C)CC2)=O)ccc2c(C)[nH]nc2c1 C1(NC(c2cn(CCC)nc2)=O)CCCN(C(c2ccc(NC(C)C)nc2)=O)C1 c1(NC(C2CNCCN2Cc2cc(Br)ccc2F)=O)ccnc(Cl)c1I N1(C(Cc2cnc(C)s2)=O)CCOCC1CC(=O)NC1CN(C2CCC2)C1 Cc1oc(C(=O)NCC2(C)OCCCO2)cc1CO c1(C(=O)NC2(CF)CCN(C(C(C)OCC=C)=O)C2)cc(=O)c(Br)c[nH]1 c1(C(N2CCC(CNC(c3c(OC)scc3)=O)C2(C)C)=O)nc2ccccc2[nH]1 c1(NC(=O)CN2CCC(c3ccc(F)cc3)CC2)nc2ccc(F)cc2s1 N1(C(c2c(C)cco2)=O)CC(CC(=O)NC2CC(C)OC2=O)C2(CC2)C1 C1(C(=O)N(C2CCN(C)C2)C2CCC2)C2CC1N(C(C1(C)CC(C)(C)C1)=O)C2 N1(C(c2ccc(C)cn2)=O)CCN(C(=O)CC2=CCCC2)C2CCCCC12 c1(C(=O)NCC2CCN(C(C3N(CC)CC3)=O)C2(C)C)scc2c1OCCO2 C#CCCC(C(=O)N1CCC(CN=[N+]=[N-])C1)NC(c1cnc(C)nc1C)=O C(=O)(C1=NOC(CNC(c2cnnc(O)c2)=O)C1)NCCC#CCC C1(CNC(CCC#C)=O)CC(C)(C)CN1C(c1ccc(C(C)=O)c(F)c1)=O CC1CN(C(c2ccc(F)c(Cl)c2)=O)CCN1C(=O)CC1CC1C C=CC1(C(=O)NCCCCC(CO)NC(=O)CCC2CCCO2)CCOCC1 S(=O)(=O)(c1cnn2ccc(=NCCn3ccnc3)[nH]c12)NC(CC#CC)C c1(CC)conc1C(=O)NCC(CC)NC(=O)C(F)(F)C1CCOCC1 N1(C(Cc2cnc(C)s2)=O)CCC2CN(C(c3cccc(Br)c3F)=O)CC12 C1(NC(c2nc(CC)oc2)=O)CN(C(c2c(Br)cncc2Br)=O)CC12CC2 CC(C)C(O)C(=O)N1CCC(C)(CNC(=O)CN2CCN(C)CC2)C1 C(=O)(N=c1cnc(I)c[nH]1)C1CCN(C(C2CC=C(C)CC2)=O)CC1 Cc1cc(Cl)ccc1OCC(=O)N(CC(C)N(C)C(C1CCC(C)(C)C1)=O)C C(CCC)(C(=O)NC1(C(=O)NCC2CC(SC)C2)CC1(C)C)=CCC Cc1c(C(=O)NCCOC2CCN(C(=O)CCS(N)(=O)=O)CC2)cccc1F C1(NC(C2C3CN(C(c4coc(C5CC5)n4)=O)CC23)=O)CCN2CCC1C2 N1(C(C2(CC#C)CCCO2)=O)CCC2(CCCN(C(=O)Cc3nccn3C)C2)C1 N1(C(c2cc(C)nc(Cl)c2N)=O)CC2CC(O)C1C2NC(c1c(OC)csc1)=O c1(C2(COC)CC2)ccc(C(=O)NCC(C)CNC(=O)CC2CSCCS2)cc1 c1(C(=O)NCC(C)(C2CCC2)NC(C(C)NC=O)=O)ccc(F)s1 N1(C(CC=CCC)=O)CCCC(C)(CNC(c2ccncc2C(=O)N(C)C)=O)C1 N1(C(C2C(=C)CC2)=O)CCC(CN(C)C(c2cn(CC3(C)COC3)nn2)=O)C1 c1(C(=O)NCC(CNC(c2ccc(C(N)=O)o2)=O)O)cccc2ncnc(O)c12 N1(C(C2CCCN(CCC)C2)=O)CCC2(CCCN2C(C2COC(C)(C)C2)=O)C1 C12(C(=O)OCC)CCC(NC(c3cc(Cl)cnc3F)=O)(CC1)C2 c1(C(N(C2CC(NC(C(Cc3c(C)cccc3)C)=O)C2)C)=O)ccc(F)c(Cl)c1 C1(C(C)NC(CC2(C=C)CCC2)=O)CCN(C(C2CCCCC2)=O)CC1 O=S(=O)(c1cnc(N2CCOCC(O)C2)c(Cl)c1)NCC1COCO1 C1(NC(c2c(C)nc(O)[nH]2)=O)CCN(C(c2cc(Cl)ccn2)=O)C1(C)C C1(c2cccs2)(C(=O)NC2CCN(CCCO)C2)CCCCC1 CN1CCC(CNCc2cc(C3CC3)ns2)C1c1ccc(F)cc1 C1(c2ccccc2Cl)(C(=O)NCC2CN(C(c3ncn(C)n3)=O)C2)CCCCC1 C(c1nc2ccccc2s1)=CC(=O)NCCN(C)C(C1CCC=CCC1)=O C1(NC(C(C)N(C(C=CC(C)C)=O)C2CC2)=O)C2CCCCCC12 C#Cc1cnn(C)c1C(=O)NC(CC(C)C)C(=O)NCC12CCC(CO1)C2 c1(C(=O)OC)ccc(NC2CCNC2c2ccccc2)c(F)c1 c1(C(=O)NCC23CC(CNC(C=CC)=O)(OC2)C3)cn2cccc(C)c2n1 c1(NCC(CC)(CC)NC(=O)CC2CC=CC2)ncc2ccnc-2[nH]1 C1(NC(CCCOC(C)C)=O)COCCN(C(=O)CC=CCc2ccccc2)C1 C(=O)(CC(=O)Nc1ccccn1)N(C)CC1(C(=O)OC(C)(C)C)CCCO1 c1(OC)ccc(C(=O)NC(C2CCCCN2C(=O)C=C2CC2)C)cc1C1CC1 C12(C(=O)NCC3CCCN(C(C(CCC)(C)O)=O)C3)CCC(OC)(CC1)CC2=O CCC(C)CC(=O)N1CCCCC1CCNC(=O)Cn1cnc(C(N)=O)n1 CCCCC(=O)C(=O)N1CC(C(=O)NC(CC)CC(F)(F)F)CCC1C Cc1cc(C(=O)N(C(C)CN(C(=O)C(C)NC(=O)CC(C)(C)C)C)C)nn1C C1(C(N2CC(CC(C)NC(Cn3ccc(C)n3)=O)C2)=O)CCC2(CCOCC2)C1 c1(C(=O)NC2(C)CN(C(=O)C(F)(F)CC3CCCO3)C2)cc2ccccc2o1 CN1CCN(C(C2CC3(C2)CC(O)C3)=O)CC1C(N1CC(F)(F)C1)=O N1(C(c2cnn(C)c2Cl)=O)CCCCCC(NC(c2n[nH]cc2C(C)(C)C)=O)C1 c1(CC)cnc(Cl)[nH]c1=NC1CN(C(c2sc(CC(C)C)nc2C)=O)CC1C c1(CN2C(C(N3CCC(O)C(F)C3)=O)CC(F)C2)c(Br)cccc1[N+](=O)[O-] C1(CNC(C(C2CCCCC2)C)=O)CN(C(c2cnc(O)n2C)=O)CC1O C1(CCNC(C2(CCOC)CC2)=O)CCN(C(=O)Cc2cnn(C)c2)C(C)C1 C1(C(=O)NCC(CNC(C(C)=C2CCCC2)=O)O)CCN(c2ccccc2)C1 c1(OC)ccc(Cl)cc1C(=O)NCC(C)(C)CN(C)C(C1CCOC1C)=O C(CC(=O)N(C(CO)C(C)C)C)(C(C)C)NC(C(C)NC(CC)=O)=O Cc1scc(C(N2CCC(N3CCN(C(C4C=CCCC4)=O)CC3)C2)=O)c1N C(CC(C)(C)C(=O)NCC(C)O)NC(c1c(C)cccn1)=O N1(C(C(C)OCCC=C)=O)CCC(CNC(c2coc(Br)n2)=O)(OC)C1 c1(C(=O)NC2CCC(N(C(c3cc(C)sn3)=O)C)C2)c(Cl)ccc(C)c1N C(=O)(C(O)C1=CCCCC1)NCCC(C(=O)NCC(CC)(CC)CO)(C)C c1(OC(C(N2CC(O)(CNC(C=CC)=O)C2)=O)C)ccc(C)cc1C CS(=O)(=O)c1ccc(C(=O)OCc2ncccc2C(F)F)o1 CCN=c1cc(-c2cn(C3CC(NC(=O)C(C)C(F)F)C3)nn2)cc[nH]1 c1(CNCc2ccc(N(CC)CC)c(F)c2)cc(=O)n2c(C)cccc2n1 C1(C2N(C(=O)Nc3c(C(=O)OC)sc(N(C)C)n3)CCC2)COCCC1(C)O C1(CCNC(C2C(C)(C)COCC2)=O)CCN(C(C2(O)COC2)=O)CCC1(F)F C(CCN=C(NCCC(C)(C)C)NC1C(C)(C)C1(C)C)SC N1(C(C2C(C=C)C2)=O)CCOC2(CCN(C(C3(COC)CCCCC3)=O)C2)C1 O=C1c2ccsc2CCC1CC(=O)NCCC1CN(C(=O)CCc2cc[nH]n2)C1 c1(C(C(N2CC(NC(C(C(C)C)NC(C)=O)=O)C2)=O)C)ccccc1S(N)(=O)=O N1(C(C(C(C)C)N(C)C)=O)CC2OCC(NC(=O)CCc3cccc(F)c3)C2C1 Cc1ncnc(C)c1CC(N1CCC(OCCNC(=O)C=CC2CCCO2)C1)=O C1(NC(C(CC)OC)=O)CCCC12CCN(C(=O)COc1ccccc1F)CC2 c1(CC(=O)NC(CC(C)C)Cn2cc(-c3nccs3)nn2)cccc([N+](=O)[O-])c1 N1(CC)CCCC(ONC(C2CCOCC2NC(=O)C=Cc2cn(C)cn2)=O)C1 c1(C(=O)NCC(C)NC(C2(CCC)CCNC2=O)=O)ccnc(O)c1F Cc1cc(C(=O)NCC(C)NC(=O)CC2NC(=O)NC2=O)n(-c2ccccn2)n1 C(=O)(CC1=CCN(C(=O)C(C)(C)CC(C)=O)CC1)NC(CCOC)C(C)C CC(C)C(CCCCl)NC1CC(C2CCC(OC)CC2)C1 CC1=C(CNC(c2nc(CNC(C3OCCC3(C)C)=O)oc2C)=O)COCC1 C1(CNC(=O)CCc2cnco2)CC2(CCOCC2)CN1C(=O)CCCC1CC1 c1(C(=O)NC2(CNC(CC(CC)C)=O)CCCC2)ccc([N+](=O)[O-])cc1C Cc1ccc(C(N2CCC(C)C(NC(=O)CCSC(F)(F)F)C2)=O)cc1C#N Nc1c(CC(N2CCNC(=O)C2c2cccc(Br)c2)=O)cccc1Br n1(C(C)C)ccnc1-c1cn(CC(C)NC(C2(C(C)(C)C)CCC2)=O)nn1 c1(CCC(=O)NCC(C)NC(c2nc(COC)sc2)=O)nnc(C)n1C c1(C(=O)NC(CCC(=O)NC(CC)CC(=O)OC)(C)C)ccc(F)c(O)c1 c1(CC(=O)NC2(CNC(C=CC(C)NC(=O)CO)=O)CCCC2)ccc(O)c(F)c1 c1(C(=O)NC2C(CC=C(C)C)CC2O)cccc(CS(C)(=O)=O)c1 N1(C(C2C(C(C)O)C2)=O)CCC(NC(c2cn3c(n2)CCCC3)=O)C12CCC2 C1(CCNC(=O)CC(C)NC(C2C(CSC)C2)=O)CCCCC1O N1(C(c2nc(OCC)oc2)=O)CC2CN(C(c3nc(Cl)sc3Cl)=O)CCC12 Cc1cc(F)cc(C(=O)NC2CN(C(c3c(O)cccc3F)=O)CC23CC3)c1C Cc1nc2cc(C(=O)NC(C3CN(C(=O)Cc4cnco4)C3)C)ccc2o1 CS(=O)CCC(=O)NCC1CCC(CNC(=O)Cc2csc(S)n2)CC1 CC1(NC(c2cc(F)ccc2F)=O)CCN(C(C2CCCCN2N=O)=O)CC1 C1(CC(=O)NCCOC2CN(C(Cc3cnn(C)n3)=O)C2)CC2(CCC2)CO1 C1(CN(C(=O)C(c2ccccn2)O)C)COCCN1C(c1ncc[nH]1)=O N1(C(c2c(CC)n(C)nc2)=O)CCC(NC(C2(C)CC2C)=O)C(CO)C1 N1(C(c2cc(SC)n[nH]2)=O)CC2(C1)CN(C(c1cccc3scnc13)=O)CCO2 Cc1cc(C)c(C(N2CC(CNC(C3(F)CC3)=O)C3(CCC3)C2)=O)c(C)n1 N1(C(C(C)=C2CC2)=O)CC(CNC(=O)COCC2CCOCC2)CC12CCC2 C1(CC=C)(NC(=O)CSC(C)C)CCN(C(c2c(C)nn(C(C)C)c2C)=O)CC1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC(CO)NC(C(C(C)(F)F)(C)C)=O C1(C(N2CCC(NC(C3(F)C(C)C3)=O)C2c2ccccc2)=O)CCC2(CC1)CC2 C(=O)(C(C)C(=O)OC)NC1CC(C(=O)NC(CCC=C)C)C1 C1(O)(C(=O)NCC2CC(COC)CN2C(=O)CCSC)CC2CCC1C2 CC1(C)CC=C(C(=O)N2CCCC(CO)(NC(C3CCS3(=O)=O)=O)C2)CC1 Cc1ccc(CC(=O)NCCOCCNC(c2occc2C)=O)c(Br)c1 C(=O)(CCN=c1[nH]c2ccccc2s1)N1C(CNC(CCC(N)=O)=O)COCC1 C1(OC)CC(C)CN(C(C2(C)CCN(C(=O)Cc3nocc3C)C2)=O)C1 c1(C(=O)NCC2(NC(C(C)n3cncn3)=O)CCOC2)csc2nccn12 CCCCC(CC(=O)Nc1ccc(C)nc1C)NC(c1cnsc1)=O C1(C(N2CCC(C)N(C(=O)Cc3cnn(C)c3)CC2)=O)CCC2(CC1)OCCO2 N1(C(CCC)=O)CCCN(C(=O)NC2(n3cc(Br)cn3)CC2)CC1 C1(NC(CCC(=O)NCCC)=O)CCN(C(=O)C(OC)OC)CCC1CO C=C(Cl)CC(C(=O)NCC(CC1CC1)CO)NC(=O)CNC(=O)CC C1(C)(C(=O)NC2C3(CC(NC(C4OCCN(C)C4)=O)C3)C2)Cc2ccccc2C1 c1(CC)c(C(=O)NCC(C)NC(=O)C=CC2C(C)C2(Cl)Cl)[nH]c(C)c1C(N)=O CC1(C)COC(C)(C(=O)NC2CCCN(C(=O)Cn3cnc(=N)[nH]3)C2)CO1 c1(C(=O)NC2(CF)CCN(C(=O)CN3CCCCCC3)C2)cc2c(s1)CCCC2 C1(CCNC(CC(CC)C2CC2)=O)CC2CCC(C1)N2C(=O)C=CC(F)F c1(C(N2CCN(C(C3CC(C)CC(C)C3)=O)CC2C)=O)cc2cc(O)ccc2[nH]1 N1(C(C(CC)C(C)(C)CC)=O)CCC2(C1)CN(C(c1cnn(C)c1N)=O)CCO2 CCCC(CC)C(=O)NC1CCC(C)N(C(=O)Cn2nnc(C)n2)C1 c1(-c2nc(C3CCN(C(C)=O)CC3)nn2CC(C)CO)cccc2sccc12 C1(F)(CNC(c2ccn(CCC)n2)=O)CCC(CNC(C2CC2[N+](=O)[O-])=O)C1 c1(CC)c(C(=O)NCc2cncc(C(=O)NCCOC(C)CO)c2)ccn1C Cc1ccc(C)c(OCCC(=O)NC(CNC(=O)CP(C)(C)=O)C(C)C(C)C)c1 N1(C(Cc2ccc(OC)cc2)=O)CC2(CNC(=O)C=C3CCCC3)CCC1CC2 c1(C(=O)NC2CN(C(CC3(OC)CCCCC3)=O)CC2O)ccc2nncn2c1 CCCCCC(O)CC(=O)N(C(C)CCNC(=O)CC1CCCN1C(C)=O)C Cc1nccc(Cl)c1C(N1CC(Cn2cc(-c3ccnn3C(C)(C)C)nn2)C1)=O c1(NCCOCCC(C)C)nc(N(CCC(C)(C)C)C)nc2sccc12 N1(C(C)=O)CCC(NC(c2ccccc2)CC2CCOC2)CC1 c1(NC(c2scc(C(=O)Nc3c(I)ccc(C)c3)n2)=O)cc(F)cc([N+](=O)[O-])c1 N(C(=NCCC1=CCCCC1)NC(c1ccco1)C)Cc1nc(COCC)on1 CCC(CC(=O)N1CC(C(N2CC(O)CC2(C)CO)=O)C(C)(C)C1)C(F)F C1(C(=O)NCC2C(C(=O)NCCc3c(C)ncs3)CCO2)CC12CCOCC2 c1(CNC(C23N(C(c4c(C)nc(CC)o4)=O)CCC2C3)=O)ccc(O)cc1C c1(C(=O)NC(C)CCN(C)C(C2(CCF)CCC2)=O)ccc(Br)nc1O C(=O)(C1=CCC(NC(c2sc(F)cc2C)=O)C1)NC(C#C)(C)C1CC1 c1(CNC(C(CCC)NC(=O)CN2C(=O)CCC2=O)=O)c(C)cccc1F c1(CNCC2CCC(F)C2)cc(O)ccc1Cl.C12(CCC1)CCCN2 c1(C(N(C2CN(C(=O)COC(F)F)CC2F)C)=O)cc(F)cc2nn[nH]c12 C1(CNC(CCN(C(=O)C=Cc2cocn2)CC=C)=O)CCCC12CCC2 N1(C(CCC2CC(NC(C3OCCN(CC)C3)=O)C2)=O)CC2CCCCC2C1C c1(C(=O)NCC(C2CCCC2)NC(C2C(C=C)CC2)=O)ccnc(Cl)c1 N1(C(CCC=C(C)C)=O)CCCC(NC(=O)Cc2cc(C)no2)CC1 c1(C(=O)NCC2C3CN(C(C(CC)C(C)C)=O)CC32)cc(C)c(C)c2ncsc12 Cc1c(C(N2CCCC2C2CCCN(C(=O)C=CCOC(C)(C)C)C2)=O)ncn1C N1(C(c2cn(CC)nc2C)=O)CC2(CC2)CC1C(=O)NC(C)(C)CC1CCC1 C1(C)(C(=O)NCCCN(C(C2CC2(C)C(F)(F)F)=O)CC)CC=CC1 N1(C(CCN(C)CCO)=O)CC2CC(NC(=O)CCc3ccsc3)C1C2 N1(C(C(C(C)(C)C)NC(C)=O)=O)CCC(C)N(C(=O)CC2CCC(=O)N2)CC1 Cc1cc([N+](=O)[O-])c(Cl)cc1S(=O)(=O)N1CC(C)NCC1C C1(C(=O)NC(C)(C)CCNC(c2ccnn2C2CC2)=O)Cc2ccncc2C1 C(CCC(O)C(=O)N1CC([N+](=O)[O-])C1)NC(C1CC(C)N(C)C1)=O C12(CNC(C(C=C)(C)CC)=O)CCCC1N(C(c1cc(CC)nn1C)=O)CCC2 c1(C(=O)NC(C2CCN(C(C=COCC)=O)CC2)C)nnc2n1CCCCC2 Cc1oc(C(N2CC3(COC(CNC(=O)C(O)C(F)F)C3)C2)=O)cc1S(C)(=O)=O c1(OCC(=O)N(CC(CNC(Cc2nnc(C)o2)=O)O)C)ccc(C2CC2)cc1 n1(CC(=C)C)nnnc1C(c1cc(C2CC2)on1)Nc1sccc1OC(C)C C1(CNC(c2snnc2C2CC2)=O)CN(C(=O)C2=COCC2)CC1C(F)(F)F O=C(CCCc1ncco1)NCCc1cc(C(=O)N(C2CCOC2=O)C2CC2)no1 C(=O)(C(CC(F)F)N(C(=O)C=Cc1cc[nH]c1)C)N(CCC(N)=O)CC C12(NC(C3CC(O)(CC#C)C3)=O)CCN(C(=O)CCC3CCCC3)CC1C2 C1(CC)CN(C(c2ccnc(OCC)c2)=O)CCC1NC(=O)CCn1cccn1 CC#CC1CCN(C(=O)C(C2CCC2)NC(C2COCC2(C)C)=O)CC1 c1(C(N(C2CCN(C(c3[nH]cc(CC)c3)=O)CC2)CC)=O)cnc2[nH]ncc2c1 CCC(CC)(CN=c1[nH]c(C2CC2)nc2c1CCC2)NCC1CC12CC2(F)F Cc1ccc(C(=O)NC2CCCCN(C(c3ccn(CC#N)n3)=O)C2)cc1F c1(C(N(C(C)CNC(c2cnc(OC)s2)=O)CC)=O)cc(Cl)ccc1[N+](=O)[O-] c1(C(=O)NCC2CN(C(C(=O)NCC)=O)CC23CC3)cc(F)c(C)cc1Cl N1(C(CNS(N)(=O)=O)=O)CCC(N(C(=O)C(F)CC2CCCC2)CCO)C1 c1(COCC)nc(-c2ccnnc2)n(C2CCCCC2C)n1 C(CCCCC(=O)NC(c1nn(C)cc1O)C)NC(C1CC(C)SCC1)=O N1(C(CS(=O)(=O)NC)=O)CCN(C(=O)C(C)C(C)(F)F)CC1c1ccccc1Cl C1(F)(CNC(CC(C=C)C)=O)CCN(C(c2cn(C(C)C)cc2C)=O)CC1 c1(C(C)C(=O)N(CCO)C(c2cccc(OCF)c2)C)ccccc1S(N)(=O)=O c1(C(=O)NCC2(C)CCN(C(COCC(=O)NC)=O)C2)cc2c([nH]1)CCC(C)C2 c1(C(=O)NC2(CC)CN(C(CCN(C3CC3)CC)=O)C2)cc(OC)c2c(c1)OCO2 C(=O)(C1CCc2nccn21)N1CCC(C(C)(C)NC(=O)Cc2cnoc2)C1 N1(C(CC(c2cccs2)NC(C)=O)=O)CCN(C(c2cscc2C)=O)CCC1C C1(NC(c2c(C(=O)OC)[nH]cc2)=O)CCCN(C(C2(C)CCCCO2)=O)CC1 CCC(C)(C)CCCC(=O)NCC1(C)CCN(C(C2CCOC(C)C2)=O)C1 c1(C(=O)NCC2CC(NC(c3ccc(CC)[nH]3)=O)C2)cc(OC)cc(Br)c1C CCC(CC(=O)NC(CC(=O)NCc1cc[nH]n1)CC(C)C)C(C)(C)C O=C(C(O)CC(F)(F)F)NCC1CCN(C(=O)CCCN2CCOC2=O)CC1 CC(CNC(=O)C(=O)NCCC1(NC(=O)C2CC2)CCC1)CN1CCCC1 C1(NC(=O)C=CC2CC2)CN(C(=O)Cc2cnc(C3CC3)[nH]2)CC1C(F)F C1(C(N(CC(C)NC(c2cc(CSCC)on2)=O)C)=O)CN2CCN1CC2C c1(CC(C)N(C(=O)C(=O)N(C)Cc2cncs2)C)ccc(F)c(F)c1 C1(F)(CNC(C=C(C)C(F)F)=O)CCN(C(c2cc(C(N)=O)cn2C)=O)CC1 N1(C(C=C(C)C)=O)CC(NC(C2(C(F)F)CCOCC2)=O)C(c2ccnn2C)C1 CC1CN(C(c2ccc(=O)n(C)n2)=O)CC1(C)CNC(=O)Cn1nnc(=N)[nH]1 N1(C(=O)COC2CN(C(=O)CSc3cn[nH]c3)C2)CCOCC1CCO C1(SC)CC(C(=O)NC(C2(C(=O)N(CC(C)C#N)C)CC2)C)C1 N1(C(C(C)OCCN(C)C)=O)CCCC(CNC(=O)C(C2CCCCC2)O)C1 Cc1ncnc(C)c1CC(=O)NCC1CCC1CNC(=O)Cc1ccc(Cl)s1 N1(C(C(C)(Cl)Cl)=O)CC2CS(=O)(=O)CC2(NC(=O)C=CC2CCC2)C1 c1(CNC(C(CC)NC(=O)CSC)=O)n[nH]c2c1CCC2 Cc1nc(CO)sc1C(=O)N(CC(O)CN(C(=O)C(O)Cc1cn(C)cn1)C)C N1(C(COCCC#C)=O)CCCC1(C)CNC(C1(F)CC(C(=O)OCC)C1)=O CC1CCN(C(C23CC2CCC3(F)F)=O)CCN1C(=O)CCc1cn[nH]c1 c1(OC)nn(C)cc1C(N1CCCC1CNC(=O)C(F)(F)c1ncccn1)=O C1(NC(c2cnc(C)s2)=O)CCN(CCNC(C2(C)CCSCC2)=O)CC1 C(Cc1ccccc1)(C(=O)NCCC(N1CCOCC1)C)OC C1(Nc2ccc(C(=O)NCC(CC(C)C)OCC)s2)CC=C(C(C)C)CC1 C1(NC(=O)COCCNC(=O)CC(Cl)Cl)CCN2CCCCC12 c1(N2CCC(N(C(C(CC)C(C)O)=O)C)C2)cc2nnc(C)n2cn1 C(=O)(CC(C)C(=O)NCC1CCC(C)CN1C(c1ccc(C)n1C)=O)OC N1(C(C(CC)=O)=O)CC(F)CC1C(=O)Nc1ncc(Br)nn1 CCC(C)C(C(=O)NCc1ncn(C)n1)N(C)C(C1CC2C=CC1C2)=O N1(C(C2N(CC)CCC2)=O)CC(CNC(c2cncnc2C(C)C)=O)CC1(C)C N1(C(CCCN(C(C)=O)C)=O)CC2(C1)CN(C(C1CC(Cl)(Cl)C1)=O)C2 n1(CC)cnc2[nH]c(=NCC(C)C(F)F)nc(N3CCC(CC(N)=O)C3)c12 c1(SC)ccc(C(=O)NC(C)CCCCNC(=O)C=Cc2sccc2C)c(Cl)c1 CC(N=c1cc[nH]cc1)C(=O)N1CCCC12CCN(C(=O)CC(C)(C)O)C2 C1(CC)(NC(C2C3CC2N(C(=O)CNC(=O)NC)C3)=O)CC(F)(F)C1 Cc1nnc(Cn2cc(Cc3[nH]nc(CC(=O)NCCOC=O)n3)nn2)o1.C(C)C c1(OCC)ccc2c(c1)CCN(CCCN(C(=O)CC(C)C)C(=O)C(F)F)C2 c1(C(C(=O)NCCCNC(C(C2CCCC2)OC)=O)(C)O)ccc(Cl)cc1 N1(C(C2(COC)CC2)=O)CCC(C2CCN(C(c3cc4cn[nH]c4cn3)=O)C2)C1 C(=O)(CC(C)(C)C(C)(F)F)N1CCC(C)C1CNC(=O)C(=O)NCC(F)(F)F C1(NC(C2CCN(C(N)=O)CC2)=O)COC2(C1)CN(C(=O)CC1COCCO1)C2 C(=O)(C#CC1(C)COC1)N(C1CN(C(c2c(C(C)C)occ2)=O)CC1(C)C)C C1(CC)CN(C(=O)CC(C)(C)N(C)C(c2cccc(F)c2N)=O)CC(CC)O1 c1(CC)cc(C(N2CCCCC(NC(C3(COC)CCOC3)=O)C2)=O)c(C)nn1 c1(C(CC)C(=O)N(C(C)CN(C)C(c2cnsc2)=O)C)ccc(Br)cc1 C(=O)(C(C)(C)CS(C)(=O)=O)N(CCCNC(C(C)N(C(C)=O)C)=O)CCO Cc1cccc(NC(C2(F)CCN(Cc3cc(C(=O)O)ccc3O)C2)=O)c1Cl C1(C(=O)NC2CCCN(C(C(C=CC)O)=O)C2C)CCOCC12CCCCC2 c1(C(CNC(CCSC)=O)N(C(=O)C(C)OCc2ccccc2)C)ccccc1 Fc1ccc2cccnc2c1CN1C(CO)CCC1Cc1ncc2[nH]cc(I)c2n1 c1(C(=O)NC2(C)CN(C(C3CC4(CCOC4)C3)=O)C2)nccc2ccsc12 Cc1cc(C2(C(=O)NCCC3CCCN(C(C4CC4(Cl)Cl)=O)C3)CC2)cc(C)c1 c1(OC)ncc(C(=O)NC2CCCC2C(N2CC3CC(C2)O3)=O)cc1Br c1(OC)ccc(CCC(=O)NCC23CC2CN(C(c2nnn(C)n2)=O)C3)cn1 CC(C)CCC(F)C(=O)NCC(C)(C)OCCNC(=O)COc1cn[nH]c1 CCC(C(O)C(C)C)NC(C1CC(CNC(=O)C(O)CC2CCCC2)C1)=O N1(C(c2n[nH]c(C)c2F)=O)CCC(CNC(=O)CN2CCC(C)CC2)C12CCC2 C(CC)(CCCO)NC(c1c(CNC(CC(=O)NCC)=O)cc[nH]1)=O C(=O)(CCC1CC1(C)C)N(CC(=O)NNC)CCNC(C1(C(=O)O)CC1)=O.C1CC1 c1(C(N2CCCC(C)(CNC(c3cn(C)nc3O)=O)C2)=O)nc2ccccc2[nH]1 C1(O)(NC(N2CC(F)(F)C2)=O)CCN(C(=O)COc2ccccc2)CC1 C(C1CN(C(C2(COC)CC(=O)C2)=O)CC1C(=O)NC1(C)CC2CCC1C2)=CC C1(OC(C(C)(C)SC2CC2)=O)CCC(OCC2CC2)CC1 CCCC(C(=O)N1CCC(C(=O)NCCc2cc(C)on2)(CO)C1)NC(N)=O C#CCC(C(=O)OC)NC(=O)C(C1(O)CCC1)NC(C1CC1(C)C)=O C1(NC(C2(C(C)C)COC2)=O)CCCN(C(C2CC(O)CN2C)=O)C1 C1(NC(C(C)OCCC(C)C)=O)CC(NC(c2c[nH]nc2C2CC2)=O)CC1O C1(CCNC(C2CSCCN2)=O)CN2CCN1CC2.c1(C(C)=O)ccc(N)c(Cl)n1 c1(NCC(C)N(C(c2c(OC)ccnc2)=O)C)ncnc2sc(C)nc12 c1(C(=O)NC(CNC(C2C(C)C2)=O)(C)C)ccc(C(O)CF)cc1 C(C(N=c1[nH]ccn2nnnc12)C(C)C)NC(c1nc(C(C)C)sc1)=O N1(C(c2cn(CC(c3cnn(CC4CCOC4)c3)O)nn2)COC)CCOCC1 c1(C(N(CC(CC)NC(=O)CC2CCCO2)C)=O)coc(CC2CC2)n1 c1(CC)n[nH]cc1C(N1CCC1C(=O)NCCCCOC(C)C)=O Cc1cc(=O)n(CCC(=O)Nc2cccc(C3CC3(F)F)c2)cn1 C1(NC(C(C2CCN(C(C3(C#N)CCOC3)=O)CC2)C)=O)CCC2CC1C2(C)C C(=O)(C=C1SCC(=O)N1C)N1C(C2(NC(C=CC=CC)=O)CC2)CCCC1 c1(NC(=O)C2=CSCS2)ccc(C(=O)O)cc1.C12C=CC(C1)NC(=O)C(=O)NC2 C1(C(C(N2C(CNC(C3CCN(CCF)CC3)=O)CC2)=O)O)CCCCCCC1 N1(C(=O)CCOc2cccc(Br)c2)CCC2(CN(Cc3cccnc3Br)C2)C1 N1(C(c2c(CC)noc2)=O)CCCC(CNC(C2(CO)CCCC2)=O)CC1 N1(C(c2cc(C)oc2C)=O)CC2CCOC2(CNC(C2CCN(C)S2(=O)=O)=O)C1 C1(NC(C=COCC)=O)CC2CN(c3nc(C(C)(C)C)nc(=N)[nH]3)CC12 C(=O)(C(CC)CC(C)C)N(C1CCN(C(c2cc(Cl)cc(C)c2N)=O)C1)CCC CC1CN(C(c2cnc(S)nc2)=O)CC(C)N(C(c2ccc(Cl)c(F)c2N)=O)C1 N1(C(C2C(OCC)C2)=O)CCCCC1CCNC(=O)C=Cc1ccc(CC)o1 c1(NC(=O)CC2CN(C(c3cccnc3Cl)=O)C2)cc(Cl)ncc1Br CC(CC(=O)NC1CC2(C1)CN(C(=O)Cc1cccc(Cl)c1F)C2)C(F)F C1(NC(c2c(C)ccn2C)=O)COC2C(NC(C3CC4(CC4)CO3)=O)COC12 Cc1ccc(CNC(=O)C(C2CCOC2)NC(=O)CN2CC3CC3C2)c(O)c1 N1(CCNC(=O)C=Cc2nccs2)CCCN(C(C2CCC2CF)=O)CC1 c1(C(=O)NCC2CC(NC(c3c(C(C)=O)ccs3)=O)C2)ccnc(F)c1Cl c1(CN2CC(N(C)C3CC3)C2)cn2cccc(Br)c2n1 Cc1cnc2n1CCN(C(=O)Oc1ccccc1F)CC2 C1(C(=O)NC23CC(CNC(c4n(CCC)ccc4)=O)(C2)C3)CCC(C)(F)CC1 CC1(C)CC(C(=O)NCCN2CCOCC2)CN(C(=O)CC(C)(C)C(F)F)C1 c1(C(N2CC3C(CNC(C(C)CF)=O)(C3)C2)=O)cc(P(C)(C)=O)cs1 N1(C(CC2N(C(C)C)CCC2)=O)CCCC(C(N2CCCCC2)=O)C1 C1(CN(C(=O)CC2CC2)C)COCCN1C(C1C2CCC1(c1ccco1)C2)=O C(=O)(C1=NNC(=O)C1)NCCN(C(c1nc(C)c(C)s1)=O)CC C1(NC(c2ccc(C)o2)=O)CN(C(c2cnc(Cl)s2)=O)CCC1CO Fc1ccc(-c2noc(-c3cccc(OC4CCCCO4)c3)n2)c(C2CCN2)c1 c1(C(=O)NC2CN(C(c3nccc(C(F)F)n3)=O)CC2O)cc2n(n1)CCCC2 N1(C(C2CCC(C)(C)CC2)=O)CCC2CCC(NC(=O)Cn3cccc3)C12 CC(Cc1ccccc1)(C(F)F)NC(C1(CN)CCC1)=O c1(OC)cc(C(=O)NC(C2CCN(C(=O)C(C)(C)c3nccs3)C2)C)ccc1O c1(CC(=O)NCC(C2CCOC2)NC(=O)Cc2cnc[nH]2)ccc2c(c1)OCO2 C1(C(CNC(CC(C)F)=O)F)CCN(C(C2(c3ccccc3)CC2)=O)CC1 C(=O)(CC(C)C(F)(F)F)NC1CC(CC(=O)NC(COC)(C)C)C1(C)C C=CCC(C)(CC)C(=O)NC1CCC(NC(c2cnc(N(C)C)c(Cl)c2)=O)CC1 N1(CC(=O)NCC)CCc2cc(-c3cccc(CC(C(=O)OCC)OC)c3)ccc21 c1(OC)ncccc1CC(=O)NCC1(F)CC(NC(c2csc(C3CC3)n2)=O)C1 C12(C(=O)NCC(=O)OCOC)CN(C1)C(=O)CONC2=O.C#CCCC N1(C(CCSCCCC)=O)CC(C(=O)NC(=O)C(CCC)N(C)C)CC1(C)C N1(C(CC2N(CC)CCC2)=O)CCC2CC1CN2C(=O)CCCN(C)C(C)=O S(=O)(=O)(c1csc(C2CC2(F)F)n1)N(CC(CC)O)Cc1ccccc1 c1(C(=O)NCC23CC(NC(C4C(OC)CCC4)=O)(C2)C3)c(C)ncnc1C N1(C(COCC#C)=O)CC(C(=O)NCCN2CCCCC2C)OC(C)C1 N1(C(C(CC#CC)NC(C2CCC(C)(C)CC2)=O)=O)CC2(CCC(=O)N2)C1 c1(C(CNC(c2n(CCOC)ncc2)=O)O)ccc(OC)c(OC)c1 c1(C(=O)NC2CC3CC2CN3C(C2CCCCC2)=O)csc2c1CCCC2 C1(NC(C2(NC(c3cc(Cl)cn3C)=O)C(C)C2)=O)CCCN2CCCC12 C1(OC)CCCCC1C(=O)NCCC(C)(C)NC(=O)CCc1cscn1 CN1CCCC1(C)C(N1CC(CNC(c2ncnn2C2CCOCC2)=O)C1)=O C1(C(=O)NCC2(C(N)=O)CN(C(=O)CCC3CCCC(=O)N3)C2)CC(F)C(=O)N1 C=CC(C(F)(F)F)NC(C1C(NC(=O)CN2CCC(OC)C2)C1(C)C)=O c1(N2C(C)CC(NC(c3cnc(Cl)s3)=O)C2)ncc(C#N)cc1Br C1(CNC(C(COCC)(C)C)=O)CC2CC(C1)N(C(c1c[nH]cc(Cl)c1=O)=O)C2 C(=O)(C1COc2ccccc21)N(C)CCNC(c1ccnc(C(F)(F)F)c1N)=O n1(CC)nnnc1C(CC)(C1CC1)NCC1CC12CC2 C12(CNC(=O)CC3CC(F)(F)C3)CCC1CN(C(=O)C(F)CC1CCCC1)C2 CC12COC(C(N3CCC(N4CCN(C(C5(F)CCOC5)=O)CC4)C3)=O)(C1)C2 C12(C(=O)NC3CC(n4cc(COC(=N)O)nn4)C3)CCCC(CC1C(=O)O)C2 N1(C(c2c(C)nc(CC)s2)=O)C(C)CC2CN(C(C3OCC4CCCC34)=O)CC12 Cn1c(O)nc2cccc(C(N3CC(CCNC(C4CCCC(O)C4)=O)C3)=O)c12 C(=O)(C1=CCCCC1)N1CC(C=C)(CC(=O)N(CC(F)F)CCOC)C1 N1(C(C2CC(C)(C)C2)=O)CCC(F)(C(=O)Nc2oncc2C#N)C1 CC1(C(N2CCCC(CNC(=O)Cc3ccc(F)cc3)CC2)=O)CCNC(=O)C1 Cc1cc(N)ccc1C(=O)NCC12CCC1CCN2C(=O)CCCNC(N)=O C1(NC(c2ccc(C)s2)=O)CC12CCN(c1ncc3c(n1)CCC3)CC2 C(=O)(C#CC1CCCCC1)NC1(C)CC(NC(=O)CC2=CCCCC2)C1 Cc1c(C(=O)COC(c2c(F)ccc(Br)c2Cl)=O)ccc(Cl)c1Cl N1(C(CCC#C)=O)CCCCC1CCC(=O)NCC(C)(C)C(=O)NC CCCCC(O)C(C)C(=O)NCCC(C)(CC)NC(=O)C(O)CCC(F)(F)F N1(CC(=O)NC2C(CNC(c3c(COC)nn[nH]3)=O)CCC2)CCNC(=O)C1 c1(CC2CN(C(=O)NC3(c4ccc(O)nc4)CCC3)C2)ccc(C(F)(F)F)cc1 C1(OC)CC(NC(c2ccc(C(C)C)o2)=O)CN(C(C2CC2Br)=O)C1 c1(N2CC(C)(C)C(NC(C3CC4CC4C3)=O)C2)c(Cl)cncc1[N+](=O)[O-] n1(C(C)C)cnnc1CC(=O)NCC(O)CN(C)C(c1cnnn1C(C)C)=O n1(CCC)cc(C(=O)N(CC(C)NC(C2CCCC2O)=O)CC)nn1 N1(C(c2n(CC)ccc2)=O)CCN(C(c2cscc2C(F)F)=O)C(C)C1 Cc1nc(CN(C2CC(C(N3CCC(CO)C3)=O)C2)C)co1 C(CC1=CCC2CC1C2(C)C)NC(c1c(C(C)C)n(-c2cccc(Cl)c2)nn1)=O Cc1nc(Cl)ccc1C(N1CCCC(n2cc(CN3CCCCC3)nn2)CC1)=O C1(C2CN(C(C3CN(C(=O)NC)C3)=O)C2)(NC(C2(C(C)C)CNC(=O)C2)=O)CC1 c1(C(=O)NCC(CNC(=O)CCC2CC2)C(F)(F)F)c[nH]c2cc(F)ccc12 c1(C(N2CCC(O)(CNC(=O)CCC3CCOC3)C2)=O)cnc2ncccc2c1 C(=O)(C(CO)C(C)(C)C)N(CCCN(C(C(C(C)C)NC(=O)OC)=O)C)C N1(C(C2CCOC(C)C2)C(=O)NC(CC)C)CC(CO)C2(CC2)C1 C1(NC(c2c(CCC)nns2)=O)(CNC(=O)CCc2ccncn2)CCOCC1 c1(C(N(CC(C)(C)NC(C2C(CC)OCC2)=O)C)=O)nc(C)n(C)c1C N1(C(CC)=O)CCC2(C1)CN(C(=O)C(C)NC(S(=O)(=O)Cc1ccccc1)=O)C2 N1(C(C23CCC(NC(CC4C(C)(C)C4)=O)(CC2)C3)=O)CCN2CC(O)CC2C1 c1(CC2(NC(=O)NC(c3cn(CC(F)(F)CO)nn3)C)CCC2)ccc(Cl)cc1 c1(CNC(c2n(C)ncc2)=O)cn(C)nc1OC(F)F C12(C(=O)NCCc3c(CNC(COCC)=O)cccc3)CCCC1C2(F)F C(c1ccc(C)s1)=CC(=O)NC1C(CNC(C2(CC#C)CCCO2)=O)COC1 CC(F)CC(=O)N1CCC(CCNC(=O)CCCF)C1 c1(NCCC(C)C)[nH]c(=NC2CSCC2C)nc2scnc12 C(=O)(C(O)C(CCC)NC(c1cc(C(F)F)[nH]n1)=O)N1CCC(F)(CC#C)C1 c1(CC)ncc(C(=O)NCC2CC(NC(c3nnsc3C)=O)C(O)C2)cn1 Cc1nc([N+](=O)[O-])cn1CC(N1CCOC(CCNC(=O)C(C)CC(F)F)C1)=O C#Cc1ccc(C(N2CCC(CC(N)=O)(NC(C3CC3COC)=O)CC2)=O)cc1 C1(N(C(=O)C(O)C2CC2)C)CC2CCC(C1)N2C(C1(C(F)(F)F)CCCCC1)=O N1(C(C(C)OCC2CCCO2)=O)CC2CC1C2CNC(=O)CC1CCOC1C C(=O)(C1c2ccccc2Oc2ccccc21)NC1C(NC(=O)CCF)C1 C1(C(N2C(CNC(=O)CCNC(c3ccco3)=O)CC2)=O)(C(=O)O)CC(F)(F)C1 C12(C(N)=O)CCCC1(C(=O)NC13COC(CNC(C4(F)CCOCC4)=O)(C1)C3)C2 CC1(C)CCC(C(=O)NCC2CCC2)(NC(C23C(=O)C4CC2C3C4)=O)C1 c1(C(=O)NCC(CNC(C2C(COC)C2)=O)OC)cc(C)nn1C1CCOCC1 C12CCC(C)N(C1)C2.c1(NC(c2cccc(SC)c2)=O)cn(C)nc1C#N Cc1cccn(CC(=O)NCC2CC(C)CCN2C(C2CCCC23CC3)=O)c1=O CC1CN(C(=O)NCCc2cnco2)CC(C)(C(F)F)O1 C1(CCNC(CC2(OC)CN(C(C3CCS(=O)CC3)=O)C2)=O)CCC(C)(C)C1 C(=O)(CCCC(CC)CC)NCC(CC(=O)NC(CC#C)CC(F)F)OC c1(OC)ccc(C2CC2)c(C(=O)NCCCCCNC(=O)C2=CCOC2)c1 c1(NCC)cc2c(C)c(Cl)ccc2[nH]1.C1CC(C)SCC(=O)N1.N(CCO)(CC)CC Cc1ccc2oc(N3CCCCC3CNC(C3C4C5CCC(C5)C34)=O)nc2c1 N1(C(c2c(C)cc(C3CC3)cc2)=O)CC2CCC1CC2NC(C1SCCCS1)=O c1(C(=O)NCC(CC)NC(=O)CCCc2nccs2)cnc(C)[nH]c1=N C1(C)(CC)CCC(C(=O)NC2C=CC(CNC(c3cncn3C3CC3)=O)C2)O1 C1(C(N2CCC(NC(c3ccc(=O)oc3)=O)(CF)C2)=O)Cc2cc(F)ccc2O1 CCCC(C(=O)NCC(O)CC(=O)NCC(=O)NOC)OCC C1(C(=O)NCCC2CCN(C(C(N3CCNC3=O)C)=O)C2)CC2(C1)CC1(CC1)C2 C1(CC(=O)NCC2N(C(CSc3n[nH]c(=N)s3)=O)CCC2)CCCC(C(N)=O)C1 C1(CCC#C)CC(CO)CN(c2nnc(CC(O)C=C)n2C)C1 c1(OC)ccc(OC)c(CCC(N2CCCC(NC(=O)CCC(F)F)C2C)=O)c1 c1(NC(C)=O)ccc(C(N2CCC(C(C)NC(c3c(C)ncn3C)=O)C2)=O)cc1 N1(C(C(c2ccc(Cl)cc2)CC)=O)CCC(NC(=O)CN(C)C2CC2)C(C)(C)C1 N1(C(C(C)Cn2ccnc2)=O)CCN(C(c2cncc(O)c2)=O)CC(C)(F)C1 c1(C(N(C2CCN(c3nncs3)C2)C)=O)c[nH]nc1C1CCOCC1 C1(C(N2CC(C)OCC2)=O)CC2CCCC2N1C(=O)CC(C)(C)C c1(NC(N(CCN(c2ccccc2)C)CC)=O)nn(-c2ccccc2)nc1C C1(CC)CN(C(C23CC(CCO2)C3)=O)CCN1C(=O)C(n1nc(C)cc1C)C C=CCC(CNC(=O)C(C)(C)C)NC(C1CCN(Cc2ccccn2)C1)=O CCCCC(F)C(=O)N1CCC(C)(NC(C2CCCN2C=O)=O)CC1 C1(C(C)C)CN(C(=O)CC2CCCC(NC(C3CCC4(CC4)C3)=O)C2)CCN1C N#CC1CCCC(C(N2CCCN(C(c3ccc(C4CC4)s3)=O)CC2)=O)C1 C1(CN(C(c2cn(C(C)C)cn2)=O)CC)CCCCN1C(=O)C(C)CSC c1(C(=O)NC(C2CN(C(C3CCCC(F)(F)C3)=O)C2)C)ccc2c(O)n[nH]c2c1 N1(C(CC(CC)C)=O)CCCC(NC(C2(C)CCOCC2)=O)C1C c1(C(N2CCCC(NC(C3CCC(OC)CC3)=O)C2)=O)ccc2ncccc2c1 C12(C(=O)NCCOCCOCC)COCC1CN(C(=O)CC1CCC(=O)N1)C2 CC1(CNC(=O)CC(C)n2cccn2)CC(NC(=O)CCOC2CC2)C1 c1(C(=O)Nc2cccc3nc(C)[nH]c32)cc(C)cc2c1NCCC2C N1(c2nc(COCC)nc(C)c2)CC2(C)CN(C(c3coc(Br)n3)=O)CC2(C)C1 c1(C(C)C)nn(C)c(Cl)c1C(=O)NCC1(NC(=O)CN2CC=CC2)CCOC1 c1(CC)cccc(CC(N2CCN(C(=O)CN(CC)CC)CC2)=O)c1 C1(CNC(c2cc(C)on2)=O)CC(C)CN(C(C2(CN(C)C)CC2)=O)C1 S(=O)(=O)(c1ccc(NC(CC2CCCCC2)CO)cc1Cl)NCC(C(C)C)(C)C Cc1cc(C(=O)NC(CNC(=O)C(C)(C)c2cncs2)C(C)C)co1 Cc1cc(C2CC2C(=O)NCCC(C)N(C)C(c2cncs2)=O)on1 c1(C(=O)NCC2(NC(c3[nH]c(=NC)sc3)=O)CCC2)c(C)nc2cccnn12 C=C1CCC(C(=O)NCc2nocc2C(=O)NC(C)(CO)C(F)F)CC1 N1(C(C(c2c(CC)cccc2)(F)F)=O)CCCC(O)(CNC(C2CC2(C)C)=O)C1 N1(C(COCCCC)=O)CCCC(NC(c2cccc(C3(C)CC3)c2)=O)C1C C12(CNC(CSCC)=O)CC1CN(C(=O)CN(c1ccncc1)C)C2 C(CCC(C)C(=O)N1CCCC(N(C)C(c2nonc2N)=O)C1)OC C1(C(=O)NC(CC=C)CC)(CC)CCN(C(C2CCCCC2O)=O)CC1 c1(C(N2CCC(C)(CNC(CC3(C)CCC3)=O)C2)=O)ccc2c(=O)ccoc2c1 c1(OC)noc(-c2nc(C3CCCC3)nn2-c2nc[nH]n2)c1Br C1(CNC(C2CCCS2)=O)CC2CCC1N2C(c1cc(Cn2cccn2)on1)=O C1(C(=O)NC2CC(NC(=O)CCCn3cccn3)C2)(OC)CCOC1 c1(C(=O)NCC(c2cccc(F)c2)NC(c2ccc[nH]2)=O)cccc2nonc12 N1(C(COC(CCC)C)=O)CCCC1(C(=O)NOCC(=O)OC)C(C)C N1(C(C2CCN(C(C=CC3(C)COC3)=O)C(C)(C)C2)=O)CCCC12CCNC2=O C1(C(=O)NC2C(C)CN(C(c3cnn(CC(F)F)n3)=O)C2)CCCCC1(F)F c1(C(=O)NCCN(C(c2cnn(C(C)C)c2Cl)=O)CC)[nH]c(C)nc1C N1(Cc2c(C)nc(-c3ccc(OC)cc3)s2)C(=O)CCN(CC2C3CCC23)C1=O c1(C(=O)NC(CC2CCOC2)C(=O)O)ccc(C(F)(F)F)c(Cl)c1 C1(C(N2CC(N(CC)CC)C2)=O)C2CC(O)C(C2)N1C(=O)CSCC(C)C c1(C(=O)NC(CN(C(c2ccc(O)nc2Cl)=O)CC)C)cc(O)ccc1Cl c1(C(N2CC3CC(CNC(C4(C)CCCCO4)=O)C3C2)=O)ccc2cncn2c1 C(=O)(CC(C(F)F)C(=O)OC(C)(C)C)NCCCC(C)NC(C1(C)CC(=C)C1)=O C1(C(=O)NC2CCN(C(C=CC)=O)C2Cc2ccccc2)CCCC2(CC2)C1 C1(CNC(Cc2cn(C(C)C)nc2)=O)CCCCN(C(c2ncccn2)=O)C1 C1(C(=O)NC(c2cccc(C)c2)C)CN(C(C2CC3(CSC3)C2)=O)CC1(F)F c1(C(=O)NCCC=C)n[nH]c2ccc(-c3cnn(CCCNC(C)=O)c3)cc12 C(=O)(CC(O)CC(C)(C)C)N1CCCCC(N(C(C(=O)NCC)=O)C)C1 N1(C(c2c(F)ccc(C)c2)=O)CCC2CCN(C(C3CCCN3C=O)=O)C2C1 c1(C(N(CCN(C(C2CC(=O)N(O)C2)=O)CC)CC)=O)cc(CC(C)C)nc(O)c1 c1(C(=O)NC(CCNC(c2n[nH]c(C)c2F)=O)(C)C)nc2c(s1)COCC2 C#CCC(C)(C)C(=O)NCC(CC=C)C(=O)N1CCC(n2cncn2)C1 CC1Cc2n[nH]cc2CN(C(c2cc(Br)c(F)cn2)C(=O)NCC2CCCO2)C1 c1(C(=O)NC(CCCNC(c2c(CC)occ2)=O)C)ccc2ccccc2n1 N1(C(CN2CC(C)(C)C2)=O)CCCC2CN(C(c3cccc(=O)o3)=O)CC12 C1(C(N(CC)CC)=O)CCN(C(=O)CC2(N(C)C)CCC2)C12CCC2 CC(C)CC(C(=O)NCC1CNC(=O)CO1)NC(c1cccc(=O)o1)=O c1(OCC)ccc(C(=O)Nc2nccc(C#N)c2OC)c2ccccc12 c1(CNC(C(CN(C(C(CC)(F)F)=O)C)C)=O)cccc(F)c1C CN1CCN(C(=O)OC(C)(C)C)C(C(=O)Nc2c[nH]c(CNCC3CCC3)c2)C1 C(=O)(CCC(=O)NC(CO)C(=O)NC(C1CCCC1O)C)NCCC Cc1cc(C(=O)NCC(O)CC(=O)NCCCC(O)CO)cnn1 N1(C(C2(C)CCC(F)(F)C2)=O)CC2(CCCN(C(c3nocc3Cl)=O)C2)C1 C1(NC(c2n(CCCSC)nnn2)(C)CCBr)CC12CCCCC2 C1(NC(CCC#C)=O)CCN(C(=O)C(C)NC(C)=O)C2CC12 C1(NC(C(CC)N(C)C)=O)CC(F)CN(C(=O)Cn2nc(C)cc2C)C1 C(=O)(C1=CCCSC1)N(CCNC(=O)C(c1cccc(F)c1)O)CC C(=O)(C1=NOC(CNC(=O)C(COC)N=[N+]=[N-])C1)N(CCOCC#C)C c1(CNCC23C(CN(C(c4cc(C)on4)=O)C2)C3)cc(F)c(Cl)cc1Cl C1(S(C)(=O)=O)(C(=O)NCCN(C(=O)CC2CCCS2(=O)=O)C)CCC1 c1(OC)cc(N)c(Cl)cc1C(=O)NCC(C)(CC(C)C)NC(=O)C=CS(C)=O CC(C)C(C(=O)NC12CC1CN(C(=O)CCCCC1CC1)C2)c1ccccc1 C1(C(=O)NCC2(CNC(CC)=O)CCCC2)CCCCC1C1CC1 c1(C(=O)NC2(C)CN(C(CC3(CSC)CC3)=O)C2)ccnc(-n2cncn2)c1.C CC1CN(C(C23CC(F)(C2)C3)=O)CC(CCNC(c2cc(Cl)cn2C)=O)O1 CC1(C)CC(NC(=O)CCC2CCC(=O)N2)CN(C(C2(C(F)(F)F)CCC2)=O)C1 Cc1cnc(C=CC(=O)NCC(C2CCOC2)NC(c2cc(C)c(Cl)s2)=O)[nH]1 N1(C(CCC)=O)CC(C(F)(F)F)OCC1CNC(=O)CCc1cccc(O)n1 C1(C(N2CCC(SC)C2)=O)CN(C(C2CC3(CCC3=O)C2)=O)CC1(F)F C(=O)(C1CCCc2nncn21)NC1(CNC(C(C)OC2CCCC2)=O)CCC1 N1(C(COCCC#C)=O)CC2(C1)CN(C(C1CC1F)=O)C2 C(=O)(C1CCCc2cncn21)NC1CCC(N(C(=O)Cn2cnnc2O)C)CC1 N1(C(=O)CC2COCCN2C(c2ccc(O)nc2)=O)CCc2ccsc2C1 N1(C(CNC(C(CC)(F)F)=O)=O)CC(C)OC(C)C1 C1(C(N(CC(CC)(F)F)C)=O)CCCC(NC(C2CC(C)CCO2)=O)CC1 N1(C(CCC(C)SC)=O)CCOCC(CNC(c2ccc(C(N)=O)o2)=O)C1 N1(C(c2snc(C)c2N)=O)CC(F)(F)CC1C(C)(C)O.C1CCN1 c1(C(=O)NCCN(C(c2c(C)snn2)=O)C)ccnnc1NC1CC1 c1(NC(C2CC3CC3N2C(c2sc(Br)cc2Br)=O)=O)cc(Cl)cc(Cl)c1F c1(CC(=O)NCC2N(C(c3cccc(OCC)c3)=O)CC2)ccc(C)c(F)c1 CCC(C)(CC(=O)OC)NC(C1CC(=O)N(c2ccccc2)C1)=O CC(c1ccsc1)=CC(=O)NC(C)CN(C(=O)CC1(c2cccnc2)CC1)C N1(C(=O)Nc2cn(-c3cccc(C)c3)nc2)CCCc2c(N(C)C)cccc21 C1(NC(c2ccnn2CC(F)F)=O)CCN(C(=O)C2=COCCC2)C12CCCC2 c1(CNC(=O)NC2C(OC(C)(C)C)CCCC2)cccc([N+](=O)[O-])c1 C1(C2CCN(C(c3nncs3)=O)CC2)(NC(=O)COCCF)CCC1 C(=O)(CC(C(F)(F)F)NC(c1cc(Cl)n(C)n1)=O)NCC1(CC)CC1 C1(Nc2nc(C(CC)C)nc(C)c2)CCC2CN(C(=O)CC3=CCOCC3)CC12 c1(C(=O)NC(CNC(c2ncn(C(C)C)n2)=O)C)ccccc1F c1(C(=O)OCC)ccc(C(N)=O)cc1.c12ccccc1COC(=O)CO2 C1(C(=O)NC(CNC(C2(CCN(C)C)CC2)=O)C(C)C)(CC)CCCO1 c1(NC(C2(NC(C3CCCC(OC)C3)=O)CCCC2)=O)cc(Cl)cnc1O Cc1c(C(=O)NC2COCC2NC(=O)C(C)(O)C2CCC2)ccn1C(C)C C(=O)(C(O)CC[S+](C)C)N(C)CC1CCN(C(C2(CCC=C)CC2)=O)CC1 C(=O)(CC(C)CNC(c1cc[n+]([O-])cc1)=O)NCc1cnc(C)o1 C1(OC)CC(NC2(C)CCN(C(=O)OC(C)(C)C)C2)C12CCCO2 C1(CC)(CNC(C2CC3CC3C2)=O)CCN(C(C2CCN2C(C)(C)C)=O)CC1 C1(CNC(c2cnc(C(=O)OC)s2)=O)CN(C(=O)C2=NOC(C)C2)CC12CCC2 c1(C(C2(C)CCCS2)(c2nnnn2C2CC2)CNCC)cc(C(F)(F)F)ncc1F N#CC1(CC(=O)NCC=CCNC(=O)CCNC(=O)Cc2ccccc2)CCC1 C1(CCNC(Cn2cc(C(C)O)nn2)=O)CSCCN1C(=O)CC1CCCOC1 CCC(C)(CC)C(=O)NCC12CC(CO1)N(C(c1cc(F)cnc1Cl)=O)C2 C=CCC(CC)C(=O)NCCOCCN(C(=O)Cc1cc(C)cc(C)c1)C C1(NCc2nccc(C)n2)CC(=O)N(c2cccc(C(C)C)c2)C1=O c1(SC)cccc(CNC(c2nnnn2C2CC2)c2ccno2)c1 CC(C(=O)NCCCNC(C1(CO)CCOC1)=O)C(=O)N1CCOCC1 C(CN(C)C)(CC(C)C)N(CC)CC.C123COC(C1)(C2)CNC(=O)C3 N1(C(C2CCN(C)C2)=O)CC2(CC(CNC(c3ccccc3CO)=O)C2)C1 N1(c2n(Cc3cc(C(C)(C)C)no3)nnn2)CCC(O)(C2CCC2)CC1 c1(C(N2CCC(O)(C(C)NC(C(C)N(CC)CC)=O)C2)=O)ccn2nccc2c1 O=C(C1=CCCOC1)NCC1CCCC1C(N1CCOCC2(CC2)C1)=O c1(OC)ncnc(C(N2CCC(NC(=O)C=Cc3ccccn3)C(C)C2)=O)c1F C1(NC(COCCOC)=O)CC12CCN(C(c1cnc(Br)o1)=O)CC2 C(=O)(C(F)CC(C)(C)C)NC1(COC)CCN(C(=O)Cc2sc(O)nc2O)C1 C(=O)(C(C)(C)C1=CCN(C(=O)CCC2OCCO2)C1)NCC(C)CC1CC1 c1(CC)ccc(CN(C)C(c2sc(-c3ccccc3O)nc2C)=O)cc1 Cc1n[nH]c(=NCC(CNC(=O)C(c2ccc(F)cc2)(C)O)C(F)(F)F)o1 N#Cc1ccc(C(=O)NCCC(O)CNC(=O)CCOCC2CC2)s1 C1(CNC(c2sc(CC)c(C)c2)=O)CC(C)(C)CN1C(C1CCCC(C)(C)C1)=O Cc1cc(NC(C2CC(F)CN(C(=O)Cc3cnc(C)s3)C2)=O)cc(Br)c1 CC(CC(=O)NC(c1ccccc1F)CNC(=O)C#CC1CCC1)C(C)(C)C C1(C(N2CC(N3CCNC3=O)C2)=O)CCC(C2CC2)N1C(=O)COCCCF.CO c1(C(=O)NCC(C)N(C)C(C2CC(C)(C)CN2C)=O)nc[nH]c2ncnc1-2 C1(N(C(C)=O)Cc2ccccc2)CCCN(CC(c2cccc(O)c2)O)C1 N1(C(c2n(CCC)nc(C)c2)=O)CCOCC(CNC(c2cnsc2C)=O)C1 Cc1cnc(C(=O)NC2C3CC2CN(C(=O)CCc2nc(=N)[nH][nH]2)C3)cc1C c1(C(=O)NCC2CCN(C(C3(F)C(C)OCC3)=O)CC2)csc2ccncc12 Cc1nc[nH]c1CC(=O)NCC=CCNC(=O)CC(C)N(C)C c1(CC)cc(NC(=O)C(C)(C)CCNC(=O)CN2CCCC2C)cc(O)c1 N1(C(CCC#C)=O)CCC2(CC2C(=O)NC(CN(C)C)C(C)(C)C)C1 C(=O)(C(O)C1=CCCCC1)NC(C(NOCC(=O)OC)=O)C1(C)CC1 O=S1(=O)C=Cc2ccc(CNCc3ccc(-c4ccco4)nc3)cc21 C1(C(C)(C)C)CCCCN1C(C1(NC(=O)CC2(O)CCCCC2)CCC1)=O C=CCC(C(=O)NCc1cc[nH]c1C(=O)NCC(C)CCC)C(C)C C1(NC(C(C)SC(F)(F)F)=O)C2CC3CN(C(=O)C=C4CCN(C)C4)C1C3C2 n1(C(CC)CC)ccc(C(=O)NCC(C)(O)CNC(c2ccc(C(C)=O)[nH]2)=O)n1 N1(C(C(C(C)(C)C)CNC(C2(Cl)CC2(F)F)=O)=O)CCN2C(=O)OCC2C1 c1(C(=O)NCCC(CNC(CC(CCC)C)=O)O)ccc2oc(C)nc2c1 N1(C(C(C)(C2CC2)OC)=O)CCOCC(C(=O)NC2(CCO)CCCC2)C1 CC1(C)CN(C(=O)C2=COCC2)CC1CNC(=O)C=Cc1ccsc1Br S(=O)(=O)(c1ccc(N(CC(C)OC)C)c2cnccc12)NC1C(CC)OCCC1 CC1CCC(CN)N(Cc2cccc(C(=O)NC(=O)OC(C)C)c2)C1 c1(C(N2CCC(NC(c3nc(C)oc3)=O)C2)=O)cnc2ccoc2c1 Cc1ccc(NC(=O)C(=O)NC(CO)C(C)NC(=O)C(n2cc(Cl)cn2)C)cc1 C(=O)(C(C)(CCC)CCC)N1CCC(OCC(=O)NC(CC#C)CO)C1 N1(C(c2cccc(C(=O)NC)c2)=O)CC2CN(C(C3(C(N)=O)CCC3)=O)CC2C1 Cc1cnc(NC2CC(CNC(C3(C)CCCNS3(=O)=O)=O)C2)nc1S(C)(=O)=O Cn1ccc(C=CC(N2C(C(=O)NCCC(=O)NC3CC3)CCC2C2CC2)=O)c1 c1(C(N(CC(CC)NC(=O)CC2CCCOC2)C)=O)ccc2cnccc2c1 C1(C(=O)NCCCCCN(C(c2cc(OC)no2)=O)C)CNC(=O)C(C)(C)C1 c1(OCC)ncc(C(=O)NC2CN(C(=O)C=C3CCC3)CC2C)cn1 C1(NC(c2csc(C(F)(F)F)n2)=O)COCCN(C(=O)C(F)(F)C2(O)CCC2)C1 c1(NC(COC)C)nc(CO)no1.c12nnnn1CCCCC1CC(C1)C2SC C(CCC(=O)NC1(CNC(=O)C(C)NC(=O)CC)CCCC1)OCCC C1(C2(NC(=O)Cc3ccns3)CC2)CCCN1C(C1CC2(CC2)C1)=O C1(C2(O)CN(C(=O)C(CO)C(C)C)C2)(CNC(c2c(C)ccc(N)c2)=O)CC1 c1(C(=O)NCC)ccc(CN(C)Cc2ccccc2F)cc1.N12CCCC1C2=O C1(C(=O)NC2C(NC(c3cc(C)ns3)=O)CCOC2)CCc2nc(C)[nH]c2C1 c1(C(=O)NC(CNC(C(C=C)O)=O)C2CCC2)cccc(C(F)(F)F)c1 C(=O)(C(O)CCC(C)C)NC1(C(=O)NCCCCC#C)CCSC1 C1(CNC(CNC(C)=O)=O)CC2(CCN(C(=O)C=C(C)c3cnn(C)c3)C2)CO1 Cc1noc2nc(C(C)C)cc(C(=O)N(C)CCNC(C3C4CCCC34)=O)c12 c1(C(C2CCOCC2)O)nc(Cn2nccn2)n(-c2ccnc(O)c2)n1.C1(C)CC1 c1(C(=O)NC2(C)CC(NC(CCNC(=O)NC)=O)C2)cnc2c(cnn2C)c1 c1(OC)ccc2cc(C(=O)NC3CN(C(C4(CO)CCC4)=O)CCC3O)[nH]c2c1 c1(CC(=O)NCCCN(C(=O)C(C)C(F)F)CC)cc(C(F)(F)F)cc(Cl)n1 c1(C(=O)OC)nccnc1C(=O)N(C)CCN(C(=O)CC1C=CCC1)C(C)C C(=O)(C(C)(C)CC#N)N1CCC(N2CCN(C(Cc3cnn(C)n3)=O)CC2)CC1 c1(C(N(C(C#C)C)C)=O)cc(CNC(c2cc(C(N)=O)co2)=O)no1 Cc1ccc(-n2cc(C(C)NC(=O)CC3CC4CC4C3)nn2)nc1 c1(CC)cc(C(=O)NC2CC3CC2N(C(C24CCC(OC)C2C4)=O)C3)cc(O)n1 C1(C2CCN(C(c3ccn(CCF)n3)=O)CC2)(NC(C2CC(OC)C2)=O)CCC1 C1(N(C2CCOC2)C(=O)COCC2CN(CCC3CC3)C2)CCCCCC1 C1(NC(C2(C)CC=CCC2)=O)CCN(C(c2ccc(O)c(N)n2)=O)CC1F C1(CC(N2CC(CN(C(C=CC(=O)OCC)=O)CC)C2)=O)CCCC(F)(F)C1 CCCC(C)(CCC)C(=O)NC(CC1CC1)C(=O)N(C)Cc1cccc(O)c1 N1(C(c2c(OCC=C)cccn2)=O)CCCCC(NC(=O)CCCC(=O)OC)C1 N1(C(c2[nH]cc(C)c2)=O)CCC2CCCN(C(c3nnn(C)c3N)=O)C2C1 C1(C(C)C)CC(C(=O)N(C)Cc2cn(-c3ccccc3Cl)nn2)CCO1 c1(C(=O)NCCN(C(=O)CC2(COC)CC2)CC)ccc(C(C)C)nc1C N1(c2nc(C)cc(OC)n2)CC(NC(=O)CN2CCCCCC2)C2CCCCC12 C(=O)(CCOC1CN(C(=O)Cc2ccsc2)C1)NCC(C)CC1CC1 C1(C)(CC)C=C(C(=O)N2CCC(CC(=O)NCC(F)(F)C(F)F)CC2)C1 c1(NC(CNC(C=Cc2n(CC)ncc2)=O)C)c(F)cc(C#N)cc1[N+](=O)[O-] c1(C(=O)NCC2OCC3(CN(C(C(C)C(C)O)=O)C3)C2)c(F)ccc2occc12 N1(C(Cc2cccc(C)c2)=O)CCCC2(CCN(C(C3CC4(CCC4)C3)=O)C2)C1 N1(C(C2CCC3(CC3)N2C(C2CC(O)C(F)C2)=O)=O)CC=CC12CCOCC2 C12OCCC1CNC2=O.C1(CNC(C2(CCC)CCC2)=O)CCC1(OC)OC C1(NC(c2c(CC)oc(C)c2)=O)CCN(C(=O)CC2CSCCO2)CC1(C)C C1(CC)CCN(C(=O)C(O)c2ccco2)C1CNC(=O)CC1CC(C)=NO1 c1(OCC=C)cccc(CN2CC(NC(c3ccc(CC)o3)=O)C(F)C2)c1 c1(CCOC)ncc(C(C(=O)NC2(C)CC2)N(C2CC2)Cc2cn[nH]c2)s1 n12nnc(c1C#N)OC(=O)C2.C1(NC(C)(C)C)CC2(CCC2)C1 c1(C(N2C(C(=O)O)CSC2c2ccncc2)=O)sc2sccc2c1Cl N1(CCOC)CC(C(=O)NC2C(C)CCC2)CC1=O.C(=O)(C=CCOC)NCC Cc1nc(CC(C)C)oc1C(=O)N(C(C)CCNC(=O)CNC(N)=O)C N1(C(CC2(OC)CCC2)=O)CC2CC1CN(C(c1c(C)ccc(F)c1O)=O)C2 C(=O)(CN=c1ccc(Cl)n[nH]1)N1C2CN(C(C3CCCC4(CCC4)O3)=O)CC1CC2 N1(C(CNC(C2C(C)C2)=O)=O)CC(NC(=O)C2=NOCC2)C(N=[N+]=[N-])C1 C1(NC(c2cc(N(C)C)ncc2)=O)CCCCCN(C(C2CCCCC2)=O)C1 C1(C(=O)NC2(CC(=O)OC)CCC2)CN(C(c2cnccn2)=O)CC(C)O1 C1(C#N)(C(N(C2CCN(C(C3COCCO3)=O)CC2)C)=O)CC2CCC1CC2 c1(SC)cccc(CC(N2CCCC(Cc3cnc(C(C)(C)C)nc3)C2)=O)c1 c1(OC)ccc(C)cc1C=CC(=O)N(CC(C)NC(=O)CC1C(=O)NN=C1C)C C12(C(=O)NC3C(NC(c4ncccc4O)=O)CCOC3)CCC(CC1O)C2 CCCCC(O)CC(=O)NCCN1CCCN(C(c2cc3sccc3s2)=O)CC1 CC1CCC(S(=O)(=O)NC(c2cccc(F)c2)c2nccn2C)C1 c1(OC)cc(C(N2CCCC(NC(C3CC(C)C3)=O)C2)=O)ccc1C CN1CCC(C#N)(C(=O)N(C2CC(NC(=O)C(C)(F)F)C2)C)CC1 C1(C(N2CC(OCC(=O)NCCc3ccccn3)C2)=O)CC2CC1CC2=O c1(C(=O)NCC2C(NC(CC3CCN(C)C3)=O)COC2)c[nH]c(=O)c2ccnn12 c1(CCC)cc(CNC2(CC(F)F)CCC2)ccc1O CCC(C)(C)C(O)C(=O)NCC1(CNC(c2cc(CO)[nH]n2)=O)CC(F)(F)C1 CC(CC(=O)NC(CNC(=O)COc1c(F)cccc1F)C1CC1)CC(F)(F)F Cc1ccc(SCC(=O)NC2CCC(N(C)C(c3c[nH]c(Br)c3)=O)C2)cc1 C(=O)(C#CC1CCOC1)N1CCN(C(CN(C2CC2)CC)=O)CC1CC1CC1 N1(C(CC)=O)Cc2ccccc2C(CNC(c2cnc(O)n2C)=O)C1 N1(C(CCC(C)NC(C(CCC)C#N)=O)=O)CCCC12CCOCC2 C1(CCNC(c2cnc(C(C)C)[nH]2)=O)CN(C(c2cc(CO)[nH]n2)=O)CC(C)O1 N1(C(CCOCC(C)C)=O)CCC(C2CCN(C(=O)Cc3cnc[nH]3)C2)C1 C1(C(=O)Nc2ccc(C#C)nc2)CCCCCCN1C(=O)CC1CCCOC1 N1(C(c2c(C(C)=O)cccc2)=O)CCOC(C)(CNC(=O)CCn2cnnn2)C1 C=CCCC(F)(F)C(=O)NC(CCC)CCCNC(c1[nH]nnc1C1CC1)=O c1(C(=O)NC(CNC(c2[nH]nc(OC)c2Cl)=O)C)ccc(C)c(F)c1Br c1(C(=O)Nc2cccc(NC(C3(SC)CCC3)=O)c2)nccc2c(C)cccc12 N1(S(CC)(=O)=O)CC(C(=O)NCc2ccccc2F)Oc2ccccc21 c1(C(=O)NC(C(C)C)CNC(C2C3(CC3)C23CC3)=O)cc([N+](=O)[O-])cc(Cl)c1Cl N1(C(CCCOC)=O)CCN(C(=O)C(C)NS(C)(=O)=O)C(C2CC2)C1 c1(OCC(=O)N(CC(C)NC(CSCC#C)=O)CC)ccc(F)nc1 C1(CC(=O)N(C2CC(NC(=O)CCC3CC(F)(F)C3)C2)C)COC(C(F)(F)F)C1 C1(CNC(C(CC)OC2CCCCC2)=O)CC2CCCCC2N1C(=O)CCOC C12(CC(=O)N(C3CCCN(C(=O)CS(=O)(=O)N(C)C)C3)C)CC3CC(CC(C3)C1)C2 Cn1nc(C(=O)NCC(C2CC2)NC(c2c(Cl)n[nH]c2C2CC2)=O)cc1CO c1(C(=O)NCc2oc(C)c(C(=O)O)c2)cc2c(s1)CCC2=O CCC(N=c1[nH]c2c(c(=NCc3cc(Cl)cc(Br)c3)[nH]1)CCCC2)C1CCCC1 C(=O)(C1=C(C2CCNC2)N(c2ccc(Cl)cc2)C(=S)NC1c1ncco1)OCC c1(C(=O)NCCOC2CN(C(C3(C)CCOCC3)=O)C2)cnn2c1OCC(F)C2 c1(-c2nc(C(C)OCC)nn2CC)cc(C(F)F)ccc1F C1(C(=O)NC(C2(O)CCN(C(c3cnc(N)cn3)=O)C2)C)Cc2ccccc2O1 C1(C(C(=O)N(CCCCN(C(C(c2cnccn2)C)=O)C)C)F)CCCCC1 CCCC(CNC(c1c(C)ccn1C)=O)C(=O)NC(C)CC(C)(C)OC c1(C(=O)NCC2CC(C)N(c3ncc(F)cn3)C2)cnc(N)c(N)c1 O=C(CC1CCc2ccccc21)NC1(CNC(C2CC2C2CCCC2)=O)CC1 c1(CC(=O)NC2(CNC(C3CC(F)C(=O)N3)=O)CC2)c(F)cncc1Cl N1(C(CCC(C)N(c2ccccc2)C)=O)CCN(C)C(CN2CC(F)CC(F)C2)C1 N1(C(=O)COC2CCC(F)(F)CC2)CC2CN(C(=O)CC34CCCC3C4)CC2C1 N1(C(CC(CC)C2CC2)=O)CCN(C(c2csc(C(C)(C)C)n2)=O)CC1C(F)F C(=O)(CCC(C)(C)F)NCC(C)NC(=O)C(c1ccccc1)N(C)C c1(C(N2CC(CNC(c3n(OC)cnc3C)=O)C3C2C3)=O)cnc2[nH]cnc2c1 Cc1cn(CC(=O)NC2CCCC2NCCN2CCCOCC2)c(=O)nc1O C(=O)(C1=CCSC1)N(CCC)CCNC(=O)CNC(C)=O.N1(C(C)=O)CCCCC1 C1(N(C(=O)CCc2cnco2)C)CCCN(C(=O)C(c2cccnc2)N(C)C)C1 Cc1nn(C)c(CC23OCC(Cn4cccn4)C(C2)C3)c1Cl.n1(C)cc(C)nn1 CC1CN(C(=O)CCc2nccs2)CC(C)N(C(c2ccc(C3CC3)nc2)=O)C1 C(=O)(C(C)(C)CC(=O)N1CCC(CN(C)C(c2nccc(F)c2Cl)=O)C1)OC c1(C(N(CC(C)CNC(=O)C(C)C=Cc2ccccc2)C)=O)nnc(O)cc1O c1(OC)cccc(CNC(c2cc(-c3ccc(CCCCO)cc3)ccn2)=O)c1 C(C(=O)N1CCC(C(N2CC3CC3(CO)C2)=O)(CC)C1)(C(C)C)SCC c1(C(=O)NCC(CNC(COC)=O)F)cnc(NC(=O)OC(C)(C)C)cn1 N1(C(C=C(C)C2CC2)=O)CCOC(C(C)NC(C2CCN(C)C2)=O)C1 N1(C(=O)CC2CC(Cl)(Cl)C2)CCc2ccc3ccccc3c2C1 N12CCOCC1CC2=O.C1(COC(=O)CC2CSC2)C=CCOC1 C=CCC(CN)C(=O)N(c1ccc(-c2cncnc2)cc1)C C(=O)(C#CC(C)C)N1C(C(=O)NC(CCC)c2nn[nH]n2)CC1C c1(C(=O)NC(CC)CN(C(=O)C(CCSCC)OC)C)ccc(O)nc1C C12(C(=O)OC)CCCCC1(C(=O)N(Cc1ccco1)CC1CCCO1)CC2 CCC(C)CCCC(=O)N1CCOCC1CNC(=O)CCCC(N)=O CCCC(CC(C)C)C(=O)NC1CCN(CC(C)CC)CC(C)(C)C1 C(=O)(C1c2c(Br)cnn2CCN1Cc1nc(C)c(C)[nH]1)OC C#Cc1cncc(C(=O)NC(C)C=CC(=O)NC(c2ccccc2)CC)c1 C1(C(=O)NCC(=O)NCC2(Sc3ccc(Cl)nc3)CCOC2)Cc2nncn2C1 C(=O)(CC(C)(C)C#N)N1C(CCCNC(C(C)Cc2ccc(F)cc2)=O)CCC1 C(=O)(NNc1cc(C(F)(F)F)nc(CO)n1)Nc1c(OC)c(N)ncn1 c1(OC)ccc(C(N2CCC(NC(c3cc(Cl)cc(I)c3)=O)C2)=O)c([N+](=O)[O-])c1 CC(C)(O)C(F)C(=O)NCC(O)CC(=O)NCC(O)CNC(N)=O C1(CNC(C(CC)O)=O)CCC(NC(c2cnc(C(C)(C)C)s2)=O)CC1 CC1CC(N2CCC2)CN1C(=O)CC1CCCC1.N12CC(C1)C2=O Cc1ncc(C(=O)NCC2(F)CCN(C(=O)CN3CC(=O)NC3=O)C2)n1C c1(C(N(CC(O)CN(C)C(C2CCOC2)=O)C)=O)cn(C)c(=O)c2cncn12 CC1CC(C(=O)N(C)Cc2ccncc2F)CN(C(C2C=CCS2)=O)C1 OCC1(c2ccccc2)CCC(NCCCOC2CCOC2)CC1 C(C(CO)(CO)NC(=O)C=CC=Cc1ccccc1)N(C)C(C1CCC2CC12)=O C1(NC(c2c(C)n(C)nc2)=O)CC1C1CCN(C(C2CCOC(=O)N2)=O)CC1 c1(NC)ccc(F)cc1C(=O)NC(CNC(=O)C(C)=C1CCC1)C(C)C N1(C(c2occ(C)c2C)=O)CCCC(CNC(c2cccc(C(N)=O)n2)=O)CC1 c1(C(=O)NCC2CN(C(C3(CC(C)=O)CC3)=O)CC2C)cc(F)c(F)cc1F C(CC(C(C)C)NC(C1CC1c1cccs1)=O)N(C(c1c(C)snn1)=O)C C(=O)(C(=O)CC(C)C)NC(CCOCC)C(=O)NC1CCCC1C(N)=O c1(C(=O)NCCC2(CNC(C3C(CC)C3)=O)CC2)cc2n(n1)CCCC2O CCCCC(O)C(C)C(=O)NC1(CCC)CCN(C(=O)CC2(O)CCC2)CC1 N1(C(C2(OCC)CCOCC2)=O)CC2CN(C(c3cncc(O)c3)=O)CC2(C)C1 Cc1cc(C(N2CC(CC(C)NC(c3cc(CO)[nH]n3)=O)C2)=O)c(F)cc1Cl C(CCCC(=O)N(CCCN(C)C(c1scnc1C)=O)C)OCC c1(CC(=O)N(CC(C)O)CCNC(C2ON=C(CC)C2)=O)ccc(Cl)nc1C c1(C(N(CCN(C(C23C(C)OC(CC2)C3)=O)C)C)=O)ccc2cccc(F)c2n1 CCCCC(C(=O)N1CC2CC2C1CNC(=O)C=C(C)C)C(C)C C1(NC(C2CCC2)=O)CCC(O)CN(C(C2OCCOC23CCC3)=O)C1 N1(C(c2nn(CC)c(C)c2)=O)CC(NC(C2CCOC(=O)N2)=O)CC1(C)CC Cc1nc(C)c(C(=O)NCCN(C)C(c2cc([N+](=O)[O-])c[nH]2)=O)c(C)n1 N1(C(C(C(C)C)CO)=O)CC(C)OC2(CCN(C(=O)CC3CC(C)(C)CO3)C2)C1 C1(C(=O)NCC(C(=O)OC)C)CCC2CCC1CN2C(=O)CCCn1cccc1 c1(C(N2CCC(N(C(CCC(=C)Br)=O)C)C2)=O)cc(-n2ccnn2)ccc1F C1(NC(N2CCOC(C3CC3)CC2)=O)CC[Si]2(CCCC2)CC1 c1(C(N2CCCC(CCNC(C3COC(=O)O3)=O)C2)=O)ccc(Cl)nc1O N1(C(c2ccc(=NC)[nH]c2)=O)CC2CCC(N(C)C(c3cc(C#N)c[nH]3)=O)C2C1 c1(OC)ccc2c(CCNC(=O)C(N3CCCC3c3ccccc3)=O)c[nH]c2c1 C1(C(=O)NC2(C)CC(F)(F)C2)CC(NC(=O)Cn2cccnc2=O)C12CCC2 N1(C(C2(NC(C)=O)CCC2)=O)CCC(CCC(C)(C)NC(=O)C(O)C(C)C)CC1 C(CNC(c1ccncc1OCC)=O)(CC(F)(F)F)NC(C(C=C)OC)=O c1(C(=O)NC(C2CN(C(C3(F)CCOC3)=O)C2)C)cc(-n2cnnc2)ccn1 c1(C(CNC(C=CCNC(CN(CCC#C)C)=O)=O)C)ncc[nH]1 C1(CCC(=O)NCCCSCC)CCCN(C(=O)C(O)C2CCCC2)C1 CN1CC(SCO)C(F)(F)C1.C1(=O)C(O)C2CCN1C2 C1(C(N(CCCNC(C2C(CCC)C2)=O)C(C)C)=O)CS(=O)(=O)CC(=O)N1 CCC(O)C(C)(C)C(=O)N1CCC1CNC(c1c(-c2ccccc2)c[nH]c1C)=O c1(CC(=O)NC2CCN(C(CCNC(COC)=O)=O)C2)c(C)cc(OC)cc1C c1(OCCCCC)ccc(C(=O)NC2CC(NC(C3(C)CC3(C)C)=O)C2)cc1 C#CCCCCCC(=O)NC(c1ccnn1C)C(=O)N(C)CCOCC1CC1 C1(NC(C2(NC(C)=O)CCCCC2)=O)CC2CN(C(c3cc[nH]c3)=O)CC12 C(N=c1nc(NC2CC(C)n3ncnc32)c2c([nH]1)CSC2)c1cnc(C)n1C S(=O)(=O)(C(F)(F)F)NCCC(N1CC(NC(C2CC2(F)Cl)=O)C1)=O C(c1ccc(F)cc1F)=CC(=O)N(CCCNC(=O)CC1CC1(C)C)C(C)C c1(C(c2nnnn2C2CC2)N(CC(F)(F)F)CC(=O)OC)ccc(F)cc1 c1(C(=O)NC(CC=C)CNC(=O)Cc2ncc(C)o2)cc(F)cc2cc[nH]c12 c1(OC)c(C(=O)NC2CC(CC(=O)Nc3cccnc3C(C)C)C2)cnn1C c1(CC(=O)NC2CC(F)(CNC(C(C)=C3CCC3)=O)C2)ccc(C)c(Cl)c1 C1(NC(c2ccc3cc[nH]c3c2)=O)CC2CC1CN(C(=O)C=CCO)C2 C1(=CC(=O)NC2C(CNC(=O)CC3CCCCC3)COC2)CN2CCC1CC2 c1(C(N2CC(C)C(CNC(=O)CC3CC4(CCC4)C3)C2)=O)ccc(Cl)cc1Cl N1(C(=O)NC2CCC(C(N)=O)C2)CC2(CCC2)C12CCC2 C1(CNC(C2=C(C)CC2)=O)CN(C(=O)CC2CCCC(C)(C)O2)CCC1(C)C C(=O)(CP(C)(C)=O)NCCN(CCOC)C(c1cnc(COC)nc1)=O C=CCCCCCC(=O)N1CC(NC(c2coc(Cl)c2)=O)CC1(C)CC C1(C)(C(N2CC(OC)(CNC(=O)C(C)CCN(C)C)C2)=O)C(C)(C)C1(C)C CC1(C)CCCN(C(=O)CCc2ccccc2Cl)C1CNC(c1cccnn1)=O c1(SCC2C(C)C2)cn2c(n1)CCCC2.c1(NCC)ccccc1 Cc1c(NC(C2CCCN(C(=O)C(C)CO)C2)=O)cccc1[N+](=O)[O-] CC1=NOC2(C1)CC(c1nc(-c3cccc(C(F)F)n3)nn1-c1ccn(C)n1)C2 C12C3CCC(C3)C1NCC2.C1(CCCCC)CCCCN1C(c1cccnc1)=O C(CS(=O)(=O)c1ccc(F)cc1)N(C(C(=O)OC)COC(C)C)C C1(NC(CSCC#C)=O)CCCC(NC(c2nn(CC)cc2Cl)=O)CC1 N1(C(C2(OCC)CCOCC2)=O)CC2(CNC(C3CC(C)CO3)=O)CCC1CC2 N1(C(c2n[nH]c(C)c2N)=O)CC2CC(NC(=O)CC3CCSCC3)C2C1 C(=O)(CCCC(=O)NCCC1CCCN(C(=O)Cc2nc(C)sc2C)C1)OCC C1(C(N2CCC(NC(CCc3n(C)ccn3)=O)C2)=O)C(C2CC2)C1(F)F c1(N2CCN(c3c(OC)c(F)ccc3)CC2)nc(Cl)nc2c(F)cc(F)cc12 C1(CNC(c2cc(OC)c(Br)s2)=O)CCN(C(=O)C=CC(C)C)C(C)C1 C(N=c1ccnc(-c2ccccn2)[nH]1)C1CC(NC(C=C(C)C2CC2)=O)C1 C1(C)(C(C)C)CCN(C(=O)CONC(=O)CN2CCN(C)CC2)CC1 CC(CC(=O)N1CCC2C(NC(=O)CC34CCCN3CCC4)CC12)P(C)(C)=O N1(CC(=O)NCCN(C(=O)C(F)CC2CCOC2)C)CCOCC1 N1(C(c2cncc(OCC)c2)=O)CC(NC(C=CC(=O)OCC)=O)C(C)(C)C1 Cc1c(NC(C)C(C)C(=O)O)cnn1C c1(CC)nc(C(=O)NC2CC(NC(c3cnc(OCC(F)F)cn3)=O)C2)c(C)o1 C(=O)(C(CC)CCOC)NC(C(=O)NCC(COC)(C)C)(C)C C#CC1(CNC(=O)C(C)(C)C2CCCN2C(c2ccsc2OC)=O)CCCC1 C(=O)(CC(C=C)CCC)N1CCC(C(C(=O)N(CC#C)CCOC)C)CC1 CCC(CO)C(=O)NCC(C1CC1)N(C)C(c1ccnn1CCOC)=O CN1CCN(C2CN(CC(N3CCCCC3C3CN(C(=O)C4CC4)C3)=O)C2)CC1 c1(NC2c3ccc2o3)ccc(F)c(OC)c1.c1(CC)nnnn1COC C(C)(C)(CC(=O)N1CCCC(C(C)NC(=O)C(C)=CC2CC2)C1)SC C1(NC(=O)CCc2ccc(F)cc2)CCCC12CCN(C(C13CC(CO1)C3)=O)C2 c1(CC)nc(C)[nH]c1C(=O)NC(C)CN(C(=O)CC1CCCO1)C c1(OC)ccc(F)cc1C(=O)N(C1CN(C(=O)COCc2cccs2)C1)C C1(C(N2CC(OC)C(NC(=O)Cc3cc[nH]c3)C2)=O)CCc2cc(C)ccc2O1 C1(CC=C)(NC(=O)CCCCCO)CCCN(C(=O)Cc2ncccc2C)C1 n1(CC)cnc2c(N3CCn4ncc(Cl)c4C3)nc(N(C)CC3CN(C)C3)nc12 N1(C(c2c(CC)non2)=O)CCN(C(=O)C=Cc2csc(Br)c2)CC1C CC1(C)OCC2CC12C(N1CCC(CO)(CNC(c2coc(CO)c2)=O)CC1)=O C(=O)(C(C)C(C)C(C)(C)C)N(CCCNC(CC1(CNC(C)=O)CC1)=O)C N1(C(c2nccc(OC)c2)=O)CC2CCC1CN2C(C1(F)CC2(CCC2)C1)=O N1(C(CCNC(C)=O)=O)CCC(C)(C)C1CC(=O)NCC1CCCC12CC2 C1(NC(C2C(C(=O)OCC)C2)=O)CC2CCC1CN(C(C1CC(C)(CC)C1)=O)C2 c1(OC)ccc2[nH]c(=NC(C)CCSC)[nH]c(=NC3C=CCC3)c2c1 Cn1cc(C#N)cc1C(N1CCC(CCNC(c2c(Cl)nsc2Cl)=O)C1)=O C(N=c1[nH]nc(CC(C)C)s1)C1OCCN(C(C(=Cc2cn[nH]c2)C)=O)C1 N(C1CCCc2ccc(O)cc21)CC1(C)CN(C)C1 Cc1cn2c(n1)CCC(NC(=O)NCC(c1ccc(Br)cc1F)F)C2 c1(C(=O)NC2C(C(C)C)CN(C(=O)C(C)(C)CO)CC2)ccc([N+](=O)[O-])c(Cl)c1 C1(NC(C(CC)CCOC)=O)CN(C(C2(C)CC(C)(C)C2)=O)CC2(CCC2)C1 C(=O)(C(O)CCCNC(C1(O)CC1)=O)NC1CCN(CCC)C1 CC1CC(=O)NCCN1C(c1cc(CCNC(=O)CCCn2cccn2)on1)=O CC(C)CS(=O)(=O)CCC(=O)NCC(C)CN(C(=O)CSc1cccc(O)c1)C N1(C(c2nc(C)[nH]n2)=O)CC(NC(C2CCC2(F)F)=O)C(C(F)F)C1 c1(C(=O)NCC(C2CCOC2)NC(c2cnc(C)o2)=O)c(C)nn(C)c1C(F)F C1(CNC(=O)NCc2n(CC)ccn2)CCC(C(F)(F)F)CC1 C1(NC(C2(c3cn(C)nc3)CC2)=O)CCCC(NC(=O)CN2CCS(=O)CC2)C1 C(C(C)(C)CCNC(c1ccc(C)n1C)=O)NC(C1(CC=C)CCC1)=O c1(CNCC2(CC)CC=CC2)ccc(OC)c(OC)c1OC CC(=O)CCCC(=O)N1CCN(C(c2ccnnc2O)=O)CC1c1ccncc1 c1(-c2c(F)ccc(NC(c3c(OC)ccc(C)c3)=O)n2)ccc2occc2c1 N(C1COc2c(F)cccc21)C(c1ccc(Cn2cc(COC)nn2)o1)=O C12(NC(c3c(OC)ncc(Cl)c3)=O)CCCCC1N(C(=O)CCC(F)(F)F)CC2 C1(N(C(c2n(C)ncc2)=O)CCO)CCN(C(c2cnc(C(N)=O)cn2)=O)CC1 C(=O)(C(C(=O)N1CCCC(CN(C)C(C2(CO)CC2)=O)C1)C(C)(C)C)OCC c1(C(N(CCN(C(C(C)c2ncco2)=O)C)C)=O)cnc(N)c([N+](=O)[O-])c1 N1(C(CCC2N(C(=O)OC(C)(C)C)CCC2)=O)CCOC(c2n[nH]c(CO)n2)C1 c1(C(=O)NCC(CNC(c2c(C)snn2)=O)CO)ccc2c(c1)CC(=O)NC2 N1(C(C2C(C)C2)=O)CC(NC(=O)CC(C)(C)C(F)F)CC12CCOCC2 C1(CNC(CC(C=C)C)=O)Cc2ccccc2CN1C(c1cc(F)cnc1O)=O c1(C(N2CCC(N(C(C(c3ccc(C)cc3)C)=O)CCO)C2)=O)c(C)nn(C)c1Cl C(C(=O)N1CC(O)CCO1)(C1CCCO1)NC(Cc1c(C)ncs1)=O N1(C(c2c(C)csc2Cl)=O)CC(C2CCCN(C(c3ccc(Cl)[nH]3)=O)C2)C1 C1(C(CC)=O)(C(=O)N(C)CCNC(=O)C(C)OCCOCCC)CCNC1=O C1(N2CC(COC)OCC2)CC2(C1)CN(C(c1cc(C)n(C(F)F)n1)=O)C2 c1(C(N2C(CNC(=O)CCC3CCCO3)CCC2)=O)ccncc1Cl c1(NC(N2CCOC(CC3CC3c3ccccc3)C2)=O)ccc2ncccc2c1 Cc1cc(C(=O)NC(C2CN(C(=O)C(C)OCCC(C)C)C2)C)cc(C)c1 c1(C(=O)NC(CC)C(C)C)cc(O)nc2c1CN(C(C1(O)CC1)=O)CC2 c1(C(c2ccccc2)OC(C2(NC(=O)OC(C)(C)C)COC2)=O)ccc(O)nn1 c1(C(=O)NC23CC(CNC(C(CC)CC)=O)(C2)OC3C)cc2ccncc2[nH]1 c1(C(=O)NC(CNC(Cc2cc(C)no2)=O)(C)CC(C)C)cc2c[nH]cnc-2n1 N1(C(C(CC=C)N(C)C)=O)CCC(NC(=O)CCN2CCOC2=O)C12CCCC2 C1(C(C)C)CCN(S(=O)(=O)NC(C2(C(F)(F)F)CCCCCC2)=O)CC1 c1(C(N2CC(NC(C3CC(N(C)C)C3)=O)C2)=O)cc2c(C3CC3)cccc2[nH]1 c1(CCCCC)cc(C(=O)N(CCC(C)NC(=O)CC2(C)CCOC2)C)n[nH]1 C(=O)(CCCC(=O)NCC(C1CC1)NC(=O)CCc1ccc(Cl)s1)NCC c1(CCC(=O)N(CC(CNC(C(C)C2CCOC2)=O)(C)C)C)ccc(F)c(F)c1 c1(C(=O)NC(CC(C)NC(c2cc(CCOC)on2)=O)C)cnc2n1CCOC2 C1(CCNC(C2CC23CCCC3)=O)CCCN(C(=O)C(=C2CCCCC2)F)C1 C1(C(N2CCN(C(C(c3cccc(Cl)c3)C)=O)CC2)=O)C2CC3C(C2=O)C13 C1(CC=C)(C(=O)NCC2(O)CCN(C(C3(O)CC(F)(F)C3)=O)C2)CCOCC1 C1(NC(C(C)OCC#C)=O)CCN(C(c2cc(O)nc(Cl)c2)=O)CC(C)(C)C1 C(=O)(CN=S(C)(C)=O)NC(CN(C(=O)Cc1ccoc1)C=O)C1(c2ccccc2)CC1 C(=O)(C(CC(C)C)C(C)C)N1CC(OC)(CNC(=O)Cc2cccn2C)C1 C(=O)(CCCC(C)C)NC1CCN(C(C(C)OCc2cccc(C)c2)=O)C1 c1(C(CCC)NC(=O)NCC2CC2)cc2c(s1)CCC2.n1(C2CC2)nccn1 c1(OC)ccc(OC)c(C2CCN(CC(N3CC(O)CCC3C(=O)O)=O)CC2)c1 c1(OCC(=O)N(C2CCC(NC(=O)CC3(C)CC3(F)Cl)CC2)C)ccc(F)cc1 c1(C(N(c2ccncc2)C)=O)cc(Oc2ccccc2)cn1C CC1CC=CCC1NC(=O)C(c1ccco1)NC(=O)C=CC(F)(F)F CCCCCCC(C)C(=O)NC(COC)CC(=O)NC(CC)C(=O)OC C1(CC(N2C(CN(C(C(CCSC)O)=O)C)CCC2)=O)CCC(=O)NC1=O c1(-c2cn(CCNC(Cc3nc(COC)on3)=O)nn2)ccc(C)cn1 CCC(CC(=O)NC1CN(C(c2ccc(CO)o2)=O)C2(CCOC2)C1)CC(C)C c1(OC)ncc(Cl)cc1C(=O)NCC(C)CNC(C1CC(N2CCOCC2)C1)=O C1(C)(NC(CSCC=C)=O)CCCN(C(c2nc(Br)c(C)s2)=O)C1 C12(NC(c3cnc(SC)n3C)=O)CC3CCC(C1C2)N3C(C1(C)CCC1)=O Cc1cn2cccc(NC(=O)OC(C)(C)C)c2n1.C12CC3(COC1C3)C(=O)N2 c1(COCC(=O)NC(C(C)=O)C)ccccn1 c1(C(=O)NCCNC(c2c(C)noc2C)=O)ccc2c(ccn2C)c1 c1(C(=O)NC(CC(C)C)C(=O)O)cn2c(n1)CCN(CCC(=O)NCC(=O)O)CC2 N1(C(CC=CC=C)=O)CCC(CC(C)NC(c2csc(C(C)=O)c2)=O)CC1 Cc1scc(C(N2CCN(CCNC(=O)CC3(C)CC3(F)F)CC2)=O)c1C1CC1 Cc1cc(C(=O)NC2CCCC(N(C)C(c3cc(C(C)(C)C)on3)=O)C2)n(C)n1 c1(NC(C2N(C(CCCSC)=O)CC(F)C2)=O)c(C)cc(C#N)cc1C C1(N(C(C=CC)=O)C)CCCC(N(C)C(c2cnc(-c3cccs3)o2)=O)C1 C1(CC=C)(C(=O)N(C)Cc2nc(C3CCCC3)no2)CCCNC1 c1(C(c2n(CC)nnn2)NCc2ncoc2C(F)F)cnn(C)c1C(C)C C=CCC(C)(CC)C(=O)N1CC(CNC(c2csnc2Cl)=O)C(F)(F)C1 N1(C(c2cn(C3CCC3)nn2)=O)CCN(C(=O)C(F)C(F)(F)F)C2CCC12 c1(N(C)CCO)ccc(C(=O)NCC2(C3CC3)COCCN2)cc1 c1(C2(C(N(CCNC(C(C)c3cncs3)=O)C)=O)CC2)ccnc(O)c1 C1(C(=O)NCc2cc[nH]n2)CC(F)(F)CN1C(c1cc(F)ccc1F)=O Cc1ccccc1C(=O)N(C)CC1(O)CN(C(=O)CC2CCC(C)C2)C1 CC(C)(CN(CC(=O)Nc1ccccc1Cl)OC(c1ccccc1Cl)=O)C(=O)O c1(C(C)C(=O)NC2CC(CNC(C3CCC(C)O3)=O)C2)ccc(Cl)c(Cl)c1 C(=O)(C1=C(C2(C)CC2)N(c2ccc(C)cc2Cl)C(=S)NC1c1cnc[nH]1)OC C1(CNC(CC(=O)OCC)=O)CN(C)CCN1C(C12CC=CC(C1)OC2)=O c1(C(=O)NCC2CN(C(c3ccc(C)nc3C)=O)C3C2C3)ccc([N+](=O)[O-])cn1 N1(C(C(=O)N(CCC(N)=O)CC(C)C)=O)CCC(CCNC(CSC)=O)CC1 C(=O)(C1CCc2c[nH]nc21)N1CC(NC(c2c(N)sc(C)c2C)=O)CC1(C)C C(C(N=[N+]=[N-])C(=O)N1CC(C(=O)NCC(F)C2CCC2)C2(CC2)C1)OCC C12(NC(c3n(-c4ccc(OCC)cc4)nnn3)(CC)C3CC3)CCCC1OCC2 C1(C(=O)NCC2CC(NC(C3CC(F)(CO)C3)=O)C2)CCCCCC1(F)F c1(C(=O)NC2(C)CN(C(C3CCn4nncc4C3)=O)C2)cc2cccc(Cl)c2s1 C1(c2cn(CCCCOC(C)=O)nn2)CN(C(=O)CO)CCN1C O=C1CC2=NNC(CC(F)C)C(=O)N1CCC2 N1(C(COCCC=C)=O)Cc2n[nH]cc2C1C(=O)NCc1cc(CC)[nH]n1 c1(C(=O)NCC2CN(C(CSC)=O)C(C)C2)ccc(C)c(O)c1 C(C(C)(C)C(=O)N(C1CC1)Cc1cn(-c2cnccc2Cl)nn1)NC(C)=O Cn1cc(C(N2CC(F)(CNC(C3CCC(C)(C)OC3)=O)C2)=O)n(C)c1=O c1(C(N2CC(NC(C(C)C#N)=O)C(CC(C)(C)C)C2)=O)cc2cnccc2o1 c1(C(=O)NC(CNC(c2cnc(C)o2)=O)(C)C(C)C)cccn2ncc(Br)c12 c1(OC)cccc(OC)c1CN1CCCCC1C(=O)Nc1ncccc1Cl C12(CNC(c3ccns3)=O)CC1CN(C(=O)Cn1ncc(Br)n1)C2 c1(C(=O)OC)cc(C(N2CC(O)CC2CNC(c2[nH]nnc2C)=O)=O)cc(F)c1 Cc1ccc(C(=O)NC(C)CCNC(=O)C(c2cccc(Br)c2)(C)C)c(N)c1 C(C1CC(C)Oc2ccccc21)NC(c1c(OCC(=C)C)cccc1)=O C1(NC(c2cc(C(C)C)on2)=O)CCCN(C(C2CC3(C2)CC(O)C3)=O)C1C C1(C(N(CCN(C)C)CC)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CC1O C1(CC(=O)NCC2(C)CCCN2C(c2cc([N+](=O)[O-])n[nH]2)=O)CC(F)(F)C1(F)F C(=O)(C(C)(C)CCC#N)NC12CC(NC(CCCn3c(C)cc(C)n3)=O)(C1)C2 Cc1nc(N2CCC(C(C)NC(C3(O)CC3)=O)CC2)c2scc(C)c2n1 N1(C(CC2C=NN(C)C2=O)=O)CCCC(F)(C(=O)NCC(C)(CO)CO)C1 c1(C(N2CC(CC(C)NC(C(C=CC)O)=O)C2)=O)csc(C)c1Br c1(CN(C)C(c2cc(C3CC3)no2)=O)ccc(CNC(=O)C(C)(C)Br)cc1 C(=O)(CC1=CCCCC1)NC(C1CN(C(C2(COC(C)(C)C)CC=CC2)=O)C1)C C1(C)(C(=O)NC(C2(CNC(=O)C(C)N(CC(F)(F)F)C)CC2)C)C=CCC1 C(=O)(C(C#N)C(C)(C)C)N1C(C)CC1C(N1CC(c2ncccn2)C1)=O C=CCC(CNC(=O)CC1CCN(C(=O)C(C)(F)C(C)(C)F)CC1)CC(C)C C(=O)(C(C)(C)CCC(=O)NC1CC1NC(C1COCC1(C)C)=O)OC N1(C(C2(C)CCOCC2)=O)CC2(C1)SCCC2NC(c1csc(C(F)F)n1)=O c1(C(=O)NC23CC(C(=O)N(c4ccsc4)CCO)(C2)C3)cc2ccccc2[nH]1 CC1CC(C)N(C(=O)CC2CCC2)CCN1C(=O)C#CC1(C(F)(F)F)CC1 N1(C(c2c(C)csn2)=O)CCCCC(C2CN(C(c3ncn4c3CCC4)=O)C2)C1 C1(CNC(c2c(C)n(C3CCOC3)nn2)=O)CCC(C)CN1C(=O)CC1CC1 C1(CC=C)(NC(c2c[nH]c(C)cc2=O)=O)CCCN(C(=O)C(C)COC)C1 C1(C(C)NC(c2scnc2C(F)(F)F)=O)CCN(C(=O)CNC=O)CC1 C1(COC(C(CC=C)N(C)C)=O)CCC(C)(C)CC1 C1(NC(c2cc(CC(C)C)[nH]n2)=O)COCCN(C(=O)C=Cc2ncc[nH]2)C1 CC1(C)CN(C(C2CCCC(F)C2)=O)CC1NC(C1C2CCC(=O)C12)=O Cc1nccnc1C(C)NC(=O)C(C1CCCN(C(=O)CC2(C)CC2)C1)C C(C(=O)N1CCN(C(c2cc3sccc3[nH]2)=O)C(CC2CC2)C1)(C(C)(C)C)SC Cc1cccc(N(CC(=O)O)C(c2ccccc2)=O)c1.C1(C)C(=O)N1 C1(C2CCN(C(C3CCCS3(=O)=O)=O)CC2)(NC(Cc2c(C)nn(C)c2)=O)CC1 c1(C(=O)NCC(=O)NC2(CNC(C3(F)CSC3)=O)CC2)ccc2c(c1)OCCO2 N1(C(CS(CC)=O)=O)CCC(C2CC2)(CNC(c2conc2C2CCC2)=O)C1 C1(OC)CC2CC1CN(C(=O)C(F)CC(C)(C)NC(=O)CCc1nccs1)C2 C(=O)(C(C)(CC(C)C)NC(=O)OCCOC(C)(C)C)Oc1cccc(SC)c1 c1(CC(=O)NCC(C2CC2)NC(C2CCN(C)C2)=O)csc2c(F)cccc12 c1(C(=O)NCC(c2ccccc2)C)cccc(NC2=NCCS2)c1 C1(C(=O)NCCC2(CO)CCC2)CC2C=CC1N(C(=O)C=Cc1ccncn1)C2 C(c1cocn1)=CC(=O)N(CC(C)NC(C1CC2(CC2)C1)=O)C CCCCC(F)C(=O)N1CC2CC1CN2C(=O)C(CN(C)C)CC c1(CCC(=O)NC(C)CN(C(=O)CCc2ncc[nH]2)C)nnc(O)nc1O C(C(O)C(=O)Nn1cnc2ccccc12)NC(C(CCC)C)=O c1(CC(=O)NCC2N(C(CCCC)=O)CC(C)CC2)ccc(Br)c(Cl)c1F c1(OC)ccc(C(=O)NC2CC23CC(NC(C2CCCOC2)=O)C3)cc1O c1(C(N(C(CC)CC(=O)NC2CCCC2(C)N(C)C)C)=O)coc2c1COC2 O=C1C2CC3C1C3C2C(N1CC(NC(C2(O)CCOC2)=O)CC(O)C1)=O Cc1cnc(CNCCCC2C=CCC2)nc1 N1(C(CC2CC(SC)C2)=O)CCC(C(=O)NCC(C)CC2CC2)(CO)C1 n1(CC)nccc1C(=O)NC1(CNC(=O)CN2CCC(C)C2)CCC1 C(=O)(N=c1[nH]oc(C(C)(C)C)c1C#N)NCC1(COC)CCCCO1 c1(OC)ccc(C2CCCN2C(c2ccccc2SCc2cccs2)=O)cc1F C1(CNC(c2c(CC)nc(=N)[nH]c2)=O)CC2(CO1)CN(C(=O)C(C)(F)F)C2 c1(SC)ncc(N)c(C(=O)NCC2CCCC2NC(c2cc(C)ncn2)=O)n1 C=C(Cl)CC(C(=O)NCCSC(C)C)NC(c1cccs1)=O c1(C(N(C)CC2CCCN(C(C3(C)CCCCO3)=O)C2)=O)nccc(N)c1Cl N(C(=NCCC1(C)CC1(Cl)Cl)NCC1CCS(=O)(=O)N1)CCC(=O)N(C)C C1(C(=O)NCC2(SC)CC2)CC12CCN(C(=O)C(c1ccccc1)=O)CC2 C(=O)(C1CCCc2cccnc21)NC(CNC(CCC(=O)NCCC)=O)C(C)C C(c1ccc(OC(F)F)c(OC)c1)=CC(=O)NC1CCN(CC(=O)NCC)CC1 C1(NC(C2CC(C)(C)C2)=O)CCC2CCN(C(c3ccccc3CO)=O)C1C2 CC1C(NC(C2CC(N(C)C)C2)=O)CCCN1C(c1cc(N(C)C)ccc1N)=O C1(C(N(CC(=C)C)CCOC)=O)CCCN1NC(=O)CCC1CC1C Cc1ccc(Br)cc1NC(C1COCCN1C(=O)CCCn1ccnc1C)=O c1(C(=O)NCC2CC(NC(c3c(NC)snc3C)=O)C2)nccn2cc(C)nc12 C1(NC(C2(NC(=O)C=CCO)CC(O)C2)=O)CC2(CNC(=O)O2)C1 c1(C(Cc2ccccc2)C(=O)NCCCC(=O)c2ccccc2)ccc(F)cc1 c1(C(=O)Nc2ccc(CN3C(=O)CCC3=O)cc2)ccc2ncccc2c1 N1(C(Cn2ccc(C)n2)=O)CC(NC(C2(C)CC2c2ccccc2)=O)C2(CC2)C1 O=C1NCC2(CCCN(C(=O)C3=CCNC3)C2)O1 c1(N2C(CNC(C3(CO)CC3)=O)CC3(CC3)C2)cc(C(F)(F)F)nc2ncnn12 C(=O)(CCCCC(N)=O)N(C(C)CN(C)C(c1cc(-c2ccco2)c[nH]1)=O)C c1(C(N2CC3(C(C(=O)Nc4ccno4)C3)C2)=O)c(F)cncc1F C12(NC(C3C(=C)C3)=O)CC(CNC(c3cc(C4CC4)[nH]n3)=O)(C1)OC2C CC1(C(=O)NC2CN(C(=O)CC3CC3)CCC2O)CCC(F)(F)CC1 c1(OC)ccc(NC(C2CC(NC(=O)Cc3cccc(C)c3)C2(C)C)=O)cc1C c1(C(=O)NCCC(C)N(C(C(C=C)c2ccccc2)=O)C)ccccc1C(C)C N1(C(C(C(C)C)NC(CCCOC(C)=O)=O)=O)CC2CC1CN2C(C)C C(=O)(C(C)(C)CC#C)N1CCC(N(C(CCC#C)=O)CCOC)CC1 CC1OCCCC1C(=O)NCCCN(C(=O)CCOC1CCCC1)C C12(NC(c3n(CC)c(O)nc3)=O)CCC(C1)N(C(=O)COC1CCC1)C2 CC(CC(C)(F)F)C(=O)NCC(CO)NC(=O)COc1ccc(Cl)c(Cl)c1 c1(C(CC)N(C2CCCN(C(c3cn(C)nc3C)=O)C2)CC)ccc(F)cc1 c1(CN(C)C)ccc(NC(C2CNCC2C(F)(F)F)=O)cc1Cl c1(C(=O)NC2(c3ccccc3)CN(C(C3(C)CC3Br)=O)C2)cc2n(n1)CCOC2 CC(C)CC(CNC(C1(CCNC(C2CC2(C)C)=O)CCC1)=O)OC C(=O)(CCCCCCc1cn(CC2COC(=O)C2)nn1)N(C1CCCC(C)C1)CC NS(=O)(=O)c1ccc(C(=O)NCC(F)CNC(=O)Cn2cnnn2)o1 N1(C(=O)NC(CC)CN(C)C)CCCC(C(N)=O)(N(C)C)C1 C(=O)(C1=CCCSC1)NC1CC(CNC(CC2(OC)CCC2)=O)CC1O c1(C(=O)NOCCC2CCCCO2)n[nH]cc1CNC(C1CCCO1)=O c1(C(C(=O)N(CC(C)NC(C2(C)CCC(C)C2)=O)C)C)cccc(F)c1 c1(C2(C(N3CC(OCCNC(=O)CCC4CC4)C3)=O)CC2)ccc(F)cc1Cl N1(C(CCC=C)=O)CC(CNC(=O)CC2(N3CCCC3)CC2)C2(CC2)C1 c1(C(=O)NC2CCC(NC(C(C)OCC)=O)CC2)c(C)[nH]c2ccc(Cl)cc12 Cc1cc(C(N2CC=C(C(=O)N(c3cnn(C)c3)C)C2)=O)nnc1C N1(C(c2n(CC#C)ccc2)=O)C(C)CN(C(=O)C=C(Cl)Cl)CC1C N1(C(C2C(C)(C)CO2)=O)CC(CO)C2(C1)CN(C(c1cncc(Cl)c1Cl)=O)C2 c1(CC(C)(C)C)ccc(C(=O)NCCC(O)CNC(=O)C(CO)N(C)C)cc1 c1(CC)nc(C(=O)NCC2CCN2C(c2ccns2)=O)cs1 C(C(=O)OCC(C1(C)CC2CC2C1)=O)(C(C)C)n1ncc(C)c1 N12CCOC3CC(CCC13)C2=O.C1(NC(C)=O)CCOC(C)(c2ccccc2)C1 c1(C(=O)NC(C(=O)NC(CCC)C(=O)NC)CN(C)C)cc(C)n(C)c1C C=CC1(NC(C2CCCN(C(c3cn(C)c(C)n3)=O)C2C)=O)CCCCC1 C1(CCC)CN(C(c2c(Cl)c(CC)nn2C)=O)CCN1C(=O)CCOC C12CCN(CC1)C(=O)C1(CCC1)C(=O)N2C.CC1CCC1CN1CCCC1 c1(C(=O)NC23CC(NC(C(C(CC)CC)C)=O)(C2)C3)n[nH]c2nccc(Cl)c12 C=CCC(C)C(=O)NCC1(F)CN(C(c2ccc(COc3ccsc3)cc2)=O)C1 c1(NC)cncc(CNC(C2CC(C)N2C(c2cccc(CC#N)c2)=O)=O)c1 C12(CNC(CSCCC#N)=O)CCCC(CN(C(c3ccc([N+](=O)[O-])s3)=O)C1)C2 C1(NC(C(COC)O)=O)CCCCC1CNC(C1CCCC1)=O c1(OC)ccc(C(c2cn(CC(C)NC(=O)CC3(O)CCC3)nn2)OC)cc1 N1(C(C(COC)C)=O)CCCC1(C)CNC(c1ccc[nH]1)=O c1(C(=O)NC(C)CN(C)C(c2csc(=N)[nH]2)=O)cccc(CCO)c1 c1(OC)ccc2c(c1)C(C(=O)NC(C)C(C)(C)NC(=O)CCCNC(N)=O)CC2 C(=O)(CC1=CCCCC1)NCC(=O)NCC(CC(C)C)NC(C1(CF)CC1(F)F)=O C1(C(N(CC(=O)NCCCOCC(F)F)CC)=O)CN(C)CCC1O C1(NC(C2C(OCC)C2)=O)CN(C(C23CC(CO2)C3)=O)CC1C1CC1 c1(OC)ccc(F)c(CN2CC3CC2CN3C(C2CCSCC2)=O)c1F Cc1cc(C(=O)NC(CC2CC2)CC(=O)NCCCCN2CCC2)c(C)o1 CC1(NC(=O)C(=O)NCC(F)(F)F)CN(C(C2CCC2(F)F)=O)C1 N1(C(C(N2CCNC2=O)C)=O)CCC(CF)(NC(c2cncc(CO)c2)=O)C1 Cc1cc(C(=O)NCC(=O)NCCCN(C(=O)C2=NOC(C)C2)C)cc(C)c1 C(=O)(CC(C)(C)CC(C)=O)N1CC2(CN(C(C3CCC(CC)O3)=O)C2)C1 c1(C(=O)NC2CCCC(CN(C(c3c(C)nns3)=O)C)C2)cc2n(n1)CCC2 c1(C(C(=O)NC(C2N(C(CCOC(C)=O)=O)CCC2)C)C)ccc(Cl)cc1 C1(C(=O)NCC(CNC(COCCOCC)=O)OC)CCOCC1(C)C c1(NC(CC2CCN(Cc3ccc(OC)cc3)C2)=O)c(C)nn(C(F)(F)F)c1C CC1(C)CC(CNC(c2ccon2)=O)CN1C(C1CC2CCC2C1)=O C=CCC(C)(O)C(=O)N1CCC(NC(=O)C(C)C2CC2)C(OC)C1 c1(C(=O)NCC2CN(C(CCSCCCC)=O)C2)nnn(-c2ccn(C)n2)c1C C1(C(N2CC(F)(c3cn(CC4CCC4)nn3)C2)=O)(OC)CCCC(C)C1 N1(C(CC(C)C)=O)CCOCCC1C(=O)NCC(C)(O)C1CCC1 C(=O)(C1=CC2CCC=CCCC12)N1CC(Nc2nccc(SC)n2)C(C)C1 N1(C(c2ccc(OC)cc2C)=O)CC(NC(=O)CCS(C)=O)Cc2ccccc21 C(CC(N)=O)(C(=O)NCC1CCC(CO)CC1)NC(C(CC)O)=O Cc1ccc(F)c(C(=O)NC23CCCC(NC(=O)C(C)CS(C)=O)(C2)C3)c1 C(=O)(C1=CS(=O)(=O)CCC1)NC1CC(NC(c2cc(C(C)C)on2)=O)C12CCC2 N1(C(C)C(N)=O)CCC2(CC1)CC2(C)C(N1CCN(C2CCOCC2)CC1)=O c1(N2CC(O)(C(C)NC(c3c(Cl)nc(OC)s3)=O)C2)nn(C)cc1[N+](=O)[O-] c1(CN2CC(=O)N(CCOCCOC(C)(C)C)C2=O)c(F)ccc(Br)c1Cl c1(C(=O)NCc2cn(CC(N3CC(C(C)O)C3)=O)nn2)ccncc1F C(=O)(C(F)CCC)NC.N12CCC1C(=O)N(C)CCCN2C.C(C)(C)(C)OC(=O)N Cc1[nH]c(=NCc2cccc(O)n2)sc1C(=O)Nc1cccc(Br)n1 Cc1nsc(C(N2CCCC2C(C)(C)NC(C2COCC2(C)C)=O)=O)c1N N1(C(COCCOC)=O)CCC(F)CC1C(N1CCSCC1C)=O C1(CC)CCCN(C(c2cnc(C)nc2C)=O)C1C(=O)NCCC[Si](C)(C)C C1(C(=O)OC)CC(CN(C2CSC2)C)CCO1 CCCC(CC)C(=O)N(C(C)CN(C)C(c1cc(=O)n(C)cn1)=O)C c1(NC(C(CC)(C)O)=O)ccc(NC(=O)CCC(=O)N2CCOCC2)c(F)c1 N1(C(CC=CC=C)=O)CC2CCC2(NC(c2ccnc(CC)c2)=O)C1 C1(C(N(C)CC2CC2Cl)=O)(NC(C2CCC2)=O)CC1(C)C N1(C(C=C2CCC(C)CC2)=O)CC2CCC1C(CNC(C1CCC(O)CC1)=O)C2 c1(C(=O)NCC2N(C(C(C)OC)=O)CC(F)(F)C2)c(C)sc2ccccc12 Fc1ccc(COc2nc(-c3ccsc3)nn2-c2ccc(OC(F)F)cc2)cc1Cl C(c1ccc2occc2c1)=CC(=O)NCC(CNC(C1C(C(C)C)C1)=O)(C)O Cc1cccc(C(=O)NCC(CC2CC2)C(=O)N(C)CC2CCC2)c1N c1(OC)cc(C(=O)NC2CCC(NCc3c(F)cccc3Cl)C2)c(OC)cc1Cl c1(C(N2CC(O)(CCNC(CCOC(C)C)=O)C2)=O)cn(C)c2ccccc12 c1(C(=O)Nc2c(CN(C(C)=O)C)cccc2)c(C)nn(C)c1Cl C1(CC)CN(C(c2cnc(O)cc2C)=O)CCC1NC(=O)CCc1ccco1 C(=O)(CCCN=[N+]=[N-])NCCCOC(C)COc1ccccc1 Cc1cc(F)ccc1C(N1CCC(CN(C)Cc2ccc(O)nc2)C1)=O CC(CC1CC1)C(=O)NCC(c1ccccc1)CNC(=O)Cc1ccn(C)n1 C(=O)(C(CC(C)C)CC(C)C)N1CC(NC(CCCOCC=C)=O)C(C)C1 c1(C(=O)OCC)ccc(N2CCN(C3CCN(CC)C3=O)CC2)nc1C Cc1[nH]c(=N)sc1C(N1CC=CC(NC(=O)C=CCOC2CCOCC2)C1)=O CC1CC(C(N2CC(c3ccccc3)(NC(C3CC4CCC3C4)=O)C2)=O)CCO1 Cc1ccsc1CC(=O)NC(CN(C)C(C1CC1F)=O)Cc1ccccc1 c1(C(=O)NC)cccc(CNC(=S)Nc2nc(-c3ccccc3)cs2)c1 c1(C(N2CCC(C)(NC(=O)CCC3CCOC3)C2)=O)cc(S(N)(=O)=O)ccc1N C1(C2CCCCC2)(C(=O)NC(CCNC(C(C(C)C)OC)=O)C(C)C)CC1 N#Cc1cc(C(N2CC34CCCC3(CNC4)C2)=O)c2ccccc2c1 N1(C(C(C)(C2CC2)OC)=O)CCC2(CCC2)C(CNC(=O)CCCF)C1 c1(C(=O)OC)c(C(N2CC(NC(=O)C3CC3)C2)=O)n[nH]c1C.n12cc(nn1)C2 C1(NC(c2c(C)cc[nH]2)=O)CCN(C(C2CCC(C(F)(F)F)CC2)=O)CC1C C1(CCC(=O)N(CC(CC)NC(c2c(CC)nns2)=O)CC)CCC(=O)NC1 c1(OC)ccnc(OC)c1C(=O)NC1CC2CC1N(C(=O)C(C#N)C(C)C)C2 CCC(C#N)(CC)C(=O)N1CC(NC(=O)C(C)Cc2ccnn2C)C(O)C1 CCC(Cc1ccc(C)cc1)N(C)N1CC(C)OC(C)C1C c1(C(=O)NC(C)C(=O)N(CC(C)O)CC2CC2)cccc2ccnn12 c1(CCC(=O)NC2CN(C(c3nc(C)nn3C)=O)CC2O)nc2ccccc2[nH]1 c1(C(N2C(C(=O)N(C3CC3)C)CCC2)=O)csc(=NC)[nH]1.C1(CCC)CCCC1N C(=O)(C(F)n1ccnc1)NCC(=O)NCC(c1ncc[nH]1)O N#Cc1ccc(CC(N2CC3CC3(CNC(=O)CC3NC(=O)NC3=O)C2)=O)cc1 C1(C(c2n(CC)nnn2)NCC2CC(CC(C)(C)C)C2)C(C)(C)C1(C)C c1(C(N2C(CN(C(CCSCCCC)=O)CC)CCC2)=O)cccc(CCF)c1 N1(CCNC(N(CC(CC)O)C)=O)CCOC(C)C1 CCC(C)C(CC(=O)NCCS(=O)CC)NC(=O)C(CC1CC1)OC c1(C(=O)NCC(C2CC2)NC(C2CCC(C(N)=O)O2)=O)ccc([N+](=O)[O-])s1 c1(NC(C2(C)CCN2Cc2cnc(Cl)nc2)=O)cnn2ccc(Cl)nc12 N1(C(CCCCCCNC(C(c2ccn(C)n2)C)=O)=O)CC2(C1)NC(=O)NC2=O Cn1nc(C(=O)NC2COCCC2NC(=O)Cn2cnnc2)cc1C(F)(F)F C=CCCC(C)(C)C(=O)NCCC1CN(C(=O)CC2CCN(OC)CC2)CCO1 C1(COC)CN(C(c2ccc(Br)cc2)=O)CCN1C(=O)CSCC(C)C C1(C(N(C2CC(C)(C)C2)C)=O)CC2(CC2)CN1C(=O)Cn1cccc1 Cc1nc(C2CCCC2)sc1C(=O)NCC1CC(NC(C2CN(S(C)(=O)=O)C2)=O)C1 CCCCCCC(CNC(c1ncoc1C(F)(F)F)c1nnnn1CC)CC c1(C(=O)NC(C(=O)NC(C(=O)OCC)C2CC2)C2CCCO2)nc(C)sc1C N1(C(CCCC(=C)C)=O)CCC2(CC1)CC2NC(=O)CCN(C)CCO c1(C(N2CCCC(C)(NC(C3CC4CC4C3)=O)C2)=O)cc2c(nc1N)CCCC2 c1(C(N(CC(CNC(CC(COC)C)=O)C)C)=O)cc(OC)ccc1F c1(C(N2CCCN(C(C(C)NC(=O)NC)=O)CC2)=O)ccc2nn[nH]c2c1 c1(CC=C(C)C)cc(C(=O)NC2CCN(C(C3(C)CC3C)=O)CC2O)ccc1F C1(C)(NC(C(CCC)O)=O)CCN(c2nc(OC)cc(OC)n2)CC1 CC(C)C(CNC(c1occ2c1CCC2)=O)N=c1[nH]nc(C2CC2)s1 C1(C(N(C2CCCC(O)C2)C)=O)CC(C)(C)CCN1C(C1CCNC(=O)C1)=O N1(C(C2C(C)(Br)C2)=O)CCC(c2cn(Cc3cc(C4CC4)no3)nn2)C1 C(C(CC(F)(F)F)NC(c1c[nH]cc1Br)=O)NC(CCCN(C(C)C)C)=O O=C1CN(C(=O)CN2CCn3nnc(Br)c3C2)c2ccccc2N1 c1(C(N(CC(CN(C(C(CCC)C)=O)C)O)C)=O)cccc(C#N)n1 c1(C(=O)NCCCCC(=O)NC(CC=C)CC)c[n+]([O-])c(C)cn1 c1(-c2c(CN(CCN(C)C)C)cc(Cl)cn2)ccc2c(c1)C(=O)C(=O)N2 c1(C(=O)NC(C(=O)NC(c2n(C)cnn2)CO)C2(C)CC2)cc(Cl)cn1C c1(C(N2C(C(=O)Nc3cnn(CC)c3)CC(=C)C2)=O)cnc(Cl)cc1OC C1(C(N(CCN(C)C(C2CC(=O)N(C3CCC3)C2)=O)C)=O)CCC2(CCC2)CO1 C(=O)(C(C(C)O)NC(C1CCCN1CC)=O)NC1CCN(CCC)C1 Cc1cn2c(n1)C(C)CC(C(=O)NCC1CN(C(C3OCCCO3)=O)CC1O)C2 c1(C(=O)NC2CN(C(C(=COCC)C#N)=O)C(C)C2)ccc(F)c(Cl)c1F C(=O)(CCC(=O)NN(C)C)NC(C1CN(C(C2CC3CCC2C3)=O)CCO1)C Cc1nc(C)c(C(=O)OCc2nc(CS(C)(=O)=O)n[nH]2)c(C)n1 c1(C(=O)NCC(C2CCCC2)NC(c2c(CC)occ2)=O)ccn2ccnc2c1 C1(NC(=O)C(F)=C2CCCC2)CCCC(NC(c2ccc(C3CC3)nc2)=O)C1 N1(C(CN(C(Cn2c(C)nc(C)n2)=O)C(C)C)=O)CCN(C)C2(CC2)C1 C12(NC(=O)CSC(F)F)COCCC1CN(C(=O)CCOc1cccnc1)C2 Cc1c(C(=O)NCCC(O)CNC(=O)CC2CCCOC2)sc2[nH]cnc(=O)c12 N1(C(C2CCC(CO)CC2)=O)CCN(C(=O)CCC2CCCC2)C(CCO)C1 C12(C(=O)NC3CC(C)N(C(=O)CSCc4ccncc4)C3)CCCC(C1)OC2 CC(CC(=O)NCc1csc2ccc(Cl)cc12)CC(C)(C)C C1C(CO)(CO)N1C(=O)C(C)NC(=O)C(C)SC.c1(C(=O)NC)ccco1.CO c1(CCC)cnnc(C(N2CC(CC(C)(C)CNC(C3(C(N)=O)CC3)=O)C2)=O)c1 c1(C(N(C(C)C)CCNC(=O)C(c2ccccc2)F)=O)cncc(C(F)F)c1 O=C(C#CC1CCCC1)N1CC(O)CC1C(=O)Nn1ccnn1 C(CCCC(=O)NCCCCC(=O)NC(C)CC(C)O)OC CC(C)(C)C(=O)NC1CC1C(=O)NCC1COC(=O)N1 c1(-n2cc(C(C)NC(=O)C(F)CC3CCOC3)nn2)cncc(Cl)c1 C(C(=O)N1CCC(C)C1CNC(c1cc(C(N)=O)c[nH]1)=O)(C(C)C)NC(=O)OC Cc1noc(C(=O)NCC(C2CC2)NC(=O)CCC2CC2(F)F)c1C C1(NC(=O)OC(C)(C)C)CCN(Cc2cccc(CO)c2)CC1CC#N C(C1=NOC2CN(C(c3nocc3C(C)(C)C)=O)CC12)NC(COCCC=C)=O C(=O)(C(C)(C#N)CC)N1CCC(C(C(=O)NCCN(CCC)CCC)C)CC1 N1(C(Cc2cc(C)[nH]n2)=O)CCC(C(=O)N(C)Cc2cn[nH]c2)C(C)(C)C1 c1(C(=O)NC(C(C)(C)NC(CC(C)n2ccnc2)=O)C)ccc(=O)n(C)n1 C(=O)(CCCC(C)=O)NCC1(C(F)(F)F)CC(=C)C1 N1(C(C(c2cccc(C(F)(F)F)c2)C)=O)CCCNC(=O)C1 C(C(=O)NC1CCN(c2cc(C)ncn2)C1C)(C(C)C)NC(C)=O c1(C(C(=O)N(C(C)CNC(=O)CCN2CCOC2=O)C)C)c(C)noc1C C(=O)(CCCC(F)F)N(CCCOCCNC(C1CC(CCC)C1)=O)C C1(NC(C2C(C)(CC)C2)=O)CC2(CCN(C(=O)CC3=CCCC3)CC2)C1 C1(CC(=O)N(C)CCNC(=O)COCC2CCCCO2)(COCC)CCCCC1 N1(C(COC(C)=O)=O)CC2CCC(C1)C(NC(C1CCC(=O)N3CCCC13)=O)C2 N1(C(CC2N(C(CCC(CC)OC)=O)CCOC2)=O)CCCNC(=O)C1C N1(C(C(C(C)C)CO)=O)CCC(C)N(C(c2ccc(-c3cnn(C)c3)o2)=O)CC1 Cc1cc(C(C(=O)NCC(C)C)N(CCC(=O)N(C)C)C)c2ncccc2c1 N1(C(c2c(C)cco2)=O)CC(NC(C2CCC(N(C)C)CC2)=O)C2(CC2)C1 N1(C(Cc2cc(C)on2)=O)CC2CCN(C(c3cc(Cl)c(Br)cc3Cl)=O)CC2C1 c1(CC)cc(C(N2CCC(CNC(=O)C(C3CCCC3)OC)C2)=O)n(C)n1 CC(C)CC(C(=O)NCC1(F)CC(NC(c2ncoc2Br)=O)C1)C(C)C C1(CC=C)(NC(C2CCC2(F)F)=O)CCN(C(=O)C(c2cnn(COC)c2)=O)C1 N1(C(CC(C)OC)=O)CCC2(CC1)C(NC(=O)CC1(CO)CC1)CS(=O)(=O)N2C N1(C(COCCNC(c2c(CC)cncc2)=O)=O)CCCC2(CC1)CC2 c1(C(N(CC(C)N(C(=O)CCC(C)(C)C)C)C)=O)cnc(N)c([N+](=O)[O-])c1 CCC(CC(=O)NCCC1CN(C(c2nc[nH]c3ncnc2-3)=O)C1)CC(C)C C1(CCCCNC(Cc2c(C)ocn2)=O)CCCN(C(=O)CC(C)N(C)C)C1 C(S(=O)(=O)CCCC(=O)N=c1cc(C(F)F)n(C)[nH]1)C1CC(OC(C)C)C1 C1(NC(c2scnc2Br)=O)CCCN(C(C2C3(CC3)C23CC3)=O)CC1 N1(C(C2N(C)CCCC2)=O)CC2(CCC2NC(=O)CN2C(=O)CNC2=O)C1 C1(NC(=O)CNC(=O)CN2CCCC2)CCOC1C(N1CC(N2CC(O)C2)C1)=O C(N=c1cccc(S(=O)(=O)N2CCOCC(C)C2)[nH]1)c1c(OC)ccnc1 N1(C(C(F)=CC)=O)CCOCC(CNC(=O)CC2(OC)CCCC2)C1 c1(OCC)n[nH]cc1C(=O)NC1(CCNC(=O)Cc2cnnn2C)CCC1 C(CC(=O)N1CC=CC(NC(=O)C=Cc2scnc2C)C1)(C(C)C)OCC c1(C(N2C(C(=O)NC(c3ccc(F)cc3F)CO)CC2)=O)c(Cl)cc(Br)cc1Cl C1(CC(C)NC(c2cc[nH]n2)=O)CCN(C(c2cncc(F)n2)=O)CC1 C(=O)(C1=CCN(C(C2(C(C)(C)O)CCC2)=O)CC1)NC(CCOC)C N1(C(CCCN(C(C)=O)C)=O)CCCN(C(=O)C=CC2CCCN2C)CC1C C1(NC(c2cc(Cl)cc(Cl)n2)=O)CCN(C(=O)CCC[N+](=O)[O-])CC1F C(=O)(CCCC1OCCO1)NCC1(NC(C(C)SC(C)C)=O)CCC1 c1(C(=O)NC2CCCN(C(CCCOCCC)=O)C2)ccc(O)c(C(C)=O)c1 c1(C(N2CCCC(NC(C3C(C)CC3)=O)CC2)=O)ccc([N+](=O)[O-])cc1Br c1(CNc2c(C(=O)Oc3ccc(C(=O)OC)cc3)n[nH]c2)ccc2n[nH]cc2c1 N1(C(C23OCC(C)(C2)C3)=O)CCCC(F)(CNC(c2csc(Cl)n2)=O)C1 c1(C(N2CCN(C(CC3CN(C)CC3O)=O)C(CO)C2)=O)ccc(N)c(Cl)c1O C(=O)(CCCC(C)(F)F)NCC(C)N(C(C(C)Oc1ccc(Cl)cc1)=O)C CON(CCO)C(=O)C1CCC(NC(=O)C2=C(C)CC2)C1 C(=O)(C1CCCc2cncn21)N1CC2CCC(NC(Cc3c(C)non3)=O)C2C1 Cc1n[nH]c2cnc(C(=O)NC3CN(C(=O)Cn4cccc4)CC3O)cc12 Cc1ccc(S(=O)(=O)Nc2ccccc2C(=O)Nc2ccc(CO)nc2)cc1C C1(C#C)(CNC(C(CC#C)NC(c2cnc(Cl)s2)=O)=O)CCOCC1 C=CCC(C(=O)N1CC=CC(NC(c2nnn3c2CCCC3)=O)C1)C(C)C C1(C(C)C)CN(C(C2CCC(N(C)C)CC2)=O)CCN1C(=O)C(=O)N(C)C C1(NC(C2CCCN(CC)C2)=O)CC2(CCCN(C(=O)COCCCF)C2)C1 C(=O)(C(CNC(C1CNC(=O)N1)=O)C(C)(C)C)NCC1N(C)C(=O)COC1 c1(C(=O)NC(C(C(=O)OC)(C)C)c2ccccc2)ccc2nccc(=O)n2c1 N1(C(CC2CC(=O)OC2)=O)CC2CCCN(C(c3cn(CC(N)=O)nn3)=O)C2C1 CC1CCC(NC(c2ccc(C(F)F)cn2)=O)CN1C(c1ncc(Cl)nc1Cl)=O c1(CCC)c(C(=O)NC2CC(NC(c3cnccn3)=O)C2)cnn1C1CCCC1 Cc1c(C(N2CCC(CCC(=O)N3CC(N4CCC4)C3)C2)=O)ncn1C c1(C(=O)NCC2(O)CC(C(=O)NCC(C)C(C)(C)C)C2)ccn2cncc2c1 CCCCCCC(CC)NC(=O)NC1(C)CC2CCC1C2 CCC(CC(=O)NC1CC2(C1)CC2NC(c1coc(Cl)n1)=O)C1CC1 C1(CNC(c2c(C)ccc(C)c2)=O)CN(C(C2COCCOC2)=O)CCC1(F)F c1(C(=O)NCC2CCN(Cc3cc(C(N)=O)cc(F)c3)C2)cc2cccn2cn1 Cc1cc(NC(C(c2ccn(CC(=O)C(=O)OC(C)(C)C)n2)N(C)C)=O)ccc1Cl C1(C(N2CC3CN(C(C(COC)C)=O)CC32)=O)Cc2ccccc2CN1C n1(CC)ncc(C(=O)NC(Cc2ccccc2)C(=O)N2CCCCC2)c1Cl C(C)(N(C)N1CCOC(C(F)(F)F)C1)c1ccc(OC)nc1 CN1CCOCC1C(=O)NCC1(C)N(C(=O)C(C)(C)N2CCCCC2)CCC1 C1(NC(Cc2ccc(C)s2)=O)CC2CCC(C1)N2C(=O)COC1CCOCC1 CC1CCCCC1(C)C(=O)NCCn1ccc(C(=O)N(C2CC3CCC2O3)C)c1 C1(CC(=O)NC(CN(C2CC2)CC)C)CCCCN1C(=O)CSc1nc[nH]n1 Cc1ccc(C(N2CC(NC(=O)Cc3sc(O)nc3O)C(C)C2)=O)c(O)c1 N1(C(C2CSCCS2)=O)CCN(C(c2cncs2)=O)C(c2cccc(F)c2)C1 Cc1ccnc2nc(C(N3CCCC(NC(=O)CCOCC4CC4)C3)=O)nn12 C(C(C)(F)C(C)(C)F)(c1n(-c2ccc(OC)cc2)nnn1)NCC(Br)=C(C)C N1(C(C)C(=O)NC2(CO)CCCC2)CCN(C(c2ccoc2Cl)=O)CC1 c1(C(N2CCC(CCNC(c3c(C)cc(SC)o3)=O)C2)=O)ncc(C)cc1C C(=O)(CC(C(F)(F)F)NC(C1(C(C)(C)O)CCC1)=O)NC(c1ncccn1)C CC1CCC(CCN(C)C)N(C(=O)C(=O)NC2(c3cccs3)CC2)C1 C1(C(N2CCCC(CN(C(c3cc(C)sc3)=O)C)C2)=O)CC12CCOCC2 c1(OC)cc(C(=O)OCc2ccc(O)c(Cl)c2)nc(C(C)C)n1 CCCC(CCC)C(=O)NCC1(CNC(C2CCN(C3CCSC3)CC2)=O)CC1 C(=O)(C(CCSC)NC=O)N(CCN(CCNC(CC)=O)C)C(C)C c1(C(N(CCC(C)NC(=O)Cc2cnns2)C)=O)ccc([N+](=O)[O-])cc1F Nc1cc2c(cc1C(N1CC3(CNC(=O)CC4CCCO4)CCC1C3)=O)CCC2 C1(C2CCCC2)(C(=O)NC(C(C)(C)O)Cc2ccc(F)cc2)CCNC1=O N1(C(c2oc(CC)c(C)c2)=O)CC(NC(=O)C(COC)OC)CC12CCC2 CCCCCC(=O)N1CCC(CCOC)(NC(=O)CCCn2ccccc2=O)C1 c1(OC)c(C(=O)NOCCSc2cn(C3CCCC3(F)F)nn2)ccc(Br)c1F c1(OCCNC(=O)Oc2ccc(OC(C)=O)cc2)c(C)cnnc1O O(NC(=O)C(=O)OCC1N(C)CCC1)CC1CC(F)(F)C1(Cl)Cl c1(C(CC)C(=O)N(CC(O)CN(C)C(C2CCCC2CC)=O)C)cccc(Cl)c1 C#CCCC(C(=O)NCC1CC2CCC(C1)C2)NC(c1cc(C)[nH]n1)=O N1(C(C(CCCCC)F)=O)C2CCCC1CN(C(=O)C(c1ccccc1)=O)C2 c1(C(N2CCN(C(C(CC)(C)C#N)=O)CC2C(C)C)=O)ccc2ccccc2n1 CS(=O)(=O)c1ccc(C(C(F)(F)F)NC(c2nccnc2Br)=O)cc1Cl c1(C(C)=O)cnn(C)c1C(N1CCC(CNC(c2cnc(C)s2)=O)C1)=O c1(CC)ccccc1OCC(=O)NCC(CNC(=O)C(c1ccc(Cl)cc1)C)OC c1(OC)nc(NCC2(F)CCCN(C(C34CC5CC3C4C5O)=O)C2)cc(C)n1 Cn1ccc2cc(C(=O)NCCC3CCCN(C(=O)COC(F)F)C3)cnc12 C#CCC(C)(CC)C(=O)NCCCNC(C1CCCC1C(C)C)=O C1(C)(C(=O)NC(C)(C)C)CC12CCN(C(=O)Cc1ccccc1O)CC2 C(=O)(CC(C)(C)C(=O)OC)NCC1N(C(C(CC)=CC)=O)CC(C)(C)C1 NC1CCc2cc(C(N3CCC(Oc4ccc(Cl)cc4)CC3)=O)ccc2C1 c1(C(=O)NCC2CN(C(c3c(C)[nH]cc3)=O)C2)ccc([N+](=O)[O-])c(N(C)C)c1 C(=O)(CC1NC(=O)c2ccccc21)NCCN(C(=O)Cc1ccn(C)n1)CC Cc1cc(C(=O)NC2CC(NC(C3(CO)CCOC3)=O)C2)c(F)cc1Cl Cc1ccc(CC(=O)NC2CCCC2NC(C2(C)COC(=O)OC2)=O)cc1Cl N1(C(C(C)OCC(F)(F)F)=O)CC(C)(CNC(=O)COC2CC=CC2)CC1(C)C CCC(C)C(O)CC(=O)NC(CNC(C1(C2(O)CCC2)CC1)=O)C1CC1 C(=O)(CC(C)(C(F)(F)F)N(C)C)NCC(CCCC)NC(=O)CCCN(C)C CCC(O)C(F)(F)C(=O)NCCCNC(=O)CCc1c(F)cccc1Cl CC1CCN(Cc2nc(C(C)(C)C)cs2)CC1NC(=O)CNc1ccccc1.OC c1(C(N2C3C(NC(C(CC)CC)=O)CC(C3)C2)=O)cc2ccccc2s1 C(=O)(C(C)(O)C(C)C)NC(CC)CN(C(=O)CSCc1cccc(C)c1)C c1(C(=O)NC(CNC(C(C)SCC)=O)C)ccc(C(=O)NC2CC2)cc1F N12CCOCC(C1)C2=O.c1(OC)n[nH]cc1C(N1CCCC1CN(C)C)=O N1(C(CC(C)(O)c2ccccc2)=O)CCC(NC(=O)C=CI)C(CO)CC1 c1(C(N2CC(OC)C(NC(c3ccc(C(F)(F)F)o3)=O)C2)=O)ccc(N)c(F)n1 C1(=O)CCCNCC2CC1C2.N1(C(C)C)CC(C(=O)NCCNC(=O)N(C)C)C1 C1(NC(C(C2CCCCC2)NC(C(C2CCOC2)OC)=O)=O)(CO)CCOCC1 CCCC(CNC(=O)C(C1CCC1)OC)NC(c1c[nH]nc1C(C)(C)C)=O C(=O)(C1=NOC(C)C1)N1CCC(OC)(CNC(=O)CC2(OC)CCCCC2)C1 N1(C(c2cc(C)sn2)=O)CCCC2(C1)CN(C(c1ccnc(C)c1C)=O)CCO2 c1(OC)cc(NC(=O)CC2CCN(Cc3ccc(Cl)o3)CC2)c(C)cc1[N+](=O)[O-] C1(C(N2CCC3C2CCCN3C(c2ccccc2)=O)=O)CCc2nccn2CC1 c1(C(=O)NCC2N(C(C(C)=C(CC)C)=O)CCC2)cccc(OC)c1O N1(C(C(n2c(C)ccn2)C)=O)CCC(F)(C(=O)NC2(CO)CCCCC2C)CC1 c1(C(N2CCCC(NC(C3CC(=C)C3)=O)C2C)=O)cccc(SC)c1[N+](=O)[O-] CC(C)(CCCCNC(=O)C(O)Cc1ccccc1)C(=O)NNC(=O)C(C)(C)O Cc1ccc(C(=O)NCC23CC(NC(C4OCCOC4C)=O)(C2)C3)cc1C C(=O)(C(CC(F)F)NC(C1CC(C)(C)CO1)=O)NCc1cc(C)ns1 C1(CC(=O)NC2(CNC(CC3CC(C(C)(C)C)C3)=O)CCC2)CCC2(CC2)CO1 C=CCCCCCCC(=O)N(Cc1cn(CC)nn1)Cc1n[nH]c2cc(Br)ccc12 N1(C(CCC)=O)CCCN(C(c2nnc(S)n2C)=O)CC1C(C)C C1(C(=O)OC(C)C(c2ccc(Cl)cc2)=O)C2CCC1(c1ccc(Br)cc1)C2 O=C(CC1CCc2ccccc21)NC1CCN(C(=O)Cn2cc(Cl)cn2)CC1F C1(NC(CCCNC(=O)NCC#C)=O)CN(C(=O)C#CC2CC2)CC2CCCC12 n1(CCCOC)cc(CCNC2(c3n(NC(=O)N(C)C)nnn3)COC2)nn1 c1(C(=O)NC(C2CCCN2C(C2CCCCS2)=O)C)cnc(N2CCCC2)cn1 C1(COCC)CCCN(C(=O)NCC2CCCN2c2ccccc2)C1 c1(C(N2C3CCC(NC(C(C#N)C4CC4)=O)(C3)C2)=O)cc2ccnc(Cl)c2[nH]1 N1(CCNC(C2CC(C)(C)OCC2)=O)CCN(C(C2CCC2Cl)=O)CC12CCC2 O=C1NC(C(=O)NCC2CC2NC(c2cccc(Sc3ccccc3)c2)=O)CC1F Cc1cc(C(=O)NCC2(C(N)=O)CN(C(C3(C4CCCO4)CC3)=O)C2)oc1C N1(C(c2cn(CC)nc2)=O)CC(CNC(=O)C(N2CCNC2=O)C)C(F)(CO)C1 C1(CNC(Cc2c(C)nc(S)s2)=O)CC2CCC1N2C(c1ccc(=O)n(C)n1)=O c1(CN(C2CCCC(n3ccnc3)C2)CC)ccc(C#N)cc1F C1(NC(c2c(OCC)oc(C)n2)=O)CN(C(=O)C(C)(O)CC)CC1S(C)(=O)=O C1(C)(C(N2CCC(N(C(Cn3c(C(C)C)ncc3)=O)CCO)C2)=O)CC(C)(C)C1 c1(C(=O)NCC(C2N(C(C(C=CC)O)=O)CCC2)(C)C)cnn2ccsc12 C1(NC(Cc2cn(C)nc2)=O)CCOCC1NC(C1(C(F)F)CC(O)C1)=O c1(CNC(C(C)(C)NC(C=CCC)=O)=O)cnc(OC)nc1 c1(C(N2CC(CN(C(=O)C(C3CCCCC3)F)C)C2)=O)ncoc1C1CCCO1 c1(OC(C)CNCC(c2ccccc2)C)ccccc1C(F)(F)F c1(COC)cc(=NCC2CCC(NC(=O)CCCC3CCC3)C2)[nH]cn1 CCCC(C)(C)CC(=O)NCC(CNC(C12CCCC1C2(F)F)=O)S(C)(=O)=O CCC(CC)C(C(=O)N1CCCOC(CCNC(C2(C)CC=CC2)=O)C1)OC C1(NC(CCc2n(C)ncn2)=O)CC2CCC1N2C(=O)COCC1CCCOC1 CN1CC(C)(C)CC1C(=O)NC1CCCCN(C(C2(C)CCC2)=O)C1 c1(C(N2CCC(C)C2CNC(C2CCC(O)C2)=O)=O)cccc(C#N)c1 C(=O)(C(C(=O)N1CCC(CNC(=O)CCCC2CCC2)CC1)C(C)(C)C)OCC N1(C(C=CCCC)=O)CC2CCC1C1CN(C(=O)Cc3csc(C(C)=O)c3)CC21 c1(OC)ccc(C=CC(=O)NCC2CC(NC(c3cc(CF)on3)=O)C2(C)C)nc1 CCCC(C)C(=O)NCC1N(C(c2ccccc2Br)=O)CCSC1 CN1CC(NC(=O)C(C)(C2CC2)N(C)C(c2ccc(=N)[nH]n2)=O)C(=O)N1 c1(C(=O)NCCCCNC(C(CCSC)O)=O)cc2ccccc2nc1C(F)F C1(CCNC(=O)CCNC(=O)C2CC2)(NC(C2C(=C)C2)=O)CCOCC1 C1(NCc2sc(C(=O)OCC)c(C)c2)CCCCC(c2nnnn2C2(C)CC2)C1 CC1CCN(C(=O)CC2CCC(=O)NC2)C(CNC(=O)CCc2cnco2)C1 c1(NC)ccccc1C(=O)NCCC1CC(C(=O)Nc2ccsc2C(C)C)C1 N1(C(CSCC#C)=O)CCC(NC(=O)CN2CCn3ccnc3C2)CC(O)C1 CC(CCCCCO)NC(=O)C(C1CCCO1)NC(=O)CCc1ccccc1 c1(CC)nc(C)c(C(N2CC(CNC(c3c(Cl)cnn3C(C)C)=O)CC2C)=O)s1 Cn1cccc(C(=O)NCC2CCCCN2c2nnc(-c3ccccc3)o2)c1=O CC1C2C(CCN2C(c2csnc2Cl)=O)CN1C(=O)C(C)n1cncn1 C1(C(N2CC(C3(NC(C4CSC4)=O)CC3)C2)=O)CCOC2(CCCC2)C1 CC1CN(C)CC(C(N2CCC(NC(c3c(C(F)F)cnn3C)=O)C(O)C2)=O)O1 N1(C(c2ccc(C)nc2)=O)CC2CCC(CNC(C3CSCCS3)=O)C2C1 Cn1cnc2c1CCC(C(N1CC(NC(C3SCCCS3)=O)C(C)(C)C1)=O)C2 Cc1cc(=NCCCN2CCCC2)[nH]cc1S(=O)(=O)NCC1C(F)(F)C12CCC2 C1(OCc2nc(OC)nc(C)c2)CC12CCc1ccccc12 c1(CC(=O)NCC2(O)CCN(Cc3n(C)cnc3)C2)ccccc1[N+](=O)[O-] c1(CC(=O)N(CCC(C)NC(c2c(SC)cccc2)=O)C)cc(F)cc(F)c1 c1(C(N(C(CNC(c2c(OC)n[nH]c2)=O)C2CC2)C)=O)ccc(C)c(Br)c1C c1(-n2c(C(C)OCC)nc(-c3ccc(Cl)s3)n2)ccc2nccnc2c1 S(=O)(=O)(c1ccc(NC(=O)C(C(C)C)NCCNC(=O)OC)cc1)NC C(=O)(C1=C(Cl)CCOC1)NCCCN(c1cc(C(C)(C)C)nc(Cl)n1)C c1(C(=O)NC2(C)CCN(C(Cc3ccn(C(C)C)n3)=O)C2)ccc2cc[nH]c2c1 Cc1c(C(=O)NCCN(C(=O)CCc2ccccc2)CC2CC2)n[nH]c1C1CC1 Cc1ccc(CC(N2CCC(CNC(C3C4CCCC34)=O)C2)=O)cn1 C12(CNC(COCCC)=O)CCC1CCN2C(c1cccc(NC(C)=O)c1)=O C(CCC(C(=O)NCCN(C(C)C)CC)NC(=O)C(C1CCOCC1)F)OCC Cc1cc(=O)cc(CNC(c2cn(CC(F)(F)F)cn2)=O)[nH]1 c1(CCNC(C(C)SC(C)C)=O)ocnc1CNC(C1CCC(C(N)=O)O1)=O C1(NC(CC2(OC)CCC2)=O)C2COCC1CN(C(=O)C=CC1CCCO1)C2 N1(C2CCN(C(C)(C)C)C2=O)CCC2(CCN(C(=O)CN3CC4CC4C3)C2)C1 N1(C(C2OCCN(CC)C2)=O)CCN(C(c2ccn(C(F)F)n2)=O)C(C(C)C)C1 CC1CCC(CNC(c2c[nH]c(=N)o2)=O)N(C(c2ccc(CO)nc2)=O)C1 c1(NC(=O)NCC2(NC(c3cc(C)[nH]n3)=O)CC2)ccccc1Br c1(C(C(=O)NC(C)(C)C)N(CC(F)F)CC)cc2c(cc1OC)CCC2 C(CN=c1[nH]nc(C2CC2)o1)(CC(C)C)NC(C1CCN(C(C)=O)CC1)=O C1(N(C(c2c(C)snn2)=O)C)CN(C(c2cc(-c3ccccc3)no2)=O)CC1O c1(OCC)nc(Cl)ccc1C(N1CCC1CNC(=O)CC1CCC1(C)C)=O c1(C(N2CCCC(NC(C(C)c3ccsc3)=O)CC2)=O)cc2c(O)cccc2[nH]1 c1(Nc2nnn(CC)c2C)nc(=NC2CCC3(CC3)C2)[nH]c2c(C)nn(C)c12 c1(C(=O)NCC2CN(C(C3C(=C)C3)=O)CC23CC3)nn(CC(F)F)cc1[N+](=O)[O-] N1(C(C=C(CC)CC)=O)CCC2C(CCCN2c2cc(SC)nc(SC)n2)C1 c1(NC(C2C=CC(NC(c3c(CC)n(C)cc3)=O)C2)=O)cc(C)c(C)c(C)c1 N1(C(CC2(C)CCCC2)=O)CCCC(CNC(=O)CC2CCC23CCC3)CC1 CC(O)(CNC(=O)CCCC1CC1)CNC(C1CCCCC1)=O Cc1nnc2n1C(C(=O)NC(C)CCNC(c1cccc3c1CCCC3)=O)CC2 C1(COC)(NC(C2CCOC2)=O)CCCN(C(=O)C=Cc2cnccc2C)C1 C1(N(C(C2C3COCC23)=O)C2CC2)CC2(NC(=O)CN3CCCC3)COC1C2 C#CC(CNC(=O)CCCCCNC(=O)Cc1ccccn1)CC(C)(C)C CC1(C)CC2(CC(C(N3C(CNC(c4ccnnc4)=O)CC4COCC34)=O)C2)C1 C1(C2=CCCCCC2)(C(=O)NCC2(F)CCN(C(C(CCC)(C)C)=O)CC2)CC1 c1(C(=O)NCC2C(NC(CC(C)CF)=O)CCCC2)cc(F)c(Cl)cc1Cl C1(CNC(c2cncs2)=O)CCN(C(=O)C(O)Cc2ccc(F)cc2)CC1 C1(NC(c2c(C)noc2)=O)CC(F)CN(C(c2ccc(NC(N)=O)cc2)=O)C1 N1(C(CC=C)=O)CC2C3CCC(C2C1)N(C(=O)Cc1c(CC)noc1CC)C3 n1(CC(=O)NC2CN(C(C(C)P(C)(C)=O)=O)C(CO)C2)cc2ccccc2n1 N1(c2cccc(S(=O)(=O)NCCN(OC)C)n2)CCc2ccc(C#N)cc2C1 c1(CC(N2CCC(C)C2CNC(=O)Cc2ccnn2C)=O)c[nH]c2cnccc12 N1(C(CC(n2ccc(C)n2)C)=O)CCC(C)(C)C1CNC(=O)CC1CCOCC1 Cc1nc(C)c(CC(N2CCCC(C)(NC(C3CCCC(F)C3)=O)C2)=O)c(O)n1 c1(CNCc2ccc(C3CCN(C)CC3)cc2)cc2c(Br)cccc2s1 C1(C(=O)OC)C=CCN(C(C2CCCN2C(c2ccc(O)nc2)=O)=O)C1 c1(CN2C(C)(C(=O)NCc3nc(Cl)ccc3F)CCC2)ccc(F)c(C#N)c1 C(=O)(C1CCSc2ccccc21)NCC1(NC(CCC(C)(C)O)=O)CCCC1 c1(C(=O)NC2CC(F)(CNC(C(C)OCC=C)=O)C2)ccc(Br)c(N)c1 C1(C(=O)NCC(CC(C)C)C)CC(NC(=O)C2=CCN(C)C2)C12CCC2 Cc1nccc(C(=O)NC2CC2CNC(=O)CCCSc2ccccc2)n1 N1(C(C2C(OC)CN(C(CCCCCC)=O)C2)=O)CCCC(C2(C)CC2)C1 c1(C(N2CC(CC)(NC(=O)CCN3CCCCC3)C2)=O)coc2c1CS(=O)(=O)C2 n1(CC)c(C)cc2c1CCCC2NC(c1c(C)oc(C)c1C)C C1(CC(=O)N(CCC(C)NC(C=CCOC)=O)C)Cc2ccccc2C1=O c1(C(N2CCCC(NC(c3ncc[nH]3)=O)CC2)=O)[nH]cc2c1CCCC2 c1(C(N2CCOCC(NC(C=CC(C)C)=O)C2)=O)nnc(O)c2ccccc12 C(=O)(C1CCc2c[nH]nc21)NCCCCNC(c1cncc(OC)c1)=O c1(CC=C)cccc(C(=O)N(CCC(=O)NCC2C3COCC23)CC)c1 C12(C(=O)NC3CC(NC(C4CS(=O)(=O)C4)=O)CC3O)CCC(CC1F)C2 CCC(C)CCC(=O)N1CCN(CCNC(=O)CC(C)(C)C2CC2)CC1 C1(CC=C)(NC(=O)CC(C)OC)CCN(C(C2C(C)OC(C)C2C)=O)CC1 N1(C(c2ccc(F)cc2F)=O)CC2(C1)CN(C(C13CCC1CC3)=O)CC2CO C(=O)(CCCC(F)(F)C(F)(F)F)NCC1COCCN(C(C(C(C)C)C#N)=O)C1 c1(C(N2CC(N(C(C(C)S(C)(=O)=O)=O)C)C(O)C2)=O)coc2c1CCCC2 C1(C(N2C(C)CC(NC(COC(C)C)=O)C2)=O)CCCCC1(F)F C#Cc1ccc(C(=O)N(C(CNC(=O)CCC2CCCC(O)C2)CC)C)cc1C C12(CCNC(C(F)=C(C)C)=O)CCC1CN(C(C1(c3cccs3)CC1)=O)C2 c1(CC)cnc(C(=O)NCCN(C(c2cc(-c3ccco3)on2)=O)C2CC2)cn1 C1(C(=O)NC(CC(C)(C)OC)C)CN(C(C2CCC2C#N)=O)CC12CCC2 CC(CNC(=O)CC1(C2CCCO2)CC1)(C1CC1)NC(=O)CSCC(F)(F)F c1(N(C)Cc2cscn2)[nH]c(=NC2CCCC(O)C2)nc2c1cnn2C C1(C)(CCC(=O)NC2C(CNC(C3(C)CC3)=O)CC2)CCC(=O)N1 c1(C(=O)NC(CC(C)NC(c2ccc3sncc3c2)=O)C)cc(S(N)(=O)=O)co1 C#CCCC(C(=O)N1CCC(F)(CO)C1)NC(c1cccc(C)c1O)=O c1(OC)cnc(NC(c2ccsc2CSC(C)C)=O)nc1CO C(=O)(C(C)(C)C#N)NC1C(NC(C(C)CSCc2ccccc2)=O)C1 C(CCCN=c1[nH]c2cc(Cl)cc(Cl)c2o1)NC(C1(OCC)CCCC1)=O C1(CNC(C=NOC)=O)CC(C)(C)CN1C(=O)CS(N)(=O)=O c1(OC)cc(CNC(c2ccncc2F)c2nccn2C)ncc1C O=C(C1CCc2cccc(O)c21)NCC(O)CNC(C1(C(F)F)CC(F)(F)C1)=O C1(CC(N2CC(CCNC(=O)C(O)CC3CC3)C2)=O)COc2ccccc2O1 CCC1=NOC(CC(=O)NCCN(CC(C)O)C(=O)C=C(C)c2ccco2)C1 C1(C(=O)NCCC(=C)CNC(c2cc(C)sc2C)=O)CCc2nc(C)[nH]c2C1 C1(c2nnnn2C2COC2)(NC(CC=C)CC)CSCCSC1 C(=O)(C1=CCC2CCC1N2C(C1(CCOC)CC1)=O)N1CCCC(COCC)C1 C1(C)(CNCC(C)CC2CC2)C(C)(C)C1(C)C C1(C2(NC(c3cccc(F)n3)=O)CC2)CCCCN1C(C1CCC=CCC1)=O CC(C)(F)C(C)(F)C(=O)NCC1CC(NC(c2cncc3ccsc23)=O)C1 N(C1CCCc2c1cnn2-c1ccccc1)C(=O)NCc1c(C)scc1 CC1COCCCN1C(=O)C(CC(F)F)NC(=O)Cc1ccon1 C(N=c1[nH]c(=N)[nH]c(=NCC2(c3ccccn3)CC2)[nH]1)c1c(C)nccc1 C=CCC(CNC(=O)CSc1n[nH]c(O)n1)NC(=O)CCC1CCC(C)O1 N1(C(C2(COC)CC=CC2)=O)CC(N(C)C(C2CCCO2)=O)C(C)(C)C1 c1(C(N2C(C)CN(C(C3(C)CC3Br)=O)CC2)=O)ccc2ncsc2c1 c1(C(N(CCN(C(=O)COc2ccc(Cl)nc2)C)C)=O)cccc2nc(O)[nH]c12 N1(C(c2cn(C(C)C)nn2)=O)CCOCC(NC(C2(CCF)CCC2)=O)C1 S(=O)(=O)(c1csc(C(=O)NC2(C)CC(NC(C34CCN(CC3)C4)=O)C2)c1)NC N1(C(C=CCC)=O)CCCC(C(C)(C)C(=O)NC)C1.C1CCCN(C)CO1 C1(NC(C(=O)NCC)=O)COC2C(NC(C3CNC(=O)N3)=O)COC12 c1(NC(=O)Nc2ncccc2Oc2ccc(F)cc2)cc2cccnc2cn1 c1(C(=O)NC(C)CN(C(=O)CCc2nccs2)C)sccc1S(N)(=O)=O N1(C(c2c(CC)cco2)=O)CC2CCCC(NC(=O)COc3cnn(C)c3)(C2)C1 c1(CC)c(C(=O)OC(C)(C)C)cccc1C.C(CCO)N1C(=O)C2C(C2)C1 N1(C(C(COCC)C)=O)CC(OC)CC1CNC(=O)Cc1c(C)cnn1C C1(C(F)(F)F)(C(N(C)CCNC(=O)COC2CCCCC2)=O)CCOCC1 c1(C(N2CC=CC(C(N3CC(OC)C(O)C3)=O)C2)=O)cc(O)ccc1C c1(C(CC)O)nc(-c2nnn(CC)n2)n(C2CC2)n1 c1(OC)cc(CC(=O)N(C)CCN(C(=O)C(C)(C)CF)C)cc(F)c1 c1(CC(=O)NC(CC(C)C)CNC(C23CCC2C3)=O)ccc(F)cc1F S(=O)(=O)(c1ccc(NCC#CI)cc1)N(C)CC C(=O)(CCC(=O)N1CCC(C)C1CNC(=O)CCCc1sccc1C)NC c1(SC)cc(C(=O)NC2CC(CNC(c3[nH]cnc3C)=O)C2(C)C)c(C)o1 C1(C(=O)NC(c2ccco2)C)CC(O)CN1C(C1C=CCC1)=O Cc1nnc(C(N2CC(c3ocnc3-c3cn(C4CCOC4)nn3)C2)=O)s1 N1(C(=O)NCCCCl)CC2CC1CN2NC(c1ccccc1N(F)F)=O c1(CNC(C=CCCC)=O)cc(C)c(C(N2CCC(CC3CCCCO3)C2C)=O)o1 c1(C(=O)NCC(C)NC(C(CC#C)C)=O)cnc2cnccc2c1 c1(C(=O)NCCC2CN(C(CCCC(N)=O)=O)C2)cccc2[nH]ccc12 C1(C)(C(=O)NCC2C(C)CN(c3ncnc(=N)[nH]3)CC2)CCCNS1(=O)=O N1(C(C2(Cc3ccccc3)CCC2)=O)CCC(NC(C2CC2C2CCC2)=O)CC1 c1(CC(=O)NCC23C(CN(C(C(C(C)C)C)=O)C2)C3)ccc(C#N)cc1F c1(C(=O)NCC2(CNC(C=C(CCC)C)=O)CCC2)nn(C)cc1C C=CC(C)CC(=O)NCC(CC)(CC)N.C(=O)(C(CCC)SC)C(=O)CCC=CC NS(=O)(=O)C1(C(=O)NCC2(F)CCC(NC(C3CCNC3=O)=O)C2)CCC1 N1(C(CC)=O)CC2CN(C(c3cc(C4(C)CC4)ccc3Cl)=O)CC2C1 C(=O)(C1=C(Cl)CCOC1)N1CC(CCNC(c2ccc(F)s2)=O)OCC1 C(=O)(C1=CN=C2N=CNN2C1)N(C1CCCCC1)CCNC(C1=CC(C)(C)C1)=O C1(CNC(C(C)(C)n2cccn2)=O)CC2CN(C(=O)CC3CNC(=O)C3)CC2C1 C(=O)(C(C)(C)C(C)O)N1CC(C(C)NC(C2(C)CC(C#N)C2)=O)C1 Cn1c(C(N2CC3CC2C3CNC(C2C=CC=CC=C2)=O)=O)cccc1=O c1(C(=O)NC(CNC(CC2(C=C)CCC2)=O)CO)ccc(O)nc1Cl C=CC(CCC)CC(=O)NC(C(=O)NCC1([Si](C)(C)C)CC1)C1CCCC1 C1(C(N2CCC(CNC(c3cc(F)n[nH]3)=O)C2)=O)CC2CCC(C1)S2 c1(C(N2C(C(C)NC(CC)=O)CCC2)=O)cnc2ccncc2c1 CCCC(O)C(=O)N1CCC(N(C(=O)CCc2c(C)noc2C)CCOC)CC1 N1(C(=O)OC(C)(C)C)CCC(NC(=O)CC2CC2(C)C)C(O)C1 C(CCC(C)C(=O)NC1CC(NC(c2ncoc2C)=O)C1)OC C1(CC)COCC1N=c1[nH]c(=N)[nH]c(=NCCCOc2ccc(C)cc2)[nH]1 N1(CC(=O)N(CCC(=O)NCC2(CF)CCC2)C2CC2)C(=O)CNC1=O CN1CCCC(CNC(=O)C(CC2CC2)c2ncco2)C1c1ccccc1 c1(C(=O)NCC(CC=C)NC(=O)C(F)(F)CC2CCCO2)cn(C)nc1C C1(N(C(=O)CCCNC(=O)C(CO)NC(N)=O)C)CCC(C(C)(C)C)CC1 Nc1ncnc2c1ncn2CCNC(c1ccccc1-c1ccc(F)cc1)=O C(CC1=CCN(C(=O)CN2CCOCC2)CC1)NC(=O)CC(C1CC1)C1CC1 c1(OCC(=O)NC(CN(C(C(C)OCC#C)=O)CC)C)cccc(Br)c1 c1(C(=O)NC(c2cncnc2)C)coc(CNC(=O)CCCN2CCCC2)n1 c1(C(N2CC3CC(NC(c4cccnn4)=O)C3C2)=O)cncc2c(O)nccc12 S(=O)(=O)(c1ccc(Cl)nc1)N1C(CC#N)CN(C(C2C=CC(=O)N=N2)=O)CC1 C1(C(=O)NCCC(C)NC(C2CCN(CCC)CC2)=O)CCc2n[nH]cc2C1C c1(C(C(=O)NCCC(C)N(C(=O)Cc2ccsn2)C)(C)C)cc(Cl)ccc1F N1(C(C(CC=C)C)=O)CCC2C(NC(=O)Cc3ccsn3)C2C1 C1(NC(C2(CCC)CC2)=O)(COC)CCCN(C(=O)C=CC(C)(C)C)C1 C1(C(=O)NCC(CC)NC(C2(O)CCCC2)=O)C(c2ccccc2)C1(F)F N1(C(C(=O)Nc2ccccc2)C2CC2Cl)Cc2ccc(Br)cc2C1 c1(OC)ccc(C(=O)NC2(C3CCCN3C(c3ccc[n+]([O-])c3)=O)CC2)c(F)c1 n1(C(C(=O)N(C(CC)C)CC(=O)Nc2snc(O)c2Cl)C)c(C)cc(O)cc1=O CC1CCC(CC(=O)NC2CC(C)(NC(=O)CCC(C)N(C)C)C2)OC1 N1(C(C)C(=O)N(C)CCN(C(=O)C(C)Oc2cccnc2)C)CCCCC1=O N1(C(c2c(CC)csc2)=O)CCN(C(=O)Cc2cccc(Cl)c2Cl)CC(O)C1 N1(C(c2cc(C(=O)OC)sc2C)=O)CC(C)N(C(C2CC2F)=O)C(C)C1 n1(C(=O)NCc2cn(C3CN(C(C(CC)OCC)=O)C3)nn2)ccc([N+](=O)[O-])n1 C(=O)(C(F)CC(C)(C)NC(=O)CC1CSCCO1)N1CC(C(=O)OC)C1 Nc1ncc(Br)nc1C(=O)NCC1CCC(NC(C2CN(C3CCC3)C2)=O)C1 C(=O)(C1=CCCN(C(C2CCCSC2C)=O)C1)N1CCC(C=C)(O)C1 N1(C(c2cnn(CC)n2)C(=O)NCCCF)CCc2oc(C)nc2C1 c1(C(N(C(C)C(C)(C)C)C)=O)cc(CNC(=O)CC(C)C2CCCO2)nn1C C1(C)(CNC(CC2CCN(C)CC2)=O)CCCN(C(c2cc(F)ccc2O)=O)C1 C1(NC(=O)CCCF)CCC(C(=O)NC2CCCCC2CC(F)(F)F)CC1 Cc1ncnc(C)c1C(=O)NC1CCC(CCNC(c2ccc(N)c(Cl)c2)=O)C1 C1(N(C(=O)CCNC(=O)OC(C)(C)C)C)C2CCC1N(C(=O)COCCF)C2 N1(C(=O)NC(c2onc(CC)n2)C)CCC(C)N(CC)CC1 N1(C(c2nccc(CNC(Cc3c(C)occ3)=O)c2)=O)C2CCC1CC(O)C2 c1(C(=O)NCC(=C2CN(C(c3cnc[nH]3)=O)C2)F)cnn2ncccc12 C1(NC(CC2CN(C)C2)=O)CC2CCCC(C1)N2C(c1cnns1)=O C1(NC(C=C(C)C2CC2)=O)C2CC(NC(C3(C)C=CCC3)=O)CC12 CC(C)CC(C(=O)NCC(O)CCNC(c1ccc(C#N)o1)=O)C(N)=O c1(C(CC)NC(=O)C(=O)Nc2nccn2Cc2cccc(Cl)c2)ccccc1Br c1(OC)cc(C)c(C(=O)N(C)CC2CCN(C(c3cnoc3C)=O)C2)cn1 C1(CCC)CN(C(=O)CC2OCCO2)CC1C(N1CC2(CC2)C1)=O C1(CC(=O)NCC2CCCC2NC(c2cncs2)=O)CC(=O)NC1=O C(=O)(CC(C(C)C)C(C)C)N1CC(OC)C(NC(=O)CCC2CCN(C)CC2)C1 c1(C(=O)NC2CCCC(NC(=O)COC(F)F)C2)ccc(C(C)(C)C)cn1 Cc1cn(C(C)C)cc1C(=O)NCCCC1(NC(=O)Cc2ccc(F)cn2)CC1 C1(C2CCN(C(C3CSC3)=O)C2)(NC(=O)C(CC(F)F)C2CCC2)CC1 c1(C(=O)NC2CN(C(C)=O)C(C)C2)coc2c(C)cccc12 C1(C(=O)Nc2cc(OC)cc(OC)n2)CC12CCN(C(=O)CCSC)CC2 CS(=O)(=O)c1ccc(CC(=O)NC2CCCC2CNC(c2cc(F)cs2)=O)cc1 O=C(CCCCCO)NC1CCC(CNCC2(N3CCOCC3)CCOCC2)C1 N1(C(C2(C)CCN(C(C#CC(C)C)=O)C2)=O)CC2(COC(C)(C)C2)C1 c1(C(N(CC(C)NC(C2CCC2C(F)F)=O)C)=O)c(C(F)(F)F)ncn1O N1(C(C(=O)NC(c2ccc(C#N)cc2)CC(C)C)=O)CCN(C2CC2)C(=O)C1 CC1=CC(C)CN(C(C2C(C)CN2C(C2CCN(C)C2)=O)=O)C1 Cc1cccnc1CNC(=O)CC1CCC(NC(=O)C=CC2CCOC2)C1 C=CC1(CC(N2CCOC(CNC(=O)CCOCCOC)C2)=O)CCCCC1 N1(C2C(NC(C)=O)CCC2)CCN(C(c2cncc(N(C)C)c2)=O)CC1 C1(NC(CSc2cccc(C)c2)=O)CS(=O)(=O)CC1NC(c1cc(C#N)on1)=O c1(OC)ccc(C)c(C(N2CCCC(N(C(=O)CCc3cnoc3)C)C2)=O)c1N N1(C(c2ccc(CC)cc2N)=O)CCN(C(c2cn(CCO)nn2)=O)C(C)C1C N1(C(c2c(C)ccc(C)c2)=O)CCC2CCC(C1)N2C(=O)C(O)C(C)(C)C C1(CC(=O)NCC(C2CCCC2)N(C(=O)COCCCOC)C)COC2CC1C2 Cc1ccccc1C(C)CC(=O)N1CC(C)(NC(c2cc(O)n(C)n2)=O)C1 c1ccc(NC2(NCCCC3CCCCO3)CCC2)cc1 c1(C(=O)NC(C2CCOC2)CNC(C2(C(C)=O)CC2)=O)ccc(C(C)(C)C)[nH]1 c1(CNC(COCC(=O)NC(C)(C)CC2CC2)=O)cccc(F)c1O C1(C(=O)NC2C(C)(CN(C)C(c3cnn4c3CCC4)=O)CCC2)CC(S(C)(=O)=O)C1 C=CC1(CC(=O)NCCc2cccnc2F)CN(C(C2C(C)C2C)=O)C1 c1(C(N(C)CC2N(C(CCC)=O)CCCC2)C)nc(C(F)(F)F)cc(C)n1 C#Cc1cnc(C(=O)NCCN(C(C2(c3ccno3)CCC2)=O)C2CC2)c(C)c1 C1(C(=O)NCC(CO)NC(C(F)OC)=O)CN2CCC1CC2 N1(C(C23N(C(=O)CN4CCC(O)CC4)CC(C2)C3)=O)CC2C3CCC(O3)C2C1 C(=O)(C#CC1CCCCO1)N1CCN(C(C=C(CCN(C)C)Cl)=O)CC1C1CC1 c1(SCC(=O)NCCC(C)(C)NC(CC=CC)=O)nc2ccc(C)cc2[nH]1 CC1CCN(C(C2(C)C(C)(C)C2(C)C)=O)CCN1C(=O)CN(C1CCSC1)C N1(C(CN(C(C(C)C)=O)C)=O)CC2(CC2)CC1CNC(C1CC12CCSCC2)=O c1(NC(C2C(C(=O)NC3(C(=O)OC)CC3)C2)=O)cccc(C(F)(F)F)c1N CCC(CN(C)C)CC(=O)NCC(C)(C)NC(=O)C=Cc1cncs1 c1(C(=O)NC(CC)CNC(=O)C=C2CCC(C)CC2)cncc2ccccc12 CN1C(=O)NCC1C(N1CC2C(NC(C3CSC3)=O)C2C1)=O C(N=c1[nH]cnc(NCC23CCC(CC2)CC3)c1C)c1scc(CC)n1 N1(C(C=CC=CC)=O)CCC(C)C1CNC(=O)COCc1nc[nH]n1 CC(C(C)C(=O)NCC1CCCC1NC(=O)Cc1cc(F)ccc1F)S(C)(=O)=O c1(CN(C)C)cc(C(=O)NCC2(CN(C(=O)CCC3CCCOC3)C)CC2)no1 C1(N(C(C2CCCC2)=O)CC)CCCN(C(=O)CC2CCS(=O)(=O)C2)CC1 CCCC(C#N)C(=O)NCCCCc1cn(-c2ccc(C)c(Br)c2)nn1 c1(C(N(CCNC(C(F)(F)C2(OC)CCC2)=O)C(C)C)=O)cnc2cccnn12 C1(NC(c2cncc(C)n2)=O)CC2CN(C(C3CN(C)CC(C)O3)=O)CC12 c1(C(=O)OCC2N(C(=O)OC(C)(C)C)CC2)cc2c(s1)CCCCCC2 C1(NC(CCN(CC)CC)=O)CS(=O)(=O)CC1NC(=O)Cc1ccc(OC)nc1 c1(OC)cccc(C2CCN(Cc3cc(Cl)ccc3N(C)C)C2)c1F c1(CNC(=NCC)NC2CC(OCC)C2(CC)CC)nnc(O)c2ccccc12 CN1CCc2[nH]nc(C(=O)NC3C=CC(CNC(=O)C#CC4CCCO4)C3)c2C1 CN1Cc2ccc(-c3cnc(C(=O)NCCc4ccsc4)nc3)cc2C1=O C1(SCC(=O)N(C2CN(C(c3cc(Cl)ccn3)=O)C2)C)CCS(=O)(=O)C1 c1(-c2cncc(C3CCN(C(CCOCC)=O)CC3)c2)ccc2sc(C)nc2c1 C(C(C)(C)C(=O)NCC1CCN1C(=O)CCn1cnc(=N)[nH]1)SC Cc1nc(C(N2CCCC2CC(=O)N(c2ccccc2F)C(C)C#N)=O)sc1C N1(C(CSC)=O)CCCC2C(CCCN2C(C2(c3ccc(F)cn3)CC2)=O)C1 N1(C(C(N2CCC(NC(=O)CN3CC(C)OC(C)C3)C2)C)=O)Cc2ccccc2C1 N1(C(c2nc(CC)sc2)=O)CCCC(C2(NC(C3(OC)CC3)=O)CC2)C1 N1(C(C2(SC)CC2)=O)CCC(CNC(=O)CCN(CC(C)C(C)C)C)C(O)C1 O(NC(=O)C(F)C(C)(F)F)C(C(=O)NCCCN(OC)C)CC(C)C c1(C(C)C)nc(NCCC(C)(C)c2ccccc2)cc(=NC2CC2C(C)(C)C)[nH]1 CCC(CC)(CC)C(=O)Nc1ccc(CC(C)NC(=O)NN2CCCC2=O)cc1 C1(NC(C(CCC)C)=O)CC2CCC(C1)N2C(C)C(=O)N(C1CCCCC1)C C(N=c1cc(C(F)F)nc[nH]1)C1CC(C)N(C(c2csc(Cl)c2)=O)C1 Cc1cccc(C(N2CCOC(C(=O)NC(c3ccc(Br)cc3)CO)C2)=O)c1O C1(CCNC(C2C(C)CC(C)O2)=O)CCCN(C(c2nnn(C)c2N)=O)CC1 C(=O)(CCCCC(C)(C)OC)NCC(CNC(=O)C(C(C)C)NC(C)=O)OC C1(N(C(C=C(C)C(F)F)=O)C)CCCN(C(C2CC(N3CCCC3)C2)=O)C1 c1(C(=O)NC(C23CC(NC(C)=O)(C2)C3)=O)cc(NCC2CC2CF)ccc1Cl O=C(CC(F)(F)C(F)(F)F)NC1CCC12CN(C(c1cccc3[nH]ncc13)=O)C2 n1(CCC(N2CCC(N(C)C(c3nocc3Br)=O)C2)=O)ncc2c1CCCC2 C(=O)(CCCCN=[N+]=[N-])N(C)CC1CCCN(C(=O)Cn2cncn2)C1 N1(C(C(CSC)O)=O)CCC(C(C)CNC(C2CC(F)(F)CS2)=O)CC1 Cc1ccc2sc(N3CCC(CNC(=O)C(C)O)C(F)(F)CC3)nc2c1C Cc1nn(CCO)cc1C(N1CCN(CCCF)CC1)C(=O)NCC1CC1 c1(C(=O)N(C2CCSC2)CC2CCCO2)csc2cccc(F)c12 C1(CC(F)F)(C(=O)NC2CC(CC(C)(C)C)C2)CCNC1 c1(CNC(=O)NC2(CCO)CCCOC2)ccc(Cl)c(F)c1F c1(CNC(C(N2CCCC(O)(CN(C)C)C2)=O)=O)cccc2c1C(=O)OC2 C(N=c1[nH]c(N2CCOC(CCF)C2)nc2c1COC2)C1(C)COCCO1 CCCC(O)CCNC(C1(CNC(c2sccc2F)=O)CC(C)(C)C1)=O N1(C(c2n(CC)ncc2Cl)=O)CCN(C(=O)Cn2nccc2C)CC(CO)C1 C(CCC(C)(C)C(=O)NCC1(O)CCCC1(C)C)NC(C(C(=O)OC)C)=O C1(O)(C(=O)NCCN(C(C(C)CC(F)F)=O)CC2CC2)CN2CCC1CC2 c1(N2CCC(CNC(C(CC)(CC)CO)=O)C2)ncc([N+](=O)[O-])c(=N)[nH]1 N1(C(C(C(C)C)OCC)=O)CCC2CCC(C1)N2Cc1ccc(C#N)cc1F Cc1ccc(F)cc1CN1CCOC(C2CC2)C1.C12CC(C1)C(=O)N2 c1(C(N(CCCO)C(C)C)=O)cn2c(n1)CN(C(c1c(F)ccc(Cl)c1Cl)=O)CC2 c1(CC(=O)NCC(C2CC2)NC(c2c(C)coc2C)=O)ccc2c(c1)CCCO2 C(=O)(C1=CCCCC1C)NC1CC(C)(CNC(Cc2c(C)cco2)=O)C1 CCC(CC)C(C)C(=O)N1CCC(C)(CNC(c2ncccc2SC)=O)C1 CC1N(C(C2(C(C)NC(c3ncccc3O)=O)CC2)=O)CCOC1(C)C c1(COC)ccc(C(=O)N(CC(=O)NC(CC)C(C)O)C2CC2)o1 c1(C(=O)NCC(O)CCNC(c2ccc(O)nc2Cl)=O)ccc2c[nH]nc2n1 C12(C(=O)NC3CC(C(C(=O)NCC(CCOC)O)F)C3)CCC(CC1)C2 CCCCCC(C(C)(C)C)NCc1cnc(C(F)F)s1 c1(C(=O)NCCN(C(c2ccc(C(=O)OC)[nH]2)=O)C2CC2)cc2n(n1)CCCO2 c1(C(N(C)CCNC(C2CCCC(C(N)=O)C2)=O)=O)cc(C(C)(C)C)ccc1N c1(C(N2CCN(C(CS(CCC)(=O)=O)=O)CC2)=O)cc2cccc(C)c2s1 c1(SC)ncc(C(=O)N(C2CN(C(=O)C(C)C3CCC3)C2)C)n1C c1(SCC(=O)NC(CNC2(OC)CCSC2)C)ccc(C(C)(C)C)cc1 CN1CCc2ccc(C(=O)NC3C4CN(C(c5ccc(Br)cc5)=O)CC34)cc21 Cc1cccn2cc(CC(N3CCN(C(=O)C=CC4CC4)C4COCC34)=O)nc12 Cc1ncc(CC(=O)NC2CCCC(NC(c3cc(CCO)on3)=O)C2)c(O)n1 N1(C(C2C(=C)C2)=O)CC2CCCN(C(c3cc(SC(F)(F)F)c[nH]3)=O)C2C1 C1(CCNC(C2C(C)C2C)=O)CCCCN1C(=O)C(C)C1CCCC1 N1(C(C2CCN(C(c3cc(CCC)[nH]n3)=O)C2C)=O)CCCCCCCCC1 C(=O)(CCOCCCNC(=O)C(O)C1CCCC1)NCC(=O)OC C1(NC(C(COC)O)=O)CN(C(=O)C=Cc2cncc(O)c2)C(C)(C)C1 C1(NC(CC2C(C)CCC2)=O)CC(Nc2nccc(-c3cnccn3)n2)C1(C)C c1(C(=O)NCC2CCN(C(C(CC(N)=O)O)=O)CC2)[nH]nc2ncccc12 N1(C(C2(C(N(C)C)=O)CC2)=O)CC2CC2(NC(C2CCC(=O)NC2)=O)C1 C1(C(c2cn(C)nn2)C(=O)NCCCC(CC=C)CC)CCC2CC1C2(C)C C1(C(N2CCC(C(N(CCC(=O)OC)CC)=O)C2)=O)CCC(=O)NC1 C(=O)(C1=Cc2ccccc2C1)N1CCC(NC(c2ncc(Cl)cc2Cl)=O)C(O)C1 C1(CN(C(CC2CC(SC)C2)=O)CC(=O)O)CCc2ncnc(C)c2C1 Cc1ccc(C(=O)NCC2(C)CCCN(C(=O)CC3CC3C)C2)c2c1NCCC2 Cc1cc(=NC(=O)C=CCCCNC(=O)CC2CCC(C)(C)C2)[nH]n1CCO C(=O)(C1=NOC2(CCC2)C1)N1C2CC(NC(c3ccc(C)cc3O)=O)CC1CC2 CC1(C)COC(CCC(=O)NC2CC3(C2)CC3NC(c2coc(CO)c2)=O)C1 c1(C(N(C)CC2CCN(C(CSCC#C)=O)CC2)=O)cc(C(=O)OC)ccc1Cl N1(C(c2c(CNC(C3(CC#C)CCOC3)=O)ocn2)=O)CCCC2CC12 C(CCCC)(CC(=O)NCC1(C)CCCC(=O)N1)N(C(C=CC=CCC)=O)C1CC1 C1(NC(CC2(CSC)CC2)=O)C(C)CCN(C(c2cc(Br)co2)=O)C1C C(C(=O)Nn1cnn(CCOC)c1=O)N(C(=O)CC1CCOC1)CCC Cc1nc(Cl)sc1C(=O)N(C1CC2(CNC2)C1)Cc1nccnc1Cl C12(CNC(C(C(=O)OCC)F)=O)CCC1CN(C(c1cc(Cl)ccc1F)=O)C2 c1(C(=O)OC2CCCC(C(C)NC3CC(OCC)C3)C2)cc(N)cc(F)c1 N1(C(C(CCC)OC)=O)CC2CC(CNC(C3(N(C)C)CCC3)=O)C2C1 C1(CNC(C(C2CC2)SC)=O)CC(F)(CNC(=O)C(C)(C)c2cnsc2)C1 CC(Cc1ccco1)C(=O)NCC1CC(CNC(C2CCCN2C)=O)C1 c1(CC)cccc(C(N2CCC(O)(CN(C)C(C3(OC)CCSC3)=O)C2)=O)c1 c1(C(=O)NC(C(C)C)CNC(C2CC=CC2)=O)cccc(N=c2cncc[nH]2)c1 N12C(CCC1(C)C)C2=O.C(CC#N)NC(=O)NCCN(S(C)(=O)=O)C c1(C(N2CCC(C(=O)NCCC(C)(O)C3CC3)(CC)C2)=O)ccn2cncc2c1 n1(C(C)C)ncnc1C(=O)NCC1(CO)CN(C2CCC2)C1.C1(C(=O)N)(C(F)F)CC1 CC1(C)CC(=O)NCC1C(=O)NCC=CCNC(c1ocnc1C1CC1)=O c1(C(=O)NC(C(=O)NC(C#C)C(C)C)CO)cnn(C)c(=O)c1 c1(CC)noc(CC)c1CC(N1CCC(NC(C2(CO)CCC2)=O)C1C1CC1)=O C1(NC(c2nc(COCC)sc2)=O)CC12CCN(C(C1CC13CCC3)=O)C2 CN(C)S(=O)(=O)NC(C1(CC(F)F)CC1)=O.C1(C2CNC(=O)N2)CCCC1 C(CC(C)(C)C(=O)NCC1CCC(NC(C2CCOC2(C)C)=O)CC1)NC(C)=O N1(C(C(C2CCCCC2)OC)=O)CCCC(CC(N2CCC(C(C)O)CC2)=O)C1 O=C1Cc2cnc(N3CC4CC4(C(=O)Nc4cc(Br)ncc4F)C3)nc2N1 CCCCCC(O)C(=O)NCC12CCC(CC1)N(C(=O)CC(C)(C)O)C2 c1(CNC(c2n(CC(=C)C)nnn2)c2csnc2C)sc(Cl)cc1Br C1(C(C)O)CCCCN1C(C1(C(C)(C)C)CCCO1)=O c1(C(=O)NCC2(C)OCCN(C(C(C)OCOC)=O)C2)cccc2c1CC(=O)N2 c1(C(N2CCC(NC(c3nc(C)oc3)=O)C(F)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(C(=O)O)CCCN(C(c2ncoc2C2CCCNC2)=O)C1 Cc1c(C(=O)NC(CO)C(C)NC(c2cc(C3CC3)no2)=O)nn2ccccc12 c1(C(=O)NCC(=O)NC)ccc2c(n1)CCN(C(=O)C(O)C(C)C)C2 c1(OC)cncnc1C(=O)NCCC1CCN(C(=O)Cc2cccn2C)C1 C12CC(=NO1)C(=O)NC2.c1(CONC(Cc2cn(CC)nc2)=O)nc(C)sc1C C1(CC(=O)NC(CO)C2CCC2)CCN(c2ncccn2)CC1 Cn1cc2c(n1)CC(C(=O)NCC(C(C)(C)C)NC(=O)Cc1ccoc1)CC2 c1(N(C)CC2CCN(C(=O)CC3CCCOCC3)CC2)nc2ncc(Cl)cc2o1 C1(CNC(C(CC2CC2)OC)=O)(CO)CCN(C(=O)CC2CC(OC)C2)C1 C1(CCC(=O)N(CC(CC)NC(=O)C(C)(C)n2ccnn2)C)CC(C)(C)CO1 c1(C(=O)NCC(CNC(C(CCSC)OC)=O)C)c(N)nn2ccccc12 c1(OC)ccccc1C(CNC(=O)CNC(=O)C1CC1)NC(C1(Cl)CC1)=O CC1(C(=O)NC2COC(c3ccccc3)C2)CCCCO1 C(=O)(CCC(C)(C)C)N(C1CCCC(N(C(CCc2nc(C)sc2)=O)C)C1)C N1(C(c2ncc(OC)nc2)=O)CC=C(C(=O)NCC2(O)CC(O)C2)CC1 c1(NC(C(C)NC(=O)C(=O)NCc2ccccc2)=O)ccc(Cl)cc1C(F)(F)F CCC(C)CC(C(=O)NCCC1(OC)CCC1)NC(c1ncccc1CO)=O C=Cc1ccc(C(=O)NC(CN=[N+]=[N-])C(=O)NCCC2CCCC2(C)C)cc1 CC(CC(=O)NCC1CCCN(C(C2CCC3(CCC3)CC2)=O)C1)C(C)(C)C C(N=c1[nH]c(=NCC2CCCC2)c2ncccc2[nH]1)C1ON=C(C)C1 N1(C(c2c(C)non2)=O)CC(N=[N+]=[N-])CC1C(=O)NCC(F)(F)C(C)(C)O c1(SC)nc(C(=O)NCCCCCN(C(=O)CSC2CC2)C)c2ccccn12 CC(F)(F)C(F)(F)CC(=O)NC1CCCC1NC(=O)CCc1nc(=N)[nH][nH]1 c1(NC(C(N2CC(O)CC(C)C2)=O)=O)cc(F)c(Br)cc1F N1(C(=O)CN2CCS(=O)CC2)CCCC(O)(CC2CC2CN=Cc2cnc[nH]2)C1 N1(CC)CCCC1CCC(C)C.c1(C(C(=O)N2CCC(C)C2=O)C)nc(C)cs1 N1(C(C2(S(C)(=O)=O)CCC2)=O)CCN(C(c2ccc(O)cc2F)=O)CC12CCC2 O=C(CC1OCc2cc(Cl)ccc21)NC1CN(C(C2CCCC2)=O)C1 C1(C(N2C(C(=O)NCc3n(CC)cnn3)CC(=O)C2)=O)CCCC1C1CC1 N1(C(c2n(C)cnc2)=O)CC(NC(c2cnco2)=O)C(C#N)C1 c1(OC)cc(C(=O)NCCN(CC(C)O)C(=O)Cc2cn(C)nn2)cc(Cl)c1 c1(C(=O)NC2CCC(NC(c3ccn(COC)n3)=O)C2)noc(C)c1C(=O)OC C(=O)(CCCCCC#N)NC1CN(C(c2cnc(C)c(N)c2)=O)CC1C c1(NC(=O)NCC(C2CCCCC2)OC)cccc(S(=O)(=O)C(F)F)c1 c1(CCC(N2CC(C(=O)OC)C(N)C2)=O)c(I)ccnc1O C(CC)(CCCC(=O)NCc1nn[nH]c1C1CC1)NC(CSCCC)=O c1(C2(C(C)NCc3ccnc(Br)c3)CC2)c(F)cccc1F C(=O)(CC(C(F)F)NC(C1(C)CCN1C(=O)C(=O)N(C)C)=O)OC C1(n2cc(-c3c(C)nn(C)c3)nn2)CCN(C(=O)Cc2cccs2)CC1O N1(C(C2CC(SC)C2)=O)CC=C(C(=O)NCCCn2cnnc2C)CC1 Cc1cn(C)cc1C(=O)NCc1cccnc1CNC(c1ccc(=N)[nH]c1)=O CC1CC(NC(=O)CN(C)C(c2ccoc2)=O)CN1C(=O)C=Cc1cnn(C)c1 C(=O)(C1CCCn2cnnc21)NCC(CO)NC(CCNC(=O)NC)=O C1(NC(C2(SCC)CC2)=O)CN(C(=O)CNC(c2ccnc(O)c2)=O)CCC1C N1(C(c2nccc(OC)c2)=O)CCC(F)(F)C(CNC(=O)Cn2cc(Cl)cn2)C1 Cc1nc2c(N3CC4CN(S(=O)(=O)CCCl)CC34)ncnc2[nH]1 C(C)(CO)(C(=O)NC1CC=CCC1)NC(Cc1c(CC)con1)=O C1(CNC(C2(C=C)CCCC2)=O)CCC2(CCC2)C1NC(c1cccnc1C)=O c1(CC(=O)NCc2ccc(Cn3cc(Br)cn3)o2)csc(-c2ccccn2)n1 c1(OC)cc(NC(c2cn(C)cn2)=O)nc(C(F)(F)F)n1.N12CCC3C(CC13)C2=O CCN=c1ccc([N+](=O)[O-])c[nH]1.CC(=O)NN(C)C(=O)NC(C)=O C(=O)(CC(C)(C)C)N(CC(C)(CC)NC(C(F)=CC)=O)CC C1(NC(C(C)CF)=O)CCS(=O)(=O)C12CN(C(c1c3c(c[nH]c1=N)CCC3)=O)C2 C1(C(=O)NCC(C)CN(C)C(c2ccco2)=O)CCS(=O)(=O)C1.C1(=O)C(C)(C)N1 N(C(=NCCCc1nnc2ccccn12)NC1CCCCC1)C(C#C)C c1(C(=O)NC2(CCNC(C3CCC4CCC34)=O)CCC2)nccc2[nH]ccc12 N1(C(CCC2N(C)CCC2)=O)CC2CC1CN2c1nc(C2CCCCC2)ns1 C=CCCC(C(=O)NC1(c2ncc[nH]2)CC1)NC(C1CC(=O)N(C)C1)=O CN(C)S(=O)(=O)N(C)CC(N1CCCC(O)(CCNC(c2ccns2)=O)C1)=O c1(C(N2C(C)(OC)CC2)=O)ccc(Cn2nccn2)cc1 n1(CCC)nccc1C(c1nnnn1CCC)NC1(c2cccs2)CC1 C1(C(N2CCC2C(N2CCC(OC3CC3)CC2)=O)=O)CCC(C2CC2)C1.C1(O)CCC1 C1(CNC(=O)CC2CC=CC2)CC2COCC2N1C(c1ccc2cc[nH]c2c1)=O C(C1CCCCCC1)=CC(=O)N(CC(C)NC(c1cnn(C)c1)=O)C N1(C(C(C)n2cccn2)=O)CCC2(C1)CN(S(=O)(=O)c1ccn(C)n1)C2 c1(OC)ccc(C(=O)NC2CC2CNC(C2(F)C(C)(C)C2(C)C)=O)c(N)c1 N1(C(CC(C=C)C)=O)CCC(NC(c2cn(C)nc2C)=O)CC1c1ccccc1 c1(N2CC(CC)SCC2)ncnc(N(CCCC(=O)NC(C)C)C)c1C C(=O)(CCC(C)(F)F)N1CCC(CN(C(c2cc(C)nc(C)n2)=O)CC)CC1 C=CCC(C(=O)NCC(C)NC(=O)CC(C1CCCCCC1)C)c1ccccc1 c1(C(N2CC(NC(C3N(CC)CCC3)=O)C(C)C2)=O)ccnc2ccsc12 CCC(CCCC(=O)N1CC(N(C(=O)C=CC2CC2)C)C1)NC(=O)OC(C)(C)C c1(NC(C2(c3ccc(F)cc3Cl)CCC2)=O)cnc2c(c1)CCC2 C1(C(=O)NCCC2CCN(C(C3(CCC)CCC3)=O)C2)CC2COCC(C1)C2 N#Cc1ccc(C(N2CCN(CC3CCC3)CC2)C(=O)NC2CCOC2)c(F)c1 C12(CNC(C(C#C)(C)C)=O)CCCC1N(C(c1nn(C)cc1C#C)=O)CCC2 CCCCCCC(F)C(=O)NC1CN(C(=O)Cn2cc(F)ccc2=O)CC1F N1(c2ccccc2)CCN(C(=NCCc2cn[nH]c2)NCC2CC2)CC1 c1(C(=O)OCC)ccc(C(N2CC3C(C2)C3(C)C)C(=O)NCCOC)c(Cl)c1 C(=O)(C(C)(O)CC(F)(F)F)NCCC1(O)CN(C(c2cn(C)nn2)=O)C1 C1(C)(C(=O)NC2(C)CC(=C)C2)CCCN1C(C1CC(=C2CC2)C1)=O C(CC(C(=O)NC1(CCNC(=O)CCc2cn(C)nc2C)CCC1)N(C)C)SC N1(C(C(C)OCC(C)C)=O)C2CCC1C(CNC(=O)Cc1ccsc1Cl)C2 O=C(C1=CSCCO1)NCC1CCN1C(=O)COC1CCCC1 Cc1ccc(C)c(C(=O)NCC2CCN(C(=O)C(O)Cc3ccccn3)C2)c1 c1(C(=O)NC(C)CN(C(=O)CCSc2ccc(Cl)cc2)C)cccn(C)c1=O c1(C(=O)NCc2c(=N)cc[nH]c2)cnn2cnnc2c1 C12(C(N(C)CC3CN(C(=O)CCC(C)(C)C)C3)=O)CCCC1CC(F)(F)CC2 CN=c1[nH]c(=NCC2CC23CC3(F)F)[nH]c(=NC2COC(C)(C)OC2)[nH]1 Cc1ccc(NC(=O)CNC(=O)C(=O)N(C)Cc2ccc(F)cc2)cc1 C1(C(=O)NCCC)CCCN1CCC(=O)NCCC(C)(F)F C12(CC)CN(C(c3c(C)ncn3C)=O)C(CNC(=O)C(c3cncn3C)O)(C1)C2 N1(C(C(CC)(C)OC2CCCC2)=O)CCCN(C(=O)COC)C(C(C)C)C1 C(C(C)(O)CNC(=O)COCC1CCCO1)N(C)C(c1cnn(C2CC2)c1)=O c1(OCC)cccc(C(C(=O)NCCC2(C)CC2)N(C(CC)CC)CC)n1 CN1N=C(CC(=O)N(C)CC2CN(C(c3ccc(F)c(C#N)c3)=O)C2)CC1=O N1(C(C(=O)NCCNc2ccc(OC(F)F)cc2)C2C(C)C2)CCCC(C#N)C1 C1(CCNS(CCOC)(=O)=O)CCCN(C(=O)Nc2ccn(C3CC3)n2)C1 C1(F)(CNC(=O)C=CCn2cncn2)CCCN(C(C2CCS2(=O)=O)=O)C1 C1(C)(C(=O)NCCC2N(C(c3cccc(OC)n3)=O)CCOC2)CCC(=O)NC1 c1(CCC)ccc(C(=O)N(CC(CC)NC(=O)CC2CCCO2)CC)cc1 Cn1nc(O)cc1C(N1CC(C)(NC(C2CCC(=O)NC2)=O)C1)=O C1(CC(N2CC(CC(=O)OC)C2)=O)C2CCCC2N1C(C1CCOC1)=O CC(CN=c1[nH]c(=N)[nH]c(=NCCc2ccc(OC(F)F)nc2)[nH]1)N(C)C1CC1 C1(CC(=O)NCCC2(NC(C3CNC(=O)N3)=O)CCOCC2)CCC(F)(F)CC1 CCCCC(COC)NC(=O)CNC(=O)CNC(c1nnn(C)c1N)=O C(=O)(CCC(=O)C(C)(C)C)NCCN(CCC)C(c1ccc(CN(C)C)nc1)=O N#Cc1cccc(Cl)c1C(=O)NCCc1ccnc(O)c1 c1(C(N(CCNC(=O)CCCc2ccc(F)cc2)C2CC2)=O)cc(Cl)ccc1F CC1CC(NC(C2COC3(CCC3)C2)=O)CCN1C(=O)CC(F)(F)F N1(C(c2c(C)nc(CC)s2)=O)CC2CCC1CN2C(c1cc(F)c(F)cc1O)=O C1(C)(CC)CCCN1N(CC1CCCO1)Cc1ccc2c(c1)OCO2 c1(CC(C)C(=O)NC2CCCC(CNC(=O)CC(C)(C)O)C2)ccc(Cl)cc1 CCC(CC)(CC)C(=O)NCC(C)NC(c1sc(-n2cccc2)nc1C(C)C)=O c1(C(N2C(CNC(=O)CCNC(C3CCC3)=O)CCCC2)=O)cc2scnc2[nH]1 Cc1nn(C)c(=O)c(C(N2CCC(NC(=O)CN3C(=O)CCCC3=O)C2)=O)c1C c1(C(N2CCC(O)(CNC(C3(C)CCCC3)=O)CC2)=O)ccc2c(c1)COCO2 n1(C(C)C)cnc(C(N2CCCC2CNC(C2CC2F)=O)=O)n1 c1(C(=O)NCC(C)CN(C)C(c2cnc3c(c2)COC3)=O)cc2c(nn1)CCC2 C(N=c1nc(N2CCC(C)CC2)c2c([nH]1)CSC2)CS(CC)(=O)=O C1(C(N2C(NC(C34CC(C(=O)OC)(C3)C4)=O)CC(OC)C2)=O)CC12CCOCC2 N1(C(CC(CC)O)=O)CCCC(C(=O)Nc2ccc(N3CCOCC3)nc2)CC1 C1(CC(=O)NCC(CNC(COCC(=C)C)=O)CO)CC2CC(=O)C1C2 C(c1ccc(Cl)cc1Cl)=CC(=O)NCC(C)NC(C(CC=C)CC)=O C(=O)(CC1CCc2ccccc21)NC(CC(C)NC(c1c(C)cc(F)nc1)=O)C N1(C(c2cccc(SC)c2)=O)CCCN(C(=O)C(C)n2cccn2)CC1C c1(NC(C)=O)ccc(C(N2CCN(C(=O)Cc3c[nH]nc3C)C3CC23)=O)cc1C C(C)(CCNC(C1CC1(C)Br)=O)NC(C=CCOC)=O N1(C(c2n(C(C)C)ccn2)=O)CCC2(CCCN2C(c2cc[nH]n2)=O)CC1 CCC(C)(C#N)C(=O)NCc1ccc(Cn2cc(CCC(=O)OCC)nn2)cc1 c1(C(=O)NCC(CC(=O)NC2C(C)(C)C2(C)C)O)cc2occc2[nH]1 c1(C(=O)NCC(CNC(c2c(C)c(Br)no2)=O)C)c[nH]c2cccnc12 c1(C(=O)NCCC2CCCN2C(=O)Cc2cc[nH]n2)sc(F)cc1Br Cc1ccc(NC(=O)C(C)NCCC2CCCC2(F)F)cc1 N1(C(C(C(CC)O)C)=O)CCC2(CCN(C(=O)CN3CCc4ccccc43)C2)C1 C(C)(CN=c1[nH]cnc2c1CCCC2)NC(c1c(C)[nH]nc1Cl)=O c1(NC2(CO)CCCN(C(C3CC(C#C)(O)C3)=O)C2)cc(C#N)nc(C)n1 S(=O)(=O)(c1cc(C(=O)NC2(C)CCCN(C(C3(F)CC3)=O)C2)ccc1F)N(C)C CC1CCC(C)N1CC(N1CCCC1CN(C(=O)CCSc1ccccc1)C)=O c1(C(=O)NC(CCCNC(CSCCC(C)C)=O)(C)C)ccc2occc2n1 Cc1ncc(Cl)cc1C(=O)NCC(O)CCNC(=O)C(C)Cc1ccccc1 C(CCN=C(NCCC1CCCC1C)N(C)Cc1cccc(Cl)c1)SC c1(C(=O)OCC)cnc(N2CCCC(c3n[nH]cc3N)C2)nc1-c1ccco1 C1(C)(CNC(CC(C)CF)=O)COCCN(C(c2cnc(N)c(N)c2)=O)C1 C1(CC(=O)NCc2c(C)cco2)CC(C)(C)CN1C(C12CC1CNC2=O)=O N1(C(=O)C=CC2CC2)CCC2(C1)c1[nH]cnc1CCN2C(C1CCCOCC1)=O c1(C(C)F)ccc(C(=O)N(C2CN(C(=O)C=Cc3ccncn3)C2)C)cc1 c1(C(N2CCC(C)C2CNC(=O)C2=CCSC2)=O)ccc2c(c1)C(=O)NC2 c1(C(=O)NCC2N(C(CCOC)=O)CC2)cccc(Cc2nc[nH]n2)c1 C1(CNC(c2c(CC)csc2)=O)CN(C(C2CC23CC3)=O)C(C)(C)C1 O=C(C1=CCCSC1)NC1CC(NC(C2CCCCN2CC(F)F)=O)C1 c1(CC(N2CCCC(NC(C(CC)OC)=O)(CC)C2)=O)noc2ccccc12 C1(C(=O)Nc2c(C(=O)OC)cnn2C)CCN(N2CCOC(C)(C3CC3)C2)CC1 c1(CNC(N2CCC(CO)C2)=O)nc2ncc(Br)cn2n1 c1(C(C)C)ccc(C(=O)N(CCCCNC(=O)C(C2CCCO2)OC)C)c(O)c1 C1(NC(=O)CO)C2CC(CN(C(=O)C(F)C(F)(F)F)C2)C1CO.C(=O)CCOCC1CC1 C#CCCN=C(NCCC1CCCC1)N1CCC(C)(c2ccc(F)cc2)C1 c1(C(N(C(C)CCNC(=O)CSC(F)F)C)=O)cccc(=O)o1 C1(NC(CC=CCC)=O)CCC2(CCN(C(c3n[nH]c(C(C)C)n3)=O)C2)C1 C1(C(=O)NCCNC(=O)CC2COCC2O)CCCCC1c1ccccc1 c1(N(c2nccc(N3CCN(c4ccc(C)c(Cl)c4)CC3)n2)C)ccc(Cl)cc1N N1(C(CN(C)C)=O)CCCC(CN(C)C(C2CCN2S(C)(=O)=O)=O)C1 c1(C(=O)NCC(CC)(C)NC(C2(N(C)C)CCC2)=O)cc(OC)cc(OC)c1 C(C(CC(C)C)C(=O)NC1CC2(C1)CC2C(=O)N(C)Cc1cccc(F)c1)OC CCC(C)C(C(=O)NC1CNC(=O)C12CC2)NC(c1csc(=N)[nH]1)=O C1(C(=O)NCCC(C)NC(=O)OC(C)(C)C)(Cc2ccccc2)CC1(F)F C#CCCC(C(=O)NOCCOCC)NC(=O)Cn1[nH]cnc1=N C1(OC)(CNC(C2COCCN2C)=O)CCN(C(c2nc(Cl)cs2)=O)CC1 Cc1ccc(F)c(C(N2CCC3CN(C(C4(C)CCC(=O)CC4)=O)CC23)=O)c1F c1(C(N2CCC(CNC(C(CC)(C)CO)=O)C2)=O)cc(C)c2c(O)n[nH]c2n1 CC1(C)CN(CCC(N2CC(O)(CNC(=O)CCC3CCCCO3)C2)=O)CCS1 N1(C(C2N3CC(C)N(CC3)C2)=O)CC2(CCCCN2C(C2CCCN2N=O)=O)C1 c1(C(=O)NCCNC(CC2N(C(C)=O)CCC2)=O)cccc2c1CCC2 N1(C(c2c(C)scc2)=O)CCCC2(C1)CN(C(c1cnc(=N)[nH]c1)=O)CCO2 N1(c2cc(COC)ncn2)CC2CN(C(c3ccncc3O)=O)C2C1 CC1(C(=O)NC2(C(F)(F)F)CC2)CC(O)CN1C(c1ccsc1)=O C(=O)(C(CCCC)N1CCCC1=O)N(CCCCCCNC(C(C=C)O)=O)C C1(CC(=O)NCCCNC(=O)OC)COCCN1C(=O)CC(C)SC CC12CC(C(N3CCC(CCCN4CCOCC4)CC3)=O)(C1)C1(CCC1)O2 C1(C(N(CCC)CCO)=O)CC12CCN(C(c1sc(F)cc1C)=O)C2 N1(C(c2ncc(OC)cn2)=O)CC(NC(c2cc(Br)c(C)o2)=O)C2(CC2)C1 CCCCC(CNC(=O)Cc1ccccc1OCC(F)(F)F)NC(=O)CCF C(=O)(CCCCCC#N)NCC(C(=O)NCCN1CCC2CC12)N(C)C C1(C2CCCN(C(c3ccc(N)cc3)=O)C2)(NC(C(CC)=CC)=O)CC1 C(=O)(CCCCCC(C)O)N(C1CN(C(CCOC(C)C)=O)C1)C CC1(CNC(=O)C(CNC(C2CCC=CCC2)=O)CC2CCCC2)CCCC1O C1(CNC(CC(c2ccc(C)cc2)C)=O)CC(F)(F)CN1C(=O)C(C)CF N1(C(c2c(=O)ccn(C)c2)=O)CCC2(NC(c3ccc(O)nc3)=O)CCCCC12 C1(CNC(C2CCCN(C)C2)=O)(NC(=O)CCCC(F)(F)F)CCC(C)(C)CC1 CC1(C(=O)Nc2ccnn2-c2ccc(F)cc2)CCCN(CC(F)F)C1 N1(C(CC2CCN(C(C(=O)NC3CC3)=O)CC2)=O)CCC(O)C(F)(F)C1 c1(C(=O)NC(C2CCCN2C(=O)CCOC2CC2)(C)C)nc2cccnc2s1 N1(C(C2CC(SC)C2)=O)CCCCC(NC(c2cccnc2SC(F)F)=O)C1 n1(CC)nc(C(=O)NC2COCC2C(N2CCSCC2CO)=O)cc1O CCCCC(C)C(=O)NC1CN(C(c2cnc(Cl)cn2)=O)CC1(C)C N1(C(C23CC(CC)(C2)C3)=O)CC2CN(C(C3(C)C=CCC3)=O)CC2C1 C12(C(=O)NC3C(CNC(=O)CCCCC4CC4)CCCC3)CCCC1OCC2 CCC(CC)C(F)C(=O)NC(CNC(=O)CC1CC1)C1CCC1 Cc1cc(C(N2CCCC(CO)(Nc3ncnc4sccc34)C2)=O)cc(C)c1F CN1CCCCC(C(=O)NCC(O)CNC(c2cc(C(F)(F)F)ncn2)=O)C1=O C(=O)(C(CCC(C)(C)C)N(C1CCOC1C)C1CC1)NCCOCC Cc1cc(=NC2CCCN(CP(C)(C)=O)C2)[nH]c(NCCn2ncc(Br)n2)n1 Cc1nccc(C(=O)NC(C)CCNC(c2ncsc2Br)=O)c1Cl C1(CCNC(C=CCN(C)CC)=O)CC(OC)CN1C(=O)CCc1nncs1 C(CC(C)N=c1cc(C)c(C#N)c(C)[nH]1)NC(c1nc(OCC)oc1)=O CCC(CC)(CCNC(=O)C=C1CCCCC1)NC(c1ccoc1)=O N1(C(=O)CSC2CC2)CC(NC(C2(C3CCCCO3)CCOCC2)=O)CC(F)C1 n1(CCNC(C(N)=O)=O)cc(C(N2CC(n3ccnc3)C2)=O)cn1 c1(C(=O)NC(C(=O)NCCS(CC)=O)COC(C)C)sc(C)cc1C c1(C(=O)NCCCCCNC(C2(C)CCC2)=O)ccc(Cl)nc1 N1(c2n(CCOCC=C)c(-c3ccccc3Cl)nn2)CC(CCO)OCC1(C)C C#CCC(C)C(=O)NCC1CCCN1C(=O)Cn1cnnc1-c1ccc(=N)[nH]c1 CN1C(=O)COCC1CNC(C1C(NC(C2CCCCC2F)=O)C1(C)C)=O Cc1nc(N2CCC(C)C2CNC(c2ccn(C(C)(C)C)n2)=O)cc(O)n1 c1(CCC(=O)NCC(CNC(Cc2ccc(C)o2)=O)C)ccc(=N)[nH]c1 C=CCCCCCCC(=O)N(C)CC1CCCCN1C(=O)CC1CC2CCC1C2 N1(C(c2c(C)[nH]c(=N)s2)=O)CCC2(CCC(NC(C3CC3c3ccco3)=O)C2)C1 C(=O)(C(N)COC)NCC(c1ccco1)N(CC)CC.c1ccccc1 C(C(C(=O)N1CCC(C(C)NC(C2(CO)CCC2)=O)C1)C(C)(C)C)OCC(=C)C C=CC1CN(C(c2cccc(N)c2C(F)F)=O)CC1NC(c1cc(C#N)c[nH]1)=O c1(C(=O)NC(CN(C(C(C)OCC)=O)C)(C)C)ccoc1Br C1(C(=O)NCC(CNC(c2n(C)ncc2)=O)(C)O)CC2(CO1)CC(F)(F)C2 C1(C(C)C)CN(C(=O)C(O)C(F)(F)F)CCCN1C(c1ns[nH]c1=O)=O C(=O)(C(F)(F)CC)N(CCNC(C12CC(CCC)(C1)C2)=O)CC1CC1 c1(C(C(=O)NCCC#N)N(C2CCC2)CC2CC2)n[nH]c2c1CCCC2 C1(CN(C(C=C(C=C)C)=O)C)CCCN(C(=O)C(c2cccc(OC)n2)(F)F)C1 c1(-c2cccc(C(N(CC=C)Cc3ccncc3)=O)c2)cc(Cl)c(N)c(Cl)c1 C(C(C(=O)NC1CC(O)C1OC)N(C)C)NC(C1C(=C)C1)=O CC1CN(C(=O)C2=COCCC2)CC(CCNC(=O)CCc2ncco2)O1 c1(OC)ccc(-c2ccc(CNC(c3ncccc3Cl)=O)cn2)cc1OC Cc1nc(C(=O)NC(C(N2CC(S(C)(=O)=O)C2)=O)C2CCC2)ccc1C#N c1(CC)oc2ccccc2c1C=CC(=O)NCCNC(=O)C=C(C)C1CC1 C=Cc1cc(C(=O)NCCCNC(c2cccc(COC)c2)=O)cc(F)c1 C1(CC(=O)NCCCC(C)NC(Cc2c(C)scc2)=O)CCCN(C)C1 c1(NC(CC2CC(C)N(C(=O)CC3C(C)(C)C3(C)C)C2)=O)cc(Cl)cnc1O Cc1cccc(C(N2CCOCC(CNC(c3ccc(F)nc3F)=O)C2)=O)c1C c1(C(N2CCCC(CCC)(NC(=O)CC(C)CF)C2)=O)nccc2occc12 C(=O)(C(C)(C)CCC#N)NC1CC(C)CN(C(=O)COc2ccc(F)cc2)C1 C(=O)(CCCCCCNC(C1CCCS1)=O)NCC(C)Cn1cccn1 Cc1nn(CCO)cc1C(=O)NC1(C)CC(NC(=O)C(C)CN2CCCCC2)C1 N1(C(C(N2CCCC(C)C2)=O)=O)CCN(C(C2(O)CCOCC2)=O)CC1CO N1(C(C(C(CC)CC)C)=O)CCC(NC(=O)CCn2ccnn2)C(F)(F)CC1 N1(C(C(C)=O)=O)CCn2c(C(N3CCC4(CNC(=O)O4)C3)=O)cnc2C1 N1(C(C2(C)ON=C(C)C2)=O)CCC(C)(NC(C2CCCC(C(F)(F)F)O2)=O)CC1 C(=O)(C1=NOC(c2ccccc2)C1)N(CC(C)(C)NC(c1c(C)nns1)=O)C N1(C(CCC=C)=O)CC2(CCCCN(C(C3CC34CC(OCC)C4)=O)C2)C1 Cc1c[nH]c(C(=O)NC2(CN(C)C(c3c[nH]c(C(F)(F)F)c3)=O)CC2)c1 N1(C(c2ccncc2Cl)C(=O)NC)CCN(C2=NCC(C)S2)CC1 Cc1ccc(CC(=O)NCCN(C(=O)Cc2ccc(Cl)c(F)c2)C)cc1Cl c1(NC2CCC(NC(C(C)C3CCCC3)=O)CC2)ncc2c(n1)CCCC2 C=C1CCC(CNC(C2CC2c2cnn(CC)c2)=O)C1 N1(C(C(C2CC2)OCC)=O)CCC(C)C(CC(=O)Nc2cc(CO)ccc2C)C1 c1(C(=O)NCC=CCNC(C(CC)N(C)C)=O)cnn2c1CCCC2 N1(C(C2C(C)(C)C2)=O)CCC(C)(NC(=O)COCCc2ccccc2)C1 c1(CN(C(=O)CC2(C)CCN2C(=O)CSC(F)(F)F)C)ncccn1 c1(C(N(C2CCN(C(C=CCN(CC(F)(F)F)C)=O)C2)CC)=O)scc(C)c1Cl C1(C(=O)NCC2CC3CN(C(c4scc(C)c4C)=O)CC32)CN2CCN1C(C)C2 Cc1cn2c(C(=O)NCCC3CCN(C(=O)C(C)CC(N)=O)CC3)cnc2s1 C1(NC(c2c(CC)c[nH]c2)=O)CC2C1CCN2C(=O)CCC1C(=O)ON=C1C c1(C(=O)NC2CCCCN(C(C=C(COC)C)=O)C2)c(Cl)ccc2ncccc12 Cn1nnc2c1CCC(C(N1CCC(NC(c3cccnc3OC(F)F)=O)C1)=O)C2 CCCCCC(CC)C(=O)N1CCCN(C(=O)CN2CCNC(=O)C2)C(CO)C1 c1(NC(C(C)OC(C(=C)C)=O)=O)ccccc1CC#N C1(CC(C)Nc2ccn(C3CCCNC3)n2)CCCCN1 C(=O)(C(C)OC)N(CCNC(=O)CCNC(=O)OC)CC N1(C(C(C)n2ccnn2)=O)CC(C2CC2)(C(=O)NCC2CCOCC2(C)C)C1 Cc1ccc(C=CC(=O)N(C2C3CN(C(=O)Cc4nc(=N)[nH][nH]4)CC23)C)o1 c1(C(N2CCC(NC(CCCOC)=O)C(CO)CC2)=O)nn(C)c2ccccc12 C=CC1(CC(=O)NCCN2C(=O)CCC2=O)CN(C(=O)COC2CN(CC)C2)C1 N1(C(C(c2ccc(Cl)s2)C)=O)CC(F)(CNC(=O)C=CC2CCCO2)C1 C=CC1(CC(=O)NC2CCC2C(=O)Nc2cc(COC)on2)CCOCC1 C(C(=O)Nc1cc(C)ccc1C)(C(C)(C)C)NC(c1c(CC)[nH]cc1)=O N1(C(c2nc(C)oc2C)=O)CCC(C)(C)C1CC(=O)Nc1ccc(O)c(C)c1 C1(C(=O)NCc2cc(C)on2)CCCC12CCN(c1ncnc3sc(Br)cc13)C2 c1(C(=O)NC2C(NC(C(C)CC(F)(F)F)=O)COCC2)ccc(=O)n2c1CCC2 C1(CNC(C(CC)(C)CO)=O)CCC2(CN(C(C3CSC3)=O)C2)O1 N1(C(=O)C=CC2CCCCC2)CCN(C(c2cncnc2C2CC2)=O)C(CO)C1 C1(CNC(CC2CC(SC)C2)=O)CCN(C(c2cc[nH]c(=N)c2)=O)CC1C C1(C(N(C(C(=O)OC(c2c[nH]c(C)c2)=O)C)C)=O)CCC(C(C)C)N1CC CCC(O)C(C)C(=O)N(C(C)CNC(c1cc(C)n(C)c1C)=O)C c1(C(=O)NCCC2(CNC(CCCC(C)=O)=O)CC2)cc2n(c1)CCCNC2=O c1(CN(C(CC)(C)C)CCC#N)cccc(F)c1F n1(CCCSC)nnnc1C(c1cc(SC)[nH]n1)NCCC1C=CCC1 C12(C(=O)NCC3CC(NC(Cc4c(C)noc4Cl)=O)C3)CCC(F)(CC1)C2 C12(C(N(C)CC3CCC(NC(c4cc(CC)[nH]n4)=O)CC3)=O)CCC(F)(CC1)C2 c1(CC(=O)OCC(c2ccsn2)=O)c(F)ccc(Cl)c1Br c1(C(C)OC)ncc(C(=O)NN(c2scc(CSC3CC3)n2)C)s1 C(C1CCOCC1)=CC(N1CC(C)(C(=O)NCCOCC#C)C1)=O C1(CSC)CCN(C(=NCCc2ccc(F)c(F)c2)NCC(F)F)C1 CC1(C(=O)NC(CC(=O)NCCC2(C)CC2(F)F)C2CC2)CC(=O)C1 C1(C(N(CC(C)(C)O)CCC)=O)C(NC(=O)C(C)OCCOC)C1(C)C c1(C(C)O)ccc(-c2nnc(N3CCC3)n2CCCOCC2CCOC2)cc1 N(C(=NCCSC)N1CCC(C2(O)CC2)CC1)C1CCC2(CC(OC)C2)CC1 c1(OC)ccc(F)c(C(N2CCCC(C(C)NC(=O)C(Br)=C(C)C)C2)=O)c1F C(C(C)N=c1cccc(S(=O)(=O)N2Cc3nc(C)sc3C2)[nH]1)(C1CC1)OC CCCC(C(=O)N1CC(OC)C(NC(c2ccc(Br)cn2)=O)C1)OCC CCCC(C)(C)CC(=O)NCCCOCCN(C)C(C1(CO)CCOC1)=O CN1C(=O)OCC12CCN(C(c1cnnn1C)C(=O)NCCC1(C)CC1)C2 C12(NC(c3c(C)nc(O)[nH]3)=O)CCCN(C(C3(C(F)(F)F)CC3)=O)CC1C2 c1(-c2n(CC)cnn2)ccc(-c2noc(C3CC3(C)C)n2)cc1 N1(C(CC=CCNC(C(C)OC2CCCC2)=O)=O)CC=CC1CF C1(CC)C(NC(c2occc2C)=O)CCCN1C(=O)COCc1cccc(C)c1 Cc1n[nH]c(C)c1CCC(=O)NC1CCCC(CNC(=O)CC2CCC(C)C2)C1 C1(CN(C(c2c(CC)csc2)=O)C)CCCCN1C(=O)Cc1nncn1C(C)C Cc1nc2cc(C(N3CCN(C(=O)C(C)C#N)CC3C3CC3)=O)cc(Br)c2o1 c1(CC(C(=O)NCC(CN(C(=O)COC2CC2)C)(C)C)(C)C)ccc(C#N)cc1 N1(C(CC)=O)CCC(C)(CNC(C2CC(NC(=O)CO)C2)=O)C1 N1(C(C2(NC(CCOCCOC)=O)CCCC2)=O)CC2(CC(CO)CO2)C1 CC1CN(C(=O)CCC2CCCN2C)CC(C)C1Nc1nccc(Cl)n1 C1(NC(=O)NCc2cnc(C)nc2O)CC12CCC1(CC1)CC2 CC(C)CS(=O)(=O)CC(=O)NC1CC2CCC1N2C(C1(C)CNC(=O)C1)=O Cc1ccc(C)c2c1OCCC2Nc1ccc(Br)cc1C(F)(F)F N1(C(c2cc(C)[nH]n2)=O)CC2CC(NC(=O)CCNC(c3ccncc3)=O)C1C2 C1(CNC(CC(COC)(C)O)=O)CC2(CCC2)CN1C(=O)CCc1cc(C)on1 C(=O)(C(F)(F)Cc1ccc(Cl)cc1)N1CC(C(C)N)C1 N1(C(C)C(=O)NCc2ccc(O)nn2)CCC(Cc2ccccc2Cl)CC1 CCCC(CCC)CC(=O)NCCN(C(=O)CCc1ncc[nH]1)CC1CC1 C(CCC(N)=O)(C(=O)NC1CC1NC(=O)CCCCCc1cccs1)NC(C)=O c1(C(N2CCN(CC(C)NC(=O)C(O)CC(F)F)CC2)=O)cc(F)cc(F)c1O C1(NC(COCCCC)=O)CC(NC(C2CC=CCO2)=O)C(O)C1 Cc1c(C(N(C2CC3(CNC3)C2)Cc2cc(F)ncc2N(C)C)=O)cncc1Br N1(C(CN(C(C)C)C)=O)CCCC1(C)CNC(=O)CCOCCOCCCO c1(OCC)nc(N2CC(C(C)NC(=O)C(C)(C)c3ccccc3)C2)ncc1Cl N1(C(CC2CC(OCC)C2)=O)CCCN(CCc2cn(CCC3CC3)nn2)CC1 c1(CC)c(NCCC2CC(NC(c3cnn(CC4CC4)c3)=O)C2)ncnc1Cl N1(C(CCSC)=O)CCC2CCCC(C1)N2C(=O)C(c1cnn(C)c1)C C1(CC(=O)NC(C(C)NC(CC(CC=C)(C)C)=O)(C)C)Cn2ccnc2NC1=O c1(C(=O)NC(CC)C(=O)NCc2[nH]ccc(=O)c2O)cc(C)ncc1C CS(=O)(=O)c1nccc(=NC2CN(Cc3cccc(O)c3Cl)CC2C#N)[nH]1 C(=O)(C1CCc2c(Cl)cccc21)NCC1N(C(CC2CC=C(C)CC2)=O)CCC1 N1(C(C(CC)(C)OC)=O)CCN(C(c2ccc(-c3ccco3)o2)=O)CC12CC2 C1(NC(c2ccc(OC)nc2Cl)=O)C2CCC1CN(Cc1ccnn1C)C2 N1(C(c2cccc(F)c2F)=O)CCN(C(C2OCC3COCCC23)=O)CC(O)C1 Cc1ccc(S(N)(=O)=O)cc1C(=O)NC12CC1CN(C(C1(C#N)CC(C)C1)=O)C2 N1(C(C2(OC(C)C)CCC2)=O)CCOCC2(COCCN2C(c2ccc[nH]2)=O)C1 c1(C(=O)NCC(=C)CCNC(C2CCCO2)=O)cc(Br)cc2scnc12 CC1(C)C(CC(=O)NCC2(NC(C3CNC(=O)N3)=O)CCC2)CC1O N1(C(C)=O)CS(=O)(=O)CC1C(N1CCC(CNC(C2(C)CCCC2)=O)C1(C)C)=O C1(C(N2CCC3C(NC(c4cc5cnccc5[nH]4)=O)C32)=O)OCC2COCCC12 C(CCC(O)C(=O)NOC1CCCC1)NC(c1c(OC)cnnc1)=O CC(C)CC(C(=O)N1CCN(C(c2sccc2C#N)=O)CC1C)C(C)C C(=O)(C(C)(O)Cc1ccccc1)NCC(C)(C1CC1)NC(c1n(CC)ccc1)=O CCC(CC)C(C)C(=O)NCC1CN(C(=O)Cc2cc(F)ccc2OC)C1 Fc1cccc2c(N3CC4CSCC4C3)nc(N3CC4CCNCC4C3)nc12 N1(C(c2c(C)nc(C(C)C)cc2)=O)CC2CN(C(c3cnoc3C)=O)CC2(C)C1 N1(C(CCC(N)=O)=O)C(C(=O)NCc2cc(O)cc(F)c2)CCC12CC2 C1(C(N2CC(CC#C)OCC2)=O)N(C(c2cc[nH]n2)=O)CC12CCCC2 C1(CC(=O)NCC(CCC)NC(c2cn(CC=C)nn2)=O)CCCC(=O)C1 Cc1cc(C)nc(NC2CN(C(c3c(I)ccnc3F)=O)CC2C)n1 c1(CC(N2CC(OC)(CNC(C3CC(N=[N+]=[N-])C3)=O)C2)=O)ccccc1[N+](=O)[O-] C(=O)(C1=C2CCN=C2NC=C1)N1CC(CNC(Cc2cc(CC)no2)=O)OCC1 N1(C(c2nccc(OC)c2F)=O)CCCC12CCN(C(=O)Cc1ccccc1)C2 C1(C(=O)NCC(CCOC)NC(c2ccc(C(N)=O)cc2)=O)CC=C(C)CC1 N1(C(C2(CC)CC2)=O)CCC(C)C(NC(c2cc(C3CCCCC3)[nH]n2)=O)C1 c1(OCCCCC)ccc(CN2CCC(C(C)NC(=O)CCOC)C2)cc1 c1(CC(=O)NCC(N(C(C2C(=C)C2)=O)C)C2CC2)c[nH]c2cccc(OC)c12 CC1(NCC2CCCC(F)(F)CC2)CC(F)(F)CN1C(=O)OC(C)(C)C CCCC(CC)C(=O)N1CC(C(=O)NCCOCC(F)F)C(C)C1 C1(CNC(c2c(CC)occ2)=O)CN(C(=O)CSc2n[nH]c(O)n2)CCO1 C1(C(N(CCCNC(c2ccc(C(C)C)o2)=O)C2CC2)=O)CC2(C1)CC21CCC1 CCCCC1CC(=O)N1.C12(NC(=O)C=C(C)COC)CC(C1)C2 c1(OCC=C)ccc(Br)cc1C(=O)NC(c1nc(C2CC2)no1)(C)C N1(CC(=O)N(CCO)Cc2scc(C)c2)CCc2c(Br)cccc2C1 N1(C(CN(CC(C)C)C(C2CC3(CCC3=O)C2)=O)=O)CC2(CCC1CO)CC2 c1(C(C)C)ncoc1C(=O)NC(C1CCOC1)CNC(c1cc(Cl)ns1)=O C(=O)(C(O)C(C)(C)CC)N(C1CC2CN(C(C3(C(=O)OCC)CC3)=O)C1C2)C c1(C(CN(C(C=CCSCCOC)=O)CCN)C)cnn(C)c1 CCCCC(F)C(=O)NCCC1CC(C(=O)N(C2CCCCC2C)C)C1 C=CC(CC)CC(=O)NCCC1CCCN1c1nc(C)ns1 Cc1c(C(=O)N(C)CC2C3CN(C(=O)C(O)C(C)(C)C)CC23)cccc1F C1(CC(=O)NC2(C)CCN(c3cc(OCC)ncn3)C2)C(=O)N(C)N=C1C CC(CC(F)(F)F)C(=O)NC1CCC(CNC(c2ccc3[nH]ccc3n2)=O)CC1 c1(C(=O)NCCC(C)N(C(c2cc(C)cc(O)n2)=O)C)ccnc2cc[nH]c12 Cc1nc(=NCC2CCN(C(c3c(C)nc(O)nc3S)=O)C2)[nH]cc1Br C#Cc1cccc(C(N2CCCC(CN(c3ccncn3)C)C2)=O)c1 N1(C(C=Cc2ccn(C)c2)=O)CCCC12CCN(C(C1CCC(C)(C)CO1)=O)C2 N1(C(c2[nH]cc(C#N)c2)=O)CCC(O)CC1CC(=O)NC1CCC(F)(F)CC1 C1(C(=O)NCC2(OC)CC2)COCC1NC(C1(CO)CCCO1)=O C1(C)(NC(CC(C)C2CCCO2)=O)CCN(C(=O)C2=CSCS2)CC1 c1(C(=O)NCCCC2(NC(c3cncc(F)c3)=O)CC2)cnc2[nH]cnc2c1 N1(C(C2N(C)CCC2)=O)CCCC(O)(CNC(c2ccc(C(F)F)cc2)=O)CC1 C1(CNC(C(C=C)(F)F)=O)(CO)CC12CCN(C(c1coc(N(C)C)n1)=O)CC2 c1(C(=O)NC2CN(C(c3cncs3)=O)CC2O)cc(Cl)c2cc[nH]c2c1 c1(C(N2C(C)CC(NC(=O)CCOC3COC3)C2)=O)cc2c(F)cccc2s1 Cc1cccnc1C=CC(=O)NCC(C)N(C(=O)CC(C(F)F)n1ccnc1)C c1(CC)cscc1C(=O)NC1CCCC1CC(=O)NCC1SCCS1 C1(CN(C(C(Cn2ccc(C)n2)C)=O)C)COCCN1C(c1cc(Cl)cn1C)=O C1(NC(c2ccc(COC)o2)=O)CN(C(=O)C(F)CC2CCOC2)CC1C c1(C(=O)NCC(CO)NC(c2ccc(C)cc2O)=O)cc([N+](=O)[O-])c(C)cc1C C1(C(N2CCN(C(=O)NC3(C)CNC(=O)C3)CC2)=O)CCC(F)(F)CC1 c1(C(N(CCNC(=O)C(c2ccccc2)O)C2CC2)=O)c[nH]cc1Br C12(NC(=O)C=C3CCCC3)CCCC(CN(C(C3CC4(C3)CC43CC3)=O)C1)C2 c1(C(N2CC(C)C(NC(=O)CN(C)C)C(C)C2)=O)cc2cccc([N+](=O)[O-])c2[nH]1 N1(C(CC2C3CN(C(C(C)OCOC)=O)CC32)=O)CCOCC(O)C1 N1(C(C=CC)=O)CC2(CC(CC(=O)NCC3CCCCC(O)C3)C2)C1 Cc1[nH]c(Cl)nc(=NC2CN3CC23)c1C#N.C1CC1 N1(C(=O)Cc2cc[nH]n2)CCC2(CC1)CN(C(c1cc(F)cc(Cl)c1O)=O)C2 Cc1cc(C(=O)NC(c2cccc(C(=O)O)c2)Cc2ccccc2)nn1C Cc1cc(C(C)NC(=O)C(=O)NCc2cnn(C)c2)c(C)s1 CCC(C(=O)NCc1csc(C(=O)NC(c2ncc(C)s2)C)c1)OC N1(C(CC(CC)OC)=O)CCC(C2CC2)(CNC(C2CCC(CC)CC2)=O)C1 N1(C(C(=O)NCC(F)F)C2C(CC)C2)CCC(c2cccnn2)C1 C1(C(F)(F)C(=O)NC2CCC2NC(=O)CSCC(C)C)(OC)CCCC1 N1(C(C2(C#C)CCCC2)=O)CC2CC(NC(C3(C)CCN(C)C3)=O)C1C2 C1(CC)CCN(C(=O)C(C)N=[N+]=[N-])C(C(=O)NCCOC(C)=O)C1 C(=O)(C(C(C)C)n1ncc(N)n1)NCC(=C)CCNC(C1C(C)C1C)=O c1(-c2c(OC)c(F)ccc2)n[nH]c2cccc(C(=O)Nc3cnnc(C)c3C)c12 C1(C(=O)NCC(CC)(CC)NC(=O)C(C)N2CC(C)C2)CC2C=CC1C21CC1 C1(CNC(C=C(COC)C)=O)CN(C(c2sc(OC)nc2Cl)=O)C2COCC2O1 Cc1ccc(C(=O)NC2CCC2NC(=O)Cc2ccsn2)c(O)n1 C(=O)(C1Cc2ccc(Cl)cc21)NCC1N(C(c2ccc(OC)cc2O)=O)CCC1C N1(C(c2c(N)non2)=O)CCOC(CCNC(C2CC3CC2C3)=O)C1 C(CC(CNC(=O)C(C)(C)N(C)C)NC(=O)C(Cc1ccsc1)NC=O)OC c1(C(=O)NCC2C3CN(C(C4CC(=O)N4)=O)C2CCC3)ccc2cnccc2c1 C12(NC(CC3(C=C)CN(C(=O)CC(C)C4CC4)C3)=O)CCCC1OCC2 CC1=NOC(C(=O)N(C2CC(C(=O)NCCc3cnc(C)[nH]3)C2)C)C1 CC(C)C(C)CC(=O)N1CCC(CNC(=O)C(c2ccccc2Cl)O)CC1 N1(C(c2cccc(C)c2O)=O)CCC(C2(NC(=O)CCn3cc(Cl)cn3)CC2)C1 Cc1cc(C(N2CCN(CCNC(c3ccc(F)s3)=O)CC2)=O)c2c(c1)CCC2 c1(CC)nn(C)c(C(N2CC3CC3(CNC(=O)CN3CSCCSC3)C2)=O)c1Cl CC1CN(C(=O)CC2CC2C(F)(F)F)CCCN1C(=O)C=CCO Cc1cc(C)c(C=CC(=O)NCCCC(C)NC(C2CC(CF)C2)=O)c(C)c1 CCC(CC(=O)N1CCCCC(NC(C2(SC(C)C)CCC2)=O)C1)C(C)(C)C C12(C(=O)NC3CCC(CCNC(Cc4nc(C)[nH]n4)=O)C3)CC3CC1C2C3 n1(CCC)nccc1C(=O)NC1CCCC1CNC(=O)C(C)Cc1cnc[nH]1 c1(CN(C(CCC2(NC(C(C)OC(C)=O)=O)CCC2)=O)C2CC2)cnn(C)c1 c1(C(N(CCC(C)NC(=O)Cc2cc[nH]n2)C)=O)cc(Cl)c(F)cc1N O(N(C(=O)C1CC(C)CN1C(=O)CCn1cncn1)C(C)C)CC N1(C(C2(CSC)CC2)=O)CC(CNC(C2(C)CC=CC2)=O)C(F)(F)C1 C1(CN)CCCS1(=O)=O.n1(C(=O)NC)nnnc1CCc1csnc1C Cc1ccc(C(CCO)Nc2cc(NCC3CCCS3(=O)=O)ncn2)cc1 CC1(C)CC=C(C(=O)NC2CC3(C2)CC(NC(=O)CSCC(N)=O)C3)CC1 CCC(C)CC(C(=O)NC(C1CC1)C1CC1)NC(=O)CCn1cncn1 c1(C(N2CCCC(N3CCN(C(C4CCCO4)=O)CC3)C2)=O)ccc(F)cc1F C12(NC(C3CC(C#N)C3)=O)CCCC1CN(C(C1(CO)CC1)=O)C2 c1(OC)ccccc1NC(=O)C(c1cccc(Br)n1)N1CC=CCC1 c1(C(=O)NC2(CCF)CCC2)ccc2n[nH]cc2c1.C12CCOC1C(=O)NC2 N1(C(C(C(C)C)O)=O)CCC(n2cccn2)(CNC(c2cc(C#N)no2)=O)CC1 N1(C(c2ccc(C(C)=O)[nH]2)=O)CCOCC1CN(C(=O)Cc1cnoc1)C c1(C(=O)NC(CC)C(OC)OC)cc(S(=O)(=O)N2CCC2)ccc1F c1(C(N(CCNC(C=CC(=O)OC)=O)C2CC2)=O)cc(S(=O)(=O)N(C)C)c[nH]1 c1(-c2nnc(C)o2)ccccc1C(=O)NC(CNC(=O)C(C)NC(N)=O)C(C)C N1(Cc2nccc(C)c2)CC2(CN(C(=O)Cn3cc(CO)nn3)CC2C(=O)O)C1 C1(C(N2CCCC(CCNC(C3(C)CC3(F)F)=O)C2)=O)CCCC12CCOCC2 C(CN=C(NCC1(c2ccc(F)cc2Cl)CC1)NC1CCNC(=O)C1)OCC c1(CNCC(CN(CC)CC)O)cccc(C#N)c1 c1(C(=O)NC(CCC)CC(=O)N(CC(C2CC2)OC)C)cccc2[nH]ncc12 N1(C(c2cnc(C(C)C)s2)C(=O)NC2(C)CC2)CCc2cc(F)c(F)cc2C1C c1(NC(CC2(OC)CN(C(C34CC(CO3)C4)=O)C2)=O)nnccc1C Cc1cc(C(=O)NC(Cn2cccn2)C(N2CCN(C(C)C)CC2)=O)ncn1 C1(NC(C(C)C(F)F)=O)CN(C(c2ccnc(OC3CC3)c2)=O)CC(C)(C)C1 C1(C(N(C)Cc2c(C)nsc2)=O)COCCC1NC(c1cc(CCO)on1)=O c1(CC)n[nH]cc1C(=O)NC1CCC(N(C)C(c2cc(-c3ccco3)on2)=O)C1 c1(NC(c2cc[nH]n2)C)[nH]c(=NCCCC(F)F)nc2c1cnn2C C1(C(=O)NC2(CC=C)CCCN(C(=O)CCC)C2)CC2(CCCC2)CO1 Cc1sc(-c2ccncc2F)nc1CN1CCN(C(c2ccccc2)=O)CC1 C(CCCCCCO)(C(=O)NCC(=O)NC1CCOCC1)N1CCC(C2(C)N=N2)C1 c1(C(=O)NC(CN(C(C2N(C(C)=O)CC2)=O)C)C)cccnc1 C1(C(=O)NC2C(F)CCN(C(Cc3c(C)scc3)=O)C2)CCc2[nH]nc(O)c2C1 c1(C(=O)NC2C(NC(C3(OC)CC(C)(C)C3)=O)CCOC2)cn(C)c(=O)n1C c1(CC)cc(C(=O)NC(C)(CNC(C2CCS(=O)(=O)N2)=O)C2CCC2)ccc1F N1(C(c2cnc(C(C)C)s2)=O)CCC(NC(=O)CCCN2CCCCC2)C(O)C1 CC1(C)CCC(C(=O)NC2CCOC3(CCC3)C2)N(C(=O)OC(C)(C)C)C1 C1(NC(CCC(=O)NC)=O)CCN(C(c2c[nH]ccc2=N)=O)C12CC2 C(=O)(CCCCCC(C)(C)C)N1CCC2CN(C(c3c(SC)ccs3)=O)CC2C1 CC1CN(C(=O)CSc2ccccc2)CC1NC(=O)Cc1nncn1C Cc1nn2c(c1C(=O)N(CCCN(C)C(c1coc(Cl)n1)=O)C)CCCC2C c1(C(=O)NCCCN(C)C(C2CCC(C)(C)OC2)=O)ccc(Cl)c(C#N)n1 C1(CNC(C2(CC#C)CCCO2)=O)CCCC2(CN(C(=O)CC#N)C2)O1 c1(C(N2CCC(C(=O)Nc3ccc(O)nc3)C2)=O)cccc2ncccc12 N1(C(c2ccc(CC)s2)=O)CC(F)CC1CNC(C1(COC)CCCCO1)=O CN1CCN(C(C2CN(C(=O)COc3ccc(O)cc3Cl)CCO2)=O)C(CO)C1 C12(CNC(CC(C)OC)=O)COC(CNC(=O)Cc3cc(C)[nH]n3)(C1)C2 C1(C(=O)NCC(=C2CN(C(C3CCCN3C3CC3)=O)C2)F)CC2CCC1C2 C1(C(N2CCC(N(C(CCc3c(C)noc3C)=O)C)C2)=O)CCCC(F)(F)CC1 Cn1cnnc1CCCC(=O)NC1COCC1NC(c1cc[nH]c1C1CC1)=O C1(C(=O)NC2CCN(C(=O)CN3CCCC3CO)CC2)CCCC2(CC2)C1 CC(F)(F)C(C)(C)C(=O)NC1COCCC1NC(c1coc(C(F)F)n1)=O c1(-c2ccc(SCC)s2)ccc(-c2cnoc2)c(C)c1.N12OCC(C1=O)C2 C(C)(C)(CC(F)C(=O)N(C)Cc1cscn1)NC(C(C(C)C)SC)=O c1(C(N2C(C3CCN(C(CSC(C)C)=O)C3)CCC2)=O)cc2ccccn2c1 Cn1cc2c(C(N3CCC4(NC(=O)C5=NOC(C)(C)C5)CC4C3)=O)cccc2n1 Cc1ncccc1CC(=O)NCCCOCCN(C(=O)CN1CCCC1=O)C C1(NC(C2(OCC)CCC2)=O)CN(C(=O)Cn2ncccc2=O)CCC1CO C1(C)(C(N(CCC(=O)OCC)CC=C)=O)CCN(C)C1=O C1(NC(NCC2CCC(C(N)=O)O2)=S)CCC(=O)NC1 c1(C(N2CC(O)(CNC(C(C(C)(C)C)OC)=O)C2)=O)c(C)cc(O)cc1C C1(NC(C(C=CC)O)=O)CC2(CCN(C(c3cccc4nncn34)=O)C2)C1 c1(OC)ccc2nc(C)c(C(=O)NC(C)C(C)NC(c3ncoc3C)=O)cc2c1 C(CC(=O)NNC(=O)C(C)(C)CCCCNC(=O)CCCCC1CC1)OC C1(NC(C2CN(CCC)C(=O)C2)=O)CCN(C(c2c[nH]nc2OC)=O)CC1O C(CCC(=O)NC(c1n[nH]c(CO)n1)C)(C(C)C)NC(C(c1ccc(C)o1)C)=O C1(C(C)=O)(C(=O)NCCOCCN(C(C)COC(C)(C)C)CCOC)CC1 CC1CCCC(C)C1N(C(c1cnc(Cl)s1)C(=O)NCCOCC1CC1)C C1(C(N2CC3C(CNC(C4C=C(C)CS4)=O)(C3)C2)=O)CC2CCCC2C1 C1(C)(NC(C2C3N(C(c4c(C)csn4)=O)C(CC3)C2)=O)CN2CCC1CC2 C1(CCNC(c2nc(C)sc2)=O)CCCCN1C(c1cnnn1C)=O Cc1cn2c(n1)CC(C(N1CC(NC(=O)Cc3c[nH]nc3O)CCC1C)=O)C2 N#Cc1ncc(Br)cc1NC(C1C2CC1N(C(=O)CC1CCCC1)C2)=O CCCC(CNC(c1c(C)nsc1N)=O)C(=O)NC(c1nc[nH]n1)C1CC1 c1(Oc2cccc(-c3ccc(NC(C4CCCCO4)=O)s3)n2)ccc(Br)cc1F N1(C(C2CCN(C(CC3CCCC(C)O3)=O)C23CC3)=O)CCc2c(nnn2C)C1 CN1CC(C(=O)N(CCNC(=O)C(c2ccccc2)=O)CC2CCCCC2)NC1=O C(CC(C(C)(C)C)NC(C1CCCC1C1CC1)=O)N(C)C(c1c[nH]c(Br)c1)=O C1(C2C(C(=O)NCC(C)(C)C3CCC3)C2)CCCN1C(=O)CSCCC#N N1(C(C2(C)CC(=C)C2)=O)CC2(C1)OC1(CO)CC2(NC(=O)CC2(C)CC2(Cl)Cl)C1 CC1OC(=O)NC1C(N1CCCC(CNC(=O)CC2C=CCC2)C1)=O c1(NC2CC(NC(c3c(C)[nH]nc3Cl)=O)C2)ncnc2cccc(Br)c12 C1(C(=O)NC(CC=C)C2CC2)CC12CCN(C(=O)C=Cc1cc[nH]n1)C2 c1(C(N(CCC)C)=O)cnc2nc(NC(=O)C=Cc3ccc(C)o3)ccc2c1 N1(C(C2CC(C(=O)OC)C2)=O)CCN(C(=O)C=C(C2CC2)C2CC2)CC(C)(F)C1 N1(C(C)=O)CC2CCC(C1)C2CC(=O)Nc1c(C(N)=O)cccc1C CP(C)(=O)c1cccc(S(=O)(=O)NC2(C(F)(F)F)CC3C=CC2CC3)c1 Cc1cc(C)nc(SCC(=O)NCC2CC2CNC(c2cc(Cl)c[nH]2)=O)n1 C1(C(N(C)CC2CCCN2C(C2(C)CCC(=O)N2)=O)=O)CSC(c2ccccc2)=N1 C1(NC(CCC)=O)CCCN(C(c2ccnn2C)C(=O)NCCC2CC2)C1 CCC(CC(=O)NCC1CCOC1(C)C)NC(=O)CC(C)n1cccc1 c1(-c2scc(C(=O)NCC(CN(C(CC(C)N(C)C)=O)C)O)n2)cccc(Cl)c1 NS(=O)(=O)c1ccsc1C(=O)NCC1CCC(NC(C2CC(F)(CO)C2)=O)C1 Cc1cccc2c1CC(C(=O)NC1CN(C(C3(C)CCCCCC3)=O)CC1C)N2 C1(C(=O)NCC(C)NC(C2CCN(c3ccccc3)C2)=O)COC(C)C1 c1(N2CCC(NC(C3(C)CC=C(C)CC3)=O)C(C)C2)cc(C#N)ccc1[N+](=O)[O-] c1(C(N2C(CNC(=O)COC(F)(F)F)CC(OC)C2)=O)ccc2nc(C)cn2c1 N1(C(c2c(CNC(C3CC(C)(C)C3)=O)ccs2)=O)CC2CC=CC1C2 C1(NC(c2c(C)cco2)=O)CCCCN(C(c2cc3ccncc3s2)=O)CC1 N1(C(Cc2n(C)ncc2)=O)CC2CCN(C(c3cc(-c4ccco4)[nH]n3)=O)CC12 c1(C(=O)NCC2COCCN(C(C3(C)N(C)CCC3)=O)C2)coc(S(C)(=O)=O)c1 CCCCCCN(CC(=O)NC1CC(NC(=O)Cn2cc(C(=O)OC)cn2)C1)C C1(C(C(=O)N(CC(=O)OC)C)C)CCN(C(=O)C(C)(C)N2CCCC2)C1 N1(C(CC)C)C(=O)NC(c2cn(C)nc2C)C(C(=O)OC)=C1C1CC1C CON=Cc1ccc(C(=O)NCC2CN(C(=O)CC=C(C)C)CC23CC3)cc1 C1(NC(c2cscn2)=O)(CF)CCN(c2ccnc(CO)n2)C1 C(=O)(C1Cc2ccc(Cl)cc21)NC1C2CN(C(c3c(C)cns3)=O)C(C2)CC1 C1(CC(=O)NC(C2CN(C(=O)CC3(C)CCOC3)C2)C)CC(N(C)C)C1(C)C N1(C(Cc2nc(C)sc2)=O)CCCC2(NC(c3cnn(C)c3F)=O)CC2C1 C1(NC(C(C)Sc2ccc(Cl)cc2)=O)CC2C1CCN2C(=O)Cc1c[nH]nc1O N1(C(C2CC(=C)C2)=O)CCC2C(CCN2Cc2ccc([N+](=O)[O-])cc2O)C1 C1(NC(Cn2c(C)ncc2)=O)CC(NC(=O)C(F)(F)CN2CCCC2)C1(C)C C12(C(N3CCC(CN(C(=O)CC4(C)CC4(F)Cl)C)C3)=O)CC(CO)(C1)OC2C Cc1cc(C(=O)N(C)CCNC(c2c[nH]nc2C2CCC2)=O)c(N)c(F)c1 CC(C)C(CN(C)C)N=c1[nH]c(=NCc2c(Cl)cncc2Cl)[nH]c2cccnc12 C1(C(N2CCC(NC(CCc3ccc(SC)cc3)=O)C2)=O)CN(S(N)(=O)=O)C1 c1(C(N2CC3N(C(C4C(=C)C4)=O)CCC(C3)C2)=O)[nH]c2ccc(OC)cc2c1C C(=O)(N=c1ccn(CC(N)=O)[nH]1)C1N(C(C2N(C(=O)OC)CC2)=O)CC(O)C1 C(=O)(C(C(C)C)NC(=O)OC)N1CC(O)(C(C)NC(C(C)OCC)=O)C1 C1(=CC(=O)N(CCNC(C2(C)C(C)OCC2)=O)CC2CC2)CCC(C)(C)CC1 N1(C(c2c(CC)non2)=O)CCN(C(=O)C2=CCC(C(F)(F)F)OC2)CC(O)C1 C1(C(=O)OCC(N2CCCC2)=O)(SCC)CCCN1C(=O)C(C1CCC1)OC N1(C(C(COC)OC)=O)CC(OC)CC1CNC(=O)CCCN1CCCCC1 CC1(C)CC(CC(=O)NCC2CCN(C(c3cnc(C(F)(F)F)s3)=O)C2)CCO1 O=C(C1=CCN(C(=O)COC2CCCC2)CC1)NC12CCCCC1C2 C1(CCNC(C(C)OC)=O)CN(C(c2cc(-c3ccc(F)cc3)ns2)=O)CCO1 O(S(=O)(=O)c1ccccc1)c1cn(N2C(=O)N(c3ccc(Br)cc3)CC2)nc1 c1(C(=O)NCCC2CC(NC(c3cncnc3)=O)C2)cc2c(cc1F)NCCC2 C1(NC(CCCC(N)=O)=O)CN(C(=O)CNC(c2ccncc2)=O)C2CCCC12 c1(C(N2C(CNC(C(C)SCC)=O)C(CC)CC2)=O)nccc(N)c1Cl Cc1cc(C(=O)N(C)CC2COCCN2C(=O)CCCC2CC2)ccc1F C1(NC(C=C(C)C(F)F)=O)CCN(C(c2cccc(C3CC3)c2)=O)CC1C(C)C N1(CCC(=O)N(C(CC)CF)C)CCCCC1c1nc(O)n[nH]1 C(=O)(C(C)(F)CCCC)N1CCC(CN(C(C(C=C)(C)C)=O)C)C1 c1(C(=O)NCC2CCC(NC(C3C(C)OC(=O)N3)=O)C2)ccc(C(F)F)cc1F Cc1nccc(C(N2CC(NC(=O)CC3CCCNC3=O)C(O)C2)=O)n1 C1(C(N(CCC(=O)NCC(c2nccs2)C)C)=O)CC1C1CCCC1 C1(CNC(c2n(C)ncc2)=O)CN(C(=O)CONC(=O)OC(C)(C)C)C2CC12 N1(CC(=O)N(CCCCCNC(=O)COCc2ccccc2)CCl)CCOCC1=O C1(C(=O)NCC(C)(CO)NC(c2coc3c2COC3)=O)CCc2[nH]nc(O)c2C1 c1(C(=O)NCC(CN(C(c2cncc(OC)c2)=O)C)C)ccc2oc(C)nc2c1 N1(C(C(C)C#N)=O)CC(C(=O)Nc2cc(C#N)ccc2F)C2(CCC2)C1 c1(OCC)ncc(C(=O)NCC2CCN2C(=O)CCCOCCN(C)C)s1 CC(C(Cc1ccsc1)CO)O.C(=O)(CNC(=O)N(C)CCN)N(C)C CC(C)(CO)C(C)(C)NC(C1CCCCN(C(=O)CN2CC(=O)NC2=O)C1)=O C1(N)CC(F)CN(C(=O)CC2CC2)C1.C1(C=O)CCCN1C(=O)C1CC1 N1(C(C2N(CC)CCC2)=O)CCC(C(N2CC(CO)C(C)C2)=O)(CF)C1 C1(=CC(=O)NCCC2(C)CCN(C(C(=O)NCC)=O)C2)CCC(C)(C)CC1 c1(OC)ccc(NC(C2(NC(=O)CC3CCOC3)CCSC2)=O)cc1 N1(C(C(C)(C2CC2)OC)=O)CCC(CNC(c2c[nH]cc2C(C)(C)C)=O)C(C)C1 C1(C(N2CCOCC(F)(CNC(=O)C=C(Cl)Cl)C2)=O)CCOCC12CCC2 C#CC1(C(=O)NC2CCOC(C)C2)CCN(C(=O)CCCC2CC2C)C1 c1(C(CCCC)=O)ccc(O)c(CN2CCOC(C3CCCCC3)C2)c1 C(=O)(C(N=[N+]=[N-])C(C)C)N1C(CN(C(C2CC(CC(=O)OC)C2)=O)C)CCC1 N(C1CC2(CN(C(c3c(C)cnn3C)=O)C2)n2ccnc21)C(C(C(=C)C)(C)C)=O Cc1cc(C(=O)NC2CC(CNC(=O)C(F)=C3CCC3)C2)c2[nH]cnc2c1 CC1(C)CN(C(=O)Cn2cnnn2)CC(CNC(c2cc(Cl)ns2)=O)O1 C1(C(=O)NC(C)CC#N)CCCC(Nc2cc(-n3ccnc3)ncn2)C1 c1(C(=O)NCC2CCN(C(CNC(=O)NC)=O)C2(C)C)cnnc2ccccc12 C(=O)(C(=O)CC(C)CC)NC1CCCC(C(=O)NC(CC#C)CO)C1 c1(C(=O)NCC(CC)N(C(=O)C(O)CCC(C)C)C)c(C)cc(C)cc1C Cc1ccnn1C(C)C(N1CCCC1C(C)(C)C(=O)NCC(=O)NC(C)C)=O CC1CC(=O)NCC1C(=O)NCCN1CCC(NC(=O)Cn2cnnn2)CC1 C=CCC(C)C(=O)NCC1(C(N)=O)CN(C(C2(CF)CC2(F)F)=O)C1 C1(OC)C2CC3CN(C(C4CCCSC4)C(=O)NCCC4CC4)C1C3C2 c1(C(=O)NCCOCCN(C(=O)Cc2cnccn2)C)ns[nH]c1=O Cc1nc2cc(C(=O)NCC(C)(CO)NC(=O)CC3CCC(=O)N3)cnc2[nH]1 Cc1cc(C(N2CCC(CCC(=O)Nc3cnc(Cl)nc3C)CC2)=O)ccc1O c1(N(C)C)ccc(NC(=O)CC2CN(Cc3cccc(CO)n3)C2)cc1 C(=O)(C(O)CC[S+](C)C)NC1CCN(C(c2nccc(OC)c2OC)=O)C12CC2 n1(CC2(C)CCC2)nc(CS(C)(=O)=O)nc1-c1ccc(-c2cccc(Cl)c2)cn1 N1(C(c2c(COC)cccc2)=O)CC2CN(C(C3CC3(F)F)=O)CC2(C)C1 C#CC1(C(=O)NCCc2noc(=O)n2C)CCN(C(c2ncccc2F)=O)C1 c1(SC)ncc(Cl)c(C(N2CCN(C(c3cc4ncsc4[nH]3)=O)CC2C)=O)n1 N1(C(=O)NCC(C)Oc2ccc(Br)cc2)C2CCC1C(N)C2 c1(CN(C)CC)ccc(C)cc1.c12cn(nn1)CCC1CN(C1)C(=O)C2=O CCC(C)C(O)C(C)C(=O)N(C1(C(=O)N(CCCO)C)CCC1)C1CC1 N1(C(C2CCS(=O)(=O)C2)=O)CCC2CCN(C(C3(O)CCCC3)=O)CC2C1 C1(NC(C(C)N(C(CC)CO)Cc2cccc(Br)c2)=O)CC2CC3C(C2)C13 N1(C(C2N(C(CCn3ccc(C)n3)=O)CCC2)=O)CCC(F)(CNC2CC2)CC1 C1(C(=O)NCC(CC(=O)NCC2COCCO2)C2CCC2)CC2(CCO1)CC2 c1(C(=O)NCC2C(NC(c3ccc(N(C)CC)cc3)=O)C2)ccc2nncn2c1 c1(N2CCC(NC(CC)=O)C2)nc(N2CC3(C)COCC3(C)C2)nc2c1COC2 C1(CC)CN(C(=O)Cn2cc(C(c3ccccc3)OC)nn2)CC1N(C)C N1(C(CN(CCCCCC)C)=O)CCC(CNC(=O)CC2OCCC2C)C(C)C1 N1(C(COCC=C)=O)CCN(C(=O)Cc2ccsc2C)C(COC)C1 C1(NC(c2c(C)n(C)c(C3CCCC3)c2)=O)CC(=O)N2CCCCC12 C1(CC)CN(C(C2(OC)CCCC2)=O)CCC1NC(=O)C=C1CCCCC1(C)C O=C1NCCc2occ(C(N3CCCCC3c3cn(C4CC4)nn3)=O)c21 Cc1nc(Cl)ccc1S(=O)(=O)N(CC1CC1c1ccccc1)CC1COCCN1 S(=O)(=O)(c1ccc(NCC(c2ccsc2)C)c(F)c1)NC(COC)C(C)C C(=O)(CCCC(CC)NC(=O)CC1(OCC)CCC1)NCC1(CCC)CC1 N1(C(C2N(C(c3ccc(C#N)[nH]3)=O)C(C3CC3)CC2)=O)CCC2C(C(N)=O)C2C1 N1(C(COCCSC)=O)CCC(C=CC(=O)NCCOCC(F)F)CC1 Cc1ncnc(C(=O)NCCC2(C(=O)N(C)CC3CCCOC3)CCC2)c1C N1(C(C2ON=C(C)C2)=O)CCC(NC(c2cc(Br)c[nH]2)=O)C(C)(C)C1 CCCC(C(=O)NC(CCC(C)C)C(=O)NCCSCC(C)C)C(C)C c1(SCCC(=O)NC2CC(CCNC(CCC=CC)=O)C2)ccccc1Cl C(=O)(C(C)CC(C)C)NCCC1N(C(c2n(CC)ncc2)=O)CCSC1 C1(NC(c2c(CSC)cccn2)=O)CCCN(C(=O)CCC2CCN(C)C2)CC1 N1(C(C2C(CC)CCC2)=O)CC(C)(C)CC1CNC(=O)CC1CC(O)C1(C)C C(=O)(C(O)P(C)(C)=O)NC(CCC)C.C1(=O)C=CCOCCN1CC c1(N2CC(C)(CNC(c3c(OC)cc(Cl)nc3)=O)C2)ncc2cn[nH]c2n1 C1(CNC(=O)CCCN2CCCC2)C2CC1N(C(=O)C=CCN1CCOCC1)C2 Cn1cc(C(=O)NCCN(C(C2C3COCC23)=O)C2CC2)c(C(C)(F)F)n1 c1(C(=O)NC(CCCC)CNC(=O)CC2(C)CC(F)(F)C2)cc(O)nc(O)n1 Cc1nc2ccc(C(N3CC4CCCN(C(C5CC(C)CO5)=O)C4C3)=O)cc2o1 C1(CC(=O)NCC(CN(C(c2cnc(CCCC)s2)=O)C)(C)C)CCCCC1F c1(C2(C(=O)NCCC3CCN(C(=O)C(F)(F)CO)C3)CC2)ccc(F)c(Cl)c1 N1(C(C(=O)NCCC2(O)CN(C(C3N(C(C)=O)CCC3)=O)C2)C)CCCC(O)C1 c1(NC(=O)OC)cc(-c2n[nH]c(C)n2)ccc1C.c12cc(ccc1Cl)C(=O)N2 c1(C(N2CCC(F)(CNC(=O)C3CC3)C2)=O)cccc(C2CC2)n1 N1(C(C2CN(C(c3c(CC)nccn3)=O)C(C)CC2)=O)CC2CC(OC)C(C2)C1 C(COCc1ccccc1)(C(=O)NC1CC(F)(CNC(C2CCCO2)=O)C1)OC C1(C(=O)NC(C(CO)NC(Cc2c(C)cccn2)=O)C)COc2ccccc2O1 C1(OC)CC2CC1CN(C(C1CCC(C)C1)C(=O)Nc1ccc(F)cc1C)C2 C(=O)(C1CCCc2n[nH]cc21)N1C(CNC(c2ccc(CC)cc2F)=O)C=CC1 CC1c2ccccc2CC1C(=O)NC1(CO)CN(C(c2cc[nH]c2)=O)C1 C1(CC(N2C(CNC(CN(C)C3CC3)=O)CCC2)=O)Sc2ccccc2NC1=O N1(C(C(CC(=C)C)C)=O)CC(NC(=O)Cc2ccccc2Cl)CC2(CC2)C1 c1(CCC)cc(C(=O)NCCNC(=O)Cc2cccnc2C)ccn1 CCC(C(=O)N1CCCC1CN(C(C1CC1C)=O)CC)N(C)C c1(OC)ccnc(C(=O)NCC(C)CC(=O)N2CCC2CO)c1 CC#CCC(C(=O)Nc1cnn(CCF)c1)NC(c1cccc(C)c1)=O N1(C(C(CCC(C)C)F)=O)CCCC2C1CCCN2C(=O)CCN1CCCC1 CC1=C(C(=O)N2CC(F)(C(=O)NCC3CCOC3)C2)CCC1 n1(CC(=O)N(C2CCN(C(C3CCC(F)(F)C3)=O)C2)C)ccc2ccc(F)cc12 c1(N(C)CC2C(C)C2)nc(N2CCCC(CNS(C)(=O)=O)C2)nc2c1cnn2C C12(C(N3CCC(NC(C(CSC)(C)C)=O)C(O)C3)=O)CC3CC(C(=O)N1)C2C3 C12(NC(C=CC(=O)OCC)=O)CCC(CN(C(c3cc(C)c(C)s3)=O)C1)C2 CCCC(C(=O)N(C1(C(N2CCC2CF)=O)CC1)C)OC N1(C(CCN(C(=O)C2=NN(C)C(=O)CC2)C(C)C)=O)CCC2(CCN(C)C2)C1 CC(O)(CC(=O)N1CC2=C(C1)CN(C(=O)COC(F)(F)C(F)(F)F)C2)C(F)(F)F N1(C(C(C)n2cccn2)=O)C2CCC1CC(F)(CNC(=O)CN(C)C)C2 c1(C(=O)NC2CCN(C(C3C(CC)N(C)CC3)=O)C2)cc(O)nc2cnccc12 Cc1cc(N)ccc1C(N1CC(N(C)C(c2cnc(O)c(F)c2)=O)C2(CC2)C1)=O C1(CCNC(C(C)(C)C2CCC2)=O)CCN(C(=O)C(N2CCCC2)C2CC2)CC1 C1(CNC(C2(C=C)CC2)=O)COCCN(C(=O)C(C)(C)c2cncs2)C1 Fc1ccc(Br)c(CCNCC2C3CCC4C(C3)CC24)c1 c1(CNC(C2CCCN(C(c3ccn(CCOC)n3)=O)C2)=O)ccc(F)nc1C C1(C(N2C(COC)C(C)(C)C2)=O)CNC(=O)CN1C(=O)Cc1scnc1C c1(C(N2C(C)CC(NC(=O)CCC3CCC(C)O3)C2)=O)ccn2nncc2c1 N1(C(COCCC)=O)CC(F)(C(=O)NCC(C)OCCO)C1 c1(C(C2(C)COC2)NCCSCC(C)Cn2cccn2)nnnn1C1CCC1 C1(CCNC(c2cn(C(F)(F)F)cn2)=O)CCCN1C(=O)CNc1ccccn1 C(=O)(C1CCc2sc(CNC(=O)NCCC3CCC(F)(F)C3)nc21)OCC CC(C)C(N=[N+]=[N-])C(=O)NCC1COC(CNC(=O)CCc2cncs2)C1 C1(NC(C(n2ncc(C)c2)C)=O)CCC12CN(C(c1cccnc1C)=O)C2 c1(C(=O)NC2C=CCN(C(C3C(CC)CCO3)=O)C2)cc(C)c(F)cc1Cl c1(NC(C2CC(NC(C(C)C)=O)C2)=O)cc(Cl)c(C#N)cc1[N+](=O)[O-] N1(C(C#CC2(CC)CC2)=O)CCC2CN(C(c3cnc(C)cn3)=O)CC2C1 Cc1cc(NC2CC3CC3C2)ncc1S(=O)(=O)N1CCC(C)C(F)(F)CC1 N1(C(C2C(C(=O)OC)CC2)=O)CCC2CCCC12C(=O)NC(C)CN=[N+]=[N-] C(=O)(CC(C(F)F)NC(=O)CCC(N)=O)N1CCC(NC(C)=O)CC1 c1(-c2ccc(C(C3CC3)NC(C=C(C)C)C)cn2)ccc(F)c(F)c1 c1(C(N2CCC(N(C(c3csc(C(F)(F)F)n3)=O)CC)C2)=O)ccc(F)nc1F c1(CS(C)=O)c(CN2CC2CNC(=O)OCC2CCCO2)oc2ccccc12 C1(C(=O)NC(CSC)(C)C(=O)NC(CN(C)C)CO)CC(=O)OC1(C)C c1(NC(C23CC(Cc4ccccc4)(C2)C3)=O)ccc(C2=CCC(O)CC2)cn1 C(c1cccc(Cl)c1)=CC(=O)NC1(CO)CN(c2nc(C3CC3)ns2)C1 C1(C(N2CC(NC(c3c(CC)nco3)=O)(CO)C2)=O)CCC(C(F)F)CC1 c1(OC)ccc(CC(=O)NC2CC(NC(c3cc(Cl)nc(Cl)c3)=O)C2)cc1Br C1(NC(C(CC)(C)C)=O)CN(C(C2CN(S(N)(=O)=O)C2)=O)CC1C1CC1 Cc1nn2c(C(N3CCC(CNC(c4ncccc4Cl)=O)C3)=O)c(C)nc2s1 c1(C(N(C2CC2)Cc2ccc(OC(C)=O)cc2)=O)cc(C)nc(Cl)c1 C(=O)(C(C)C(=O)N1CCOCC1c1ccc(C(=O)N(C)CC2(C)CC2)n1C)OC C(=O)(CC(C)CC(=O)N1CCCC1CN(C)C(c1cccc(F)c1SC)=O)OC C1(C(N2CCC(N(C(C(C)OCC=C)=O)CC)C2)=O)SC2C=CC1CC2 C(=O)(CCC(C)(C)NC(c1ncncc1Cl)=O)NC(C(C)O)C c1(CNC(C2(C)CC=C(C)CC2)=O)nc2c(s1)CN(C(c1ccoc1)=O)CC2 N1(C(CC=CCNC(C2C(CCC)C2)=O)=O)CC2C(C(=O)OC)C2C1 C1(NC(C(c2cccc(C)c2)C)=O)CCC(C)N(Cc2cc(C)on2)C1 C(=O)(C1Cc2c(Cl)cccc21)N1CCC(CCNC(CCC=C)=O)C(F)(F)C1 c1(C(=O)NCC2(F)CN(C(C34CCC(CC3)CO4)=O)C2)cc2ccc(Cl)cc2o1 N1(C(CCCN(CCC)CCC)=O)CC2(CC(NC(C3CCN(C)C3C)=O)C2)C1 C1(C(=O)NC(CNC(C2(CCCC)CCC2)=O)(C)CO)CS(=O)(=O)CC(=O)N1 CC(C)(C)C(=O)C(=O)N1CCCC1C(C)(C)CNC(C1(Cl)CC12CCC2)=O C1(C(N2CCC(O)(C(=O)NC(C)C)C2)=O)(COC)CCN(C)CC1 S1(=O)(=O)c2ccc(cc2)N1.CC1(C)CN(S(=O)(=O)C(F)(F)F)CCC1CO N1(C(C(C=C)(F)F)=O)CCC2(CCN(C(=O)CC(CC)C(C)(C)C)CC2)C1 N1(C(c2cn(CCCC)nn2)=O)CC2C3CCC(C2C1)N(C(=O)CNC(C)=O)C3 CCC(C)(C)CC(C(=O)NCCCF)N1CCOC(C(N)=O)C1 C=CC1(CC(=O)NC2(C(=O)O)CCC2)CCC1 C1(C(N2CC(NC(C(C)(C)N(C)C)=O)C(F)CC2)=O)Cc2ccccc2S1 C=CCC(C)(O)C(=O)NCc1cccc(C(=O)NCC2(C)NC(=O)NC2=O)n1 C(=O)(C(C)N(OC)C(=O)CCN(OC)C(=O)C1CN(CCC2CC2)C1)OC C=CCC(C(=O)NCc1nnc(C)n1CC)NC(=O)CCSCCCC c1(C(N2CCC(=C)CC2C(N2CCCC(CCC)C2)=O)=O)cccc2ccnn12 C(COC(=O)C(Cc1ccccc1)C(=O)OC(C)(C)C)(CC(C)C)OC c1(C(=O)NCC2CCN(C(c3n[nH]c(CC)c3Cl)=O)C2)cc2cccn2cn1 CC(C)C(CCc1ccc(Cl)cc1)(c1nnnn1CC(F)F)NCCC1CSC1 N1(C(c2cc(C)cc(Br)c2)C(=O)NC(C(=O)OC)C)CCc2ccc(F)cc21 N1(Cc2n(C(F)F)ncc2)CCC(F)(F)CC12CCC2 N1(C(C(CN(C)C)N(C)C)=O)CCC(C)(C)CC1C(=O)NCc1ccncc1F C(CN=c1[nH]c(=NCc2cccc(C3CC3)c2)[nH]c2c1CCC2)C1(C)CCCO1 CC(C)(O)C(O)C(C)(C)NC(=O)C(CCCc1nn[nH]n1)NC(=O)OC(C)(C)C c1(C(=O)NC(CCNC(C(F)=C(C)C)=O)(C)C)ccc(-n2cnnn2)cn1 CCCCCCC(C)C(=O)NC12CCC(CNC(=O)C3=CCCCC3)(C1)OC2 C12(NC(C(CCCC)C)=O)CCCC1N(Cc1nc(-c3ccccc3)no1)CC2 C=Cc1cc(C(N2CC(NC(=O)CCc3nc(CSC)no3)CC2C)=O)cc(F)c1 N1(C(C2(C)CCCS2(=O)=O)=O)C2CCC1CC(CN=c1ncc(F)c[nH]1)C2 Cc1ccc(Br)c(CN2CCC(F)(C(=O)NC(C#N)C(N)=O)C2)c1 CC1CCCC(CC(N2CCC(CC(=O)NC34CCN(CC3)C4)C2)=O)O1 C1(C(N(CC(C)NC(c2nccc(C)n2)=O)C)=O)CC(C2CCC2)C1 C1(NC(CCCOC(C)C)=O)C2CCC1N(C(=O)CC1CCCCN1C)C2 c1(CNC(=O)C(O)CC2CCCCC2)cccc(NC(C2CCC3(CC3)C2)=O)c1 C(CCNC(C1CN(C2CCC2)C1)=O)(C(=O)NCC1CC(C)(C)CO1)OC CCC1=NOC(C(=O)NC2(C)CC(NC(c3cc(C)oc3C)=O)C2)C1 c1(CC)ccc(C(C)=CC(=O)NCCN(C(=O)C(=O)NC2CC2)CC2CC2)cc1 C1(OC)(CNC(c2csc(-c3cnn(C)c3)n2)=O)CCN(C(=O)CNC(N)=O)C1 C12CCCC(C1)NC2=O.c1(OC)cc(C(=O)NC2CN(C(COC)=O)C2)on1 c1(C(c2ccsn2)NCCCNC(N)=O)nnnn1CC1CCOC1 Cc1cnccc1N1CCN(C(=O)NC(c2ccc(Br)cc2)C(F)(F)F)CC1 CC(CC(=O)N1CC(S(C)(=N)=O)C1)CC(C)(C)C.C1CCC(=O)NC12CCC2 c1(C(N(C)CC2CCN(C(C(C)S(N)(=O)=O)=O)CC2)=O)ccc(F)c(O)c1F C(=O)(C(C)(O)CC(C)C)NC1CCN(C2CCN(Cn3c(C)ncc3)C2)CC1 c1(C(=O)NCC(CC(=O)OCC)C)cc(I)ccc1O Cn1nnc2c1CC(C(=O)NCC1(O)CCCN(C(C34CC(C3)C4)=O)CC1)CC2 CC1CC(NC(c2c[nH]nc2CNC(=O)CCC2CC2)=O)C(C)CN1C C(N=c1[nH]c(=NCCNS(=O)(=O)NC(C)C)[nH]c2c1COCC2)C1C(CC)C1 C1(F)(C(=O)NC2CC(NC(C3CCC(C)CC3)=O)CC2O)CCCN(C)C1 CCS(=O)(=O)N1CC(C(=O)NCCC(c2cccs2)NC(=O)COC2CCOC2)C1 C(=O)(CCCS(C)(=O)=O)N1CC(N(C(C2CC=C(C)CC2)=O)C)C2(C1)CC2 C1(C(N2C(CNC(C=Cc3nc(C)c(C)[nH]3)=O)C=CC2)=O)CC2OC(=O)OC2C1 c1(CC)cnccc1C(=O)NCC(C)CN(C)C(c1nc(Br)c[nH]1)=O C(=O)(C(CC(F)F)NC(C1C=CCC1)=O)NCC(C)(O)CO C(=O)(CC(C)n1cccn1)NC(C(=O)NCCC(=O)N(CC)CC)c1cccs1 C1(C(N2CC(OC)C2)=O)C(C)CCN1C(c1cnccc1C)=O c1(C(N2CCN(C(=O)Cn3ccnn3)C(C(F)F)C2)=O)cnc2ncccc2c1 c1(C(C)=O)ccc(Cl)cc1S(=O)(=O)NC1CCC[Si](C)(C)C1 C#Cc1ccnc(C(=O)NC(CC(=C)C)C(=O)N(C)Cc2ccnn2CC)c1 n1(CC(=O)NC2CCC(NC(CN3C(C)CC3)=O)CC2)cc(C#N)c(O)nc1=O Cc1cc(=NCC2(S(=O)(=O)NC(C)(C)C)CC2)[nH]c(=NCC2OCCC2C)[nH]1 N1(C(C(C(C)(C)O)NC(C(C)OCCOCC)=O)=O)CCC12CCOCC2 C1(C(=O)NC(C)(CNC(c2ccc(CO)nc2)=O)CO)CCc2nc(O)[nH]c2C1 c1(C(=O)NCC2N(C(c3ccc(CC)o3)=O)CC2)cc(F)c2cn[nH]c2c1 C1(CNC(c2ccc(CCF)cc2)=O)COCCN(C(=O)CC2CCCC2)C1 C1(NC(c2ccn(C(F)F)n2)=O)CCOCC1NC(C1CC(C(F)F)C1)=O CC(C)C(=O)C(=O)N1CC2C(CNC(c3cccnc3)=O)C2C1 C=C1CCN(C(=O)CC2CC=CC2)C(C(=O)NC2CC2C2CCC2)C1 c1(CN(C2CCN(CC)CC2)CC2CCN(C(C)=O)C2)ccc(S(C)=O)cc1 c1(NCC(=O)NCC2CCC(NC(=O)COC3CC=CC3)C2)ccc(F)c(F)c1 c1(C(=O)NC2CN(C(c3ccc(C(OC)OC)o3)=O)C2)nccc2n[nH]cc12 C1(CNC(c2n[nH]c(C)c2Cl)=O)CN(C(C2COC(=O)N2)=O)CCC1(C)C C(CC(F)(F)F)SCC(=O)NCC(C)CNC(C1(Cc2ccccc2)CC1)=O CC1CN(C)CCCN1C(C1CC2CC1CN(C(C1SCCS1)=O)C2)=O C1(C(N(C2CC(C#N)C2)CC(=O)NCC2CC(F)(F)C2)=O)CCC(CO)CC1 C1(NC(CC2(CC)CCC2)=O)CC(C(=O)NC2CC2O)CC1O CN1CCCCC1C(=O)NO.c1(-n2cc(CN)nn2)ccc(OC(F)(F)F)cn1 C1(C(=O)NC(c2nc(C)[nH]n2)(C)C)(NC(=O)C(C)C2CC2)CCN(C)C1 N1(C(=O)CCC=CBr)CCN(C(c2cc(F)c[nH]2)=O)C2CCCCC2C1 C(=O)(C1CCCc2ncnn21)NC1C(CNC(=O)CCn2cccnc2=O)CC1 N1(C(C2CCN(CC)C2)=O)CC(C)C(C)(CNC(c2[nH]cc(C)c2C)=O)C1 C1(NC(c2c(C)nc[nH]2)=O)CCN(C(c2c(N)ccc(F)c2C)=O)CC(C)(C)C1 C1(NC(C(C)(C)C2CCCCC2)=O)C=CCN(C(c2nc[nH]c2C(F)(F)F)=O)C1 Cc1ccccc1C(=O)NCC(=O)NCCCCCNC(C1(C)COC(=O)C1)=O C1(C(=O)NC2C(OC)CN(C(c3c[nH]nc3C)=O)C2)COCC2(CCC2)O1 C1(C(N2CC(=C)C2)=O)CCC(C2CC2)N1C(C1(n2cnnn2)CC1)=O C1(C(N2CCC(N(C(CCCN=[N+]=[N-])=O)CCO)C2)=O)CCn2cncc2C1 c1(C(=O)NCC(CN(C(=O)CC2CCCN(C)C2)C)O)cccc(CF)c1 Cc1c(Cl)c(C(=O)NC2(CNC(C34COC(CF)(C3)C4)=O)CCOC2)nn1C Cc1cc(Cl)c(C(N2C3CCC2CC(NC(C2(C(C)C)COC2)=O)C3)=O)cc1C N1(C(c2cc(CCC)nn2C)=O)CCN(C(C2(CC)CCCC2)=O)CCC1C CC(=O)CCCC(=O)N1CCC(CCC(=O)O)CC1 Cc1cccc2cc(-c3ccc(CNCc4c(F)cccc4F)cc3)c(O)nc12 N1(C(CSCCOC)=O)CC(NC(c2c[nH]c(Br)c2)=O)C2CC12 c1(C(=O)NC(CC)CN(C(=O)C(C)OCC2CC2)C)cccc(CC(F)(F)F)c1 n1(CCO)nc(C(=O)N(CC(O)CNC)C)ccc1=O.N1(CC)CCCC(C)C1 CC1CN(C(C2(C)CC3CCC2C3)=O)CCC1NC(C1CC2CCC1C2)=O c1(C(N2CCCN(C(c3cnc(C)s3)=O)C(C)C2)=O)cnn2c1C(=O)CCC2 N1(CC)CC2CC(OC)(C2)C1.C12(C)C=CC(C1)NC2=O Cc1cc(F)c(C(N2C(C(=O)Nc3cnn4cccnc34)CCC2C)=O)c(F)c1 n1(CC(C)C)ncc(C(=O)NC(C)C(C)NC(C2(c3cccnc3)CC2)=O)c1N C1(NC(C(CCC)F)=O)CCCN(C(c2cccc(F)c2N)=O)C1C c1(C(N(C2CCN(C(c3ccnnc3)=O)C2)CC)=O)ccnc2cc(Cl)ccc12 c1(N(n2ccnn2)C(CN2CC(O)(c3nccs3)C2)=O)cccc(Cl)c1 c1(CC(=O)NCC2CC(CNC(=O)CCc3cc(Cl)cs3)C2)ccc(F)cc1.C N1(C(C(N)Cc2csc3ccccc23)=O)CC2(CCC2)CCC1CO C(=O)(C(C)(C)C(O)C(C)C)NC1C(O)C=C(C(=O)NC(C2CCCC2)CC)C1 C(=O)(C(C)=Cn1ccnn1)NC1CC(F)(CNC(C=CCCC)=O)C1 N#Cc1ccc(C2CCN(CC3(C(F)(F)F)CC3)C2)s1.c1(S)ccc(N)cc1 c1(C(N(C2CCN(C(c3cc(C(N)=O)cs3)=O)C2)C)=O)c[nH]c2ncnc(O)c12 C1(CNC(C(C=C)(C)O)=O)CC(C)(C)CN1C(=O)C(c1ccc(Cl)cc1)C c1(C(=O)NC2C(NC(C3CC(=C)C3)=O)CS(=O)(=O)C2)cccc2c1oc(=O)n2C C1(NC(c2c(C)noc2)=O)CCCCN(C(C2CCC2)=O)C1 N1(C(c2nnc(C)s2)=O)CCOC(CNC(c2c(C)nsc2Br)=O)C1 Cc1sc(C(=O)NC2(C)CC(NC(c3ccnc(C)c3N)=O)C2)c(C)c1Br c1(CNC(C(CNC(C2(Cl)C(C(C)=O)C2)=O)O)=O)ccc(C)c(O)c1 n1(CC)cccc1C(=O)NCC1CC(F)(CNC(=O)C=CC(c2cnn(C)c2)=O)C1 CC(C)CC(O)C(C)C(=O)NCc1cc[nH]c1C(N1CC(O)CC1(C)CO)=O N1(C(c2nc(OCC)sn2)=O)CCC2CCN(C(c3cc(CC)no3)=O)CC12 c1(C(=O)NCC(C(=O)OC)N(C)C)cc(Cl)c(C)cn1.C12(CCCSC1)C(=O)O2 CC1OC2(C)CC1(C(=O)NC13CCC1CN(C(c1ccc(N)c(Cl)c1)=O)C3)C2 c1(SCC)cccc(CNC(=O)C(n2cc(C(N3CCNC3=O)C)nn2)C)c1 N1(c2nnc(C3(OCC)CCC3)n2CC)CCC2C(C1)C2(F)F C(=O)(C1=NN(C(C)C)C(=O)CC1)NCC1N(C(c2occ(C)c2)=O)CC2(CC2)C1 C1(NC(c2c(CC)non2)=O)CC(NC(C23CCC(OC)C2C3)=O)C(O)C1 C1(C(N2CC(OCCNC(C(C(C)O)C)=O)C2)=O)CCC2(CCCC2)C1 C1(C(N2C(C(=O)Nc3c(C)nsc3)CCC2)=O)OCCCC1(C)C N1(C(CCSCC(N)=O)=O)CCCN(C(c2cnc3nccn3c2)=O)CCC1 c1(OCC(=O)NCc2cn(C(CCCC)CC)nn2)ccc(F)cc1N c1(C(=O)NCCOC2CCN(C(c3c(CC)nc[nH]3)=O)C2)ccc(C)nc1O C1(CC)C(C(=O)NC(c2ncccn2)CC)CCCN1C(c1c[nH]c(=O)cn1)=O CC1=C(C(=O)N(CCCCCCNC(C2CC(n3ccnn3)C2)=O)C)COCC1 N1(C(C2C(C)(C)N(C(=O)C(F)CC3CCOC3)CC2)=O)CCc2cccc(O)c21 O=S(=O)(c1cccc(N2CCC(CO)CC2)n1)NCC1(F)CCC1 C1(O)(C(C)NC(C=CCCC)=O)CCN(C(=O)CC2CCC(C)CO2)CC1 Cc1cc(C(=O)NC(C(N2CC3(CCCO3)C2)=O)C2CCCC2)ncc1N C1(OC)(OC)CCCN(N2CC3CC2CC3CO)C1 c1(C(=O)NC2CN(C(C3N(C)CC(O)CC3)=O)CC23CC3)ccnc2c1CCO2 C(=O)(C(C)CC(C)C)N(CC(C)NC(C1CC(OC)C1)=O)CC C1(C)(C)C=CC(=O)N1.C1(CCC)CC1(C(=O)NC(c1ccco1)C)C(=O)OCC C(=O)(C1CC(C)(C)Oc2ccccc21)NC1CN(C(C(COC)N(C)C)=O)C1 c1(C(=O)NC23CCN(C(c4c(C)nc[nH]4)=O)CC2C3)cc2c(o1)CCCNC2=O c1(CC(=O)NCC2CCCN2C(=O)CCN2CCOC2=O)ccc(CO)cc1 C1(C(=O)NC(C)CSC(F)F)CCCCCC1NC(c1cc(O)nc(O)n1)=O C(=O)(CCCC(F)(F)CO)N(C1CCCN(C(=O)CC2CCC(C)CO2)C1)CC c1(C(C)OC)nc(C)c(C(N2CC(NC(c3cnc(CC4CC4)s3)=O)C2)=O)s1 c1(NC(C2CCC(NC(=O)CCC3CC3)CO2)=O)cc(F)c([N+](=O)[O-])cc1F c1(SCC)ccccc1C(=O)NCCN(C(=O)CC1CC1)CC1CC1 c1(C(N2CCC(NC(C(c3ccc(Cl)cc3)C)=O)CC2)=O)c(Cl)nn(C)c1Cl C1(NC(C2N(CC#C)CCC2)=O)CC2CC(C1)N(Cc1csc(C3CC3)n1)C2 c1(C(N2C(CNC(=O)COC(F)(F)F)CCCC2)=O)c(F)ccc2n[nH]cc12 N1(C(c2scc(C#N)c2)=O)CC(F)(F)CC1CNC(=O)CC1COCCO1 c1(CC)c[nH]c(C(=O)NC(C)C(c2ccccc2)NC(=O)C=CC(=O)N(C)C)c1 N1(C(CC(C=C)C)=O)CCC2(CC2NC(c2cnn(C3CCC3)c2)=O)C1 c1(OC)ccccc1C(CNC(C1(CCO)CC1)=O)NC(c1nc(C)sc1C)=O c1(OC)cc(C(O)CNC(=O)Nc2ccc(C(N)=O)nc2SC(C)C)ccc1C c1(C(N)=O)ccc(Cl)c(NC(=O)NC2CCCC2CC2(O)CCCOC2)c1 C(CC(C)(C)C(=O)N1CCC(N(C)C)C(C)C1)NC(C1C(C)CC=CC1)=O N1(C(=O)OC(C)(C)C)CCCC(Cc2nn[nH]n2)C1.N12CC3CC1(C3)C2=O Cc1cc(S(=O)(=O)N2CC(C)(C)OC(C)(C)C2)ccc1-c1cccnc1 C#Cc1ccc(C(=O)NCC2CCN2C(=O)C(C)N(C)C(C)=O)cc1 N1(C(C=NOC)=O)CCC2(CCN(C(c3cnc4c(Cl)cccn34)=O)CC2)C1 c1(C(N(C2CC(NC(C3C(=C)CC3)=O)C2)C)=O)cc(Cl)cs1 CS(C)(=O)=NC(=O)CNC(=O)NCc1ccc(Cl)cc1Cl N1(CCNC(C2CC(CNC(C3C(=C)C3)=O)OC2)=O)CCCC(O)C1 c1cc2n[nH]cc2cc1-c1nnc(CCC2CCCCC2)o1 c1(C(=O)NCc2nc(-c3cccc4c3COC4=O)cs2)ccc2c(c1)C(=O)NCC2 C1(C2CN(C(C3CC3Cl)=O)C2)(NC(C2CCCCC2)=O)CC1 C1(C(C)NC(c2cnc(CC)s2)=O)CCN(C(=O)COCc2cccnc2)CC1 CCCC(C(=O)NC1C2CN(CC(CC)OC)CC12)S(N)(=O)=O c1(CN)cccc2c1CCN2C(c1cnnn1-c1cc(Cl)ccc1Cl)=O c1(C(=O)NC(C2CCN(C(CC3(CC)CCOCC3)=O)C2)C)cccc(F)c1N c1(CCC(=O)N(CCOCCNC(C2C(CCC)C2)=O)C)cc(C(C)=O)c(C)o1 c1(C(N2C(CNC(C(CCCOC)C)=O)CC(F)C2)=O)cc(C)c(O)c(C)c1 C(CCC)(CCCNC(=O)C(F)=CCCF)NC(C(C)SCC)=O N1(C(CCCN(C(C)C)C)=O)CCN(C)CC1C(=O)NC1CN(C(N)=O)C1 N1(C(CC(CCSC)O)=O)CC(NC(=O)C=CCN2CCCC2)CC12CCC2 c1(C(=O)NC(c2cnn(C)c2)C(=O)NC(c2cncnc2)C)cnn(C)c1N c1(C(N2CC(O)CC(NC(C3CC4(CCC4)C3)=O)C2)=O)c(Cl)ccc2ccoc12 C=CCCC(C)(C)C(=O)NC(C)CC(C)NC(c1cc[nH]c1C(=O)OC)=O N1(C(Cc2ccc(C(C)C)cc2)=O)Cc2[nH][nH]c(=NC(=O)c3cnco3)c2C1 c1(C(=O)NC2(CNC(COCCOC)=O)CC2)cccc(SC(C)C)c1 N1(C(=O)CCNc2ccccn2)CC2CCCN(C(c3cnc(CO)s3)=O)C2C1 Cc1cc(Cl)c(C(=O)NC2CN(C(=O)C(C)n3ccnn3)CC2O)cc1C C1(C(C2CCCC2)C)CCCN(CC(=O)N(CCOCC(F)(F)F)C2CC2)C1 Cc1cc(CC2CCN2C(=O)NC(C2CCCC2)C)n(C)n1 CC1NC(=O)CCC1CNC(C1CCN(C(C2CCCCC2)=O)CC1)=O CC1OCCC1C(N1CCC(CC(=O)NCC2CC(F)(F)C2)C1)=O c1(C(=O)NC(CSCC)C(=O)N(C)CC2CCCCC2)nc(C)ccc1C C#CCCCCS(C)(=O)=NC(=O)c1ccc(C)c(C(=O)O)c1 CC1CC(NC(=O)C=CC2CCCN2C(=O)CSC(F)(F)F)CCC1(C)C C1(C(=O)NC2CON(CC)C2=O)CN(C(=O)CC(C)N(C)C)CCC1(C)C C1(NC(C2C(NC(C(CCC)OCC)=O)CCOC2)=O)CCC(N=[N+]=[N-])CC1 c1(CC)ccccc1-n1nc(Cc2ccccn2)nc1C(C)OCC(F)(F)F Cc1ccc(-c2nc(C)c(C(=O)NCC3OCCC3C(=O)O)s2)cc1.C(C)(C)(C)O c1(-c2cc(C(=O)NC3C(NC(C(CSC)O)=O)C3)on2)ccc(Cl)cc1 N1(C(c2n(C)ccn2)=O)CCC2C(CCN2C(=O)Cn2cnc3ccccc23)C1 S(=O)(=O)(c1c(F)ccc(C)c1F)Nc1sc(CC)c(-c2ccccc2)n1 CC(CCCN=c1[nH]c(=NC(CF)CF)c2c(F)cccc2[nH]1)c1ccccc1 C1(CN(C=O)Cc2cccc(OC(F)(F)F)c2)CC2OCCC2O1 c1(N(C)C)cc(NC2CC3C4C=CC4(C2)C3)c(Br)cn1 c1(C(N(C2CCN(C(c3nc(CCC)oc3)=O)C2)OCC)=O)nnn2c1CCC2 N1(C(c2c(F)ccc(OC)c2)=O)CCCCC(NC(=O)CC(C)SC)CC1 c1(CNc2cc(N3CCCC(CS(C)(=O)=O)C3)ncn2)nnn2c1CCC2 N1(C(Cc2c(C)n[nH]c2C)=O)CC23CCCC2(C1)CN(C(=O)CSC(F)(F)F)C3 C(=O)(CC(C)(C)C(F)F)N1CC(C)C(CNC(=O)CSc2nncs2)CC1 C1(CNC(C2(C)CCC(C)C2)=O)CCC(C(=O)NCCN2CCC(OC)C2)CC1 Cc1cccc2nc(CCC(=O)NC3(C)CCN(C(=O)CCCC4CC4)C3)[nH]c12 Cc1nn(C)c2ccc(C(=O)NC3CCCC3NC(C3CC34CC4)=O)cc12 C1(COC)(CNC(c2n[nH]c(C)c2C)=O)CCCN1C(c1[nH]cnc1C)=O Cc1cc2[nH]c(C(=O)NC3C4CC3CN(C(c3ccc(F)cc3Cl)=O)C4)cc2o1 C=CC1OCCCC1C(=O)NCC1CCN(C(=O)C=C(C)Cl)C(C)C1 CCC(CCC(=O)NC(C(=O)Nc1cccc(OCF)c1)C1(O)CCC1)OC c1(SC)nc(N2CCC(NC(C3CCN(C)CC3)=O)C(C)C2)cc(Cl)n1 c1(CN(CC(=O)NC(C)CCc2ccncc2)C)ccc(N(C)C)cc1 C(CC(=O)NC1CC1c1cncs1)(CC(C)C)NC(c1c(C)nncc1)=O C(c1ccc(OC)cn1)=CC(=O)NC1C2CN(C(COCCC=C)=O)CC21 c1(OC)ccc(N(Cc2ccc(Cl)cc2)Cc2c(C)ccn2C)cc1 C=CCC(C)C(=O)N1CCC(C(CO)NC(C2CC(C(F)(F)F)C2)=O)CC1 c1(C(=O)NCC2N(C(C(N3CCCCCC3)C)=O)CCC2)cncc(N)n1 CC(C)(C(=O)N1CC2(CCN(C(c3coc(CS(C)(=O)=O)n3)=O)C2)C1)S(C)(=O)=O c1(C(=O)NC2C(NC(C(C)OCC(F)(F)F)=O)C2)ncc(F)cc1N c1(CC(=O)N(C2C(N(C(=O)C(O)C(F)F)C)CCCC2)C)ccn2cncc2c1 C1(CNC(c2cnc(CC)s2)=O)CCN(C(C2CC2c2sccc2C)=O)CC1C C=C1CC2(C1)C(=O)NC2.C(=O)(C(C)CN(C)C)NCC1CC(n2cncn2)C1 Cc1csc(C(N2CCC(CC3CC3)C2)C(=O)NC(c2ccccc2)C2CCC2)n1 c1(C(C(=O)NC2C(NC(C(CSC)(C)C)=O)C2)C)ccc(F)c(Cl)c1 Cc1nc(C)n(CCCC(=O)NCCC(C)NC(=O)C=CC(=O)N(C)C)n1 c1(C(=O)NC(C(=O)NC2(CCOC)CC2)CCF)cc(C)nc(C)c1 BrC1=CC=CCC2C3(CCOC1CNCCC2)CC3 C1(CNC(CCC#C)=O)COCC2(CCN(C(C3(C)CCN(C)CC3)=O)CC2)O1 c1(NCc2c(C)ncs2)[nH]c(=NCC2CCCC3(CC3)C2)nc2c1ncn2CC CC(C)(O)C(C)(O)CNC1CC(c2ccccc2)CN1 CC(F)(F)C(C)(C)CC(=O)N1CCC2CC1CN(C(c1ccc(Cl)c(F)c1)=O)C2 N1(C(CN(C)S(N)(=O)=O)=O)CCOC2(CCN(C(C3CCC(CO)CC3)=O)C2)C1 Cc1c(C(N2CCC(CCCNC(=O)C(CO)NC(N)=O)CC2)=O)ncn1C C1(CC)CN(C(c2ccc(OC)nc2Cl)=O)CCN1c1ncccn1 CC1CCCCC1Cn1cc(C2(C(=O)OC(C)(C)C)CCN(C(=O)OC)C2)nn1 c1(C(=O)NCC23C(CN(C(C(N)=O)=O)C2)C3)cc(C(F)F)ccc1[N+](=O)[O-] c1(C(C(=O)NCC(=C)C)N(C(C)C)C2CC2)cncn1C C(=O)(C1CCCc2ccccc21)N(c1cc(C2CC2)ncn1)C.C12CCCN1C2 CC(C)(CNC(C1CCCO1)=O)CCNC(c1ncoc1C1CC1)=O C#CCC(C(=O)NC(CCF)C(=O)NC(c1ncc(C)cn1)C)C1CC1 c1(C(=O)NC(CC)(C)CNC(C2CC2C(C)(F)F)=O)cncc(C#N)c1 C12(NC(Cc3c(C)cccc3Cl)=O)CCCN(C(C3CCCC3)=O)CC1C2 C(=O)(C#CC(C)(C)O)N(C)CC1CCCCN1C(c1cn(C(C)(C)C)nn1)=O c1(CC)ncc(C(=O)N(C2CCC(NC(c3nc(O)sc3C)=O)CC2)C)c(O)n1 C(N=c1[nH]cnc(Cl)c1OC)C1(C)CCC(NC(CC(COC)C)=O)CC1 CC1(CNCc2cn(CC(N3CCCC3CC(N)=O)=O)nn2)CC2CCC1C2 C12(C)CCN(C1)C2=O.C1(C(=O)NC2CCC(N(C)C)C2)(NC(=O)NC)CCCC1 c1(C(N2CC(C(C)NC(C(C)OCC)=O)C2)=O)cc(C#N)c(F)cc1F C1(NC(C=CSC)=O)(CNC(=O)CCC2CCCC(O)C2)CCCCC1 C12CCCCC1N2.C(N=C(NS(C)(=O)=O)NC1CCOCC1)C1C(C)(C)C1 C1(C)(OC)CCCN(C(=O)CONC(C2CC(=O)OC2(C)C)=O)CC1 N1C(=NCCc2ccsc2)NCC1.Cn1nc(C(F)F)nc1C(F)(F)F C(=O)(CC(C)C(F)(F)F)N1CCC(OCCNC(C2(COC)C=CCC2)=O)C1 CCCC(O)C(CO)NC(=O)C(CC1CC1)NC(C1CC(CC2CC2)C1)=O N1(C(Cc2nn(C)c(Cl)c2)=O)CC(NC(=O)CCS(C)=O)C2CCCCC12 N1(C(c2c(CC)n(C)cc2)=O)CC2CCCC1CN(C(=O)Cn1cnnn1)C2 C1(C(=O)NCCN(C(=O)CSC(F)(F)F)C)CCC(O)CN1C N1(C(c2ccn(C)c2CC(=O)O)=O)CCn2cc(C(=O)Nc3cn[nH]c3)nc2C1 N1(C(C2(CCC)CCCC2)=O)CC2(C)CN(C(C3(NC(N)=O)CC3)=O)CC2(C)C1 N1(C(CC=C=C)=O)CCC2(C1)CN(C(c1cn3cccc(C)c3n1)=O)CC(C)O2 N1(C(CC(C)C2CC2)=O)CCC(CNC(c2ccn3ncnc3c2)=O)C12CCC2 N1(C(c2cc(Cl)ns2)=O)CCC2(C1)CN(C(C1CCC1c1nc[nH]n1)=O)C2 C1(NC(=O)CCc2cc(Cl)cs2)CC2CCC1(NC(=O)C(C1(O)CCCC1)F)C2 N1(C(C(=O)NCC#C)C)CCC(NC(=O)COC(c2cn(CC=C)nc2)=O)CC1 C1(CNC(c2nccc(C)n2)=O)COCCN(C(=O)C(C)C2(O)CCC2)C1 c1(CC(=O)NC2CC3CC2N(C(c2ccco2)=O)C3)ccc(Br)cc1F Cc1ccc(CC(=O)N(C)CC2C3CN(C(=O)C(C)(C)CO)CC23)cc1Br CCC(CCC(=O)N1CC(Cn2cc(C(C3CCOCC3)C)nn2)C1)OC c1(-c2onc(-c3cc(Br)sc3)n2)cc(OC2CCCC2)ccn1 C(CCN=C(NCCN1CCCC1)NCC1CCC(C)O1)SC N1(C(c2ccc(OCC)nc2O)=O)CCC(=C(F)F)CC1 N1(C(CCC=CC)=O)CC(NC(C2(OC)CCSCC2)=O)CC1C N(C1CCCn2cnnc21)C(C1CC(F)CCN1C(c1cc(F)cc(F)c1)=O)=O N1(c2nc(C)nc(Cl)c2)CC(NC(=O)C2=C(Cl)CC2)C2CCCCC12 C1(C#C)(C(=O)NCCCC#C)CCN(C(=O)C(C)C(C)C)C1 C1(NC(c2c(C)nco2)=O)CCCN(C(C2CCCC2c2nnc(S)n2C)=O)C1 N1(C(CCC(C)(C)NC(C(n2ccc(C)n2)C)=O)=O)Cc2cccc(F)c2C1 c1(N(C(C2C(NC(CCOC)=O)CCC2)=O)C)cc(C)cc(F)c1 C#Cc1ccc(C(=O)NC2(CCOC)CCN(C(c3conc3CC)=O)C2)cn1 c1(CC(=O)NC2(CCN3CCC(c4ncc[nH]4)CC3)CCC2)ccc(CO)cc1 CC1CN(C(=O)CCOCC2CC2)CCC1NC(C1(C)CCSCC1)=O C1(C(=O)NCC(CC=C)CC=C)CN(C(c2cc(C)nc(O)n2)=O)CCC1(C)C N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)C(c2ccc(Cl)cc2Cl)O)CC1C(F)F N1(C(=O)CCc2ccoc2)CCC2C1CCN2C(C1Cc2ccccc2O1)=O C1(C(=O)NCC(C)N(c2ncc(C)c(O)n2)C)CC2(C1)NC(=O)NC2=O N1(C(CC(C(=O)OC)(C)C)=O)CCC2(CCC(NC(C3CC4(CCC4)C3)=O)C2)C1 N1(C(CCN(CC#C)C(c2ccn(COC)n2)=O)=O)CCCC2(CC2)C1 N(C)(S(=O)(=O)N(C)C)CC(=O)NC1(CO)CN(C(C=Cc2nc(C)sc2)=O)C1 C1(N(C(C(C(C)C)SC)=O)C)CCCCN(C(c2ccc(C)nc2O)=O)C1 C1(C(=O)OCC2CC3CCC23)CCN2CCOCC12 c1(C(=O)NCC(=C)CCNC(=O)CCc2ccccn2)ccc(Cl)c(F)c1 C12(CNC(C(=Cc3cn(C)nc3)F)=O)CCC1CN(C(C1(C)CNC(=O)N1)=O)C2 c1(NC=O)ccc(C(=O)NC2CN(C(c3cc[nH]n3)=O)CC2F)cc1 N(C1c2ccccc2CC1NC(c1ccoc1Cl)=O)C(c1cncn(C)c1=O)=O N1(C(CC2(OCC)CC2)=O)CC(O)CCC1C(=O)NC(c1nncn1C)CO c1(C(=O)NC(CN(C(C(C2CC2)OCC)=O)CC)C)cc(I)c[nH]1 C(N=C(NCCC1(O)CCOC1)NC1CCCCC1)c1ccc(C(N(C)C)=O)s1 N1(C(c2n(CCOC)ncc2)=O)CCC(C)(NC(c2cc(Br)ccc2F)=O)CC1 CS(=O)(=O)c1nccc(Nc2cnc(F)cc2C(N2CCC(C#N)CC2)=O)n1 N(C1CCCc2cc(Nc3ccnc(C#N)n3)ccc21)C(=O)OC(C)(C)C C12(NC(CC3CC(SC)C3)=O)CCCCCC1N(C(=O)C=Cc1ccn(C)c1)CC2 CCCC(CCO)NC(=O)CCN(C(c1nonc1C)=O)C(C)C c1(C(=O)NC2CN(C(CCCCC)=O)C(C)(C)C2)cnc2n1CCOC2 N1(C(CSC)=O)CCC2(CCOC2)C(CNC(c2n[nH]c3cc(C)ccc23)=O)C1 c1(C(=O)NCC2(NC(CN3C(C)CC3)=O)CCOC2)ccc(Cl)cc1Br CC1(CNc2cc(CC#N)ncn2)CCN(C(=O)CCC2CC2)CC1 n1(CC)nc(C(C)C)cc1C(N1CCN(C(=O)N(C)C)CC1)=O.C1(=O)CC(C)O1 CC(CC(=O)N1CC(NC(=O)CCc2ccc(Cl)cc2)CC2(CC2)C1)C(F)(F)F N1(C(c2c(CC)[nH]cc2)=O)CCCCCC1C(=O)NCc1ncnn1CCOC C(C)(C)(C(C)CC(=O)NCc1noc(C)n1)NC(CC(CC)SC)=O C1(C(N2CC(CNC(C(C)OCC3CCCCO3)=O)C2)=O)CCC(C)(C)CC1 CCCCC(CCCC)NC(C1C(C)OCCN1C(c1ccnn1COC)=O)=O N1(C(Cc2c(C)n[nH]c2)=O)CC2(C(=O)NC(C)(C)C(O)CO)CC1CO2 C1(C(N(CCNC(C2(NC(=O)OC)CCCC2)=O)C)=O)CCCC(C)(C)CC1 N1(C(C2=C(C)CC2)=O)CC(O)C(O)C1CNC(=O)C(C)OC1CCCC1 c1(C(N2CC(O)(Cc3cn(CC(=O)OCC)nn3)C2)=O)cc2c(Cl)cccc2[nH]1 c1(-c2ccc(CNCC34COCC(C)(C3)CO4)s2)ccc2c(c1)OCCO2 C1(NC(C2N(C(c3c(C)cco3)=O)CCSC2)=O)CN2CCC1CC2 N1(Cc2cn(CC(=O)OC(C)(C)C)nn2)CC2C(C(=O)SC3CCNC3=O)C2C1 c1(CC(N2CC3C(CNC(C(C=CC)O)=O)(C3)C2)=O)c(C)[nH]c2ccnn2c1=O CCC(CC)CC(=O)N1CCCCC1CN(C)C(c1cnc(S)[nH]1)=O CC1CN(C(c2nn[nH]c2Cl)=O)C(C)CN1C(C1CC2CCC1CC2)=O C1(NC(C(=Cc2cnc[nH]2)C)=O)CCC(F)(CNC(=O)Cn2cnc(C#N)n2)C1 CON1CC(C(N2CCCC2C2(O)CN(CC3CC4(CCO3)CC4)C2)=O)CC1=O c1(C(C(=O)NCCC2(C)CC2)N(C2C(C)CCC2)C)cccc2c1OCC(=O)N2 c1(C(N2CC(NC(C)=O)(CO)C2)=O)sc(C(C)=O)cc1Br S(=O)(=O)(CCC(F)(F)F)NC1CC2(CN(C(C3C4COCC34)=O)C2)C1 N1(C(C(CCC)c2ccc(Cl)cc2)=O)CC2(CNC(=O)C=C(C)C)CC1CCO2 c1(CCNC(=O)C(=O)NC2CCCC2)ccc(F)cc1Cl N1(C(C(C)OC)=O)CCCCC1C1CCN(C(C2CN(C)C2)=O)CC1 C12(CCCSC1)NC2.S(=O)(=O)(CCN(C)C)N(CC)CC C1(C(=O)NCCOC(=O)OCC)CN(C(=O)C(C)(C)OC(F)F)CCC12CCC2 CC(F)CC(=O)N(CC(Cc1ccccc1)NC(=O)Cc1csc(Cl)n1)C CCCC(C)C(=O)NCCN(CCC1CCCCCC1)C1CC1 CCC(CC(=O)N(C)CC1(NC(=O)C(C(C)C)n2ccc(C)c2)CC1)C1CC1 C1(N(CC(C)C)C(=O)CSCCN(C)C)CCN(C(C2CCCCO2)=O)CC1 c1(OC)ncc(C(=O)NC(C)CCCNC(c2coc(C(C)=O)c2)=O)c(C)n1 c1(C(=O)NCC2(NC(CC3CCCN(C)C3)=O)CCOC2)cc(F)c(Cl)cc1Cl c1(OC)cc(C(=O)NCC2(O)CCN(C(=O)C(F)C3CC3)C2)nc(Br)c1 N1(C(C2N(C(c3ccn(C)c3)=O)CC(O)CC2)=O)CC2(CCCCC2)C1 N1(C(C)=O)CC(O)CC1C(=O)NC(C)CC1CN(C(=O)CCCc2nc(C)cs2)C1 N1(C(C(CC#C)NC(c2ccc(CF)cc2)=O)=O)CCN(CC)C(C)C1 CCC(C)C(=O)NCC(C(C)C)NC(C1(C(=O)OCC)CC=CC1)=O N1(C(COCC)=O)CCC2C(CCN2Cc2ccc(C)nc2Br)C1 S(=O)(=O)(c1ccc(NCc2c(CC)noc2)cc1Br)N(C)CC1(C)CC1 C1(C(N2CCC(C(C(=O)NC(CC#C)C)(C)C)C2)=O)CC(=O)OC1(C)C C1(C(N(CC)CC)=O)CCc2nc(-c3cccc(C)c3OC)sc2C1 N1(C(C2N(C(C3N(C)C(=O)CC3)=O)CC=C2)=O)CC(F)(F)C(F)(F)C1 C1(C(N(C2CCCN(C(C3CC(=C)C3)=O)C2)CCO)=O)CCc2ccccc2C1 c1(NC2C(SCC)CCC2)cc(N2CCCC(F)(CO)C2)nc(C)n1 CC1CCCn2c(C(=O)NCC3CC(NC(=O)CCn4ccnc4)C3)cnc21 C12CCN(C(C(=O)NC(CO)C3CC3)C1)C2=O.C1(CC)C=CCC1 C(=O)(CC(CC1CC1)NC(=O)CC(Cl)Cl)NC(C#C)(C)C1CCC1 Cc1nn(C)c(C(=O)NC23CC2CN(C(=O)CSc2ccccc2)C3)c1[N+](=O)[O-] c1(C(N2CCC(N(C(C3CC(Cl)(Cl)C3)=O)CC)C2)=O)ccc2ccsc2c1 c1(CC(=O)NC2C(CNC(C(c3n(C)ccc3)=O)=O)C2)ccc([N+](=O)[O-])cc1Cl N1(C(C2(C(=O)Nc3cccc(SCC)c3)CC2)=O)CCS(=O)(=O)CC1.C1(=O)CN1 N#Cc1c[nH]c2c(F)ccc(F)c2c1=NCC(O)CNC(=O)Cc1cscn1 c1(OC)c(C(=O)N(C)CC2CCCN2C(C2CC23CCOCC3)=O)cccc1Cl C1(NC(c2cn(CCC)nc2)=O)CC2CCC1N(C(=O)Cc1ccncc1Cl)C2 n1(C2CC2)ncc2c1Sc1nc-2on1.c1(SCCOCCOC)ccccc1 N1(C(C2CN(C)C(=O)CC2)=O)C2CCC1CN(C(=O)Cc1cnns1)C2 c1(C(N2CC(n3cc(CCCCC)nn3)C2)=O)cccc2nnn(C)c12 c1(C(N2CCC(NC(c3n[nH]cc3[N+](=O)[O-])=O)CC2)=O)cc2ccccc2cn1 C(=O)(C(C)C(O)C(C)C)N1C(CNC(c2ncc(OC)cn2)=O)CCC1 C1(C(C(=O)NC2(C(N(CCCC)CCCO)=O)CCC2)F)CCOCC1 Cc1cnc(Cl)c(C(N2CCCC(NC(=O)CC3CC3(Cl)Cl)C2C)=O)c1 C1(NC(C2CC(OC)C2)=O)CC(C)(NC(=O)C=CC2CCC2)C1 c1(NC)cncc(C(=O)NC2CC(N(C)C(c3ccc(C(N)=O)nc3)=O)C2)c1 Cc1ccc(C(=O)NC(CNC(=O)C(C)Oc2ccc(F)cc2)C(C)C)nc1 C1(CNC(C(C)(C)OCC)=O)CC(OC(C)C)C1(C)C.C1(=O)CCOCCCN1 N1(C(c2cnc(OC)nc2C)=O)CC(C)CN(C(c2csnn2)=O)CC1C C1(CNC(COCCN(C)C)=O)(CO)CCCN(C(C2CCCO2)=O)C1 C1(C(=O)NCCC2N(C(c3cnc(C)nc3)=O)CCCC2)CCC=CCCC1 c1(N(C)CC2CCCC2)nc2c(c(=NC3CCN(C)C(=O)C3)[nH]1)SCC2 CC1CCC1CC(=O)N(CCC(=O)N1CC(n2cnnc2)C1)C1CC1 CCCCCC(C)(C)C(=O)NCC(C)(O)CNC(c1c(C)[nH]c2ncccc12)=O c1(N2CCN(C(COC)=O)CC2)[nH]c(=NCc2cnc(C)cn2)nc2sccc12 C1(CC(N2CCC(N(C(CCOCCOCC)=O)CCO)C2)=O)CCS(=O)(=O)C1 C1(N(C(C2CCC(C)(CC)O2)=O)C)CCC2CN(C(c3ccc(F)s3)=O)CC12 C1(CC(=O)N(C)CC2(CNC(c3ccccn3)=O)CC2)CCCCCCC1 N#Cc1cc(C(F)(F)F)cc(N2CCN(c3ncc(C4CC4)s3)CC2)n1 Cc1cc(NCC2(CO)CC3CCC2C3)ncc1S(=O)(=O)NC1C=CCC1 CC1=NNC(=O)C1CC(N1CCC(CCC(=O)N(C(CF)CF)C)CC1)=O CCCCCC(CC)C(=O)N1CC(NC(c2ncsc2CC)=O)CC12CCCC2 c1(-c2onc(-c3c(CSC)cccc3)n2)ccc(S2(=O)=NCCC2)cc1 CC(C)(O)C#CC(=O)N1CCC(C(N2CC(C3CCCCC3)C2)=O)O1 CS(=O)C=CC(=O)N(CCNC(C1CSCCS1)=O)Cc1cccc(Cl)c1 Cc1cc(C(N2CCC(N(C(=O)COC(F)(F)F)C3CC3)CC2)=O)c(C)n1C N1(C(Cn2c(C)ncc2)=O)CCC2C1CCCN2S(=O)(=O)CCC(F)(F)F N1(C(CC=CCCCCC)=O)CCC(C2(NC(c3cc(COC)on3)=O)CC2)C1 C1(CCOC)(NC(=O)C(F)C(F)(F)F)CCN(C(c2coc(N(C)C)n2)=O)CC1 c1(Nc2ccc(NC(C3N(C)C(=O)OC3)=O)cc2)ncc2ccsc2n1 c1(-c2cccc(CC(=O)N(C(C)C)C(C)C)n2)cccc2c([N+](=O)[O-])cccc12 c1(OC)ncnc(OC)c1CNc1cnc(F)cc1C(=O)Nc1c[nH]nc1C#N N1(C(CCC=C)=O)CC(NC(=O)Cc2c(CC)noc2CC)C(F)(F)C1 c1(C(=O)NCC2C(NC(c3cncn(C)c3=O)=O)C2)cn2cccc(F)c2n1 Cc1ccc(NC(C2CN(C(c3cc4sccc4s3)=O)CCC2O)=O)c(C)c1 C(C)(C1=CCN(C)CC1)NC(CN(C(=O)Cc1cn(C)cn1)C(C)C)=O C1(C(=O)NCc2cccc(OCC(C)C)c2)CC=C(C(F)(F)F)CC1 N1(C(C2C(C)=C2)=O)CCN(C2CCN(C(c3cnc(Cl)cc3Cl)=O)CC2)C(=O)C1 C1(O)(CNC(C(C)N(CC)CC)=O)CCCN(C(c2cc(CO)on2)=O)CC1 N1(C(C2N(C)C(=O)CC2)=O)CC(NC(c2nocc2C(C)(C)C)=O)CC1(C)C C=CC1(CO)CCN(C(=O)C(c2ccco2)NC(c2cn[nH]c2)=O)CC1 c1(NC2(CNC(c3ccc(O)nc3Cl)=O)COC2)ccc([N+](=O)[O-])c(O)n1 N1(C(Cc2cc(C)nn2C)=O)CCC2(CC2C(N2CCS(=O)(=O)CC2)=O)C1 CCCC(C(=O)NCC1CC(NC(=O)CC23CCC(CC2)C3)C1)NC(N)=O C(C(=O)N(O)Cc1cn(C(C)C(=O)N2CCCC2)nn1)NC(CC)=O c1(C(N(C2CN(C(C(C)SC)=O)CC2(C)C)C)=O)c(C)ccc2n[nH]cc12 CS(C)(=O)=NC(=O)C(=O)N1CC2(C1)CN(C(c1cc[nH]c1C1CC1)=O)C2 N1(CCOCC)CCN(C(c2ccn(C)c2)C(=O)NCC2CCCO2)CC1 CN1CCN(C(c2cc(=O)n(C)cn2)=O)CC1CNC(=O)Cn1cccnc1=O C1(NC(C2(CCC=C)CCCC2)=O)CN(C(C2C3CCC2CC3)=O)CCC1C N1(C(Cc2c(C)ncc(Cl)c2)=O)CCN(C(c2c[nH]c(C#N)c2)=O)C(C)C1C N1(C(=O)COCC2CCCC2)CCC2CN(C(c3ccc4[nH]ccc4n3)=O)C2C1 C1(CNC(C(C)C2CCOC2)=O)CC2(CCN(c3ncnc4[nH]cnc34)C2)CO1 CN1CC2(CCN(C(=O)C(CCF)NC(=O)C(O)CC(C)(C)C)CC2)C1 N1(C(c2cc(C(F)F)[nH]n2)=O)CCC(C(N2CCOCC2CCO)=O)(CO)C1 c1(C(=O)NC(C(=O)NC2CC(C(C)(C)C)C2)c2ccco2)ccc(C#N)[nH]1 c1(NC(=O)NC2CCCC(CCCC)C2)cc(C)ccc1OCCO N1(C(C(C)CC2CCC2)=O)CCN(C(c2cc(O)cnc2N)=O)C(C)C1 C1(C(C)NC(=O)COC2CN(C(=O)CC3(C)CC3)C2)CC(F)(F)C1 c1(NC(C2N(Cc3cccc(N(C)C)c3)CCC2O)=O)c(F)ccc(Br)c1F N1(C(c2c(C)oc(CO)c2)=O)CCOC2(CCN(C(=O)C#CC3CCOC3)C2)C1 C1(C(N2CCC(COC)CC2)=O)C2CCC1CN(C(C1(F)CCCC=C1F)=O)C2 N1(C(C=CC)=O)CCC2CC1CN(C(=O)Cc1ccc3ccncc3c1)C2 C1(NC(c2n(CC)ccc2)=O)C2CCN(C(C3SCCS3)=O)CCC12 C1(NC(C(CC(C)=O)C)=O)CN(C(c2cc(F)cc(Cl)c2C)=O)CC(F)(F)C1 C1(C(=O)NC2CC(N(C)C(c3cc(C(N)=O)[nH]n3)=O)C2)COCCN1C C(=O)(C(C)(C)CNC(C1CCC(C2CC2)N1C(=O)C(Cl)Cl)=O)OC CC(CF)CC(=O)NCC1(C(C)(C)C)CCNC1=O C(=O)(C1c2c[nH]nc2CN1C(=O)CC1CCC(O)C1)N(CC(C1CC1)OC)C c1(CNC(C(C)C2CCCO2)=O)nc2c(s1)CN(C(c1cnc(N)cn1)=O)CC2 c1(NC(N=c2scc(-c3c(OC)ccc(OC)c3)[nH]2)=O)nc2c(s1)CC(O)CC2 n1(CCOC)cc(C(=O)NCC(CC)(CC)NC(=O)C(F)OC)c(=O)cc1C c1(-n2c(C(c3c(OCC)nsc3)NCC=C(C)C)nnn2)ccc2c(c1)OCO2 C(C)(CCCC(=O)N1CCN(C)CC1)NC(C1(CC=C)CC1)=O N1(C(CCC(C)(F)F)=O)CC2(CNC(=O)C(CO)C(C)(C)C)CC1CCO2 C(=O)(C(F)C(C)(F)F)NC1CC(N(C(C=Cc2ccc(C)o2)=O)C)C1 Cn1ncc(S(N)(=O)=O)c1C(=O)NCC1(C)CCCN1C(c1cncnc1)=O Cc1cnnc(NC2CN(c3ncccn3)C2)c1 c1(OC)c(Cl)cc(C(=O)NC2CCCN(C(C3COCCO3)=O)C2)nc1Cl Cc1ncc(C(N2CCC(C)(NC(=O)COCC(C)C)C2)=O)cc1C#N C12(CCCCC1C)NC2.C(=O)(C(C)(C)C)NC(C)C(=O)Nc1nncs1 N1(C(C2(OC)CC2)=O)CCN(C(=O)CCCc2ccc(Cl)c(Cl)c2)C(C2CC2)C1 c1(OCC)ccc(C(=O)NCC2(Nc3ccnc(C)n3)CC2)c(F)c1F C(=O)(CC(F)(F)CC(=O)N1CC2CC(C1)CN(C(=O)CNC(C)=O)C2)OC C1(CNC(=O)C(c2ccccc2)O)CC2(CO1)CN(C(=O)Cc1cc[nH]c1)C2 C(c1ccccc1)=CC(N1CC2CC1C2C(=O)NCc1ncccn1)=O c1(C(N2CC3C(C(=O)Nc4cc(OC)c(Br)cc4)(C3)C2)=O)cc(F)cc(C)c1O C1CC(C)(C)C(=O)N2CCC(C2)O1.c1(C2C(CC(=O)OC)C2)ccccn1 Cc1c(C(=O)NCC2C(C)CCN2C(c2c[nH]c(C#N)c2)=O)ccc2cncn12 C(=O)(CC(C)(C)CC(F)F)N1CCC(C2(NC(CCC3N(C)CCC3)=O)CC2)C1 CC1(C)CCC(CNC(c2cncnc2C2CC2)=O)N(c2ncc(I)cn2)C1 c1(OC)ccccc1C(C)NCC1CN(c2ccc(C(F)(F)F)cc2)C1 c1(C(=O)NCC2C(NC(CCCC(N)=O)=O)CCC2)coc2c1C(O)CCC2 CCC(C)CCCCC(=O)NCC1CC1C(=O)NCCc1ccnc(O)c1 O=C1Nc2cc(C(N3CCOCC(CNC(C4C=CCC4)=O)C3)=O)ccc2C1=O N1(C(C2(CCCC)CCC2)=O)CCC2(CCC2CNC(=O)C(C)O)CC1 C(=O)(C(F)C(C)(C)O)N(CC(N1CCCC(OCC)C1)=O)C1CC1 Cc1csc(C(N2CC(CNC(=O)C=C3CCCCC3)C3CC23)=O)c1C C1(NC(C2(CC)CCCCC2)=O)CCCN(c2cc(C(=O)NC)ncn2)CC1 N1(C(C(COC)(C)OC)=O)CC2C=CC1C(C(N1CC(C(C)(C)O)C1)=O)C2 N1(C(CCC=C=C)=O)CCC(NC(=O)COc2cncc(Cl)n2)C(CO)CC1 C(=O)(C1=CCc2ccccc21)NC1CC2CN(C(=O)OC(C)(C)C)CC(C1)C2 c1(C(N(C(C)CCNC(C2(N(C)C)CCC2)=O)C2CC2)=O)cccc(=O)n1C c1(CN(C(=O)CNC(c2ccsc2CO)=O)C)cn(CCc2ccccc2)nn1 N1(C(C(C(C)O)C)=O)CCN(C(c2nccc3cc[nH]c23)=O)C2(CCC2)C1 N1(C(C2CC3C=CC2CC3)=O)CCCN(C(C2CCC23CCC3)=O)CC1 C1(NC(C(C)=C(CC)C)=O)CC2CC(C1)N(C(c1cc(O)ncc1F)=O)C2 Cc1cc(C(N2CC(N(C)C(C3CC4CCC3O4)=O)C(C)(C)C2)=O)cc(N)c1Cl C1(NC(C(CC=C)N(C)C)=O)CC2CC(C1)N(C(=O)Cn1ccc(C(F)F)n1)C2 Cc1ncc(C=CC(N2CCC(C)C2CNC(=O)Cn2cc(C3CC3)nn2)=O)s1 c1(C(CNC(c2c(CCC)n[nH]c2)=O)NC(=O)C(C)SC(C)C)cccc(C)c1 c1(CNC(C(C)CN(C(=O)CCN2CCCC2=O)C)=O)ccccc1C#N C(=O)(CC(O)(c1ccccc1)C1CC1)NCC(C(C)C)NC(=O)CNS(N)(=O)=O c1(OCCOC)ccc(NC(=O)C(=O)Nc2cnc(CCSC)nc2)cc1 CC1CN(CC(=O)NCC(C)(C)OCC(=O)N(C)CCF)C1 N1(C(c2ccc(CC)cc2F)=O)CCCC(C)(C)C1CNC(=O)CN1CCC1 N1(C(C=C(CCC)CCC)=O)CCOC2(CCN(c3ccc(C#N)nc3)C2)C1 C1(C(N2C(CNC(CCOC)=O)CC(F)(F)C2)=O)CC2CC1C1C2C1(F)F N1(C(Cc2nc(C)sc2)=O)CCN(C(c2coc3c2COC3)=O)C(CF)C1 c1(C(N(CCNC(C2CCN(CC)C2)=O)CC)=O)cc2n(c1)CCC2 C1(C(N(C2CCN(C(c3nc(CCC)sc3)=O)C2)CC)=O)CCC(=O)NC1 c1(CNC(C(C=C)(F)F)=O)ccc(CNC(C2(C)CCC2)=O)cc1F N1(C(C(C(C)C)O)=O)CC2CS(=O)(=O)CC2(NC(=O)C#CC(=O)O)C1 Cc1ccc(C(=O)NCC2(NC(c3ccnc(C(C)(F)F)c3)=O)CCCC2)nn1 C=CCC(CC=C)C(=O)NC(CC=C)C(=O)NCCC1CC=CC1 c1(C(N(CC(C)(C)NC(C2CC(C)(C)CCO2)=O)C)=O)n[nH]c2ccccc12 c1(C(c2ccns2)NC(=O)NC23CC(C(F)(F)F)(C2)C3)cccc(F)c1 c1(NCC(CC)(CC)C(N)=O)[nH]c(=NCC(C)(C)NS(C)(=O)=O)nc2sccc12 C1(CNC(C(C)CN(C(=O)CC2(O)CCCC2)C)=O)CC12CCOCC2 C#Cc1ccc(C(=O)NC(CC#CC)C(=O)N2CCCCC2CO)cc1C S(=O)(=O)(c1ccc(NC(=O)NC(C)C)cc1)N(CC(O)C(=O)OC1CCNC1)C C(C)(C(C)(C)C(=O)NCC(CC)OC)NC(C=C(CCC)C)=O N1(C(CNC(N)=O)=O)CCC(O)CC1C(=O)NCC(C1CCCC1)O C1(NC(C=CC(C)C)=O)CCCC(CC(=O)NCC2(F)CCOCC2)C1 S(=O)(=O)(c1ccc(C(=O)NCC2CC2NC(=O)C2=CCCS2)cc1)NC(C)(C)C C1(C)(C(=O)NCC(C(C)C)NC(c2ccccn2)=O)CC(C2CC2)=NO1 c1(-c2scc(C(=O)NC(c3ncc(F)cc3F)C)n2)c(Cl)cccc1Cl CC(F)(F)CC(=O)NCC1CCN1C(c1ccc(Nc2ccc(Cl)cc2)nc1)=O Cc1cc(C(=O)N(C)CCOCCNC(c2cn(C(C)C)nn2)=O)nnc1O Cc1c[nH]ccc1=NC(=O)c1cc(NC(C2CCC(F)(F)CC2)=O)cn1C C(CNC(=O)Cn1nnc(C2CC2)n1)(CC(F)(F)F)NC(Cc1c(C)n[nH]c1C)=O c1(C(=O)NC2C(C)CCN(C(c3cccn3C)=O)C2C)cccc2c1nnn2C c1(CC(=O)NCCCOCCNC(C(C)C2CCC2)=O)ccc(C(N)=O)cc1 C1(C)(C(N2CC(O)(CCNC(C3(OC)CCCOC3)=O)C2)=O)CCC(C)C1(C)C C(=O)(C1CCCn2cncc21)N(C)CCNC(c1cn(C)ccc1=O)=O c1(C(=O)NC2(C#N)CCN(Cc3cc(I)ccc3O)C2)cc2ccoc2cn1 CC(c1cnn(C)c1)=CC(=O)NCC1C2CN(C(=O)CC3CCC=CCC3)CC12 c1(-c2nc(NC(c3ccc4c(c3)OCO4)=O)sc2)cccc2ccnn12 c1(C(=O)NC(CNC(c2ccc(C#C)cn2)=O)CCOC)cnc2ncccn12 C1(CNC(c2c(CC)onc2)=O)CN(C(=O)C(C)CC(C)(F)F)C2CCCC2O1 C1(NC(C2CCC=CCCC2)=O)CCCN(C(c2ccc(C3CC3)cc2)=O)CC1 Cc1sc(C(=O)Nc2csc(-c3ccc(C(C)O)cc3)n2)cc1[N+](=O)[O-] CCC(CC(=O)NC1CC(NC(=O)CC2CCCN2CC)CC1O)C1CC1 N1(CCC#C)CCC(NC(=O)NCC(c2ccncc2C)C)CC1 c1(C(=O)NCC(C)(C2CCC2)NC(C2Cc3nccn3C2)=O)cc2n(n1)CCC2 c1(C(=O)NC2CC3CN(C(c4cn(CC=C)nn4)=O)CC32)cnn2ccn(C)c12 CC(C(=O)N1CCN(C(C2CCCCN2C)=O)CC1)S(C)(=O)=O N1(C(C2CCCN(C)C2)=O)CCC2C(CCCN2C(c2ocnc2C(F)F)=O)C1 c1(OC)ccc(C(CNC(C23CC(C2)C(C)O3)=O)NC(=O)CCC(C)C)cc1 C1(CN2CCCN(C(C)=O)CC2)Cc2ccc(C(=O)O)cc2O1 O=C1C2Cc3ccc(F)cc3N2C(=O)N1CC1(Br)CCOCC1 N1(C(CC2C(CC)C2)=O)CCOC2(CCC(NC(=O)C(C)(C)OC(C)C)CC2)C1 CC(=O)CCCC(C)C(=O)NC1CCCC(NC(C2CC(C)CCO2)=O)C1 C(C)(CCC(=O)NCC1(NC(c2cccnc2Cl)=O)CCC1)OC c1(C(N2C(CC)CC(C)(C)C2)C(=O)NCCCSC)cc(S(N)(=O)=O)cs1 C1(CC#C)(C(=O)NC(CCNC(C2CC2C(C)(F)F)=O)c2cccs2)CCCC1 C1(NC(CS(=O)(=O)NCC)=O)C2CCC1CN(C(C1CC13CC3(F)F)=O)C2 C12(NC(CNC=O)=O)CCC(C1)N(C(=O)CSc1nnnn1CC(F)(F)F)C2 C1(C(=O)NCC23CC2CN(C(=O)Cn2cnnn2)C3)CCn2cnnc2C1 c1(C(N(C(C)C(=O)NC(CO)CCF)CCC)=O)ccc(=O)n(C)c1 C1(N(C2(CNC3CCCS3)CCC2)C(c2ccncc2)=O)CCCCCC1 C(=O)(CCCCNC(=O)CCC1CC(F)(F)C1)N(C)Cc1cncn1C Cc1ccc(C(=O)Nc2cn[nH]c2)cc1Br.C12CCCN1C(=O)COC21CC1 c1(C(=O)NCC(C)N(C(CCN(C(CCC)C)C)=O)C)cc2ccncc2s1 CC(F)(F)C(F)C(=O)NC1CC(COc2ccccc2)C1 Cc1ccc(C(=O)NCC(C)(F)CNC(=O)C(C)C#N)cc1F C12(NC(=O)Cc3cnns3)CCCCC1N(C(=O)CS(=O)(=O)C1CC1)CC2 c1(C(=O)NC2CC(NC(=O)CC(c3ccc(F)cc3)O)C2)ccnc2ncnn12 N1(C(C2N(C(c3c(C)n[nH]c3)=O)CC2C)=O)CCc2cccnc2C1 C(=O)(C(O)CCC(C)C)NC1CC(NC(c2c(SC)csc2)=O)CC1O CC(C)C(CNC(C1(C)CC1(C)C)=O)C(=O)N(C(C)CCO)C C1(CNC(CS(CC)=O)=O)CC12CCN(c1snc(Cl)c1C#N)CC2 c1(OC)ccc(Cl)cc1C(N1CC2CC1CC2NC(=O)Cc1cnnn1C)=O C=CCC(CNC(C1CCCN1CC(C)C)=O)NC(c1cc(CC(C)C)[nH]n1)=O c1(CC(=O)NCCN(C)C(c2ccc3nonc3c2)=O)cncc2ccccc12 C1(SC)CN(C(C2CC(n3cccn3)C2)=O)CC1NC(=O)CNC(C1CCC1)=O C(=O)(CCCCC(F)(F)F)NCC1C(C)(C)CCN(C(CCCOCC=C)=O)C1 C1(N(CCC)C(=O)N(C2CCCN2C)C)CC(O)CC(C)(C)C1 C1(NC(CCC(C)OCC)=O)CCC(C)N(C(=O)Cn2ccsc2=N)C1 C1(O)(C(C)NC(c2occc2CN)=O)CCN(C(=O)CCSc2ccccn2)C1 C1(CNC(C(C=C)O)=O)CC12CCN(C(=O)CCCCC#N)CC2 C1(C(=O)NCC2(F)CC(NC(C3CN(C)C3)=O)C2)CCC(F)(F)C1 Cc1ncnc(O)c1C(N1CCC(CCCNC(C2(CO)CCCO2)=O)CC1)=O Nc1ccc(C(=O)NC2CCCC2NC(=O)CC(F)(F)Br)nc1 n1(C2(C(N3CC(CNC(C4(CO)CC4)=O)C3)=O)CCC2)cc(Br)cn1 C1(C)(C(=O)NC2C=CC(C(=O)NC(c3cn(C)nc3)CO)C2)CCSCC1 c1(SCC)cccc(C(N2CC(C(C)(C)O)(CNC(=O)CCC(C)OC)C2)=O)c1 Cc1cc(C(=O)NCC(CC(F)(F)F)NC(=O)CC2CCCCN2C)cc(C)n1 N1(C(C(C)(C)CF)=O)CCC(C2(O)CC(NC(C3C=CCCC3)=O)C2)CC1 N1(C(C(CCCC)O)=O)CCN(C(c2cc(C(F)F)ncn2)=O)CC(C)(F)C1 c1(SC(CNC(c2n(C)ccn2)=O)(C)Cn2cccn2)cccc(I)c1 c1(C(=O)N(C(C)(C)C)CCl)ccc(-c2cncnc2C(N2CCOCC2)=O)cc1F CC(C)CC(CNC(=O)CCc1ccc[nH]1)NC(=O)CC1CCN(C)C1 Cc1cc(Cl)n[nH]c1=NC(=O)C1CCCN1Cc1cnc(C(C)C)s1 C1(OC)CCN(C(=O)CC2(OC)CN(C(C3CC4(CCC4)C3)=O)C2)CC1F c1(CN(c2n(CCC#C)c(C(C)O)nn2)CC)ncc2n1CCCC2 N1(CC)C(=O)CCC1CC(=O)NC1CCN(C(c2sc(C(C)C)nc2C)=O)C1C C1(NC(c2c(C)cnnc2)=O)CC2CCC1N2C(C1(C(F)F)CCCC1)=O N1(C(C2C(CC)CCO2)=O)CC2(NC(=O)COCc3nc(C)no3)CCC1CC2 C1(CNC(c2c(C)oc(-c3ccccc3)n2)=O)C(C2CC2)CCN1C(=O)CC#N Cc1c(CNC(c2nccc(Cl)c2F)=O)oc2ccccc12 C(=O)(C(C)(C)CCC(C(=O)NCCC#N)N1CCOCCC1C(C)C)OCC c1(CNC(=O)NCC(=O)OC(CC(O)CO)C)ccc(OCCF)cc1 c1(CC)ccc(F)cc1NC(=O)CCCCNC(=O)C=Cc1ccn(C)c1 C1(NC(CC2(CS(C)(=O)=O)CC2)=O)CCCN(C(=O)C2=C(Cl)CC2)CC1 c1(C(=O)NCC(C(C)(C)C)NC(CNS(CC)(=O)=O)=O)cc(N)c(F)cc1F c1(CNC(c2n(CC(=C)C)nnn2)C2(CF)CC2)ccc(-n2cncn2)c(F)c1 N1(Cc2ccc(N(C)C)cc2O)CC2CN(C(c3ccc(F)c(Cl)c3)=O)CC2C1 c1(-c2nc(CNCCn3c(C(=O)OCC)cc(C)n3)c(C)o2)ccc(Cl)c(Cl)c1 C1(CC(=O)NC(CC#C)CCOC)N(C(c2ncc(CC)cn2)=O)CCC1(C)C c1(C(=O)NCC2CCN(C(Cc3cccc(OC)c3)=O)C2)nc(Br)cnc1N N1(C(C2(CSC)CC2)=O)CCC(C(C)C(=O)NC2CC(C)C2)CC1 c1(C(=O)NC(CC(C)NC(c2cn(CCF)nn2)=O)C)cccc2nnn(C)c12 CCCCCCC(F)C(=O)N(CCNC(=O)CS(=O)(=O)N(C)C)C1CC1 Cc1c[nH]cc(C(N2CCC(NC(C3CN(C4COC4)C3)=O)CC2)=O)c1=O C1(CC(N2C(C)CC2)=O)COCCN1C(C1CCCC(=O)C1)=O c1(N(C)C(c2ccccc2Oc2ccccc2)=O)ncnc2cc[nH]c12 c1(CC)ncc(C(=O)NCC2C(C)CCN2C(=O)C#CC(=O)N(C)C)c(O)n1 c1(C(C)C)cccc(CNC2CCCC(CCN)C2)c1 C1(NC(C2C(C)(C(C)C)C2)=O)C=CCN(C(=O)C(C)n2cccn2)C1 c1(C(N(CC(O)CNC(=O)CN(C2CCCC2)C)C)=O)cc(=O)n(C)cn1 N1(C(C(CC)(C)C)=O)C2CCC1CC(CC=C)(NC(c1ccn(C)c(=O)c1)=O)C2 c1(CC)cc(C(=O)NC2CCC(NC(c3cnc(C(N)=O)s3)=O)CC2)cc(O)n1 O=C(CCCCC(F)(F)F)NCC1(F)CCN(C(C2CCCOC2)=O)CC1 C12(NC(CC=C)=O)CCN(C(c3cccs3)=O)CCC1C2 N1(C(C)=O)CCOC(C(=O)NCCC(C)C)CC1.CCCC1C(=O)N1 c1(NC(C(N2CCC(F)(C(=O)OC)C2)=O)=O)ccc(F)cc1C(C)C N1(C(C(C)(C)CNC(C2CC3C=CC2C3)=O)=O)CCC(CO)C(O)C1 c1(NC(N2CC(C(C(=O)OCC)F)C2)=O)ccccc1OCC c1(N2CC(C)(CNC(Cc3n(C)cnc3)=O)OCC2)ncc([N+](=O)[O-])cc1CO N1(Cc2c(C)noc2-c2ccccc2)CCN(C)c2ccc(C(=O)O)cc21 N1(CCc2c(C)cccn2)C(=O)CN(Cc2cccc(OCC(F)(F)F)n2)C1=O C(CCN(C)C(c1ccc(C(F)F)o1)=O)(C(C)C)NC(c1cn(CC=C)nc1)=O N1(C(c2ccc(CC)s2)=O)CCC(C)(C)C1C(=O)NCCF C1(NC(C2CC(C3CCC3)C2)=O)CCCCN(C(c2ccco2)=O)C1 Cc1cc(C(N2CCC(NC(c3cc(O)cc(F)c3)=O)C2)=O)cc(C)c1F C1(NC(CC2N(C)CCC2)=O)CCC12CCN(C(c1cscn1)=O)CC2 CC1(C)CCN(C(=O)C#CC2CCC2)C1C(=O)NCc1ncc(F)cc1F c1(C(C)C)ccoc1C(=O)NCC(C)(O)CNC(=O)CCC1CCCOC1 c1(C(=O)NCC2(O)CCN(C(CCCCOC)=O)C2)cc(Cl)c2ccccc2n1 C12(CNC(C3C(C)(C)C3(F)F)=O)CCCC1N(C(c1cocn1)=O)CC2 CC(C)CNC(=O)CN(C(N)=O)C1CC1.C1C(=O)N1C(C1CCC1)C C(=O)(CC(C)(C)CCOC)N1CC(N(C(c2c(CC)[nH]cc2)=O)C)C1 C(=O)(CC(=O)NC(C)(C)COCCCNC(C1CN(C2COC2)C1)=O)N(C)C N1(C(CCc2cc(C)on2)=O)CC(O)CC1CNC(=O)CC1CCN(C)C1 C(C)(C(C(=O)NCCC1CCOC1)NC(c1cc(C)sc1N)=O)OC c1(C(N2CC(C(C)NC(c3ccc(Cl)s3)=O)C2)=O)cn2c(n1)CCCC2 c1(C(N2CCN(C3CC3)C(=O)C2)C(=O)NC2CCCCC2)cc(F)cc(I)c1 N1(C(C2CN(C(N)=O)C2)=O)CCCCC1C1CCN(C(=O)CCc2cn[nH]c2)C1 C1(C(N2C(CC)(CC)CC2)=O)CN(C(C2CC(=O)C2(C)C)=O)CCN1C C(=O)(CCCCCC#N)NC(C1CCN(C(C2CCCC(F)C2)=O)C1)C Cn1cnc(C=CC(=O)NCCCCC2CN(C(c3cc(C(F)F)cs3)=O)C2)c1 C1(CN(C(=O)CSCc2cccnc2)C)CC(F)CN1C(=O)C(Cl)=CCl CN1CCN(C(c2occc2CNC(c2cc(C(N)=O)co2)=O)=O)CC(O)C1 c1(C(=O)NCCCn2cc(CC(c3ccccc3)C)nn2)c(C#N)cnn1C N1(C(C2CCC(C)O2)=O)CC2CCC(C1)C2CC(=O)N1CCC1 C1(NC(c2csc(O)n2)=O)CC2(C1)CN(C(c1cnc(-n3cccn3)cn1)=O)C2 c1(-n2ccc(C(N(CCNC(=O)C(C)(C)SC)CC)=O)n2)ccc(F)c(Cl)c1 C1(NC(C=CC)=O)C(C)(C)CN(C(C2CN(C(=O)C(C)(C)C)CCO2)=O)CC1(C)C c1(C(=O)NC(CNC(C2CN(CC)C(=O)N2)=O)C(C)C)cccc2c1CNC2=O N1(CCNC(=O)C(F)CC2CC2)CCCN(C(C2CCN(C3COC3)C2)=O)CC1 c1(OC)cc(CN)ccc1CNC(N1CC(CO)OCC1C)=O N1(C(c2c(CC)scn2)=O)CCOC2(CCN(C(c3cc(Cl)cnc3C)=O)C2)C1 C1(C(N(CC#CC)C)=O)(NC(=O)C(=Cc2ccco2)C)CCSC1 Cc1cncc(C)c1C(N1CCC(C(=O)NC2CCCNC2=O)C(C)C1)=O c1(OC)cc(F)c(C(N2CC(NC(C3C(C)(C)C3(F)F)=O)CC2(C)C)=O)cc1N S(=O)(=O)(c1ccc(=NCc2ccno2)[nH]c1)NCc1cccc(OCC)c1 c1(C(N2CCC(NC(=O)C(Cl)=CCl)CC(O)C2)=O)cncc2cnccc12 C1(C)(C(N2CC(OCCC(=O)NCCS(=O)(=O)N(C)C)C2)=O)COCCO1 C(=O)(C1=NN(CC)C(=O)CC1)N1CCC(C(C)(C)NC(C(CC)C(F)(F)F)=O)C1 C12(CC(=O)NCC3(C(N)=O)CN(C(C4CC5CCCC45)=O)C3)CCCCC1C2(F)F N1(Cc2ccc(Cl)cc2OC(F)(F)F)CC(NC(c2n(C)ccn2)=O)C2(CC2)C1 C1(C(=O)NCC2(NC(C3NC(=O)OC3)=O)CC2)CCC(C2CC2)C1 CC1CN(C(=O)C(CCC2CCC2)NC(c2cocc2Cl)=O)CC1(F)F C(C#Cc1cn(CC2C(CO)C2(C)C)nn1)NC(c1ccc(C)c(I)c1)=O C(=O)(CC(C(F)(F)F)NC(C1CN(C)CC(C)O1)=O)NC(CC)CCO CCC(C(=O)NC1CCC(NC(C2(OC)CCCCC2)=O)C1)C(C)C c1(C(=O)NC2CN(C(C(C)NC(N)=O)=O)CC2C)cc(O)nc(N(C)C)n1 C(=O)(CC(C)(C)C(F)F)N1CCC(C(N(CC)CC2CC2)=O)OCC1 Cn1c(=O)oc2cc(C(N3CC4COC(=O)C4C3)C(=O)NCCC3CC3)ccc12 N1(C(C2(N(C(c3nc(C)c(C)s3)=O)C)CC2)=O)CCCC2(CCC2)C1 N1(C(c2cn(C)nn2)C(=O)NC(CC)C)CCCCC1c1nncn1C N1(C(C2(NC(C3CN(C)C3)=O)CC(O)C2)=O)CC(CO)C2(CCC2)C1 Cc1cccc(C)c1OCC(O)CNC(c1ccnc(NC(=O)C2CC2)c1)=O C1(NC(Cc2c(C)nc[nH]2)=O)CCCN(C(=O)CC2CCCC2(F)F)CC1 CCCCC(C(=O)N1CC(C(=O)OCC)C1)NC(=O)C(CCC)NC(N)=O N1(C(C(N)=O)=O)CCN(C(C2CC3CCC3C2)=O)CC1c1cn[nH]c1 C(CCC(C)(F)F)N(C)C(C1CN(C(c2ccc(C(N)=O)o2)=O)CCO1)=O N1(C(c2c(Cl)cc(C)s2)=O)CC(NC(=O)C(Cl)=CCl)C(C)(C)C1 CC1CC(CNC(c2nc(C(F)(F)F)cs2)=O)CCN1C(C1CC12CCC2)=O N1(C(C)C)CCC(N(C(=O)C(C2CCN(C(=O)Cn3cnnc3)C2)C)C)C1 c1(-c2cn(C(C)C)c(=O)cc2)ccc2cc(C(=O)NCCC(O)CO)cn2c1 N1(CC)CCOC(C(=O)NCC(C)(C2CC2)NC(c2ccc(C(F)(F)F)[nH]2)=O)C1 CC1CN(CC2CC=C(CN(C)C)CC2)CCC1CO CC1(C)COC(CC(=O)NC2(CF)CCN(C(=O)CC3CCCCC3O)C2)C1 N1(C(c2c(C#N)scc2)=O)CCCC2(NC(C3CCCOCC3)=O)CCCC12 c1(C(N2CCC(N(CCC)C(c3cccc(OC)c3)=O)C2)=O)ccc(N)c(N)n1 C1(NC(CCn2c(C)ncc2)=O)CCN(C(C2CC(n3ccnn3)C2)=O)C12CC2 c1(NC(c2nnnn2C2CCOC2)C2(CC)CCC2)cc(Cl)c(Br)cn1 CC(C(=O)N1CC(OCCOC(=O)C=CBr)C1)n1cccn1 c1(-c2[nH]nc(C(=O)NCc3nc(CNC(C(N)=O)=O)sc3)n2)ccc(F)c(F)c1 C1(Cn2cc(C3CCN(C(c4c(C#N)csc4)=O)C3)nn2)CCC(F)(F)CC1 c1(C(N2CC=CC(NC(C3CCCCS3)=O)C2)=O)ccc(F)c(O)c1 c1(C(=O)NCC(C(C)(C)C)NC(CCC#C)=O)cc2n(n1)CC1(CC1)C2 C(=O)(CC1=CCN(C(=O)C(C)S(C)(=O)=O)CC1)N1CCCC(C)(CC)C1 c1(C(=O)NC2(C)CC(NC(C3C(CC)OCC3)=O)C2)cc[n+]([O-])cc1 Fc1ccc(C(CN2CCCC2)NCC2CC3CC3C2)nc1 N1(C(CCCOCC)=O)CCN(C(=O)COc2ccc(OC)cc2)C2CC12 CC(C(C)C(=O)NC1CC2(CCN(C(c3coc(Br)c3)=O)CC2)C1)S(C)(=O)=O CCC(CNC(c1c(CNC(c2cc(C3CC3)no2)=O)nnn1C)=O)CCO C(CCCCC(=O)N1CC(C)OC(C)C1)N(C(CC(C)OC)=O)C c1(N2C(C3CCN(C(C4C(C(=O)OC)C4)=O)CC3)CCC2)ncncc1C#N n1(CC2CCN(CCCN3C(=O)CCCCC3)CC2)cnc2cc(Cl)ccc12 c1(CC(=O)NCC(C23CCC(CC2)C3)NC(c2ccc(Br)o2)=O)ccc(F)cc1 CCC(C)C(C(C(=O)NCCC1CC1)N(C)CCc1cccc([N+](=O)[O-])c1)OC CC1=CCC(NC(=O)C(Cc2cc[nH]n2)NC(=O)CC23CCCC2C3)CC1 Cc1nnccc1C(=O)NC(C1CCCC1)CNC(C1(C2(C)CC2)CC1)=O N1(C(c2cc(C)c(Cl)cc2)=O)CCC(C)N(C(c2nocc2Br)=O)CC1 C(=O)(C1=C(Cl)CCCC1)NCC1CN(C(C(C)NC(=O)Cc2ccccc2)=O)C1 c1(OC)cc(CCNC(C2CNCCO2)=O)cc(F)c1OC C1(NC(CN(C(C)C)C)=O)COCC1CNC(C1CCOC1)=O c1(CN2C(CC#N)CN(c3ncccn3)CC2)ccc([N+](=O)[O-])cc1F CCC(C)(CC)C(=O)N(CC(C)N(C)C(c1cc(Br)ccn1)=O)C c1(NC(N2CC3CCCC(C3)C2)=O)cnc2[nH]cnc2c1 C1(OC)(CNC(c2cn(C(C)C)cn2)=O)CCN(C(=O)C(C)C(C)C)CC1 c1(CCCC(=O)NCC2(C)CCN(C(C=C(C)C(F)F)=O)C2)ccc(O)c(F)c1 c1(C(C)OCC)ncc(C(=O)NC2CCN(C(=O)C(C)NC(=O)C(C)(C)C)C2)s1 C1(C(C(C)C)NC(=O)CCCF)CCN(C(=O)CC2(C)CC2(F)F)CC1 Cc1ccc(C=CC(=O)NC2CC(N(C)C(C3CCCN3c3nccs3)=O)C2)s1 c1(-c2cc(C(=O)NCc3nc(NC)sc3)no2)c(Cl)cccc1Cl C(=O)(CCC(CF)CF)NC(CC#C)(C)C(=O)NCc1ccc(Cl)cc1 O=C(CC(F)(F)C(F)F)NC(CNC(c1ccnn1C1CC1)=O)CO N1(C(C(C)OCOC)=O)CCCCC(C(=O)NC(c2ncccn2)C)C1 C1(C(N2CCC(NC(=O)C3=CCCCCC3)CC2)=O)Cc2c(F)cccc2O1 C(=O)(C(C)CCC(C)(C)C)NC1CC2(CC(C(=O)NCCNC(C(C)C)=O)C2)C1 N1(C(CC(C)OC)=O)CC2CCN(C(=O)Cc3ccc(OC(C)(C)C)nc3)C2C1 C1(C(NOC(=O)NC)=O)C(C)OCCN1C(=O)C(C)OC Cc1ccc(N2CCCC2)c(C(=O)NCC2CCN2C(c2cc(N)ccc2O)=O)c1 N1(C(C(=O)NCCCC=C)=O)C2CCC1CC(F)C2 C1(C(=O)NCC(CO)NC(c2cc(C(F)(F)F)n[nH]2)=O)CCn2ncnc2C1 C1(C(N2CCCC(C(=O)NC)C2)=O)COCCN(C(C2CN(C(N)=O)C2)=O)C1 C#Cc1cnc(N2CCC(CNC(c3cnc(F)c(F)c3)=O)C2(C)C)nc1 C1(C2CN(C(=O)CCCC(F)F)C2)(NC(C2CCCC(C)C2)=O)CC1 N1(C(C(CC)COC)=O)CCCN(C(c2cc3sccc3[nH]2)=O)C(C)C1 c1(N2C(C)(CNC(C3(C)CCCS3(=O)=O)=O)CCC2)nccn2nnnc12 c1(CN(C)C(C2CCOC(CNC(=O)OC(C)(C)C)C2)=O)c(Cl)cncc1Cl N1(C(c2ncc(C)cc2C)=O)CC(C)(C)OC2(C1)CN(C(c1[nH]cnc1C)=O)C2 C(c1ccc(C)nc1)=CC(=O)N(CC(CC)NC(C1CCC=CCCC1)=O)CC Cc1ccc(F)c(C(N2CC(NC(=O)COC3CCCCC3)CC(O)C2)=O)n1 CCCCC(CNC(c1sccc1C#N)=O)NC(=O)CC1CC2CC2C1 CCC(CC(=O)NC(COC)C(C)C)N(C)C(c1cc(C)c(C)[nH]1)=O C1(C(N2CC(F)(CNC(CCSCC(C)C)=O)C2)=O)CCC(C(N)=O)CC1 Cc1ccn(C)c1C(=O)NC(CNC(=O)CSc1c(C)n[nH]c1C)C(C)C Cc1cc(CC(N2CC(CNC(c3conc3C3CC3)=O)C2)=O)no1 N1(C(COC)=O)CC(CC(=O)NCC(C2CCC2)OC)CC1(C)C Cc1nnn(CC(=O)NC(Cn2cccn2)C(=O)N(CCC(F)(F)F)C)n1 C1(NC(C2CCC(CCC)CC2)=O)CC1C1CCCN(C(c2cnc[nH]2)=O)C1 N1(C(c2ccn(CC)n2)=O)CCC(F)(CNC(C2C3CC4C(C3)C24)=O)C1 C12(NC(=O)Cc3ccc(CO)cc3)CCCC1CN(C(=O)C1=COCC1)C2 N1(C(Cc2nc(C)[nH]n2)=O)CCC2CN(C(=O)Cc3cc(C)sc3C)C2C1 CCCCCCOCC(N1CCC(OCCNC(C2CCCSC2)=O)C1)=O C12(NC(COCCC#C)=O)CCC(C(=O)NCC3CCCC3CF)(CC1)C2 C(CCN=c1[nH]c(=NCc2cccnc2N(C)C)[nH]c2ccsc12)N(C(C)=O)C N1(C(c2c(CC)cncc2)=O)CC(C(=O)NCCCn2cnnc2)CCC1C c1(CC(C)C)ncc(C(=O)NCC2CCN2C(c2cn(CC(N)=O)nn2)=O)s1 c1(C(N(CCC2N(C(C=CC(CC)C)=O)CCCC2)C)=O)cc(Cl)ccc1C c1(C(=O)NCC2C(C)CN(C(=O)Cc3cc[nH]n3)C2)ncc(N)cc1Cl N1(C(C(CC)OCC)=O)CCN(C(=O)CN2CC(=O)NC2=O)CC1CCO c1(C(=O)NC2CCCC(N(C(CCOCC#C)=O)C)C2)ccc([N+](=O)[O-])cn1 C1(OC)CN(C)C(C)(C(=O)N(C2CCN(C(c3ncc(Cl)s3)=O)CC2)C)C1 C1(NC(C23CC(CNC(C(C)(F)F)=O)(C2)C3)=O)CCN(C2CC2)C1=O c1(N(CC)CC)ccc(C(=O)NC23CC(C(=O)NC4CCO4)(C2)C3)cc1 N1(C(Cc2c(C)noc2C)=O)CCC2(CCCN2C(=O)CC2CCC(C)(C)C2)C1 c1(C(N2CC3N(C(C(CC)=O)=O)C3C2)=O)cc(F)c(Cl)c([N+](=O)[O-])c1Cl Cc1cc2[nH]c(C(N3CCCN(C(=O)CNc4nccs4)C(C)C3)=O)cc2o1 c1(CC(=O)OCC)cc(Cl)ccc1NC(c1csc(N(c2ccccc2)C)n1)=O C1(CNC(C2CC(=O)N(C3CCCC3)C2)=O)CC(NC(c2cccs2)=O)C(O)C1 c1(-c2cn(CC)nc2)cc(C=O)ccc1C(=O)OC N1(C(c2ccc(O)c(Cl)n2)=O)CCN(C(=O)Cn2ccnn2)C2CCCCC2C1 CC(C)C1=CCC(C(=O)NC2CCN(C(c3ccc([N+](=O)[O-])o3)=O)C23CC3)CC1 C1(NC(c2c(OCC)cccn2)=O)COC2(CCCN(C(=O)CC3(C)CC3)C2)C1 C1(C(=O)NCCN(C(=O)Cc2ccnc(O)c2)CC)CCC(C(C)C)CC1 c1(CCNC(=O)NC(C)CCCOc2cccnc2)c[nH]c2c(F)c(F)c(F)cc12 c1(NC(c2c(-c3cnn(CCC)c3C)c[nH]n2)=O)cccc([N+](=O)[O-])c1Cl N1(C(CCC#C)=O)CCCC2(C1)CN(C(=O)CC(C(C)C)C(C)C)CCO2 N1(S(CC)(=O)=O)CCOCC1C(=O)NC1CN(C(=O)C=Cc2ccco2)CC1C N#CC1(C(N2CCCN(C(=O)COCC3CCCO3)CC2)=O)CCSCC1 c1(OC)ccccc1C(=O)NC1CCCC1C(=O)Nc1ccccc1N(C)C C(c1c(C)nn(C)c1Cl)=CC(N1CC(CNC(CC2CC(CC)OCC2)=O)C1)=O CCC(COCC1CC1)N=c1[nH]c(=NC)[nH]c(=NCC2(C)CC2(C)C)[nH]1 N1(C(C2(N(C)C(=O)OC(C)(C)C)CC2)=O)CCC(O)C12CCCC2 C(=O)(CC1=CCN(C(=O)COc2ccon2)CC1)NCC1N(C(C)=O)CCC1 c1(C(=O)NC(CC2CN(C(C(CC)C)=O)C2)C)cc(Br)c(Cl)s1 C1(C(=O)NCC(C2CCCC2)NC(C(C(C)C)(C)C)=O)CCCCN1S(N)(=O)=O N1(C(C2CN(C(CC(C)SC)=O)CC23CC3)=O)CCC2(CCCC2)C1 C1(NC(=O)Cc2cc(C3CC3)on2)CC2CCC(C1)N2C(C1CCCC12CCC2)=O c1(C(=O)NCC2N(C(C3(OC)CCCCC3)=O)CCC2C)cn2c(n1)SCC2 c1(C(=O)NCCCCC(C)NC(=O)C=C2CCN(C)C2)ccn2ccsc12 C12(C(=O)NCC3CC(C)N(C(C4C(C)(C)C4(F)F)=O)C3)CCC(F)(CC1)CC2 N1(C(CCC)=O)CCCC(C(=O)N(CCCNC(=O)C=Cc2cnc(C)s2)C)C1 C=C=C(C)CC(=O)NCC1(CNC(=O)C(c2ccc(Cl)nc2)(F)F)CCCC1 C(=O)(C1=CCN(C(c2cnn(C3CC3)c2)=O)C1)NCCC1C(C)C1 c1(OC)cc(NC(c2n[nH]cc2NC(c2ccc(Cl)c(F)c2)=O)=O)cc(Br)n1 Cc1cc(=NCc2cccc3sccc23)[nH]c(N2CCC(N(C)C)C2)n1 Cc1nn(C)c(C)c1C(=O)NCC1(F)CCCN(C(C2C3CCC(=O)C23)=O)C1 c1(N2CCN(C(C)=O)CC2)nc(=N)nc(N(CCC#N)C)[nH]1 CC(C)=C=CC(=O)N1CC(O)CC1CNC(C1CC2(CC2)CO1)=O CCC(CC)CC(=O)NC1(CNC(C2CC23CCCOC3)=O)CCCC1 Cc1cc(F)c([N+](=O)[O-])cc1C(N1CC(NC(=O)CCS(C)(=O)=O)C(O)C1)=O Cc1cc(C(=O)NC2CN(C(=O)C(C)C#N)CC2S(C)(=O)=O)c(S(N)(=O)=O)s1 N1(C(C2CCN(C(CC(CC(C)C)O)=O)C23CCC3)=O)CCc2cccnc2C1 Cn1cc(C(F)(F)F)c(NC(C2CC2NC(C2(c3cn[nH]c3)CC2)=O)=O)n1 N1(C(C(C=C)O)=O)CCCC2C1CCN2C(c1cc(Br)cn1CC)=O Cc1nc(C(=O)NC2CC(NC(C3CCOCC3)=O)C23CCC3)c(C)n1C c1(C(N2CC(NC(=O)Cc3ccc(Cl)cc3Cl)C3C2C3)=O)cncc2[nH]ccc12 Cc1cc(Br)cc2cc(C(=O)NCCNC(C3CCOC(=O)N3)=O)oc12 C#Cc1cc(C(=O)NC2(C)CCN(C(c3ccnn3C(F)F)=O)C2)cc(F)c1 C1(NC(Cn2nc(C)c(Cl)c2)=O)C2CC1N(C(c1cn(C3CC3)cn1)=O)C2C CC(C(=O)N1CCC(O)C1)P(C)(C)=O.C1(CCNC=O)CN(C(=O)OC(C)(C)C)C1 CC1CCCCN1Cc1ccc(SCCC(N2CCC(CC(=O)OC)C2)=O)cc1 CCCC(C)(O)C(=O)N(CC(O)CN(C(=O)Cn1nc(O)ccc1=O)C)C c1(CCC)ccc(C(=O)NC2CCC(NC(=O)CCc3ccc(Cl)cc3)C2)cc1 C1(C(N2CC(C=C)OCC2)=O)CC2CCC(C1)N2C(=O)CC(C)(C)OC c1(CC(=O)NCC2(F)CC(NC(CCCOC)=O)C2)c[nH]ccc1=O N1(C(COC2C(C)CCCC2)=O)CC=C(CCNC(=O)Cc2ccccn2)CC1 N1(C(C2CN(C(c3cc(CC)nn3C)=O)CC2F)=O)CCC(CO)C1(C)C Cc1cccc(C(=O)NC(C2CCCCN2C(c2ccc(CO)cc2)=O)C)c1F c1(SCC(N2CC(CCC(F)(F)F)C2)=O)scnc1C1CCCC1 CC(CCNC(=O)C=Cc1nnc(C(C)C)o1)CCNC(=O)C=CC1CC1 N1(C(CC2N(C(C(C)C3(O)CCC3)=O)CCC2(C)C)=O)CC2CSCC(C2)C1 N1(Cc2c(OC)nsc2)C2CCCC1CN(C(c1cncnc1)=O)C2 c1(C(N(C)CCOCCN(C)C(C2CC(F)C(=O)N2)=O)=O)cc(N)ccc1Cl c1(OC=S)c(F)cc2c(c1F)N2.c1(CN(CC2=CCSC2)C(C)=O)ccccc1Cl c1(C(=O)NC(C)CCCNC(=O)C(O)c2ccco2)ccc(C(F)F)cc1Cl c1(C(=O)NCc2cc(I)cs2)cn(C2CCN(Cc3ccccc3)C2)nn1 N1(Cc2cccc(C(=O)Nc3ccc(C)cc3)c2)CC2(COC(C)C2)C1 S(=O)(=O)(c1cccnc1N(C)Cc1cn(C)cn1)N1CCCC(CC)CC1 N1(C(CNC(CCC)=O)=O)CCC(C2(O)CN(C(=O)C3=C(C)S(=O)(=O)CC3)C2)CC1 N1(C(C(C(=O)OC)C)=O)CCC2(CCCN(C(=O)Cc3ccnc(F)c3F)C2)C1 CC(O)(CNC(=O)CC1CCCO1)CNC(C1(C(N)=O)CC1)=O CCCCC(CNC(C1CC1C(N)=O)=O)NC(c1oc(CCC)nc1C)=O c1(C(N2CC(NC(c3cnc(C)nc3)=O)C(C)C2)=O)cnc2ncnn2c1C C12CCCC(C1)OC2.n1(CCC(=O)N(C)CC)cc(COC)nn1 c1(C(=O)NCCC(C)(C)NC(=O)C(F)C2CCC2)ccc2oncc2c1 C1(C(=O)NCC2(COC)CCCN2C(c2cccnc2)=O)CC(C)CC(C)(C)C1 N1(C(c2c(CC)ocn2)=O)C(C(=O)NCCCNC(=O)C(C)C)C2CC(O)C1C2 Cc1c(NC(c2n[nH]c(=N)s2)C)ncnc1N1CCOC(C)C1 C(N=c1cccc(NC(=O)C(C)(C)C)[nH]1)c1ncn(CC)n1 N1(C(c2cc(C)ns2)=O)CCCC(F)(C(=O)Nc2cnc(C)nc2C)C1 N1(C(c2c(Cl)cn(CC)n2)=O)CC2(CCCC2NC(c2cn(CCO)nn2)=O)C1 N1(C(CC2(C)CCN(C(c3ccc(C=C)cc3)=O)C2)=O)Cc2ccnn2CC1C N1(C(C2(Cl)C(C(C)=O)C2)=O)CC2OCC(NC(c3ccnnc3)=O)C2C1 C1(CNC(=O)CSCC(N2CC(F)C2)=O)CCCC(F)C1 N1(C(c2nccc(CNC(CCCC3C(C)C3)=O)c2)=O)CC2C(C1)C2(C)C c1(OC)ccc2oc(C(C(=O)NC)N(C)CCOC)c(C)c2c1 C(CNC(c1ccncn1)=O)(CC(=O)Nc1ccc(CO)nc1)OC c1(CCC(=O)NCCN(CCOC)C(C2COCC(C)O2)=O)ccc(C)cc1C CC1CC(C)CN(N2CCCCC2c2ncc[nH]2)C1 c1(SC)ncc(Br)c(N(C(=O)Cc2ccc(Cl)cc2F)CC2(F)CCCNC2)n1 c1(C(C)=O)ccc(NC(c2csc(=NCc3cc(C)ccc3Br)[nH]2)=O)cc1O N1(C(c2n(C)cnc2)=O)CCC2(CC(NC(C3CCC3)=O)C2)C1 c1(C(=O)NCC2(F)CCN(C(c3c(C)c(Cl)ccc3)=O)C2)cc2cnccc2[nH]1 c1(C(=O)NC(C2CCCC2)CNC(=O)CCOC2COC2)ncoc1C1CCCO1 N1(C(COC)=O)CC2CC1(CNC(c1ccc(-n3ccnc3)nc1)=O)C2 CC(C)C(F)(F)CC(=O)NC1CCN(C(c2cn(Cc3ccccn3)nn2)=O)C1 c1(C(N2CC3C(NC(C(CC(C)C)F)=O)C3C2)=O)cccc2nccnc12 C1(CC)CN(C(c2ccc(C3CC3)cc2)=O)CCN1C(=O)C(CC)N(C)C CC1(NC(c2snnc2C2CC2)=O)CC(NC(c2ccoc2C2CC2)=O)C1 N1(C(C(CC)OC)=O)CCC2(CCCN(C(=O)CNC(C3CCC3)=O)C2)CC1 c1(OCCC(=O)NCCc2nc(-c3cccc(F)c3)no2)ccc(Br)cc1 c1(C(=O)NCC2(NC(C3CC4CC4C3)=O)CC2)ccc(CO)o1 C1(C(=O)NC(C)C(CO)NC(=O)Cc2ccsc2C)(CC)CC(C)(C)C1 C1(C(=O)NC2(CNC(=O)COC3CCC3)CCC2)CC(F)C(=O)N1 CCC(CCC(=O)NCc1cccc(COC)c1)NC(=O)C=CCN(C)CC Cc1cc(C(=O)NCC2CC(CNC(=O)Cn3ccnn3)CO2)ncc1F Cc1ccc(C)c(C(N2CCC(CNC(C3CCCN3N=O)=O)C2(C)C)=O)c1 c1(OC)c(C)cc(NC(=O)CSCC2CCC3(CCC3)O2)cc1Cl N1(C(Cc2c(OC)nccc2)=O)CC(NC(=O)C=Cc2cscn2)C(C2CC2)C1 c1(C(N(C=O)CC2CN(C)C2)C2CC2)ccc(F)cc1 C1(N(C(=O)CCc2nc[nH]n2)CC)CCCN(C(c2ncccc2C)=O)C1 C=CC(CCC)CC(=O)N1CCC(NC(c2ccccc2N2CCCC2=O)=O)C1 C#Cc1ccc(C(N2CCCC(CC)(NC(=O)CCNC(=O)C=CCl)C2)=O)nc1 N(C1COc2cccc(F)c21)S(c1ccc(NCc2c(C)ocn2)nc1)(=O)=O C1(CC)CN(C(=O)CC23CCC(CC2)OC3)CCC1NC(=O)CCCCC1CC1 CCCC(O)C(CO)NCc1ccc(C(F)F)cc1 N1(C(CNC(c2c(C(C)C)onc2)=O)C)CCN(C(=O)CC2(O)CCOC2)CC1 c1(-c2cn(CCCOCC(=O)NC(CC)(C)C3CC3)nn2)scc(C)c1C(=O)O N1(C(C=Cc2c(N)cccc2)=O)CCC2(CCN(c3nc(C(F)F)nc(=N)[nH]3)C2)C1 C=CCC(CC(C)C)C(=O)N1CCCC1CCCNC(c1n[nH]cc1CC)=O C1(C(=O)NC23C(CN(C(C=C(C)C)=O)C2)C3)CCC(F)(F)CC1 N1(C(c2c(CCC)[nH]cc2)=O)CCCCC1C1(NC(C2CCN(C)C2=O)=O)CC1 C(=O)(C(C)(CNC(c1n[nH]cc1CC)=O)CC)N1C(C#C)CCC1 Cn1ncc(C(=O)NCC2COC(CNC(=O)Cc3ccoc3)C2)c1C(N)=O N1(C(CCS(C)(=O)=O)=O)CC2CCC(C1)N2C(c1ccc(F)cc1Br)=O n1(CCCCNC(C(F)=CCC)=O)cc(CC(C(=O)OC)C2CC2)nn1 c1(CC(N2C(CN(C(=O)Cc3ccon3)C)CCC2)=O)ccc(Br)nc1 C1(CNC(c2cccc(OC(F)F)c2)=O)CC2CC2N1C(=O)C=Cc1ccco1 N1(C(C(N2C(C(=O)NCCOCCOC)CC3CC32)=O)(C)C)CCS(=O)(=O)CC1 c1(C(N2CC(N(C)C(c3ccsc3)=O)C3(C2)CC3)=O)ccnc2c1ncn2C CCC(CNC(c1sc(NC2CC2)nc1C)=O)(CC)NC(C1CC=CCO1)=O N1(C(=O)C2=CCOCC2)CC2CCC(NC(C3CC4CCC(C3)S4)=O)CC2C1 c1(CC)c(C(N2CCCC(CN(C(=O)C=CSC)C)C2)=O)cccc1C c1(C(=O)NCC(CNC(CC=CC=C)=O)C)cc2cccnc2s1 C(=O)(C(CC=C)C(C)C)N1CCCC(CCNC(c2nccc(C#C)c2)=O)C1 C1(CNC(c2nc(N(C)C)oc2)=O)CN(C(C2(C)CCCN2C)=O)CCC1(C)C C1(CC(=O)NC(C)CCN(C(=O)CSc2ccccc2O)C)CC2(CCC2)CO1 Cc1n[nH]c(C)c1C(C)C(=O)N(C(CNC(=O)C=CC1CC1)C1CC1)C c1(C(=O)NC2CCC(C(N=c3cc(C)o[nH]3)=O)CC2)c(F)ccc([N+](=O)[O-])c1F N1(CC(C)C)CCCC1C(N1CC(C(C)NC(=O)C=CSc2ccccc2)C1)=O c1(OC)ccc(C(=O)N(C(=O)CC2CCC(C(F)(F)F)N(C)C2)C2CC2)nc1Br c1(C(N2CC(NC(c3cc(C)nnc3O)=O)C3C2C3)=O)cc(F)cc([N+](=O)[O-])c1 C(C(C)(C)CC(=O)N1CC(n2cnnn2)C1)NC(c1cc(C)nn1C)=O c1(C(=O)NCC2CCC(NC(C3(CC)COC3)=O)C2)ccc(-c2ccsc2)cc1 C1(C(=O)NC2CCC(NC(=O)CN3CCSCC3)CC2)CCc2ncnn2C1 Cc1nc2c(n1C)CN(C(c1ccc(C(F)F)o1)C(=O)NCC1CCCO1)CC2 O=C(C1=CCOC1)NC1CN(C(c2cc(-c3ccccc3)on2)=O)CC1C(F)F Cc1csc(=O)n1CCC(=O)NCC1CCC(NC(=O)CSC2CC2)C1 CC1=C(C(=O)NCC2CN(C(=O)C(C)Cc3cnco3)C(C)(C)C2)CCO1 c1(N(C)CCN2CCCCC2)ccc(-c2cc(CN)[nH]n2)cc1 C1(NC(c2ccc(C(F)F)cc2)=O)CN(C(=O)Cc2sc(O)nc2O)C2CC12 CC(C)C(C)(CNC(c1cc[nH]c1)=O)NC(C1CC1F)=O C1(CCOC)(C(=O)NCCN2CCC(C)C2)CCN(C(=O)C=CC(C)(C)C)CC1 Cn1nc(Br)cc1C(=O)NCC1(C)CCCC1NC(C1CC1(C)C)=O C1(C)(C(NOCCCOC)=O)CC(O)CN1C(c1c[nH]nc1C1CC1)=O c1(C(N(C(C)CNC(=O)CCN2CCCCC2)C)=O)cc(N)cc2ccccc12 C1(CNC(C#CC(C)(C)C)=O)CN(C(=O)CC2CCSC2)C2(CCC2)C1 C=CCCC(=O)N1CCCC1C(C)(C)CNC(c1cnn(CC=C)c1)=O c1(CC(=O)N(CCCNC(C2(C)CC(F)(F)C2)=O)CC)c[nH]c(=N)nc1O C1(NC(=O)C=Cc2ccoc2)CCN(C(C2(F)CC2)=O)CCC1c1ccccc1 N1(C(C(CCC)CCC)=O)CCc2sc(CNC(=O)COCC3CC3)nc2C1 N1(C(C(COC)(F)F)=O)CCC(CNC(c2cn(C)cn2)=O)C(F)(F)CC1 N(C(=NCC1C(C)(C)C1(C)C)NC(c1cccs1)C)CC1(C#N)CCC1 c1(C(C)NC(C(=O)Nc2c(C(=O)OC)cccc2)=O)nc(Cl)ccc1Cl CCN=c1[nH]c(C)c(C(=O)NC2CN(C(=O)C(C)(CC)CO)CC23CC3)s1 c1(OC)ccc(Cl)c(C(=O)N(C(C)CNC(c2csnc2C)=O)C)n1 C=CC(C)(O)C(=O)NCC(C1CC1)N(C(=O)C(F)(F)Sc1ccc(F)cc1)C c1(C(=O)NCCC(C)NC(c2cc[nH]c2-c2ccccc2)=O)ccc(F)cc1Cl C(=O)(CC1=Cc2ccccc2C1)NC1(CO)CCN(C(C=CCN(C)C)=O)CC1 N1(C(c2[nH]ccc(=N)n2)=O)CCN(C(=O)C2=C(Cl)CC2)C2CCCCC2C1 C(=O)(CC(CC(C)C)NC(=O)Cc1ccc(C#N)cc1)NC1CCN(C(C)=O)C1 N1(C(C(CC(N)=O)O)=O)CC2CN(C(c3scnc3Cl)=O)CC2C1 N(C1CCCn2cnnc21)C(=O)CC1CCN(C(C2CC3CCCC3C2)=O)CC1 c1(NC(C2N(C(c3ccc(C(C)O)cc3)=O)CC2)=O)ccc(S(N)(=O)=O)cc1Cl C=CCCCCCCNC(C1(NC(C2C(C)(C)C2(F)F)=O)CCC(C)(C)C1)=O C(CCCC(=O)NC(C)CCC1CC1)N(C(C(C)C1CCOC1)=O)C C(=O)(CC(C(F)(F)F)NC(c1ccc(F)cc1C)=O)N1CC2C(CC)(C2)C1 C1(COC)(NC(C2CC2(C)C)=O)CN(C(c2cnn(C)n2)=O)C1 c1(C(=O)NC2COCCN(C(c3nccc(C#N)c3)=O)C2)ccc2cnnn2c1 C1(CNC(c2cc(C)ncn2)=O)N(C(=O)CN2CCCC2C)CCC1(C)C N1(C(CCS(=O)(=O)NC)=O)CCC(C2CC(NC(=O)Cc3cncn3C)C2)C1 C12(C(=O)NCCN(C(CCCNC(=O)OC)=O)C(C)C)CCCCC1NC(=O)C2 C1(C(=O)NCCCC(C)NC(c2c(C)ccs2)=O)COCCN1CC(F)F c1(OC)cc(-c2ccccc2OC(F)=C(F)F)c2cc(CO)[nH]c2c1 Cc1cccc2cc(NC(C3CN(C(C45CCC(CC4)C5)=O)CCC3O)=O)[nH]c12 N1(C(C2(SC(C)C)CCC2)=O)CCN(C(=O)C(C)N(C)C)C2(CCC2)C1 N1(C(CC2CCC(OC)CC2)=O)CCC(C)(NC(C2CCCS(=O)(=O)C2)=O)CC1 O=C(Cn1nnc2cc(C(=O)O)ccc12)NNC(=O)N=c1cc2n([nH]1)CC(O)CO2 CCC(O)C(C)C(=O)NCC1(O)CCN(C(c2cnc(C(C)=O)s2)=O)C1 N1(C(c2c(C)csc2Cl)=O)CC(CNC(C2(C)CCC(=O)NC2)=O)C2(CC2)C1 C(N=c1[nH]c(N2CCC3(C2)CN(C)C3)nc(=N)[nH]1)C1CCC(C)(CC)O1 N1(C(c2ncccc2Cl)=O)CCC2C(C1)CN2C(=O)CCSCc1ccccn1 N(C(=NCCc1ccc(F)cc1)NCC(=C1CCOCC1)F)C1C(C)C1 c1(NC)cnc(Cl)cc1C(=O)NC1CC(C)CN(C(c2cc(C)nc(C)n2)=O)C1 C(CC(C(=O)NCC1(C(C)(F)F)CC1)NC(C12CC(F)(C1)C2)=O)N(C)C c1(NC(CC2CCN(C(c3cc(OC)c(I)cc3)=O)C2)=O)ccc2c(c1)OCC2 c1(C(=O)NCCCCC2(NC(C)=O)CC2)cnc(O)cc1C(F)(F)F C(C)(C)(C(C)CC(=O)N1CCC(C2CC2)CC1)NC(C1CN(CC)C(=O)C1)=O CC(=O)CCCCC(=O)N1CC2(CCCC2)C1C(N1CCN(CC2CC2)CC1)=O N1(C(C(CCOCC)NC(C2C=CCC2)=O)=O)CC2(CC=CC2)C1 C1(CNC(C2C(CC)C2)=O)C(C)CCN1C(=O)CCN1CCNC(=O)C1 Nc1cccnc1C(=O)NC(CC1CCCC1)C(N1CCCC(F)C1)=O c1(OC(C)C(=O)NC2CC(C(=O)Nc3c(Br)nnn3C)C2)ccc(F)cc1 C(=O)(C(F)(F)CO)N1CC(CC(C)NC(c2cnc(-c3ncccn3)s2)=O)C1 CCCS(=O)(=O)C(C)C(=O)NC1CCC(NC(c2cncc(C3CC3)c2)=O)C1 C(=O)(CCCC(=O)NC(C)C)N(C1(C)CC(NC(=O)CC(O)CC)C1)CCC C(C(CNC1(c2nnnn2CCN2CCOCC2)CCOC1)C(C)C)OC C12(CNC(C(C=C)(C)CC)=O)COCCN1CCN(C(C1(Cl)CC1)=O)C2 C(=O)(C(Cc1cccnn1)NC(c1ccsn1)=O)OC C(=O)(CC(C)(O)CCC)N(C1CCN(C(=O)COCCSC)C1)CC c12ccc(c3c1CCCC3)oc2=O.c1(C(=O)NCC)ncoc1C1CCCCC1 C1(C(N2C(C)(C(=O)NC)CCC2)=O)CCN(C(=O)C(C)=C(C)C)O1 CCCC(O)CC(=O)NCCCCNC(=O)C(F)(F)C(O)c1ccccc1 N1(C(CNC(CC(C)c2ccco2)=O)=O)CC(O)C(O)C1 Cc1n[nH]cc1CN(C)C(C1(NC(=O)CCC2CCCC2)CC1C)=O c1(N(C)CC2CC2)nc(N2CCS(=O)C3(CCC3)C2)nc2c1CCCCCC2 C1(C(=O)NC(C2CCCN2C)C)CC2CC2N1C(C1CCN(C)CC1)=O C12(C(=O)NC(C)C(CO)NC(=O)C(C)OC3CCCCC3)CCC(CC1)CC2 c1(CC)c(C(=O)NC2CC(CNC(=O)C(C)C(C)(C)C)C2)cccc1F Cc1nc(C(=O)NCC2CCCCCN2C(=O)CC2COC(=O)C2)cn(C)c1=O N1(C(C(CC=C)NC(C)=O)=O)CCC2(CC1)CC2C(=O)N(CCCF)C N1(C(C2(C)CN(C)C(=O)C2)=O)CCN(C(C2CC(F)(F)CS2)=O)CC12CC2 C=CCC(C(=O)NCC=CCNC(=O)CCOCC1CCCO1)c1ccccc1 CCC(C)(C)C(O)C(=O)NCC(CC1CC1)C(=O)N1CC(C(F)(F)F)C1 C1(C(=O)NCC2C(NC(=O)CCc3ccsc3)CC2)CCC2CC2CC1 c1(NC2CN(C(CNC(CC3(OC)CCC3)=O)=O)C2)ccnn1C(=O)OC C(C(C)(C)C(=O)N(C)CC1CCCNC1=O)NC(C(C)SC)=O N1(C(C2(COC)CCOC2)=O)CCC2C(C1)CN2C(c1cccc2scnc12)=O C1(NC(Cc2scc(C)n2)=O)CN(C(c2ccc(CO)c(F)c2)=O)CCC1C C1(C(=O)NC(C)CNC(c2ccc(CC(F)(F)F)cc2)=O)CC2C=CC1CC2 Cc1ccc2occ(C(=O)NCC34CC3CN(C(c3ccc(Cl)cc3)=O)C4)c2c1 CN1CC(O)CC1(C)C(N1CCCC(NC(c2cc(O)ccc2F)=O)CC1)=O N(C1CCc2cccnc21)C(CNC(CC(CCCC)O)=O)=O C1(CNC(C(c2c(C)cccc2C)O)=O)CC2CC(C1)N(C(=O)CC#N)C2 N1(C(C23CN(C(=O)C(F)OC(F)(F)F)C(C2)CCO3)=O)CCN2C(=O)NCC2C1 c1(C(N(C(C)CNC(=O)C=CC2CC2)CC)=O)cnc(C#N)s1 C1(C(C)=O)CC(C(=O)NC2CC(NC(=O)C(C)(C)c3cccs3)C2)C1(C)C C1(O)(CN(C(COC)=O)C)CCCN(C(C2CCC(=O)N(C3CC3)C2)=O)C1 CCC(CCC(=O)Nc1cnn(C)c1C)NC(c1cnn(C)c1CC)=O c1(CC(N2CC(F)CC(NC(c3n[nH]cc3Cl)=O)C2)=O)coc2ccc(F)cc12 N1(C(C2C(c3n(C)cnc3)C2)=O)CCC(F)(NC(c2cccc(Br)c2F)=O)CC1 N1(C(C2C=CC(NC(=O)CC3(O)CCCC3)C2)=O)CCc2ccsc2C1 CC1CC2(CCN(C(=O)C3=COCCC3)CC2)CN1C(C1CCCC(C)(C)O1)=O c1(OC)c(NC(C2C3CCC2(c2ccccn2)C3)=O)cccc1C(=O)O c1(CNC(C2CCCCO2)CF)cn2c(n1)CCCCC2 C1(SC)CCCC1n1cc(C2(C)CN(C(C3CCCN3C(C)C)=O)C2)nn1 C1(CN(C(C(C)n2cccc2)=O)C)CN(C(c2cc(C(N)=O)c[nH]2)=O)CCO1 C1(NC(C(CCCC)=O)=O)CN(C(c2cn(CCC)nn2)=O)C2(CCC2)C1 C1(CNC(CC#C)=O)CC2CCC1N(C(c1nccn1C)=O)C2 O=C(C1=C(c2ccc(F)cc2)CCOC1)NCC1CCCCCC1(F)F C1(C(N2CC(NC(C(C)(C3CC3)OC)=O)C(SC)C2)=O)CCC(C)(F)CC1 c1(C(=O)NC(C2(O)CN(C(c3ccc(C)c(F)c3)=O)C2)C)cc(C)n(C)c(=O)c1 CN1N=C(C(=O)NC2CC(NC(c3c[nH]nc3Br)=O)C23CCC3)CCC1=O CC1(C(C)(C)O)CCN(C(=O)NC2(c3ccccc3)CCC2)C1 C(C)(CCC(=O)N1CCOC(CNC(c2cn(CCC(C)C)nn2)=O)C1)OC N1(C(C(C)n2ccnc2)=O)c2ccccc2CC1CN c1(CNC(c2ccc(CCCCC)o2)=O)cc(O)nc(CNC(=O)C(O)CC)n1 c1(OC)ccc(C(=O)NCC2(C(C)(C)C)CCN(C(C3(C)CC3)=O)C2)c(C)n1 N1(C(c2nc(C)oc2)=O)CCC(NC(=O)C=CC(c2cnn(C)c2)=O)CC1C c1(OC)ccccc1COC(F)(F)F.C1(C2CNC(=O)C(F)O2)CCN(CC)C1 c1(C(=O)NCCC2CCN(C(c3cc(C(=O)OCC)n[nH]3)=O)C2)cncc(C)n1 C1(C(=O)NCCCCNC(C(C2CCCCC2)N(C)C)=O)CCc2nccn2C1 C1(NCCC2(C)N=N2)CN(C(=O)OC(C)(C)C)CC12CCC2 CN1CC(NC(=O)C(C2CCC2)NC(=O)CC(Cl)Cl)C(=O)N1 C12(C(=O)OC)CCN(C)CC1CN(c1nnc(C(C)(F)F)n1CC(C)C)C2 N1(c2snc(CCC)n2)CCC(C)C(NC(=O)C(C)(c2ccccc2)OC)C1 Cc1csc(C=CC(=O)NC23CC2CN(C(C2(c4ncco4)CC2)=O)C3)n1 N(C1CCOc2cccc(Cl)c21)C(C(n1cc(-c2cccc(Cl)c2)nn1)C)=O c1(SCC(C)=O)cccc(NC(=O)NC(c2nnc(C)o2)CC)c1 C(=O)(C1CCCc2ncnn21)NC1(C)CCCN(C(CCC#C)=O)C1 c1(CC(=O)N(CCN(C(CCOCC#C)=O)C)C)cc2ccccc2c(=O)o1 CCCC(C#N)C(=O)N1CC(NC(c2cc(-c3cnn(C)c3)on2)=O)CC1(C)C N1(C(COCC#C)=O)CC(NC(=O)C(CC#C)C2CC2)C(O)C1 N1(C(C(CC=C)CC)=O)CC2CCC1C(CNC(c1ccc(=O)n(CC)n1)=O)C2 N1(C(C2CCN(C(Cc3nc(C)sc3)=O)C2)=O)CCc2cc(F)c(F)cc2C1 c1(OC)ccc(C(=O)NCC2CC(OC)CN2C(C2CNC(=O)N2C)=O)cc1F c1(-c2nccn2C)ccc(Cl)cc1.C1(CN(CC)CC2CC2)(OC)CCCC1 CC1(C)CCC(C(=O)NC2(C(=O)Nc3cc(F)ccc3O)CCSC2)CO1 N1(C(CN(C)C(=O)C2CC2)=O)CCCC12CCN(C(c1cc(N)c(Cl)cn1)=O)C2 N1(C(CC(C)(C)NC(=O)CCN=[N+]=[N-])=O)CCC12CCC(O)CC2 Cc1ccc([N+](=O)[O-])cc1C(=O)NC1CCN(C(=O)CC=C(Cl)Cl)C(C)C1 C(C)(c1ccccc1C)=CC(N1CC(CC)C(CNC(C2CC(C)C2)=O)CC1)=O CC1(C)COC(CCNC(C2(NC(=O)C(F)F)CCCC2)=O)C1 C(=O)(C(COC)CC)N1CCC(CN(C(c2c(CCC)nco2)=O)C)C1 Cc1cccnc1C=CC(=O)NCCN1CCN(C(C2(C)C=CCCC2)=O)CC1 N1(C(CNC(c2n(CC)ncc2)=O)C(F)F)CCN(C(=O)CC2CCOC2)CC1 c1(OC)cc(N2CC3CC(NC(c4csnn4)=O)CC2C3)ccc1[N+](=O)[O-] C1(C(=O)NC2CCC23CN(C(c2cc(Cl)c[nH]2)=O)C3)CCc2nccn2C1 C1(COC)CN(C(c2ccnn2-c2ccccc2)=O)CCN1C(C1CC1(F)F)=O CC(O)C(C)(C)C(=O)NC1CN(C(C2CC(=O)N(CC(F)(F)F)C2)=O)C1 NS(=O)(=O)c1n[nH]cc1C(N1CCC12CN(C(c1ccnc(Cl)c1O)=O)C2)=O C1(O)(CC(N2CCC(Cn3cc(CN4CCCCC4)nn3)CC2)=O)CCCOC1 N1(C(c2cccc(NC(C)=O)n2)=O)CC2(CCC(CNC(C3CC3CF)=O)O2)C1 C(c1cncc(F)c1)=CC(=O)NC1CC(NC(c2cccc(Br)c2)=O)C1 C(C)(C)(CC(=O)NCC1CC2CCC1C2)NC(Cc1c(C)ncs1)=O N(C(=NCCN1CCOCC1)NCSc1ccc(Cl)cc1)CC(C)(CO)C1CC1 c1(C(=O)NCC(C)N(C(C(C)OCC#C)=O)CC)cnc(CCC(F)(F)F)s1 C(=O)(CCC(=O)N1CCC(F)(CNC(C2CCC(C)(C)O2)=O)C1)NC N1(C(C2N(C(C(c3cccc(C)c3)C3CC3)=O)CC2)=O)CCCC2(COC2)C1 N1(C(CC(C)OC)=O)CCN(C(=O)C=Cc2ccnn2C)CC1CC(F)(F)F C1(CC(=O)NCC(CCOC)NC(=O)C=Cc2ccncc2)CCCC(OC)C1 C(=O)(CCC(C)(C)C)NC1C(CNC(C2CCCN(C(C)=O)C2)=O)C1 N1(C(C2CCC(C(C)(C)C)CC2)=O)CC2CCC(NC(=O)C=C3CCC3)CC2C1 C12(C(n3cc(C4CN(C(=O)Cn5ncnn5)CCO4)nn3)CC)CCC(CC1)C2 C1(NC(C2(CCCC)CCC2)=O)CCCCCC1NC(=O)CC1CCN(C)CC1 c1(OC)nscc1C(=O)NC1CC(O)C1CC(=O)NC1(C(=O)OC)CC1 C1(NC(c2cn(CC)nn2)=O)CCN(Cc2nc(CC(C)C)no2)C(C)C1 CCC(CC)(CCC(=O)NCCCN(C(=O)CC1C=CCCC1)C)[N+](=O)[O-] C(=O)(C(O)C(F)(F)F)NCC(C)(C)CNC(C1(n2cccn2)CCC1)=O c1(C(N2C(CCNC(CC#C)=O)CCCC2)=O)ccc(NS(C)(=O)=O)cc1Cl c1(COC)nc(C)c(C(N2CC(C)(NC(=O)C(C)NC(=O)COC)C2)=O)s1 N1(C(C(C2CC2)OC)=O)CC(C2CN(C(c3ncc(Cl)cc3Cl)=O)C2)C1 CCC(C)(CNC(=O)C(F)(F)C1CCOCC1)NC(=O)CN1CCOC1=O C1(C(N2CC(CCCCNC(c3c(C)ccnn3)=O)C2)=O)CCC2(C1)CC2(F)F Cc1ccnc(C(=O)NC(C)CC(C)NC(=O)Cc2ccc(C(N)=O)nc2)n1 CC1(C)CCOC1C(=O)NCCC1(C)CCN(C(c2cccc[n+]2[O-])=O)C1 CCCCC(CC)C(=O)N1CCC1C1CCN(C(c2cc3n(n2)CCO3)=O)CC1 O=C1COc2cc(F)c(C(N3CCC(NC(C4CNC(=O)N4)=O)C3)=O)cc2N1 C1(C(=O)NCC(C)NC(=O)C(=O)NCC(F)(F)F)CCCN1C1CCCC1 C1(CNC(c2ccc(C)cn2)=O)COCCN(C(C2(C)COC(=O)C2)=O)C1 c1(CN(C2CCC3(CCC3)C2)C=O)ccc(F)c(C(F)(F)F)c1 c1(OC)c(C(N2CCC(CNC(c3cc(=O)cc[nH]3)=O)CC2C)=O)ccnc1Cl c1(C(N2C(CNC(=O)CCc3cnoc3)CC3(CC3)C2)=O)cnc2[nH]ccnc1-2 O=[N+]([O-])c1cnn(CC(O)CN2CCOC(C3CCCCC3)C2)c1 c1(C(=O)Nc2c(F)cc(I)cc2F)n[nH]c2c1CN(c1ncc(F)cn1)CC2 c1(OC)ccc2ncc(C(=O)NCC3CC3CNC(=O)C=CC3CCOC3)n2n1 N1(C(CCC2CC(OC)C2)=O)CC(C2CN(C(=O)C(C(C)(C)C)NC(N)=O)C2)C1 c1(C(=O)NCc2cc(C(=O)NC(C34CCC(CO3)C4)C)on2)ccnc(CO)c1 Cc1cc(-c2cn(CCCC(=O)NC3CCCOC3(C)C)nn2)c(C)cc1Cl CCC(C)(COC)CNC(=O)C(c1cn(C)nn1)NC(=O)C=CC1CC1 C(=O)(C1CCc2cccnc21)N1CCCCC(NC(c2cscn2)=O)CC1 C1(C(=O)NCC(C)(C2CCC2)NC(=O)CC23CC(C2)C3)CC2(C1)CC(F)(F)C2 N1(C(c2nnn(CC)c2C)=O)CCN(C(c2csc(Cl)n2)=O)CC1CC(C)(C)C C1(C)(C(=O)NCCCNC(c2c(OCC(C)C)nccc2)=O)CCCC1(F)F C(=O)(C(C)Cc1ccncc1)NC1C(NC(CCOCCC)=O)CC1 CC1CCC(C(N)=O)CN1C(C1(C)CCCN1C(=O)CC1(C)CCC1)=O CCCC(C)CC(=O)N(CC(=O)NCC(C)OC)CCn1cc(C)cn1 c1(C(=O)NC2CC(F)(CNC(CC(C)C)=O)C2)cnn2c(=O)cc[nH]c12 C(C(C(C)(C)C)NC(=O)Cn1ccc(C(F)(F)F)n1)NC(C1C(C)C1)=O C(C)(C)(CCC(=O)N1CCC(n2cccn2)C1)NC(C1N(C)CC1)=O C1(CNC(C(n2ccc(C)n2)C)=O)CC2(CCC2)CN1C(=O)OC(C)(C)C N1(C(C=C(C)C(C)(C)C)=O)CCC(O)(CNC(=O)CCc2ccnc(Cl)c2)C1 C1(NC(=O)C(c2ccc(F)cn2)(F)F)CC12CCN(C(c1coc(Cl)n1)=O)CC2 c1(CNC2C(C(N3CCCC(OC)C3)=O)C2)cccc2ncnn12 c1(CC)ccoc1C(=O)NC(CNC(C1CC1(F)F)=O)C(C)C c1(C(=O)OC)ccc(NC2CC2C(=O)NCc2cccc(C(=O)OC)c2)cc1Cl C1(C(=O)NCc2cccnc2F)CCC2(CC2)N1C(c1csc(Cl)c1)=O CC1(C)CN(C(C2(OCC3CC3)CC2)=O)C(C)CO1.c1(C(=O)N)coc(Cl)c1 N1(C(c2c(CC)cco2)=O)CCC(C)CC1C(=O)NCC(C)(F)C(C)C N1(C(C(C)(C)SC)=O)CCCC(F)(CNC(c2cc(C)c(O)nn2)=O)C1 C#CC1(C(=O)NCCCC(O)CO)CCN(C(=O)C(C)CSC)C1 C1(CNC(C2C(C)N(C)CC2)=O)CC2(CCN(C(c3cncs3)=O)CC2)C1 N1(C(CC2C(C)(C)C2)=O)CC(C2CN(C(c3ccc(C(F)F)c(F)c3)=O)C2)C1 C1(NC(CCc2cn(C)nc2)=O)CCN(C(=O)CN2C(=O)CNC2=O)C12CCC2 C1(C#N)(C(N(CCCCN(C(C2N(C(C)=O)CCCC2)=O)C)C)=O)CCCOC1 N1(C(C(C)=C(C)C)=O)CCCCC1CC(=O)NCc1nn[nH]n1 c1(C(N2CC(C(=O)Nc3ccc(CC#N)cc3)C2)=O)cc(Cl)cc(Cl)n1 Cc1cc(C(=O)NC2(CNC(c3cc(C)n(C(F)F)n3)=O)CCC2)c(C)c(C)c1 c1(CC(=O)NC(C)CCCNC(c2c[nH]cc2Br)=O)noc2ccc(F)cc12 c1(C(=O)NCC2N(C)CCN(c3ncnc(Cl)c3F)C2)cc2cccnc2s1 N1(C(C(C)C2CCCO2)=O)CC2CC3CC2C1C3NC(c1cn[nH]c1)=O C1(CC=C)(C(N2CCOCC2C)=O)CCCN1C(=O)C(O)C=CC C1(C(N(C(C=C)C2CC2)C)=O)C2CCCC2CN1C(c1nccnc1N)=O CC1(C(=O)NCCNC(=O)Cc2csc(-c3ccc(Cl)s3)n2)CCC(=O)N1 C(=O)(C1=CC2CCC(C1)C2)NC(c1cccnc1)C(N1CC(C)CN(C)CC1)=O c1(CC)ocnc1C(=O)NC(C)C(=O)NCCN1CCC(C)C1 c1(CN(C(C(=O)N(C)CC2CCCO2)=O)CC(F)F)cccc(F)c1 C(C(O)CNC(=O)CCC1CCCO1)N(C(=O)C(C1CC1)C1CC1)C C1(C2CC2)(C(=O)NC2C3CCC(F)C23)CCC1.Cn1nccc1C1CC(=O)N1 c1(C(N2C(C(N3C(CCC)CCC3)=O)(CC)CCC2)=O)n[nH]c2c1COC2 C1(CNC(CC2CC(CC)C2)=O)CC12CCN(C(=O)COc1cncc(C)n1)CC2 N1(C(c2c(C)nncc2)=O)CCC2CN(C(c3oc(Br)nc3C)=O)CC12 N1(C(COCC=C)=O)C2CCC1(CNC(=O)Cc1c(C)cccc1C)CC2 c1(C(N2CC(NC(C(CCCC)C)=O)C(O)CC2)=O)ccc2nccnc2n1 N1(S(C)(=O)=O)CCCC1C(=O)NC1CCCC1NC(=O)CCCF c1(OC(C)C(=O)NCC=CCNC(=O)CC(C)n2cccn2)ccccc1C#N C1(CN(C)C)CC(O)CN1C(C1CCOCC1NC(c1cnn(CCO)c1)=O)=O C(C)(CCCCCC)NC(C1(CC=C)CN(C(c2cn(COC)nc2C)=O)C1)=O N1(C(c2c(C)nc[nH]2)=O)CCC2CC1CN(C(c1cnccc1Cl)=O)C2 Cc1cc(C(N2CCCC(CNC(=O)C(C(C)C)N3CCCC3=O)C2)=O)n(C)n1 c1(C(N(C(C(C)C)C)C)=O)occc1CNC(=O)CN(C1CCCC1)C C1(NC(C(C)(C)F)=O)CCN(c2cncc(Cl)n2)CCC1CO Cc1csc(C(=O)NCCC(Cc2ccccc2)NC(=O)Cc2nncn2C)c1 C1(C(N(CCCCCCCC)C)=O)CN(C(=O)COC(C)CC)CC12CCC2 C(=O)(C1=NOC(C)C1C)N1CC(C(=O)Nc2cnn(CC)c2C)(CC)C1 CC1CCC(C(=O)NCCC2CN(C(=O)C(C3CCCCC3)N(C)C)C2)O1 N1(C(C2C(C)CC(=O)NC2)=O)Cc2[nH]nc(C(=O)NCCCC3CC3C)c2C1 N1(C(=O)Nc2c(C(C)C)ocn2)CCOCC1CNC(=O)C(Cl)(Cl)Cl CC1CC(NC(C2CCC(F)CC2)=O)CN1C(C1CC(=O)N(c2cn[nH]c2)C1)=O C(=O)(C(CC1CCCC1)NC(=O)C(C)OCOC)NCCCC c1(C(N2CC(C(=O)OC(C)(C)C)C2)=O)ccccc1Cc1csc(Cl)n1 C1(CCNC(CSSC)=O)CN(c2cc(C)nc(COC)n2)CCS1(=O)=O C(CCCCCCNC(=O)Cc1ccsc1C)n1cc(CSC)nn1 N1(C(C(C)c2cncs2)=O)CC2(CNC(=O)CCCOC(C)(C)C)CC1CO2 C1(CC)CN(C(C2CN3CCC2C3)=O)CCO1 c1(N(C2CN(C(C3CCCN3C3CC3)=O)C2)C)ncnc2c(Br)nn(C)c12 C=CCC(C)(C)CC(=O)N1CCCC(C)(C)C1CNC(c1cc(=O)n(C)cn1)=O C(CC(C)C)(C(=O)NCC(C)C)N(C(COC)=O)C N1(C(c2scc(C)c2)=O)Cc2c([nH][nH]c2=NC(=O)c2ncccc2Br)C1(C)C N1(C(CCC)=O)C(C(=O)NC(C)C(=O)NC2CC2)C2CC(F)C1C2 N1(C(CC(CCCC)O)=O)CCC2(CCCN2C(=O)C(C)c2ccsn2)CC1 n1(C(C)(C)C)ccc(C(=O)N(C2CC2)CC2CC2NC(=O)CC2CCOCC2)c1 C1(NC(c2cc(CO)ccc2O)=O)CC2(CCN(C(C3C4CCCC34)=O)CC2)C1 CC1ON=C(C(=O)N2CCN(C(C3(Br)CC3)=O)CC2c2ccccc2)C1C Cn1ncc(Cl)c1CC(=O)NC1CCC(CNC(=O)C(O)CN(C)C)CC1 C1(NC(C(C#C)(C)C)=O)CCN(C(=O)CCN(CC(F)(F)F)C)CC1(C)C Cc1ncc(Cl)c(C(=O)NC(C)CC(C)NC(=O)COCCc2ccccc2)n1 N1(CC(=O)NCCCC)CCCC(CC)C1.C(=O)(C(C)OCC)NCCN C#Cc1ccc(C)c(NC(c2ccc(CNC(c3ccc(NC)s3)=O)cn2)=O)c1 CC(CCNC(=O)CCc1cccc(F)c1)CCNC(C1CC1(C)C(F)F)=O c1(OC)ccc(I)cc1NC(=O)NCCCc1nc(C2CC2)n[nH]1 CC(C(=O)N(C)CCN(C)C(C1CC(CN=[N+]=[N-])C1)=O)=CC(C)(C)C N1(C(c2ccn(COC)n2)=O)CC2CCC(C1)N2C(c1cncc(C2CC2)c1)=O CCC(CC)CC(=O)NC1CCC(NC(c2cccc(C3(O)COC3)c2)=O)CC1 Cc1ccc(O)c(CNC(C2(NC(=O)CCCNC(=O)C3CC3)CCOC2)=O)c1 CON=CC(=O)N1CCC(OCCNC(=O)C(C)=C2CC2)C1 c1(NC(C2C(C(C)NC(C(C)N(CC)CC)=O)C2)=O)cc(C)cc(Cl)c1 N1(C(COCc2c(C)cccc2)=O)CCC(NC(=O)CN=S(C)(C)=O)C(C)C1 Cc1cc(C)c(C(N2CCN(C(=O)C(C)C(O)C(C)C)C(C3CC3)C2)=O)cc1N C12(C(=O)NCCCC(c3ccccc3)NC(c3ncc[nH]3)=O)CCCC1C2(F)F C1(NC(c2cc(C3CC3)no2)=O)CC2CCC1CN(C(C1CSCCS1)=O)C2 C(C)(CC(=O)NC1CCCC1CC(=O)N(CC(C)C)C(C)C)SC C(CCC[Si](C)(C)C)N(C(=O)C(C)(C)Nc1cccc(F)c1)C C1(C(=O)NCC2C(CNC(=O)CCC3OCCO3)C2)CC2C=CC1C21CC1 C1(NC(C=CC(C)(C)C)=O)CN(C(=O)Cc2cccc(O)c2F)CC2(CCC2)C1 N1(C(C2CC(OC)(OC)C2)=O)CCC(CC(=O)N(CC(F)(F)Cl)C)CC1 N1(CC(=O)NCC(C)(C2CCC2)NC(c2c(C)ncs2)=O)CCCCCC1=O c1(C(=O)NCC2N(C(C(C)=O)=O)C3C(C2)COC3)cnc2c(Cl)cccn12 Cn1nc2c(c1C(=O)NCC1C=CCN1C(=O)CC1CCOC1)CSCC2 c1(N(CC(Cl)Cl)C)cc(Br)ccc1S(=O)(=O)NC1CCOC(c2cnn(C)c2)C1 c1(C(=O)NC2C3CCN(C(C=Cc4n(C)ncc4)=O)C3C2)cnc2c(c1)COC2 c1(C(=O)NC2CCC(C)(CNC(C3(COC)CCC3)=O)C2)cccc2[nH]ncc12 C(=O)(CCCCN=[N+]=[N-])N1CC2C(CC(=O)NC(c3nc[nH]n3)CC)(CC2)C1 c1(C(N(C2CCN(C(c3ccn(C)n3)=O)C2)C)=O)nccc2ncccc12 C(F)(C(=O)NCCN(CC(=O)NCC(F)C1CCC1)CC)=CC Cc1cccc(CCC(N2CCOC(CCNC(C3CC4CC4C3)=O)C2)=O)c1 N1(C2CCN(C(=O)Nc3ccc(-n4c(C)ncc4)nc3)CC2)CC(C)CS1(=O)=O C1(CNC(C(c2c(C)cccc2)C)=O)CN(C(c2nocc2C)=O)CC1(C)C C1(C(=O)NC(C2CN(C(=O)CC(C)(C)O)C2)C)CCC2(CC1)CC2 n1(NC(CN(C2CNC(C(=O)O)C2)C)=O)c(-c2cscn2)nc2ccccc12 N1(C(c2c(C)cn(C)n2)=O)CCC(NC(=O)C(C#N)=CC(C)C)C(C)C1 N1(C(C(C)NC(=O)NC)=O)CC2CC1CCC2NC(=O)Cc1ccon1 C1(C(=O)NCC(CSC)OC)CCCN(C(=O)C(C2CCCCC2)=O)C1 c1(N(C(=O)CCC=CBr)C(C2CN(C(C)=O)C2)C2CC2)ccccc1[N+](=O)[O-] C1(C(C)(C)C)CC(CNC(=O)C(=O)C=CCN=[N+]=[N-])CCO1 c1(C(N2CCC(CCOC)C2)C(=O)NCC2CC2)cccc2c1COCC2 c1(CC(=O)NC(C(=O)N(C(C)CNC(C)=O)CC)C)csc(COC)n1 c1(C(N2CCCC(C)(C(C3CC3)NC(C)=O)C2)=O)ccc(C(F)(F)F)nc1N N1(C(C(C)OCCCC)=O)CCC(NC(c2sc(N(C)C)nc2Cl)=O)C12CCC2 C(CC(F)CN=[N+]=[N-])NC(C(CC=CC)NC(C1CCCCN1C)=O)=O C1(C(=O)NCC(CCCC)NC(c2nc(Cl)c(Cl)s2)=O)CCOC2(CCCC2)C1 C1(C)(CNC(CCCC=C)=O)CN(C(=O)C=Cc2cncs2)CCO1 C(=O)(CC(C)NC(c1cnn(CCNC(c2cc(C3CC3)on2)=O)c1)=O)NCC C1(C(N2CCC(N(C(=O)CC3CC(C)(C)C3)CC)C2)=O)CC(=O)OC1(C)C N(C1CS(=O)(=O)c2ccccc21)Cc1nc(-c2ccc(SC)s2)sc1 C1(C(=O)NCc2ccc(C)cn2)N(C(=O)Cc2c(C)noc2C)CCC1(C)C C=CC1COCC1NC(=O)C(C(C)C)NC(C1C2CCCCC12)=O C(C(C)(C)CC(=O)N1CCCCC1CCNC(=O)CCCc1ccsc1)N(C)C C=C(C)CC(=O)NCC(CC)N(C)C(C1CCCC1)=O N1(NC(c2ccc(Cc3ccccc3)[nH]2)=O)CCCC(NC(c2ccsc2)=O)C1 N1(C(CC(C)(C)OC)=O)CC(C)N(C(=O)CC2(n3cccn3)CC2)CC1C C1(N(C(c2ccc(C)n2C)=O)C)CN(C(=O)C(O)C2CCCC2)CC1(C)C CC(C(O)C(F)F)NC(=O)C=CC1CCCN1C(c1ncccc1N)=O c1(C(=O)NC2CC(C(=O)OC)C2)ccc(C)cc1.c12ccc(cc1)NC2 C1(C2CCN(C(C3CSCN3C)=O)C2)(NC(c2ccc(OCC)c(C)c2)=O)CC1 C1(N(C(COCC(=C)C)=O)CCOC)CCCN(C(C2(n3cccn3)CC2)=O)C1 C1(C(=O)NC(CC)(C)CNC(=O)Cn2ncnn2)CNC(=O)C(C)(C)C1 n1(-c2ccc(C(=O)NC(C)C(c3ccccc3)C)s2)nnc2ccccc12 C(=O)(C1CCc2cccnc21)N(C)CC1(O)CN(C(C2CC(F)C2)=O)C1 CS(=O)c1cc(C(N2CC(O)(C3(CNC(C4CC4(F)F)=O)CC3)C2)=O)cc(N)c1 C1(C(=O)NCC2(O)CN(C(C3CC4CCCC34)=O)C2)(COC)CCOCC1 Cc1cc(C(N2CCC(NC(C3CC(C)(C)C3)=O)C2C(C)(C)C)=O)ncc1C#N N1(C(C(C)NC(=O)NC)=O)CCC(NC(C2(C)CC3CCC2C3)=O)C(F)C1 CC(C)(CC(=O)O)NC(c1ccc(C(F)(F)CN)cc1)=O CC(C(=O)NCCCCC(C)NC(C1CCC2(CCC2)O1)=O)S(C)(=O)=O CN1CCN(C(C2(C)CCCO2)=O)CC1C(=O)NC1CCCC1C#N N1(Cc2n(C)cnc2)CC(=O)N(CC2(c3cnn(C)c3)CC2)C1=O C(CCCN=c1nc2c(ncn2C(C)C)c(N2CCC(C(N)=O)CC2)[nH]1)OCC C(=O)(C1CCCc2nc[nH]c21)NCC#CCNC(C1=NOC(C)C1)=O C1(NC(=O)C2=COCCC2)CCOC2(CCN(C(C34CCC(C3)C4)=O)CC2)C1 C(C(C)(O)CC(=O)N1CCN(CC(=O)Nc2c(C)cccc2O)CC1)OC c1(C(N2CC(C)(C)C(CNC(c3cncs3)=O)C2)=O)ccc2cncn2c1 N1(C(c2ccc(=N)[nH]n2)=O)CCC2CCN(C(C3CCCCCCC3)=O)C2C1 N1(C(CCC=CCC=C)=O)CC2CC2(NC(=O)CSc2ccccc2Cl)C1 C=CCCC(C(=O)NCCCCCN=[N+]=[N-])NC(=O)C(C)NC(C)(C)CC N1(C(c2csc(C)c2C)=O)CC(C)CCC1CNC(c1ccc(C(N)=O)s1)=O CC1(C)C2CC(C(N3CCCC3(C)Cc3ccccc3Cl)=O)CC12 C1(C(=O)N(C)CC2CCCCN2C(=O)CSCCC(C)C)(CC)CCC(O)CC1 c1(C(N2CCC(=CCNC(C(C)SCCCC)=O)CC2)=O)coc2c1CCCC2 N1(C(CC(CC)C)=O)CCC2(CCCCC2NC(=O)Cc2csc(S)n2)CC1 ClC(Cl)CN=c1[nH]c(=NCC2CCCCO2)[nH]c2c1COC2 C(CC(C(=O)NC(C)C(=O)NC1CCC(CCOC)CC1)OC)OC c1(C(N2CCN(Cc3cccc(OC)c3)CC2)C(=O)NCCC)cccnc1C C1(C(=O)NCC(C)N(CC(N2CCCC2)=O)C)N(C(=O)OC(C)(C)C)CCC1(C)C c1(C(=O)NCC(CNC(=O)CCC2CCCC2)OC)c(Cl)sc(C)c1C C(C(=O)NCC(F)CNC(=O)CSC(F)F)(C(C)C)OCC(C)C Cc1noc(C)c1C(C)C(N1CCC(Cn2cc(Cn3ccsc3=O)nn2)CC1)=O O=C1OCC2CCN(C(c3cc(C4CCCN4)[nH]n3)=O)C12 c1(C(N2CC(CO)C(CO)C2)C(=O)NCCCCCC)cn2cc(F)ccc2n1 c1(NC(C(CCCOC)NC(C2OCCC2(C)C)=O)=O)cnc2ccnn2c1 C12(NC(c3n(C)nnc3)=O)CCOCC1CN(C(c1cc3scnc3[nH]1)=O)C2 CCCCC(=O)C(=O)NC1CCC(NC(=O)COc2cc(C)ccc2F)C1 CC1CN(C(c2ccoc2)=O)CCC1CNC(C1(CC#N)COC1)=O C(=O)(C(C)(C)N=[N+]=[N-])NCC(CC(=O)N(CC(Cl)Cl)C)O c1(SCC)cnc(C(=O)NC(C(=O)NC2CC3(CSC3)C2)c2ccco2)nc1 c1(NC(N2CCC(C3(C(F)(F)F)CC3)CC2)=O)cc(-c2cccc(F)c2)ccn1 C1(C(N(CC(COCC)O)C)=O)CN(C)CCN1C(c1cnc(O)c(C)c1)=O C1(OC)CCCC(NC(=O)CC2(OC)CN(C(=O)Cn3ccnc3C)C2)CC1 C1(C(N(CCC)CCNC(=O)CC2CCCCC2O)=O)Cc2nccn2C1 N1(C(C(CCCC)O)=O)CC2CCC1C1CN(C(=O)Cc3cc(Cl)n(C)n3)CC21 c1(C(N2CCC(CNC(C3CCC(CC)C3)=O)C2)=O)ccc(NS(C)(=O)=O)nc1 C(C(C(C)(C)C)NC(=O)C(C)(C)N(C)C)NC(c1ccc(C(C)=O)o1)=O N1(C(C=Cc2n(C)ncc2)=O)CCC2CN(C(c3nocc3Cl)=O)CCC2C1 c1(C(N2CC(C)C(NC(c3cccc4nonc34)=O)C2)=O)cc2ccncc2s1 c1(C(=O)NCC=CC(=O)OC)cc2cccc(N)c2cn1 N1(C(c2c(C)ccnc2)=O)CCN2CCN(C(c3ccsc3C(F)F)=O)CC2C1 N1(C(c2cc(SC)oc2)=O)C(C(N2CC(C)(N(C)C)C2)=O)CCC1C1CC1 N1(C(C2(C(CC)=O)CC2)=O)CC2(C)CC1(C(N1CC3CC3C1CO)=O)C2 C=C(Cl)CCC(=O)NCCN(C)C(C1CCN(c2ccc(Cl)cc2)C1=O)=O N1(C(Cc2nc(CC)sc2)=O)CCOCC1CN(C)C(C1(C)CCCOC1)=O N1(C(c2ccc(C#C)o2)=O)CCC(NC(=O)C2=CCCCC2C)C(CO)CC1 C(=O)(C1=CCOCC1)N(CCN(C(c1cnc(C(C)C)nc1)=O)CC)CC N1(C(CC(C=C)c2ccccc2)=O)CCN(C(=O)Cc2ccc(Cl)cn2)C(C)C1 N1(C(c2c(CC)noc2)=O)CCC(C)C1CNC(C1(NC(C)=O)CCC1)=O C(CC(C(=O)N1CCC(n2cnnn2)C1)N(C)C(c1ccccc1)=O)SC C1(C(=O)NC2CN(C(C(C)C3CC3)=O)CC2F)CC(S(C)(=O)=O)C1 N1(CC)C(C)CN(C(=O)CC(C)NC(c2n[nH]cc2[N+](=O)[O-])=O)CC1C c1(C(=O)NC2C(CNC(CCSC)=O)CC2)ccc(C2(F)CC2(F)F)cc1 CC1(C)C2CCC1(NC(=O)C=C1CN(C(=O)OC3CC(OC(C)(C)C)C3)C1)CC2 c1(C(N2CC(CNC(CCOCCCOC)=O)C2)=O)noc2cc(Cl)ccc12 CC1(C)CC2(CC(C(=O)NC3CCN(C(C4CC5CCCC(C4)C5)=O)C3)C2)C1 Cc1ccccc1C1(NC(C2CC(c3cccc(Cl)c3)(O)C2)=O)CCC1 C1(NC(c2cc(C(C)C)on2)=O)CN(C(=O)CC2(N(C)C)COC2)CC(C)(C)C1 C(=O)(CC(O)CC(C)(C)C)NC1COCCN(C(C=Cc2occ(C)n2)=O)C1 c1(C(=O)NCCCN(C(C)C)C(C2CCCCC2F)=O)ccc(F)cc1C(F)F CC(CF)N=c1ccn2ncc(S(=O)(=O)N3CCOC(C)CC3)c2[nH]1 CS(=O)(=O)c1ccccc1CC(N1CCCCC1CNC(=O)CCCCCF)=O Cc1cncc(C)c1C(=O)NC1C2CN(C(C3CCCN3C=O)=O)CC12 C1(O)(CCNC(C2(CCOC)CCC2)=O)CN(C(=O)C(C)C2CCC2)C1 N1(C(C2C(C3C(C)C3)C2)=O)CCN(C(=O)C(C)O)CC(C)(C)C1 c1(C(=O)NCC2CC(=O)N(C)C2c2cccc(Cl)c2)ccc2c(c1O)CCCC2 c1(C(=O)NC2C(C)N(C(c3ccc(C(C)(C)C)nc3)=O)CC2)ccc(F)cc1F C1(NC(CP(C)(C)=O)=O)CN(C(=O)C=Cc2ccccc2F)CCC1CO c1(C(=O)NC(CCN(C(CC(C=C)CC)=O)C)C)ccn2cc(C)nc2c1 Cn1ncc(C(N2CC=CC2C(N2CC(CO)C3(CC3)C2)=O)=O)c1C#N Cc1cccc(Cl)c1C(N1CC(NC(c2cncc(Cl)c2)=O)C(C)(C)C1)=O c1(C(N2CC(NC(CCC)=O)CC2(C)C)=O)ccc(Br)c2c1OCCC2 c1(C(=O)NCCOCCNC(c2cc(C)on2)=O)nc(Cl)c(Cl)s1 C1(NC(CCOCCN(C)C(C2CCS(=O)CC2)=O)=O)CCCC(O)C1O C(CC(O)C(=O)NC(C1CCOC1)C)NC(Cc1cnc(C)s1)=O C(N=C(NCC1CCCO1)NC1CCOc2ccccc21)c1cc(C)nn1C c1(C(N2CCC(C(N3CCC(CCOC)C3)=O)(CF)C2)=O)cccn(C)c1=O c1(CN(C)C(C2CCN(C(=O)C(N)CC(N)=O)CC2)=O)ccc(F)c(Br)c1 C1(CNC(N(c2ccc(Cl)cc2)C(C)C)=O)CCCC(C)CC1 N1(C(=O)OC)CCC(N=c2[nH]c(N(C)Cc3c[nH]nc3C)nc3c2COC3)C1 C(=O)(C#CC1CCOC1)N1CCC(CC(=O)NC(c2nncn2C)C)CC1 C(CC(=O)NC1(CC(C)C)CC1)N(C(CSCCOC)=O)C(C)C C1(F)(C(=O)OCC(=O)Nc2n(C)cnn2)CCS(=O)(=O)C1 N1(C(c2c(C)nc(C)s2)=O)CC(C)CN(C(C2CC3C=CC2C3)=O)C(C)C1 CC1=C(CNC2CS(=O)(=O)CC23CCC3)C(C)N2NC=NC2=N1 c1(CC(N2CCC(=Cc3cccs3)CC2)=O)ccc(Cl)c(C(F)(F)F)c1 c1(C(=O)NC(C)CCN(C(=O)CNC(c2cccs2)=O)C)cccc2c1CCN2 N1(C(C(C(CC)C)O)=O)CCC2CN(C(c3cc(C(N)=O)co3)=O)CC2C1 CC1(C)CCN(C(C2CCOC2(C)C)=O)C1C(=O)NCc1ncc[nH]c1=O CCCN=C(NCc1cc(C)on1)NCc1cc(C2CC2)on1 CC(C)CC(C(=O)NCC1CCC1CO)ONC(C1(C)CCC(=O)C1)=O c1(C(=O)NCc2cccc(CNC(C(C)=CC)=O)c2)ccc2nc(Cl)nn2c1 N1(C(c2ncc(C3CC3)cn2)=O)CC2CC(C(N3CCCC3)=O)(C2)C1 N1(C(CCN(CC)CC)=O)CC2(CC(NC(c3ccccc3C#N)=O)C2)C1 C1(n2cnnn2)(C(=O)NCC(CO)NC(=O)C(C2CCCCC2)O)CCOCC1 C(=O)(C(O)CC(F)(F)F)NCC(CC)NC(c1cc2sc(C(=O)OC)cc2[nH]1)=O C=C1CN2C(=O)CCC2(C(=O)Nc2cccc(NC(=O)C(C)c3cccs3)c2)C1 C(=O)(C(CC(F)F)N(C)C(c1coc(C(F)F)c1)=O)NCC(COCC)C Cc1csc(C(N2CCCC(C(=O)Nc3cn(C)nc3C)C2)=O)c1C c1(C(=O)NC2CCN(c3cccc(C)c3)C2=O)cc(C)c(Br)c(C)c1 N1(C(C(C)OC2CCOC2)=O)CCCCCC1CNC(C1CC12CC2)=O N1(C(C2(C)ON=C(C)C2)=O)CCCC2(C1)CN(C(C1OC(C)CC1C)=O)CCO2 N1(C(c2scc(C)c2)=O)CCC(C2CCN(C(=O)C=C3CCC(C)(C)CC3)C2)C1 N1(C(C=Cc2ccc(C)o2)=O)CCC2(CC1)CCN(C(=O)C(C)CS(C)(=O)=O)C2 C1(CNC(CC=CC=C)=O)CN(C(=O)CC(c2ccc(F)c(F)c2)C)CCN1C c1(C(=O)NCCC(C)NC(c2cc(-c3cnn(C)c3)no2)=O)cn2c(n1)SCC2 c1(C(N2CC(C)(NC(=O)CC3(C)CCS(=O)(=O)N3)C2)=O)cc(Cl)c(F)cc1O C1(C(N(C)CC2CC2(C)C)=O)N(C(c2cnn[nH]2)=O)CCC1(C)C CC1CCn2cc(C(N3CCCC(CN(C)Cc4cccc(Cl)n4)C3)=O)nc2C1 C#CCC(C(=O)NCC(C)(C)CC1CC1)NC(=O)C(C(C)C)C1CCC1 C1(CC(N2C3CN(C(c4n(C)ncc4)=O)C(C3)C2)=O)Cc2cccc(Cl)c2O1 C(C(=O)NCCCC1CCCN1C(=O)CCn1ccnc1)(C(C)C)OCC(C)C N1(C(C(CCC)C(C)C)=O)CCC2CCN(C(c3nn[nH]c3Cl)=O)CC12 c1(C(N2CCN(CC(F)(F)F)CC2)=O)n[nH]c2c1CN(C(C1CC1F)=O)CC2 Cc1c(F)ccc(C(=O)N(C)CCNC(=O)C(C)C(C)(C)C)c1C c1(NCC(CCCC)NC(C2CCN(C)C2=O)=O)nc(Cl)nc2[nH]cnc12 c1(C(N(CCC(=O)NCCN=[N+]=[N-])C2CC2)=O)cn2c(n1)CCC2 Cc1ccnc2nc(C(N3CCC(O)(CCNC(=O)C4=CCOCC4)C3)=O)nn12 Cc1ccc(CO)cc1CC(N1CCN(C(=O)C(O)C(C)C)CC1C(F)F)=O Cc1cc(C2CC2)ccc1C(=O)NC1CC1NC(C1CN2CCC1CC2)=O N1(S(CCOCC)(=O)=O)CCCCC(C(C)OC)CC1 C1(C(N2CC(CNC(CC(C=C)(C)C)=O)C3C2C3)=O)Cc2cncn2C(=O)N1 CCC(CC)CC(F)C(=O)N1CC(NC(c2cncnc2)=O)CC(F)C1 c1(C(=O)NC(C(C)C)CNC(=O)CCNC(N)=O)c(Cl)cc([N+](=O)[O-])cc1Cl C1(NC(C(CCSC)O)=O)CCN(C(c2cc(O)cc(O)n2)=O)C(C)C1 C(=O)(C(C)CC1CCCCC1)NCC(C)NC(c1cnn(-c2ccccc2)n1)=O C1(C(=O)NC2CCCN(C(c3csc(C)c3C)=O)C2)SC2C=CC1CC2 C1(C(NOCCC(C)C)=O)CCCN(C(=O)Cn2cnnc2O)C1 Cc1cc(F)ccc1NC(=O)C(CC(C)C)ONC(c1ccc(F)s1)=O CCC(C(=O)OC)C(=O)N1CSCC1C(=O)NC1(C)CCC(C)(C)C1 C12(CNC(c3c(C)noc3)=O)CCCCC1N(C(c1ccn(C(F)F)n1)=O)CC2 N1(C(C(C)(CO)NC(C)=O)=O)C2CCC1C1CC1(NC(c1cc[n+]([O-])cc1)=O)C2 C1(C(=O)OCC)(CC)CCCN(C(CC2CCOCC2)C(=O)NC(C)CC)C1 C(CCCC(CO)NC(=O)C(COC)CC)NC(CNS(NC)(=O)=O)=O c1(NCCCSC)ccc(-n2cc(C)c(O)n2)c(F)c1 c1(C(=O)NCC(CN(C)C(C2CCC(F)(F)C2)=O)O)cc2cccnc2nc1O CCC(C(=O)N1CCN(C)C(CNC(C2CNC(=O)O2)=O)C1)C(C)(C)CC c1(C(=O)NC(C2CCN(C(CC(=C)C)=O)CC2)C)ccc2nc(OCC)[nH]c2c1 c1(NC(C(N2CCN(C3CC3)CC2)CC)=O)c(Cl)nc2ccccn12 n1(CCNC(=O)CNc2ccc(Br)cc2)cccnc1=O N1(C(CCCOC)=O)CCN(C(c2ncc(C(F)F)s2)=O)C(C(C)(C)C)C1 c1(NC(CCOC)Cc2cccc(Br)c2)cc(C(N)=O)ccc1NC(C)=O N1(C(C(CNC(=O)OC)(C)C)=O)CC(C(=O)NCC(C)(C2CC2)OC)CC(C)(C)C1 CCCCCC(C)(C)C(=O)NCC1CN(C(=O)Cc2cc(F)ccc2Cl)CC1C C1(NC(C2CC3(CC(=O)N3)C2)=O)CCCC12CCN(C(c1ncccn1)=O)CC2 c1(-c2cn(CC(c3ccc(CCC=C)cc3)=O)nn2)cc(F)cc(Cl)c1 C(=O)(CC(C)C(C)(C)NC(c1cccc(O)c1F)=O)NCc1ccc(C)nc1O N1(CC)Cc2ccc(NC(C3CCNC3c3ccccc3)=O)cc2C1 C12(NC(C3CN(C)C3)=O)CCC1CN(C(c1ccc(NCC(N)=O)cc1)=O)C2 C(=O)(C(CNC(=O)C(C1CC1)SC)CC1CC1)NC(CCOC)(C)C C1(C(=O)NC2C(SC)COC2)CCCCCCN1C(=O)CCCc1ncco1 C1(C(=O)NCc2cn(CC)nn2)CN(C(=O)CC2CCCCN2C)C2(CCC2)C1 c1(COC(NOC2CCC(C)C2)=O)cc(O)nc(COc2cccc(CO)c2)n1 CCC(O)(C(=O)NCC1(C)CCN(C(c2cc(Cl)cs2)=O)C1)c1ccccc1 CCCCC(CNC(C1(CNC(C2CCOC2(C)C)=O)CCCO1)=O)CC C1(N(C(c2occ(C)c2)=O)C)CCC(NC(C2CC2c2ccsc2)=O)CC1 C(=O)(CC(C)(C)C)NCC(C)N(C(=O)CN(c1cnc(C2CCCO2)s1)C)CC c1(CC)ccc(C(=O)NC(CNC(c2cnn(C)c2C)=O)CC(C)C)c(Cl)c1 C(=O)(C(O)CCC(C)C)N1C(CNC(C(CC)N(CC)CC)=O)CC(OC)C1 c1(OC)cnc(N(Cc2c[nH]nc2C2CCCNC2)CC2CN(C)CCO2)nc1C C1(C)(COC)CC(NC(=O)C2CC2)CN1C(c1c[nH]cc(Cl)c1=O)=O C1(NC(=O)Cn2ccnc2)(N)CCC1.CC(C)CC1CC1C(=O)NCC Cc1c(Br)ccc(-c2noc(CSc3cccc(F)c3Br)n2)c1F O=S(=O)(c1ccc2[nH]c(=NC3C=CCCC3)sc2c1)NCCCn1nccn1 O=C(CC1OCc2cc(Cl)ccc21)NC1CCN(C(C2CSC2)=O)CC1O Cc1ccc(NCC(=O)NCC(O)CNC(=O)COC2CC2)c(C)c1 C12(NC(c3ncn(C)c3)=O)CCC(CC1)N(C(C1CCC3CCC(=O)N13)=O)C2 N1(C(=O)NCCCN2Cc3ccccc3C2)CC2CS(=O)(=O)CC(C1)O2 S(=O)(=O)(c1c[nH]c2ncncc12)NCC(C12OCCC(N)(C1)C2)N1CCOCC1 C#CC1(C(=O)NCC2CC(CC)C2)CCN(C(=O)C=C(C)CCC)C1 c1(-c2cn(C3CCN(C(C4CCS(=O)(=O)C4)=O)C3)nn2)ccc(F)nc1 C1(NC(c2n[nH]cc2F)=O)CN(C(c2cnn3c2CCC3)=O)CC12CCOCC2 N1(C(CS(CC)=O)=O)C2CCC1CN(C(=O)Cc1cnns1)C2 c1(C(C)OC)nc(C(=O)NCC2(OC)CN(C(c3conc3C)=O)C2)co1 CC1(CNC(C2CCC(OC(F)F)CC2)=O)CCCN(C(c2ncccn2)=O)C1 c1(C(C)NC(C2(CN)CC(O)C2)=O)c(C(=O)O)oc2ccccc12 Cc1ncc(C(=O)NC(C2CN(C(c3cc(C(C)C)on3)=O)C2)C)n1C CC1CN(C(c2cscc2C#N)=O)CCC1C(=O)NC1CC(N2CCC2)C1 S(=O)(=O)(c1ccc(Cl)c2nonc12)Nc1c(C(=O)NCc2ccc(Cl)cn2)scc1 C1(NC(C2CC3CC3C2)=O)CCC2CN(C(c3ccc4cnsc4c3)=O)CC2C1 c1(OC)ccc2cc(C(N3CC(C(N4CCCC5(COC5)C4)=O)C3)=O)ccc2c1 N1(C(C2(C(=O)OCC)CCC2)=O)CC2CCC2(CCNC(c2cscn2)=O)C1 N1(C(CCC)=O)CCC2(CCCC2NC(=O)Cc2ccc3c(c2)CCC3)CC1 c1(OC)cc(N2CCC(C)C(NC(C3CC(C)C3)=O)C2C)c(Cl)cc1[N+](=O)[O-] CC(C)C(C(=O)N(C(C)CCNC(C1CCCC1C(C)C)=O)C)n1cnnc1 C1(CNC(=O)CCc2ncccn2)CCC2(CCC2)CN1C(=O)C=CCF C(=O)(CC(C(F)F)n1ccnc1)NC(C)CNC(C1(c2ccnc(O)c2)CC1)=O Cn1ccc(=NC(=O)c2cnn(CCNC(=O)C(CO)C(F)(F)F)c2)[nH]1 C1(C(=O)NCC(C(C)(C)C)NC(=O)C(F)CC2CCCC2)CCc2c[nH]nc2C1 C1(CNC(c2c(C)coc2)=O)(NC(C2(F)C(C)(C)C2(C)C)=O)CCC(C)(C)CC1 N1(C(C)C(N2CCCCC2)=O)CCN(CC(c2ccc(F)cc2)O)CC1=O N1(C(=O)CSC2CCCCO2)CC2=C(C1)CN(C(C13CC(F)C1C3)=O)C2 C1(CNC(C=C(C)C)=O)C(C)CCN1C(C1CCCN(C)C1)=O c1(NC(C23CC(NC(COc4cccc(C)n4)=O)(C2)C3)=O)cnc(C)c(Br)c1 c1(CC)cc(Cl)ccc1C(N1CCCC1CCNC(c1cnnn1C)=O)=O C1(C)(OC)CC2CC1CC2NCC1CC2(C1)N=N2 N1(C(C2(NC(=O)CN3CC(C)(C)C3)C(C)CCC2)=O)CCCNC(=O)CC1 C1(CC)CCN(C(=O)CCC2CCC(NC(C3(OC)CC(C)(C)C3)=O)C2)CCO1 Cc1csc2nc(CC(=O)NCC3(O)CC(CNC(C4CC5CC5C4)=O)C3)cn12 c1(NC2C(C)C2)nc2c(c(=NCC3Cc4ccccc43)[nH]1)CCC2 C1(CNC(CNC(C)=O)=O)CN(C(=O)COc2cncc(Cl)n2)C2CCCC2O1 N1(c2nc(C)cc(OC)n2)CC(NC(=O)CC(C)(O)C2CC2)CC2(CCC2)C1 c1(SC2CC(c3n(CCCSC)nnn3)(NCC3CC3(Cl)Cl)C2)ccc(C)cc1 Cc1cc(C)c(CN2CCC(CNC(=O)CN(C)C(c3cccs3)=O)CC2)s1 C(=O)(CC1=NN(C)C(=O)C1)NC(CCC)CCCNC(=O)CCCN1CCCC1 N1(CC)CCOCC1C(=O)NCCCN(C(=O)C(n1ccnc1C)C)C(C)C C1(CNC(=O)COC2CCCCC2)C(C2CC2)CCN1C(=O)C(F)C1CCC1 c1(NC(C2C(C)CC(C)N2C(=O)OC(C)(C)C)=O)cn(C)c(=O)nc1O c1(C(=O)NCC2(F)CCC(NC(C3(C)ON=C(C)C3)=O)C2)cccc(N)c1O C1(NC(Cn2ncc(C#C)c2)=O)(CNC(=O)CNC(=O)NC)CCCCCC1 CC(C)CCC(O)C(=O)N1CCC2(CC2)CC1C(=O)NCC=C(Cl)Cl c1(C(=O)OC)cc(NC(=O)NC2(CO)CC(C)C2)c(C)s1 c1(C(N2CCC(CNC(C(CN(C)C)N(C)C)=O)C2)=O)c(F)cccc1F Cc1cc(C(N2CC(F)(C(=O)Nc3cccc(N4CCCC4)c3)C2)=O)cnc1O c1(C(=O)NCCCN(CCCNC(=O)COC2CC2)C)cnn2ccccc12 C#CCCCC(C)(c1nnnn1C)NC1(C)CN(C(N)=O)C1 Cc1conc1CC(=O)NCC#CCNC(c1c[nH]nc1F)=O c1(CC)nc(C)c(CCC(N2CC(CNC(C3(F)CC3)=O)CC2C)=O)c(O)n1 Cc1nnccc1C(=O)NC(C)C(C)C(=O)N(CC(C)C)CCO C1(C(N(CC=C)CCC)=O)CCCN(C(=O)CS(=O)CC)C1C c1(C(N2C(CNC(C(CCC)OC)=O)CC(O)C2)=O)sc2ccc(Cl)cc2c1C c1(C(N2C3CC(NC(C4CCNC4=O)=O)CC2CC3)=O)cc([N+](=O)[O-])ccc1O c1(C(=O)NCC(C)CNC(=O)CNC(=O)Cn2cncn2)cnc(N)c(CO)c1 N#Cc1cccc(C=CC(=O)NCc2ccc(Br)nc2)c1.C12CC1C(=O)N2 C=C(Cl)C(C)(C)C(=O)NC1CCC(NC(C2(F)CC=CC2)=O)C1 C=CCC(C)(CC)C(=O)NC1COCC1NC(C1(CCO)CC1)=O c1(C(=O)NCC(C)NC(=O)COC(F)F)ccnc(N2CCCC2)c1 c1(C(N(C)CC2CN(C(C3(C)CC=CC3)=O)CCO2)=O)cc(C(C)C)cnc1O CC(C)C(CCC(=O)N1CCCC(F)C1)NC(c1cc(C(N)=O)[nH]n1)=O c1(C(=O)NCC(CCOC)NC(c2[nH]c(C3CC3)nc2C)=O)ccc(C)nn1 C(CC(=O)N1CCCC1(C)C(=O)OC)(C(F)(F)F)NC(C1(CC#C)CCC1)=O N(C(=NCC(C)C)N1CN(C)C(=O)C1C)Cc1c(C)ccc(F)c1 c1(C(CNC(=O)COCC2CCCCO2)O)ccc(C(F)(F)F)cc1 O=C1CCN(C(c2nccc3cc(Cl)ccc23)=O)c2cc(Br)ccc2N1 CC(c1ccsc1)=CC(N1CCC1CNC(c1cn(C2CCC2O)nn1)=O)=O N1(CCCOCC)CC(=O)N(C2CCC(CCC(N)=O)CC2)C1=O c1(OC)cc(C(=O)NCC2CN(C(c3c[nH]c(C#N)c3)=O)C2)cnc1O C=CCCCC(=O)NC(C)CCCNC(=O)CCc1nncn1C c1(CC)cccc(F)c1C(N1CCC(C(F)(F)F)C(CNC(=O)C(C)O)C1)=O Cc1ccc(N)c(C)c1C(=O)N(CCCCN(C(=O)C(C)C(F)(F)F)C)C CC1=C(C)CC(C(=O)NC2CCCCN(C(=O)CN(C)C(=O)C3CC3)C2)CC1 c1(C(=O)NC(C(=O)NCc2c(OC)cccc2)CC2CC2)cc(F)cc(F)c1 c1(OCCC)cc(C(N2CCC(OC(C)C)CC2)=O)cc(C(C)C)c1 N1(C(C(C(C)C)NC(C)=O)=O)CC2CC(C1)N(C(=O)C(C)(C)OC(C)C)C2 CC(CC(F)F)C(=O)N1CCC(NC(=O)COc2ccccc2C(C)(C)C)C1C N1(C(CCC=CCC=C)=O)CC(NC(c2conc2C2CCCO2)=O)C(C)(C)C1 C1(NC(C2CCCC(C)(C)C2)=O)CCN(c2nc(Cl)c(C#N)s2)CC12CCC2 CCC(CC)(CO)C(=O)NCC1CCCCC1NC(c1nc(=O)n(C)[nH]1)=O N1(C(CNS(NC)(=O)=O)=O)CC23CCCCC2(C1)CN(C(C1(C#N)CC1C)=O)C3 c1(C(C)N(C(=O)C(F)CC2CCOC2)C)c(F)cccc1F c1(C(=O)NC(CN(C(c2cnn(CC)c2Br)=O)CC)C)cnc(NC)cn1 C1(C(N2CC(C)C(C)C2C)=O)(CC)CCN(C(=O)C=CC(=O)NC2CC2)CC1 c1(C(N2CCC(CC(=O)NC(C)C(F)(F)F)C2)=O)cc(Cl)nc(Cl)c1F c1(CC)[nH]nc(C(N2CCC(F)(CNC(=O)CCCC3CC3)C2)=O)c1Br C(N=c1nc2sccc2c(N2CCCCC(C)(F)C2)[nH]1)c1nn(C)c(Br)n1 C1(NC(C(C)OCCC#C)=O)CN(C(=O)CC2CS(=O)(=O)C2)CC1CC(C)(C)C C(=O)(C(C(C)(C)C)NC(=O)CC(C1CC1)C1CC1)NCC1(CO)C(C=C)C1 N1(C(CC2(C(=O)OC)CCOCC2)=O)CCCC(CNC(c2ccns2)=O)CC1 C1(NC(=O)NCC(C)S(C)=O)CCCC1P(C)(C)=O CC1CN(C(C2C3CC4C(C3)C24)=O)CC2(CCN(c3nccnc3F)C2)O1 C1(CCC)CN(C(=O)C(C)CC(=O)OC)CCN1C(c1cccc(C)c1F)=O c1(C(=O)NCC(C)CN(c2ccnc(-c3ccccc3)n2)C)ccc(F)nc1 N1(C(CNC(C(C)(C)C)=O)=O)CCC2(CCC(NC(=O)C(C)(C)S(C)(=O)=O)C2)C1 C=CCCC(O)CNC(C1CC1C(C)NC(c1c[nH]nc1C(C)C)=O)=O C1(NC(CCN(S(C)(=O)=O)C)=O)COCCN(C(c2cncnc2)=O)C1 CC1(C)CCN(C(=O)CCNC=O)C1CC(N1CCCC(O)(C(N)=O)C1)=O CC(C)C(CNC(C1CN(C(C)C)C1)=O)C(=O)NCCCN1CCCC1C c1(NCC(C)C(F)(F)F)ccc(S(=O)(=O)NC2CN(C)CC2(C)C)cc1C#N C1(CNC(C=C(C)C)=O)CN(C(=O)Cc2c(C)noc2Cl)CC1(C)C C12(CNC(C(CC)C3CCC(=O)N3)=O)CC(CN1C(=O)C(C)(C)COC)C2 CC12CC3CC(CC(C(N4CCCC(O)(CNC(C5CC5F)=O)CC4)=O)(C3)C1)C2 c1(C(N2C3C(NC(C(C)NC(N)=O)=O)CC(C3)C2)=O)ccc([N+](=O)[O-])cc1N c1(C(=O)NC(CCCNC(C(C)NC(CC)=O)=O)CO)c(C)cccc1Cl N1(C(c2cc(C)oc2)=O)CCCN(C(=O)CC2CCC3(CCC3)O2)CC1C(C)C Cc1cnc2n1CCCC2C(=O)N(C)CC1(O)CCN(C(=O)CSC2CC2)C1 CC(CC(C)NC(=O)C=CCN1CCOCC1)NC(c1ccc(C(F)(F)F)o1)=O c1(CN2CCC(N(C)C)(C(N)=O)CC2)c(C(=O)O)oc2ccccc12 c1(C(=O)OC)c(C)[nH]c(C(N2CC(NC(c3ncc(C)cn3)=O)C2)=O)c1C C1(CCOC)(C(N2CCC(CNC(c3cnsn3)=O)C2)=O)CCCC1 N1(C(C=COCCNC)=O)CCC2CC1CN(C(c1csc(C(=O)NC)n1)=O)C2 CP(C)(=O)CCC(=O)N1CCC(C(=O)Nc2ccc(C3CC3)nc2)C1 Cn1c(=O)[nH]c(NCCNC(=O)Cc2cncnc2)c(C#N)c1=O C1(C(N(C)Cc2ccc(CNC(C(C)(C)OCC)=O)cc2)=O)CC(=O)N(OC)C1 c1(NC2C3(C(C(=O)OCC)NCC3)C2)ccc2c(c1)CCCO2 C1(NC(c2n(C)nnc2)=O)CCC(CC(N2CCC3CC23C)=O)CC1 C1(CC)(CC)CC(NC(=O)C#CC(C)(C)C)CN1C(=O)C(F)N(C)C N1(C(C)C(=O)NC2COCC2CNC(c2cc(Cl)cs2)=O)CCCCC1=O C(CC(CC)C(=O)N1CCC(CO)(CNC(=O)CC2(C)CCCCC2)CC1)=CC Nc1ccc(C(=O)CCC(=O)N(CCc2nn[nH]n2)CC2CCCO2)cc1 Cc1noc(N)c1C(=O)NC1CCN(C(c2coc(-c3ccccc3)c2)=O)CC1 C(CC1CCCCC1)(C(=O)OC1CC(CC(N)=O)C1)NC(=O)OC(C)(C)C N1(C(C2(CC)CCCNC2)=O)CCNC(=O)CC1c1ccccc1 Cc1cccc(C(C)C(=O)NCC2CCCN(Cc3ccc(C4CC4)cc3)C2)c1 N1(C(c2cc(C(=O)OCC)c(C)[nH]2)=O)CC2(CCC(NC(C3(C)CC3)=O)CC2)C1 N1(C(C(C)OC)=O)CCN(C(=O)C(F)(F)CCn2ccnn2)CCC1C Cc1nc(C(=O)NC(C)CNC(c2coc(Cl)n2)=O)c(C(F)(F)F)[nH]1 c1(NCC(C)CCO)cc(Br)ccc1S(=O)(=O)NCCCCCF c1(C(=O)NCC2(C)CCCN(C(=O)CC3C=CCC3)C2)cc(C#N)ccc1O N1(C(C(CO)NC(N)=O)=O)CCN(C(c2ccc(F)cc2)=O)CC12CCC2 c1(CNC(C(CN(C(c2n(CC)ccc2)=O)C)C)=O)ccc(C)nc1 c1(C(=O)NCC2C(CNC(Cc3cn(CC)nn3)=O)C2)ccc2nn[nH]c2c1 C1(CC(=O)NCC2N(C(CC)=O)CCC2)SC(=N)NC1=O CC1(CNC(C2CC(=O)CCO2)=O)CCN(C(=O)CC(=O)NC2CC2)C1 c1(OCCCCC)cc(C)ccc1CNc1ccc(NC(=O)C2CC2)cn1 C1(CNC(C(C)Nc2scc(C)n2)=O)CCCN(C(C2(CC(C)C)CCC2)=O)C1 C12CCN(CC1C)C(=O)O2.c1(NCCOCCCC)ccsc1C c1(CC)ccc(C(=O)NC(C)C(CO)NC(C2(C(C)C)CCC2)=O)c(C)n1 c1(CNC(c2n(CCCOC)nnn2)C2CCCSC2)cn2cccc(F)c2n1 C#CCC(C(=O)N(C)Cc1ncco1)NC(c1csc(Cl)c1)=O Cc1nc2c(o1)CCN(C(=O)NCc1noc(C(N)=O)n1)C2 C1(CC=C)(C(=O)NC(C)CCCCO)CCN(C(c2cc(CC)sn2)=O)C1 c1(C(=O)NC2(CCNC(C(C)n3ccnn3)=O)CCC2)ccc(N)c(F)c1F N1(C(=O)C=C2CCCCC2)CCC2(C1)CN(C(=O)CCc1cccc(F)c1Cl)C2 c1(C(=O)NCCOC2CN(C(C(C(C)C)SC)=O)C2)nn(C)c2ccc(F)cc12 CCC(C)(CNC(c1ncoc1C1CC1)=O)NC(c1cc(C2CCC2)[nH]n1)=O C1(NC(c2cc(-c3cn(C)nc3)no2)=O)CCN(C(C2(C)CC=CC2)=O)CC1O C1(NC(C(N2CCOCC2)C)=O)CC2CC(C1)N(C(C1CC1C)=O)C2 C(=O)(C(C)CC(C)(C)C)NC(CCCC)C(N1CC2(CCC2)CC1C)=O c1(COC)nc(CC2CCCCC2)n(-c2ccccc2F)n1 C1(O)(C(CNC(C2(COC)CC=CC2)=O)C)CCN(C(c2csc(C)n2)=O)C1 C1(C)(CNC(C(C)Cc2cccnc2)=O)CCN(C(C2CCCCS2)=O)C1 S(=O)(=O)(c1cccc(C(=O)N(C)C)c1)N1C2C(N3CC(C)C4(C3)CNC4)CC(C2)C1 N1(c2c(C)cnc(C)n2)CC2CCC(NC(c3cccnc3F)=O)CC2C1 N1(C(C2CC(O)CN2)=O)CC2CC2(CNCc2cncs2)C1 N1(C(CCCC=C)=O)CC(NC(C2(C)CC2C(=O)OC)=O)CC12CCOCC2 C1(NC(C2(CCOC)CCN(C(=O)C(F)F)CC2)=O)CC2CCCCCC12 c1(CC(=O)NCCCC(C)NC(Cn2cc(C(=O)OC)nn2)=O)ccc(C)cc1F Cc1ccc(CNCC(=O)NC(=O)NC2CCCC2)nc1Br C1(CC(=O)NCCCN2C(C)CCC2)CCN(C(c2scnc2Cl)=O)C1(C)C CC(C)CC(C(=O)N1CCCCCC1C)NC(c1nnc(O)nc1O)=O Cc1ccc(C=CC(=O)NC(C)C(C)NC(c2ccc(Br)s2)=O)cc1C C(C1CCOCC1)=CC(=O)N(C)CC1CCCN1C(C1CCC1(F)F)=O c1(CCC(=O)NCC2(O)CN(C(C3C(C)CC3)=O)C2)ccc(Br)c(Cl)c1 C(CCCCc1ccccc1)NC(=O)NCC=C(C)C c1(C(=O)NC(CCN(C(C(CC)(C)O)=O)C)C)oc(P(C)(C)=O)cc1C N1(C(C(C)N(CC)CC)=O)CCOCC(NC(=O)C(C2CC(F)(F)C2)OC)C1 C1(C)(NC(C2CC(OC)C2)=O)CCCN(C(C2CC2C2CCC2)=O)C1 c1(C(=O)NC(C(C)NC(=O)C(c2ccccc2)F)CO)cc(Cl)ccc1O N1(C(C)=O)CCCC(C(=O)NC(CNC(=O)C=CSc2ccccc2)CO)C1 N1(C(C(C)N(C)C)=O)CC2CCN(C(C3CCOC3c3ccncc3)=O)CC12 c1(C(=O)NC(C(=O)N2C(COC)CC2)CCF)cc2occc2[nH]1 C1(COC)CC(CNC(c2csc(C)c2C)=O)N(C(=O)CCc2cncn2C)C1 c1(C(=O)NCC(C)CC2CC2)ccc(CNC(=O)CCOC2CC2)nc1 c1(C(N2CC3C(CNC(C(C)C(C)(C)C)=O)C3C2)=O)cccc2sncc12 C(CCCC(C)NC(C1(F)CCCCC1)=O)NC(c1c(C)scc1)=O O=C(C1=C(Cl)CC1)NC1CCOC(C(=O)NCCC#CCO)C1 c1(C(N2CC(CNC(C(C3(O)CCCCC3)CC)=O)C(C)C2)=O)ccn(O)c(=O)c1 C=C=C(C)CC(=O)NCC1CCCCC1C(=O)Nc1cncnc1O C#Cc1ccnc(C(=O)NC2CN(C(=O)CNS(=O)(=O)N(C)C)C(C)(C)C2)c1 C1(NC(c2[nH]cc(C#N)c2)=O)CCC2CCN(C(c3ccc4cncn4c3)=O)C12 C(CCC(C)(C)C(=O)N(C1CC(C(=O)Nc2cncc(C3CC3)c2)C1)C)OC c1(N2CC(COC)OC(C)(C)C2)nc(C)cc(=NC(C)c2ccc(Cl)c(F)c2)[nH]1 C1(N(C)C)CC(NC(C2(NC(C3COCC3C(N)=O)=O)CCCC2)=O)C1(C)C N1(C(C(=O)NC(c2ccncc2Cl)C)=O)CCC(C)C(N)C1 c1(C(N2CCC(F)(CNC(c3n(C)ccn3)=O)CC2)=O)ccc2ncncc2c1 c1(N(CCNOC)C(N2CCOC(C)C2)=O)nc(OC)c(F)c(Cl)n1 C1(C(=O)NCC(CC)NC(C2(CCC=C)CC2)=O)CCC(CN2CCOCC2)O1 N1(C(C(C)OCOC)=O)CCCN(CCNC(=O)CCc2cscn2)CC1 c1(SC)ccc(N2CC(C(=O)NC3CCN(C(=O)C=C4CCC4)C3)CC2=O)cc1 C1(C(N(C(C)CNC(=O)C(C)(C)n2cc(Br)cn2)C)=O)CC2CCC1C2 C12(NC(=O)CCc3cncc(F)c3)CCC(CC1)N(C(=O)C=Cc1cocn1)C2 N1(C(COC(CC)(C)C)=O)CC(CNC(=O)CC2CC3(CC3)CO2)C(O)C1 C(N=c1[nH]nc(C(N)=O)s1)C1C(C)CN(C(C2(C)CC2)=O)C1 c1(OC)cc(C(N2CC(C)(CC(=O)Nc3cc(F)cc(F)c3)C2)=O)ccc1I CCC(CC)C(C)C(=O)N1CC(CCNC(=O)CC23CCC(CC2)OC3)C(C)C1 C1(C)(C(=O)OCC)CCN(C(C)=O)CC1 C1(NC(=O)CSc2nnc(S)s2)CCCC(NC(=O)CN2CCCC2)C1 C1(C(=O)NC(C2CCOC2)CNC(=O)C(F)=CCCF)(NC(C)=O)CCCC1 C(=O)(C(CC(C)C)C(C)C)NCC1C(NC(C(C)N(C(C)=O)C)=O)C1 C(=O)(CCCCCCCCCO)N(C(C)CN(C(=O)C(Cl)=CCl)C)C c1(C(=O)NC2CN(C(C=CC=CCC)=O)CC2O)ccc2ccc(Cl)cc2n1 N1(C(c2c(OC(C)C)nccc2)=O)CCCN(C(=O)C(C)n2cncn2)CCC1 c1(C(C)C)ccc(F)cc1CN1CCNCC1NC(=O)NCCc1ccccc1 c1(C(=O)NC2C(C)CCN(C(CC(CCC)O)=O)C2)c(C)nc(O)nc1C C1(CNC(CCOC)=O)(NC(=O)CN(S(C)(=O)=O)C)CCCCC1C.C(C(C)C)N CCCC(C(=O)NC(CO)C(C)NC(c1ncn(-c2ccccc2)n1)=O)OC N1(C(c2cn(C(C)C)nc2)=O)CCC(C(=O)NCCn2ccnn2)C1C c1(C(N2CCC(N(CCO)C(C3(C4CCC4)CC3)=O)C2)=O)cc2c[nH]cnc-2n1 N1(C(c2c(CCC)nns2)=O)CCC2CN(C(C3CCSC3)=O)CC12 N1(C(=O)OC)C2CCC1CN(c1nnc(-c3n[nH]c(C)c3Cl)n1CC1CC1)C2 c1(C(=O)NC2C(NC(COC(C)C)=O)CCCC2)nn(C)c2c1CC(F)(F)CC2 N1(C(c2nnn3c2CCC3)=O)CC2CCN(C(C3CCCCC3)=O)CC2C1 c1(C(c2n(CCSC)nnn2)NCCc2nc(C)cs2)cncc2ccccc12 C1(CC)CCCC(N=c2[nH]c(=NCC3(C)CCN(C)CC3)[nH]c3c2SCC3)C1 C(=O)(C1=CCCOCC1)N1CC(C)(C)C(NC(=O)Cc2ccc(Br)s2)C1 Cc1nc2sccn2c1C(=O)NC1CC12CCN(C(=O)CC1CC1C1CC1)CC2 CCC(CC)(CO)C(=O)NCCC1CCCN(C(=O)C(F)C2CCOC2)C1 C1(C(=O)NCC(C2CCC2)NC(c2ccc(CO)o2)=O)CC2CCC1C2 c1(C(N2CCC(CCNC(c3nc(C4CC4)cs3)=O)C2)=O)ccc(O)cc1 C1(C(C)NS(=O)(=O)Cc2ccccc2)CC2(C1)CN(Cc1ccc(O)nc1)C2 Cc1ccc([N+](=O)[O-])c(-n2cc(CNC(c3ccccc3)C)nn2)c1 N1(C(C=CC)=O)CCCC2CN(c3ncc(C#N)cc3Cl)CCC12 N1(C(c2cc3cccnc3[nH]2)=O)CCC2CCN(C(C3(C(F)F)CC3)=O)CC12 C(=O)(CC1OCc2ccccc21)NCC(C)(C1CC1)NC(=O)C1=CCS(=O)(=O)C1 C#Cc1ccc(C(=O)NC2CN(C(c3ccc(SC)s3)=O)CCC2C)nc1 C1(C(=O)OCC)CCOC(C)(CC(=O)Nc2ccc(C(=O)OC)cc2)C1 N1(C(C2CC(C(C)C)C2)=O)CC2CC1CN2C(c1sccc1Cl)=O C1(CNC(C=COCC)=O)CCCC(NC(c2cc(Br)oc2C)=O)C1 c1(C(N(C(CCNC(C2CC(N(C)CC)C2)=O)C)C)=O)cccc2[nH]nc(O)c12 C1(C(=O)NC2(CCOC)CCC2)CCCN(C(C2CCNC2=O)=O)CC1 CC#CCCCC(=O)NCC1(OC)CCN(C(=O)CC(=O)OCC)C1 N1(C(C2CC(C)CN(C(=O)C3=CC(C)(C)C3)C2)=O)C2CCCC1COC2 C1(c2ccc(OC)cc2C)NC(=O)N(CCC2CC2)C2=C1C(=O)NCC2 N1(C(N(C)Cc2ccccc2)=O)CCC2CCNC(=O)C2C1 c1(-n2cc(C(=O)NCC(CCOC)OC)nn2)ccc(F)c(OC)c1 Cc1ccc(CNC(C2(F)CCC2)C)c(=O)n1C C1(CNC(c2c(C)ccn2C)=O)C(O)C(O)CN1C(c1cnc(CC(C)C)s1)=O c1(CNC(C2(C=C)CCC2)=O)nc2c(s1)CN(C(=O)Cc1ccsc1Cl)CC2 O=C(CCCC1CCCO1)NC(c1ccccc1)C(=O)NC1C=CCC1 C12(C(N3C(C4CCN(C(c5nncc(C)c5)=O)C4)CCC3)=O)CCC(F)(CC1)CC2 C1(C2CCOCC2)(C(N2C(CNC(C(C)c3cccs3)=O)CCC2)=O)CC1 N1(C(CCOC)=O)CC(C)N(C(C2CCCC(C)C2)=O)CC1C N1(C(C(C)(C)SC)=O)CC2(NC(c3cc(N)cnc3Cl)=O)CCC1CC2 CC(CC(=O)NC1CC(O)(CNC(c2cc(C(N)=O)co2)=O)C1)N1CCCC1=O C1(C)(C(N(C(C)(C)C)CC2CC(NC(NCCC)=NC)C2)=O)CCCCO1 CCC(CN(C)C)C(=O)NCCCC(=O)Nc1cnn(C(C)(C)C)c1 O=NN1CCCC1C(=O)NCC1CN(C(=O)CCc2cnc(C3CC3)o2)CCO1 N1(C(C2N(CC)CC2)=O)CC2CC1C2CNC(=O)CCC(C)N(C)C c1(C(=O)NCCN(C2CCCC2)C(C=CC(C)(C)C)=O)cc2sccc2n1C c1(C(C)C(=O)NCCOC2(C)CC2)ccccc1S(N)(=O)=O C1(CCC)(NC(c2cn(C)cc2C)=O)CCN(C(c2cnnn2CC)=O)CC1 C1(OC)CCN(C(=O)CSCCNC(=O)Cc2ccnc(O)c2)CC1C C1(CNC(C(C)(C)NC(=O)CCn2cccn2)=O)CCC2(CC2)C1 N1(C(CCOC)=O)CCC(COC)(NC(c2cnc(Cl)[nH]2)=O)C1 c1(C(N2CC3C(C(=O)NC4CC4)C3C2)=O)ccc(NC(C2CC(=O)N2)=O)cc1Cl CC1CCc2ncc(C(=O)NC3CC3CNC(=O)CCc3csc(=N)[nH]3)n2C1 c1(C(=O)O)coc2c1CN(C(C1CCC(Oc3ccncc3)C1)=O)C2 c1(C(N2C3CN(C(c4c(CC)nns4)=O)C(C3)C2)=O)nnc2ccccc2n1 C1(C)(C(=O)NCC2C(C)CN(C(c3cccc(O)n3)=O)CC2)CC2(C1)CC2(F)F n1(CC(=O)N(C)CC2N(C(C3C(C)=C3)=O)CCC2)ccc2c(N)cccc12 Cc1ncc(Br)c(C(=O)NCCCN2CCN(C(C3CCCCCC3)=O)CC2)n1 C1(NC(CCc2c(C)nccc2)=O)CC(CO)C12CCC2 c1(NC(N(CCC)Cc2ccccc2)=O)c(Cl)cc(Cl)nc1C c1(OC)cc(C(=O)NC2CC(C)N(C(c3ccc(C(C)(C)C)o3)=O)C2)nn1C C(=O)(CCCC(=O)NCC1CN(C)CCN1C(C1CC1[N+](=O)[O-])=O)OC c1(C(=O)OC)cc(NC(=O)CC2CCN(c3ncncc3Br)C2)cc(Br)c1 c1(SC)cc(C(=O)NCc2nc(CNC(=O)C(C)(F)F)cs2)c(C)o1 CCCC(C)(CC)C(=O)NCC1CCC1NC(c1c[nH]c(=N)c(C)c1)=O N1(C(C=CC(C)C)=O)CC(OC)C(NC(=O)CNC(=O)CCc2ccccc2)C1 C1(NC(CC2(OCC)CC2)=O)CC(c2ccccc2)(NC(=O)Cc2cc[nH]c2)C1 c1(C(N2CC(OC)C(NC(=O)C(F)C3CCC3)C2)=O)nnn2c1C(=O)NCC2 c1(CC(=O)NC(CNC(c2cnc(OCC)s2)=O)C2CCC2)cc(O)nc(O)n1 C(=O)(C(F)C(C)C)Nc1nnc(OCC)s1 C(C(=O)N(C)CCOCCNC(=O)CCC1CCCO1)(SC)SC C1(NC(c2c(C)cco2)=O)CN(C(=O)C2=C(Cl)CCOC2)C2(CCCCC2)C1 C1(C)(NC(CC2CC(=C)C2)=O)CCCCC1C(=O)NCc1ccnc(C(=O)OC)c1 N1(C(C(C(C)(C)O)F)=O)CCC2CC(NC(c3ccn(CCF)n3)=O)CCC2C1 N1(C(c2cn(COC)nc2)=O)CC2(C)CN(Cc3noc(C4CC4)n3)CC2(C)C1 c1(C(N(CC(C)(C)NC(CC2C(CC)C2)=O)C)=O)cc(Cl)c2n[nH]cc2c1 c1(C(=O)NC2(C)CN(C(c3cc(OC)cc(OC)c3)=O)C2)cc2sc(F)cc2[nH]1 CC(CC(=O)NC(C1CCN(C(c2scnc2C(C)(C)C)=O)CC1)C)P(C)(C)=O CCC(CC(C)C)C(=O)N1CCC(C2CCCN2C(=O)CC2(CO)CCC2)CC1 C12(CNC(CN(CC)CC)=O)CCCCC1N(C(=O)C(C)CCOC)CCC2 Cn1cnc(C=C(F)C(N2CCCC2CC2C(C)(C)C2(C)C)=O)c1 c1(CNC(C2CCCN(C(=O)Cc3cccs3)CC2)=O)cccc2occc12 C12(C3CNC(=O)N3)CCC(CC1)C2.Cc1cnn(CC2(O)CCSC2)c1 Cc1nn(CC(C)C)c(C)c1CN1CCN(C(=O)NC(C)(C)C)CC1C(F)F c1(C(N(C2CN(C(=O)C(C)(C)F)C2)C)=O)cc([N+](=O)[O-])ccc1Br CC1CC(C(=O)N2CCC(OCC(=O)NCCCC(F)F)C2)=NO1 CCCC(C)(O)CC(=O)N1CCOC(CN(C(=O)Cc2occc2C)C)C1 c1(C(C(=O)NC(C)C(=O)NC2CC2Cc2ccccc2)=O)cnn(C)c1 C12(C(N(CCCNC(c3ccc(COC)cc3)=O)CC)=O)CCC(O)(CC1)CC2 N1(C(=O)Cc2coc(C(F)F)n2)CC2CCN(C(=O)Cn3ncnn3)C2C1 Cc1nocc1C(=O)NC(C(=O)N1CC(c2nncs2)C1)C1CCCO1 C(=O)(CC(C)CC(C)C)NCC1(OC)CN(C(c2nnsc2N)=O)C1 c1(C(=O)NC2C(NC(c3cnn(CCC)c3C)=O)CCC2)ccc(C#N)cc1C c1(C(=O)NCCOC2CCN(C(C(C)(C3CC3)OC)=O)C2)cc2c[nH]nc2s1 C1(C(=O)NCC2CC(F)(CNC(CN3C(C)CCC3)=O)C2)CC(=O)OC1(C)C CC1CN(C(=O)CN(C)CCO)CCCN1C(c1ccc(OC(F)F)nc1)=O c1(OC)cc(C(=O)Nc2cccc(F)c2Cl)c(NCc2cc(Cl)cnc2C)cn1 N1(c2ccnc(NCCCc3c(OC)cccc3)n2)CC2(C1)CN(C)CCO2 CC1CC(C(=O)NC(C)(C)CF)CN(C(=O)Cc2ccnc(O)c2)C1 CC1(C)CCN(C(c2nc(Cl)cs2)=O)C1C(=O)NC1CCCC1N=[N+]=[N-] Cc1cccn2cc(C(=O)NCC(O)CN(C(=O)C(O)Cn3cncn3)C)nc12 Cn1cc(C=CC(=O)NC2(C)CC(NC(c3cn(CC(F)(F)F)cn3)=O)C2)cn1 N1(C(C2N(C(C)=O)CSC2)=O)CCCC(N(C)C(C2COCCO2)=O)C1 C(=O)(C(C(C)C)N(C)C)N1CC(C(C(=O)NCCCc2cncnc2)OC)C1 C=CC(C)(CC)C(=O)N1CC(CNC(C2CCC3(CC2)CC3)=O)C(F)(F)C1 C=CC(CCC)CC(=O)NCCN(C)C(c1c(F)cc(OC)cc1Cl)=O CC(O)(Cc1ccccc1)C(=O)NCCCN(C(=O)CN1CCOCC1)C1CC1 N1(C(c2cccc(SC)c2)=O)CCN(C(=O)C(C)(C)N(C)C)CC1CC(F)(F)F C1(OC)CN(C(=O)C(C)(CSC)NC(C2CC(SC)C2)=O)CC12CC2 Cc1cc(Cl)c(C)c(C(N2CC(CO)(NC(=O)CCC=CC(C)C)C2)=O)c1N CC1(C)CN(CC2CCNC(=O)O2)CC1c1cccc(C(F)(F)F)c1 c1(C(N2CCC(CN(C(C3(CCC=C)CC3)=O)C)C2)=O)ccc(Br)cc1 c1(NCc2cc(C)ncn2)nc[nH]c(=NCc2ccc(F)c3ccccc23)c1C Cc1cn2c(C(=O)NCC3CCN(C(C4CCCS(=O)(=O)C4)=O)C3)c(C)nc2s1 CC(=O)CCCC(C)C(=O)NCCC(=O)N(C)C(c1nccs1)C NS(=O)(=O)c1ccc(F)c(NC(=O)CCCc2cccc(Cl)n2)c1 C=C(Cl)CCC(=O)NC1CN(C(=O)C(C2CCCC2)OC)CC1n1cccn1 C(=O)(CCC(CF)CF)N1CC2C(C(N3C(C(C)C)CC(O)C3)=O)(C2)C1 C#Cc1ccccc1CNC(=O)CCC(CC)NC(C1(OC)CCSC1)=O NC12CCOCC1CN(C(=O)C(=O)NCC1(c3ncccc3F)CC1)C2 C1(C)(C(=O)NC(c2nc(CC)[nH]n2)C)CCN(C(=O)C(O)CSC)C1 N1(C(Cc2ccc(C)o2)=O)CC(CCNC(=O)CC2(C#N)CC2)OC(C)C1 C12(CNC(c3ccc(CC)cc3)=O)CC(NC(c3ncccc3Br)=O)(CCO1)C2 C1(NC(C2(N(C)C)CCC2)=O)C2CC1N(C(C1CC1c1cccc(Cl)c1)=O)C2 CCC(C)C(O)CC(=O)N1CCCC(C)(C(=O)NC2CCN(C)C2)C1 c1(C(=O)NCC2N(C(COCCC(C)C)=O)CCC(C)C2)nccc2n[nH]cc12 N1(C(C(C)=CC2CC2)=O)CCC(F)CC1C(=O)N(C1CC(C)C1)C N1(CC(C)(C)NC(C(CN(C)C)O)=O)CCN(C(=O)CC2CCC(=O)N2)CC1 S(=O)(=O)(c1cccnc1NCCc1csc(C(C)(C)C)n1)NC1C(CC)CCC1 C(=O)(C1=CC2(CCOC2)C1)NC1CN(C(Cc2nc(CC)sc2)=O)CC1C1CC1 Cc1cccn2cc(C(=O)NCC(CO)NC(=O)C(CO)C(C)(C)C)nc12 CCCCCCCC(F)C(=O)NC1C2CC(NC(C3(C)CS(=O)(=O)C3)=O)CC12 N1(C(c2c(C)nccc2)=O)CC(C)N(C(=O)CCCN=[N+]=[N-])C(C)C1 C(=O)(C(C)(CC)C(N)=O)NCC1N(C(CS(=O)(=O)N(CC)CC)=O)CCN(C)C1 C(C)(C)(C(C)CC(=O)N1CCSCC1)NC(c1nc(C)oc1)=O C1(NC(C=CCOC)=O)CC(C)CN(C(=O)CSCCC(C)C)C1 c1(C(N2CC=C(CCNC(CS(=O)(=O)NC)=O)CC2)=O)ccc2cn(C)nc2c1 C(CC(C)(C)C)(C(=O)Nc1cnc(F)c(C)c1)NC(CCNC(=O)OC)=O c1(C(=O)NC(CCNC(C(C)C#N)=O)C)cc(Cl)ccc1OCC(F)(F)F c1(CC(N2CCC(CCNC(c3ccccn3)=O)CC2)=O)ccc2nc[nH]c2c1 c1(N(CCCCOC)C)cccc(S(=O)(=O)NC2CCS(=O)(=O)C(C)C2)n1 CC(C)CCC(=O)NC(C)C(=O)NCc1ccccc1Br c1(OC)ccc(CC(C)C(=O)NC(CO)C(C)NC(c2ccns2)=O)cc1OC C12(NC(C=C(C)C)=O)CC1CN(C(=O)CCc1ccccc1OC(F)(F)F)C2 C1(C(N)=O)CN(C(c2ccc(CNC(=O)COC3CCCCC3)s2)=O)CCO1 C1(C(N2C(C)(C(=O)OC)CC2)=O)CC(NC(=O)CNC(=O)CC(C)C)C1(C)C CN1CCC(C(=O)NCCC2(O)CN(C(c3[nH]ccc3-c3ccccc3)=O)C2)C1 c1(C(N)=O)ccc(CCC(N2CCCC2c2cccc(Br)c2)=O)cc1 C1(C(=O)NCc2ccc(CNC(=O)Cn3cncn3)o2)COC2(CO)CC1C2 c1(CC)c(C(=O)NCCCCNC(=O)CCN2CCNC(=O)C2)nnn1CC N1(C(c2c(CCOCCCC)ocn2)=O)CCC(NC(=O)C2=CCSC2)CC1C Cc1nc(NC2(C3CNC3)CC2)ncc1[N+](=O)[O-] C=C(Cl)CC(C(=O)N(CCN(C)C)CC)NC(=O)CC1CCC(C)(C)O1 C(=O)(CS(=O)(=O)C(C)(C)C)NCC1CCC(NC(CCSCCC)=O)CC1 c1(CC(N2CCC(N(C(C=CC)=O)C)C2)=O)ccc(OC)cn1 C12(C(=O)OC)CCC(C(=O)Nc3ccc(Cl)cc3NCC(=O)N(C)C)(CC1)O2 c1(C(=O)OCC)cc(NCc2cn(C)nc2C(F)F)ccc1C C(=O)(C1CCc2nnc(C)n21)NCCC1N(C(Cc2cc(C)no2)=O)CCSC1 c1(CC)cccc(NC(c2ccc(NC(=O)C(=O)N(C)C(C)C)nc2)=O)c1C C(=O)(C(F)(F)C(F)(F)C(F)F)NCC(CNC(CCC(CC)OC)=O)C N1(Cc2cc(C(=O)OC)n[nH]2)CCC2C(C1)NC(=O)CCN2C C(CNC(C1COC(C)(C)C1)=O)(CC)(CC)NC(c1nc(CCC)oc1)=O C1(CC(=O)OC)COC(C)(C)CN1C(=O)Nc1ccc(-n2cnnn2)c(C)c1 c1(C(=O)NCCC(=O)NCC2CCCC2)cc2c(s1)CCCCCC2 C#Cc1cccc(CC(=O)NC2CC3C(NC(C4(OC(C)=O)CC4)=O)C3C2)c1 C(=O)(CC(C)C(C)(C)C)NCC(C)(CC(C)C)NC(c1c(SC)scc1)=O C(=O)(C1=NOC(C)C1C)NCC12N(C(CCN(CCC)C)=O)C(CC1)CC2 N1(C(CCC)=O)CCCC(C(N2CCCC2CCN(C)C)=O)C1CC C=CC(C)CC(=O)NC(CCOC)C(=O)NC1(C(=O)NCC)CC1 c1(CNC(=O)Nc2ccc(OC)c(F)n2)c(O)cc(F)cc1F C1(C(N2CC(OCCOC)C2)=O)CC12CCN(C(c1ccsc1C)=O)CC2 C1(C(=O)NC(CC(=O)NC)C)CCC(C(C)C)N1C(=O)CCn1cnnn1 CC1(C)C(C(N2CC(CCCCNC(c3ncsc3C3CC3)=O)C2)=O)C1(C)C CC1CC(C(=O)NC2CC3CN(c4ccnc(C#N)n4)CC23)=NO1 C12(C(C3(SC)CC3)=O)CC(C)(C1)OC21CCOCC1.C1(NC2CNC2)CCOCC1 N12CC(CCC1C)NC(=O)c1ccc(cc1)C2C.Cc1ccccc1CO N1(C(C2(CSC)CC2)=O)CCC(F)(C(=O)NC2(CF)CC2)C1 C1(C(=O)NCCC2CCCC2(C)C)(SC)CCN(C(=O)C(C)SC(C)C)C1 c1(CC(=O)NC2CN(C(Cn3ncc(C)c3)=O)C2)ccc2ncnn2c1 N1(C(C(CC)C2CCOCC2)=O)CCC(C)(CCNC(c2c(C)ncn2C)=O)C1 c1(C(=O)NCC2CC3(CC(NC(C4C(C)(C)C4)=O)C3)C2)cc(O)ccc1[N+](=O)[O-] N1(C(c2ccccc2)C)CCC(C)(CNc2cn(-c3cccc(Br)c3)nn2)C1 CC(C)(C(=O)NC1CCCC(CNC(c2c[nH]nc2Cl)=O)C1)C(F)F C(=O)(C(C)(C)CCCO)NC1(CC=C)CN(C(c2coc(C(F)F)c2)=O)C1 c1(OC)cc(C(=O)NCC(C)CNC(C2(c3cnccc3C)CC2)=O)ccc1C c1(C(=O)NCC(C)CNC(=O)C(C)C2CCCO2)ccc(C2CCC2)nc1 C1(C(N2C(CNC(C3C(C4C(C)C4)C3)=O)CC2)=O)CNC(=O)CC12CCOC2 c1(SC)ncc(N)c(C(=O)NCCCCNC(c2cc(F)cnc2O)=O)n1 C(=O)(N=c1cc(C(F)(F)F)[nH][nH]1)C1CCC(NC(c2c(OC)nsc2)=O)CO1 CC(C)CC(=O)C(=O)NCCC1(C(N2CCC(CCO)C2)=O)CCC1 C12CCCC(C1)CN(C)C2=O.c1(CNC(CN(C2CCCC2)C)=O)ccsc1 C(N=c1ccnc(CNC(=O)CSc2nncs2)[nH]1)C12OCC(CC3CC3)(C1)C2 C(=O)(CC(CC)C(C)(C)C)N1CCC(N(C(c2ncc(C#C)cc2C)=O)C)C1 c1(C(=O)NCC(CN(C)C(c2ccccc2F)=O)O)ccc(Br)c(F)c1F c1(C(N2C(C(C)(C)C)CCC2)=O)ccc(-n2cc(-c3ccnc(F)c3)nn2)cc1 c1(C(=O)OCC)ccccc1CNCC1(CNC(C)=O)CC1 O=C(CC(C(F)F)c1ccccc1)NCCN(CCO)C(c1ncsc1C1CC1)=O C1(C(=O)OC)CCC2(CC2)N1C(=O)C(=O)NCC1CCC12CCC2 N1(C(C(CCC)OC)=O)C2CCC1CC(F)(CNC(C1(CC)CCC1)=O)C2 Cc1cc(C(=O)NC2(CNC(=O)C(C)NC(=O)C(C)(C)C)CCC2)c(C)n1C1CC1 C1(OC)(CNC(=O)C=CCCc2ccccc2)CCN(C(C2(C)CC2C)=O)C1 C1(C(N2CC(C(=O)NCC(=O)N(C)CC)(COC)C2)=O)CC2CC(=O)C1O2 c1(CC)cc(C(=O)NCCc2ocnc2CNC(c2nnsc2SC)=O)on1 c1(C(=O)NCCC(C)N(C(=O)CCOCC(F)F)C)ccc(-n2cncn2)cc1 c1(NC(CCCCC)C2CC2)nc2ccccc2nc1NC1CCN(CC)C1 C1(C(N2CC(OC)C(NC(c3cnc(SC)s3)=O)C2)=O)CC(S(C)(=O)=O)C1 C1(NC(C(CO)NC(N)=O)=O)CCCCN(C(c2ccncc2N)=O)C1 c1(OCC)cccc(NC(C2CC(F)CN2C(C2CC2C(C)(C)C)=O)=O)c1 c1(C(=O)NCCCCC(C)NC(=O)C(C)N(C)C)ncnc2c1cnn2C c1(C(=O)NC2CN(C(c3c(SC)csc3)=O)CC2(C)C)cccn2nncc12 C1(C(=O)NCCN(C)CC)CC(NC(=O)CN2CC(=O)NC2=O)CCO1 c1(C(=O)NC(CN(C(=O)CC2CC3CC3C2)C)(C)C)ccc(S(N)(=O)=O)s1 C1(NC(CSc2ccc(OC)cc2)=O)CN(C(=O)CC2CCN(C)C2)CCC1F Cc1ccc(CC(=O)NC2CC2CNC(c2cn(C(C)(C)C)nc2C)=O)c(C)c1 c1(N2CCN(C(C)C(N)=O)CC2)nc(-c2ccccc2)nc(=NCCC2CC2)[nH]1 C1(c2nnnn2C2(C)CC2)(NC(c2cccc(NC)c2)=O)CCOCCC1C c1(CC(C2CC2)NC(=O)NC2CCCCC2)ccccc1 CC(C(=O)NC1(C)CC(NC(=O)CCOc2ccc(F)c(F)c2)C1)S(N)(=O)=O CCCC(C)(CC)C(=O)NCC(C)(C)CNC(c1ccc(=O)n(CC(C)O)c1)=O N1(CC)CC(NC(=O)C(CC2CC2)NC(c2cc(CO)c(C)o2)=O)CCC1=O C#Cc1cncc(C(=O)NCC2CCC(C(=O)NC(c3nc(C)cs3)C)O2)c1 C1(CNC(CC(C)SC)=O)CCN(C(c2cc(Cl)nn2C)=O)C1(C)C N1(C(C(COCC)(C)C)=O)CCC2CN(C(=O)C(C)=C3CC3)CC2CC1 c1(C(C)=O)ccc(CC(=O)NC(=O)C(=O)N(C)C)cc1.C12CCC1COC2=O n1(CC)cnc2[nH]c(=NC3CCS(=O)C3)nc(N(C)CC)c12.C(CCC(F)(F)F)N C1(NC(C(C)NC(N)=O)=O)CCC(CNC(=O)CCCn2ccnn2)CC1 C(C)(CN=c1nc(C2CCCCC2)nc[nH]1)N(C(C(C)CN1CCOCC1)=O)C c1(C(=O)NC2C(NC(C=CCC)=O)CCC2)ccc(C)c(C(=O)OC)c1 c1(C(C)C)n[nH]cc1C(=O)NC1COCC1C(=O)N(C)Cc1ccon1 CCC(CC(F)F)C(=O)N1CCOCC(NC(C2(C)CCC(=O)NC2)=O)C1 C1(NC(c2c(C)nc(CO)s2)=O)COC2(CCN(C(c3ncn(C)c3C)=O)C2)C1 C(CC(F)(F)F)(C1CCCOC1)OC(C(F)=CC)=O C(c1cccc(C)c1)=CC(=O)N(CCNC(=O)CC(C)(O)C1CC1)CC N1(C(C)C)CCN(CCC(=O)NCC#CCNC(C2(C)CC2C)=O)CC1 C(C)(C)(C(=O)NCCCCCN(C)C(C1CC(F)(CO)C1)=O)OCC C1(CNC(C2CN(C(C)=O)C2)=O)CC(C)CCN1C(=O)C(O)C1=CCCC1 c1(C(=O)NCc2ccc(C(=O)O)cn2)cc(Cl)nc(Cl)c1F c1(C(N2CCCC(CNC(CCCC)=O)C2)=O)ccn2c(O)nnc2c1 C1(C(N(CCCC)CC)=O)(NC(c2cncn2C)=O)CC(O)C1 CCC(C)C(CC(=O)N(C)C(C1CCCC1)C)NC(C1CCC(C)(C)OC1)=O C1(C)(C(N2CC(CC#C)(C(=O)NCC(C)OCC=C)C2)=O)CC2CCC1C2 c1(C(=O)NC2C3CN(C(c4cocn4)=O)CC23)ccc(Br)cc1I N1(C(CCOC(CC(C)C)C)=O)CCCC(N(C)C(C2(O)CCOCC2)=O)CC1 CCCCC(CNC(=O)Cc1sc(SC(F)F)nc1C)NC(=O)CCCOC C1(NC(Cc2ccc(CC)cc2)=O)CN(C(C2CC(C)CC(=O)N2)=O)C(C)(C)C1 Cc1cc(C(=O)NC2CC(C)(NC(C3CCCCO3)=O)C2)c(C)n1-c1ccon1 c1(NC(C)C)ncccc1C(=O)NC1CC(CNC(=O)CCCCNC(N)=O)C1 N1(C(C2C=CCN(C(CNC(=O)NC)=O)C2)=O)CCC(C)(C)CC1C(=O)NC C1(C(C)CO)CCN(C(C2C3CN(Cc4cc(Cl)ccn4)CC23)=O)CC1 C1(C(CNC(C=C(CCC)C)=O)(C)C)CCN(C(=O)CCC(C)SC)CC1 C1(CCC)CN(C(c2ccc(=O)n(C3CC3)c2)=O)CCN1C(C1CCOC1)=O C#CCC(O)C(=O)N(CCCOCCNC(c1n[nH]c(C)c1Br)=O)C N1(C(=O)NCC2CCCN2CCCO)CCCCC1Cc1ccc(F)cc1 C1(CCCC)(C(=O)NCC2CCN2C(C2CC3CC3C2)=O)CCCC1 Cc1cc(C(N2CC(NC(c3c(C)ncn3C)=O)CC(C)C2)=O)ncc1N N1(C(c2cc(C)n(C)n2)=O)C2CCCC1CN(C(=O)C(F)CC1CCOC1)C2 c1(C(=O)NC2(COC)CN(C(C3CCCS3)=O)C2)ccc2nnc(S)n2c1 C(CO)(C(=O)NCC1CCCN1C(=O)OC(C)(C)C)N(C)C(C1CC1(F)F)=O N1(C(c2c(CCC)[nH]cc2)=O)CCC(C(=O)NCCc2ncccn2)C(O)C1 c1(C(N2CCC2CNC(C2C(=O)NCCC2C)=O)C)cccc2ccccc12 N1(C(c2nccc(N)c2)=O)CCC2(CC1)CC2NC(C1CC12CCCCC2)=O C#CCC(C)(CC)C(=O)NCC(C)(C)C#CC(=O)Nc1ccc(F)nc1 Cn1nc(Br)c2ncnc(NCCC3CCCN(C(C4CNC(=O)N4)=O)C3)c12 CC1SCCCC1C(=O)NC(C)(C)CN(C)C(c1cc(-c2cnn(C)c2)on1)=O c1(C(N2CCC3CN(C(C4C5CCCOC45)=O)C3C2)=O)cccc2nc(Cl)cn12 C(=O)(CC(C)(C)CC(=O)OC)N1C2C(NC(C(CCC)NC(C)=O)=O)CC(CC2)C1 c1(C(N2CC3C(N(C(C=CC=CC)=O)C)C3C2)=O)cc(O)ccc1CC C1(NC(=O)CCN2CCOCC2=O)CC2CC1CN2C(=O)Cc1ncc(F)cn1 CCCCS(=O)(=O)CC(=O)NC1CCCC(NC(c2nc(C)c(N)cc2C)=O)C1 C1(CNC(CC=CCC)=O)CN(C(=O)COc2cc(C)on2)CC1(F)F C(C1(C)Cc2ccccc21)NC(CCCn1cc(CNC(C(C)O)=O)nn1)=O C(c1ccncc1)=CC(N1CC2C(CC(=O)NCc3cc(C4CC4)no3)C2C1)=O C1(CNC(CCCNC(C)=O)=O)CCN(C(c2cc(C(F)F)nn2C)=O)CC1C C(=O)(C1CCc2nccn21)N1CCN(C(C2(C)CSC2)=O)CC1CO C#CCC(C)(CC)C(=O)NC(C)CCNC(c1ncc(C(N)=O)cc1Cl)=O C(=O)(CC(C)(C)CC=C)NCC1(C(=O)NC(CC=C)CC)CC12CCC2 c1(C(=O)NC2CC(CNC(COc3cccc(C)c3)=O)C2)cn(C)c(=O)nc1O C(=O)(CCC1(NC(c2cnns2)=O)CCC1)NCC(=O)N(C)C C1(NC(COC(C)=O)=O)CCCC12CCN(C(c1cccc3nsnc13)=O)CC2 N1(C(C(Cn2ccc(C)n2)C)=O)CC2CCC(C1)C2NC(c1cn[nH]c1)=O C(=O)(C1=NNC(C(F)(F)F)C1)NCC1C2CN(C(c3nn(C)c(Cl)c3)=O)CC21 c1(C(N2CC(C(=O)NCC3CC34CCC4)(COC)C2)=O)cc(OC)ncn1 Cc1ccccc1C(C)CC(=O)NCC1CCCN1C(=O)C(C(C)C)NC(N)=O N1(C(C(C(CNC(C2(CCC)CCC2)=O)C)F)=O)CCC([N+](=O)[O-])CC1 CN1C(=O)CSC1=CC(=O)N(C)CC1CN(C(C2(C3CCC3)CC2(F)F)=O)C1 CCCC(CC)CCC(=O)N1CCOC(C(=O)NCCCCCCF)CC1 c1(C(N2CCC(C)(CNC(C(C)SC(C)C)=O)C2)=O)cc(S(N)(=O)=O)c[nH]1 c1(C(=O)NC(CNC(CCOCCC)=O)(C)C)ccnc(OCCOC)c1 c1(N(CC(=O)OC(c2cccc(Cl)c2Cl)C)S(C)(=O)=O)cccc2ccccc12 N1(C(C2(COC)CCOC2)=O)CCC2CCC(C1)N2C(C1CC(O)C1)=O c1(OC)ccc(-c2cnccc2C(=O)Nc2sncc2C(N)=O)c(OC)c1 c1(C(=O)NC(C(=O)NCP(OCC)(C)=O)CC(C)C)cc2cccnc2[nH]1 N1(C(C(C2CCC2)NC(Cn2ncc(C#N)c2)=O)=O)CC(=O)NC(=O)C1 n1(CC)cc(Cl)cc1C(=O)NC(C1CCN(C(C2CCOC2)=O)C1)C C1(c2cccc(F)c2)(NC(=O)CCF)CCN(C(=O)CC(O)C2CCCC2)C1 C1(NC(c2c(C)c[nH]c2)=O)CC(O)CN(C(c2cn(C)nc2-c2ccoc2)=O)C1 c1(C(N(CCNC(C2N(CC)CCCC2)=O)C)=O)c(Br)nc2n1CCC2 N1(C(C(CC)Sc2nc(=N)[nH][nH]2)=O)CC(CNC(=O)Cc2cnsc2)C2(CC2)C1 C(CCC(C)CC(=O)NC1C2CN(C(=O)CS(=O)(=O)N(C)C)CC12)=C(C)C C(C1CCCc2ccccc21)c1cn(-c2nc(C)cs2)nn1.FCF c1(CNC(C(n2cc(CS(C)(=O)=O)nn2)C)=O)ccccn1 c1(C(N2C(C(C)(C)NC(=O)CC3CC=CCC3)CCC2)=O)ncncc1Cl N1(C(CC2N(C(CC(C(=C)C)OCC)=O)CC2)=O)CCCN(C)CC1CC c1(C(=O)NC2CC2CNC(=O)C(F)F)nc2c(cc1Br)OCCO2 C=CCC(CC(C)C)C(=O)Nc1ccccc1OCc1cccs1 c1(CN2CC3N(C(c4c(C)c(F)ccc4)=O)C(C3)C2)cnc2[nH]ccc2c1 Cc1cc(C)n(C(C)CC(=O)NC(CCNC(=O)Cc2cnc(C)s2)C(C)C)n1 CC(CC(=O)N1CC=CC1CF)C(=O)c1cccc(F)c1 c1(CC)cc(F)ccc1C(=O)NC(CNC(=O)C(CSC)c1ccccc1)CC Cc1cc(F)c(C(=O)NCC(CO)CC(C)(C)C)c(Br)c1 Cc1ccc(OCCC(=O)NC2C=CCN(C(C3CCCCN3C)=O)C2)c(C)c1 N1(C(c2ccn(C)c(=O)c2)=O)CC2=C(C1)CN(C(C1CCc3ncsc3C1)=O)C2 CC1CC(=O)NCC1C(=O)NC(CNC(=O)CCC(C)O)C1CC1 C(=O)(C(C)(C)C(F)(F)F)NC(CC1CN(C(CC2CC(OCC)C2)=O)C1)C c1(C(C)NC(C(C)NCC)=O)nc2cc3ccccc3cc2[nH]1 c1(C(=O)NCCC(C)N(C)C(C23CCC(CC2)C3)=O)cc(N)cc(S(C)(=O)=O)c1 N1(C(CC2CC(=C)C2)=O)Cc2n[nH]cc2C1C(=O)NCC1C2CCCC12 c1(C(N2CCC(CNC(C(C)NC(C)(C)C)=O)CC2)=O)csc2nccn12 C1(C2(NC(CCNC(N)=O)=O)CC2)CCCCN1C(=O)CC1CC2(CC2)CO1 C1(CC(=O)N(CC)CC2CCOC2)(NC(=O)C(C)N=[N+]=[N-])CCCCC1 c1(CN(CCOC)CC2(Cc3ccc(F)cc3)CC2)ccnc(F)c1 c1(C(=O)NC(CCNC(c2cc(OC)ncn2)=O)C)cc2sccc2[nH]1 c1(C(=O)NC(C(C)NC(=O)C(C2CCOCC2)O)CO)c[nH]c(=N)c2[nH]ccc12 Cc1sc(C(=O)NC2CC(C)(NC(=O)Cc3c(Cl)cnn3C)C2)cc1[N+](=O)[O-] O=C(C1=Cc2ccccc2OC1)NC1C2CN(C(C3C4CCC(F)(F)C34)=O)CC12 c1(C(=O)NCC(CNC(c2cc(C)sn2)=O)OC)nccc2ccncc12 c1(C(N2CCC2(C)C(C)C)C(=O)NC)sc(Cl)nc1C N1(Cc2cc(C)ns2)CCCC2(CCN(C(=O)C3CCCc4c3ncn4C)C2)C1 C(=O)(CCC(C)(C)NC(=O)C(C)OCC(C)C)NCCOCC N1(C(=O)Cc2ccc(O)cc2)CCCC2(C1)CN(C(c1cnn[nH]1)=O)C2 CCCCC(CC)CC(=O)NC1CC(CC(=O)NCCOCC)C1(C)C N1(C(=O)OC(C)(C)C)CCC(C(c2ccc(F)cc2)CC(=O)O)CC1 C(=O)(CCCC(=O)N(C1CN(C(C2CC(F)(CO)C2)=O)CC12CC2)C)OCC C1(CCC(=O)NCc2snc(C)n2)CCCCN(C(=O)CCC2CCOCC2)C1 N1(C(C2N(CC)CC2)=O)CCC2CN(C(c3cc(C)cnc3N)=O)CC2CC1 CN1CCC2(CC1)CC2C(N1CCOCC(C(=O)NCCC(=O)N(C)C)C1)=O Cc1ccnc2nc(C(=O)NCCC3CCN(C(=O)CC4CN(C)C4)CC3)nn12 N1(C(C2C(CC)C2)=O)CCN(C(=O)CC2(C(F)(F)F)SCCS2)C(C2CC2)C1 c1(OC)noc(C)c1NC(C1CC(NC(=O)CNC(C2CC2C)=O)C1)=O C1(N(C)C)CCCN(N(C)C2CN(c3ccccc3)CC23CC3)C1 N1(C(C(C=C)(C)C)=O)CCC2(CC1)CN(C(=O)CC1CCC(=O)NC1)C2C(C)C Cc1ccnc(C(N2CC3CC2(CNC(C2CN4CCN2CC4)=O)C3)=O)c1N C(=O)(CC(CC)NC(c1ccn(CC)n1)=O)N(CC)Cc1ccoc1 c1(CC(=O)NC(CC)(C)CNC(C2CCS2(=O)=O)=O)ccc(OC)cc1C c1(C(=O)NC2CC(CNC(C(C)(C)OC(C)=O)=O)C2)n[nH]c(C)c1Cl CC(CC(N)=O)C(=O)N1CCC(CCN(C)C(c2ncncc2N)=O)CC1 C1(CNC(c2nc(C)sc2C)=O)CCC2(CN(C(C3CCC(C)(C)O3)=O)C2)O1 c1(C(=O)OC)ccnc(NC2CCN(C(=O)C(C)NC(C3CCCCC3)=O)C2)c1 c1(CC(=O)NCC2CCC(C)C2)cc(F)ncc1Br C(=O)(CCCC(C)C)NCC(c1c(OC)cccc1)NC(C1(C)CC1(C)C)=O N1(C(C(C)(F)F)=O)CCCC(N(CCO)C(C2CCN(S(=O)(=O)C(F)F)CC2)=O)C1 N1(C(CCCCCC)=O)CCc2nc(CNC(=O)C(CC(C)C)C(C)C)sc2C1 c1(C(=O)NC2CN(C(COCCC#C)=O)C(C)C2)cc(Cl)c2ccccc2c1O N1(C(c2ccc(C)cn2)=O)CC2CC(NC(c3ccc4sncc4c3)=O)C(C2)C1 c1(C(N(C2CCN(C(c3cc(C)[nH]c3C)=O)C2)CC)=O)cc(C)n(C)n1 C1(C(=O)OCC)CC(CSc2ccnnc2O)C12CCCC2 C1(=CCNC(C(C)C2CC2)=O)CCN(C(C2(c3ccccc3)CC2(Cl)Cl)=O)CC1 Cc1cccc(CC(=O)NCCOCCOCCCNC(C2CC2(F)Cl)=O)c1F CC(C)C(C(=O)NCC(CC1CC1)C(=O)N(CC(F)Cl)C)C(C)C C1(C(C)NC(=O)CSCc2ncc[nH]2)CCN(C(=O)CCc2cnccn2)CC1 C(=O)(C1=C(Cl)CCCC1)NC(CNC(c1ccc(C#C)nc1)=O)CC=C N1(C(Cc2cc(C)no2)=O)CC(N(C(=O)Cc2c(C)n[nH]c2C)C)C2(CC2)C1 C1(n2cc(CC(=O)OC)nn2)CCCN(C(C2CCOC(C)C2)=O)C1 c1(C(=O)NCC(C)N(C(=O)CCN2CCC(F)C2)CC)cc(C)nn1CC c1(N2CC3N(CCF)C(CC3)CC2)nc2ccccc2c(=NCc2ccoc2)[nH]1 CC(C(=O)NCc1ccc(C(NC[Si](C)(C)C)=O)o1)C(C)(C)C C(CC(C(=O)NCCNCCN=[N+]=[N-])NC(=O)C(C)CC1CCC1)SC C1(C(N(C(C(=O)NC(CN(CC)CC)C)C)CC)=O)C2CCC(C2)C1C c1(OC)ccc(C(N2CC3CC(NC(=O)C(C)C4CCC4)C2C3)=O)cc1O CN1CCCC(C)(C(=O)NC2CC=CCC2C(=O)NCc2ccc(Cl)o2)C1 O=S(=O)(c1ccc(Cl)cn1)NCC1CCCCN1c1ncnn2ccc(Br)c12 C1(C(=O)NCC2CCC(NC(CCC(=C)C)=O)C2)CN2CCN1CC2C C1(NC(C=C(C)C2CC2)=O)CCCC(CNC(=O)C=CC2CCOCC2)C1 CC1(O)COCCN(C(=O)COC(C)(C)CNC(=O)CCC2CCCOC2)C1 c1(C(=O)NCC2(C)CCN(C(c3c(CC)ocn3)=O)CC2)cc(F)c(F)cc1N Cc1nc2ccc(C(=O)N(C(C)CCNC(C3CN4CCN3CC4)=O)C)cc2o1 Cc1c(C(N2CCCC(NC(c3nsnc3O)=O)CC2)=O)sc2[nH]cnc(=O)c12 Cc1ccncc1C(=O)N(C1CCCN(C(=O)Cc2ccoc2)C1)C c1(OC)ccccc1SCC(N1CCCC(C(C)NC(=O)CN2CCCC2)C1)=O C(=O)(C(O)CC(C)(C)C)NCC(CC)NC(c1nc(CC)oc1C)=O N1(C(c2c(CC)noc2)=O)CCN(C(c2[nH]cc(C)c2C)=O)C(CC)C1 C(C(C)(CC)CC)(c1n(CCOC)nnn1)NCC1(NC(=O)OC)CC=CCC1 c1(C(=O)NCC2(C)CCCN2C(=O)Cc2cscn2)c(F)cc(C#N)cc1F c1(C(N2CCC(C)(CNC(C(C=C=C)C)=O)C2)=O)ccc(Cl)c(OC)c1F C1(C(=O)NCC2CN(C(C(C3CC3)SCC)=O)C2)CCN(C(=O)C(C)C)CC1 C12(NC(CCC)=O)CN(C(c3cccnc3C(F)(F)F)=O)C(COC)(C1)C2 Cn1nc([N+](=O)[O-])cc1C(N1CCC2CCCC12CNC(c1ccc(F)o1)=O)=O C1(CNC(C(C)(F)F)=O)Cc2ccccc2CN1c1cc(C2CC2)nc(Cl)n1 N1(C(C2CC(OC)C2)=O)CCSCC1C(=O)N(C)CC1CC1 c1(C(=O)NCC(C)N(C(=O)C2=CCCS2)C)cc(C#N)ccc1F C(C(CC(F)(F)F)NC(c1cccc(C(F)F)n1)=O)NC(c1cccc[n+]1[O-])=O c1(C(N2C(CN(C(C3(CC#C)CC3)=O)C)CCC2)=O)nc[nH]c2ncnc1-2 N1(C(C=CSC)=O)CC2(C1)CN(C(=O)Cn1cnc([N+](=O)[O-])c1)CC2CO C(C1=CCCN(C(c2ccc(OCF)cc2)=O)C1)NC(C1CC=CCO1)=O C1(C(N2CC(n3cc(CNC(C(CC)(C)C)=O)nn3)C2)=O)(OC)CCC(C)(C)CC1 O=C1NCC(C(=O)NC2CC(CCC(=O)NC3CC(F)(F)C3)C2)N1 C(CC(=O)N1CCC(NC(c2cccc(N)c2O)=O)CC1C)(C(F)(F)F)OC c1(SC)cc(C(N2CC(C(=O)NCCNC(=O)CCF)C2)=O)co1 C(=O)(C1CCc2cc(Br)ccc21)NC1C(CNC(c2cn(CC)nn2)=O)CC1 C(C(C)(O)CC(=O)N1CC2C(NC(C3C4CC5C(C4)C35)=O)C2C1)OC c1(C(N2C(C(N3CCC(CO)CC3)=O)CSCC2)=O)cccc(F)c1Br C1(C(=O)NCCCN(C(=O)CN2CCCCCCC2=O)C)OC(C)(C)OC1(C)C C(c1ccc2c(c1)OC(F)(F)O2)=Cc1cc(Br)cc(OCCC)c1 c1(C(=O)NCC(C(C)C)NC(CC(c2ccc(C)cc2)C)=O)cc(Cl)ccc1F C12CCN(CC1)CCOC2c1ccccc1F.c1(C(=O)O)cscn1 c1(NC(C2CCCN(C(c3ccnc(C)n3)=O)C2)=O)cc(F)c(F)cc1[N+](=O)[O-] C1(C(=O)NCCCCNC(c2ccc(C#N)o2)=O)CCC(N=[N+]=[N-])CC1 c1(C(C(=O)NC2CCN(CCS(=O)(=O)NC)C2)(F)F)ccccc1C C(N=c1ccnc(NCc2cc(NC3CC3)ncc2F)[nH]1)C1(CCC)CCC1 C=C(C)CCCC(=O)NC(C(=O)N1CCN(C)CC1CCO)C(C)(C)C C12(C(N(CCCCNC(C(C)Cc3ccccn3)=O)C)=O)C=CC(CC1)C2 Cc1c(Br)sc(CNC(c2cc3n(n2)CCC3)c2nnnn2CCC2CC2)c1C C1(CNC(CN(C2CCSC2)C)=O)COCCN1C(=O)Cc1cncc(F)c1 C12(NC(c3c(C)scn3)=O)CCCC1N(C(=O)CC1CC3(CC3)CO1)CCC2 c1(C(N2CC(O)(C(C)NC(C3CCC3(F)F)=O)C2)=O)cccc(C(F)F)c1F C(CC)(CC)(CCNC(C1(CF)CC1)=O)NC(C1CC(O)(CC#C)C1)=O c1(C(=O)NC(CC#C)(C)C)cc(Br)ccc1C1CC1 N1(C(C)C)N=C(C(=O)NC2(C3CC3)CCN(C(=O)Cc3csnn3)C2)CCC1=O c1(CC(=O)NC(C)CCNC(C2CC(F)C2)=O)ccnc(O)c1 C(CCCNC(c1cccs1)=O)(c1ccccc1)NC(C1(CC#C)CCC1)=O N1(C(C=C(C)C(F)F)=O)CCC2CCCC12CNC(c1ncc(C(F)(F)F)s1)=O C1(C#N)(C(N2CC(C(C)(C)O)(CNC(CCNC(COC)=O)=O)C2)=O)CC(C)C1 c1(C(=O)NCCN(CC(=O)NCCCC)C2CC2)cc(C(F)(F)F)nn1C Cc1oc(C#N)cc1C(=O)NC(C)C(=O)NC1(C)CS(=O)(=O)C1 c1(C(C)C)ccc(NC(=O)C(=O)NC(C2CCCCO2)C2CC2)cc1 C1(C)(CNC(c2n(CCC)nnn2)c2cc(COC)on2)C=CCCC1 CC1(CC(=O)NCCCC2CCCN2C(=O)CCc2ncc[nH]2)CCCCCC1 c1(C(=O)NC2CC2CNC(c2ccccc2C(F)F)=O)cc2cccnc2o1 C(=O)(C1=CCCOCC1)NC1CCN(C(c2n(CC#N)ncc2)=O)CC1O CCCCCC(=O)N(C1CCN(C(=O)CC2OCCC2C)CC1)C C1(C(N(C)CC2(Br)CC2)=O)CCCCC1CNC(=O)CN1CCSCC1 C1(C(N2CC(C)C(NC(=O)C=C3CC3)CC2)=O)CC2C=CC1C21CC1 C1(C(=O)NCc2c(C(N(CC(N)=O)CC)=O)nco2)CCC(C2CC2)C1 C1(C(=O)NCC(CCC)NC(=O)C(C)(C)O)CCCC(F)(F)C1 C(c1ccccn1)=CC(=O)NCC(C)(C)NC(C1C(C)(C)C1(F)F)=O C12(C(N3CCC(NC(C(c4ccccc4)N(C)CC)=O)C3)=O)CC(C1)C(C)O2 C1(NC(CC2C(C)(C)C2)=O)C2CC3C(C2)C13C(=O)N1CC(O)CO1 CC1(C)CC(C(=O)NCCOCCC(=O)NCC2CC3CCCC3C2)CCO1 c1(C(=O)NCC(CC=C)NC(=O)CCC2CC(C)(C)CO2)ncc(N(C)C)cn1 c1(C(=O)NCC2C(NC(C=C(CCC)C)=O)C2)cc(C)nc2[nH]nc(O)c12 CN1Cc2c(-c3nc4c(s3)CC(C(N3CCC(Br)C3)=O)CC4)cccc2C1=O N1(C(C(CNC(c2cc(C(N)=O)co2)=O)OC)=O)CC2(CCOCC2)C1 N1(C(C(=O)N(c2ccccc2)C)=O)CC2CCN(C(=O)C(F)CC3CCOC3)C2C1 c1(N(C)C(C2CN(C(=O)NC3CC3CO)C2)=O)c(Br)cc(C(F)(F)F)cc1I O=C(CCC(=O)N1CCCC1C1CCCCCC1)c1ccncc1 CC1(C(N2CCC(CNC(C3CCC(F)C3)=O)C2)=O)C=CCCC1 C(=O)(CC(C)C(F)(F)F)NC1CCC(C)(NC(CC(=O)OC)=O)CC1 c1(C(=O)NC(C(C(C)C)NC(C2C(C)(C)C2(C)C)=O)C)noc2ncccc12 N1(C(=O)OC(C)(C)C)CC2CC(C(N3CCCC(C(C)(F)F)C3)=O)CC(C1)C2=O c1(C(=O)NC(CC2CN(C(C3CC=C(C)CC3)=O)C2)C)cc2n(n1)C(C)CCC2 C1(NC(C)=O)CN(C(C2(NC(C3(CC4CC4)CCC3)=O)CCC2)=O)CCC1O C1(NC(=O)NCC(CCSC)N)CCC(C)(C)CC1CSc1ccccc1 N#CC1CCN(C(C2CC(NC(c3cc(Oc4ccccc4)ncn3)=O)C2)=O)C1 c1(C(=O)NC2CCCN(C(C3CC34CCSCC4)=O)CC2)scc2c1CCCC2 C1(NC(C2CCC(C(C)C)CC2)=O)CCCCN(C(C2(F)CCOCC2)=O)C1 C1(C)(CNC(c2c(C)onc2)=O)CCN(C(C2CCC(CC(F)(F)F)CC2)=O)C1 N1(CC)CCCCC1C(=O)NC1CCN(CCNC(=O)N(C)C)CC1 c1(NC(c2c(CNC(C(CC=C)(C)O)=O)noc2)=O)cccc([N+](=O)[O-])c1 C1(CNC(c2c(CC)ncs2)=O)(CO)CCN(C(=O)Cc2cc(C3CC3)no2)C1 C=CCC(C)(C)CC(=O)NC1CCN(C(c2cc(C)cc(Br)c2)=O)CC1F N1(C(C(c2cccc(Cl)c2)(C)C)=O)CC2CC1CN2C(=O)CCc1cncnc1 CC1(C)CCCC(C(=O)NC2CCC(CS(C)(=O)=O)CC2)O1 c1(NC(=O)C2CC2)ccc(Cl)c(C#N)c1.CN1CC(N2C3(CCC3)CC2=O)C1 CC1CCCN(C(c2cc(CF)on2)=O)C1CCNC(c1ccc(N)c(N)n1)=O c1(OC)c[nH]c(C(N2CCC(C(C)N(CC(F)F)C)CC2)C(=O)NCC)cc1=O N1(CCC(=O)NCC(c2c(C)nn(C)c2C)=O)CCOC2(CCC2)C1CO C(=O)(C(O)CCC(C)C)NCC(C)(C1CCC1)NC(c1nc(OC)c(F)cn1)=O CCCC(CC)CCC(=O)N1CCC(OC2CN(CC3CCCOC3)C2)CC1 n1(CC)ccc(C(N2CCC2CC(N2CCC(Br)C2)=O)=O)n1 c1(OCC(CCC(=O)N2CCCC(C(=O)OCC)C2)=O)cc(C)c(O)nn1 C(N(O)C(=O)Cc1cccc(Cl)c1)c1cn(C(C)CO)nn1 N1(C(C2N(C(C3N(C)C(=O)CCC3)=O)CC(O)C2)=O)CC2C=CCC(C2)C1 CC1(CC(N2CC(CNC(c3cn(C(F)(F)F)cn3)=O)C(O)C2)=O)CCCCC1 C1(OC)CCCC(NC(c2nc(-c3cnccn3)no2)C(C)C)C1 CC12CCCN1S(=O)(=O)C(C(=O)NCCCCCNC(=O)CCF)C2 N1(C(CCN(CCOCCOC)C)=O)CC(NC(=O)C(F)(F)CO)C(C)C1 C1(C2CC2)(NC(CC(C=C)C)=O)CCN(C(c2noc3c2CCCC3)=O)C1 CC1(C)CCC(CNC(=O)CC2CSCCO2)(NC(C2CCC3(CCC3)O2)=O)C1 Cc1ccnn1C(C)C(=O)NC(C1(O)COC1)C c1(C(C)(C)OC)ccc(C(N2CC=CC2CNC(C2(O)CCC2)=O)=O)cc1 C1(CNC(C(F)=CC)=O)CCCC2(CN(C(=O)C(C(C)(C)C)N(C)C)C2)O1 C12(SC)CC(C(=O)NC(C3CCCN3SCc3cscn3)C)(CO1)C2.C1(=O)CN1 c1(C(N2C3CN(Cc4nccc(OC)c4)CC32)=O)onc2ccccc12 C1(C(C)C)CN(C(C)=O)CCN1C(=O)C(Cc1ccc(O)cc1)NC(N)=O CC1(C)CC(CC(N2CCC(NC(C3CC(F)(F)C3)=O)C(F)C2)=O)NC1=O C1(CNC(C(C(C)C)NC(COC)=O)=O)COCCN(C(c2cc(C)c[nH]2)=O)C1 N1(C(CC(C)NC(C)=O)=O)CCC(NC(=O)C(=O)N(C)C)CC1 C1(NC(c2ccc(CO)o2)=O)CCCN(C(C2CC(n3ccnn3)C2)=O)CC1 c1(C(=O)NC2CN(C(c3cc(C)ncc3)=O)CC2(C)C)cc2nccn2c(O)n1 C(=O)(CCCc1sccc1C)NCC(CC)NC(C1(n2ccnc2)CCCC1)=O C12(CNC(CC(CC)CC)=O)CCCC1N(C(=O)C=C1CCCC1)CCC2 C1(=O)C2=NOC(C2)CN1.c1(CCC(=O)NCCC2(O)COC2)ccc(CO)cc1 CC(C)S(=O)(=O)C(C)C(=O)N1CCC2(C1)CN(C(c1cc(Cl)c(F)c(Cl)c1)=O)C2 Cc1cccc(C)c1C(=O)NC1CC1C(=O)OC(=O)C(C)N(C)C CCC(C(=O)NC(c1ccccn1)C)N(C(=O)Cc1cnsc1)C C(CCCC(=O)NCc1occc1C(N1CCOC(CCF)C1)=O)OCC C1(NC(Cn2c(C)cc(C)n2)=O)CC2CC1CN(C(c1onc(Br)c1C)=O)C2 C1(C(=O)NC2CCN(C(CC3(C)CC(F)(F)C3)=O)CC2F)C2CCCCCCC12 c1(CC)nc(C)c(C(=O)NCC2CC(NC(=O)C(F)(F)Cn3cccn3)C2)s1 c1(C(N(C)CCNC(=O)CC2CC=CCC2)=O)ccc(C(F)(F)F)cc1C1CC1 c1(CC)nc(C)oc1C(=O)NC12CC1CN(C(c1csc(C(C)C)n1)=O)C2 C(=O)(CCC(F)(F)F)N1C(C(=O)NC(COC)C2(C)CC2)CCC1 C(=O)(CCCC(CC)NC(=O)Cc1c(C)cnn1C)NCCCC=C C1(O)(CCNC(=O)COC2CC=CC2)CCN(C(C2CC3CCC3C2)=O)C1 c1(CN2CC(C(=O)NC(c3ccccc3)C(N)=O)OCC2)cc(Cl)c(F)c(Cl)c1 c1(C(N2CC(CCNC(C(COCC)C)=O)C2)=O)cc(Cl)c2n[nH]cc2c1 c1(C(=O)NC(C)CCNC(=O)C(c2cccc(F)c2)C)cnc2n(c1=O)CCS2 c1(C(=O)NCCC(=C)CNC(c2n[nH]cc2CC)=O)cncc2[nH]ccc12 C=CCCCC(C(=O)NCC(C)C(F)(F)F)NC(C1COCOC1)=O c1(CNC2CCC(C(=O)Nc3ncc(C#C)nc3)C2)n[nH]c2ccc(Br)cc12 c1(CC(N2C(CNC(CC=C)=O)C=CC2)=O)ccc(F)c(Br)c1 c1(NC(C)CNC(=O)C(C2(O)CCCCC2)(F)F)nc(O)n(C)c(=O)c1[N+](=O)[O-] c1(C(C(=O)NCC)N(c2ccccc2)C(C)=O)cccc(Cl)c1 C(c1ccc(OC)c(F)c1)=CC(=O)NC(C(=O)OC)Cc1cn(C(C)(C)C)nn1 CC1=C(C(=O)N2CCCOC(CNC(C3(F)CCC3)=O)C2)CCO1 N(C1CCc2cc(CNC(C3(C)COC3)=O)ccc21)C(c1cc(CC)n(C)n1)=O N1(C(C2CCC(C)O2)=O)Cc2ccccc2C1CNC(=O)CC(C)(C)O c12c(cnn1CC)C(=O)NC2.c1(OCCNCC(=O)NC)ccc(OC)cc1 C(C)(C(=O)NCCCCO)N(CCC)C(C1CCO1)=O C12(CN(C)C(c3cnc4cnccn34)=O)CCCC1CCN2C(=O)OC(C)(C)C C1(NC(Cn2ncc(CC)c2)=O)CCC(C)(C)CC1CNC(c1nnsc1C)=O C(=O)(C1CCCCc2ccccc21)NC1CC(CNC(=O)C2=CCOC2)C1 C12(CCNC(C(C)(C)CF)=O)CCC(C1)N(C(=O)C(F)CC1CCCCC1)C2 CC(=O)C(C)CC(C)C(=O)N1CC(NC(c2ccc(O)nc2C)=O)CC12CCC2 C1(CNC(C(CCOC)C)=O)CCCCN(C(c2cc(C3CCC3)no2)=O)C1 c1(OCC)ccc(-c2n[nH]c(C(=O)N(CCCSCC)C)c2Br)cc1 c1(C(=O)OC)nc(CCN(c2ccccc2)C(=O)C(C2CCCCC2)F)oc1C C(=O)(CC(C)(C)C)NC1C(NC(C(C)OCCCC)=O)CC1.C12(CC1)C(=O)NC2 C(CCCCCNC(C1CCOC(CC)C1)=O)N(C(COC(CC)CC)=O)C Cc1cc(C(N2CC(O)CC2CNC(C23CCC2C3)=O)=O)ccc1[N+](=O)[O-] c1(C(C)NC(C2(CC(N)=O)CC2)=O)nocc1C(=O)NCCC(C1CC1)C1CC1 C1(NC(C(=O)NCC2CC2)=O)CCCC2CN(C(c3nccc(Cl)c3F)=O)CC12 N1(C(c2c(CC)c[nH]c2)=O)CCN(C(=O)CC2=CCN(C)CC2)C(C)CC1C CC1(C)CC(NC(c2cccc(Cl)c2F)=O)CN1C(C1CCC(=O)C1)=O CCS(=O)(=O)CC(=O)NCC(CC)CC(=O)NC(CF)C(F)(F)F c1(CNC(C2(NC(c3n[nH]c(C)c3Cl)=O)CCOCC2)=O)ccnc(F)c1F C(C)(C(CC(=O)Nc1cnc(C)c(Cl)c1)NC(=O)CCC1(C)N=N1)OC CC1CN(C(c2ccnc(N(C)C)c2)=O)CCC1NC(=O)NCCO C(C(=O)N1CC=CCO1)C1C(C)CCN(C(C2CCC(CCC)CC2)=O)C1 N1(C(C2CC(CNC(C(C)OC)=O)OC2)=O)CCCN(C)CC1 c1(C(=O)NC(C2CN(C(c3c[nH]c4cccnc34)=O)C2)C)ccc2[nH]ccc2n1 Cc1n[nH]c(=NCC(C)(C(C)C)NC(=O)CC2CCNC2=O)s1 c1(-c2onc(C)n2)ccc(C(=O)NC(C)CN(C)C(c2nocc2Cl)=O)cc1 CC1CN(Cc2ccccc2)CC(C)N(C(c2ccc3ocnc3c2)=O)C1 C1(NC(C2C(c3ccn(C)c3)C2)=O)COCCN(C(c2cc(C3CC3)cs2)=O)C1 CC1CC(NC(c2ccno2)=O)CCN1C(c1ncccc1Cl)=O CC1=NN(C)C(=O)C1CC(N1CCC1CNC(=O)CCOC1CCC1)=O C(=O)(CCCCC(=O)NC1CC(F)(CNC(C2CCc3cnnn3C2)=O)C1)OC C12(CC(N3C4C(NC(CC(=O)OCC)=O)C(CC4)C3)=O)CC3CC(CC(C3)C1)C2 CC1(C(N2CCC(OC3CN(C(=O)CCF)C3)CC2)=O)COCCO1 c1(Nc2c(C(F)(F)F)ncc(C(=O)OCC)c2)cnc2c(Br)n[nH]c2c1 C(=O)(C(O)CC(C)(C)C)NCCNC(C1CCCN(C(CCC(=C)Cl)=O)C1)=O C(=O)(CCCC(=O)N(C)C)NCC(C(=O)NCC1(O)C(C)CCC1)N(C)C c1(OCCC(=O)NCCCNC(CSCCC#N)=O)ccc(F)cc1Cl Cc1cc(C(=O)Cn2cc(C(=O)CC(=O)NCCCCCCO)nn2)ccc1Cl c1(OC)cnc(F)c(C(=O)NCC2CC(F)CN2C(=O)C(O)C(C)C)c1 C1(C(N2CCC(CCCC)C2)=O)CCN(C(c2sccc2CC)=O)C(CC)C1 C1(C(C(=O)N(CCCN(C(Cc2c(C)n[nH]c2)=O)C)C)(C)C)CCCN(C)C1 C1(CC)C(NC(c2cccnc2C)=O)CCCN1C(=O)CN1CCC(OC)C1 C1(C(N2C(COC)C=CC2)=O)CC2CC2N1C(=O)C(n1ccnc1C)C c1(SC)nc(N(C2CCNCC2(C)C)C(=O)CN2CC(=O)NC2=O)cc(C)n1 C1(NC(c2c(C(C)C)cccc2)=O)CC2CCC(C1)N2C(C1(N=[N+]=[N-])CC1)=O N1(C(C(C)CCO)=O)CCN(C(=O)CSc2n[nH]c(O)n2)CC(O)C1 C1(C(=O)NCC2CC2CNC(c2c[nH]nc2C)=O)(OC)CC(C)CC(C)C1 Cc1cn2c(C(=O)NCCN(C)C(c3ccnc4ccccc34)=O)c(Cl)nc2s1 C(=O)(C(C)CCO)NCC(C(C)C)NC(=O)C(c1ccc(Cl)s1)C c1(C(=O)NCC(C)N(C)C(C2COC3(C)CC2C3)=O)cccc(C(F)(F)F)c1O C1(CC(=O)NC(CN(C(c2ccoc2CC(N)=O)=O)CC)C)CCCS(=O)(=O)C1 C1(CC)CN(C(C2CCCC(CF)C2)=O)CC1C(=O)NC1CCCC1O C1(C(=O)NCC2(CO)CCN(C(CCC=CC)=O)CC2)CS(=O)(=O)CC(=O)N1 C1(NC(c2ccc(-c3onc(CC)n3)cc2)=O)CN(CC)C2CCCCC12 S(=O)(=O)(c1c[nH]ccc1=NC(C)C1CCCCN1CC)N1CCC(CC)(CO)C1 N1(C(=O)OC(C)(C)C)CCC(NC(C23CSCC2C3)=O)C1(C)C C1(NC(C2(Nc3ccccc3F)CC2)=O)C2CN(Cc3ccccc3)CC12 N1(C(C(N2CCSCC2)C)=O)CCC(NC(C2CN(C)CC(C)O2)=O)CC1C CC(C(=O)NNc1ccc(Br)nn1)c1c(F)cccc1Cl c1(-c2onc(C(=O)O)n2)ccc(Oc2ccc(Cc3ccccc3)cn2)cc1Cl C1(Cc2cn(Cc3c(C(=O)O)cco3)nn2)CCN(C(C2(Br)CC2(F)F)=O)CC1 C1(NC(c2ccc(CC)cc2)=O)CN(C(c2cccnc2)=O)CCC1(F)F N1(C(c2n(CC)ncc2)=O)CCC(C)(CNC(c2ccc(COC)s2)=O)CC1 C1(O)(CNC(C2C(C)(C)C2NC(c2ccc(C(F)F)o2)=O)=O)CCCOC1 CN1CCN(C(=O)C(CNC(C2OC3CCC2C3)=O)N(C)C)CC1CO c1(C(=O)NCC2C3CN(C(C(C=C)O)=O)C2C3)cc(S(N)(=O)=O)c(Cl)cc1Cl c1(N(CCC)CC)ccc(C(=O)N(C(C)CN(C(=O)C(C)CC2CC2)C)C)cc1 C#Cc1ccc(OCC(N2CCN(C(=O)C(C)NC(N)=O)CC2C(F)F)=O)cc1 CCCCC(CNC(=O)C(C)CCOC)NC(c1onc(Br)c1C)=O C1(C(=O)NCCNC(Cc2cn(CC)nc2)=O)CCCS1(=O)=O N1(C(CNC(C(CC)C)=O)=O)CCN(C(c2cc(C)n(CCOC)n2)=O)CC1 CCC(CC(F)F)C(=O)N1CC(CNC(c2cn(CCO)nn2)=O)CC1(C)C N1(C(CSC)=O)CC2CCC2(CC(N2CCCC2CCO)=O)C1 c1(NC(C2C(NS(c3cn(C)nc3)(=O)=O)C2)=O)cccc2c([N+](=O)[O-])cccc12 C1(C(=O)NCC2N(C(C3(C4CC4)CC3)=O)CCC2)CC12CCOc1ccccc12 c1(NC(C(c2ccccc2I)CC)=O)cc2ccc(SC)cc2cn1 c1(C(=O)Nc2ccc(-c3cnn[nH]3)cc2)ccc(O)cc1Cl c1(C(=O)NCC2CCN(C(=O)CC3CCC3)C2)cccc(CN2CCOCC2)c1 c1(CN2CC3N(C(CCC=C(C)C)=O)C3C2)ccc(F)c(C(=O)O)c1F c1(C(N2CC(OC)CC(NC(C(C=C)(C)C)=O)C2)=O)ccc2nn[nH]c2c1 N1(CC(=O)NCC(C(=O)NC2CC(O)C2)O)C(=O)CCC1=O CC(C)(C)CS(=O)(=O)N1CCCC(c2ocnc2C(=O)O)C1 C1(CNC(=O)NCCCc2nnco2)CCCC12OCCO2 N1(CCNC(Cc2cc(C)no2)=O)CCN(C(C2CCCC23CC3)=O)CC1 c1(C(N(CC(CN(C(C)=O)C)O)C)=O)n[nH]c2ccc(Cl)cc12 c1(CC)ccc(C(N2CCC(NC(c3cc(COC)on3)=O)C2(C)C)=O)cc1F N1(C(C2CC3(ON=C(C)C3)C2)=O)CCCCC2(C1)CN(C(=O)C(C)SC(C)C)C2 NS(=O)(=O)CCC(=O)NC1CCCC1C(=O)NCCCCC(=O)N(C)C C1(C(=O)NCC(C)N(C)C(C23CCC2CC3)=O)C(C(=O)OC(C)(C)C)C1(C)C CC(C)(C)S(=O)(=O)CC(=O)N1CCN(C(C2COCCOC2)=O)C2CC12 c1(C(N2CC(C(C)NC(c3c(C(C)C)nns3)=O)C2)=O)cc2ccsc2[nH]1 Cc1ccc(C=CC(=O)NCC(C)CN(C(=O)CC2CCCS(=O)(=O)C2)C)cn1 N1(C(c2cnc(C)nc2C)=O)CCCC2(NC(c3cncc(Cl)n3)=O)CCCC12 Cc1ccc(N)cc1OCC(N1CCC1CNC(=O)C(c1ccc(Cl)s1)O)=O N1(C(C2(OC)CCC2)=O)C(C(=O)NC2CCC3CCC23)CCC12CC2 N(C1CCc2c(Cl)cc(Cl)cc21)CC1(Nc2cnccc2)CC2(CCC2)C1 C1(C(=O)NC(C2CCN(C(C3CC(C(=O)OC)C3)=O)C2)C)CCC(C)(C)OC1 c1(N(CC(C)C(F)(F)F)C)ccc(S(=O)(=O)NC2CC2C2CCOCC2)c(Br)c1 C=CC1(CC(=O)NCC23CCC(CC2NC(=O)Cc2cn[nH]c2)C3)CCCCC1 c1(NC(C)=O)ccc(C(=O)NC(C)CNC(C2(C#N)CC(C)C2)=O)c(Cl)c1 C1(C2(NC(Cc3ncc(C)s3)=O)CC2)CCCCN1C(C1C2CCCC12)=O N1(S(c2ccc(C(=O)OC)cc2)(=O)=O)CCCC2(CCN(C(=O)CN(C)C)C2)C1 c1(NCCCC(N)=O)nc(N2CCSCC2)nc2scnc12 C1(NC(CCC2(C)CC2)=O)CC2CCC1N2C(c1ccc(OC2CCC2)cc1)=O C(=O)(CCCS(C)(=O)=O)NC1CCC(NC(CC(CC)C2CCC2)=O)C1 CC(C)C(C(=O)NC1C=CCN(C(C2CC(=O)C2(C)C)=O)C1)NC(N)=O N1(CC(C)(C)NC(CCCOCC)=O)CCN(C(c2ccc(F)cn2)=O)CC1 CCC(C)(C(=O)N(C(C)C(=O)NCCC(C)N1CCC1)C1CC1)OC N1(C(c2c(C)n(C)nc2)=O)CC2CN(C(c3ccnnc3S)=O)CC2(C)C1 c1(C(=O)NCC(CC)NC(C2CNC(=O)N2)=O)c[nH]nc1C(C)(C)C c1(OC)cc(Cl)c(C)cc1COC(=O)C(F)(F)CC(C)C c1(CC)c[nH]c2cc(COC)ccc12.C12(CCCNCC1)CO2 CC1CN(C(=O)CC(F)(F)F)CCN1C(C1CCOC1c1ccncc1)=O N1(C(c2cc(C#N)sc2)=O)CCCC2(CCCN2C(c2ccc(Cl)nc2O)=O)C1 N1(C(Cc2ncc(C)s2)=O)CC(C2CN(C(c3cc(F)c(F)cc3O)=O)C2)C1 Cc1cncc(C(N2CC(CC(=O)N(CC(C)O)CCO)C(C)C2)=O)n1 CCCC(C)(C)C(=O)N1CCC(C)(NC(C2CCC23CCOCC3)=O)C1 CCCC(CCC)CCCC(=O)N1CC(CCNC(=O)CN(C2CCSC2)C)C1 C1(C(=O)OC)CC(=O)CN1C(c1sccc1SC)=O c1(CCC(=O)NCC(CNC(C2=C(C)OCC2)=O)C)cccc(S(N)(=O)=O)c1 O=C(C(Cl)=CCl)NC1CCC(CCNC(C2CC2(F)F)=O)C1 CCC(CN(C)C)CC(=O)NCC1(CNC(=O)C(c2ccc(F)cc2)SC)CC1 CN1CCc2c(NC(=O)N(C3(O)CCC3)Cc3ccccc3)cccc2C1=O Cc1ncc(CC(=O)NC(C2(O)CN(C(C3CC3[N+](=O)[O-])=O)C2)C)[nH]1 C1(CCC(=O)NCC2(C(=O)NC(C3CCCC3)C)CC2)CCC(=O)N1 C(=O)(C1=CCCOC1)NC(C(C)C)CCN(C)C(c1cnc(C(F)(F)F)cn1)=O c1(N2CCC(O)(CCNC(c3sccc3Cl)=O)CC2)c(Br)cccc1[N+](=O)[O-] c1(NCc2cc(C)ns2)cc(NCC(Cl)=CCl)ncn1 c1(CCC(N2CC(C)C(NC(=O)Cn3nnc(=O)[nH]3)C2)=O)ccc(F)cc1Cl CC(O)(CC(=O)N1CC(NC(=O)COc2cccc(F)c2)C(O)C1)C1CC1 C(=O)(C(C)(C)CC(=O)NC(C)CNC(c1ccccc1C(C)(C)C)=O)OCC CCC(C)CCCCC(=O)N1CCC(N(C(=O)CCCN(C)C)CC)C1 CC1(C)C2CCC1(C)C2C(=O)NC1CN(C(=O)Cc2cc(F)ccc2Br)C1 c1(CC)cc(C(=O)NCC2CCC(C(=O)NCCC(C)(C)F)O2)n[nH]1 O(C=C(C#N)C(=O)N1CC(NC(c2cc(C3(C)CC3)on2)=O)C(C)(C)C1)CC C1(C(N2CCCC(O)C2CCc2ccccc2)=O)COc2ccccc2C1 c1(NCC(=O)NCCN(C(=O)C(C)(C)C)CC)nc(C)nc2sc(C)c(C)c12 N1(C(C2CCCN(CC(=O)OC)C2)=O)c2ccc(Br)cc2NC(=O)C1C C(C(COC)C(=O)NCC1CCCN(C(C2(N(C)C)CCCOC2)=O)C1)OC c1(NCC)ccc(C(C(=O)NCC2CCCO2)N(CC(F)F)C)c(Cl)c1OC.CO C1(C(=O)NCCN(C(=O)CC2CCC(O)C2)C(C)C)CCc2nnn(C)c2C1 c1(C(=O)NC2C(NC(C(C)NC(C)(C)C)=O)CCOC2)cn2c(n1)CCC2 CCC(C)C(C(=O)NCC1(CC(=O)N(C2CC2)CC2CC2)CC1)OC Cc1ccc(NC(=O)CSCCNC2CN(C3COC3)C2)c(C)n1 C#Cc1ccc(C(N2CCC3CC23C(=O)NC(CC2CC2)C(=O)NC)=O)cc1 N1(C(CC(CCC)C)=O)CC2C3CCC(C(NC(=O)Cc4sccc4C)C3)C2C1 N#CCCCC(=O)N1CCCC1C1CCN(C(C2CC(F)(CO)C2)=O)C1 CC1CC(C(=O)N(C)CC2CCN(C(=O)CCC3(C)CC3)CC2)Cc2nn[nH]c21 C1(C)(C(=O)NCCC(CC)(C)NC(C2COCCO2)=O)CCCN(C)C1 C1(OC)CCCN(C(=O)C(CC(C)C)ONC(c2cccc(F)c2)=O)CC1 C1(NC(C2CCC3(CCC3)O2)=O)CCC12CCN(C(=O)C1=CCCOC1)CC2 c1(N(CC)CC)nc(N(C)C2CC2)c2c(n1)CCC2.c1(CN)cccc(N)c1.c1cnco1 c1(C(N(C(CNC(=O)Cc2cn[nH]c2)C2CC2)C)=O)ccc(Cl)c(Cl)c1N CCC(CC(F)F)C(=O)NCC1(NC(c2ccn(C(C)(C)C)n2)=O)CCOC1 C1(CNC(CC2(CSC)CC2)=O)C(C)CCN1C(c1ccc(CN=[N+]=[N-])o1)=O C1(NC(CN2CC(OCCCCC)C2)=O)CCCC(F)(F)C1 C1(NC(CN(C2CCSC2)C)=O)CC(C2CCN(C(C3(C)CC3)=O)C2)C1 CC1C(C)N(C(c2cccc(C#N)c2Br)=O)CCN1Cc1ccccc1 c1(C(C(=O)NCC2CC2)N(CCCOC)CC(C)C)nc(Br)ccc1OC n1(CC)cc(Br)cc1-c1nc(C2CC=CCC2)nn1CC1CCS(=O)(=O)C1 C1(CNC(c2[nH]cc3c2CCC3)=O)CN(C(=O)C(F)(F)CO)CCC1(F)F C1(CNC(N(C)CC2CC2C)=O)C=CCC1 O=C1CCC(CC(=O)NCC(C2CCCCC2)NC(C2CCS(=O)(=O)N2)=O)CN1 C(=O)(C(O)CCC(C)C)NCC1C(N(C)C)CN(C(C2COCOC2)=O)C1 C1(OC)CCCCC1CC(=O)NCCc1nc(-c2ccncc2)no1 Cn1cc(C2CCC2)c(NC(C2CCC(CN)OC2)=O)n1 c1(CCNC(N2C3CN(CC)C(C3)C2)=O)cccc([N+](=O)[O-])c1 CCCCC(C)(C1CCCO1)NC(=O)CSCc1nnc(C)o1 C1(CC(=O)NC(C2CCN(C(C3(CO)CC3(F)F)=O)CC2)C)CCC(=O)NC1 Cc1n[nH]c(=NC2CCC(N(C(=O)C(C)NC(c3cccc(F)c3)=O)C)CC2)o1 C1(NC(C2CCCN(C(c3ccc(C(=O)OC)s3)=O)C2)=O)CCNC(=O)CC1 c1(C(=O)OC)cccc2[nH]c(CNC(=O)CC3CC(C(=O)OC)C3)cc12 c1(C(N2C(C)CC(NC(c3c(C)c(N)n(C)n3)=O)C2)=O)ccc2cncn2c1C c1(C(=O)NCC2CC(F)CN2C(c2cc(Br)n[nH]2)=O)csc2ccncc12 C1(C(=O)NC2CC(NC(C=C3CCC(C)CC3)=O)CC2O)CCCCCN1C C1(CN(CC(=O)NCCC)C)CCN(C(=O)C(CC)SC)CC1 C1(OC)C(NC(C2(CNC(=O)Cn3cncn3)CC=CC2)=O)CC12CCC2 N1(C(CCCOC(C)(C)C)=O)CC2(CCCCN(C(C3(Cl)CC3(F)F)=O)C2)C1 CC(C)(C(=O)N1CCC(NC(c2cnn(C(F)(F)F)c2)=O)C(CO)C1)S(C)(=O)=O C1(NC(C(F)OC)=O)CCC2CCN(C(C3CC34CCSCC4)=O)C1C2 C1(CCNc2c(Br)ncc(C(C)C)n2)CN(C(=O)OC(C)(C)C)CCS1(=O)=O CC1(C)CC(=O)NC1CNC(C1(C)CCN(C(c2c[nH][nH]c2=N)=O)C1)=O CC1CCCC(C(=O)NCCNC(=O)C(=O)OC(F)F)CC1 C1(CC)CCCCN1C(=O)C(=O)NCc1ccccc1CC1CC1 C1(NC(CC2N(C(c3c(C)n(C)cn3)=O)CCCC2)=O)CC1C1CCCC1 C1(C(=O)Nc2cnn(C3CCCCC3)c2)(CC)CCNC1 N1(C(COCCC=C)=O)CCCC(CCC)(NC(c2cccn2C)=O)C1 n1(CCC#C)c(N2CC3CC2(c2nc(C)no2)C3)nnc1C(c1ccncc1)O C1(NC(C(=O)NC(c2ccncc2)CC)=O)CCCN(Cc2cccc(F)c2)C1 Cc1sc(C)c(C(=O)NCC2(C)CCC(NC(c3cnc(C4CC4)[nH]3)=O)C2)c1C#N C(=O)(C(F)(F)c1cscc1Br)NC(C)CNC(C1(C)CCC1)=O C=CC(F)(F)C(=O)NCCC(C)NC(C1C(CN=[N+]=[N-])C1(C)C)=O Cn1cncc1CCC(=O)NC1CCCC1NC(C1COCCO1)=O N1(C(C(C)=C(CC)C)=O)CC(OCC)C(NC(=O)CNC(=O)C(C)(C)C)C1 Cc1ccc(CN2CC3CC3(C(=O)NCC3CC3C3CC3)C2)cc1Cl c1(CC(=O)N(C)C)ccc(Cl)cc1S(=O)(=O)NC1CC(C(F)F)C1 CCC(CCC(=O)NC1CCN(C(c2coc(Br)c2)=O)C1(C)C)OC C1(C)(NC(C(CCOCCO)NC(CN(C2CC2)CC)=O)=O)CN2CCC1CC2 c1(OC(CC)C(=O)NC(C)(C)C(C)NC(=O)C(C)NC(=O)NC)cccc(C)c1 c1(SC(CCCC)C(=O)O)ccc2c(c1)n(CC(C)C)c(=O)n2C1CC1 c1(C(=O)NC(N2C(C)(C(N(CC)CC)=O)CC2)=O)ccc(-c2nncn2C)cc1 N1(C(c2c(C)nc(COC)s2)=O)CCN(C(=O)CC(C)SC)CC1CO N1(C(C=CCC)=O)CCN(C(c2conc2CC)=O)CC1C(F)F C1(C)(C(N2CC(n3cc(C(C)(C)NC(C4CC(O)C4)=O)nn3)C2)=O)COCCO1 N1(C(C2(C=C)CCN(C(=O)Cn3cccc3)C2)=O)CCCC(C)(C)CC1 C(C(N=c1cc(CC(N)=O)n(C)[nH]1)c1nnnn1C1(C)CC1)(OCC)OC c1(C(=O)NCC(CCCC)NC(=O)C(C)N2CC(C)C2)nc(C)c(C)nc1C C1(CC)C(C(=O)NCCN2CC(C)(O)C2)CCN1C(=O)C=C1CCCCC1 CC1CCC(NC(c2cccc(C3CC3)n2)=O)CN1C(C1COC2(CCC2)C1)=O Cc1c(-c2ccc(-c3cnn(C)c3C)cc2)oc2ccccc12 C#CCCCCC(=O)NC1(CNC(c2cc(C(=O)C(F)(F)F)c[nH]2)=O)CCOC1 c1(SC(C(=O)NCCNC(CCCc2onc(C)n2)=O)C)ccc(F)cc1 c1(C(N2C(C)CC(CNC(c3cccc(OC)n3)=O)C2)=O)ncc(Cl)cc1Cl C#Cc1ccc(-c2nc(-c3ccc(Cl)cn3)nn2C)nc1 N1(C(COCCC)=O)CC(CNC(c2csc(C(N)=O)n2)=O)OC(C)(C)C1 c1(OC)nccc(C(=O)NC2(CN3CCN(C(=O)C(C)CC(F)F)CC3)CC2)c1F c1(CNC(CSC(C)C)=O)ccc(C(=O)NCC2(O)CCN(C)C2)cc1 C1(CC)(CC)CN(C(=O)C(n2cc(-c3ncc(C)cc3C)nn2)C)CCS1(=O)=O C1(CNC(c2c(OC)nsc2)=O)N(C(C2CC2C(C)(C)C)=O)CCCC1(C)C C=CCC(CC(C)C)C(=O)N1CCCC1(C)C(=O)N(C1CCC1C)C c1(CNC(c2n(C)ccc2)=O)nc(CNC(C2C(C3CC3)C2(F)F)=O)cc(O)n1 Cc1cc(C)c(CC(=O)NCC2CC(CS(C)(=N)=O)C2)c(C)c1Br N1(C(C(C(CC)O)C)=O)CC2(CCCCN2C(=O)C(C)NC(=O)C(C)(C)C)C1 Cc1cc(CN(C=O)Cc2ccc(O)c(Br)c2)ccc1N(C)C Cc1ccc(C)c(CC(=O)NC(C2CCCCN2C(=O)C(C)OCC2CC2)C)c1 N1(C(c2ncoc2C)C(=O)NCC=C)CCc2sccc2C1c1cccs1 c1(C(=O)NCC2=CCN(C(CN3C(C)CCC3)=O)CC2)cccn2nncc12 c1(C(=O)NCC2(O)CN(C(C3CCCO3)=O)C2)cccc(N2CCCC2)n1 c1(C(N2CCC(NC(C3C(C)C3)=O)(CN(C)C)CC2)=O)cc2c(F)cc(F)cc2[nH]1 C=CC(C)(CC)C(=O)NCc1cn(C2CN(C(=O)CSCC(N)=O)C2)nn1 N1(C(CNC(=O)OCC=C)=O)CCC(NC(C2CCCCN2N=O)=O)C(C)C1 c1(NC(C2CC2C(=O)Nc2cccc(Cl)c2)=O)cc(Cl)ccc1N1CCCC1 c1(C(=O)OC)ccc(C)nc1NC1CCN(C(c2cc(C)cs2)=O)C1C CC1CCCCN1C(=O)C=CC(C)NC(=O)C(CO)N(C)C N1(C(CN(CC)CC)=O)CC(NC(C2CCC2C(=O)OC)=O)CC(C)C1 C#Cc1cccc(C(=O)N(CC(C)NC(c2cc(F)c(O)c(F)c2)=O)C)c1Cl c1(CNC(C(C)(C2CC2)OC)=O)ccccc1CN(C)C(c1c(C)cnn1C)=O Cc1cnncc1SC(N1CCOCC1c1ccccc1Cc1ccccc1)=O c1(C(N2C(C)CCN(C(=O)C(F)OC(F)(F)F)CC2)=O)c[nH]c2cc(F)ccc12 Cc1nc2ccccn2c1CC(=O)NCCN(C(=O)C(C)C(C)(F)F)C N1(C(C(C(=O)OC)C)=O)CCC2CCN(C(=O)C(=O)NC(C)C)CC12 c1(C(=O)NC2(C)CCCN(C(C3C(CC)CCC3)=O)C2)cccc2ccncc12 c1(CC)cc(C(=O)NC2CC(CO)N(C(C3CCC(C)O3)=O)C2)ncn1 Cc1ccc(-c2nc(C)c(C(C)NC(C)C(=O)OC(C)(C)C)s2)cc1 c1(C(=O)NC(C2CCN(C(C(C)SC)=O)C2)(C)C)cc(Cl)c(F)c(Cl)c1 CC1CN(S(=O)(=O)N2CCN(Cc3n[nH]c4c3CNCC4)CC2)CC(C)O1 C12(C(N(C)CCC3CCN(C(C4(N=[N+]=[N-])CC4)=O)CC3)=O)CCCC(CO1)C2 C1(C2CCC2)(CNC(C=Cc2cn(C)nc2)=O)CCN(C(=O)Cc2cncs2)CC1 C12(CN(C(C(c3ccc(N(C)C)cc3)C)=O)CCO)CCCC1OCC2 Cc1nn(CC(C)C)c(C)c1S(=O)(=O)NC1CCC(C(=O)O)CC12CCC2 C1(n2cc(-c3ccc(C(=O)OCC)o3)nn2)CCN(S(=O)(=O)CC(C)C)CC1 N1(C(C2CC(=O)NC2)=O)CCC2CCCC12C(=O)NCC(O)C1(Cl)CC1 C1(C(=O)NCC(C)NC(c2cn(C(C)C)c(=O)cc2)=O)CCc2[nH]nc(O)c2C1 c1(OC(C)C)ccc(C(C2CCCO2)NCc2ccc(F)cc2)cc1 c1(C(=O)NC2CC3(C(C(=O)NC(C(=O)OCC)C)C3)C2)cnc(C)nc1C C1(C(=O)NCc2nn(CC)nc2C)C2CCC(C2)C1NC(=O)Cc1nonc1C N1(C(C2(F)CC(C(=O)OCC)C2)=O)CCC(CC(=O)NC2C3CCCCC23)CC1 c1(C(=O)NCC2C(NC(C)=O)CCC2)ccc(-c2cncnc2)cc1F c1(C(=O)NC(CC)CNC(=O)CCC2CCC(=O)N2)cncc2[nH]ccc12 C(=O)(CCS(C)(=O)=O)NC(C)C(C)NC(=O)C(F)(F)c1ccsc1Cl C(=O)(C(CC(=O)O)N1CCOC(CN2CCOC2=O)C1)NC(=O)OC(C)(C)C C1(C(N2CCC(NC(CCC3CC(C)C3)=O)CC2)=O)CC(O)c2ccccc2O1 c1(C(=O)NC2CC(NC(c3c(C)nc(C(C)C)o3)=O)C2)c(Cl)nn(C)c1Cl c1(NC(c2nc(-c3c(C)ccc(OC)c3)sc2C)=O)ccc2scnc2c1 n1(CC(=O)NC2(C)CC(NC(C(C)(C)OC)=O)C2)c(O)nc2ccccc12 C1(NC(CN2CCN(C)CC2)=O)CCN(C(=O)Cc2cccc(Cl)c2)C12CC2 Cc1nc(Cl)ccc1CC(N1CCN(C(=O)CC2CCCOCC2)C(CO)C1)=O O=S1(=O)CCC(NC(=NCc2ccn(C3CCCC3)n2)NCC2CCOC2)C1 Cc1cc(C(N2CC(O)(CCNC(=O)CC3CC3)C2)=O)ccc1F C1(CC(C)CNC(=O)C#CC2CC2)CCN(C(c2ccoc2)=O)CC1 c1(NC(=O)CC2CCCN(C(=O)CC3CCOC3=O)C2)cccc(F)c1F CCC(C(=O)NC1CC(C(F)C(=O)N(C)Cc2cncn2C)C1)N(C)C C12(NC(c3c(Cl)cncc3Cl)=O)CCCC1N(C(=O)CC1CC1)CCC2 c1(C(N2CC3C(CCNC(C=CC)=O)(CC3)C2)=O)cc(C)c(Cl)c(C)c1 C1(C(N2C(C(=O)Nc3cc(O)nc(C)n3)CC(=C)C2)=O)CCc2nc[nH]c2C1 c1(C(=O)NC(C)CC2CCC2)c(Cl)cncc1Br CC1CN(C(=O)CC2CCCC2)CCC1CNC(=O)CCCCN1CCCC1 N1(C(C2C(CC)N(C(=O)Cn3cccc3)CC2)=O)CC(O)CC1(C)C C(=O)(C(=O)C(F)(F)F)NCCC1CCN(C(C(C)CC2CCC2)=O)CC1 c1(C(=O)NCC2(C3CC3)CCN(C(C(CC)OC)=O)C2)cc(S(N)(=O)=O)oc1C c1(C(=O)NCCCN(C(=O)Cn2cnnn2)CC)cnn(CCC(F)(F)F)c1 C1(C(=O)NC2(C(F)(F)F)CS(=O)(=O)C2)CCn2c(O)nnc2C1 C1(NC(Cc2c(C)nc(C)s2)=O)CCCC2CN(c3ncnc(Cl)c3CO)CC12 C12(NC(CCC3CCN(C(c4cc(C)ncc4)=O)C3)=O)CCC(C1)OC2C c1(NC(=O)NC(C)(CN)C2CC2)ccc2cccnc2c1 N1(C(c2ccc(OC)c(F)c2)=O)CC(NC(=O)CCC(C)N(C)C)C(C2CC2)C1 C1(C(=O)NC(C)CNC(c2cnn(-c3cccnc3)c2)=O)COCC2(CCC2)O1 C#CC1(O)CCN(C(=O)CC2CC2CNC(=O)C(COC)CC)C1 c1(C(=O)OC)ccc(NCCCNC(=O)CC2CC3(CCC3)CO2)c([N+](=O)[O-])c1 c1(C(=O)NC(CC)(CNC(C2(CCOC)CCC2)=O)CC)ccc(F)c(C)c1N N1(C(c2ccc(C#C)o2)=O)CC(F)(F)CC1C(=O)NC1(C)C(C)(C)C1(C)C c1(C(=O)NCC(C)(C2CCC2)NC(=O)CCS(C)(=O)=O)cccc2[nH]nc(O)c12 c1(C(CC)NCC2CC(=O)N(C)C2)cc(Cl)ccc1OC CC(C)(O)C(=O)NC(C1CCCCC1)CNC(=O)Cc1ccccc1 c1(N2C(NCC3C(F)(F)C3)CCC2)ncc(Cl)cn1 O=C1NCC2(CCN(C(=O)CC3(NC(C4CC(O)C4)=O)CCCCC3)C2)O1 N1(c2n(CC(=O)N(CC)CC)nnn2)CCC(N=c2[nH]c(=N)[nH]n2C)CC1 N1(C(C2(C)C(C)C2)=O)CCCC(CCCCNC(=O)CC2(C)CCCC2)C1 C1(CNC(C2=CCC(C)CC2)=O)CN(C(c2cc(Cl)ns2)=O)C2COCC2O1 N#Cc1cn(CC(N2CCCC23CCN(C(=O)C2=CCCC2)C3)=O)c(=O)nc1O c1(CC)cc(Cl)ccc1NC(C1(O)CCN(C(c2ccc(Cl)s2)=O)C1)=O C(=O)(C(C)C(F)(F)C(F)F)N1CCC(CCNC(C2(CC#C)CCOCC2)=O)C1 C1(NC(c2c(CC)nns2)=O)CCN(C(C2(N=[N+]=[N-])CC2)=O)CC1CC N1(C(CCOC)=O)CC(C)CCC1C(=O)N(C)CCc1cnn(C)c1 c1(C(=O)NCCN(C(c2cc(C3CCOC3)[nH]n2)=O)CC)cn(C2CC2)nn1 c1(C(C)OCC)nc(C(=O)NC2(C)CC(NC(c3snnc3C)=O)C2)cs1 C(c1ccc(C(=O)OCC(=O)NC2C3CCC(O3)C2N)cc1)=CC(=O)OC c1(C(=O)NC(CNC(C(C)NC(C2CCCC2)=O)=O)C2CC2)ncc(F)cc1N C(=O)(CS(=O)(=O)CC)N1CCC(N(CC#C)C(C2C3CN(C)CC23)=O)C1 N1(C(Cc2cnc(C)[nH]2)=O)CCCC(C)C1CNC(=O)CCc1ccn(C)n1 C1(NC(c2c(C)scc2)=O)C(CNC(c2cc(C(N)=O)[nH]n2)=O)CCC12CCC2 c1(OC)sc(C(=O)NCC2CC2CNC(c2ccnc(C)c2)=O)cc1Br N1(C(c2[nH]cc(C(C)=O)c2)=O)CCCCC(N(C(=O)C(C)NC=O)C)C1 c1(C(=O)NCC2CCN2C(=O)C(O)c2cnc[nH]2)csc2c1CCCCCC2 C1(NC(c2nc[nH]c2C(F)(F)F)=O)CCCCCN(C(C2CC2F)=O)C1 c1(C(N(CC(C)CNC(=O)COCCc2cccs2)C)=O)ccc(F)c(N)c1 c1(CNC(C23CC(OC)C2C3)=O)ncccc1CNC(c1cnccc1C)=O N1(c2nc(=NC)[nH]c(=NCC3(C)CC3)[nH]2)CCOc2ccc(Br)cc2C1 N1(C(CNS(C)(=O)=O)=O)CCOC2(CCCN(C(C3CCC=CO3)=O)C2)C1 Cc1cc(=NC(=O)C2CCN(Cc3cc(Br)ccc3F)CC2O)[nH]c(Cl)n1 Cc1ncc(CCC(=O)NC2(CNC(C3CCCN3CC(F)F)=O)CC2)s1 C(=O)(CCC1=CCCCC1)N1CC(C#C)(C(N2CCc3c[nH]nc3C2)=O)C1 C(CCCCC(=O)NC1CN(C(=O)Cc2nccn2C)CC1(C)C)NC(C)=O S(=O)(=O)(c1ccc(C#N)cc1Cl)N1CC2N(C(C(=O)N(C)C)=O)C(COC2)C1 c1(C(N2CCN(Cc3cnn(CC)c3C)CC2)=O)cc(C)c(Br)cn1 CC1C(C)N(C(=O)CC2CCCC2)CCN1C(=O)CCc1cc(Cl)cc(Cl)c1 C1(N(C(=O)CC2(OCCO)CCC2)C)CN(C(c2cc(=O)cc[nH]2)=O)CC12CC2 C1(CNC(c2c(OC)nsc2)=O)COCCN1C(=O)CC(C)c1ccco1 N1(C(C2C(C)CCC2)=O)CCCC2(CCN(C(=O)C=CC(C)(C)C)CC2)C1 c1(OC)ccc(O)cc1C(N1CC(O)(C(C)NC(c2csc(Cl)c2Cl)=O)C1)=O c1(N2CCC(CNC(c3cc(CC)cc(F)c3)=O)C2)ccc([N+](=O)[O-])cc1F CCC(CN(C)C)CC(=O)N1CC(CO)(NC(C2CC3CC3C2)=O)C1 C(C(C(=O)NCCC(F)F)NC(=O)Cn1ccnc1C)SCC C1(C(=O)NC2(CC=C)CCN(c3nnc(C(N)=O)s3)C2)CCC(C)(C)CC1 N1(C(C2CC(OCC)C2)=O)CC2CN(C(c3ccc(O)cc3)=O)CCC2(CO)C1 CC(C(=O)NCC1CC2CCC1N2C(c1cc(C(F)F)ccc1F)=O)C(C)(F)F C(=O)(C(C)CC(F)F)N1CCC(N(C(=O)C(C)C)CCOC)CC1 N1(C(C2(OC)CS(=O)(=O)C2)=O)CCN(C(=O)C=C(C)C)C(CO)C1 c1(C(N2CCC(C)(CNC(C(c3ccc(C)cc3)=O)=O)C2)=O)ccc(F)cc1C c1(NC(CC2(N(C(C3N(CCC)CCC3)=O)C)CC2)=O)ccc(C#N)cc1O C1(OC)COCC1n1cc(C(=O)NCCC(C)NC(c2ccnn2C)=O)nn1 c1(C(=O)NCC(C)CNC(c2cn(C)c(O)n2)=O)cc(Cl)cc(F)c1N Cc1cc2c(C(=O)NCC3CN(C(=O)CCCOC(C)C)CCO3)cccc2o1 C1(C(N2CC(COC)(NC(c3csc(C)c3)=O)C2)=O)COC2(CCC2)C1 c1(C(c2nnnn2C2CC2)NCCC2(C(F)(F)F)CCC2)ccc2ncsc2c1 c1(CNC(CC=CC=C)=O)nocc1C(=O)NC(C)CC(N)=O C1(C(=O)NCCCCNC(c2ncc(Br)cn2)=O)CCCC(F)(F)C1 N1(C(C2CCN(Cc3c(C(=O)OC)cc(Br)cc3)C2)=O)CCC(O)C(C)(CO)C1 C1(CNC(c2c(CNC(C3CCN(C)CC3)=O)ocn2)=O)CCC(C)(C)CO1 c1(C(CC)C)ccc(C#N)c(N2CCC(N(C(=O)C=Cc3cscn3)C)C2)n1 c1(CNC(C2C(C(=O)NCCC)C2)=O)ccccc1C(C)(C)NC(=O)CC1CC1 N1(C(C2(OC)CC2)=O)CCC(C(F)(F)F)C(NC(=O)C=CC2CCC2)C1 CS(=O)CCC(O)C(=O)NC1CC2(C1)CN(C(=O)Cn1nnc3ccccc13)C2 N1(C(c2c(C)ccs2)=O)CC(CNC(c2cc(CO)c(C)o2)=O)C2(CCC2)C1 CS(=O)(=O)c1cccc(S(=O)(=O)NC2CC2c2ccc(F)nc2)c1 CC1(C(=O)NCc2ccc(-n3cccn3)cc2)CCNC1=O C1(C)(C(N2CC(CC)C(CNC(c3cc(C)ns3)=O)CC2)=O)CC(C)OC(C)C1 C1(C(=O)NCC2(C3CC3)CCCO2)CC=CCC1C(=O)Nc1cncs1 N1(C(c2ccsn2)=O)CCN(C(=O)C=CC2CCCO2)CC(CO)C1 c1(CCC(=O)N(CCN(C(C(C2CCCC2)OC)=O)C)C(C)C)c(C)n[nH]c1C c1(C(N(C2CN(C(C3CCSCC3)=O)C2)C)=O)cccc(Cn2ccnn2)c1 Cc1nc(C(=O)N(CC(O)CN(C(=O)CCNc2ccccc2)C)C)cs1 c1(CC(=O)OCC)cc(Br)c2c(c1)CCO2.c12ccsc1CNC(=O)C2 C(=O)(C(F)(F)C(F)F)NC1CN(C(C(CC=C)OC)=O)CC1F O=C(C(O)C(F)(F)F)NCc1cccc(-c2cc[nH]n2)c1 N1(C(CC2C(CNC(CC=CCC)=O)C2)=O)CCCC(CCO)CC1 Cc1noc2ncnc(N(CC(O)CN(C)C(C3CCC(C)C(C)C3)=O)C)c12 C1(NC(C=CC=CCC)=O)CCN(C(=O)C(C)(C)C)CC1CO c1(C(C(=O)NCC(=C)C)N(C)CCC2(C)OCCO2)nc(Br)cs1 C1(CNC(CN(CC(=O)NC(C)C)C)=O)COC2COCC12.C12(C)CCCN1C2=O CC1CCN(C(=O)Cn2cc(C3CCOC3)cn2)C(C)C1NC(=O)C=CC(N)=O C(=O)(CCS(=O)(=O)NC)N(CC(C)NC(=O)C1=CCCSC1)C.C(C(N)=O)NCC#N CCC(C)C(O)C(=O)Nc1cccc(NC(N2CCCC2)=O)c1 c1(NC(C2CCN(Cc3c(C(=O)OC)cccn3)C2)=O)cc(F)c(Cl)cc1F Cc1nc(C(C)C)nc(O)c1C(=O)NC(CCN(C(=O)C1=CCCS1)C)C(C)C Cc1nc2c([nH]1)CC(NC(c1[nH]ccc1-c1ccccc1Br)=O)CC2 Cc1c[nH]c(C(=O)NCC2(C(=O)NC3CC(CC(N)=O)C3)CCCO2)c1C c1(C(N2CC3(CC(C(=O)Nc4c(SC)cccc4)C3)C2)=O)cc(Br)cc(Cl)c1F C(C)(C(CC(=O)NCC1CCOC1C)NC(C1CCC1C(C)(C)C)=O)OC N1(C(COC(CC)(C)C)=O)CC(N(C(=O)CN2CCC(O)CC2)C)C(O)C1 C(=O)(CCC(N)=O)NCC1(NC(c2n(COC)ncc2)=O)CCOC1 N1(C(C2(SC)CCC2)=O)CCC(C2CCN(C(c3cc4scc(C)c4[nH]3)=O)C2)C1 c1(C(=O)OC)ccc2c(c1)C(NC(=O)NC(C)C(=O)NC(C)(C)C)CC2 N1(C(c2c(OC)scc2)=O)CC2(NC(C3OCCC3C)=O)CCCC2(F)C1 C1(CN(C(=O)C(N2CCCC(F)CC2)=O)CC2CC2)CCC2(CCCCCC2)O1 N1(C(CC2(NC(CCC)=O)CC2)=O)CCC(CCCO)C1.C1C(=O)N1 CS(=O)c1ccc(CC(=O)NC2CC(NC(c3ccc(N)c(Cl)c3O)=O)C2)cc1 C=C(F)C1(CC(N2CCN(CCNC(=O)CSc3n[nH]c(O)n3)CC2)=O)CCC1 C(=O)(C=C1SCC(=O)N1C)N1C(C)CC(CNC(=O)C2=CC3CCCC23)C1 c1(OCCC(=O)NCCCCNC(c2ccc(C)cn2)=O)ccccc1[N+](=O)[O-] N1(C(C(C(C)C)F)=O)CC(N(C(=O)C=CSCc2ccco2)CCO)CC1(C)C c1(CC(=O)N(CC(CNC(C(CC)C)=O)(C)C)C)c[nH]c2cc(F)ccc12 c1(CCC(=O)NCC2CC(CNC(C=CCCC)=O)OC2)ccc(O)cc1 C1(C)(C(=O)NCC(n2cc(C3(C)CCCC3)nn2)C)CCCS1 N1(C(=O)C=CC2CCCCCC2)CC2CCN(C(C3C=CCS3)=O)C2C1 Cc1cc(C(=O)NCC2CC(F)(CNC(=O)C(C)Oc3cccnc3)C2)sn1 c1(Nc2c(C)c(N3CCC(C4CCCC4)C3)ncn2)ccc2oc(=O)n(C)c2c1 c1(C(=O)NCCCOCCCNC(C(C(C)(C)O)F)=O)cn2cccnc2n1 Cc1cc(C(=O)NCC(C)CC(=O)NC2CC3CC3C2)nc(O)c1 n1(CCC(=O)NCCN(C(=O)CC2CCC3CC23)C)cc([N+](=O)[O-])cn1 N(C(=NCCC(C)C)NCc1cn(C2COC2)nn1)CC1CCC(=C)CC1 c1(C(N2C(CNC(c3ccc(=N)[nH]c3)=O)CC(OC)C2)=O)cc(C)c(C)c(F)c1 C=CCCCCCC(=O)N1CCN(C(=O)C(C)(CC)OC)CC(CO)C1 N1(CCNC(C2C(CNC(Cc3cn(CNC)nc3)=O)CC2)=O)CC2CCC1C2 N1(C(C(c2cccc(C)c2)O)=O)C2CCC1CC(O)(CNC(=O)CCF)C2 c1(OC)ccccc1CCC(=O)NC1CC(NC(=O)Cc2ccc(Br)nc2)C1 C1(C)(CC)CCCN(C(=O)CC2CCCC2NC(=O)Cc2ccc(C)cc2)C1 C1(C(=O)NC2(CC)CCN(C(C3CC34CCC4)=O)CC2)CCCCN1S(N)(=O)=O CC1=C(C)CC(C)(NC(c2cc(CN(C(C3(CCCF)CC3)=O)C3CC3)[nH]n2)=O)CC1 C(=O)(CC(C)C(C)(C)C)N1CCC(C=C)(C(=O)NCC(c2cnc[nH]2)C)C1 C1(C2CCN(C(=O)Cc3cc[nH]c3)C2)(NC(c2cc(CCC)c(C)s2)=O)CC1 N(C(=NC)N1CCC(SC(C)(C)C)C1)Cc1[nH]nc(COCC)n1 C12CN(CC(C)(C)OC1=O)C2.C1(OCC)CC(CN(C)CCC2CC2)C1.C1CO1 CC(C)CC(O)CC(=O)NC(C)(CNC(=O)C=CCO)Cn1cccn1 Cc1cc(F)sc1C(=O)NC(C)CNC(C1CC12CCC2)=O CC(C)C(O)C(=O)N(CC(C)CNC(=O)Cc1ccc(SC2CC2)cc1)C c1(C2N(C(Cn3cc(-c4nc(CC)sc4)nn3)=O)CCC2)cccc(C(C)C)c1 N1(C(C2C(C)C2C)=O)CCCC1CCNC(=O)C(F)n1ccnc1 C1(c2ccc(C)cc2)NC(=O)N(CCCNC(c2nnnn2C)=O)C1=O c1(C(N2CCN(C(C=CC=CC)=O)CC(O)C2)=O)ccnc2c1ccn2C c1(C(=O)NC(C)CNC(=O)CC2C=CCC2)ccc(CC(=O)OC(C)(C)C)cc1 C12(C(N(CCCNC(c3c(C)nc(C(C)C)s3)=O)C(C)C)=O)CC=CC(C1)OC2 CC1CCN(C(c2cccc3nn[nH]c23)=O)C(C)C1NC(c1cncc(Cl)n1)=O C1(C(=O)OC)C2CCC1CN(C(=O)CN(C)C(=O)Nc1cc(Cl)cc(Cl)c1)C2 c1(N2CCC(OCCNC(C3C(CC)C3)=O)C2)cc(C)nc(C(C)(C)C)n1 C1(OC)(CNC(=O)N(C)Cc2oc(CO)cc2C)CCCC(C)C1 C=C(C)C(CC(=O)NCCOCCS)OC.C(=O)(CS(=O)CC)N1CC(N)C1 CN(CCCC(=O)NCC1CC1NC(=O)Cc1cc2ccccc2o1)N=O C1(C(=O)Nc2ccc(CCF)cc2)(CC)CCCN(C(c2ccn(C)c2)=O)C1 CC(F)(F)C(F)C(=O)NCCCC1CN(C(C2CCC(CN=[N+]=[N-])C2)=O)CCO1 N1(C(C2CC(F)CN2C(c2cc(F)c(F)c(Cl)c2)=O)=O)Cc2ccc(F)cc2C1 C1(CC(=O)NCC(CC)NC(c2ccc(OC)c(C)c2)=O)CCCC2(CCC2)O1 c1(C(=O)NC23C(CN(C(C(C)(C)c4ccc(Cl)s4)=O)C2)C3)cc(N)c(Cl)cn1 N1(C(C2(CC)CCC2)=O)CC(NC(c2cc(N)ccc2Cl)=O)C2(CC2)C1 N1(C(CN(C(C(C)C)=O)C)=O)CCC(C)(NC(C2(C(C)C)CCCO2)=O)C1 C1(NC(C2(CCCC)CCCC2)=O)CCN(C(c2cnoc2C)=O)CC(O)C1 CC(CCN=c1ccc(S(C)(=O)=O)c[nH]1)NC(=O)CCc1cn[nH]c1 O=C(C1=C2CCN=C2NC=C1)NCCN(C(C1CCCCC1)=O)Cc1cccs1 C1(C)(NC(CC2C(NC(C3(OCC)CC3)=O)CC2)=O)CCCC1O N(C1CCCc2occc21)C(C1CCCCN(C(C(CCC=C)(C)C)=O)C1)=O N1(C(c2cc(C)[nH]c2)=O)CCCC(C(=O)NC(c2cc(C)on2)C)CC1 C(=O)(C1=CCCN(C(=O)C=C2CCCCC2)C1)NCC(C#C)CC C1(C(=O)NCC(C)NC(c2cccc3c2OCCO3)=O)Cc2c(F)cccc2O1 C1(ONC(=O)C2CC2)(NC(=O)CC2CCC(=O)O2)CCCCC1 N1(C(C(CC)Nc2nc(C)cs2)=O)CCC(C2CN(C(=O)CCSCC)C2)CC1 Cc1c(C(F)(F)F)cc(C(N2CCN(C(=O)CCF)C3CCC23)=O)cc1[N+](=O)[O-] C1(NC(C2CCC(C)CC2)=O)CCCN(C(C2(c3ccno3)CCC2)=O)CC1F Cc1cc(NC(=O)NCC(c2ccc(F)cc2)C)cnc1C c1(CCC)sc(C(N2CC(CNC(=O)CC(C)O)C(O)C2)=O)cc1CC N1(C(C(C)OCCOC)=O)CCCC(CO)(NC(=O)C(C)c2cccs2)C1 c1(N2CC3N(C)C(CCC3)C2)nc(=NCC2(N(C)C)CC2)[nH]c2ccsc12 c1(C(=O)OC)cnn(C(C)(C)C)c1Cl.C12COC(C1)CNC(=O)C(=O)N2 C1(C(CNC(COCCSC)=O)(C)C)CCN(C(C2CCCC2OC)=O)CC1 c1(C(=O)OCC)c(N2CCN(C(C3CC3C(C)O)=O)CC(O)C2)cc(C)nc1O CCCCC(=O)C(=O)N(CCCN(C(=O)C(C)c1cc[nH]n1)C)C N1(C(C2CC(=C)C2)=O)CC2CC(NC(=O)C(C)(O)c3ccccc3)C(C2)C1 c1(CNCC(N2CCCC(NC(C3(SC)CC3)=O)C2)=O)ccsc1[N+](=O)[O-] N1(C(c2cc(C)ncc2C)=O)CC2CCC1C(CNC(C1CC1F)=O)C2 C12(CN(c3cccn3C)CCNC(C)=O)CC3CC(C1)CC(O)(C3)C2 c1(C(=O)NCCOC)ccc2[nH]c(C(=O)Nc3c(C)cc(C)nc3Br)cc2c1 Cc1cc(C)c(CC(=O)N(C2CCN(C(=O)COc3ccc(F)cc3)C2)CC)s1 C1(c2cn(CCC3CN(C(C4OCC(C)C4)=O)C3)nn2)CCCC(F)(F)C1 CCC(CCC(=O)NCCn1cc(C(=O)NCCNC(=O)CC)cn1)OC N1(C(c2c(NC)cnnc2)=O)CCCC(C(C)C)CC1.N12CCCC1C=CC2=O NS(=O)(=O)CCCC(=O)N1CCC(O)C(NC(=O)C(O)c2ccsc2)C1 CCC(O)(CC(=O)N1CC(NC(=O)CCn2ccnn2)C(O)C1)c1ccccc1 Cc1cn(C)nc1C(=O)NC1(C(=O)NC(C(N)=O)C2CCCC2)CC1C Cn1[nH]c(C2CCN(CCN3CCOCC3)CC2)nc1=N N1(C(CC2(C)OCCO2)=O)CCC(CF)(NC(=O)Cc2cc(C3CC3)no2)C1 Cc1ccc(COCC(=O)NCCCCN2CCN(C(C3(Cl)CC3)=O)CC2)cc1 Cc1cc(C(=O)NC(C)CC(C)NC(=O)Cn2ccsc2=N)c2c(c1)CCO2 CCC(C)C(CC(=O)OCC1N(C(=O)COC(C)(C)C)CCCC1(C)C)OC c1(CC)cccc2c(F)c(C(N3CC4C(NC(=O)C=C(Cl)Cl)C4C3)=O)[nH]c12 Cc1ccc(Cl)cc1C(=O)NC1(CNC(C2CCN(CC(C)C)C2)=O)CCCC1 N1(C(c2c(F)ccc(N)c2)=O)CCCC(C2CCCN(C(=O)C(F)(F)CO)C2)C1 c1(OC(C)C)n[nH]c(C(=O)NC2CN(C(=O)Cn3cnc(=N)[nH]3)CC2F)c1Br C=CCCC(F)(F)C(=O)N1CCC1(C)CC(=O)NCCN1CCCC(O)C1 c1(NC)ccc(C(=O)NC(C)C(C)NC(=O)C(C)N(C)C(C)=O)cc1[N+](=O)[O-] N1(C(c2ncc(C)nc2)=O)CCC(CNC(=O)CN(C)C(N)=O)C(C)C1 C1(NC2CC(C(F)F)(OC)C2)CCCCC(F)(F)C1OC(=O)OC(C)(C)C c1(C(N2CCC(F)(CNC(C3(CF)CCC3)=O)C2)=O)cccnc1F C=CCCCC(C)(C)C(=O)N1CC2CCC(C1)C2NC(C1CCN(C)C(=O)C1)=O C1(C)(CCOC)COCCN(C(c2cn(C3CC3)nn2)=O)C1.C1(NC=O)CCCC1O c1(C(C)NC(C2N(C(C(CSC)OC)=O)CCCC2)=O)ccc2ccccc2c1 C(=O)(CC(F)(F)C(C)C)N1CC(CCC)N(C(c2nnn(C)c2C(F)F)=O)CC1 C1(C(C)NC(c2ccc(C3CCCCC3)o2)=O)CN(C(=O)C2CC2)CCO1 CC(CS(C)(=O)=O)C(=O)N1CC(O)(CN(C)C(C2(CO)CCOCC2)=O)C1 c1(C(N(C2CN(C(C3CC4(CSC4)C3)=O)C2)C)=O)nnc2ccccc2c1N C1(CNC(C(COCC)C)=O)CN(C(c2ccccc2OC2CC2)=O)CCN1C c1(C(N2CC(NC(CC3(C)CC3(F)F)=O)C2)=O)ccc(C(=O)CF)cc1 c1(CC(N2CCC(C(=O)Nc3cn(CC4CC4)cn3)C2)=O)cc(C2CC2)nn1C c1(C(N(CC(C)N(C(=O)CC2CCN(C)C2=O)C)C)=O)cc2n(n1)CCC2 Cc1nc(N2CC3CCCC(NC(C4CC(C(C)C)C4)=O)C3C2)ccc1[N+](=O)[O-] N1(C(CN(C(C(C)C)=O)C)=O)CCC2CN(C(=O)CN3CCN(C)C(=O)C3)C2C1 C1(CC(=O)NCC2CC(=O)NC2)CC(NCC2CC(F)(F)C2)CCO1 CC1(C)COCC1C(=O)NC1CN(C(C2CC3CCC(C2)C3)=O)CC1O CCC(C)(CNC(C1CCC(=O)O1)=O)C(=O)NC(c1nnc(C)o1)C C1(CC(=O)NC(C2CN(C(C3C4CCC(=O)C34)=O)CCO2)C)CC2(CCC2)C1 c1(OC)cc(C(=O)NC2(C)CN(C(c3cnccc3C)=O)C2)c(F)c(Cl)c1 c1(OC)ccc(C2CCN(C(c3cc(-c4cccc(F)c4)on3)=O)CC2)nc1 CCC(CC(F)F)C(=O)NCC1CN(C(=O)CC(C)C(=O)OC)CC(C)(C)O1 C(CC(C)N=c1[nH]c(C(C)C)nc2[nH]ccc12)NC(c1c(C)ccnc1)=O C1(C(=O)NCCC2CC(NC(CC(C)O)=O)C2)CCC(C)(C)OC1 c1(CCOC)nc(=NCC2(O)CCCN(C(=O)CCNC(C)=O)C2)s[nH]1 Cc1cc(C)c(C(=O)NCCC(C)N(C(=O)CCC(F)F)C)cc1N C1(C(=O)NCC2CCC(C(N(c3ccc(OC)cc3)C)=O)C2)CCOC(=O)CC1 Cc1cccc(CC(=O)NC(C)CCNC(C2(S(C)(=O)=O)CC2)=O)c1Br Cc1ncc2n1CCC(C(=O)NC(C)CNC(C1CC1C(C)O)=O)C2 N1(Cc2scc(C)n2)C2CCC1CC(NC(c1cccnc1Cl)=O)C2 c1(C(=O)NC2CC3CN(C(C=CC)=O)C(C2)C3)cccc2[nH]nc(O)c12 N1(C(C(=Cc2cn[nH]c2)C)=O)CCOC(CCNC(=O)CC2CCC(=O)N2)C1 c1(C(=O)OC)ccc2c(c1)CCN(C(C1CC1NC(c1cc(C)nn1C)=O)=O)C2 C(CC(C(C)(C)C)NC(C1CC1c1ccco1)=O)N(C(C(C=C)(C)C)=O)C C1(=CC(=O)N(CC(C)NC(=O)CSCCN(C)C)C)CC2CCC(C1)N2C C(CCC)(C(=O)N(C1CCCC1C)C)NC(COCCCC#C)=O C(=O)(C1CCCc2n[nH]cc21)N(CC(C)CNC(=O)Cc1cccnc1Cl)C c1(C(N2CCN(Cc3c(C)nn(C)c3Cl)CC2CC#N)=O)nc2ccccn2n1 Cc1nc(C)c(C(=O)NCCOCCOCC(O)CN(C)C)o1 c1(C(N2C(CCC#C)CCC2)C(=O)NCC)ccc(N(C)CC=C)c([N+](=O)[O-])c1 C=CCC(CC)C(=O)NC1CCN(C(c2cc(OC)cc(F)c2)=O)C1C(C)(C)C c1(OC)ncccc1N(C(=O)CSc1cccc[n+]1[O-])C c1(OC(C)C)cnc(C(=O)NCCCCNC(=O)CC2CC3C=CC2C3)cn1 c1(C(N(CC(C)(C)NC(CC2CC(=C)C2)=O)C)=O)cc(Br)cs1 CCC(C)C(O)CC(=O)NCC1CC(NC(=O)CNS(=O)(=O)c2cccnc2)C1 CC1(C(N2CC(OC(=O)Nc3cccs3)C2)=O)CCc2ccccc2C1 C(C(CC(C)C)C(=O)NCc1ccc(C(=O)NC(C2CCCO2)C)nc1)OC c1(C(=O)N(C(C#C)C2CC2)C2CC2)occc1CNC(=O)Cc1cccs1 N1(C(C(C)C2CCOC2)=O)CCC2(CC1)CC(Nc1snc(Cl)c1C#N)CO2 c1(CC(=O)NC2C=CCN(C(c3cc(O)ncn3)=O)C2)cc(F)cc(Br)c1 C(C(=O)N1CC(O)(C(C)(C)CNC(C2(C3CCCO3)CC2)=O)C1)(C(C)(C)C)SC CC(CCC(=O)N1CCC(CNC(=O)Cc2cncnc2)C12CC2)S(C)(=O)=O C1(C)(CC)CN(C(c2[nH]cnc2C)C(=O)Nc2ccc(F)cc2C)CCO1 CCCC1C(=O)N2CCN(CC2)O1.C1(NC(C2(SC)CC2)=O)CCN(C)CC1 C1(CNC(CCCC(C)=O)=O)COC(C)(C)CN1C(=O)CC1CCOC1=O C(C(O)C(=O)NC(C)CC(=O)NCCc1ccon1)=CC N1(C(C2C(CNC(c3ccc(CC)nc3)=O)CCO2)=O)CC(O)CC12CCC2 C(=O)(C(CC1CCCC1)NC(=O)CC(C)N(C)C)N(CC(=O)NCCC)C c1(C(N2CC(Cn3cc(-c4c(F)cncc4F)nn3)C2)=O)ccnc2ncnn12 N1(C(C2(OC)CCC2)=O)CC(CCNC(=O)C(O)Cn2cncn2)C(C)C1 N1(C(=O)CC2CCCO2)CCC(O)(C2(NC(C34CCCC3C4(F)F)=O)CC2)CC1 CC1(C)CCC(CC(=O)NCC2(NC(C3CC(C#N)C3)=O)CC2)OC1 Cc1cnc(C(N2CCOCC2CNC(=O)CCS(C)(=O)=O)=O)c(C)c1 N1(C(C(COC)OC)=O)CCCC(CO)(NC(=O)Cc2cnoc2)C1 C1(NC(c2csc(Cl)n2)=O)CC2CCC1CN(C(=O)C1CCc3c[nH]nc31)C2 N1(C(C(C2CCCCC2)C)=O)CC2CC(NC(c3ccc(Cl)s3)=O)CC1C2 c1(OC)cnc[nH]c1=NCC1(O)CCCN(C(c2ccccc2SCCO)=O)C1 C(=O)(C(C)(C)C(=O)N1CCCCC1CNC(c1csc(C(F)F)n1)=O)OC n1(CC)nnc2c1C(C(=O)NCc1ccc(F)cc1F)CN(C(C1CCC1)=O)C2 Cc1cc2nc(N(C(C)C(C)C)Cc3cccnc3)sc2cc1C O=C(C1CCc2ccccc21)NCC1CCCN1c1nc2c(F)cc(Cl)cc2s1 c1(N(C)CCn2cnnc2)nc(NCCc2cccc(F)c2)c2ccsc2n1 n1(CC(=O)NCC2(F)CCC(NC(C(CCCC)O)=O)C2)ncc2ncccc12 N1(C(c2[nH]cc(C)c2)=O)CC(NC(C2(C(F)F)CCCO2)=O)CCC1C C(C(F)(F)C(=O)N1CC(C)(c2ccccc2)C1)OC N1(C(c2c(C)cn(C)n2)=O)CC2CC1CCC2NC(=O)Cc1c[nH]nc1C Cc1cnc(C(N2CC(NC(C3CC34CC4)=O)CC23CCC3)=O)cc1C#N N1(C(C(C)Cc2ccc(Br)cc2)=O)CCOC2C(C(=O)OC(C)(C)C)CC12 c1(C(N2CCCC(N(C(C(C(=O)OCC)F)=O)C)C2)=O)nc2ncc(C)cn2n1 N1(c2ncnc(CC)c2F)CCC2C(CCN2C(c2cccnc2)=O)C1 NS(=O)(=O)CCc1cn(C2CCN(C(c3ccn(CC(F)F)n3)=O)C2)nn1 C1(NC(C(C)OC)=O)COC2(C1)CN(C(c1c(N)cc(Cl)cc1Cl)=O)C2 N1(C(CNC(CNC(C)=O)=O)=O)CCOC(CNC(C2(CO)CCOC2)=O)C1 C1(NC(c2c(NC)cncc2)=O)CCN(C(=O)C(F)(F)COC)CC1F c1(CCC(=O)NCCC2CCN(C(C3(F)CCOC3)=O)C2)ccc(F)cc1 c1(OC)ccc(C2(C(=O)N(c3nccs3)C)CC2)cc1OC C1(NC(c2cc(C)n(C)n2)=O)CC2CC(NC(c3cnc(Cl)c(N)c3)=O)C1C2 C(=O)(C(C)C(C)COC)NCC1(NC(c2n[nH]c(CC)c2Br)=O)CC1 Cn1cnc(=N)[nH]c1=NCc1ccn(C2CCCCCC2)n1 Cc1cccc2c(N(C(=O)C=Cc3ccc(F)cc3)CC3CCNC3)ncnc12 C(=O)(CC1=CCCC1)N(C(C)CNC(=O)C(c1cc(Cl)ccc1F)(C)C)CC Cc1ccc(CNC(C2CC2C(=O)Nc2oncc2C#N)=O)c(F)c1 Cc1cc(C)nc(N2CC(NC(c3cn(CC4CCCO4)nn3)=O)CC2C)n1 N1(C(CCC2CC(NC(C3(C)N(C)CCC3)=O)C2)=O)CC2CC3CC2C1C3 C1(CNC(c2c(CC)scc2)=O)CCN(C(c2c(C)nsc2C)=O)CC1C C1(NC(COCCCC(C)C)=O)C2CC3CN(C(C4CCCC4(C)C)=O)C1C3C2 c1(C(=O)NC2C(C)N(C(=O)CC3CC3(C)C)CC2)c(Cl)c([N+](=O)[O-])nn1C C1(NC(c2nc(CC)sc2)=O)CC2CC1CN2C(c1ccccc1CC)=O CCCCN=c1[nH]c(=NCCC2CCCCN2C)[nH]c2cccc(F)c12 C(=O)(C(CC(C)(C)C)NC(c1cc(O)n(C)n1)=O)NC1CN(C)C(=O)C1 C(C(=C)CCNC(c1n[nH]cc1C)=O)NC(C=CC)=O C1(N(C(=O)COCc2ccccn2)C)CN(C(=O)CN2CCSCC2)CC1(C)C C1(S(=O)(=O)c2ccccc2)(C(=O)OCC2CCCCCO2)CCC1 C(CC1=CCCCC1)NC(C1CCCN(C(CCSC)C(=O)O)CC1)=O c1(CC(=O)NC(C2CN(C(C(COC)(C)OC)=O)C2)C)cc(F)ccc1C C1(C(=O)NCC2(NC(CCC=C)=O)CC3CCC2CC3)Cc2c(C)cccc2O1 c1(C(=O)NC2CCN(C(c3cc(CC)on3)=O)CC2)cc(C)c(O)c(C)c1 CN1C(=O)CCC1CC(=O)NCc1ncccc1C(N1CCC(C)(F)C1)=O c1(C(=O)NCCOCCNC(C2CN(C)C(=O)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(C(N(C2CCCN(C(=O)CCCc3ccsc3)C2)CC)=O)CCOC(C)(C)C1 C1(N(C(=O)C(F)(F)F)C2CN(C(C(CC=C)CC)=O)C2)CC2(CCNCC2)C1 Cc1cc(C(=O)NCC2CC2NC(=O)CC2(n3cncn3)CC2)cnc1C(F)F C(=O)(C1=NN(C)C(=O)CC1)NC1CCC(N(C(c2nc(CCC)oc2)=O)C)C1 C(C(C)N=c1[nH]c(CC)nc(Cl)c1C)(C1CCCCC1)OCC C1(NC(CCC2CCN(C(COCCCCC)=O)CC2)=O)C(C)(C)C(O)C1(C)C C1(C2(O)CCN(C(=O)C=CCF)CC2)(NC(C(C)NS(C)(=O)=O)=O)CC1.C(C)(C)C C(=O)(CCCC(C)=O)N1C(C(=O)NCC2(F)CCCCC2)(COC)C=CC1 c1(OCC)cccc(C(=O)NC2CCC(CNC(=O)CNC=O)C2)c1N C1(NC(c2cnc(OCC)nc2)=O)CN(C(=O)CC(=O)OC(C)(C)C)C(C)(C)C1 C(C1(O)CCc2ccccc21)NC(=NCC(C=C)C)NCC1CCC1 c1(NC(C2CN(Cc3cccc(Br)c3Cl)CCC2O)=O)cccc(F)c1[N+](=O)[O-] C1(C(C)N(C)C(C2CC(CCNC(=O)CC(C3CC3)C3CC3)C2)=O)CCOCC1 CC1CN(C(=O)CCC2(C)CN(C(C3CCN(C)CC3)=O)C2)CC1(F)F CC1COc2c(C(=O)NC3CCCC3NC(=O)CCCC(N)=O)cccc21 CC1(C)C=C(C(=O)N2CC(NC(c3cc(-c4cccs4)[nH]n3)=O)CC(F)C2)C1 c1(C(=O)Nc2c(C(=O)NCCOCCOC)scc2)cc(Br)ncc1Br C12(CC(=O)NCC3C(CNC(c4nn(C)c(F)c4)=O)C3)CCC(CC1)CC2 c1(C(N2CC(C)C(CNC(=O)CCCC(F)F)C2)=O)coc2c1C(=O)NCCC2 C1(C(=O)NC2(CSC)CCC2)CCN(C(c2cnnc(O)c2)=O)CCO1 C1(OC)CC(CNC(C2CCN(S(C)(=O)=O)CC2)=O)N(C(=O)CC2CC(F)C2)C1 C1(C(N(C)CC2CCSC2)=O)CN(C(C2(C#N)CCCO2)=O)CCN1C c1(OC)cccc(CCC(=O)NC(C)CC(C)NC(c2ccsn2)=O)c1F N1(C(Cc2ccc(C)c(C)c2)=O)CCC2CN(C(C3(C)CCCN3C)=O)CC2C1 C1(C#N)(C(=O)NCC#CC(=O)N(C)CC2CCCS2)CC(=O)C1 c1(SC(C(=O)OC(CCC)C)C)ccc(Cl)cc1 C1(C)(NC(C(CNC(C2N(CC)CCC2)=O)N(C)C)=O)CC(C)(C)C1 C1(NC(CC2(C)N(C(c3cc(C)cc(O)n3)=O)CCC2)=O)CCn2ncnc2C1 c1(C(=O)NCC(CC(C)C)NC(C(C(CC)O)C)=O)nc(N)cc2ccccc12 CC1(C2CC2)CN(C(c2cc(CNC(=O)CCN=[N+]=[N-])cs2)=O)CCO1 C1(NC(C2CCN(C)C2)=O)CN(C(c2cc(C(C)(C)C)on2)=O)CC2(CC2)C1 C1(C(=O)NCC(CSC)(C)C)C2CCC(C2)N1C(=O)C(C1CCCCC1)C c1(NC(C2CCC(NCc3cccc4cc[nH]c34)CC2)=O)c(Cl)cc(Cl)cc1Br C#CCCCCCC(=O)N1CC=CC1CNC(=O)Cc1cc(F)ccc1Cl N1(C(c2c(C)c(Cl)ccn2)=O)CCC2(CCCCC2NC(c2cc(Cl)no2)=O)C1 N1(C(C2C=C(C)CS2)=O)CC(C(=O)Nc2cc(C)cc(O)c2)CCC1(C)C c1(N2CCCC(CSC)C2)nc(N(CCS(N)(=O)=O)C)nc2ccc(Cl)cc12 c1(C(=O)NC2C(C)(C)CN(C(=O)CCC(F)(F)F)C2)ccc([N+](=O)[O-])cc1F N1(C(CCc2nc(C)sc2)=O)CC(NC(=O)CCc2scnc2C)CC12CCC2 C1(NC(c2cnnc(O)c2)=O)CCN(C(C2(O)CCCCCC2)=O)CC1CO Cc1cc(-c2csc(C(N3CCn4cccc4C3)=O)n2)c(F)c(F)c1 C1(CC)CN(C(C2CN(C(C)C)C2)=O)CC1C(=O)NCCSC c1(CC(=O)NC2C(NC(C3(CC)COC3)=O)C2)cccc(OC)c1 O=C(CCCC(=O)C1CC1)NCc1cc(C(=O)NCc2cncs2)on1 C1(C(=O)NC2CN(C(=O)CC3CNC(=O)O3)CC2CO)(CC)CCCC1O C#CCC(C)(C)C(=O)N1CC(CNC(c2ccccc2C(C)C)=O)C(O)C1 Cc1ccc(F)c(CC(N2CCC(C)(NC(C3CC34CC4)=O)CC2)=O)c1 c1(C(=O)NCCOCCNC(CC2(C)CCCO2)=O)cc(Cl)ccc1-n1cncn1 Cc1cc(C(=O)NC2CC(NC(=O)Cc3cc(C)on3)C2)c(C)cn1 CC#CCCCC(=O)NC(CC)CCC(=O)NC(C)(COC)CO N1(C(c2cnc(SC)s2)=O)CCOC(CN(C(=O)C=Cc2cnc[nH]2)C)C1 Nc1cc(F)cnc1C(N1CCN(C(=O)CSc2ccccn2)C(C(F)F)C1)=O C1(CCNC(C2C(C(=O)OC)CCC2)=O)CN(C(=O)Cn2nnnc2C)CCO1 CC1(C)CCCC(C(=O)NCC2CN(C(c3ccnc(F)c3N)=O)C2)CC1 C1(C(N(C)Cc2ncn(C)n2)=O)(CNC(=O)CC2CCCO2)CC12CCC2 c1(CCC(=O)N(C(=O)CSc2ccccc2)CC)cc(C)nc(C)c1 C(=O)(CCCNS(C)(=O)=O)NCCN(C(C(C)OC1CCCC1)=O)CC(C)O C1(C(N(C(C)COc2cnn[nH]2)CC)=O)(CC)CN(C(=O)C(C)OC(C)C)C1 C(C)(C(=O)N1CC(NC(=O)C(C)(C)CO)CC(F)C1)(C(C)C)OC N1(C(C(C)OCC=C)=O)CCC(CCCCNC(C2C3CC4C(C3)C24)=O)CC1 c12nc(cs1)CC(=O)NCCN2C(=O)C(C)=CC1CC1.C(=O)OCC.OC CCC(C)C(C(=O)NC)N(C=O)Cc1cncc(OC)c1 N1(C(CN(c2ccncc2)C)=O)CC(CNC(C2CCCSC2)=O)C2(CCC2)C1 Cc1cc(=O)oc(C)c1C(N1CC2CC1C2NC(C1CCC(C)(C)O1)=O)=O C1(O)(CNC(=O)CCc2cn[nH]c2)CCN(C(c2ccccc2SC(F)F)=O)C1 C1(OC)CC2(C1)CN(C(=O)CNC(=O)C(F)CC1CCC1)C2 C(C(C)(O)CC(=O)NC1(CCNC(c2cnc(-c3ccco3)s2)=O)CCC1)OC N1(C(C(C(C)C)(C)C)=O)CC(NC(C2(C)CC2(F)F)=O)CCC(O)C1 c12cc(cc(F)c1)CNCC1C(C1)C(=O)NC2.OC(F)(F)F.O=C(CNCC)OC c1(CCCNC(C(N2C(CC)CCC2)=O)=O)nn(C)c2c1CCCC2 c1(C(=O)NC2C(NC(=O)CC3CCCOCC3)CC2)csc2nnsc12 N1(C(C2CC(=O)NCC2)=O)CCN(C(c2cccc3nccn23)=O)CC(O)C1 N1(C(c2n(COC)ncc2)=O)CC=C(C(C)(C)C(=O)N2CCC(F)(C#N)C2)C1 c1(SC)cc(C)c(C(=O)NCC(CNC(C2CC2(F)F)=O)CO)o1 N1(C(Cc2ncc(C)s2)=O)CCC(NC(C2CC23CC3)=O)C(O)C1 c1(C(=O)NC(CNC(C2CC(C)=C(C)CC2)=O)CO)n[nH]c2c1CCSC2 C1(C(=O)NC2CCN(C(C(C)OCCOC)=O)CC2C)CCC(C2CC2)CC1 c1(SC)ccccc1C(N1CC(CCCCNC(C2CN(C)CCO2)=O)C1)=O N1(C(CNC(C(CC)C)=O)=O)CCOC(C)(CNC(=O)CCS(C)(=O)=O)C1 Cc1cc([N+](=O)[O-])ccc1C(=O)NCC(C(C)C)NC(C1CC1C#N)=O Cc1cccc2cc(C(=O)NCC3CCCN3C(c3cc(Cl)ncc3O)=O)sc12 CCC(O)C(=O)N1CCC(C(=O)NC2CSC2)C1 c1(C(=O)OC)ccc([N+](=O)[O-])c(NC2CC(N(C(=O)C(C#N)=CC3CC3)C)C2)c1 c1(CC)ccc(C)cc1NC(=O)C(O)C(C)(C)NC(=O)OC(C)(C)C N1(C(=O)COCCc2nccc(-c3ccccc3)n2)CCN(CC(O)CO)CC1 c1(C(=O)NCC(CC)NC(c2conc2C)=O)c[nH]c2cccc(F)c12 C1(C(N2C(CN(C(Cn3c(C)nnn3)=O)C)COCC2)=O)CC2(C1)CC21CC1 N1(C(c2c(CC)cno2)=O)CC2CCOCC2(NC(c2cncc(NC)c2)=O)C1 C1(CNC(c2ccc(Cl)nn2)=O)CCN(Cc2cc(Cl)c(O)cc2F)CC1(F)F C(=O)(C1=Cc2ccccc2C1)N1CC(C(=O)NCC(COC)(F)F)CC12CCC2 CC1C(C(=O)NCCC2CC2)CCCN1C(c1cc(F)cc(Cl)c1)C(=O)N(C)C Cn1cc2c(n1)CC(C(=O)NC1CCC(CCNC(=O)CNC=O)C1)NC2=O CC(F)CC(=O)N(C(c1ccccc1)CNC(=O)Cn1ncnn1)C c1(CN(C2CCC2)C(C2CCN(Cc3cnn[nH]3)C2)=O)ccn(C(C)(C)C)c1 CC1CCC2(CC1)CCC(CSc1nc(C3CNC(=O)CC3(F)F)no1)O2 c1(C(=O)NC2C(CNC(c3c(C)n[nH]c3)=O)CCC2)cc2cccnc2nc1O C#CCC(C)C(=O)N(CCCNC(c1ccoc1I)=O)C c1(N2C(CCCNC(C(C)NC(COC)=O)=O)CCC2)nc(Cl)nc2[nH]cnc12 c1(CC)nocc1CN(C(=O)COCCNC(=O)Cc1ncoc1C)C N1(C(C23CC(n4cc(COc5cccc(N)c5)nn4)C2C3)=O)CC2COCC2C1 CC1(C)COCC1C(=O)NC1CC2(C1)CC2NC(C1CC1c1ccco1)=O C1(c2nc(C)on2)CCCN(N2CCCC2(C)C2CCCCC2)C1 CCC(C)CCCCC(=O)NCC1CCC2(CN(C(c3ccc(F)cc3)=O)C2)O1 c1(C(C)=O)cc(CNC(CC2N(C(C34CC(CSC)(C3)C4)=O)CCC2)=O)oc1C CON=Cc1ccc(C(N2CCC(C)(NC(=O)C#CC3CCCO3)CC2)=O)cc1 C(=O)(C(CCOC)NC(C12CCCC1C2)=O)NCC1CC(CCOC)C1 Nc1cc(C(=O)NC2CCC2NC(c2n[nH]cc2Cl)=O)c2ccccc2c1 N1(C(Cc2ccc(C)cc2)=O)CCC(NC(c2cc([N+](=O)[O-])c[nH]2)=O)C(C)C1 C1(C(N2CCC(C(C)C)(C(=O)NCCc3cnn[nH]3)C2)=O)CC(=O)CC(=O)N1 c1(OCCC)cccnc1CC(=O)NCCC1(O)CN(C(=O)CCC=C(C)C)C1 N1(C(C(CC)CC)=O)CC(NC(=O)NC2CCc3ccnn3C2)CC12CCC2 c1(C(N2C(C(C)C)CCC2C(=O)N(C)CCO)=O)ccc2[nH]ccc2c1 c1(C(N2CCOCC(NC(C3C(=C)CC3)=O)C2)=O)cc(C)nc(Cl)c1N c1(CCCC(=O)NC2C(NC(c3c(OC)cccc3)=O)CC2)ccc(Cl)c(Cl)c1 CC(C)(C)S(=O)(=O)CC(=O)N1CC2CCC1CN2C(=O)CC1CCOC1=O N1(C(c2scc(C(N)=O)c2)=O)C2CCC1CC(CNC(=O)C(O)C(F)(F)F)C2 C1(O)(C(=O)NCCCNC(=O)Cc2cncs2)CCC(C(F)(F)F)CC1 c1(C(N2CC(NC(CCC(C)C)=O)C(F)(F)C2)=O)ccc2ccccc2n1 C1(NC(C2CC(C)(CC)C2)=O)CCN(C(c2ccc(C(N)=O)cc2)=O)CC1 C(CC(=O)N=c1ccn(CC(N)=O)[nH]1)N(C(CCCOCC)=O)CC CCC(C)(C(=O)N1CC2(CNC(=O)C(C)(C)C)CC1CO2)C(N)=O C12(NC(C(CC)=CCCC)=O)CCCC(CN(C(c3cnc(C4CC4)s3)=O)C1)C2 N1(C(C(C(C)C)NC(C)C)=O)CC2CCC1C(NC(C1(O)CC1)=O)C2 C=CC(C)CC(=O)NC(Cc1ccccc1Br)C(=O)NCC(=O)N(C)O c1(OC(C)C(=O)NCC(F)CNC(=O)CC2CC(=O)C2)ccc(Cl)cc1Cl C1(NC(=O)N(CCOC2(CNC(CC)=O)CCOCC2)C)CNC(=O)CC1C C1(NC(c2c(CCC)nco2)=O)CCN(C(=O)Cc2ccoc2)CC1CO N1(C(c2c(OC)scc2)=O)CCN(C(=O)CSC2CC2)C(c2cn[nH]c2)C1 C1(NC(C(c2ccnn2C)C)=O)CCC(NC(c2cn(C(C)(C)C)nn2)=O)CC1 n1(CCOC)cc(C(=O)NC2CC(CCNC(C3CCC(C)C3)=O)C2)c(C)n1 CCC(CNC(=O)C(C(C)O)NC(=O)C=CC1CC1)C(C)(F)F c1(C(N2CCC(O)(CN(C(c3c(OC)noc3C)=O)C)C2)=O)cc(C)cc(C)c1 C(=O)(CS(=O)(=O)c1ccccc1C)N1CC(NC(CC2CC(OC)C2)=O)C(F)C1 c1(CNC(=O)NCC2CCN(CCC)C2)ccnc2[nH]ccc12 C1(C(N2CC(CC=C)(NC(=O)C(CCC)=CCC)C2)=O)CCc2nnnn2CC1 Cc1nc2[nH][nH]cc-2c(=NC2CCC3CN(C(=O)C(F)(F)C(C)(C)O)CC23)n1 CC(C)(O)C#CC(=O)NCC1CCN1C(=O)CSc1ccc(F)cc1 C1(NC(C(Cc2ccc(C)cc2)C)=O)CCN(C(=O)CCc2ccco2)C(C)C1 C1(O)(C(N(CCNC(=O)Cc2cccnc2)C2CC2)=O)CC2(CCOCC2)C1 c1(N2CCC(=C)C2)ncnc2n[nH]cc12 c1(OC)cc(C(=O)NCC2(O)CN(C(=O)C(O)CN3CCCC3)C2)ccc1C N1(C(C(=O)NCCOC)=O)CCC(NC(c2sccc2C)=O)C1 c1(-c2cccc(CC(=O)N(c3cccc(F)c3Br)CCO)n2)c(O)cccc1O N1(C(CCc2nc(C)c(C)o2)=O)CCC(F)C(NC(C2(CO)COC2)=O)C1 N1(C(c2ccc(CSCC)cc2)=O)CCC(O)(CO)CC1.C1(=O)C(C)(CC)N1 C1(CNC(C(C)N(C)C)=O)CCN(C(=O)C(CO)N(C)C)C(C)C1 N1(C(c2ncc(OC)nc2)=O)CCCCC(C(=O)NC(C)C(C)(C)CN(C)C)C1 c1(C(=O)NCC2(F)CCC(NC(Cc3cnc(C)s3)=O)C2)cnn2c1NCCC2 C1(NC(C(C(C)C)CO)=O)CN(C(c2ccc(=O)n(C3CC3)c2)=O)CC2(CCC2)C1 NC(=O)CCCCC(=O)N1CCC2(CC1)CC2NC(c1ccc(=O)oc1)=O C(=O)(C(O)CCC(C)C)NCC1C(CC(=O)NCc2ncc(C)[nH]2)C1 c1(C(N2CCN(C(CCC=C)=O)C(C)CC2)=O)ccc(C#N)c(F)c1Br Cn1cc(S(=O)(=O)NC(C2(C)C=CCC2)=O)ccc1=O N1(C(c2cc(CC)c(CC)o2)=O)Cc2nccn2CC(NC(C2CC2(Cl)Cl)=O)C1 CC(C)CCCCC(=O)NC1CN(C(=O)C(c2ccc(Cl)cc2)(C)C)C1 N1(CCNC(C#CCNC(C=CCOC)=O)=O)C(=O)CNC1=O c1(C(N2CC(N(C(C(C(C)C)n3cnnc3)=O)C)C2)=O)cc(F)cc2nn[nH]c12 C(=O)(C(C)(C)C(C)C)N1CCC(CC=C)(NC(=O)C=Cc2ccc(C)s2)C1 S(=O)(=O)(c1ccccc1F)N1CCC(NS(c2c(C(=O)O)ncs2)(=O)=O)CC1 N1(CCCCOc2ccccc2)CCC2(CC1)CNCCO2 Nc1ccc(F)c(F)c1C(N1CC(NC(=O)Cc2cnns2)CCC(O)C1)=O Cc1sc(Br)cc1C(=O)NCC#CCNC(C1CCS(=O)CC1)=O C1(CNC(C(COC)NC(=O)C(c2ccnn2C)C)=O)(CO)CCN(C)C1 c1(C(=O)OCCC(CCC(=O)OC)(F)F)ccc2nnc(C(C)(C)C)n2c1 Cc1c(NC(C2C3CN(S(=O)(=O)c4cccs4)CC23)=O)cc(Cl)cc1[N+](=O)[O-] CC(CC(C)(C)O)C(=O)N1CCC(C(=O)N=c2ccn(CC(N)=O)[nH]2)(C)C1 C#CCC(C)(C(=O)Nc1cccc(C(C)C)c1)NC(C1CC(=O)CCO1)=O N1(C(C2C(C(=O)OC)C2)=O)CC(F)(CNC(=O)C(F)(F)Sc2cnn(C)c2)C1 N1(C(CSCCCC)=O)CC2CC2(CNC(C2CC2F)=O)C1 CC(C)(CN1CCCCC1)C(=O)Nc1cccc(NC(c2csc(C#N)c2)=O)c1 Cc1cccc(C(=O)NC2CC2CNC(c2cncc(N(C)C)c2)=O)c1C S(=O)(=O)(c1cccc(=NCC(C)c2ccncc2)[nH]1)NCC(CCC)C C1(C(=O)NCC2(CCC)CC2)CC(NC(C2CCC(F)CC2)=O)CCO1 N1(C(Cc2c(OC)cccc2OC)=O)CC2CCC1CN2Cc1ncsc1Br CCC(CC)C(C(=O)NCC1COCCN1C(C1OCCCO1)=O)OC c1(C(=O)NC23CN(C(CCSC)=O)C(C2)C3)ccc(N(c2ccccc2)C)cc1 C1(O)(C(=O)NC2CC3CC2N(C(=O)CC2CCCC2)C3)CC2(CCOCC2)C1 c1(NC2CC(F)(CNC(C3CCCC(C)C3)=O)C2)ncc2c(n1)CCOC2 C(C(C)(O)CC(=O)OC(=O)NCCC(C(C)C)N(C)C)OC CC1CC(NC(c2cc(OCC(F)F)ccn2)=O)CN1C(C1CC(F)(F)C1)=O C1(CC)CCC(C(N2CCOC(CNC(=O)C(O)CSC)C2)=O)CC1 C1(NC(=O)CC2C=CCCC2)COC2(C1)CN(C(C13CCCC(C1)OC3)=O)C2 N1(C(c2c(C)ccc(F)c2)=O)CC(C2CN(C(c3cc(C(C)(C)C)c[nH]3)=O)C2)C1 C=C=C(C)CC(=O)N1CCC(C2CCCCN2C(c2ccccc2Cl)=O)C1 C(=O)(CC1=NNC(=O)C1)NC1(CNC(CCC(=O)N(C(C)C)C)=O)CCCC1 CC1CN(C(=O)C(C2(C)CC2)NC(C2CCC2C)=O)C(C)C(C)(C)O1 C(=O)(C(F)(F)C(F)F)NC1CN(C(C2C(C(=O)OCC)C2)=O)CC1C(F)F C(=O)(NNc1cc(C(F)(F)F)ccc1F)NC1CC(OC)CN(C(C)=O)C1 c1(OC(C)C(=O)NC2CC2CNC(C2CC(C)(C)C2)=O)cccc(Cl)c1Cl c1(CNC2CC3CC(C(=O)OC)C2O3)c(C)cc(CO)cc1C C1(CC)(CNC(C2CC(O)CN2C(=O)CNc2cccnc2)=O)CCOCC1 C1(CC)CN(C(=O)CC(F)(F)F)CCN1C(=O)C(F)CC1CCCCC1 C=CC(C)(C)NC(=O)CCOC1CN(C(=O)C2CC2)C1 c1(C(=O)NCCCCNC(C2C(C)(C(C)C)C2)=O)cnnc(C2CC2)c1 CCC(CC(=O)NCCCc1cccs1)N(C(=O)C(CSC)OC)C c1(-c2cncc(C)c2)ccc(C(=O)Nc2ccccc2C(=O)NC2CC2)c(C)n1 c1(C(N2C(CNC(=O)CCC3CCOC3)C3CCC2C3)=O)cccc2c1OCO2 C(=O)(C1=CCS(=O)(=O)C1)N1CC2(CC(NC(=O)C(F)CC3CCCCC3)C2)C1 c1(C(=O)NCC(CC)N(C)C(c2nc(Cl)oc2C)=O)ccncc1OC CCC(CC)C(C)C(=O)N1CC(NC(=O)C=Cc2ccccc2)C(C2CC2)C1 c1(N2CCCCC(NC(c3ccc4cncn4c3)=O)C2)ncc2cccnc2n1 Cc1cc(C)c(C(=O)NCC2COCCN2C(c2cnc(O)n2C)=O)s1 CC(C)(CCCNC(C1CCCO1)=O)C(=O)NC1C2CCCCC12 Cn1c([N+](=O)[O-])cnc1NC(=O)CSc1ccc(F)cc1 Cc1ccncc1C=CC(=O)NC(C1(O)CN(C(C2CC3CC3CC2C)=O)C1)C N1(C(C(COC)C)=O)CCN(C(c2ccccc2-n2ccnn2)=O)CC(O)C1 c1(SCC(=O)NCCC(O)CNC(C2CCCCO2)=O)ccc(F)cc1 C#Cc1ccc(C(=O)NCc2ccc(C(=O)NCC3(C4(O)CCC4)CC3)o2)cc1 C(C)(N=c1nc2sccc2c(NCC2CSCCS2)[nH]1)c1c(SCC)cccc1 c1(C(N(CC(CN(C(CC(C(=O)OC)C)=O)C)O)C)=O)cnc2cc[nH]c2c1 c1(C(N2C(CNC(CC(CC)C)=O)CCC2)=O)ccc(F)cc1C#N c1(C(N2C(C)CCC(NC(c3cc(OC)ns3)=O)C2)=O)cccn2nccc12 c1(C(=O)NC2CN(C(C3CNC(=O)O3)=O)C(CO)C2)cc2ncsc2[nH]1 c1(C(C)C)cccc(F)c1C(=O)NCCNC(=O)Cc1ccco1 C1(C(NOCCC=C)=O)(CNC(c2cc(Cl)ns2)=O)CCCO1 C1(CNC(c2nnc(CC)s2)=O)CCN(C(=O)CSC(F)(F)F)CC1C C12CN(C(=O)OC(C)(C)C)C(C)(C1)N2.C(C)(C)(CCC=C)N(C(C#C)=O)C C(C)(CC(=O)NC1CC(=CC(=O)NOCC)C1)OCC CCCCC(O)CC(=O)N1CCC(F)(CNC(=O)CCc2cc[nH]n2)C1 c1(CC(C(=O)NC(C(CO)NC(C2(C(CC)=O)CC2)=O)C)C)ccccc1C c1(C(=O)NCC(CNC(c2cc(Cl)cc(C)c2N)=O)O)ccc2c(c1)CCC=C2 CCC(C)CC(C)C(=O)N1CCC(CCNC(C2CC(C)(C)C2)=O)CC1 c1(C(N2C(C(=O)Nc3cc(OC)ncc3)CCCC2)=O)ccn2cncc2c1 Cc1cc(N)c(C(N2CCC(OC3CN(C(C4CC(F)C4)=O)C3)CC2)=O)cc1C CCCC(C(F)(F)F)NC(C1CCCN(C(c2cc(C)nn2CCC)=O)CC1)=O C1(C#N)(C(=O)NC(C2CN(C(c3cnn(CCN(C)C)c3)=O)C2)C)CCC1 C1(CNC(C2C(OCC)C2)=O)CC2(CC2)CN1C(C1CC12CCSCC2)=O N1(C(C(CC)OCC)=O)CCC(C(C)C(=O)N(C2CCCC2O)C)CC1 c1(C(N2CC(CNC(C(=C(C)C3CC3)F)=O)C2)=O)c(N)sc2c1CCSC2 Cc1cc(CC(=O)NC(C)CCCNC(=O)C(C)Cc2cnc[nH]2)c(C)s1 S(=O)(=O)(c1ccc(Cl)cc1F)N1CC(C(=O)NCc2nc[nH]n2)NCC1 CC1CCc2[nH]nc(C(N3CC4CC(NC(=O)CCCC(N)=O)C3C4)=O)c2C1 C1(Cc2ccccc2)CCCN1C(c1nc(CN(C(C)C(=O)N(C)C)C)no1)C C(=O)(C1=Cc2cc(Cl)ccc2OC1)NC1C(NC(COCCCCCC)=O)COC1 C1(C(=O)NC(C)CCNC(=O)C(C)CCO)CC(=O)CC1(C)C c1(CN(C)Cc2cn(-c3cc(C)c(Cl)c(N)c3)nn2)cccc2cccnc12 S(=O)(=O)(c1nccs1)N1CCC(NC(c2cccc(Br)c2F)=O)C1 N1(C(CC(C)n2ccnc2)=O)C2CCCC1CN(C(=O)C(F)(F)CO)C2 C(=O)(CCS(=O)(=O)CC(C)C)N1CCC(CNC(CCC(CC)C)=O)C12CCC2 N1(C(C2(C(N(C(C)C)C)=O)CC2)=O)CC(NC(c2cnn[nH]2)=O)CC2(CC2)C1 C12(CNC(c3ccc(C)s3)=O)CCC(NC(c3cc(=O)cc(Cl)[nH]3)=O)(CO1)C2 c1(C(c2nnnn2Cc2ccccc2)NCCSCC)ccc(F)c(Br)c1 N1(CCN(C(CC2(NC(C(C)C3CC3)=O)CCC2)=O)C)CCCCC1 c1(C(N2CC(NC(C(C)C3CCCO3)=O)(CO)C2)=O)cc2c(Cl)cc(F)cc2[nH]1 C(=O)(C(CCC(N)=O)N(C)C)NC1(CNC(CCC(=O)NCCC)=O)CCOC1 C=C(C)CN=C(NCC1(OC)CC1)N(C)CC1CCOC1 C1(CC)CN(C(c2nn(CC)cc2Cl)=O)CCC1NC(C1(O)CCSCC1)=O N1(CC)CC(C(=O)NC2CN(C(=O)CCc3nc(C)no3)C2)CCC1=O c1(C(=O)NCCC(C(C)C)NC(c2cscn2)=O)c(F)cccc1[N+](=O)[O-] N1(C(c2cc(C)nnc2)=O)CCN(C(=O)CCCCCF)CC1C(C)C C(=O)(CC1=CSC2=NCCN12)NC(CC(C)NC(=O)CCCc1cccs1)C CC(=O)CC(C)(C)C(=O)N1CCC(OCCNC(=O)CCCC(F)(F)F)C1 C12(CC(N3C(C(=O)OC)CC3)=O)CCC1CN(C(=O)CCC1CCCCC1)C2 c1(NC(CCSC)C)ccc(S(=O)(=O)N(C)CCc2c(F)cccc2Cl)c(Cl)c1 C(C(C)C)(C(O)C(=O)N(C(CNC(c1cccc2cncn12)=O)C1CC1)C)OC CCC(C(=O)N(C1CCCCN(C(=O)C(=O)NC(C)C)C1)C)C(C)(F)F c1(CC(=O)NCCC(C)NC(C(C(CC)C)NC(C)=O)=O)ccc([N+](=O)[O-])c(N)c1 N#CCCCCC(=O)N1CCC(NC(C2CC3CCC2O3)=O)CC1 c1(CC)nc(C)sc1C(N1CCSC(C(N2CC(O)C(O)C2)=O)C1)=O CCCCCCCC(=O)NC1CCN(C(=O)C(c2c(C)noc2C)C)C12CCC2 Cc1cc(NC(=O)C(CO)(CO)NC(=O)C#CC2CCC2)cnc1Cl c1(C(=O)NCC2C(C(N(CC(COC)(F)F)C)=O)C2)cccc(C)c1N N1(C(C2CCN(CC(C)C)CC2)=O)CCN(C(=O)CC2CC2(C)C)CC(CO)C1 CCCCC(C(=O)NC1CCC(NC(=O)C(C(C)(C)C)OC)C1)N(C)C c1(C(=O)NC(CN(C(=O)CCn2cccn2)CC)C)cnn(C(C)C)c1Br C(CC(C)C)(C(=O)NCC(O)C(=O)NC)N(C(C1C(=C)C1)=O)C N1(C(CN2CCN(CC)CC2)=O)CC2(NC(=O)CC(C)(C)CC)CC2(C(=O)O)C1 O=C1C2CC3C1C3C2NC(Cc1cc[nH]n1)C(=O)N1CC(n2cc(CO)nn2)C1 c1(C(N(CCC(C)NC(c2cc(N3CCCC3)ccn2)=O)C)=O)ccncc1O C1(NC(=O)C(F)C2CCC2)CC2(C1)CN(C(C1(n3cccn3)CC1)=O)C2 C1(OC)CN(C(=O)C(CNC(=O)CSC(C)C)CC2CCCC2)C2(CCC2)C1 CN1CCC(C(=O)NCC2CCC(NC(c3cc(C(F)(F)F)cs3)=O)C2)CC1=O C(N=c1ncc2cc(F)ccc2[nH]1)C1C(N)C1 c1(N2CCC(CNC(C#CC(C)(C)C)=O)C2)ccc([N+](=O)[O-])cc1F C(CNC(C1CCC(c2ccccc2)C1)=O)(C(C)(C)C)NC(c1cc(C)sc1)=O N1(C(C2(C#N)CC2)=O)CCC(NC(=O)Cc2ccc(F)cn2)C2(CCC2)C1 CC(C)CCCC(C)CNC(=O)C(c1ccccc1)NC(C1(O)CCSC1)=O c1(N2C(C(=O)Nc3cccc(O)c3Cl)CC2)ncc2cc(Br)ccc2n1 N1(C(c2cccc(C)c2)=O)CC2CC(CNC(=O)CN3CCOCC3)CC1C2 c1(C(C(=O)N(C(=O)C=Cc2ccc(Br)s2)CC)(C)O)ccc(F)cc1 C(CC1=CCCCCC1)NC(CC1CC(NC(C2(CC(C)C)CC2)=O)C1)=O c1(CC(=O)N(C2CCCN(C(c3c(CC)nns3)=O)C2)C)ccc(C#N)cc1 C=C=CCC(=O)NC1COCC1NC(=O)C(F)F c1(C(=O)NCC(CO)NC(C(C=C)(C)C)=O)c(F)ccc(C)c1Cl C1(C(N(C2CCN(Cc3sncc3Br)CC2)CCC)=O)CCCC(F)C1 CC1(C(=O)NCC2(NC(c3cccc(CC(F)(F)F)c3)=O)CCC2)COCCO1 Cn1nc(C(=O)NCCNC(C2(NC(=O)OC(C)(C)C)CCC2)=O)cc1Br c1(C(=O)NCCOC2CN(C(C3(C(=O)NC)CCC3)=O)C2)c(C)ccc(C)c1O N1(C(C(CCC)(C)C)=O)CCC2(CCCC2NC(c2nnc3ccccn23)=O)C1 Cc1cc(NC(c2ccc(NC(C3(n4ccnc4)CC3)=O)cn2)=O)ccc1Br c1(C(N(CCNC(=O)COc2ccsn2)C2CC2)=O)ccn2ccnc2c1 N1(C(CCNS(CC)(=O)=O)=O)CC(C)CN(C(c2ccc(Cl)c(O)c2)=O)CC1C c1(NC(C(=O)N(CCCNC(C=CC)=O)C2CC2)C)ccc(F)cc1.C(C)=O C1(NC(=O)OC(C)(C)C)CC2CC(NC3CCN(C4CC4)C3=O)CC12 c1(SC)ccc(C(N2CC3C(NC(c4cn5c(n4)SCC5)=O)C3C2)=O)c(Cl)c1 CC1(NC(c2ccncn2)=O)CN(C(=O)C(F)=C2CCC2)C1 C(C(O)CC(F)(F)F)NC(C(C(C)NC(c1cccc(CO)n1)=O)C)=O Cc1nc(CNC(C2CC(NC(C3CC(CF)C3)=O)CCO2)=O)sc1C CCCCC(CNC(c1ccc(C(F)(F)F)nn1)=O)NC(C1CC1F)=O c1(C(=O)NCC2(COC)N(C(C(CCCC)O)=O)CC2)ccc2c(C)noc2c1 CCCC(CNC(c1cnc(OC)s1)=O)C(=O)Nc1ccc(CC)c(O)c1 c1(COCC(=O)NCCC2(NC(=O)C(=Cc3c[nH]cn3)F)CCC2)ccccn1 C1(NC(c2ccc(OC)s2)=O)CCCCC1CNC(c1c(C)[nH][nH]c1=N)=O c1(CNc2cccc(C(=O)Nc3ccc(O)cn3)c2)ccnc(Cl)c1Br c1(C(CN(CC(C)=O)CCC)=O)cc2c(Br)coc2cn1 c1(C(=O)NCC2CC(CC(=O)OC)C2)c(Br)ccc(F)c1I C12(NC(N3CCC(Oc4ccccn4)C3)=O)CCCC1C2(F)F C1(C(N2CC3(CCNC3=O)C2)=O)N(C(C2CC23CC3)=O)CC12CCCC2 C(C)(CNC(c1ccsc1)=O)(CC(C)C)NC(c1cccc(SCCC)c1)=O N1(C(c2nc(C(C)NC(=O)C=CC(F)F)oc2)=O)CCC2(CC1)N=N2 c1(C(C)=O)cc(C(N2CC(Cn3cc(C(C)(C)F)nn3)C2)=O)c[nH]1 C1(NC(CSCCC(C)C)=O)C=CC(C(=O)NC(C)CC(C)O)C1 CCC(C)CC(=O)N(CCNC(=O)C(N1CCC(O)CC1)C)C(C)C c1(C(N2CCC(CO)C2)=O)c(-c2cnc(NC(=O)C(F)(F)F)nc2)cncc1F N1(C(C2(CC)CCOCC2)=O)CCC(C)C(NC(c2ccncc2)=O)C1 CCC(CC(=O)N(CC(O)CN(C(=O)C(F)n1ccnc1)C)C)OC C1(NC(C2(CNC(C(CC=C)NC(C)=O)=O)CC3(CC3)C2)=O)CCOC(C)(C)C1 C1(NC(CCCC2CCC2)=O)CN(C2CCCC2)CCC1c1ccc(F)cc1 c1(C(=O)NC(C(C)C)CNC(=O)CC2CC=CCC2)ccc2c(=O)cc[nH]c2c1 c1(C(=O)NC(C2CCCN(C(CN(C)CC)=O)C2)C)ccc(C(C)(F)F)nc1O C1(=CC(N2CC3C(NC(=O)C=CCn4cncn4)C3C2)=O)CN2CCC1CC2 c1(C(N2CCCC(NC(C3C(C)C3)=O)(CO)C2)=O)cccc(Cl)c1[N+](=O)[O-] C1(NC(CC2N(C)CCC2)=O)CCCCN(C(c2cncnc2)=O)CC1 CC(CN(C(=O)C(F)C(C)(C)O)C)N=c1ccn2c(Br)cnc2[nH]1 c1(OC)cc(Cn2nc(C(C)O)nc2-c2ccc(OC)cn2)cc(OC)c1OC c1(-n2cc(C(CCC)NC(c3ccc(C(C)=O)nn3)=O)nn2)ccc(F)cc1C N1(C(c2[nH]cc(CN(C)C)c2)=O)Cc2ccccc2C(NC(=O)C=CCF)C1 c1(N(CCN(C(c2n(CC)nnc2)=O)C)C)ccccc1OC C#CC1(C(=O)NC2CN(C(c3ccncc3Br)=O)CC2C)CCCC1 Cc1noc(Cl)c1CC(=O)N(CC(C)O)CCNC(c1conc1CC1CC1)=O c1(C(=O)NC(CN(C(c2cc(CCC)ncc2)=O)CC)C)cc(C)cc(C)n1 C1(N(C(C(=O)NC2COC2)c2cscn2)C)CCC(C)(C)C1 CN1CCC(C(=O)NCCCCNC(C2NC(=O)C3CCC23)=O)c2ccccc21 c1(CNCC)ccc2ccc(Cl)cc2n1.C12(CCCCC1)C(=O)N2 C=CC1CCCCN1C(=O)C(C(C)(C)C)NC(C1CC(C)N(C)C1)=O c1(OCC(c2n(CC)nnn2)(C)NCCOC)ccc(CCSC)cc1OC Cc1oc(CNC(=O)CCCC#N)nc1C(N1CCC(C(C)C#N)CC1)=O Cc1cn(C(C)(C)C(=O)N2CCC2CC2CCC(CNC(=O)C(F)(F)F)C2)cn1 C(CC(O)CCO)NC(C(C1CCCC1)NC(=O)CCc1ccccc1)=O c1(C(=O)NCC2CCN2C(=O)C=C(Cl)Cl)ccc(=O)n(CCO)c1 CC(C)(CCCF)C(=O)NC1C2CC3C1C3C2C(N1CC(O)C(O)C1)=O [N-]=[N+]=Nc1cc(F)ccc1C(=O)OCCC1=CCC2CC1C2(C)C CC(O)(CC(=O)N1CC(NC(=O)CC(c2cccs2)n2cccc2)C1)C(F)(F)F C(CC(C)C(=O)N1CSCC1C(N1CCCC1C1(C)CC1)=O)=CCC c1(CCC(=O)NC(C2CC(CNCC)(Cc3ncon3)C2)=O)cccc(F)c1Br c1(C(=O)NC(CCCC)CNC(c2ccn(C3CC3)n2)=O)ccc(O)nc1Cl N1(C(CC#N)=O)CCC2(C1)CN(C(=O)Cc1csc3cccc(F)c13)CCO2 C1(NC(C2CN(C)C(=O)CC2)=O)CCC2CN(C(=O)CN3CCOCC3=O)CC12 c1(COC)ncc(C(N2CCCC(NC(c3n[nH]c(SC)c3Cl)=O)C2)=O)c(O)n1 Cc1cc(C(=O)NCC23CCC2CN(C(C2C=CCCC2)=O)C3)cc(F)c1 CC(F)(F)C(=O)NCCCCC1(NC(C2CC2[N+](=O)[O-])=O)CC1 CC(C)C1=CCC(C(=O)NCC2CC(CNC(c3ccc([N+](=O)[O-])s3)=O)C2)CC1 C1(NC(c2ncn(C)c(=O)c2)=O)(CNC(=O)C(=O)NC(C)C)CCC(F)(F)CC1 CCCCCC(c1nnnn1C1CCOC1)Nc1cccc(N2CCOC2=O)c1 n1(CC(=O)NC2(CNC(C3(C(F)F)CC3)=O)CCCC2)ncn(O)c1=O N1(C(c2cc(C)no2)=O)CCC(C)(CNC(=O)C(C)(C)C2CCOCC2)C1 CC1CN(C(c2cn(C3CCOC3)cn2)=O)CC1CNC(C1(CF)COC1)=O C(C(=O)O)(C(O)c1cccnc1)NC(=O)Cn1cc(Cl)cn1 c1(C(=O)NC(C2(O)CN(C(C=CCC)=O)C2)C)cc(C)c(Cl)cc1C N1(Cc2cccc(OCC)n2)CC2(CCC(NCc3cc(C)cc(Cl)c3)C2)C1 c1(C(c2n(CCCCCC)nnn2)NCC(=O)NCCC)ccc(Cl)cn1 C=CCCCC(C)(C)C(=O)N1CCN(C(C2OCC3COCCC23)=O)C(CC)C1 C1(NC(c2cn(CCOC)nn2)=O)C=CCN(C(=O)C(F)C2CCC2)C1 Cc1c(C(N2CC(NC(=O)CCN3CCC(O)CC3)C(C)(C)C2)=O)nn(C)c1N C1(c2ccc(CC)cc2)CN(C(C2(CCO)CC2)=O)CCN1C(C1SCCS1)=O C(C)(C)(CC(F)C(=O)NC(C)C(=O)N(C)CC)NC(c1c(CC)cco1)=O C(=O)(CCC(C)(C)C#N)N1C(C(C(=O)N(CC(C)C#N)C)(C)C)CCC1 Cc1ccc(CO)cc1C(N1CC(CCCCNC(=O)CN2CCCC2C)C1)=O C1(C(=O)NC(C)C(C)(C)NC(=O)CS(=O)(=O)C2CC2)Cc2cc(Cl)ccc2O1 c1(CC)noc(C(N2CCC(N(C(=O)Cc3ccoc3C)C)CC2)=O)c1C Cc1cccc(C(=O)N(CC(C)C(=O)NCCC2CCCN2C)C)c1F N1(C(c2c(C)cccc2N)=O)CC(C2CCCN(C(=O)Cc3cnccn3)C2)C1 C1(CCNC(c2cc(C)on2)=O)CSCCN1C(=O)COc1ccsn1 c1(C(=O)NC2CN(C(c3cncc(OC)n3)=O)C3C2C3)cc2n(c1)CCSC2 n1(CC)nc(C(N2CCCC2CNC(=O)C(F)OC(F)(F)F)=O)c(Br)n1 c1(C(=O)NCC2OCCN(C(C=CCCC)=O)C2)cc2nc[nH]c2cc1F c1(C(=O)NCC(CC(=O)N(CC(CC)CC)C2CC2)C2CCC2)ccc([N+](=O)[O-])o1 c1(CC(N2CC3CN(C(c4c(C)c[nH]n4)=O)CC3C2)=O)ccc([N+](=O)[O-])cc1F N1(c2[nH]c(=NCc3c(C)nccn3)[nH]c(=N)n2)CCCC1C1OCCO1 c1(C(N(C(CNC(C=CC(=O)OCC)=O)C)C)=O)c(C(F)(F)F)cccc1CC c1(C(N2CC(CNC(CCC=C)=O)N3CCC2C3)=O)ccc(=O)n2c1CCC2 c1(NC(c2ccc(OC)cc2)=O)scc(O)c1C#N.c12ccc(cc1)C(=O)NC2 C#CCCCC(C)C(=O)NC1C2CC1N(C(c1cnc(C3CC3)nc1)=O)C2 c1(C(C(=O)NCC(CNC(Cc2nc(C)[nH]n2)=O)C)(C)O)ccc(F)cc1 CCC(Cc1cccc(F)c1)C(=O)NCC(c1cn(C2CC(O)C2)nn1)(C)O c1(CC(=O)NC2CCCC2NC(C2COCCO2)=O)ccc2nc[nH]c2c1 C#CC1(C(=O)NCc2nonc2C)CCN(C(=O)C(O)C2CC2)CC1 N1(C(N(CC)Cc2cc(O)n(C)n2)=O)CC2(C(=O)OC)CC(c3ccccc3)(C1)C2 CC(C)(CNC(=O)C(C1CCOCC1)N1CCCC1)Cn1cc(C2CC2)nn1 CC1(C)CC(NC(=O)C=CCO)CCN(C(C2CC3(CCCC3)CO2)=O)C1 C(=O)(C(C)C(F)(F)C(F)F)NCC(CC)(CC)NC(C1CC1(C)C(F)F)=O c1(C(N2CCN(C(CSCCCC)=O)C(C)CC2)=O)c[nH]c2c(CC)cccc12 N1(C(C(CCCC)C)=O)CC2(C1)CN(C(=O)CCCOCCOC)CCO2 C1(NC(=O)Cn2ccnn2)CN(C(C2CC2c2ccncc2)=O)CCC12CCC2 Cc1ccc(O)cc1CN1CC2(CC2)CC1C(=O)OC(C)(C)C Nc1c(C(=O)NC(c2ccccc2Cl)CCO)cc(F)cc1Br C#CCCCC(C)C(=O)N1CC(NC(=O)C(C)CN2CCOCC2)C(CO)C1 O=C(C#CC1CCCCO1)N1CCN(c2ncnc(O)c2Br)CC1 C(=O)(C1=COCCO1)NCC1(CNC(=O)CCc2cnc[nH]2)CC12CCC2 c1(N2CCC(O)(C(C)NC(c3cnc(Cl)cn3)=O)C2)nc(C(F)F)nc(=N)[nH]1 N1(C(COc2ccc(C)cc2C)=O)C2CCC1C(F)C(NC(=O)CC1CCC1)C2 C=CC1(C(N2CCC(C(C)C(=O)NCC(C)(C)C3CC3)C2)=O)CCOCC1 c1(C(=O)NC2C(NC(CN3CC(C)C3)=O)C2)ccc(-c2cn[nH]c2)cc1 N1(C(C2C(OC)(OC)CC2)=O)CC(CNC(c2ncoc2C)=O)CC1(C)C CC1CCN(C(=O)CCCc2ccsc2)C(CNC(=O)CCC2CCCCO2)C1 C1(C(=O)NCC(CNC(=O)CC(C2CC2)C2CC2)CO)CCCC2(CCC2)O1 c1(C(N2CC(C(N(C)CC3C(C)C3)=O)OCC2)=O)cc(F)ccc1F c1(C(N)=O)ccc(C(=O)NCC(O)CNC(c2ccc(C3CCOC3)s2)=O)[nH]1 c1(CN(C)CC2(C)CC2(F)F)cc2cc(Cl)ccc2s1 CC(C)(O)CC(=O)NC1(CCC(=O)NCCC(N)=O)CCCC1 c1(OC)cc(C(F)(F)F)ncc1C(=O)NC1CC1C(=O)N(C)C C1(C)(CC)C=C(C(=O)NCC2CN(C)CCN2C(c2csc(C(C)=O)n2)=O)C1 C(C(=O)N(C1CCCN(C(c2c[nH]c(Br)c2)=O)C1)CCO)(C(C)C)OC C=C(C)CC(C(=O)NCCCNC(c1ccc(CC2CC2)s1)=O)NC(C)=O c1(C(=O)NC2CCC(NC(c3c(N)cccn3)=O)CC2)ccnc2c1CCC2 N1(C(C(n2c(C)cc(C)n2)C)=O)CCCC(C)(NC(=O)CSCc2cccs2)C1 N1(CC(=O)N(CCC)CCC)CCCCC(CCCc2ccc(F)c(Cl)c2)C1 C1(CCNC(CNC(=O)OCC)=O)CC(OC)CN1C(=O)C(C)(C)SC C1(OC)CC(C)CN(C(c2ccnc(CNC(C3CCCC(OC)C3)=O)c2)=O)C1 N1(C(=O)CN2CCOC2=O)CC2(C(N3CCCC(CO)CC3)=O)CCC1CC2 C1(NC(CNC(c2ccc(C)s2)=O)=O)CC2CN(C(C34CCC(C3)C4)=O)CC12 C1(NC(c2n(C)cnn2)=O)CN(C(c2cc(O)ccc2F)=O)C2(CCOCC2)C1 N1(c2snc(SC)n2)CCCC(C)(C)C1CNC(=O)CN1CC2CC2C1 C1(NC(CSCC)=O)CN(C(=O)C=Cc2cncc(O)c2)C(C)(C)C1 N1(C(C(C)OCCC=C)=O)CCC2(CCOCC2)C(NC(=O)CC(C)CCC)C1 C(=O)(C(C#N)CC)NC(CCC)CNC(c1ccncc1OCC)=O CCC(C(=O)OC)C(=O)NCC1(CO)CCN(C(=O)C(=O)NCCC(N)=O)C1 c1(C(=O)NCC(C)O)cccnc1CNC(=O)CCOCCSC1CCC1 N1(C(c2cnc(C)s2)=O)CC2(CCN(C(c3ccc(Cl)cc3)C)CC2)C1 c1(C(=O)NC(C(C(C)C)C)CNC(c2ccc(Cl)cn2)=O)cnc2[nH]ncc2c1 C(C(O)(C(=O)NC1CC(NC(=O)CN2CCCCCC2)C1)C(F)(F)F)N(C)C C1(NC(C(F)=C(C)C)=O)CCN(C(=O)C(C)C2CC2)CC1F c1(C(=O)NCCNC(COCc2cccc(OC)c2)=O)csc2cc(C)sc12 C1(NC(Cc2c(C)cccn2)=O)CC(F)CN(C(C2CCC(=O)N2)=O)C1 CC1C(=O)N(C)CCN1C(C1(C)CN(C(c2ccncc2O)=O)C1)=O C(=O)(C(C)(C)C(=O)NCC(C1CCN(C(c2cnc(O)c(C)c2)=O)CC1)O)NC N1(C(c2c(CC)ncs2)=O)CCCC2CN(C(=O)C(c3ccccc3C)C)CC12 c1(CN2CCCC(N(C(C=CC=CC)=O)C)CC2)cc(=O)c2ccccc2[nH]1 C1(NC(C2CC=CCO2)=O)CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)CC1O c1(C(=O)NC2C(NC(C3(C(F)(F)F)CC(=C)C3)=O)CCC2)cc(F)cnc1OC N1(C(C#CCNC(C2CCCCCC2)=O)=O)CCOC2CCCCC12 c1(C(=O)NCCCOCCN(C(C(C2CCCCC2)C)=O)C)cscc1Cl Cc1ncc([N+](=O)[O-])n1CCNc1cnn(C2CNC2)n1 CC1=C(C)CC(C(=O)NCC(C(=O)N(C2CCC2)CCO)C(C)C)CC1 CC1Cc2cc(C(=O)NC34CCC(C3)N(C(C35CCC(C3)C5)=O)C4)ccc2O1 C1(SCC)CCCC(NC(=O)NC(c2ncccc2F)C)C1 c1(C(=O)NC(C2CCN(C(c3c(C)c[nH]n3)=O)C2)(C)C)nn(C(F)F)cc1Cl C(=O)(C(CCC)C(C)C)N1CCN(C(c2cn(CC=C)nn2)=O)CC1CC(F)F C1(CN(CC)CC)CCCCN1C(=O)CCc1ccc(N(C)C)nc1 N1(C(C(C)(C)OC(C)C)=O)CCN(C(C2(C)CCCS2)=O)CC12CCC2 n1(CC)cc(Cl)c(C(=O)NC(C(C)NC(c2conc2COC)=O)C(C)C)n1 c1(C(=O)NCC(CCOC)NC(c2cc(C(=O)OC)nn2C)=O)cc2occc2[nH]1 c1(C(N2C(C)CC(NC(CC(C=C)(C)C)=O)C2)=O)ccc2oc(N(C)C)nc2c1 c1(-c2c(C(=O)OC)noc2)ccccc1CC1(C(=O)NC(C)(C)C)COC1.C(=O)(N)O C12(NC(CN(C3CC3)CC)=O)CCC(CC1)N(C(C1CCCS1(=O)=O)=O)C2 n1(C(C)C)ncc(C(=O)NCC2CCCC2C(N2CCC2C2CCCC2)=O)n1 c1(CC(N2CC(CC(C)NC(c3c(CC)cno3)=O)C2)=O)ccc(F)cc1 c1(C(=O)NCCC2(O)CN(C(C(CC)C(C)O)=O)C2)ccnc2[nH]ncc12 N1(C(c2cnc3n2CCCC3)=O)CCC2(CCCN2C(=O)C2=CCOCC2)C1 N1(C(C(CCC)=CCC)=O)CCn2c(CNC(C3CC3(C)C(F)F)=O)nnc2C1 C1(NC(c2c(CC)nc(C)o2)=O)CN(C(=O)Cc2ccccc2O)CCC1C C#Cc1ccc(F)cc1C(=O)NCCCC(C)(C)NC(c1oc(SC)cc1C)=O C1(CNC(c2ccc(SCC)nc2)=O)CCC(C)CN1C(=O)CNC(N)=O c1(SC)cc(C(=O)NCCC2(O)CCCNC2)cc(SC)c1 N1(C(CCCNC(C)=O)=O)CCN(C(=O)Cn2nccc2C)C2CCCCC2C1 C1(CCNC(c2cc(OCC)no2)=O)CC(F)(F)CN1C(=O)C(N)=O C1(NC(C2(C(C)C)CC2)=O)CC2CC1CN2C(C1(Cc2ccccc2)CC1)=O C1(C(=O)NCC2CCCN(C(c3ccc[nH]3)=O)C2)CC12CCC(F)(F)CC2 C1(c2nnc(Nc3ccncn3)o2)(NC(c2ccccc2)=O)CCOCC1 C1(CC(=O)NC(CC=C)CNC(c2cnc(CC)nc2)=O)CCCS(=O)(=O)C1 C(=O)(C(C)C(O)C(C)C)NCCN(CC(C)O)C(c1nc(C(C)C)oc1)=O CC1(C)CCC(CC(=O)Nc2cccc(NC(=O)CC3C=CS(=O)(=O)C3)c2)C1 CCC(CC)C(C)C(=O)N1CC2(CCC(CNC(=O)CN(C)CCO)O2)C1 c1(C(N(C2CC(NC(CC3(CC)CCC3)=O)C2)C)=O)nc(C)oc1C N1(C(C(CC(C)C)C)=O)CCCN(C(=O)Cc2csc(C3CC3)n2)CC(CO)C1 c1(C(=O)NCC2(F)CN(C(C3C(CC)CCC3)=O)C2)cccc(C(C)(F)F)n1 N(C1CCCc2sccc21)C(CCCCCO)c1n(CCSC)nnn1 C1(C)(CC)CC1C(=O)NCC1CC(C(=O)NCC(C)(C)n2ccnc2)C1 CCC(CC(=O)N(C)CC1CN(C(C2OCCC2(C)C)=O)CCO1)OC C1(OC)(CNC(C2CC(F)(CO)C2)=O)CCN(C(=O)CC2OCCC2(C)C)C1 C(=O)(C(C#N)C(C)C)NCC(c1ccccc1)N(C(c1[nH]cc(C)c1)=O)C c1(OCC)cnc(C(=O)NC(CNC(=O)CCOC2COC2)CC(C)C)cn1 c1(C(N2CC(C(C)(C)O)(CNC(Cc3c(C)non3)=O)C2)=O)nccnc1N C1(C(=O)NCc2cn(-c3ccccc3C(F)(F)F)nn2)CNC2(CC2)CO1 CC(C)CC(C(=O)NCCCN1CCC(O)C1)NC(c1ccccc1)=O Cc1c(F)cc(C(=O)NC2CCCCN(C(=O)C=Cc3cscn3)C2)c(F)c1N Cc1ncsc1C=CC(=O)Nc1cccc(NC(=O)C(F)(F)c2cncs2)c1 C1(CC)CCC(C(=O)NCC(C(=O)NC(c2nc(=O)o[nH]2)C)N(C)C)O1 N1(C(C(CC)C)=O)CC2(C(=O)NC3CC(c4ncc[nH]4)C3)CCC1CC2 N1(C(C(C)=NOCC#N)=O)CCCC(CCNC(=O)C=Cc2ccc(C)o2)CC1 C(=O)(C(C)(C)CC(=O)N1CC2CCCC2(NC(c2ccoc2C)=O)C1)OCC C#CC(C)(C)C(=O)N1CC2CC2(CNC(C2(COC(C)C)CC2)=O)C1 c1(C2(C(=O)NC3C(NC(C(C)SC(C)C)=O)C3)CC2)cc(F)cc(C#N)c1 c1(-c2ccc(SCCN(C)C(C3CCCNC3)=O)[nH]2)cc2ccccc2o1 c1(C(N2CC(CNC(C(C)(C)OCC)=O)C3C2C3)=O)nc(C)ccc1C C1(C(=O)NCCC(CNC(=O)CNC(=O)C2CC2)O)CCC(OCF)CC1 N1(C(COCCCC#C)=O)C(CNC(=O)C2=C(Cl)CCOC2)CC2CCCC12 N1(c2cc(-c3occc3)nc(N3CCCCC3)n2)CCc2c(O)nc(O)nc2C1 C1(C(=O)NCC(CN(C)C(c2ccoc2C(F)(F)F)=O)(C)C)CCCCS1(=O)=O CCN=c1ccc(C(=O)NCC(C)(C(C)C)NC(=O)CC2CC23CC3)c[nH]1 C1(NC(C2C(CC)OCC2)=O)CC12CCC(NC(=O)C=C1CCN(C)CC1)CC2 Cc1cc(C)c(C(=O)CCCC(=O)OCCc2cc(C)n(C)n2)c(C)c1 O=C1CCOC2(CCN(C(=O)CCOc3cc(F)cc(F)c3)CC2)C1 N1(C(CC(c2ccc(Br)cc2)C)=O)CC2C(N(C(=O)CCF)C)C2C1 c1(C(N2CC(F)CC(NC(CC(C(=C)C)OCC)=O)C2)=O)cc(C)c(C)c(C)c1 Cn1nc(CNCc2cc(Cl)ncc2Br)c2ccccc2c1=O [N-]=[N+]=NCC(C(=O)N1CCSC2(CC2)C1)NC(=O)C(O)C1CCCC1 CC1CC(CCNC(=O)C(C)N(C(=O)COCCF)C2CC2)C1 c1(OC)ccccc1C(CNC(=O)CC1CCC1)NC(c1ncc(F)cn1)=O N1(C(C(=O)NCCC)C(C)C(C)(C)C)CCn2c(nc3ccccc23)C1 CCC(CC(=O)NC1(CCNC(=O)CN(C)CCOC)CCOCC1)SC1CC1 C1(C(N2CC(O)(CCNC(COC3(C)CCC3)=O)C2)=O)CC(C2CCCC2)C1 c1(NCC)cnc(C(=O)NC(C)CCCNC(c2sccc2Br)=O)cn1 C(=O)(CC(C)(O)C(F)(F)F)NC(C)CN(C(=O)C(C)CCc1cccc(F)c1)C c1(C(=O)NCCN(C(C(c2ccccc2)SC)=O)C)cc2cc(Cl)ccc2s1 C(=O)(C#CC1(C)CCCO1)N1C(C(=O)Nc2c(OC)n(C)nc2C)CC1 C1(NC(c2cnc(C3CC3)s2)=O)COCCN(C(c2ccccc2Br)=O)C1 c1(CN(CC(=O)O)C(c2nncn2C2CCOCC2)=O)cn(C2CCC2)nn1 C1(C(=O)NCC2N(C(CCC(=O)N(C(C)C)C)=O)CCC2C)CCCCC1(F)F c1(CC(=O)NC(C(C)NC(C2CC2(F)F)=O)CO)ccc(Cl)c(Cl)c1 c1(C(=O)NCC=C(C(=O)NCc2c(CC)noc2)C)cccc2cncn12 C#Cc1ccc(C(=O)NC(CC(N)=O)C(=O)N2CCN(CC(C)C)CC2)cn1 c1(SC)ccc(C(N2CCN(C(=O)CCc3nnc(S)n3C)CC2)=O)cc1 C=C(C)CCCC(=O)NCc1nc(C2CCN(C(C3CC3(F)F)=O)CC2)n[nH]1 N1(C(C=Cc2c(C)n[nH]c2)=O)CCC2(CCCN2C(=O)COCC(F)F)CC1 CC(C)C(C)(CNC(=O)CC12COC(CF)(C1)C2)NC(=O)Cc1cncs1 CC1CC(=O)NCCN1C(C1CCC2(C1)CC2(F)F)=O C1(NC(C(CCOC)C)=O)CC2CC(C1)N(C(c1cc[nH]c3nccc1-3)=O)C2 C=C=CC(C)C(=O)N(C)CC1COCCN1C(c1cn(CCO)nc1C)=O c1(N(C)CCC2CC2)ccc(S(=O)(=O)NCC(O)CCC2CC2)c(Br)c1 C=C(CNC(=O)COCc1ccccc1)CCNC(C1CSCCS1)=O c1(OC)ccc(Cl)c(C(N2CCC3C(NC(=O)Cn4cnccc4=O)C23)=O)c1 C=CC(C)(CCOC)C(=O)NC(C)CCCNC(=O)CC1CCCNC(=O)C1 C1(CNC(c2c(COC)cc[nH]2)=O)CN(C(C2CCCNC2=O)=O)CCCO1 N1(C(C2C(=C)C2)=O)CCCCC1CN(C(=O)C(CC)=CCCC)C C=Cn1nccc1C(=O)NC1CC(CNC(c2ccc(C(C)(F)F)nc2)=O)C1 c1(-c2nccc(C(C(C3CCN(C)CC3)C#N)=O)c2)ccc(Cl)c(Cl)c1 C(=O)(CCCN=[N+]=[N-])NC(C=CC(=O)Nc1c(C)n(C)nc1)C C1(C(C(=O)NCCN(CCC)CCC)C)CCN(C(=O)C#CC2CC2)CC1 N1(S(CC)(=O)=O)CCC(C(N2CC(CNC(c3cn[nH]c3)=O)(OC)C2)=O)CC1 CCC(CC)CC(=O)NCCOCCN(C)C(C1CCC1C(N)=O)=O c1(NC(C2(NC(CCOCC)=O)CC(F)(F)C2)=O)ccc(OC)c(OC)c1 CCC(C(=O)NC(C1CCN(C(c2cnc3n2CCC3)=O)C1)(C)C)C(C)C C1(C(N2CCC(c3nn[nH]n3)C2)=O)C2CCC(C2)N1C(=O)Cc1ccccc1F C(=O)(CCCCCn1cc(-c2ccnn2C)nn1)NC(C(=O)OC)C1CC=CC1 CC(C)C(C)(CN=c1[nH]c(=N)[nH]c(Cl)c1[N+](=O)[O-])NC(c1coc(C(N)=O)c1)=O n1(CC(N2CCC(NC(CC=C=C)=O)CC2C)=O)cc([N+](=O)[O-])nc1C c1(OC)cccc(C(CNC(C)=O)NC(C2C3CCC2(c2ccccn2)C3)=O)c1 c1(C(N(CCCNC(C(C(CC)C)C)=O)C)=O)cc2c(cc1C)OCO2 c1(CN(C)C)ccc2c(c1)CN(N1CCC([N+](=O)[O-])CC1)C2 O=C1NCC2CN(C(C34COCC3CN(C(=O)CCCC3CCC3)C4)=O)CCC12 C1(C(N2C(CN(C(c3c(CC)ocn3)=O)C)CCC2)=O)CCCCC(C)(C)C1 N1(C(=O)Cn2cc(CO)nn2)CC(C2CN(C(c3cnc4ccccn34)=O)C2)C1 CC(CC(=O)N(CCCCN(C(=O)CN1CC2C=CC1C2)C)C)CC(C)(C)C c1(C(=O)NCC23OCC(CNC(CC(C)CF)=O)(C2)C3)cc(F)c(O)c(F)c1 c1(CC)n[nH]c(-c2nc(CCCCN(C)C)nn2-c2cccc(Cl)c2)c1Cl c1(C(N(CCCNC(CCN(CC)CC)=O)CC)=O)ccc(C)c(P(C)(C)=O)c1 c1(NC(C2CCN(C(c3cccc(OC)c3F)=O)C2)=O)cc(OC)ccc1C#N C1(NC(C(=O)N(C)Cc2ccc(C)cc2)=O)CC(O)CN(C(=O)OC(C)(C)C)C1 CC(C)CC(C)(C)C(=O)NC1(CC(N2CCC(CO)CC2)=O)CC1 O(NC(=O)CC(C1CC1)NC(=O)COc1ncccn1)CC C12(CNC(CC(C)SC)=O)CC1CN(C(c1cnn(CC(C)C)c1)=O)C2 Cc1cc2ccc(C(N3CCC(CNC(=O)CC4(C)CC(F)(F)C4)C3)=O)cn2c1 [N-]=[N+]=NC1CCCN(C(c2cccc3c[nH]nc23)C(=O)NC2CCOC2)CC1 N1(C(CC(=O)OCC)=O)CC2CCN(C(c3cc(CCCl)c[nH]3)=O)CC12 C1(CNC(C(C)=CC)=O)CN(C(c2ccnc(C)c2)=O)CC(C)(C)O1 C1(O)(CN(C(=O)CC2CCCN(C)C2)C)CCN(C(=O)CC2CC2)C1 N1(C(c2c(C)ccn2C)=O)CCC(C2(NC(=O)C(N3CCNC3=O)C)CC2)C1 c1(NC(c2csc(C(=O)Nc3cccc4cc[nH]c34)n2)=O)ccc2ncsc2c1 N1(C(C#CCNC(C2(C)CC(=C)C2)=O)=O)CCC2(CCOC2=O)C1 C(CC(C)(C)CC(=O)NC1CCC(N(C)C(c2nnc(O)cc2C)=O)CC1)OC c1(C(=O)NCC2CCCCN(C(C(C)=CC3CC3)=O)C2)cc(C)cc([N+](=O)[O-])c1 c1(C(=O)OCC)cccc(C(=O)NC(c2ccc(CC(F)(F)F)cc2)C)c1O c1(OC)ccc2c(=NCCC3CC=CC3)[nH]c(=NCc3cccc(O)n3)[nH]c2c1 C1(CNC(Cc2cn(C)nc2)=O)CC(O)CN1C(=O)CSCc1cscn1 N(C1CCc2c(C(=O)O)cccc21)C(C(CC)OC1CCCCCC1)=O c1(C(N2CCN(C(CS(CC)(=O)=O)=O)CC2CCO)=O)nccn2nccc12 C1(NC(=O)NCc2ncccc2Br)CS(=O)(=O)CC1c1ccccc1 C1(CNC(c2cnc(C)nc2)=O)COC(C)(C)CN1C(C1CCCN(C)C1)=O C(=O)(C1=C(Cl)CC1)NC(CC)(C)CNC(=O)CCc1ncc[nH]1 N1(C(C2C=CCC2)=O)CCC2CCC(C1)N2C(c1ccc(O)cc1Cl)=O N12CCCC(C1)C2=O.C1(CNC(C)=O)CCC(NC(=O)COc2cnn(C)c2)C1 CC1CN(C(c2cncc(C(C)(C)C)c2)=O)CC(C)CN1C(=O)C(CO)C(C)C N1(C(Cc2cnc(C)s2)=O)C2CCC(C(N3CCCCC(CO)C3)=O)C1CC2 Cc1nc(=N)[nH]c(=NCC2CC(CNC(c3ccncn3)=O)CO2)[nH]1 N1(C(C2CCCN(S(CCC)(=O)=O)C2)=O)CCOC2(C1)CN(C(=O)CN(C)C)C2 C1(CNC)CCCN(C(=O)CC2CCOC2(C)C)C1 C1(OC)CC(C)CN(C(C2CCCN(C(=O)CC3CCC(=O)C3)C2)=O)C1 N1(C(c2cc(C)sc2C)=O)CCC(C)C(CNC(c2nccc(C)c2F)=O)C1 CC1(C(=O)NCc2ccc(C(=O)NCC3CC4C=CC3C4)cn2)CCC(O)CC1 C1(CNCc2c(C)ccs2)CC12CCc1ccccc12 Cc1nn(C2CC2)cc1C(=O)NCC1(O)CC(NC(=O)COCC(F)F)C1 c1(C(C(=O)NCC2CC(CF)C2)NC(=O)Cn2ccnn2)cccnc1 C(N=c1[nH]c(=NCC(CC)C(C)(F)F)c2sccc2[nH]1)c1c(SC)cc(C)cc1 Cc1ncsc1C=CC(N1CCCCC1CCCNC(C12CC(F)C1C2)=O)=O O=c1ccc2cc(NC(c3nnnn3C3COC3)C3CC3(Cl)Cl)ccc2o1 N1(CC)CCC(C(=O)NC(C)CCN(C)C(C2(CN(C)C)CC=CC2)=O)C1 CN1CC(=O)N(CC(=O)NC2CN(C(=O)CSCc3ccncc3)C2)C1=O c1(C(N(C2CCCN(C(COCCC=C)=O)CC2)C)=O)cnn2c(=N)[nH]cnc12 N1(C(CCOCCOC)=O)CCN(C(=O)COC2CCC2)CC1c1ccccc1 C1(C(N2CCC(CCNC(c3cc(C)sc3C)=O)CC2)=O)CC2(CCC2)CO1 N1(C(C2(C(C)C)CNC(=O)C2)=O)CC2(C1)CN(C(=O)CSC1CC1)CCO2 C1(NC(Cc2ncn(C)c2)=O)CN(C(=O)CC2=CCCC2)CC2(CC2)C1 C=CC(C)(C)CC(=O)NC1CCN(C(c2ccc(CN(C)C)nc2)=O)C1(C)C N1(C(C=C(CC)CC)=O)CCc2[nH]nc(CNC(c3ccncc3Br)=O)c2C1 c1(-c2scc(NC(c3ccc(F)cc3F)=O)n2)cc([N+](=O)[O-])ccc1F Cc1cc(CC(=O)NC(C)(CNC(c2c(C)n[nH]c2C)=O)C(C)C)n(C)n1 n1(CC(=O)NC2(CNC(c3cocc3Br)=O)CC2)cc(C(F)(F)F)cn1 c1(C(=O)NCC(C)NC(c2cc3cc(F)ccc3[nH]2)=O)n[nH]c2c1CN(C)CC2 CCCC(C)C(=O)NCCCCCN1CCN(C(=O)CC2CCCN2CC)CC1 c1(C(=O)NC2CCCN(C(c3[nH]c(=NC)sc3)=O)CC2)ccc2nccnc2c1 C1(C(=O)NCCC(C)NC(C=C(C)Cl)=O)(C)CCCC1.c1(N)ncn(C)n1 C1(C(=O)NC2CCC(C(=O)NC3C(C)(C(F)F)C3)CC2)CC12CCOCC2 N1(C(CCC(=O)OC)=O)CC(CNC(=O)C(C)C(=O)N2CCOCC2)OC(C)(C)C1 Cn1nnc(C(=O)NC2CCN(C(C3CC(C)(c4ccccc4)C3)=O)C2)n1 c1(C(N2C(CNC(c3c(C)csc3Cl)=O)CCC(C)C2)=O)ccc2nncn2c1 C1(O)(C(=O)NCC2C(NC(c3cnc(CC)s3)=O)CCC2)CCCC(C)(C)C1 CC1(CNC(c2conc2CNC(c2ccncc2O)=O)=O)CCC(=O)N1 c1(C(=O)NC2(C)CC(NC(COC(CC)C)=O)C2)cccc(C)n1 N1(C(=O)NCCCOC(C)(C)C)CC(F)(F)C1C1CCC1 c1(OC)ncc(Cl)c(=NC2CC(NC(C3CC4(CC4)C3)=O)C2)[nH]1 C(=O)(CCCC(F)(F)C(F)(F)F)N(CCCNC(c1c(C)con1)=O)C CCC(C)(C)CC(=O)NCC(CC(=O)NCC1(CCO)CC1)OC CC1(NC(C23CC2CN(C(c2ncncc2N)=O)C3)=O)CCC(=O)NC1=O C(CCC(C)C)(C(=O)N(C1CCN(C(c2cnc(N)c(N)c2)=O)C1)C)NC(C)=O C(N=c1nc2c(Br)csc2c[nH]1)C1CCN(Cc2c([N+](=O)[O-])cccc2)CC1 N1(C(c2nccc(CC)c2)=O)CCC2CN(C(=O)CSCCC(C)C)CC12 n1(C(C)C(=O)NCCC2CC2(Cl)Cl)cc(C2(C)CCCO2)nn1 N1(C(CCC)=O)CCCCC(N(C(=O)COCc2ccnn2C)C)C1 CCCC(C(=O)N1CCCC(CCNC(C2(CO)CCOCC2)=O)C1)S(N)(=O)=O N1(C(C(CC(=C)C)C)=O)CCCCC(C2CN(C(c3cncc(Cl)c3Cl)=O)C2)C1 c1(C(N2CCN(C(C(C)=C(C)C)=O)CC2C)=O)cnc2c(cnn2C)c1O N1(C(CC2CCC(C)O2)=O)CCC2(CC2)CC1C(=O)N(CC(F)F)C C12CC3(CCN(C3)C(=O)C=CCN3CCC3C(=O)N1)C2.c1(CC)cccc(OC)c1 N1(C(C(CSC)C)=O)CCN(C)CC1C(=O)NCc1ncn(C2CC2)n1 c1(C(=O)NC(C(C)NC(C2CCC2(C)C)=O)(C)C)ccc(C(F)F)cc1F C1(NC(C(C2CN(C(=O)CCC3CCCC3)C2)OC)=O)CC12CCCCCC2 CC1=C(C(=O)N2CCC(CC(C)C(C3(C(=O)N(C)C(C)C)CC3)=O)CC2)CCC1 c1(C(=O)NCC(NOCC(=C)Cl)=O)ccc(NC)cc1 C12(CNC(c3c(C)noc3)=O)CC(NC(=O)C3=C(Cl)CC3)(CO1)C2 n1(CC)ncc(C(=O)N(C2CCC(CNC(=O)CCC(C)SC)CC2)C)c1C C=CCN(OC)C(=O)c1cn(CCN(C(=O)C(CCC)OCC)CC)nn1 C(CCC(C(=O)NC(C)CCOC)NC(C1CCC2(CC1)CC2)=O)OC c1(C(=O)NC(c2cn(Cc3cccc(C)c3)nn2)C)cc2c(C)sc(C)c2s1 C(=O)(C(C)C(C)C(C)(C)C)N1CC2(CC(NC(c3cc(C)c(C#N)cn3)=O)C2)C1 C1(NC(C2C(C)OCC2)=O)CN(C(c2cnn3cccnc23)=O)C2CCCC12 N1(C(C(C2CCN(C(C3CC(O)(CC#C)C3)=O)C2)F)=O)CCC=CC1COC C1(CC)CC(NC(=O)C(c2ccc(-c3ccccc3)cc2)(C)C)CCN1 N1(C(c2cnn(C)c2C(F)F)=O)CCCOC(CNC(=O)COC2(C)CCC2)C1 Cc1cc(CNC(=O)C(C)(CO)NC(=O)CC2CCCSC2)cc(O)n1 N1(C(c2nc(CC)sc2)=O)CC(NC(C2CC2c2cccnc2)=O)C(O)C1 C=CCN=c1[nH]cc(C(N2C(CNC(=O)C#CC(C)(C)C)CC3COCC23)=O)s1 CC1=C(C(=O)NC2CCC(NC(c3cncc(C(F)F)c3)=O)C2)CCO1 C(=O)(C1=CCC2(COC2)OC1)NC(C(C)NC(=O)Cn1ccc(C(F)(F)F)n1)C N1(C(C(COC)O)=O)CC2CC3CC2C1C3NC(C1Cc2cc(C)ccc2S1)=O N1(C(COCCOCC#C)=O)CCC(COC)C(O)C1.N12CCOCC1CC2=O CC1CN(C(=O)CC2(N(C)C(c3ncc(F)cc3N)=O)CC2)CC(CO)O1 c1(OC)c(F)ccc(C(N2CC3CN(c4nccc(C)n4)CC3C2)=O)c1F N1(c2n(C)c(=O)nc(O)c2)CCC2CCC(C1)N2C(=O)CCCC1CCCCC1 c1(C(=O)NCC2(F)CCC(NC(C)=O)C2)cc(NC(N)=O)ccc1Cl C1(CC)C(=O)NCCCN1C(=O)CC=CCNC(c1cc(C)c[nH]1)=O Cc1ccc2ncc(C(=O)NC3CCC(CNC(C4CC(C)CO4)=O)CC3)n2c1 C(=O)(CC(C(=O)NCCC(C)CCNC(c1cncc(C)c1)=O)NC(C)=O)OC c1(SC)ccc(C(=O)N(C(C)CCNC(=O)C(C)(C)c2cnco2)C)s1 C(c1ccc(F)cc1)=CCC(N1CC2C(CNC(CCSC)=O)C2C1)=O N1(C(CCN(C)CCO)=O)CCC(C2CC2)C1C(=O)NC1CC2(CCOC2)C1 C1(CNC(C2C(CCOC)C2)=O)CCN(C(C2(C#N)CC3(CC3)C2)=O)CC1(F)F C(N=c1ncc(I)c[nH]1)C1CCCCN(C(C2C(=O)NCC2)=O)C1 N1(C(Cc2c(C)n[nH]c2C)=O)CCCN(C(C2CCN(C3CC3)C2=O)=O)CC1 c1(OC)ccncc1C(N1CCCC1C(C)NC(c1nccnc1N)=O)=O CC(O)C(C)(C)C(=O)Nc1cccc(NC(C2CC3CC2C3)=O)c1 CCCC(CCC)=CC(=O)N(C)CC1(NC(=O)C(C)OCc2ccccc2)CC1 c1(C(N(C2CC(C#N)C2)CC(=O)NC(c2ncc[nH]2)CC)=O)ccc(Cl)o1 C1(C(=O)NC(C)CCCNC(=O)C(C)(C)O)CCC2CCCCC2C1 c1(NC(CN(C(=O)COc2ccccn2)CCO)=O)coc2cccc(Br)c12 C1(CNC(C(C)(C)SC)=O)C2CCC1CN(C(C1CCS(=O)(=O)CC1)=O)C2 N1(C(C(C)(OC)OC)=O)CCC2(CC(C(=O)N=c3[nH]ccn4nccc34)=NO2)C1 C(=O)(C1CCN(C)c2ccccc21)N(CCNC(c1c(OC)ccnc1)=O)C1CC1 O=C1CN(CC(=O)NC2CCCCC2NC(C2CC3CC2CO3)=O)C(=O)N1 C1(c2cn(CC(CC)O)nn2)CN(C(C2CC=CCC2)=O)CCO1 C(=O)(C(C)(C)c1nccs1)NC(C1(O)CN(C(=O)CCCC2CC2)C1)C C(=O)(CCC(C)NC(c1ncn(C)n1)=O)NCc1ncc(C)o1 C=CCCCCCC(=O)N1CCCC(NC(=O)CC2CCCCO2)C1C C1(N(C)C(c2csc(-c3nc[nH]n3)n2)=O)CN(C(C23CC(F)(C2)C3)=O)CC12CC2 N1(C(c2n(CC)nnc2C)=O)CCCC2(CCCN2C(C23CCN(CC2)C3)=O)C1 C1(C(=O)NCC2CC2NC(c2n[nH]cc2C2CC2)=O)(CC)CCCO1 CC1CC(=O)NCC1C(=O)N(CCC(C)(C)NC(=O)CCOC1CCCC1)C C1(NC(CC2(C)CC2(F)Cl)=O)CCC(NC(=O)C=CCOC2CCOCC2)CC1 C1(C)(C(=O)NCC(n2cc(C(C(C)C)O)nn2)C)CC(F)(F)C1 c1(C(N2CC3CN(C(CC(C)CN(C)C)=O)CC3C2)=O)cc2c(=O)[nH]ccn2n1 N1(C(C2CC=C(C)CC2)=O)C2CCC1C(NC(c1cc(C)n(CCO)n1)=O)C2 c1(CC(N2CC3(CN(C(=O)CCc4cnn[nH]4)C3)C2)=O)cncc2ccccc12 C1(CNC(CNC(CC)=O)=O)CC2CCC1N2C(c1coc(Br)n1)=O c1(C(=O)NCC2CCCN2C(=O)CC2CC3CCC2O3)cccn2ncnc12 C1(CC)CN(C(c2cc(C)c[nH]2)=O)CCC1NC(C12CC3CC1C2C3)=O N1(C(c2c(COC)nn(C)c2)=O)CCOCC(C(=O)NC(CO)C(C)(C)C)C1 N1(C(c2ccc(N)cn2)=O)CCC(NC(=O)CC2CC(O)C23CCC3)C(O)C1 c1(C(N(C)CC2CCN(C(c3c(C)nc(CC)o3)=O)C2)=O)cc(F)cc(Cl)c1N O=C(C#CC1CCCCO1)N1CCC(CCCO)CC1 CCCC(C(=O)NCC(CC)NC(c1ccn(CCN(C)C)n1)=O)C(C)C N1(C(COCCOC)=O)CC(C(=O)NC(C2CCCO2)(C)C)C(C(C)C)C1 C1(NC(CCc2ccc(C3C(C)C3)o2)=O)CCN(C(=O)C=CC(C)(C)C)CC1C C(CCO)(C(F)F)NC(CC1(NC(CC2(C)OCCO2)=O)CC1)=O C1(NC(C2CCOC2)C)CCCN(C(=O)CN2CCOCC2)C1 N1(C(C2(OCC)CCCC2)=O)CC2C(CC(=O)NCC3COCCN3C)C2C1 N1(C(C=CC(CC)C)=O)CC(CC(=O)N(C2CCCC2C)C)CC1(C)C C12(NC(CCNC(=O)OC)=O)CC(C(=O)NCCCc3ccoc3)(C1)C2 C(CN=c1[nH]c(=NCCc2nc(-c3ccncc3)n[nH]2)[nH]c2ccsc12)OCC N1(C(=O)CN(C(=O)CC2CCC2)C2CC2)CCC(c2ccco2)C1 c1(C(=O)NCC2(F)CC(NC(C3C(C(N)=O)CCC3)=O)C2)c[nH]ccc1=O C1(N(C)C(c2cscc2F)=O)CCCC(NC(=O)Cn2nnnc2C2CC2)C1 c1(N2CC(C(C)NC(c3c(CC)cc(Cl)cc3)=O)OCC2)ncc(C#N)cc1Cl Cc1ccc(C=CC(N2CCC(F)(CNC(=O)CCC3CC3)C2)=O)s1 C1(C)(CC)CCC(C(=O)NCC(C2CCCC2)NC(=O)CCc2cn[nH]c2)O1 c1(OC)ccc(Br)c2c1C(NCC1CCNC3(CCC3)C1)CC2 C(=O)(C(C)CS(C)(=O)=O)NCC1N(C(CNC(CC(C)C)=O)=O)CC2(CC2)C1 Cc1cc(C(=O)NC(CNC(=O)Cn2nccc2C)C(C)C(C)C)cc(C)c1Cl CC(C)CCC(=O)NCN.C1(CC(=O)N)CCOC1=O.C1C(=O)N1CCCN(C)C c1(C(N(C)CC2(NC(C(C(C)C)SC)=O)CC2)=O)cc(F)cc2cnccc12 O(NC(=O)C(CCC(C)C)NC(=O)C(C)NC(N)=O)C(CC)CC c1(OC)ccc(C(CN(C)C)NC(=O)NC(C(F)(F)F)C2CC2(C)C)cc1 C=CCC(C(=O)OC)NC(=O)Cn1cc(-c2cccc(SC(F)(F)F)c2)nn1 C=CC1(C(=O)NCc2cnns2)CCN(C(=O)CC(C)C(F)F)C1 N1(C(C(COC)(C)C)=O)CCN(C(=O)CSCCc2ccccc2)C(CO)C1 N1(C(C(=O)N(C)C)=O)CCC(NC(=O)Cc2ccn(C(F)F)n2)C(F)C1 Cc1cc(=NC(=O)CN2CCC(F)(F)C(CNC(=O)CC3CC3(C)C)C2)[nH]o1 C(CCO)(C(C)(C)C)NC(C=CCN(C)C(c1cnc[nH]c1=N)=O)=O N1(C(C(C)(C)CO)=O)CC2CN(C(C3(S(C)(=O)=O)CC(O)C3)=O)CC2(C)C1 CC1CN(C(c2ccccc2-n2cc(C)nn2)=O)CC1(C)C(=O)OCC(N)=O c1(C(N2CCCC(N(C(C3CC(C)N(C)C3)=O)C)C2)=O)c2c(nn1C)CCOC2 N1(C(C(COCC)N=[N+]=[N-])=O)CCCC(C2CN(C(c3cc(=O)cc[nH]3)=O)C2)C1 Cc1nc2c(s1)CCCC2C(=O)NCCCN(C)C(c1coc2c1CCCC2)=O c1(CC(=O)N(C(CCNC(C(C)OCCC#C)=O)C)C)cc(C)n(C)n1 n1(CCN(C)C)cc(C(=O)NC2CC2CNC(C2(N3CCOCC3)CC2)=O)nn1 C1(C(N2C(CC(=O)OC)CCC2)=O)CC12CCN(C(c1cc(F)n(C)n1)=O)CC2 CCCC(CCC)C(=O)N(C)CCOCCNC(C1CCCC1C1CC1)=O c1(C(=O)NC2(CCCC(=O)NCC(=O)NCC3CC3)CCC2)cc(O)ncn1 C#Cc1ccc(F)c(C(=O)NCCC(CC)(CC)NC(=O)CC2CCOCC2)c1 c1(CNc2ccc(-n3cc(C(=O)O)nn3)cc2)c(F)ccc2occc12 C1(C(=O)NCC(CCCC)NC(CC2(C=C)CCC2)=O)CCOC(=O)CC1 C=C(F)C1(CC(N2CCC(NC(=O)CCCn3nc(C)cc3C)C2C)=O)CCC1 C12(CNC(=O)C(O)Cc3ccccc3)CC1CN(C(=O)CC1(CO)CC1)C2 c1(OCC(N2CCC(C)(C(=O)OCC)C2)=O)c(-c2nn[nH]n2)cccc1Cl C1(NC(CN(CCC#C)C)=O)CCCN(C(c2cccc(N)n2)=O)C1C C(C)(C)(CC(=O)N1CCN(C(C)CNC(c2cc[nH]c2C2CCC2)=O)CC1)OC C#CCCCCCCC(=O)N1CC2CC1(C(=O)NCc1nc(C3CC3)no1)C2 Cc1ccc(NC(=O)COC(C2(c3cn(C)nn3)CCC2)=O)cc1 c1(SC)ccc(Cl)c(C(=O)NC2CCN(C(=O)Cc3ccc[nH]3)CC2C(C)C)c1 c1(C(C(=O)NC2CN(C(c3cc(C)cc(F)c3)=O)C2)C)cn(C)c2ccccc12 N1(C(c2c(CC)ccc(F)c2)=O)CCC2(NC(=O)Cc3cccnc3)CCCC12 C1(C(=O)N(CCCNC(c2sccc2SC)=O)CCO)(NC(=O)OC)CCCC1 C1(C(=O)NCc2c(COC)ocn2)CC(C)CCN1C(C1C2CCC(F)(F)C12)=O c1(C(N2CCCCC(NC(CN(C)C)=O)C2)=O)cc([N+](=O)[O-])c(Br)cc1F C1(NC(c2c(CC)scc2)=O)CN(C(=O)CSc2nncn2C)CCC1O C1(C(N(C)CC2CN(C(c3ccc(C)o3)=O)C2)=O)CCC(=O)NC1 Cc1nc(C(=O)NCC2CN(C(c3sccc3C#N)=O)CC2C)ccc1[N+](=O)[O-] CN1CC(C(=O)NC2(CCNC(c3nc[nH]c3C(F)(F)F)=O)CCCC2)NC1=O c1(C(=O)NCC2C(NC(C(n3ccc(C)n3)C)=O)C2)cc(Br)c(C)cn1 C(CCCC(=O)NC(C(=O)NC(c1cnc[nH]1)C)c1cccs1)SC c1(-n2ccc(C(=O)NCC3CCN3C(c3ccc[nH]3)=O)n2)ccc(F)c(F)c1F C12(C(=O)NC(C(C)F)C)CCCC1CCN2C(=O)C(c1cnn(C)c1)C C1(NC(c2c(CC)cccc2)=O)CN(C(C2(C3CC3)CC2)=O)CC2(CCC2)C1 C=CC(CC)C(=O)NC(C(=O)N(C)CC1(OC)CCC1)c1ccoc1 N1(C(CCc2onc(CSC)n2)=O)CCC2(NC(=O)Cc3cnn(C)n3)CCCC12 N1(CC)CC(NC(=O)C(CC2CCC2)NC(=O)C=CC2CCCC2)CC1=O c1(C(C(=O)NC(C2(O)CN(C(C3(O)CC(C)(C)C3)=O)C2)C)CO)ccc(F)cc1 C1(OC)CC2CCC1CC2C(N1CCC(O)(CCNC(C2CCSCC2)=O)C1)=O c1(SC)ccc(C)c(C(=O)NCC2(O)CCN(C(=O)Cc3ncc(F)cn3)C2)c1 C1(C(N(CC(C)NC(c2c(C(=O)OC)n(C)nc2)=O)C)=O)CN2CCC1(C)CC2 N1(C(CS(=O)(=O)NC)=O)CCC2C(C1)CN2C(=O)CC(C(F)(F)F)OC c1(CC(C(=O)NCC(CNC(CC(=C)C)=O)C)C)ccccc1Cl Cn1cc(CCC(=O)NC2CC2CNC(=O)CC2(C3CC3)CC2)nn1 Cc1coc(C(=O)NCC2CN(C(C3(C)CCCO3)=O)C2)c1 N1(C(CCc2ccn(C)c2)=O)CCC(NC(c2nc(Cl)sc2Cl)=O)C(CO)CC1 C=C(C)CCCC(=O)NCCC1CN(C(=O)COc2ccccc2Cl)CCO1 C1(N(C(=O)C(c2ccccc2Br)F)CC2CCC2)CNC(C(F)(F)F)CO1 Cc1cc2cc(C(=O)NCC3CN(C(=O)C(C)(C)S(C)(=O)=O)C3)ccc2cn1 C1(CC(=O)NC2C(N(C)C)COC2)CCOC1(C)C S(=O)(=O)(c1ccsc1C(N1CCC(NC(=O)C=Cc2cn[nH]c2)C(O)C1)=O)NC Cc1ccccc1C(=O)NCC(=O)NCC(F)CNC(c1sccc1Cl)=O CC1(C)OC2(C(=O)NCCCCCNC(C34CCCCC3C4)=O)CCC1CC2 c1(C(=O)OC)c(C)ccc(C)c1C(=O)NCCNC(=O)C(F)(F)c1cncs1 N1(C(C2(CC(=O)OCC)CCCC2)=O)CCOCC(NC(=O)C2=COCCO2)C1 c1(C(N2CC(O)(CNC(c3ccc(SC)o3)=O)C2)=O)cnc2c(c1)CNC(=O)N2 S(=O)(=O)(c1ccc(F)c(Br)c1)N1CCN(C2CCN(C(=O)C(F)F)C2)CC1 C1(NC(CCC2N(C(C=CC(CC)C)=O)CCC2)=O)COC2(CCCC2)C1 N1(C(C(c2cnn(C)c2)C)=O)CCC(O)(C(C)CNC(c2nccn2C)=O)C1 C1(CC)C(NC(=O)C(C)Oc2cccnc2)CCN1C(=O)CCC=CC(C)C c1(C(=O)NC(C=C)C)ccc(Cl)c(C2=CC(=O)CC(C)(C)C2)c1 c1(C(N2C(C(C)NC(c3cnc(O)o3)=O)CCCC2)=O)cccc2oc(O)nc12 N1(C(C(c2cc(F)cc(F)c2)(C)C)=O)CCCC(NC(C2CCNC2=O)=O)CC1 N1(C(c2c(C)cccn2)=O)CC2CCC(CNC(C3(F)CCOC3)=O)C2C1 C1(C(=O)NC(CCCCNC(=O)Cc2ccns2)CO)CC2CCCC(C1)C2 c1(CC)ccc(C(=O)NCC2(O)CN(C(c3cc(OC)no3)=O)C2)s1 Cc1[nH]nc2cc(C(=O)NC(C)(C)CC3CCC3)ccc12 c1(C(=O)NC2CCCN(C(C3CC34CC4)=O)CC2)c[nH]c2cc(O)ccc12 C1(NC(c2ccsn2)=O)CC(NC(c2ccnc(O)c2Br)=O)C12CCC2 CCC(CC(C)C)C(=O)NC(CN(C)C(c1sc2ccsc2c1C)=O)CC C1(NC(C2CCN(C(C)C)CC2)=O)CCN(C(c2cnc(N)c(Cl)c2)=O)C1(C)C C1(S(=O)(=O)NC(C2CNCCO2)C)(C(=O)OCC)CCC1 c1(CC(=O)NC(C)CCCCCO)cccc(Cl)c1Cl C12(C(N(C3CCN(C(C4CC5CC4C5)=O)CC3)CCO)=O)CCOC1CCOC2 Cc1nn(CC(=O)NC(C(C)NC(C2(CO)CCC2)=O)C(C)C)c(C)c1[N+](=O)[O-] CC(C)(C)C(CNC(=O)CCC(F)(F)F)C(=O)NC1CCC2CCC12 c1(NC(c2cccc3nccn23)=O)cccc2ccoc12 C1(NC(C(Br)=C(C)C)=O)CN(C(=O)CCC(C)C#N)CCC12CCC2 CCCCCS(=O)(=O)CC(=O)NCC(C)CN(C(=O)CC12CC(C1)C2)C C(C(F)(C(=O)NCCCC(=O)NC1CC1)C(C)C)NC(c1c(CC)cccc1)=O CC(C)C(C(=O)NC(C)CNC(=O)Cc1n[nH]c(=N)s1)c1ccncc1 c1(OC(C)(C)C)ccc(NC2CCC(C)(c3ccccc3)C2)cc1CNC(N)=O N1(C(C2(O)CC(C)(C)C2)=O)CCCC(C2CN(C(c3c[nH]c(=N)o3)=O)C2)C1 CN1C2CCC1CN(C(=O)C(CO)NC(c1ccncc1N)=O)CC2 Cc1cc(C(F)(F)F)ccc1C(=O)NCCN(C(C1CC1(F)Cl)=O)C(C)C c1(OC)cnncc1C(=O)NC(C1CCN(C(C2CCC(=O)N2)=O)C1)(C)C CC1CCC(NC(c2cnc(-c3ccccc3)[nH]2)=O)CN1C(=O)CNS(N)(=O)=O c1(C(N2CC(C)N(C(=O)CN3CCCC3=O)CC2)=O)c(F)ccc(N)c1F CCCC(C)CCCC(=O)NCCCNC(=O)C(c1cccnc1)O C(=O)(CCCCCF)N1CCC(C(C)NC(Cc2cccc(OCC)n2)=O)C1 C(CCC(C(=O)NCC)N1CCOC(CC2CCOCC2)C1)OCC C(CSC1CC1)(C(=O)NCCC1COCCO1)NC(=O)OC(C)(C)C CCCC(CC(C)C)C(=O)NC1C=CC(CC(=O)NC2CCC(C(=O)NC)C2)C1 N1(C(c2c(C(C)(C)C)ccs2)=O)CCC2CCN(C(C3CC(=O)N3)=O)CC2C1 C(CCCCCCO)NC(C(C1CCCN(C(=O)CCC2(C)N=N2)C1)C)=O Cc1cc(NC(C2(C)CCCC2)=O)ccc1NC(=O)COCCC(C)C N1(C(c2cnn(C)c2N)=O)CC2CCN(C(C3CC(n4cnnc4)C3)=O)C2C1 c1(C(N(C)CC2N(C(C=C(C)C(C)(C)C)=O)CCC2)=O)ccc(C#N)cc1O Cc1cccc(C(=O)NC2(CCNC(=O)C(F)C(C)(C)O)CCCC2)c1C CN1CCN(C(c2cnc(N)c(O)c2)=O)CC1CNC(C1CCCSC1)=O c1(CC(=O)N(C(CNC(C2(C(=O)OCC)CCC2)=O)C)C)cscc1Br C(=O)(C(C)(C)n1cc(Cl)cn1)NC(C1CCN(C(=O)CNS(=O)(=O)C2CC2)C1)C N1(C(c2n(CC#C)cnn2)=O)CCN(C(c2scnc2Cl)=O)C(CC)C1 C1(C(=O)OC)CC(C(=O)O)CC(C(N2CCC(C(=O)OC)CC2)=O)C1 Cc1cc(C(=O)NCC2CCCC(NC(=O)COCc3scnc3C)C2)n(C)n1 C#Cc1ccnc(C(N2CC(N(C)C(c3ncsc3NC)=O)C(C)(C)C2)=O)c1 C(CC(C)C)(C(=O)NCC=C1CCSCC1)ONC(c1c(CC)n(C)cc1)=O c1(C(CC)NC(c2ccccc2[N+](=O)[O-])C)cc(Cl)cc2c1OCC2 CN1C(=O)CC(C(N2CC=CC2CNC(=O)CC23CCCC2C3)=O)NC1=O CCC(O)C(C)C(=O)N1CCC(C(C)(C)NC(=O)Cc2cnn(CC)c2)C1 C1(C(=O)NCc2onc(COC)n2)CCCC(NC(=O)CNc2ccsc2)CC1 C(C1CCCCCC1)=CC(N1C(CO)CC(NC(Cc2c(C)noc2)=O)C1)=O C1(NC(C(C)Sc2cncnc2)=O)CCCCC1(F)F.C12(C(C)C)CN(C1)C2=O C1(CNC(CNS(N)(=O)=O)=O)CC2(CO1)CN(C(c1cc(Cl)c([N+](=O)[O-])[nH]1)=O)C2 c1(OC)ccc(C=CC(=O)NC2CCC(N(C(=O)C(C)OC)C)CC2)cc1O c1(C(=O)NC2C(OC)(OC)CCCC2)cc2c(C)nn(C)c2s1 C1(CNC(COCCCCC)=O)COC(C)(C)CN1C(c1cccc(C)c1)=O C12CN(CCC1C)C(=O)C2.C1(CCC)(CC)CCCN1C(=O)CCC1CC1 Cc1ccc(N(C(C2CSCCN2C(c2cccc(OC(F)F)c2)=O)=O)CCO)nc1 C1(NC(CC(c2c(C)n[nH]c2C)C)=O)CC2CC(C1)N(c1nnc(C#N)s1)C2 c1(CC(=O)N(CC(c2nn[nH]n2)C)C)ccccc1OCCCC#N CC(C)C(O)CC(=O)NCC(F)CNC(c1cc(-c2ccncc2)no1)=O C=CC(CC)CC(=O)N1CCCC(CNC(c2coc(-c3cn[nH]c3)c2)=O)C1 C1(C)(C(N(C)CC2N(C(c3ncc(OC)cn3)=O)CCOC2)=O)CCCCCC1 c1(C(=O)NCCC2CC(NC(=O)Cc3cnsc3)C2)cc2cccnc2o1 c1(C(=O)NCC2COCCN2C(=O)C#CC2CC2)cc(=O)c2ccc(Cl)cc2o1 N1(C(=O)NCCCc2cncc(F)c2)CCNc2cc(Br)ccc2C1 c1(OCCC)cccc(C(=O)NCCC2CCN(C(=O)C(C)c3ccsc3)C2)c1 Cc1cc(C(=O)NC2CCN(C(c3ncccc3C)=O)C(C)C2)nc(C(F)F)n1 C1(CNC(C2CC(CC)C2)=O)C2CN(C(=O)CN(C3CCC3)C)CC12 N1(C(C(C)Oc2ccc(C)cc2Br)=O)CCCC2CCCCC12 N1(C(C(CSC)O)=O)CCC2(CC1)CCN(C(C1CCC3(CCOCC3)C1)=O)C2 c1(C(=O)NCC(c2cc(OC)c(F)cc2)O)cc2c(F)c(F)cc(F)c2[nH]1 c1(C2(C(=O)NC3(CF)CCC3)CC2)ccc(C(N)=O)nc1.C(=O)(C=CCF)NCC CC(O)(C(=O)N1CC(NC(=O)CCCc2ccc(F)cc2)C(F)(F)C1)C(F)(F)F C(=O)(C1=CCc2ccccc21)NCCC(CCNC(CC(=O)OCC)=O)C c1(C(=O)NC2CC(CNC(C3C(C)(CC)C3)=O)C2)cc(C)nn1C c1(C(=O)NCC2(F)CCN(C(c3ncc(OC)nc3)=O)C2)ccc2c(c1)CCC2 c1(C(=O)NC2C3(CC(NC(CCNC(=O)NC)=O)C3)C2)cccc(C)c1C C1(C2(C)CC2)CC(O)CN1C(C1CCCN1C(C1CCC(F)(F)C1)=O)=O C(=O)(C(C)(C)C(=O)NCC(CC)NC(C1(F)CCC1)=O)NC C1(N(C(C2CC(SC)C2)=O)C)CN(C(=O)C=C2CCN(C)C2)CC1F C#CCCCC(C)C(=O)NC1(CC=C)CN(C(c2cc[nH]c2)=O)C1 c1(-c2nc(C)sc2)cccc(C(=O)NC(C)(C)CNC(C2OC3CCC2C3)=O)c1 c1(C(C)C)nnc(N2CCOC3CC23)n1C1CCCN(C(=O)OC(C)(C)C)C1 c1(C(=O)Nc2ccc(-n3c(C)ccn3)cc2)cc2cccc(C)c2s1 C1(CCNC(CCCOC)=O)C(C)CCCN1C(C1CCCCC1)=O N1(C(C(CO)OC)=O)CCCN(CCNC(=O)C(F)CC2CCCC2)CC1 N1(C(c2[nH]cc(CC)c2)=O)CC2CCC(C1)N2C(C1(C2CC2)CCOCC1)=O C1(CNC(CSCCC)=O)CC2(CCC2)CN1C(c1sccc1C)=O C(C)(C(C)(C)C(=O)NC1(c2cccs2)CC1)NC(C(CO)OC)=O CN1CC(C(=O)NC2CN(C(=O)C=Cc3ccc(=N)[nH]c3)CC23CC3)CCC1=O N1(C(c2c(C)cc(F)s2)=O)CCC2CC(NC(c3csnn3)=O)CCC2C1 c1(NC(C(n2cc(CN3CCC(=O)CC3)nn2)C)=O)cc(=O)[nH]c2cc(F)ccc12 C1(CNC(C(C)OC(C)C)=O)CCC2(C1)OCCO2 N1(C(C2CN(C(C)=O)C2)=O)CC2CC3CC2C1C3NC(c1n[nH]cc1Br)=O c1(C(=O)NC2(CNC(c3cnc(Cl)[nH]3)=O)CC2)ccc(F)c(Br)c1F CCCC(C)(CCC)C(=O)NCCNC(C1CN(C(C2C=CC=CC=C2)=O)C1)=O N1(CCCC23N(C(=O)OC(C)(C)C)CCC2C3)CCCC(C)(C(N)=O)C1 c1(NC)c(C(=O)N(C(C)CCNC(c2c[nH]cc2C(F)(F)F)=O)C)cccc1F C1(C(=O)NCCC(C)NC(=O)CC=CC(C)(C)C)OCCN(C)C1=O c1(CN2CC(O)(CNC(c3c(C)cc(Br)cc3Cl)=O)C2)ccc2nc(O)[nH]c2c1 c1(NC(C2C(NCc3c(O)ccc(C)c3)CCCC2)=O)cc(Cl)c(Cl)cc1I C12(NC(=O)C3=CCCO3)CCCC1N(C(c1nc3ccccn3n1)=O)CC2 Cc1cc(CC(=O)NCCCC2CCN(Cc3ccccc3)CC2)n(C)n1 CC(C)(CC(=O)N1CCC1CNC(C12CCC1CC2)=O)C1CCCCC1 c1(C(=O)NCC2OCCN(C(CC3(C)CCC3)=O)C2)cccc2c1CCC2 C1(OC)CC2CC1CN(C(c1conc1CNC(c1cnccn1)=O)=O)C2 N1(C(c2c(CC)con2)=O)CCCC(CCC(=O)NCC(CC)CCO)C1 C1(O)(CN(C)C(C2(F)CCOC2)=O)CCN(C(=O)CCc2ccc(Cl)cc2)CC1 c1(C(=O)NCC(C)N(C(c2cnc(NC(C)=O)o2)=O)C)nn(C)c(N)c1C c1(C(C)NC(C2C(CC)CCO2)=O)ccc(CNC(C2CCN2CC)=O)cc1 C(=O)(CCC(=O)N1CC(NC(=O)Cc2c[nH]nc2O)CC1C)N(CCC)CCC N1(C(C(CC(C)C)O)=O)CCN(C(=O)C(=CC2CCCC2)O)C2CCCC12 C1(C(C)NC(C2(C(N)=O)CC2)=O)CCN(C(c2ccc(CCF)cc2)=O)CC1 CC1(C)CC1(c1ccccc1)C(=O)NCC1CN(C(C2(CF)CCC2)=O)C1 c1(C(=O)OC)ccc(OC(C)CCF)c(C)c1 N1(C(c2cnc(CC)s2)=O)CCCN(C(=O)CCCC(=O)N(C)C)CC1C Cc1cc(F)c(C(N2CCC(C)C(NC(c3csc([N+](=O)[O-])c3)=O)C2)=O)cc1F c1(C(=O)NCC2(F)CC(NC(C(=O)NC3CC3)=O)C2)ccc2nnc(O)n2c1 C1(O)(CCC2(C)CN(Cc3cccc(N4CCOCC4)c3)C2)CCCCC1 C(=O)(CCC(C)C#N)N(CCC(=O)OCC)C1CC1 N1(C(C2CC(NC(C(n3cc(CC4CC4)nn3)C)=O)C2)(C)C)CCCC1C(C)O C1(C)(NC(C2C(OC)C2)=O)CCN(C(c2cc(C3CC3)on2)=O)CC1 N1(C(C2(CC#C)CCCO2)=O)CC(OC)C(OC)C1CNC(c1cccn1C)=O N1(C(C(CSC)OC)=O)CC2CC1CN2C(c1cncn(C)c1=O)=O c1(C(=O)OC)ccc(COC(C23CC(N=[N+]=[N-])C2C3)=O)c(OC)c1 C1(S(N)(=O)=O)(C(N(C)CC2CN(C(C3CCCCN3C)=O)C2)=O)CCC1 C1(CNC(Cn2ncc(CC)c2)=O)CCC2CN(C(=O)C(F)=CC3CC3)CC12 N1(C(CC(C)SC)=O)CCC(CCC(=O)NC2CN(C)CC2C)CC1 N1(C(Cc2c(SC)cccc2)=O)CCC2(CC1)CN(C(=O)CC1CCOC1=O)C2 C#Cc1cccc(C(=O)NC2CC(CCNC(c3ncccc3F)=O)C2)c1F c1(CCC)onc(C)c1C(N1CC(NC(=O)CC(C)F)C(C)C1)=O C1(CNC(CCCC#C)=O)C(C)CCCN1C(=O)C(C)N(CC(F)(F)F)C N1(c2ccnc(C(=O)OCC)n2)CCCN(C(=O)C(C)(O)C2CCC2)CC1 C1(NC(c2cc(CO)[nH]n2)=O)CCC2CCN(C(C3(CO)CCC3)=O)C1C2 N1(C(C2C(C)(COC)C2)=O)CC2CC(C1)C2NC(c1cc(O)cc(F)c1)=O Cc1[nH]nc(C(=O)NCCCCC(C)NC(=O)C(C)C(F)(F)F)c1[N+](=O)[O-] C1(NCC(c2cccs2)C)CCC(NC(C2(C)CC(C(F)(F)F)C2)=O)C1 C1(CNC(c2ccncc2)=O)CSc2ccccc2O1 c1(C(CC(=O)N(CCCN(C(CC(C)O)=O)C)C)C2CC2)ccc(F)c(F)c1 C(=O)(CCCC(=O)NC1(C)CCN(C(=O)CC2CCCN2C(C)C)CC1)OCC N1(C(C2(CNC(=O)C=CCCC)CC(=C)C2)=O)CC2CC(OC)C(C2)C1 c1(C(c2nnnn2C(C)(C)C)NC(CCCC)CCC)sc2ccccc2c1Cl N1(c2ncc(C)cn2)CC(NC(=O)C(CO)c2ccccc2)CC(C)C1 CC(C(=O)NCC(O)CC(=O)N1CC(C(N)=O)C1)C(C)(C)C c1(C(=O)NCC2N(C(C(C)OCC#C)=O)CCCC2C)c(F)cccc1[N+](=O)[O-] c1(C(=O)NCC2(F)CN(C(CC3(C=C)CCC3)=O)C2)cn2c(n1)CCCC2 C1(NC(c2cc3n(n2)CCO3)=O)CC2(C1)CC(NC(C1(c3nccs3)CC1)=O)C2 C1(C(N2CC(C)(NC(C(C(C)C)C)=O)C2)=O)CC(c2ccccc2[N+](=O)[O-])=NO1 C(C(C)(COC)C(=O)N(C)CC1CN(C(c2nnn(C)c2N)=O)CCO1)OC N1(C(c2ccc(OC)cc2)=O)CCCC(NC(c2cc(C)sc2C)=O)C1C c1(CCC(N2C(CCCNC(C3CCSC3)=O)CCC2)=O)nc2ccccc2[nH]1 N1(C(C2(OCCOC)CC2)=O)CCN(C(c2conc2C(C)(C)C(F)F)=O)CC1 N1(C(C(C)SCC)=O)CC2CCC1CN2Cc1c(C)[nH]c(C(=O)O)c1C Cc1cc(C(N2CCCC(C)(NC(=O)C(O)C(C)C)C2)=O)c2occc2c1 N1(C(C(C)O)=O)CC2(CCN(C(c3ccc(F)cc3Br)=O)CC2)C1 C1(CC(=O)NC(C(C)C)CCNC(=O)Cc2cccnc2F)CCC(C)(C)CC1 n12ccc(n1)C(=O)Sc1nc(cs1)C1CC21.C1(CCC(=O)NC2CC(OC)C2)CCCCO1 C1(C(N)=O)CCCC(C(N2CC(O)(CN(C(=O)CC3CCOC3)C3CC3)C2)=O)C1 C(=O)(CS(=O)(=O)C1CC1)NCC1OCCC(NC(CN(CCC)C)=O)C1 C(=O)(C(F)CC(C)(C)C)N1CCC(C(=O)NC(C)CCCCCO)(CF)C1 N1(C(c2c(CC)c[nH]n2)=O)CCN(C2CCN(C(=O)CN3CC(C)C3)C2)CC1 Cc1cnc(C)c(C(=O)NC(C2CCCN2C(=O)CC2CCCCC2)C)c1 c1(OC)ccc(C(=O)Nc2nc(CC(=O)Nc3cnccc3Br)cs2)c(C#N)c1 c1(C(N(C(CNC(c2cnc(CCCC)s2)=O)C)CC)=O)cc(OC)n(C)n1 CCC(C)(C(=O)O)N(c1ccccc1F)C(=O)CCCSc1cccc(Cl)c1 c1(CNC(C2(CNC(Cc3ccc(OC)nc3)=O)CC2)=O)cc(F)c(C)cc1Cl C(C)(CCC(=O)NC1(CNC(=O)C(C2CCCO2)SC)CCC1)OCC c1(OC)ccccc1CCC(N1CCOCC1CNC(=O)C=CC1CCOC1)=O C(=O)(C1COc2ccccc21)N(CCCN(C(=O)CC1CCCC12CC2)C)C N1(C(c2nccc(C)c2)C(=O)NCC2CCCO2)CCOCC(C2CCC2)C1 C(C(C(=O)Nc1cncnc1O)C(C)C)NC(c1c(C)cnnc1)=O N1(C(CCP(C)(C)=O)=O)CCN2C(=O)C(NC(c3cnc(=N)[nH]c3)=O)CC2C1 C(=O)(C1=NNC(=O)C1)NCCC1CCC(NC(c2c(CC)cco2)=O)C1 CC1(C)CC(C(N2CC=CCC2)=O)CCN1C(=O)CCn1cccc1 N1(C(C2(CNC(c3cncc(-n4cccn4)n3)=O)CC2)=O)CCC2CCCCC12 c1(C(=O)NCCCc2onc(CC(=O)N(C)C)n2)ncccc1N(C)C C1(CC(=O)NCCSCC)CN(C(c2ccnc(SCC)c2)=O)CCO1 c1(C(=O)NC2C(CNC(C3(COC)CCOC3)=O)CCC2)nn(C)cc1COC c1(C(N(C2CCC(NC(C3CC34CCC4)=O)CC2)C)=O)cc(Cl)cc(F)c1N C(=O)(CN=c1[nH]c(=NCCC2CC2(Cl)Cl)c2ccc(OC)cc2[nH]1)NCC C=C(C)C1OCCCC1C(=O)NC1CCC1NC(c1cc(Cl)cs1)=O CC1OCCC1C(=O)NCC(=O)OC1CC(C(=O)N(C)C)C1 Cc1c(F)ccc(C(=O)NCC2CCCN2C(=O)Cc2ccc(Cl)cc2F)c1Cl c1(CCC(=O)N(CC(CN(C)CC2CC23CC3)O)C)nc(C(C)(C)C)no1 n1(C(C)C)ncc2cc(NC(=O)C(C)Cc3ccnn3C)ccc12 CS(=O)(=O)c1ccnc(NCC2CN(C(C3C=CCC3)=O)C2)n1 C1(CNC(C2N(C(Cc3n(C)ccc3)=O)CC=C2)=O)CC12CCOCC2 C(C1=CCN(C(=O)CCN2CCCC2)CC1)NC(c1cncc(CC)c1)=O CC(=O)CCCC(=O)NCC1CN(C(=O)CCSC(F)(F)F)C2CC12 C1(C)(NC(c2cnc(CC)s2)=O)CCCN(Cc2cnc(OC)nc2C)C1 C1(CC(=O)NC2(CNC(c3n(CC#C)cnn3)=O)CCCC2)CC(C)(C)C(=O)N1 N1(C(C(C)=C(C)C)=O)CCC(C(=O)NCc2ccnc(O)c2)CC1(C)C N1(C(C2C(OC(C)(C)C)C2)=O)CCC(F)C(NC(c2cc3occc3s2)=O)C1 C1(OC)CC2CC1CN(C(C1(CNC(=O)COCCN(C)C)CCCO1)=O)C2 C1(CNC(c2ccn(CC)n2)=O)CC(C)CN(C(c2ccc(Cl)s2)=O)C1 c1(C(=O)NC2CCC(CNC(Cc3nn(C)c(Cl)c3)=O)C2)cnn2c1CCCC2 c1(C(N2C(CN(C(=O)Cc3cnn(C)c3)CC)CCC2)=O)ccc(C)nc1N c1(C2CC(F)C2)cccc(Br)c1.C1(C(CN2CCOCC2)(F)F)CCCN1CC(=O)NC CCC(C(=O)N1CCC(CCOC)(NC(=O)C2=C(C)CC2)CC1)C(C)C c1(NC(C2CC(NC(C3(C(=O)OC)CC3)=O)C2)=O)c(C(F)(F)F)cnn1C C1(C(=O)NCCC2(O)CCN(C(=O)C(O)CCSC)C2)(CC)CC(C)(C)C1 N1(C(C2(CCC)CC(=O)C2)=O)CCC(F)(C(N2CCC2CC(C)(C)C)=O)C1 Cc1cccc(C(C)(C)C(=O)NCC2CCCC(NC(=O)C3=NOCC3)C2)c1 c1(C(CNC(=O)NC23CCCC2NCC3)F)cccc(Cl)c1F N1(C(C(C(C)C)C)=O)CCn2ncc(CNC(C34CC(C3)C(C)O4)=O)c2C1 C1(CNC(CCOCCOCC)=O)(COC)CCN(C(C2OCC2(C)C)=O)CC1 N1(C(C(c2cn(C)nc2)O)=O)CC2CCCC2(Nc2cnc(C#N)cn2)C1 C1(NC(C2C(C(=O)OC)C2)=O)C2CC3CN(C(c4[nH]cnc4C)=O)C1C3C2 CC(Cc1cnc[nH]1)C(=O)NCc1ncoc1C1CN(C(=O)C(C)C2CC2)C1 C(=O)(CCCC(=O)N(CCCN(C(=O)CC1CCCCN1C)C)C)OC C1(Cl)(C(N(CCC(C)NC(C2CC(=C)C2)=O)C)=O)CC2CCC1O2 CCC(CC(F)F)C(=O)NCc1cn(C2CCCCN2c2ncc(Br)cn2)nn1 N1(C(CCc2n(C)cnc2)=O)C2CCCC1CN(C(C1CCCCS1(=O)=O)=O)C2 Cc1nc(C2CCCOC2)sc1C(=O)N(CC(C)Cn1ccnc1)CC1CC1 N1(C(c2nc(C)co2)C(=O)NC(c2ccccc2)C)CC(CO)OCC1C C1(C(=O)NCC2N(C(CCCNC(N)=O)=O)CCC2)Cc2cccc(F)c2O1 Cc1[nH]nc(C(C)C)c1C(N1CC2CC2(NC(=O)C(C2CC2)C2CC2)C1)=O C(Cc1ccco1)(C(=O)NCCC1CCCC1)NC(C1C(C(C)(F)F)C1)=O c1(C(N2CC(C)C(CNC(=O)CC3CCOCC3)CC2)=O)c(N)cc(Cl)cc1F CCCCCCC(=O)NCC1C2CN(C(=O)CCc3nc(C)c(C)o3)CC12 C(=O)(C(C)CC(F)(F)F)N(C1CCCN(C(c2sc(CC)c(C)c2)=O)CC1)C Cc1cnc2n1CCC(C(=O)NCCCN(C(=O)C(C)Oc1ccccn1)C)C2 N1(C(c2cc(NC(C)=O)ncc2)=O)CCC2(CCCC2NC(c2cscn2)=O)C1 Cc1ccc2nc(C(=O)NC3CN(C(=O)CN4CCC4C)CC3C)ccc2c1 c1(C(N(C(CN(C(CC2ON=C(CC)C2)=O)C)C)C)=O)cc(C)c2c(c1)CCC2 C1(C(N2CCC(C)(CNC(c3cncnc3C)=O)C2)=O)(CC)CNC(=O)C1 C(CCCCCC(=O)NC(C)CN(C(=O)CC1COC2(CCC2)CO1)C)SC N1(C(C(CNC(=O)CCN2CCOCC2)O)=O)CC2CC1CS2=O c1(CC)ccc(C(=O)N(CCNC(=O)C(C)OCCOC)C(C)C)c(N)c1 C1(c2n(-c3c(CC)cccc3)nc(C3CC34CC4)n2)CC2(CCC2(OC)OC)C1 C12CCN(CC1)C2=O.C1(C(C)(C)C)(CN(C(=O)Cc2cn(C)nn2)C)CCCC1 c1(CC)ccc(C)c(C(=O)NC(C2CCCC2)CNC(c2cc(Cl)no2)=O)c1 C1(C2CC2)(NC(COCCC#C)=O)CCN(C(=O)C(C)SCC)C1 c1(CC)conc1CC(=O)NCC1CCCN1C(=O)CC1CCC1 n1(CC)ccc(CC(=O)NC2CCC2CC(=O)N(CC(CC)OC)CC)n1 C#CCC(C)(C(=O)NOCC=CC=C)NC(c1ccc(C#C)cn1)=O C1(C)(C(=O)NC2(C)CN(C(=O)C(F)=C3CCCC3)C2)CCN(C(N)=O)C1 c1(C(=O)OCC)ccccc1COC(=O)C(F)(F)c1nc(C)cs1 C1(CCN(C(=O)CCNC(c2ccncc2)=O)C)CCCCN1C(=O)CCCF CCCCCCCCCCCCCCC(O)CNCCc1ccsc1Br C1(C(C)CNC(=O)Cn2ccnc2)CCN(C(=O)C(C2(O)CCCCC2)O)CC1 C1(COC)(CNC(=O)CCn2ccc(C)n2)CCCN1C(c1ccccc1)=O c1(C(N(C(C)CNC(=O)C(C(C)O)N(C)C)CC)=O)ccc(=O)n(C)n1 c1(C(=O)NC(CNC(c2cc(C)ncn2)=O)C(C)C(C)C)ccc(C)c(Cl)c1Cl C1(O)(CNC(c2c(CC)nn(C)c2Cl)=O)CCCN(C(=O)CCC(C)OC)CC1 C1(C(=O)NOCCCF)(CC)CCN(C(=O)C(C)(C(C)C)OC)CC1 N1(C(CCC=CC)=O)CC2CC1CN2C(C1(CNC(c2ccccc2)=O)CC1)=O C1(C(=O)NCc2c(CNC(CC(C)C(F)F)=O)cccc2)CC2CCC(C1)C2F c1(C(=O)NC(C2CCCCN2C(=O)C2=CCCC2)C)cccc[n+]1[O-] C#CCCC(C(=O)NCCc1ccc(C)nc1)NC(C1C=CCC1)=O C1(C(N(C(C)CNC(=O)COCCOC2CCCC2)CC)=O)CCSC(C)C1 C1(CC#C)(C(=O)O)CCN(C(C2CCCN(Sc3ccc(Cl)cc3)C2=O)=O)CC1 C1(O)(C(C)NC(C=CSC)=O)CCN(C(C2CC(C)CO2)=O)CC1 C(=O)(C(CC(C)C)n1ccnc1)NCCCCN(C(C(F)=CCC)=O)C c1(C(=O)NCC(CNC(C(COC)C)=O)O)cn(C(C)C)c(=O)nc1O C(=O)(C1=C(c2ccccc2)CCCC1)N(CCNC(=O)Cc1conc1C)CC CC(CNC(N1CCOCC(C(=O)O)C1)=O)CC(F)(F)F c1(CC)cc(C(=O)NC2CC2NC(=O)CN(C)C(C)=O)ccc1F N1(C(C2CCC(CC)CC2)=O)CCC2CCCC(C1)N2c1ccnc(OC)n1 CC1=C(C(=O)NC(C(=O)NCC2=CCCC2)C(C)(C)C)CCC1 C1(NC(CC2CC(=C)C2)=O)CC2CCC1CN2C(c1cnc(OC)nc1C)=O C1(OC)C(O)CC1N=c1[nH]c2ccccc2nc1N1Cc2ccncc2C1 CC1(C)CCC(C)(C)N(S(=O)(=O)Cc2cn3cc(Cl)ccc3n2)C1 c1(OC)cccc(NC(=O)C(C2CC=CCC2)NC(=O)CCc2cn[nH]c2)c1F C(CCC(=O)N(CCC(=O)NC(C)(CO)C1CCC1)CCCO)C1C(C)C1 CCC(O)C(C)(C)C(=O)N1CCN(C(c2ccnc(S)c2)=O)C(CO)C1 N1(C(CS(=O)(=O)NCC)=O)CCN(C(=O)CCC2CCOC2)CCC1C CC(C)C(C(=O)O)N1CCC(CC(=O)N(N2CCCC(C(N)=O)C2)C)C1 N1(C(C(C(COC)C)C)=O)CCCN(C(=O)Cc2cc(OC)ccc2Cl)CCC1 C1(CC=C)(NC(C2CCOC(CC)C2)=O)CCN(C(c2nnn(C)n2)=O)C1 C1(C(=O)NC2CCCN(C(C3(CC(=O)OC)CC3)=O)CC2)CCN2CCOCC12 CC1(C)NC(=O)CC1C(N1CCCC(C)(CNC(c2ccnc(S)c2)=O)C1)=O N1(C(CCOC(C)=O)=O)CC2CCC(CNC(=O)CC(C)c3ccco3)C2C1 CCC(CC(=O)NCCCCC1CN(C(=O)C=CCn2cncn2)C1)C(C)C N1(C(C(=O)NC(C)C)CC2CCC3CC23)CCCC(CO)(CO)C1 c1(COC(C2(C3CCCO3)CCOCC2)=O)ncc(F)cc1F C(C(C)(COC)C(=O)N1CCC(C(C)C(=O)NC(c2nccs2)C)C1)OC N1(C(C(C)NC(c2ccco2)=O)=O)CCC2CCN(C(=O)CSC3CC3)CC12 CCC(CC(=O)N1CC(CCNC(=O)C=Cc2cnc(C)s2)(OC)C1)C1CCC1 C1(NC(C=CCOC)=O)COC2C(NC(c3c(F)ccc(F)c3OC)=O)COC12 S(=O)(=O)(c1ccc(Br)cc1)NCCC(=O)NC1CCSC2(CCC2)C1 C(CCC1CC1)(C(=O)NCc1ccc(O)cc1)NC(c1cn(CC)nc1)=O Cc1nn(C)c(Cl)c1CNC(C1CC1NC(=O)CCOc1cccc(C#N)c1)=O N(C(=NCCOCc1ccccc1)NCC1C2COCC12)CC(=C)C CCC(C(C)C)C(C(=O)NC(C)(C)C)N(c1nc2c(s1)CC(C(=O)OC)CC2)C c1(C(N2CC(C)(CCC(=O)NC3C(C)C3)C2)=O)cc(O)cc(F)c1 c1(N2CC(C)(NC(=O)C(=O)Nc3ncc[nH]3)C2)nccc(S(C)(=O)=O)n1 N1(C(C(=O)NCCOCCCC)=O)CC2CC2(NC(=O)C(C)C2CCC2)C1 C(=O)(CCCC(C)=O)NC(COC)C(=O)N(C)CC1CCC(C)CC1 C(=O)(CCCC(=O)NC1CC(NC(c2ccc(C(C)(F)F)nc2)=O)C1)OCC C1(CCNC(CNC(N)=O)=O)CC(F)(F)CN1C(C1OC2CCC1C2)=O c1(N(CCC)C)nc(N(CCC(=O)NCC)C)nc2ncn(CCN3CCCC3)c12 C1(C2CCC2)(C(=O)NC2C(OC)CN(C(=O)C(C)(CO)OC)C2)CC1(F)F Cc1ccc(CC(C)C(=O)N(CCC(C(C)C)NC(c2csc(F)c2)=O)C)cc1 C(=O)(C#CC1CCOCC1)NCC1(NC(C2C(OC)C2)=O)CCC1 N#CC1CCCC(C(N2CCCC(C(=O)NC3CCC=CCC3)C2)=O)C1 c1(C(=O)NCC(C(N2CCCC(C(=O)OC)C2)=O)O)ccc(=O)n(C)c1 Cc1cc(CC(=O)NCC2(O)CCCN(C(=O)CS(=O)(=O)N(C)C)C2)ccc1Cl N1(C(CCCOCC)=O)CCC(O)(C(C)CNC(c2cccc[n+]2[O-])=O)C1 N1(C(Cc2ccc(C)nc2)=O)CCN(C(c2n[nH]c(C)c2Cl)=O)CC1C c1(C(N2CCCC(N(C(C(C)NC(=O)NC)=O)C)C2)=O)cc2n(n1)CCNC2=O c1(OC)cc(Cl)c(Cl)cc1CNCC1(C(=O)Nc2cc(C(F)(F)F)ccc2C)CC1 c1(CCCC(=O)N2CC(=C(CNC(C3CC(C)(F)C3)=O)F)C2)ccc(F)c(F)c1 Cc1ccc(CCC=O)cc1Cl.N1CCN(C(=O)Cc2ccsc2)C(C2CC2)C1 CON1CC(C(=O)NCC2(O)CC(CNC(=O)CC(C)(C)C3CC3)C2)CC1=O N1(C(CC(C)OC)=O)CCC(C)(C(=O)NCCC(F)(F)F)C1 CC1CCN(C(=O)C=Cc2cnc[nH]2)CC1NC(=O)C=CCN1CCCC1 c1(C(N(C2CCN(C(Cc3c(C)n(C)cn3)=O)CC2)C)=O)ncc([N+](=O)[O-])n1C c1(C(N(CCN(C(CC(CC)C)=O)C)C)=O)cccn(CC(C)C)c1=O C(C(F)C(=O)NC1CC1NC(C1(c2ccccc2)CCCC1)=O)N(CC)CC.O C1(C)(C(=O)NCC2(COC)CCCN2C(=O)CCCC2CCC2)CCCNC1=O C1(NC(CCC(=O)NC)=O)CCC2CN(C(c3ccn(C)c3)=O)CC2C1 N12CCC3C1CCN3C(=O)C(C)C2=O.c1(SC(c2ccccn2)C)ccccn1 C12(C(=O)NCC(CC)(C)OC)CC(CN(C(c3cn(C4CC4)nn3)=O)C1)C2 c1(C(N2CC(COC)N(C(=O)CCS(C)=O)CC2)=O)cc2c(C)ccc(F)c2o1 Cc1cc(CC(=O)NCC2CN(C(C3(C#N)CC3C)=O)C2)nn1C C=C(Br)CC(C)(C)C(=O)NCC1CC1NC(c1ccn(CC(C)C)n1)=O CC(C)(CNC(c1cccc(=O)o1)=O)CC(=O)NC1(CCO)CCOC1 C1(NC(CC(CC)(C)C)=O)CC2CN(c3cc(C)c([N+](=O)[O-])cn3)CC2C1 n1(CC)cc(C(N2CCC(CN(C(=O)C(C)CC(C)C)C)C2)=O)c2ccccc12 c1(C(=O)NCC2C(NC(C(C)c3cccs3)=O)COC2)cnn(C)c1Cl c1(C(=O)NCC(CNC(c2c(CCC)nsc2N)=O)C)cccc2cncn12 N1(C(C(CCCC)N(C)C)=O)CCC2(CCN(C(c3ccnnc3)=O)C2)C1 c1(C(=O)NC2CCC(N(C(CCC=C=C)=O)CC)CC2)cnc2c[nH]nc2c1 N1(C(CCC=C)=O)CCOC2(CCN(C(c3cnc4cc(C)nn4c3C)=O)C2)C1 c1(C(=O)NC(C(=O)OC)C)n[nH]cc1CNC(=O)CCOC1CCCC1 C(C)(C)(CC(F)C(=O)NCC(C)(O)COC)NC(C=C(CCC)CCC)=O C1(CNC(=O)CSc2cccnc2)CC(F)(F)CN1C(=O)CC1CC(F)(F)C1 c1(OC)cc(NC(=O)C(C)(C)O)cc(OC)c1C(C)C C1(C(=O)NC(C)CNC(c2ocnc2C2CC2)=O)(N(C)C)CCCOC1 CCCC(O)CC(=O)NC1CCN(C(=O)Cn2ccc(C)n2)C1 CC1CCC(CC(=O)NC2CC(O)(CNC(c3nocc3Br)=O)C2)CC1 N1(C(C2CCN(C)CC2)=O)CCCCC12CN(C(c1cc(CCCO)on1)=O)C2 c1(C(=O)NC2CC(CCNC(C(C)CC(C)(C)C)=O)C2)ccc([N+](=O)[O-])c(N)n1 n1(C(C)C)ncc(C(=O)NC2CCCN(C(=O)CC3SC(=N)NC3=O)C2)c1Cl N1(C(CC)CC)C(=S)NC(c2cc(OC)c(O)cc2F)C2=C1C1(CCC1)NC2=O N1(C(C2OCCN(C)C2)=O)CC2CCCC2(C(=O)NCc2nccs2)C1 C(C(=O)NC1(CNC(=O)C2=CSCCO2)CCC1)(C(C)(C)C)OC O=S(=O)(c1nc(N2CCC3(CCCCC3)C2)ccc1Br)N1CCSCC1CCO N1(C(c2c(C)c(Br)no2)=O)CCOCC(NC(C2(C)CCCS2)=O)C1 N1(C(CSCCCC)=O)CCC(CO)(CNC(c2cncs2)=O)CC1 N1(C(CCC2CCCN(C(CCC(=O)NCCC)=O)C2)=O)CCCC(C)(O)CC1 c1(CC)c(C)[nH]c(C(=O)CN(CC#N)C(C)C)c1C N1(C(=O)Nc2cn(Cc3ccc(OC)cc3)nc2)CCCC12CCCC2 CCC(CC(=O)OC)NC(c1oc(CNC(=O)Cc2ccn(CC)n2)cc1C)=O c1(C(N2CC(CNC(CNC(CCC)=O)=O)N(C)CC2)=O)cc2nnn(C)c2s1 C#Cc1cn(C)nc1C(N1CC2(C)CC1(C(=O)NC1CCC(C)(C)C1)C2)=O C1(NC(CCC=C)=O)CCN(C(=O)C(c2ccc(F)cc2)F)C(C)C1 c1(C(=O)NCCC2(CNC(c3n(CC)nnc3)=O)CC2)cc2c(s1)CCCC2 CC1CN(C(=O)CN2C(=O)OC(C)(c3ccccc3)C2=O)Cc2cccc(Br)c21 C(=O)(C1=CCCC1C)N1CCC(C(=O)NCC2(CC)CCOCC2)C1C C1(N(C(CCC#CC)=O)C)CCN(C(c2ccc(C)cc2Cl)=O)CC1C c1(N2C(C(=O)Nc3cc(I)ccc3F)CC3CC32)ncc2c(n1)CCC2 C(CCC(C)C)(C(=O)N(C)CC1CCOCC1)NC(CC(CC)C1CC1)=O C1(NC(C(CSC)O)=O)CC2CCC(C1)N2C(c1ccoc1C)=O c1(C(N2CC(NC(CC(CC)O)=O)C(F)(F)CC2)=O)ccc(C)cc1[N+](=O)[O-] C=CCCCCCCC(=O)NCCOCCC(=O)NCCc1cnc(C)[nH]1 C(=O)(C(C)(C)CNC(C1OCCC1CNC(C1CCSC(C)C1)=O)=O)NCC C(=O)(C1CCc2cc(F)ccc21)N1CCC(NC(c2n(CC)nnc2)=O)CC1C CCCCCCNC(C1(NC(=O)CC2C=CCCC2)CC(F)C1)=O c1(C(=O)NCCCN(CCC)C(c2cc(C)nn2CC)=O)ncc(C)cc1C N1(C(c2c(C)cc(CC)o2)=O)CCCC(CC)(NC(=O)Cc2cncc(F)c2)C1 c1(CNC(C(CC)SC)=O)cncc(NC(=O)C(=O)Nc2ccccc2F)c1 Cc1ccc2sc(C(N3CC4CC(C3)C4NC(=O)CC3CCCO3)=O)c(C)c2c1 C(=O)(C1=C(Cl)CCC1)NC1CCC(CNC(=O)CC(O)Cc2ccccc2)C1 N1(C(CC2(NC(C)=O)CC2)=O)CCC(C(=O)NCC(O)C(C)(C)C)(CC)CC1 C#Cc1cccc(NC(C)C(N2CCN(C(=O)C(F)n3cccn3)CC2)=O)c1 C1(NC(COCc2cc(C)on2)=O)CCC12CN(C(c1cc(Cl)ccn1)=O)C2 N1(c2nccc(OC)n2)CC(NC(=O)Cn2c(C)cc(C)nc2=O)CC2(CC2)C1 O=C1CC(=O)NC(C(=O)NC2C=CC(C(=O)NCc3ccncc3Cl)C2)C1 Cc1cc[nH]c1C(=O)N(C1CN(C(=O)C(F)n2cccn2)C1)C c1(N(C(=O)CN2C3COCC2C3)C(c2cnccc2Br)=O)ccccc1F C1(CNC(c2cocn2)=O)C(C2CC2)CCN1C(c1csnc1Cl)=O C12(CNC(c3ccc(C)cn3)=O)CCC1CCN2C(=O)CSc1nncn1C C=CC1CN(C(=O)CNS(=O)(=O)CCCC)CC1NC(=O)Cc1ncccc1C c1(CC)cccc(CC(=O)NCCN(C(c2cc(C)c(Br)o2)=O)C2CC2)c1 c1(C(N2CC(C)C(NC(CCC=CC)=O)C(C)C2)=O)cnc2cccc(C)n12 C(=O)(C1CCCc2nc[nH]c21)NCC1(F)CC(CNC(=O)CCOC2CC2)C1 CC1C(=O)CC1C(=O)NCC1(NC(=O)CC2CCSC2)CCC1 C1(CNC(CCc2ccn(C)n2)=O)CC2COCC2N1C(c1cc(O)cs1)=O Cc1ccc(C(=O)NC(C)C(N2CC3(CC3)CC2C)=O)cc1O C(CCC(=O)N1CCCC1CC(=O)NCC(C1CC1)SC)OC C1(C(=O)NCCC#C)CC(O)CN1C(=O)C(c1ccccc1Br)O.C(C)(=O)OCC N1(C(c2cnc(OC)nc2)=O)CC2CN(C(c3cc(C)c(O)nn3)=O)CC2(C)C1 c1(OC)c(C(=O)NC(CNC(=O)Cc2ccoc2)C(C)C)cccc1C(F)F c1(OC)ccn2c(C(N3CCC4CC3CN4C(C3(F)CCOC3)=O)=O)cnc2c1 N1(C(C(CC)CC)=O)C2CCC(C2)C1CC(=O)NC1C=CC(COC)C1 Cc1nnn(CC(=O)N(CC(O)CN(C)C(C2(O)CCOC2)=O)C)n1 C1(C(=O)NCC2CC(NC(C(CC(C)C)C)=O)C2)CN2CCN1CC2C C1(NC(C2CC3CCC2O3)=O)CCN(C(c2ccnnc2O)=O)CC1 c1(OC)ccc(CC(=O)NC(C)CNC(=O)CC2CC(C)(C)CCO2)c(C)c1 c1(C(=O)NCC2CC(NC(c3cnn[nH]3)=O)C2)c(Cl)ccc2c[nH]nc12 C(=O)(C(O)CCCc1ccccc1)NC(CC)CNC(C1(N(C)C)CCC1)=O FC(F)(F)C(F)(F)Cn1nc(-c2nc[nH]n2)nc1-c1ccc(-n2ccnc2)nn1 C1(CC(C)NC(=O)CC2(C)CC2(Cl)Cl)CCN(C(c2nnn(C)n2)=O)CC1 CC1(C)CCCOC1CC(=O)NCC1(CNC(c2cc(Cl)ccc2F)=O)CC1 C1(CCCNC(c2cccc(=O)o2)=O)CCN(C(c2ccncc2F)=O)CC1 C(=O)(C1=CCCCO1)NCC1CCCC(CNC(=O)C2=COCC2)C1 C(=O)(C1=C(C#N)CCC1)N1CC(NC(c2c(C)cccc2F)=O)CC(OC)C1 c12cccc(c1)CO2.C1(NC(c2[nH]nc(C(=O)OC)n2)=O)CCCC(N(C)C)C1 C1(CN(C(=O)C2=CCOC2)C)COCCN1C(=O)CCCc1ccsc1 N1(C(C(C)C)=O)CCC(N(C(=O)COc2ccc(Br)cc2Cl)C)C(C)C1 Cc1ccc2[nH]c(C(=O)NC3(C)CCCN(C(c4sc(C)cc4C)=O)C3)cc2c1 CC(=O)CCCC(C)C(=O)NCC1(C(N2CCC3(CCC(O)C3)C2)=O)CCCC1 c1(C(=O)NC2CC(CCNC(CSCC(=O)OC)=O)C2)cnc(O)o1 C1(C#N)(C(=O)NCCNC(C2C(=C)CC2)=O)CC12CCC2 C1(C(=O)NC(CC#C)C)CC(C2CN(C(C)(C)C)C2)C1 n1(CC(=O)N(CC(C)CNC(=O)C2=COCCO2)C)sc2ccccc2c1=O C1(C)(C(=O)NCC2CCCN(C(C3C(C)OCC3)=O)C2)CCN(C)C1=O N1(C(C(Br)=C(C)C)=O)CCC(C(C)CNC(=O)C(C)Cn2cccn2)CC1 c1(C(N2CCC(C(C)N=c3nc(C(C)(C)C)[nH]s3)C2)=O)ccc2ccncc2n1 C1(NC(c2ccc(C)nn2)=O)CCC12CN(C(=O)CC1CCCCN1C)C2 N(C1CCCc2c1cnn2-c1ccc2c(c1)COC2)Cc1onc(CC)n1 CC1=C(C(=O)N2CCSCC2CCNC(=O)CCn2cncn2)S(=O)(=O)CCO1 CCC(CC)(CO)C(=O)N1C2CCC1CN(C(=O)CC13CCCC1C3)C2 C(C(C)(F)C(C)(C)F)n1cc(CNC(C2(C)CC3(CC3)C2)=O)nn1 c1(C(C(=O)NCCCSC)N(CC(=O)OC)C(C)C)ccc(C(F)F)cn1 c1(COC)ccc(C(=O)N(C2CCN(C(C3C=C(C)CS3)=O)C2)CCO)s1 CC(C)CCCC(C)C(=O)NCC(C)(C)C(=O)NC1CC(C(F)(F)F)C1 C1(NC(CCCCN(C(C)=O)C)=O)C2CCC1CN(C(=O)C(=O)N(C)C)C2 N1(C(CC(=O)OC)=O)CC2(CO)CC1(C(=O)NC(CO)CC(C)(C)C)C2 CCC(CCC(=O)N(C)CCOCCC(=O)N(CC(O)CC)C)OC n1(CC)nc(C)c(NC(C2CC23CCN(C(=O)CN2CCCCC2=O)C3)=O)c1C C1(NC(c2c(CC(C)C)nc(C)s2)=O)CC(O)CN(C(=O)COCCF)C1 C(=O)(C1Cc2ccc(Cl)cc21)NCC1C(NC(C2(CS(C)(=O)=O)CCC2)=O)COC1 Cc1ccc(F)cc1-c1nnc(CN2CCCC2c2ccco2)o1 C(C1CC1)(C1CC1)=CC(=O)N(CC(C)C(=O)NC1CCN(CC2CC2)C1)C Cc1cccc2c(C(=O)NC(CNC(=O)C(N)=O)CO)coc12 CC1CN(C(=O)C(F)(F)c2cccnc2)CCN1C(=O)CC1CCCC1 N(C1CCCc2ccoc21)C(C1=CCN(C(CCC=CC)=O)C1)=O c1(C(=O)NC2CCC2NC(c2cccc(C3CC3)c2)=O)ccc2oc(S)nc2c1 CC(CC(C)(C)C)C(=O)N1CC(C)(C)CC1C(N1CCOC(C)(CO)C1)=O C(=O)(C(C)(C)C(C)NC(c1cnns1)=O)NC1C(CCOC)CCC1 C1(NC(c2cccc(Br)c2F)=O)CCN(CCOCC2CC2)CC1O n1(C(CC)C)nc(C(N2CCCC(NC(=O)C(C)N(C)C)C2)=O)cc1C C12(NC(Cc3cc(C)no3)=O)CCCC1CN(C(c1cc(C)c(C)nn1)=O)C2 CC1CC(NC(c2cc(C(C)(C)C)nn2C)=O)CN(C(c2nn(C)cc2Cl)=O)C1 C1(OC)CNCC1.C1(C(F)(F)F)(C(=O)OC(C)(C)C)CC1 C1(C(C)NC(=O)C(C)(C)c2cn(C(C)CCC3CCOC3)nn2)CCCC(=O)C1 N1(C(c2c(C)nnn2C)=O)CCC2(CC1)CN(C(=O)Cn1cccc(N)c1=O)C2 Cc1cc(NC(=O)C(O)CCNC(C2(C)CCC(=O)NC2)=O)cnc1O C(=O)(C(O)CC(C)(C)C)NCC1N(C(c2nc(C)c(C)s2)=O)CC1 C1(C#N)(C(=O)NCC2C(CC(=O)N(C)Cc3n(CC)ccn3)C2)CC1(C)C CCCCC(CC)C(=O)N1CC2CCC(C(=O)N(C3CCC3)C3CC3)(C2)C1 N1(CC(=O)N(C(CNC(C2(SCC)CC2)=O)C2CC2)C)CCOCC1 N1(C(C(CC=CC)C)=O)CC2(CC(NC(C34CCC(OC)C3C4)=O)C2)C1 CCCCC(CNC(=O)CC(C)n1cc(Br)cn1)NC(=O)CCSC Cc1[nH]c(C#N)cc1C(N1CCC(CF)(NC(=O)Cn2cccn2)C1)=O C1(O)(CC(N2CCC(CCO)CC2)=O)CCN(C(=O)CCn2cncn2)CC1 c1(OC(CC)C)ccccc1C(N1CC(NC(c2cc[nH]c2C)=O)C(C)C1)=O N1(C(C2CCC(CNC(c3ncc(C)[n+]([O-])c3)=O)CC2)=O)CC2(CNC(=O)C2)C1 C1(CNC(COC2(C)CCCC2)=O)CCCC(NC(c2cccnc2)=O)C1 Cc1ccn(C)c1C(N1CCCC(CNC(c2cc(Cl)ccn2)=O)C1)=O Cc1nc(C(N2CCCC(CO)C2)=O)ccc1-c1nc(CC2CC2)cs1 Cc1cnc(NC(C2CC2NC(=O)Cc2cc(Br)cs2)=O)c(Cl)c1 C1(C(N2C(CO)CC(NC(COCC=C)=O)C2)=O)CN2CCC1(C)C2 c1(C(N)=O)ccccc1C(N1CCC(C(=O)NCC(CO)CO)C1)=O C12(C(=O)NCCC3(O)CN(C(c4c(OC)nsc4OC)=O)C3)CCCN1CCC2 N1(C(C2CC3(CC3)CO2)=O)C2CCC1CC(NC(=O)C(F)(F)C(O)C1CC1)C2 Cc1cc(C(=O)N(CCCC(=O)NC2CCN(C(C)(C)C)C2)C)c(C)n1C CC(N=c1[nH]c2c(c(=NCc3cncs3)[nH]1)SCC2)c1ncnn1C c1(C(=O)NC2(C)CCCN(C(C3(CC4CCC4)CC3)=O)C2)cnn2cnnc2c1 c1(C(N2CCC(CCNC(C(CC)OC)=O)C2)=O)ccc(OC2CC2(F)F)cc1 c1(Nc2ncc(C(=O)OCC)[nH]2)cnc(Cl)cc1C(=O)NCc1ccc(Cl)cc1 C1(NC(C(CC)=CC)=O)CC2CCC1CC2NC(=O)COCCCC(C)C N1(C(CCCOC)=O)CC(CNC(=O)C(C)Cc2ccccc2)CC(C)(C)C1 C(C1=NOC2CN(C(c3ns[nH]c3=O)=O)CC12)NC(=O)C=Cc1nccs1 CCC(CC)C(=O)NCC1CCCN1CC(=O)Nc1ccccc1NC(C)=O n1(C(CC)C)ncc(C(=O)NC2(CF)CCN(C(=O)CCOCCOC)C2)c1C c1(C(N)=O)cocc1C(=O)NCC1CCCN1C(=O)CC1CC2(CC2)C1 C1(O)(CCNC(CCC(C)OC)=O)CCCN(C(c2cnccc2C(F)F)=O)C1 C#CCCCCCCC(=O)NCC(CC=C)C(=O)NCCSC(F)F C1(NC(c2c(OC)ccs2)=O)CCCC(C(=O)NCC2(CCO)CN(C)C2)CC1 C(N=c1nc2sccc2c(N2CCC(C)(N(C)C)C2)[nH]1)c1c(F)ccc(C)c1 CCCCCCCC(=O)NCC(c1ccccc1)NC(=O)C(c1cccn1C)=O Cn1cc(C(N2CCN(C(C3CCC4CC34)=O)CC(O)C2)=O)c2cc(Cl)ccc12 N1(C(C(CCC)NC(C)=O)=O)C2CCC1CN(C(C1CC(OC)C1)=O)C2 c1(CN(C2CC2)Cc2ccc(N)cc2)ccc([N+](=O)[O-])cc1Cl C1(NC(c2[nH]c3nc(C)sc3c2)=O)CCN(C(=O)C(C)NC(N)=O)CC(C)(C)C1 c1(C(N2CC(NC(c3ccc(I)c(Cl)c3)=O)C(F)C2)=O)csc2ccccc12 C(=O)(C1CCCn2cnnc21)N(C)CC1CCCN1c1ncns1 c1(OC)cc(C(N2CCCC2CCCNC(=O)CSCC2CCCCO2)=O)sn1 C1(NC(c2c(CC)n(-c3ccccn3)nc2)=O)CC2COCC(C1)C2 O=[N+]([O-])c1c(Br)cccc1S(=O)(=O)N1CCC1CO c1(C(N2CCC(C(C)C(=O)NCc3cscn3)C2)=O)ccc(O)c(F)c1 C1(c2nnnn2CC)(NCCOCC=C)CC2CC(O)C(C1)N2C c1(Nc2ccc(CNC(=O)C3CC3)cn2)ccc(-c2cscn2)cc1 C1(CNC(C2(C)CC(C)C2)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC1C N1(C(CCS(=O)(=O)NC)=O)CCC(C)(C)C(NC(=O)Cn2nnnc2C)C1 C(=O)(C(C)(C)CN(C(=O)C(C)CC1CCCCC1)CC(C)C)OC C(=O)(C1CCc2c[nH]nc21)N1CC(CC(CNC(c2c(C)sc(O)n2)=O)(C)C)C1 C1(NC(=O)C=CC2CCCC2)CC2CC(NC(c3csc(Br)n3)=O)CC12 c1(C(=O)NC23C(CN(C(C4(C)CC(F)C4)=O)C2)CC3)cc([N+](=O)[O-])cnc1N C(CC(O)CNC(=O)CCN(CCC(C)(C)C)C)NC(C(C)=CC)=O.C(=O)(CCC)N C1(OCCCNC(C2CCCCO2)=O)CCN(C(=O)CCC2CCC(=O)N2)CC1 CC(=Cn1ccnn1)C(=O)NCCC1CN(C(=O)CC2CCCCN2C)CC1C C#Cc1cccc(NC(N2CCOCC2(C)Cc2cccc(C(=O)OC)c2)=O)c1 C1(CC)CN(C(C2CCCCN2C)=O)CC1NC(c1ccc(C(N)=O)cn1)=O C(CCCC(=O)NC(C1CCCN1C(=O)C(C)C)C)(OC)OC C1(NC(c2cc3cnccc3o2)=O)CCN(C(C2(CCF)CC2)=O)C12CCCC2 CC1CC(=O)NC1C(=O)NCC1(CNC(c2cccc(Cl)c2)=O)CC1(F)F C1(OC)CCCN(C(C2CCCC2CNC(=O)C(C)(F)c2ccon2)=O)C1 C(=O)(C(O)C1=CCCCC1)NCCCC(C)NC(c1c(Cl)ccc(Cl)c1O)=O N(C1CCC(NC(=O)C(CC)(CC)OC)c2ccccc21)C(CSCCC)=O C1(NC(CNC(C2C(COC)CC2)=O)=O)CCC(C#N)CC1 N1(C(=O)COCc2ccncc2)CCC(C2(NC(C34CCC(C3)C4)=O)CC2)C1 N1(C(C2CCCC(C)C2)=O)CC2CC(NC(c3cccc(N(C)C)n3)=O)C(C2)C1 C1(C(=O)NCC(CO)NC(C2OCCO2)=O)(OC)CCCOC1 C1(NC(C2(CC=C)CCCC2)=O)CCCCC1NC(C1CCC(C)CC1)=O C1(SC)CN(C(c2ccc(C#N)[nH]2)=O)CC1NC(C1CS(=O)C1)=O c1(C(=O)NC(CNC(CC(=C)C)=O)(C)C2CCC2)cc(=O)n(C)cc1Br C1(C(C)NC(C(C)C#N)=O)CCCN(C(=O)C(C)(C)OCC(F)(F)F)C1 c1(C(N2C(C)(CNC(c3c(OCC)cccc3)=O)CCC2)=O)oc(C)nc1C#N C(CCCCC(=O)NCCOC1CCCC1NC(=O)CCOC1CCCC1)OC C1(N(C(c2c(COC)noc2)=O)C)CN(C(c2c[nH]c(C#N)c2)=O)CC1O c1(CNC(=O)NC(c2ccccc2F)C)ccc(C(C)(C)C)cn1 C(=O)(C(CC(C)C)C(N)=O)N1CC(CNC(c2c(CC)nc(C)o2)=O)(OC)C1 NC(=O)C1=NOC(CNC(=O)C(C2CCC2)NC(c2cccc(F)c2)=O)C1 N1(CCNC(C(C2CCCC2)NC(C=CCCC)=O)=O)CCCCCC1 C#CCCCCC(=O)N(CC)CC1C(O)CCN1C(=O)OC(C)(C)C c1(CCC(=O)Nc2ccc(OC3CC3(F)F)cc2)c(F)cccc1Cl Cc1ccc(C)c(C(=O)NCC2(CNC(c3oncc3C)=O)CCC2)c1C c1(CC(N2CC(CNC(C=CC3N(C)CCC3)=O)C2)=O)ccc([N+](=O)[O-])c(N)c1 CS(C)(=O)=NCC(=O)NC1CCN(C(=O)C=Cc2ccccn2)C(C2CC2)C1 C(N=c1cc(C)[nH]c(=NCC2(CC)CCCCO2)[nH]1)C1(COCC)CCCSC1 C1(O)(CN(C(c2c(C)nns2)=O)C)CCN(C(c2ccncn2)=O)C1 C1(OC)CN(C(c2cn(CCO)nn2)=O)CC1C(N1CCC1C1CCC1)=O C1(C(N(CC(=O)NC2(CCC)CC(=O)C2)C)=O)(OCCOCC)CCCCC1 C1(NC(C=CSC)=O)CCOC2(CCN(C(C3CC3CC(C)C)=O)CC2)C1 c1(C(N2CC(CO)CCC2C)C(=O)NC)nc2ccc(Br)cc2s1 c1(C(=O)NCC2C(C)CN(C(C3C=CCS3)=O)CC2)cnn2ccccc12 C(C(C(=O)N(C)Cc1cnc(C)s1)NC(=O)Cc1cnnn1C)OC c1(CC)cnccc1C(=O)N(C)CC1C2CN(C(=O)CSCC(N)=O)CC12 c1(N(CCCNCCC(c2c(C#N)cnn2C)OC)CCC)ccc(=O)n(C)c1 N1(C(COCCCCCC)=O)C(CNC(=O)CCOCC)CC2COCC12 N1(c2n(C)c(C3CC3c3ccc(F)cc3)nn2)CCC(C2CC2)C1C(n1cccn1)C C(CCCCCC(=O)NCCC1(O)CCC1)NC(C(N1CCOCC1)C)=O C1(CNC(C(CC)C(C)(F)F)=O)CCC2(CCN(C(c3cc(Cl)c[nH]3)=O)CC2)O1 CCC(C)(CO)C(=O)N1CC(NC(=O)COc2ccc(F)cn2)C2(CC2)C1 C12(C(N3CCC(C(C)C#N)CC3)=O)CC(CO1)N(C(C1(CO)CC(C)(C)C1)=O)C2 CC1C(C(=O)NCc2nc(N(C)C)n[nH]2)CCCN1C(=O)C(=O)C1CCCC1 CC(C#N)C(=O)N1CC(N(C)C(c2cc(C3CC3)no2)=O)C1 C1(NC(=O)Cc2ccc(Cl)nc2)CN(C(=O)CC(F)(F)F)C2(CCC2)C1 C1(C(=O)NCCC2CN(C(c3c(C)noc3)=O)CC2C)CCCCC12OCCO2 C(CNC(C1CC1COC)=O)(CC)(CC)NC(CNC(C(CC)C)=O)=O c1(NC2CCC(C(=O)NCCN3CCOCC3)CC2)ncnc(C(F)F)c1Br C1(CCNC(c2ccc(OC)s2)=O)CC2CCC(C1)N2C(C1CC2(CC2)C1)=O C1(CC)CN(C(c2cnc(C(C)=O)s2)=O)CCN1C(=O)Cc1ccn(C(F)F)n1 c1(C(=O)NCCN(C2CCCC2)C(=O)CC2CCNC2=O)cncc(C2CC2)c1 CC1CCC(NC(C2(C#N)CC2)=O)CN1C(c1cc(-c2cccs2)n(C)n1)=O N1(C(CCCCOCC)=O)CC(C)(C)OC2(C1)CN(C(C1CCC(F)CC1)=O)C2 C(=O)(C(C)(F)C(=O)NCCC(C)(C)NC(=O)COC1CCOC1)OC c1(C(CNC(c2n(CC#C)cnn2)=O)NC(=O)CC(C)OC)cccc(OC)c1 c1(N(CC(=O)OCC)CC2CCCO2)nccc(=NCCC#N)[nH]1 c1(C(C(=O)NC2CCC2)N(C2CCCCC2)C)csc2ccccc2c1=O C1(NC(C2CCC(NC(C3(C=C)CCCC3)=O)C2)=O)CCCCNC1=O n1(CC(N2CCCC(CN(C)C(c3nc(Br)cs3)=O)C2)=O)ccc2ccccc12 c1(C(N2CC(CNC(=O)Cc3cnc[nH]3)C2)=O)cnc(COc2ccccc2)s1 N1(C(c2cc(C(=O)OC)ncc2F)=O)CCC2CN(C(c3ccoc3)=O)CCC12 C1(CNC(c2c(C)coc2)=O)(NC(C2CCNC2=O)=O)CCCCC1 CC1(C)CCC(C(=O)NC(C)(C)C(F)(F)F)CN1C(=O)CC1COCC1O CCCC(C(=O)NC(C)CN(C)C(c1nsnc1O)=O)S(N)(=O)=O CS(=O)(=O)c1cc(C(N2CCC(C3CC3)(NC(c3cc[nH]n3)=O)C2)=O)cc(N)c1 C(=O)(CCCCCNC(c1coc2c1COC2)=O)N(CC(C)(C)C)C1CC1 O=C1CCC(=O)NCc2cc(no2)C(=O)NCC(CO)N1.C1(C(=O)O)CCCC1 C(C)(CCC(=O)NC(C)C(CO)NC(=O)Cc1ccnn1C)SC C(C(=O)N(C)OCCC)N(CC(=O)OC)C(=O)CC1CCCC1O c1(C(=O)NC2CCN(C(C(CC)C(C)C)=O)CC2)cc(N)c(Br)c(F)c1 N1(C(C2CC3CC3C2)C(=O)NCCCSC)C2CCC1CN(C(C)C)C2 c1(CN(C(C)C(O)Cc2ccccc2)C=O)ccc(C(F)(F)F)c(F)c1 C(=O)(C1CCCc2nn[nH]c21)NC1C(CNC(C(CC)(C)CC)=O)CCCC1 C1(CC(=O)NC(C(=O)NCC2C(OC)CCC2)CC2CCC2)CCC(C)(C)O1 CCN(OC)C(=O)C(CC1CC1)NC(c1ccn(C)c1C)=O c1(OC)ccc(C(N2CCCC(O)(CCNC(=O)Cn3cnnn3)C2)=O)c(O)c1 c1(-c2cn(CCC)nc2)cccc2[nH]c(C(=O)Nc3coc(Cl)n3)cc12 N1(C(C(=Cc2ccccn2)C)=O)CC2CCC1C2NC(=O)C1=CSCS1 CCCCC(CNC(=O)C=C(CC)CC)NC(=O)CC1(O)CCOC1 c1(NCC(N2CCN(CC)CC2)(C)C)ccc(Cl)c(C)c1Cl c1(C(=O)NC(CCNC(c2cc(C)nc(O)c2)=O)(C)C)cc(F)c(C#N)c(F)c1 c1(NC(C(C)N(C)CC)=O)sc2c(c1C(=O)N(c1cn[nH]c1)CC)CCC2 C12(CNC(CCCCCSC)=O)CCC(CN(C(=O)C3=CCC(C)CC3)C1)C2 N1(C(C)=O)CC(NC(=O)NCCCCc2cnn(C)c2O)C(C)(C)C1 C1(CC)(CC)CC(C(=O)NC(COC(C)C)C(=O)NC2CCN(C(C)C)C2)C1 c1(CNC(C(=O)Nc2cccc(C3CCCN(C)C3)c2)=O)ccc(F)c(N)c1 Cc1cccc(Cl)c1C(=O)N(C1CCC(NC(c2cc(Cl)cn2C)=O)CC1)C Cc1cnn(C(C)C)c1C(=O)NCC(C)N(C(=O)CC1(C)CCCO1)C c1(OC)cc(NC(c2ccc3c(cnn3C(F)F)c2)=O)cc([N+](=O)[O-])c1 C1(CNC(C2C(C(C)(F)F)C2)=O)CCCC(NC(=O)CCc2csnn2)C1 N1(C(CCCOCC)=O)CCCC(NC(c2cn3ccsc3n2)=O)C1C N1(C(CCC(=C)Cl)=O)CCN(C(C2CCC3(CC3)C2)=O)CC1C(C)C N1(C(c2cccn3c(CO)nnc23)=O)CCn2c(n[nH]c(=O)c2=O)C1 Cc1nc(C(C)NC(=O)CC(C2CC2)NC(c2cc(Cl)cs2)=O)n[nH]1 c1(OC)ccc2cc(C(=O)NC3CN(C(c4cnn(C)n4)=O)CC34CC4)[nH]c2n1 C1(O)(C(N(C)CC2CCCN(C(C3(CSC)CC3)=O)C2)=O)CCC(C)(C)CC1 C=C(Cl)CCC(=O)NC(CN(C)C(c1coc(-c2ccccn2)n1)=O)CC CC1COc2c(C(=O)NCC3CCN(C(=O)CC4(CO)CC4)CC3O)cccc21 C(=O)(CCCC(C)N(C)C)N1C(CNC(CN(S(CC)(=O)=O)C)=O)CCC1 Cc1cccc(C(O)C(N2CCC(NC(c3nccn3C)=O)C2)=O)c1 C(c1nc2ccccc2s1)=CC(=O)NC1CCC1NC(C1CCCCC(=O)N1)=O N1(CC(CC)CC)CCCC(C(=O)NC2CCSCC2)C1 Cc1cc(F)c(C(=O)NC2CC(NC(=O)C#CC3CCC3)C2)c(Cl)c1 c1(C(=O)NC(C2CC3CC3N2C(=O)C(O)C(C)(C)C)C)c(F)cc(Cl)cc1F CCC(C)(C)C(O)C(=O)NCC(C)NC(c1coc2c1CCCC2)=O c1(C(N2CCCC(CNC(CC(=O)N(C)C)=O)C2)=O)cc2ccsc2c(O)n1 C1(C)(CNC(c2c(C)n[nH]c2)=O)CN(C(C2CCOC2=O)=O)C(C)(C)C1 C(=O)(CCCCCCN=[N+]=[N-])N(C)CC1CN(C(C(C2CCCCC2)OC)=O)C1 NS(=O)(=O)c1n[nH]cc1C(N1CCCC1CNC(c1cncs1)=O)=O N1(CC(CC(CC)(C)C)=O)CCCC(N=[N+]=[N-])CC1 N1(C(CC2(C)CCCO2)=O)CCN(C(=O)C(F)n2cccn2)CC1.O=C N1(C(c2nccc(CC)c2)=O)CCC2C(CCCN2C(c2[nH]nnc2CC)=O)C1 c1(OCc2ncc(C)o2)cccc(NC(=O)NCc2c(C)coc2C)c1 C1(C(C(=O)N(C2CCCC2)CCN(C(=O)COCC(F)F)C2CC2)F)CCCCC1 C=C(Cl)C(C)(C)C(=O)N1CC2(C1)CN(C(=O)C(C)CC1CCCO1)C2 N1(C(C(COC)(C)C)=O)CCC2(CCCCN(C(=O)C(C)(C)CC(C)(C)C)C2)C1 c1(C(N(C2CCN(Cc3nc(CC)sc3)C2)C)=O)cnn2cccnc12 c1(CC(=O)N(C)CC2CCN(C(CCC(=C)C)=O)C2)c(F)cccc1Br c1(CNC(C(=O)NC(CC=C)C)=O)cnc(CNC(=O)OC(C)(C)C)s1 c1(C(=O)NC2CC3(C2)CN(C(C2CCCCS2)=O)C3)cc(Cl)cc([N+](=O)[O-])c1O C(C(C)(C)C(C)(F)F)NC(C1(NC(CCSC)=O)CC1)=O.C(C)(=O)O Cc1nn(C)c(C(=O)NCCNC(C2CC2c2ccc(Br)cc2)=O)c1Cl C=CCC(C)(C)CNC(=O)CCC1CCN(C(C2CC(N(C)CC)C2)=O)C1 C1(N(C(=O)C(C)(C)C2CCOCC2)C)CCN(C(c2ccc(Cl)o2)=O)CC1 c1(C(C)C(=O)NC2(C)CC(NC(C3CCC3)=O)C2)ccc(-c2ccccc2)cc1 N1(C(CSc2n(C)cnn2)=O)CCCC12CCN(C(c1c[nH]c(C(N)=O)c1)=O)C2 c1(C(N2C3CC(CNC(C=CC=CC)=O)C2CC3)=O)cc2nccc(Cl)c2s1 c1(OC)nc(=NCc2nc3c(s2)COCC3)nc(Oc2cc(F)cc(F)c2)[nH]1 N1(C(C(CC)C)=O)CC2(C)CC1(C(=O)N(C)CC)C2 N1(C(Cc2c(C)noc2C)=O)CC(NC(=O)C(C)OCC2CC2)CC12CCCC2 C1(NC(c2cc(C)nn2C(F)F)=O)COCCN(C(C23CC(C)C2C3)=O)C1 c1(CC)nc(=N)[nH]c(=NCCC2CCN(C(c3nc4nccc(C)n4n3)=O)C2)[nH]1 C1(CNC(c2c(CC)scc2)=O)CC2(CCC2)CN1C(=O)C(C1CCOCC1)C C1(C(=O)NCC2(NC(C3CC4CC3CO4)=O)CCCCC2)CCCCNC1=O C#CCCCC(=O)N1CCC(C(=O)N(CCCC#C)C)O1 Cc1c(C(=O)NC2CCCCC2NC(c2cn(C)nc2C(C)C)=O)cnn1C1CC1 c1(C(N2CC=CC(NC(CCc3c(C)n[nH]c3C)=O)C2)=O)ccc2nccn2n1 c1(C(N2CC(C(C)NC(CCNS(CC)(=O)=O)=O)C2)=O)ccc(C2CCC2)nc1 N1(S(CC)(=O)=O)CCC(C(=O)NC2C3CN(C(=O)CCC(=O)N(C)C)CC23)CC1 c1(CC(=O)NC2C3CCC2N(C(=O)C2=CCCC2)C3)ccc2nc(O)[nH]c2c1 CN1C2CCC1CC(CC(N1CCC(CNC(=O)CC3CC4(CCC4)C3)C1)=O)C2 N1(C(C2N(CC)CC2)=O)CC(CO)(NC(c2n[nH]cc2SC)=O)C1 CC(C)C(O)CCN=c1[nH]c(=NCc2ccnc(OCCO)c2)c2[nH]ccc2[nH]1 c1(C(C(=O)NC2C(n3cc(-c4c(C)ocn4)nn3)CCC2)O)ccc(Br)cc1 c1(C(=O)NC(CC(C)NC(Cc2c(C)n(C)nc2)=O)C)n[nH]c2c1CCSC2 Cc1ccc(C(=O)NCC2C=CCN2C(=O)Cc2nncn2C)cc1C C1(C(=O)NCC2(CO)C(C=C)C2)CCN(C(c2c[nH]c(=NC)s2)=O)C12CC2 C(=O)(C1=CCCN(C(=O)CCOC(C)(C)C)C1)NCc1ncc(OC)o1 c1(C(C(=O)NCC2C(NC(CCC3CC(OC)C3)=O)C2)OC)ccccc1Cl C1(NC(C2(N(C(c3cc(OC)no3)=O)C3CC3)CCC2)=O)CC(C)OC1=O N1(C2C3CN(C(c4c(C)nccc4)=O)C(C3)C2)CC(F)(F)OC(F)(F)C1 C1(C(=O)NC2C(NC(C3(OC)CC3)=O)C2)CC(C(C)C)C1 c1(CC)cc(C(=O)NC23CCN(C(c4cc(F)ccc4C)=O)CC2C3)cc(O)n1 C(=O)(C(C(=O)N(C1CCCCC1NC(C12CC(C)(C1)C2)=O)C)C(C)(C)C)OCC C1(C(=O)NCC(C2CCCCC2)NC(c2ccc(C(C)C)s2)=O)CC=CCC1C CCCCCC(C)CC(=O)NCC1CC(O)(CNC(=O)CCF)C1 N(C1CCCn2ccnc21)CC1N(Cc2ccccc2)CC1C1CC1 N1(C(CC(=O)NCC#C)=O)CC=C(CNC(C2CNC(=O)N2C)=O)CC1 Cc1oc(-c2cnn(C)c2)nc1C(=O)NCC1CCCCN1C(=O)CS(N)(=O)=O c1(C(N2CC3C(CCNC(CC=C)=O)(CC3)C2)=O)nc2ccccc2cc1Cl C(C1CCCN1C)=CC(=O)NCC1(C(=O)NCC2CCCN2C)CC(=C)C1 Cc1nccc(C(=O)NC2C=CC(CC(N3CCC(C)(C(N)=O)C3)=O)C2)n1 C1(N(C(c2cncnc2)=O)CC)CCCN(C(=O)C(C2CC2)C2CC2)C1 C1(O)(CC#C)CC(C(=O)N(CC(C)C(=O)N(C)CC2CC(O)C2)C)C1 c1(C(=O)NC(CN(C(C2C(C)OCC2)=O)C)(C)C)ccc(C#N)[nH]1 c1(C(C)C(=O)N(C2CC(NC(=O)C(F)(F)c3ccnn3C)C2)C)ccc(F)cc1 Cc1cc(C)c(NC(N2CCC3CN(C(c4c(C)n[nH]c4C)=O)CC23)=O)c(C)c1 Cc1cc(CNC(C2CCCC(NC(=O)Cc3cnoc3)CC2)=O)cc(C)n1 CC1(C)CCC1C(=O)NCC1C=CCN1C(=O)CSCc1ccccc1 c1(C(=O)NCC23C(CN(c4cc(N(C)C)ncn4)C2)C3)ccc(C#N)c(Cl)c1 C1(NC(Cc2ncc(C)s2)=O)CCCN(C(c2c(Cl)c(C)nn2C)=O)CC1 c1(C(=O)NCC(C)(C)CNC(C23CCCCC2OCC3)=O)cccc2ccoc12 c1(C(=O)NCC2(O)CN(C(C3CC(=O)N3)=O)C2)ncc(Br)cc1F C#Cc1ccc(C(=O)NCC(C2CCCC2)NC(=O)CCNC(=O)CO)cc1 N1(CCN(C)C)CC(C(=O)NCC(F)CNC(=O)CCn2ccnn2)CC1=O c1(C(=O)NC2CCC(C)N(C(c3nccnc3N)=O)C2)c[nH]c2cc(Cl)ccc12 N1(C(CCSCC(C)C)=O)C2CCC1CC(CCNC(=O)C(F)n1cccn1)C2 c1(NC(C23CC(C(N4CC5CC4CO5)=O)(C2)C3)=O)ccc(Br)c(C(F)(F)F)n1 C(=O)(C1=C(C)OCCS1(=O)=O)N1C(CC)CN(C(=O)CN2CCOCC2=O)CC1 Cc1cccc(CC(=O)NCCC2(CNC(C3CC(C)(C)O3)=O)CC2)c1C CC(C)C(O)C(C)C(=O)N1C2CCC(C(=O)NCC3(C)CC3)C1CC2 C1(NC(c2c(C)cno2)=O)Cc2ccccc2C1NC(=O)C(C)CS(C)(=O)=O CCC(C)CC(=O)C(=O)NC1CCCC(NC(c2c[nH]cc2C(C)C)=O)C1 C1(NC(C(CC2CN(C(C3(OC)CCCCC3)=O)C2)F)=O)CCC(=O)N(C)C1=O C(=O)(C(C)OC1CCCC1)N(C1CCCC1)CCC C1(NC(C2C(C)=CCS2)=O)CCC(C)(CNC(=O)CN2CCN(C)C(=O)C2)CC1 c1(OCC(=O)NC(CCN(C(C)=O)C)C(C)C)ccc2c(c1)CCCC2=O C12(CNC(CC3(C=C)CC3)=O)CC3CC(CC(C3)C1NC(=O)C(F)CC1CC1)C2 Cc1cc(C(=O)NC2CCN(C(C3(O)CCCC(C)(C)C3)=O)C2)c(F)cc1F C1(C(N2CCN(CCN(C(c3c(C)occ3)=O)C)CC2)=O)CCC2(C1)CC2(F)F c1(C(=O)NCC(CCC)NC(C2CCC(NC(N)=O)CC2)=O)cccc(Cl)c1 N1(C2CN(C(C3(C(N)=O)CCC3)=O)C2)CCN(C(C2(N=[N+]=[N-])CC2)=O)CC1 S(=O)(=O)(c1c(Cl)cc(Cl)cc1Cl)N1CCC2(CCCN(C(C(CC)C)=O)C2)C1 N1(CC#CC)CCN(C(C2CCOC2CNC(=O)C(=O)NOC)=O)CC1 c1(C(=O)OC)ccc(C(=O)NCC(O)CNC(c2csc(C3CC3)n2)=O)[nH]1 Cc1ccc(F)c(C(=O)NC(CCN(C(=O)CCCCCF)C)C(C)C)c1O CCCC(C)(CCC)C(=O)NC(c1ccc(C)cc1)CNC(c1cocn1)=O NC1CCCC12CCN(C(=O)CN1CCc3[nH][nH]c(=N)c3C1)CC2 C1(CNC(=O)CCF)CC=CCN1C(=O)C(O)CC1CC1 c1(C(C(=O)OC)C)ccc(OC)c(OC)c1.C#CCC1C(=O)N1 C=CCCCCCC(=O)N1CCC(C(=O)Nc2cnccc2CO)C(CC)C1 N1(C(c2cnc(OCC)s2)=O)CC(NC(=O)CCCc2cnn[nH]2)C(C(F)F)C1 C=CCCCC(C(=O)NCC(=O)NC(C)(C)C)NC(C1CC12CCCC2)=O c1(C(N2CC3(CCN(C(c4cccc(C)n4)=O)C3)C2)=O)cc2ccc(Cl)cc2o1 c1(C(N2CCC3(NC(c4scc(C)c4)=O)C(C2)C3)=O)cc2c(ncn2C)[nH]1 C1(NC(C=CSC)=O)CC(NC(C2CC2c2cn[nH]c2)=O)C(O)C1 C(=O)(C(Cc1cc[nH]n1)NC(c1ncoc1C)=O)N(C(COC)(C)C)C N1(C(c2c(NC(CCOC)=O)cccc2)=O)CCC(C)C(CC(=O)O)C1 C1(CNC(=O)COC2CCOC2)CCC(CNC(C2C3CCC(F)C23)=O)CC1 N1(C(c2cc(C)c(N)cn2)=O)Cc2nccn2CC(NC(=O)CC2CC2(C)C)C1 Cn1cc(C(N2CC(CNC(=O)CNC(C3CCOCC3)=O)C2)=O)c(C(F)F)n1 Cc1ocnc1C(=O)N(C)CCOCCCNC(c1cc(C2CC2)on1)=O c1(C(N2CCC(N(C(C3CCC(O)C3)=O)CC)CC2)=O)cc(OC)nc(OC)c1 CC1(C)CC(C(=O)NCC(O)CN(C)C)CN1C(C1CCC(CO)CC1)=O N1(C(c2occ(C)c2)=O)CC2(CCN(C(=O)C=Cc3ccccc3Cl)C2)C1 N1(C(C(c2ccccc2)N(C)C)=O)CCC(CNC(=O)CC2CC=CC2)C1 CN1CCOC(COC(NOC(c2ccccn2)=O)=O)C1.N(C)C C(=O)(CN=c1[nH]c2ccccc2s1)NCCOCCN(C(C(COC)C)=O)C CC1CC(NC(=O)CCSc2ccccc2)CN(C(c2n[nH]cc2I)=O)C1 C(CCCCC(=O)N1CCN(C(c2n[nH]cc2C(C)C)=O)CC1)SC C(CCC(=O)N(CC(O)CCC)C)N(C(CCSCCCC)=O)CCO O=C1NCC2CCC1N2N1CCCC(C(c2cc(F)ccc2F)=O)C1 n1(C(C)C)cc(C(c2nnnn2C2CCCC2)NCCc2cnn(C)c2)cn1 N1(C(COCCCC(C)C)=O)CCC(NC(C2CC(CC(F)F)C2)=O)CC1C CC(N=[N+]=[N-])C(=O)N1CCSCC1C(=O)NCC12CC(CCO1)C2 c1(CC)cc(N2CCN(C(c3sc(C)nc3C)=O)CC2)nc(-c2ccncc2)n1 C(=O)(C(CC(F)F)NC(=O)C=Cc1cnccn1)NCC(C)(C)n1cccn1 O=C(CCS(=O)(=O)c1ccc(F)cc1)OCc1cscc1C(F)(F)F C1(CNC(C(C)c2ncco2)=O)CC12CCN(C(c1ccoc1Cl)=O)CC2 C1C(C(F)F)CC(=O)N1.C1(C)(C)C(=O)O1.S(=O)(=O)(Cc1ccon1)N(C)C C(=O)(C1Cc2c(Cl)cccc21)NC(CNC(C1=C(CC)OCCC1)=O)(C)C1CC1 C(Cc1ccccc1)(CC(F)(F)F)N(C)C(=O)Nc1cnn(C)c1CCC(F)(F)F N1(C(CN(C(C)=O)C)=O)CCC(N2CCC(CC3CC3)C2)C2(CC2)C1 N1(C(c2ccc(SCCC)cc2)=O)CC2CCC1C2NC(=O)C(O)C(F)F Cc1ncsc1CNC(=O)C=CC(C)(C)NC(=O)CC1CCC2CC12 C(C)(c1ccccc1OC)=CC(N1C2C(CNC(C(CC)(C)CO)=O)C(C2)C1)=O C=CCCC(C(=O)NCC(C)CC(=O)NC)NC(c1cnc2n1CCC2)=O c1(CC)sc(C(N2CCCC2C2CCCN(C(=O)C=CCOC)C2)=O)cc1C N1(C(C=COCC)=O)CCC(C2CCN(C(c3cn(C4CCC4)nn3)=O)C2)C1 CCC(C)(CN=c1[nH]c(N(CCCc2cnccn2)C)nc(=N)[nH]1)C(C)O c1(C(N(CC(C)O)CCNC(C2(C)CCCCC2)=O)=O)ccc2c(c1)nnn2C C(C1=Cc2cc(Br)ccc2OC1)NC(C)(C)CC1CCOC1 C1(NC(Cn2c(C)ccn2)=O)CCCC(NC(=O)C(c2ccc(Cl)s2)C)C1 O=C(CS(=O)(=O)CCO)NCC1CCCN(C(C2CC3CCC2C3)=O)C1 c1(OCC)cc(N2CC(=C(F)CNC(=O)CCC3CCOCC3)C2)ccc1[N+](=O)[O-] CC1(C)CC(C(N2CC(OCCNC(C3CC=CCC3)=O)C2)=O)CNC1=O N1(C(C(c2c(C)n[nH]c2C)C)=O)CCN(C(C2CC2(C)C(C)C)=O)C(C)C1 C(CC(=O)NCC1(C(C)C)CC1)(C(F)(F)F)NC(CCC=CC)=O S(=O)(=O)(c1cnn2ccc(NCC3CCOCC3C)nc12)N(CCCC(C)C)C C1(C(=O)NCCN(C(=O)CCCc2ccco2)C)CC2CCC1C2.C12(CC1)C(=O)N2 C1(CCCNC(CCN(C(C)=O)C)=O)CCN(C(c2ncsc2N(C)C)=O)CC1 CN=c1[nH]cc(C(N2CC(OC)CC2CNC(=O)C2=CCOC2)=O)o1 c1(-c2nc(C)c(-c3nc(S(=O)(=O)c4ccc(Cl)s4)no3)s2)c(C)ccc2ncccc12 c1(C(=O)NC2CCCN(C(CC=CCC)=O)C2)ccc2c(c1)oc1ccccc21 c1(C(N2CCC(C(CNC(C(CC)O)=O)(C)O)CC2)=O)ccn2cncc2c1 N1(C(c2c(C)con2)=O)CCN(C(=O)Cc2ncncc2Cl)C2COCC12 CCC(C)(O)C(=O)NCc1c[nH]nc1C1CCN(C(c2cc(C(F)F)no2)=O)C1 C(=O)(C(C)CS(C)(=O)=O)N(C(CC)CNC(=O)CS(=O)(=O)CC)C N1(C(c2cnn(C)n2)=O)CCC2CC1CN(C(=O)CCn1cncn1)C2 C(=O)(C(CCS(C)=O)N(C)C)NCC1CCC(CN(C(C(C)C2CC2)=O)C)CC1 c1(CNC2CCC(C(=O)Nc3cc(C)c(Cl)cn3)OC2)c(O)cc(F)cc1F CCC(CC)(CN=c1[nH]c(C(C)(C)C)nc(=N)[nH]1)NC(c1cscn1)=O C1(C)(C(N2CC(OC)C(F)C2)=O)CC12CCN(c1nc3cccc(F)c3s1)CC2 O=C1Cc2c(C(=O)NCC(F)CNC(=O)Cn3cnnn3)ccnc2N1 N1(C(C(C)NC(=O)NC)=O)CC(O)CC1C(=O)NCC1(OC(C)C)CCCCC1 c1(CN(CCCC(=O)OCC)C(c2ccc(OC)cc2)C)ccc(Cl)cc1 N1(C(C2=C(C)CCC2)=O)CC2=C(C1)CN(C(=O)C(C)(C)C(N)=O)C2 C(=O)(C1CCCc2sccc21)N(C1CN(C(CC=CC=C)=O)C(C)(C)C1)C1CC1 C(CC(N)=O)(C(=O)NCCOCCN(C)C(C1(F)CCCN(C)C1)=O)NC(C)=O c1(C(=O)NCC(CC)NC(c2cccc(=O)o2)=O)c(OC)c(Cl)cc(O)c1Cl C1(CC)CN(C(C2(C)CC(=C)C2)=O)CC1NC(=O)C(c1ccc(F)cc1)O S1(=O)(=O)c2ccc(Br)cc2N1.N1(Cc2ccc(C3(C)CC3)o2)CCCCC1CO c1(OCC)ccc(NC(C2CCC2NC(C2CC(O)CN2C)=O)=O)cc1 C#CCCCCCC(=O)NC1CCN(C(c2cnc(C)[nH]c2=N)=O)C1(C)C c1(C(N(c2ncc(F)c(OC)n2)C(C(=O)OC)C)=O)ccc2occc2n1 N1(C(CCC(C)=O)=O)CC(NC(C2CC2C2CCCCC2)=O)Cc2ccccc21 C1(NC(C2CCN(C(C)=O)C2)=O)(CF)CCN(C(c2cncnc2)=O)C1 C(=O)(C1COc2ccc(F)cc21)N1CC(NC(C2(CC#C)CCCC2)=O)C(O)C1 C1(CNC(c2ccn(C)n2)=O)CC2COCC2N1C(c1ccccc1)=O C1(CCC)CCCN(C(C2CC23CC(NC2(C(=O)NCC)CCC2)C3)=O)CC1 Cc1cnn(C(C)C)c1NC(=O)NC(C1CCOC1)CO C1(C(N(C2CCC(CNC(c3cc(C)[nH]n3)=O)CC2)C)=O)CC(=O)NC(=O)N1 C(=O)(C(O)C(C)(C)CC)N1CC(NC(CC(CC)CNC(=O)OC(C)(C)C)=O)C1 N1(C(COCC)=O)CCC(N2CCN(C(c3csnc3Br)=O)CC2)CC1 N1(C(C(C#C)(C)C)=O)CCC(C2CCN(C(c3cncc(C4CC4)c3)=O)C2)C1 N1(CC)CC(COC(=O)Cc2csc(C(C3CC3)Sc3ccccc3)n2)OC1=O N1(C(C(C2CC2)SC)=O)CC(CC(=O)NCCC2CCOC2(C)C)CC1C c1(C(c2nnnn2-c2ccccc2)NCC(C)OC)cc(F)c(F)c(F)c1 c1(OCC)ccc(NC(=S)Nc2cnc(C(C)O)cn2)cc1OC(C)C c1(C(N2C(CC(=O)NCC3(c4cccs4)CCCC3)CC2)=O)ccc(F)cc1Cl c1(C(=O)N(c2nn[nH]n2)CCO)occc1Br.CC(F)(F)F c1(NC(C(CC)(C)O)=O)ccc(CNC(=O)C(C)(C)N2CCOCC2)c(C)c1 N1(C(C2(OC)CCC2)=O)CCC(COC2CCN(C(C3(Cl)CC3)=O)C2)CC1 Cc1ccc2c(N(CC(O)CN(C)C(C3NC(=O)CC3C)=O)C)ncnc2c1 C1(NC(c2cccc(OCCF)n2)=O)CN(C(=O)C=Cc2cccs2)CC12CC2 N1(C(C(CSC)O)=O)CCCCC(NC(=O)CCOc2ccccc2SC)CC1 Cc1cc2c(SCCC3SC(=O)NC3=O)csc2s1 c1(NCC(=O)N(C2CC(CNC(=O)C(F)C3CCCC3)C2)C)ccc(C#N)cc1 Nc1c(C(=O)NCC2(NC(C3CC4(CCC4)CO3)=O)CCCCC2)cccc1F N1(C(CSCC(C)C)=O)CCCC1(C)CNC(=O)Cn1ncn(C)c1=O c1(-c2cnc(C3N(C(CCS(C)=O)=O)CCC3)[nH]2)ccc(Cl)cc1Cl C12(CNC(C(CC)C(C)C)=O)CCC(CNC(=O)CC34CCCC3C4)(CC1)CO2 n1(CC)nc2c(c1C(=O)NCC1CC(NC(=O)C(C)CC(F)F)C1)CCCC2 Cc1scnc1C(C1CC1)NC(=O)CNC(=O)Cc1cnoc1 CC(C)CC(C)(CO)NC(=O)COC1CN(C(C2CCCCCCC2)=O)C1 Cc1oc(-c2ccccc2)nc1C(N1CCOC(CS(N)(=O)=O)C1)=O c1(C(=O)NCCN(C(c2cn(CCC)nc2C)=O)C)cnc(O)c2cccnc12 N1(C(c2cn(C)[nH]c2=N)=O)CCC(CO)(CNC(C2(Cl)CC23CCC3)=O)CC1 c1(OC)ccc(C(N2CCOC(CNCc3ccc(OC(F)F)cc3)C2)=O)c(C)c1 C1(COC)(NC(=O)Cc2cccn2C)CN(C(=O)CCC2CCOC2)C1 C#CCCC(=O)NC(C1CC1C(=O)NC(c1nn[nH]n1)C1CC1)C N1(C(CN(S(C)(=O)=O)C)=O)CCCC(NC(C23CC(C)(C2)C3)=O)CC1 C1(NC(c2ccc(SCCCC)cc2)=O)CCN(C(=O)C(C)(C)F)CC1CC C(=O)(C(O)CC1CCOCC1)NCCN(C(=O)C(O)CC1CCOCC1)C(C)C c1(C(N2C(CNC(CCC=CCC=C)=O)COCC2)=O)cnn2cc(C)cnc12 O=C1CC(Cn2cc(C(C3CC3)NC(=O)Cc3csc(-c4nc[nH]n4)n3)nn2)CO1 C1(NC(c2c(OC)ncc(Cl)c2)=O)CN(C(=O)CSCCC#N)C2(CCC2)C1 N1(c2[nH]c3cccc(C#N)c3c2)CCC2(CCCCN(C(C3(C4CCCO4)CCCO3)=O)C2)C1 c1(C(=O)NC2CC(Cn3cc(C4CC4)nn3)C2)cccc(C2(F)CC2(F)F)c1 C(CC(O)CNC(c1ccc(C2CCCCC2)o1)=O)NC(COCCCOC)=O c1(C(=O)NCC(C)(C2CC2)NC(c2ccncc2N)=O)ccc2ncccc2c1 N1(C(=O)Cc2nc[nH]n2)CCN(C(c2ccc(OC(F)F)c(F)c2)=O)C(C2CC2)C1 N1(C(c2c(NC)nccc2)=O)CC2CCC2(CC(N2Cc3c[nH]nc3C2)=O)C1 N#Cc1cccc(S(=O)(=O)Nc2cc(N(C)C)ncn2)c1.N12CCC(O)(CC1)C2 CC1CN(C(=O)C(C2CC2)N(C(=O)Cc2ccccn2)C)CCS1=O C1(C(=O)NCC(CNC(c2cnn(CCN(C)C)c2)=O)OC)CCCCO1 c1(N2CCC(NC(CC3CN(C)C3)=O)C(F)C2)nc2ccc(O)cc2s1 Cc1cc(C(N2CCC(F)(CNC(=O)CC34CCC(CC3)C4)CC2)=O)cc(N)c1 N1(C(c2nc(C(C)C)sc2)=O)CC2CC1C2NC(=O)COc1ccsc1Cl c1(CCCC=C)ccc(-c2nc(-c3ccc(CN(C)C)cc3)nn2C(C)C)cc1 C12(NC(CC=C)=O)CCC(CC1)N(C(=O)CCc1cccc(C)c1Br)C2 c1(C(=O)NCC2(NC(C3C(C(C)(C)C)C3)=O)CCC2)ccc2nccnc2c1 C(c1ccncn1)=CC(=O)NCC(CNC(C(c1ccccc1)OC)=O)(C)O C1(CC(=O)NCC2C3CC2N(C(c2nocc2C2CC2)=O)C3)CCS(=O)(=O)C1 C=C(CNC(c1cnn(CCOC)c1)=O)CCNC(=O)CC1CCCC1C c1(NC(CN(C)C(c2cc(C(N)=O)no2)=O)(C)C)cc(O)ncn1 C12(NC(=O)C#CC3CCCC3)CCCC(CN(C(=O)CCn3ccnc3)C1)C2 c1(SCC(=O)NC2(CCCNC(C3(CC)CC3)=O)CC2)ccc(O)cc1 Cc1nncn1NC(=O)C1C(C)CCN1C(=O)Cn1cc(Cl)cn1 c1(N(C)C)ncc(Br)c(C(N2CC3CC(C2)N3C(C2CCCC2O)=O)=O)n1 C1(C(=O)NCC2(CC(=O)NCCCCC#C)CC2)CCCCC1O C1(C(C)CC)CC(=O)N1.C#Cc1c[nH]nc1C(N1CC(C)CC1CC)=O c1(SC)ccc(C(=O)NC2CC2NC(c2n[nH]cc2C(F)(F)F)=O)s1 N1(C(C(CCN(C)C)NC(=O)C#CC(C)(C)C)=O)Cc2cccc(O)c2C1 CCCC(CC(C)C)C(=O)N1CCC(C(=O)NC2(C)CCC(O)CC2)C(C)C1 C1(NC(c2sc(CC)c(C)c2)=O)CCN(C(C2CCN(C(=O)NC)C2)=O)C1(C)C c1(-c2nc(C(CC)C)nn2C(C)C(C)C)[nH]c2ccc(Br)cc2c1Cl c1(CNC(=O)NCCCc2ccc(O)nc2)cc(F)c(Cl)c(Cl)c1 N1(C(C(CCC)O)=O)CC(NC(c2ccc3oc(S)nc3c2)=O)CC12CCCC2 c1(C(=O)NC2(CNC(=O)CC3(O)CCOCC3)CC2)ncnc2c1CCCC2 C1(CC)CCc2[nH]nc(C(N3CCOC(CN(C)C(=O)C4CC4)C3)=O)c2C1 CN1C(=O)CCC1C(=O)NC1C2CC1N(C(C1CC1(C)C(F)F)=O)C2 c1(OCC(=O)N(CCNC(C(CCC)OC)=O)CCOC)c(C)cccc1Cl C1(C(N(CC(CC)C)C)=O)CCN(C(C2CCCOCC2)=O)CC1 c1(OC)ccnc(C(=O)NCC2CCCC(C(N3CCC3CO)=O)C2)c1OC C1(OC)CN(C(C2NC(=O)OC2C)=O)CCC1NC(c1scnc1C(C)C)=O C1(C(=O)NCC=C(C)C)CCC(CC2(NC(CC3N(C)CCC3)=O)CCOC2)CC1 O=C(C1=CCCOCC1)NC12CCCC1N(C(c1cnns1)=O)CC2 O=C1CCN(C(c2cccc3ncnn23)=O)C2CCCCC12 C1(OC)CC(CC(=O)NC(C(=O)NCCC(=O)NC(C)(C)C)C2CC2)C1 c1(C(N2C(CNC(CC3(C)CC3)=O)COC(C)(C)C2)=O)cc([N+](=O)[O-])ccc1N N1(C(c2ccc(C(C)C)o2)=O)CCCC(O)(CNC(c2cn3ccnc3s2)=O)C1 c1(C(=O)NC2C(NC(C(c3ccccc3O)OC)=O)CCC2)ccc([N+](=O)[O-])[nH]1 C1(CCC)CN(C(C2(Cl)CC2(C)C)=O)CCN1C(c1cc(OC)no1)=O C(=O)(C1=NOC2COCC12)NC(CCN(C(C=C(C)Cl)=O)C)C(C)C C(=O)(C#CC1CCOC1)N1CCC(C(=O)Nc2cccc(F)c2)OCC1 C1(CC=C)(NC(=O)Cn2cnnn2)CCN(C(=O)CSc2ccccc2Cl)C1 CC(CC(=O)NCC12CC=CC(C1)OC2)C(C)(C)NC(c1ccn(C)n1)=O CC1CCC=C1C(=O)N(C)Cc1ccccc1.C12CSCN1C2=O c1(C(N(CC(C)O)CCNC(c2cc(SCC)[nH]n2)=O)=O)ccc(OC)c(Cl)n1 CCC(CCC(=O)NCCOCC1CC1)NC(=O)C(C)NC(C)(C)C C1(CC)CNC(=O)CN1C(=O)C(CC(F)F)NC(=O)CCc1ccsc1 CC1=C(C)CN(C(=O)CC2CC3(C2)CN(C(c2ccoc2Cl)=O)C3)CC1 c1(OC)ccc2c(=O)c(C(N3CC(CS(C)=O)C3)=O)c[nH]c2c1OC CS(=O)(=O)c1ccc(C(F)C(=O)NOCCCC(F)(F)F)cc1 C(=O)(C(O)(C(F)(F)F)C1CC1)N(CCCN(C(C(CCCC)N(C)C)=O)C)C Cc1nc(C2CC2)ncc1C(=O)NC1CCN(C(C2(C3CC3)CC2)=O)CC1C C1(CC(=O)NCCN(C(C2CCCCCC2)=O)CC)CCC(F)(F)CC1 C(=O)(CCCCC(=O)NCCCC1CCCCN1C(c1nnc(S)n1C)=O)NC c1(CSCC(=O)NC(CNC(=O)C=Cc2cn[nH]c2)C2CC2)cccc(Cl)c1 c1(C(=O)NCC(CC=C)NC(c2c[nH]cc(C)c2=O)=O)c(F)ccc(C#N)c1F C1(CC)CC(O)CCN1C(C1(C)CC(O)CN1C(=O)CSc1nc[nH]n1)=O c1(COCC(=O)NCC2CN(C(c3c(C)noc3C)=O)C2)nn(C)cc1[N+](=O)[O-] C(=O)(C(CCF)NC(c1nc[nH]n1)=O)NC(C)CN=[N+]=[N-] N#Cc1ccc(S(=O)(=O)Nc2ccc(Cl)cc2)c(NCCN2CCCC2)c1 C1(C(=O)NC2CC(OCC(=O)NCc3ccc(F)c(O)c3)C2)CCCC12CCC2 C1(NC(C2(C=C)CCOCC2)=O)CCN(C(=O)CC2C=CCC2)CC(O)C1 CCCC(C(=O)NC1CCOCC1NC(C1(C(N)=O)CC1)=O)C(C)C C1(C(=O)NCCCCC)CC(=O)CN1C(C1CC=CCO1)=O c1(C(=O)NCCCN(CCCCNC(C2C(CC)C2)=O)C)ccc(CN(C)C)o1 C(=O)(C(CCc1ccccc1)C(F)(F)F)N(CC(CC)C)CC(F)(F)F C1(CNC(c2c(COC)cc[nH]2)=O)CCCN(C(c2c(Cl)cnn2C)=O)C1 CN1CCn2nc(C(=O)N(C3CCCC3)CCc3nn[nH]n3)cc2C1 N1(C(C2C(NC(c3cnn[nH]3)=O)C3CCC2C3)=O)CCC(C2CCC2)C1 c1(C(N2CC3CC(NC(C4(CCF)CCC4)=O)CC3C2)=O)ccn2cncc2c1 Cc1cc(C(=O)NC(CC2CCCC2)C(=O)NCCC2(C)CCOC2)ccc1O c1(C(=O)NCC2C(CNC(c3ncn(CC)c3)=O)C2)cccc(N2CC=CC2)c1 Cc1cc(C=CC(=O)NCC(C)N(C)C(c2cc(C(F)F)ccn2)=O)ccc1F N1(C(C(C)CSc2ccccc2)=O)CCCC(CO)(NC(=O)C2=CSCCO2)C1 C1(C)(CC)CC(NC(C2CC=CC(NC(=O)CCC3CC3(C)C)C2)=O)CCO1 C1(NC(C(CCC)OCC)=O)CCCN(C(c2nn(C)nc2C(F)(F)F)=O)CC1 c1(OC)ccc(C=CC(=O)NC(C)CN(C(=O)C(F)CC2CC2)C)c(OC)c1 c1(NC2C(C)CCCC2)ccc(S(=O)(=O)NC2(c3ncccn3)CCC2)cc1Cl Cn1ncc(C(N2CC(NC(=O)C3=CCCC3)CC(C)(C)C2)=O)c1S(C)(=O)=O C(=O)(C(F)(F)C(F)(F)F)N(CC(C)(C)NC(c1cc(C)[nH]c1C)=O)C CC(CO)C(=O)N(C(CNC(c1csc(-c2ccccc2)c1)=O)C1CC1)C c1(C(C(=O)NCC(CC)NC(c2cocn2)=O)(C)C)ccc(Cl)cc1 N1(C(C2C(C)CC2)=O)CCC(C)(C)C(C(=O)NCC2(O)CCSC2)C1 c1(C(N(C2CCCC(NC(c3cc(C)c(C)[nH]3)=O)C2)C)=O)cnc2nccn2c1 Cc1ncc(CCC(=O)NC2(c3ccc(Br)cc3)CCCOC2)c(O)n1 C(=O)(CC1=CCCC1)NCC1C(C)CCN1C(=O)COCc1ccccc1 c1(C(N2CC(NC(c3ccc(Br)cn3)=O)C(F)C2)=O)ccc2c(Cl)ccnc2c1 C1(NC(CCc2cc(C)n(C)n2)=O)CCN(C(c2nnn(C)n2)=O)C12CC2 C1(C(C)NCc2ccc(NC(C)=O)cc2)CC12CCCCC2 C1(NC(C(=O)NCC)=O)CC12CCN(C(=O)Cc1cc(OC)c(O)cc1F)CC2 C1(NC(=O)CC2CCOC2)CCN(C(=O)CNC(C2CCC2)=O)CC1CO N1(C(Cn2cc(NC=O)nn2)=O)CC2(CCN(N3CC4CCCC3C4CO)C2)C1 N1(CCC(CC)(C)C)CCC(=O)N(Cc2ccc(CC(N)=O)cc2)C1=O CCCCNC(=O)CSC1CCC1 N1(C(CC(C)(C)N(C)C(C2(C)CCCOC2)=O)=O)CCn2ccnc2C1 C#CC1CCN(C(=O)C(CC)NC(c2c[nH]c(C(N)=O)c2)=O)C1 c1(C(=O)NCC(CNC(Cc2c(C)ccnc2)=O)F)c(F)ccc(F)c1Cl S(=O)(=O)(c1ccccc1[N+](=O)[O-])N(CCN(CCC)C(c1ccnc(OC)n1)=O)C c1(CN(c2ccc(C)c(Br)c2)CCCC)ccc(OC)c(OC)c1 C#Cc1ccc(C(=O)NCC2CCN(C(=O)Cn3cc(Br)c(C)n3)C2)c(C)c1 CCC(C)C(=O)C(=O)NCC1CC2(CC(NC(=O)CC3CC=CCC3)C2)C1 N1(C(C2(COCC)CCC2)=O)C(C(=O)NCC2CCCS2)CCC12CC2 C1(NC(C23CC(NC(C(CC)OC)=O)(C2)C3)=O)CCCC(C(C)C)C1 N(C(=NCCCCl)N1CCC(c2nncs2)C1)C1C(OCC(F)(F)F)C1 N1(C(CCC)=O)CCCCC1C(N1CCC(N(C(c2ccncc2)=O)CC)C1)=O C(=O)(CC1OCc2ccccc21)N1CC(C(N)=O)(CNC(CC(C)O)=O)C1 N1(CC(=O)N(CCC(C)NC(=O)C(F)=CC2CC2)C)CC(=O)Nc2ccccc21 N1(C(C2C3CCCCC23)=O)CC(C2CC2)(C(N2CCOC3CC23)=O)C1 C1(C(=O)NCCCCC2C(C)C2)CCCCC1NC(c1cc[nH]c1)=O c1(C(=O)NCC2(NC(C(C(C)C)NC(COC)=O)=O)CC2)c(O)nnc(C)c1C C(=O)(C1=CCCCC1)N1C(CC=C)(C(=O)OCC)CCC1.C(=O)CCCn1ccnc1 C1(C(=O)NCCCC(C)NC(C(C)Cn2cccn2)=O)CCC(O)CC1 CC1CCC(CO)(NC(=O)CCN(C)C(c2cccc(CC#N)c2)=O)C1 N1(C(C2CC2c2csc(Br)c2)=O)CC2CCN(C(C3(F)CC3)=O)CC2C1 C1(CC=C)(NC(=O)CC(F)(F)F)CCCN(C(=O)CCC2(C#N)CCC2)C1 Cc1oc(C(N2CCC(CNC(=O)C(O)Cn3cncn3)C2)=O)cc1Br Cc1cc(C#N)nc(N(Cc2cccc(F)c2Br)CC2CCCNC2)n1 N1(C(=O)Cc2ccc(C(=O)OC)cn2)CC2CC(C1)C2C(=O)OC c1(-c2cn(C(C(=O)NCC(CC)(C)CO)C)nn2)ccc(C)c(F)c1 CC1=C(C(=O)N2CCC(CNC(=O)CN(c3cnccn3)C)C2(C)C)CCO1 N1(c2cc(C(=O)OC)cc(OCC)n2)CCC2CNCC2C1 c1(COC)cc(C(=O)NCC(C)(CO)NC(=O)CNS(N)(=O)=O)c(C)o1 N1(C(C2(CC)CCCC2)=O)CC(N(C(=O)Cc2n[nH]cc2Br)C)C(O)C1 C1(CC=C)(C(=O)N(CC(=O)OC)C)CCN(C(=O)C(COC)N(C)C)C1 c1(CC)nn(C)c(C(N2CCC2CNC(=O)CC2CCC3(CCC3)O2)=O)c1Cl N1(C(C(=O)NCCOCC)C(C2CC2)OC)CCC2OCCCC2C1 N1(C(C(c2cncnc2)C)=O)CCC2(NC(=O)Cc3ccc(O)nc3)CCCC12 Cc1ccc(Cl)cc1NC(=O)C(C1CCN(C(C2C(C)(C)C2(F)F)=O)C1)F C1(NC(CC(C)CF)=O)CCC2(CC1)CC2NC(=O)CCN1CCC(O)CC1 c1(C(=O)NC(CNC(c2nnc(C)s2)=O)CO)ccc(=O)n2c1CCCCC2 N1(C(CC2C(NC(c3cc4n(n3)CCO4)=O)CC2O)=O)CC(=O)N2CCCC2C1 c1(N2CCC(NC(c3cc(SC)c(F)cc3)=O)C(O)C2)ncc2c(n1)COC2 c1(C(N2C(C)CN(C(c3cc(C(N)=O)c[nH]3)=O)CC2)=O)cnn2cccnc12 c1(C(N(CCCCNC(C(C)OCCC=C)=O)C)=O)c(Cl)cc(C#N)cc1Cl Cc1oc(-c2ccccc2)cc1NC(=O)NCC(C1CCCO1)N(C)C CCS(=O)(=O)CC(=O)NC1CCCC1(C)CN(C)C(c1ncnc(C)c1C)=O C(=O)(C(C)CS(C)(=O)=O)N1CC2(N(C(CCCCCOC)=O)CC2)C1 C1(C(=O)NCCN(C(=O)CC2CCCC(C#N)C2)CCC)CC2CCC1C21CC1 Cc1cc(C2CC2)ccc1C(N1CCC(C)(CNC(c2cnncc2O)=O)C1)=O N1(C(CN(C(=O)OCC)C)=O)C2CC=C(C(=O)N(c3cccnc3)C)C1CC2 C1(CN(C(c2c(CC)occ2)=O)C)C2CN(C(=O)Cc3csc(C)n3)CC12 C12(C(=O)Nc3cc(SC)n[nH]3)CC1CN(C(c1ncoc1C)=O)C2 Cc1c(Cl)ccc2cc(C(N3CCN(C(=O)CC4(O)CC4)C(C)C3)=O)cnc12 C1(CNC(C2C(CNC(C3(OCC)CC3)=O)CCO2)=O)CC(O)C(O)C1 C(CCC(=O)NC(C)CNC(=O)C(C)(C)C1CC1)NC(=O)OC CC1CN2CCN1CC2C(=O)NC1CCCCC1CNC(C12CCCC1C2)=O C1(C(=O)NOCC(O)CO)CC2CCC1CC2(F)F N1(C(C(C2CC(C)(C)C2)OC)=O)CCCN(C(c2cnsc2)=O)CC1 c1(C(=O)NCC2(OC)CN(C(C3CCC(F)C3)=O)C2)cnn2c1CCC2 C1(C(N2C(CCC)COCC2)=O)CC(C)(C)CCN1C(C1CC(=O)CCO1)=O c1(C(=O)NC(C)C(F)(F)F)ccnc(CNC(C2CCCC(F)C2)=O)c1 c1(C(=O)NC2(C3CCCN3C(=O)CCn3cccc3)CC2)cc2n(n1)CC(F)C2 N1(C(C(C2CCC2)OC)=O)CCN(C(=O)CCc2conc2C)CCC1C c1(C(N2CC(NC(C(C=C)c3ccccc3)=O)C2)=O)c(C)cc(C)oc1=O Cc1cccc2ccc(C(=O)NC3CCC(NC(=O)C(C)O)C3)nc12 Cc1cccc(N)c1C(=O)NC1CCCC(NC(=O)C=CBr)CC1 CCCCC(CCC)NC(=O)C(=O)Nc1cccc(COCCC)c1 C1(CNC(C(CSC)(C)C)=O)CN(C(=O)CC(F)(F)F)CCC1C c1(NC(C2CC3(CC3)CN2C(C2CC=CCC2)=O)=O)cc(Br)cc2[nH]ncc12 Cc1cnc(C(=O)NCCC2CN(C(C3C4CCCC34)=O)CCCO2)cc1Cl c1(OC)ccc(C=CC(N2CCC(NC(c3ccc(SC)o3)=O)C2)=O)c(C)c1 c12ccc(cc1)c(=O)n2CCCNC(C)=O.c1(N)cncc(C(F)(F)F)n1.CO C(=O)(C(C(F)(F)F)C(F)(F)F)N1C2C(CNC(C(C(C)C)O)=O)CC(CC2)C1 c1(C(=O)NCC2CN(C(CCC(C)C)=O)C(C)(C)C2)cnc2ncnn2c1O N1(C(Cc2c(C)cccc2C)=O)CCC2CN(C(c3ccnnc3S)=O)C2C1 N1(C(C(CC=C)C)=O)CCN(C(c2cc(C)c(C)o2)=O)C(C2CC2)C1 C1(CNC(C2(OC)CCC2)=O)CCC(C)(C)CN1C(c1ccncc1)=O c1(CC)ncc2c(n1)CCC(C(N1C(C(=O)O)CCC3OCCC13)=O)C2 C1(NC(c2coc(CO)c2)=O)CCCCCN(C(=O)C(F)(F)C2CCOCC2)C1 Cc1cc(C(=O)O)cc(N2CCCC(C(N3CC(c4ccccc4)C3)=O)C2)n1 C=CCC(CC)C(=O)NCCOC(C)(C)CNC(=O)C(C1CCC(C)(C)CC1)C C12(C(N3CC4CCN(C(Cc5c(C)nc[nH]5)=O)CC43)=O)CCC(C#N)(CC1)CC2 CC(C)C(CNS(=O)(=O)N)C1CC1.C(CCCCn1cncn1)N(C1CCCC1)CC c1(C(N(CCNC(C(C2CCC(=O)N2)C)=O)C)=O)cc(=O)n(C)o1 c1(CN(C(Cc2c(C)cco2)=O)C)cccc(CNC(c2occ(C)c2C)=O)c1 C(=O)(CC(O)C(C)C)NC1C2CCN(C(CCc3cc(C)[nH]n3)=O)C21 C=CC(CCC)CC(=O)NCC1CCC1NC(c1cc(C#N)c[nH]1)=O C(=O)(C(F)(F)C1=CCOCC1)NCC(C)N(C(=O)CC1CCC(=O)N1C)CC N1(C(c2c(C)nc(C3CC3)s2)=O)CCN(C(=O)C2=CCCC2)C2CS(=O)(=O)CC12 c1(SC2(CNC(C3(N(C)Cc4c[nH]c(=N)s4)CC3)=O)CC2)ccc(Br)cc1 C12(NC(C3CCCN(CC)C3)=O)CC(CNC(=O)C(N)=O)(C1)OC2(C)C c1(C(N)=O)ccc(NC(=O)C(c2ccccc2)NC(=O)COC)cc1C(=O)O N1(C(C=CC)=O)CC(OC)CC1(C)CNC(=O)CCSc1n[nH]c(C)n1 C1(C(=O)NCC(CC)NC(c2cc(C)n(-c3ccc(C)cc3)n2)=O)CCCN(C)C1 c1(C(C(=O)NCCCF)N(CCCOC)C)sc(C(=O)OC)cc1C Cc1cccc(OCCC(=O)N(CCNC(C2C3CNC(=O)C23)=O)C2CC2)c1C c1(CC(=O)N(CCC(=O)NCC(C)NC(C=CC)=O)C)ccncc1 C=CC(CC)CC(=O)NC1CN(C(C2CCCC2F)=O)C(C)(C)C1 Cc1cc(CC(=O)NC(C)CC(C)NC(c2cnsn2)=O)ccc1CO CCCCC(C)C(=O)NCc1cccc(CN(C(=O)C=C(C)C(F)F)C)c1 N1(C(C(C)N(C)C)=O)CC(C(N)=O)(CNC(C2CC2(C)Br)=O)C1 CCC(C)(C)C(C)NC(=O)C(C)(C1CCC1)NC(=O)Cn1ccnc1 c1(C(=O)NCC2(CN(C(C(CSC)O)=O)C)CC2)cc2c(F)ccc(F)c2[nH]1 C(=O)(CC1=CCCCC1)NCCC(=C)CNC(=O)C(C1CCCC1)OC C12(CNC(C3C(CC)C3)=O)CCC(CC1)N2C(=O)CC(C)C(=O)OC N1(C(c2c(Cl)cc(C)s2)=O)CCC(C)C(NC(C2CC3CCC2CC3)=O)C1 C1(CC(=O)Nc2cccc(O)c2F)CC2OCCC2O1 S(=O)(=O)(c1ccc(NCc2csc(CO)n2)c(F)c1)NCC1C(C)OCC1 N1(C(C(CC)NC(=O)CCCCN(C)C(C)C)=O)C(C)CCCC1C C#CCCCCCCC(=O)N1CCCC(C)(NC(=O)COC(C)=O)CC1 C=CCC(F)(F)C(=O)N1CC(CCNC(=O)C(C)NC(C2CCCC2)=O)C1 N1(C(C(C(C)C)OC)=O)CC2CCC(C1)C(NC(=O)C(N)=O)C2 C1(NC(c2ncc(OC)cn2)=O)CC2(C1)CC(CNc1nccnc1C#N)C2 CC(C)CCCCCC(=O)N1CCC(C)C1C(=O)NCCN1CCOCC1 C1(C)(CNC(CC2CC(OCC)C2)=O)CN(C(c2cnc(C)c(N)c2)=O)CCO1 C1(C(N(C2CCN(C)CC2)C)=O)CCC(O)CN1C(c1nnc(S)n1C)=O C=CC(C)(C)CC(=O)NC(C)CCN(C(=O)C(F)C1CCCC1)C O=C(CC1=CCCCC1)NCC1CCCC(NC(C2CN(CC(F)(F)F)C2)=O)C1 C1(CNC(c2cnn(-c3nccs3)c2)=O)CC(F)CN1C(=O)CO CN1CCC(C(N2CCCC(O)C2)=O)(NC(c2sccc2CO)=O)C1 C1(c2nnnn2Cc2ccco2)(NCc2ccc(CC)cc2)COC2(COC2)C1 N1(C(C(COC)OC)=O)CC=CC(NC(=O)Cc2csc(-c3ccccc3)n2)C1 N1(Cc2ccc(Cl)cc2)CCOC2(CCCC2)C1.c12ccccc1NCC2 C1(CC)CCCCN1C(=O)COCCNC(c1cn(C(C)C)cc1C)=O c1(C2CCCN(C(C3CCNC(C(F)(F)F)C3)=O)C2)c[nH]c2ccccc12 Cc1cncc2nc(CC(=O)NCC3(F)CCCN(C(=O)C(C)C(F)F)C3)cn12 CC1(C)CCC1C(=O)NCC(C1CCCC1)NC(c1cnc(C(N)=O)s1)=O CN=c1ccc(Br)c(C(=O)NC(C)CN(C(=O)CCC(C)C)C(C)C)[nH]1 c1(C(N)=O)c(NC(N2CCC(CC3CCCO3)C2)=O)cccc1N1CCCC1 C(=O)(CC(C(=O)N1CCC(C2CCCN2C(c2ccns2)=O)CC1)N(C)C)OC N1(C(c2c(C)cc(C)[nH]2)=O)CCN(C(C2CC3(CSC3)C2)=O)CC1CS(C)(=O)=O C1(OC)CC(NC(=O)COC(C)C)CN(C(C2CC3CCC(C2)C3)C)C1 C=CCC(CC)C(=O)N1CCN(C(=O)COc2ccon2)C(C2CCC2)C1 Cc1ccc2c(C)c(C(=O)NCC34CC3CN(C(=O)CC(C)CF)C4)[nH]c2c1 c1(-c2cncc(C(=O)NCC3(CC)CCC(=O)N3)c2)ccc2c(c1)oc(=O)n2C C1(C(N2CC(CNC(=O)Cc3ccno3)C2)=O)CC12C(=O)Nc1ccccc12 C(=O)(C(CO)C(F)(F)F)NCCC(=O)NCc1nccc(OC)n1 C(=O)(CC(C1CC1)NC(C1(CC)CCOC1)=O)NCC(=C)CC C(=O)(CCCCCNC(C)=O)NCCN(C(C1(C(=O)OC)CC1C)=O)C1CC1 C1(NC(C=C(C)C(F)F)=O)CCN(C)C12CCCN(C(C1CCC(C)C1)=O)C2 C(CC(C)(C)C(=O)N1CCCOC(CNC(C2NC(=O)OC2C)=O)C1)OC c1(CNC(NC(CC=C)C)=NC)cc(OCC2CCC2)cc(F)c1 c1(-n2cc(C(=O)NCC3C(OC)CCC3)nn2)ccc(Cl)cc1 C(C1=CCN(C(C2(C)CC2Br)=O)CC1)NC(C(CC)Oc1ccccc1)=O C(CCCC(=O)N1CCC1C(C)O)N(C(C(C)(C)OC(C)=O)=O)C C1(C(N(C(C)C)CCN(C)C(C2CCC(F)C2)=O)=O)CCn2ncnc2C1 C1(C(=O)NCCCCCNC(c2cnc(C(C)(C)C)[nH]2)=O)(COC)CC=CCC1 N1(C(C(=O)NCCOC)=O)CCC12CN(C(c1ccc(C(C)=O)nn1)=O)C2 C1(NC(Cn2c(C)cnc2)=O)CCCC(NC(c2c(Br)cnn2C)=O)C1 C1(C#C)(C(=O)NC2(CC#C)CC2)CN(C(C2CC2C2CCC2)=O)C1 c1(C(N2C(CC)C(NC(c3csc(C)c3)=O)CC2)=O)csc2ccccc12 C1(C2CCOCC2)(C(N(C)CCN(C(=O)C(C)(C)C(N)=O)C)=O)CCOCC1 N1(C2CN(C(C3C(CCC)C3)=O)C2)CC(NC(=O)CCn2ccc(C)n2)CC1=O C1(CC)CCCN(C(=O)C(C)NC(N)=O)C1C(=O)NC1(C(=O)N(C)C)CC1 Cc1cccc(C(=O)NC(C2CN(C(c3cc(Cl)ccn3)=O)C2)C)c1[N+](=O)[O-] C1(NC(C(COC)(C)C)=O)CC12CCN(C(C1CC(CF)C1)=O)CC2 N1(C(=O)Oc2ccccc2)CCS(=O)(=O)N2CCOCC12 CC1(C(N2CC=CC(NC(c3ccncc3F)=O)C2)=O)CCC2(CC1)OCCO2 C12(C(=O)NCC3CCN(C(c4cc(C)ncn4)=O)C3)CC(CO)(C1)OC21CCC1 c1(C(=O)Nc2nc(C)c(C(=O)Nc3cc(Cl)ccn3)s2)ccc2cc[nH]c2c1 CCCCCCCCCC(C(=O)NCC)N1CCC1(C)c1ccccc1 C1(CC(=O)N(CCOCC=C)C)COCCN1C(=O)CC1(O)CCCOC1 C1(O)(CCC)CCN(C(c2c(CNC(=O)C(C)NC(C)=O)nnn2C)=O)CC1 N1(CC)N=C(C(=O)NCC(O)CCNC(=O)CC2CSCCS2)CCC1=O Cc1nc(N(c2cnn(C3CNC3)c2)C(c2ccc(Cl)c(Br)c2)=O)ncc1F C1(N(C)C)CCN(C(=NCC2CCCN(C3CCCC3)C2)NC2CC2)C1 c1(C(N2CCC(NC(C(C)SCCCC)=O)C2)=O)cccc(C)c1[N+](=O)[O-] N1(C(C2(COC)CC2)=O)CC2CCC1C(CNC(=O)C(O)CC(C)C)C2 CC1CCN(C(=O)C(C)N(C(C)CNC(=O)CCOC2CC2)C)CC1 c1(SC)cc(C(=O)NCC2CN(C(=O)CCC3CC3(C)C)CCO2)c(C)o1 N=c1nnn(CC(=O)NCC(=C2CN(C(c3cn(CC(F)(F)F)nn3)=O)C2)F)[nH]1 CC12CN(C(c3ccc(OC(F)F)cc3F)=O)CC1CN(C(C1CNC(=O)C1)=O)C2 C1(CNC(C(C=C)O)=O)CN(C(C2CSC2)=O)CCN1C c1(C(=O)NC2CC(N(C(CC(c3ccc(F)cc3)C)=O)C)C2)c[nH]ccc1=O CCC(CC(=O)NCC(c1ccccc1F)NC(=O)C(C)(C)COC)CC(C)C c1(C(=O)OC)ccc(O)nc1NCc1nc(C)cs1.C1(CC=O)CCCCCC1 N1(C(C23C(CN(C(C(C)CO)=O)C2)C3)=O)C2CCC1CC(CO)C2 C(c1c(C)cc(C)cc1C)=CC(=O)NC1C(NC(C2(C=C)CC2)=O)CS(=O)(=O)C1 N#Cc1cc(N(CCNC(c2csc(Cl)c2Cl)=O)C2CC2)nc(C2CC2)n1 Cc1ccc(C(C)C(=O)NC(C)(C)CNC(c2sccc2F)=O)s1 Nc1ccc([N+](=O)[O-])cc1C(N1CCC(NC(=O)CC2CCOC2)C1)=O C1(CNC(N(CCO)CC)=O)CCCN(c2nccn2C)C1 CC(C)CC(CC(C)C)C(=O)NCCC1(NC(=O)CN2CC(C)(C)C2)CCC1 Cc1ccnc(CNC(C2CC3CC3N2C(=O)CC2CCOC2)=O)n1 C12CCCC(C1)CC(=O)N1CC(n3cc2nn3)C1.C1(OC)(OC)CC(CO)C1 c1(CCNc2nc(C)nc(N3C(C)CC4CNCC34)c2)ccc2ncccc2c1 C(CN=c1[nH]cnc2ccc([N+](=O)[O-])cc12)NC(=O)CC(C1CCC1)C1CCC1 c1(C(N2C(C)CCC(NC(c3c(C)coc3)=O)C2)=O)cc(C)cc2c1CCC2 Cn1ncc(C(=O)NC2CC(F)(CNC(c3ccc(CO)cn3)=O)C2)c1F C(=O)(CS(=O)(=O)C1CC1)N1C(C(C)C)C(NC(c2cc(F)cnc2O)=O)CC1 c1(SCC(=O)NC(C(C)(C)NC(CC2(NC(C)=O)CC2)=O)C)ccccc1F N1(C(C)=O)CC(F)(F)CC1C(=O)N(C(c1ccccc1C)=O)Cc1ccccc1 C(=O)(C1CCCc2nn(C)cc21)NCC1(O)CC(NC(c2n(CC)ccc2)=O)C1 C#Cc1ccc(F)cc1CNC(=O)C(=O)NCC(C)Sc1ccccc1 C(CCC(O)CO)NC(c1ccc(CNC(C2CC(=C)C2)=O)s1)=O n1(CC(=O)NCC(CCNC(C(C)CSC(F)(F)F)=O)O)sc(=O)c2ccccc12 c1(C(N(CCCNC(c2c[nH]cc2-c2cnn(C)c2)=O)C)=O)ccc(N)cn1 Cc1ncc2n1CC(C(=O)NC(C)CC1(O)CCC1)CC2 N1(C(C2(C(C)(F)F)CC2)=O)CCCCC(NC(c2ccc(CO)cn2)=O)C1 c1(C(=O)NCCN(C(c2cccc(OC)n2)=O)CC)ccc2c(c1N)CCCC2 N1(C(COCCC=C)=O)CCN(C(=O)C(CCC)NC(C)=O)C(C)C1 C1(CCC)CCCCC1N(C1(O)CN(C(=O)CCCn2cncn2)C1)C(=O)C1CC1 N1(C(c2n[nH]c(C)n2)C(=O)NCC=C)CC2C(CN=[N+]=[N-])C2C1 c1(C(=O)NCCNC(=O)Cc2cn[nH]c2)c(F)cccc1F c1(C(N2CC(CC(=O)NCCOc3ccccn3)C2)=O)ccc(C(F)F)cc1F c1(C(N(C)CCC2CCN(C(c3ncc(Cl)cn3)=O)CC2)=O)cnc(O)nc1O Cc1cc(Br)c2nc(CN3CC(c4ccccc4)C(F)C3)ccc2c1 C(CNC(=O)Cc1cncc(C)c1)(CC(C)C)NC(C1CCC(OC)C1)=O C1(NC(c2ccncc2F)=O)COC2(CCN(C(=O)C3=CCOCC3)CC2)C1 c1(OCC)cc(-c2nc(CC(C)(C)C)nn2C2CCCC(C)C2)cc(Cl)c1OC N1(C(c2nc(CC)oc2)=O)CC(OC)CC1(C)CNC(c1cc(C)cc(C)c1)=O C1(CC)CCC(O)(C(=O)NC2CC(CNC(c3cnn(C(C)(C)C)c3Cl)=O)C2)C1 N1(CC(=O)NC(C(C)C)CCN(C)C(C2CC=CC2)=O)CCS(=O)(=O)CC1 C(=O)(CC(C)(O)CCC)NC1CCN(c2ccc(C(C)=O)cn2)C(C)C1 CCC(C)CCC(=O)NCC1(OC)CN(C(c2c[nH]nc2Cl)=O)C1 C1(NC(C2CSCC(=O)N2)=O)CC2CN(C(c3cc(Cl)c(Cl)[nH]3)=O)CC12 Cc1cc(C(=O)N(C2C3CN(C(c4nocc4Cl)=O)CC23)C)cn1C(C)C Cc1cc(Br)cnc1C(=O)N(C)CCN(C(=O)CC1OCCC1(C)C)C C1(CN(C)C(C2(NC(=O)CN3CCCC3)CCC2)=O)COC(C)(C)C1 CCCCC(C)C(=O)NC1(COC)CCN(C(=O)C(C2CCCCC2)O)CC1 C=C(C)C(C)(O)C(=O)NCC1CCN1C(C1(C(F)F)CCC1)=O C(=O)(C1Cc2ccc(F)cc21)NC(COCCNC(C(c1cn(C)nc1)O)=O)(C)C c1(OC)ccccc1C(=O)NCC(C(C)(C)C)NC(=O)CCc1cc(C)n(C)n1 c1(C(c2n(CCCCCC)nnn2)NC(C)C(C)CC)nc(C)c(C)o1 N1(C(C(CCOC)(C)C)=O)CCN(C(=O)COC2(C)CCC2)C2CCCCC12 C(=O)(CCN(C(=O)CN(C)C)CCOC)NC(C#C)C1CCC1 N1(C(c2cnc(OCC)nc2)=O)CCOCC(NC(=O)CC2CC(C)C2)C1 N1(C(Cn2cc(CNC(C3N(CCC)CCC3)=O)nn2)=O)CCS(=O)CC1C c1(C(=O)NCC(CNC(C(c2ccnn2C)C)=O)F)ccc(OC2CCC2)cc1 c1(C(=O)NCc2cn(C3CN(C(C=CC)=O)C3)nn2)ccc2cnc(C)n2c1 C12(NC(C(C)OC3CCCC3)=O)CCCC1N(C(c1cc(C#N)on1)=O)CC2 C(=O)(C1=CNS(=O)(=O)N=C1C)NC1CCN(C(C(CCCC)(C)F)=O)C1 c1(-n2cc(CNC(c3ccc(F)c(F)c3)C)nn2)cc(N)ccc1Cl C(=O)(C(O)CC(F)(F)F)NC1CC(CNC(c2nsc3ccccc23)=O)C1 N1(C(C(C)(C)c2ccno2)=O)CCCC(CNC(=O)CSc2ccccc2O)C1 c1(CC)ccc(C(=O)NCCCCCNC(=O)Cc2cnccn2)c(F)c1 c1(C(=O)NCC(CNC(CCC(C)OC)=O)OC)ccnc(C)c1C N1(C(=O)OC(C)(C)C)CCOC2(CCCN(C(=O)NCc3cc(F)n[nH]3)C2)C1 N1(C(C2(C)CC2Br)=O)CCOC2(CCCN(C(=O)Cc3cnns3)C2)C1 CCC(C(=O)NCC1CCCN1C(C1CCC=CCCC1)=O)C(C)C N1(C(CCCCC(N)=O)=O)CCC(C2(NC(C3(F)CCOCC3)=O)CC2)CC1 Cc1ccc(O)c(C(=O)NC(C)(C)C(C)NC(=O)CCC2CC(C)C2)c1 c1(C(=O)NC2CC(NC(c3c(OC)c(Cl)ccc3)=O)C2)cc2ncn(C)c2cn1 c1(C(N2C(C)(CNC(CN3CCC(C)CC3)=O)CCC2)=O)cnc(O)n(C)c1=O CCCC(O)CC(=O)N(C1CCCCN(C(c2ccc(O)c(CC)c2)=O)C1)C c1(CC(=O)NC(C(=O)NC(C(C)SC)C)(C)C2CCC2)ncccc1F C=C(C)CN=C(NC(c1cc(OC)ns1)C)N1CCC(C(=O)N(C)C)C1 c1(C(C(=O)NC2CCN(C(c3cnsc3)=O)CC2)(F)F)cc(Cl)ccc1F c1(C(=O)NCC(c2ccccc2)C)sccc1CNC(=O)Cc1ncnn1C c1(NC(CC)C(C)C)ccc(NC(N2CCC(O)CC2)=O)cc1F CCC(C)CCC(=O)N(C(C)(C(=O)NOCC=C(C)C)C1CC1)C c1(CC(=O)NCC2N(C(C3C(C)CCC3)=O)CCOC2)noc2ccccc12 C(=O)(C1CCC(C)(C)c2ccccc21)N(CCN(C(c1scc(C)c1C)=O)C)C C1(C#CC(=O)NCC2(C)CC(NC(=O)CNC(c3ccc(C)s3)=O)C2)(CC)CC1 C1(C(C2(O)CCOCC2)C)NC(=O)N(CCc2nccs2)C1=O c1(OCCC(=O)NCc2cc(OCC)c(O)cc2)cc(C)cc(C)c1C C(=O)(C(O)CC[S+](C)C)N1CCC(N(C(=O)CSC(C)(C)C)C)C1 Cc1cn2c(n1)CC(C(N1CCCC(NC(=O)CSC(F)F)C1C)=O)CC2 Cc1cc(OCCC#CCN=[N+]=[N-])cc(C)c1S(N)(=O)=O c1(NC(CC2(OC(C)C(=O)NC34CC(C)C3C4)CCCC2)=O)ccccc1Cl c1(C(c2n(CCCC)nnn2)NCc2cnn(CCF)c2)cnc(OC)c(F)c1 C1(n2c(COC)ncc2)CCN(C2CNC(C)C2)CC1 C1(C(C)(C)O)(CNC(=O)CSc2cn[nH]c2)CN(C(C2(C)CCOC2)=O)C1 N1(C(Cn2cc[n+](C)c2)=O)CCN(C2CCN(C(=O)COCC(F)F)CC2)CC1 S(=O)(=O)(c1cccc(N2CCCC(CCO)C2)n1)NCCC(=O)NCC C1(c2cn(C)nc2)COCCN1C(=O)Cn1nc(C(=O)O)cc1C C1(C)(CNC(CN(C(C)C)C)=O)CCN(C(c2ccc(Br)cc2Cl)=O)CC1 c1(C(=O)NCC23N(C(CCCC)=O)CCC2CCC3)cc2ccccc2c(O)n1 C(N=c1[nH]c(=NCCCCS(C)(=O)=O)[nH]c2c1SCC2)C1(CC)CCC(=O)N1 C(=O)(N=c1ccn(Cc2ccc(C#N)cc2)[nH]1)Nc1cccc(CC(=O)OC)c1 C1(CCCNC(C(C2CCC2)OC)=O)CN(C(=O)CC2CCCC(C)O2)CCO1 CCCC(C(=O)NC(c1cccc(C)n1)C)NC(c1ccoc1)=O Cc1cc(C(N2CCC(C)(NC(=O)Cn3cnnc3)C2)=O)ncc1Br C1(C(=O)NC(CC)CNC(c2ccnn2CC2CCC2)=O)CC2C=CC1C21CC1 C(CCCC(=O)NCCC1CC(NC(c2cccc(-n3ccnn3)c2)=O)C1)SC c1(C(=O)NC)cc(-c2nc(C(N3CCC(SC)CC3)=O)cs2)ccc1F N1(C(C(C=C)OC)=O)CC2(C1)CN(C(c1cnn(C)c1SC)=O)CCO2 c1(OC)cccc(C(=O)NC2(C3CN(C(C4NC(=O)CC4C)=O)C3)CC2)c1O C(Cc1ccccc1)(C(=O)N(C1CCCNC1)c1ccccc1)NC(C)=O CCCCCC(C)CC(=O)NC1CC(F)(CNC(c2cnc(C(C)(C)C)o2)=O)C1 N#Cc1cc(S(=O)(=O)N2CCC(F)(C(=O)O)C2)ccc1C(=O)O N1(C(COC(CNC(c2ncc(NCC)nc2)=O)(C)C)=O)CC2(CNC(=O)C2)C1 Cc1cc(C)c(C(=O)NC2CCN(C(C3CC4C=CC3O4)=O)C2C)c(S)n1 c1(OC)cc(C(F)(F)C(=O)NC2CC(CCNC(C3CC3C#N)=O)C2)ccc1C C1(CNC(CCc2ccc(SC)s2)=O)CCCCN1C(=O)C(C)CC1CCCC1 C(C(C)(CC(C)C)NC(c1cnc2n1CCC2)=O)NC(c1c(C)sc(Cl)n1)=O Cc1c(C(=O)NC(Cn2cccn2)C(=O)NCc2scnc2CO)nnn1C C(=O)(CCC(=O)N1CCCC(N(C(=O)CCC(F)F)C)C1)Nc1nnc(CC)s1 c1(C(C)C)n[nH]c2ccnc(C(=O)NCC3CN(C(C4C(C)C4C)=O)CCO3)c12 C(C)(CC(=O)N1CC2(C1)CN(C(=O)C(N)=O)C2)(C(F)F)N(C)C C(N=c1[nH]c2ccc(C)nc2s1)CC1N(C(C2(CC)CCOCC2)=O)C2C(C1)C2 c1(C(=O)NCCC(C)NC(=O)Cc2nnc(O)s2)cc(Cl)cc(Cl)c1 C1(C(=O)OC)CCC(C(N2CCCC2CCNC(=O)C(C)SC(F)(F)F)=O)CC1 N1(C(C(CC)OCC)=O)CC2CCC(C1)C2NC(c1ncn(C)n1)=O N1(C(C2CCC(C)(C)CC2)=O)CC2COCCC2(NC(C2COC2)=O)C1 C1(NC(CNC(CCC(=O)OCCC(C)C)=O)=O)CCC(C(F)(F)F)N(C)C1 N#CC(C(=O)N1CCCC1CNC(=O)C(c1ccccc1)O)c1ccccc1 N1(CC(C)COc2ccccc2)C(=O)CN(CCc2cc(Br)cs2)C1=O C1(c2n(CC=C)nnn2)(NCc2n[nH]c(C3CC3)n2)CC2CCCCC12 N1(C(C2CCN(C(c3c(CC)n[nH]c3)=O)C2)=O)CCC2(CCOC2=O)C1 N1(S(=O)(=O)c2cc(C(F)(F)F)cs2)CCc2cc(F)ccc2C1 C(=O)(CCC(C)NC(c1cnn(C)c1N)=O)NC(C)C(=O)NCCF c1(C(=O)NCC23CCC2CCN3C(c2cc[nH]c2)=O)[nH]nc2ncc(Br)cc12 C(c1ccccc1)=C(C(c1n(CCOCC)nnn1)NC1CCN(C)C1=O)C C1(c2ccc(NC(CS(CC)(=O)=O)=O)cc2)C2Sc3cc(C)ccc3C12CO c1(C(N(CCNC(c2cnn(CCOC)c2)=O)CC)=O)cc(Cl)sc1Cl C(=O)(C1CC(=O)c2cccc(OC)c21)NCC(C)NC(CCC=C)=O c1(C(=O)NCC2(NC(C3CC(=O)OC3)=O)CCOC2)ccc2nc[nH]c2c1F c1(C(N(C(C)C)CCNC(=O)CCc2cnco2)=O)ccc2ncsc2c1 C(=O)(C1=CCCOC1)NCC(c1ccccc1)NC(C12C(CN(C(C)=O)C1)C2)=O C1(C(N2CCN(C(CC(C)C)=O)C(C3CCC3)C2)=O)CN(S(=O)(=O)N(C)C)C1 Cc1c(C(=O)NCC2CCC(NC(c3occc3Br)=O)C2)c(Cl)nn1C C(=O)(CCCC(=O)N(C)C)NCC=CCNC(CCC=CC(C)C)=O S(=O)(=O)(c1cc(Br)c(F)cc1F)NC1CCCN(Cc2ccc(F)c(C)c2Cl)C1 c1(CC(=O)NC(CC=C)CNC(=O)C2CC2)cc(Br)ccc1C N1(C(C2(O)CCN(C(C(C)c3cccs3)=O)C2)=O)Cc2c(O)n[nH]c2C(F)(F)C1 c1(OCC(=O)NCC(C)(C)CNC(c2csc(O)n2)=O)ccc(F)nc1 c1(CC(=O)NCC2CCCC(NC(=O)CSC(F)(F)F)C2)cccnc1Cl CC(C)CC(C(=O)N(C(C)C(=O)NCC1CNC(=O)CO1)C1CC1)C(N)=O CC(C)(C(=O)NCCCC1(NC(=O)CC2(C)CC2(F)Cl)CC1)c1cccs1 C1(NC(CCCC)=O)CCCC(C(=O)N(C2CCCOC2)CC)C1 c1(C(N2C(CC(=O)NC(C)CC(N)=O)CC(F)C2)=O)c[nH]c2ncccc12 c1(NC(=O)CC2CCN(C(c3ccc(O)cc3)=O)C2)ncnc2[nH]c(Br)nc12 CCN=c1[nH]cc(C(=O)NC2CCC(CNC(=O)CC3CCCCC3C)CC2)s1 c1(CCC(=O)NC2C(NC(Cc3nc(C(=O)OC)sc3)=O)C2)ccc(OC)nc1 c1(CC(=O)NCC(CC)NC(=O)CC2CC(O)C2(C)C)cccc(F)c1F C(=O)(C(O)CC(N)=O)N(CCCC(N1C(COC)C=CCC1)=O)C c1(SCC)ccnc(C(=O)NS(=O)(=O)CCCn2cnnn2)c1 c1(C(=O)NC2CC(NC(C3C4CNC(=O)C34)=O)C2)cc(Br)ccc1F C=CC1(CNC(=O)C(CC)NC(=O)CC2CCC(=O)N2C)CCOCC1 c1(COC(C(CSC)C)=O)ccc(O)c(C)c1C C(=O)(CCP(C)(C)=O)NC(C1CCN(C(=O)C(C)NC(=O)C(C)(C)C)CC1)C c1(OC)ccc2c(c1)C(NC(=O)NC13CCCCC1NC(=O)C3)C(=O)N2 C1(CNC(C2(NC(CCCOC(C)=O)=O)CCOCC2)=O)CC1C1CCCC1 c1(C(=O)NC2C=CC(CNC(c3csnn3)=O)C2)cc(Cl)cnn1 c1(CC)c[nH]nc1C(N1CC(O)(C(C)(C)CNC(C2CCOC2)=O)C1)=O c1(C(N2CC3CC2CN3C(c2cnc(Cl)c(F)c2)=O)=O)cc2ncccn2n1 CC(C(=O)N(C)Cc1ccc(CNC(c2cc(Cl)no2)=O)cc1)C(C)(C)C c1(CC)nn(C)c(OC)c1C(c1nnnn1C1COC1)NCC1CCSC1 Cc1cn2cc(C(N3CCCC(CO)(NC(C4CCSC4)=O)C3)=O)cc(C)c2n1 c1(C(N2CCC(NC(CCC=C)=O)CC2C2CC2)=O)ccnc2c1cnn2C Cc1cc(C(N2CCC(O)(CNC(c3onc(C)c3C)=O)CC2)=O)c(Cl)cc1F C(N=c1cc[nH]cc1S(=O)(=O)NCC1CC12CCOC2)c1c(OC)cccc1F c1(C2C(C)(C(=O)NCCCOCCNC(=O)CCNC(N)=O)C2)ccccc1 Cc1cc(CCNC(c2ccnc(Br)c2)C)cc(C)c1 N1(C(C2(C)CC(=C)C2)=O)CCC2CN(C(C3CC(C(=O)OC(C)(C)C)C3)=O)CC12 N1(C(C2CCC(C)N2c2ncccn2)=O)CCC(F)(F)C(CNC(=O)NCCCl)C1 c1(OC)nc(C(N2CCC(NC(c3ccc(C)c(C)c3)=O)CC2C)=O)cc(O)n1 c1(C(C)NCCc2cc(C3CC3)nn2C)cc(Br)ccc1F C(=O)(C(C)CC(C)C)N1CCC(N(C(=O)C=Cc2cnc(OC)nc2)CC)C1 CCCCC(C)(F)C(=O)NCC1CCCCN(C(c2cn(C)nc2C)=O)C1 N1(C(CCC(=O)N(C)C)=O)CCCCC(C(=O)NCc2ccc(CO)cc2)C1 N1(C(C(COCC)C)=O)CC(C)(C)CCC1CNC(c1cscc1C(F)(F)F)=O C(CS(=O)(=O)CC(=O)N(C)CC1CN(C(=O)Cc2nnc3n2CCOC3)C1)OC N1(C(c2cc(F)c[nH]2)=O)CC2(CCN(C(c3ccccc3C3CC3)=O)CC2)C1 C=C1CCC(C(=O)NC2CC3(C2)CC3C(=O)NCCN(C(C)C)C2CC2)CC1 CC1CC(CNCCCN2CCCN(C(=O)OC(C)(C)C)CC2)CC(C)C1 c1(CC(=O)NCCCCCCNC(C2N(C)CCC2)=O)ccc2cccnc2c1 c1(C(=O)NCC(CNC(=O)CN2CCC(C)C2)OC)ccc2nccnc2n1 CC1=C(F)CN(C(=O)C(O)CNC(=O)Cc2cc(C)n(C)n2)CC1 c1(C(N(CCCNC(C(C)SCC)=O)C(C)C)=O)cn(C)c(=O)cc1OC CCCCC(O)C(C)C(=O)NCC(CNC(c1cnc2cc[nH]c2c1)=O)CO N1(C(C(C2CN(C(C3(C#N)CCOC3)=O)C2)OC)=O)CCOC(C)(C)CC1 c1(CC(N2C(C(=O)NCC3CCCS3)CC(F)C2)=O)c[nH]c2ccc(Br)cc12 N1(C(c2ccc(C)nc2)=O)CC(O)CCC1C(N1CCC(CO)CC1)=O N1(C(C2CC(C(=O)OC)C2)=O)CC(CC(=O)NCCC2CCCN2C)CC1(C)C N1(C(C(c2ccc(C)s2)C)=O)CC(NC(C2CC2C)=O)CC(C)(C)C1 c1(C(=O)NC2CC(CNC(C3(C)CCCCO3)=O)C2)cc(N)ccc1Br c1(N(c2c(C)ccc(C)c2)C)nc2c(c(=NC(C)c3cnn(C)c3)[nH]1)CSC2 C1(NC(c2nc(CC)oc2)=O)CC(NC(=O)CN2CC(=O)NC2=O)CC1O N1(C(c2cnc(C)[nH]2)=O)CC(CNC(c2n[nH]c(C)c2Br)=O)C2(CCC2)C1 C1(NC(c2ccsc2C(F)F)=O)CC2CN(C(=O)C=Cc3ccc(Cl)cc3)CC12 N1(C(C2CCC(OC)C2)=O)CCC2(CC1)CC2NC(c1cnc(N(C)C)s1)=O CCC(COC)C(=O)NC(C)CCNCc1ccc(C(C)C)cc1.C1(=O)CN1 c1(CNC(C(c2ccsc2Br)N(C2CCC2)C)=O)cccc(Br)c1 c1(COC)nc(NCCNC(=O)OC(C)(C)C)cc(N2CCOC(C)CC2)n1 N1(C(C2(COC)CCCCO2)=O)CC2CC(NC(=O)CC3=CCCCC3)CC2C1 CCCCC(O)C(=O)N1CCCC1CC(=O)Nc1c(OC)ncnc1OC N1(C(C(C)(C(C)C)NC(C)=O)=O)C2CCCC1CN(C(c1cnccn1)=O)C2 c1(C2C(CNC(=O)CCn3ccnc3)C2)c(F)cccc1F C1(CNC(=O)Cn2cc(Cl)cn2)CCC12CCN(C(=O)Cc1ccno1)CC2 C1(C)(CNC(CCOCC(C)C)=O)CC(NC(C2CCC(O)C2)=O)C1 N1(C(=O)NC(CC(C)C(F)F)C)CCCCC(C)(F)C1 C1(C(C)NC(CCC#C)=O)CCN(C(C2(CO)CCCC2)=O)CC1 C1(NC(C2C(OC)CC2)=O)CC(CNC(c2c[nH]nc2OC)=O)C12CCC2 c1(C(N2CCC(NC(C(CC)=CC)=O)(CF)C2)=O)cc(OC)cc(C)n1 c1(C(N(C2CCN(C(C(COC)C)=O)C2)C)=O)cncc2[nH]ccc12 CC(C)(CC(F)(F)F)C(=O)NC1CCC1NC(=O)CCc1cccnc1Cl C(=O)(CC(C)C(C)(C)C)N1CCC(O)(CNC(c2c(CC)ccs2)=O)C1 C1(C(=O)NCCc2ncccn2)(NC(C(C)C2CC2)=O)CC1(C)C C(=O)(C1=NOC2COCC12)N(C1CN(C(=O)CCn2cccn2)CC1(C)C)C N1(C(C=CC=C)=O)CCCCCC1CNC(C1(C=C)CC1)=O C1(NC(CCNC(CC(C)C)=O)=O)CC(CNC(=O)CC=C(Cl)Cl)C12CCC2 c1(C(N2C(CNC(c3cnn4cc[nH]c34)=O)CCC2)=O)cccn(O)c1=O c1(C(N(C)Cc2nc(C(C)(C)C)cs2)=O)ccc2c(c1)NCCNC2=O N1(CCCC=C)CC2CCC1C1CN(C(c3cc(C)ccc3[N+](=O)[O-])=O)CC21 c1(-c2cnc(CNC(c3ncc(C#C)nc3)=O)nc2)ccc2c[nH]nc2c1 C1(O)(CNC(C2(C)CC2(Cl)Cl)=O)CCCN(C(=O)C(F)(F)C(F)F)C1 CCC(CC(C)C)C(=O)NCCN(C(C1C(F)(F)C12CC2)=O)CC1CC1 N1(C(C(C)(C)OCC)=O)CCCC(C(C)C(=O)NC(c2cn(C)nn2)C)C1 C1(C(N2CCC(NC(C34CCC(F)(CC3)C4)=O)CC2)=O)CCCCC(F)(F)C1 c1(C(=O)NCCCN(C)C(c2ccc(Cl)cn2)=O)ccc(C(F)(F)F)c(N)c1 C(=O)(CC1COc2ccccc21)N1CCC(NC(C=CC(C)C)=O)C12CC2 c1(N(C)C(C23CC2COC3(C)C)=O)nccc(C(C)(C)C)n1 c1(C(=O)NC(C(C2CC2)OC)C)cc(CNC(C2(Cl)CC2)=O)on1 c1(CCC(=O)NCC2N(C(c3cnc(C)o3)=O)CC2)c(C)noc1C CC1=C(C(=O)N2CC(NC(c3cccc(CO)n3)=O)CC2(C)C)SCCO1 C1(CC(=O)NC(C(NS(=NC)(C)=O)=O)C2CN(C(C)=O)C2)CCCC12CC2 c1(C(C)C)nc(C(=O)N(C(C)C(=O)NC(c2nncs2)C)C)co1 c1(C(N2C(CNC(CCCCCOC)=O)CC(F)C2)=O)sc2ccccc2c1C CCCCC(CNC(=O)C(c1ccc(Cl)cc1)=O)NC(=O)CCc1cnn(C)c1 CC(C)C(C(=O)Nc1cncc(C(=O)NC(C2CCOC2)C)c1)c1ccccc1 CCCC(CC)CC(=O)NCC(CNC(c1ccc(CO)c(Cl)c1)=O)CO c1(C(N2CCC(NC(=O)C=CSCc3ccco3)(CO)C2)=O)c(F)ccc(F)c1Cl N1(C(CCCC(C)=O)=O)CCC(O)(C2(NC(c3cc(Br)no3)=O)CC2)CC1 C1(NC(C(C)OCC#C)=O)CC2CCC(C1)N2c1ncns1 C1(OC)CC(CNC(=O)C(C2CC2)N(C)C)N(C(C2CC3(CC3)CO2)=O)C1 CNS(=O)(=O)N1CCN(C(=O)C(Cc2ccco2)NC(=O)OC(C)(C)C)CC1 N1(C(C2N(CC)CC2)=O)CCCC(C2CC2NC(c2ccsc2)=O)C1 N1(C(C2C3(CC(NC(C(C)SC)=O)C3)C2)=O)CCCC(C)(C)C1 C1(CC(=O)NCC#CCC)CN(C(c2cc(F)ccc2O)=O)CC12CC2 c1(C(N(CC(CNC(CCOCC(C)C)=O)C)C)=O)sc(=N)[nH]c1C1CC1 c1(CCC(=O)NC2C(NC(C(C)NC(CC)(C)C)=O)C2)ccc(OC)c(O)c1 C1(NC(c2cc(SCC)ncc2)=O)CCCCN(C(C2(CO)CCCO2)=O)C1 C(=O)(C1CCc2nccn21)N1C(CCOC)CN(C(=O)CC2CCOCC2)CC1 NS(=O)(=O)c1cccc(-c2ccc(=NCC3CC3)[nH]c2)c1 Cc1ccc(SCCC(=O)NCC2CC2CNC(c2ccc(C3CC3)o2)=O)cc1 C1(C(N(C)CC2(CNC(c3cnco3)=O)CC2)=O)CCCCS1(=O)=O C12(C(=O)NCCC(=O)NCC#C)CC(CN(C(c3cn(C)cn3)=O)C1)C2 C1(n2cc(COC)nn2)CCC(NC(=O)Cc2cn(C)nn2)CC1 C1(CNC(C2N(C(C)C)CCC2)=O)CCCCN(C(=O)C(C)c2cccs2)C1 C1(C(=O)NC(C)(C)CCNC(c2ccnn2C2CCCCC2)=O)CCC12CCC2 N1(C(CCOc2ccc(OC)cc2)=O)CC2CC1CC2NC(=O)C(C)=C1CCC1 C(=O)(CCCCC#N)N(C(C)CNC(=O)CCNC(C1CCC1)=O)CC c1(C(N2CC(NC(c3ccc(OC)c(O)c3)=O)C(F)C2)=O)cc2ccccc2o1 Cc1ccc(C(CNC(c2ccccc2N2CCN(C)CC2)=O)N(C)C)c(C)n1 N1(C(c2ccc[n+]([O-])c2)=O)CC2(CCCN(C(c3ncncc3Br)=O)C2)C1 N1(C(Cc2ccc(C)s2)=O)CC=C(CC(=O)NCC2(O)CCC(C)C2)CC1 c1(N2CCC(C)(C(N3CCC(O)C(F)C3)=O)CC2)ccn2nccc2n1 N1(C(c2c(C)[nH]cc2)=O)CCC2(CC1)CC2C(=O)NCCC1CCOC1 c1(-c2n(CCC(N)=O)ccn2)cccc(S(=O)(=O)N2C(=O)CCC2=O)c1 c1(-c2nc(C(=O)NC(c3ccsc3)(C)C)sc2)c[nH]c2ncc(Br)cc12 C1(C(N2CCC(n3cc(-c4n(CC)ccn4)nn3)CC2)=O)Cc2nnc(C)n2C1 CC(C)(C)C(=O)C(=O)NCC1(CNC(C2(OC)CCCOC2)=O)CC1(F)F S(=O)(=O)(c1ccc2ccccc2c1)N(C1CCCNCC1)Cc1onc(CC)n1 C1(NC(CCC(=O)NCC(c2ccc(F)cc2)C)=O)C2Cc3ccc(Br)cc3C12 Cn1nc(-c2cccnc2)cc1C(=O)NC1CC1NC(c1ccon1)=O CC#CCC(C(=O)OC(C)(C)C)NC(=O)NCc1c(OCC)cccc1C C1(CCOC)CCCCN1C(c1c(C2CC2)cnn1C)C(=O)NC1CCCC1 c1(C(N2CC(NC(CN(C)CC)=O)C(CO)C2)=O)ccc(C)cc1O N1(C(Cc2cn(CC)nc2)=O)CCN(C(C2C3CCCC23)=O)C(CC2CC2)C1 C1(C)(C(N(CCOC)C)=O)CN(C(=O)CNC(c2ccc(F)cc2)=O)C(C)(C)C1 Cc1ccc2c(c1)CN(CC(C1CCC1)NC(=O)OC(C)(C)C)CC2 N=c1ccc(C=CC(=O)NCC(O)CNC(=O)COC2CCOC2)c[nH]1 c1(C(N(C(Cc2ccc(C(C)=O)cc2)=O)C2CC2)=O)cc2[nH]cnc2cc1F c1(C(N(C2CCN(C(c3ccoc3Cl)=O)C2)CCO)=O)cc2c(Cl)cccn2n1 C(c1c(Cl)cccc1Cl)=CC(=O)NCC(CNC(C(C)(Cl)Cl)=O)F C12(C(N3CC4CCN(C(c5ncn(C)c5)=O)CC43)=O)CCCC(=O)N1CCC2 c1(CNC2C(O)C(F)CCC2)c(F)ccc(Cl)c1Br CC(C)(C(=O)NCc1cc(C(=O)NC2CCN(C(N)=O)C2)n[nH]1)C(F)F Cc1nc(NCCc2nc(C3CCCO3)n[nH]2)cc(=NCC2(C)C=CCCC2)[nH]1 N1(C(C(CC)NC(N)=O)=O)CC(=O)CC1C(=O)NCC12CCC(CC1)O2 c1(C(N2C(CNC(C=C(COC)C)=O)CCC2)=O)sccc1C#N C1(NC(=O)CCF)CC2CC(C1)CN(C(=O)C(c1ccc(F)cc1Br)O)C2 C1(NC(=O)CN2C(=O)CCC2=O)CCCN(C(=O)C=CC2CCCCCC2)CC1 CC1=C(C(=O)N2C(C(=O)Nc3cc(C(C)C)ccc3C)CCC2C)CCO1 c1(C(N2CC(NC(c3cc(OC)c(C)cc3)=O)C(C)C2)=O)cccc([N+](=O)[O-])c1 C1(NC(COC2C(C)CCCC2)=O)CCSC12CN(C(=O)C(C)(C)C1CCC1)C2 c1(NC(C(C(C)NC(CCC=C)=O)C)=O)c(C)ccc(O)c1C C12CN(CC1(C)C)C2=O.c1(NC(C)=O)ccc(NC(c2cccn2C)=O)cn1 C1(c2n(CCC)nnn2)(NC2CCC(NC(C)=O)CC2)CCN(C(C)C)CC1 c1(C(C(=O)NC2C(NC(c3c(CCC)nns3)=O)CCC2)C)ccc(F)cc1F C#CC1(C(=O)NCCOCCC(=O)NC2CC(C)C2)CCCCC1 C1(C(=O)NC(c2cnn(C)c2)C)CC12CC(NC(c1ccncc1Cl)=O)C2 c1(NC(c2ncc(-c3cccc(C)n3)nc2)=O)ccnc2c1CCO2 C(CC(C)(C)C)(C(=O)N1CC(C)(C(N)=O)C1)NC(C(C(C)C)C1CCC1)=O C1(C(=O)OC)CC(C)(C)CCN1C(c1cc(-c2cc(OC)ccn2)oc1C)=O C1(NC(c2c(C)ncs2)=O)CCCC12CCN(C(c1cc3n(n1)CCCO3)=O)C2 C1(C(N(CCC(C(C)C)NC(C(C=C=C)C)=O)C)=O)CC2CC(C1)CC(F)(F)C2 Cc1n[nH]cc1CC(=O)NC(C)C(C)(C)NC(=O)C=CCOCc1ccccc1 C(=O)(C1=CCCC1)N1CCC(N(C(=O)CN(CC(=O)NC(C)C)C)CC)C1 CC(c1ccccc1F)=CC(=O)NC(Cc1ccccc1)CCC(=O)O CCC(C)(CCNC(=O)C(=CC1CCCCC1)F)NC(C1CC(C2CC2)C1)=O C(CC(C(=O)NCP(C)(C)=O)NC(=O)Cc1cnc(C)s1)=CC N1(C(C(=O)NC(C)C)=O)C(C)CC2CN(C(c3ccc4ncncc4c3)=O)CC12 C1(C(N2CCC(C(C)C(N3CCOC(C(C)(C)C)C3)=O)CC2)=O)CC2(CC2)CO1 C1(CC(=O)NCC2C=CCN2C(c2ccnnc2O)=O)(OC)CCCCC1 c1(NC(C2CCCN(Cc3ccc(CC(=O)OC)cc3)C2)=O)c(O)cccc1O N1(C(C=Cc2n(CC)ccn2)=O)CCCC(NC(C2(CC(C)C)CCC2)=O)C1C C1(CNC(C2CCS(=O)(=O)C2)=O)CC2(C1)CN(C(=O)Cc1cccnc1)C2 C1(C(N2CCC(CCC(=O)NCC3COC(=O)N3)C2)=O)(OCC)CCOCC1 O=C(C#Cc1ccc(Cl)cc1)NC1CCCN(C(c2cc(F)c(F)cc2I)=O)C1 CCCC(C)(O)C(=O)NC1(CN(C(=O)CCCOc2ccc(C)cc2)C)CC1.CCO Cc1cccn2ncc(C(=O)NCC(C3CC3)NC(=O)C(C)(O)CC(C)C)c12 c1(C(N2C(C)(CC)CC(N)C2)=O)c[nH]c2c(F)c(Cl)ccc2c1=O Cc1ncnc(C(N2CCC(C(C)(C)NC(c3c[nH]cc(F)c3=O)=O)C2)=O)c1C c1(NC(C)C(C2CCCCC2)NC(=O)CCC2CCCCCC2)ncc(I)cn1 c1(C(=O)NC2(CNC(=O)CC3(O)CCOC3)CCC2)sc(Cl)cc1Cl CCC(CC)CCC(=O)NCC(C(N1CCC(C(COC)C)CC1)=O)N(C)C c1(C(=O)OC)ccc(N2CCN(C)CC2)nc1C.c12nccnc1C(=O)N2 C(c1ncco1)=CC(N1CCC1CNC(=O)C(c1ccccn1)C1CCCC1)=O Cc1c(N)ccc(C(=O)NC2CS(=O)(=O)CC2NC(c2cocn2)=O)c1F C=CCC(C(=O)N1CC(N(C)C(C2(OC)CCOCC2)=O)C1)c1ccccc1 C1(C(N2C(C)(CNC(=O)Cc3csc(=N)[nH]3)CCC2)=O)CCCS(=O)(=O)C1 CCCCCCCCC(=O)N1CC2(C1)CN(C(C1CC(OC)C1)=O)C2 CC1CCC(NC(c2ccc[nH]2)=O)CN1C(c1cc(Cl)ncc1O)=O Cn1nc(Br)c2ncnc(N3CC=CC(NC(=O)CC4CC(O)C45CCC5)C3)c12 N1(C(C(CC#C)O)=O)CC(NC(c2[nH]c(=N)ccc2C)=O)C2(CC2)C1 c1(OC)cccc2cc(C(=O)NC(C)CC(C)NC(=O)C(C)(C)N3CCCC3)[nH]c12 C1(C(N2CCC(CC(C)NC(c3occ(C)c3)=O)CC2)=O)CCC(N=[N+]=[N-])CC1 c1(C(C(=O)NC2C(NC(C(CC)(C)C)=O)CCC2)(C)C)ccc(F)cc1F C1(NC(CCN(C)CC)=O)C(CNC(=O)Cc2ccccc2Cl)CCC12CCC2 c1(CC)cc(C(=O)Nc2cccc(NC(=O)CN3CCCCC3C)c2)oc1CC N1(C(C2(COC)N(C(C3C(=C)C3)=O)CC=C2)=O)CCC2(CCOCC2)C1 N1(C(C2N(C(C(C)C)=O)CCCC2)=O)CCN(C(=O)C#CC2CC2)CC(C)(F)C1 c1(C(=O)NC(C2CN(C(C3CCCCC(=O)C3)=O)CCO2)C)nc(Cl)ccc1Cl S(=O)(=O)(C1CN(C(C2(O)CC2)=O)C1)N1CCN(C(C2CCCC(C)C2)=O)CC1 c1(SC)ccc(C=CC(=O)NCC(C)N(C(=O)CCC2(C)CCC(=O)N2)C)s1 C1(C)(C(=O)Nc2cn(CC)nc2)CC12CCN(Cc1cnc3ncccn13)CC2 C12(C(=O)NCC3(O)CCN(C(CC(C)CF)=O)C3)CC3CC(CC(C3)O1)C2 Cc1cc(C)c(C(=O)NCC2CC(O)CN2C(c2cnn3c2OCC3)=O)cc1N C=CC(F)(F)C(=O)NCC(C1CCCC1)NC(=O)CC1(CC(=O)OC)CC1 C1(F)(CNC(C2(C)C(C)(C)C2)=O)CCN(C(c2n[nH]cc2C2CCC2)=O)C1 C1(O)(CNC(c2cn(C3COCC3F)nn2)=O)CCN(C(=O)Cc2cnsc2)C1 c1(C(=O)NC2C(C#N)CN(C(c3csnn3)=O)C2)ccc2[nH]nc(Br)c2c1 c1(N(C(C(C(C)C)n2cncn2)=O)CC(C)C)ccc(Cl)c(Cl)c1 C1(CC)(NC(=O)CN(c2ccccc2)C)CCCN(C(=O)Cc2ccc(C)o2)C1 CON=C(C(=O)NCCC(C)NC(=O)CC(C)(O)C1CC1)c1ccco1 CCC(C)(O)C(=O)N1CC(C(NCP(C)(=O)OCC)=O)C(C)C1 N1(C(C(CC)(C)CNC(c2cc(C)c(C)s2)=O)=O)CCCC2C(=O)NCC12 c1(CC(=O)NC23CC2CN(C(C2(CO)CC2)=O)C3)nsc2ccccc12 C(=O)(C#CC1CCOC1)NC1C(CCC)CN(C(c2cc(C)cnc2O)=O)C1 CCC(C)C(C(=O)NCCOC1CCCC1)N(C(=O)C1=CCCCC1)C c1(CCNC(C2CCC(F)(F)C2)=O)cccnc1O N1(C(C(CC)(C)C)=O)CCC2(NC(c3cn(CCCC#N)nn3)=O)CCCC12 C1(NC(CSNC(c2cnc(C)s2)=O)=O)(CO)CCN(C(=O)CC(O)C(C)C)CC1 N1(C(C2CC2(F)Cl)=O)CCC2(CC1)CC2c1cn(Cc2ccc(O)c(O)c2)nn1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(C1CCCC(NC(c2nnc(C)s2)=O)C1)C c1(C(N2CCN(C(CCOC)=O)CC2c2ccnn2C)=O)cc2c(s1)CCOC2 C1(C(=O)NC(CN(C(c2cnc(CC(C)C)[nH]2)=O)C)C)Cc2ccccc2S1 N1(C(c2cc(CC)[nH]n2)=O)CCC(NC(=O)C(C)CCC(C)(C)C)C2(CCC2)C1 C1(CNC(c2n(CC)cc(Cl)c2)=O)N(C(=O)C(F)=C2CCCC2)CCCC1(C)C N1(C(C(=O)Cc2ccc(F)cc2)=O)CC2(CC2)CC1CNC(=O)Cn1nccn1 C1(NC(C(C)SC)=O)COC2(CNC(=O)C(c3ccc(C)cc3)(F)F)CC1C2 c1(C(N(C(CNC(=O)Cc2cccs2)C2CC2)C)=O)cn(-c2cnn(C)c2)cn1 c1(C(N2C3C(C(=O)NCCC4C(C)CCCC4)C(C3)C2)=O)cc(F)c(F)cc1Cl N1(C(CCC=C=C)=O)CC2CCC(N(C(=O)C=CCOCC(F)(F)F)C)C2C1 c1(C(=O)NC2C=CCC(C(N(C3(COC)CC3)C)=O)C2)cccc(O)c1C N1(C(CC(=O)OC)=O)CCC(C)C1CNC(=O)CC1CCC(C)CO1 C1(NC(=O)Cc2cc(C3CC3)on2)CN(C(=O)C2=C(Cl)CCC2)CCC1O C1(CC(N2CCC(CC(C)NC(=O)C(C)CC)CC2)=O)(CSC)CCOCC1 S(=O)(=O)(c1ccc(-n2ncc(Cl)c(Cl)c2=O)cc1)N1C(C(C)C)CN(C)CC1 C=CCCC(CC(C)C)C(=O)NCCC1CCN(C(c2ccc(O)c(C)c2)=O)C1 CCN=c1[nH]cnc2cc(C(=O)Nc3ccc(C(C)=O)cc3)ccc12 Cc1cccc(OCCC(N2CC3CC3(NC(c3cc(CO)oc3C)=O)C2)=O)c1 c1(C(=O)NC(C2(O)CCN(C(c3cc(Br)n[nH]3)=O)C2)C)noc2ccc(Cl)cc12 O=C1CCC2C(C(=O)NCc3ocnc3C(=O)NCC=CCl)C12 c1(C(CCCC2(NC(=O)C(=O)N(C)C)CC2)C)ccc(C(C)(C)C)cc1 C(=O)(C1CCCc2n[nH]cc21)NCCC(C)N(C(c1nccc(SC)n1)=O)C CC(CC(C)(C)C)C(=O)NC1CCC1C(N1CCC(O)(C(N)=O)CC1)=O C(=O)(C1=C(C)OCCS1)NC(CC)(C)CCNC(=O)C=Cc1ccc(C)s1 N1(C(c2c(C)noc2C)=O)CCC(NC(=O)Cc2c[nH]nc2O)C(C(C)C)C1 CC1CCC(NC(c2cn3c(n2)SCC3)=O)CN1C(c1cc(C(F)F)nn1C)=O C(=O)(CCCCCOC)N1CCC(CCC(=O)NCC2CC(CC)C2)CC1 C1(NC(c2cc(Cl)ns2)=O)CCCC(CNC(C2(c3cccnc3)CCC2)=O)C1 c1(CNC(c2cc(C)cc(C)c2)=O)ccc2c(c1)CN(C(c1cncnc1)=O)C2 c1(-c2nc(C3NCC(=O)NC3)on2)nc2c(s1)CCC2 n1(C(CC)CC)ncc(C(=O)N(CC(C)CNC(=O)C(O)CC)C)c1C C1(C(=O)NCC(C)(C)CNC(=O)CC2(C)CC2(Cl)Cl)NC(=O)OC1(C)C C#Cc1ccc(OCC(=O)NCCCCNC(C2CC(O)C2)=O)c(OC)c1 O=C(CC1=CCCC1)NCC1C2CN(C(=O)CCOCC(F)(F)F)CC12 c1(C2C(c3cn(C)nn3)C2)nc(-c2cc[nH]n2)nn1C1CCOC1 C1(NC(CSCCOC)=O)CC(NC(=O)C(c2cccc(Cl)c2)(C)C)C12CCC2 c1(C(N2CCOCC(NC(C3C(C)CC(C)O3)=O)C2)=O)cccc2c1ncn2C Cc1ccn2nc(C(N3CC(C)C(NC(C4CCSCC4)=O)C(C)C3)=O)nc2n1 c1(C(N2C(C)CC(NC(c3cc(C)sn3)=O)C2)=O)cc2ccccc2c(O)n1 C12(C(=O)NC(C3CCN(C(=O)CC=CC(C)(C)C)C3)C)CC3CC1C2C3 CCC(C)(C)C(C(=O)NCC(C)CNC(c1cc(N)cc(F)c1)=O)OC CCCCC(CNC(c1ccc(-c2cccs2)s1)=O)NC(c1nc(O)sc1C)=O C1(F)(CNC(c2cnc(O)s2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)O)CC1 c1(C(CC)NCc2c(F)cc(F)c(F)c2F)cccc(S(N)(=O)=O)c1 c1(C(=O)Nc2ncc(C(C)=O)cn2)ccc(N(C)Cc2ccc(Br)cc2C)cc1Cl Cc1cnc(C)c(C(=O)NC(C2CCN(C(C3CCCC(O)C3)=O)C2)(C)C)c1 C1(CNC(C2CC=CCC2C(F)(F)F)=O)CC2(CCC2)CN1C(=O)CO N1(C(c2n(CC(C)C)ncc2)=O)CC2CCC(NC(=O)Cc3cn[nH]c3)CC2C1 C=CC(CC)CC(=O)NCCCCC1CCCN(C(=O)Cc2cn[nH]c2)C1 c1(C(=O)NCC2(C)N(C(c3ncc(OCC)nc3)=O)CCC2)c(C)[nH]c(C)c1C c1(OC)c[nH]c(C(=O)NCCN(C(C2CCOC(C)C2)=O)CC2CC2)cc1=O c1(C(=O)NC)ccc(C(=O)N(C)CC2(O)CN(C(=O)C=CCCC(C)C)C2)cn1 N1(C(C(=O)N(CC(=O)NCSc2nn[nH]n2)CCC)C)CCNC1=O C1(CC#C)(C(=O)Nc2ccc(N(C)C)cc2)CCN(c2nnc(C(=O)OC)s2)C1 C(c1ccc(I)o1)=CC(=O)N(C(=O)C(CC)c1ccccc1)CCOC C(=O)(CC(C)(C)CC(=O)OC)NC1CC(F)(CNC(c2c(COC)noc2)=O)C1 C1(CNC(c2c(CC)[nH]c(=N)s2)=O)C(C)CCCN1C(=O)C(O)C(C)C c1(CC)cc(C(=O)NC2CC23CCN(C(=O)CCCF)C3)cc(O)n1 Cc1cc(C(=O)N2CCCN2C(C2CC(C)C2)=O)ccc1N1CCOCC1.CCO N1(C(=O)CC(F)(F)F)CCC2CCN(C(C3(F)CC4(CCC4)C3)=O)CC2C1 N1(C(C=COCC)=O)CCC2(CCC(CNC(C3CN(C)C3)=O)O2)CC1 C(=O)(C1=CCSC1)NCC1(CNC(C(N2CCCCC2=O)C)=O)CCCO1 C1(NC(C(CCCC)NC(C2CC3CCC3C2)=O)=O)CCCC(C2CC2)C1 c1(CNC(c2n(C(CC)C)nnn2)CC(C)C)cccc(Cl)c1Br c1(C(=O)NC(C2CCCN2C(=O)CC2CCN(C)C2)C)c(C2CC2)cnn1C C1(C(C)C(=O)NCC(C)(C)F)CCCN(C(C2(CF)CC(=O)C2)=O)C1 N1(C(C(C(C)C)(C)O)=O)Cc2ccccc2CC1CNC(=O)CC1CCN(C)C1 Cc1oc(C)c(C(N2CC(NC(=O)C(n3cc(Br)cn3)C)C(C)C2)=O)c1C c1(C(N2C(CN(C(CCOCCOCC)=O)C)COCC2)=O)cccc(C)c1F C1(NC(c2nnc(C)s2)=O)CC(O)CN(C(c2cc(C3CCOCC3)no2)=O)C1 C1(C#N)(C(N2CCC(OC)(CNC(C3CCC3(F)F)=O)C2)=O)CCCCCC1 C1(C(=O)NC2(COC)CCN(C(=O)Cc3occc3C)C2)CCc2nc[nH]c2C1 C1(NC(CN(CC(C)(C)OC)C(COC)=O)=O)CC(F)(F)C1(C)C CS(=O)(=O)c1sccc1CNC(N1CCCC2OCCC12)=O N1(C(c2c(C)n(C)nn2)=O)CCN(C(=O)CC(C)NC(C2CCCC2)=O)CC1C c1(-c2onc(-c3n(C)nnc3Br)n2)csc2c1CCCC2 C(=O)(CC(C(C)C)OCC)N1CCC(N(C(C2CC(CC)(CC)C2)=O)C)CC1 C1(OC)CNCC(C(=O)NCCc2csc(C(F)(F)F)n2)C1 c1(CC)cc(CC(N2CC(CC(F)C(=O)NCCCCc3cnc[nH]3)C2)=O)on1 CCCCC(CC)CC(=O)NC1COCCN(c2nc(C)nc(C)c2C)C1 c1(C(N2CCC(O)(C(=O)NCCC)CC2)=O)ccc2c(c1)NC(C)CC(=O)N2 C(c1ccc(F)cc1)=CC(=O)NC1CCC(N(C)C(c2ccco2)=O)CC1 N1(c2ncnc(=N)[nH]2)CCCC1C1CCCCN1C(C1CCN(C(N)=O)CC1)=O c1(-n2ccc(C(N(C3(C(=O)O)CCOC3)CC)=O)n2)cccc(C(F)(F)F)c1 C1(C)(CCC)CCN(C(=O)C(C)(C)CNC(C2CC=CCO2)=O)C1 c1(C(=O)NCCCOCCCC)ccnc(CNC(=O)C(C2CCOC2)SC)c1 c1(C(=O)NC2(CO)C(C)C2)cccc(Cn2cc(-c3ccccn3)nn2)c1 CC1(C)CCCCC1CC(=O)NC12CCC(CC1NC(c1ccc(C#N)o1)=O)C2 N1(C(C2(C#C)CCCC2)=O)C2CCC1C(CNC(c1cc(COC)[nH]n1)=O)C2 C1(C(=O)NC(CNC2(C(C)(F)F)CC2)CO)CCN(C(c2cc(CO)on2)=O)CC1 C1(NC(C2CC(NC(C3C(C)CC3)=O)C2)=O)CCC(CN(C)C)CC1 CCCCC(C)C(=O)NC12CC1CN(C(c1conc1C1CCC1)=O)C2 c1(C(N2C(C(=O)Nc3cc(C)cc(O)c3)CC2C)=O)cc(C#N)ccc1C c1(C(N(C(C=CC(=O)N(CC(C)C)CCOC)C)CC)=O)ccccn1 N1(C(C2(n3ccnc3)CC2)=O)CCC(n2nccn2)CC1 CC(C)S(=O)(=O)C(C)C(=O)N1CC(NC(c2nc(=O)n(C)[nH]2)=O)C(C(F)(F)F)C1 N1(C(=O)OC(C)(C)C)CCN(C(=O)Cc2ccccc2OC(F)F)CC1CF C1(CNC(c2ncccc2Cl)=O)C2CN(C(C3(CF)CC3)=O)CC12 N1(C(C2(C(=O)OC)CC2C)=O)CCC(C)(NC(=O)C(=Cc2cccnc2)C)C1 C(=O)(C(=O)N=S(C)(C)=O)NC(CCCNC(CN1C(C)CCC1C)=O)(C)C C(=O)(C(F)C(C)(F)F)N1C(C2(C(=O)NCc3n(C)cnc3)CC2)CCC1 C(=O)(CCCC(=O)N(C)C)NC1CC(C)N(C(=O)COCc2ccnc(O)c2)C1 CS(=O)(=O)c1ccnc(N2CCOCC2CC(=O)Nc2cc(C#N)ccc2Br)n1 N12C3CCC1CC(C3)C(=O)NCC2.N1(C(C)=O)CCC(O)CC1 Cc1cnc2ccc(C(=O)NC3(CNC(C4(Cl)CC4(C)C)=O)CC3)cn12 Cc1nn(C)cc1CN1CCC(CCNC(=O)CCOc2cccc(Cl)c2)CC1 c1(CC=C)cccc(C(=O)NCC2C=CC(NC(c3ccc(C4CC4)o3)=O)C2)c1 N1(C(c2c(C)ncs2)=O)CCCCC1CN(C(=O)C(C(C)C)n1cccc1)C Cc1nc(C(C)C)nc(O)c1C(=O)NCC1C2CN(C(=O)CCNC(N)=O)CC12 C12(C(=O)NCC3(NC(CCN4CC(=O)NCC4)=O)CC3)CCCC1C2(F)F N1(C(c2cn(CCC)nc2C)=O)CCCN(C(C2CCCCO2)=O)C(CO)C1 c1(CNC(C2(CC)CN(C(CSCCCC)=O)C2)=O)ccc(OC)cn1 Cc1cncc(C)c1C(=O)NCC(C)(C(C)C)NC(C1CC2CCC1CC2)=O C1(F)(C(=O)OC)CCN(Cc2nncn2CC(F)(F)F)C1 N1(C(C(C)=C2CCC2)=O)CCC(CCC(=O)N(C2(CCO)CC2)C)C1 c1(CC(C(=O)OC)n2cc(Cn3cc(C)cn3)nn2)ccc(C)c(C)c1 c1(OCC(=O)N(CC(C)O)CCNC(CCc2nc(C)sc2)=O)ccccc1O CCCC(CCCNC(=O)C(C)OCCOCC)NC(c1snc(C)c1N)=O C=C1CCC(C(=O)NCCC2CCN(C(C3CC(OC(C)(C)C)C3)=O)C2)CC1 C1(NC(CSC(C)C)=O)COC2(CCN(C(C3(C#N)CC3(C)C)=O)CC2)C1 CCC(C)CCCCC(=O)NC1C(C)(C)C(NC(c2ocnc2C)=O)C1(C)C c1(C(=O)NCCCC(C)NC(C2(CC)CCCCO2)=O)nccc(C)c1F N1(C(c2c(C)ncnc2)=O)CC2(NC(c3cccn3C)=O)CCC1CC2 Cc1ccc2sc(C(=O)NC(C)CNC(c3ccc([N+](=O)[O-])cc3Cl)=O)cc2c1 N1(C(CN(C(=O)OC)C)=O)C(C(=O)N(CC(O)C2CCC2)C)CCC12CC2 C1(NC(c2c(SC)scc2)=O)CCCCC1NC(c1[nH]c(C)nc1C)=O O=C(CCCCCNC(C1(F)CC2(CCC2)C1)=O)NCCOc1ccc(Br)cc1 Cc1csc2ncnc(N3CCC(C)C3CNC(C3CCCCS3)=O)c12 N1(C(C(C)OCC)=O)CCCC(N(C(=O)C(c2ccccc2Cl)C)C)C1 CC(C)CC(C(=O)NC1CCOC(CNC(C2(F)CCC2)=O)C1)C(N)=O C12(NC(C34N(C(CN5C(C)CCCC5)=O)CC(C3)C4)=O)CCCN(CCC1)C2 CC(CCN1CCC(CS(N)(=O)=O)C1)C(=O)NC1CCCCC1 C12(CNC(CC3N(CC)CCC3)=O)CCC1CN(C(=O)Cc1c[nH]nc1O)C2 c1(OC)cncc(N(C)C(C2CCCC2CNC(c2cnsc2)=O)=O)c1 C1(NC(C(Cn2ccnn2)NC(Cn2nnc(C)n2)=O)=O)CCN(C)CC1 c1(NC(=O)NC(C(=O)NCC2N(C(C)=O)CCCC2)CO)cc2ccsc2s1 c1(OC)cc(OC)nc(C(N2CCC23CC(c2ncc[nH]2)C3)=O)c1 c12noc(n1)C2C.c1(NC(=O)NCC(COCC)C)cnn(CCOC)c1 c1(SCCC(N2CCCC(N(C(C(CSC)O)=O)C)C2)=O)ncnc2[nH]cnc12 Cn1cccc(C(=O)NCC2(C(N3CCOC(CCF)C3)=O)CC2)c1=O C=CCC(C(=O)N1CC=C(C(=O)N(C2CCNC2=O)C)C1)C(C)C C(=O)(CCCCCC(C)O)NC1C(CNC(c2ccc(CC)cn2)=O)COC1 N1(C(C)C)CCC(C(=O)NC(C)(CNC(C2CC2F)=O)CO)CC1 CC(C)C(C)C(=O)N1CCC(CNC(C2CCCC(CF)C2)=O)CC1 CCC(C)(CC(=O)NCCN(CC(C)O)C(c1cccc(COC)c1)=O)C(=O)OC N1(C(C2C(C)C2)=O)CCCC12CCN(C(c1cc3c(s1)CC(C)(C)C3)=O)C2 C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NC1OCCOC1c1ccccc1.c1(S)cn[nH]c1.C1(=O)CO1 C(C(C(C)(C)C)Nc1cc(CN2CCC(CO)C2)ncn1)NCc1ccc(C)o1 c1(OC)cccc(NC(=O)CCN(CC2CC2)CC2CCCO2)c1 N1(C(C=C(C)C)=O)CC(C)CN(C(c2cn(C)nc2C)=O)C(C)C1 CC(CNC(=O)C(F)(F)c1ccccn1)(Cn1cccn1)N=c1cc(Cl)c(O)n[nH]1 O=C1CC2(CCN(C(=O)Cc3cccc(OC4CC4)c3)C2)CN1 c1(NCCN(CCC)CC)cc(Br)ccc1S(=O)(=O)N(C)Cc1cccc(Cl)c1 Cc1noc(C(F)(F)Cl)c1C(=O)NC1CN(C(=O)C#CC2CC2)CC1F c1(C(N2CCC(N(CCC)C(C3CC3CC)=O)C2)=O)ccc2cn(CC)nc2c1 CCC(O)C(F)(F)C(=O)NC(C)CC1CN(C(c2cc(=O)n(C)cn2)=O)C1 CCC(CCC(=O)NCCc1ccncc1F)NC(C1CNC(=O)O1)=O CC#CCCC(=O)NC1CC(CNC(=O)CCCCC2CCCCC2)C1 C(=O)(C(C)(C)C(=O)NC1CCC(C(N2CCC2(C)CC)=O)C1)OCC CCC(C)(CNC(C1CCC(C)N1C(C12CCC(C1)C2)=O)=O)CO C1(C(N2CCC(N(c3ccc(C#N)nc3)C)C2)=O)CCc2cncn2C1 N1(C(C(CC(C)C)F)=O)CCC2OCCN(C(=O)CCC(=O)c3cccs3)C2C1 c1(-c2cn(Cc3ccc(N4C(=O)NCC4)cn3)nn2)ccc2nccnc2c1 C1(C(N2CCC(N(C(Cc3ccc(OC)cc3)=O)C)C2)=O)Cc2ccccc2C1 c1(C(=O)OC)[nH]nc(NC(=O)NC(CO)C(O)c2ccccn2)c1Cl C1(C(N2CC(C#C)(F)C2)=O)CC(F)CCN1C(=O)Cc1nc(=N)[nH][nH]1 c1(NC(C)=O)ncc(S(=O)(=O)NC2CN(C(c3nccs3)=O)CC2F)s1 N1(c2ccnc(SC)n2)Cc2[nH]nc(NC(c3cccc4[nH]ccc34)=O)c2C1 c1(C(=O)NCCCCCN(C(c2c(CC)ccs2)=O)C)cc(OC)cc(C)n1 C=CCC(CC)C(=O)N1CCN(C(c2cncc(C)c2Cl)=O)C(CCO)C1 c1(OCC(N2CC(CN(C3(C)CCCCCC3)C)C2)=O)ccccc1[N+](=O)[O-] CC1CCCN(C(=O)CCn2ccnn2)C1CCNC(=O)CN1CCN(C)CC1 C1(c2n(CCOCC)nnn2)(Nc2cc(C)cc(Cl)c2)CC2CC1CC2F CCC(C)C(O)C(C)C(=O)N1CCC(OCCNC(=O)CCc2csnn2)C1 Cc1cc(C(=O)NCCC2(O)CN(C(c3cn(C)nc3Cl)=O)C2)cc(C)c1F C1(C(N2CC(F)(CNC(C(C)(C)CO)=O)C2)=O)CC12C1CC3CC(C1)CC2C3 c1(C(CNC(c2ccnn2CC(C)C)=O)NC(C(=O)NCC)=O)cccc(C)c1 C1(OC)CN(C(=O)COCC2CC2)CC1NC(C1CCCCCS1)=O C1(CNC(c2sccc2Cl)=O)CCCN(C(c2cccnc2OCC(F)F)=O)C1 c1(C(=O)NCC(C)CNC(=O)C(C(C)(C)C)n2ccnn2)ccc([N+](=O)[O-])cc1 C1(F)(C(N2CCN(C(C(C)C3CCCC3)=O)C(C)C2)=O)CCC(F)(F)CC1 N1(C(c2ccn(C(C)C)n2)=O)CC(C(=O)NC2CCCSC2)C(C)(C)C1 Cc1nc(Cl)ccc1C(N1CC(O)CC1C(=O)Nc1cnc(Cl)c(Cl)c1)=O CC1CCN(C(c2ccc[nH]2)=O)CCN1c1ccnc(C2CC2)n1 Cc1ncn(C)c(=O)c1C(N1CC(O)(CNC(C2(C#N)CC3(CCC3)C2)=O)C1)=O C1(OC)CC2(C1)CC(C(=O)NCC(CO)NC(=O)CC1CCC(F)(F)CC1)C2 C=C(C)C(C)(C)C(=O)NC1CN(C(c2coc(C3CCCC3)n2)=O)CCC1CO N1(C(CC(CC)(C)C)=O)CCCN(C(=O)Cc2ccccc2C(=O)OC)CC1C N1(C(C(CCC2CCC2)NC(c2ccn(CC)n2)=O)=O)CCc2ncncc2C1 C(c1c(Cl)cccc1Cl)=CC(=O)N(CC(C)(C)NC(c1c(C)snc1)=O)C c1(OC)c(NCc2cccnc2OC(F)F)cc(Cl)cc1C(N)=O Cc1nsc(N2CCC(NC(=O)CC3CC=CCC3)C2)n1 CCCCC(O)C(=O)NC1CN(C(=O)CCN(c2ccccc2)C)CC1O CC1CC(CNC(=O)CC2CC=CC2)CN1C(=O)Cc1cccc(O)c1 N1(C(CC(CCC)C)=O)CC(NC(=O)Cn2ncc(Br)n2)CC(C)(C)C1 c1(C(=O)NC(c2ccc(C)cc2)CNC(c2ccco2)=O)cc(N)c(F)cc1C C1(C(N(CC(C)NC(C=CCC)=O)C)=O)CC(=O)NC(=O)C1 C(=O)(CC1(O)CCOc2ccccc21)NC1CCN(C(C(CCC)CCC)=O)C1 N1(C(CC2(OC)CCC2)=O)CC2(CC(NC(c3ccccn3)=O)c3nccn32)C1 C1(C(=O)NCC2(O)CN(C(c3cc(OC)c(F)cc3)=O)C2)CC2C=CCC(C1)C2 c1(C(N2CC(C(C)(C)O)(CNC(CCCCCC)=O)C2)=O)cc2n(n1)CCCO2 c1(CNC(COCC#C)=O)cc(C(=O)NC2(C(N)=O)CC(CO)C2)n[nH]1 c1(N(C)CC23CCCC2OCC3)nc(=NCC2CSCCO2)[nH]c2ccsc12 Nc1cc(Cl)nnc1C(=O)NC1CS(=O)(=O)CC1NC(=O)Cc1c[nH]nc1O C(CC(=O)NCC(O)CNC(c1cnn(CC(C)C)c1CC)=O)(C(C)C)OCC n1(SCCN2CCN(C(CN)=O)CC2)c(=O)oc2cccnc12 CCC(N=c1nc2c(cnn2C)c(N(C)CCc2cnc[nH]2)[nH]1)c1ccncc1 c1(C(=O)NCC(CO)NC(C(C(C)C)O)=O)cc2ccnc(Cl)c2s1 CCC1=C(C(=O)NCC(C2CC2)NC(c2cc3nc(=O)ccn3[nH]2)=O)CCCO1 c1(C(=O)OC)cc(-c2cn(CC3CCCC(C)C3)nn2)cnc1OC CCCC(C(=O)NC(C)CC(C)NC(c1ccc(C(C)=O)[nH]1)=O)C(C)C C(=O)(CC1=CSC2=NCCN12)NCC1(O)CCN(C(C2CCCC(C)C2)=O)CC1 S(=O)(=O)(c1c(C)cccc1Cl)NC1C2CN(C(CCCC=C)=O)CC21 N1(C(C(N2CC(CC)(NC(=O)OC(C)(C)C)C2)=O)=O)CCn2cncc2C1 Cc1ccc(N2C3CCC2CC(NC(c2nccnc2N)=O)C3)c([N+](=O)[O-])c1 C1(CC=C)(C(=O)NCC(=O)N2CCCO2)CCN(C(=O)C(F)C(C)C)C1 c1(C(=O)NC2CCC(CNC(CCC#CC)=O)C2)cc(OC)c(S(N)(=O)=O)s1 C1(C(N2C(CN(C(C=NOC)=O)C)CCCC2)=O)OC2CCC1CC2 c1(OC)ccc(NC(=O)C(=O)NC(C)C(=O)NO)cc1S(C)(=O)=O CC(C)(C)C(C(=O)NCC1CCC(F)(F)C1)NC(=O)CC1CC1C1CC1 c1(C(N(C2CCCN(C(=O)C(C(C)C)SC)C2)CC)=O)cc2ccccc2s1 CC1CC2(CCO1)CCN(C(c1cccnc1-n1cccn1)=O)C2 C1(C(N(CC(C)NC(C2CC(NC(c3ccco3)=O)C2)=O)C)=O)CCCOC1C c1(NC(CC(N2CCCC2)=O)=O)cccc(-c2cnn(C3CCOC3)c2)n1 C1(O)(CNC(C(C)S(C)(=O)=O)=O)CC2CCC(C1)N2C(=O)Cc1cncnc1O N1(C(c2ccc(CNC(C=C(C)C)=O)cc2)=O)CCN(C)C(=O)C1C C12(CNC(C(CC)OCC)=O)CCC(NC(c3cccc(CCO)c3)=O)(CO1)C2 C1(NC(C(C)Cc2ccc(F)cc2)=O)CN(C(C2CCOC2)=O)CC2(CC2)C1 c1(CC(=O)NC2(CCCC)CC2)ccc2c(c1)CC2.C123CC(CO1)(C2)CNC3=O C1(CNC(CC2N(CC)CCC2)=O)CC2CCC1N(C(=O)CP(C)(C)=O)C2 N1(C(=O)C=CI)CCC2(CCCN2c2nc(C3CCOCC3)ns2)CC1 CC1CCN(C(=O)CSCc2ccccc2Cl)C(CNC(c2cc[nH]n2)=O)C1 N1(C(c2ccns2)=O)CCC(C2CCN(C(c3cnc(C(F)(F)F)s3)=O)C2)CC1 N1(C(C(C)N(C(CCCOCC)=O)CC)=O)CCC(F)(F)C(C)C1 c1(C(N(CCC(C(C)C)NC(=O)CC(C)(C)C)C)=O)ccc2c(c1)CN(C)CC2 Cc1sc2ncnc(N3CCCC(C)(CNC(=O)C=Cc4cnc[nH]4)C3)c2c1C N12CCOC(C1)C2=O.CC(C)(F)C(=O)N1CCC1(C)CC(c1ccccc1)=O C(=O)(C1CCCc2c[nH]nc21)NC1(CC)CCN(C(C2CCC(C)C2)=O)CC1 Cc1ccc(-c2nc(C(N3CC(F)CC3CNC(=O)C=CC3CC3)=O)cs2)cc1 C12(C(=O)NCCCCNC(C=CCN(CC)CC)=O)CCCN1CC(O)C2 c1(C2C(NC(c3c(Br)n[nH]c3Br)c3n(CC=C)nnn3)C2)ccc(F)cc1 CCCC(C)(CCC)C(=O)NCC(CC(C)C)NC(c1cnn2c1OCC2)=O Cc1cc(C(N2CC=CC2C(=O)NCC2COC(=O)N2)=O)c(C)s1 C1(NC(C(C)OCC#C)=O)C2CC1CN(C(=O)C(N1CCC(C)C1)=O)C2 C1(NC(c2sc(CC)c(C)c2)=O)CN(C(c2ccc(F)cc2O)=O)CC12CC2 C1(CC)(NC(=O)COCC2CC2)CCCCCC1.C12CC(C1)C(=O)NC2 Cc1cnc(C(=O)NCCN(C(c2n[nH]c(C)c2F)=O)C(C)C)c(Br)c1 C=CCCCCCN=c1ccn2ncc(S(=O)(=O)NC(C)CC(N)=O)c2[nH]1 C1(NC(c2nc(Cl)ccc2Cl)=O)(CO)CCCN(C(C2(Br)CC2)=O)C1 C(CO)(C(C)NC(c1cc(CNC(=O)CSCCC(C)C)[nH]n1)=O)SC c1(C(=O)NCc2c(C(=O)NC(CCSC)CO)con2)cnn(C)c1Cl n1(CC)cc2ccc(C(=O)NC3CN(C(c4cc(Cl)n(C)n4)=O)CC3C)cc2n1 C1(CNC(C2(CC)CCNC2=O)=O)CN(C(C2(C)CCC(=O)N2)=O)CCC1(F)F C(=O)(C1CSc2ccccc21)NC1C(NC(C=Cc2c(C)n(C)nc2)=O)COC1 C1(c2ccccc2)(NC(C)CC2CN(Cc3cc(I)n(C)n3)C2)CCCC(=O)N1 N1(C(CC(C=C)C)=O)CC(CC(=O)NCc2cc(OC)nn2C)CC1(C)C c1(CC(N2C(CN(C(C(C(C)C)SCC)=O)C)CCCC2)=O)ccc(Cl)nc1C CCCCC(CNC(C1CN(C(=O)CCc2ncnn2C)CC(C)O1)=O)CCC N1(CC(=O)NC(C2CCOC2)C#C)CCN(C(C2(CC)CC(F)(F)C2)=O)CC1 c12ccc(cc1Cl)CCCN2S(C)(=O)=O.c1(CC(=O)OC)cnn(C)c1 C1(NC(c2cccc(=O)o2)=O)CCC2(CC1)CC(NC(=O)C(O)CC1CC1)C2 c1(C(N(C2CCCCC2)C(C(=O)OCC)C)=O)cnc(SCC(F)(F)F)o1 c1(CC)cc(C)c(C(=O)NCCC(C)(C)CNC(=O)CC2(O)CCCCC2)o1 c1(C(=O)NCC(CC)(CC)NC(=O)C(O)C(C)OC)c(Cl)nc2ccccn12 c1(C(N(C2CC(C(F)C(=O)NCC(C)(C)C3(O)CCC3)C2)C)=O)ccn(C)n1 N1(C(C(C)NC(CCC)=O)=O)CCC2(CC(NC(c3c(C)cccc3Cl)=O)C2)C1 N=c1c(C(=O)NCCC2CCN(C(=O)Cn3ncnn3)C2)c[nH]c2ccccc12 NC(=O)CC(O)C(=O)NC1CC2(C1)CC2C(=O)NCCOc1ncccn1 C1(C(N2CC(CNC(C3(CC#C)CCOCC3)=O)C2)=O)CC12CC(F)(F)C2 N1(C(c2c(Br)cn(CC)n2)C(=O)NC2CCCCC2)CCCSc2cc(C)ccc21 C1(O)(C(=O)NCC2C(NC(=O)CSC3CC3)CC2)CCc2ccccc2C1 N1(C(c2cncc(CC)c2)=O)CC(C(=O)N(C)Cc2ccoc2C)CCC1(C)C c1(NC(=O)NC(CCOC)(C)C)c(N)cccc1Br Cc1c(C(=O)NCc2cn(CCNC(C3CCC3C)=O)nn2)cnn1C(C)C c1(CN(C(=O)C(C)(C)N(C)C)C)ccccc1CNC(=O)C(C1CCCCC1)F c1(C(=O)NC2CC(F)(CNC(C(c3ccc(F)cc3)CC)=O)C2)csc(=NC)[nH]1 CCC(C(=O)NCC(C)CNC(c1ccc(C)s1)=O)N(C)C Cc1ccc(OCCC(=O)NCC(C(C)(C)C)NC(c2nn(C)cc2N)=O)cc1 CC(C(=O)N1CCC(CNC(=O)COCC2CCCC2)C1)S(N)(=O)=O N1(C(Cn2c(C)ncc2)=O)CC(NC(c2cc(C(F)(F)F)cc(F)c2)=O)C(C#N)C1 C1(COC)(NC(C2CCC(=O)N2C)=O)CCN(C(C2CC(C)(C)C2)=O)CC1 C(CCCCCNC(c1ccc(Cl)cn1)=O)NC(c1c(COC)ncs1)=O C(c1ccc(F)cc1)=C(C)C(N1CC2CC1(CNC(=O)C(C)CF)C2)=O C1(CC(=O)NC(CC)C(=O)NC23CC(F)(C2)C3)CCOC1(C)C N1(C(=O)NC(C)(C)CCCO)CCNC(=O)C(F)(F)C1 N1(C(c2c(CC)c[nH]c2)=O)CC(N(C(=O)CCC2CCOCC2)C)C(F)C1 CC(C(=O)NCCN(CCCO)C)N1CCCC1.C12CC(C1)C(=O)NC2 Cc1c(NCc2ccccc2-c2ncc[nH]2)ncnc1N1CCC(C2CC2)C1 N1(C(c2ccc(OC)c(OC)n2)=O)CCN(C(=O)C(C)S(N)(=O)=O)C2COCC12 c1(SCC(=O)NC(C(C)NC(Cn2ncc(CC)c2)=O)C)ccc(C(F)(F)F)cn1 C1(O)(CNC(=O)CN2CCCS2(=O)=O)CCCN(C(=O)C(c2ccccc2)O)C1 N1(CCCCCCC(N)=O)CCC2(CC1)NC(=O)N(CC(=O)O)C2=O C=C(C)CC(C(=O)NCC#CC(F)(F)F)NC(=O)CCn1ccnn1 c1(C(N2CC3(CC(NC(C(C)n4cccn4)=O)C3)C2)=O)cc2cccnc2[nH]1 c1(NCC(=O)Nc2cn(C)nc2)ccc2c(c1)OCCO2 C(=O)(C(C)CCC(C)(C)C)NC(CNC(C1CCN(CC(C)C)C1)=O)C C1(NC(C(CC)N(C)C)=O)CC1C1CCCN(C(c2cc(C)n(CC)n2)=O)C1 C(=O)(C1=CS(=O)(=O)CCC1)N1CCCC(O)(CNC(c2[nH]cc(CC)c2)=O)CC1 O=C(CC1=Cc2ccccc2C1)NC1C=CCN(C(=O)Cc2cncnc2)C1 CCCC(CC)C(=O)NCC(C1CCN(C(=O)C(C)(C)c2ccsc2)CC1)(C)O c1(CC)ncncc1C(=O)NC1CC1CNC(c1ccc(CO)s1)=O CN1CCCCC1CC(=O)N(CC(=O)NC1CCOC1=O)C1CCC1 N#Cc1ccc(C(N2CCC(C3CC3)(CNC(C3(CO)CCC3)=O)C2)=O)c(O)c1 CC(CCC(=O)N1CCC(C)(O)C1)NC(=O)CSC1CC1 C1(NC(c2c(SC)cc(F)cc2)=O)CN(C(=O)Cc2ccno2)C2(CCOC2)C1 c1(C(=O)NCCC2CCN(C(C)=O)C(C)C2)c(F)ccc2[nH]ccc12 CC1(C)OCCC1C(N1CCSCC1C(=O)NC1C=CC(CO)C1)=O c1(C(=O)NC2CC3(CC(NC(C(COC)C)=O)C3)C2)nc(Cl)c(Cl)c(N)c1Cl C1(CC(=O)NCc2cc(C(N)=O)no2)CCN(C(=O)C2=NOCC2)CC1 C1(CC(=O)NCCC2CC(NC(C3(CC=C)CCCC3)=O)C2)CC(CC)=NO1 c1(NCC(=O)NC2(NC(=O)C=CCOCC3CC3)CCOC2)cc(F)cc(F)c1 C12(C(=O)NCCCCCNC(C(CC=C)CC)=O)CC(CO)(C1)OC2(C)C c1(C(C(=O)NCC)N(CC(=O)OC)CC(=O)OC)ccc(C2CC2)cc1 c1(NCC2(C)CC(F)(F)C2)ccc(S(=O)(=O)NC2C3COCC23)cc1Cl c1(C(N(C)Cc2nc(C(C)OC)sc2)=O)cc(Cl)nnc1Cl CC1CCCC(NC(=O)CCCNC(=O)C(=O)C2CCCC2)C1 c1(C(=O)NCC23CC2CN(C(c2cnc(S)[nH]2)=O)C3)ccc2oc(O)nc2c1 C1(NC(C2CC(=C)C2)=O)CCC(NC(=O)C(c2cncn2C)O)C1 n1(C(C)C)ccc(CNC(=O)CC2CCN(C(=O)C=Cc3ccoc3)C2)n1 C1(NC(C2(C)CC=CCO2)=O)CCN(C(c2scnc2Cl)=O)CC1O c1(C(=O)NC2C(N(C)C)CC2)cccc2cncn12 N1(C(C2(C)CC(=C)C2)=O)CC2CCCC2(NC(c2onc(OC)c2Br)=O)C1 N1(C(c2c(C)c(=O)cc[nH]2)=O)CC2OCCN(C(=O)C(C)C(C)O)C2C1 C1(C(F)(F)F)(C(=O)NCC(C)CNC(=O)C(F)=C2CCCC2)CCOCC1 c1(NC)cncc(C(N2CCCC2C(=O)NCC2C3CCCOC23)=O)c1 C1(C(=O)NCC2C(NC(c3ccc(-c4ccccn4)s3)=O)C2)CCC(F)CC1 CC(C)CC(=O)C(=O)N1CCC(CNC(=O)C(F)C(F)(F)F)C1 c1(NC)ncccc1C(=O)NCCCC(C)NC(=O)CCC(=O)N(C)C N1(C(CC2(C#N)CC2)=O)CCC2CCC(NC(=O)C(O)Cc3cnc[nH]3)C1C2 C1(C(=O)OC)CCN(C(=O)CC2(NC(CC(=O)NCC)=O)CC2)CC12CCC2 C(=O)(C1=CNS(=O)(=O)N=C1C)NC1CC2CN(C(CCN(C)CC)=O)C1C2 CCCCC(CNC(c1cc(C)n(CCO)n1)=O)NC(C1CCCO1)=O CCC(CC)C(=O)N(C)CC1CCN(C(=O)Cc2ccnnc2O)C1 c1(CC)ccccc1C(=O)N(C1(CC(=O)N(CC(N2CCOCC2)=O)C)CC1)C C(=O)(C1CCc2ccc(C(=O)O)cc21)N1C(c2cn(C(C)CO)nn2)CCC1 c1(Nc2ncccn2)ncc2[nH]ncc2n1.c12csc(n1)NC(=O)C2 C(CCN=c1ncc(C(F)F)c[nH]1)NC(C(C)Nc1ccc(C)cc1)=O Cc1nn(C)cc1C(O)C(=O)NCCC(C)NC(c1nn[nH]c1C(F)(F)F)=O CCC(CN(C)C)C(=O)N1CCC(C)(NC(c2ccoc2)=O)C1 C(=O)(CCC(F)F)NC(C)CCCNC(C1(C)CC1C(F)(F)F)=O Cn1nc(I)c2cc(C(N3CC(CC(=O)NCC(C)(C)CO)C3)=O)ccc12 N1(C(CCCOCC)=O)CCOC2(C1)CN(C(c1cccc(Cl)c1F)=O)C2 N1(C(CCC(N)=O)=O)Cc2ccc(CNC(c3cn[nH]c3)=O)cc2C1 c1(C(N(C(CNC(CSCC#C)=O)C)C)=O)ccc(NS(=O)(=O)CCCC)cc1 Cc1cc(C(=O)NCCCN(C)C(c2cn(C)nc2C2CC2)=O)nnc1O N1(C(c2c(CCNC(c3ncn(C)c(=O)c3)=O)n[nH]c2)=O)CCSC2CCCC12 c1(OCC(=O)NCC(CO)N(C)C(c2cnn(CC3CC3)c2)=O)ccc(F)cn1 c1(C(N2CC(NC(c3cc(C)c(C)[nH]3)=O)CC(OC)C2)=O)sccc1S(N)(=O)=O N1(C(C(c2cccnc2)OC)=O)CC(NC(=O)C(O)CC(N)=O)C2(CC2)C1 C1(C(=O)N(C2CCC3CC23)C)(CC)CCN(C(C2CC2(F)F)=O)C1 N1(C(c2c(C)cccn2)=O)CC(C(=O)NC2CC(O)C2ON)C2(CC2)C1 N1(C(C(C(C)C)NC=O)=O)CCCC2(CCN(C(C3CCC(C)(C)OC3)=O)C2)C1 C12(C(N(CCN(C(C)C)C(c3cccc[n+]3[O-])=O)C)=O)CC3CC(C(=O)N1)C2C3 CC1Cc2ccccc2N(C(=O)C=Cc2ccc(C(C)(C)C)cc2)C1 N1(c2cc(C(C)C)ncn2)CCC(NC(c2ccc(C(C)C)s2)=O)C2(CCC2)C1 CC1CN(C(=O)CC2CCOC2=O)C1C(=O)Nc1cnn(C2CC2)c1 C1(CNC(C2(C)ON=C(C)C2)=O)(CO)CC12CCN(C(c1cocn1)=O)CC2 N1(C(C2CC(NC(C(C)(C)OCC)=O)C(O)C2)=O)CC(C2CCCCC2)C1 N1(C(CC(COC)C)=O)CC=C(C(=O)NC2C=CC(CO)C2)CC1 N1(S(C(C)C)(=O)=O)CCOC2(CCCN(C(c3ncc(Cl)cc3Br)=O)C2)C1 CCC(CC(=O)NC(C)C(=O)NCC(C)(F)F)OC C1(C(N2C(C)CN(C(C3(O)CCOCC3)=O)CC2)=O)CC2CSCC(C1)C2 C1(C(N2CCC(N(C(=O)C=CCO)CCO)C2)=O)CCc2nnc(C(F)(F)F)n2C1 c1(CC(=O)NCCCNC(C2C(OC)CC2)=O)cnn(C(C)(C)C)c1 c1(C(C)(C)SC)cn(C(C)C(=O)NC(CCN2CCCC2)=O)nn1 C1(NC(c2n(C=C)nnc2)=O)CN(C(=O)CCN2CCNC(=O)C2)C2(CCC2)C1 Cc1ncc(C(=O)NC(C)CCCNC(C2(C(C)(F)F)CC2)=O)[nH]1 N1(C(C(c2c(C)cccc2)(F)F)=O)CCS(=N)(=O)C(C)C1 N1(C(C=CC)=O)CCC2(CC1)CN(c1ccnc(C(=O)OC)n1)CCO2 N1(C(C2C(CC)OCC2)=O)CCCC(N(C)C(C2CCOC(C)(CC)C2)=O)CC1 N1(C(C(=O)NC(C)CN2CCCC2=O)=O)CCC2CCC12c1ccccc1 c1(NC(C2C(NCc3scc(C)n3)CCC2)=O)cc(Cl)cnc1O CCC(C)C(C(=O)N1CCCOC(CNC(c2cc(C)c(C)[nH]2)=O)C1)OC N1(C(c2c(CCC)n(C)nn2)=O)CC(NC(=O)CN2CCSCC2)C(C2CC2)C1 c1(OC)cnc(Cl)cc1C(=O)NC(C1(CNC(=O)CCC(F)(F)F)CC1)C CC#CCCC(=O)NC(C1CCN(C(C2(c3ccc(Br)cc3)CC2)=O)CC1)C CC(C)C(CCC(=O)NOCC=CCl)NC(C1CCCCC1O)=O CCC(C(=O)N1CCCC1CNC(=O)C(C)=C1CCC1)SC N1(C(CC(C)(C)SC)=O)CC2CC(C1)N2C(C1CC1C(F)F)=O c1(C(N2CCC(C)C(NC(=O)Cc3cncnc3)C2)=O)cc(F)c(O)c(F)c1 c1(C(N(CC(O)CF)CC)=O)ccc(CNC(C2CC(=O)N(C)C2)=O)cn1 Cn1ccc2nc(N(C3CCCCNC3)C(c3cccc(Br)n3)=O)ncc12 C1(C(=O)NCCOC(CC)CC)COC2(C1)CN(C(=O)CC(C)=C(C)C)C2 n1(CC)[nH]cnc1=NC(=O)C(=O)N(C(C)CF)C N1(C(c2nc(C)n(C)n2)=O)CC2(CCN(C(C3(N=[N+]=[N-])CC3)=O)CC2)C1C(C)C C(=O)(C1=CS(=O)(=O)CCC1)N1C(C)CCC(NC(=O)C=Cc2ccc[nH]2)C1 C1(C(C)C)CC(CC(=O)N(CC(C)(C)CNC(=O)CC2CC(C)(C)C2)C)CCO1 N1(C(c2cc(C)cc(O)n2)=O)C2CCC1CC(CNC(=O)CC13CCCC1C3)C2 CCC(C)(CO)C(=O)N1CC2CC2(CNC(=O)CNC(c2ncccc2O)=O)C1 N1(C(CC(C=C)CC)=O)CCCCCC(NC(=O)Cc2occc2C)C1 c12cccc(c1)NC(=O)C2C.C12CC(C1)NC2C.CCCCSC(C1CCC1)=O N1(C(C(C)Sc2ccc(C)cc2)=O)CC2=C(C1)CN(C(c1coc(C)n1)=O)C2 c1(CC(N2CCN(C(CC(=O)OC)=O)CC2)=O)ccc(F)c(C(F)(F)F)c1 C1(NC(C2(CCNC(C3CCC(=O)C3)=O)CCC2)=O)CCC2(CCC2)C1 CC1=C(C(=O)N2CC(NC(C3CN(CC(F)(F)F)C3)=O)C2)Cn2nnnc2N1C Cc1noc(C)c1C(=O)NCC1C=CCN1C(=O)COCC(F)(F)F C(=O)(C1CCCc2nc(C)[nH]c21)NCC(C)(CO)NC(c1cncc(C)c1)=O c1(CN2CCC(C)(C(N3CCS(=O)CC3)=O)C2)cc([N+](=O)[O-])ccc1Br c1(SCC)ccc(C(N2CCCC2C2(c3ccc(COC)cc3)CC2)=O)cn1 CN1CCN(C(Cn2cc(C)nn2)=O)CC1.c1(C(C2CC2)N)ccccn1 C12(C(=O)NCCOCCN(C)C(c3cc(Cl)c(Cl)[nH]3)=O)CC1COC2(C)C C1(C(N(C)CC2CCCN(C(C34CC(OC)C3C4)=O)C2)=O)C2CCC3C(C2)CC13 N1(C(c2c(C)cccc2Cl)=O)CCC2(CCC(NC(C34CC3CNC4=O)=O)C2)C1 Cc1ccn(C(C)C(=O)N(C(C)CN(C(=O)CN(C)C(N)=O)C)C)n1 c1(C2N(C(C3CC(F)(F)C3)C(=O)NCC)CCC2)ccc(C(C)(C)C)cc1 c1(NC(=O)NCC(F)Cl)ncc2nccnc2n1 Cc1cc(C(N2CCOCC2CN(C(=O)Cn2cncn2)C)=O)c2n[nH]cc2c1 C1(NC(CCSC)=O)Cc2ccccc2C1NC(c1ccc([N+](=O)[O-])cc1F)=O CCCCCS(=O)(=O)CC(=O)NC1CN(C(C2CCCN2C=O)=O)CC2(CC2)C1 c1(CN2C(NS(CCCC)(=O)=O)COCC2)cc(OC)c(OC)cc1C C1(C(=O)NC(C(O)CO)C2CC2)CC(O)CN1C(=O)CCc1cncnc1 N1(C(c2nccc(OC)n2)C(=O)Nc2ccc(F)cc2)CCC(C)(C2CC2)C1 C1(CC(=O)NC2CCN(C(=O)NC3(c4ccncc4)CCC3)C2)CCCC2CC12 c1(C(N2CCC(CNC(C3C4CC5C(C4)C35)=O)CC2)=O)cc2scnc2[nH]1 c1(C(N2C(CC(=O)NC(C#C)C(C)OC)CCC2)=O)cccc(CC)c1 C1(CNC(c2ccnn2C(F)(F)F)=O)CC(F)CN1C(=O)COC1CCCCC1 C(CCCC(=O)N1CC(N(C(=O)C(C)CCOC)C)C1)OCCC=C c1(C(=O)NCC(CNC(c2c(CCC)nco2)=O)O)cncc(OC(C)C)c1 N1(C(c2c(OC)cccc2Cl)=O)C2CCC1CC(CNC(c1n[nH]cc1Br)=O)C2 c1(OCC)ccc(C(N2CCC(F)(CNC(=O)CNC(=O)OC)C2)=O)cn1 C(=O)(CC(=O)NCC(C)N(C)C(c1cnn(C2CC2)c1)=O)OC c1(CCN(C2CCN(CC3COC3)CC2)C)ccc(S(=O)(=O)NCC(=O)OC)cc1 C(=O)(C1=CCCCN1C(=O)OC(C)(C)C)NCC1CC(CN(C)C)C1 c1(NC(=NCc2ccc(C(F)(F)F)cc2)NC2CCCC2)ccc2occc2c1 C(C1=CCN(C(=O)C(c2ccccn2)O)CC1)NC(C=C(C)Cl)=O C(=O)(C(O)P(C)(C)=O)NC1C2CN(C(c3cc(OC(C)(C)C)ncc3)=O)CC21 c1(CC(=O)NCC2CC(F)(CNC(CN(C)CC)=O)C2)ccc(C)cc1 N1(C(=O)CCc2cncnc2)CC2CC2(C(=O)NCCc2cccc(Br)c2)C1 C1(C(N(CCC(C)NC(=O)C2=CCOCC2)C)=O)CC12CCOCC2 C1(C(CC)NC2CCN(CC(=O)O)CC2)CCCC(C)(C)C1 C#CC1CCCN(C(C2CCN2C(=O)CN(C)CCOC(C)=O)=O)C1 CC(CNC(C12CC(C#N)(C1)C2)=O)C(F)C(=O)NC1CN2CCCC1C2 N1(C(COCP(C)(C)=O)=O)CCOCC(NC(=O)C(c2cccnc2)O)C1 C1(C(N2CCCC(C)C2CCO)=O)(OC)CCN(C(=O)CCc2ncc[nH]2)CC1 Cc1cc(C(=O)NC2CC2NC(c2nocc2C(C)C)=O)sn1 C1(CCC)CC(C(N2CC3C(CNC(=O)COc4cc(C)on4)C3C2)=O)CCO1 c1(C(C(=O)NCCOCC)N(C(C)CCC(C)C)C)nn(C)nc1Br c1(C(N2CCC(F)(C(=O)NC3CCN(C(C)C)CC3)C2)=O)c(Cl)cccc1Cl C1(CNC(C2CCCN(C(C)C)C2)=O)CC2(C1)CN(C(=O)COc1ccon1)C2 C12(C(=O)NCc3c(CNC(C(CC)COC)=O)cccc3)CCC(F)(CC1)CC2 CCCC(CCC)C(=O)N1CCCC1CN(C(=O)COCc1nc(C)no1)C C1(C(=O)NCC(CCNC(c2cc(OC)ncc2)=O)O)Cc2cc(Cl)ccc2O1 c1(OC)cccc(Cn2nnnc2C2(NCCC=CBr)CCC3CC23)c1 c1(CC)ccc(F)c(C(=O)NCC2(C)CCN(C(c3nc(C4CC4)cs3)=O)C2)c1 Cn1ncc(C#N)c1C(N1CCC2(NC(=O)Cc3cnc[nH]3)CC2C1)=O N1(C(c2cncc(OCC)c2)=O)CCC2(CC(NC(=O)C(C)(C)S(C)(=O)=O)C2)C1 c1(CNC2CC2)nc(Cl)ccc1F.c12ccsc1CNCC(O)CNC2=O c1(NCCN(CC)CC)cc(=NC(C)c2ccc[nH]2)[nH]c(C(C)C)n1 c1(Cc2nnc(-c3ccc(OC)cc3OC)o2)cn2cc(Cl)cc(Cl)c2n1 N1(C(C2C(CNC(c3ccc(O)nc3)=O)CC2)=O)CCC2CCCC2CC1 N1(CC(N2CC(CC(F)C(=O)NCc3ccc(O)cc3)C2)=O)C(=O)CCCC1=O CC1(C)CC(=O)N(CC(=O)NCC2CCC2NC(C2(C3CCC3)CC2)=O)C1=O c1(CNC(=O)NC2C(C)(CC3CC3)CCC2)cc(Br)cnc1O c1(OC(C)CC(=O)NCc2cnnn2Cc2ccccc2)ccc(Cl)cc1Br C12(C(N3C(C(=O)NCCOCCCC)CCCC3)=O)CCC(CO)(CC1)C2 CC1CC(C)N(C(c2cn(C)ccc2=O)=O)CCN1C(c1cc(O)cc(=O)o1)=O C1(CN(C)C(c2ccncc2F)=O)COCCN1C(=O)CCc1cncc(F)c1 C(CC(=O)NCC1(F)CCOCC1)(C(F)(F)F)NC(C(COC)C)=O C#Cc1ccccc1CNC(=O)CC1(C)CCN(C(=O)CCCC#CC)C1 CC(C(=O)NCC1(NC(=O)C(F)=C2CCCC2)CCOC1)C(=O)N1CCOCC1 C1(C(=O)NC2(C)CN(C(c3cc(C(F)(F)F)cnc3O)=O)C2)CC2CC1C1CC21 CC(O)C(C)(C)C(=O)N(CCCN(C)C(C1CCN(C)C1)=O)C Cc1ccc(Cl)cc1C(N1CC(C)(NC(C2CCC3CC23)=O)C1)=O C1(NC(c2csc(Cl)c2)=O)CCOCC1NC(C1CC(F)(F)C1)=O c1(CC(N2C(CNC(C3C(C)CCC3)=O)CC(C)(C)C2)=O)ccc(C#N)cc1F N1(C(CNS(C)(=O)=O)=O)CC2ON=C(CNC(c3ccc(C(N)=O)cn3)=O)C2C1 CCC(C(=O)NN(C(=O)OC)c1ccco1)c1ccc(OC)c(OC)c1.C(C)(C)(C)O C(=O)(C1c2ccccc2C2CC1C2)NCC1C(CNC(C2(CCC=C)CC2)=O)C1 C(=O)(C1(C)CCCc2ccccc21)N(C1CC2CCCC(C1)N2C(=O)C1CC1)C c1(C(=O)NCCN(C(C)C)C(c2cccc(N)c2F)=O)ccc(F)cc1F C1(NC(CSC(=N)N)=O)COC2(C1)CN(C(c1cc(C(F)(F)F)on1)=O)C2 C1(NC(=O)NC2(c3cccc(Cl)c3)CCC2)CC2C(C1)C2(F)F c1(C(N(C2C(C)CCN(C(c3c(CC)ncs3)=O)C2)C)=O)n[nH]c2ccccc12 CC1CCN(C(C2CCSC2)=O)CCN1C(c1ccc(CO)c(F)c1)=O C1(NC(C=C(COC)C)=O)CC2C1CCN2C(c1nnn(-c2ccccc2)n1)=O Cc1cc(C(=O)NCC2CCN(C(=O)CCC3CC3(Cl)Cl)C(C)C2)cc(N)c1O N1(C(c2c(N)n(CCO)nc2)=O)CCC2C1CCCN2C(=O)C1=CCCS1 CC1C2CCCCC2CN1C(C1CC12CCN(C(=O)Cc1cn(C)cn1)C2)=O C1(NC(C2CC(OC)C2)=O)CCC(Cn2cc(C(C)(O)C=C)nn2)C1 c1(C(=O)NCCCCNC(CCCc2nc(C)sc2)=O)nccc2c1NCCC2 C(CC1c2ccccc2CCN1C(=O)CSC)NC(C1N(CC)C(=O)CC1)=O C1(C(C)(C)NC(C2CC2(F)F)=O)CCN(C(=O)CCc2ccccc2)C1 c1(C(=O)NC2CN(C(C(=CC3CCCC3)C)=O)C2)ccc(Br)cc1O C12CCCC3CN(CC13)C(=O)N2.CC(CCC1CCCC1)NC(=O)OC(C)(C)C c1(CCC(=O)NCCN(C(=O)CN2CCCNC2=O)CCC)cncc(F)c1 c1(NCC2CC(C)(COC)C2)ncnc2onc(C)c12 CCC(C(=O)NC1CC(NC(=O)Cc2c(Br)ccc(F)c2F)C1)C(C)(F)F C(=O)(C(CC(C)=O)NC(=O)CCOC)Nc1cccc(C(=O)OCC)c1 N1(C(CC(=C=C)C)=O)CCCC(N(C)C(c2csnn2)=O)CC1 c1(NCc2nnc(C)s2)cc(=NCC23CCCC2OCC3)[nH]cn1 c1(CN2CC(=O)N(CCc3nnn(C)n3)C2=O)nc2cc(F)c(F)cc2[nH]1 Cc1ccccc1C(C)C(=O)N(C)CC1COCCN1C(C1CC1(F)F)=O Cc1nncc(CNC(=O)CC2C3CCCC3N2C(=O)CC2(C)CCOC2)c1C C1(C(N(C2CN(C(=O)C(F)=C3CCC3)C2)C)=O)CCC(=O)N2CCCC12 C1(C(=O)NC2CC(O)C2)CN(C(c2ccc(Br)cn2)=O)Cc2cccn2C1 Cc1cc(-c2cn(CC3CCCN3C(=O)CCOC(C)C)nn2)sc1C N1(C(C2CC(N(C)CC)C2)=O)CCC2(CCC(NC(=O)CN3CC4CC4C3)C2)C1 Cc1nnn(NC(=O)C(Cn2cncn2)NC(C2CC2C2(C)COC2)=O)c1C CC1(C)CCC(=CC(=O)NCC2CN(C(C3(Cl)CC34CCC4)=O)CCO2)CC1 c1(OCCC)ccccc1C(=O)N(CC(O)CN(C(=O)C(C)(C)CC1CC1)C)C c1(-n2c(C3C(C)C3)nc(Cc3cccc(Br)c3)n2)cc(Cl)ccc1CO c1(C(=O)NCC2(C)OCCN(C(Cc3cn(C)nc3)=O)C2)cnc2[nH]nnc2c1 CC1=C(C(=O)NCC2CCCN(C(=O)CCc3ccoc3)C2)CCCC1 c1(C(=O)NCCCC(C)NC(c2c(OC)n[nH]c2)=O)nn(C)nc1C C1(c2c(OC)cccc2)(CN2CCOCC2)CN(N2CCOCC2C(C)C)C1 C1(C(=O)NCCC#C)CCC2(CN(C(c3cc(F)c(Cl)cc3C)=O)C2)O1 c1(C(=O)NC2CCN(C(c3c(C)cc(C(F)(F)F)s3)=O)C2)c(C)cc[nH]c1=N CC(C)(C)C#CC(=O)N1CC(CNC(c2ccc(NC3CC3)nc2)=O)C(O)C1 C(=O)(C1=CC2C=CC(C1)C2)N1CC(CC(C)NC(C(C(CC)C)NC=O)=O)C1 Cc1ccc(C(c2nnnn2C2COC2)NC2CC(=O)N(O)C2)c(C)c1C N1(C(=O)OC(C)(C)C)CCCC12CCCN(c1ccc(=N)[nH]c1F)C2 Cc1cc(C#N)ccc1NC(c1cnn(-c2ccccn2)c1C)=O N#Cc1cc(C(=O)NCC2CCN(C(c3cc(F)c[nH]3)=O)CC2)ccc1[N+](=O)[O-] c1(C(=O)NCC2CN(C(CC=CCC)=O)C(C)C2)cn(C)c2ncccc12 c1(C(N2CC(NC(C(CN(CC)CC)F)=O)(CO)C2)=O)cc2ncccc2o1 CC1(c2nn[nH]n2)CCN(Cc2csc(-c3cccc(C(N)=O)c3)n2)CC1 C1(C(C)C)C(C(=O)NCCC2CCC(C)(C)C2)CCN1C(c1ncccn1)=O Cc1nc(C(=O)NCCn2cc(CCc3ncccc3F)nn2)c(C)o1 c1(C(=O)NCC2CC(NC(C(C)N(CC(F)(F)F)C)=O)C2)c[nH]nc1C(C)(F)F c1(C(=O)OC)c(C)nc2ccc(C(N3CC4C5C=CC(O5)C4C3)=O)nn12 c1(CC2(CC)CN(C(=O)NC(c3ccc(Cl)cc3)C(C)C)C2)ccccc1NC N1(C(c2oc(C)c(Br)c2)=O)C2CCC1CC(CNC(C1CC1(C)C)=O)C2 C1(C(=O)NCCN(C(C(C)OCC2CC2)=O)CC(C)O)CCC(N(C)C)CC1 Cc1nc(Cl)[nH]c(=NCC2CN(C(=O)COCC3CCOC3)CCCO2)c1F C1(C(N2CCC(CNC(=O)CC3OCCO3)C2)=O)(OC)CC(CF)C1 c1(OC)nc(N2CCC2CNCc2nccnc2Cl)nc2[nH]cnc12 c1(CC(C)C)cc(C(=O)N(CCCNC(C2(C)CCCO2)=O)CCO)no1 N1(C(c2nc(OCC)sn2)=O)CCC(N(C(C2(C(C)(F)F)CCC2)=O)CC)CC1 C=CCC(CNC(=O)CN1CC=CC1)C(=O)NCc1ccc(OC)nc1 C1(NC(c2cnnc(O)c2)=O)COC2(C1)CN(C(=O)Cc1cscc1F)C2 C12(CNC(C(CC=C)(F)F)=O)CCCCC1CN(C(c1cc(OC)nn1C)=O)C2 C1(NC(c2c(CC)ocn2)=O)CN(C(C2(C)COC(=O)C2)=O)Cc2ccnn2C1 c1(NC(C2CC23CN(c2cc(C(F)(F)F)ncn2)C3)=O)ccnc(F)c1Br c1(CC(=O)NC2CC2CNC(c2nc(Cl)cs2)=O)coc(-c2cccs2)n1 C(=O)(C(F)C(C)(C)O)N1CC2C(CNC(c3c(C)oc(-c4cccs4)n3)=O)(C2)C1 c1(C(N2C(CNC(CCCNC(C)=O)=O)CCC2)=O)cccc2c1NCC(C)C2 Cc1nc(O)sc1C(=O)N(C1CN(C(=O)C(C)C(C)C)C1)C C(=O)(C1Cc2ccccc21)N(CC(C(=O)N1CC(n2cc(OCC)nn2)C1)O)C C1(C(N(CCOC)CC)=O)CCCCCN1C(c1cnncc1OC)=O C1(CNC(C2CC(C(C)C)OC2)=O)CCN(c2nc(C(=O)C(C)C)ns2)C1(C)C N1(C(C(C)(C)C2CCN(C(C3CCCC(=O)N3)=O)C2)=O)CCCC2(CC2)C1 c1(CNC(C(CSC)(C)NC(=O)COCCC(C)C)=O)ccc(C)c(O)c1 C1(CNC(C(C=C=C)C)=O)CN(C(c2ccn(CCCC)n2)=O)CCC1(F)F C1(NC(=O)C=Cc2ncc[nH]2)CC2CCC(C1)N2C(c1ccc(F)c(Cl)c1)=O N1(C(C(CC=C)(C)C)=O)CCC(N=c2cc(C)[nH]c(-c3cccs3)n2)C(C)C1 C(=O)(Nn1ccccc1=O)C1(CNC(C2CC(C)OC2)=O)CCCC1 CC(O)CCC(=O)N1CCCCC1CCNC(c1nsnc1O)=O c1(CC)cc(C(=O)NC23CCCN(C(=O)CC(=O)OC)C2C3)c2ccccc2n1 N1(C(CC(CC)CC)=O)CCCC1C(C)(C)CNC(=O)C(=O)NCC(F)(F)F N=c1[nH]cnc2c(C(N3CCC4(CC3)CC4CNC(c3cn[nH]c3)=O)=O)cnn12 c1(C(=O)NCC(C)CNC(C2(C(F)(F)F)CC2)=O)ccc2c(c1)CCCS2 N1(C(C(CCSC)N(C)C)=O)C2CCC1CC(NC(=O)CCP(C)(C)=O)C2 C1(NC(=O)C(N2CCC3(CC3)C2)=O)COC2(CCCC2)C1 C(CCC(O)C(=O)NC1CCC(F)CC1)NC(c1c(C)noc1)=O C(=O)(C(CO)C(C)(C)C)N1CCC(NC(COCCCCCC)=O)C1 C(C(C(=O)N1CCC1C(N)=O)C(C)(C)C)NC(c1cnc(C)o1)=O C1(COC)(NC(c2cnc(SC3CC3)cn2)=O)CCCN(C(c2occc2C)=O)C1 CC1(C)CN(C(c2cccc(Br)c2F)=O)CC1NC(c1ccncc1N)=O C(=O)(C(C)(C)C(=O)NC1(CNC(C2(OC)CCSC2)=O)CCCCC1)NC CC1(C)CN(C(C2CC3CCC2O3)=O)CC1CNC(c1cc(C(N)=O)ccn1)=O c1(CC)ncccc1C(=O)N(CCCCNC(=O)COC1CC=CC1)C C1(SC)CCC(CC(N2CCC(F)(CO)C2)=O)CC1.C12(CC1)C(=O)N2 c1(CCC(=O)NCC2CC(F)(CNC(=O)OC(C)(C)C)C2)ncccc1F c1(NC(C2COCCN2C(c2ccc(C3CC3)nc2)=O)=O)ccc(Br)nc1F c1(C(=O)NC2CCN(C(C(C)=C3CCC3)=O)C(C3CC3)C2)ccc(S(C)(=O)=O)o1 CC(CC(F)(F)F)(C(=O)OCc1cnccc1Cl)c1ccc(F)cc1 N1(C(CC2C(C)CCO2)=O)CCC2CN(C(c3cc(Cl)ncc3Cl)=O)CC2CC1 N(C1CCCc2n[nH]cc21)C(CCC1(C)CN(C(C2CC2(F)F)=O)C1)=O CC1(C)C(NS(=O)(=O)CC2CC(F)(F)C2)CC1CC(=O)O Cc1cc(C(=O)N(C2CCC3CC23)C)c(O)c(C)n1 C1(O)(CCNC(=O)Cc2nc[nH]n2)CCN(C(=O)CC2CC(=O)NC2=O)CC1 N1(C(c2ccn(CCCC)n2)=O)CC(C)N(C(=O)CCN2CCOCC2)CC1C c1(C(N2C(C)CCC(NC(COC)=O)C2)=O)cc(Cl)c(OC)cc1C c1(C(N(C2CCC(NC(c3cc(C(N)=O)no3)=O)C2)C)=O)ccnc(C(N)=O)c1 N1(C(CC=C=C)=O)CCN(C(c2cc3sc(C(=O)OCC)cc3s2)=O)CCC1C C1(CC(=O)NC2(CNC(=O)COC3CCCCC3)CC2)Cc2ccccc2C1=O C#CCC(C)C(=O)NC1CCC(N(C(c2ccc(COC)s2)=O)CC)CC1 c1(C(=O)NCC2N(C(CC(CCC)C)=O)CCC2CC)cc2ccccn2c1 c1(OC)ccc2c(c1)N(C(=O)CCC1OCCO1)CCN2C c1(C(=O)NCC(C)N(C(=O)C(O)C(F)F)C)ccc2c(c1)CCCC(=O)N2 c1(OC)ccc2ccccc2c1CN1CCC1C(=O)NC1CSC1 C(C1Cc2ccccc21)NCSCCC[Si](C#C)(C)C C(=O)(C(C)(Cc1ccc(Cl)cc1)NC(=O)C(c1cccc(C)c1)=O)OC N1(CCNC(c2c(C)snc2)=O)CCC(NC(c2cncc(N)n2)=O)CC1 CCCCC(C)C(=O)NC(C1CCCN(C(=O)CNc2ccccc2)C1)C C(=O)(C1COc2ccccc21)N1CC(C(=O)NCCNC(C2CCNC2=O)=O)C1 Cc1[nH]nc2c(C(N3CCCC(NC(=O)C(C)N4CC(C)C4)C3C)=O)cccc12 C1(CC(=O)NC2CCS(=O)CC2)CC(N=c2[nH]c(C(F)F)nc3ccccc23)C1 C1(NC(C(CC(C)C)NC(CCC(=O)NC)=O)=O)(OC)CCC(C)(C)C1 N1(C(C2CC3N(C(c4ccc(C)cc4)=O)C(CC3)C2)=O)CC(C2CCCCC2)C1 c1(N2C3CC(=O)NCC2CC3)nc(=NCCc2ncccc2F)[nH]c2c1COC2 C=CCC(C)(CNC(=O)C(c1ccoc1)NC(=O)C(F)n1ccnc1)CO N1(C(CCc2cc(C)on2)=O)CCC(N(CC(C)C)C(C2CC2Cl)=O)CC1 N1(CCC)CCCC(C(=O)NCC2CC(F)CN2C(c2cn(C3CC3)nn2)=O)C1 C(=O)(CC(C)CNC(C1(C)CC1(C)C)=O)NCCN1CC(OC)C1 N1(C(COCCOCC)=O)CC(N(C)C(C2CC3CCC2CC3)=O)C(C)(C)C1 C1(C(N2CC(CNC(CN(CCCCCC)C)=O)C2)=O)CC(C(C)=NO)C1(C)C C1(C)(CNC(c2c[nH]c(=NC)s2)=O)CN(C(C2(C)C=CCCC2)=O)CC1C Cc1nc(Sc2ccncn2)nc2ccccc12 C1(NC(c2ccc(SC)s2)=O)(CO)CCN(C(c2nc(C)ccc2C)=O)CC1 c1(C(N2C(=O)NC(CC(C)C)C2=O)C)ccccc1[N+](=O)[O-] c1(C(=O)NC(C(C)NC(C(c2ccc(C)cc2)OC)=O)(C)C)nn(CC)cc1Cl c1(C(N2CC(NC(c3sccc3Cl)=O)C(O)C2)=O)cc(F)c(F)cc1Cl C1(NC(c2ccc(C3CNC3)cc2)=O)CCCCC12CCCNC2 N1(C(C2CC(C)(CC)OCC2)=O)CCCC2(C1)CN(C(=O)Cn1cc(C)cn1)C2 c1(C(=O)NCCCN(C(=O)CCC(=O)NC)C(C)OC)cc(Cl)c(OC)c(Cl)n1 c1(C(N2CCC(N(C(=O)CC=CC(C)(C)C)C)CC2)=O)cc(F)c(CO)c(F)c1 N1(C(c2sc(C)c(O)n2)=O)CC(NC(=O)C(O)C2CCCC2)C2CCCC12 N1(C(c2cccc(CC=C)c2)=O)CC2CCN(C(c3cc(C)c(Cl)s3)=O)C2C1 Cn1cc2c(n1)CCCC2C(=O)NCC1(C)CCN(C(c2ncc(F)cn2)=O)C1 C1C(F)(C(C)C)C(=O)OCC(C)C(=O)N1.C(C)(C)(CC(=O)OCC)NCC c1(C(N(CC(CO)(CO)NC(C=C(C)Cl)=O)C)=O)cccc2ncsc12 N1(C(C2CN(C(C)=O)C2)=O)CCCCCCC1C(=O)NC1CCNC(=O)C1 N1(C(c2c(OC)scc2)=O)CCCC(C2(NC(C3COC4COCC34)=O)CC2)C1 C1(CC)CCCCCCN1C(=O)C(C)NC(C1CC(=O)C12CCC2)=O N1(C(CCC#CC)=O)CCCOC(CCNC(=O)C(F)C2CCCC2)C1 N1(C(CCCOCCC)=O)CC(C(F)(F)F)CC1CNC(=O)C(CC)SC C1(CC(=O)N(C2CCN(C(c3cnc(Cl)s3)=O)CC2)CC#C)CCCS1(=O)=O C1(OCC)CCCNS1(=O)=O.C12(CC(=O)NCC(=O)NCC)CN(C1)C(=O)O2 CCC(C(C)C)NC(=O)C#CCNC(c1cnc(C)o1)=O C1(N(CCOC)C(C2(C)CC2C(=O)O)=O)CCNCC1 C1(C(N)=O)CCCCN1C(=O)COC(C1CCN(c2cccc(F)c2)C1=O)=O C(=O)(C1=C(C)CCOC1)NCCCN(C(CCC(=C)C)=O)C CCCCCC(C)(C)C(=O)NC(C1CC=CCC1)C(=O)NCCc1cnn(C)c1 CCC(CC(=O)NCC(CNC(=O)Cn1cc(Cl)c(C)n1)S(C)(=O)=O)C(C)(C)C c1(C(=O)NCC(CNC(C(C)OC)=O)CO)ccnnc1O Cc1ccc(C(=O)NCC(C)(C)CN(C)C(C2CS(=O)(=O)C2)=O)cc1Cl C(CCCCNC(C1CN(CC(C)C)C1)=O)N(C(C(C)SC)=O)C c1(C(N2CCC(C(C)(C)NC(c3[nH]n(C)c(=O)n3)=O)CC2)=O)ccc(O)c(Cl)n1 N1(C(C2(COC)COC2)=O)CCC(C)C(NC(c2ccncc2C(F)F)=O)C1 C1(CC=C)(NC(c2cc(C3CCC3)on2)=O)CN(C(c2[nH]ccc2C2CC2)=O)C1 C12(C(C(F)(F)F)NC(=O)NC3C(CC)C3)CC3CC(CC(C3)C1)C2 c1(C2(NC(c3ccnc(OCC(F)(F)F)c3)=O)CCCC2)cccc(F)c1F N1(C(COCCSC)=O)CC2CC2C1C(=O)NCCC(O)CO c1(C(=O)NC(CCCNC(c2c(C)cco2)=O)C)cnc(CC2CC2)nc1O c1(C(=O)NC(CCOC)CNC(=O)CCC2CCOC2)c(C)cccc1O N1(S(=O)(=O)c2cccc(N3CC4CC3CN4CCF)n2)CCOc2c(Cl)cccc2C1 c1(C(=O)OC)cc(I)c(Cl)cc1NC(c1sccc1NC(c1c[nH]c(Br)c1)=O)=O Cc1ccc(C)c(OCC(N2CC(CC(=O)O)CC2C)=O)c1 C1(NC(c2cccnn2)=O)CN(C(c2snc(O)c2Cl)=O)CC2(CC2)C1 C1(CC)(COC)CCN(N2CCC3CCN(C)C(=O)C23)CC1 c1(OC)ccccc1C1CN(Cc2noc(C)c2Br)CCO1 c1(CN(C)Cc2snc(C)n2)cccc(Cl)c1Cl c1(C(N2CCOCC(NC(C3CC34CCSCC4)=O)C2)=O)cc(Cl)cc(F)c1F c1(CC)c(C(=O)NC(C)C(CO)NC(c2csc(C(F)(F)F)n2)=O)nnn1C C(CCCCC(=O)NCc1c[nH]nc1C(=O)NC1COCCC1(F)F)OCC CC1OCCC1CC(=O)NCc1cc(C(=O)NCCc2c[nH]nc2O)co1 c1(NCc2c(CC)nns2)ccc2ccccc2c1 C1(NC(CCC)=O)CCC2(CC1)CC(NC(c1cc(C)c(OC)c(C)c1)=O)C2 N1(C(COC)C)CC2CC1CN2C(C1CCOC(C)C1)=O c1(CC(C(=O)NC(C)CCCNC(c2cn(C)[nH]c2=N)=O)O)cc(Cl)cc(Cl)c1 N1(C(CCCNC(C)=O)=O)C2CCC1CN(C(C1COCC1C(F)F)=O)C2 C1(CNC(CCCN(C(C(C)CC2CC2)=O)C)=O)CCCOC1(C)C n1(CC(=O)NCCC2CN(C(=O)COC(F)F)C2)cnc(Br)c1 n1(CCCCNC(CCN(C(COCCC=C)=O)CC=C)=O)ccnc1C CCCC(C(=O)NC(C1(O)CN(C(=O)Cc2nc(C3CC3)cs2)C1)C)N(C)C C=C1CCN(C(=O)C(N2CCCCC2)C)C(C(=O)NCCc2c[nH]nc2C)C1 C1(NC(CCCCC=C)=O)CCN(C)C12CCCN(C(=O)CN1CCOCC1)C2 CC1(F)CCN(C(C2CC(CNC(C3CC34CCOCC4)=O)C2)=O)CC1 c1(NC(c2n(C(CC)(C)C)nnn2)C2CN(CC(F)F)C2)ccc2nccn2c1 n1(C(=O)NCCOCCC(=O)OC)cc(NCC2(n3cc(C)cn3)CCC2)nn1 C1(NC(CSCC(C)C)=O)CC2CN(C(=O)C(C)SC3CCOCC3)CC12 O=C(C1=CCSC1)NCC1(C(=O)NCc2nn[nH]c2C2CC2)CCCO1 c1(SCC(N2CC(NC(=O)C=C(Cl)Cl)(CO)C2)=O)nccc2ccccc12 c1(C(N2CCC23CN(Cc2c(F)cc(Cl)cc2Br)C3)=O)cccc2c[nH]nc12 N1(C(C2C(C)(CC)C2)=O)CCCC(NC(=O)CNS(N)(=O)=O)C1CC CCCCC(O)C(=O)NC1C2CC1N(C(C1CCN(C3CCSC3)CC1)=O)C2 c1(C(=O)NC(C2CCN(C(CSC)=O)C2)(C)C)cc(C(=O)OC)oc1C CCCC(O)C(=O)N1CCC(CNC(c2ccc(-c3nnc(O)o3)cc2)=O)C1 CC1OC2(C(=O)NC3CN(C(=O)Cc4cnccn4)CC3C)CCC1CC2 C(CC(C)(C)CC(=O)NCc1cnc(OC)cn1)OC c1(C(=O)NCCN(C(C2C(C)(C(=O)OC)C2)=O)CC2CC2)ccc(OC)c(OC)c1 CCCCCCC(CC)C(=O)NCC1CCN1C(C12CCC(CC1)C(C)O2)=O C1(NC(C(N2CCC(O)CC2)C)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CC1F C1(OC)CC(C(=O)NCC2CCC2NC(=O)CNc2ccccn2)N(C(C)=O)C1 C1(OC)CCN(C(C2(F)CCN(C(c3cncc(C)n3)=O)C2)=O)C12CCC2 c1(CNC(C2CSCN2C(=O)CC2CCCC2)=O)ccncc1Cl C=CCCCC(C)(C)C(=O)N1CC2CC2(C(=O)Nc2ccccc2CCO)C1 CC1=C(C(=O)NCC2CC(C)CN(C(=O)CCC3CCCO3)C2)CCC1 C1(CC=C)(C(=O)NCC(=O)NOC)CCCN1C(=O)CCC1CCCCO1 c1(CC)c(Cl)nc[nH]c1=NCC1(O)CCN(C(c2cnn3cc[nH]c23)=O)CC1 c1(C(=O)NCC(CC)NC(=O)C(O)c2cnc[nH]2)cc(OC)c(Cl)cc1Cl CCC(C)(C(=O)NC1CC2CCC(C1)N2C(=O)C=C(C)Cl)C(F)F c1(NC(c2c(C)nn(C)c2I)c2nnnn2C)cccc2c1OCCC2O C1(NC(=O)CCCc2cccs2)CN(C(c2cnns2)=O)CCC1CO c1(C(C(=O)NCCC(C)N(C(=O)C(C)=C2CC2)C)OC)ccccc1C(F)(F)F c1(OC)nc(C(N2CCC(OCC(=O)NCC(C3CCCC3)O)C2)=O)co1 CC1CC(C(=O)NCC2CCN(C(c3cnn(CCF)c3)=O)CC2O)CC(=O)N1 C1(CNC(CN(C2CCSC2)C)=O)N(C(C2SCCS2)=O)CCCC1(C)C N1(C(CCC=C)=O)CCC(C(=O)NCc2ccnc(F)c2)C(C)(C)C1 c1(N2CCCC(C)C2)cc(S(=O)(=O)NCCS(=O)(=O)N(C)C)ccc1C#N c1(CC(=O)NC2C(CNC(C3(COC)CCCO3)=O)C2)cccc(OC(F)F)n1 C(CC(F)F)(C(=O)N1CC=CC(O)C1)NC(CN=[N+]=[N-])=O.n1(CCCN)nccn1 N1(C(CC=C=C)=O)CC2CCN(C(c3scnc3C(C)C)=O)CCC2C1 N1(C(CN(C(C)C)C(C2Cc3nccn3C2)=O)=O)CCC(F)C(O)C1 CC(C(=O)O)C(C)(O)CNCC(=O)NC(=O)Nc1ccccc1 c1(C(N2CC(C(=O)Nc3cc(C)c(F)cc3)CC2(C)C)=O)cc2cccnn2c1 N1(C(C2(c3cc(C)no3)CC2)=O)CCCCC(NC(C2CSCCS2)=O)C1 C(=O)(C1=CCCCC1)N1CCC(C)(C(=O)NC(CCO)C(F)F)C1 CCC(C)CC(=O)C(=O)N1CCC1CC(N1CCCC(C)(C)C1)=O C#CC1CCN(C(C2COC(CNC(=O)C(O)C3CCCC3)C2)=O)C1 N1(C(CSC)=O)CC(C(F)(F)F)OCC1CNC(c1cc(C)c(C(F)F)cn1)=O C(=O)(CCC(C)=O)NCC1C(C(=O)NCC(COC)(F)F)OCC1 C#Cc1cnn(CC(N2CCC(C(=O)NC(C)Cc3cccs3)(CF)C2)=O)c1 C(=O)(C(C)(C)C(=O)NCCC1CCN(C(=O)Cc2cnc[nH]2)C1)OC c1(C(=O)NCCCC(C)(C)NC(C2C(=C)CC2)=O)c(C)ccc([N+](=O)[O-])c1C c1(OC)ccc(-c2cn(C3CCN(C(C4CC(O)C(F)C4)=O)C3)nn2)cc1Br c1(C(=O)NC(C2CCN(C(=O)Cc3sc(O)nc3O)C2)C)cncc(C2CC2)c1 c1(C(=O)NCCC2CCC(NC(=O)C3=COCCO3)C2)cccc2ccsc12 c1(C(N2CC(NC(=O)NCC)C2)=O)cc(CNC(c2csc(Cl)c2)=O)ccn1 c1(C(N2CC(NC(C3(OC)CC3)=O)C2)=O)ccnc(C)c1Cl C1(CCC)CCCN(C(=O)CCN(C(=O)CC2CCOC2)CC)CC1 c1(C(N2C(C(=O)NC(C#C)C)CC3CC32)=O)cc(Br)c(C)c(Br)c1 NS(=O)(=O)c1ccc(CCCNC(C2CC2c2cc(F)ccc2F)=O)cc1 N1(C(=O)NCc2nn(CC)c(O)c2)CCC2(CC1)CC(C(=O)OC(C)(C)C)C2 C(CCN(C)C(c1ccc(C)nc1O)=O)(C(C)(C)C)NC(CC(=C)C)=O c1(CN2CC(C)C(NC(=O)CCc3ccc(F)cc3)CC2)cccc2nsnc12 c1(CNC(C2CC(=C)C2)=O)n[nH]c2c1CN(C(=O)CCCOCCOC)CC2 Cc1nc(C)c(F)c(=NCC2C(C)CCCN2C(=O)Cc2nc(C3CC3)cs2)[nH]1 C1(CC)CCOCCN1C(C1CC2C(C1)C2(F)F)C(=O)NC C1(NC(CCCCCC)=O)(CNC(=O)CC(C)COC)CCC(F)(F)CC1 C(CO)(CCCCNC(=O)C=C1CC1)NC(CCOC(C)C)=O CN1CC=CCC1CC(N1CCC=CC1C(=O)N(C1CCCC(O)C1)C)=O CCC(O)C(F)(F)C(=O)NC1CC2(C1)CC(C(=O)NC1CC(=O)NC(=O)C1)C2 C1(C(=O)N(CCCCNC(=O)CCC2CCCCO2)C)(COC)CC(=O)C1 Cc1cncc(C(=O)NCC2C(C)CCN2C(c2cnn(C(C)C)c2)=O)n1 C#CC1(C(=O)NCCCN2CCC2)CCN(C(=O)CC2(COC)CC2)C1 C12(N(C)C(=O)NC3CCCN3CC3(c4ccccc4)CC3)CCC(CC1)CC2 N1(C(CSCCC(C)C)=O)CCCC1CN(C(C1CCCC1)=O)C1CC1 C1(NC(C2CC23CCOCC3)=O)(CO)CCCN(C(c2ccn3ccsc23)=O)C1 N1(C(C(C)=CC)=O)CCCC2(NC(c3cccn4nncc34)=O)CC2C1 c1(CN(C(=O)Cc2cncnc2SC2CC2)CCC2CC2)c(Cl)nsc1Cl C(=O)(C1=NNC(=O)CC1)NCC1CCN(C(C2C3CC(C)(C3)OC2)=O)C1 Cc1ccc(-c2noc(C(=O)N(C)C)n2)cc1F.N12CC(CC1CO)C2 C(=O)(CC(C)CCC(=O)N1CC=C(CNC(c2cccc(Cl)c2Cl)=O)CC1)OC C#CCCCCCCNC(=O)C(C)CNC(=O)CC1(O)CCOCC1 CC1CCN(C(=O)CC2(N3CCCC3)CC2)C1CNC(c1cc(Br)n[nH]1)=O C1(C(=O)OC(C)(C)C)CC(CO)N(CC(N2CCCCC2)=O)C1.c12cccn1C2 N1(C(CC#C)=O)CCCCC1CCNC(c1cncc(Br)c1)=O c1(NC(c2cccnc2Br)C)ncc(S(=O)(=O)NC2CCN(C)C2)cc1Cl N1(C(C(C)CN(C)C)=O)CC2(CNC(c3ccc(CC4CC4)o3)=O)CCC1C2 c1(C(=O)NC2CCN(C(c3ccn(C(C)C)n3)=O)C2)n[nH]c2c1CCOC2 C=CCC(CNC(c1cnc(=N)[nH]c1)=O)C(=O)NC(C)(C)CCF c1(C(C)C(=O)NC2CC2NC(=O)CC2=NNC(=O)C2)ccc2ccccc2c1 N1(C(Cc2n(C)ccn2)=O)CC(O)CC1C(=O)NC1CN(C(N)=O)C1 C1(NC(C2(CC=C)CCCCC2)=O)CC(NC(C2(OC)CCCC2)=O)C12CCC2 C1(CNC(C=CCC)=O)CC(NC(c2ccn(CC)n2)=O)C(O)C1 c1(OC)c(C(=O)NCC(CO)NC(c2ccc(C(C)(C)C)[nH]2)=O)cc(Cl)cc1C N1(C(CC2(OC)CC2)=O)CCCC2(C1)CN(C(=O)C(C)N=[N+]=[N-])C2 C=CCC(C)(C(=O)NC1(CNC(c2cc(OC)cc(C)n2)=O)CC1)N(C)C N1(C(CC2N(CC)CCCC2)=O)CCC2CC1CN2C(=O)CC(=O)OC C12(C(=O)NC(CCNC(c3cc(C(C)C)nn3C)=O)(C)C)CSCC1C2(F)F c1(C(=O)NC(CN(C(C(C=C)(F)F)=O)C)C)cncc2ccccc12 c1(C(=O)Nc2ccc(NC(c3cccc(C)n3)=O)cc2C)c(C)cc(O)cc1C Cn1cc(C(=O)NC2CCN(C(C3(C#N)CC3)=O)CC2)c(C(C)(C)C)n1 CCC(CCOC)C(=O)NC(C)(C)C(C)NC(=O)CN(C1CCC1)C C1(C(N2CCN(C3CCN(C(c4c[nH]c(=N)o4)=O)C3)CC2)=O)CC1C1CCCC1 Cc1cccc(NC(C2(NC(C3CC(=O)C3)=O)CCCC2)=O)c1 c1(C(N(C(CNC(c2cc(C(C)C)n(C)n2)=O)C)C)=O)nn(C)c2c1CSCC2 C1(NC(c2c(C)nc(O)[nH]2)=O)COCCN(C(=O)C=CSc2nc[nH]n2)C1 N1(C(C)=O)CCN(C(=O)Cc2cc(=O)n(-c3ccc(C)cc3)[nH]2)C2CCC12 CCC(CC)C(C)C(=O)NC1CC(C)CN(C(c2c(C)nn(CC)c2C)=O)C1 c1(C(N2CCC(OCC(=O)NC3(CCCCO)CC3)C2)=O)cc(O)nc(O)n1 C12(CNC(C(CC)F)=O)CCCC1N(C(c1ccc(Br)c(F)c1)=O)CC2 C(=O)(C(CC(F)F)NC(c1nccnc1N)=O)NC(C#C)CC(C)C C(=O)(C(CC(=O)OC)NC(C)=O)NC1CC(NC(COCCCC)=O)C1 c1(OC)ccc(C(N2CC(CNC(C3CCN3C(C)(C)C)=O)C2)=O)cn1 CC(F)(F)C(C)(C)C(=O)NC1CC2CC(NC(=O)C(=O)NCC(F)F)CC12 CC(C)CC(C)CN=c1[nH]c(N2CCOC(C(=O)N(C)C)C2)nc2cc[nH]c12 C(=O)(CCC1=CCCCC1)NC1CCC(CC(N2C(C)CCC2(C)C)=O)C1 C1(CN(C(c2cnc(CC(C)C)[nH]2)=O)C)CCCN(C(=O)CC2CCNC2=O)C1 CCS(=O)CC(=O)NC1CCN(C(c2cccc(C(C)(F)F)c2)=O)C1C(C)(C)C N1(C(C2(F)CN(Cc3ccncc3Cl)C2)=O)CCc2nc[nH]c2C1 c1(C(N2C(C)CC(CNC(c3cc4scnc4[nH]3)=O)C2)=O)ccc2c[nH]nc2c1 N1(C(c2ccc(C(=O)OC)[nH]2)=O)CC2CCCN(C(=O)CN(C)C(C)=O)C2C1 c1(C(N2C(CCC)CN(C(C3(CO)CCCC3)=O)CC2)=O)ccc2occc2c1 c1(CC)nc(C(=O)NCCC2CCCCN2C(=O)CC(O)C2CC2)c(N)s1 c1(C(N2CC3CC2(CNC2CN(c4n(C)ccn4)C2)C3)=O)cnc2n1CCC2 C1(CNC(C(CC)OCC)=O)(NC(=O)CCCSC(C)(C)C)CCCCC1C N1(C(c2c(C)c(Cl)ccc2)=O)CCC(NC(=O)CC2CCCCO2)C(CO)CC1 C1(C(N(C2CCN(C(CCc3c(C)nn(C)c3)=O)C2)C)=O)OCCN(C)C1=O c1(C(N2C(CN(C(CC3C(CC)C3)=O)CC)CCC2)=O)cccn2ccnc12 C1(CC(N2CCC(N(C(=O)CCF)CC)C2)=O)CCCCN1C C(C(C)(C)C1=CCCC1)NC(CC1CC(C)N(C(=O)CC2=CCCC2)C1)=O C(C)(CO)(C(=O)N(C)CCNC(C1CCC(O)C1)=O)OC c1(C(C(=O)NCc2ccc(F)cc2)N(C(CC)C#N)C)nc(Br)ccc1OC CC1OCCC1(C)C(N1CC(OCCNC(=O)Cc2ccnc(O)c2)C1)=O c1(N2CCN(C(c3c(C(C)C)nns3)=O)CC(O)C2)ncnc2c1SCCC2 N#Cc1cn(Cc2ccco2)c(=O)n(C(=O)COC2CCCCC2)c1=O N1(C(CCC2(C)CC2)=O)C2CCC1CC(NC(=O)CC13CCCC1C3)C2 C(=O)(CCC(C)S(C)(=O)=O)NCC(C)(C)NC(CC(COC)C)=O Cc1cccc(C)c1-n1cc(C2CCCCN2C(=O)CC(C)C(C)C)nn1 N#Cc1cc([N+](=O)[O-])ccc1CN1CCN(S(=O)(=O)c2ccc(Cl)s2)C(C#N)C1 C12(NC(=O)CCSC(F)(F)F)CCCN(C(=O)Cc3cnoc3)CC1C2 CC1SCCC1(c1nnnn1CC1CC1)NCCCc1cccs1 CC1CC(O)CCN(C(C2CCCN(C(C3C4CN(C)CC34)=O)C2)=O)C1 C1(CC(=O)NCCOCC(=O)NC(CCC=C)C2CC2)CCCC(O)C1 N1(C(C(CC)N(CC)CC)=O)CCC(C2N(C(=O)C(C)CO)CC2(C)C)CC1 CC(c1cnn(C)c1)=CC(=O)NC(C)CNC(c1cn(C)c(C)n1)=O C1(C)(C(=O)NCC2(CCNC(c3c(C)n(C)cn3)=O)CC2)CCC(F)(F)CC1 Cc1cc(C(=O)NCC(C)(C)CNC(C2(N(C)C)CCCSC2)=O)c(F)cc1Cl C1(NC(CCCCC)=O)CCCCCN(C(=O)CCc2ccncn2)C1 C1(NC(CCSCCC)=O)CCN(C(c2ccccc2C)=O)C12CCC2 C(=O)(CC(O)CC(C)(C)C)N1CCN(C(CCCc2ccc(C)cc2)=O)CC1C c1(OCC(F)F)ccccc1C(c1nnnn1C1CCC1)NC1CC2(CCC2)C1 c1(NCC2(NC(C(CC(CC)C)C)=O)CCCC2)nc2c(cc1C#N)CCCC2 c1(C(=O)NCC(CNC(Cc2ccc(C)o2)=O)F)ccc2ncccn12 N1(C(CC(C(=C)C)OCC)=O)Cc2occ(C(=O)NOCC=CCl)c2C1 CCC(C)C(O)C(=O)NCC1(c2ccccc2)CCN(C(C2CC2F)=O)CC1 N1(C(C(CSC)C)=O)CCC2(C=C(C(=O)NCc3cc(C)ns3)C2)C1 CCC(CCOC)C(=O)NCCC1(O)CN(C(=O)COc2cc(C)cc(C)c2)C1 CC1(C)CCC(NC(C2COCCC2NC(=O)Cc2cncs2)=O)C1 c1(C(=O)NC(C)C(c2cccc(Cl)c2)C)ccc2cc[nH]c2n1 C1(C(N2CCC(C)(NC(C(C)c3ccco3)=O)C2)=O)CCc2ncnn2C1 C1(COC)CN(C(=O)C(C)O)CCN1C(c1[nH]nc(OC)c1Cl)=O c1(NC2CCN(c3ccc(C)cc3)C2)cc(C#N)ccc1OC(F)F C(C)(N=c1nc2sccc2c(NCC2(CCO)CCOC2)[nH]1)c1ncc(C)cn1 c1(NC(c2nccc(OC)c2)c2nnnn2C(C)C)ccc(Cl)c(F)c1 c1(C(N2CCN(C(C(C)OC(=O)C3CC3)=O)CC2)C)c(F)cccc1Cl C(=O)(C(C)(C)S(C)(=O)=O)NCC(CCOC)NC(C12CCC(CC1)O2)=O Cc1ccc(SCC(N2CCC(CNC(c3occ4c3CCC4)=O)C2)=O)c(C)c1 c1(CCC)cc(C(N2CCC(C(C)(C)C)(CNC(C3CC(=O)N3)=O)C2)=O)nn1C c1(CC(=O)NCC2CC(NC(=O)C3=C(Cl)CC3)C(O)C2)ccc(C(F)F)c(F)c1 c1(CC(N)=O)ccccc1C(=O)NCC1(O)CC(CNC(=O)C#CC2CC2)C1 C1(NC(CNS(N(C)C)(=O)=O)=O)CC2CC1N(C(=O)CC1CN3CCC1CC3)C2 CN1C(=O)CCC1C(N1CC2CC1C2NC(C1(C)CCCS1)=O)=O C1(C(=O)NCC=C2CCN(C(=O)CC(C)(C)O)CC2)(OC)CCC(C)C1 c1(CC(=O)N(C2CCCN(CC(C)CS(C)(=O)=O)CC2)CC)ccc(F)cc1Cl C1(NC(C2C=CCN(C(=O)CCc3nc[nH]n3)C2)=O)CCCC2(CC1)CC2 CC1(C(=O)NCc2ncoc2C2CN(C(c3c[nH]c(C(N)=O)c3)=O)C2)C=CCC1 C#CCCCC(C)C(=O)N1CCN(C(c2occc2COC)=O)C(C)C1 N1(C(C(C)OCCC(C)C)=O)CCCN(C(C2CC3CCC2O3)=O)CC1 N1(C(c2ccc(Cl)cn2)=O)CC2CCN(C(=O)COC3CCCCC3)C2C1 C(=O)(C(C#N)C(C)(C)C)N1C2CC(NC(c3cc(CC)no3)=O)C1CC2 c1(C(N2CCC(CN(C(C(c3ccccc3)C)=O)C)C2)=O)cccc(O)c1F C(=O)(CC(C)C(C)(C)C)N1CCC(C(=O)NCc2c(OC)nn(C)c2)CC1 c1(CC)ccc(C(=O)NC2CCC(CCNC(c3sccc3OC)=O)C2)c(F)c1 N1(C(C(C)S(C)(=O)=O)=O)Cc2ccccc2C(CNC(=O)C2=NOCC2)C1 n1(CC(=O)NCC2OCCN(C(C(CC)(C)OC)=O)C2)ccc(=O)n(C)c1=O Cc1nn(C(C)(C)C)cc1C(N1CCC(NC(=O)C=Cc2cc[nH]n2)C1C)=O C(=O)(CCC(=O)N1CC(CNC(C2(C)CCNC2=O)=O)C1)NCC C(=O)(C1=C2CCCN=C2NN1)N(C)CC1CCN(C(C2CCCC(C)C2)=O)CC1 C(C)(C(C(=O)Nc1cnn(CC)c1)C(C)C)NC(CCC)=O c1(NC)ccccc1OC.c12ccc(o1)C(C(=O)NC1CCC1C)N2C C1(N(C(=O)C(CC)N(C)CC)CC#C)CCN(C(c2cnc(Cl)s2)=O)CC1 C12(NC(C)=O)CCN(C(c3ncc(Br)cn3)=O)CC1C2 CCCCC(CC(=O)NC1CC(C(C)O)C1)NC(C1(CO)CCCC1)=O C(CC(F)F)(C(=O)NCC1CC12CCCCC2)N(C(c1c(C)[nH]cc1)=O)C c1(-c2nc(C(C)O)nn2C2CCCOC2)ccc2ncn(C)c(=O)c2c1 C1(O)(CC(=O)NCCN(CCOCCCC)CCOC)CCCCC1 C1(CC(NOCCOCC)=O)CCCCN1C(=O)CC1CCOCC1 C12COCCN1C(=O)C=CCC1(CC1)NC(=O)C2.c1(CC)ccncc1N c1(CC)nc(C)c(C(N2CCCC2(C)C(=O)N(CC)CC2(O)CCC2)=O)o1 O=C(C1=CS(=O)CCC1)NCC1(O)CN(C(C2CN(CC3CCCCC3)C2)=O)C1 C(CC(=O)N=c1ccn(C)[nH]1)C12CN1C2.C12(OC)CCCC1C2(F)F C(C(CC(=O)NC1CC(C)(NC(c2ccc3nn[nH]c3c2)=O)C1)C(F)F)N(C)C C1(C(=O)NC2(CCNC(C3CCC=CCC3)=O)CCOCC2)CC2C(C1)C2(F)F C1(CC)CCCCC1C(=O)NCCOCCOCCNC(c1n[nH]c(C)n1)=O C1(C#N)(C(=O)NCC(CNC(c2cccc(OC)n2)=O)OC)CC2(CCC2)C1 CC1C(NC(C2(C)CCCCC2)=O)CCN1C(C1CCC1CF)=O C1(CNC(C(c2cccnc2)NC(CNC(N)=O)=O)=O)CC2(CCC2O)C1 N#CC1CCN(C(=O)COC2CCN(C(=O)CC3CCC(=O)N3)C2)C1 N1(C(C2CCC(=O)NC2)=O)CC2CC(CNC(=O)Cc3ccc(O)cn3)C2C1 NC(=O)C(F)(F)CNC(=O)CNC(c1cn(CCO)nn1)=O C(=O)(C(F)CCC(=O)O)NCCC1(CC(=O)OCC)CC1 c1(NC(C2CCN(Cc3noc(C4CC4)n3)C2)=O)cc2c(-c3nn[nH]n3)cccc2[nH]1 C1(CNC(C(CC)NC(N)=O)=O)CC2CCC(C1)N2C(=O)CC(C)(C)OC C12(NC(CCCCCCC)=O)COCCC1CN(C(c1ccoc1C)=O)C2 N1(C(CNCC2C(CC)C2)=O)CCCN(C(C)=O)CC1 c1(C(C)(C)C)cnc(CCC(=O)NCC2(NC(C3CSCCS3)=O)CCOC2)o1 c1(C(N2CCC(C(C)(C)NC(=O)Cc3cc[nH]c3)C2)=O)ccc(C2CC2)nc1 c1(C(=O)NCC2N(C(C3(CCOC)CCC3)=O)CC2)cn(C)c(=O)cc1C N1(C(=O)CC(F)F)CCC=C(c2cccnc2)C1.c1(-c2nccs2)ccc([N+](=O)[O-])nc1 C1(CC)(NC(c2cnsc2C)=O)CCN(C(c2c(C(=O)OC)cnn2C)=O)CC1 C#CCCCC(C)C(=O)NCCCCCCN(C(=O)C=CC(C)(C)C)C C1(C(N)=O)CC2(CCN2C(=O)CN(C(=O)C(F)C(C)(F)F)C2CC2)C1 Cc1cnc(Cl)c(S(=O)(=O)NC2CN(C(c3cc(Br)c(C)s3)=O)CC2F)c1 c1(CCC(=O)NC(CC)CNC(=O)C(CO)N(C)C)n[nH]c2c1CCCC2 CCCCCS(=O)(=O)CC(=O)N1CCCN(C(c2ccc(Cl)c(C)c2)=O)CCC1 CCC(C)(C)CCCC(=O)NCCC(C)N(C(=O)Cc1cc(C)cs1)C Cn1ncc(C(N2CCOCC2CC(=O)NCC2=CCCCC2)=O)c1Cl c1(C(=O)NC2C(OC)CN(C(=O)CN3CCC(C)C3)C2)c(C)cncc1F c1(C(=O)NC2CCC(C(=O)Nc3ncc(F)c(Cl)n3)OC2)c(Cl)cnc(Cl)c1Cl C(=O)(CCCC1CCC1)NC(C(=O)NC(C)Cc1ccco1)C1CCC1 CC1(C)CN(CCOc2cc(Cl)cc(Cl)c2)CCC1O CCC(C(=O)N1CCN(C(c2c[nH]c(=N)s2)=O)CC1CO)C(C)(F)F C(=O)(CC(C)(C)C(F)F)N(CCOCCCNC(c1cnc(CC(C)C)[nH]1)=O)C CC(C)C(C)(CNC(c1ncc(Br)cn1)=O)NC(=O)CC(=O)OC(C)(C)C S(=O)(=O)(c1cccnc1NC1CCCCC1C(F)(F)F)NCC(CN(C)C)(C)C c1(C(=O)NCCN(C(c2n(COC)ncc2)=O)C(C)C)nccnc1C(=O)OC C(=O)(C(C(C)(C)O)NC(c1cnn2c1CCC2)=O)NC(c1nccs1)C N1(C(C2C(C=C)C2)=O)CCN(C(c2cccnc2-c2ccc(C)o2)=O)C(CC)C1 C=Cc1ccc(C(=O)NC23CC(C(=O)NC(CCC)CCCC)(C2)C3)cc1 S(=O)(=O)(c1ccc(=NCCc2ccns2)[nH]c1)NCCN(CC(F)F)C c1(C(N2CC(O)CC(NC(CS(=O)(=O)NC)=O)C2)=O)ccnc2cc(F)cnc12 c1(OC)c(NC(C2CN(Cc3cc(Cl)ccc3O)CCS2)=O)cccc1F c1(C(N2C3CCC2CC(NC(=O)C(F)(F)C(F)F)C3)=O)cnc2ncccn12 Cc1cn(C)nc1CC1(O)CN(C(C2CCN(Cc3cn(C4CC4)nn3)CC2)=O)C1 Cc1cc(NC(=O)CCc2cnn(C)c2)ccc1NC(=O)CC1CCC1C C1(C(C)C)CC(NC(=O)N(CC(O)C(F)(F)F)C(C)C)CCO1 C1(NC(=O)Nc2nccc(CC)c2)CCc2nnc(Cc3ccccc3)n2C1 CC(CCC(C)(C)C)C(=O)NC1(C(N2CC(OCCO)C2)=O)CCSC1 C(=O)(CCCCCCN=[N+]=[N-])NCC1N(C(C(CCC)N(C)C)=O)CCCC1 N1(C(CN(C(C(C)N(C(C)=O)C)=O)CCO)=O)CCN(C(=O)CSC(F)F)CC1 C1(C)(CNC(c2c(CC)oc(C)c2)=O)CN(C(=O)CC2C=CS(=O)(=O)C2)CCO1 c1(C(C(=O)NCCCNC(=O)CC2CC=CC2)(F)F)cccc(Cl)c1 N1(C(C23C(CN(C(c4cccc(C)c4F)=O)C2)C3)=O)CCCCC(F)(F)C1 N1(C(CC(C)C2CC2)=O)CCCC(C(=O)NCC(C)OC2CCCC2)CC1 C(=O)(C1=CCC(C)CC1)N1CCN(C(C2CCN(C(C)=O)CC2)=O)C(CCO)C1 c1(C(N(CC(C)NC(C(C)O)=O)C)=O)cccc(OCF)c1 C1(CNC(C(CC)SC)=O)(NC(=O)C=Cc2cnn(C)c2)CCCCC1 C(=O)(N=c1[nH]n(-c2ccccc2)cc1C#N)c1cnn(CC)c1NC(=O)C(N)=O c1(C(=O)OC)c(Cl)nc[nH]c1=NCCC1CCCCN1C(=O)CC1CCOCC1 c1(NC)cnccc1C(=O)NCc1cc(C(=O)NCC2CCC3(CC3)C2)ccn1 Cc1cccc(N)c1C(N1C2CCC1C(CNC(=O)CCF)C2)=O C1(NC(c2c(C)cns2)=O)CCOC(C(=O)NCCS(N)(=O)=O)C1 c1(CC)cc(NC(C2(CNC(=O)CN3CSCC3=O)CC23CCC3)=O)ccc1F C1(OC)CC(CCNC(c2c[nH]nc2C(C)C)=O)N(C(=O)C(C)c2cccs2)C1 c1(C2CCN(c3ccnc(NCC4(C(C(C)C)O)CC4)n3)C2)cc(F)cc(Cl)c1 C(=O)(CS(=O)(=O)c1ccccc1C)NCC(CNC(C1CC(C(=O)OC)C1)=O)O C1(C)(C(=O)NC2C(NC(c3cc(COC)on3)=O)CCC2)CCNC(=O)C1 CCCC(CC)N=c1cc(C)[nH]c(=NCc2cc(C)cs2)[nH]1 C1(C(C)NC(CNC(C2(C(C)(C)CCCl)CC2)=O)=O)CCC(CO)CC1 CCCCC(C)NC(C1CCN1C(c1cncnc1)=O)=O c1(C(=O)NCC23OCC(CNC(C(C(C)C)(C)O)=O)(C2)C3)sccc1S(N)(=O)=O C1(C(N(OC)C(C)C)=O)CC2CCCC2N1C(c1n[nH]c2cccnc12)=O Cc1ccc(C(C)C(=O)NC2(CNC(c3c(Br)noc3C)=O)CC2)cc1 c1(C(C)(C)NC(C2CCCN2CCSC2CCC3CC23)=O)nnnn1C1CCC1 c1(C(=O)NCC(C2CC2)NC(C(CC=CC)C)=O)cc(C(C)(C)C)n(C)c1C c1(CNC2C(C)CN(C(=O)C(c3cnn(C)c3)=O)C2)ccc(F)c(O)c1F CCC(C)CC(C)C(=O)N1CC(CN(C(=O)CN(c2ccc(Cl)cn2)C)C)C1 c1(C(=O)Nc2cc(C)nn2-c2ccccn2)cnn2cccc2c1 C1(OCC(C)C)CCN(C(c2csc(Br)n2)C(=O)NCC2CCCO2)C1 CC1CN(C(=O)C(F)(F)C(O)C2CC2)CCC1CNC(=O)CSC(C)(C)C C#CCCCC(C)C(=O)NC(CC(C)(C)C)C(=O)Nc1ccc[n+]([O-])c1 c1(OC)ccc(CC(O)CN2CCCCC2C2CC2)cc1 c1(C(=O)NCC2CCC2NC(C2CCC(=O)N2C2CC2)=O)cccc2occc12 CC1(C(=O)NCCNC(=O)CC2CCCCO2)COC(=O)N1 N1(C(c2cc(CC)nn2C)=O)CC2CC(NC(=O)CC3CCC(O)C3)C2C1 N1(C(c2csc3ccccc23)=O)CC(CO)C2(C1)CN(C(C13COCC1C3)=O)C2 C1(C(C)(C)NC(COCC(=O)OC)=O)CCN(C(=O)Cc2cc[nH]n2)C1 C1(O)(CCNC(=NCC)NCCOCCF)CC2CCC1C2 C=Cn1nccc1C(=O)NCC1CCCCN1C(c1cnn(CC(F)F)c1C)=O S(=O)(=O)(c1cccc(=NCCC2CC=CC2)[nH]1)N(CC(C)C)CC1(CC(C)C)CC1 C1(C(N2C(C(N3C(CN(C)C)CCC3)=O)C(O)CC2)=O)CCCC(=O)CC1 C12(C(=O)OC)CC(CNC(=O)Nc3cccc(OC)c3C)(C1)OC2(C)C C(=O)(CCN=C(NCC(C(C)(C)C)OC)NCCc1cc2ccccc2o1)NC C(=O)(C1=NOC2COCC12)N1C(C)CC(NC(C2CCNC2=O)=O)CC1 Cc1ccsc1CCCC(=O)NCCN(CC(C)O)C(=O)C=CC(=O)N(C)C N(C1c2ccccc2CC1NC(c1ccc(C2CC2)o1)=O)C(C1C(C)CCO1)=O N1(C(C(C)SC)=O)CCC2(CCN(C(c3cc(N)ccc3Cl)=O)C2)C1 C1(CC(=O)NC(CC(C)NC(CN(CCC#C)C)=O)C)C(=O)ON=C1C CCCCCCCCCCC(C)NC(=O)Nc1cc(Cl)cc(Br)c1F C1(c2ccccc2)(NC(C(C)SC(C)C)=O)CCN(C(=O)CCF)C1 n1(CC)c(C)cc(C(=O)NC(CNC(=O)CC23CCC(CC2)C3)CCOC)c1C C(c1ccncc1)=C(C)C(N1CCOC(CN(C)C(C2CC2C(F)(F)F)=O)C1)=O C1(NC(C(C)CC2CC2)=O)(CO)CCN(C(c2coc(CO)c2)=O)CC1 c1(C(CC)C(=O)N2CC(NC(c3ccc(CN(C)C)o3)=O)C2)ccc(F)cc1 C1(NC(c2c(C)cc(C)o2)=O)CC12CCN(C(=O)C(N1CCCCC1)C)C2 N1(C(c2cc(Cl)ccc2C(F)(F)F)=O)CCn2ncc(C3=CCCC3)c2C1 c1(C(N2CCCC(NC(c3cc(O)ccc3Br)=O)CC2)=O)ccc2sccc2c1 N1(C(CN2CCN(C)CC2)=O)CCN(C(=O)CCS(C)=O)C2CCC12 N1(C(C(C)Cc2ccnn2C)=O)CCN(C(=O)CSc2cn[nH]c2)CC(C)(F)C1 N1(C(c2cccc(Cl)c2)C(=O)NC2COC2)CC(O)C2(CCCC2)C1 c1(C(=O)NCC=CCNC(c2c(C)cccc2F)=O)[nH]nc2ncccc12 c1(NCC2N(C(=O)OC(C)(C)C)CC2)cc(CO)no1 c1(OCC)cc(=NC(=O)CC(=O)N2CCC3(CC(O)c4ccccc4O3)C2)[nH]o1 CC1CN(C(C2C(C)(C)C2(C)C)=O)CC(C)C1NC(c1cc(Cl)c(Cl)s1)=O C1(C(CC)C)CCCN1C(=O)C(C)N(C(=O)CCNC(=O)CO)C1CC1 N1(C(c2nc(COC)oc2)=O)CC(C)(C)CC1CNC(=O)CC1CCC(C)CC1 c1(C(N2CCC(CCNC(C(C)CC(N)=O)=O)C2)=O)cnn2c1CCCC2 C1(CC)(NC(=O)CC(C)N(C)C)CCN(C(=O)Cc2cc(C)ccc2F)CC1 C1(CNC(C2CCSC2)=O)CC(N=c2[nH]c3cccc(F)c3s2)C1 N1(C(C#CC(=O)N(C)C)=O)CC(C2(NC(C3CCCNC3=O)=O)CC2)C1 c1(C(N2CCC(CNC(CCCCCSC)=O)C2)=O)cc2n(n1)CC(C)NC2=O N1(C(CCCC=C)=O)CC2CN(Cc3ccc(O)c(C)c3)C2C1 c1(C(=O)NCc2c(C)nc(F)cc2)n[nH]c2c1CN(C(C1(C)CCOC1C)=O)C2 N1(C(C(CC(C)C)OC)=O)CC2CC(C1)C(CO)C2NC(=O)Cc1nc[nH]n1 CCCCCC(C)(CC)C(=O)NCCCCCCn1cc(CC2CCCC2)nn1 N1(C(CC(CC)CC)=O)CC2(CCC2)CC1CNC(c1c(C)ccc(C)c1C)=O C=CC(C)(O)CC(=O)N1CCCC(CN(C(c2ocnc2CC)=O)CC)C1 C1(CC(=O)NC(C(=O)OCC)C)CC2(C1)CN(C(=O)CN(C)C(=O)C1CC1)C2 CCCCC(C)(C)NCC(c1cn(CCOC)nn1)CC C(=O)(N=c1cnn(C2CCC2)[nH]1)c1cccc(CN(CC)Cc2ccccc2)c1 C=C=CCCC(=O)NCCC(=C)CNC(c1occc1Br)=O c1(CNC(c2cn(CCF)nn2)=O)ccccc1CNC(c1ccc(O)cn1)=O C1(NC(c2cnc(C(C)C)nc2)=O)CC(C)CN(C(c2cc(Cl)ccc2N)=O)C1 C=CCCCCC(=O)NC1(C(=O)NCCCC(=O)N(C)C)CC1(C)C C=C(C)CC(C(=O)NC(C)CCC(=O)NCCc1ncoc1C)OC Cc1ccc2c(c1)CC(C(=O)OCC1CCCN1)S2(=O)=O CC1=C(C)CC(C(=O)NC2CN(C(=O)Cn3cc(C4CCC4)nn3)CC2C)CC1 CC1(C(c2ccc(Cl)cc2)c2csc(CNC(F)(F)C(F)(F)F)n2)CC(F)(F)C1 c1(SC)nc(C)c(CSCC(=O)NC(c2ccccc2C)(C)N)s1 c1(C(N2CC(NC(C(C)OCCOCC)=O)C2)=O)cc2c(nc1O)CCOC2 N1(C(CNC(N)=O)=O)CC(C2CC2)(C(N2CC(O)(c3nn[nH]n3)C2)=O)C1 N1(C(C=C(C)C(F)F)=O)CCOC2CN(C(c3cc4[nH]ccc4s3)=O)CC12 c1(-c2cnc(NC(c3cccc(OC)c3O)=O)c(O)c2)cccc2c1OCC2 C(=O)(C(O)C(F)(F)F)NC(CC(N1C(CNC(C)=O)CCC1)=O)C1CC1 c1(C(=O)NCC2C3CN(C(c4ns[nH]c4=O)=O)CC23)cncc2sccc12 N1(C(CCC(=O)NC)=O)CCCC(OCCNC(CCOCC)=O)C1C N1(C(CC(=C)Br)=O)CCN(C(c2nnccc2C)=O)C(C)C1C C1(NC(c2c(C)nsc2C)=O)CC2CC(C1)N(C(C1CN(C3CCCCC3)C1)=O)C2 S(=O)(=O)(c1cc(C2OCCO2)cs1)NCCNc1c(C)noc1-c1ccccc1 c1(CC(=O)N(CCC(C)NC(CSCC)=O)C)nc(Br)n(C)c1C C1(CC(=O)NCC2(NC(CCc3cc(C)[nH]n3)=O)CCCC2)CCCCC1(C)C c1(CC)cccc(-c2nc(C(O)CC)nn2-c2cccc(OC)c2)n1 C1(C(N2CC(NC(=O)C(c3ccc(Cl)nc3)(F)F)CC(F)C2)=O)CN2CCC1CC2 C(N=c1[nH]c(N2CC3CC2C(F)(F)C3)nc2cccnc12)c1scc(C)c1 Cc1c(CCC(N2CC(NC(=O)C(C)C3CC3)C(O)C2)=O)cnn1C c1(NC(CC(CCC)NC(=O)OC(C)(C)C)=O)ccc2ccn(C)c2c1 CC1(C)CC(NC(=O)CC(CNC(=O)Cc2cncs2)C2CCC2)C12CC2 Cc1cc(CNC(C2(CC(C)C)CCN(C(=O)C(C)OC(C)C)C2)=O)cc(F)c1 c1(C(N2CC(NC(C(C)(CO)OC)=O)C(C(F)(F)F)C2)=O)cccn2nccc12 C(=O)(CCC(C)(C)C#N)N1CC(CC(=O)N(C2C3CCCC23)C)C2(C1)CC2 N1(C(C(CC)C2CCOCC2)=O)CCN(C(C2(C#N)CC2)=O)CC(C)C1 N1(S(c2c(C)nn(C)c2)(=O)=O)CCC(C2CCCN(C(=O)CN3CCCC3)C2)C1 C(=O)(C1=C(C2(C)CC2)N(CC(=O)O)C(=O)NC1c1ocnc1C(F)(F)F)OC Cn1cnc2c1C(C(=O)NNC(=O)c1ccc(OCC(F)(F)F)cc1)CCC2 C1(C)(COC)CC(NC(=O)C=CSC)CN1C(c1oc(C)nc1C)=O c1(C(=O)NC2C(NC(CC=C=C)=O)CC2)ccc(C#N)c(Cl)c1 c1(C(=O)NCC(CC)N(C(=O)CC2CSCCO2)C)cn2ncccc2n1 C1(c2nnnn2CC2CCCO2)(NC(CC(C)(C)C)C)CCC=CCC1 c1(-c2ccc(CC)o2)nc2ccc(C(=O)Nc3ccc(C#N)o3)cc2[nH]1 CCCC(CCC)CC(=O)NCC(CO)NC(=O)CCOc1ccc(OC)cc1 CCCCCCCC(=O)NC1CC(C(=O)N(CC(=O)OC)C)=CC1O c1(C(=O)NCC2(C(=O)NCC3CCN(CC)CC3)CC2)cc(F)cc(Br)c1F C1(C(=O)NC(CC)COC)CC2CCCC2N1C(C1CC(=O)N(C)C1)=O C1(NCCCC)CCCN(N(C)C(C)CCC)C1 c1(C(N(c2nc(SC)c(Br)cn2)C2CCNCC2)=O)cc(Cl)cc2nc[nH]c12 C12(CNC(C3C(C=C)C3)=O)CCC(NC(=O)CC3(NC(C)=O)CC3)(CC1)CO2 c1(CN(C(C)C(=O)NCC(F)CNC(c2ccccc2)=O)C)ccccc1 c1(CN(CC(=O)O)C(C2CC2C(=O)O)=O)cn(CC(F)F)cn1.c12cn-1nn2 c1(OC)ccc(C(N2CC(CNC(=O)CCc3cnc(C)s3)C2)=O)cc1C1CC1 N1(CC(=O)NC2(C3CN(C(=O)CC=C(Cl)Cl)C3)CC2)CCCCC(O)C1=O c1(C(N(CCOC)CCNC(=O)Cn2cccn2)=O)c(F)cc(C)cc1F C12(C(N3CC(COC)C3(C)C)=O)COC(C1)C(NC(c1c(C#N)ncn1C)=O)C2 c1(OC)oc(C)nc1C(=O)NC(C1CN(C(=O)C2=C(C)CC2)CCO1)C CC1(C)CCN(C(=O)C(C2CC2)C2CC2)C1C(=O)NCC(Cl)Cl C1(C(=O)NCCCCC2(NC(c3cnc(N(C)C)s3)=O)CC2)CC2(C1)CC(O)C2 C(=O)(C(CO)C(F)(F)F)N1CC2C(C(=O)NCCc3nc(C)[nH]n3)C2C1 C(=O)(C(O)CNC(=O)CCCC1CCCO1)N(C(C(=O)OC)C)C c1(C(=O)NCC2C(NC(c3cccc(C(C)C)c3F)=O)C2)ccc2c(c1)NCC2 C(=O)(CC(C(=O)N(CC(O)CNC(=O)CN1C(=O)CCC1=O)C)NC(C)=O)OC c1(C(N(C(C)CCNC(c2cc(Cl)cnn2)=O)C)=O)ccnn(C)c1=O c1(C(=O)NC2C(CNC(Cc3cn(C)nc3)=O)CCC2)cc2n(n1)CCCC2=O C1(C(=O)NCC(C)Cn2ccnc2)CN(C(C2(C(N)=O)CCC2)=O)CCO1 C1(NC(=O)NCC(C)C2CC2)CCCN(S(=O)(=O)N(C)C)C1 CCS(=O)CC(=O)N1CCC(C)(CCNC(=O)Cc2ccnn2C2CCCC2)C1 c1(C(=O)NC(CC#C)C)ccoc1CNC(c1cnn(CCN(C)C)c1)=O N1(C(c2cn(CC)nc2)=O)CCC2CCN(C(=O)CC3=CCCC3)C2C1 C1(NC(C2C(C)CCO2)=O)CCCC(CNC(c2cccn2C)=O)C1 c1(-c2nc(O)cc(C)n2)nc(C2COc3ccccc32)nn1CC1CCCO1 Cc1nc(O)ccc1C(=O)NC1COCCN(C(C2CC2C)=O)C1 n1(CC(C)C)[nH]c(CC(=O)NCCCC(C)NC(C2CCCOC2)=O)cc1=O C1(C(N2CCC(CCC(=O)N(C)CC3(O)CCC3)C2)=O)CN2CCN1CC2 C#CCCCCC(=O)NCCN(C(=O)Cc1ccc(F)cc1C)CCOCCO S(=O)(=O)(CC(=O)NCC(C1CCC1)NC(=O)C(=O)C(C)C)NCC N1(C(C2C(CC)CCC2)=O)CC2CC(C1)CN(C(c1cnc(S)nc1)=O)C2 C(=O)(C1CCS(=O)(=O)c2ccccc21)NC1CC(CNC(c2cc(C)no2)=O)C1 CCC(C)(CNC(c1n[nH]cc1Cl)=O)NC(C1CC(=O)C1C(C)(C)C)=O c1(N(C)C)cnc(C(N2CCCC(CNC(c3cocc3C(N)=O)=O)C2)=O)cn1 c1(OC)cc(Cl)c(Br)cc1NC(CCC(C)C)C(=O)OCCCF C1(C(=O)NCCC2(CNC(C(C)OCC=C)=O)CC2)CCOCC=C1 N1(C(CC(C)(C)C)=O)CC2(CCCC2NC(c2noc3ccccc23)=O)C1 Cc1c(C(=O)NC2(CO)CN(C(C3(C)CC(F)(F)C3)=O)C2)cccc1[N+](=O)[O-] N1(C(c2c(C)nn(C)c2)=O)CC2(C)CC1C2NC(c1c[nH]nc1C1CC1)=O N1(C(C2CCN(CC)C2)=O)CCC(NC(c2snnc2C)=O)C12CC2 C(=O)(C(C)S(N)(=O)=O)N1CC(C(N(C(c2ccncc2)C)C)=O)C(C)C1 c1(C(=O)OCC)ncc[nH]c1=NCc1ccc(-c2ccnn2C(C)C)cn1 c1(C(C)C)ccc(C(=O)NC(C)CC(C)NC(c2ccc(C3CC3)cc2)=O)cc1 N#CC1(C(=O)CNC(=O)C)CCC1.C1(=O)CN(CCO)C(=O)OC1.C(C)(C)(C)O n1(CCC(N2CC(OC)(CNC(=O)CCC3CC3C)C2)=O)cnccc1=O C1(CC#C)CCCCN1C(=O)CC=CCNC(=O)C(C1CC1)OC c1(C(=O)NCC(CC)NC(c2cnc(C3CC3)nc2O)=O)cccc2nsnc12 c1(C(N2CCC(CNC(C3(C)CC(=C)C3)=O)C2)=O)cc2c([nH]1)CCC2 c1(CNc2c(CC(N3CCC(F)CC3)=O)cccc2)cccc2nccnc12 C1(C)(C(N2C3CCC(NC(c4ccnc(C)n4)=O)(C3)C2)=O)CC(C(F)(F)F)=NO1 C(=O)(C(C(C)(C)C)OC)N1C(C(N2C(C)(CC)CC2)=O)CSCC1 C12(NC(=O)COCc3noc(C45COC(C4)C(O)C5)n3)C3C4C1C1C2C3C41CO CCC(CNC(C1CCN(C(C)=O)C1)=O)(CC)NC(c1cc(C(N)=O)[nH]n1)=O C1(CNC(CC2(CSC)CC2)=O)(CO)CCCN(C(=O)C(O)C(F)(F)F)C1 C1(N(C)C(C2CCNC(=O)C2)=O)CCCN(C(C2CCN(C3CC3)CC2)=O)CC1 N1(C(C)=O)CCC(C(=O)OCCOCC)c2ccccc21.C1(=O)CCCCCO1 N(C(=NCC1CC1)N1CCc2c(Cl)cc(F)cc2C1)C(C)Cc1ccccc1 C(=O)(CC(F)(F)CS(C)(=O)=O)NC1C2(CCN(C(c3c(C)ccnc3)=O)CC2)C1 N1(C(C2N(C(C)=O)CC(O)C2)=O)C2CCC1CC(NC(c1ncccc1Cl)=O)C2 C1(CNC(C(C)SC(C)C)=O)CCC2(CN(C(C3CCC4(CCC4)CC3)=O)C2)O1 C1(C(N(C(C)CNC(c2coc(C(F)F)n2)=O)CC)=O)OCCC1C(F)(F)F Cc1sc(C(=O)NCCOCCNC(=O)Cn2[nH]cnc2=N)c(C)c1C Cc1cc(C(=O)NC2CC(CCNC(=O)CCCC(F)F)C2)c(C)c(C)c1 N1(C(C(P(C)(C)=O)O)=O)CCC(C2CCN(C(=O)Cn3cnnc3O)CC2)C1 C1(C#CC(=O)N2CCC(C(C)NC(c3nc(C)ccc3C)=O)CC2)(CC)COC1 Cc1cccc(CCC(=O)NC2CCC(N(C)C(C3NC(=O)OC3C)=O)CC2)c1 C(CC(C)C)(C(=O)N1CCCC(N(CCO)C(c2ccc(Cl)s2)=O)C1)NC(C)=O C12(C(N(C)CC3CCCN3C(c3cnoc3C3CC3)=O)=O)CC(C1)S(=O)(=O)C2 c1(C(N(C2CN(C(C(C)=C(CC)C)=O)CC2F)C)=O)cc(F)c(F)cc1OC c1(C(=O)NC(C)(CO)C(=O)N2CCC(n3ccnc3)C2)cccc2cc[nH]c12 C1(CCC)CN(C(c2cn(C)nc2OC)=O)CCN1C(=O)CC1CCC(=O)N1C c1(OC(C)C)cccc(CNC(c2c[nH]nc2CCNC(=O)C(C)C#N)=O)n1 c1(C(CNC(=O)C(O)CC2CCCCC2)NC(C=CCC)=O)cccc(OC)c1 c1(C(N2CC(CNC(c3n[nH]c(C)c3Cl)=O)C(O)C2)=O)cc(Cl)c(F)cc1F c1(C(N2CCC(C(=O)NC(COC)C(C)C)C2)=O)c(OC)cccc1C N1(CC(=O)N(CC(=O)NCC2CCN(CCC)C2)CCC)C(=O)CCC1=O S(=O)(=O)(c1cccc(C(F)(F)F)c1)N(n1ccnc1C(=O)OC)CC=C CCC(CC)CCCNC(c1c(Br)ncn1C)c1nnnn1CCCSC N1(C(C2(C)CC=C(C)CC2)=O)C2CCC1CN(C(c1nnn(C(C)C)c1C)=O)C2 c1(C(N2CCN(C(C(F)=CCC)=O)CC2C)=O)cc2ccccc2c(OC)n1 CCS(=O)c1ccccc1OCCCNC(=O)N(C)C C1(NC(c2ccc(CCC)s2)=O)CC2CCC1C(NC(=O)C#CC(C)(C)C)C2 C1(CCC)CCN(C(=O)C(F)C2CC(NC(C3CC3Cl)=O)C2)CC1 N1(C(CC=C=C)=O)CC(NC(C2(C)CCN(C)C2)=O)C(N=[N+]=[N-])C1 c1(NCC2C(C)C2C)[nH]c(=NCc2ccccc2C(C)(F)F)nc2ncn(C)c12 C1(C(=O)NCCCN(C(C(C)NC(CC)(C)C)=O)C)COc2ccccc2C1 C1(CCC)CN(Cc2cccnc2)CCN1C(=O)Cc1cccc(Br)c1 c1(C(=O)NC23CC(CNC(c4n(C)ncc4)=O)(C2)C3)nccc(F)c1Cl N1(CCC)CCN(C(=O)C(C(C)O)NC(C2CC(C)(F)C2)=O)CC1 c1(C(N2C(C(=O)NCC(CC)C(C)C)CC(OC)C2)=O)cc(C)nc(C)n1 N1(CC(C)(C)N)CCN(C(C2C(C(F)F)C2(C)C)=O)CC1 CC1=C(c2ccncc2)CN(c2nc(N3CCC(C)(C)C3)c3c(n2)CSC3)CC1 c1(CC)ncnc(CC)c1C(=O)NC1CC1NC(=O)Cc1c(C)noc1C C1(CN(CCCCCCC=C)C=O)CCc2ccccc2O1 N1(C(C(CCC)(C)O)=O)C2CCCC1CC(NC(=O)CSc1nc[nH]n1)C2 C1(C)(CN(c2n(CC(=C)C)nnn2)C(C)C)CCCCC1 c1(C(=O)NCCCCNC(c2ccccc2OC2CCC2)=O)ccc(Cl)cn1 c1(C(N2CCC(O)(C(C)NC(CNC(C)=O)=O)C2)=O)c(C)ncc2ccccc12 c1(N(CC(F)(F)Cl)C)nc(N2CCN3CC4(CC4)CC3C2)nc2ccsc12 CC1=NN(C)C(=O)C1CC(=O)NC1CC(NC(c2cn(C)cc2C(F)(F)F)=O)C1 c1(C(=O)NCC2CCC(NC(C3(CC(C)C)CCC3)=O)C2)cnn2cnnc2c1 C(c1ccncc1)=C(C)C(=O)NC1CC1NC(=O)C(C(C)C)N(C)C N1(C(CCC2N(C(Cc3c(C)n[nH]c3)=O)CCCC2)=O)CCOCC(O)C1 C1(C(=O)NC2(CNC(COC3(C)CCC3)=O)CCCC2)CC12CCOCC2 Cc1cc(Cl)c(Cl)cc1C(N1CCOC(C(C)NC(=O)C=CCN(C)C)C1)=O N1(CC(=O)NC(C)C2CC2)CCN(C(C2COC2)=O)CC1 C1(NC(C2(C)CCCN2C(=O)CC2(C#N)CC2)=O)CCCOC12CCC2 c1(C(C)C(N2C(CNC(=O)C3=COCCO3)CC(O)C2)=O)c[nH]c2ccccc12 C=CCC(CC(C)C)C(=O)NC1(C(=O)NC2CC2O)CCC1 c1(CNC(C2CCC(C)C2)=O)ccc(CCNC(c2n[nH]c(C3CC3)n2)=O)cc1 C1(CN(C(CN(C)C)=O)C)COCCN1C(=O)CC1CCC(O)C1 c1(C(N2C(C)(CNC(Cc3ncc(C)o3)=O)CCC2)=O)ncnc2c1CCCC2 CN1CC2(CCN(C(C3CC4CC4N3S(=O)(=O)c3ccc(Br)cn3)=O)CC2)C1 C1(NC(C2(C(=O)OC)C(=C)CC2)=O)CN(C(=O)C2=NOC(C)C2)CC12CCC2 N1(C(C(c2ccncc2)C)=O)CCC(C)C(CNC(c2cccc(Cl)c2)=O)C1 c1(OC)cnc(Cl)[nH]c1=NC1CCC2CN(C(=O)Cc3cc(C4CC4)on3)CC12 C1(C(=O)NC(CNC(Cc2nc(C)sc2)=O)C(C)C)CC2CCC1O2 Cn1nc(C(=O)NC(C)(C)CNC(C2C(C(F)F)C2(C)C)=O)ccc1=O CC(CCC(=O)N1CCC(F)(CNC(C2(Cl)CC2)=O)C1)N(C)C c1(OC)ncnc(C(=O)NCC2=CCN(C(C3CN4CCN3CC4)=O)CC2)c1F C#CCCCC(C)C(=O)N1CCC(C2CC2)(NC(c2cccc(C(N)=O)n2)=O)C1 N1(C(C(=O)NCC)=O)CCn2c(CNC(C3CCN3C)=O)nnc2C1 N1(C(c2nn(C)cc2I)C(=O)NCCOC)CCCCCC1c1cccc(C)c1 N1(C(c2cnc(CC)o2)=O)CC2CC(NC(c3ccc([N+](=O)[O-])s3)=O)C1C2 CON1CCC(C(=O)NCC(O)CN(C)C(C2COCC2(C)C)=O)CC1 C(=O)(C1=CCCSC1)NCCC(C(=O)N1CC(CN(C)C)C1)O C1(NC(c2cncc(NC)c2)=O)CC2CC(NC(c3cc(C)n(C)n3)=O)CC2C1 c1(C(N2CC(CCNC(Cc3cc(=N)[nH]cc3)=O)C2)=O)coc2cc(F)ccc12 CCCCCCC(C)NC(C1(F)CCCN(C(c2cnc3n2CCC3)=O)C1)=O C1(CC=C)CCCCN1C(=O)C(Cc1ccccc1Br)NC(=O)Cc1ccsn1 O=C(CCCn1cc(CC2CCCC2)nn1)NC1CN(c2n[nH]cc2Br)C1 C1(C2CCCCC2)(NC(=O)CCOCCCNC(C2COC(=O)N2)=O)CC1 c1(NC(C2C(NC(c3ccc(C)cc3F)=O)CCC2)=O)ncc2ccccc2n1 C(=O)(C1CCc2nccn21)NCCN(C)C(C1CN2CCN1CC2)=O C=C(Cl)C(C)(C)C(=O)N1CCCC(N(C(=O)Cc2cccc(Cl)c2F)CCF)C1 CN=c1[nH]c(=NCc2cc3cc(Br)ccc3[nH]2)[nH]c(=NCC2(C)CC(C)C2)[nH]1 CCC(CN=c1nc2c(ncn2CC)c(NCC(C)(CC)OC)[nH]1)OC c1(C(N2C(C(=O)NCCOCCC#C)CCC2)=O)cc(CO)ccn1 Cc1ncccc1C(=O)NC(c1ccccc1)C(=O)NCCn1cccnc1=O c1(NCC2OCCN(C(c3c(CC)c(Br)ccc3)=O)C2)cc(F)cc(C)c1O CC1(NC(=O)NCc2cccc(Cl)c2F)Cc2ccccc2C1 Nc1ccc(C(=O)NC2CC23CC(NC(c2ncc(Cl)cc2Cl)=O)C3)c(Cl)c1 O(NC(=O)C(C)(C)C(C)NC(=O)C(C)c1ccco1)CCOC C12(NC(c3ccc(SC)o3)=O)CCC(CNC(c3cnsn3)=O)(CC1)OC2 N1(C(c2c(C)nn(C)c2N)=O)CCC2(CC1)CN(C(c1occc1Cl)=O)C2 N1(C(=O)CC2CNC(=O)O2)CC2CC(C1)N2C(C1(O)CCCC1)=O c1(C(=O)NCC2(C(C)NC(C(C)OCCOC)=O)CC2)ccc(N)c(Cl)c1 CC1N(C(=O)C(C2(O)CCC2)NC(C2COCOC2)=O)CCCC1(C)C N1(C(c2ncc(OCC)nc2)=O)CC2CCC1CN2C(c1cnc(N)cn1)=O C1(CNC(CN(C)CC)=O)CCCC1NC(c1cc(Cn2cc(Cl)cn2)cs1)=O C1(CNC(=O)NCC2(C#C)CC2)CCN(Cc2ccccc2Br)CC1C C=C1CCC(C(=O)N(C2CCCN(C(=O)C(F)OC)C2)CCF)CC1 C12(C(=O)NCC(CCOC)NC(c3nnc(C)s3)=O)CCC(CC1)CC2 C1(NC(C2(NC(C)=O)CCC2)=O)CC2(CCCCN2C(C2SCCC2C)=O)C1 N1(C(C(CO)NC(N)=O)=O)CC2(CC(NC(=O)CN3CCCC3=O)C2)C1 C1(C(=O)NCCN(C(C2C(OCC)C2)=O)C(C)C)CCC(O)CC1 c1(C(C)C)cc(C(=O)NCC2CC(C(=O)NCc3cn(C)nn3)C2)on1 c1(CCC(=O)NC2C(NC(CCC#CC)=O)CCCC2)c(Cl)cccc1[N+](=O)[O-] N1(C(c2c(SC)scc2)=O)CCC2(CC1)CN(C(=O)C(C)CCCC(C)C)C2 N1(C(C2(C3(C)CC3)CC2)=O)CCC(C=CC(=O)NCC(C)(F)C(C)(C)F)CC1 N1(C(=O)Nc2ccc(OC)cc2)CCC(C)C(NC(C2C=CS(=O)(=O)C2)=O)C1 C(C(=O)NC1CCN(C(=O)CC2CCCC(=O)C2)C1C1CC1)(C(C)C)SCC C1(NC(c2ncn(C)n2)=O)CN(C(C2Cc3nccn3C2)=O)C2CCCC12 c1(C(CC(=O)NCCC2CC(NC(C=C(CC)CC)=O)C2)O)cccc(F)c1 N1(C(=O)NC2CCN(C(=O)Cc3cn[nH]c3)O2)CC23CCC2(COC3)C1 C=CCC(C)C(=O)NCc1ccc(CN(C(=O)CC(C)COC)C)cc1 C(N=c1c(Cl)c[nH]c2c(Br)cccc12)c1ccc(S(=O)(=O)N(C)C)cc1 Cc1nc(C)c(CC(=O)NC(C)CN(C)C(c2ccnc(C)c2O)=O)c(O)n1 N1(C(C(CCC)NC(c2ncn(C)n2)=O)=O)CCC(C)=C(F)C1 c1(C(=O)NCC(C2CCOC2)NC(c2cc(C(=O)OC)on2)=O)ncncc1Cl N1(C(C2(C#C)COC2)=O)CCC(NC(C2CC3CCC2CC3)=O)C(C)(C)C1 c1(C(=O)NC2CCCC(Nc3ncc(I)cn3)C2)cc2ccccc2oc1=O c1(C(=O)NC(CCOC)C(=O)N(C)CC2CCCO2)cnn2ccccc12 N1(C(C(C=C)CC)=O)CCC(COC)(NC(c2ccc(=N)[nH]n2)=O)CC1 c1(NC2CCN(C3CC3)C2)ccc(F)cc1.c12ccoc1C(N(C)C)C(=O)NC2 Cc1ccc(C(N2CC(O)(CN(C)C(c3c(C)cccc3N)=O)C2)=O)c(C)c1 CC1CCCCN(C(=O)C(C(C)(C)O)NC(=O)COC(C)(C)C)C1 C1(C)(C(=O)NC(CN(C(=O)CNC(=O)NC2CCCCC2)CC)C)CC2CC2C1 C#CCCC(O)C(=O)NCC1(F)CCC(NC(=O)CCCCc2cnc[nH]2)C1 C(=O)(C(C)(C)CC(F)F)NCCC(CNC(CCCCCOCC)=O)O CCCC(CCCNC(c1ccc(OC)cc1Cl)=O)NC(C1(Cl)CC12CCC2)=O N1(C(CN(C)CC)=O)CCC(CNC(=O)C(C(C)C)n2cncn2)(COC)C1 C1(C(N(C)Cc2n(CC)ccn2)=O)CN(C)CCN1C(=O)C(C)CN(C)C c1(C(=O)NCc2c(C(N3CCC(CC(N)=O)C3)=O)scc2)ccccc1Cl C1(C(C)N(C)C)CCN(C(=NCC2CCCO2)NCc2cccc(Br)c2O)C1 N1(C(CC(C)C2CC2)=O)CC2CCCCC2(NC(=O)Cn2ncnn2)C1 c1(-c2cn(CCC(=O)NC(C)CCN(C)C)nn2)ccc(C(F)(F)F)cn1 CC(C)(C)CC(C)(C)C(=O)NC1CCCN(C(=O)CCCc2cnccn2)CC1 Cc1cc(C)n(-c2cccc(C(F)(F)C(C)(F)F)c2)n1 CCCC(O)C(CO)NC(=O)CN(C(c1cc(C)nnc1C)=O)CC1CC1 N1(CC(C)(C)NC(=O)C=Cc2cccnc2)CCN(C(C2CCNC2=O)=O)CC1 C1(NC(C2(CC=C)CCOCC2)=O)CCN(C(C2(C#N)CC2)=O)CC1F S(=O)(=O)(c1cccc(NCC(C)Oc2ccc(F)c(Br)c2)c1)N(CCC(C)C)C c1(OC)cc(CN2CC3C(C2)N3C(c2c[nH]c3ccccc23)=O)cc2c1OCO2 C1(NC(C2(c3c(C)cc(F)cc3)CC2)=O)CCN(C(=O)C#CC2CC2)CC(O)C1 n1(CC)c(-c2nc(C3CCCO3)nn2-c2nccn2C)cnc1O CC1(C)CCCCCC1NC(C1(NC(c2cc[n+]([O-])cc2)=O)CC1(C)C)=O Cc1cnccc1C(N1CC(c2ccccc2)(NC(C2COC(=O)C2)=O)C1)=O C=CCC(CC)C(=O)NCCCOCCN(C(=O)C(C)C)C N1(C(CN2CC(C)C2)=O)CC2CC(C(=O)NC(C)(C)C)CC(C2)C1.C1(=O)C=CCN1 C1(C(c2nnnn2C2CC2)(C)NCC2CCCC(C)(C)C2)Cc2ccccc2C1 CC1CCCN(C(=O)CCc2cn(C)cn2)C1CNC(=O)CN1CCC(C)(C)C1 c1(C(c2occc2Br)N(CCNC(=O)C(C)(C)C)CC)ccccc1F c1(CC(=O)NC(CNC(C(C)OC)=O)C2CCC2)ccsc1Cl O(NC(=O)CN(C(=O)CC)CCN(C)C)CCC.C1(C)CCCO1 CN(CCCC(=O)N1CC(NC(c2cnn(C(C)(C)C)c2)=O)C2(CC2)C1)N=O CC1CN(C(=O)CS(C)(=O)=O)CCC1NC(=O)C(F)(F)C1(O)CCCC1 c1(C(C(C)NC(c2c[nH]c(C(F)(F)F)c2)=O)C)ccc(C(F)(F)F)cc1 c1(C(NOC(c2nn[nH]n2)C)=O)ccc(NC(C(F)(F)F)C2CC2)nc1 C1(NC(C2C(CC)OCC2)=O)CCS(=O)(=O)C12CN(C(=O)C=C(Cl)Cl)C2 C(=O)(CCCC(F)F)N(C(CNC(C1CCN(C)C1)=O)C1CC1)C CCCCCC(C)(C)C(=O)NCCCCN(C)C(C1CC(=O)N(C(C)(C)C)C1)=O CC1CN(C(C2CCC(F)CC2)=O)C(C)CN1C(=O)CCc1ccccc1C#N CCC(CC(=O)N1CCC(CNC(=O)Cc2cnc[nH]2)(COC)CC1)C(C)(C)C N1(C(=O)C2=CCOC2)CCN(C(c2ccc(-c3cccs3)o2)=O)C(C2CCC2)C1 C1(CC(=O)NCC(CNC(C2(C(C)C)CCCO2)=O)(C)C)CCCCCC1 N1(C(C2(O)C(C)(C)C2)=O)CCC2(CCOCC2)C(NC(=O)Cc2cn[nH]c2)C1 N1(C(c2c(C)cc(Cl)nc2)=O)CCC(N=c2ccnc(C(C)(C)C)[nH]2)C1 n1(CC(COC)OC)c(N2CCN(c3ccccc3Cl)CC2)nnc1C(C)C c1(-c2ccc(C3(C(N4C(CCCCC)CCC4)=O)CC3)s2)ccc(F)cc1 Cc1cnc(C(=O)NC2CCCN(C(=O)CCc3nnc(C4CC4)o3)C2)c(F)c1 C1(NC(c2cnn(C)c2Cl)=O)CN(C(C2CC(=O)N(CC3CC3)C2)=O)CC1(C)C C1(NC(C(=O)N(C)C)=O)CC2CC(NC(=O)CCc3ccc(O)nn3)C1C2 C1(C(=O)NCCC(O)CNC(=O)CC2CCCC2O)(COC)CC(=O)C1 C1(C)(CSC)CCN1C(=O)C(F)CC1CN(C(=O)COc2cc(C)on2)C1 C1(N(C(=O)Cn2nnc(C)n2)CC)CCCN(C(C2CC3CCC2O3)=O)C1 C1(CNC(CC(=O)OC)=O)CCN(C(c2nn(C(C)(C)C)cc2Cl)=O)C1(C)C c1(NC(C2CC2NCc2ccc(F)s2)=O)ccc2sc(Cl)nc2c1 C(=O)(C(C)(C)C(=O)OC(C)(C)C)N1CC2C(N(C(CC=C(C)C)=O)C)C2C1 C1(CC)CN(C(=O)C(C2CCC2)NC(=O)COCC2CCC2)CC1O N1(C(C2N(C(c3c(C)cccc3O)=O)CCC2)=O)CC(=O)NC2(CC2)C1 N1(C(c2cncc(O)c2Cl)=O)CCCC(C2CN(C(=O)C(O)C(F)F)C2)C1 CCCC(C)(C)C(=O)NC1CC(F)CN(C(=O)Cc2cccc(C(N)=O)c2)C1 CCC1=NOC(C(=O)NC2(C)CCCC2NC(=O)Cc2csnn2)C1 CCCC(C#N)C(=O)N1CCC(C)C1c1cn(CCOCc2ccccc2)nn1 c1(SC)nc(Cl)cc(=NC2CC(F)(CNC(c3cnn4ccn(C)c34)=O)C2)[nH]1 C(=O)(C1=CC2(CCOCC2)C1)NCC1(F)CC(NC(C2C(CC)C2)=O)C1 c1(C(=O)NCCCN(C(C(C=CCCC)O)=O)C)cc2c(Cl)nccc2s1 N1(C(c2scc(C(C)=O)c2)=O)CCC(C(C)NC(C2(F)CC=CC2)=O)CC1 N1(C(Cc2c(C)con2)=O)CC2CC(NC(C3CCOC4(CCC4)C3)=O)CC1C2 n1(CC)cc(C(=O)NC(C)(C)C=CC(=O)NCC(F)(F)CC2CC2)nn1 Cc1cccc(F)c1C(=O)NC1C=CC(C(=O)NCCCCc2ccccc2)C1 C#Cc1ccc(C)c(NC(=O)NC(CSC)C(=O)N2CCCCC2)c1 c1(NC(C(C)OC(=O)CCn2cccn2)=O)c(Cl)cccc1F Cc1cccc(CC(=O)NCc2cc(C(N3CCCC3CN(C)C)=O)co2)c1 C1(CCC2N(C(c3nc(C)sc3)=O)CCC2)CCN(C(=O)CC2(CO)CC2)CC1 c1(N(C(N(CC=C)CC2CC2)=O)CCO)cccc(CN2CCSCC2)c1 C1(CNC(C2N(N=O)CCC2)=O)CC2CCC1N2c1cc(C(F)(F)F)nc(Cl)n1 C(C(C)(CNC(=O)CCN(C(c1ccc(C#N)s1)=O)CC1CC1)CO)OC N1(C(C#CC(C)C)=O)CCC(O)(C(C)NC(=O)CCCCCn2cnnn2)CC1 CC1CCN(C(=O)N(C)Cc2ncnn2C)c2ccccc21 C1(C(=O)NC(C2CCN(C(C3(C)CCCC3)=O)C2)C)CCC1(C)C C1(NC(CCC(=O)NC)=O)CCCC12CN(C(C1CC3(C1)CC3F)=O)C2 N1(C(C2(C(C)C)COC2)=O)CC(CO)(NC(=O)CSc2nncs2)C1 C12(NC(c3c(C)cc(C)o3)=O)CCCC1N(C(=O)Cc1ccc(Cl)cc1C)CC2 C12(C(N(C3CCN(C(C45CCCN(CC4)C5)=O)C3)C)=O)CCC(CC1)CC2 CC1(C)CCCC(CC(N2CCC(CCNC(=O)Cn3cnnc3O)C2)=O)C1 c1(CC)cc2c(NCC3(NC(c4ccc(CC)o4)=O)COC3)ncnc2s1 n1(CCC)cc(C(=O)NCC2(CN(C(=O)CC(C)OC)C)CC2)c(C)n1 c1(CN2CCC(CNC(=O)C=Cc3ccc(Br)cc3)C2)c(Cl)cccc1B(O)O Nc1cc(F)c(C2CC(N3CC(=O)N(CC(=O)Nc4ccc(F)cc4F)C3=O)C2)c(F)c1 N1(C(C(CC=CC)C)=O)CC(CC(=O)NCC(C)(O)CSC)CC1(C)C CCCCCC(O)CC(=O)N1CCC(C(C)NC(C2CC3(C2)OCCO3)=O)CC1 C1(NC(CCCC)=O)CN(C(=O)C(C)NC(=O)OC(C)(C)C)C2CCCC12 CC(CC(=O)N1CC2CN(C(c3nc(Cl)ccc3N)=O)CCC12)C(F)(F)F CC1(O)CCN(CC(=O)NC2CCCCC2NC(=O)C(c2cccnc2)O)C1 C(CC(N=c1cc[nH]cc1C#N)C(C)C)N(C(Cc1ccc(C)nc1)=O)C C(CCC(C)C)(C(=O)NC(CCNC(c1n[nH]c(C)c1F)=O)C(C)C)NC(C)=O C1(NC(CC2(OC)CN(C(c3ccc([N+](=O)[O-])s3)=O)C2)=O)CCCCC1(C)C c1(C(N2C(C)CN(C(=O)CC3CCCNC(=O)C3)CC2)=O)nc2cccnc2s1 O=C(C1=CCCN(C(=O)CCCCCBr)C1)NCc1cnc(Cl)s1 N1(C(C2CC2c2c(Cl)cccc2Cl)=O)CC2(CCOCC2)C1c1ccco1 c1(OCC)ccc(C(=O)Nc2cccc(C#N)n2)cc1OC.C12CC(C1)NC2=O C1(N(C(c2cn(CCCOC)nc2)=O)C)CCN(C(C2CCC(C)S2)=O)CC1 Cc1nn(CC(=O)NC(C2CCCN2C(=O)CC2CCSC2)C)c(=O)o1 c1(CNC2C(C(=O)NC(C)C)CCCC2)ccc(F)cc1O C1(NC(=O)CC2CSC2)C(CNC(C2CC2c2ccco2)=O)CCC12CCC2 C1(C(=O)NCC2C(C(=O)NCC(C)NC(=O)OC)C2)CCCCC(=O)C1 C1(NC(CCCC(=O)NC2CC2)=O)CN(C(=O)C=CC2CCC2)CC12CCOCC2 C1(C(=O)NC(C)CN(C(C2(F)CCCCC2)=O)CC)(OCC)CCCOC1 c1(CN(CC(CNC(C2CC2CO)C)O)C)ccccc1 c1(SC)ccccc1C(c1nc(C)cn1C)N1CCC(c2ccccc2Cl)C1 c1(C(=O)NC2C(C)(CNC(c3coc(CO)c3)=O)CCC2)ccnc2[nH]cnc12 c1(C(=O)NC2CCN(C(CCc3ccc(C(=O)OC)[nH]3)=O)C2)ccc(Cl)c(C)c1 N1(C(C2(NC(CC(C)C3CCCO3)=O)CC(O)C2)=O)CCC(C2=NOCC2)C1 C=CCCN=C(NCc1cc(C)c(C)s1)NC(C)C1CC1 N1(C(c2cc(C)c(C)o2)=O)CC(C2CCN(C(C3CCOC3(C)C)=O)CC2)C1 C1(N(CC#C)C(C2CC2CF)=O)CCN(C(C2(C(F)(F)F)CCCC2)=O)CC1 c1(C(=O)NC(C)C(=O)NCCCNC(C2C(Cl)(Cl)C23CC3)=O)ccccc1Cl N1(C(CCOCC)=O)CC(NC(c2nscc2C)=O)C(n2ccnn2)C1 CCCC(C(=O)N1CCCCC1CNC(=O)C(C(C)CC)OC)S(N)(=O)=O CC1CN(C(=O)C=Cc2cnc[nH]2)CC1NC(=O)CCOc1cccc(F)c1 Cn1ccc(-c2noc(C3(C4CCNCC4)CCC3)n2)n1 N(C)(S(=O)(=O)N(C)C)CC(=O)NC1C2CN(CC(=O)N(C3CCCC3)CC)CC21 c1(C(=O)NC(C)CCNC(=O)C(c2ccccc2F)O)cccc(P(C)(C)=O)c1 CC(=Cn1ccnn1)C(=O)NC1COCCC1NC(C1CCC(F)(F)CC1)=O C1(C(=O)NCC2(CNC(C(C)CN(C)C)=O)CCCC2)CCc2nn(C)cc2C1 N1(C(C(CCC)=CCC)=O)C2CCC1(CNC(c1cnc(O)s1)=O)CC2 CC(C)C(CCN(C(=O)CCc1cc[nH]n1)C)NC(C1(O)CCCC1)=O C1(CCNC(C(C)SC)=O)CN(c2nccc(C#N)n2)CCCO1 C(CCN(C(=O)C(c1ccc(F)cc1)CO)C)(C(C)C)NC(c1c(C)cc[nH]1)=O N1(C(C2C(CC)N(C(c3ccc(F)cc3)=O)CC2)=O)CC(OC)CC(C)C1 C1(C(=O)NCCCN(C(C2C(C(=O)OC)C=C2)=O)C)CCCCN1C Cc1ccc(C(C)(C)C(=O)NC2CN(C(=O)CC(=O)N(C)C)C3CC23)cc1 c1(C(N(C(C(N2CCCC(OC)CC2)=O)C)C2CC2)=O)c[nH]c2cnccc12 Cc1ccc(S(=O)(=O)NCC(N2CC3CCC(C2)C3O)=O)c(F)c1 c1(CCNC(C2CC2F)=O)ccc(CNC(C2CC(F)C2)=O)cc1 C(CCF)(C(=O)NCCCc1nccs1)NC(C1C(C)OCC1)=O c1(C(N(CC(CC)NC(c2cc(C(CC)CC)no2)=O)C)=O)nnc(O)cc1O C(=O)(C(=O)NCC(C)CNC(C1CCN1C(=O)OC(C)(C)C)=O)NC c1(C(N2CC(O)(CC)C2)=O)ccc(CNC(=O)CSc2ccccc2)cc1 C1(C(N2CCC(COC)(CNC(=O)C(O)C(C)C)CC2)=O)CC(C(C)(C)C)=NO1 C1(C(=O)NCCc2nnc(C)s2)CC(C)CN(C(C2C=CC=CC=C2)=O)C1 C=CCN(OC)C(=O)C12C(NC(=O)CCc3csnn3)C3CC1C2C3 C1(C(=O)OCC)CC12CCN1C(CCO2)C(C)(CCCOC)NC1=O c1(OC)ccnc(OC)c1C(=O)NC1CCN(C(C2COC(=O)O2)=O)C1 C1(C(=O)NCC2CCC(NC(CS(CC)(=O)=O)=O)CC2)COC2(CCC2)CO1 N1(C(c2c(C)cnn2C)=O)Cc2nccn2CC(NC(=O)CCc2ccoc2)C1 c1(SCC)cccc(C(=O)NC2CN(C(=O)C(O)C(F)F)CC2C(F)F)c1 S(=O)(=O)(c1cscc1F)Nc1c(CC(=O)OC)cccc1 c1(OC)c(C(=O)N=CC(=O)NC2(CO)CC(OC3CCC(O)CC3)C2)cnn1C C1(CC(=O)NC(C=C)(C)CC)CC2(CC2)CN1C(=O)CSC(C)(C)C c1(OCCC(=O)N(CCNC(C(CC)COC)=O)C(C)C)ccc(Cl)cc1Cl C=CCCC(C(=O)OC(C)(C)C)NC(=O)CC1CCCCN1C(C1CC1OC)=O C1(NC(C(C)OCC#C)=O)CN(C(c2sccc2C2CC2)=O)CC1S(C)(=O)=O C(=O)(CCC(F)F)NCC(CNC(=O)Cn1ccc(C(F)(F)F)n1)O [N-]=[N+]=NC1CC(C(=O)NC2CC3CCC2O3)N(C(c2ccc(C#N)cc2)=O)C1 Cc1ccc(-c2ccc(C(=O)NC3CC(F)(CNC(c4ccsn4)=O)C3)s2)s1 C1(C(=O)O)CN(C(c2cnc(O)c(Cl)c2)=O)CC12CCCC2 c1(C(N2CCC(CNC(CSC)=O)C(F)(F)C2)=O)ccc2nc(O)[nH]c2c1 C(=O)(C1=Cc2ccccc2C1O)N(C1CCC(NC(=O)CC2CCC2)CC1)C C1(N(CC(=O)NC)C)CCN(C(=O)C(C)n2cccn2)C1(C)C c1(OCC)c(CC(c2nnnn2NC(C)(C)C)C2CSC2)cccc1Cl C1(NC(CN(c2ncccn2)C)=O)CC2CC(C1)N(C(=O)Cc1ccc(Cl)s1)C2 C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)CSc2nnnn2C)CC1C C#CCC(O)C(=O)N(C)CC1CC(F)CN1C(C1CC(F)(F)C1)=O N1(C(C(c2ccccc2Cl)(C)C)=O)CC2CC2(CNC(c2ccsc2C#N)=O)C1 C1(NC(C(COC)OC)=O)CN(C(C2(C)CCOCC2)=O)CCC12CCOCC2 C1(NC(C2(CC#C)CCC2)=O)CC(CNC(C2CCC(=O)N2C(C)=O)=O)C(O)C1 Cc1ccc(C(=O)NC2CCCC2NC(C2(C(C)(F)F)CC2)C2CCC2)c(Cl)c1 N1(C(C(CCOC)C)=O)CCN(C(c2cn(CC(F)(F)F)nn2)=O)C(C)C1 Cc1cc(C(c2nnnn2C2COC2)Nc2cn(CCF)nc2C)sc1C C1(C(=O)NCC2(CN(C(=O)C=C3CCC(C)C3)C)CC2)(OC)CCC(C)(C)CC1 c1(OC)ccc(Cl)c(C(=O)NCCC2CCCCN2C(c2cccnc2C)=O)c1 N1(C(C(CC(C)C)O)=O)CCCCCC(NC(c2ccc3ncnn3c2)=O)C1 c1(N2C3CC(CNC(C(C)O)=O)CC2CC3)ncnc(N(C)C)c1[N+](=O)[O-] c1(C(N2CC(F)CC(NC(C(C=C=C)C)=O)C2)=O)ccc2cc(O)ccc2n1 CCCCCC(O)C(=O)NCC(C)(CC(C)C)NC(=O)CCSc1ccccn1 CCC(CCC(=O)N1CCSCC1CCNC(c1cc(Cl)cs1)=O)OC N1(C(C(C)=CC=C)=O)CCC(C(C)C(=O)NCC2CN3CCC2C3)CC1 C=C=CC(C)C(=O)NCC(C)NC(c1c(C(F)(F)F)coc1CC)=O c1(C(=O)NC2CN(C(C(C)(C)NC(C)=O)=O)CC(F)C2)c[nH]c2ccc(Br)cc12 C1(NC(c2c(C(C)C)c[nH]n2)=O)CCN(C(=O)COC2(C)CCCC2)CC1F C1(CCC)CC(C(=O)NC(C)(C)CNC(c2nc(C)oc2C)=O)CCO1 N1(C(C(CC2CC2)NC(C(CC=C)(F)F)=O)=O)CCC2(CC1)CN(C)C2 C1(CNC(c2cccc(CNC(C3CC4C=CC3C4)=O)n2)=O)CCC(CO)CC1 C1(NC(C2CCN(C(C)=O)C2)=O)CC2(C1)CC(NC(C1CNC(=O)N1C)=O)C2 C(=O)(C(CC(C)C)CC(C)C)NCCN(CCC)C(c1cc(F)ccc1NC)=O c1(C(N2C3(CNC(C(COCC)N=[N+]=[N-])=O)CC(C2)C3)=O)nc(C)c(C)[nH]c1=O N1(C(COCC)=O)CCCC1CNC(=O)C(C1CC1)N(C)C c1(C(N2CC(NC(c3cc(CCOC)on3)=O)(CO)C2)=O)cc(O)ccc1C S(=O)(=O)(c1cccc(Cl)c1)N1CC(CC(N2CCC(F)C2)=O)OCC1 C12(CNC(c3ncc(C)nc3)=O)CCCC1CN(C(=O)C(C)C1CC1)C2 C#CC1(C(=O)NCC2(N(C)C)CCC2)CCN(C(=O)CC(C)(O)C=C)C1 N1(C(CSCC(N)=O)=O)CC(NC(C2CC(OCC3CC3)C2)=O)C(O)C1 c1(C(N(CC(CC)NC(C2CC2c2ccsc2)=O)C)=O)ccc(F)cc1[N+](=O)[O-] C1(NC(c2cc(CC)no2)=O)CCC2(CCN(C(C3(C(F)F)CC(=O)C3)=O)C2)C1 c1(C(=O)OC(C)(C)C)conc1C(N1CCC(NC(C2CC2(Cl)Cl)=O)C1)=O N1(C(C(=O)Nc2ccc(C)cc2)=O)CC(C)N(C(c2cccc(Cl)c2)=O)CC1C C1(CNC(c2cc(C)no2)=O)CN(C(c2cnn(CC3CC3)c2)=O)CCC1(C)C C(C(C)N=c1[nH]c(Cl)nc(C)c1F)NC(Cc1ccc(C)cc1Cl)=O c1(NC(N(C(C)C(C)(C)c2ccccc2)CC#C)=O)n[nH]nc1OC N1(C(c2cc(CC)c(C)s2)=O)CCCC1C1CCCCN1C(=O)COC(C)(C)C C(CC(=O)NCCCCCC(C)C)(C(F)F)NC(c1ccc(C(C)=O)[nH]1)=O c1(CC)ccc(C(=O)NCC2CC(NC(=O)C(C)(O)CC(C)C)C2)cc1[N+](=O)[O-] S(=O)(=O)(c1ccc(Cl)cc1Cl)N1CCN(C(C=C(C)C)=O)C2(C1)CC2 CCC(O)CC(=O)NC1CCN(C(c2nc(Cl)sc2C)=O)C1 C1(CC(N2C(CC)CC(C)C2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C N1(C(CC2CN(C(Cc3ccc(C)s3)=O)C(C)C2)=O)CC2CCC(C1)C2O N1(C(CC(C=C)CCC)=O)CCCCC2(C1)CN(C(=O)CC(F)(F)F)C2 C1(C(=O)NC(CC(C)NC(c2cnc(C)[nH]2)=O)C)CCCCN1N=O c1(COC)cc(C(N2CC(O)(C(C)NC(=O)CCCc3csc(C)n3)C2)=O)n[nH]1 Cc1cccc(C(=O)N(CC(=O)O)Cc2cn(CC(c3cccnc3)O)nn2)c1C c1(C(N2CC3CN(C(C4(n5ccnn5)CC4)=O)CC3C2)=O)cc(Cl)c(F)cc1Cl N1(C(c2cc(SC)oc2)=O)CCC2(C=C(C(=O)NC(c3c(C)n[nH]c3C)C)C2)C1 c1(C(N(C(C)CNC(=O)C2=C(C)CCC2)CC)=O)c(F)ccc(F)c1O CCC(C)C(C(=O)NCC1CCCCO1)NC(c1ccc(=N)[nH]n1)=O c1(C(N(CC(C)CNC(=O)CC2COC(=O)C2)C)=O)ccnc2[nH]cnc12 c1(C(C)C(=O)N2CC(OCCNC(C3CC34CCC4)=O)C2)ccccc1Br C(=O)(C(CO)c1ccccc1)N(CC(C)(C)NC(=O)C(N)=O)C n1(CC=C)ccnc1C(=O)NCC(C)N(C(c1ccc(CNC(C)=O)s1)=O)CC C1(CC(=O)N(CCn2cc(C(C)(C)C(=O)O)nn2)C2CC2)COc2ccccc2O1 c1(OC)cccc(NC(=O)C(c2nocc2CC2CC2)N(C)CC2CC2)c1 Cc1ccc(OC(C)C(=O)NCCCN(C(c2cnnn2C)=O)C2CC2)cc1 CC1(C(N2CC3C(C(=O)NCc4cccc(Cl)n4)C3C2)=O)COC(=O)N1 c1(CCC)cc(C(=O)N(C)CC2CN(C(c3cnn(CC)n3)=O)CCO2)nn1C C(=O)(C1=CCCSC1)N1CCC(CCCCCNC(c2c(C)ocn2)=O)CC1 N1(C(CN(C)C(N)=O)=O)CC2CCCC(C1)N2C(C1CC12CCOCC2)=O c1(C(C)(C)C)ncc2c(n1)CC1CCC2N1C(=O)CC1CCC(C(F)(F)F)CC1 C12(C(=O)NCCC3(NC(C4CCCC(CF)C4)=O)CC3)CCC(CC1)CC2 C1(NC(c2c(C(C)C)occ2)=O)CCC2(CCCN(C(=O)Cc3cncs3)C2)C1 c1(C(=O)NC(CNC(C=C(CCC)C)=O)(CC)CC)nc2n(c1Br)CCC2 c1(OCC(C)C)ccc(C(N2CC(O)(CCNC(C3(C)CSC3)=O)C2)=O)cc1 C1(c2nnnn2C)(Nc2c(OC)c(C(N)=O)ccc2)CCc2ccccc2OC1 C1(Cc2cn(C3CN(CC(=O)NN4CCCCC4)C3)nn2)CCS(=O)(=O)C1 C(C=CC(=O)NC1(CNC(=O)CNS(N)(=O)=O)CC1)(CC)=CC C1(NCC(C)C2CCC2)CCNCCC1CO N1(C(C(C#N)=CC(C)C)=O)CCC2CN(C(=O)C(C)Cc3cnc[nH]3)CC2CC1 C(CC(F)(F)Cn1cc(CCOC)nn1)CNCCCC=C C1(NC(C(C)OC)=O)CC2CN(C(C3(COCC(F)(F)F)CC3)=O)CC12 CC1CCC1N=c1ccnc(N(CCCn2ccnc2)C)[nH]1 Cc1n[nH]c2cnc(C(=O)NCC3CN(C(C4CC5CCCCC45)=O)C3)cc12 n1(CC)ccnc1C(N1CC(O)(CNC(=O)CC2CCOC2C)C1)=O S(=O)(=O)(c1ccc(Cl)cc1Cl)N1CCC2CN(C(C=CC)=O)CC21 C1(c2cn(CC3CC(CF)C3)nn2)(N(C)C)CCOCC1.C1(C(=O)N)CCCO1 C(C)(C(O)C(=O)NC1CC(NC(c2cccc(N)n2)=O)C1)OC N1(C(CN(C)C(N)=O)=O)CCC(CNC(=O)C=Cc2cn(C)nn2)C1(C)C c1(NC)ccccc1C(=O)OCC(C)C(=O)Nc1ccccc1OC n1(CC)c(N2CCC(Oc3cncc(Cl)n3)CC2)nnc1C(C1(C)CC1)O C1(OC)CCCC(NC(C2CCN2C(C2(NC(C)C)CC2)=O)=O)C1 c1(C(C)(C)NC(=O)NC(C)C(C)(C)C#N)ccc2c(c1)OCCO2 C1(CNC(CC(CCC)O)=O)CCN(C(=O)Cn2ccnc2C)C12CCC2 c1(CNC(CC(=C=C)C)=O)c(C)nn2c1CN(C(c1csc(C(C)C)n1)=O)CC2 C(=O)(C1=C(Cl)CCCC1)NC1(C(N2CC(CC(C#C)C)C2)=O)CCCCC1 Cc1occ(C(F)(F)F)c1C(N1CCC1C(=O)NC(c1cnn(C)c1)C)=O c1(C(=O)NC2(CC)CCN(C(c3cc(C)n(C)c3)=O)CC2)cc(F)c(C)cc1F c1(NCC(F)(F)Oc2cccnc2)nccc(=NCC2=CCCOC2)[nH]1 Cc1nc(-c2cccc(Cl)c2)[nH]c1C(=O)N(C1CC(NC(=O)C2=COCC2)C1)C N1(C(c2nc(C)[nH]n2)=O)CCCC(C2CCCCN2C(=O)CC2CCNC2=O)C1 c1(C(N2C(C)CC(CNC(c3c(NC)scn3)=O)C2)=O)cnc(O)c(C)c1 C(CCC(C)(C)C(=O)N1CC2CCC(C(N3CC(OCC(N)=O)C3)=O)(C2)C1)OC C(=O)(C1=CC2CCC(C1)C2)N1CC2=C(CN(C(C(N=S(C)(C)=O)=O)=O)C2)C1 Cc1ccn(CC(=O)NCC2(CNC(c3cncc(Cl)c3Cl)=O)CC2)c(=O)c1 Cc1cn2c(C(=O)NCC(C)(O)CNC(C3CC3C)=O)cnc2s1 N1(C(c2cncc(C)c2)=O)CC2C(NC(c3ccc(-c4ccco4)[nH]3)=O)CC2C1 N1(C(c2ccc(-c3ccc(C)o3)s2)=O)CC=CC(NC(=O)C(C)CO)C1 c1(OC)ccc2[nH]c(=NCCCC(C)(F)F)nc(N3CCC(OC)C(C)C3)c2c1 N1(C(COC(C)C)=O)CCCC2C1CCN2C(=O)Cc1csc2nccn12 C=C(C)C1OCCC1C(N1CCC(CCC(N2CCCC2C(O)CO)=O)C1)=O c1(C(N2CCC(C(C)NC(=O)CCF)CC2)=O)cc2n(n1)CC(F)C2 Cc1cccc2cc(C(=O)NC3C4CCN(C(=O)CC(C)(C)O)C34)oc12 N1(C(CCCOCC=C)=O)CCCC(OCC2(c3ccccc3F)CC2)C1 c1(C(N(CC(CNC(Cn2ncc(C)c2)=O)O)C)=O)cc(F)c(Cl)cc1F Cc1ccc(Cl)c(OCC(N2CC3CC3(CNC(C3(CO)COC3)=O)C2)=O)c1 C(=O)(CCC1=CCc2ccccc21)N1CCC(NC(C=CC=CCC)=O)C(F)C1 c1(CC(=O)NCc2csc(CNC(c3cnn(CCF)c3)=O)n2)ccc(Cl)cn1 c1(C(=O)NCC2CN(CC)C(=O)C2)cc(Cl)c(Cl)c(C(N)=O)c1Cl c1(C(N2C(CNC(=O)CC3C=CCC3)CC2)=O)ccc(-c2ccccc2)nc1 C1(CNC(C2(CC)CCOCC2)=O)CN(C(C2(CC)CCNC2=O)=O)CC12CC2 Cc1cc(Br)cc(C(N2CCOCC2C2CCC2)C(=O)NC2CC2)n1 Cc1cc(NC(=O)C2CC2)sc1C(=O)NC1CN(C(=O)Cn2cnnn2)CC1F N1(C(C(CC)OCC)=O)CC2(CCC(NC(=O)C(=Cc3c[nH]cn3)F)CC2)C1 c1(CCC)ncc(C(C(=O)NCCCSC)N(CCOc2ccccc2)CC)s1 c1(C(=O)NCC2(O)CCN(C(C(C)(C)C3CCCO3)=O)C2)ccn2ccnc2n1 c1(CC(=O)N(C2CCC(NC(CCCC)=O)C2)C)ncn2c1CCC2 C1(N(C(C(C2CCC2)OC)=O)C)CCCCN(C(c2ccc(C(N)=O)cn2)=O)C1 C1(CC(=O)NCc2c(C(N(c3cccc(O)c3)C)=O)n(C)nc2)CCCC2CC12 C(C(C)C)(C(C)C)NC(C1(NC(CN(C(=O)OCC)C)=O)CCSC1)=O.OCC c1(NC(C2CCN2Cc2cc(F)c(F)cc2Br)=O)cc(Cl)c(O)cc1Cl CC1CC(NC(=O)Cc2cncc(F)c2)CN1C(=O)COC1CC=CC1 c1(C(N2C(CCOC)CN(C(c3cc(Cl)no3)=O)CC2)=O)cc(C)c(C)cc1C c1(C(=O)NCC2C(NC(C(C)NC(C)=O)=O)CC2)ccc(S(=O)(=O)NOC)cc1 C=CC(CC)CC(=O)N(CCCNC(=O)Cc1ccc(CC)c(F)c1)C c1(CNC(C2(C=C)CCC2)=O)cc(C(=O)NCC(C2CCCC2)O)ccn1 C12(C(=O)NC3CN(C(CNC(=O)CC(F)(F)F)=O)CC3O)CCCC(C1)OC2 CC#CCCCC(=O)NCC(C)(C)C(=O)N(CC(=O)N(C)C)CC c1(C(N2CC(C3N(C(CC=C)=O)CCC3)(O)C2)=O)cc([N+](=O)[O-])nn1C C(=O)(CCCC(=O)N1CCC(=CCNC(=O)C(O)C2CC2)CC1)N(CC)CC N1(C(c2ccc(C3(C)CCO3)cc2)=O)CC(NC(=O)CCF)CC12CCOCC2 C1(CNC(CC)=O)CN(C(c2cccnc2OC(C)C)=O)CC1C CC1=C(C)CC(C(=O)NCc2cc(C)c(C(=O)NCc3cccnc3C)o2)CC1 C12(C(N(CCCNC(c3ncc(OCC)nc3)=O)C3CC3)=O)CCC(CC1)OC2 N1(C(CCC)=O)CC(NC(=O)CCC2CC2(Cl)Cl)CC2(CCC2)C1 N1(C(C2C(C)(C)COC2)=O)CC2CC1CN2C(=O)CCOCC(F)(F)C(F)F C12(NC(=O)CNCC3(O)CN(C(=O)CC4C=CCC4)C3)CC3CC(CC(C3)C1)C2 N1(C(c2nc(CCC)oc2)=O)CCC(C)(C)C(NC(c2ccc(OC)cc2)=O)C1 CCCCCC(=O)N(CCC(=O)NCCC(=O)NC1CC1)C(C)C c1(C(N2CCC(CN(C(c3c(C)scc3)=O)C)C2)=O)ccc2c(c1)CC2 CC1(C)CC(CO)N(C(c2ccc(CNC(C3CC3[N+](=O)[O-])=O)nc2)=O)C1 C(=O)(CCC(C)O)NC(CNC(CCN(CC)CC)=O)C(C)C c1(OC)ccc(C(C)C(N2CC(NC(=O)Cc3cnc(C)o3)C(C)C2)=O)c(C)c1 Cc1ncc(C(=O)NC(Cc2ccoc2)C(=O)NCC(C)CO)n1C C1(C(N2C3CC(C(N4CCCC5(CC5)C4)=O)C2CC3)=O)C2Sc3ccccc3C12 N1(C(C(CC)n2cncn2)=O)CCC2(CCCN2C(=O)CCNC(=O)C=CCl)C1 N1(CCc2n(C)ncc2)CCCCC(N=c2nc[nH]cc2C#N)C1 c1(N(C)C)nc(Cl)c(C(=O)NCCCCCNC(C2(CO)CCOC2)=O)s1 C1(NC(c2n(CCCC)ncc2)=O)CC(O)CN(C(=O)CC2CCC=CCC2)C1 N1(C(C(CC)(F)F)=O)CCCC(F)(C(=O)NCCOCCOCCO)C1 N1(C(c2c(OC)nc(C)cn2)=O)CC2(CCCN(C(C3CC3Cl)=O)C2)C1 c1(COC)cc(C(=O)N(CC(C)NC(c2snnc2C2CC2)=O)C)n[nH]1 C1(NC(c2nc(CCC)oc2)=O)CC2CC(C1)N(C(C1(C)CC(O)CN1C)=O)C2 C1(NC(=O)C(F)C2CCOC2)CC1C1CCCN(C(c2c[nH]cc2C2CC2)=O)C1 N1(C(c2ccc[nH]2)=O)CC(NC(C23CC(CO2)C3)=O)C(O)C1 C1(CC)(Nc2nccc(C(C)(C)C)n2)CCN(C(C2(CCO)CC2)=O)CC1 CCC(C)(CNC(c1cc(C)sc1N)=O)C(=O)N1CC(C)(O)CO1 C1(NC(CCCOCC#C)=O)CCCC12CN(NC(C1(C(=O)OC)COC1)=O)C2 N1(C(C(C=C)c2ccccc2)=O)CCC(C)C(NC(=O)CC(C)(C)CC)C1C Cc1cnc(C(=O)NC2CCCC(N(C)C(C3CCC(C(C)C)CC3)=O)C2)cn1 N1(C(CC2C(C)CN(C(C3CC4(CC4)CO3)=O)C2)=O)CC(C)C(F)(F)C1 C=CCC(CC(F)F)NC(C1C(CC)CCCN1C(=O)COC1CCOCC1)=O CC(C)CCC(C(=O)N(C1CC(OC)C1)C)NC(=O)CCC(C)(C)N(C)C N1(C(Cc2c(C)ocn2)=O)CCOC(CN(C)C(C2CCC(=O)N2C)=O)C1 N1(C(C(C=C)C)=O)CCN(C(=O)CC2CC3(CCC3)C2)CC(C)(F)C1 C1(NC(C2(CCCC)CCCC2)=O)CCC(C)N(C(=O)Cn2ccnn2)C1 CC1CN(C(=O)C(C2(O)CCCC2)F)CC1NC(=O)Cn1cc(C#N)cn1 Cc1ccc2nnc(CNC(=NCCC(C)C)NC3CCOC(C)C3)n2n1 N1(C(c2c(C)n(C)c(-c3ccccc3)c2)=O)CC23CCCC2(COC3)C1 C(=O)(C1CCc2cccc(OC)c21)NC(CC=C)CNC(=O)Cn1cc(Cl)cn1 CC1(C)CC(C(=O)NC2CCC2O)CCN1C(=O)C=CC(F)(F)F Cc1[nH]cc(C(=O)NC2CN(C(=O)C(C)C3(O)CCC3)CC2(C)C)c(=O)c1Cl C1(C(=O)NC(CN(C(c2occ(C)c2)=O)C)(C)C)CC12CC(O)C2 C#CC1(C(=O)Nc2ccc(OC)nc2)CCN(C(=O)C#CC2CC2)CC1 C(=O)(CCCCNC(=O)CCC1CCCCN1C(c1ccc(F)s1)=O)OC(C)(C)C N1(CC(=O)Nc2ccc(-c3nc(C)sc3)cc2)CCC2(CC1)CC(CO)=NO2 C1(C(=O)NCCN(C(C2(O)COC2)=O)C2CC2)CCCC1n1cccc1 C1(CNC(C2COC3COCC23)=O)CCC2(CN(C(=O)CC3CCOCC3)C2)O1 Cc1ncc(N)cc1C(=O)NCC=CCNC(=O)Cc1n[nH]cc1Br c1(C(=O)NC2CN(C(C(C(CC)O)(F)F)=O)CC2O)sc2cccc(F)c2c1Cl C1(NC(c2c(C)ncn2C)=O)CC2CC(C1)N(C(c1ncsc1S(N)(=O)=O)=O)C2 Cc1nccc(CNC(=O)C=CCC(C)(C)NC(=O)Cc2cc[nH]n2)n1 C(=O)(CCCC(CC)NC(=O)C1=C(C)OCCS1)N1CCC(CC)C1 c1(C(N2C(CNC(C(C=CC)O)=O)CCC2)=O)cnc2cnn(C)c2c1 C1(C(=O)Nc2scc(C)n2)CC12CCN(c1ncnc(C)c1Br)C2 N1(C(c2ccc(OCOC)cc2)=O)CCCC(SC)CC1 C(=O)(C=C1SCC(=O)N1C)N1CC(NC(C(CC=CCC)C)=O)C(OC)C1 C12(C(N3C(C=C)CCC3)=O)COCC1CN(C(c1n[nH]cc1CC)=O)C2 c1(N2C(C)(CNC(C(C)NC(C)=O)=O)CCC2)ncc([N+](=O)[O-])cc1F CCCC(C)(C)C(=O)NCC1(O)CCCN(C(c2nccc(Cl)c2O)=O)C1 C1(NC(CCSCC)=O)CC2CCC(C1C)N2C(=O)CCOCCOC C1(OC)CC(CNC(C2(CO)CC2)=O)N(C(=O)C=Cc2cn(C)nn2)C1 n1(CCC)nc(-c2cscn2)nc1-c1cscc1OC c1(CCC(=O)NCC(C)(O)CNC(C2CCC23CCC3)=O)c(F)cccc1F c1(NC(C2(C)N(C(c3cc(C)on3)=O)CC2)=O)ncc(Br)nn1 C1(C(N2CC(C(=O)NCC(C3CCCCC3)C)(SC)C2)=O)CC2C(C1)C2(C)C C1(NC(=O)CN2CCCC2)C2CN(C(c3csc(C(F)(F)F)n3)=O)CC12 C(=O)(CCCCC(C)(C)C)NC1CC(C(C)NC(C(C)NC(C2CCC2)=O)=O)C1 C1(C(=O)N(CC(O)C2CCC2)C)(SC)CN(C(c2ccc(Cl)s2)=O)C1 C(C1CCCC1)=C(C)C(=O)NC(C)C(=O)NC(C)Cc1nn[nH]n1 c1(CN(C(CN2CCC(CCCC)C2)=O)C)ccccc1Cl C1(NC(c2cc(C)nn2C)=O)CCN(C(c2sc(=N)[nH]c2C)=O)C(C)C1 N1(C(C(C)NC(=O)NC)=O)CC2CCC1CC2NC(C1CCC(F)(F)C1)=O N(C(=NCCCOc1ccc(F)cc1)NCC1CCCOC1)C1C(C)C1 N1(C(=O)Cc2ccsc2)CC2CC1CN2CC1CCCCO1 Cc1nn(-c2ccccc2)cc1C(=O)NC12CC1CN(C(c1cc[nH]c1C)=O)C2 C1(NC(c2ccc(C)cc2)=O)CCN(C(=O)CC#N)CC1(C)C c1(C(=O)NCC2C(C)CN(C(c3cccnn3)=O)C2)cc(S(C)(=O)=O)ccc1Cl C1(CCC(=O)NCC2N(CC(=O)N(C)CC)CC2)CCCN1C CCC(C(=O)NC(C1CCN(C(c2[nH]nnc2C2CC2)=O)C1)C)c1ccccc1 C1(CNC(c2c(C)nns2)=O)CN(C(=O)CCc2nncs2)CC1O C(=O)(C(N=[N+]=[N-])C(C)C)N1CCC(CC)CC1C(=O)N(CC(F)F)C c1(C(N2CC(NC(c3cnc(CC)[nH]3)=O)C(C)CC2)=O)ccc(Cl)cc1[N+](=O)[O-] C1(NC(C2(C)CN(C(C3CCC(CC)O3)=O)C2)=O)CN2CCC1(C)CC2 CC1(C)CCCC(NC(c2ncoc2CNC(C2CC3(CC3)CO2)=O)=O)C1 C1(C(N2C(CCNC(=O)CC3CCC(=O)N3)CSCC2)=O)COC2COCC12 C(CC(=O)NCC(C)(CC(C)C)NC(c1cnn[nH]1)=O)(C(F)(F)F)OC c1(N(C)Cc2ccc(OC)nc2)nc(N2CCC(F)CC2)nc2c1COCC2 c1(N2C(=O)CC(NC(CCC#C)(C)C)C2)ccc(Cl)c(Cl)c1 C1(NC(c2ccc(CN(CC(N)=O)C)cc2)=O)CCOC12CCOCC2 c1(C(c2nnnn2C2(C)CC2)NCC2C(CCC)C2)cnn(-c2ncccn2)c1 C1(C(N(C2CCN(C(=O)CC3(O)CCCOC3)C2)C)=O)CCC(C(F)(F)F)CC1 Cc1c(C(N2CCOCC(CNC(C3(C)CCCN3C)=O)C2)=O)sc2cncn12 CC1CN(C(c2csc([N+](=O)[O-])c2)=O)CC1(C)CNC(=O)C(c1ccccc1)F C1(CC(=O)NC(C(C)n2cccn2)C)CCCCN1C(C1OC2CCC1C2)=O N1(C(C2C(=C)C2)=O)CC2CCC1CC2NC(=O)C(C)(C)CF CCCC(C(=O)NOCCCN(C)C)NC(c1cnc(O)n1CC)=O C1(C(=O)NC(CNC(c2cnn(C)c2Cl)=O)C2CC2)Cc2cc(F)ccc2O1 C(=O)(C(CC(C)C)CC(C)C)NC(CCNC(c1cc(C)c(Cl)cc1)=O)C(C)C Cn1nc2c(c1C(N1CC3C(NC(=O)CCc4cnn[nH]4)C3C1)=O)CSCC2 CC1CCCN(C(=O)C2=CCOC2)C1CCNC(=O)CNC(c1ccncc1)=O c1(C(=O)NC2CCC(NC(C(CC(=C)C)C)=O)C2)cc(S(N)(=O)=O)cs1 CCCC(CC)CCC(=O)NCC1(O)CCCN(C(C2(C)CC=CC2)=O)C1 N1(C(C(CNC(CCCCC=C)=O)C(C)C)=O)CCC(C2CCC2)CC1 C1(CC(=O)NC)CN(C(C2CSCCN2C(=O)C(C)Cn2cccn2)=O)CCO1 C(=O)(CC1=NNC(=O)C1)NCC1(C)CCCN1C(c1cc(Cl)nc(=N)[nH]1)=O Cc1cc(F)c(C(=O)NC(C)CCNC(=O)CSCC(F)(F)F)cc1Br C1(C(=O)NCC(C)N(CC)CC)CCN(C(c2ccoc2)=O)C1 C1(C(=O)NCCc2ncc(C)o2)CC2(CCN(C(=O)C(N3CCNC3=O)C)C2)C1 c1(C(N(CCNC(c2c(Cl)ccc(OC(C)C)n2)=O)C)=O)ccc2ccsc2c1 CC(=O)C(C)(C)CC(=O)NC(Cc1cc[nH]n1)C(=O)NCC1(C)CCN(C)C1 c1(C(=O)NCC(C)C(=O)O)ccc(F)c(-c2cn(C3(C(=O)O)CC3)nn2)c1F c1(C(=O)NC2C(OC)COC2)oc(CNC(C2(CO)CCCC2)=O)nc1C C#CCC(C(=O)NC(c1cnn(C)c1)C)NC(c1coc(C(C)C)n1)=O C1(F)(C(=O)NCC(C)(C2CC2)NC(=O)Cc2cnc[nH]2)CC1(F)F CC(O)CCCCCC(=O)N(CCN1CN(CO)C(=O)C1C)Cc1ccccc1 C1(NC(C2(CCCC)CCC2)=O)CN(C(c2cccc(CF)c2)=O)CC1O c1(C(=O)NCCC(CNC(c2c(C)ccnn2)=O)O)c[nH]c(=N)nc1C N1(C(CNC(=O)NC)=O)CCN(C(c2cc(O)nc(C)n2)=O)C(C(F)F)C1 CC(C)CCCC(C)C(=O)N(C)CC1CCN(C(C2COC(=O)N2)=O)CC1 C1(NC(=O)CCC2CCC2)CCCC2CN(C(=O)CNS(N)(=O)=O)CC12 CCCC(C)C(=O)N1CCC(F)(C(=O)Nc2nccnc2C)C1 c1(OC)ccc(C(N2CCC(C)(C(N3CCC(C)(O)C3)=O)CC2)=O)c(F)c1 C1(NC(C(CCN(C)C)O)=O)(CO)CCCN(C(=O)C(c2cccc(N)c2)O)C1 N1(C(C(C(CC)CC)C)=O)CC(CNC(=O)C=Cc2ncc[nH]2)OC2COCC12 C1(C(=O)NCCN(C(c2cc(COC)on2)=O)CC)CCOC(C)C1 CC1CCN(C(C2CC(NCc3cc(Br)c(F)cc3F)C2)=O)CC1(F)F C1(NC(=O)CCC2CCCC2)CN(C(C2(CC3CC3)CCCO2)=O)CC1F c1(OC)ccc(CC(=O)NC2CC(F)CN(S(=O)(=O)C(C)COC)C2)cc1F C1(NC(C(C)N2CCC2)=O)C(C)CCN(C(c2cscc2C(F)F)=O)C1C C(C1=CCN(C(C2(F)CCCCCC2)=O)CC1)NC(c1ncccc1C(F)F)=O C(CC(=O)NCc1cccc(CO)c1)(C(C)C)NC(CSCC#C)=O C1(C)(C(=O)NCCOCCN(C)C(C23CCC(CC2)C3)=O)CCCS1(=O)=O C1(CNC(=O)C(O)C2CC2)COCCN1C(C1CCCC1Cc1ccccc1)=O C1(NC(=O)CCOCC(F)(F)F)CS(=O)(=O)CC1N=c1ccnc(C2CCC2)[nH]1 N1(C(c2c(NC)snc2C)=O)CC(NC(=O)CCc2ccccc2)CC(O)C1 C1(CNC(CC2(C=C)CC2)=O)CC(NC(c2cn(C3CC3)nn2)=O)C12CCC2 c1(C(N2C(C(=O)NC(C(C)C)CO)CCC2)=O)cccc2ccoc12 N1(C(C(C(C)C)O)=O)CC(CNC(c2nccc3ccsc23)=O)OC2(CCC2)C1 C(c1ccc(C#N)cc1)=CC(=O)NC1CCC(C)N(C(c2cccc(=O)o2)=O)C1 N1(C(C=C(C)CCc2ccccc2)=O)CC2OCC(NC(=O)C3=CCCS3)C2C1 CCC(O)C(F)(F)C(=O)NCCC1CC(NC(c2csc(-c3ncc[nH]3)n2)=O)C1 c1(NC(C(c2cc(O)cc(Cl)c2)N2CCC(NC(C)=O)C2)=O)ccc(Cl)cc1F C1(C(N(CC(C)N(C(C(C2CC2)SC)=O)C)C)=O)CC2(C1)OCCO2 c1(C(N2C(CNC(c3c(CC)noc3)=O)C(C)CC2)=O)cncc(S(N)(=O)=O)c1 N1(C(c2c(C)n(C)nc2)=O)CC(F)(F)CC1(C)CNC(=O)Cc1ccnnc1O C1(NC(C=CC)=O)CCC(N(C(=O)C(C(C)C)Oc2ccc(Cl)cc2)C)CC1 C12(C(N3C(CNC(c4ncsc4C4CC4)=O)CCCC3)=O)CCCN(CCC1)C2 c1(C(N(CC(N2CCC(C)(C(C)C)CC2)=O)CC(=O)O)=O)ccccc1[N+](=O)[O-] C12(CNC(=O)Nc3c(C)c(Cl)ncn3)CCC(CC1)C(C)(C)O2 N1(C(c2cnc(C(=O)OC)s2)=O)CCOC(C(C)NC(=O)CC2CCCC2)C1 Cc1[nH]nc2c1CC(C(N1CC(CNC(=O)CCCCNC(N)=O)C1)=O)CC2 CCCC(C(=O)NC1CCN(C(=O)C=CC(=O)OCC)CC1F)S(N)(=O)=O Cc1ccnc(N2CCC(C(C)NC(=O)Cc3sc(C4CCC4)nc3C)C2)n1 CC1CN(C(c2ccc(CNC(=O)CS(C)(=O)=O)cc2)=O)CCC1O C1(C(N)=O)CCCCN1C(C1C=CC(NC(=O)Cc2cccnc2)C1)=O Cc1cc(C(=O)NC2COCCC2NC(C2CCC(C)(C)CO2)=O)cc(C)c1N CCC(CC)(CN=c1c(C#N)c[nH]c2c(C)cc(F)cc12)OC c1(C(N(C2CN(C(C(CC=CC)CC)=O)CC2(C)C)C)=O)[nH]cc2c1CCCC2 c1(C(N2CC(C)(NC(C(CC)C(C)C)=O)C2)=O)cc2c(o1)CCCNC2=O C12(C(=O)NC(C)CCO)CCC(CC1)N(C(=O)Cn1cccn1)C2 CCCCCC(=O)NCC(N1CCCC1(CNC(C1CCC(C)CC1)=O)COC)=O c1(C2C(C(N(CC(C)NC(=O)C(=Cc3c[nH]cn3)F)C)=O)C2)ccc(Cl)nc1 Cc1ccc(C(=O)NC2CCOCC2NC(=O)CCNC(C2CCC2)=O)c(F)c1 c1(OC)cc(C(=O)NC(C)CCCNC(c2ccc(N(C)C)nc2)=O)ccn1 C(CC(C)C(F)(F)F)NC(=O)NCC1CC(C)SCC1 C1(NC(c2ccc(C)cn2)=O)CCC2CN(C(c3cc(Cl)cnn3)=O)CC2C1 c1(C(N2CCC(CNC(CCc3ccc(C)s3)=O)C2)=O)cnn2c1CCCN2 N1(C(C(COC)O)=O)CC2(CC(NC(c3cnc(OC)cc3C)=O)CO2)C1 c1(C(=O)NC(C2(O)CN(C(C3CC(F)CN3C)=O)C2)C)c[nH]c2ccc(F)cc12 C(=O)(C1=Cc2ccccc2OC=C1)N1CCC(CN(C(C(C=CC)O)=O)C)C1 Cc1ccn2ncc(C(=O)NC3CC(NC(c4cc(CO)[nH]n4)=O)C3)c2c1 C1(CNC(c2csc(S)n2)=O)CCN(C(C2CCN(C3CC3)CC2)=O)C12CC2 C1(C(=O)NC23C(NC(C(C)=C4CC4)=O)CC(CC2)C3)CCn2nnnc2C1 C#CC(CC(C)(C)C)NC(c1[nH]ccc1CNC(C1(C)CC(C)(C)C1)=O)=O N1(C(c2cc(C3CCCC3)no2)=O)CCCC(N(C(=O)CCC(F)F)CCO)C1 c1(C(C)(C)C)ccncc1NC(C1CC(c2cccc(F)c2)(F)C1)=O N1(C(CC2(CC=C)CCCC2)=O)CCC2CCN(C(c3c(C)[nH][nH]c3=N)=O)CC12 c1(NC2C(NC(C3(C(=O)NC)CCC3)=O)CCCC2)cc2nncn2c(C)n1 Cc1nc(-c2ccccc2)oc1C(=O)NC(C)CNC(=O)CC(C)CN(C)C Cc1cc(C(=O)NCC(=O)NCC2CC2NC(C2C3CNC(=O)C23)=O)n(C)n1 CCCC(CCC)C(=O)N1CCC(NC(c2c(F)ccc(Cl)c2F)=O)CC(O)C1 C1(CNC(COCCOCCOC)=O)C(O)C(O)CN1C(=O)CCS(C)(=O)=O N1(C(CCC2N(C)CCC2)=O)CC2CC2(CNC(=O)C(C)(C)c2cc[nH]n2)C1 C=C(C)C1OCCC1C(=O)NC1C2CC1N(C(c1cnncc1C)=O)C2 C1(NC(C2C(C)OCC2)=O)CCN(C(C2CNC(=O)C2)=O)CC1(C)C C(=O)(CC(C(=C)C)OCC)N(C1(C(N(C(CC#C)C)C)=O)CCC1)C1CC1 C1(C(N2CCC(CN(C(=O)Cc3cnsc3)C)C2)=O)CC(c2ccncc2)=NO1 C1(CNC(c2c(C)n(C)nn2)=O)CN(C(=O)CC2CCCOC2)CCN1C N1(C(C=C(C)CCc2ccccc2)=O)CC(NC(=O)CC(C)C)CC(C)(C)C1 C1(C2CCCC2)(NC(C2C(NC(C3CCC=CCC3)=O)CCO2)=O)CC1 c1(SC(CC)C(N2CCCC(CCCC#N)C2)=O)ncnc2c1ncn2C1CC1 C=CC1CCCN1C(=O)C(C)(CO)NC(C1COCC1C(N)=O)=O C(=O)(C(O)C(F)(F)F)N(C)CCNC(=O)CCc1cc[nH]n1 c1(OC)cccc(C(=O)NC2CCN(C(=O)C(O)CC3CC3)C2C)c1F CC1CN(C(C2OCCC2NC(=O)CC2CC(F)C2)=O)CCC1(F)F C1(C(C)NC(=O)CCSc2cccs2)CCN(C(=O)CC(=O)N(C)C)CC1 N1(C(CN(C2CC2)CC)=O)CC(C)(CNC(=O)C(c2ccnn2C)C)CC1(C)C c1(CC(=O)N(C(CNC(C2(CC)CCOC2)=O)C)C)sc(C2CCCC2)nc1C C(=O)(C1=NOC(CNC(c2ccc(C(N)=O)[nH]2)=O)C1)N(CCOCC)C N1(C(C(=O)NCC)=O)CC(C)C(NC(=O)Cc2c[nH]c3ccccc23)C(C)C1 C1(CC=CC)CCCN(C(c2ccc(Br)cn2)C(=O)NCCCC2CC2)C1 CCC(COC1CCCC1)N=c1[nH]c(=NCC(CC)C2CC2)[nH]c2cc[nH]c12 N1(C(C(C)OC2CCCC2)=O)CC(O)C(O)C1CNC(=O)C(C)(F)F N1(C(C2CC(=O)NC2)=O)CCCCC12CCCN(C(C1CCCCO1)=O)C2 N1(C(C2C(=O)NCC2)=O)CC2CCN(C(=O)Cn3nccn3)CCC2C1 C(=O)(CC(C)(F)F)NCC(CN(C)C(c1ccc(CS(C)(=O)=O)o1)=O)O c1(CC(=O)NCCCCCNC(c2ccc(C(C)=O)o2)=O)ccc2[nH]ccc2c1 O=C(C1c2ccccc2CN1C(c1csc(Br)c1)=O)NCCCCCCCCO c1(CC)ncc(COC(=O)Cc2cccc(NS(C)(=O)=O)c2)cc1C C(=O)(C1=CCC2CCC1N2C(=O)Cc1ncccc1F)N1CCC(C)(F)C1 c1(OCC(=O)NC(CNC(=O)CSC2CC(N3CCCC3)C2)CO)cccnc1 CCCCCCCCC(C)C(=O)N1CCCC(C2CN(C(=O)C(C)C(C)O)C2)C1 C1(CCNC(c2cc(CCC)ncc2)=O)C(C)CCCN1C(c1cc(Cl)c[nH]1)=O C(=O)(C(C)CCC(C)(C)C)NCC(C)(CO)NC(Cc1ccc(SC)cc1)=O c1(OC)cncc(CCC(=O)NCC(O)CCNC(C2CCCC2C(C)C)=O)c1 N1(C(CC(=O)NC)=O)CCC2(CCCN(C(c3cc(C#N)ccc3C)=O)C2)C1 N1(C(C(=O)NC(c2cnc(Br)s2)C)=O)CCC(c2ccccc2)CC1C Cc1cc(-c2ccc(CN(C)Cc3ccncc3)cc2C)ccc1C=O c1(C(=O)NCC(CC)NC(c2ccccc2COC)=O)c(C)nn(CC)c1Cl Nc1c(C(=O)NCCNC(c2[nH]nnc2-c2ccccc2)=O)cccc1F C1(C(C(C)NC(C2(Br)CC2)=O)NC(CC)=O)CCCCC1 c1(C(=O)NC2C=CCN(C(C3CCC(C)(C)C3)=O)C2)cscc1S(C)(=O)=O C1(NC(C=C(C)C2CC2)=O)C(CNC(c2cnn[nH]2)=O)CCC12CCC2 c1(NC2(COCC)CC2)cc(SC)cc(N)c1.C1CO1 C(=O)(C(F)C1=CCCCC1)N1CC2CN(C(c3c(C)nsc3N)=O)CC2C1 C1(NC(C2CC(C)(C)C2)=O)CCN(C(=O)CCCCNC(N)=O)CC1O N1(C(C=COCC)=O)CCN(C(C2CCC(=O)N(C(CC)CC)C2)=O)CCC1C c1(C(N2CCC(COC)(NC(=O)CCc3nnc(C)o3)C2)=O)cc2n(n1)CCC2 c1(NC(c2c(C)n(C)nc2N(C)C)=O)nn(C)c2ccccc12 N1(C(C(COC)(C)C)=O)CCCC2(C1)C(NC(=O)C1=CSCCO1)CCN2C C#CCC(C)(C(=O)Nc1cc(C)cnc1O)NC(=O)CC1CCC(C)(C)O1 N1(C(c2n(C)ccn2)=O)CC2CCC1C1CN(C(=O)CCc3ccnn3C)CC21 c1(C(N2CC(CNC(c3c(C)csc3)=O)OCC2)=O)cc(Br)c(F)cc1F C1(c2cccc(Cl)c2)(C(=O)NCC2C(NC(C(C)SCC)=O)CC2)CCCCC1 c1(C(=O)NC)ccc(C(=O)NCc2c[nH]nc2C2CCN(C(=O)C(C)O)C2)cn1 C(CCCCC(=O)NCC1(C)CCCN1C(=O)Cc1ccc(F)cc1C)OC NS(=O)(=O)c1cc(C(=O)NCCCN(C(=O)C(F)(F)CO)C2CC2)co1 n1(C(C)C(=O)N(C2CCCS2)C)cc(C2(O)COC2)nn1 N1(C(C2C(C)CCO2)=O)CCOC(C(=O)NC(C2CCOC2)CO)C1 N1(C(CC2CN(C)C(C(F)(F)F)CC2)=O)CCC23CCCCC2(C1)C3(F)F N1(C(C(=C)F)=O)CCC12CN(C(c1ccccc1OC)=O)C2 c1(OC)nscc1C(=O)NCc1cc(C(=O)NCCCCCC2CC2)no1 c1(C(=O)NCC(C(=O)N(c2ccc(OC)cc2)C)OC)ncnc(O)c1F C(CC(C(=O)NC(C)C(O)C(F)F)NC(=O)C(O)Cn1cncn1)OCC c1(C(=O)NC2CC(NC(=O)CCc3nnc(C(F)F)o3)C2)snc(Cl)c1Cl c1(C(=O)NC2CCN(C(C(C)OCC#C)=O)C2(C)C)ccc2c(c1)B(O)OC2 c1(C(=O)NC2(C3N(C(C4C(CC)C4)=O)CCC3)CC2)c(OC)ccc(OC)c1N N1(C(=O)Nc2csc(Br)c2)CC(CO)CC12CCOCC2 CC1(C)CCN(CCNC(c2ccc(CNC(C3CC(=O)C3)=O)o2)=O)C1 c1(C(C)=O)ncc(C(N2CCC(C3CCCN3C(=O)CC3CC(C)(C)C3)C2)=O)s1 C1(c2nc(C3C(C)(COC)C3)on2)(c2ccncc2)CCCCC1 c1(OC)ccc(C(=O)NC2CC3CC2N(C(=O)C(C)(C)C#N)C3)cc1C(F)F CCCCCCCCC(=O)N1CCOCC1CN(C(=O)C(C)(CC)CO)C CC1(C)CCCC1CNC(c1[nH]ccc1-c1ccccc1)=O C=CCCCC(C(=O)NC(CC)C(C)(C)C)NC(=O)COCCF c1(NC(=O)NNC(=O)c2ccccc2Br)cc(F)c(F)c(F)c1 C(=O)(CCCNC(c1cccnc1)=O)NC(C1CN(C(C23COC(C2)C3)=O)C1)C c1(C(=O)NCCC2CN(C(=O)C3=CSCCO3)CCO2)ccnc2ccccc12 C#CC12CCC(C(=O)NC3CN(C(=O)CC4CC(=O)C4)CC(C)(C)C3)(CC1)CC2 C(CNC(C1(C2CCCO2)CC1)=O)(CCOC)NC(CC1(OCC)CCC1)=O C1(C(=O)NC2C3CN(C(CC4CC(=O)NC4)=O)CC2C3)CCCC2(C1)CC2(F)F CC(C)S(=O)(=O)c1ccccc1NC(=O)CC1(C)CCN1Cc1cccnc1Cl N1(C(c2ncn(CC)c2)=O)CCC2(NC(c3ccn4ccnc4n3)=O)CCCC12 c1(C(=O)NC2CCN(C(C3CC(C)N(C)C3)=O)CC2)c[nH]c2ccncc12 c12cccc(c1)NC(=O)C2C.C1(C(N(C(=O)OC)C(C)C)C)CCC1 N1(C(C=Cc2nc(C)c(C)[nH]2)=O)CCCC2CN(C(=O)CC(O)CN(C)C)CC12 C12(NC(=O)CN3CC=CC3)CCOCC1CN(C(c1cccc(CO)c1)=O)C2 c1(NC(C2CCOC2CNC(C2C3CCC(=O)C23)=O)=O)ccc(CO)cc1 CC(C(=O)NCC1CN(C(C2(C)CC=CC2)=O)C1)S(N)(=O)=O CCC(C)C(C(=O)NC1CC(NC(c2coc(-c3ccccc3)c2)=O)C1)OC c1(C(=O)NC2C(NC(c3cn(CCC=C)nn3)=O)COC2)cncn(C)c1=O N1(C(c2oc(C(=O)OC)c(C)c2)=O)CCCC(CO)(NC(=O)COCCF)C1 C1(COC)CN(C(c2c(C3CC3)noc2C)=O)CCN1C(c1cscc1C)=O C(=O)(C1=NOC(C)C1)NCC1CN(C(CCOc2c(CC)cccc2)=O)CC1C C1(C(N2CC(C)CC(NC(c3c(C)coc3C)=O)C2)=O)CCc2nncn2C1 C1(NC(C(C(C)C)OC)=O)CCN(C(c2sc(C(C)(C)C)nc2C)=O)CC1F Cn1cnc(CC(=O)NCC(C2CCOC2)NC(=O)COC2CCC2)c1 c1(C(N2CC(CCNC(C(C(CC)C)O)=O)C2)=O)ccc(F)c(S(N)(=O)=O)c1 c1(NCCCC)ccccc1C(=O)NCC(C1CCC1)NC(=O)CCC(C)OC CC(C)CCC(=O)NCC(=O)NC1C=CCN(C(=O)CSC2CCOC2=O)C1.OC n1(CC)c(CNC(=O)CN(C(=O)CC2CCOCC2)C2CC2)nnc1O C(=O)(C(CC(C)C)OC)NCC12C(CN(C(c3c(CC)nc(C)[nH]3)=O)C1)C2 c1(OC)ccc(CO)cc1C(=O)N(C1CCC(NC(c2cc(=O)cc[nH]2)=O)C1)C c1(C(N2CCC(OC)(CNC(C3CC=CCC3)=O)C2)=O)ccc(S(C)(=O)=O)s1 C1(NC(C(OC)OC)=O)CCN(C(C2CC3CC2C3)=O)CC1O Cn1ncc(NC(C2COC(CNC(=O)CC3(C)CC3)C2)=O)c1Cl c1(C(=O)NCCCN(C(=O)C(C)OC)CC)ccc(C(N)=O)cc1[N+](=O)[O-] C1(CCNC(c2cc(C(F)(F)F)no2)=O)CCCN(C(=O)CC2CCOC2=O)C1 CC1CCCCC1(CNC(=O)Cc1cnccn1)NC(=O)CCCN=[N+]=[N-] c1(C(=O)NC2CCC(CNC(c3occ(C)c3C)=O)CC2)ccc2nccn2c1 c1(C(N(C2(CNC(=O)CC3(C(F)F)CC3)CC2)C)=O)cnco1 C1(C(=O)NCCC2CC(NC(c3ccc(=O)oc3)=O)C2)CC2CCC1O2 C(C)(C(=O)NC1CCN(CC(=O)Nc2ccc(C)cc2C)C1)(C(C)C)OC C#CCC(C)(C)C(=O)N(CCNC(=O)C(CCSC)NC(N)=O)CCOC C1(CC)CN(C(=O)C=CCN(CC)CC)CC1C(=O)Nc1ccccc1Cl CC1(C)CCC(C(=O)NC2C3CN(C(=O)C(C4CC4)C4CC4)CC23)O1 c1(C(=O)NC(C(C)NC(C2SCCS2)=O)C)ccncc1C(F)F CC(CN(C)C)C(=O)N1CC(C(O)C(=O)N(C)CCF)C1 c1(C(=O)NC(CC)(C)CNC(=O)CC2C=CCCC2)cc(COC)c(C)s1 C1(NC(C2(CNC(C3(NC(C)=O)CC3)=O)CCCC2)=O)CC(C)(C)C12CC2 C(CC(=O)NCCC(C)OC)(C(F)F)NC(C1(CC)CC(C)(C)C1)=O C1(C(=O)NCC2(C)N(C(c3cc(C)sn3)=O)CCC2)CCc2ccnn2C1 c1(N(CCOC)CCNC(=O)CCN2C(=O)CCC2=O)nccc(C)c1[N+](=O)[O-] c1(NC(C2C3CC2N(C(=O)CCc2ccc(Br)c(F)c2)C3)=O)ncc(Cl)cc1O c1(C(=O)NCC2CCN(C(=O)Cc3ccc(Cl)cc3F)C2)ccc(Cl)c(Br)c1 c1(C(=O)NCC=CCNC(C2CCN(C)S2(=O)=O)=O)cc(F)c2ccccc2c1 N1(C(C(C=C)(C)C)=O)CC(CC(=O)NC2CN(C)CC2C)C2(CC2)C1 C1(NC(COC)=O)CCN(C(c2cc(Br)sc2Cl)=O)C(C)C1 O=C(C1=CC2CCCC12)N1CCN(C(c2ccc(-n3cccn3)c(Cl)c2)=O)CC1 C(=O)(CCCCCS(N)(=O)=O)NCC1CN(C(c2ccc(OC(C)C)nc2)=O)C1 C(=O)(CC(O)CC(C)(C)C)N1CC2N(C(c3n(CC)ncn3)=O)C(CC2)C1 C=C(C)CCN=C(NCCc1ccc(Cl)c(F)c1)NCc1cccs1 N1(C(c2cnn(C(C)CC)c2)C(=O)NCC)Cc2ccccc2C1CCO CCCCC(CC)CC(=O)NCc1cc(C)c(C(=O)NC(CCC)C(F)(F)F)o1 N1(C(C2C(C)OC(C)C2C)=O)CCC(NC(=O)CCCCCO)C2(CCC2)C1 C1(CNC(CCCCOCC)=O)COCCN(C(=O)C2=CCCCC2)C1 N1(C(C(CC)SC)=O)CCCC1(CNC(=O)C(C)(C)c1cccnc1)COC C12(CNC(=O)CC3=CCCC3)CCCCC1N(C(=O)COc1ccccc1)CC2 N1(C(C2(C)CCCS2)=O)CCC(O)C(NC(c2cc(C3CC3)ccc2F)=O)C1 N1(C(c2n(CC)nc(C)c2)=O)CC(CNC(c2cnc(SC)s2)=O)CC1(C)C N1(C(=O)CC2CCC3(CCC3)O2)CCCCC2(C1)CN(C(C1CCCS1)=O)C2 C1(OC)CS(=O)(=O)C2CN(C(=O)NCC(c3cc(Cl)sc3Cl)(F)F)CC12 Cc1cc(C(N2CCC(CN(C(=O)COCCCF)C)CC2)=O)c(C)nc1C c1(CNCC(C)C2CNC2)ccccc1CNS(C)(=O)=O CCC(C)C(C(=O)NC1CN(C(C)C)CC1C)N(C(=O)C=C(C)COC)C c1(C(CC)NC2CCN(c3ncco3)CC2)ccc(Cl)c(F)c1 C(=O)(CCCCC(F)F)N1CC(NC(c2ccccn2)=O)C2C1C2 c1(C(N2CC3C(N(C)C(C4CCS(=O)(=O)N4C)=O)C3C2)=O)cc(O)cc(C#N)c1 C1(NC(C2CCN(C(=O)CCCC3CC3)CC2O)=O)CC2(CCCC2)C1 C(=O)(CCCS(C)(=O)=O)NCC1N(C(C(c2cccc(O)c2)C)=O)CC(OC)C1 C1(NC(c2c(OC)csc2)=O)COC2(C1)CN(C(=O)C(C)(O)c1ccccc1)C2 C12(C(=O)NCC(C)CN(C)C(c3cc(F)cnc3O)=O)CCCC1CC(=O)CC2 c1(CC(N2CCOCC(NC(CCC(=O)N(C)C)=O)C2)=O)nnc2n1CCCC2 c1(SC)ccsc1C(=O)NCC#CCNC(=O)CC1C=CCCC1 C(C(N)=O)(C(F)(F)F)NC(C(C)c1nn[nH]n1)=O Cc1n[nH]c(C)c1C(C)C(=O)N(CC(C)NC(c1ncccc1C(F)F)=O)C C1(C(=O)NCC2CCC(NC(c3scnc3C3CC3)=O)C2)C(F)(F)C12CCC2 N1(C(c2cccc(N(C)C)c2)=O)CC2CC1CC2NC(c1cc(O)cc(Cl)c1)=O C12CC(c3ccccc3)(C1)NC2=O.C1(CNC(C2CC(SC)C2)=O)CCCC1O C=C1CCC(C(N2CC3CC3(CNC(c3nc(C)oc3OC)=O)C2)=O)CC1 C1(C(=O)NC2CC2(F)F)COC2(CCN(C(c3ccncc3Br)=O)CC2)C1 c1(NC(C2OCCN(C(CSCC)=O)C2)=O)c(F)c(F)c(Cl)c(F)c1F C1(C(=O)NCC2CCN2C(=O)CN(C(=O)C(C)C)C)(SC)CCC1 C(=O)(C(=O)NOC)NC(c1ccccc1)C(=O)NC1(C=C)CCC1 c1(C(=O)NCC(C2CCN(C(=O)CCN3CCOC3=O)CC2)C)ccncc1Cl N1(C(C=CCNC(c2cscn2)=O)=O)CCC(n2cncn2)C1 C1(C(=O)OCC(=O)N(CC#N)Cc2cccc(Br)c2)COC2(CCC2)C1 CCCC(C(=O)OC)C(=O)N1CCOCC(NC(=O)C(C)(C)C2CC2)C1 c1(-c2n(CC(=C)C)nc(-c3ccc(OC)cn3)n2)cnn2c(OC)cccc12 c1(CC(C)C)cc(C(=O)NCC(C)(C(C)C)NC(=O)C#CC2CC2)cc(O)n1 CC1(C)CC(C)(C(=O)NC2CC=CCC2)CN1C(c1ccc2[nH]ccc2c1)=O Cc1cccc(-c2cn(C3CCN(C(C4CCCCS4)=O)C3)nn2)c1F C(C(C(=O)N1CCC(CSC)C1)NC(c1cnn(CCO)c1)=O)SCC C(=O)(C(C)CC(N)=O)Nc1c(C2N(C(Cc3cc(C)no3)=O)CCCC2)n[nH]c1 O(NC(=O)CCC(C(C)C)NC(=O)C(CSC)CC)CCOCC c1(CC)nc(CNC(c2nnnn2CC2CCOCC2)(C2CC2C2CC2)C)cs1 Cc1c(C(=O)NC2CC2NC(=O)C(F)(F)C2(O)CCCC2)cncc1Cl c1(C(=O)NC2C(CNC(c3ccc(OCC#C)cc3)=O)CC2)cc(C)cnc1C c1(C(N2C(CC(=O)Nc3c(OCC)cccc3)CC2)=O)ncc(F)cc1N Cc1nnc2n1CCC2(C)C(=O)NC(C)Cn1cc(CCO)nn1 c1(CCC(=O)NCCC2CCCN2C(c2cnc(C3CC3)o2)=O)cccnc1 O=C(C1=CCCCO1)NC1CCN(C(c2ccc(-n3cncn3)c(F)c2)=O)C1 N1(C(CS(C)(=O)=O)=O)CCCC2(C1)CN(C(C1CC3CC1C3)=O)CCO2 N1(C(C2C(C(C)(C)C)C2)=O)CSCC1C(N1CCC1)=O n1(C(=O)NC(C)CCCCNC(=O)C(C)N(C)C)cc2ccccc2n1 N1(CC)CC(C(=O)N(CCCNC(C2CCCN(C(=O)OC)C2)=O)CC)NC1=O CC(CC(=O)NC(C)CN(C)C(c1ccnc(Cl)c1)=O)C(F)F CC(C)CCCC(=O)NC(CCN(C(=O)CC1CC1(C)C)C)C(C)C N1(C(=O)COC(F)F)CCN(C(c2ccc(C(F)(F)F)nc2)=O)C(C2CC2)C1 N1(C(C2CCCC(=O)O2)=O)CC(NC(=O)C=Cc2cncnc2O)CC2(CC2)C1 c1(C(=O)NCC(CC(C)C)NC(C2CNC(=O)N2C)=O)c(O)cccc1Cl C(C(=O)N=c1cc(C)o[nH]1)N1CCC(CCCNC(CCCC=C)=O)CC1 c1(C(=O)NCCCC2N(C(C(N3CCCC(O)C3)C)=O)CCC2)nc(Cl)c(Cl)s1 c1(OC)cc(C(=O)NC2CCN(C(=O)C(C)(C)CF)CC2CO)c(Cl)cc1Cl c1(CC)sc(=N)[nH]c1C(=O)N(C1CCN(C(=O)CN2CC(OC)C2)CC1)CC c1(C(=O)NCC2CC(NC(CC(CC=C)(C)C)=O)C2)cc(S(N)(=O)=O)c(C)o1 N1(C(CC(CC)C(F)F)=O)CC(NC(C2SCCCS2)=O)CC12CCOCC2 N1(Cc2nnc(C)o2)CC2CN(C(c3ccnc(N(C)C)c3)=O)CC2C1 C1(CNC(C(C)OCC2CC2)=O)(CO)CCN(C(=O)CNS(=O)(=O)C2CC2)CC1 c1(C(N2CCC(NC(c3c(C)nn(C)c3)=O)C2)=O)ccc(=O)n(C(C)C)c1 c1(C(N2C(C)C(O)CC2)=O)cc(O)nc2c1CN(C(C1CCN(C)C1C)=O)CC2 Cc1ncnc(C)c1C(=O)NCC1=CCN(CC(=O)NCC(C)C)CC1 N1(CCC)CCCC1C(N1CCC(C(=O)NCc2cccs2)C1)=O C1(NC(C(c2cccc(F)c2)C)=O)CC2(C1)CC(CNC(C1CSCCS1)=O)C2 C1(C(=O)Nc2cccc(COC)c2)N(C(=O)CCc2cccs2)CCC1(C)C C(=O)(C(CC)C(C)(C)CC)N1CCN(C(c2cn(CCOC)nc2)=O)CC(O)C1 C1(CNC(C(C)NS(C)(=O)=O)=O)CN(C(c2ccc(F)cn2)=O)CC(C)(C)O1 CC1(C)CN(C(C2CCN(S(=O)(=O)C(F)F)CC2)=O)C1C1CCCO1 CCCCCC(O)CC(=O)NCc1ocnc1C(N1CCCC1(C)COC)=O C1(CC)CN(C(C2CC(=O)N(C)C2)=O)CC1NC(c1cccc(OC2CC2)c1)=O CC1(NC(c2cccc(OCC3CCCO3)c2)=O)CCCN(C(=O)CCC#N)C1 N1(C(C(C2CCOCC2)OC)=O)CCOCC(NC(c2cccc(CO)c2C)=O)C1 Cc1ccc(C(=O)NCc2cn(C3CN(C(c4cnc[nH]4)=O)C3)nn2)c(Cl)c1 CCCCCC(C)CC(=O)N(CCC(=O)Nc1cccc(C(C)F)c1)C CC1CCC(CNC(=O)CCCc2ccccc2)CN1C(c1csnc1Cl)=O Cc1c(C(N2CCN(C(=O)CC(C)C)CC2CC(F)(F)F)=O)sc2ccccc12 N1(C(c2cnn(C)c2Cl)=O)CCC2(CCN(C(C3CC(=O)CCO3)=O)C2)C1 CC(F)(F)CCC(=O)N1CCC(N2CCN(C(=O)Cc3ccsn3)CC2)CC1 c1(C(N2CCC(NC(C(C)C3CC3)=O)C2)=O)ccc2c(c1)OCCO2 C1(O)(CN(C)C(C2CC(=O)CN2C(C2(C)CCCO2)=O)=O)CCCCC1 C(=O)(C1COc2ccc(Cl)cc21)N1C2CC3(NC(C(=O)N(C)C)=O)C(C1CC2)C3 O=C1CCN(CCOCC2CC3(CCC3)CO2)C(=O)C(Cc2cccs2)N1 C1(C(N(CCNC(=O)CCCn2ccnc2)C2CC2)=O)Cc2n[nH]cc2C(=O)N1 C(CN=c1cccn[nH]1)NC(N1CCC(n2ccnn2)C1)=O N1(C(CCS(C)=O)=O)C2CCCC1CN(C(C1CCC(=O)O1)=O)C2 c1(N2C(C)CN(C(c3nccc(Cl)c3F)=O)CC(C)C2)ncnc2c1SCCC2 Cc1ocnc1C(=O)NC(C(=O)NCc1cn(C)cn1)C1CCOC1 N1(C(C(CCCC)C)=O)C2CCC1C(F)C(NC(=O)Cc1cncn1C)C2 C1(C(N(CC(O)CNC(=O)CCc2ccoc2)C)=O)CC(C)(C)SC(C)(C)C1 c1(NCC2C(CNC(CCC3CCC(C)O3)=O)C2(C)C)ncc(S(C)(=O)=O)cc1Cl C=CC(CCC)CC(=O)N1CC2(CCC2)CC1CNC(c1cc(F)cnc1O)=O n1(CC(=O)NCC=C)cc(CNC(=O)CC2CCCCO2)nn1 c1(C(=O)NCC(CC)NC(=O)C(c2ccccc2)OC)ccc(OC(C)=O)cc1 c1(C(=O)NCC2C(NC(C(CC)OC)=O)CC2)ccc2c(c1)S(=O)(=O)NC2 N1(C(C2(C#C)CCC2)=O)CC(NC(=O)CCc2cc(C)cc(C)c2)C2(CC2)C1 c1(C(=O)OC)ccc(CCNC(=O)CCCCON)cc1 C1(NC(COCCC(C)C)=O)C2CCC(C2)C1C(N1CCC(CO)CC1C)=O N1(C(C2CC(OCC)C2)=O)CCCC1c1cn(C2CC(O)C2)nn1 N1(C(CNS(CC)(=O)=O)=O)CC2CC1CN(C(C1CCC(C(N)=O)CC1)=O)C2 N1(C(=O)Nc2c(NC(c3cc(F)ccc3O)=O)nccc2)CCCC(F)(F)C1 C(=O)(C(CCC)OC)NCCCC1(NC(C(C=C)c2ccccc2)=O)CC1 C#Cc1cccc(OCC(=O)NC2CN(C(=O)CN3CCCCC3)CCC2F)c1 N1(C(C(CNC(C(C2CC2)OC)=O)C)=O)CC=CC12CCOCC2 c1(C(N2CCC(N(C)C(c3ccc(I)c(F)c3)=O)C2)=O)cc(F)c2cc[nH]c2c1 C(CCC(=O)NC1(CN(C)C)CCOC1)=C(C)C.c12ccc(s1)C(=O)NC2 C(=O)(C#CC1CCCOC1)NCCCCCCN(C(=O)CN1CCOCC1)C C1(C(CNC(CN2CC(C)(C)C2)=O)(C)C)CCCCN1C(c1cnsn1)=O N1(C(C2(F)C(C)C2)=O)CCC(NC(=O)Cc2ccc(F)c(Cl)c2)C(F)(F)CC1 C12(C(=O)NC(C34CCC(CC3)C4)C)COC(C1)C(NC(=O)C#CC1CCC1)C2 C1(NC(CCC2C(C)C2)=O)CN(C(c2cc(Br)cn2C)=O)CC12CCOCC2 c1(C(N2CCC(F)(CNC(C3(C)C(C)C3)=O)C2)=O)ccc2c(c1)CC(C)(C)C2 c1(C(N2C(CNC(C(C)NC(C)(C)C)=O)CC2)=O)c2n(c(=O)n1C)CCCC2 Cc1ccc(C)c(C(N2CCC(N(C)C(c3cc(=O)n(C)cn3)=O)CC2)=O)c1N N1(C(c2cn(C)nc2O)=O)CC(NC(C2C=CCS2)=O)CC2(CCC2)C1 c1(CC)cc(C(=O)NCCCN(CCO)C(c2cnsc2)=O)ccc1C C1(NC(c2cc(Br)no2)=O)COC2CN(C(c3ccnnc3)=O)CC12 C(=O)(CCC(C)N(C)C)NC(C1N(C(C(=O)NCC)=O)CCC1)C c1(CC)noc(CC)c1CC(=O)NC1CC(CNC(=O)C(C)(C)OC)C1 C1(O)(CNC(C2C(C)(COC)C2)=O)CCN(C(c2cnc(C3CC3)s2)=O)CC1 c1(C(N2C(C)(CNC(c3cc(CO)on3)=O)CCC2)=O)cc([N+](=O)[O-])n[nH]1 Cc1nn(-c2ccccc2)cc1C(N1CCCC1C1(NC(=O)C=C2CC2)CC1)=O C1(C(=O)NC2C=CC(C(N(C(C3CCC3)C)CC)=O)C2)CC12CCOCC2 C(=O)(CCCCC(C)(C)C)NC(C(C)NC(=O)C(=O)N(C)C)CCc1ccccc1 N1(C(c2c(CSC)cccn2)=O)CC2CCN(C(C3CC(SC)C3)=O)CC2C1 c1(NC(C2C=CC(NC(c3cccc(Cl)c3Cl)=O)C2)=O)ccc(CO)cc1F C(=O)(C(C)(C)c1cncnc1)OCCOCC(=O)Cc1ccccn1 CC1COC(C)(C)CN1Cc1cc(O)nc(-c2ccccn2)n1 N1(C(CC(C(F)F)NC(C(CC)C(C)C)=O)=O)Cc2ccc(C)nc2C1 N1(C(C(C)OCCCCCC)=O)CCCCC1CN(C(=O)C(C)CC)C C(c1cncc(-c2cccc(C(N3CCCCC3)=O)c2)c1)=CC(C)(C)N(C)C C1(C(N(CC=C)OC)=O)CCC2CCC1N2C(=O)Cn1cc(Cl)cn1 c1(C(N(C)CC2CCN(C(=O)Cn3cnnc3)CC2)=O)cc([N+](=O)[O-])cnc1O CCC(F)C(=O)N1CCC(N(C(=O)CCC=CCC=C)CC)C1 C1(C(=O)NCC(CC)NC(=O)COCC2(F)CC2)CCC(C(C)(C)C)CC1 c1(C(N2C(CNC(C(C(CC)O)C)=O)(CC)CCC2)=O)ccc2nccn2c1 Cc1oc(C(=O)NC2CCCC(NC(=O)CCCn3ccnn3)C2)cc1CO C(=O)(C(CC1CCCC1)CC)NC(c1c(C(=O)NCC(CCC)O)con1)C N1(C(C2(C)CC2)=O)CCC2(CCCN(C(c3cc4ccnc(Cl)c4s3)=O)C2)C1 c1(C(N2CC3(CC(NC(=O)CC4CS(=O)(=O)C4)C3)C2)=O)noc2cc(Cl)ccc12 c1(OC)c(C(=O)N(CCCCN(C)C(C2CCCC(C)O2)=O)C)nc(O)nc1O N1(C(CC(C(C)C)NC(CC(CC)O)=O)=O)CCC12CCCSC2 c1(CCNC(=O)NC2CCCC2n2cccn2)cccc(F)c1 c1(CNC(C)CCN=c2[nH]nc(C(F)F)s2)ccc(S(N)(=O)=O)c(C)c1 CC1(C)CCCC(C(=O)NC(CNC(c2cnc(=N)[nH]c2)=O)C2CC2)O1 c1(OC)ccc(F)c(C(N2CCCC2CCNC(c2cnc(S)[nH]2)=O)=O)c1 C(CC(=O)NOCC(C)O)C1(CNC(c2cc(C(C)=O)[nH]n2)=O)CC1 Cc1cc(F)c(C(=O)NC(C2CCOC2)CNC(=O)CC(C)(C)C)cc1F C1(OC)CC(OC(=O)Cc2ccc(OCC(C)C)cc2)C1(C)C C#CC1(NC(C2CCC(CNC(=O)C=CCN3CCC3)C2)=O)CC(F)(F)C1 C1(O)(CNC(CP(C)(C)=O)=O)CCCN(C(c2nscc2Br)=O)C1 c1(C(=O)NC(CCN(C)C)C(N2CCC(F)(CF)CC2)=O)c[nH]c2ccccc12 CC(C)CC(O)C(=O)N1CCN(CCCNC(c2cc(Cl)no2)=O)CC1 n1(CC)c(C(N2CCNCC2C(N)=O)=O)cc2ccccc12 c1(C(=O)NCC(CNC(CC2CCC(C)C2)=O)(C)C)cc(S(C)(=O)=O)co1 C(=O)(C(O)CCCNC(=O)CC1(C#N)CC1)NC(C)(C)C(N)=O c1(OCC=O)ccc(N(CC)CC)cc1C.C(=O)(C(C)N(CC)CC)N N#Cc1ccncc1C(=O)NCC1OCCC1C(=O)NCCN1CCCC1 C(=O)(CS(=O)(=O)C(C)(C)C)NCCC1(O)CCN(C(C2(C(N)=O)CC2)=O)C1 N1(C(C(C)Cn2ccnc2)=O)CCOC(C(=O)Nc2ccc(F)cc2O)CC1 C(=O)(CCN=C(NCCN1CCNC1=O)NC1CCOC(C)(C)C1)NC N1(C(C(=O)NCCOC)=O)CCN(C(=O)C(F)=C(C)C2CC2)CC1C1CC1 C(=O)(C1=CCC(NC(c2cc[nH]c2)=O)C1)NCCC1C(C)CCO1 CC(C(=O)NNc1ccc(Br)c(F)c1F)OCC1CCCO1 N1(C(=O)NC(C(=O)OC)C)CCC2(CC(C(=O)NC3(C#N)CCOCC3)=NO2)C1 c1(CC)nc(-c2nc(CO)nn2CCn2cncn2)sc1-c1ccccc1 CCCCCC(O)C(C)C(=O)NC(C)CCCNC(=O)C(C)(C)CC c1(C(=O)NCC2N(C(Cc3nc(C)[nH]n3)=O)CCCC2C)ncc2ccccn12 c1(SC)ccc(CCCC(=O)NC2C3CC2N(C(=O)CC2CCC(=O)O2)C3)cc1 C1(C(=O)NC(C)(C)CNC(=O)C=C2CCCCC2)(CC)CCC(F)(F)CC1 CC1(O)CN(C(C2(NC(=O)CCCC3CCCO3)CC(O)C2)=O)C1 c1(CSCC)cccc(C(=O)NCC2CC2CNC(c2ccncc2Cl)=O)c1 C(CC(C(C)(C)C)NC(c1cccc(C(F)F)n1)=O)N(C)C(c1cnn(C)n1)=O CC(C)CC(C(=O)N1CC2CC2C2CC12)ONC(=O)CC1C=NN(C)C1=O c1(C(=O)NCC2(C(C)(C)C)CCN(C(COC)=O)C2)c(C)cnnc1O c1(C(N2CCC(N(C(=O)C3=CC(C)(C)C3)CC)C2)=O)ccc(CO)c(F)c1 C1(C)(NC(C=CC(C)NC(C2(C(N)=O)CCC2)=O)=O)CC1(C)C c1(NC(CNC(c2c(C)nc(CC3CC3)o2)=O)C)cc(C#N)c(F)cc1[N+](=O)[O-] Cc1c(NC(c2nc(-c3ccccc3)oc2C(C)C)=O)cnn1CCO C1(C(N2CCC(O)(C(C)NC(CSC)=O)C2)=O)CCC(O)CN1C C(=O)(CC(C)(C)C#N)N1C(C(N2C(CC)CC2)=O)C=CC1 c1(SC)ncc(-c2cccc(CC(=O)NCc3cccc(C(F)(F)F)c3)n2)cn1 N1(C(C2C(NC(c3scc(OC)c3)=O)CCO2)=O)CCOC(C(N)=O)C1 c1(OC)cc(OC)cc(CN2CCC(C)(C(=O)Nc3cc(F)cc(Br)c3)C2)c1 N1(C(C2(CC#C)CC2)=O)CCC2CCN(C(c3cc(O)nc(O)c3)=O)CC2C1 CC(C)C(=O)CCCN1CCN(C2CCCCC2)CC1 c1(C(=O)NCc2cncc(C(=O)NC(CO)C(F)(F)F)c2)cc2n(n1)CCC2 C(=O)(C#CC1CCC1)N1CCC(C(C)NC(c2ccn(CC)n2)=O)C1 C(=O)(C(CC(C)C)C(N)=O)N(C(C)C(=O)NC1COCC1N=[N+]=[N-])CC c1(C(=O)NC(N(c2ccccc2)CC2CCCC(CC)C2)=O)ccnc(C)c1Cl c1(C(=O)OC)cc2c(c(S(=O)(=O)NC3(c4cccc(C(=O)O)c4)CC3)c1)CCC2 CCC(C)C(C(=O)N(C(C)(C(=O)NC1CC1CC(C)C)C1CC1)C)N(C)C c1(NC(C2CC2C(N2CCOCC2)=O)=O)ncc(Br)cc1Br Cc1cncc(C(=O)N(C)CC2CN(C(=O)CSCc3csc(=N)[nH]3)CCO2)n1 C1(C(=O)NC(C2C3CC4C(C3)C24)=O)CC12CCN(C(C1(C)CC(F)(F)C1)=O)C2 C(=O)(CC1=CCCCC1)NC(CCCNC(=O)Cn1cnnn1)c1ccccc1 c1(C(=O)NC2C(NC(=O)C3=CCCOC3)CCCC2)ccc2c(c1)COCCN2 N1(C(CC2C(OC)COCC2)=O)CC2CC(NC(=O)C(c3ccc(F)cc3)=O)C1C2 C1(C)(CNC(CCN(C)CC)=O)CCN(C(=O)CNC(c2cscn2)=O)CC1 C1(CCC)CN(C(c2cc(C(=O)OC)cs2)=O)CCN1C(c1cccnc1Cl)=O N1(C(C(COCC)C)=O)CCCC(O)(CNC(C2(C)CCC(F)(F)CC2)=O)CC1 c1(-c2cnc(SCC(=O)NCC3CC4CCC3C4)o2)ccccc1F C(=O)(CCC(C)(C)NC(c1cn(C)c(=O)n1C)=O)NCc1c(C)nn(C)c1 CCC(CC(F)(F)F)C(=O)N1CCC(C(C)Nc2cnc(C(=O)OCC)cn2)C1 C1(c2ccc(F)c(F)c2)Cc2cn3c(n2)SC(=N1)N3.C(F)(F)F Nc1cc([N+](=O)[O-])ccc1C(=O)NCC1CC1NC(c1ccccc1[N+](=O)[O-])=O N1(C(c2ccn(C3CCC3)n2)=O)CC2CN(C(C3(O)CCCCC3)=O)CC(C1)O2 C#Cc1ccc(C(N2CCC(C=CC(N3CCC(C(N)=O)C3)=O)CC2)=O)cn1 C(=O)(C1CCCc2ncccc21)NC1CCN(C(Cc2c(C)nn(C)c2Cl)=O)C1 c1(C(N2CC(NC(C=CC(CC)=CC)=O)C3C2C3)=O)ccc2nncn2c1 Cc1cccc(C(=O)N(CCNC(=O)C(n2nccc2C)C)C(C)C)c1Br C(C(N=[N+]=[N-])C(=O)N1CCCC12C(=O)NOC2)OCC.C1(C)(CO)CC1 N1(C(c2cc(C)oc2C(F)(F)F)=O)CCC2CN(C(C3CC3C3CCC3)=O)CC12 S(=O)(=O)(c1ccc2c(c1)CN(C(C1CC(C)(C)C13CCC3)=O)C2)N(C)C Cc1nc(NCc2ccc(N(C)C)c(C)c2)cc(=NCC2CCOCC2)[nH]1 C12(CNC(C3CC(O)C3)=O)CCCOC1CCN(c1ncnc3cnccc13)C2 C(=O)(NNc1ncnc2sccc12)C12N(C(=O)OC(C)(C)C)CC(CC1)C2 N1(C(CCSCCC)=O)CC2CCC2(CCNC(c2nccnc2C(N)=O)=O)C1 C1(OCC)CCN(C(=O)CC2(OC)CN(C(=O)CC3(COC)CC3)C2)CC1C c1(C(N(CC(=O)NCc2c(C)nc(C)s2)C)=O)ccc(C)c(O)c1 n1(CCC)nc(C)cc1C(=O)NCC(C1CCCC1)NC(C)=O c1(C(=O)NCC2CCCC2NC(C2CC3CC3C2)=O)cc(Cl)cc(Cl)n1 C1(C)(NCCCC(=O)NNC(c2cscn2)C)CCN(Cc2ccccc2)CC1 c1(C(c2nnnn2CCCC)NC(CCCC)COC)ccc(N(C)C)cc1F c1(C(=O)NCCCNC(=O)C(F)Cc2ccccc2)cnc2[nH]nnc2c1 C1(C(=O)NC2C(CCOC)CCC2)CC(O)CN1C(=O)C=C1CCOCC1 C=CCCCCCC(=O)NC1CCN(C(=O)COC2(C)CCC2)CC1F c1(C(N2C(C)CC(c3ccccc3)C2)=O)cc2cccc(Br)c2cn1 c1(C(=O)NC2CCCC(C(=O)Nc3cnoc3)C2)cc(F)cc([N+](=O)[O-])c1 c1(C(N2C(CO)CC(NC(c3c(CC)onc3)=O)C2)=O)cc(C)nc2ncnn12 N1(C(COC(C)=O)=O)CCC2(NC(=O)Cc3ccc(F)cc3Cl)CCCCCC12 CCC(CC(=O)N1CC2C(CNC(c3cncc4c[nH]nc34)=O)C2C1)C(C)C N1(C(=O)NC(C)C)CCC(C)(C)C1C(N1CCCC1)=O N1(C(CC(CC)C(F)F)=O)CCC2(CCCCC2NC(=O)CN(C)C)CC1 n1(CCOC)cc(NS(=O)(=O)CC2COCCO2)c(C)n1 C1(C(N2C(C(C)C)C(NC(C3CC(=C4CCC4)C3)=O)CC2)=O)CN(S(N)(=O)=O)C1 c1(CCNC(C(CN(C)C)NC(=O)CN2CCCC2=O)=O)cccnc1O N1(C(C(CC2CC2)OC)=O)C2CCC1CC(C(N1CCC1C(C)C)=O)C2 c1(C(=O)NC2CC(CNC(C=C(CCC)CCC)=O)C2)cc(F)c(N)cc1OC Cc1cc2c(cc1NC(=O)CC(C)N(C)C(=O)NC(C)(C)C)CCO2 N1(C(C(C2CCC(=O)N2)C)=O)CCCC(CO)(NC(C2CCCCC2)=O)C1 Cc1noc2ncc(C(N3CC(NC(C4(C)CC4)=O)C(O)C3)=O)cc12 C1(NC(CCCN=[N+]=[N-])=O)CC(N=c2nc(C3CC3)[nH]s2)C1 C1(N(C(c2c(OC)csc2)=O)C)CN(C(=O)CCP(C)(C)=O)CCC1O Cc1nnc(CNC(c2ccncc2)C2CCNC2)n1C O=S(=O)(c1ccc(N2Cc3cccc(Cl)c3C2)cc1Br)NCc1cc(Br)no1 c1(NC(C)CCC(F)(F)F)ccc(S(=O)(=O)NCC2(C)CCCOC2)cc1C#N N#CC1(C(N2CC(CCCCNC(C3CC34CCCCC4)=O)C2)=O)CCSCC1 c1(OC)ccc(C(=O)NCC2C3CN(C(C4CCO4)=O)CC23)c(OC)c1Cl C(=O)(C(Cc1ccccc1)CC(C)C)NC1CCCC(NC(C(CC)CC)=O)C1 C1(CC)CCCN(C(=O)CCC(C)C)C1C(=O)N(C1CC1C1CC1)C N1(C(=O)CCc2ccc(Cl)s2)CC(C2CN(C(C3CC3F)=O)C2)C1 CCC(COC)C(=O)N1CCC(C(C)(C)NC(C)=O)CC1 Cc1cc(C(=O)NC2CCC2NC(c2csc(Cl)c2Cl)=O)ncn1 CC(C)C(CCNC(C1(n2cccn2)CCC1)=O)NC(=O)Cn1ccccc1=O C1(CNC(CC2CC(C(C)=O)C2(C)C)=O)CC(C)CN(C(=O)Cc2ccns2)C1 CC1CCCCC1(CNC(=O)CCCC(N)=O)NC(=O)CC(C)(C)F Cc1cc(O)nnc1C(=O)NCCC1CN(C(C2(O)CCC2)=O)CC1C c1(C(=O)NC(C2CC(NC(C3(CC(F)F)CCOCC3)=O)C2)C)cccc(O)n1 C12(Nc3cc(NCCc4nc5cnccc5[nH]4)nc(C)n3)CCCCC1CCC2 N1(CC(=O)N(CC)CC2CCCO2)CCC12CCOC(C)(C)C2 C1(C2CC2)(CNC(C2C(OC)C2C)=O)CCN(C(=O)COCC2CCCOC2)C1 C1(C(=O)NCCOCCNC(Cc2n(C)ccn2)=O)CCCCC1C#N N(C1CC2(CCN(c3nnc(O)s3)C2)Oc2ccccc21)C(C=C(C)Cl)=O C(=O)(C(C)CC(N)=O)NC1CC(F)(CNC(c2c(C(C)C)scn2)=O)C1 C1(NC(C(C(C)(C)C)NC(C)=O)=O)CN(C(c2n[nH]c3c2CC3)=O)CCC1(C)C C1(CNC(CCc2n(C)ccn2)=O)(NC(=O)CC#N)CCOCC1 c1(C(=O)NC(CNC(CC2CCC(C)C2)=O)(C)C2CC2)ncc2ccccn12 C1(C(N(CCC#N)Cc2ccccc2F)=O)C2C=CC(C2)C1C(=O)O N1(Cc2cccc(C)c2)CCCC(N(C(=O)CNC(=O)CC(C)(C)C)C)CC1 C1(NC(c2nnn(CC)c2C)=O)CC(NC(c2occc2Br)=O)C12CCC2 N1(C(C2C(C)CCC2)C(=O)NC2CCCC2)CCCC2(C=CCO2)C1 c1(CC(N2CCCC2)C)nnc(C(c2cccs2)O)n1CCN(C)C C1(CC(=O)NCC2N(C(CSc3n(C)ccn3)=O)C3C(C2)C3)CN2CCN1CC2 N1(CC(c2nnnn2C2CC2)(C)NCC2(C)CSC2)CCc2ccccc2C1=O c1(-n2c(C(=O)NC3CC(CNC(CCOCC#C)=O)C3)cnc2)ccccc1Cl C(=O)(C1CCCc2nncn21)N1CCC(O)(CN(C)C(C2(C)CCOC2)=O)CC1 N1(C(C(CC=CC)CC)=O)CCC2CN(C(=O)C=Cc3sc(Cl)nc3Cl)CC12 c1(C(N2C(CNC(c3n(C(C)C)ncc3)=O)CCC2)=O)c(Br)cc(F)c(F)c1F CC(CC(=O)N1CCCC1CC(=O)N(C)CC1(C)CC1)C(C)(C)C c1(OCCC)ccc(C(N2CCC(C)(CNC(=O)CCOCC(F)F)C2)=O)cc1 C(=O)(CCCCC#N)NCC1(F)CCC(CNC(C(C)Sc2ccccc2)=O)C1 C(=O)(CC(F)(F)C(C)(F)F)NCC1CCC2(CN(C(CC(CC)CC)=O)C2)O1 C1(CNC(C(=O)Nc2ccc(OCC(=O)OCC)cc2)=O)Cc2ccccc2O1 Cc1cc(C)c(C(N2CC(CNC(C3CCCC3)=O)C(C(F)(F)F)C2)=O)c(=O)o1 Cc1cc(C)c(NC(C2CC23CC(NC(=O)CC(C)n2cccc2)C3)=O)c(C)c1 N1(C(=O)Nc2nc(Br)cc(C)n2)CCC2(CC(C#N)C2)C1 C1(CC)C2CCCC1N(C(=O)CCc1nnc(C(=O)NCc3ccsc3)o1)C2 C1(NC(CCC=C(C)C)=O)CC12CCN(C(c1nn(C)cc1N)=O)CC2 CC1Oc2c(F)cccc2C1NC(c1ccc(C#N)cc1Br)=O C1(C(=O)N(C)CCC2CCC2)(SC)CN(C(C2CCCC2O)=O)C1 C1(NC(C2CC23CC3)=O)CCN(C(C2SCCS2)=O)CC1O C1(C(N2C(C3(NC(CN4CC(C)(OC)C4)=O)CC3)CCC2)=O)CC2(CCCC2)C1 CCC1=C(C(=O)NCCOCCCN(C)C(C23CC4CC2C3C4)=O)SCCO1 N1(C(C(CC)OC)=O)CC2C(CN(C(=O)CCC3CCCCC3)C)C2C1 C1(C(N(CC(=O)NCC2CC(C)(O)C2)CC2CC2)=O)Cc2nccn2C1 c1cc2c(NC3CCCC4(C3)OCCO4)[nH]c(=NC3CCSCC3)nc2s1 c1(CN2CCC(C(C(=O)Nc3nc(C)sc3)C)CC2)cc(F)ccc1[N+](=O)[O-] N1(C(c2c(CC)csc2)=O)CCCC12CCN(C(c1cscc1OC)=O)C2 C1(CCC)CN(C(c2c(C)cnn2C)=O)CCN1C(C1CC1c1ccccc1)=O C1(C(=O)NC2CN(C(c3ncn(C)n3)=O)CC2O)CCCCNC1=O C#CCC(C)(C)C(=O)NC(C)CCN(C(=O)C(C)Oc1ccc(Cl)cc1C)C C(=O)(CCCC(C)(C)NC(=O)C1=CCCCC1C)N1C(C(=O)NC)CC(O)C1 C1(NC(=O)Cn2cccnc2=O)CCN(C(=O)Cc2cnccn2)CCC1CO C(=O)(C(C)CC(C)(C)C)NCC1N(C(C2N(C(C)=O)CSC2)=O)CCCC1 c1(C(=O)NCC2(C)CCOC2)cccnc1CNC(C1CCC(F)C1)=O c1(SC)nc(C)cc(=NCC(CC(C)C)NC(=O)C(CC)NC(c2ccco2)=O)[nH]1 N1(C(C(c2cccc(F)c2)C)=O)CCC12CN(C(=O)Cc1cncn1C)C2 C1(C(=O)NCC(C)OC)COC2(C1)CN(C(c1ccc(=N)[nH]c1)=O)C2 C1(CN(C(=O)CCCCN2CCCCC2)C)CCCN(C(=O)COCC2CC2)C1 c1(CC(=O)NCC2CC3CNC2C3)ccccc1OCc1ccccc1 Cc1[nH]nc(C(=O)NCCC2CCN(C(=O)Cc3cc(C4CC4)no3)C2)c1F C(=O)(C(C)(C)C(N)=O)NC(C1(C(=O)NC2CCN(CC(=O)OC)C2)CC1)C1CC1 C(N=c1[nH]c2c(c(=NC3CCc4cccc(C(N)=O)c43)[nH]1)COC2)c1c(C)nco1 C(CCCCC(=O)N1CCCC1CNC(c1cc(C#N)no1)=O)OCC C1(CC(=O)N(CCC(=O)NCC(N)=O)CC=C)CC2CC2C1 c1(C(N2C(CNC(CC3(C)CCOCC3)=O)CCC2)=O)cnn2cccc(Cl)c12 C(CNC(c1n[nH]c(O)n1)=O)(C(=O)NCC(CC1CC1)CO)OC c1(CN=C(NC(COC)C)NCCn2ccnc2)ccc(F)c(O)c1 N1(C(C(CCC)OCC)=O)CC2(CCN2C(=O)CCC2CCC2)C1 N1(Cc2ccc(CN3C(=O)CNC3=O)cc2)CCCC2(C1)OCCO2 N1(CC(=O)NCC(C)C)CC(NC(c2cnsn2)=O)CCC1C CC1CC(CNC(=O)CS(C)(=O)=O)CCN1C(C1CC2CCC(C1)S2)=O CC1(C)CNC(=O)OC12NC(=O)N(C1CC1c1nc(C(F)(F)F)no1)C2=O N#Cc1cc(C(=O)NCC2CCN2C(c2nccc(Cl)c2F)=O)n2c1CCCC2 C=CC1(CC(N2CCC3CC23)=O)CN(C(=O)CSC(F)(F)F)C1 CCCCC(CC)CC(=O)N1CCC(C)(C)C(C(=O)NC2CC(O)(CO)C2)C1 CCCCCC=CCCNC(=O)NC(C)C(=O)NC1(C(=O)O)CCOC1 O=C(CCC(F)F)NCC1CCC(NC(=O)C=Cc2ccco2)C1 c1(CN2C(CC(N3CCC(c4ccccc4)C3)=O)CCC2)cc(Br)c([N+](=O)[O-])s1 c1(C(N2CCC(C(N)=O)C(C)(C)C2)C(=O)NC)ccc2c(c1)CC(C)O2 Cc1cc(C#N)cc(C)c1C(N1CCCC1CNC(=O)C(c1cnn(C)c1)O)=O c1(C(=O)NCC(CC)NC(=O)C(C)S(C)(=O)=O)coc2c(F)c(Cl)ccc12 c1(C(=O)NC(CCCNC(Cc2ccc(C)cc2F)=O)C)cccc2c1NCC2 CCC(CCCC(=O)NC1CC2CC1C(O)C2O)NC(c1cc(C)sc1N)=O C(CCCCC(=O)N1CCC(CC)C1C(=O)NCC(C1CCCC1)OC)OCC C#Cc1ccc(Cl)c(C(N2CCCC(CN(C(=O)C(C#N)CC)C)C2)=O)c1 n1(CCC(=O)Nc2cnn(C(C)C)c2C2CC2)c(=O)oc2ccccc12 N1(C(c2c(OCC)scc2)=O)CCC(C)(NC(=O)COCCCOC)CC1 N1(C(C2(C(=O)OC)CC2)=O)CCC(C(F)F)(CNC(=O)CC23CCN(CC2)C3)C1 N1(C(=O)NC(c2ccc(F)cc2)CCC)CCCC1C1OCCO1 CCCCC(O)C(=O)NC1C2CN(C(=O)Cc3ccc(Br)cc3C)CC12 C1(CNC(C=C(C)C(F)F)=O)CCC(CN(C(=O)C=C2CCCCC2)C)CC1 c1(OC)nc(Cl)ccc1C(=O)NC(C)C(c1ccc(C)c(F)c1)O N1(C(c2ccc(CCCC)cc2)C(=O)NCCCC2CC2)CCOC2CCCC12 Cn1nc(C(=O)NC2CC(C(=O)NCCC(N)=O)C2(C)C)cc1O n1(CC(N2CC(C(=O)NCc3ccsc3Br)C(O)CC2)=O)nnc2ccccc12 N1(C(c2cc(C)cc(Br)c2)C(=O)NC(C)C(=O)OC)CCC(C2CCOC2)CC1 Cc1cc(NC(c2coc(CNC(c3cnn(C(C)C)c3)=O)n2)=O)cc(CO)c1 C(=O)(CC(O)C(C)(C)C)NC(C)CN(C)C(c1ccccc1)=O C1(CC)C(C(=O)NCCOC2CCN(C(=O)Cc3cn(CC)nn3)C2)CCN1C CC1C(NC(=O)C(F)(F)C(F)F)CC2CCC1N2C(=O)CCc1ccccn1 CC1C(NC(=O)C(C)(C)C2CCCCO2)CCN1C(=O)CC1CCOC1 CCC(CC)CC(=O)N1CCC(CCC(N2CCC(C)C2C(=O)OC)=O)C1 N1(C(=O)Cc2ccno2)CCC2CCCN(C(=O)CCC3CCCCCC3)C2C1 C1(C)(NC(COCC=C)=O)CC(NC(c2csc(C(C)(C)C)n2)=O)C1 N1(C(Cc2ccc(C)c(Cl)c2)=O)CCC2CN(C(=O)Cn3cnnc3O)CC2C1 C1(CCO)(NC(C(C)SCCCC)=O)CN(C(=O)C(CO)c2ccccc2)C1 C(=O)(C(O)C(C)(C)C)NC1(CC(=O)NCc2ccc(OC)cn2)CCC1 C1(C#N)(C(=O)Nc2cccc(CNC(C(CCC)OC)=O)c2)CC12CCCC2 C1(CC(=O)Nc2cccc(C3CCOCC3)c2)CCCS(=O)(=O)C1 Cc1ccnc(C)c1NC(C1CCC(NC(=O)C(C)Cc2ccccn2)C1)=O CC(C)(C)CC(=O)NC(C1CC=CCC1)C(N1CCCC(CO)C1)=O C1(C(=O)NCC2C3CN(C(=O)C=CC=C(Cl)Cl)CC23)CCCCCS1(=O)=O Cc1ccc(C)c(-n2nc(C3CC34CC4)nc2C(O)Cc2ccc(F)c(Cl)c2)c1 N(C(=NCCSC(F)(F)F)NCC1(C(C)(C)C)CCCO1)Cc1nnn(CC)n1 C1(NC(C2CC(C(C)C)C2)=O)CC2(CCN(C(C3(N4CCOCC4)CC3)=O)C2)C1 CCC(C)C(C)C(=O)N1CC(c2ocnc2NC(=O)CC2(O)CCCCC2)C1 C(=O)(C1CC(=O)Nc2nc3ccccc3n21)N(C1CCSCC1)C C1(CNC(=O)CC(C2CC2)C2CC2)CC2CCC1N2C(c1ccsc1Br)=O N1(C(C2(C)CC2)=O)CCCC(C2CC2NC(=O)CCCCCn2cnnn2)C1 C12(CNC(C3(CO)CCN(C(C(C)SCCCC)=O)C3)=O)CCCC1CCC2 C(=O)(CCCCCCBr)N1C(CC(N2CCN(CC(F)F)CC2)=O)COCC1 C1(CC)CN(C(c2c(CNC(=O)C=Cc3cnccn3)cnn2C)=O)CCO1 C1(C(=O)NC(C2CCOC2)(C)C)COCCC1NC(c1cccc(CO)c1)=O c1(C(N2CCC(O)(C(C)NC(CCSCC(C)C)=O)C2)=O)occ2c1CCOC2 c1(CC(N2CC(C(C)NC(c3c(C#C)c[nH]n3)=O)C2)=O)c[nH]c2cnccc12 N1(C(C2(C#C)CCCC2)=O)CCC2(CCC(CNC(C3CC3(Cl)Cl)=O)O2)CC1 N1(C(C2COC(C)C2)C(=O)NC(C)C)CCC2(O)CCOCC2C1 CCC(CC(=O)NC1(COC)CCCN(C(c2nc(C)oc2OC)=O)C1)C(F)F C(CCCCC(=O)NC1CC1C(F)(F)F)NC(C1C(C)CC1)=O O=C(N=c1cc(Cc2ccc(F)cc2)[nH][nH]1)c1cccc2c1COC2 Cc1nc(Br)cnc1NC(C1CCCN(C(=O)CC#N)CC1)=O Cc1c(NCCCc2ccsc2)ncnc1N1CCC(CC2CCC2)C1 C1(NC(C(C)CC2CCC2)=O)CCC2(CCCN2C(=O)CC(C)(C)C(F)F)CC1 N1(C(c2c(C)ocn2)=O)CCC(C2CCN(C(c3ccnn3CC(F)F)=O)C2)C1 CCCCCCC(C)C(=O)NC1CC(C)(NC(c2cncc(Cl)c2)=O)C1 N1(C(C2C(C(C)O)C2)=O)CCCC(C2(NC(C3(O)CCCCC3)=O)CC2)C1 Cc1nnc(C(=O)NC2CCCC2CNC(c2ccc(CO)o2)=O)s1 C1(N(C(CN(S(CC)(=O)=O)C)=O)C)CN(C(=O)OC(C)(C)C)C2(CCC2)C1 CCCC(C#N)C(=O)NC1CCCCN(C(c2cc(C)nn2C2CCC2)=O)C1 N1(C(c2c(C)onc2)=O)CCN(C2CCCC2NC(C2(C)CC=CCO2)=O)CC1 N1(C(=O)Oc2c(C)cccc2)C2CC1CN(Cc1ccnc(F)c1)C2 c1(C2CC(C(=O)NCC3CCC(NC(c4sccc4F)=O)C3)C2)ccccc1 C1(NC(CCC=C)=O)CC2CC(NC(C3CCCC34CCC4)=O)C2C1 C1(C(N2CC(CCC)N(C(c3csnc3C)=O)CC2)=O)CCCN2CCCCC12 c1(C(=O)NCCC2CCCN(C(=O)C(F)C3CC3)CC2)ccc2nn[nH]c2c1 N1(C(=O)CCOC2CC2)CCCC2(CCN(C(=O)CC3CC4CC4C3)CC2)C1 C(=O)(C1=C(C)N(C)c2nnnn2C1)N1CC(NC(=O)NC(C(=O)OCC)C)OCC1 Cc1nc(O)[nH]c1C(=O)NCC(C)(C)CN(C)C(c1ccc(Cl)o1)=O c1(C(=O)NC(C(C)C)CNC(C2(C3CC3)CC2)=O)ccc2c(c1)OCC2 Cc1cnc(N2CCOC(C(C)NC(c3cc(C4CCC4)on3)=O)C2)nc1O c1(CC(=O)NCC(C)NC(CC2C(C)=NOC2=O)=O)ccc(F)cc1F C(=O)(CCCC(N)=O)NCCC(C)(C)NC(=O)CC12CC(C1)C2 c1(CC)ccc(F)c(C(=O)N(C)CC2CCN(C(c3conc3CC)=O)CC2)c1 c1(C(=O)NCC2(CN(C)C(C34CC(CO3)C4)=O)CC2)c[nH]nc1C1CCOCC1 N1(C(C2(COCC)CC2)=O)CCC(C(=O)Nc2ccccc2C(C)O)CC1 CC1CN(C(C2C(NC(c3ccc4[nH]ccc4n3)=O)C2(C)C)=O)CC(C)(C)C1 N1(S(C(C)(C)C)(=O)=O)CC2CC1CC2NS(=O)(=O)CC#N C#CCCCCCC(=O)N1CC(C2CN(C(c3ccc([N+](=O)[O-])n3C)=O)C2)C1 c1(CC(=O)NC(CCC)CNC(C2CCC2C)=O)cc(F)cc(F)c1 N1(C(c2c(CC)cccn2)=O)CCN(C(c2ccc(CC(C)C)s2)=O)CC(O)C1 C#CC1COCCN1C(=O)CCC(CC)NC(=O)CCN(C)CCC N1(C(c2c(C)cc(F)cn2)=O)CCC(N(C(=O)C=C2CCOCC2)C)C2(CC2)C1 C1(NC(C(Cn2ccnn2)NC(CCC(C)N(C)C)=O)=O)CCCN(C)C1=O C12(C(N3CCC(C(C#C)C)CC3)=O)CCCC1CCN2C(c1sncc1CC)=O N1(C(c2c(C)nccc2)=O)CCC(C)(C)C1C(N1CC(c2cc(O)n[nH]2)C1)=O C1(C)(C(=O)NCC2(NC(CCC(C)(F)F)=O)CCOC2)Cc2ccccc2C1 c1(OCCOC(=O)OCC)ccccc1S(C)=O C1(C(N2CCC(O)(CNC(=O)CCc3cc(Cl)cs3)C2)=O)CC2C(C1)C2(F)F c1(OC)ccc(NC(=O)N(C2CC2)Cc2ccc(C)cc2)c(C(F)(F)F)c1 c1(OC)ncccc1C(N1CCOCC1c1ccc(C)o1)C(=O)NC1(C)CC1 C1(C(N2CC3CC(CNC(=O)Cc4ccco4)C3C2)=O)CCc2ncsc2C1 N1(C(C2CCN(CC)CC2)=O)C2CCC1C(C(=O)NC(C)CCCO)C2 C(C)(CC(=O)NC1CCN(CCOC)C1)NC(COCC(=C)C)=O c1(C(=O)NC2C(CCC)CN(C(C3(SC)CCOCC3)=O)C2)cn(C)ccc1=O C(CCO)(C(C)(C)C)NC(CN(C(Cc1cc(C)[nH]n1)=O)C)=O c1(CC(=O)NC(C2CCN(C(COC(CC)C)=O)C2)(C)C)ccc(F)cc1F Cc1ncncc1C(=O)NCC1COC(CNC(C2CCCN2C(C)C)=O)C1 c1(OC)c(F)ccc(F)c1C(=O)NCC1CC1NC(C1(P(C)(C)=O)CC1)=O CC(C(C)(C)C)=CC(=O)NC1CC(NC(=O)C(C)(Cl)Cl)C1 Cc1cc(C)n(C(C)C(=O)NC2CCCC2(C)NC(=O)Cc2cncs2)n1 C1(C(=O)OCCN(C)C)CCN(CC2CCCC2C(C)(C)C)CC1 CCC(F)(F)CCN=c1nc2scnc2c(NCCOC2CCCCO2)[nH]1 OC1CN(Cc2c(F)ccc(CC3CC3)c2Cl)CC(c2cncnc2)CC1O C(=O)(CCS(C)(=O)=O)NC1CCC(C(=O)NCC(c2ncc[nH]2)C)CC1 c1(OC)ncc(CC(=O)NC2(CNC(c3cccnc3OCCO)=O)CC2)cn1 c1(C(CNC(CC2CC(OC)C2)=O)CNC(=O)CN2CC=CC2)ccccc1 n1(CC)ccc(CC(=O)N(CCCNC(=O)C(C)OC(C)(C)C)CCO)n1 C1(CCNC(c2cccc(C)c2C)=O)CN(Cc2nc(=O)n(C)[nH]2)CCS1(=O)=O N1(C(Cc2cn(CC)nc2)=O)CCCCC(NC(c2nn[nH]c2Cl)=O)C1 C1(C(=O)NC(C2CCCC2)CNC(C2(CC(C)C)CC2)=O)CC=CC1 c1(C(=O)NC2C(C)CCN(C(=O)Cn3cccn3)C2)cc(F)c2c(c1)nnn2C C1(OC)CN(C(=O)OC)CCC1O.C12CCN(C1)C2=O C1(C(=O)NC2CN(C(c3ccc(C(N)=O)o3)=O)CC2CO)CCCCC1C1CC1 N1(S(CC(=O)OCC)(=O)=O)CCC(F)(F)C(NC(c2cnn(C(C)(C)C)c2)=O)C1 N1(C(CC2=NN(C)C(=O)C2)=O)CCC(C2CCCN(C(C34CC(C3)C4)=O)C2)C1 C1(C(N(C(CC(=O)N(CC#C)CC2CC2)(C)C)C)=O)CCC(C)=C(C)C1 CC1CN(C)CCC1N(C(c1cc(Cl)ccn1)C(=O)NCC1CCCO1)C C(C(F)C(=O)NC1(CCO)CN(C(C2CCN2C2CCCC2)=O)C1)N(CC)CC N1(C(c2nnn(Cc3cc(C)no3)c2C)=O)CCC2(O)CCOCC2C1 c1(CN2CCCC(CNC(c3ccc(OC)cc3)=O)C2)ccc(O)c(C)c1 n1(CCC)cc(Cl)c(C(N2CC(NC(=O)C(C)(C)OC)C2)=O)n1 n1(CC(C(=O)NCC(C)N(C(c2cc(SC)oc2)=O)C)(C)O)c(C)cccc1=O N1(C(c2cc(Br)cs2)C(=O)NC(C(=O)OC)CC(C)C)CCC(C#N)CC12CC2 C1(C(N2C(CC(=O)NC(CSC)(C)CO)CCC2)=O)CC2(CC2)CO1 C(c1ccc2[nH]ccc2c1)=CC(=O)NC(C)C(C)NC(c1coc(C(F)F)c1)=O Cc1ccc(C(=O)N(C(C)(C(=O)N(C)CC2CCCCO2)C2CC2)C)c(C)n1 Cn1cc(C=CC(=O)NCC2(C(=O)NC3CCC=CCC3)CC23CCC3)cn1 Cc1cc(F)ccc1CC(N1CCCC(CNC(C2CC(C(C)C)=NO2)=O)C1)=O C1(CNC(C(C(C)C)(C)C)=O)CN(C(c2ccnc(F)c2N)=O)CCC1(C)C Cc1cccc(OCOC(C)C)c1C.C(C(C)(C)CN(C)C)N(C(CO)=O)C C(=O)(C(C)S(C)(=O)=O)N(C1CCN(C(C2CCCC(OC)C2)=O)C1)CC O=S1(=O)CC2CN(Cc3ccc(Br)c(Cl)c3F)CC2(c2ccccc2)C1 CC1CN(C(=O)CC2(O)CCCC2)CC1CC(=O)NC1CC(=C2CC2)C1 CC1CN(C(c2ccc(C(N)=O)o2)=O)CC1NC(=O)C(C)(C)OC(C)C CCCCC(CC)CC(=O)NCC1(F)CC(CNC(=O)CC2CCCC23CC3)C1 c1(C(N2CC(COC)(CNC(=O)CN(C)CCO)C2)=O)cnn2c1CCC2 N1(C(C(CC)=CCCC)=O)CCCC(CCC)(NC(c2cccc(O)c2F)=O)C1 C(CCCCCC(=O)N(CC(C1CCC1)OC)C)NC(C(C)N(CC)CC)=O c1(N2CCC(C)(OCC)CC2)nc(C)cc(=NCCc2ncn(C)n2)[nH]1 c1(C(C)C)ncncc1C(=O)NC(C)CN(C)C(C1CCSC1)=O C1(NC(C2(CSC)CCOCC2)=O)CCN(C(C2(C)CC2(F)F)=O)CC(C)(C)C1 Cc1nc(O)ccc1C(N1CC(O)(C(C)NC(c2cccc(C3CC3)c2)=O)C1)=O N1(C(Cc2n[nH]c(=NC)s2)=O)CCC2C(C1)CN2C(=O)CCOC1CCOCC1 CCC(C)CC(C(=O)NCC1(CF)CC1)NC(=O)CC1CCC1 C1(CCNC(=O)C=Cc2cocn2)CN(C(C2CC(n3ccnc3)C2)=O)CCO1 Cc1nccc(C(=O)N(C)CCOCCNC(=O)CC2CCCCC2C)c1Cl c1(OCC(C)C)ccc(-c2cscc2C(=O)N(C2CC2)CC2CCN(C)CC2)cc1 Cc1cccc(C(N2CCCC2CNC(=O)CC2OCCCO2)=O)c1F c1(OC)ncc(C(N2CCC(O)C2C(=O)Nc2ccc(I)cc2F)=O)cc1F N1(C(c2cc(N)cc(F)n2)=O)CCCC2CN(C(=O)CC3COCCO3)CC12 N1(CC)CCN(C(c2cc(OCc3ccccc3)ccc2O)C(=O)O)NC1=O C(CS(=O)(=O)c1ccc(C(F)(F)F)cc1)NC(N1CCCC(N(C)C)(CO)C1)=O C1(C)(OC)COCCN1C(c1ccnc(C2CC2)n1)=O CN1CC(NC(C2CC(F)(CN)C2)=O)CC12CCCC2 Cc1cc(O)n2ncc(C(=O)NC3CC(NC(=O)CC4(C)CCCC4)C3)c2n1 C#Cc1ccc(F)cc1C(=O)NC(CC)(CC)CCNC(C1(COC)CC1)=O N1(C(CCNC(=O)OCC)=O)CCN(C(=O)NOCC(O)CO)C(=O)C1 c1(C(N2CCN(C(CCC(=C)Br)=O)C(C)C2C)=O)ccc2nc(O)oc2c1 c1(C(C2(Cc3nnnn3C3CC3)CCC2)NC(C)C)ccc(C(Cl)Cl)cc1 c1(C(=O)NCC(CNC(=O)COc2cccnc2Cl)O)ccnc2cc[nH]c12 c1(C(N(C(C)C(N2CCCC2CN(C)C)=O)CCC)=O)ccnc(OC)n1 CCC(C)C(O)C(=O)NC(C)(C)CN(C)C(c1ccc(SCCN(C)C)cc1)=O N1(C(C2(C(C)(F)F)CC2)=O)CCC2CC2(C(=O)Nc2cccc(O)c2)CC1 c1(N2CCC(C)C(NC(c3ccco3)=O)C2C)ccc([N+](=O)[O-])cc1Br C1(C)(C(=O)NCCN(C)C(c2cc(OC(F)(F)F)cc(Cl)c2)=O)CCC(=O)NC1 C1(C(N(CC(=O)NCC=CC)C(C)C)=O)COCCC1C c12cc(nn1C)NC2=O.c1(CN(CC(C2CC2)OC)CC)cc(C2CCC2)n[nH]1 c1(NC(C2CC(NC(c3ccc(Br)c(Cl)c3)=O)C2)=O)nc(Cl)ccc1O n1(CCCNC(=O)N=c2ccn(Cc3ccccc3)[nH]2)c(=O)oc2ccccc12 C12(C(N3C(C(N(c4cccnc4)C)=O)CC(O)C3)=O)CC3CC(CC(C3)C1)C2 C(=O)(C(C)CCCC(C)C)NCC1=CCN(C(C2N(CCC)CCC2)=O)CC1 C(=O)(C(C)CC(C)C(C)=O)N1C(C(=O)NC2(C#C)CC(F)(F)C2)CC=CC1 c1(C(=O)NC2CCC(C)N(C(=O)CC3(C)CCOCC3)C2)ccc2oncc2c1 N1(C2CCCc3ccccc32)CC1.C1(C(=O)O)CC1(F)F c1(C(=O)NC2CCCC(NC(COC(C)C)=O)CC2)cnc2[nH]c(O)nc2c1 CC(C)C(O)C(=O)NC1CC1CNC(=O)CCc1nnc(C2CCCC2)o1 c1(OC)ccccc1NC(=O)C(c1ccc(CCC(=O)OC)o1)NC(C)C(C)C N1(C(C2C(C(C)C)C2)=O)CCC(C)C(N(C(=O)C(=Cc2cccc(F)c2)F)C)C1 N1(C(C(CC)COC)=O)CCOCC(NC(=O)CC(C)(C)CN(C)C)C1 c1(C2(C(N3C(C(N)=O)CC(F)C3)=O)CC2)c(Cl)cccc1Cl C=C1CC2CCC(C1)N2C(=O)C(c1cccs1)NC(=O)CC(CC)C(C)C N1(C(c2cc(Br)c(C)s2)C(=O)NCCCCCC)CCC(O)C(F)C1 CCCCCC(O)CNC(C1C2CC3C(C2NC(C2CN4CCN2CC4)=O)C13)=O N1(C(C(CC=C)CC)=O)CCCC2(C1)CN(C(C1COCCOC1)=O)C2 C1(NC(c2cnc(CC)s2)=O)CCN(C(=O)CCCCN(C)C)CC1C c1(C(=O)NC2C(NC(=O)Cc3ccc(Cl)cc3F)C2)csc2ccccc12 c1(C(N2CC(NC(CCC(C)N(C)C)=O)C2)=O)ccc2c(c1)CCCS2 CC(C)(C(=O)N1C(CNC(c2cc(Br)c[nH]2)=O)CC2COCC12)S(=O)(=O)C1CC1 C(F)(F)(CN=c1ccc(Br)c(S(=O)(=O)NCC(C)CO)[nH]1)c1cn(CC)nc1 Cc1cc(C(=O)NCC2CCN2C(=O)CCSCC(C)C)nn1C(C)C c1(-c2c(OC)c(F)ncc2)cc2c(s1)CCN(Cc1ncc[nH]1)C2 c1(C(N2C(CN(C)C(C3CC34CCC4)=O)CC(F)C2)=O)ccnc2c1CCC2 C1(C(N(CC(C)NC(=O)CN2CSCC2=O)CC)=O)CC2(C1)CC(C)(C)C2 N1(C(c2c(CC)con2)=O)CC(NC(=O)C(CCSC)NC(N)=O)CC12CCC2 C(=O)(C1CC(=O)c2c(F)cccc21)N(C1CCN(C(c2cc(OC)ns2)=O)C1)C C#Cc1ccc(F)cc1C(=O)NCC1CN(C(C2C3CCC2(C)C3(C)C)=O)C1 c1(C(=O)NCC2N(C(C(C)CN3CCOCC3)=O)CC2)cc([N+](=O)[O-])n[nH]1 N1(C(c2cc(C)c(C)[nH]2)=O)CC2CC3CC2C1C3NC(=O)C(C)SC(F)(F)F C(=O)(C1CCc2ccccc21)NC1CC(C)N(C(=O)C(C)Cc2ccccc2)C1 N1(C(C(C)(O)C2CC2)=O)CC2(C1)CN(C(C1CC13CCCCC3)=O)C2 c1(OC)ccc2c(c1)OCCC2NC(c1ccc(Br)c2c1OCCC2)=O N1(C(C(C(CC)C)NC(c2cc(CO)on2)=O)=O)CCC2(CCOC2)C1 c1(C(=O)NCC2(CCNC(C3CC(CF)C3)=O)CC2)cc(O)cc(Cl)c1Cl N1(Cc2cn(C(C)C)nn2)CCC2(CCO2)CC1 c1(C(N(CCC#C)C)=O)ccc2c(n1)CN(C(=O)CC1CCCCC1O)CC2 Cc1cnc2c(C(=O)NC3CN(C(C4CC4(Cl)Cl)=O)CC3O)cnn2c1 N1(C(c2c(CC)nccc2)=O)CC2CCN(C(=O)Cc3nc(=N)[nH][nH]3)C(C2)C1 C1(CNC(c2ccc(Br)cn2)=O)COCCN1C(=O)CC1C=CCC1 N1(C(CNC(C)=O)=O)CC(C)CC1c1cccc(F)c1 N1(C(CCCCC)=O)CCCC2(C1)C(NC(c1ccc(Br)o1)=O)CCN2C c1(CC(=O)NCCOC2CCN(C(C(CC)n3cncn3)=O)C2)c(C)noc1Cl C1(F)(CNC(CCC)=O)CCCN(C(C2(CC)CCOCC2)=O)CC1 C1(NC(C=C(CCC)C)=O)CC2CCC1CC2NC(C1(C)CCCC(F)(F)C1)=O c1(OCOC)noc(Cc2cn(C3CC3)nn2)n1 O=C(C1CCCn2cnnc21)NCCCCC1CN(C(c2nc(Cl)c(Cl)s2)=O)C1 Cc1cnc(COCC(=O)NCC2(CNC(c3[nH]cnc3C)=O)CCC2)o1 N1(C(CC#N)=O)CCCC2(NC(=O)Cc3ccc(Br)s3)CCCC12 C1(CNC(CC(CC)(C)C)=O)CC2(CCOCC2)CN1C(C1CC(C#N)C1)=O c1(C(N2CC(CC=C)(NC(c3cc([N+](=O)[O-])c[nH]3)=O)C2)=O)ccc(F)c(C#N)c1 C=Cc1ccc(C(N2CC(NC(=O)C3=C(Cl)CCC3)C3CC23)=O)cc1 C1(CCNC(C=Cc2ncc(C)[nH]2)=O)CN(C(C2(C)CCC(=O)N2)=O)CCCO1 C(=O)(CS(=O)(=O)C1CCCC1)NCC(CO)NC(=O)CCCC1CCC1 CC1=C(C)CN(C(c2sccc2CNC(c2ccn(C(F)F)n2)=O)=O)C1 c1(CCC(=O)N(CC(C)CNC(=O)C(F)(F)CN(C)C)C)c[nH]c2ccccc12 C=C(Cl)CCC(=O)N1CC2C(CNC(c3c[nH]cc3-c3csc(C)n3)=O)C2C1 c1(C(N2CC3(CC(NC(C(C#C)(C)C)=O)C3)C2)=O)cc(Br)c2[nH]c(C)nc2c1 c1(CN=C(NCC(COC)F)NC(C)C2CC2)nnc2cccnn12 C(=O)(C1=CC2CCC(C1)C2)N1C(C(N(C)CCc2nccs2)=O)CCCC1 CCCCS(=O)(=O)NC(C)C(=O)NCCN(C)C(c1cc(C(C)(C)C)n(C)n1)=O N1(C(C2CC(C)OCC2)=O)CCC(C(=O)NOCCCCC2CC2)C1(C)C N1(C(C2C(=C)C2)=O)CC(NC(C2(COC)CC=CC2)=O)CC(C)C1 C1(N(C(c2cc(COC)no2)=O)C)CN(C(=O)CS(N)(=O)=O)CCC1O N1(C(c2c(C)ccnc2)=O)CCC2CCN(C(=O)C3=CCCCC3)CC2C1 C12(CNC(C(n3c(C)ncc3)C)=O)CCCC1N(C(c1cscn1)=O)CC2 CCCC(C(=O)NCC#CCNC(C1(n2cccn2)CCC1)=O)S(N)(=O)=O C(CN=c1[nH]c(=NCCC(O)c2ccccc2)[nH]c2ccccc12)NC(C)=O Cn1ncc2c(NC3CN(C(=O)Cc4cccs4)CC3(C)C)ncnc12 N1(C(C(CC)C)=O)CC(CO)C2(CCN(C(=O)Cc3c[nH]nc3O)CC2)C1 c1(C(N2CCC(NC(C(C=C)O)=O)C2)=O)ccc(-c2ccc(F)cc2)n1C C1(C(=O)NCC2N(C(CCOCCOC)=O)CCC2C)CCCC(C)CC1 c1(N(C(C)CSC)C)nc(=NC2CC(F)(C(=O)OC)C2)nc(N2CCOCC2)[nH]1 c1(C(=O)NCCC(=O)NC(C)(C)C)cc(Br)cc2nn(C)cc12 N1(C(CCc2ccn(C)n2)=O)CCCN(C(=O)CCC2CCC(=O)N2)CCC1 C(c1cc2ccccc2n1C)=CC(=O)NC1(CCNC(CCCCC)=O)CCC1 c1(C(=O)NCC2CC(C)N(C(C3CCC3)=O)C2)nc2n(c1Cl)CCCC2 n1(C(CC)C)nnnc1C(c1ncc(I)s1)Nc1cnn(CCOC)c1 c1(Cc2c(C)nc3ccccc3c2)[nH]c(=NCc2cocn2)nc2c1ncn2C CCCCCC(C)(CC)C(=O)N1CC=CC(NC(=O)CSCCCC)C1 C(=O)(CC(P(C)(C)=O)c1ccccc1)NCC1N(C(CCC)=O)CCC1 Cc1ccc2c(CC(=O)NCC(CO)NC(C3(n4cccn4)CC3)=O)coc2c1 C(=O)(C1=CCCOCC1)N(CC(CN(C(=O)CSc1nncn1C)C)O)C Cn1cc2c(CN3CCC(O)C(C(=O)Nc4cccc(Br)c4F)C3)cccc2n1 Cc1cc(CC(=O)NCCOCCn2cc(-c3nc(C4CC4)cs3)nn2)sn1 O=C(CN=c1cc[nH]cc1)NC1CCCC(NC(=O)C(F)(F)C2CC2)CC1 Cc1c(C(=O)NC(C2CCCN2C(=O)C(C)NC=O)C)cnn1C(C)C C=C(C)C(C)(O)C(=O)OC1CC(C(=O)NC2CCCCNC2=O)C1 c1(NC(c2cc(-c3ccccn3)c[nH]2)=O)cccc(C2CCOC2)c1 Cc1cc(CNC(=O)CC2CCCC(C)C2)oc1C(=O)N(C(C(N)=O)C1CC1)C N1(c2n(C)nnn2)CCC2(CC1)CC(NC(c1cnc3c(cnn3C)c1)=O)C2 c1(Nc2cc(COC)cc(C(N)=O)c2)nn2ncccc2c1C(=O)OC c1(OC)cc(C(N2CC3CC2C3NC(=O)C(=Cc2ccco2)C)=O)ccc1C#N C1(C(=O)NCCNC(=O)NC)CCCN(C(c2ns[nH]c2=O)=O)C1 c1(CC(=O)NCCCN(C(c2nnn(C)c2N)=O)CC)cc(F)ccc1OC CCCC(CCCO)C(=O)N1CCC(C)C1CNC(=O)CCCn1cccn1 C1(C(NOCC(N)=O)=O)CC2(CC2)CN1C(c1ccc(=N)[nH]n1)=O N1(C(C(COC)Cl)=O)CCC12CCN(C(c1ccc(Cl)c(Br)c1)=O)CC2 C1(C(=O)NC(c2ncccn2)CC)CC(=O)CN1C(c1csc(C#N)c1)=O c1(N2CCC(CC(N3CCC(O)C3)=O)C2)[nH]cnc2nc(Br)cc1-2 C1(CCNC(c2ncn(CC)c2)=O)CC(F)(F)CN1C(C1CC(C(=O)OC)C1)=O c1(CC(=O)NCC2(NC(=O)C(O)CN3CCCC3)CCCC2)cccc(O)c1 C(=O)(CCN(OC)C(=O)C=C1CCCCC1)N1C2CC(=C)CC1CC2 N1(CC)CCC(C(=O)NC(C2(CNC(=O)COc3ccccc3C)CC2)C)CC1 C(=O)(C(C)C1=CCCC1)N(C1CCCN(C(Cn2ncc(C#C)c2)=O)CC1)C C(=O)(C1=C(C#N)CCC1)N1C(C(C)(C)C(=O)NC2CN(C3CC3)C2)CCC1 C(C)(C)(CC(=O)NCC1CN(C(C2CC2c2nc[nH]n2)=O)CCO1)N(C)C c1(C(N2C(COC)(CNC(c3csnn3)=O)CCC2)=O)ccc2c(c1)C(C)CO2 C(=O)(C1=CCCC(C)(C)C1)NCC1COCCN(C(c2c(C)onc2)=O)C1 C(C(C)(C(=O)NCC1NC(=O)NC1=O)NC(c1cc(C)co1)=O)SC C1(CC(=O)NCC2(O)CN(C(c3cc(C)[nH]n3)=O)C2)SC(=N)NC1=O Cc1ncnc(C)c1C(=O)NC1CCC(C(=O)NC2CCCC3(C2)N=N3)CC1 CC1CCC(C(F)(F)F)N1N1CCN(c2cc(Cl)ccn2)CC1 N1(C(C(CC)CC)=O)CC2CCCC(CNC(=O)C#CC3CCCCC3)C2C1 Cc1nc[nH]c1CC(O)C(=O)NC1COCC1CNC(=O)C=CC(F)(F)F C(=O)(CCCCCCCCCO)N1CCC(NC(C2C(CC(C)(C)C)C2)=O)C1 C1(NC(CCOCCOC)=O)CC2(C1)CC2NC(=O)C(C(C)C)c1cccnc1 C1(C(=O)NC(CC(=O)OC)C)CN(C(=O)CCCCC2CC2)CCN1C c1(C(=O)NC(CN(C)C(C23CC(C2)C3)=O)(C)C)cn(C)nc1Cl C1(N(C(C2(O)CCC2)=O)CC)CN(C(=O)C=CC(C)=O)C1 CC(C)C(C(=O)Nc1cn(C)nc1C#N)C(C)NC(C1CCC2(CC2)C1)=O C1(OC)CN(C(c2ccco2)=O)CC1NC(C1CCC(C(F)F)CC1)=O C#Cc1cccc(C(=O)NC2CC2CNC(=O)C(c2ccc(Cl)c(Cl)c2)C)c1C N(C1CCOc2c1ccc(Cl)c2Cl)S(=O)(=O)c1c(F)cc(Cl)cc1F C12(C(=O)NC3CC(N(C)C(c4cnn(C5CC5)c4Cl)=O)C3)CCC(CC1)CC2 C1(C(=O)OC(C)(C)C)(C(=O)NCC2(S(C)=O)CC2)CCOCC1 Cc1nc(O)ccc1C(=O)N(CC(C)O)CCNC(=O)CCc1cccc(O)c1 C(CCC(C)(C)C(=O)NCC1(CO)CC1)NC(C1N(C)CCCCC1)=O C(C(=O)NC1CC(CCNC(C2(n3ccnn3)CC2)=O)C1)(C(C)C)NC(C)=O c1(C(N2CC(CC)N(C(C3CCC3CF)=O)CC2)=O)cc2c(s1)CCOC2 Cc1ccc2nc(CNCC(O)CC3CCCC3)cc(=O)n2c1 CN1NC2=NC(c3nnnn3-c3ccccc3Cl)CC1=N2.C1CCOC1 CC1CCCCC1(C)C(=O)NCC1CC(CNC(=O)Cc2c[nH]nc2O)C1 C1(NC(CC2(C=C)CN(C(C3CCC3(F)F)=O)C2)=O)CCN(C)CC1C#N N1(C(C=C(NC(C)=O)C)=O)CC2CC1CCC2NCc1ccc(NC(N)=O)cc1 c1(NCCC2CCC(NS(c3ccn(C)n3)(=O)=O)CC2)[nH]nc2c(Cl)cccc12 C=C(C(=O)N1CC2CC1C2CNC(c1c[nH]nc1-c1ccc(Br)s1)=O)C(F)(F)F C1(n2cc(C(C)NC)nn2)CCCN(C(c2ccc(Cl)c(C(F)(F)F)c2)=O)CC1 CC(C)(N=c1[nH]cc(C#N)o1)C(O)c1ccc(I)cc1 CC1C(O)CCN1C(=O)CC1CCCCN1C(c1ccc(CO)cn1)=O C1(NC(C2(C)CN(C(C(C)NC(C)=O)=O)C2)=O)CN(C(C)C)CC1C c1(C(N(C2CCCC(NC(=O)C(C)(C)C(F)(F)F)C2)C)=O)cc2c([nH]1)CCCC2 Cc1ccc(C(=O)NC(C)(C)CCNC(=O)CC2CC3CC3C2)c(C)c1 C(=O)(C(CC1CC1)NC(=O)C=CC(F)F)N(CCN=[N+]=[N-])CC Cc1nn(C)cc1C(O)C(=O)NC(CNC(=O)CN1CC2CC2C1)C(C)C C(=O)(CCCC(C)C)N1CC(CCC)C(C(=O)NCCc2cc[nH]n2)C1 c1(C(N2CCN(C(C(C)OC)=O)CC2CCO)=O)cncc2nc(C)[nH]c12 Cc1cc(N)cc(C(N2CC(CNC(=O)Cc3cccnc3Br)C2)=O)c1F C(C)(CC(=O)NC1C=CC(C(=O)N(C(C)CO)C2CC2)C1)OC N1(C(c2cc(CC)cc(C)n2)=O)CCC2CN(C(C3C4CC5C(C4)C35)=O)CC12 C1(NC(CC(CCC)C2CC2)=O)CN(C(=O)CCC(=O)NCC)CC(C)(C)C1 c1(SC(C(=O)NCC=CCNC(CCNC(CC(C)C)=O)=O)C)cccc(Cl)c1 c1(C(=O)NC2C(NC(C(C=C)(C)C)=O)COCC2)nccc2ccccc12 Cc1nn(C)c(C(=O)NC(C)CNC(=O)C(c2ccc(F)cn2)(F)F)c1[N+](=O)[O-] Cc1cc(C(C)C(=O)NC23CC(NC(=O)Cc4cc(C)on4)(C2)C3)cc(F)c1 C1(C(N(CC(=C)C)CC)=O)CC2CC1CC2NC(=O)CNC(=O)OC C1(C(=O)NCCNC(CC)=O)CC(C)(C)CCN1C(=O)C(O)CCN(C)C C1(C(N2CC(C)C(CO)CC2)=O)CC2CN(C(=O)C(C)OC(C)(C)C)CC2C1 N1(C(c2ccc(N(CC)CC)cc2)=O)CC2CCC2(NC(C2CC(O)C2)=O)C1 C1(CNC(C2OCCN(C)C2)=O)COCCN(C(c2cc(Br)co2)=O)C1 C1(CNC(C2(CC)CCCO2)=O)(NC(=O)COC2CC=CC2)CCC(C)(C)CC1 C(c1cc[nH]n1)=CC(=O)NC(C(N1CCC(n2ccnc2)C1)=O)c1ccoc1 O=C(C1=C(Cl)CC1)NCC1CCN1C(=O)Cc1cc(Cl)sc1Cl C=CC1(C2(C(=O)NC3CCC(CNC(c4ncncc4Cl)=O)C3)CCC2)CCC1 c1(C(=O)NCC2C(NC(CNS(NC)(=O)=O)=O)C2)cc2c(Cl)cncc2s1 C1(NC(c2c(SC)cnn2C)=O)CCCC(NC(c2cc(C(N)=O)no2)=O)CC1 c1(C(N2CCC(C(c3ccccc3)O)CC2)=O)cc(Br)ccc1Cl CC(C(O)C(F)F)NC(=O)CC1CCCC1NC(c1cc[nH]n1)=O CC1CC(NC(=O)NC2CCC(NC(C3CCCCC3)=O)C2)CC(C)O1 C(=O)(CC1=NN(C)C(=O)C1)NC(CCC(=O)NC(CC(C)(C)OC)C)C(C)C c1(OCC2CC2)cccc(C=O)c1.C(=O)(C(C)C(C)O)NCCOC1CCN(CC)C1 CCC(C)CC(C(=O)NCCC(C)(C)O)NC(c1cocc1C)=O C(CCN(C)C(c1ccnc(C(C)(C)O)c1)=O)(C(C)(C)C)NC(CC(C)F)=O c1(OC)cc(C(=O)NC2(CCCCNC(c3cc(C)[nH]n3)=O)CC2)cc(C)n1 C12(CNC(c3cc(C)ns3)=O)CCC1CN(C(c1cc(C)n(C(C)C)c1C)=O)C2 C1(C(=O)NC2(CCOC)CCN(C(=O)C=C3CCSCC3)C2)CCC2CC2CC1 C1(C)(C(N2CC(OCCNC(c3c(F)ccc(C)c3)=O)C2)=O)CCS(=O)(=O)CC1 c12ncc(cc1F)NCC1C3CN(CC13)C2=O.CC1CC(C(=O)N(C)C2CC2)C1 C(=O)(CC(C)(C)C#N)NC(C)C(C)C(=O)N(CCO)CCO C#CCCCC(=O)NCc1ccccc1CNC(=O)C(C)C(=O)OCC CCCCC(C)(F)C(=O)NC(C)C(=O)N(C)CCc1cnc[nH]1 c1(C(C)NC(c2cn(-c3cc(C)sc3C)nn2)=O)c(CC)cccc1C c1(C(=O)NC(C(C)NC(C2C(COC)C2)=O)(C)C)oc2ccc(Cl)cc2c1C N=c1[nH]c(Cl)c(Cl)cc1C(=O)NCCC1(O)CN(C(=O)Cc2cnc[nH]2)C1 C1(OC)CN(C(=O)CCOC2CCCC2)C(C)(CNC(=O)CCF)C1 CON(CCC(=O)N1CC2(CC=CC2)C1)C(=O)C1CCC(=O)O1 N1(C(C=CSC)=O)CC(C2CN(C(=O)CC3CCC34CCC4)C2)C1 c1(CC)cc(C(N2CCCC(NC(=O)Cc3cncn3C)CC2)=O)ccc1OC C1(NC(C(C2CC2)NC(c2cnc(CC)o2)=O)=O)CCCCCC1 c1(C(N2CCC(CCNC(c3nccc(C)c3)=O)C2)=O)ccnc2c1cnn2C N1(C(C2N(C(CC)=O)CSC2)=O)CCN(C(c2cn(CCOC)cn2)=O)CC1C c1(C(N2C(C(C)(C)NC(C3C4COCC34)=O)CCC2)=O)cc(Cl)c(F)cc1O N1(C(C2(NC(c3c(OC)ccs3)=O)CCCC2)=O)CCCC2(CC2)C1 CC(CCCCNC(C1(O)CCOCC1)=O)NC(=O)C(N1CCCC1)C1CC1 Cc1cc([N+](=O)[O-])ccc1OC1CCN(C(c2cncc(Cl)c2Cl)=O)C1 C1(c2scc(CC)n2)CCCN(C(=O)CNC(=O)Cc2nncs2)C1 N1(C(c2ccnc(OC)n2)=O)CCN(C(C23CC(C)C2C3)=O)C(CC(F)F)C1 C1(NC(c2cc(CC)ncn2)=O)CC2CC(NC(=O)Cc3ccsc3)C2C1 c1(C(N2CC(O)CC(NC(CC(C=C)(C)C)=O)C2)=O)cnn2ccncc12 N1(C(CCC)=O)CCCN(C(=O)Cc2cccc(Cl)c2OCC)CC1C c1(C(=O)NCC(C(C)C)NC(C2CC=C(C)CC2)=O)cc(Cl)cc(Cl)n1 c1(C(N2CCC(CC(=O)NC3CC4CNCC34)C2)=O)cncc(C(F)F)c1 N1(C(C=C(C)C(F)F)=O)CC2(C1)CN(C(c1coc(O)n1)=O)C2 N1(C(C(C2CCN(C(c3c(CC)cco3)=O)C2)F)=O)CCC(F)(CF)C1 C(=O)(CCCC(F)(F)F)N(C)CC1(NC(c2ncncc2F)=O)CC1 O=C(N=c1ccnc2[nH][nH]cc1-2)C1CC2CC2N1C(c1csc(C(F)(F)F)n1)=O CC(C)CCC(C)N(C(=O)C(=O)NCC1CCN(S(C)(=O)=O)C1)C C(=O)(C(F)(F)CCn1ccnn1)NC(C(C)C)(C)CNC(C1(C#N)CCC1)=O c1(CC(N2CCC3(C(NC(CCN(C)CC)=O)C3)C2)=O)c(C)nc(O)nc1O c1(C(N2CC(C)C(CNC(c3cnccn3)=O)CC2)=O)cn2cccc(Cl)c2n1 N1(C(=O)C2=C(Cl)CCCC2)CCC2CCN(C(C3CC4(CCCC4)CO3)=O)C2C1 c1(C(=O)NCCCCCN(C(C2(CC#C)CC2)=O)C)cc(C(=O)OC)c(C)[nH]1 c1(NC(=O)NC2C(C#N)CCC2)c(C2CC2)cccc1F c1(OC)ccc(NCCC(=O)NC(C2CCCN2C(c2csnn2)=O)C)cc1 CC(C1=CCN(C)CC1)NC(C1CC2CN(C(=O)C(C)(Cl)Cl)CC2C1)=O CCCCC(C(=O)N(C1CCCCCC1)CCNC(C1CC=CCO1)=O)C(C)C C(=O)(C1CCCn2ccnc21)N1CCC(OC)(CNC(=O)CNC=O)C1 N1(C(CC(C)F)=O)CCOC(C(=O)N(C2CCCCC2O)C)CC1 C1(c2ncc(-c3c(C)cccc3)o2)CN(C(=O)Oc2ccccc2)C(C)CO1 S(=O)(=O)(c1ccc2[nH]c(=NCC(F)F)sc2c1)N(CCC(F)(F)F)C Cc1cccc(C2=CCN(C(=O)NC3CCN(CCN(C)C4CC4)CC3)CC2)c1 C1(C(=O)NCc2c(CC)noc2C)CCCCCN1C(=O)C(C)NC(C)=O C(C(=O)NC(CC(C)C)C(=O)NCC1CCCCCC1)(C(C)(C)C)OC CC(C)CC(C)(C)C(=O)NCC(F)CNC(=O)Cc1ccc2nn[nH]c2c1 C1(F)(CNC(C(=Cc2ccco2)C)=O)CCN(C(=O)Cn2ncn(C)c2=O)CC1 N1(C(C(C2CN(C(=O)C(n3ccc(C)n3)C)C2)OC)=O)CCC2(C=CCO2)CC1 C1(O)(C(=O)NC(c2cccc(Br)c2)C)CCN(C(C2CCC(F)(F)C2)=O)C1 c1(NC(C(N2CC(OC)C(c3ccncc3)C2)=O)=O)cc(F)ccc1C C1(NC(=O)Cn2cnnn2)CCN(CC(F)F)CC1.C12CCN(CC1)C2 c1(CCC(=O)N(C)CC2CCCN(C(C3C(C=C)CC3)=O)C2)c(C)ncnc1O c1(C(=O)NCC(C)CNC(C2(O)CCC2)=O)cccc(C2CC(F)(F)C2)c1 CC1CCC(C(N2CCC(N(C(c3ccco3)=O)CC3CC3)CC2)=O)C(=O)N1 C1(C(N(CCC)CCC)=O)CN(C(c2cc(Br)ccc2C)=O)CCC1(F)F Cn1nc(C(=O)N(CCCNC(C2(C(C)(F)F)CCC2)=O)C2CC2)cc1Cl C12(C(N3C4C(NC(CN(C)C(N)=O)=O)C(CC4)C3)=O)CCC(C)(C(=O)O1)C2(C)C c1(N2CCC(C)(NC(=O)CC(c3cccc(F)c3)O)C2)ncnc2c1CCC2 C1(C(N2CC(C=C)(CC(=O)NCCC(O)C(F)F)C2)=O)CCCCCN1C C#CC1(C(N2CCCC(CC)CC2)=O)CCN(C(c2ccsc2)=O)C1 C(CCCC(=O)N1CC(CC(=O)NOC(C)C)CC1C)SC c1(C(=O)NCC(C)N(CC(N)=O)C)ccc(C(F)(F)F)o1 N1(C(c2c(C)n(C)nc2)=O)CCCC(C)C1CCNC(=O)C=C1CCN(C)C1 N1(C(C(c2ccc(F)cc2)C)=O)CCC(NC(C2CCN2C)=O)C12CC2 C1(C)(C(=O)NCC(C(=O)NCCn2c(CC)nnc2)O)CCN(C)CC1 C12(C(N3CC4(CN(C(CCc5nc(C)c(C)[nH]5)=O)C4)C3)=O)CC1Cc1c[nH]nc12 c1(C(N2CC(O)(C(C)NC(=O)CN(C)C)C2)=O)cc(F)ccc1NC(=O)C1CC1 CCC(C)(C)C(=O)C(=O)NC1CCCC(C(=O)N(CC(C)(C)N(C)C)C)CC1 c1(CCn2cc(C3CC(C(=O)OC)(OC)C3)nn2)c(Cl)n(C)c2cc(C)ccc12 c1(C(=O)NCCC2(O)CCN(C(C3C(C#C)C3)=O)C2)cc2[nH]nnc2cc1OC N1(C(C(C=CCCC)O)=O)C2COCC1CC(NC(C1CC(C(F)(F)F)C1)=O)C2 N1(CC(N2CCN(C(c3c(C)nncc3)=O)CC2)=O)CC(=O)N(C)C1=O Cc1noc(C)c1C(N1CCCC1CN(C)Cc1ccnc(Cl)c1)=O c1(OCC)ccc(C(=O)NCCCCCCNc2ncnc(O)c2Br)cc1C CC1(C)CCOC1C(=O)NCCC1(NC(C2CCCC2(F)F)=O)CCC1 c1(C(=O)NC2CCN(C(C(=O)NCC)=O)C2)ccc(F)c(Cl)c1N N1(C(c2ccc(-c3cc(C#N)on3)cc2)=O)CC2OCCOC2C1 C(C(C)(C)CCl)(c1n(CCCCCC)nnn1)NCCC(=O)N(C)C C1(C(=O)NC2CCCC2)CC2CC2N1C(C1CC1c1ccc(Cl)cc1)=O CC1C(C)N(C(c2nn(C)cc2N)=O)CCN1C(C1CC2(CSC2)C1)=O CC(C)CCC(C(=O)NCCc1ncccn1)NC(c1cc(F)cc(F)c1)=O C12(NC(c3cncc(C)n3)=O)CCOC(CNC(c3csc(C)c3N)=O)(C1)C2 C(=O)(C(CO)C(F)(F)F)N1CC(C)(CCC(N2CC(=O)NC(C(N)=O)C2)=O)C1 CC(C)C(CC(=O)NC(C)(CO)C1CCCC1)NC(C1(n2cccc2)CC1)=O N1(C(C(C)NC(=O)NC)=O)CC(C)(C)CC1CNC(c1ccc(CO)c(F)c1)=O Cc1ccc(C(N2CCCCC(N(C)C)C2)C(=O)NCc2cccs2)nc1Br C12(NC(c3cc(C)c(O)nn3)=O)CCCC1N(C(c1cnn(C)c1Cl)=O)CCC2 c1(C(=O)NCC2(NC(C3C(OCC)CC3)=O)CCCC2)ccnc(S)c1 N1(C(COCC(=O)NC)=O)CCC2(CCCC2CNC(C2CCCC(=O)O2)=O)CC1 C12(NC(c3c(Cl)nc(OC)s3)=O)CCN(C(=O)CCn3cccnc3=O)CC1C2 S(=O)(=O)(c1ccc(CCCc2nc(C(C)(C)C)cs2)cc1)N1CCCC(C)CC1 c1(OC)ccc2c(c1)CN(N1CCC(ON3CCCCC3)C1)CC2 c1(C(C)C)n[nH]cc1C(=O)NCc1n[nH]cc1C(N1CCC(CN(C)C)C1)=O N1(C(C2CCCCN(C(CC(=O)OC)=O)C2)=O)CCCC2CCCCC12 CC(C)C(C(=O)N(CCO)CCO)NC(=O)OC(C)(C)C.C12CCCN1C2 N1(C(C(COCC)N=[N+]=[N-])=O)CCC2(CC1)CC2C(N1CC(C(N)=O)(OC)C1)=O N1(C(c2c(CC)ncnc2)=O)CC2CCC(CNC(=O)C(C(C)C)N(C)C)(C2)C1 c1(OC)ccc2cc(C(C)NC(=O)N(C3CCCOC3)CCF)oc2c1 C1(C(=O)NC2CC=C(C)CC2)CC2CCC(C1)C2 N1(C(c2cc(C)c(C)c(C)c2)=O)CCCC2(CCCCC2O)C1 N(C)(C(=NCC1=C(C)OCCS1)NC(C)C)C(c1ccc(NC(C)=O)cc1)=O C(C(=O)NOC1CCCCC1)(C1(C)CC1)NC(=O)C=CC1CCOC1 CC1CCCC(CC(=O)NC2CC3(C2)CC3C(=O)NCC2C3CN(C)CC23)O1 C1(NC(CN2CCC(OC)C2)=O)CC(C(=O)NC2CC3(CCOC3)C2)=CC1O N1(C(C2(C=C)CCN(C(=O)Cc3c[nH]nc3C)C2)=O)CC2(CO)CCC1CC2 c1(C(=O)NC(CCOC)CNC(=O)C(O)CC(C)C)ccc2cc(Cl)ccc2c1 C1(NC(CC2CC(SC)C2)=O)CC(CC(=O)NC2(CN(C)C)CC2)C1(C)C N1(C(CC(C(F)F)NC(CC(CC(=O)OC)C)=O)=O)CC(C)c2ncccc21 C1(NC(=O)Cc2cscn2)CS(=O)(=O)C2CN(C(=O)CN3CCCS3(=O)=O)CC12 C1(N(CC(=O)NCCN(C(C2CC2c2cccnc2)=O)CC)C)CCCCCC1 C1(SC)CN(c2ccnc(NCC3(NC(=O)OC(C)(C)C)CC3)n2)CC(C)S1(=O)=O CC1CC(CC(=O)NCCC(O)CNC(c2ccc3c(c2)CC3)=O)CC(C)(C)C1 c1(CC)ncc(C(=O)NC(CCNC(=O)C(c2ccc(Cl)s2)C)C(C)C)cn1 N1(C(c2c(C)nns2)=O)CCCCC1CNC(=O)Cc1ccn(C)n1 C#CCCC(O)C(=O)N1CC(NC(c2c(Cl)cnn2C)=O)C(c2ccccc2)C1 N1(C(C)C)C(=O)COCC1C(=O)NCC1C2CC1N(C(=O)Cn1cncn1)C2 C=C(C)CCCC(=O)NC(c1cccnc1)C(=O)NC(C)CC N1(C(C2CN(C(C)=O)C2)=O)CCCC(NC(=O)C#CC2CC2)C1 Cc1cnnc(O)c1C(N1CC(CN=c2[nH]nc(C3CC3)o2)(O)C1)=O C#Cc1cccc(C(N2CCC2CNC(=O)Nc2ccc(F)cc2C)=O)c1 C(CCO)(C(F)(F)F)NC(CC1(C)CCN1C(=O)CC1CCOCC1)=O N1(C(C(c2cnn(C)c2)C)=O)CC(n2cc(-c3c[nH]c(C(=O)O)c3)nn2)C(O)C1 C(=O)(C1=Cc2ccccc2C1)NC1(CNC(C2(F)CCC(C)CC2)=O)CCCC1 c1(C(C(=O)NC(C)CC)N(CCOCC)C)ccc(CC)c(C)c1 C1(C(=O)NCCN(CCOC)C(C2SCCCS2)=O)CCC2(CC1)CC2 c1(C(=O)NCC(C2CCC2)NC(c2c(COC)cco2)=O)ncncc1OC CC(CO)CCN=c1cc[nH]cc1S(=O)(=O)NC1CCCC(O)CC1 C(=O)(C1CCC(=O)c2ccccc21)N1CCN(C(c2ncn(C)n2)=O)C(CO)C1 CN1CC(C(=O)NCC23CC(CCO2)C3)N(C(=O)COCC2CCCOC2)C1 N1(C(C(=O)NC(c2cccc(Br)n2)COC)=O)CC2C(C1)C2(C)C c1(NC(C2CC(F)CN2Cc2ccc(Cl)nn2)=O)ncc(Br)nc1Br c1(C(c2nnnn2C(C)C)OCC)cn(CC2(CCCC)CC2)cn1 C12(NC(CN(C)CC)=O)CC3CCC(C1C2)N3C(=O)CCc1c[nH]c(C(N)=O)c1 n1(CC(=O)NCC(CNC(CCCc2nc(C)sc2)=O)(C)C)cc(F)ccc1=O C#CC1CC1C(=O)N(CCNC(C1CCC1CF)=O)CC CCC(C)CC(C)C(=O)N1CCC(CNC(c2cccc(OC(C)C)c2)=O)C1 C(=O)(CC(C)(C)C=C)NCC1(CNC(CCCOCC=C)=O)CCCCC1 CC1(C)COC(C(=O)NCC(C)(CO)NC(=O)CC2COCC2(C)C)CO1 C1(CNC(c2cc(COC)sc2)=O)CN(C)CCN1C(c1cc(O)ccc1F)=O N1(C(=O)Cc2ccncc2)CC2CCC(C1)N(Cc1cc(Br)c(F)cc1Cl)C2 C(CCC(=O)NC(CNC(=O)CCCC1CCOCC1)CO)=CCC=C C1(C(=O)NC2CN(C(C3C(C)(C)C3CN=[N+]=[N-])=O)C2)CCC2(C1)N=N2 CC(F)CC(=O)NC(CC12CC(C1)C2)C(=O)NCCC(O)CO N1(C(C2CC(C)OC2)=O)CC(C2CCCN(C(c3cnc(O)nc3O)=O)C2)C1 C=CCCCCCC(=O)N1CC(O)(C(C)NC(=O)C(CO)c2ccccc2)C1 C1(C(=O)NCC2(NC(C3CSCN3C(C3CCC3)=O)=O)CCC2)CCOCC1 C=CCC(CC(C)C)C(=O)NCC1(NC(=O)CCc2ncccc2C)CCC1 c1(C(N2CC3CC3(C(=O)Nc3cncc(F)c3)C2)=O)c(C(F)(F)F)cccc1Cl Cc1c(C(N2CCC(O)(CCNC(C3(C)CCCO3)=O)C2)=O)sc2nccn12 c1(NC(C(=O)NC2CCCN(C(=O)OC(C)(C)C)CC2)=O)c(Br)cc(Br)c(O)c1Br C12(C(N3C(CNC(C4N(C(C)=O)CCCC4)=O)CC3)=O)CCC(C)(C(=O)O1)C2(C)C c1(C(N2CCCC(C(=O)NCCC#C)C2)=O)cccc(Br)c1O c1(CNC(C2CC(OC)CN2C(C2CCN(C)C2)=O)=O)c[nH]c2cnccc12 C12(CNC(c3cc(C)cc(O)c3)=O)CN(C(C34CCC(C3)C4)=O)CC1CCO2 N1(C(=O)NC)CCC(C(N2CC(NC(C3(N4CCOC4=O)CC3)=O)C3CC23)=O)CC1 N(C1CCCc2nn(C)cc21)C(C(C)(CC)CC)c1n(CC)nnn1 C(=O)(CC(C(F)F)NC(c1c(C)nccn1)=O)NC12CCCC1C2 C1(NC(C(COC)OC)=O)CCC(O)CN(C(=O)CN2CCN(C)CC2)C1 c1(C(=O)NCC(CC)NC(C2C3CCOCC23)=O)cn(C)nc1C1CCCC1 c1(C(=O)NCCC2C(C)C2)cc(CNC(=O)Cc2nccn2C)cs1 C1(C(N(CCCNC(=O)CC2CCCC2C)CCC)=O)CC(F)(F)C1(C)C C1(c2ccccc2)(NC(=O)NC(C)C(N)=O)CC(F)(F)C1 CCCCCC(C)(CC)C(=O)NCC1CCN(C(=O)C=CI)C1 C1(O)(CNC(C(C2CCC2)OCC)=O)CCN(C(c2ccc(N(C)C)nn2)=O)C1 CC1(C)C2CN(C(c3ccc(NC(c4ccc(N(C)C)cc4I)=O)cn3)=O)CC12 c1(N(C)C)nc2cccc(C(N3CCCCCC3CNC(C3(O)CC3)=O)=O)c2o1 c1(CC(N2C3CN(Cc4cccc(F)n4)CC23)=O)ccccc1[N+](=O)[O-] C(F)(C(=O)NCCC1CC(NC(=O)C(C)n2cnnn2)C1)OC C1(NC(CSCC(=O)OC)=O)CC2(CCN(C(c3ccns3)=O)C2)C1 C1(C(N(C)Cc2cn[nH]c2)=O)CC12CCN(C(c1cnc(S)nc1)=O)C2 c1(C(=O)NCC2N(C(Cc3cnc(C)s3)=O)CCC2)cccc(N=S(C)(C)=O)c1 CCCCC(C)C(=O)NC(C)CC(C)NC(c1cn(CCO)nc1C)=O C12(C(=O)NC3(CO)CN(C(C=CC)=O)C3)CCCC1(C(=O)O)C2 N1(C(C(c2cccs2)NC(c2c(C)n(C)cc2)=O)=O)CC2CC3CC2C1C3 S(=O)(=O)(c1cccc(C(N2CCC(F)C(NC(=O)C3CC3)C2)=O)c1)NC C(=O)(CC1=NNC(=O)C1)N1CCOCC(CNC(=O)COCC2CCC2)C1 C1(C)(C(N2CC(CC(=O)NCC(C(C)C)O)OCC2)=O)C(C)(C)C1(C)C C(N=c1ccn(CC(=O)NCc2cccc(Br)c2)c(O)n1)c1ccc(C)cc1F C=Cn1nccc1C(N1CC(CC(=O)NCC(C2CCC2)OC)(OC)C1)=O C(CC(F)F)(C(=O)N1CCN(C2(C)CC2)CC1)NC(c1ccnc(C)n1)=O CC1CC(=O)NC(C(N2CC(=O)NCC2C(=O)NC2CCC=CCC2)=O)C1 C1(NC(C2C(CC)OCC2)=O)CC(C)N(C(=O)CC2CC3(CCC3)C2)C1 c1(OC)ccc(F)c2[nH]c(C(N3CC(CNC(=O)CN4CCCCC4)C3)=O)cc12 C12CCCCN1C(=O)CCCC1(CCC1)N(CCC(=O)OC)C(=O)C2.CN.OC C1(C(=O)NCCNC(c2nccc(CC)c2)=O)CC2CCCC(C1)C2=O N1(C(c2ccn(CC)n2)=O)CCCCC(CNC(=O)Cc2conc2C)C1 CCCCCC(C)CC(=O)NCCOCC(N1CCCCCC1C(C)C)=O N1(C(c2c[nH]c(=NC)o2)=O)CCC(C)(C)C1C(=O)NC(c1ncc[nH]1)CO C1(CC(=O)NC2(C=C)CCC2)CCN(C(=O)C(C)CN(C)C)C1(C)C C1(CNC(c2c(C)ncs2)=O)C2CCCC1N(C(=O)CSc1cn[nH]c1)C2 C1(C(=O)NC2CC(C)(CNC(C3CC(O)C3)=O)C2)CCCC(C)(C)CC1 C(c1cncc(F)c1)=CC(=O)NC(C1(O)CCN(C(c2cnc(CC)s2)=O)C1)C C1(NC(c2cnc(Cl)s2)=O)CC12CCN(C(=O)CN1CC=CC1)CC2 S(=O)(=O)(c1ccc(Br)cc1)N1CCC(NC(=O)OC(C)(C)C)C12CCC2 c1(OC)ccc(F)c2cc(C(=O)NCC(C)CN(C)C(C3CC3C(N)=O)=O)[nH]c12 N1(C(C(CC#C)C)=O)CCCC2CN(C(C3CC(SC)C3)=O)CCC12 C1(SC)CN(C(=O)Cc2scnc2C)CC1NC(c1csc(C(C)(C)C)n1)=O N1(C(C(N2CCCCC2=O)C)=O)CC(NC(C2CC3CC3C2)=O)CC12CCCC2 N1(C(c2nc(CC)oc2)=O)CC(CNC(c2ccc(C(C)=O)nn2)=O)CCC1C C1(CNC(C(CC=C)(C)C)=O)CN(C(c2ccc(CC)[nH]2)=O)CCC1(F)F CCC(CC(F)(F)F)C(=O)N(CC(C)NC(C1CC2(C1)CC(C)(C)C2)=O)CC N(C1CN(C(=O)C2=CCC(C)(C)CC2)Cc2ccccc21)C(C)=O CC1(C)CC(C(=O)NC2COCC2C(=O)NCCOc2ccncc2)CCO1 C(=O)(C(C)CS(C)(=O)=O)NC(CC)CNC(=O)CC1CCCN1C(=O)OC C=CCC(C)(C)C(=O)NC1CCN(C(=O)C=Cc2ncc[nH]2)C(C)C1 c1(OC)ccc(NC(C2CN(C)CCN2C(C2CC23CC3)=O)=O)cc1C C(C1c2ccsc2CCN1C(c1sccc1F)=O)NC(CSCC=C)=O N1(C(=O)NC2CCCCN2)CCc2nc[nH]c2C1c1ccc(F)cc1 C1(C(=O)NC(C)CCNC(=O)CC23CCC(CC2)CC3)CS(=O)(=O)CC12CC2 N1(C(C(C(C)C)NC(C)=O)=O)CCC12CN(C(C1CC(=O)NC(=O)N1)=O)C2 CCCCC(C(=O)NCCOCc1ccccc1)NC(=O)C(C)(C)Cl C(C(=O)N=S(C)(C)=O)NC(c1ccncc1C)c1n(CCCSC)nnn1 C=CC1CCCN(N2CCN(c3nc(Cl)ns3)CC2)C1 CC(C)(C)C(O)C(=O)NC1C2CC(NC(=O)C(C)(F)CC3CCCC3)CC12 C1(C(N2CC3C(CNC(=O)CCC4CCOCC4)(C3)C2)=O)(CF)CC2(CCC2)C1 c1(N(CC)CC)cccc(CCC(=O)NC23CC2CN(C(=O)CC(C)OC)C3)c1 CC1(C)COCCC1C(N1CCC(CNC(=O)Cc2csc(C(F)F)n2)CC1)=O CC(C)(C)C1CCNc2c(NC(C3(Oc4ccccc4)CCC3)=O)cnn21 N1(C(C=C(COC)C)=O)CCC(NC(=O)CSC2CCCCO2)C1C1CC1 C12(NC(C(CC=C)NC(C)=O)=O)CCC(CNC(c3ccsc3)=O)(C1)OC2 C1(CC(N2CC=CCC2c2cccnc2)=O)CNC2(CCOCC2)CO1 C1(C)(CNC(Cc2cnn(C)n2)=O)CC(F)(F)CN1C(c1cccc(Cl)c1O)=O C1(C(C)C)CN(C(C2COCC2NC(C2CCC3CC2CO3)=O)=O)CCCO1 C1(CC)CCCN(C(c2ccc(CO)o2)=O)C1C(=O)NCC1(O)CCN(C)CC1 N1(c2nc(N3CCC(CCO)C3)cc(C)n2)CCC2(CCCCO2)C1 C(=O)(CC(CC)N(C(=O)C(C)O)C)NCC1(CCC)CCC1 N1(C(CCNC(C)=O)=O)CCCCC1C(C)NC(C1CC(CC2CC2)C1)=O C1(CNC(c2cc(OC)ns2)c2nnnn2C2CC(F)(F)C2)CC(C)(C)C12CC2 C1(NC(C(CC)CC)=O)C2CCN(C(=O)CC3CCCO3)CC12 c1(C(N(C(CNC(C2CCC2C(C)(C)C)=O)C2CC2)C)=O)cc(Cl)c(Cl)n1C C1(NC(C(C)(C)CC#N)=O)CCC2(CC1)CCN(C(c1conc1C1CC1)=O)C2 c1(CNC(C=C(C)C)=O)ccc2c(c1)CCC2NC(=O)C(F)(F)c1nccs1 CCCC(C(N)=O)NC1CN(C(=O)CCn2cc(CCOC(C)=O)nn2)C1 C(=O)(CC(C)C(=O)OCC)N(CCCNC(c1cc(OC)no1)=O)CCC C=C=CCCC(=O)NC(C)(C)C=CC(=O)NCC(N1CCOCC1)=O c1(C(=O)NC2(CC=C)CCN(C(=O)C=CBr)CC2)[nH]c2c(C)cccc2c1C c1(OC)c(F)cc(C(=O)NCC(C2CC2)NC(C2CCC(C)(C)CO2)=O)cc1Cl c1(C(CC)N(C)C(=O)NC2CC2(CC)CC)noc(C)n1 Cc1csc(=NCC(=O)N2CCC3C(NC(=O)C(O)CC(F)(F)F)CC23)[nH]1 c1(C(=O)OCC(c2ccc(C)n2C)=O)cc(O)cc(=O)o1 N1(C(C2CN(C)C(=O)N2)=O)CC2CCC1(CNC(=O)CCCS(N)(=O)=O)CC2 N1(C(C(C=C)(F)F)=O)C2CCCC1CC(NC(c1ccccc1S(C)(=O)=O)=O)C2 CCC(C)C(O)CC(=O)NCC1(NC(=O)C2=C(C#N)CCC2)CCCCCC1 CC(C(C)C(=O)N1CCC(NC(=O)CSCC2CCCCO2)C(C)C1)S(C)(=O)=O N1(C(C2C(C(C)O)C2)=O)CC(CNC(C2CC2(C)C)=O)C1 c1(C(=O)NCC(C(=O)NCc2ccnn2C(C)C)OC)cccc(Cl)c1 N1(C(C(N2CCC(C)C2)=O)=O)CCCC(O)(CNC(C2(C(N)=O)CC2)=O)CC1 C12CCC(CC1)NC(=O)C2.C1(CC(=O)OC)CC(NC(=O)COC(C)C)C1 c1(C(=O)NC2C(CNC(CNC(C)=O)=O)CCC2)ccncc1Br N1(C(C(C(C)NC(c2ccccn2)=O)(C)C)=O)CC2CCC(O)C(O)C12 c1(NC(C)C(C2CCCCC2)NC(C2CCOC2)=O)ncc(C#N)cc1Br N1(C(CC(CC)O)=O)CCC(NC(c2c(C)coc2C(C)(C)C)=O)C(CC)C1 C(=O)(C(CSC)NC(=O)CCCn1cncn1)OCC.C1(NC=O)CCC1 C1(F)(C(=O)NCC2C(C(NOCC3(C)CC3)=O)CCO2)CCOCC1 Cc1c(NC(=O)C(CCC2CC2)NC(c2csnc2Cl)=O)cnn1C N1(C(C(F)=CC)=O)CCC(CNC(c2n[nH]cc2-c2ccccc2)=O)C(C)C1 c1(C(N2CCN(C(C3CC=C(C)CC3)=O)CC2)=O)cccc(Br)c1N N1(CC)CC(C(N2CCC(O)(CNC(C3CN(C(C)C)C3)=O)C2)=O)CC1=O Cc1nn(C)cc1C(O)C(=O)NC1CN(C(c2nocc2Cl)=O)CC1C C1(CNC(C2(CCC)CC2)=O)CN(C(c2occc(=O)c2OC)=O)C(C)(C)C1 C1(C(=O)Nc2c(C)nsc2)(NC(c2cc[n+]([O-])cc2)=O)CCCC1C NC1COC2(C(N3CCOC(c4ccc(F)c(Cl)c4)C3)=O)CC1C2 C(=O)(C1=CC2CCC(C1)C2)NCC1(CNC(C(CC#C)(C)C)=O)CC12CCC2 c1(OC)cc(N2CC(NC(C3CC4CC3C3CC43)=O)CCC2C)ccc1[N+](=O)[O-] C=C(C)CC(C(=O)N(C(C)CSC)C)NC(c1ncoc1CC)=O C1(C(N)=O)CN(C(C2CCCC2NC(=O)C#CC2CC2)=O)CC12CC2 C1(C(=O)OC(C)(C)C)(C(=O)NCCNC(=O)CC2CCCC2(F)F)CCOCC1 c1(OC)nc(=NCC2CCC2(F)F)[nH]c(OC)c1[N+](=O)[O-] C(=O)(C1=CCCCCC1)NC(CC#C)C(=O)NCC(C)(O)CN(C)C c1(C(N(C)Cc2cc(Cl)ccc2Cl)=O)cc2c(ncc3ccccc23)s1 C(N=c1[nH]c(=NCCCN2CCC(O)C2)c2ncccc2[nH]1)c1n(CC)ncn1 c1(C(N2C(CNC(C(CCC)OC)=O)CC2)=O)c(F)ccc2nc[nH]c12 N1(C(CCCOC)=O)CCC2(CC1)CN(C(c1ccc(F)c(C)c1)=O)CC2CO C1(CC(=O)N(CC(=O)NCCN(CC(F)(F)F)C)CCOC)CC1(C)C C(=O)(CC(C)(C)CN(C)C)NC(C)C(C)C(=O)NCCS(N)(=O)=O c1(-n2ncc(C(N(CC(CNC(C(CC)(C)C)=O)O)C)=O)c2)ccc(F)cc1F N#Cc1ccc(CNC2(c3nnnn3CC(F)F)CCNCC23CC3)cc1F C1(NC(C2C(=C)C2)=O)CCC(CN(C(=O)CCCc2cnccn2)C)CC1 C1(C(=O)NC(COCC)C)CC=CCC1NC(C1(COC)COC1)=O c1(OC)cc2c(cc1OC)C(=O)C(SC1CN(S(C)(=O)=O)C1)C2 c1(C(N2CC(CNC(c3nocc3C3CC3)=O)C2)=O)ccc(-c2cn[nH]c2)cc1 C(C(CC(F)(F)F)NC(C1CC(=O)NC1(C)C)=O)NC(C(C=C)CC)=O N1(C(CCCC)=O)CC(C(=O)NC23CC(F)(C2)C3)C(F)(F)C1 O=S(=O)(c1cccc(N2CCOC(C(F)F)CC2)n1)NCCCOC1CCCC1 N1(C(C(C)(C)OC(C)=O)=O)CC2(CCN(C(=O)C3=C(Cl)CCCC3)CC2)C1 C1(C(=O)NCCCn2ccnc2)CC(O)CCN1C(c1cc(F)cnc1O)=O C=C1CC(C(=O)NCC(C)C#N)(CNC(=O)COCC)C1 c1(C(=O)NCCC2CCN(C(CC)C(N)=O)CC2)ccc(OC)nc1C C1(CC)CN(C(=O)CN(C2CCC2)C)CCC1NC(c1ccnc(N(C)C)c1)=O C1(NC(NCC(COC)(C)C)=NCC2CCCO2)CCn2c(C(F)(F)F)nnc2C1 c1(CNC(C(C(C)OC)NC(=O)CC2CNC(=O)O2)=O)nn(C)c(=O)n1C CN1CCC(CC(=O)NC(c2ccccc2F)CNC(=O)CO)CC1 C(=O)(CC(C(F)(F)F)n1ccnc1)NC1CC(CN(C(C)C(=O)NC2CC2)C)C1 N1(C(c2c(C)cccn2)=O)CCC(NC(C2CCC(=O)N2)=O)C(CO)CC1 c1(OCC)ccc(-c2cccc(NC(=O)CN(C)C)n2)cn1.c12ccccc1N2 c1(N(C)C(c2cnn(-c3ccc(O)nn3)c2C(F)(F)F)=O)nc2ccccc2o1 Cc1ccc(CNC(c2ccn(CC(F)(F)F)n2)=O)c2ccccc12 c1(OC(C)C(=O)NCC(CO)NC(c2cnc[nH]2)=O)ccc(F)cc1 C(=O)(C1CCC(=O)c2cccn21)NCCN(C(C=CCCC)=O)CC(C)O c1(CC)onc(C)c1NC(=O)C(C)N(C(=O)CCN1CCOC1=O)C1CC1 C(=O)(C1=CCC(F)(F)CC1)NCCCOCCNC(C1CCCC(=O)N1)=O C(C(C(=O)N(CCCOCCNC(C1CC1C)=O)C)C(F)(F)F)OC c1(C(=O)NCC2C(CNC(c3c(CC)nns3)=O)C2)cc2c(F)cc(Cl)cc2[nH]1 CC(N=c1nc2c(cnn2C)c(NCc2ccc(C(F)(F)F)o2)[nH]1)C1CC1 N1(CC)N=C(C(=O)N2CC=CC2CNC(c2cnc(C(C)(C)C)s2)=O)CCC1=O Cc1nccc(C(=O)NC23CC(NC(=O)CC4CCCN(C(C)C)C4)(C2)C3)c1Cl CC(C)CS(=O)(=O)CC(=O)N1CCOCC(CNC(=O)C(F)C2CCOC2)C1 C1(N(C(C(CC)O)=O)C)CCN(C(c2cccc(N)c2F)=O)CC12CC2 CC12CCC(C(=O)NCc3cccc(NC(=O)C(=O)c4cccs4)c3)(CO1)C2 C1(NC(=O)C=Cc2ccccn2)CC2CC(C1)N(C(c1cnc(C3CC3)[nH]1)=O)C2 C1(CC(=O)NC(CCOC)CNC(=O)C(C)N(C)C(C)=O)CCCCCC1 C(C(CNC(c1cnn(CCNC(c2cccc[n+]2[O-])=O)c1)=O)C(C)C)OC Cc1ccccc1CC(=O)NC(C)(C)CC(=O)N(C)CCN(C)C1CC1 C1(CNC(C(C2CC2)OC)=O)CN(C(=O)CCc2nc[nH]n2)C2(CCC2)C1 c1(C(=O)NC2CC(CO)NC2=O)cccc2ccc(Br)nc12 Cc1c(C(N2CCCC(C)(CNC(C3CSCN3C)=O)C2)=O)cnc2ncnn12 C1(NC(CC2(O)CCCN(C)C2)=O)CC2(CCCN(C(C3CC4CC4C3)=O)C2)C1 Cc1ccc(F)c(CS(=O)C(C)C(=O)N(Cc2ccccn2)Cc2ccco2)c1 N1(C(c2c(C)nn[nH]2)=O)CCCC(NC(c2cn3c(n2)CCC3)=O)C1C CC(=O)C(C)(C)CC(=O)NC1CCC(NC(=O)C2=CCCSC2)C1 N1(C(C(CC2CC2)OC)=O)CCC2OCCN(C(=O)C(=O)C(C)(C)C)C2C1 N1(C(CSCC)=O)C2CCCC1CN(C(C1Cc3ccccc3C1)=O)CC2 c1(CNC(C2CC=CC(NC(C3(C(N)=O)CC3)=O)C2)=O)cccc(F)c1O N(C(=NCCCOCC)NC1CCN(CCN(C)C)C1)N(CCCC)C C1(C(=O)N(c2c(OC)cc(C)cc2)CC#N)CC2CCC1N(C(=O)CC#N)C2 c1(CC(=O)NC(C=CC(=O)NCCC=CC=C)C)c(C)noc1C C12(CNC(C(=O)Nc3c(CN(C)C)cc(F)cc3)=O)CCCCN1CCC2 C1(C(N2CCC(NC(CC(CCC)O)=O)(COC)CC2)=O)CCc2nccn2C1 C(c1c[nH]nc1C)=CC(=O)N(CCNC(=O)C(C)OC)CC C#CC1CCCN1C(=O)C(CC1CC1)NC(=O)C(C)(CO)OC c1(OC)ncccc1CCC(=O)NC1CCN(C(=O)CN2CCNC2=O)C1 N1(C(CC(C)N(C)C)=O)CCC2C(C1)CN2C(=O)C(=O)NCCC(N)=O c1(C(N2CCC(C3(NC(C4C=CCC4)=O)CC3)C2)=O)ccc2cnccc2c1 Cc1[nH]nc2ccc(C(=O)N(C(C)CN(C)C(C3CCCCCC3)=O)C)cc12 C1(C(F)(F)C(=O)N2CCC(N(C)C(c3ccncc3Cl)=O)C2)(OC)CCCCC1 N1(C(C(N2CC3C(C(=O)Nc4nc(O)cc(C)n4)C3C2)C)=O)CCc2n[nH]cc2C1 C(=O)(C#CC1CCCO1)N1CCC(N(C(=O)C#CC2CC2)C)C1 C1(OC)(CNC(c2ccsn2)=O)CCN(C(c2ccnc(O)c2)=O)CC1 C1(CCOC)CCC(C(=O)Nc2ccc(-c3nn[nH]n3)nc2)CC1 C(=O)(C1=CCN(C(C2CC=C(C)CC2)=O)CC1)NCC1(SC)CCC1 CCCC(C(=O)NCC(C)CC1CCCC1)NC(C1(OCC)CCOC1)=O C12(C(=O)OCC(N3CCN(Cc4ccc(F)cc4)CC3)=O)CCC(CC1)CC2 N1(C(c2c(F)ccc(OC)c2)=O)CCN(C(=O)CNC(N)=O)CC(C)C1 Cc1cc(Cl)cc(N)c1C(=O)NC1CCN(C(=O)C(C)CC(F)(F)F)C1 CC1CC(C(N)=O)CN(C(c2ccc(CNC(=O)C3=COCCC3)nc2)=O)C1 C=CCC(CNC=O)C(=O)Nc1c(C)ccnc1OC C1(NC(CC2N(C(Cc3ccc(C)o3)=O)CC2)=O)CC12CCCC2 N1(C(c2ccc(OC)cc2)=O)C2CCC1CC(C(=O)NOC(=O)C(C)N=[N+]=[N-])C2 C1(CNC(CC(C)=C(C)C)=O)CC(C(=O)NCC=CC(C)(C)C)=NO1 C1(C(N(C2CN(C(c3cnc(SC)s3)=O)CC2O)C)=O)CCc2nnc(C)n2C1 c1(C(=O)NC2C(CNC(c3cc(CC)on3)=O)CC2)ccc(=O)n(CCOC)c1 CC(CNC(c1cccc(=O)o1)=O)C(F)C(=O)NCC(C)(C)C(C)(F)F n1(CC)ncc(Cl)c1C(=O)NCC(C)N(C(=O)CC(C)C1CC1)C C(c1cccc(Cl)c1)=C(C(=O)NCC1CCN(C(c2c(C)nc(OC)s2)=O)C1)C c1(COC)cc[nH]c1C(=O)N(CCC(=O)N1CC(F)C1)C1CC1 N1(C(c2cc(C)nc(C)c2)=O)CCC2(CCCN2C(C2CCOC2(C)C)=O)C1 c1(NC(=O)NC2C(CNC(=O)OC(C)(C)C)C=C2)nccn2nccc12 C12(C(N3CCC(C(N4CCC(C(C)(C)C)CC4)=O)C3)=O)CCC(CC1)CO2 C(C(O)C(F)(F)F)N(C)Cc1cn(Cc2cccc(Cl)c2)nn1 C1(CC=C)(C(=O)NCC=CCSC)CCN(C(c2nc(C)sc2C)=O)C1 Cc1nc(=NCCN(C(=O)CCC2CCCCC2)COC2CCCO2)[nH]cc1Br c1(C(=O)NCCN(C(=O)C(N2CCC(C)C2)=O)CC)ccn2nccc2n1 CN1CCCC(C)(CNC(=O)Cn2cc(CC3CCCNC3=O)nn2)C1 O=S(=O)(c1cccnc1N1CCC2CC2C1)NCC1(CCO)CCCC1 C(c1cccnc1)=CC(=O)NCCOCCNC(c1cn(CCCC#N)nn1)=O C(CC(C)C)(c1cccnc1)NC(=O)NC(c1nccn1C)CC C(C(CC(=O)O)CC(C)C)NCc1ccc(OC(C(=O)NC)C)c(Cl)c1 C(=O)(C1CCCc2cncn21)NC(C1CCN(C(C2COC(C)C2)=O)CC1)C C1(NC(C(C)(C)C2CCN(C(=O)C(C3CCCCC3)=O)C2)=O)COCC(C)(C)C1 c1(C(=O)NCC(CNC(=O)CNC(c2ccco2)=O)OC)n[nH]c2c1CCCC2 c1(C(N2CCC(C(=O)N=c3cc[nH][nH]3)(O)C2)=O)cc(F)c(Cl)cc1Cl C1(NC(C(C)OCC(F)(F)F)=O)CCC12CN(C(c1cn(C)[nH]c1=N)=O)C2 O=C(CC1=CCOCC1)N1CC(OCCC(=O)N2CC(N3CC(O)C3)C2)C1 CCCCCC(O)CC(=O)NC12CC(C(=O)Nc3sc(C)cc3Cl)(C1)C2 C#CCCCC(C)C(=O)NCC(C)(C)CN(C)C(C1CCc2n[nH]cc2C1)=O N1(C(C2OCCN(C)C2)=O)CCCN(C(c2cc(C#N)cn2C)=O)C(CO)C1 c1(CC)onc(C(=O)NCC(CNC(=O)CC2CC(OC)C2)OC)c1C N1(C(CSCCCC)=O)CCC(CO)(CNC(c2nn(C)cc2C)=O)CC1 C1(NC(C2CC=CC2)=O)CC(C(F)(F)F)CN(C(c2cc(Br)ccc2I)=O)C1 N1(C(c2cnc(OC)s2)=O)CCCCC(N(C)C(C2(C)CCN(C)C2)=O)C1 CC(C)CCCC(=O)N1CCC(CCC(=O)NC(CN(C)C)CO)CC1 N1(CC2CCC(CC)O2)CC2CCC1CN2C(c1cnn(CC(F)(F)F)c1)=O N1(C(C(C)C(C)O)=O)CCOCC(CNC(c2scnc2Cl)=O)C1 N1(C(=O)CCC2CCCCCC2)CCC2CN(C(C3(O)CCOCC3)=O)CC12 c1(CNC(C2CC(C)(F)C2)=O)nc(CNC(=O)CS(C)(=O)=O)cc(O)n1 CCC(C)(CNC(C1CN(C(C2CS(=O)C2)=O)CCO1)=O)CO C(CC(N)=O)(C(=O)NC1CCCC1CN(C)C)NC(c1nccc(OC)c1)=O c1(OC)cc2[nH]cnc2cc1C(N1CCCC(C)(OC)C1)=O C1(CCC(=O)NCCn2ncc(C)c2)CCCCN1C(=O)CC(C1CC1)C1CC1 c1(C(C)(C)C)ccc(C(N2CCC(NC(C3CC(C)(CN)C3)=O)CC2)=O)c(N)c1 C1(CC(C)O)CCCN1C(C1(CCNC(=O)CN2CCOC2=O)CCCC1)=O Cn1[nH]c(C(=O)NCCC2(NC(=O)Cn3nnc(-c4ccco4)n3)CC2)nc1=O Cc1ccc(C(N2CC(C3CCN(C(C4CC5CC(=O)C4O5)=O)CC3)C2)=O)c(O)n1 c1(C(=O)NC(C(C)NC(c2cnc[nH]2)=O)C)ccc(Cn2ccnc2)[nH]1 Cc1cccc(C)c1CNC(=O)C(N1CCOC(C)(C(F)F)C1)CCOC(C)C N1(C(C(C(CC)O)C)=O)CCC=C(C(=O)NCC2CC(F)(F)C2)C1 CCCCC(O)C(=O)N1CC(CNC(=O)C(C)C(O)Cc2ccccc2)C1 C1(C(=O)Nc2cn(C)nc2)CCC(NC(=O)CCN2CCOC2=O)CC1 c1(CNC(C2C(NC(C3COCC(C)O3)=O)CC2)=O)cccc2ccnn12 c1(C(N2CC(CC(C)NC(C3(C)CCCCO3)=O)C2)=O)ccc(O)c(Cl)n1 Cc1cc(-c2cnc(CNC(c3ccc(C(F)(F)F)nc3C)=O)nc2)cc(C)c1 N1(C(CC(CCC)C)=O)CC2CCC(C1)N2C(C1(Cc2cccs2)CCCC1)=O c1(OC)ccc(S(=O)(=O)N2CCN(Cc3nc4ccccn4c3C)C3CC23)cn1 c1(N2CC(CC=C)(NC(c3cncc(C)c3)=O)C2)ncnc2c1ccn2C1CC1 N#Cc1cc(CNCC2(Nc3ccnc(C4CC4)n3)COC2)ccc1Br Cc1cc(CC(N2CC(CO)(NC(=O)COc3ccsc3)C2)=O)no1 c1(CCNC(C2C(C)C2)=O)ccc(NCc2ncc(Br)cn2)cc1 Cc1onc(C(=O)NC(C)C(C)NC(c2ncc(F)cn2)=O)c1[N+](=O)[O-] N1(C(CCC)=O)CC(NC(=O)CC(C)(C)CC)CC2(CC2)C1 c1(C(=O)NCC2C(CNC(CN(C)C(=O)C3CC3)=O)C2)csc(C#N)c1 c1(C(=O)NC(CC(=O)NCCOC(CC)(C)C)C2CC2)cc(C)cc(F)c1 CC1=NNC(=O)C1CC(=O)NCC1(F)CCC(CNC(c2ccc(F)cn2)=O)C1 c1(NC(C)=O)ccc(F)c(C(=O)NC(C)C(C)NC(C23CC(C2)C(C)O3)=O)c1 C1(C(N(C)CCOCC(=O)NCCc2nnc(O)o2)=O)COC(=O)N1C c1(CSC)cc(C(=O)N(CCCNC(C2CC2(C)Br)=O)CCO)sc1C C(=O)(C1=COCCC1)N(C1CN(C(C2(n3nccn3)CC2)=O)CC1F)C C(C(CC(C)(C)C)NCc1nccn1CCc1ccccc1)OC CCC(C)C(C(=O)NCC1C2CN(C(=O)C3=NOC(C)C3)CC12)N(C)C C(C(=O)N(C)CC1CCCN(C(=O)CSCCC(F)(F)F)C1)(C(C)C)OCC C1(N2CCCC2)(CC)CCN(C(C2CC(=O)N(C(C)C)C2)=O)CC1 N#Cc1cccc(F)c1C(=O)NCC1COC(CN=c2[nH]cncc2Cl)C1 N1(C(=O)OC(C)(C)C)CCC(NC(CCc2cn(C(C)(C)C)nn2)=O)CC1 c1(CNC2CCN(C(c3ccn(C)n3)=O)CC2F)cc(F)c(C#N)c(F)c1 c1(C(C(N2CC(NC(c3n(CC)ncc3)=O)C(C)C2)=O)(C)C)cccc(Cl)c1F CCC(C)C(C(=O)NCc1ccc(C)o1)N(C(=O)COc1ccsn1)C C(=O)(C1=C2CCCN=C2NN1)N1C2C(NC(c3ccc(CF)cc3)=O)C(C2)C1 CC(N=[N+]=[N-])C(=O)N(CC(C)NC(C1(c2cc[nH]n2)CC1)=O)C Cc1nc(N2CC3CCC2CN3C(C2CCS2(=O)=O)=O)ccc1C#N c1(C(N2CCC(NC(c3cccc(C)c3Cl)=O)C2)=O)ccc2c(c1)COCC2 c1(C(N2CCCN(C(C(C)C)=O)CC2C(C)C)=O)cc2cc(F)cc(F)c2o1 N1(C(CC=CC)=O)CC(CC(=O)N(CC)Cc2ccccc2)CC1C c1(C(N(CC(C)NC(c2ccccc2)=O)C)=O)cncc2cnccc12 N1(C(c2ncc(C)o2)C(=O)NC(C)C)CCC(C2CCCC2(C)C)C1 C1(C)(C(=O)NCCOCCOCCNC(c2c(C)n[nH]c2)=O)CC(C)OC(C)C1 N1(C(C(CC2CC2)OC)=O)CCC2(CC1)CN(C(=O)CC(O)c1ccccc1)C2 N1(C(C(C=CC)O)=O)CCN(C(=O)CCCc2nc3ccccc3o2)CC(O)C1 C1(COC)(NC(c2cnc(O)o2)=O)CCCN(C(c2cccc(OC)n2)=O)C1 C1(F)(C(=O)NC2CCC(NC(C(c3cccc(OC)c3)C)=O)C2)CCS(=O)(=O)C1 O=C1C(Cc2cccc(Cl)c2O)CCCN1CC(N1CCCCCC1c1ccco1)=O C12(NC(c3cscc3C(F)F)=O)CCCC1CN(C(=O)C1=C(Cl)CCC1)C2 Cc1cc(C)c(C(=O)NC2CCC2CNC(c2ccn3nccc3n2)=O)c(O)n1 N1(C(C2(OC)CCC2)=O)CCC(C)C(CC(=O)NC2CC2c2cc(C)on2)C1 O=C(C1=CCN(C(C2(C3(O)CCC3)CC2)=O)C1)NC1CCOCC1 C1(C(=O)NC(c2ccnc(F)c2)C)(NC(C2C(C)(C(C)C)C2)=O)CCOCC1 C(CCC(C)Cc1nc(-c2cccc(Br)n2)nn1C(C)C)=C(C)C [N-]=[N+]=NC1CC(C(=O)NC2CC(CNC(c3ccnn3CC(F)(F)F)=O)C2)C1 C(=O)(CCS(N)(=O)=O)OC(C1(C2CN(CCON)C2)CC1)C CCC(C)(C)CCCC(=O)NC(C)C(C)C(=O)NC1CNC1 C1(NC(c2ccncc2O)=O)CC2(C1)CC(NCc1ccc(F)cc1O)C2 N1(C(c2occ(C(=O)OC)c2)=O)CCCC(C(=O)NCC2(CO)CCCC2)C1 C(=O)(C#CC1CCOCC1)N1CCCN(C(C(CC)OC2CCCC2)=O)CC1 c1(NC)ccc([N+](=O)[O-])cc1C(N1CCC(C)C(NC(=O)CCCCOC)C1)=O c1(OC)ccc(-c2nc(C3CCC(F)CC3)n(C3CCCSC3)n2)nc1 C1(C(N2C(CC(=O)NC3CC=C(C)CC3)CCC2)=O)CCCCCN1C C1(C(=O)NC2CCC(NC(=O)CC3CCC(=O)N3C)C2)(OC)CCCCCC1 N1(C(CC(CC)(F)F)=O)CC2(CCN(C(c3cc(Br)n[nH]3)=O)CC2)CC1C c1(OC)ncc(NC(C2(C)CCN2C(c2[nH]cnc2C)=O)=O)cc1F C1(NC(N(C)Cc2ccc(C3CC3)cc2)=O)C2CC3CC(C2)CC1(CO)C3 C1(C(=O)OC)(CC)CCCCN1C(c1ccc(NC)cc1)=O N1(C(C(CO)NC(N)=O)=O)CC2(C1)CN(C(=O)CC=Cc1ccccc1F)C2 C#Cc1ccc(C(=O)NCC=CCNC(c2sc(CC3CC3)nc2C)=O)cc1F c1(C(=O)OCCOc2ccc(F)cc2F)ccc(Cl)c(C(F)F)c1 S(=O)(=O)(c1c(C)nn(C)c1C)N1CC(NC(c2c(C)c[nH]c2)=O)C(C#N)C1 C=CC(CCC)CC(=O)NC(CCC1CCC1)C(=O)NC1CC(=O)N(C)C1 N12CCCCC1CNC(=O)C2.C1(C(N)=O)CC(CNn2ccnn2)C1 N1(C(c2cc(Br)ncc2Br)=O)CCCC2C1CCN2Cc1ccc(F)c(F)c1F c1(NC(C2(CC)CCOC2)=O)ccc(NC(=O)C(C)C(C)(C)C)cc1C S(=O)(=O)(c1cccc2cccnc12)N1CCN(C(C=CC(C)C)=O)C2(C1)CC2 C(=O)(CC(C(F)(F)F)n1cccn1)N(C1CCCN(C(c2c[nH]c(=N)s2)=O)C1)C N1(C(C(CC)OC2CCCC2)=O)CCC(C)(C(=O)N(C2CC3(CCC3)C2)C)C1 c1(C(=O)NC2C(NC(c3cnnc(O)c3)=O)COC2)n[nH]c2c1COCC2 c1(C(=O)NCC2(C(C)NC(=O)Cc3ccc(F)cc3)CC2)[nH]nc([N+](=O)[O-])c1Cl N(C)(C1CN(C(=O)C=CSC)CCc2ccccc21)C(CCOCCCOC)=O N1(C(c2c(C)c[nH]n2)=O)CCN(C(=O)Cc2ccccc2[N+](=O)[O-])CC(C)(C)C1 C1(NC(C2CCC(CNC(c3cc(C#N)[nH]c3)=O)CC2)=O)CCc2nn[nH]c2C1 N1(C(Cc2c(C)nsc2)=O)C2CC1CN(C(c1sccc1CC#N)=O)C2 C12(C(N3CC(N(C)C)C4(C3)CC4)=O)CCC(CC1)N(C(c1cnc(S)nc1)=O)C2 C=C1CCN(C(=O)C(C)C(F)(F)F)C(C(N2CC(c3nncs3)C2)=O)C1 O=[N+]([O-])c1cnc2c(F)cccc2c1SC1CNC2(CCOCC2)C1 c1(C(N2C(Cn3cc(CC=C)nn3)C=CC2)=O)ccc(C(C)C)c(C(F)(F)F)c1 N#Cc1cc(F)c(C(=O)NCCCNC(C2CCc3nncn3CC2)=O)c(F)c1 C(CC(=O)NCC1CCN1C(c1cccc(N)c1)=O)(C(F)(F)F)NC(C)=O CCS(=O)(=O)NNC(=O)c1c(F)cncc1Br C(CN=c1[nH]c(N2CCN3CCCCC3C2)nc2c1COCC2)N(CCC)CC CC1CN(C(c2cscc2C2CC2)=O)CC(C)N(C(=O)CN2CCC(O)CC2)C1 C=CCC(C)(CC)C(=O)N(C1CCCC1)C(c1nnn(C2CCCCC2)c1C)=O C1(C(=O)NCC2(C)CCC(=O)N2)CCN(C(=O)COCC(F)F)O1 c1(C(=O)NC(C(C(C)C)NC(=O)C2=CCCCO2)C)ccc2nsnc2c1 C1(CN(C)C(C2CC2Cl)=O)CCN(C(C2CCCN(c3cnccn3)C2)=O)CC1 C(C(O)C(=O)NC(C)(C)C(=O)N(C)Cc1ncn(C)n1)N(C)C C(C(C)(C)C(C)(C)C)NC(CC1(OC)CN(C(=O)CSCC(F)F)C1)=O O=S(=O)(c1ccc(O)nc1)N1Cc2cnc(C3CC3)nc2C1 C1(C(=O)NC2CC3C(NC(c4c(C)ccc(Cl)c4)=O)C3C2)CC(C)(C)OC1(C)C C(=O)(CCCCCC(C)C)NCC1N(C(c2c(C)scc2)=O)CCCC1C CCCCC(C(=O)N1CC(C2(NC(=O)C(O)CC(C)C)CC2)C1)C(C)C C=CCCC(C)(C)C(=O)N1CCCC(C)(NC(c2cnn(CC=C)c2)=O)C1 CN1CC=CCC1CC(N1CC(O)(CCNC(C2(C)CNC(=O)N2)=O)C1)=O c1(OC)ccc2c(N3CCC4CCC(C3)S4(=O)=O)nc(=NCC(Cl)(Cl)Cl)[nH]c2c1 N1(C(C2(NC(CC3(C)CCOC3)=O)CC(O)C2)=O)CC2CCC(C1)O2 CC1CC2CN(C(C3(NC(=O)CCC4CC(C)C4)CC(CO)C3)=O)CCN2C1 C1(C(=O)Nc2cn(CC)nn2)CC(O)CN1C(c1ccc(SC)cc1)=O c1(NC(C(CCC)N(C(=O)C(=O)C(C)(C)CC)C)=O)ccc2ncccc2c1 C1(C)(C(=O)NCC(CC2CC2)OC)CC(O)CN1C(c1ccc(F)cc1F)=O N1(C(C(C)NC=O)=O)CCC2(CC1)CC(C(=O)Nc1ncc(C#N)cn1)CO2 N1(C(CC2N(C)CC=CC2)=O)CCCC(C)(C)C1CNC(C1CCC1)=O CC1=C(C(=O)NCC(C2CCC2)NC(C2C3CCC4C(C3)CC24)=O)CCCO1 C1(CN(C(C2(C)CC2(C)C)=O)CC)CCCN(C(=O)CC2CN(C)C2)C1 C(=O)(CC(C)(O)COC)NCC(CC)NC(c1sccc1C(C)=O)=O N1(C(C=CCC)=O)CCC(O)(C(C)NC(C2CCC(=O)N(C)C2)=O)CC1 C1(CC(=O)NC2(CN(C(=O)CSC(F)(F)F)C)CC2)CCOC1=O CCCCC(CC)CC(=O)NC(CC)CCC(=O)NCc1nnc(O)o1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CC2(C1)SCCC2NC(=O)CC1C=CCC1 N1(Cc2n(CC=C)c(Cc3cnn(C)c3C#N)nn2)CCc2ccc(Br)cc2C1 c1(CC)cccc(CC)c1CC(=O)N(CC(C)N(C)C(c1ccncc1F)=O)C c1(OCCNC(CCC)(c2nnnn2C2CCOC2)C2CC2)ccc(C)c(F)c1 c1(C(=O)NC(CC=C)CNC(=O)C(C)NS(=O)(=O)CC)ncc(CC)cn1 N1(C(CN(CCOC)C)=O)CCC(NC(c2cccc(SC)n2)=O)C2(CCC2)C1 C1(C(=O)NC(C#C)(C)CC)CC2CC2N1C(=O)C(N1CCCCC1)C N1(C(C2(CC)CCNC2=O)=O)CCC2CN(C(=O)C=CBr)CC2C1 c1(C(N2CC=CC23CCCC3)=O)coc2c(Cl)cc(Cl)cc12 N1(C(COCC)=O)CCN(C)C(CNC(=O)CCc2nncn2C)C1 C(C(C)(C)CN(C(=O)C(F)(Cl)c1ccccc1)C)NC(C(c1ccn(C)n1)C)=O c1(C(=O)NC2(C)CCN(C(c3c(Br)cc(C)s3)=O)C2)cccn2nncc12 c1(CC(=O)NCC(C)CN(C)C(C2CCCCC2O)=O)ccc2c(c1)CCO2 Cc1ccc(OC(F)F)cc1C(=O)NCC(C(C)C)NC(=O)CNC=O N1(C(c2n(C(C)C)cnc2)=O)CC=C(C(=O)NCC2(F)CC(CO)C2)CC1 N1(C(CC(CNC(COC2(C#C)COC2)=O)O)=O)C2CCCC1CC2 N1(C(C2C(CC)OCCC2)=O)CCCN(C(=O)C(C)(C)CN2CCOCC2)CC1 C1(N(C(C(C2CCOCC2)C)=O)C)CCN(C(c2coc(Br)c2)=O)CC1 C1(C)(C(=O)NC23CC(NC(CCCOCC)=O)(C2)C3)CCN(C)C1=O c1(C(=O)NCC)ccc(C(=O)NC(C)C(c2ccc(Br)cc2)OC)cc1 N1(C(c2c(CC)ccs2)=O)C2CCC1C(C)C(NC(=O)CC1CCC(C)CC1)C2 Cc1[nH]nc(C(=O)N(CC(=O)NC2C(=O)OCC2CO)C)c1C CC1CCn2ncc(C(=O)OCC(c3c(Cl)nc4ccccn34)=O)c2C1 N1(C(Cc2cnc(C)o2)=O)CCCC(C2CC2NC(C2(C)CCC2)=O)C1 C1(CO)COCCN(Cc2ccccc2)C1.C12(CCC1)C(=O)NOOCCC2 c1(C(C)C)cccc(C(=O)NC(C)Cn2cc(COC3CCOC3)nn2)c1F Cc1cnc(F)c(CNC(C2CC23CC(NC(c2c[nH]c(C)c2)=O)C3)=O)c1 c1(C(C2CC=CCC2)NC(CC2(C(N)=O)CCOC2)=O)ccccc1 c1(C(=O)NCCCCCCNC(C2C(C=C)(C(F)(F)F)C2)=O)c(C)nc(C)n1O CC1(C)CCC(CNC(=O)CS(=O)(=O)CCO)N(C(C2CCC(C(N)=O)O2)=O)C1 c1(-n2c(CC(C)C(C)C)nc(CC)n2)ccc(Cl)c(C)c1 C1(C(=O)NCC(F)CO)COCCN(C(c2ccccc2O)=O)C1 C=CCC(CC=C)C(=O)NCC=CCC(=O)NCC1CC1(Cl)Cl c1(CNC(c2ccc(OC)cn2)c2n(CC=C)nnn2)cccc(C(N)=O)c1 C(=O)(C1=CCC(F)(F)CC1)N1C2C(CNC(c3c(C)nc(C)[nH]3)=O)CC(CC2)C1 c1(C(N2C3CCN(C(CCC(N)=O)=O)C(C3)C2)=O)nncc2c1CCCC2 c1(OC)ccc(NC(C2CCN(C(=O)Cn3nc(C)cc3C)C2)=O)c(C)n1 C1(NC(COCCC#C)=O)CC(O)CN(C(=O)CCc2nnc(S)n2C)C1 CCC(C)(C)C(=O)C(=O)NOCC(=O)NCc1ccccc1F C(C(=O)NC1CCCCC1C(=O)NCc1nc(C)oc1C)(C(C)C)OCC n1(CC(N2CCC(CN(C(CC3CC(C)C3)=O)C)C2)=O)cc([N+](=O)[O-])ccc1=O N1(C(C2CC(C#C)(O)C2)=O)CC(NC(=O)C(F)n2cccn2)CC2(CC2)C1 C(=O)(CC(C)COC)NC(CC)CNC(c1cnc(C(C)=O)s1)=O Cc1cc2c(cc(C(=O)NC3C(O)CC3O)n2CC(F)(F)F)s1 Cc1cc(C)c(C(=O)NCC(F)CNC(c2[nH]c(=N)ccc2C)=O)c(C)n1 C1(CC)CN(C(c2cn(CNC(C3OCCC3C(C)C)=O)cn2)=O)C(C)CO1 CC(C(=O)NCC1CC(F)CN1C(c1cc(Cl)cnc1O)=O)C(F)(F)F Cc1nc2ccc(NC(=O)C3=CCCN(C(=O)C(C)O)C3)cc2o1 C1(C(=O)NCC2N(C(C(C3CCOCC3)=O)=O)CCC2)CCCC2CCCCC12 c1(C(=O)NC(CN(C(c2cn[nH]c2)=O)CC)C)ccc(OC2CCC2)cc1 C1(CNC(C2CC(=C)C2)=O)CC2CCCCC2N1C(=O)COCCCOC O=C(C1=CCCOCC1)NCCCNC(=O)CC1CCCC(O)C1 C(=O)(C(F)C(F)(F)F)N1CCC(CCN(C(=O)CSC2CCCC2)C)CC1 c1(OC)ccc(-c2cnc(NCC3CCCCC3C(C)(C)C)o2)cc1 c1(C(=O)NC2CN(C(C3(CC)CCCC3O)=O)C2)cc(F)cc2nn[nH]c12 c1(C(=O)NC(CNC(COCCC#C)=O)(C)C2CCC2)nn(C)nc1Br C1(CC)CN(C(=O)Cc2cncn2C)CCC1NC(=O)CC1CCCCC1(F)F c1(C(=O)NC2CC(C)N(C(c3cc(Cl)ccc3N)=O)C2)nc2ncccn2n1 C1(C)(CNC(C2(OC)CCCOC2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)CC1 Cc1cc(C(N2CCCC(c3nc(C)cs3)C2)C(=O)NC(C)C)cc(F)c1 CC1CN(CCCCNC(=O)C(=O)NCc2ccc(F)cc2F)CC(C)O1 C1(NC(c2ccccc2O)=O)CC(O)CN(C(=O)C=C2CCCC2)C1 c1(N2CC(F)CC(C(=O)NCc3cccs3)C2)ncc(Br)c(N2CCCC2)n1 c1(C(=O)NCC2CC(NC(C(CC)NC(C)=O)=O)C2)cncc(OC(C)C)c1 C=CC(C)(O)C(=O)NC1CC(NC(=O)C=CC=CCC)C1 C(CC(C)(C)CC(=O)N1CCC2C(NC(=O)CNC(C3CCCC3)=O)C12)OC CCCC(CNC(C12CCC(c3nn[nH]n3)(CC1)C2)=O)CCO C1(C(=O)NC2CCC(CNC(c3[nH]nnc3C3CC3)=O)C2)C2CCC(F)(F)C12 C(=O)(CCCCCCNC(c1cc(C)[nH]n1)=O)N1C(CSC)CCC1 C1(C(=O)NCC2CCCC2NC(c2nocc2C)=O)(COC)CC1(F)F CC1CN(Cc2ccccc2)CC1C(N1CCC1NCCCc1ccco1)=O Cc1ccc(F)c(C(N2CSCC2C(=O)NCCCOCC(F)F)=O)c1 N1(C(CS(CC)=O)=O)CC(NC(c2conc2C2(C)COC2)=O)CC1(C)C c1(C(N2CC(C3(NC(C4(C(N)=O)CC4)=O)CC3)C2)=O)ccc2c(c1)C(=O)CCC2 C(=O)(C(C)(F)CC1CCCC1)NCC(C)NC(c1cc(CCOC)on1)=O N1(C(C2OCCC(C)C2)=O)CCCC(C2CN(C(C3(F)CCN(C)CC3)=O)C2)C1 N1(C(C(CC)n2ccnc2)=O)CCC(CN(C(=O)CC2(N(C)C)COC2)C)CC1 N1(C(c2occ(C)c2)=O)CC2(CCC2)CCC1CNC(=O)Cc1ccc(Cl)cn1 C#Cc1ccc(C(=O)NC(C)(CO)C(=O)NC(C=C)C(F)(F)F)cn1 N1(C(c2ccc(OC)nc2)=O)CC2(CC2)CC1CNC(C1CNC(=O)C1)=O C(=O)(C(CC(F)F)NC(C1CCCC(CF)C1)=O)NCC1(COC)CC1 N1(C(C2CCN(C(c3cc(CC)ncc3)=O)CC2C)=O)CCCC2(CC1)CC2 N1(C(C2C(c3ccc(C)cc3)C2)=O)CC2(CC(OCCC(=O)CC(C)(C)O)C2)C1 c1(C(=O)NCC2CC(CNC(C=C(C)Cl)=O)OC2)ccc2ccncc2c1 N1(C(C(C2CC2)NC(=O)OC(C)(C)C)=O)CCOCC12CCS(=O)(=O)C2 C1(C(N2CCC(CCNC(C3N(S(C)(=O)=O)CCC3)=O)C2)=O)CSCC(=O)N1 N1(C(CC(=O)OC)=O)CCC2(CC1)CC2NC(C1CC=C(C)CC1)=O c1(C(=O)NC2CC(C(C)C)OC2)cc(Cl)c(Br)cn1 c1(NC(=O)NC(C)C)cccc(F)c1NC(=O)CC(C)C(=O)c1ccc(Cl)cc1 N1(C(C2COCCC2(F)F)=O)CC2CCC(C1)N2C(c1nncn1C1CC1)=O C=CCCC(C(=O)N1CCCC(C)(O)C1)NC(c1c[nH]nc1C)=O C1(C(=O)NC2CC3CN(C(CC(=O)N(C)C)=O)C2C3)CC2(CO)CCCC12 Cn1cccc1C(=O)NCC(C1CCCC1)NC(c1ncoc1C(C)(C)C)=O c1(SCC(=O)NC(c2ccccc2)CC#C)ncccc1C c1(C(=O)NCc2c(C(=O)NC(C)C#N)cco2)cc2cccn2cn1 c1(C(N(C2CCN(C(=O)CNC(=O)C3CC3)C2)CCC)=O)cn(C(C)C)cn1 Cc1ccc(C(N2CCCC(C)(NC(c3cc(Cl)n(C)n3)=O)C2)=O)c(C)n1 c1(CN2CC(CC(N3CC(C)CC(COC)C3)=O)C2)cccc(Cl)c1[N+](=O)[O-] CC1CN(C(=O)C(n2ccc(Br)n2)C)CC1CNC(c1cnccn1)=O N#CC(C(=O)NCC1CCCN1C(c1cnc(Cl)s1)=O)C1CC1 n1(CC)ncc(C(=O)NCC2C3CN(C(c4ccnc(C)c4)=O)CC23)c1C1CC1 n1(CC(=O)CC)cnnc1O.C(=O)(CCc1ncc[nH]1)N1CC(=O)NCC1.C(C)N CCCC(CC)C(=O)NC(CNC(c1cc(C)n(CCO)n1)=O)CC(C)C C1(CCCNC(=O)Cn2nnc(=O)[nH]2)CCCCN1C(=O)Cn1cnnc1 CCCCCCC(CC)C(=O)N1CC(COC)(NC(=O)C(CC)C(F)(F)F)C1 c1(CC)nc(C(=O)N(C)CC2CCN(C(c3cnc(O)n3CC)=O)CC2)c(C)o1 c1(OC)ccc(C)cc1C(N1CCC(C)(C)C1CNC(=O)CC12CCCC1C2)=O C1(CN(C(C2C3CCC(=O)C23)=O)CC)CCCN(C(=O)CNS(=O)(=O)N(C)C)C1 c1(C(=O)NC2C(NC(c3c(C)n(C)nc3)=O)CCC2)cc(Cl)cc(F)c1F N1(C(C=Cc2ccc(CC)o2)=O)CCN(C(C2CCCC(CF)C2)=O)CC1CC C=CC1(C(=O)NCc2c(C)n[nH]c2C)CCN(C(C2CCCOC2)=O)C1 C(=O)(CC(O)CNC(=O)CCc1cc(C)no1)NC1(C(N(OC)C)=O)CC1 c1(CNC(NCCC(=C)Br)=NC)cc(C(C)(C)C)no1 C#CCCC(O)C(=O)N1CC(OC)CC1CCNC(=O)CC1COC(=O)C1 C1(O)(C(N(C2CS(=O)(=O)C2(C)C)C)=O)CC2(CCCN(C(=O)OC(C)(C)C)C2)C1 C(=O)(C(CCF)NC(c1c[nH]nc1Cl)=O)NCC1C(C)(C)C1 C(CN=c1[nH]c(=NCC2CCCCC2O)c2cc(Cl)ccc2[nH]1)NC(=O)NC N#CC1(C(=O)NCCCCCC(=O)N2CCN(C3CC3)CC2)CCCOC1 C1(O)(C(=O)NCC2CCCO2)CC(F)(F)C1 c1(SC)cccc(C(N2CC(CNC(c3cn(C4COC4)nn3)=O)CC2C)=O)c1 C#CCCCC(C(=O)NC(C)(C)C)N1CCCC(CCF)C1 N1(C(C(CC=C)NC(C)=O)=O)CC2CCN(C(=O)Cn3cnc(=N)[nH]3)CC(C2)C1 N1(C(CC2CC(SC)C2)=O)CCCC(NC(c2cc(O)ccc2F)=O)C1C c1(CCC(C)C(=O)NCCC2CN(C(=O)CO)CCO2)ccc2ccccc2c1 C(=O)(C(C)(C)COC(C)(C)C)N(CCN(C(=O)CCC1CCN(C)C1)C)C C12(NC(c3ccc(O)nc3Cl)=O)CCCC1N(C(=O)C(O)(C1CC1)C1CC1)CC2 C1(C(C)C)CCCN(C(c2sccc2Br)C(=O)NCc2csc(Br)c2)C1 C1(NC(c2n(CCSC)nnn2)c2cncs2)CS(=O)(=O)N(C)C1(C)C c1(C(N2CCC(C)(CC(N3CC4(CN(CC)C4)C3)=O)C2)=O)ccc(C#N)cc1C N1(C(C2(CC)CC2(F)F)=O)CCC2(CCCC2NC(=O)CC2CC=CC2)CC1 C1(C(CNC(C(C2CCC(=O)N2)C)=O)O)CCN(C(=O)Cc2ccccc2)CC1 C1(CC(=O)NC2CC2)CCCN(C(C2CCCCCCC2)=O)CC1 c1(SCC(=O)NCC2CC(CNC(C3CCS3(=O)=O)=O)C2)nc2ccccc2s1 C#CCC(O)C(=O)NCC1CCN1C(c1ccc(C(F)(F)F)[nH]1)=O C1(Cl)(C(=O)NC2(C(=O)OC)CC2)CC1C(C)=O.C1(=O)CC2(CC2)N1C c1(C(N2CCC(NC(C(C3CC3)OC)=O)C2)=O)ccc(C)c(F)n1 c1(C(C)NC(=O)Nc2ccc(C(N3CC4C(CO)C4C3)=O)nc2)ccccc1Br c1(CC)ccccc1C(=O)NC(C1CCCN1C(=O)CCC(=O)OC)C C12(CN(C)C(c3cnn(C)n3)=O)CC(CO1)N(c1nnc(-c3ccccc3)s1)C2 c1(NC(C(C)N(C(C2CCCC(OC)C2)=O)C)=O)cc(C)ccc1F c1(OC)ccc(C(N2CC(OC)C(NC(c3c(C)cnn3C)=O)C2)=O)c(Cl)c1 C(=O)(CC(C)C(=O)NC(C(N1CC(C)(C(N)=O)C1)=O)C1CC1)OC CC(C)(C)C(C)(C)C(=O)NCCN1CCN(C(=O)C#CC2CCCC2)CC1 C12(NC(C(C)(C)F)=O)CCCC1N(C(c1cnc3ccccc3n1)=O)CCC2 CC1OCCC1(F)C(N1CCC(CCN(c2ncccn2)C)CC1)=O c1(C(=O)NCC2CCCC(OCC)C2)c(O)ccc(F)c1Br N1(C(CC=C=C)=O)CC2CC2(NC(c2cnc(S)nc2)=O)C1 Cc1cccc(CC(N2CCC(N(C)C(C3(C)CCN(C)C3)=O)C2)=O)c1C C1(C(N(CCCN(C(CC(=O)NCC)=O)C)C)=O)CCCC(C(=O)OC)C1 C=CCC(C)(C)C(=O)N1CCC(NC(=O)Cn2ncn(C)c2=O)C(C(N)=O)C1 c1(OC)c(NC(=O)C(N2CCC(OC)CC2C)=O)cc(Cl)cc1C C(=O)(C(F)(F)Cc1ccc(F)cc1)NC1CC(CNC(C=CC=CCC)=O)C1 n1(CC)ccnc1C=CC(=O)NC1CC(CO)N(C(=O)CCC(=O)N(C)C)C1 Cc1nc(C2(NC(C3(NC(=O)C(C)N4CCCC4)CCC3)=O)CC2)no1 CC#CCC(C(=O)NCC=CC)NC(C1CC=CCO1)=O C1(NC(CN(C2CCC2)C)=O)CC2CCC(C1)N2C(C1CCCC1(C)C)=O C1(C(=O)NCC(=O)N(C2CC(C(N)=O)C2)C)(COC)CCC1 C1(N(C(CCCOC)=O)C)CCCN(C(=O)C(C(C)O)N(C)C)C1 c1(C(=O)NCC2CC3CC(NC(C(CC)(C)O)=O)C3C2)c(C)cc(OC)cc1C C=CC1CCCN(C(c2nnc(C)s2)C(=O)NCC(C)C)C1 C1(C(N(C2C3CN(C(c4nnsc4N)=O)CC23)C)=O)CC2CCC2C1 c1(CC(C)C)cc(-c2nc(-c3cncnc3)nn2CC2CCSC2)n(C)n1 O=C(C#CC1CCCOC1)NCC1COCC1NC(=O)CC(C1CC1)C1CC1 c1(C(N(CCNC(=O)C(F)C2CCOC2)CC)=O)cnn2c1N(C)CC2 c1(C(N2CCC(N(C(CCCC(C)=O)=O)C)C2)=O)ccccc1S(C)(=O)=O O=C(C1=CCCCO1)NCC1(O)CCN(C(=O)CCC=Cc2ccccc2)C1 CCC(C)(C)C(=O)N1CC(CNC(c2cncnc2-c2ccccc2)=O)C(O)C1 CC(C)C(C(=O)N1CCCC(CN(C(=O)C(F)(F)C2CC2)C)C1)c1cccnc1 c1(CC)ccc(O)c(NC(=O)CC(CC)NC(c2cc(C(N)=O)[nH]n2)=O)c1 C1(CC(=O)NCC(=O)N(C2CN(C)C2)C)CCCN1C(C1CC1F)=O CCC(O)C(F)(F)C(=O)NCC1CN(C(=O)CC2CCC3CC23)C1 C1(C(=O)NC2CCC(NC(c3ocnc3C3CCC3)=O)CC2)CC2COCC2C1 CCCC(C)(C)C(=O)N1CCCC(C(C)NC(c2nc(C)[nH]c2C(F)(F)F)=O)C1 c1(CCC(=O)NCC2CC(F)(CNC(C=C(CC)CC)=O)C2)ccc(Cl)c(F)c1 C(CCCCCC(=O)N(C1CCCC1)CC)NC(c1c(CC)ncs1)=O C(=O)(C#CC1CC(F)(F)C1)N1CCC(C)CC1CNC(c1ccc(C(N)=O)cc1)=O n1(CC(N2CC(N(C(=O)C3=CCOCC3)C)C(F)C2)=O)ncn2nccc2c1=O C(c1cccc(F)c1Cl)=CC(=O)NC1C(NC(C=CC(CC)=CC)=O)CCOC1 CC1(NC(C23CC(F)(C2)C3)=O)CCN(C(C2CC2C(C)(F)F)=O)CC1 n1(C(CC)C)nc(C(=O)NCC(CNC(=O)Cc2ccsc2)CO)cc1C C(C)(CNC(=O)CCCN1C(=O)CCC1=O)(C(C)C)NC(CNC(CCC)=O)=O C1(CSC)CC(NC(=O)C(=O)NC(C)Cn2cncn2)C12CCC2 c1(CC)ccccc1Cl.C12CCN(CC1)C(c1ccc(C(F)(F)F)cc1)C(=O)N2 c1(C(=O)NCC(C)(C)CNC(c2cncnc2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 c1(CC(=O)NC2(CN(C)C(C3CN4CCN3CC4)=O)CC2)c(F)cccc1C#N n1(CCC)cc(Cl)c(C(=O)NC2CCN(C(=O)CC3OCCC3C)C2)n1 Cc1cc(=O)n(C)nc1C(=O)NCCNC(c1cccc(Br)c1F)=O c1(N(CC(C2CC2)OC)C)nc(NC2CCOC2)c2cnn(C)c2n1 C(=O)(CCC(C)(C)C)N(CCC(=O)NC(c1cncc(F)c1)C)CC C1(NC(C(CC)OCC)=O)CC2CC(NC(c3cccnn3)=O)CC12 C=C1CCN(C(c2cnn(CCNC(c3ncoc3C)=O)c2)=O)C1 C(=O)(N1OC2CCC1C2)C1(NC(Cc2c(C)ccnc2)=O)CCC1 Cc1ncc(C(N2CCOC(CNC(C3C4CNC(=O)C34)=O)C2)=O)c(=N)[nH]1 c1(CC)ncccc1C(N1CCC(NC(C2(N(C)C)CC2)=O)C1C)=O N1(C(c2c(C)cc(CC)o2)=O)CCCC(C)(C(=O)NCC2(C(C)(C)OC)CC2)C1 c1(C(=O)NC2C(C)(C)CN(C(=O)CCCC3CCC3)C2)nc2ccc(Cl)nn2n1 c1(CC)cc(NC(=O)C(C2(O)CN(C(=O)CCCCCN(C)C)C2)F)cc(O)c1 c1(N2CC(CNC(C3C(CC)OCC3)=O)(OC)C2)nccc(S(C)(=O)=O)n1 C1(C)(CCNC(CC2CC(CC)OCC2)=O)CCN(C(C)=O)CC1 c1(C(N2CCN(C(C=CCC)=O)C(CC)C2)=O)ccc2n[nH]c(CCC)c2c1 c1(COC(N(C(C(=O)NCCNC(CC=CC=C)=O)C)C)=O)ccccc1 C1(N(C(C(C2CC2)OCC)=O)C)CCCN(C(c2ccc(NC)cc2F)=O)CC1 C1(C(N2CCC(C)C2CNC(c2cccc(CCO)c2)=O)=O)CC2(C1)OCCO2 c1(C(=O)NCC2C(NC(Cc3ccc(C)cc3Br)=O)C2)cc2ncccc2o1 C1(CNC(C(C)(C)OCC)=O)C(C)CCN1C(=O)CCC1OCCO1 C(=O)(C(CNC(C1OCCC1(C)C)=O)C(C)(C)C)N1CC(CC(C#C)C)C1 C1(NC(COc2cn(C)nc2)=O)CN(C(=O)C(=O)NCC2CC2)C2(CCC2)C1 CC1CC(NC(C2CC(O)C2)=O)CCN1C(c1cccc(C(F)F)c1Cl)=O c1(C(N2CCCC2C(c2ccccc2)O)=O)ncc(C2OCCO2)s1 C(=O)(CCCCC(C)C)NC(CC=C)CC(=O)NCCc1cnco1 C1(C(N2C(C)(CNC(c3ncc(C(F)F)s3)=O)CCC2)=O)Cc2cccnc2C1 C=CCCC(=O)NC(C1CC=CCC1)C(=O)NC(c1nc[nH]n1)C1CC1 C1(CC(=O)NC2CC(F)(CNC(C3(CC4CC4)CC3)=O)C2)CCCCCC1 N1(C(C(C(C)C)F)=O)CCC(C2CCCN(C(c3ccc(F)o3)=O)C2)CC1 c1(C(=O)OCC)ccc(NC(=O)CCc2cc(C)ccc2C)cc1OC c1(CC(=O)NCC2C(NC(C(C)c3ccco3)=O)CC2)sc(O)nc1O C1(CC=C)(NC(C2COCCC2(F)F)=O)CCCN(C(=O)CC(C)(C)CC)C1 N#Cc1ccccc1C(=O)NCC(CC(=O)Nc1ccsc1)C1CCC1 CCC(C)CCCCC(=O)NC1CC(NC(=O)CC23CCCC2C3)C(O)C1 C1(O)(CNC(C(F)=C(C)C)=O)CC(NC(=O)C(O)c2cnc[nH]2)C1 c1(C(N2CCC(O)(C(CNC(C=CCOC)=O)C)C2)=O)cc(C)c(C(F)F)cn1 c1(C(C(N2CC(N(C(c3c(C)n[nH]c3)=O)C)C2)=O)C)cc(Br)ccc1F C1(C)(COC)CN(C(=O)C(C)(C)C2CCN(C(=O)CCOCC(C)(C)C)C2)C1 C1(C(N2CC(COC)(CNC(=O)CCN3CCCC3=O)C2)=O)CCCC(=O)C1 c1(OCCC(=O)N(C(C)CNC(C2CC3CC2C3)=O)C)ccc(S(C)(=O)=O)cc1 C(=O)(C(C)C(C)COC)N(CCCNC(CCC)=O)C(C)C.c12ccc(cc1)s2 N1(C(C2(OC)CCCC2)=O)CCC(NC(=O)Cn2nnnc2C)CC(C)(C)C1 C1(CNCC)CCCCC1CNC(c1ncc(Cn2cc(CCCO)nn2)s1)=O c1(C(C)NCc2ccc(C(=O)OC)o2)cc2ccccc2[nH]1 n1(CC)cc2ccc(C(=O)NC(C)C(C(C)C)NC(c3c[nH]cc3C)=O)cc2n1 c1(NC(c2ccccc2)COC)ncnc(NCCSc2cccc(Cl)c2)c1C c1(CC)nc(C)c(C(=O)NCC2(F)CCC(CNC(c3n[nH]cc3CC)=O)C2)s1 C(CCCC(=O)NCC1C=CCN1C(C1CCC1Cc1ccccc1)=O)SC C(=O)(C1=C(Cl)CCCC1)NCc1ccc(C(=O)NC2CCN(C(=O)C3CC3)CC2)s1 Cc1ccccc1SCC(=O)NCC1CC2CC2N1C(=O)Cc1sc(O)nc1O c1(COCC)nc(C)c(C(=O)NCC2CN(C(c3cccn3CC)=O)CC2C)s1 CCCC(CCCNC(c1sccc1C(C)C)=O)NC(=O)C(C)C(F)F N1(C(CCCN(C)CC2CCCO2)=O)CCC(NC(C2CCC=CCC2)=O)CC1 c1(NC(C(CSCC)NC(C=CC)=O)=O)cccc2c1OCO2 Cc1nnc2n1CCCC2C(=O)NC1CCN(C(=O)CCCC#N)CC1 N1(C(c2ccoc2Cl)=O)CCC2CCCN(C(=O)COCC(F)(F)F)C2C1 N1(C(CCN(C)CCO)=O)CC2C3CCC(C2C1)N(C(=O)CC(=O)NC1CC1)C3 c1(CC)ccc(NC(=O)C(C)N(C(=O)C(C)(C)n2ccnn2)C2CC2)cc1O C=CC1(C(=O)NCC[Si](C)(C)C)CCN(C(C2CCS2(=O)=O)=O)C1 N1(C(CCC=C)=O)CC(NC(=O)C(C)(O)C(C)c2ccccc2)CC2(CC2)C1 c1(CCCC(=O)N(C(CNC(CC(CC)C)=O)C2CC2)C)nc2ccccc2o1 C1(CCC=C)(C(=O)NCc2ncnn2C(C)C)CN(C(c2ccc(OC)o2)=O)C1 C#Cc1ccc(OC)c(C(N2CCC(NC(=O)CC3CC3C(F)(F)F)C2C)=O)c1 C(C(C)C)(C(O)C(=O)NCCC1CCN(C(C2CC3(CCC3O)C2)=O)C1)OC C1(C(N(C)CC2(O)CCN(C(c3cc(C)oc3)=O)CC2)=O)Cc2cccnc2C1 Cc1nc2cncc(NC(c3cnc(C(F)(F)F)s3)=O)c2nc1C C(=O)(CCC(C)(C)F)NC(CN(C)C)C(N1CCCCC1C(C)(C)C)=O c1(C(C)(C)C(N2CCC(C)(NS(=O)(=O)C(F)F)C2)=O)cccc(C#N)c1 N(C1CCCn2nncc21)CC(C1CCN(C(=O)OC(C)(C)C)CC1)C.C1CN1 C12(NC(C3CC34CCOCC4)=O)CCCC1(F)CN(C(=O)C(F)(F)C(F)F)C2 c1(C(=O)NCC(CNC(c2cn(C)nn2)=O)CO)cncc(C(C)(C)C)c1 C1(C(F)F)(OC)CC(C(=O)N(CCCCN(C)C(C2(O)CCSC2)=O)C)C1 C1(NC(c2c(CC)scn2)=O)CS(=O)(=O)CC1NC(=O)CCCn1cc(C)cn1 C1(C(N(c2nc(C)cs2)C(C)=O)=O)CC(=O)N(CC(F)(F)F)C1 C1(CNC(c2n[nH]c(C)c2C(F)(F)F)=O)CC(N=c2ccc(C#N)c[nH]2)C1 N1(C(C(=O)NC2CCC(C)O2)=O)CC2CN(C)CC2(C)C1 C(=O)(C1CCc2ccccc21)NCC(CNC(=O)COC1CCCOC1)OCC Cc1cc(C(N2CC3CC3(CNC(C34CC(C3)C4)=O)C2)=O)cc(C)c1Cl c1(C(N(CCC(=O)N(CC(C)C)C)C)=O)ccc2occc2c1 C(=O)(C1CCCc2nncn21)NCC(C1CCCC1)NC(c1occ(C)c1C)=O c1(C(=O)NC2CN(C(c3c(F)ccc(C)c3)=O)C(C)C2C)cnc2[nH]nnc2c1 C1(C(N2CC(C(N)=O)C2)=O)COCCN1C(=O)CCc1cncnc1 c1(C(N2C(C(C)C)CN(C(=O)CCC(=O)N(C)C)CC2)=O)cc(Br)cc(F)c1O C(=O)(CCCC(C)(C)C)N1C(CN(C(c2nc(O)nc(O)c2F)=O)CC)CCC1 c1(C(=O)NCCCC(C(=O)Nc2c(CC)cc(O)cc2)O)ccc2cc[nH]c2c1 C1(NCCc2ncn(CC)c2)CCNC2CC12 c1(N2CCCC(OC)(CO)C2)nc(C)cc(=NCc2c(Cl)cccc2Cl)[nH]1 C1(NC(c2c(C)cc(F)cc2)=O)C2COCC1CN(C(c1ncccc1Cl)=O)C2 CC1(C)CCN(C(=O)C(N)=O)C(C(=O)NC2(C)CCC(=O)NC2=O)C1 c1(C(C)C)nc(NC(c2cn[nH]c2)C)cc(=NCc2cncc(C(N)=O)c2)[nH]1 c1(N2CCC(C)C(NC(=O)CCC(N)=O)C2)nccc(S(C)(=O)=O)n1 N1(C(C(CC)=CC)=O)CCC(CCNC(C2(C(=O)C3CC3)CC2)=O)CC1 N1(C(CNC(c2cccs2)=O)=O)CC(CNC(C2CC3CCC2O3)=O)C(O)C1 c1(CC(=O)NC2CC(F)(CNC(=O)CCC3CCCO3)C2)ccc(O)cc1 c1(CC)ccc(C(N2CCOCC2CN(C(=O)CC2CSCCS2)C)=O)cc1N C12(NC(C(C)n3cncn3)=O)CCCC1N(c1ncnc3[nH]ccc13)CC2 C1(CNC(c2cc(C)cc(Cl)n2)=O)CC2COCC2N1C(C1CCCSS1)=O C(Cc1ccccc1Br)(CC(=O)NN=c1ccn(C)[nH]1)NC(c1cnc(C)s1)=O C=C(C)C(C)(O)C(=O)NCC1CC2CCC1N2C(=O)CCn1nc(C)cc1C c1(C(=O)NCC(C)CN(C(=O)CC2CC2(C)C)C)csc2cc(Cl)cnc12 c1(C(C)=O)ccc(CNC(=O)C(Cn2cncn2)NC(=O)OC(C)(C)C)o1 N1(C(C2N(C(c3n(CCC)ncc3)=O)CCC2C)=O)CCC(C)(C2CC2)C1 N1(C(c2c(OCC)cccc2)=O)CCN(C(c2[nH]cnc2CC)=O)CC2(CC2)C1 Cc1nn(C(F)(F)F)c(C)c1CNC(=O)NC(CO)C(O)C1CCCCC1 c1(NCC2(COCC=C)CNCCO2)cc(NC)ccc1OC CC(C)(CC(=O)NC1CCCN(C(=O)CNC(=O)C2CC2)CC1F)CC(F)F c1(N2CC(C)(NC(CCNC(=O)NC)=O)C2)c(C(N)=O)cccc1[N+](=O)[O-] c1(C(N(C)CC2CCN(C(C(C(C)(C)C)OC)=O)C2)=O)cnc2ccncc2c1 Cc1c(C(N2CC(NC(=O)CCCCc3cnc[nH]3)C(C)C2)=O)ccn1C1CC1 C(=O)(CC1=CCCCC1)N1CCCC(NC(C2CC(=O)N(C3CCCC3)C2)=O)C1 C12(C(N3CC(NC(C4(COC)CCCCC4)=O)C3)=O)CC3CC(C(=O)N1)C2C3 C(=O)(CC1OCCc2ccccc21)N1CC(CCNC(c2c(CC)[nH]cc2)=O)C1 C#CCC(C)(C)C(=O)NCC(CCCC)NC(=O)Cc1cc(C(F)(F)F)n(C)n1 Cc1nc2ccc(CN3CCN(C(=O)Cc4cccc5[nH]ncc45)CC3)cc2[nH]1 c1(OC)cnc(C(N2CCC(OCCc3ccccc3)CC2)=O)c(F)c1 Cc1ncc(Cl)cc1C(N1CC2CC(NC(=O)Cc3cc(O)nnc3O)C1C2)=O c1(C(N2CC(CCC)N(C(=O)CC(C)F)CC2)=O)ccc(C#N)c(O)c1 C(C)(C)(C(=O)NCc1n[nH]cc1C(=O)NCCc1cocn1)OC(C)C C1(NC(=O)COC(F)F)CN(C(=O)CCCC2CCCC2)CCC1C(F)(F)F c1(C(N2CCC(O)(CC)C2)C(=O)NCC)nn(CC(=O)OC)cc1C C1(=O)C(O)COCCC1=O.c1(O)ccccc1.CCCC(=O)NCC1CC(N)C1 C(c1c(Cl)nc2sccn12)=CC(N1CC(NC(c2cc[nH]c2)=O)C(CO)CC1)=O N1(C(C2C(C)(C(F)F)C2)=O)CC2CC1C2C(=O)Nc1cnccc1C(N)=O Cc1cnc(F)cc1C(=O)NC1CCC(NC(=O)C(C(C)C)OCC(C)C)CC1 C(=O)(CCCCC(F)F)N1C(CNC(C=Cc2nnn(C)n2)=O)CCCC1 C1(C(N2CC(NC(=O)COc3cccnc3)(CO)C2)=O)CN2CCN1CC2 C1(C(N2CCSCCC2C)=O)(CC)CCCN(C(c2ccc(C(C)=O)[nH]2)=O)C1 C1(C(N(CCNC(=O)Cc2cc(O)nnc2O)CC)=O)CCc2nn[nH]c2C1 C1(C(N(C)CC2(CNC(C3CCCC3)=O)CC2)=O)CC2CCCC(C1)C2 C1(C(=O)NC(CNC(c2cc(C(=O)OC)ncc2)=O)C2CC2)CC2CCC(C1)C2 c1(OC)ncc(C(=O)NCCCN(C(=O)CCc2cnc(C)o2)C)cc1C CCC(CC(F)F)C(=O)NCC1CCN(C(c2cc(C(N)=O)cc(C)c2)=O)CC1 C1(NC(c2c(CC)onc2)=O)CN(C(C2(F)CC2c2ccccc2)=O)CC1O c1(C(C(=O)Cc2c(C(=O)NCC3(CC)CC3)cco2)OC)ccc(NC)cc1 c1(Cn2cc(C3C(OC)CN(C(C(C)=CC)=O)C3)nn2)cc2c(s1)CCC(C)C2 C1(C(NOC(CC)CC)=O)CCOCC1NC(c1ocnc1C)=O C1(C)(NC(Cc2cn(CC)nc2)=O)CCCN(C(c2cc(F)cnc2OC)=O)C1 c1(OC)ccc2cc(C(=O)NCC3CC3CNC(c3ccc(C)cn3)=O)sc2c1 C12(C(N3CCC(N(C(CCc4onc(CC)n4)=O)C)CC3)=O)CCCC(C1)OC2 C1(C(N(CCCNC(C(C2CC2)OCC)=O)C)=O)CCCC2(CCC2)O1 C1(C)(OC)CN(CC(=O)NCC2CC(F)(CNC(C3CCCN3C(C)C)=O)C2)C1 C(CC(C)C(=O)N(CCNC(C1CC(=O)N(C2CCCC2)C1)=O)C(C)C)=CCC c1(COC)nc(Cl)cc(=NCC2CN(C(=O)CN(C3CCSC3)C)CC2C)[nH]1 N1(CCC(N2C(CN(C(=O)C=Cc3ccco3)CC)CCC2)=O)CCC(C)CC1 C1(C(=O)NCCCN(C(C(Br)=C(C)C)=O)C2CC2)CCN(C2CC2)C1=O C12(NC(C(C)N(C)CC3CC3)=O)CC1CN(C(c1sccc1-n1ccnn1)=O)C2 C12(C(=O)NC(C(C)NC(=O)C=C(Cl)Cl)CO)CCC(CC1)C(C)(C)O2 CC1CCN(C(=O)CN(C)CCN(C)C(C2(CO)CCC2)=O)C1 C(N=c1[nH]c2c(cc1C#N)COCC2)C1C(NC(c2cc(C)oc2C)=O)CCC1 C(=O)(C(C)(C)COCC(F)F)NC(C)C(C)NC(c1ccncc1F)=O N1(C(C(C)Sc2ccc(C)cc2)=O)CCC(C2CN(C(c3cnccn3)=O)C2)C1 N1(C(CC(CC)C2CCC2)=O)CCN(C(c2ccc(C)nc2C)=O)C(CO)C1 c1(NC(=O)NCc2ccc[n+]([O-])c2)ccc2ccc(Cl)cc2n1 C1(C(N(C2C3CN(C(C4(CC=C)COC4)=O)CC32)C)=O)CCc2c(cnn2C)C1 N1(C(C2CCC(NC(c3nccc(C#C)c3)=O)C2)=O)CC2CCC(O)CC2C1 C1(C(=O)OC)CCOC2(CCCC2)C1.N12CCN(CC(O)C1)C(=O)c1nsc2n1 C1(C(N(CCN(C(C2CCN(C(C)=O)C2)=O)C(C)C)C)=O)CCC(C(N)=O)N1C C(=O)(C(O)C(F)(F)F)N1CC(NC(=O)CCCCc2ccc(Br)cc2)C1 N1(C(C2C(C)OCC2)=O)CC2CCN(C(=O)CCCn3ccnc3)C2C1 Cc1cc(C(F)(F)F)cc(C(=O)NC(C)CC(C)NC(=O)C=CC2CCCC2)n1 C1(CC(=O)NCC2CCCN(C(=O)COc3cnn(C)c3)C2)(OC)CCCCC1 C(=O)(C(CC(N)=O)NC(=O)CC1CC(=O)C1)NC1CCN(C(C)=O)CC1 c1(C(=O)NCC(C)C(F)C(=O)NCc2conc2C2CC2)cncc2[nH]ccc12 c1(C(=O)NC(C)CCNC(c2ccc3c(c2)COC3)=O)ccc2c(c1)C(C)CO2 N1(C(c2cnc(N(C)C)c(Cl)c2)=O)CC2CC1CCC2NC(c1cc(Cl)no1)=O N1(C(c2c(C)cccc2O)=O)CCCC(C2CN(Cc3ccc(Br)c(O)c3)C2)C1 CC1CCN(S(=O)(=O)CC(=O)NC2CC3(C2)CC3NC(=O)COC(C)C)CC1 c1(CC(C)C)ccccc1C(N1CC(NC(C2CC2[N+](=O)[O-])=O)C(C(F)F)C1)=O C=C(C)c1cn(C2CCC(C(=O)NCCc3ccc(C(=O)OC)cc3)CC2)nn1 c1(CC(=O)OCC)nc(C)c(C(N2CCC2CNC(c2ccon2)=O)=O)s1 c1(C(N2CCN(C(CC(C)C(F)F)=O)CC2CC2CC2)=O)c[nH]c2ncccc12 C1(C)(C(=O)NCCN(C(=O)C(C(C)O)N(C(=O)C2CC2)CC)CC)CCC(=O)NC1 CCCC(O)(CSCCc1cccc(CCOC)c1)CCC C(=O)(C(C)C(O)C(C)CC)N(C(C)CNC(c1ccccc1)=O)CC c1(CCC(=O)N(CC(CC)NC(C2CCC(=O)O2)=O)C)cncc(F)c1 CCCCCC(O)CC(=O)NC1(C)CC(NC(c2coc(CO)c2)=O)C1 c1(-n2c(Cc3cn(CC)nc3C)nc(C3CC34CC4)n2)cccc2cccnc12 C(=O)(C1=C(C)N(C)c2nnnn2C1)NC1CCN(C(c2c(CC)c[nH]c2)=O)C1 N1(C(c2ncc(OC)cn2)=O)CCC(NC(=O)C=Cc2cncc(F)c2)C(O)C1 C(C(CCCC)NC(=O)C(C)C(C)C)NC(c1cn(CC=C)nn1)=O C(CCO)(C(=O)N1CCOC(CNC(=O)C=Cc2nccs2)C1)N(C)C C1(C(N2CCC(CNC(C3CN(CC(F)(F)F)C3)=O)C2)=O)COCCC1(F)F Cc1nc2ccccc2cc1CN(C(C1COCCN(CC2(CO)CC2)C1)=O)C N1(C(C)=O)CCCC(C(N2CC(CNC(C3(CN(C)C)CC(F)(F)C3)=O)C2)=O)C1 C(=O)C1CCCn2nccc21.CCN1C(=O)Cc2ccc(C(=O)N(C)C=O)cc21 N1(C(CNCC=C)=O)CCC2(C1)OCc1ccccc12 C1(NC(C(F)OC)=O)CN(C(C2(C)CS(=O)(=O)C2)=O)CCC1C CCCC(CNC(=O)Cn1nc(C)nc1C)C(=O)N1CCC=CC1C(=O)OC C1(C(N2C(CN(C(=O)C(F)(F)C3(O)CCCC3)C)CCC2)=O)CC12CCOC2 N1(C(C=CCOC)=O)CCC(C(N2CCC(C(C)C)(CO)C2)=O)C12CC2 C(C)(CC(C)N(C(=O)CCOC1CCC1)C1CC1)NC(CN(CC)CC)=O c1(CCC)nc(C)c(CNC(=O)NCC(C)OC(F)F)o1 c1(NC(C2C(NC(c3ncn(CC)c3)=O)CC=CC2)=O)ccc2nccn2c1 CC(C)C(F)(CNC(C1CCCCCC1)=O)C(=O)NC1CCOC2(CCC2)C1 c1(C(=O)NCCNC(c2cnc(-c3cn(C)nc3)s2)=O)cccc(C2(C)CC2)c1 C1(COC)CCN(C(=O)C(c2ccoc2)NC(c2cccnc2S)=O)CC1 C1(NC(=O)Cc2c(Cl)cccc2Cl)CCN(C(=O)CCc2cn[nH]c2)C12CCC2 Cc1cc(N)n(CC(N2CC(CNC(c3sccc3C)=O)C(C)C2)=O)n1 C1(CN(C)C(c2cc(CF)on2)=O)CCN(C(C(C2CCOCC2)OC)=O)C1 C1(C(=O)NCc2ccc(O)nc2)(CNC(C2(C)CC(C(F)F)C2)=O)CC=CCC1 N1(CCc2n(C)cnc2)C(=O)CCN(CC(Cl)C(F)(F)F)C1=O C(c1ccccc1F)=CC(=O)NC(CC)(CNC(c1cnn[nH]1)=O)CC c1(OCC(=O)OC)cccc(C(=O)NC2CN(C(C3SCCC3C)=O)C2)c1 N1(C(C(c2ccc(C)s2)C)=O)CCC2(CCC(NC(=O)CCC3CCC3)C2)CC1 C1(C(=O)NCC2CCCN2C(C2CC2C(F)(F)F)=O)CCCCC(F)(F)C1 C1(=O)C(F)=CC(=O)N(C)C(C2CC2)CN1.C(CCC=CC1CC1)=C(C)C C1(N(C)C(c2ccc(C(F)(F)F)s2)=O)CN(C(=O)C(F)F)CC1F CP(C)(=O)c1ccc(C(N2CCC2CNC(c2nsc3ccccc23)=O)=O)cc1 N1(C(C(CC2CC2)NC(c2c(C)cnnc2)=O)=O)CCOCC(C)(F)C1 C#CCCCCCCC(=O)N(C)CCOCCC(=O)N1CC(OCCCOC)C1 C12(C(N3CCCC(NC(Cc4cc(C)on4)=O)C3)=O)CCCC1CC(=O)C2 C(c1ccc(C)cn1)=CC(=O)NC1C(NC(C(CCC)C)=O)C1 N1(Cc2n(C(C)C)ncc2)CC2(CN(C(=O)CCc3ccc(Cl)cc3)CCO2)C1 C1(C(N2C(C(=O)NCC(C)C#N)CSCC2)=O)CC2C(C1)C2(F)F c1(C(=O)NCCC(C)OC)cccc(CNC(=O)CC2CC(SC)C2)n1 C1(C(=O)NC(CCOC)CO)CCCN(C(c2cnc(O)c(C)c2)=O)C1C C1(CNC(C(C=C)O)=O)CN(C(=O)C(O)CCSC)CCC1C N1(C(C(C)SCCCC)=O)CC2C(C(=O)NC(c3nncs3)C)C2C1 c1(C(C(=O)NCCCOC)N(C(CC)CC)C)c(C)noc1C c1(C(N2C3C(NC(Cn4nnc(C)n4)=O)CC(C3)C2)=O)ccsc1S(C)(=O)=O c1(NC(c2cc(-c3nc[nH]n3)ccc2F)=O)c(F)cc(F)cc1Br C1(CC)CCN(C(C2CC2CF)=O)C1CNC(C1CSC1)=O c1(C(=O)NC2(CNC(C(C)=C(CC)C)=O)CCOC2)cn(C)c(=O)nc1O c1(NC(C(C)C)CCO)ccc(S(=O)(=O)N2C3CCC2CC3)c2ccncc12 C1(C(=O)NC(C(=O)NC(CCC(=O)OC)C)Cc2cnc[nH]2)C2CCC(F)(F)C12 c1(C(=O)NN2CC(CC)N(Cc3ccc(C(=O)O)s3)CC2)cccc2c[nH]nc12 c1(C(N2C(C(CNC(C(CC(C)C)C)=O)(C)C)CCC2)=O)cccc2c1NCC2 C(=O)(C=CS(C)(=O)=O)NC(C)CCNC(=O)CCC1NC(=O)NC1=O Cc1ccc2c(CC(N3CC(CNC(C4C=CCCC4)=O)C(C)C3)=O)c[nH]c2c1 C(c1ccccc1F)=CCC(N1C(C(C)NC(C2CCCS2(=O)=O)=O)CCC1)=O N1(C(c2c(OC)c(Cl)sc2)=O)CC(NC(c2ccnn2C)=O)CC(O)C1 N1(C(C(N2CCOCC2)C)=O)CCN(C(C2CCC=CCCC2)=O)CC12CCC2 N1(C(C2(C)CN(C(CC3C(C)(C)C(O)C3)=O)C2)=O)CCC12CC(C)(CO)C2 C1(C(N2CCC(CNC(=O)Cc3cnn(C(F)F)c3)C2)=O)C2CCCCCCC12 C12(C(N3CC(C4(NC(C5C(OCC)C5)=O)CC4)C3)=O)CCCCC1CS(=O)(=O)C2 c1(C(=O)Nc2nc(CNC(C)CC3CCCCO3)[nH]n2)ccc(Cl)cn1 C(=O)(C(C)(O)C(F)(F)F)NCCSCC(=O)NCCn1c(C)cnn1 c1(C(=O)NC2C(NC(=O)CN3CCOC3=O)CC2)ccn2nnnc2c1 Cc1ncc(C(N2CCC(CC(=O)N(C(C)CC(C)C)C)C2)=O)c(=N)[nH]1 CC(C)C(C(=O)N(C1CCCCC1O)C)NC(=O)COc1cccnc1 CS(=O)C1CN(C(c2cc(CNC(C3CCCCC3)=O)no2)=O)C1 CCCCC(CNC(c1ncc[nH]c1=O)=O)NC(=O)CC1(N2CCCC2)CC1 CC1C(C)N(C(c2nccc3nn[nH]c23)=O)CCN1C(=O)C(=O)C(C)(C)C c1(CN(C(=O)C(=O)N(C)CC2CC3CCC2C3)CC=C)ccc(F)cc1 c1(C(N(CC(C)CNC(C2CC23CC(F)(F)C3)=O)C)=O)cccc2[nH]ncc12 C1(CNC(CC=CC)=O)CCCC(CNC(c2cc(C(C)C)nn2CC)=O)C1 N1(C(C(=CC2CCCC2)C)=O)CC2(C1)CN(C(=O)CC(C)O)CC2CO N1(C(CC2(C)CCCO2)=O)CCCC12CCN(C(c1csc(F)c1)=O)CC2 CC1COC(C(=O)NC(C)(C)CN(C)C(c2csc(C(N)=O)n2)=O)C1 Cc1nn2ncccc2c1C(=O)NC1CC1CNC(=O)CCOCC(F)(F)F Cc1ncc(C(=O)N(CCNC(C23CC(C)C2C3)=O)CCc2ccccc2)o1 c1(C(N2CC(O)CC2CNC(C2(CC(F)F)CCC2)=O)=O)cn2ncccc2n1 c1(C(=O)NCC(C)CN(C)C(c2nn(C)cc2C(C)=O)=O)nc2ccccc2[nH]1 C12(C(N3CC4C(NC(C(C)(C)OC(C)C)=O)(C4)C3)=O)CC=CC(C1)OC2 N1(C(c2c(C)nc(CO)nc2)=O)CCN(C(=O)CC2CNC(=O)C2)CC12CCC2 C(C(C(=O)NC1CCCCC1NC(C1CC2CC1C2)=O)C(C)(C)C)OCC=C N1(C(CNC=O)=O)C2CC1CN(C(=O)CCCC1OCCO1)C2 c1(C(=O)NCC2C(N(C)C)CN(C(C(C)=CC)=O)C2)cc2cccc(C)c2nn1 c1(C(=O)NC2C3(CCN(C(C(C)(C)F)=O)CC3)C2)c[nH]c2cc(Cl)c(Cl)cc12 Cc1cc(Cl)c(C(N2CCC(NCC(N3CCS(=O)(=O)CC3)=O)C(C)C2)=O)cn1 CC(C(=O)N1CC(NC(C2(CCF)CCOCC2)=O)C(F)C1)C(C)(F)F N1(C(C(CSC)C)=O)CCN(C(C2(O)CC2)=O)CC1CC(F)F C(C(F)(F)F)(C(F)(F)F)N(Cc1c(C)onc1)Cc1cccc(Cl)c1 C1(C(N2CCCC(CCF)C2)=O)CC(F)(F)CN1C(C1CCOC1)=O c1(N2CCC(C(C)NC(=O)C=Cc3ccccc3Br)CC2)cc2ncnn2cn1 CCC(CC(=O)NC(C(=O)NOCCOCCOC)C1(C)CC1)C1CC1 CCCCCCC(F)C(=O)NC(C)CN(C)C(c1cn(C)[nH]c1=N)=O N1(C(C2CC(C(=O)NC3(c4cccc(Cl)n4)CC3)C2)=O)CCOC2CC12 N1(C(C2CC(OC)C2)=O)CCC(C(C)(C)C)(CNC(=O)CN2CCC(C)(O)C2)C1 c1(NCc2ncc(C)s2)cc(=NCc2cc(Br)cc(C)n2)[nH]cn1 c1(C(N(CC(CC)NC(C(CCC#C)O)=O)C)=O)c(C)c(C)cc(C)c1C N1(C(c2c(C)nc(C(C)C)s2)=O)CC(C)N(C(c2ccc(C#N)o2)=O)CC1C n1(CC(=O)NCCC2CC(NC(CC3C(=O)NC(=N)S3)=O)C2)ccc([N+](=O)[O-])n1 c1(OC)ccc(OC(C)CNC(=O)NC23CC(F)(C2)C3)c(Br)c1 C12(C(N3C(CNC(CC4CC(C)(C)C4)=O)C=CC3)=O)CCCC1C2(F)F C1(C(N(CCCNC(=O)Cc2c(F)cccc2F)CC)=O)CCCC1S(C)(=O)=O Cc1ccc(C(N2CC(NC(C3Cc4nncn4C3)=O)CC2(C)C)=O)c(O)c1 C1(S(C)(=O)=O)(C(=O)NCC2CN(C(C3=C(C)OCC3)=O)C(C)CC2)CCOCC1 c1(C(=O)OCC)ncc(C(=O)NC2CC(C)(NC(C3CC3C(N)=O)=O)C2)s1 C1(CNC(C(C(C)C)SC)=O)COC(C)(C)CN1C(c1ccc(F)c(O)c1F)=O C12(C(=O)NCCC3CN(C(C(C4CCC4)OC)=O)C3)C=CC(CC1)C2 c1(CC(=O)NC(C)(C)C=CC(=O)Nc2cnc(F)nc2)cccc(F)c1F CC(C)C(O)C(=O)NCC1CC(F)CN1C(=O)COCC1CCOC1 Nc1cc(Br)cnc1C(=O)NC1CCCN(C(C2(CF)CC2)=O)CC1 CC1=NN(C)C(=O)C1CC(=O)NC1COCCN(C(C2CCOC(C)(C)C2)=O)C1 N1(C(C(CC)N(CC)CC)=O)CCN(CCNC(C2(C)CC3(CC3)C2)=O)CC1.C(C)=O C(=O)(C(CC1CC1)NC(=O)CCN1CCOC1=O)NC(c1ncc(C)[nH]1)CC c1(C(N2CCC(NC(c3c(C)noc3C)=O)C(O)C2)=O)cc(Cl)cc(Cl)c1O Cc1cc2nc[nH]c(=NCC3CC(CNC(c4ccoc4Cl)=O)CO3)c2[nH]1 Cc1oc(C(F)(F)F)c(C(N2CCN(C(C3(C)CCCN3C)=O)CC2C)=O)c1C CCC(F)(C(=O)OC)C(=O)N1CC2CC1CC2CNC(=O)CCC(C)C C=CC(C)(C)CC(=O)NC1(C(=O)NCC2C3CCCCCC23)CCSC1 N1(C(c2c(COC)cccc2)=O)CCCC(COC)(NC(=O)C#CC(C)(C)C)C1 Cc1ccc(-c2cc(C(=O)NC(C)CCN3CCCCC3)no2)c(C)c1 C1(C(N(CCCNC(C=C2CCC(C)CC2)=O)C)=O)CCC2C(CC1)C2(F)F N1(C(C(CC(C)C)N(C(=O)CC2CCC(C)(C)O2)C)=O)CCCC(C)(C)C1C c1(CCC(=O)N(CCCNC(c2csc(O)n2)=O)C)cc(F)cc(F)c1 N1(C(COCCOC)=O)CC(NC(C2CCC(c3ccccc3)O2)=O)C(O)C1 c1(Cc2nc(-c3ccc(C(C)C)nc3)n(CC3CC3)n2)cn(C)c2ccccc12 c1(NC(CC(=O)Nc2c(C(C)C)cccc2)C)ncc2[nH]ncc2n1 C(C(C)(C(N)=O)NC(C1(CNC(=O)CN2CCC(=O)CC2)CCCCC1)=O)OC C(=O)(CC(C)CC(C)(C)C)N(C)CC1N(C(Cc2cn(CC)nc2)=O)CCCC1 C1(CCC(=O)NC(C(=O)OC(C)C)C)CCCN(C(=O)CC2C=CCCC2)C1 C1(N(C(=O)CSCCC#N)CC#C)CCN(C(=O)CCSC2CCCC2)C1 Cc1ccc(OC2CCN(C(=O)C(c3ccc(F)cn3)(F)F)C2)cc1 C1(C(=O)NCCN(C(CC2(COC)CC2)=O)CC(C)O)CC2(CCCC2)C1 C1(C(=O)NC(CN(CC)CC)C)CCC(C)(C)N(C(c2cc(CO)nn2C)=O)C1 C1(C(N(CC(CC)NC(=O)C=C(C)C(F)F)C)=O)(COC)CCCCO1 C(=O)(C1=NOC(c2ccccc2)C1)NCCCNC(C(c1cnccn1)C)=O CC1CN(C(C2(CCF)CCC2)=O)CCCN1C(c1cnn(C2CC2)c1)=O c1(CC)ncc(C(=O)N(C)CCN(C(=O)CCc2cnc(C)s2)C)c(O)n1 c1(C(=O)NCC(CO)NC(c2cccc(OC(C)C)c2)=O)n[nH]c2c1COC2 C1(Nc2scc(C=C)n2)CN(C)CC(F)(F)C1 c1(C(N(C(CC)CO)C)=O)ccncc1-n1cc(CC(C)(C)C)nn1 C12(NC(C#CC(C)C)=O)CCCC1N(C(=O)CSCc1csc(=N)[nH]1)CC2 N1(CC)OCC(N(C2CCOC(c3ccc(F)cc3)C2)C)C1=O CC1CC(CC(N2CCC2CC2CC2)=O)CN1C(=O)Cn1cccc1 c1(CNC(C2CCCC2O)C)ccc(Br)s1 c1(C(N2CCC(C(C)NC(c3c(C)coc3)=O)C2)=O)cc(C(N)=O)ccn1 C#Cc1cnc(C(=O)NC23CCN(C(c4cncc(C)c4)=O)CCC2C3)c(C)c1 N1(C(Cc2c(C)non2)=O)CC2(CC2)CC1CNC(=O)C(C)(F)F C1(Nc2ncc(C#C)cn2)CC2CC(C1)N(C(C1CCCCC1C(F)(F)F)=O)C2 C1(C(N(CCN(C(=O)CCCc2ccncc2)C)C)=O)C(C)(C)C1(F)F N1(C(c2cn(CC)nc2C)C(=O)NC(C)C)CCS(=O)C(C)C1C C(=O)(CC(C)C(F)(F)F)NCC(=C)CCNC(=O)Cc1cccc(C2CC2)c1 CC(CC(=O)NC1CCOC1C(N1CC(CC2CC2)C1)=O)N(C)C n1(CCC)ncc(CNC(C(C)(C)CCN(C)C)c2nnnn2C2(C)CC2)c1C c1(CCC(=O)NCCN(C(c2c(NC)c(F)ccc2)=O)C)cccc([N+](=O)[O-])c1 c1(C(=O)N(C)C)ccc(C=CC(=O)NC2CCCC2NC(c2cnc(C)o2)=O)cc1 n1(CC)cnc2c(NC(C)CC(N)=O)[nH]c(=NC(C)c3ccccc3)nc12 N1(C(C2CC(C)C(C)CC2)=O)CC(O)(C2(CNC(C3(CO)CCC3)=O)CC2)C1 C#Cc1cccc(CC(=O)NC(C)(CO)C(=O)NCC=CBr)c1 c1(NC(N(CCn2cc(CNC(C)=O)nn2)CC)=O)cc(Br)c([N+](=O)[O-])[nH]1 c1(C(C)C)ncc(C(=O)NCC(C)N(C(=O)C=CCO)C)n1C c1(CNC(N2CCSCC(CO)C2)=O)cc(O)cc(Cl)c1 c1(C(CC)C)nc(NC2CCCCC2NC(C2CCC3CC3CC2)=O)cc(C)n1 C(=O)(CCCCCn1cc(CN2CCCCC2)nn1)NC(c1ncccn1)CC Cc1nc(C(N2CCCC2CNC(c2ncc3ccccn23)=O)=O)c(=O)[nH]c1C c1(-c2nc(CCC(=O)NC(C)(CNC(=O)C=CBr)CO)on2)cccc(Cl)c1 CC(CCNC(=O)Cn1cc(Cl)cn1)CCNC(c1cc[nH]n1)=O c1(-c2cn(C(C)C(=O)O)nn2)cccc(NS(=O)(=O)CC(=O)OC(C)(C)C)c1 C1(NC(c2cc(SC)oc2)=O)C(C)CCN(C(=O)Cc2ccc(Cl)cc2)C1C N1(C(c2cc(C)c(O)nc2)=O)CC2CN(C(c3cc(O)nc(O)n3)=O)CC2(C)C1 c1(C(=O)NCC(CC(=O)OC)NC(C(C(=O)OCC)OC)=O)ncc(Cl)cc1Cl N1(C(C2N(C(=O)OC(C)(C)C)CC2)=O)CCC2(CC2NCC2CCCCC2)C1 C1(NC(Cn2cccc(C(=O)OC)c2=O)=O)CCCN(C(=O)CC2(O)CC2)CC1 c1(CCC)ccc(C(=O)NC(C2CCN(C(c3cc(C(C)=O)cs3)=O)C2)(C)C)[nH]1 CC1(C)CC(C(=O)NCCSCCCO)(CNC(=O)CCC2CC2)C1 N1(C(C(C)n2cccn2)=O)CC2(CC(NC(c3nocc3C3CC3)=O)C2)C1 C(=O)(C1OCCc2ccccc21)N1CCCCC(N(C)C(c2ccnn2C)=O)C1 N1(CC(=O)NCC(=O)NC2CC(NC(=O)CSC(F)F)C2)CCCCC1 C1(c2cn(CCCC(=O)N(CCCN(C)CCC3CC3)C)nn2)CC2(CCC2)C1 C=CC1(C(N2CCCC3(C2)N=N3)=O)CCN(C(=O)C#CC2CCC2)C1 CN1CCN(CC(=O)NC2(C)CC(NC(=O)CC34CCC(CC3)C4)C2)CC1 C(CCC(=O)NCC1CCC1NC(c1ccnn1CCC)=O)NC(=O)NCC#C c1(C(N2CCN(C(c3c(C)cc(C)o3)=O)CC2)=O)cccc2ncnc(O)c12 C(=O)(C(O)C(CCC)NC(=O)CNC(C1CC1C)=O)NC(CC#C)C(N)=O O=C1CC(C(=O)NC2CN(C(c3cnsc3)=O)CCC2C(F)(F)F)CC(=O)N1 CCCC(F)C(=O)N1CCCC1C(C)NC(=O)CCC1CC(F)(F)C1 C(C1=CCN(C(c2ccn(C(F)F)n2)=O)CC1)NC(C(C)(C)c1ccncc1)=O C(C)(C)(CC(F)C(=O)N1CC2CC1CO2)NC(C(CCC)=CCC)=O C(=O)(C1=C(C)CN(C(c2cn(C3CCOCC3)nn2)=O)C1)N(CC)CC CCCCCCCCC(CO)NS(=O)(=O)c1cccc(-c2nnn(C)n2)c1 C1(NC(C2C(C)C2C)=O)CC(C)(CNC(C2CCCCO2)=O)C1 C1(NC(C(n2c(C)cc(C)n2)C)=O)CCN(C(=O)C#CC2CC2)CC1C C(=O)(C(C)(O)C(C)(C)C)N1CCC(CN(C(Cc2c(OC)ccnc2)=O)C)C1 c1(OC)ccc(CC(C)C(N2CCCC(CC(=O)O)C2)=O)cc1S(N)(=O)=O c1(N2CCCC(NC(C3(CC)COC3)=O)C2C)ncnc2sc(C(C)C)cc12 N1(CC(C)NC(c2c(CC)scc2)=O)CCN(C(c2ncc(Br)cn2)=O)CC1 N1(C(CCC(=O)NC)=O)CCCC(C)(CNC(=O)CC2(OC)CC2)C1 C1(NC(CC=CCCCCC)=O)CCC(C)N(C(c2cccc(C(N)=O)n2)=O)C1 c1(C(N(CCC(C(C)C)NC(C(CSC)C)=O)C)=O)cc2cn[nH]c2cn1 CCCC(C(O)C(=O)N(C(C(N)=O)C1CC1)C)NC(=O)CN=[N+]=[N-] CCCCCC(C(=O)NCC1C2CN(c3c(Cl)cncc3[N+](=O)[O-])CC12)C(C)C N1(C(c2cc(C)ncc2C)=O)CC2(CCCC2)C1C(=O)NCCC(C)N1CCC1 c1(-n2cc(CCOC)nn2)cccc(C(=O)NC2(C)CCSCC2)c1 c1(CC)cc(C(N2CCC(O)(CN(C)C(c3cc(CC)c(C)s3)=O)C2)=O)nn1C n1(C(CC)C)nnnc1C(c1nnn(C)n1)NCc1cc(OC)no1 C=CCCCC(=O)NCC(C1CCOC1)NC(c1snnc1C1CC1)=O c1(NC(=O)OC(C)(C)C)cc(NC(=O)C(c2cccc(Br)n2)(F)F)cc(Cl)c1 C(=O)(CC1OCc2ccccc21)N(CCCCN(C(=O)COC1CCOC1)C)C N1(C(C2(C=C)CCN(C(c3n[nH]c(C)c3C)=O)C2)=O)CCCCCCC1CC c1(C(=O)NC2CN(C(CCC(=O)OCC)=O)CC2C(F)F)cn2ccsc2n1 C#CC1(C(=O)NCC2COCC2N(C)C)CCN(C(=O)C2=CCSC2)C1 C1(CC=C)(NC(C2CCC(C(N)=O)O2)=O)CCCN(C(c2cc(C#N)cs2)=O)C1 N1(CC#N)CC=C(CCNC(=O)CCOC2CCN(C)CC2)CC1 c1(C(=O)NC(C2CCCN(C(=O)CCc3cnn(C)c3)C2)C)ccnnc1O n1(CC(C)CO)nc(CCN(C)C)nc1-c1cn(-c2ccccc2)nn1 C1(NC(c2cnc(CC)nc2C)=O)CCN(C(=O)C(C)(O)COC)C12CCCC2 Cc1oc(CO)cc1C(N1CCC(CNC(=O)C(C)Sc2ccccc2Cl)C1)=O C1(C)(CNC(N(c2c(NC(C)=O)cccc2)C)=O)CCC(=O)NC1 c1(C(=O)N(C(C)(C)C)CC)cc(-c2cccs2)[nH]n1.c1(C(CC)N)nc(C)cs1 c1(OC)cc(C(=O)NC2CN(C(=O)CCCCCF)CC2C)cc2c1OCC2 C1(C)(CNC(C=C(C)c2ccc(OCC(C)C)cc2)=O)CCCCC1(F)F C(C)(CCC#N)(c1n(CCCOC)nnn1)NCCc1ccncc1Br CN1CC(O)CCC1C(=O)OC1CCN(C(CCOC(C)(C)C)=O)CC1 c1(C(N2CC(CC=C)(NC(c3ccn(C)c3C)=O)C2)=O)cnc(O)cc1C c1(CC#N)ccc(NC(=O)CC2CN(C(C3CC(=O)C3)=O)CCO2)cc1 CN1C(=O)C(=O)N(CC(=O)NCC2(C)CCCN2C(c2ccno2)=O)C1=O C1(C(N(C2CCCCC2)CCNC(=O)COC(=O)CO)=O)CCCOC1 Cc1nnc(CCC(=O)NC2(C)CC(NC(C3CNC(=O)N3)=O)C2)n1C c1(C(CCCOC)NCCCCOC)ccc(OC)c(F)c1 N1(CC=C)CCC(N(CCCCNC(c2cc(C3CCCN3C)[nH]n2)=O)C)C1=O c1(SCCC(=O)NC2(COC)CN(C(C3CSCC(=O)N3)=O)C2)ccc(F)cc1 Cc1c(C(=O)N(C2CN(C(C3(C)CC3F)=O)C2)C)oc2ccccc12 Cc1nc(C(=O)NCC(C2CCCN2C(=O)CCCC#N)(C)C)c(C)o1 N1(C(CC)=O)CCN(C(c2ccc(SC(F)(F)F)o2)=O)CC(C)(F)C1 N1(C(c2c(OC)nsc2)=O)CCCC2CN(C(=O)CCc3cscn3)CCC12 c1(C(=O)NC2C3CN(C(COCCN(C)C)=O)C(C3)C2)nccc2occc12 C(=O)(C(CO)C(C)(C)C)N1CC(C=CC)C(C(=O)NCc2cncc(OC)c2)C1 c1(C(N2CC(N(C(C=CCC)=O)C)C(F)C2)=O)ccc2ncccn12 N1(C(Cc2cc(C)on2)=O)CCC2(CCN(C(=O)C(F)(F)C3CC3)CC2)C1 c1(NC(CCCN)CO)ccc2ccncc2c1[N+](=O)[O-] c1(C(N2C3C(C(=O)NC4CCC(C)CC4)C(C3)C2)=O)cccc2cccnc12 c1(NC(C(=O)N(C(C)CCN2CCCC2)C2CC2)=O)ncc(-c2ccncc2)s1 C(C(C(F)(F)F)N)NC(=O)C=CCNC(C1CCC1)=O.C1(C)CCCC1 C1(C(NCP(C)(C)=O)=O)CCCC(NC(C2(C(C)(C)OC)CC2)=O)C1 C1(NC(c2cc(C(N)=O)no2)=O)CCSC12CN(C(=O)CC1CCOC1=O)C2 c1(C(N2CCC(NC(CCc3n[nH]c(=N)s3)=O)C2)=O)ccc2cnoc2c1 C1(CC)CCN(c2cc(N3CCOC(C4CC4)C3)nc(C)n2)CCO1 c1(C(=O)NCCOCC(=O)NCC2CCC(O)C2)ccc(F)c(F)c1 CC(Cc1cnc[nH]1)C(=O)N(CCCNC(c1cnco1)=O)C1CC1 C1(NC(C=CCC)=O)CCN(C(c2cc(OC)c(Br)s2)=O)CC1(C)C S(=O)(=O)(C(C)CN=c1[nH]c(=NCc2cc(C)c(C)cc2C)[nH]c2c1CCC2)NC CCCC(=O)N(CC(=O)NCCc1ncc[nH]1)CC(C)C O(NC(=O)C(CC)NC(c1ncoc1CC)=O)CCCC#C Cn1nccc1C(F)=CC(=O)NCC1CC1CNC(c1cc(Cl)ccn1)=O C1(S(C)(=O)=O)(C(=O)NCC(C(C)C)NC(C2CC=CCO2)=O)CC(O)C1 C(CCO)(C(F)(F)F)NC(c1ccc(CNC(CC(C=C)C)=O)nc1)=O C(C(N=c1c(C#N)c[nH]c2ccccc12)C(C)C)NC(c1cnc(C)o1)=O C1(NC(C(c2n(C)ncc2)O)=O)CCCN(C(C2SCCCS2)=O)CC1 N1(c2nnc(O)s2)CCC(NC(=O)C(CCC)OCC)CC1.C=C1CCC1(CO)C c1(C(=O)NC(C)C(C)(C)NC(=O)CC(C)n2cccn2)cnc(O)c2cncn12 c1(COCC(=O)NCCCCNC(C(C)n2cncn2)=O)cccc(Cl)c1 C1(C(=O)NC2CCCN(C(CSCC#C)=O)CC2)CC12CCC(C)(C)CC2 c1(C(N(C2CN(C(=O)CCc3nccn3C)C2)C)=O)cc(C(F)(F)F)cnc1N c1(C(=O)NCCC(CNC(=O)C(F)=CC2CC2)O)ccc(C2CCOC2)cc1 Cc1ccc(C(=O)NC(C2CCCN2C(c2cc(C)on2)=O)C)c(O)n1 c1(C(N2CC(C(C)NC(C3CC34CCSCC4)=O)C2)=O)csc2c1CCCC2 c1(C(N2C(C)CCC(CNC(CCCC)=O)C2)=O)cc(F)c(Br)cc1C C(=O)(CCS(=O)(=O)C(F)(F)F)N(C1CCCCN(C(C(CC)(C)C#N)=O)C1)C C1(NC(=O)CCc2ccon2)CN(C(=O)C(O)C(F)(F)F)CCC12CCOCC2 c1(CN2CC(n3ncc(NC(COCCOC)=O)c3)C2)ccc2oc(C)nc2c1 C1(O)(NCCC)CCCN(C(C2(C(=O)N(C)C)CCCC2)=O)C1 c1(NC(CN(C(C2(CC#C)CCCC2)=O)C)(C)C)ncnc(C)c1OC N1(C(c2ccc(C)s2)=O)CC(C)OC2(CCN(C(C3CCCSC3)=O)C2)C1 N#Cc1ccc(=NCC(=O)NCCCN(CCO)C(C2(F)CCOC2)=O)[nH]c1 N12CC3(CC3)CC1CNC(=O)c1nsc2n1.C(=O)(CCC(F)F)OC n1(CC)cnc2c(NCC3(C)CC(C)(C)C3)[nH]c(=NCC=C(C)C)nc12 C12(NC(CCCCSC)=O)CC(CNC(=O)CNC=O)(C1)OC21CCC1 c1(CNC(C(C)=CCC)=O)cc(C(=O)N(CC(O)CC)C)cs1 CCCCC(CC)CCC(=O)NCCCNS(=O)(=O)c1cccnc1C(=O)OC c1(C(N2CC(CCNC(C=CSC)=O)OC(C)C2)=O)cc2cc(C)ccc2o1 CC1=C(C)CC(C(=O)N(C(CNC(=O)CS(N)(=O)=O)C2CC2)C)CC1 N1(C(COC)=O)CCN(C(=O)CCS(=O)(=O)N(C)C)CC(C)(F)C1.C(C)N N1(C(CN2CCN(C(C(c3cccnc3)C)=O)CC2)=O)CCC2(CC1)CC2 C(=O)(C=CS(C)=O)NCCC1CCN(C(C2(CCOC)CCC2)=O)C1 C1(C(=O)NCC2CC2C2CCCO2)CN(C(=O)CC2(O)CCC2)CCO1 CC1=C(C(=O)NC(c2cccc(C(=O)O)c2)C(=O)O)Cn2ncnc2N1C c1(C(N(CCCNC(CCC(=C)C)=O)C)=O)nccc2ccccc12 N1(C(CC(CNC(C(C)N=[N+]=[N-])=O)C2CCC2)=O)CCCC2(CCOC2)C1 c1(C(=O)NCC(C)N(C(c2ccc(F)c(O)c2)=O)CC)cc2c(nn1)CCCO2 CC1(C)CC(=O)NC1CN(c1ccccc1)CCCN.C1(=O)C(CC(=O)O)O1 C(=O)(C(C(C)C)NC(=O)CN(C1CCCC1)C)NCC=CCC(=O)OCC N1(C(C(CCC)NC(N)=O)=O)C2CCC1C1CC1(NC(c1scnc1C)=O)C2 C1(CNC(C2CN3CCCC2C3)=O)CN(C(=O)C2CC2)CCC1(F)F N1(C(C(C=C=C)C)=O)CC(C(=O)NCCN(C)C)C2(CC2)C1 C(=O)(C(CC(C)C)NC(C)=O)NCC(CNC(CC1(C=C)CC1)=O)OC N1(C(CC(C)C)=O)CC2CCN(C(c3cc[nH]c3)=O)CC2C1 c1(N2CC(C(=O)NCC(=O)NCc3ccsc3)C(O)CC2)nc2ccccc2s1 C1(c2ccccc2F)(C(N(CCC(C)O)C2CC2)=O)CC2(CC2)C1 C1(OC)CC(CNC(=O)CCC2CCOC2)N(C(c2n[nH]c(C)c2O)=O)C1 CC1C(NC(=O)CC2(C)CCC2)CCCN1C(c1csc(C(C)(C)C)n1)=O C1(C)(CCNC(c2c(OC)csc2)=O)CCN(C(C2(C)CC(C)C2)=O)C1 c1(OC)cc(C(N2CCCC(NC(=O)C(=O)O)C2)=O)cc([N+](=O)[O-])c1 C1(C)(C(=O)NCCCN(C(C)C)C(C2CCN(CC(F)(F)F)C2)=O)COC(=O)C1 C1(NC(C(C2CN(C(C(C)SCC)=O)C2)OC)=O)CC(C)CC(C)(C)C1 C(=O)(CCCCCO)N1CCC(N(CC#C)C(C2CC2(Cl)Cl)=O)CC1 C1(NC(c2n(COC)ncc2)=O)CCN(C(=O)Cc2cnccc2C)C12CCC2 Cc1cccc(COCC(=O)NCCC2CCN(C(C3CCCC(=O)O3)=O)C2)c1 Cc1ccn(CC(=O)NC2CCCC2NC(c2cnnn2C)=O)n1 N1(C(c2nnn(CC)c2C)=O)CC2CC1CN2C(=O)C(c1c(Cl)cccc1Cl)C CCC(C)(CCNC(c1cnc(C2CC2)o1)=O)NC(c1cc(Cl)ns1)=O C1(C(N2CC(OC(C)=O)C2)=O)CCN(C(=O)c2cc(C)cc(O)n2)O1 CCCC(C)(C)CC(=O)N1CCN(C(c2cc(C#N)ccc2C)=O)C(C2CC2)C1 C1(NC(CCOCCOC)=O)CCC2(CC1)CC2NC(=O)C(C)C(C)(C)C C(C)(C(=O)NC1CC(OCC2CC2)C1)N(C(=O)Cc1ccsc1)CCC.OCC N#Cc1cccc(CCC(=O)NCCC2CN(C(C3CCSC3)=O)CCCO2)c1 c1(C(=O)NCCN(CCCCCC)C(c2cncc(C)n2)=O)cc(C)ccn1 c1(C(=O)NC2CCN(CCNC(C(CC)C(C)C)=O)CC2)ccc2nnnn2c1 n1(CC(C)C(=O)NCCCNC(=O)CC2(O)CCCCC2)ccc2ccccc12 CC1=NOC(=O)C1CC(N1CCN(CC2CN(C(c3occc3Br)=O)C2)CC1)=O C1(CCCC)CN(C(c2[nH]ccc(=O)c2C)=O)CCN1C(C1CN(C)C1)=O CCC(O)C(C)C(=O)NCCN(C(c1cncnc1C(C)(C)C)=O)C1CC1 N1(C(C2(C)CC2)=O)CCCC(C2(NC(C3CN(CC(F)(F)F)C3)=O)CC2)C1 N1(C(C(CCC)OC)=O)CC(NC(=O)CCc2ccc(Cl)cc2)CC(F)C1 c1(OC)c(F)ccc(F)c1CN1CC(NC(C2CCCS2)=O)C(F)(F)C1 C(=O)(C1CCCc2ncnn21)NC1CCC(C)N(C(c2[nH]ncc2C#N)=O)C1 c1(C(N2CC3C(C(N4CCCC(CC)(CO)C4)=O)(C3)C2)=O)cc(C)cc(C#N)c1 C(CCC(C)C(=O)NCC(C1CCN(C(=O)C=C2CCN(C)CC2)CC1)C)OC c1(C(N2C3CCC2C(CNC(=O)C(F)(F)C2CC2)C3)=O)ccc2c(c1)CCC2 N1(C(C2(CC)CCC2)=O)CCN(CC2CCN(C(C3CCC(C)C3)=O)CC2)CC1 C1(C(=O)NC(CC(=O)N(C2CCCCC2)C)C2CC2)CC2(CC2)CO1 C1(F)(CNC(c2n(C)nc(C(F)F)c2)=O)CCN(C(C2(C)CC(F)C2)=O)CC1 CC1(C(N2CCOC(CC(=O)NCC(O)C3(Cl)CC3)C2)=O)CC(C#N)C1 N1(C(C2CC(CCC)OCC2)=O)CC(C2(NC(=O)CC(=O)N(C)C)CC2)C1 c1(C(=O)Nc2occ(C)n2)sc(=NCc2[nH]c(C)nc2C)[nH]c1C N1(C(C2NC(=O)CC(=O)C2)=O)CC(C(=O)Nc2cnn(C3CC3)c2)CC12CCC2 Cc1ccc(C(=O)NC(CO)C(C)NC(=O)CC2COCC2O)cc1N N1(c2c(S(=O)(=O)NC3(CC)CCOC3)cccn2)CCN(C)C2(CCOC2)C1 C1(CNC(C(COC)(C)C)=O)(CO)CCCN(C(=O)C(C(C)(C)C)SC)C1 N1(C(C=CCCC)=O)CCCC(CCNC(=O)Cn2cc(C)cn2)CC1 CC1(C)C=CC(NC(=O)NC2CC(OCC(F)(F)F)C2)CC1 C(=O)(CC(C(C)C)NC(=O)CC1CC(C)=NO1)NC(c1nc[nH]n1)CC Cc1[nH]nc2cc(NC(c3c(-c4cnc(CO)nc4)cncc3F)=O)ccc12 C1(NC(C(C2CCC2)OC)=O)CN(C(=O)C(C)(C)C#N)CC1c1ccccc1F C12CC13CCN(C3)C(=O)CCN2.Cc1cc(CNC(C2(F)CC2)=O)no1 CCC(O)CCN=c1nc(-c2ccccc2)[nH]c(=NCc2nnnn2C)[nH]1 c1(C(N2CC(C(N3CCC(C)(CC)C3)=O)(SC)C2)=O)cc(C)n(C)c1C c1(NCC(C)CNC(=O)CNC(=O)N(c2ccccc2)C)ccn2ccsc12 O=C1CC(NC(=O)CN(C(=O)CCn2cccn2)C2CCC2)CN1 c1(C(=O)NCCC(C)NC(C2CC3C=CC2C3)=O)ccc(-c2ncc[nH]2)cc1 C1(NC(CCN(C)C(C2CCC(O)CC2)=O)=O)CC(O)C(O)C1 C1(NC(c2c(C)ncnc2C)=O)CCC2CCN(C(=O)C(C)n3ccnc3)C12 C1(C(=O)NCC(CC=C)(C)C)CC(F)CCN1C(c1ccccc1O)=O C1(NC(C(CSC)OC)=O)CN(C(=O)C=Cc2ccc(Br)cc2)C(C)(C)C1 C(=O)(CCCCC(F)F)NC1(C2N(C(c3ccc(OC)cc3)=O)CCCC2)CC1 C1(NC(C(C)OCCCC)=O)CN(C(c2cc(C(F)F)cs2)=O)CC1CC c1(C(C(=O)NCC(COC)NC(=O)Cn2[nH]cnc2=N)C)cnn(C)c1 C(N(C)N(C)Cc1csc(CN(CC)CC2CC2)n1)C1(CC)CCCC1 C1(C(=O)NCC(CNC(c2ccc(COCCO)o2)=O)CO)(CO)CCOCC1 N1(C(COC)C)CCN(C(=O)C=Cc2ccccn2)C(=O)C1 C1(CNC(CS(CC)=O)=O)(OC)CCN(C(c2c(OC)ccnc2F)=O)CC1 C1(NC(COC2CN(C(C)=O)C2)=O)CC(C)(O)C1.c12nc(no1)C(=O)NC2 C1(CNC(C(C(=O)OC)(C)F)=O)CC2CCC(C1)N2C(C1(CC2CC2)CC1)=O Cc1ccc(C)n1CCC(N1CC(O)(CCNC(C2CCCCN2C)=O)C1)=O N1(C(c2ccc(C(F)(F)F)o2)=O)CCC(Oc2cncc(Cl)n2)CC1 CCCC(C(=O)N(C1CCC(F)(F)C1)C)c1ccc(Cl)cc1 C1(NC(c2ccc3nccn3c2)=O)CS(=O)(=O)C2CN(Cc3ccccc3)CC12 c1(C(N2CC(NC(c3cc(-c4ccncc4)no3)=O)C2)=O)cc(Cl)cc(Cl)c1Cl N1(C(C2N(c3cc(OC(C)C)ncn3)CC2)=O)CCN(C2CC2)C(=O)C1 c1(C(=O)NC2CN(C(C3(F)CC3)=O)CC2O)cccc(C(F)(F)F)c1Cl Nc1c(C(N2CC3(C(=O)O)CC2CCO3)=O)cc(F)cc1Br c1(C(=O)NCC2CC(NC(c3cc(C)sc3C)=O)CC2O)ccsc1S(C)(=O)=O N1(C(C2N(C(=O)COc3ccsc3)CCC2O)=O)CCOCC(C2CC2)C1 C1(C(=O)NC(CC)CCCO)C(C)OCCN1C(C1CCCC1O)=O C1(N(C2CC2)Cc2nc(CCCC)[nH]c2Cl)CCC(C)(C)CC1 c1(NC(C2CC(F)CN2Cc2cncs2)=O)cccc(OC(F)(F)F)c1Cl CC1CN(C(=O)Cc2ccccc2)CC1NC(C1C2CCCC12)=O c1(C(=O)NCC(CC)NC(c2ccccc2OC)=O)cnc(C)nc1OC C12(C(N(C(C)CNC(C3(F)C(C)(C)C3(C)C)=O)C)=O)CCC(N(C)C)(CC1)CC2 c1(OCC)cncc(C(N2CCC(OCCNC(c3ccnnc3C)=O)C2)=O)c1 N1(C(C=Cc2occ(C)n2)=O)CCC2C(NC(c3ncccc3Br)=O)CC12 CC12CC(C(=O)NC(C3CC(N(C)CC4(O)CCCN(C(N)=O)C4)C3)=O)(C1)C(C)(C)O2 c1(C(=O)NCC(CO)NC(c2ncc(C#N)cc2Cl)=O)cnc2[nH]c(O)nc2c1 Cc1csc(C(=O)NCC2CCCC2C(=O)NC(C)Cc2nn[nH]n2)c1C CC1(COC(=O)CSCC(=O)Nc2ccccc2)CC2C=CC1C2 c1(NC(CC2CN(C(Cc3cc(C)cc(C)c3)=O)C2)=O)ncc([N+](=O)[O-])cc1Cl Cc1c(C(N2CCC(OC3CN(C(=O)C(C(C)C)OC)C3)CC2)=O)ccn1C(C)C C1(c2n(CCC)nnn2)(NCc2nnc(C(C)C)s2)CCS(=O)(=O)CC1 CCC(CC)C(C)C(=O)NC1CCN(C(c2cc(C)ncc2Br)=O)C1(C)C N1(C(COCCN(C)C)=O)CCCOC(CNC(c2ccc(N)cc2F)=O)C1 N1(C(C(c2c(C)noc2C)C)=O)CCCN(C(c2nc(Cl)ccc2N)=O)CCC1 C1(NC(c2c(C)cc(CC)o2)=O)CCN(C(c2sc(C(C)C)nc2C)=O)CC1O Cc1snnc1C(=O)NC(C1CC1NC(C1(N2CCCC2)CCC1)=O)C c1(C(N(C2C(C)CCN(C(CCC=CC)=O)C2)C)=O)cccc2c(C)ccnc12 Cc1ccc(F)cc1C(=O)CC(=O)NCC1(C2CCCO2)CCC1 C=CC1(C(=O)NCC2(C)CCC(=O)N2)CCN(C(c2c[nH]nc2Cl)=O)C1 CN1CCN(C(CC2CCCO2)C(=O)Nc2ccccc2)CC1c1cccs1 Nc1cccc(CC(=O)NCC2CCCN2C(=O)CC2CCC(=O)N2)c1N c1(CC)noc(CC)c1CC(N1CC(C(C)NC(C2(C)CC(F)C2)=O)C1)=O N1(C(CCCC(C)C)=O)C2CCC1CC(NC(c1conc1C1CCC1)=O)C2 C(=O)(C(CC(C)C)CC(C)C)NC1C(CNC(C(C=C)(C)C)=O)CCC1 C12(C(=O)NC3CC(N(C(c4c(C)nc(C5CC5)[nH]4)=O)C)C3)CCCN1CCC2 CC1COCC(CC(=O)NCc2cc(C(=O)N(C)CCN3CCCC3=O)on2)O1 C1(CN(c2nnc(-c3cccc(O)n3)n2CCC#N)C)CCc2c[nH]nc2C1 c1(C(=O)NCC(=O)N(CCCCCNC(C(CC)C)=O)C)cccc(Cl)c1 C12(C(=O)NC3CCCC(NC(CNC(=O)OCC)=O)C3)CCCC(C)(C1)OC2 N1(C(C=CCCC)=O)CC(NC(C2(CC)CCOC2)=O)CC(C)C1 N1(C(c2c(OC)ccc(F)c2)=O)CC(NC(C2CCCN2C)=O)C2CCCCC12 c1(C(=O)NC(CNC(c2c(OCCC)cccn2)=O)C)ccc2ocnc2n1 c1(C(C(=O)NCC=C)N(C2CCOC2)C)ccc(Oc2ccc(F)cc2)nc1 C(=O)(C1=CCOCC1)N1C(CN(C)C(c2cnc(C(F)F)s2)=O)CCC1 N1(C(CC2CC(CC)OCC2)=O)CCCC2(NC(=O)C(F)C3CCOC3)CC2C1 C1(NC(CC2(C(C(C)C)O)CC2)=O)CCN(C(C2CC3CCC3C2)=O)CC1C c1(OC)cc(CC(=O)NC2CCCN(C(=O)C=C(Cl)Cl)CC2)cc(F)c1 c1(C(N2C(CN(C(=O)CC3COC(=O)C3)C)CCCC2)=O)cnc2ccnn2c1 c1(CN(C(C2CSCN2C(=O)C(C)n2cnnc2CC)=O)CC)ccc(C)c(C#N)c1 N1(C(CCSCCNC(c2c(CC)nn[nH]2)=O)=O)CCC(C)C(CO)C1 N1(C(CCNC(COC)=O)=O)CC2(COC(CNC(=O)Cc3cnsc3)C2)C1 Cc1ccc(C(=O)NC(C2CN(C(=O)Cn3cnc(Br)c3)C2)C)s1 C1(C(=O)NCC(=O)N(C)C2CC2)(CC)CCCN(C(C2CCCC(C)(C)C2)=O)C1 n1(CC(=O)N(C(CNC(CCC#C)=O)C)C)[nH]cc2c(=O)ncnc1-2 C1(NC(c2ncccc2O)=O)CN(C(c2cnn(C3CC3)c2)=O)CC12CC2 CC1(NC(=O)CCC2CCC(=O)N2)CCN(c2nnnn2-c2ccccc2)CC1 CC1(C)C(C(=O)NCC(c2cccnc2)N2CCOCC2)CC12CCN2 C1(NC(C(CC)C(C)C)=O)CC2(CCN(C(=O)C#CC3CCCO3)CC2)C1 c1(C2(C(=O)NCC(=O)NCCN(C)C(c3cn[nH]c3)=O)CC2)ccc(C#N)cc1 c1(C(N2CCOCC(C)(CNC(C(CC)(C)O)=O)C2)=O)ccc2cncn2c1C C=CC(C)(CC)C(=O)NC1CCC1NC(=O)Cc1cccc(N2CCOCC2)c1 N1(C(c2ccc(C(=O)NC)nc2)=O)CCN(C(c2cccc(C#N)c2)=O)C2CC12 N1(CCC)CCCC1C(N1CC(CNC(C2COCC2C(N)=O)=O)(OC)C1)=O C(=O)(C1=CCCOCC1)NCCC(C)N(C)C(c1cncc(CN(C)C)c1)=O CC1COc2c(C(N3CC4(CSC4)C3)=O)cccc21 c1(C(N2CC3C(NC(c4nc(CC)oc4)=O)C(C3)C2)=O)cccc2nnn(C)c12 c1(C(=O)NC(C)CN2CCN(C(=O)C=C(Cl)Cl)CC2)cnc2[nH]cncc1-2 c1(OC)c(CC(N2CCC(C(C)NC(=O)CCOC3COC3)C2)=O)cccc1F CCCCS(=O)(=O)Nc1cccnc1C(N1CCN(CCC)CC1)=O c1(C(N2CCN(C(c3n(CCCC)ncc3)=O)C(C)C2)=O)sc(=NCC)[nH]c1C C1(N(C(C2(NC(=O)OC(C)(C)C)C(=C)CC2)=O)C)COCCC1C c1(NC(C2(CNC(CCCCCCC)=O)CC2)=O)ccc2cccnc2c1 C(C(=O)NN1CCCC1C(N1CC(SC(F)F)C1)=O)N(CC)CC C(=O)(CCCCCCCCC1CC1)NCC(CN(C(C(C)(C)OCC)=O)C)C c1(NC(c2nnn(C)c2C)C(CC)C)ccc(OC)cc1 N1(C(C2(C)CC(=C)C2)=O)CCC(NC(=O)CC2(C#N)CCC2)C(C)C1 C#CC1(NC(C2CCC(CNC(=O)CS(=O)CC)CC2)=O)CCCC1 c1(OCC)cccc(CC(=O)NCCCN(C(=O)C(C)CSC(F)(F)F)C)c1 C1(CC(=O)OC)CN(N2CC(c3cccc(OC)c3)CC2C)CC2(CCC2)O1 O=C1CCCCC(C(N2CCCN(C(C3CCC(F)(F)C3)=O)CC2)=O)N1 C1(C)(CC)CN(C(c2cccc(OC3CC3)c2)C(=O)NC2COC2)CCO1 CC1(C)CC(CO)CCN1C(=O)CC(O)CNC(=O)CCc1cccnc1 CS(=O)C=CC(=O)N1CC(NC(C2(CO)CC(F)(F)C2)=O)C(CC2CC2)C1 c1(CSCC(=O)NCCNC(CN(C2CC3CCC2C3)C)=O)cccc(Cl)c1 C(=O)(CC1CCOc2ccccc21)N1CC(O)CC(NC(CN(C)C(N)=O)=O)C1 C(=O)(CC(O)CC)N(CCC(=O)N(C1CCN(C)C1)C)CC=C N1(C(c2cn(CC=C)nc2)=O)CCC(NC(=O)C(CCC)=CCC)CC1C c1(NCc2ccnc(C)n2)[nH]c(=NC2CCCN3CCCCC23)nc2sccc12 N1(C(CCC=C)=O)CCC2(CC1)COC(CNC(=O)C(CCC)NC(C)=O)C2 CCCC(C#N)C(=O)N(CC(CO)(CO)NC(c1ccnc(N(C)C)c1)=O)C N1(C(c2n(CC)nc(C)c2)=O)CC2CCC2(NC(c2ccoc2Cl)=O)C1 C(=O)(C(CC(C)C)N1CCCCC1=O)NC1C(NC(C2(SCC)CC2)=O)COC1 n1(CCC)nnnc1C(C)(CCOC(C)(C)C)NCCC(Cl)Cl c1(C(N2CCN(C(=O)Nc3cc(Cl)ccc3Cl)CC2)=O)cc(F)cc(F)c1F c1(C(=O)NCC2(F)CCN(C(C(CN(CC)CC)F)=O)C2)ccc2nn[nH]c2c1 N1(C(c2cc(C(C)C)[nH]n2)=O)CCN(C(=O)C(O)Cc2cnc[nH]2)CC1C C(=O)(CC(C)(C)C)NC(C(C)C)C.C12CCN(CC1)C(=O)C1CC1C(=O)N2 CC(C)C(CN(C(=O)Cc1ccn(C)c1)C1CC1)C(=O)N1CC(C)C(C)C1C c1(C(CC)NC(=O)CCCOC(=O)C(CCN)OC)ccc(Cl)c(Cl)c1 C1(C(C)NC(c2ccno2)=O)CCN(C(c2ccc(OCCO)cc2)=O)CC1 C(=O)(C(CCCC=C)NC(=O)C(C1CCC1)OCC)NCC(CC#C)(C)CO c1(C(=O)NCC2N(c3ccnc(C(C)(C)C)n3)CCCC2)c(F)cc(Cl)cc1Cl C1(NC(COCCCC)=O)CN(C(=O)C(C)SCC)CC1C(F)(F)F N1(C(CC2CCCC(C)O2)=O)CC2(CC(NC(C3CCC(=O)O3)=O)C2)C1 C1(CCC(=O)NC(COCC)C(C)C)CCCCN(C(=O)C(C)C)C1 C=CCC(CC(=O)NC1CCOC(C(C)C)C1)NC(=O)Cc1ncccc1C c1(CC(=O)NC2C(CNC(C(COC)C)=O)CCC2)ccc2c(c1)CCN2C c1(-c2cccc(C#N)c2)n[nH]c2c1CN(Cc1ncco1)CC2 C(=O)(C1=CC2(CN(C(c3cncc(C)c3)=O)C2)OC1)NCCOCC(=O)NC N12CC3C(C3C1)CN(C)C2=O.C(C(C)(C)N1CCCC1)N(C(C)C)CCO C1(OCC)COCC1N=c1[nH]c(=NC(C)Cc2ccc(Cl)cc2)[nH]c2c1CSC2 CCN=c1cc(-c2nc(Cc3ccc(C)cc3)n(-c3ccn(CC)n3)n2)cc[nH]1 CC(C)C(C(=O)NCC(CNC(C12CCCC1(C(N)=O)C2)=O)C(F)(F)F)C(C)C C1(CNC(C(CCC)C)=O)CCCC2(CN(C(=O)CC3(COC)CCCC3)C2)O1 C=CCCC(C(=O)N1CCOCC1CN(C)C)NC(=O)C=CCF C1(NCCCN(CCCN)OCC)C(=O)N(C)CCC1C CC1CC(N=c2c([N+](=O)[O-])c[nH]c3ccc(F)cc23)CCN1C(C1CCC1)=O c1(-n2cc(C(CCC)NC(c3ccccc3C(F)F)=O)nn2)cc(F)ccc1C C1(C(N2CC(CC(=O)Nc3c(OC)nn(C)c3)(OC)C2)=O)CC2CC(=O)C1O2 Cc1cc(C(=O)NCC(=O)NCCN(C)C(c2cc(C#N)c[nH]2)=O)n(C)n1 N1(C(C(COCC)C)=O)CC2CCC2(CNC(=O)CC2(CN(C)C)CCC2)C1 N1(C(c2nc(CC)sc2)=O)CCN(C(c2ncccc2C(C)=O)=O)CC1C N1(C(CC(C=C)C)=O)CCC(NC(=O)C2=CCOC2)C1(C)C C1(CC)CC(C)N(c2nnc(-c3ccc(C)s3)n2CCS(=O)(=O)CC)C1 CC(F)(C(=O)NCCC1CN(C(=O)CCCc2ccccn2)C1)C(F)(F)F c1(C(=O)NCC(CCCC)NC(c2cc3scnc3[nH]2)=O)n[nH]c2c1CC1CC21 C1(NC(=O)Nc2scc(COC)n2)CCS(=O)(=O)C(C)C1 C1(C(=O)NCCC2N(C(c3c(C)nc(C)[nH]3)=O)CCSC2)OCC2CCCCC12 N1(C(CCCNC(C)=O)=O)CC(OC)CC(NC(c2cc(C)sc2C)=O)C1 Cc1csc(C(=O)NC2CCC2NC(C23C=CC(CC2)C3)=O)c1Cl CC1CN(C(=O)Cc2ccc(O)nc2)CCN1C(c1coc(Cl)n1)=O CC1(C)OC(=O)C(CC(=O)NC2CC(NC(=O)CSc3nc[nH]n3)C2)O1 C12(c3n(CC(=C)C)c(N(CCCCC)C)nn3)CCCCC=C1OCC2 c1(C(=O)NCC(C2CC2)NC(C2N(C)CC2)=O)cc(Br)cs1 c1(C(C)(C)OC)nc(C)c(C(=O)NC(CNC(C2CCSCC2)=O)C2CC2)s1 c1(C(=O)NC(CC)CNC(c2cccnn2)=O)ccc2nc[nH]c2c1F N1(C(C(C2CCC2)OCC)=O)CC2CC2(NC(C2CN(CC(C)C)C2)=O)C1 N1(CC(CN(CC#C)C(=O)OC(C)(C)C)O)CCN(c2ccccc2)CC1 N1(CC)CCCC(C(=O)NC(C)(CO)C(=O)N(CC(C2CCCC2)O)C)C1 C(=O)(C1=COCCO1)N1CC(C(C)NC(=O)C2=C(Cl)CC2)C1 c1(N(C)C)cccc(-n2ncc(-c3noc(-c4csc(S)n4)n3)c2N)c1 N1(C(c2csc(Cl)n2)=O)CCOC(C2CN(C(=O)C=CC=C(Cl)Cl)C2)C1 C1(CC#C)(C(=O)NC(C)C(F)(F)F)CCN(C(=O)C(C)C(C)C)C1 C=CCCCCC(=O)N1CCCC(NC(C2CCCC2F)=O)CC1 C1(NC(c2n(CC(C)C)ncc2)=O)CN(C(C2CC3CCC2O3)=O)CC2(CC2)C1 C(=O)(CC(C)C(C)(C)NC(=O)CN1CCC(C)C1)NCc1cccc(OC)c1 C(C(COC)C(=O)N1CC(F)CC1Cn1cc(C2OCCO2)nn1)OC C(=O)(N=c1cc(C)n(C)[nH]1)C1(CNC(CC(=O)NCC#C)=O)CCCCC1 Cc1cccc(CC(N2CCC(NC(=O)CC3CCCCC3F)CC2)=O)c1F C12(NC(C(C)NC(C3CN(C(N)=O)C3)=O)=O)CCC(C(F)(F)F)(CC1)C2 C1(O)(CNC(C2C3(CC3)C23CC3)=O)CCN(C(C2CCOC2=O)=O)CC1 C1(C#N)(NC(CN(C(c2cn(CCC)nc2)=O)CCOC)=O)CCOCC1 C(CN=[N+]=[N-])(C(=O)NC(C)C(=O)N(C)C)NC(CSCCOC)=O C(=O)(C(CNC(C1(n2cnnn2)CC1)=O)C(C)C)NC1(COC)CC1 CC(C(CO)NC(C1(C2CCCCO2)CC1)=O)NC(=O)CC(C)c1ccncc1 C12(NC(c3ccc(F)cn3)=O)CCCCC1CN(C(C1CC3CCC1CC3)=O)C2 c1(C(=O)OCC)sc(C(=O)NCCC(O)CNC(C2CC2F)=O)c2c1CCCC2 C1(NC(c2scc(C)c2C)=O)CN(C(C23CCCC2(C(N)=O)C3)=O)CC1(C)C c1(C(N(CCNC(C2(F)C(C)C2)=O)C2CC2)=O)cccnc1OC(F)F n1(C(C)C)ncc(C(=O)NCC2C3CN(C(=O)Cc4conc4C)CC23)c1N c1(OC)c(F)cc(F)c(NCC(C)CNC(=O)C(F)(F)C2CC2)c1[N+](=O)[O-] C(N=c1cc(SC2CCCC2)nc[nH]1)C1CS(=O)(=O)CC1O C1(NC(CCCOCCOC)=O)CN(C(c2csc(Cl)c2)=O)CC1n1ccnn1 C12(CCNC(CC3(OC)CCC3)=O)CCC1CN(C(c1cc(Br)co1)=O)C2 c1(C(N(CC(C)NC(c2cc[nH]c2)=O)C)=O)ccnc(OCCN(C)C)c1 C1(CNC(C2(CCC)CCC2)=O)CCN(C(=O)CCC=CBr)CC1C CS(=O)(=O)C1(C(N2CCCOC(CNC(c3c(O)cccc3O)=O)C2)=O)CCC1 c1(C(N(CC(CN(C(C(C)(CO)OC)=O)C)O)C)=O)cc(C)c2sccc2c1 c1(CC(=O)NCCN(C(C=CC=CC)=O)CC(C)O)nnc(O)s1 N1(C(c2c(C#C)c[nH]n2)=O)CCC(C=C)(C(N2CCCC(CC(N)=O)C2)=O)CC1 C=CC(CC)CC(=O)NC1CCN(C(=O)CNC(c2c(F)cccc2Cl)=O)C1 C(=O)(CCCN=[N+]=[N-])NC1(C(N(CC(C)C(F)(F)F)C)=O)CSC1 N1(C(c2ccc(OC)nn2)=O)CCC(C(=O)Nc2cnn(C3CC3)c2)C(O)C1 c1(C(=O)NCC(CNC(C(COC)(C)O)=O)C(F)(F)F)ccc(S(C)(=O)=O)cc1 CCCCC(CC)CC(=O)NC(C)(C)CN1CCC1.C1=CCNC1=O c1(-c2ccc(C(N3CCCCC3c3ccccc3)=O)c(O)c2)ccn2cnnc2c1 N1(C(=O)Nc2ncc(OC)s2)CC(C)SC(C)C1 N1(C(CC(CNC(C2CC=CC2)=O)OC)=O)CC2(CCC(=O)NC2)C1 c1(-c2cc(C(=O)NC3CCC(NC(=O)Cn4nccn4)C3)no2)cccc(F)c1 Cc1cccc(Cl)c1CC(=O)NCCC1CN(C(C2CCN(C)C2=O)=O)CCO1 C=C=CCC(=O)NC(C)CCNC(C1CCC(C(F)(F)F)C1)=O C#CC1(C(=O)NCC2CCCN2C(C2CC(N3CCCC3)C2)=O)CCC1 O=C(CC(O)COCc1ccccc1)NCC=CCNC(=O)Cc1cscc1F C=CCCCCCCC(=O)N1CCCC(C(=O)NCCC(C)CO)(CC)C1 c1(C(N2CC(F)(CNC(c3c(COC)ccs3)=O)C2)=O)cccc(Cl)c1Cl N1(C(Cc2cc(=N)[nH]cc2)=O)CC2CCN(C(=O)C3=CCSC3)CCC2C1 C(C(CC(C)C)NC(c1csnc1Br)=O)NC(C1(NC(C)=O)CCC1)=O C(=O)(CC(CNC(=O)C(C)(C)NC(C)=O)C1CCC1)N(N1CCCC1)CC C1(CC=C)(NC(=O)Cn2cccn2)CCN(C(C2CC2(F)F)=O)CC1 CC(C)CCC(O)C(=O)N1CCN(C(C2(CF)CCOCC2)=O)CC1CC1CC1 c1(NC2(c3n(CC)nnn3)CCC2)c(C)nn(-c2ccc(C)c(Cl)c2)c1C C(Cc1ccccc1)(CCNC(C1(Cl)CC1)=O)NC(c1cncnc1)=O Cc1nc(N2CCOCC(NC(=O)CS(=O)(=O)Cc3cccs3)C2)cc(Cl)n1 C1(COC)(CNC(C2(CO)CC2)=O)CCCN1c1nnc(-c2ccon2)s1 Cc1ccccc1-c1cn(C(C)CN(C(=O)CCN2CCCC2)C2CC2)nn1 CC(CCC(C)(C)C)C(=O)NC1(C(=O)NC2CCn3cncc3C2)CC(F)C1 N1(C(CCN(C)CCO)=O)CCCC(C2CCN(C(=O)C(C)(C)CN(C)C)C2)C1 Cn1nc(Br)c2ccc(C(N3CC(F)CC3C(N3CCCC3C(N)=O)=O)=O)cc12 N1(C(c2c(C)c(Cl)cnc2)=O)CC2CN(C(=O)CC(O)CCN(C)C)CC2(C)C1 Cn1ccc2ccc(C(N3CCCC3CC(=O)NCc3cncc(O)c3)=O)cc12 C1(C(=O)NCCCN(C(=O)CC2CCN(C)C2=O)CC)CCc2nc[nH]c2C1 CCC(CNC(C1(F)CCCN(C(=O)C(n2nccc2C)C)C1)=O)C(C)(F)F C(=O)(CCCCCO)NCCCCC(C)NC(C=CC)=O c1(C)ccc(CO)c(F)c1.N1(C(C)=O)CCCC1CNC(C1CCC(N(C)C)C1)=O C#CCC(C)C(=O)N1CCCC(N(C(=O)CCc2cnoc2)CCF)C1 C1(NC(=O)C=CC2CCOC2)CCCN(C(=O)CCc2ccco2)CCC1 C(CCCC(C)(C)C(=O)NNC(=O)C1CCCCO1)NC(C(C)C(C)(C)C)=O c1(C(=O)NCC2OCCCN(C(c3ncc(C)cn3)=O)C2)cnc(O)n(C)c1=O C1(NC(C(CC)(C)C)=O)CC(F)(F)CC1NC(C1CCCN1c1cnccn1)=O C1(NC2(c3nnnn3CCCSC)CC(CCCC)C2)CC(O)C(O)C1 N1(C(C(CCC)N(C)C)=O)CC2CC(C1)N(C(c1nn(CC)nc1C)=O)C2 N1(C(C(C)=CC)=O)CCN(C(=O)CC(O)C2CCCC2)CC1CCO c1(CC)cc(C(N2CCCC(CC(N3CCC3C(=O)NC)=O)C2)=O)ncn1 O=S1(=O)CCc2cc(CNC(=NCCCC3CC3(F)F)NC3CCCC3)ccc21 c1(OC)cccc(O)c1C(N1CCN(C(c2cc(C)c(C)o2)=O)C(C(C)C)C1)=O Cc1cc(O)cc(Cl)c1C(=O)NC1CCCCC1CNC(=O)CCCN(C)C N1(C(CCOCC)=O)CC(NC(c2cnc(N(C)C)s2)=O)CC(C)C1 c1(C(N2CCN(c3ncnc(Cl)n3)CC2)=O)cc(F)ccc1C1CC1 C(=O)(C(F)CC(C)(C)C)NC1CC(CCNC(c2c(C)n(C)nn2)=O)C1 Cc1nnc2ccc(C(N3CC(NC(C4CC5(CC5)CO4)=O)C(C)C3)=O)cn12 CC1CNCC(N(C(=O)CC(c2ccc(Cl)cc2)O)C(C2CCCCC2)=O)O1 CCCCCC(C)(CC)C(=O)N1CC2(CC(NC(c3sccc3Cl)=O)C2)C1 C1(N2CC2)C2CC3C(C2)C13.c1(C2(C(=O)O)CC2)c[nH]c(C(F)(F)F)c1 C1(NC(c2nccc(OC)c2OC)=O)C(C)CN(C(c2cnc(Cl)s2)=O)CC1C C1(NC(C(c2ccc(C)cc2)O)C)CC(C)(C)OC(C)(C)C1 N1(C(CC2(C)CC2(F)F)=O)CC(NC(c2ccc(Cl)c(O)c2)=O)CC12CCC2 c1(-c2cnc(SCc3ccc(OC)cc3)o2)ccc(C)cc1C c1(C(N2CCC(N(C(CCN(C(C)=O)C)=O)C)C2)=O)ccc(-n2cnnn2)cn1 c1(COC)nc(=NC(=O)c2ccc(C(C)(C)S(C)(=O)=O)cc2)o[nH]1 C(=O)(C1=CCCN(C(=O)CCC2CCCO2)C1)N(C1CCN(C)C1)CC c1(OC)ccc(Cl)c(CC(=O)NC2CCC(Nc3cncc(C#N)n3)CC2)c1F n1(C(C)C)ncc2c(NC(c3cnn(C)c3)C)[nH]c(=NC3CC=CC3)nc12 N1(C(CC(C)F)=O)CCc2c(c(CNC(C3CC3F)=O)nn2C)C1 C1(C(=O)NCCC2(O)CCN(C(CNC(C)=O)=O)C2)CCc2nnc(O)n2C1 c1(C(N2C(CNC(c3cnc(C)nc3)=O)CCCC2)=O)ccc2occc2c1O c1(C(=O)NC2CC(CNC(=O)C(C3CCCO3)C3CC3)C2)cccn2nncc12 C(=O)(CC1CC(C(C)C)c2ccccc21)N1CCC(NC(CCC#C)=O)C(O)C1 c1(C(=O)OC)ccc2nc(NC(c3ccc(Cl)cc3Cl)=O)[nH]c2c1 Nc1ccc2nc(N3CCCC(CO)(NC(=O)C=Cc4ccccn4)C3)sc2c1 c1(C(=O)NC2CCN(C(C3(COCC)CC(F)(F)C3)=O)C2)cc(S(N)(=O)=O)c[nH]1 N1(C(C=Cc2cn(C)nc2)=O)CCC(NC(=O)C(=O)NCC(F)F)C2(CCC2)C1 C(=O)(C(C)CC(F)F)NC(C(=O)NCc1ccc(C)cc1)C1CCC1 N(C1c2cc(F)ccc2CC1C)CC(C)=CC=C c1(OC)ccc(C(=O)NC2CN(C(C3(C#N)CC(=O)C3)=O)CCC2C)c(C)c1 N1(C(C(CC)(C)O)=O)CCC(O)(CN(C)C(C2CN(C(C)=O)CCO2)=O)CC1 N1(C(C2CC2NC(c2cnncc2C(F)(F)F)=O)=O)C2CCC1C(C(F)(F)F)C2 CCCCC(C(N)=O)NC(C1CCCN(C(=O)Nc2c(C)cccc2Cl)CC1)=O c1(C(N2CC(C(=O)Nc3c(C)c(Br)c(Cl)nc3)C2)=O)c(F)ccc2[nH]ccc12 c1(C(=O)NCC2C(NC(C(C)(C)c3ccccn3)=O)CCC2)cnc2n1CCS2 N1(C(CC=C(C)C)=O)CCC(NC(c2nccc3nn[nH]c23)=O)CC(C)(C)C1 C1(NC(CNC(C(COC)(F)F)=O)=O)COCC1C1CC1 CC(C)(CC(=O)N1CC(C2(NC(=O)CCc3ccc(F)nc3)CC2)C1)C(F)F c1(C(N(CC(CNC(C2C(C(C)C)OCC2)=O)O)C)=O)cnc2c[nH]nc2c1 c1(C(N2CC(NC(C3C(C)C3)=O)C2)=O)cc2sc(N(C)C)nc2s1 C12(C(=O)NC(CC)CN(C(C3CC3c3ccn(C)n3)=O)CC)CCC(CC1O)C2 Cc1cc(C(N2CCC(C)C2CNC(c2cc[nH]c3nccc2-3)=O)=O)c(O)cc1F S(=O)(=O)(c1ccc(NCCC(C)F)cc1Cl)NCCC1(COC)CC1 c1(-n2c(CSCCC(F)(F)F)nc(C(C)OC)n2)cc(C)nc(C)c1 CN1CC(C(=O)NCC2(F)CC(NC(C3CC(=O)N(CC4CC4)C3)=O)C2)CC1=O C1(NC(c2c(SC)ccs2)=O)CN(C(=O)C(O)CC(F)F)Cc2ccnn2C1 N1(C(C2CC(CC)C2)=O)CC(C)(C)OCC1CNC(=O)CS(=O)(=O)NC c1(NC(=O)Nc2cccc(CO)n2)ccc([N+](=O)[O-])cc1 CC(C(=O)NOCC1(C)CCC1)NC(=O)CC12CCC(CC1)C2 c1(C)nc(-c2ccoc2)nn1C1CCSCC1.Cc1ccsc1-n1ccnc1C Cc1c(Br)c(C(=O)N(C)CC2(O)CCN(C(=O)C3=CC(C)(C)C3)C2)nn1C C(=O)(C1CCCc2ncc(C)n21)NC(C1CCCC1)CNC(CNC(C)=O)=O c1(C(=O)NC2(CCNC(c3ccsc3Br)=O)CCC2)c[nH]c(=O)cn1 c1(C(=O)NCC2C(NC(c3ncn(CC)c3)=O)C2)ccc(=O)n2c1CCCC2 N1(C(C(C)N(CC)CC)=O)CCC(C(C)(C)C(=O)NC(C)C)C1.C1CCC1 C1(NC(C(C)(C)N(CC(C)(C)C)C)=O)CC2(CCN(CNC(=O)OC(C)(C)C)C2)CO1 C1(C(N2CC(C#N)C(NC(C3(Br)CCC3)=O)C2)=O)Cc2ccccc2O1 Cc1ccc(F)c(C(N2CCSCC2C(=O)NC2CC(c3ncc[nH]3)C2)=O)n1 N1(C(C2(CC=C)CCC2)=O)C2CCC1CC(CNC(C1C=CCC1)=O)C2 c1(OC)c(C(=O)NC2CN(C(c3ccoc3Cl)=O)CCC2C)nc(O)nc1O C(=O)(C(C)(C)C1=CCN(C(c2ccc(OC)o2)=O)C1)N1C(C#C)CCC1 c1(C(=O)NCCC2(NC(c3cnsn3)=O)CCC2)ncc(C(F)F)s1 C1(CC)CN(C(=O)C(N2CC(O)CC2CN)=O)CC1c1cnn(C)c1 C(=O)(C(C)C(=O)N1CCCC1CN(C)C(c1csc(-c2cnccn2)n1)=O)OC c1(N(C)Cc2ccc(OCCC)cc2)cccc(S(=O)(=O)N2CCSCC2C)n1 C(C)(CCCN=c1[nH]nc(C2CC2)s1)NC(C(C)Sc1ccccc1F)=O Cc1cc(O)cc(C)c1C(=O)NCC1CCN(C(=O)Cc2nc[nH]n2)C1(C)C N1(C(C(C)S(C)(=O)=O)=O)CCC2C(CCCN2C(=O)CCCC(N)=O)C1 C1(CC(N2CCC(OCC)C2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 C1(C(N(C2CCOC2)CC)=O)CCCN(C(=O)CCc2ccccn2)CC1 N1(C(C=CCC(C)(C)NC(C(C(C)C)C2CCC2)=O)=O)CC(O)CCC1C c1(C(=O)NC2CN(C(C(C(C)C)CN(C)C)=O)C2)noc2c1CC(C)(C)CC2 C(=O)(C(C)(C)C1=CCN(C(=O)C2=C(Cl)CCCC2)C1)N1CC(C)(C)C(O)C1 C1(C#N)(CNC(=O)C=CCNC(=O)C(F)=CC2CC2)CCC1 C(=O)(C1=Cc2ccccc2OC1)N1C2CCC(NC(c3cnc(Cl)[nH]3)=O)(CC2)C1 C(CC(=O)NCc1cc(O)ccc1F)(C(F)F)NC(CC(C)F)=O C1(CC)CCCCC1NC(c1c(CNC(=O)C(=Cc2cn[nH]c2)C)cnn1C)=O C(=O)(C1=CCC(C)CC1)NC1CCN(C(c2ccc(C)s2)=O)C1(C)C n1(CCC)nnnc1C(c1cscc1C)NCCC(F)(F)F c1(C(=O)NCC2C(NC(c3cnn(C)c3Cl)=O)CCC2)cccc(F)c1Cl C(C(C)(C(C)C)NC(c1nc(Br)c(C)s1)=O)NC(C1(C#C)CC1)=O C1(N(C(C(N2CCCCCC2)C)=O)C)CCN(C(=O)Cn2nccn2)CC12CC2 N1(C(C2(C)CC(=C)C2)=O)CCC2CCCC(C1)N2C(c1cc(C(C)=O)cs1)=O C1(C)(C(N2CCC(CCNC(c3cc(COC)no3)=O)CC2)=O)CCC(O)CC1 C1(C(=O)NC(c2nc(C)sc2)C)C2CCN(C(c3cc4n(n3)CCO4)=O)CC12 C1(C(N(CC(CC)C)C)=O)C(O)CCN1C(=O)COCC1CC1 C1(C(C(=O)NC2CC(CNC(c3ccc(SC(F)(F)F)o3)=O)C2)O)CCCCCC1 c1(C(=O)NC2CC(C)(NC(c3cnc(C4CC4)s3)=O)C2)cncc2cccnc12 C1(NC(C(C2CCC2)OC)=O)CCN(C(c2csnc2C)=O)C1C C1(C(N2CCC(N(c3ccncn3)C)C2)=O)CCC(F)CC1 Cc1nc(C)c(C(=O)N(C)CC2(O)CCN(C(c3csc(C(F)F)n3)=O)C2)o1 C(C)(CCCCN=c1[nH]nc(-c2ccccc2)s1)NC(C1C(OC)CCC1)=O N1(C(c2c(C#C)c[nH]n2)=O)CC2CCC1C1CN(C(=O)CCC3CCCO3)CC21 N1(C(C2CCCC2(F)F)=O)CCn2nccc21 CC1CN2CC(O1)C(=O)N1CCC(CC1)OC2=O.C(C#N)(C(N)=O)NC(=O)C1CC1 CC(C)(CNC(=O)CCc1ccsc1)CNC(=O)CC1(N2CCCC2)CC1 C1(C(N2CCCC(CC)(NC(c3csc(=N)[nH]3)=O)C2)=O)CC2(C1)CC(C)(C)C2 O=C(CS(=O)(=O)c1ccc(C)c(Cl)c1)OCC1COC(c2ccccc2)O1 N1(C(c2ccc(COC)o2)=O)CCCC(CN(C(=O)CCC(=O)OC)C)C1 C(CC1CCC1)(C(=O)N(CCC(=O)NC1CC2CC2C1)CCCO)OC N1(C(C(c2cc(C)sc2)(C)C)=O)CC2CC1CN2C(=O)OC(C)(C)C CCCC(C)(C)CC(=O)N1CCCC1Cn1cc(CC2CCCCO2)nn1 C(=O)(C=C1SCC(=O)N1C)NCC1CCCN(C(C2CC(C(=O)OC)C2)=O)C1 N1(C(CC(CC(=O)OC)C)=O)CCC2(C=C(C(=O)NOCC=CCl)C2)C1 C1(NC(c2ccc(CC)cn2)=O)CN(C(c2[nH]nnc2C2CC2)=O)CC1C1CC1 C1(CN(CC=C)C)CCN(N2CCCC2Cc2ccccc2)CC1 c1(C(=O)NCC2C(CNC(CCOCC#C)=O)C2)ncc(C(N)=O)cc1Cl c1(C(=O)OC)cnc2nc(NC(c3cccc(O)c3OC)=O)ccc2c1 c1(C(N(C)CC2CN(C(c3cnncc3O)=O)C2)=O)nc(O)[nH]c(=O)n1 C(=O)(C1CCNc2ccccc21)NC(CC(C)C)CNC(c1nccnc1N)=O C1(NC(Cc2nc(C)[nH]n2)=O)CN(C(C2CCCC(=O)N2)=O)CC1C C=CCCCC(=O)N1CCCC(N(C(=O)Cc2csc(C(=O)OC)c2)C)C1 c1(C(=O)NCCCC2N(C(c3cnn(CC)n3)=O)CCCC2)cccc(C)c1C c1(C(N2CCC(CNC(Cc3cc(C)no3)=O)C(O)C2)=O)ccc2nccn2n1 c1(C(C(N2CCC(NC(C=CCCC=C(C)C)=O)C2)=O)=O)ccc(F)cc1 CC1OC2(C(=O)NCCCC(C)NC(=O)COCC(C)(C)C)CC1C2 C1(C(NNC(c2c(OC)c(Br)ccc2)=O)=O)CCc2nccn2CC1 N1(C(CNS(C)(=O)=O)=O)Cc2ccccc2OC2(C1)CN(C(=O)CNC(N)=O)C2 N1(C(CS(CC)(=O)=O)=O)CC(N=c2[nH]c(Cl)ncc2C2CC2)C1 c1(C(C)C(=O)NC2(CN(C(=O)CCS(C)(=O)=O)C)CC2)cc2ccccc2s1 C(=O)(CC1=CCCCC1)NC1C(C)CCN(C(c2c(C)oc(C)c2Br)=O)C1 N1(C(c2c(OCC)scc2)=O)CC2CCC(Nc3cc(C)ncn3)C2C1 C(=O)(C1=NN(CC)C(=O)CC1)NC1C2CN(C(C(C=C)C)=O)CC21 C12(C(=O)N(C)C)CCCN1C2=O.C1(CC)CCN(C(=O)CCO)CC1 C12(C(=O)NCC(C(C)(C)C)NC(C3CCN(C)C3=O)=O)C3CCC(CC13)C2(F)F c1(C(N2CC(SC)C(n3cc(CC4(O)CCC4)nn3)C2)=O)cc(C)c(F)cc1Br C(=O)(CCCCO)NCC(=O)NCCCCNC(CCc1cn(C)nc1)=O C1(C(=O)NC(C(C)C)CNC(=O)C(C)(O)c2ccccc2)CCCCC1(F)F N1(CC(N2CCN(C(CCOC)=O)CC2CF)=O)CCCCCCC1=O C(C(C)(C)N(C)C)SC.C12(CC1)C(=O)N(CC(=O)O)C2 N1(C(Cc2cc(C)no2)=O)CCC(F)(CNC(=O)CC2CCC3CC23)CC1 N1(C(C(CCSC)O)=O)C2CCC(C2)C1CNC(=O)CSc1cccc(Cl)c1 c1(NC(c2nnnn2C(C)C)CCOCC=C)ccsc1C c1(C(=O)NCc2c(CNC(=O)CC(F)F)cccc2)cccc(=S)n1O C1(CNC(C2OCCN(C)C2)=O)CCC12CCN(C(=O)CCC#N)CC2 C1(C)(C(=O)NCCOC2CN(C(COCC(=C)C)=O)C2)CC(C#N)C1 N1(C(c2n(C)cc(I)c2)=O)CCC(NC(=O)C=CC(C)(C)C)C1(C)C N1(CC#N)CCCN(C(c2c(O)cccc2O)=O)CC1 c1(NC(=O)Nc2ncc(NC(c3ccc(Cl)cc3)=O)s2)ccc(Cl)cc1Cl C1(CC(C)(C)C)CN(C(=O)COc2ccsn2)CC1NC(C12COCC(C1)C2)=O N1(C(CCC2CCCN(C(c3cnn(C)c3N)=O)C2)=O)Cc2ccncc2C1 C(=O)(C(C(C)C)C(C)C)Oc1c(OCc2cn(CCOC)nn2)cccc1Cl N1(C(C2CC(C)(NC(C3CC(C)(O)C3)=O)C2)=O)CC(CO)C(O)C1 c1(-c2n(CCC=C)nc(-c3cccc(Br)c3)n2)cc2cnccc2[nH]1 C1(OC)CN(C(=O)C=CC2CCOC2)CCC1NC(c1cccc(OC)c1C)=O CN1CCC(N(C(=O)C(C2CC2)N(C(=O)Cc2ccc(F)cc2)C)C2CC2)C1=O c1(CCC(N2CC(CNC(C=C(C)C(C)(C)C)=O)C2)=O)ccc(N2CCC2)cc1 c1(C(N2CC(CNC(c3csnn3)=O)C(O)C2)=O)cc(F)cc2cnccc12 C1(N(C(=O)NC(C)C(C)n2cccn2)C)CCC(C)(C)C1 N1(C(C(CC=C)CC)=O)CCCC(C)(C)C1CNC(c1ccc(F)o1)=O c1(C(=O)NC2CN(C(c3cc(COC)[nH]n3)=O)C2)ccccc1CC#N c1(NCCOCC)ncc(C)cc1S(=O)(=O)NCc1cc(F)ccc1C c1(C(=O)NCC(C)(C)NC(C(C(C)C)c2cnc(C)s2)=O)nccn2nccc12 C1(C(=O)NCc2ccc(C)o2)CC=CCN1C(=O)CCc1ccccc1 CCCC(C(=O)OC)C(=O)NCC1CC(F)CN1C(=O)CC1CCC(=O)NC1=O C#CCCC(C(=O)NC1CC(=O)N(C)C1=O)NC(=O)CC1CCCCCC1 C(C1CCOCC1)=CC(=O)N(C(C(=O)N(C1CCN(CC)C1)C)C)C1CC1 CCC(CN(C)C)C(=O)N1CC(NC(c2sccc2C)=O)CC1C CCC(C)CC(C(=O)NCCc1cnco1)NC(c1c[nH]cc1C)=O C(=O)(C1Cc2ccccc21)N1C(C)CN(C(c2cccn3ccnc23)=O)CC1 CC1CCC(F)(C(=O)NC2CC(F)CN(C(c3ncc(F)cc3F)=O)C2)CC1 C1(C(=O)NC(CC)CNC(C2CCC(C)(C)CO2)=O)CCC2(CCCC2)CC1 C(C(C(=O)N(C(C)CNC(c1cc(C2CCCCC2)[nH]n1)=O)C)N(C)C)OC C(=O)(C(C)(C)CCC)NC1(CCNC(C2(CC#C)CCCCC2)=O)CCC1 C1(C(C(=O)NCCC#N)N(CCOC)C(C)C2CC2)CCC(C)C1 N1(C(C(CC=C)(C)C)=O)Cc2occ(C(N3CC(=O)NC(CC)C3)=O)c2C1 c1(N(C(=O)NCC(c2ccc(OCCN(C)C)cc2)NC)C)ccccc1Cl c1(C(N(C(C=C)C(N2CCCC(c3n[nH]c(C)n3)C2)=O)C)=O)sc(OC)nc1C N1(C(Cc2c(C)non2)=O)CCC2(CCCN(C(=O)CCC3CC3C)C2)CC1 C1(C(N2CCC(C(=O)OC)(CF)C2)C(=O)NCC(=C)C)CCCOCC1 c1(OC)c(C(=O)N(CCNC(=O)CN(C)CCO)C(C)C)cc(F)cc1F c1(COC(C2C(C)(C)CC2)=O)nc2ccc(F)cc2s1 c1(OC)ccnc(O)c1C(=O)NC1CCC(N(C)C(c2nccn2C)=O)C1 C1(CNC(c2ccc(COC)c(F)c2)=O)CCCCN(C(=O)CSC(C)C)CC1 c1(N2CCC(c3ccc(C)cc3)C2)nn2cc(C)nc2s1 c1(CN2C(c3c(C)ccc(OC)c3)CC2)cc([N+](=O)[O-])ccc1OC(C)C C1(NC(C2ON=C(CC)C2)=O)CCN(C(c2cnc(C3CC3)nc2O)=O)CC1C C1(C(N2CCC(CSC3CC3)C2)=O)CC(O)CN1C(c1cnn(C2CCCC2)c1)=O N1(C(C(COC)C)=O)CCCC(O)(CN(C)C(c2cc(SC)n(C)n2)=O)C1 c1(C(=O)NCC2(O)CCCN(C(c3ccccn3)=O)C2)cc2cc(F)ccc2o1 C1(C(N(C)CC#N)=O)CCCC(NC(c2ccccc2F)=O)C1 CC1CCC(C(=O)NCC(CC)NC(C2CCCCN2S(C)(=O)=O)=O)CC1C c1(NC(C(=O)N(CCC)CCNC(c2csc(C)n2)=O)=O)ccc(C)c(C)c1 N1(C(C2C(C)C2)=O)CCCC2(CCCN2C(=O)C(c2ccc(Cl)cc2)O)C1 N1(C(C)C(N)=O)CCC(C)(NC(=O)CC2C=CCC2)C1 N1(C(CC2CN(C(C3(CC)CC3)=O)C2)=O)CCc2c(O)noc2C1 C(=O)(C1=CC2(CCN(C(=O)C(CO)C(F)(F)F)C2)C1)N(CC(C1CCCC1)O)C N1(CC)CCCCC1C(=O)NCC1CC(NC(=O)C2=CCOC2)C1 N1(C(C#CC(OCC)OCC)=O)CCN(C(=O)Cc2ccc(C)o2)C2CCCC12 CC(CNCc1cn(-c2ccccc2)nc1C(C)(C)C)S(N)(=O)=O c1(CC(=O)NCC(CNC(CN(c2ccccc2)C)=O)O)ccccc1CO c1(C(N2CC(CC=C)(NC(=O)Cc3cnns3)C2)=O)cc(N)cnc1C c1(CCC(=O)NC(CNC(C2CCC(COC)C2)=O)(C)C2CC2)cnn(C)c1C C1(C(=O)NCCN(CCOC)C(C2CCC3CC3C2)=O)(COC)CC(F)(F)C1 c1(N2CCC(N(C)C(c3ccc([N+](=O)[O-])s3)=O)C2)nc(Cl)nc2nc(Cl)n(C)c12 C(=O)(CC(O)CCCC)NC(C(N1CC2(CC(=C)C2)C1)=O)CCC N1(C(c2cc(C)ncc2C)=O)CC(F)(F)CC1(C)CNC(=O)CCC1CC1(C)C C1(F)(CNC(C(Br)=C(C)C)=O)CC(NC(=O)CCc2ccccn2)C1 C1(C(N2CC(CC(CNC(c3c(CC)non3)=O)(C)C)C2)=O)CC1C1CC1C c1(CC(N2CCC(CCNC(C3(CCC)CC3)=O)CC2)=O)ccc(F)c(OC)c1 N1(C(C(C(C)C)SC)=O)CCCN(C(c2ccc(C(C)=O)c(F)c2)=O)CCC1 c1(C(c2nnnn2C)NCC2(C=C)CCOCC2)cccc2ccsc12 n1(CC(N2C(C)(C(C)(F)F)CC2)=O)cc(NC(=O)Oc2ccccc2)nn1 C1(C(c2nnnn2C2CCOC2)NCc2nc(C)c(C)o2)(OC)CCCCCC1 C1(C(=O)O)C(C2CC2)CCN1C(C1CC=CC(n2cc(CCNC=O)nn2)C1)=O C1(C(=O)NCCC2OCCN(C(c3c(COC)cco3)=O)C2)CCCCC1(F)F C1(NC(CCCSC)=O)CCC(C)(CNC(c2c[nH]nc2C(C)(C)C)=O)C1 c1(C(N2CCCC(C(=O)NCCC#C)C2)=O)nc2ccccc2nc1C c1(C(N2CC(C3N(C(CC(C)C4CC4)=O)CCC3)(O)C2)=O)cc(Br)n(C)c1 C1(CNC(c2ccc(-c3ncon3)cc2)=O)CCCN(C(C2CCCOC2)=O)C1 c1(C(N2CC(NC(c3c(C)ccnc3)=O)C(CO)CC2)=O)cc(C)c(Cl)c(C)c1 c1(C(N2CC(C(C)NC(C3C(CCC)CCC3)=O)C2)=O)c(C)nc2sc(C)cn12 C1(NC(c2cccnc2-n2nccn2)=O)CCN(C(c2nc(Br)cs2)=O)CC1F c1(CC)cc(N)ccc1C(=O)NC1CC(NC(=O)Cc2cn(C)nn2)C1 N1(C(CCCCCN(C(=O)CCC2CC2)C)=O)CCC2(CNC(=O)N2)C1 C1(CN(CCNC2CC2)CC)Cc2ccccc2O1 C(=O)(C1=CCC(C)(C)CC1)N(C(NNC(=O)C1C(C)C1)=O)C(C)(C)C Cc1nc2ccccc2nc1NC(=O)N(C(c1ccc(F)c(Cl)c1)CO)C C(CC(C)(C)C)(C(=O)NCCC(C)NC(=O)C(c1cn(C)nc1C)O)OC C12(NC(C3CC(C)(C)OCC3)=O)CC3CC(C1)CC(NC(C1CCCO1)=O)(C3)C2 C1(CC(C)NC(=O)CCOCCN(C)C)CN(C(C2(C)CSC2)=O)C1 Cc1[nH]c(C#N)cc1C(=O)NCC1C2CN(C(c3ccsc3Br)=O)CC12 N1(C(C2N(C(c3c(CC)[nH]cc3)=O)CCCCCC2)=O)CC(CO)C(C2CC2)C1 Cc1ccnnc1C(N1CCC(CNC(c2c[nH]c(C(F)(F)F)c2)=O)C1)=O Cc1cccc2c(C(=O)N(CCOC)Cc3ccccc3)cccc12 N1(C(C2CCC(CC)C2)=O)CCC(CN(C)C(C2(CO)CC2)=O)CC1 c1(C(=O)NC(C2CCCN2C(=O)CSCc2cscn2)C)ncc[nH]c1=O N1(C(Cc2ccn(C(C)C)n2)=O)CCC(C)(NC(C2CCC(C)CC2)=O)C1 CC(C(=O)NCCN(CCCN(C)C)C(=O)CC1CCC(=O)N1)S(N)(=O)=O Cc1cc(C)n2nc(C(N3CCC(CNC(=O)COC(F)F)C34CC4)=O)nc2n1 N1(C(C2C(COC)C2)=O)CCCN(C(=O)CC2CCS(=O)(=O)CC2)CC1 c1(N(C)Cc2c(C)cco2)nc2c(c(=NC(C)C3CC3)[nH]1)SCC2 C(=O)(C(CCS(C)=O)N(C)C)N(CCC(C(C)C)NC(c1c(C)nc(C)[nH]1)=O)C C(=O)(CC(C)CC(C)C)NCC(C1CCC1)NC(c1c(C)cno1)=O C1(N(C(=O)C=CCO)C)CC12CCC(NC(=O)CN1CCN(C3CC3)C1=O)CC2 c1(CC(N2CCC(N(C(=O)C(F)(F)c3nccn3C)C)C2)=O)ccc(O)c(F)c1 C1(NC(C(C)CCN(C)C)=O)COC2(C1)CN(C(=O)CC(C)(C)C)C2 CCCCC(CC(=O)NCCCCCF)NC(c1ncccc1F)=O c1(OC)ncccc1C(N1CCC(C(C)(C)NC(=O)CN2CC(=O)NC2=O)C1)=O c1(C(=O)NCCCCCNC(c2c(C(C)C)cccc2)=O)ccc2c(c1)OCO2 N1(C(C=CC)=O)CC(C(N2CCCC3(CCC3)C2)=O)CC(C)(C)C1 N1(C(C2C(C(=O)OC)C2)=O)CCN(C(=O)CCC2CCCCO2)CC1C C(=O)(CCCC(=O)OC(C#N)C1CC1)NC(C)(C)C c1(C(=O)NCCN(C)C(c2ccncc2N=[N+]=[N-])=O)nc2n(c1Cl)CCCC2 c1(NC(C2CC(=C)CN2C(c2ccno2)=O)=O)cc2[nH]ncc2cc1OC C1(OC)CCC2(C(N3CC(F)(C(=O)NCC4COCC4(C)C)C3)=O)CC12 C1(C(N(CCNC(c2ccsc2Cl)=O)C2CC2)=O)COCCC1c1ccccc1 c1(OCC(N2CC3C(NC(C(CCC)O)=O)(C3)C2)=O)ccc(Cl)c2ccccc12 c1(C(=O)NCCCC2(NC(C=C(C)C(C)C)=O)CC2)cn(CC2CCCO2)nn1 c1(C(=O)OC(C(F)(F)F)C2CCCO2)ccc(Br)cc1C(F)(F)F C1(NC(c2ccc(SC)s2)=O)CN(C(c2cnc(C(C)(C)C)s2)=O)CCC1C C=CCC(C)(C)CC(=O)NCC1CN(C(c2cccc(Cl)c2N)=O)CCN1C C1(CC#C)(C(=O)N(CC(C)N(C)C(c2ccn(CCC)n2)=O)C)CCOC1 c1(S)ccccc1F.C1(n2c(C3C(C(CC(=C)Br)=O)(N)C3)nnn2)CCCCCC1 c1(C(N2C(CC(N3CC(CCC)OCC3)=O)CC2)=O)cc(C)cc(O)c1 C1(NC(=O)C(CO)c2ccccc2)CC2CCC(C1)N2C(=O)CN1CCCC1 C1(C(=O)N(c2ccc(OCF)cc2)C(=O)C2CC2)C2Cc3ccccc3C12 C1(CC(=O)NCCCCN(C(=O)C=CC2CC2)C)COCC(C)(C)O1 N1(C(c2cc(=N)[nH]cc2)=O)CC(NC(=O)Cc2cnns2)CC2(CCC2)C1 c1(C(=O)NC(CNC(c2ccc(C)cc2)=O)C(C)C)cccc(C(F)F)c1Cl CCCC(C)(C)CC(=O)NC1(CC(=O)NCC(c2ccccn2)O)CCC1 N1(C(CC)=O)CCCC(C(=O)NC2C=CCN(C(C3CCCCN3C)=O)C2)C1 C1(CN(C(=O)COCC2CCCO2)C)CCCN(C(=O)C(c2cnn(C)c2)O)C1 c1(C(=O)NC2CCCC2NC(C2CCC2(F)F)=O)cnc2c(F)cccc2c1 C(C(C(=O)NCCCNC(N)=O)NC(c1cc(C)c[nH]1)=O)OCC C1(NC(CCCc2onc(C(C)C)n2)=O)CN(C(=O)Cn2cnnc2)C2CC12 CC1CN(C(C2(C)CC2(F)F)=O)CC1CC(=O)NCC12CCCC1C2 c1(C(=O)NC2(CF)CCN(C(CCc3n(C)cnc3)=O)C2)ncnc2c1CCC2 c1(C(=O)NC(CNC(c2c(CC=C)cccc2)=O)C2CC2)cn2c(n1)CCCC2 Nc1cc(C(=O)NCC2CCC(NC(c3ccc(Cl)cc3Cl)=O)CC2)ncc1F C12(NC(c3nccc4[nH]ccc34)=O)CCCC1CN(C(=O)C=Cc1cscn1)C2 C(C1=NOC2CCCC12)OC(CC(c1ccccc1)NC(C)=O)=O C(=O)(CCCC(=O)N(C)C)NC(C(C)NC(c1cccc(N)n1)=O)C CN1CC(=O)NC(CC(=O)NC2COCCC2NC(=O)C(C)(C)O)C1=O C1(CC=C)(C(=O)N(C)CCC2CC2)CCCN1C(=O)CCOC(=O)C1CC1 c1(C(=O)NCC(C)(C2CC2)NC(C(CC(C)C)OC)=O)ccnc2[nH]nnc12 C1(C(=O)NCC(C)N(C(=O)CC(C)(C)c2ccccc2)C)Cc2nncn2C1 C1(C(=O)NCCN(C(=O)OC)C)CC2CC1CO2 N1(CCC)CC2(CC(NC3CCC(C)(C)O3)C2)C1 N1(C(C(CC)OC)=O)CCC2(C1)CN(C(C13CCCCC1C3(F)F)=O)CC(C)O2 C1(C(=O)NCC2(C(=O)NC(c3cn(C)cn3)C)CC2)CC2(CSC2)C1 N1(C(C2CN(C)C2)=O)CCCCC1CCNC(c1cnn(C)n1)=O N#Cc1cc(F)c(F)cc1NC(c1ccc(CN2CC3CNC(=O)C3C2)cc1)=O Cc1nc(Cl)sc1C(N1CCN(c2noc(C)n2)CC1)C(=O)NCC1CCOC1 C(C(O)C(C)(C)C)NC(CCCn1cc(-c2cn(C(C)C3CC3)nc2)nn1)=O CC(C)CC(N)CC(=O)N1CC2CCCC1C2CO C1(NC(C2CS(=O)(=O)CC23CC3)=O)CCCC12CN(C(c1ccc[n+]([O-])c1)=O)C2 c1(C(=O)NC2CCC(NC(CC(C)C3CCCC3)=O)C2)cn2cc[nH]c(=O)c2n1 N1(C(c2cnc(CC)nc2)C(=O)NC(C)C)CCC2CCCCC2C1 Cc1cc(F)c(C(=O)NC2CCN(C(C3CCCCN3C)=O)C2)c(F)c1 c1(CC(=O)NCCN(CCOC)C(C2CN(C(C)=O)CCO2)=O)nnc(C)n1C C1(NCC(=O)NC(C)C(=O)O)CCCCC1C C1(F)(C(=O)NCC2(C)CC(NC(CCC)=O)C2)C(C)(C)C1(C)C C1(C(N2C(c3ccc(CN)s3)CCC2)=O)CC(CN)C12CCC2 C1(C(=O)NCC(=O)NCC(=O)Nc2cccc(OC)c2)CCOC(=O)CC1 C1(CNC(c2ncccc2Cl)=O)CCCC2(CN(C(=O)CN3CCC3)C2)O1 c1(CNC(C2CN(C(=O)NC)C2)=O)cc(C(=O)NCC2CCC(C)S2)on1 C1(NC(=O)CSCc2cscn2)CCN(C(=O)CC2CC3(CCC3)CO2)CC1F N1(C(c2c(C)ccnc2)=O)CC2(C1)SCCC2NC(C1CC2CC2C1)=O c1(C(N(C2CCN(C(C34CCCCC3OCC4)=O)C2)C)=O)ccc(F)c(F)c1F c1(C(=O)NCCC(CC)(CC)NC(=O)C(O)CN(C)C)n[nH]c2c1CSCC2 C1(C2CCOCC2)(C(=O)OCc2cn(C3CCCC3)cn2)CCOCC1 CC1CCCC1C(=O)NCCSCC(N1CC(C)(O)C1)=O c1(C(=O)NCCC2(C)CCN(C(=O)CC3OCCC3(C)C)C2)cccc(F)c1N C1(O)(CCNC(C2C(CNC(=O)Cc3ccoc3)OCC2)=O)CCCCC1 N1(C(C2C(C(C)O)C2)=O)CCC2(NC(c3cc(Br)co3)=O)CCCC12 C12(NC(CCCSC)=O)CCC(F)(F)CC1CN(C(C1CCC1(C)C)=O)C2 C1(NCc2cn(-c3cccc(C)c3)nn2)CCN(Cc2ccccc2)C(C)C1 C(c1ccc(Br)cc1)=CC(N1CCN(C(CNC(c2c(NC)scn2)=O)=O)CC1)=O N1(C(C(CCC)(C)C)=O)CCOC2(CCCN(C(=O)C(C)(COC)OC)C2)C1 C1(C(N(CCC(C(C)C)NC(=O)CN2CCNC(=O)C2)C)=O)CN(C)CC(C)O1 Cc1cc(C(=O)NC2COCC2NC(C2(C(C)(C)C)CCCC2)=O)ncc1CO C12(CNC(C(CC)N(C)C)=O)CCC(CC1)CN2C(=O)CCNC(=O)CO CC1CCCC1(C(=O)N(CCCN(C)C)C)NC(C1CCCC1O)=O CCC(C)C(C)(c1nnnn1C1CCCC1)Nc1cnn(CCC(C)C)c1C c1(OC)cc(F)c(C(=O)NC(C)CNC(c2ccc3c(c2)OCC3)=O)c(Cl)c1 Cc1cc(C(N2CC3CCN(C(=O)CS(C)(=O)=O)CC3C2)=O)ccc1[N+](=O)[O-] CC1(C)CCOC1C(=O)NCC1COCCN1C(=O)CSc1ccccc1O C12(NC(C3(CNC(=O)CC4CCCCC4)CCCO3)=O)CC3CC1C2C3O c1(NC(N2C(c3nc(C)c(C)[nH]3)CCC2)=O)ccccc1S(=O)(=O)C(F)F CC1CN(C(C2(C)CCCN2C(c2ccc(Cl)c(F)c2)=O)=O)C(C)CO1 N1(C(c2c(C)nc(O)[nH]2)=O)CCC2(CCCCN(C(=O)C=CC3CC3)C2)C1 c1cc(N2CC3CCC3C2)nc(N2CCC(CC3CCCC3)C2)n1 C(=O)(C(O)CCCNC(=O)COc1ccccc1)N(CC(C)CO)C Cc1ccc(C)c(OCCC(=O)NC2C3CC2N(C(c2cc(C)ccn2)=O)C3)c1 c1(C(=O)NC2CN(C(C(COC)COC)=O)CC(F)C2)cc(Cl)cc(C)c1OC C#Cc1ncccc1NC(c1ccc(N2CCN(C(C)=O)CC2)nc1)=O C1(CCC(C)C)CCN(C(c2cnc(N(C)C)nc2)=O)CC1 c1(N2CCCC(NC(c3cccnc3C3CC3)=O)C2)cccc(F)c1[N+](=O)[O-] N1(c2nc(C#N)cc(C)n2)CC23CCCC2(CN(C(=O)C2=CCCCCC2)C3)C1 c1(C(N2CC3CC(NC(C(C(C)C)N(C)C)=O)C3C2)=O)c[nH]c2cc(N)ccc12 C(=O)(C1=CC2C=CC(C1)C2)NC1CCC(CC(=O)NC(COC)C)C1 N1(C(CCCNC(=O)OC)=O)CC(CNC(=O)COCCC2CCCC2)CC1C C(=O)(CCCC(C)CC)NCCNc1sc(C(=O)OC)c(C)c1Br C1(C(N(C)CC2CCCN2C(c2cnsc2)=O)=O)Cc2cc(Cl)ccc2C(=O)O1 Cn1nc2c(c1C(=O)NCCN1CCN(C(C3CCNC3=O)=O)CC1)CCCC2 C1(NC(C=Cc2c(C)ncs2)=O)CCCN(C(=O)CP(C)(C)=O)CC1 C1(Cc2cn(CC(C)(C)C)nn2)CN(C(=O)CC2CSCCO2)CCO1 c1(CC)ccnc(C(N2CCC(C(=O)Nc3cccc(Cl)c3)C2C(C)C)=O)c1 N1(C(C=COCC)=O)CCC(NC(c2ccco2)=O)C(F)C1 c1(C(N2CC3(CCN3C(c3ccc[n+]([O-])c3)=O)C2)=O)cccc2c(Br)n[nH]c12 N1(C(c2scc(OC)c2)=O)CCCC(C(C)NC(c2nnn(C(C)C)c2C)=O)C1 C12(C(N(CCCC3CCC3)C)=O)CCC(n3cc(Cn4cc(Cl)cn4)nn3)(CC1)C2 N1(C(C2CN(C(C3(C(F)(F)F)CC3)=O)CC23CC3)=O)CC2(CCCCCC2)C1 C1(NC(C2(CC)CCN(C(C3CCC4CC34)=O)CC2)=O)CCC2(CCC2)CC1 C1(C(=O)NCc2c(C(N3CC4C(CC)(C4)C3)=O)nco2)CC12CCCCC2 c1(C(N(CC(C)N(C(C2C(CCOC)C2)=O)C)C)=O)ccc(O)nn1 C12(CNC(C(F)=CCC)=O)CC3CC(CC(NC(=O)COCC4CCC4)(C3)C1)C2 C1(F)(C(=O)NCCCCN(C(C)C)C)CCCN(C(C2CC(=C3CC3)C2)=O)C1 C1(C(=O)OC)(COC)CCCCN1CCC(=O)N(C1CCCCCC1)C C1(CC=C)(NC(=O)C(C)NS(=O)CC)CN(C(c2occc2CC)=O)C1 Cc1cccc(O)c1C(=O)NC1CCCC(NC(C2(C)COCCO2)=O)C1 C(C(C)(CO)OC)NC(CN(C(=O)CC(C)n1ccnc1)CC#C)=O c1(C(=O)NC(CCC)C(=O)N(C)Cc2ccn(CC)n2)ccc2c(c1)COC2 c1(C(=O)NC2CC3CC(NC(C4CCS(=O)CC4)=O)C3C2)cc2ncccc2[nH]1 C1(NC(=O)CC2CCOC2=O)C2CC1CN(C(=O)Cc1c(F)cccc1Br)C2 c1(C(N2CCC(CNC(C3(C#C)CCC3)=O)C2)=O)cnc(C)nc1COC CCC(CN(C)C)CC(=O)NCCCCC(C)NC(c1csc(COC)c1)=O CC1CCN(C(=O)CC2CCCOC2)CCN1C(c1csnc1Br)=O C(C(C)(CC)C(N)=O)NC(CC1N(C(COCC(=C)C)=O)CCC1)=O NC1(C(=O)NC(c2ccc(F)cc2)C2CC2)CC12CCC2 Cc1ncccc1C=CC(N1CC=C(CNC(C2CC(C)CO2)=O)CC1)=O c1(C(N2C(CN(C(=O)C(=O)C(C)(C)C)CC)CCC2)=O)ccc(OC)c(Cl)c1 N1(C(CC2(OC)CN(C(C(C)OCCC=C)=O)C2)=O)CC(CO)C(C2CC2)C1 C1(C)(CNC(C2C(OC)CC2)=O)CCCN1C(C1CC1C(F)F)=O n1(CC(=C)C)c(N(CCCn2ccnn2)C)nnc1CC1CCCC1 c1(OC)noc(C)c1C(N1CCC(C(C)NC(c2cc[n+]([O-])cc2)=O)CC1)=O N1(C(COc2c(C)cc(Cl)cc2)=O)CCC2CCCC12CNC(=O)C1=CCCS1 CC(=O)CCCC(=O)Nc1ccc(NC(C2CCCN2C(=O)OC)=O)c(C)c1 c1(C(=O)NCC2C(CC)CCC2)ccc(C)nc1 C(CCCC(=O)NC1CC(CN(C)C)C1)OC.C12CCOC1C(=O)NC2 CC1CCN(CC(=O)N(C(C)CN(C)C(c2ccn(CCF)n2)=O)C)CC1 c1(C(=O)NCC(CC)NC(C2CC(C)CCO2)=O)ccncc1N(C)C N1(C(c2ccc(SC)cc2Cl)=O)CCC2CN(C(C3CCCC(C)O3)=O)CC12 C1(C(=O)NC(C)CNC(=O)C(CN(C)C)N(C)C)CCC(=O)N1C1CC1 C(CC(F)F)(C(=O)NCCC1NC(=O)NC1=O)NC(COCC(=C)C)=O c1(C(=O)OC)ccc(CNC(=O)CCCOc2ccc(Cl)cc2)cn1 c1(C(=O)NC(C2(CNC(=O)CC3(O)CCCOC3)CC2)C)cn2cc(Cl)cnc2n1 CCC(C)CCC(=O)N1CCC(Cn2cc(-c3cccc(C(=O)O)c3)nn2)C1 C(=O)(C(O)C1=CCCCC1)N1CCN(CC(=O)NCc2n(CC)cnn2)CC1 c1(OCC)cc(CNC(=O)C(N2CCC(C)(c3cccc(Cl)c3)C2)=O)cc(F)c1 c1(OC)cc(OC)c(C(=O)N(C(C)CN(C)C(c2cocc2C)=O)C)cc1OC c1(C(C(=O)NC)N(CC(C)(C)C)CC)ccc(OC)c(SC)c1 C1(CC)CN(C(C2(C(=O)OCC3CC3)CC2)=O)CCC1NC(=O)Cn1nccn1 c1(C(N(CCNC(C2CCC(OCCC)CC2)=O)C)=O)ncc(Cl)nc1Cl C1(CNC(c2c(C(=O)OC)cn(C)n2)=O)CC(C)(C)CN1C(=O)CC=C(C)C N1(C(C2C(C)(C)OCC2)=O)CCCC(O)(CNC(C2CN(CC(F)(F)F)C2)=O)C1 c1(N(C(=O)CC2CC2)CCCN2CCOCC2)cc2nc(F)ccc2o1 N1(C(C2CC(OCC)C2)=O)CCN(C(=O)C2=NOCC2)C(CSC)C1 C1(CC)CCN(C(=O)CS(C)(=O)=O)C1C(=O)NC(C)C(C)n1cccn1 CCC(C)C(O)C(=O)NC(C)CC1CN(C(c2csc(-c3ccccn3)n2)=O)C1 C1(C(N2C(CNC(C(CC#C)C)=O)CC(F)(F)C2)=O)CC2(C1)CC(C#N)C2 c1(C(=O)NC2CCCC(NC(CCCCC=C)=O)CC2)ccc(F)c(OC)c1F Cc1ccc(-c2ocnc2C(=O)NC(CNC(C2(C)CC2(F)F)=O)C2CC2)s1 C=C(CNC(=O)CC=CC)CCNC(=O)C(O)C1CC1 C1(C(N2C(C=CC(N3C(COC)C=CC3)=O)CCC2)=O)CC(=O)CC(=O)N1 c1(C(=O)NC(CC)CNC(c2cc3cccnn3c2)=O)cnn2ccc(C)cc12 c1(C2(c3cc(-c4ccoc4)[nH]n3)CC2)ccc(Br)cc1.C12CC1C(=O)N2C Cc1cc(-c2nc(-c3ccccc3F)nn2CCOC(C)C)c(C)o1 N1(C(C(CC2CC2)NC(c2cc(C(C)C)[nH]n2)=O)=O)CCC2(CSC2)C1 CP(C)(=O)C1CCCCC1C(=O)NC1C2CC1N(C(=O)CC1CCOC1)C2 N1(C(C(c2ccccc2)OC)=O)CC2(C1)CN(C(c1nnn(C)n1)=O)CC2CO N1(C(C(C2CN(C(C3CC3C(C)C)=O)C2)OC)=O)CCCC2(CCC2)C1 N1(C(c2c(C)nco2)=O)CCC(C)C(CNC(=O)CSc2ccc(F)cc2)C1 c1(C(N2CCC(C=C)C2)C(=O)NC2CC(C(=O)OC)C2)cc(C)c(F)cc1Br c1(CC(=O)NCC2C(CCNC(C)=O)C2)coc2cc3c(cc12)CCC3 N1(C(C(COC(C)C)(C)C)=O)CCC(C(F)(F)F)C(NC(=O)C(C)(C)N(C)C)C1 S(=O)(=O)(c1c(Cl)cc(Cl)cc1Cl)NCCn1ncc(NC2CCCC(C)CC2)c1 c1(C(=O)CC2(O)CC(NC(C3(CC)CC3)=O)C2)ccc([N+](=O)[O-])c(NC2CC2)c1 S(=O)(=O)(c1ccccc1Br)NC1C2(CN(C(CC3CCN(C)CC3)=O)C2)CCC1 C(CCCCCC(=O)NC12CCC(CC1NC(C1CCCNC1=O)=O)C2)SC S(=O)(=O)(c1cnc(N2CCC(CCC)C2)cc1C)NC(CCC=C)(C)C c1(C(C(=O)NC2C(CNC(C3(OC)CCC3)=O)COC2)(F)F)c(F)cccc1F CC1(C)Cc2ccc(C(N3CC(O)CC3CNC(=O)CC#N)=O)cc2O1 C1(C(N2CC(NC(C3CC4(CSC4)C3)=O)(CO)C2)=O)COCCC1(F)F N1(C(c2n(C)c(=O)ccc2)=O)CCC2(CCCC2C(NCP(=O)(O)O)=O)C1 C(=O)(C(CC)C(=O)OC)N1C(C(N(CCOCC#C)C)=O)(COC)C=CC1 C1(C(N(C)CCC2CCOC2)=O)CCCCN1C(=O)CCC(=O)N1CCCC1 c1(C(C2CCCC2)NC(N2CC=CC(O)C2)=O)ccc(Cl)cc1O C1(CNC(CC2CN(C(C3(CNC(C)=O)CCC3)=O)C2)=O)CC(=O)N(C)C1 N1(C(c2ccc(C3CC3)nc2O)=O)CCC2(CCC2)C(O)C1 c1(NC(C)=O)ccc(CC(N2CCN(C(=O)COC(F)F)C3CC23)=O)cc1C C1(C(N2C(CNC(C3COCCOC3)=O)CC(C)(C)C2)=O)CCc2nc[nH]c2C1 C1CCCCC(=O)N2CCCCC2c2cn1nn2.N12CCC(CC1)C2.CCOC c1(-c2ccc(OC)nc2OC)cccc2nc(C(=O)Nc3nc(C)cs3)ccc12 CCC(C)C(O)C(=O)NCCN1CCC(NC(=O)CCCn2cccn2)CC1 Cc1cc(C(=O)NCC2CC2CNC(=O)CCc2cc(F)ccc2Br)cnc1O c1(C(=O)NCC2(NC(C(C(C)C)OC)=O)CCCCC2C)cncc2ccsc12 c1(C(=O)NCC2C(CNC(C(F)=CC)=O)C2)c(C)ncn(C)c1=O CC1CCN(C)CCN1C(N1CCC(CC(C)(F)F)CC1)=O CCC(C)C(C(=O)NCC(C)(C)CNC(=O)CC1(O)CCC1)NC(N)=O Cc1cn2cc(C(=O)NC34CCC(C3)N(C(=O)CC3COCCN3C)C4)nc2s1 N1(C(c2c(CCC)nns2)=O)CC2CC(C1)C(CO)C2NC(c1nonc1N)=O N1(C(=O)CC2(NCCNc3cc(Cl)ccn3)CCC2)Cc2cncnc2C1 c1(CC(=O)NC(CNC(c2c(CC)occ2C)=O)C)cccc2cccnc12 c1(OC(C)C)ccc(NC(c2cnnc(O)c2S)=O)c(Cl)c1 N1(C(C(F)=CCC)=O)CCC(NC(=O)COCc2ccccn2)C(CC)C1 c1(C(N2CC(COC)N(c3nccc(C)n3)CC2)=O)c(C)ccc(Br)c1F n1(CC(=O)N(CC(C(C)C)NC(=O)C(F)SC)CC)c(C2CC2)nc2ccccc12 CC(C(=O)NC1CCC1CNC(c1cc(C2CCCC2)nn1C)=O)P(C)(C)=O c1(C(N2CCN(C(=O)CCc3cnn[nH]3)C3CC23)=O)cccc([N+](=O)[O-])c1Cl C=CCCCC(C(=O)NC(C)(C)CCCC)NC(=O)COCCC(C)C C1(CCC(=O)N(CCCN(C)C(C2(C)CC2(F)Cl)=O)C)CCCCN1C C(CN=c1ccnc(N2CCOC3(CCSCC3)C2)[nH]1)(CC(C)C)OC C1(CCNC(CCNC(C)=O)=O)CN(C(=O)CS(=O)(=O)N(C)C)CCCO1 c1(-n2c(-c3cccc(C(C(C)C)CCO)c3)ncc2)cc(=NCC(F)CO)[nH]cn1 C1(CNC(C2(CN(C)C)CC2)=O)C=CC(NC(=O)C(C)(C)C2CCCO2)C1 C(CCC(N)=O)(C(=O)N(CCCC)Cc1nccs1)n1cc(C(C=C)(C)O)nn1 C1(C(=O)NCC(C)(CO)c2ccccc2)CCCC2(CCNCC2)O1 C=CCC(CNC(c1ccc(C2CC2)o1)=O)C(=O)N1CCCC1CC1CC1 C12(OCC)CCC(C(N3CC4(CC(CNC(=O)CC(C)O)C4)C3)=O)(CC1)C2 Cn1ccc2[nH]c(C(=O)NC3(C)CCN(C(=O)C(F)=C4CCC4)C3)cc12 C(=O)(C(C)CC(=O)OC)NC1CC(N(C(CSCCN(CC)CC)=O)C)C1 C1(NC(C2(C3CC3)CC2)=O)CS(=O)(=O)CC1N=c1[nH]ncs1 c1(C(=O)NC2C(CNC(C=CC(CC)C)=O)CC2)cccc([N+](=O)[O-])c1C C(=O)(C1=CC2CCCC12)NC1CCN(C(CC2(C(=C)F)CCC2)=O)C1C CC1OCCCC1C(=O)NC12CC(C1)N(C(=O)Cn1ncnn1)C2 c1(C(N2CC(F)(C(=O)Nc3cn(C(C)(C)C)nc3)C2)=O)cccc(Br)c1 C1(CC=C)(NC(c2ccc(SCC)cc2)=O)CCN(C(C2(CC#N)COC2)=O)C1 c1(CC)cc(C(=O)NCC=CCNC(C2(C)CCCC2(F)F)=O)cc(O)n1 C=CCC(CC=C)C(=O)N1CC(C)CCC1C(N1CC(C2CC2)(OC)C1)=O C1(c2ccc(C)o2)CS(=O)CCN1CCc1ccc(C(F)(F)F)cn1 C(=O)(CS(=O)(=O)CC(=O)NCC(CO)NC(=O)CC1C=CS(=O)(=O)C1)OC c1(C(=O)NCCC2C(C)CN(C(C3(CO)CCOCC3)=O)C2)cc(N)cc(O)c1 c1(C(=O)NCC(C)N(C(CC2(C=C)CCC2)=O)C)cccn2cncc12 C1(N(C)C)CN(C(=O)C=CCC(C)(C)NC(=O)CCc2ccc[nH]2)CC1O N1(C(C(C)(C)C2CCCCO2)=O)CC2CC(C1)CN(C(=O)CC1OCCO1)C2 C(=O)(C(CO)NC(N)=O)NCCN(N1C(C(=O)NCC)CCC1)C(C)=O C=C=C(C)CC(=O)NCCCC(=O)NCc1cccc(OC)n1 C1(CC(=O)NCCCN(C(=O)C(CC)OC2CCCC2)CCC)CCC1(C)C C=C(C)C(C)(O)C(=O)NCC1(CNC(c2cncc(N(C)C)n2)=O)CC1 O(NC(=O)C(c1cccnc1)NC(c1ccn(CCF)n1)=O)CC(C)C N(C)(C1CN(C(=O)C(=O)NC2CC2)CCc2ccccc21)C(CC(CC)OC)=O c1(C(=O)OCCCN(C(=O)Cc2ccccc2F)CC)ccc(NC)cc1 N1(C(C2(SC)CC(=O)C2)=O)CC(C(=O)NC2CC3(C2)CC(O)C3)CC(C)(C)C1 CCC(C#N)C(=O)NC(c1ccccc1)CNC(=O)C(C)(C)OCC(F)(F)F CCN(C(C)c1ccccc1Cl)N(C)C1CCN(c2cnn(C)c2)C1=O CC1(C)C(c2cccc(Cl)c2)CCN1C(C1CCC1Cc1ccccc1)=O Cc1cc(C2CCC2)ccc1C(=O)N(C1CCN(C(c2cnccc2Cl)=O)C1)C c1(C(=O)NCC2(CO)CCN(C(C3CC=CCO3)=O)C2)ccn2c1CCCC2 S(=O)(=O)(C1CCC(=O)CC1)NC1CCCN(Cc2cccc(OC)c2F)C1 C(=O)(C(C)CC)N(C(C(=O)N(C)CC)C)C.C1(=O)CO1 CS(=O)(=O)c1cc(C(N2CCC(O)C2c2cccc(Br)c2)=O)cc(N)c1 CCC(C(=O)OC)C(=O)NC(c1ccnn1C)C(N1CCC(CCOC)C1)=O c1(CC(=O)OC)c(C)nn2c1CN(C(=O)COCCCC1CNC1)CC2 C1(C(=O)NC2(CC=C)CN(C(C3(c4ccn(C)n4)CC3)=O)C2)C2CCC(=O)C12 C1(N(C(C(CCOC)NC(c2cscc2C)=O)=O)C)CCC2(CC1)CC2 C1(CC)(NC(=O)CO)CN(C(c2cncn2C)=O)C1 N(C1CCCc2c[nH]nc21)C(C(C(C)C)NC(=O)CC1(C)CCOCC1)=O CC1CCn2ncc(C(=O)NCC=C3CCN(C(=O)CCF)CC3)c2C1 c1(OC)ccc(N)c(C(=O)NC(C)CCNC(=O)COC2CCOC2)c1 C(=O)(C(CO)NC(=O)C(N1CCNC1=O)C)N(C1CC(=C)C1)C C(=O)(C(CN=[N+]=[N-])NC(c1occc1C)=O)N(C)Cc1n(CC)cnn1 c1(C(=O)NCC(CC)NC(c2cc(C(C)C)nn2C)=O)cn(CC)nc1C CCCCC(C)NC(C)(CCc1ccco1)c1nnnn1C1CCC1 N1CC(ONC(=O)CC(=CC2CCC2)C)C(C)(C)C1.C(=O)C(C)(C)CC#N c1(CCC)cc(C(=O)NC(Cc2cc[nH]n2)C(=O)NC2CC=CCC2)n[nH]1 c1(C(=O)NC2CC(CCNC(C3CC=CCO3)=O)C2)ccc2nsnc2c1 c1(C(=O)NCCCC(=O)N2CC(OCC(=O)NC)C2)cc(C#N)ccc1N c1(C(C(=O)N(CCN(C(c2cnc(SC)s2)=O)C)C)C)c(C)n[nH]c1C c1(CC(=O)NCC23N(C(C4CCC(C)C4)=O)CC(C2)C3)nn(C)c2ccccc12 C1(C(=O)NCCC#C)CCC2(CN(C(c3c[nH]cc3C)=O)C2)O1 c1(CC(=O)NCC2CN(C(c3csnn3)=O)CCCO2)csc2ccc(Cl)cc12 C1(C(=O)NCc2scnc2Cl)CCOCCN1C(=O)CC1C=CCC1 N1(C(=O)C=Cc2ccoc2)CCC2(C1)CN(C(C1CC(CCF)C1)=O)C2 c1(C(=O)NC2CC(C(C)C)SCC2)cc(C#N)ccc1Cl c1(OC)ccc(CCC(=O)N(C2CC2)CC2CCCO2)cc1CO C1(CC)(NC(=O)C=CS(C)=O)CCN(C(=O)C(C)(C)CN2CCN(C)CC2)CC1 c1(CN(C(C(CC)Cc2cccc(C)c2)=O)CC)cccc2c1CCC2 C(=O)(C(F)(F)c1csc(=N)[nH]1)NCC(CN(C)C(C1(N(C)C)CCC1)=O)O O=C(CCCC1CCCO1)NC(=O)CSCC(=O)NCCCCN1CCOCC1 c1(C(N2CCC(NC(c3cc(C)on3)=O)C(C)(C)C2)=O)cncc2nnn(C)c12 C1(C(=O)NCCOC2CN(C(C(C(C)C)F)=O)C2)CCCCC1(F)F N1(C(CC(C)c2cccnc2)=O)CC=C(CNC(c2cc(O)nc(O)n2)=O)CC1 Cc1[nH]nc2ccc(C(N3CC4(CC4)CC3CNC(=O)CC3(C)CC3)=O)cc12 c1(C(=O)NCCCC(c2ccccc2)NC(CCC#C)=O)cc(Cl)c(Cl)s1 C1(C(N(CCN(C(c2cc(C(C)C)on2)=O)CC)CC)=O)CC2COCC(C1)C2 Cc1ccnc(N(CCCNC(c2cc(O)nn2C)=O)C(C)C)c1[N+](=O)[O-] c1(C(=O)NC(CCCNC(c2n(CC)ncc2)=O)C)nc(O)nc(O)c1N C1(O)(NC(Cc2ccc(CC)cc2)=O)CCCN(C(=O)NCCCC(C)C)C1 c1(NC(=O)NCCC#C)ccccc1-n1nc(C)cc1C CC1C2CC(C2NC(C2CCN(C)C2=O)=O)N1C(=O)C1=CCCOC1 C1(C(C)C)(CO)CCN(C(=O)C(Cc2cn[nH]c2)NC(c2ncncc2Cl)=O)C1 C(CNC(=O)C(C)n1ccnc1)(CNC(=O)CC1(NC(C)=O)CC1)OC c1(CC)nc(C#N)cc(=NC(C)CNC(=O)Cc2ccco2)[nH]1 c1(CC(N2C(CNC(C3CCOC3)=O)CC(O)C2)=O)ccc([N+](=O)[O-])cc1 N1(C(CCCOCC)=O)CCCCC12CC(NC(=O)Cc1ccc(CC)cc1)C2 CC1CC2CCC(C1)N2C(=O)CC(C)NC(c1ccc2cc[nH]c2n1)=O C(=O)(C(C)(O)C(F)(F)F)OCc1noc(C)c1Br C1(C(=O)NCC(CNC(c2ccc(C#C)o2)=O)C)CC2(C1)CC2(F)F CC(C)(C(=O)NC1CNC(=O)OC1)C1=CCN(C(C2CC2C2CCCO2)=O)C1 C(=O)(C1=C2CCN=C2NC=C1)N1CCN(N2C(C(=O)NC)CCC2)CC1.C=O C1(CC(=O)NCC(C2CCC2)NC(C2(n3cccn3)CC2)=O)CCCC1O C1(NC(C=Cc2cnc(C)s2)=O)C(CNC(=O)C(C)(C)CC#N)CCC12CCC2 C12(N(C)C(c3ccc(OC(F)(F)F)c(Cl)c3)=O)CC(N=[N+]=[N-])(C1)C2 c1(OC)cc(I)cc(NCC(C)C(=O)c2ccccc2)c1[N+](=O)[O-] C=CCC(C(=O)N1C(C(N2CC(C#N)C2)=O)CC2CC12)OC c1(C(=O)NCCC2N(C(C(C)(C)O)=O)CCC2)ccccc1CO C(=O)(C(O)P(C)(C)=O)N(C1CC1)CC1CCN(C(C2N(C)CCC2)=O)CC1 c1(C(=O)NC(C2CC(NC(C3(Cl)CC34CCC4)=O)C2)C)ncccc1F C1(C)CC(C)CN1NC(c1cc[nH]n1)C.c1(N)cccc(-n2ccnc2)c1 N1(C(CC(C)n2cccc2)=O)CCC(O)C(N(C)C(C2CCCN2N=O)=O)C1 c1(C(=O)NC(CNC(CCSC)=O)(C)C)cc(C(F)(F)F)ccc1[N+](=O)[O-] C1(CNC(C=C(CC)C)=O)CN(C(c2ccnn2C)=O)CCC1C(F)(F)F C(c1nc2ccccc2[nH]1)=CC(=O)N(C(C)CNC(c1cc(C#N)cn1C)=O)C C(=O)(CC(C)(CN(C)C)C(F)(F)F)N1CC(CNC(C)=O)C(F)(F)CC1 C1(O)(CNC(C(CCC)NC(C)=O)=O)CCCN(C(C2CC(=O)N2)=O)C1 C=CCC(C)(C)C(=O)NCC1CN(C(c2cnco2)=O)CCC1C N1(C(CCC2CCN(C(c3nn(C)c(Cl)c3)=O)C2)=O)CC2OCCOC2C1 C(Cc1ccoc1)(C(=O)N(C)CCOCCO)NC(CC1(OCC)CCC1)=O C(=O)(CC1=NNC(=O)C1)N1CC2C(CNC(c3c(C)cc[nH]c3=N)=O)(C2)C1 c1(CC)ccc(-c2cnn(C(C)C)c2)c(F)c1 c1(OC)ccc([N+](=O)[O-])c(NC(CNC(=O)C(C)N(C)C)C(C)(C)C)c1F N1(C(c2cc(C(=O)OCC)n(C)n2)=O)CC2CC(C1)C2NC(=O)C(O)C(C)CC N1(C(CNC=O)=O)CC2CCC2(C(=O)NC2CC(O)C2)C1 C(=O)(C(C)C(C)C)NCCN(C(=O)COc1ccsc1)CC=C Cc1nc(C)c(C(N2CC(NC(=O)CCc3ccnc(OC(C)(C)C)c3)C2)=O)[nH]1 CN1CCN(C(c2cc(C3CC3)ns2)=O)C(CNC(C2(CO)CCCO2)=O)C1 C1(NC(Cn2c(C)nc(C)n2)=O)CC(NC(=O)CCCN(C)C)C12CCOCC2 Cc1[nH]nc2ncc(C(N3CCC(C)N(C(C4CCCC4C)=O)CC3)=O)cc12 C1(C(N(C(CNC(c2c(SCC=C)cccc2)=O)C)CC)=O)CN2CCC1CC2 Cn1cc(C(=O)NCC2(NC(=O)C=C3CCSCC3)CC2)c(-c2ccccn2)n1 c1(C(=O)NCCC2N(C(Cn3nnc(=N)[nH]3)=O)CCSC2)ccc2c(n1)CCC2 CCC(CC(C)C)C(=O)NC(Cc1ccco1)C(N1CC(=O)NC(=O)C1)=O N1(C(C(C(COC)C)C)=O)CCC2(C1)CN(C(=O)COCP(C)(C)=O)C2 N1(C(C2CC3C=CC2C3)=O)CCCC2(C1)CN(C(C1(O)COC1)=O)CCO2 N1(C(c2nc(OCC)sn2)=O)CCC(C)N(C(c2ccn(CC(F)F)n2)=O)CC1 C1(C(=O)SC)CCCN1CC(N1CC(Cn2cc(CSC3CCOC3)nn2)C1)=O c1(C(N2CCN(C(c3c(CC)con3)=O)CC2C(C)C)=O)cc2nnn(C)c2s1 C1(F)(CNC(c2c(C)ccc(C(C)C)c2)=O)CCCN(C(=O)C=C2CCC2)CC1 C1(C(N)=O)CCCN(CCC(=O)NCC2(O)CN(C(=O)CC3CCOCC3)C2)C1 c1(CNC(C(CO)NC(C2C3CC(=O)CC32)=O)=O)ccc(F)c(F)c1 N1(C(C2N(C)CCCCC2)=O)CCC2(CC(NC(=O)COc3cnn(C)c3)C2)C1 CC(C)C(C)CC(=O)NCCCC1CCCN1C(c1cnc(C2CC2)o1)=O N#Cc1ccc(N2CCC(C(=O)NCC3CC(NC(C4CCO4)=O)C3)C2=O)cc1 c1(CC(C)NC(=O)CN2CCCC(C3CCCCN3C)C2)ccc(OC(F)F)cc1 c1(OC)c(C)nc(C2CC2)[nH]c1=NCC1(F)CCN(C(=O)CC2CC2(Cl)Cl)CC1 c1(C(C(=O)NCCN(C(=O)CC(C)CN(C)C)CC)(C)O)ccc(F)cc1 C=CCCC(F)(F)C(=O)N1CC(CC(F)C(=O)NCC(C2CC(C)(C)C2)O)C1 C=CCC(C)(C)CC(=O)N1CCN(C(c2c[nH]nc2C)=O)CC(CO)C1 N1(C(c2c(C)cco2)=O)CCCOC(CNC(c2ncccc2C(F)(F)F)=O)C1 C(=O)(CC1=NNC(=O)C1)NC(c1c(OC)cccc1)CNC(=O)Cc1cocn1 c1(SC)ccccc1C(=O)N(CCCCCNC(=O)C=Cc1sccc1C)C c1(C(N2CC(F)(CNC(c3cn(C)nc3C(F)F)=O)C2)=O)ccc2ccnn2c1 C12(NC(c3[nH]cc(CC)c3)=O)CCCC1CN(C(=O)CSCCN(C)C)C2 C1(CN(C)C(c2ccc(C3CC3)nn2)=O)CN(C(=O)Cn2cnnc2O)CCO1 CC#CCCCC(=O)NCCCCO.C1CCN(C)CCCO1 c1(OC)ccc(-c2c[nH]nc2C(N2CCCC(C)CC2)=O)c(C)n1 Cn1ccc(C(=O)NC2(CNC(c3cn[nH]c3)=O)CCOC2)cc1=O C(=O)(CCCC(F)(F)C(F)(F)F)NCC1(O)CN(C(C=CS(C)=O)=O)C1 Cc1cccc2c(C(N3CC4(CC4)CC3CNC(C3CS(=O)(=O)C3)=O)=O)coc12 C(=O)(C(C)C(F)(F)F)NCC1(COC)CCCN1C(=O)CCC=CBr N1(C(C(CC2CCC2)OC)=O)CCC2CN(C(C3COC(=O)N3)=O)CC12 c1(OC)nccc(CNC(C2(C(=O)OC(C)(C)C)CCC2)=O)n1 N1(C(c2cnc(C(C)OC)s2)=O)CCN(C(C2CCO2)=O)CC2(CC2)C1 C1(CC(=O)NC(C2(O)CN(C(=O)CS(C)(=O)=O)C2)C)CCC2(CCC2)O1 Cc1nc(NCCCc2cnn(C)c2)cc(=NC(C)C2CCOC2)[nH]1 c1(CC)ncc(C(=O)N(C(C)CCNC(=O)CCOc2ccncc2)C)[nH]1 C1(C)(COC)CC(NC(c2[nH]cnc2C#N)=O)CN1C(=O)CCOCC(C)C N1(CCNC(C2(CC)CCC2)=O)C2CCC1CN(C(=O)C(C)(C)CC(C)C)C2 C(=O)(CC(C)(C)C(F)(F)F)N1CC(C)C(NC(C2CCCS(=O)(=O)C2)=O)CC1 N1(C(c2ccc(C(C)C)nc2)=O)CC2CCC1C(NC(=O)C(F)F)C2 C(CCN=c1nc(O)c2ccccc2[nH]1)N1CCc2c(C(=O)O)ccc(F)c2C1 C#Cc1ccc(C(N2CC(NC(=O)CC3CCNC3=O)CC3(CC3)C2)=O)cc1F c1(C(=O)NC2CC(CCNC(C(C3CCC(=O)N3)C)=O)C2)c[nH]nc1F Cc1ccccc1C(N1CC2C(C1)N2C(C1(c2ccc(F)cc2)CC1)=O)=O C1(C2CC2)(C(N2C(C#C)CC2)=O)CN(C(C2C3CCCOC23)=O)C1 c1(C(=O)NCCCN(C(C2(C)CC=CC2)=O)CC)cc2cccc(OC)c2[nH]1 CCCCCC(O)C(=O)NC(CC(N)=O)C(=O)NC(C)CC(C)(C)CO CC1CC(n2nc(-c3cccc(Br)c3)nc2C2CCCN2N=O)CCO1 C=C1CC(C(=O)NC(c2ccccc2)COC)N(CS(=O)(=O)CC2CC2)C1 S(=O)(=O)(C1CCCCC1)N1CCC(NC(c2cccs2)=O)CC1 c1(CC(=O)N(CC(C)NC(c2cc(C)oc2C)=O)C)ccc(O)c(C)c1 C12(C(N3CCC(COC)C3)=O)CC(CO)(CN1C(=O)C(C)c1cc[nH]n1)C2 c1(C(=O)NCC(CCOC)NC(=O)C(F)(F)C(F)F)cncc(S(C)(=O)=O)c1 CCC(CC)C(C(=O)NC1CCC(NC(c2cnoc2CC(C)C)=O)C1)OC c1(C(=O)NCC(C)(CO)NC(CCC2CC(C)C2)=O)cncc(N(C)C)c1 N1(Cc2nc(C(C)(C)C)on2)CCN(CC2CCC(F)(F)C2)CC1 N1(C(CC)=O)CCN(C(C2CCC23CCC3)=O)CC1c1cccc(Cl)c1 C1(C(=O)NCCN(CC)Cc2ncnn2C(C)(C)C)CCC2CC(C)CN2C1 C=CCC(CC)C(=O)NC1C=CCCC1C(=O)NCC Cc1ccc(C)n1CC(N1CC=CCC1C(=O)NCC1CC2CCC2C1)=O c1(CC(=O)NCC2C(C(=O)NCc3ccc(C)s3)CCC2)ncccc1F c1(CCC(=O)NCC(c2ccccc2)NC(COC(C)=O)=O)ccc(F)cc1Cl CC(N(C)N1CCC2NC(=O)OC2C1)C1(S(C)(=O)=O)CC1 C1(C(N2CCC(C(C)NC(C3(CCOC)CCC3)=O)C2)=O)CC(O)CN1C(C)=O N1(C(C2C(C=C)C2)=O)CC2CC1CN2C(c1nnn(-c2ccccc2Cl)c1C)=O c1(C(=O)NCC23N(C(C4C(C)C4)=O)C(CC2)CC3)cc2c(nn1)CCCC2 N1(C(c2c(C)nccc2)=O)C2CCC1CN(CC(O)COCc1cccs1)CC2 c1(C(N2C(c3n(-c4ccc(C)cc4)nnn3)CCCC2)=O)cc(C)nc2[nH]nc(C)c12 Cc1ccc(F)c(N)c1C(N1CC2C(NC(=O)Cc3cnc(C4CC4)[nH]3)C2C1)=O N1(C(C)=O)CCC(CC23CC(C(=O)NC(=O)C(C)(C)O)(C2)C3)C1 c1(OC(=O)COC2(CNC(C3CC(OC)C3)=O)CCOCC2)ccc(C#N)cc1 N1(C(Cc2c(C#C)cccc2)=O)CCC2CCN(C(=O)CC(C)(C)OC)CC2C1 C1(CNC(Cc2nnc(C)o2)=O)CN(C(C2CCCC(=O)N2)=O)C2(CCC2)C1 c1(C(=O)NCC2CC(NC(c3c(C#C)c[nH]n3)=O)C2)nc(OC)cc(OC)n1 CC(CC(N)=O)C(=O)N1CCCC(OCCNC(=O)CN2CSCCSC2)C1 CC(C)(C)C(C(=O)NC1CCCCC1(C)O)NC(c1cccc(F)c1F)=O Cc1nc(C(N2CCN(C(=O)Cc3csc(S)n3)C(CO)C2)=O)ccc1[N+](=O)[O-] C1(CC(=O)O)CS(=O)(=O)C2CN(CC(O)COC3Cc4ccccc4C3)CC12 C1(NC(C2(CCCC)CCCC2)=O)CN(C(c2cn(C)cc2C)=O)CC12CC2 N1(C(c2cnnc(O)c2)=O)CCC2(CCCN(C(C3CCCC3)=O)C2)C1 N1(C(CCC2CC(NC(C(C)c3ccsc3)=O)C2)=O)CCC2CCN(C)CC12 C1(C)(C(=O)NCC=CCSC)CN(C(C2C3CCC(F)C23)=O)C(C)(C)C1 C1(CC(=O)NC2CC(NC(COCCOCC)=O)C2)COCCOC1 C12(C(N3C(C(=O)OC)C4CC4C3)=O)CC(CN(C(c3cc(F)ccc3F)=O)C1)C2 N1(C(c2cn(CC)nn2)=O)CCC(C)(C)C(NC(=O)CC(C)C2CCCCC2)C1 Nc1ccc(CCCNC(=O)NCCc2cc(Cl)ccn2)nc1 N1(C(C=C(C)Cl)=O)CC2CCCC(C1)N2C(c1nc(C)sc1Br)=O c1(CNC(=O)NC(c2cccs2)CC)cc2occc2s1 c1(C(=O)NC2CN(C(CC=C(C)C)=O)C(C)C2)coc(S(=O)(=O)N(C)C)c1 CC(C(=O)N1CC2CC3CC2C1C3)C(C)C(C)(C)C Cc1noc(C)c1CCC(=O)NC(C)(CNC(=O)C(O)Cc1cnc[nH]1)CO C(=O)(C(CC(C)C)NC(c1ccc(O)nc1)=O)N1CCC(COC(C)=O)C1 N1(CC)C(=O)CCC1CC(N1CC2C(CNC(c3ccco3)=O)C2C1)=O N1(C(C(C)(C)SC)=O)CCC2C(C1)NC(=O)CN2C(=O)CC1CC(C)(C)C1 S(=O)(=O)(c1cccc(=NCc2cc3c(s2)CCC3)[nH]1)NC(C1CCC(F)(F)C1)C c1(C(C(=O)NCCC)N2CCC2C2CCOCC2)cccc(C)n1 C1(n2cc(C3CCN(C)C3=O)nn2)CC2CCC1(C(N(C(=O)C(C)(C)CO)C1CC=CC1)=O)C2 N1(C(Cc2cnc(C)o2)=O)CCC(NC(c2cnn(C(F)F)c2)=O)C(O)C1 CC1CC(=O)NCCN1C(C(=O)NC1CC1)c1ccoc1 CC1CCC(N2CCCC2)CN1C(=O)NC(=O)NCC(c1ccc(O)cc1)O c1(C(C(=O)NCCc2ccc(-n3cc(C(C)O)nn3)cc2)O)ccc(C#N)cc1 c1(C(=O)NC(C)CN(C(=O)C(C)(C)S(C)(=O)=O)C)c(F)ccc2n[nH]cc12 N1(C(c2cnc(CC)nc2O)=O)CC(NC(=O)CCNC(N)=O)C(C2CC2)C1 c1(NCCc2ccc(SC)cc2)ccc(S(=O)(=O)N2CCOCC3CC23)cc1Cl c1(OCC(=O)NC2C(CNC(c3cnc(CC)[nH]3)=O)CC2)ccc(Cl)cc1F C#CC1(C(=O)NCCC2COCC2O)CCN(C(=O)C(C)C(C)C)C1 CC1CCN(C(=O)CC(C)C(C)(C)C)CCN1C(=O)Cc1cccs1 CC(C)C(C)(CNC(c1cccc(Br)c1)=O)NC(=O)CC1CC12CC2 C1(CC(=O)NC(CC)(CNC(C2(C)CC3CC3C2)=O)CC)COC(C)(C)CO1 C1(C)(OC)CCN(C(=O)CC2(OC)CN(C(=O)CC3CSC3)C2)CC1 N1(C(CC(CNC(c2cccc3nccn23)=O)O)=O)CCCC12CCCC2 c1(C(C(N2CCC(N(C(=O)CC3CCOC3=O)C)C2)=O)(F)F)ncc(Cl)n1C CN1C(=O)CSC1=CC(=O)NCC(C1CCN(C(C2(CO)CCCO2)=O)CC1)F CCC1=NOC(CC(=O)NCC(c2ccccc2)CNC(C2OCCO2)=O)C1 c1(OC)ccc(CCCCC(=O)NCCCCN(C)C(c2csnn2)=O)cc1 C12(NC(=O)CC3CCCOC3)CCCN(C(c3cc(F)c(F)cc3F)=O)CC1C2 c1(C(=O)NCC(c2cccc(C)c2)NC(CCCOC)=O)scc(C)c1C C1(C(=O)NC(C)CNC(c2c(Br)cnn2C)=O)CC12CCC(C)(C)CC2 C(=O)(C1CCCc2sccc21)N1CC(NC(c2cccc(CO)c2)=O)C2(C1)CC2 Cc1ccn(C)c1C(N1C(C(=O)NCCc2ncnn2C)CC1C)=O C1(OC)CC(NC(=O)C(=O)N(C)C)CN(C(=O)C=Cc2ccc(C)s2)C1 Cc1nc2cc(C(=O)NCC3CCCCN(C(C4CC4C#N)=O)C3)ccc2s1 c1(CC)ccc(OCC(=O)N(C(C)CN(C(=O)C(c2csc(C)n2)=O)C)C)cc1 c1(C(=O)NCC(CC=C)NC(C2(F)CCCOC2)=O)c[nH]c2c(C#N)cccc12 C1(OC(F)F)CCC(NC(=O)OCC(=O)N(CCN(C)C)C)CC1 CC1(C)NC(=O)OC12CCN(C(c1nnc(C3CCCNC3)s1)=O)C2 CN1CCN(C(=O)C(c2ccccc2F)O)CC1CNC(c1cccnc1Cl)=O N1(C(C2(NC(=O)CCc3cscn3)C(C)(C)C2)=O)CC2(C1)CC2(F)F C1(CNC(CCOCCCNC(c2cnc(C)o2)=O)=O)OCCC1(C)C CS(=O)(=O)CCC(=O)N1CC2C(CNC(=O)C(O)COCc3ccccc3)C2C1 c1(CC)ccc(C(=O)NC(CNC(c2cc(-c3ccncc3)[nH]n2)=O)CC)o1 C1(CNC(C(C2CCOC2)NC(C(C2CC2)OC)=O)=O)CCN(C)CC1 N1(C(=O)COc2cccnc2)CC2CN(C(c3coc(Cl)n3)=O)CC(C1)O2 c1(OCC)noc(C)c1C(=O)NCC1(CNC(c2cc(CN(C)C)on2)=O)CC1 c1(OC)nccc(C(=O)NCCC2CCCN2C(C2CCCC(OC)C2)=O)n1 c1(S)ccncc1OC.C(=O)(C(CN(C)C)NC(=O)C1CC1)NCCCOC c1(C(N2C(CN(C(CCCC(C)O)=O)C)CCCC2)=O)ccc(S(C)(=O)=O)o1 N1(C(CCNC(N)=O)=O)CC(NC(c2ccc(Br)o2)=O)CC2(CC2)C1 C1(N(CCCC)C(C2CC=CC2)=O)CCN(C(C2(C)CC(C)(C)C2)=O)CC1 C(=O)(C(C)C(C)(F)F)N(C)CC1N(C(C(CC=C)NC(C)=O)=O)CCCC1 C#CC1(C(=O)NCc2n[nH]c(C)c2C)CN(C(C2CCN(C)C2C)=O)C1 C(C(C)CC(=O)NCCN(C1CC1)CC)NC(C1CC(CC)C1)=O C1(O)(COC(N(C(C)C(Cc2ccccc2)C(=O)OC)CC)=O)CCS(=O)(=O)CC1 C1(C(=O)NCCC2CCN(C)C2=O)CC(O)CCN1C(C1CC(N=[N+]=[N-])C1)=O c1(CCC)sc(C(N2CCC(C)(c3cn(-c4ccccc4)nn3)C2)=O)cc1Br Cc1ccc(OCC(=O)O)c(NC(=O)CC23CCC(CC2C(F)(F)F)C3)c1 c1(SCC(N2C(C(=O)OC)CC2C)=O)ccc(O)cc1Br C(=O)(CCCCNC(N)=O)NCC1(O)CC(C(N(CC(C)(C)OC)C)=O)C1 c1(OC)cccc(C(F)(F)C(=O)NCC(C)CNC(C2(C(=O)N(C)C)CC2)=O)c1 C=CC(C)(O)C(=O)NCC1(NC(c2ccnc(OC)c2)=O)CC1 C(=O)(C(C#N)(CC)c1ccccc1)NCC1CC(F)(CNC(C(C=CC)O)=O)C1 C12(C(N(C)CC=CC(=O)NCCC(C)N3CCCC3)=O)CCCC1C2(F)F C(C)(CCCCNC(=O)C(C(C)C)c1ccncc1)NC(c1c(C)coc1)=O C1(CNC(C(COC)OC)=O)CC2CCC1N2C(=O)C=C(C)C C1(C(=O)NCC(N(C(COC(CC)C)=O)C)C2CC2)CCc2cncn2C1 c1(C(=O)NC(CNC(C2N(CC)CCCC2)=O)C(C)C)cnc2cnccc2c1 C1(CC)CN(C(=O)COc2ccccc2)CCN1C(=O)C(CCSC)NC(C)=O N1(C(C2OCCN(CC)C2)=O)CCOCC(C(=O)NCCCC(=O)NO)C1 c1(C(CCC(=O)N(CCNC(C2CC(SC)C2)=O)C)=O)csc2ccccc12 N1(CC)CCCC(CN(S(C)(=O)=O)Cc2ccc(F)c(Cl)c2)C1c1cnn(C)c1 Cc1cc(Cl)ncc1CC(=O)NCC1CCC(OC2CCCC2)CC1 CC(C)CC(=O)C(=O)NC(c1nocc1C(=O)NCCc1cnco1)C C1(C(=O)NCC2(F)CCC2)COC2(C1)CN(C(C1CCC(F)(F)C1)=O)C2 N1(C(C2CCC(CC)O2)=O)CC=CC(NC(=O)Cc2nncs2)C1 c1(OC)cc(C=CC(=O)NC2CCCCN(C(=O)C(C)(C)C(C)C)C2)ccc1F C(=O)(CCS(C)(=O)=O)NCC#CC(=O)NCC(c1ccsc1)C CC1CN(C(C2CN(C)CCN2C(=O)CCc2ccn(C)c2)=O)Cc2nncn21 CC(C)CC(O)C(=O)NC1CCC(F)(CNC(C23CCC(CC2)C3)=O)C1 N1(C(CCSCCCC)=O)CCN(C(=O)C2=CCOCC2)CC12CC2 Cc1ccc(C(N2CC3CC2CN3C(c2cnnc(O)c2)=O)=O)cc1N c1(C(N2CCC(C(N3CC(O)(CC(C)C)C3)=O)(OC)C2)=O)cccc(C#N)c1 C1(NC(c2n[nH]c(CC)c2Cl)=O)CCC2CCN(C(C3CCCC34CC4)=O)C12 N1(C(C=C(CC)CC)=O)CCCC1C(C)(C)NC(c1ccc(COC)s1)=O C(CS(=O)(=O)c1ccccc1)NC(C1C2CCC(C2)N1C(C1CCCCO1)=O)=O Cc1nnc2n[nH]c(NC(c3cc(N)ccc3[N+](=O)[O-])=O)c2c1C c1(C(N(CCCN(C(COC(CC)C)=O)C)C)=O)c(F)ccc2ccncc12 C1(NC(CC2ON=C(C)C2)=O)CC2(CCN(C(=O)CC3CCC4CC34)CC2)C1 C1(CNC(c2nc(C3CC3)cs2)=O)COCC1NC(=O)C(F)(F)C1(O)CCCC1 Cc1cc(C2CC2)ccc1C(=O)NC(C)CCCNC(C1CCCOC1)=O CC(C)C(C(=O)NCCC(F)(F)Cl)C(C)NC(=O)C(C)N=[N+]=[N-] C1(CNC(CC#N)=O)CN(C(c2cc(C(F)F)ccn2)=O)CC12CCOCC2 C1(CC(=O)N(C2(C(=O)NCCOCCN(C)C)CC2)C)OC(C)(C)OC1=O C#CC1(O)CCCN(C(C2CC(C)N2C(=O)COc2ccn(C)n2)=O)C1 c1(C(N2CCN(C)C(c3ccc(F)cc3)C2)=O)ccc2c(c1)C(N)CC2 C1(C(N2CCN(C(C(C(C)C)(C)O)=O)CC2CCO)=O)CCOC2(CCC2)C1 c1(C(=O)NCc2cccc(CN(C(C(CC)F)=O)C)c2)ccc(CO)cc1OC C1(CNC(CCn2ncc(C)c2)=O)CN(C(=O)CCC2CCCO2)CCCO1 Cc1c(C(=O)NC2(CO)CCN(C(C3C=CCCC3)=O)C2)cnn1CC(F)F Cc1nc(C(=O)NC2CCN(CCNC(C3CCC3C)=O)CC2)c(C)s1 N1(C(CCOCC#C)=O)CC(CO)C2(C1)CN(C(=O)C(O)CC1CC1)C2 c1(OC)cc(N)c(F)cc1C(N1CCCC(NC(C2CCCC2F)=O)C1)=O O=C(NNc1cc(F)c(F)cc1F)c1cnc(Br)s1 C(c1ccc(Cl)c(C(F)(F)F)c1)=CC(=O)NCC(CC)NC(C12CC(C)C1C2)=O C1(CCC(=O)NCCC(C)NC(C2(C3CCCO3)CCC2)=O)CCC(=O)C1 C=CCC(C)(CC=C)NC(=O)C(C(C)O)NC(=O)CCN1CCCC1=O C1(CNC(C=C(C)CNC(=O)CCC2CC(C)C2)=O)CCC(O)CC1 c1(NC(C23CC(C(N4CCSCC4)=O)(C2)C3)=O)c[nH]c2ccc(Br)cc12 C1(C(=O)NCCCN(C(c2c(NC)snc2C)=O)C)CCOC2(CCCCC2)C1 C1(NC(C(C)N(CC)CC)=O)CC2CC(C1)CN(C(=O)CCC1CCCCO1)C2 N1(C(C(C2CCCC2)OCC)=O)CC(NC(=O)CCSC)C(c2cnn(C)c2)C1 N1(C(CC(C)OC(C)(C)C)=O)CCOCC1C CC(C)CS(=O)(=O)CC(=O)NCC1CN(C(=O)COC2(C)CCC2)C2CC12 c1(OC)cc(C(=O)N(C(C)(C)C)CCN)c(-c2cc(SC)cc(F)c2)cn1 C1(C(=O)NCC(C(C)O)C)CCOCCN1C(=O)CC(C)(C)O N1(C(C2(C)CCC2)=O)Cc2cccc(CNC(=O)CCc3cccnc3)c2C1 CCCCC(CO)NC(=O)CC(CC)NC(c1sccc1CO)=O CC1OCCOC1C(=O)NC(C1CCN(C(C2C=CCCC2)=O)CC1)(C)C c1(CCNC(C(C2CC(F)(F)C2)OC)=O)c(Br)cncc1Br CCC(C)CCC(=O)NCCCN(C(=O)C(c1ccccc1Cl)O)CC C(=O)(CCCCN(C)C(C1CCCC1)=O)N(C(C=C)C1CC1)C C12(C(=O)NCCC(COC)OC)CC(CN(C(=O)CCCC(C)C)C1)C2 N1(C(c2ccn(CC)n2)=O)CCOCC1CC(=O)NCC(C)(O)C1CCCC1 C1(C(=O)NC2CCCC(NC(C3(CC#C)CCC3)=O)C2)CCC(C)(O)CC1 CC(CCN=c1ccnc(NC2CC2)[nH]1)C(F)F.c12cccc(c1)S(=O)(=O)NC2 C1(CNC(CNC(N)=O)=O)CN(C(c2cc(C3CC3)cs2)=O)CC1(F)F C(=O)(CCCCCF)NCC1(CN(C(c2ccc(OCC)nc2)=O)C)CC1 c1(CC)ccc(C(=O)NC(C)C(CO)NC(c2cn(C)nc2OC)=O)c(C)n1 N1(C(C(CSC)C)=O)Cc2nccn2CC(NC(C2(C3CC3)CCCO2)=O)C1 N1(C(C(SC)SC)=O)C2CCCC1CN(C(c1cc(C#N)c[nH]1)=O)C2 CN1CCN(C(=O)CCc2cnccn2)C(C(=O)NCC2(C3CC3)CCC2)C1 C(C(CC(C)C)NC(C1CCCN1CC)=O)NC(C=CCC)=O N1(C(CC(C)(C)C)=O)CC2(CNC(c3ccc(Cl)cc3)=O)CC1CO2 C(C(C)(C)C(=O)NCC(C(C)(C)C)NC(=O)C(C)CN1CCOCC1)NC(C)=O c1(CC(=O)NCCC(C)NC(c2c(SC)cnn2C)=O)ccc2sccc2c1 C1(C)(CNC(C(C)(C)OCCC)=O)CCN(C(C2CC2C2CC2)=O)C1 c1(C(=O)NC2CCCCC2NC(c2cccnc2O)=O)cc2c(nn1)OCCS2 c1(C(N(CCc2cn(-c3ncccc3C)nn2)CC)=O)cc2cc(O)ccc2[nH]1 N1(C(C(C)=C(CC)C)=O)CCN(C(=O)Cn2nnc(C)n2)CC2CCCCC12 C(=O)(CC1OCc2ccccc21)NC1(C)CC(NC(=O)Cc2ccccc2O)C1 N1(C(c2cnc(C)s2)=O)CCC(NC(C2(F)CCS(=O)(=O)C2)=O)CC1C c1(C(N(CCCNC(COCCC)=O)C(C)C)=O)cccc2[nH]c(C)cc12 c1(C(=O)OC)cccn(CC(=O)NCC(F)CNC(=O)CC2(C)CC2)c1=O c1(C(=O)NC(C)CN(C)C(c2ccn3c2CSCC3)=O)cc2nn[nH]c2cc1F N(C1CCCc2c1cnn2CCO)C(C(n1cc(-c2n(CC)ncc2)nn1)C)=O Cn1[nH]c(=NC(=O)C2CC(F)CN(Cc3cc(Cl)cnc3Cl)C2)cc1Cl CCCC(CNC(C1CCC(=O)O1)=O)C(=O)N1CCCC1(CO)CO c1(NCc2cncc(OC)c2)cnc(F)cc1C(=O)Nc1c(C)cccc1Br C(=O)(C1CCc2ccccc21)N1CC(NC(CCc2c(C)noc2Cl)=O)(CO)C1 C1(CNC(CC(CC)SC)=O)C(OC)C(OC)CN1C(=O)CP(C)(C)=O c1(C(N2CC(NC(CCC(C)SC)=O)C(SC)C2)=O)cc2ccc(F)cc2o1 N1(C(C(C(C)C)O)=O)CC(C(N2CC(O)CC2(C)C)=O)CC(F)(F)C1 c1(C(N2CC(CN(C(C=CC(CC)C)=O)C)OCC2)=O)cn2cccc(F)c2n1 N1(C(c2c(CC)n(C)nc2)=O)CCN(C(=O)C=Cc2ccn(C)c2)C2CC12 c1(C(N2CC(N(C(c3c(CC)nnc(C)c3)=O)C)C2)=O)[nH]c2ccccc2c1C Cc1ccc(N)c(C(=O)NCC23CC(C2)C(NC(c2csnn2)=O)CO3)c1F c1(C(N2CCC(OC)(CNC(=O)C=C3CCOCC3)C2)=O)cnc2ncccn12 CN1CCN(C(c2ccsc2C(=O)NC2CC2)=O)CC1NC(=O)C(=O)N(C)C C(C(C)(C(=O)N1CCCC1C(=O)N(C1CC(CO)C1)C)OC)OC C1(NC(CC2CN(C)CC2O)=O)CCCCCN(C(=O)Cc2cncc(F)c2)C1 C(C(=O)N1CC(CCNC(C2CCN(C(=O)N(C)C)CC2)=O)C1)(C(C)(C)C)SC c1(NC(C2CCOCC2)C(=O)NC)ccc(F)c(S(N)(=O)=O)c1 N1(C(c2scc(OC)c2)=O)CCOC(C(C)NC(=O)CC2CC3CCC2C3)C1 CC(CC(C)(C)C)C(=O)NCCCN(C(=O)Cc1ncn2c1COCC2)C C1(S(N)(=O)=O)(C(=O)NC(CCNC(c2cc(C)oc2C)=O)C)CCCC1 c1(C(=O)NCC(CNC(CN(C(COC)=O)C)=O)C)cc(COCC)no1 c1(OCC(=O)NCC2(F)CCOCC2)cccc(C(F)(F)F)c1.C12CC1NC2=O C1(NC(=O)Cn2cnc(Br)n2)CCN(C(=O)CCn2cncn2)CC1O c1(C(=O)NC2C(C)CCN(C(=O)C(C)(Cl)Cl)C2)cc2n(n1)CCNC2=O c1(C(C)(C)NCc2ccc(N3CC(C)OCC3)cc2)cccc(C#N)c1 c1(C(N2CCC(n3cc(CNC(C4(O)CC4)=O)nn3)C2)=O)cc(Br)no1 N1(C(c2cc(OC)ns2)=O)CC(C2CCCCN(C(c3csnn3)=O)C2)C1 N1(c2nc(SC)nc(O)c2)CCC(NC(c2[nH]nc([N+](=O)[O-])c2Cl)=O)C(C)(C)C1 Cc1nc(-c2ccc(Cl)s2)sc1C(=O)N(CC(C1CCCC1)O)C N1(CCNC(C(c2cnn(C)c2)NC(c2c(C)non2)=O)=O)CCOCC1=O C=CCCC(c1nnnn1C(C)C(=O)OC)(C1CC1)NCc1ccccc1Cl Cc1nc(N2CCC(NC(=O)CC3CCCC(C)C3)C2)ncc1Br c1(C(=O)NCC2N(C(c3cn(C)nc3)=O)CC(O)C2)ccc(N)c(C(F)(F)F)n1 C1(NC(C2C(OCC)C2)=O)CCCCC1CNC(c1cc(C(C)(C)C)nn1C)=O c1(NCCC2N(C(c3cnccn3)=O)CCCC2)nc(Cl)nc2[nH]c(O)nc12 c1(C(N(C(C)C)CCNC(c2sccc2C(F)F)=O)=O)cccc2c1COCC2 CC(CC(=O)N1CCOC2(CCC2)C1)C(C)(C)NC(=O)CC1CNC(=O)O1 C1(NC(C2(CC=C)CCC2)=O)CN(C(C2CCC2(C)C)=O)C2CCCCC12 Cc1cc(C)c(C(N2CC3CCC3(CCNC(=O)C(=O)NC(C)C)C2)=O)c(O)n1 N(C)(C1CN(C(=O)COC)CCc2ccccc21)C(C=C(CC)C)=O C1(C(=O)NC)CN(C(=O)NCC2CC2(C)C)c2ccccc2O1 c1(C(N2CCC(NC(c3cncc(Cl)c3)=O)(CO)C2)=O)cnc2ccccc2n1 C1(C(=O)Nc2ccc(O)nc2)CCCC12CCN(Cc1ccccc1I)C2 CC(Cc1cccs1)CN=c1nc(N2CCC(F)(CN(C)C)C2)c2c([nH]1)CCOC2 N1(C(C(C(C)O)C)=O)CC2CN(C(c3csc(Cl)c3)=O)CC(C1)O2 N1(C(=O)NC2(C(=O)O)CC(=O)NC2)CC2CN(C3CC3)CC2C1 Cn1cc([N+](=O)[O-])cc1C(N1CCN(C(=O)Cc2nc(=N)[nH][nH]2)C(CF)C1)=O N1(C(C(CC(C)C)OC)=O)CCC(C(=O)N(C)OCC(F)(F)F)C(C)(C)C1 Cc1ccc(C(=O)NC2CCCCC2C(=O)NCCCC#N)c(I)c1 CCCCC(CNC(c1coc(C(N)=O)c1)=O)NC(=O)Cc1cnc(C)s1 c1(C(=O)NCC(C)N(C(CCCN(C(C)=O)C)=O)C)cc(C)cc(O)c1 C1(CN(C)CCF)CNCCOC1 Cc1cncc(C(N2CCOC(CCNC(=O)Cc3ccc(C)s3)C2)=O)n1 c1(C(=O)NCC2(CF)CCC2)cncc(-n2cccn2)n1 c1(N2CCN(Cc3cn(CCO)nc3)CC2)nccn2cnnc12 C(=O)(CCC1=NNC(=O)CC1)N1C(CNC(C2(CO)CCC2)=O)CCC(C)(C)C1 c1(C(N2CC(CNC(c3nccc(Cl)c3F)=O)C2)=O)c(F)ccc2occc12 CC(C)(O)CC(=O)NC1COCC1NC(C1(c2ccnc(Cl)c2)CC1)=O N1(C(c2cc(C)sn2)=O)C2CCC1CC(C(N1CCC3(CCCO3)C1)=O)C2 C1(CC(=O)NCCC2CC(C(=O)NC3CC3c3cncs3)C2)CCCOCC1 N1(C(=O)Cn2cc(CC3CC(Cl)(Cl)C3)nn2)CC(O)CC1C1CC1 C#CCC(C)(C(=O)N1CCC(O)C(CO)C1)NC(C1C=CCC1)=O C=CC1(CC(=O)NCC(C)OC(F)F)CN(C(c2coc(C(F)F)c2)=O)C1 c1(-n2cc(CCCC(=O)NC(CC(CC)C)C(=O)O)nn2)c(F)c(F)cc(F)c1F c1(C(N2CCCCC2C(=O)O)=O)cc(Br)c(F)cc1Cl.N12CCC1C2=O c1(C(N2CC(F)CC(C(=O)NCC3(CO)CCC3)C2)=O)ccc2c(Cl)ccnc2c1 N1(C(Cc2nc(C)[nH]n2)=O)CC2CC(NC(C3CCCC34CCC4)=O)C2C1 c1(NC(c2occ(C)c2)=O)ncc2c(Cl)cccc2n1 C=CCC(C(=O)N(CCN(C(=O)C1=CCCS1)CC)CC)C(C)C c1(CCC(=O)NC(C)C(C)NC(=O)CC#N)cnn(-c2ccccc2)c1 c1(C(N2CC3(C(C(N4CC(=O)NC4)=O)C3)C2)=O)cc(Cl)cnc1Cl n1(CC(=O)NC(CC)CN(C)C(C2CC(F)(CO)C2)=O)nc(C)c([N+](=O)[O-])c1C C1(C(=O)NCc2ccc(Cl)cc2Br)CC12CCN(Cc1ccc(C(=O)OC)[nH]1)C2 C(c1cnc(C)nc1O)=CC(=O)NC1CC(CNC(c2oc(CC)c(C)c2)=O)C1 c1(C(N2CC(CNC(=O)C3=COCC3)C3(C2)CC3)=O)ccnc2ccccc12 c1(N)nnc2ccc(C(F)(F)F)cn12.c1(NC(C)C(=O)NCCO)ccc(Cl)cc1 CCC(C#N)C(=O)NC1(C(=O)NC2C=C(C)CCC2)CCOCC1 N1(C(c2scc(C)c2)=O)CCN(C(c2ccc(C)o2)=O)CC1C#N c1(C(=O)NCCC2(O)CN(C(CN(CC)CC)=O)C2)ccc(C#N)nc1O c1(C(=O)NC2CCOCC2NC(C2CSCCS2)=O)ccc2nn[nH]c2c1 CC1CN(C(C2(C(N)=O)CCC2)=O)CCC1NC(C1CN(S(=O)(=O)C(F)F)C1)=O Cn1c(-c2nc(C(C)C3CC3)nn2CCC(C)(C)C)cc2ccsc12 Cc1ncc(C(=O)NCCc2cn(CC3CCC4CC4C3)nn2)c(O)n1 Cc1cc(NCC2CCCN(C(c3conc3C)=O)CC2)n2ncnc2n1 C1(C(=O)NC(c2cc(OC)c(O)cc2)C(=O)O)CC2(C1)C(C(=O)O)C21CCC1 CCCC(O)C(=O)NCC(CC)NC(=O)CC1(C(F)F)CC1 N1(C(C(C)=C2CC2)=O)CC(CNC(c2ocnc2-c2ccccc2)=O)CCC1C c1(N(CC(=O)N(C(CN(C(COC(C)C)=O)C)C)C)C)ccc(Cl)cc1 N1(C(CNC(=O)NCc2ccco2)=O)CCC2(CC1)CC(C(=O)O)CO2 CC1(C)CCC(C(=O)NC2CC(C(F)F)(NC(c3ccc(O)cc3)=O)C2)CC1 N1(C(c2cc(COC)[nH]n2)=O)CC(O)CC1C(=O)NCCNC(=O)OC CC1(C)CCC(C(=O)NC2CCCC2CF)(NC(=O)COC2CCC2)C1 N1(C(=O)NC2C(C(=O)OCC)COCC2)CCC(C)=C(C)C1 c1(C(=O)NCC(CC)NC(=O)C(N2CCCCCC2)C)cnc2n1CCCCC2 CC(C)C(C#N)C(=O)NC1(C(N2CCCC(CCCO)C2)=O)CC1(C)C Cc1cc(Br)c2ncnc(NCc3sccc3C(F)(F)F)c2c1 c1(C(=O)NC2(C)CN(C(C(CC)Sc3ccccc3)=O)C2)nc(C(C)=O)sc1C C1(COC)CC(CNC(=O)C(c2ccc(Cl)cc2)=O)N(C(=O)Cc2cn[nH]c2)C1 c1(OC)ccc(C(N)=O)cc1C(=O)NC1CCCN(C(C2CC2OC)=O)C1 CC1CCN(C(=O)CN(C)C(N)=O)C(CNC(C2CCC3(CCC3)C2)=O)C1 Cc1nc(Cl)c(NC(C2CC(F)CN(C(=O)C3CC3)C2)=O)c(Cl)n1 N1(C(C2CCN(CC)C2)=O)CCC(C(N2CCC3(CCCO3)C2)=O)CC1(C)C c1(C(=O)NC2(CN(C(C(C)Cn3cccn3)=O)C)CC2)cc2n(c1)CCOC2 c1(N2CCC(NC(c3ccc4cncn4c3)=O)C(F)C2)ncnc2cccnc12 c1(OC)nsc(OC)c1C(=O)NC(C)CCN(C(=O)Cn1cnnn1)C N1(C(CCOCC)=O)CCC2CCN(C(=O)C(c3ccccc3F)(C)C)CC2C1 C1(C(N2CCN(C(c3cc(C)no3)=O)CC2)=O)Cc2ccccc2C1C C1(CC)CN(c2nnc(C(c3ccccn3)(F)F)n2CCC(=O)NC)CC(C)O1 c1(NC(C2CC3CC2(c2cccnc2)C3)=O)c(Cl)cc(I)cc1Cl C(=O)(C(=O)C(F)(F)F)N(C1C(N(C(C(C2CCC(=O)N2)C)=O)C)CCCC1)C C1(NC(c2cccc(OC)c2)=O)CCN(C(=O)Cc2ccc(O)cn2)C(C)C1 c1(CC(=O)NC2CC(CNC(C3C(COCC)C3)=O)C2)c(Cl)cnn1C CC1CN(C(=O)CCN(C(c2ncccc2O)=O)C2CC2)CC(=O)N1 CC1CN(C(=O)CC(C(F)(F)F)c2ccccc2C(=O)O)CCC12CCOC2 C(=O)(CC1CCc2ccccc21)NCC1CC(C)(C)N(C(c2csc(F)c2)=O)C1 C#Cc1cnn(CC(=O)NC(CNC(=O)COCC2CCOC2)(CC)CC)c1 C1(C(=O)N(CCC(C)NC(=O)CCC(C)CN(C)C)C)(OC)CCC(C)(C)CC1 N1(C(C(C)OCC)=O)CCC(C)(C)C(NC(c2cnc(SC)[nH]2)=O)C1 C1(C)(NC(c2cn(C)nc2)=O)CCCN(C(c2cnn3c2OCC3)=O)C1 c1(N2CCC(c3nc(=N)[nH][nH]3)C2)nc(=N)[nH]c(=NCCS(=O)(=O)CC2CC2)[nH]1 C1(N(C(c2c(-c3cncc(C)c3)nccc2)=O)C)CCCCN(CCO)C1 C(CC)(CCCC(=O)NCC[Si](C)(C)C)NC(C1(CC=C)CCC1)=O CCC(C)CC(=O)N1CCC(CCC(=O)NCC2(C)CCCO2)CC1 C12(C(=O)NC3CC4C(NC(CCC(=O)N(C)C)=O)C4C3)CCCN(CC1)C2 N1(C(c2nc(CCC)sc2)=O)CCn2c(CNC(C3C=CCC3)=O)nnc2C1 N1(C(CCOCCOC)=O)CCC(O)(C(C)NC(c2cc(C(C)=O)cn2C)=O)C1 c1(C(=O)NCC(C)(C2CCC2)NC(C23COC(CCO2)C3)=O)cc(F)cnc1O C1(C(=O)NCCC(CNC(CSc2cccc(C)c2)=O)O)CN2CCN1C(C)C2 N1(C(CC(C(C)C)NC(c2ccc(CC)s2)=O)=O)CCC2(CCC2)C(O)C1 c1(SCC(N2CC3C(NC(C=CC(=O)OCC)=O)(C3)C2)=O)ccc(C)cc1C Cn1cc2ccc(C(=O)NC3COCCN(C(=O)C(C)(C)CCl)C3)cc2n1 CC1CC(NC(c2ncoc2C(C)(C)C)=O)CN(C(=O)C=C2CCN(C)C2)C1 C(N=c1[nH]c(N2CC34CCCC3(COC4)C2)nc2c1CCC2)C1(COC)CCC1 N1(C(C(C(C)O)N(C)C)=O)CC2(C1)SCCC2NC(c1cc2cnccc2o1)=O N1(C(C(CC)C#N)=O)CC(C2CCCN(C(=O)CNC(c3ccco3)=O)C2)C1 N1(C(C2C(C)(C(C)C)C2)=O)CCC(CF)(NC(=O)C(C)Cc2ccccc2F)C1 CCCCC(C(=O)N(C)CC1CCCN1C(c1ccc(O)c(Cl)n1)=O)NC(N)=O C1(C)(CC(=O)NCC2C(C)CCN(C(=O)CCC(F)F)C2)Oc2ccccc2O1 N1(C(CCCC2(NC(=O)CC3CS(=O)C3)CCC2)=O)CC2CSCC2C1 c1(C(N2CCC(C(=O)Nc3ncc(C)cc3Cl)C(O)C2)=O)ccc(I)c(F)c1F c1(CNC(C2CC(OC)(OC)C2)=O)ncccc1C(=O)NOCCC1CC1 Cc1sc(C)c2sc(C(=O)NC3CN(C(C4(F)CCCC4)=O)CC3C)cc12 N1(c2ccnc(NC3C(CCCC)CCC3)n2)CCC2(CC1)CCN(C)C2 c1(C(N(C2CCN(C(CCC=C=C)=O)CC2)CC)=O)cc(C(=O)OC)cc(F)c1F C1(C(=O)NCC(C)N(C(=O)CCc2cn(C)cn2)C)CCNC(=O)C1 C(=O)(C1=COCCO1)N(C(CNC(c1c(C)c(C2CC2)on1)=O)C1CC1)C N1(C(C2C(OCC)C2)=O)CC2C(N(C(=O)CCc3ccsc3Cl)C)C2C1 N1(C(c2nc(CC)oc2C)=O)CCCC1C1CCCN1C(c1cccnc1C)=O N1(C(CC2CCN(C(C3(C)CNC(=O)N3)=O)C2)=O)CC2CC(O)CC1C2 c1(OC)cc(C(N2CC(O)(C3CCC(=O)N3)C2)=O)sn1 C#CC(CC(C)(C)C)NC(=O)C(CCOCCO)NC(c1cccc(CO)c1)=O Cc1cc(C(=O)N(CCC(C)NC(C2CCC(=O)N2C2CC2)=O)C)oc1C N1(CC)CCN(N2CCC(S(=O)(=O)CC(=O)NC)CC2)CC1=O Cc1nc(O)sc1C(=O)NC1CCCCC1CNC(c1cc(C(N)=O)c[nH]1)=O C(=O)(C(=O)N=S(C)(C)=O)NCC1C(NC(c2ccc(COCCOC)cc2)=O)C1 CCC(C)(CCC(C)C)C(=O)N1CCn2cc(C(=O)Nc3cnnn3C)nc2C1 C(=O)(C(O)C1=CCCCC1)NC(C)(CO)C(=O)NCC1(O)CCOC1 S(=O)(=O)(c1cccc(C#N)c1F)Nc1cnc2ccc(C)cn21 c1(C(N2C(CNC(CS(CC)(=O)=O)=O)CC(F)C2)=O)cc2cccnc2[nH]1 Cc1ccc2c(=NC(C)C3CCCO3)[nH]c(=NCCc3cc[nH]n3)[nH]c2c1 S(=O)(=O)(c1cc(F)c(F)c(F)c1F)CCCCCC(c1c[nH]c2ccccc12)=O CC12CCC(C(=O)NCC3CC3NC(=O)Cc3csc(-c4ccoc4)n3)(C1)OC2 CC(C)(CCCNC(C1COCOC1)=O)C(=O)N1CC(CO)C(O)C1 N1(C(C(COC)C)=O)CCC(CC(N2CC(c3nncs3)C2)=O)CC1 C(C)(C(=O)NC1CC(OCC(=O)N(C)C(c2cccs2)C)C1)OCOC c1(OC)ccc(C(=O)N(C)CCCN2CCC(O)(CC(=O)O)C2)cc1-c1cc(F)ccc1C C1(NC(C2CC23CCC3)=O)CCN(C(=O)CCC2CCOCC2)C(C2CC2)C1 c1(-c2n(C3C(C)OCC3)nc(Cc3cnn(C)c3)n2)noc2c1CCCC2 c1(NC(C(CCC)C)C)ncccc1S(=O)(=O)N(C(CF)CF)C c1(-c2cc(C)c(O)cc2)ccc2ccnc(NCc3cn[nH]c3)c2c1 C1(N(C(c2n(CC)cnn2)=O)C)CN(C(=O)C=Cc2cn(C)nn2)CC1(C)C CC1C(NC(=O)CC2OCCCC2(C)C)CCCN1CCn1nnnc1C1CC1 CCCCN=C(NCCc1ncccc1C)NCCC1CCC2(CC1)CC2 C(C(C)(C)C(=O)NC(C)CC(C)O)NC(CNC(=O)NC)=O N1(C(C(=O)NCC2CC2)=O)CCOC2CCN(C(C3CCCNS3(=O)=O)=O)CC12 c1(OC)cc(O)ncc1C(=O)NC1CCCN(C(C2CCCC3CC23)=O)C1C C(=O)(C1=CCCCC1)NC(CNC(c1c(C)cnn1C)=O)(C)C1CC1 C1(NC(C(CC)F)=O)CN(C(=O)C=C2CC3CCC(C2)N3C)C2CCCCC12 N(C(=NCCC(C)=O)N1CCCC(CO)(CO)C1)CC(=C)CC c1(C(N2CCN(C)C(CNC(C3CC4(CCC4)C3)=O)C2)=O)[nH]cc2c1CCCC2 N1(C(C2C(C(C)O)C2)=O)CCC(NC(c2cncc(Cl)c2Cl)=O)C2(CCC2)C1 c1(C(=O)NCC(C(C)C)NC(C2C(C=C)C2)=O)cnc(C)nc1C CCCC(C)(O)C(=O)N1CCC(C2CCCN2C(=O)Cn2ccnc2C)CC1 c1(C(=O)NC2C=CC(CNC(=O)CCOC3CCC3)C2)ccc(O)c(F)c1 N1(C(CCC2(C)CC2)=O)CCC(c2nnc(CNC(=O)CC(C)(F)F)s2)CC1 N1(CC(CC)C)CCC2CCC(C1)N2C(c1cncc2[nH]ccc12)=O c1(C(=O)NC2CCN(C(c3cccnn3)=O)C2)ccc(C(F)(F)F)nc1O c1(C(=O)NC2(CO)CCCN(C(C(CCC)C#N)=O)C2)ccc2c(c1)COCC2 C(C)(C(=O)N(C)CC1CCCN1C(c1ccnc(F)c1F)=O)(C(C)C)NC(C)=O c1(C(=O)NCCC2CCN(C(C=CCCC)=O)C2)ccc2ccc(Br)cc2n1 C1(n2cc(C34N(C(C(CCC)CCO)=O)CC(C3)C4)nn2)CCC(F)(F)CC1 CC(CC(=O)N1CCCC(NC(=O)CCC2OCCO2)C1)CC(F)(F)F CCCCCCC(C(=O)NCCN(C(c1c[nH]c(=N)s1)=O)CC)NC(C)=O c1(C(=O)NCC2CC(CNC(=O)OC(C)(C)C)C2)cc(CSC)no1 Cc1cc(C(=O)NC23CCC(NC(C45CC(CO4)C5)=O)(CC2)C3)ccc1F C#CC1(C)CCCN(C(C23CN(C(=O)OC(C)(C)C)C(CF)(C2)C3)=O)C1 CCCC(C(=O)NC1CN(Cc2noc(C(C)C)n2)CCC1C)C(C)C c1(C(=O)NCC(CCC=C)O)cc(C#N)cc(C#N)c1 c12cccc(c1F)NC(=O)C13CC(C1)(C3)NC2=O.c1(CC)cnccc1N(C)C C(CCN=c1nc2scnc2c(NC2CCCC23CC3)[nH]1)N1CCC(C)CC1 Cc1cncc(CNC(C2CC(O)CN2C(=O)C=C2CCOCC2)=O)c1 N1(C(=O)Nc2ccc(SC)s2)CCCC2C1CCN2C(=O)CC1CCN(C)CC1 c1(CC2N(C(C(C)N(CCC)C3CC3)=O)CCC2)cccc2ccccc12 C12(C(=O)OC)CN(C(c3cnc(C)nc3)C(=O)NC3CC3)CC(CO)(C1)C2 C1(C(=O)NCC(C)(C(C)C)NC(Cc2c(C)cccc2)=O)CC2C(C1)C2(F)F N#Cc1cccc(NC(=O)CC2CCN(C(c3cc(O)ccc3I)=O)C2)c1 C1(C(=O)NCCN(C(CCCOCC)=O)C2CCCC2)Cc2cccnc2C1 N1(CC)CCC(C(=O)N(CCCNC(c2ccnn2C(C)CC)=O)C2CC2)C1 c1(N(C(c2cc(-c3cnn(C4CCCC4)c3)cs2)=O)C2CC2)c(O)ncnc1O O=C1CC(C(N2CCCCC(NC(c3cnn4c3SCC4)=O)C2)=O)CC(=O)N1 CCC(CC)C(=O)N(O)Cc1cn(C(C)C(N2CCCCC2)=O)nn1 c1(C(N2CCC(C(C)NC(C(CC)NC(C)=O)=O)C2)=O)c(Cl)nn(C)c1Cl Cc1ccc(C(C(=O)NCc2cccs2)N(C2C3COCC23)C)nn1 c1(N2CCCC(C)(CC)CC2)cc(Br)ccc1S(=O)(=O)NCC1CCC(O)CC1 c1(C(N2C(CNC(C(CSC)OC)=O)CC(OC)C2)=O)cn2ccc(F)cc2n1 C1(C(=O)OC)C(F)(F)C12CC(C(=O)NCC1CCC3COCC3O1)C2 N1(C(=O)Cn2ccnn2)CC2CCC(C1)N2C(C1CC(O)C(F)C1)=O C1(C(=O)NC2CNCC(C#C)C2)CCN(C(=O)OC(C)(C)C)C12CCSCC2 c1(CCC(=O)NC(C(C)NC(C2=C(C)OCC2)=O)C)c(O)nc(=N)[nH]c1C N1(C(C2N(CCC)CCC2)=O)CCOC(C(N2CCC(F)CC2)=O)C1 c1(OC)cc(CNCC23CC2CN(C(c2cncc(Cl)c2C)=O)C3)cc(Br)c1O C1(C(=O)NC2CCN(c3snc(CCOC)n3)CC2O)Cc2ccccc2CO1 CCC(CNC(=O)C=C(C1CC1)C1CC1)(CC)C(=O)NC(C)COC(C)C C1(CC(N2CCC(CN(C(=O)CC3C=CCCC3)C)CC2)=O)CCCCC1(F)F c1(OC)cc(NC(=O)COC(c2cc(C)cc(O)n2)=O)c(Cl)cc1Cl C1(CCCC)CN(C(c2ccon2)=O)CCN1C(=O)C(C(C)C)NS(C)(=O)=O C1(C(=O)NCC(CN(C(C(CC)F)=O)C)C)CCc2ccccc2O1 c1(C(=O)NCCC(C)NC(C(CC)OC)=O)nc2ccccc2nc1C(F)(F)F C1(NC(C23CC(C)C2C3)=O)(CNC(c2cccc(CO)c2)=O)CCOCC1 c1(C(N(C2CCC(NC(=O)C(F)=CCCF)C2)C)=O)ccc(P(C)(C)=O)s1 C1(N(C(CN(C(C(F)=CCC)=O)C)=O)C)CC(C)OC(C)C1 Cc1ccc(Cl)c(OCC(=O)NC2CC(NC(=O)CC3CCC3C3CC3)C2)c1 c1(C(N(CCCCC(N2C(C(C)O)COCC2)=O)C)=O)cn2c(n1)CCC2 N1(C(C(C)CO)=O)CC23CCCCC2(C1)CN(C(=O)Cc1cscn1)C3 c1(OC)cc(N)ccc1C(=O)NC1CCCC1NC(=O)C(C)CF c1(C(N2CCC3(NC(Cc4nc(C)sc4)=O)C(C2)C3)=O)cc([N+](=O)[O-])ccn1 N#Cc1ccc(CN2CC3(CC3C(=O)Nc3cnn4ccccc34)C2)cc1F c1(-n2ccc(C(=O)NCCN(C)C(C34CCCCC3C4)=O)n2)ccccc1F N1(C(c2c(CC)n[nH]c2)=O)CCC2C(C(=O)NC(C)C(C)(C)CC)C2C1 N1(C(c2ccc(C3CC3)s2)=O)CCOCC1CC(=O)NC1CC(CCOCC)C1 C1(n2c(N(C)C(=O)OC)nnn2)CCN(C(=O)Nc2ccccn2)CC1 Cn1c(C(=O)NCC2(C(C)(C)C)CCN(C(c3csc(O)n3)=O)C2)cnc1Cl c1(C(=O)NC2CC(F)(CNC(c3cnsc3)=O)C2)cncc2[nH]ccc12 c1(C(=O)NC(CC(C)NC(c2cn(CC)nc2C2CC2)=O)C)cc2ccsc2[nH]1 C(CCCCCN(C(=O)C(F)CC)C)NC(c1nc(CCCCC)sc1)=O N1(C(C2(CSC)CCCCO2)=O)CC2CCCC2(c2noc(C(C)OC)n2)C1 CC1C(=O)NC(=O)CN1C(=O)C(CO)NC(=O)Cc1ccoc1 C1(C(N2C(C(=O)NCc3ccn(CC)n3)COCC2)=O)CC(C)(C)CN1C c1(C(N2CCN(C(C3CCC(F)(F)C3)=O)CC2)=O)ccc(I)cc1[N+](=O)[O-] C(CC(C)C)(C(=O)NCCCCC1CC1)N(C(C(C(C)C)NC(C)=O)=O)C Cc1cnc2ccccc2c1C(=O)NCC1(O)CC(NC(=O)CNC=O)C1 C1(C(N(CCCOC(C)C)C)=O)CC(C)(C)CN1C(=O)CC1COCCO1 CC1CN(C(c2ccccc2C(N)=O)=O)CCN1C(c1cccnc1N)=O c1(OC(C)C)cccc(C(C)Nc2nnc(N(C)C)n2C)c1 C1(NC(C(=O)Nc2c(C)occ2)=O)(CO)CCCN(C(=O)C(C)CSC(F)(F)F)C1 c1(NC)ncccc1C(=O)NCC(C1CC1)N(C)C(c1sc(N(C)C)nc1Cl)=O c1(CN2CCC(Nc3nc(OC)c(F)cn3)CC2)cccc([N+](=O)[O-])c1 n1(CC(N2CCCC(C)(CNC(C(CCC)O)=O)C2)=O)c(C)nc2ccccc12 c1(CC)cnccc1C(=O)N(CC(C)(C)CNC(=O)C(O)C1CC1)C N1(C(CC(=O)OC)=O)CCN(C(C2CCN(S(C)(=O)=O)C2)=O)C(C2CCC2)C1 C1(F)(C(N2CC(CC(=O)OCC)C2)=O)CN(C(=O)C(C)OC(C)=O)C1 c1(C(=O)NCCC(C)N(C)C(C2Cc3nccnc3C2)=O)ccc2cncn2c1 Cc1nc(C)n(CC(=O)NCC2(C)CC(NC(=O)CC3(C(F)F)CC3)C2)n1 CC(C)C(C(=O)NCCc1cncs1)C(C)NC(c1ccsn1)=O c1(NC(N(C(c2ccccc2Cl)C(=O)O)C)=O)ncnc2c1nc(N(C)C)n2C N1(C(CCCOCC=C)=O)CCC2(CCC2)C(NC(=O)CC2CCC(=O)C2)C1 C1(CNC(C(C)SC)=O)CCCC2CN(C(=O)C=CC3(C)COC3)CC12 C=C(Cl)CCC(=O)NCC(C1CC1)NC(=O)C(C)Oc1cccc(C(C)C)c1 c1(NC(=O)NC2C(c3ccc(C(=O)OCC)o3)C2)cc[nH]c(=N)n1 C1(NC(=O)CC2CCC3CC23)CCCN(c2ccc(C3CCC3)cn2)C1 C1(O)(C(=O)NCC2(C)N(C(CC(C)F)=O)CCC2)CCCCCC1 C(C(=O)NC(COC)CC(=O)N1CCCCC1)(C(C)C)OCC N1(C(C2C(C)(C)C2)=O)CCCC1(C)CNC(c1cc(Br)ccn1)=O C1(NC(COC)=O)CC2(CCN(C(c3ccnc(N(C)C)c3)=O)CC2)C1 C(=O)(C1=CC2(CCOC2)C1)N1CCCC(CNC(CCCC#N)=O)C1 c1(OC)ccc(Br)c(CCC(=O)N(C2CCOC2)C2CCC2)c1 C(=O)(CC(C)(C)CNC(C1CC(C)(C)C1)=O)NC(c1ccnn1C)C C1(NC(CN2CCN(C)CC2)=O)CN(C(c2ccc(O)nc2)=O)CC1N=[N+]=[N-] CCC(CCC(=O)NCC(CC)(CC)OC)NC(=O)C(C)(O)COC C1(O)(C(N(C)CC2(CNC(c3cc(C)oc3C)=O)CC2)=O)CCCC(C)(C)CC1 C1(C(=O)NCC2(F)CN(C(c3n(CC#C)ccc3)=O)C2)CCCCC1(F)F N1(Cc2cn(CC3CNC(=O)O3)nn2)CCCC(NC(c2ncc[nH]2)=O)C1 C12(C(=O)NC3CC(NC(c4c(NC)nccc4)=O)CC3O)CCCN(CCC1)C2 Cc1cccc(C2(NC(c3ccc(C)n3C)=O)CCC(NC(=O)C(C)N=[N+]=[N-])C2)c1 C1(NC(CCC=C)=O)COC2(CCN(Cc3cccc4cccnc34)CC2)C1 c1(OCC)ncc(C(=O)NC2CC(CCNC(=O)CC3C(=O)NN=C3C)C2)cn1 C1(OCC)(CNC(c2sc(C)nc2NC(c2ccco2)=O)=O)CCCSC1 C(=O)(CCC1=CCCCC1)NC(CCC)CC(=O)NCC1CC(CC)C1 CC1=C(C)CC(C(=O)N(CCCNC(c2cc(O)cnc2Cl)=O)C)CC1 CC(C)C(C)CC(=O)NCC(C)C(=O)NCCCn1ccnn1 n1(CC(=O)NC2CC(NC(C=C(CCC)C)=O)C2)c(C2CC2)nc2ccccc12 C(=O)(N1CCCc2nncn21)C1C(c2c(-n3c(C(=O)O)nnn3)coc2)CCCC1 c1(C(N2CC3(OCC(NC(CC4(C)CC4)=O)C3)C2)=O)cnc2c(c1)NC(=O)CS2 N1(C(Cc2cccc(C)c2F)=O)CCCCCC(NC(c2onc(C)c2C)=O)C1 C12(C(N3CCCC(C)(NC(=O)CSCCC#N)C3)=O)CCC(N(C)C)(CC1)CC2 c1(SCC)ccccc1CC(N1CCC(N(C)C(C2CCCS2(=O)=O)=O)CC1)=O C1(NC(C(c2c(C)noc2C)C)=O)CC2CCC1N(C(c1n[nH]c(=N)[nH]1)=O)C2 N1(C(COC)=O)CCOCC1C(=O)NCc1ncsc1-c1ccccn1 c1(C(=O)NCC(CC=C)NC(=O)CC=C(Cl)Cl)cc2cccc([N+](=O)[O-])c2[nH]1 N1(C2CC(C(N3CCCC3Cn3cc(CC4COC4)nn3)=O)C2)CCCS1(=O)=O CN1CCCC12CCN(C(C1(CNC(c3cnc(=N)[nH]c3)=O)CCCO1)=O)C2 c1(C(=O)NC(CCOC)CNC(=O)CCn2cccn2)cc(Br)cnc1O C(=O)(CC(C(F)(F)F)NC(C1(CC)CCC1)=O)N1CCC(CCCC)C1 N1(C(C2C(OC(C)=O)C2)=O)CC2CC(NC(=O)CCCCC(N)=O)C(C2)C1 N1(C(C2(C)CC3CC3C2)=O)CCC2C(C1)CN2C(=O)CCc1ccccc1 Cc1cc(Br)cc(C(N2CCC(NC(c3csnc3C)=O)C(O)C2)=O)c1C c1(NC(c2cc(Br)cc(OCC)c2N)=O)nc2c(Br)cccc2s1 c1(C(N2C3C(NC(C4C(COC)C4)=O)CC(C3)C2)=O)cc(OC)cc(F)c1 C1(CNC(C(COC)COC)=O)CN(C(c2cc(C(F)F)cs2)=O)C(C)(C)C1 CCC(C)C(C(=O)N1CC=C(C(=O)N(CC2=CCSC2)C)C1)N(C)C S(=O)(=O)(c1ccc(=NCC2CC2(Cl)Cl)[nH]c1)NCc1ccc(N(C)C)c(F)c1 N1(C(C2CC(O)(CNC(c3cc(C)sn3)=O)C2)=O)CCC(C2CCC2)CC1 CCCC(C)(O)CC(=O)N1CCN(CC(C)NC(c2cc(CC)ccn2)=O)CC1 C(=O)(CCP(C)(C)=O)NC(C1CCN(C(C(C)Cc2ccc(Cl)cc2)=O)C1)(C)C C1(NC(C2CC(C(C)(C)C)C2)=O)CC12CCN(C(=O)CCc1ccccc1)CC2 c1(C(=O)NC(CC)CNC(c2nn(C)nc2Br)=O)ccc(C#N)nc1O C1(N(C)C(C2CCC(C(C)(C)C)CC2)=O)CN(C(C2CC(O)C2)=O)CC1(C)C CC1CN2CCN1C(C(=O)NCC(C)CNc1ccc([N+](=O)[O-])cc1)C2 C1(C(=O)NC2C(NC(CCNC(N)=O)=O)CCCC2)Cc2cncn2C(=O)N1 C(=O)(CCC(C)(C)C(=O)OC)NC1CCCC(NC(c2c(OC)cncc2)=O)C1 N1(C(CC2(OC)CC2)=O)CCN(C2CN(C(=O)CN3CCCC3C)C2)CC1 C(CCC(O)C(=O)NCC1(C(=O)NCCCc2nncs2)CC1)OCC C1(CNC(c2nc(C3CC3)cs2)=O)COCCN(C(c2cc(O)cc(Cl)c2)=O)C1 C#Cc1ccc(C(=O)NC(C)(C)CCCNC(c2coc(C(F)F)c2)=O)cc1F c1(C(=O)OC)cc(Cl)cc(Cl)c1NC(=O)C(N1CCCC1CSC)=O N1(C(C(=O)NC(=O)NC)C)CCC(NC(c2cnn(C3CC3)c2)=O)C(C)(C)C1 N1(C(CCC(=O)c2cccs2)=O)CCOC2(C1)CN(C(c1coc(Cl)n1)=O)C2 c1(C(=O)NCC(C)N(C(c2cc(C)sc2C)=O)C)cccc(S(C)(=O)=O)c1 N1(C(C(CC)NC(C)=O)=O)C2CCC1C(CNC(=O)C=C1CCSCC1)C2 C1(NC(CN(CCOC)C)=O)CCN(C(=O)C(c2cccc(OC)c2)C)C1(C)C c1(C(=O)NCC(C)CNC(C2CC2CF)=O)ccc(S(C)(=O)=O)c([N+](=O)[O-])c1 C(C(C(=O)NC1CCC(NC(=O)C(C)(C)O)C1)NC(C)=O)OC c1(C(N2C3C(NC(C(C)n4cncn4)=O)C(C3)C2)=O)ccc(O)nc1Cl CCC(C(=O)N1CCSCC1C(N1CCC(C(N)=O)CC1)=O)C(C)C C#CCCCC(=O)N(CCNC(c1ocnc1Br)=O)C1CC1 N1(C(COC(C)C)=O)CCC(C2CCN(C(C34CCCCC3C4)=O)C2)CC1 C(=O)(C(O)P(C)(C)=O)NCCC(C)N(C(CCC=CC)=O)C c1(CC(=O)NCCN(C(C)C)C(C2CCN(C)C2C)=O)ccc(O)cn1 C1(NC(C=CC(C)C)=O)C2CC1N(C(C1(C(C)C)CC1)=O)C2 C1(CNC(C(C)CO)=O)CC(F)CN1C(c1ccnc(OC2CCC2)c1)=O c1(C(N2CCC(CSC)C2)C(=O)NC(CC)C)nnc(-c2ccccc2)s1 c1(CN2C(C(=O)NCCC3(C)OCCO3)CCCC2)cccc2nonc12 CCCCC(C)CCC(=O)NCC1(F)CC(NC(c2cncc(F)c2)=O)C1 C(=O)(C(CC(C)C)C(C)C)NC(CC(=O)NC(CSC)(C)CO)C(F)F C1(C(=O)NC2C=CCN(C(=O)C(O)Cc3ccccc3)C2)Cc2nccn2C1 Cc1cc(C(=O)NC(Cc2ccccc2)CCNC(=O)CC(=O)N(C)C)c(C)s1 C1(C(N(CC(C(=O)N2CC(CCCCC)C2)C)C2CC2)=O)COCCC1C C(=O)(CC1=CCCCC1)N1CCC(C=C)(C(=O)NCC(F)(F)COC)C1 c1(OC)ccc(CN2CCC(F)(C(=O)Nc3cncc(C(F)(F)F)c3)C2)cc1I C1(CNC(=O)C2CC2)CC2CCC(C1)N2c1ccnc(C(F)F)n1 c1(NCC2(COCC)CC2)cc(S(=O)(=O)N2CCC(CN(C)C)C2)ccc1C#N O=C1CC(C(=O)NC2CCCCC2C(=O)NC2(c3ncc[nH]3)CC2)=NN1 c1(C(=O)NC2C(CNC(C3CC(C)(C)C3)=O)CC2)ccc2c(c1)CCCC2=O N1(C(C(C)(C)C2CC2)=O)C2CCCC1CN(C(c1cc3n(n1)CCCN3)=O)CC2 C=CC1(C(N2CC(OC)C(C)C2)=O)CCN(C(c2cnc(C3CC3)o2)=O)CC1 C(=O)(C1c2c[nH]nc2CN1C(=O)CCC1CC1C)NC1CN(CC)C(=O)C1 Cc1csc(CCC(=O)NCCOCCN(C(=O)CC2CCCC2O)C)n1 c1(COC(C(C(C(C)C)O)C)=O)c2ccccc2cc2ccccc12 Cc1nc(CNC(=O)C(CCC2CC2)NC(C2CN(C3CCC3)C2)=O)oc1C N1(C(c2cncc(C)c2)=O)CC(C(=O)NC2CC3OC(=O)CC23)C(C)(C)C1 C1(C(=O)NCCC2N(C(c3c(C)ocn3)=O)CCCC2)CCn2c(C)cnc2C1 C1(NC(=O)Cn2cncn2)CCC12CCN(C(=O)CN1CC=CC1)CC2 Cc1cc(C(=O)NC2CCN(C(=O)C(N3CCC(CO)CC3)=O)C2)cc(Cl)n1 C1(C2CCOCC2)(C(=O)NCC(CC)NC(=O)C=Cc2ccoc2)CC1(F)F c1(C(=O)NCC(C)(C)CNC(=O)CCNC(c2ccsc2)=O)ccc([N+](=O)[O-])o1 C=CCC(C(=O)N1CC(C)(C)C1C(C)C)NC(C1CC(CC)(CC)C1)=O C(C1OCCc2sccc21)NC(c1c(O)cc(OC)cc1Br)C(=O)OCC CCCC(C)(C)CC(=O)N1CC(O)(CNC(=O)CC(C)CC(C)C)C1 C1(CNCCC(c2ccnn2C)C)CC2CC1(CO)C2 C(=O)(C1=CCCOCC1)NC1(CNC(CC2N(C)CCCC2)=O)CC1 c12cc(N)ccc1SC1(CC1)C(=O)N2.C(CCCOC(F)F)OC(C)C c1(Cc2nc(CC3(C)CC3)n(-c3ccc(F)cc3)n2)cc(F)ccc1F C=CCC(CNC(C1OCCC1C(F)(F)F)=O)NC(c1cnc(C(C)C)s1)=O C(=O)(CS(=O)(=O)N1CCC(CC(=O)NCc2cc(CC)n[nH]2)C1)OCC C12(NC(CCCC3C(C)C3)=O)CCC(CC1n1cc(-c3ccncc3)nn1)C2 c1(C(=O)NC2CN(C(c3ccc(SC)cc3C)=O)CC2C)c(F)ccc(O)c1F N1(C(CC(c2ccccc2)NC(N)=O)=O)CCCN(C(=O)C2=COCCC2)CC1 N1(C(C(COC)O)=O)CC(OC)CC1CNC(c1ccc(-c2nc[nH]n2)cc1)=O CN1CC(NC(c2ccnc(CNC(=O)CCc3ccncc3)c2)=O)C(O)C1 Cc1cc(S(N)(=O)=O)oc1C(N1CC2CC1CN2C(c1cnc(O)o1)=O)=O CC(C)(F)CC(=O)N(CCCCCc1cn(CCCOCC(=O)O)nn1)C1CC1 N1(C(CCCOC(C)=O)=O)CC(CNC(=O)CN2CCCCC2C)CC1(C)C c1(CC)nc(C(=O)NC2CC(CNC(c3cnncc3O)=O)C2)c(N)s1 N1(C(Cc2cc(C)[nH]n2)=O)CC2(CCN(C(c3cnn(C(C)C)c3F)=O)C2)C1 C1(C(=O)NCCOC2CN(C(CN(C(COC)=O)C)=O)C2)CCc2nc(C)nn2C1 C(CC(C)C)(C(=O)OC)N(C(c1ncc(I)s1)C(=O)NC1CC1)C CC1(C)OCCN(C(C2C3CCCCC23)C(=O)NC2CCOCC2)C1(C)C CC(CN1CCOCC1)C(=O)N1CC(OCCNC(C2(CCC#N)COC2)=O)C1 c1(C(=O)OC(C2C(CC)C2)=O)nn(CC)cc1OC c1(C(=O)NCC2C(NC(c3ncc(OCC)nc3)=O)C2)cc2occ(Br)c2[nH]1 CCC(C)C(CC(=O)N1CC(CC)CC(C)C1)NC(=O)CNC(=O)C1CC1 c1(OC)cccc(F)c1C(=O)NC1CCC(C(=O)Nc2cccc(C)c2F)C1 Cc1c(C(N2CCC(C)(CCNC(=O)CN3CC=CC3)C2)=O)noc1C1CC1 C1(CNC(C(c2nc(C)sc2)=O)=O)CCC(C)CN1C(=O)Cn1nccn1 C1(N(C(CCCCC)=O)C)CN(C(c2c[nH]cc(F)c2=O)=O)CCC1C Cc1ccc2c(C(N3CCC(NC(=O)C4=C(Cl)CC4)C(C)C3)=O)coc2c1 N1(C(CC(CC)O)=O)CC2CC(C(N3CC4(COC(C)C4)C3)C(C)SC)C(C2)C1 Cn1c(I)cc2c(N3CC4CCCC(C3)N(Cc3ccccc3)C4)ncnc12 c1(NC(c2ccc(-c3ccc(O)cc3O)nn2)=O)ncc(F)cc1Br C12(C(=O)NC3(CO)CCN(C(=O)Cc4ccc(Cl)c(F)c4)C3)CCCC1CCC2 N1(c2nnc(C(C)(C)C)o2)CC(NC(=O)C2=CCCCCC2)CC2(CC2)C1 CCCCC(CCCC)C(=O)NC1CC2CC(NC(C3(F)CC3)=O)C1C2 c1(SCC(=O)OCC2C(C)C2(F)F)csc2ccccc12 C(=O)(C(O)CN1CCCC1)N(CC(C)C)CC(=O)NC1(C)CSC1 N1(C(C2OCC(C)C2)=O)CC=C(CCNC(C2CCCC23CC3)=O)CC1 N1(C(C=CC(C)C)=O)CC2CN(C(C3CC3F)=O)C2C1 Cc1c(NCC(C)CO)ncnc1NC1CCN(CC(F)(F)F)CC1 C(=O)(C1=CCC2CCC1N2C(C1CC1(Cl)Cl)=O)N1CC(C(=O)NC)OCC1 C1(C)(CNC(C(C)=C(CC)C)=O)CCC(NC(c2occc2C2CC2)=O)C1 CCC(C(=O)NCCc1cc(C(=O)NCC2(CO)CCOC2)no1)SC C1(NC(C2C(NC(CC3CC(CC)C3)=O)CCO2)=O)CCOCCC1C c1(C(=O)NCCN(CCC)C(C2(COC)CCOC2)=O)cnn(C2CCC2)c1 c1(C(C)C)ccc(C(C)C)c(S(=O)(=O)NCc2ccc3c(c2)C(=O)OC3)c1 N1(C(CC(C(=C)C)OCC)=O)CC2(CCC2)CC1C(=O)NC12CCC(CC1)C2 C1(CC2C(C(=O)NCCSCCCNC(C3CC3C(F)(F)F)=O)C2)CCCCC1 N=c1nc(C2CC2)[nH]c(=NC2CCCC23CN(C(C2(C(F)F)CCCC2)=O)C3)[nH]1 C(CCSC)(C(=O)N1CCN(CC(N)=O)CC1)OC N1(C(C(C2CCCOC2)OC)=O)CCC(N(C(=O)C2=CCOC2)CCO)CC1 CC(C(C)(C)O)NC(=O)C(=O)NCC1CCC1CN=[N+]=[N-] C#CC1CCCC(NC(=O)CCCCCN(C)C(C2(C#N)CC2(C)C)=O)C1 CCC(C)(C)C(=O)N1CC(NC(C2CCOC2c2ccnn2C)=O)C1 Cc1ccc(S(=O)(=O)N(c2ccccc2)CC(O)COCCCC#N)cc1 C(=O)(N=c1[nH]n(C)cc1CN)Sc1c(OCC)ccc(Br)c1 c1(CC)ccc(C(N2CC3(CC3)CC2CNC(C2(F)CCCCC2)=O)=O)c(C)c1 C#Cc1cc(C(N2CC3(C2)CN(C(C2(C)COC(C)CO2)=O)C3)=O)cc(N)c1 c1(OC)cc(NC(c2cc(NC(C)=O)[nH]n2)c2nnnn2C2CCC2)ccc1C Cc1cc(C(N2CCC(NC(=O)Cc3cn[nH]c3)CC2C)=O)ccc1Cl CC(C)CC(C)CC(=O)NC1(C)CCCN(C(C2CCCOCC2)=O)C1 N1(C(C(C)CC2CCCCC2)=O)CCC2(CCCCC2NC(c2ccon2)=O)C1 C1(CN(C)C(C2CC2F)=O)CN(C(C2CCCN2C=O)=O)CCO1 C(=O)(CC(C)CNC(c1nnnn1Cc1ccco1)c1cscn1)OC N1(C(c2c(COC)cc[nH]2)=O)CC2CC(C1)N(C(c1cc(Cl)sc1Cl)=O)C2 N1(C(c2c(SCC)cccc2)=O)CC(F)(F)CC1(C)CNC(C1C2COCC12)=O N1(C(CC=C)=O)CCC2CCN(C(c3cccc4nnn(C)c34)=O)CC12 c1(NC(C=CC(C)(C)NC(c2ncn(C3CC3)n2)=O)=O)ccc(F)cc1F c1(CC(=O)NC2CC(CCNC(C3C(C)(C(C)C)C3)=O)C2)c(Cl)cccc1Cl CC(C)CC(CNC(C1CCN(C(C2CC(O)C2)=O)CCO1)=O)CO N1(C(=O)CC(F)F)CCC(C2CCN(C(c3cccc4cc[nH]c34)=O)C2)C1 C(c1csc2ccccc12)=CC(N1C(CNC(C2CCC(C)O2)=O)C=CC1)=O N1(C(C2CC(=C)C2)=O)CCC(NC(=O)C(C)(F)F)CC1c1ccccc1 C1(C2CN(C(=O)C(C)(C)c3ccno3)C2)(NC(C2CCC(OC)C2)=O)CC1 CCC(C)(C)CC(=O)N1CCC1(C)CC(=O)N(C(CO)C(C)C)C c1(CC(=O)NC2CCCC(NC(C3(O)CCOC3)=O)C2)nc2ncccn2n1 c1(CNC(C2C(C)=CCS2)=O)nnn(C)c1C(=O)NC1CCC2CCC12 C12CCN1CC(O)CNC(=O)COCCCC2.CCCCN(CC(=O)OC)C(C)=O C1(CC(=O)NC(=O)C=Cc2cnc[nH]2)CC(O)C12CCC2.C12(CC1)C(=O)N(C)C2 C1(C)(CNC(C(=O)NCCOC)=O)CN(C(C2(Cl)CC2(F)F)=O)CCO1 C1(NC(C(C)CF)=O)CCC(C)(C)CC1CNc1cc(O)nc(O)n1 N1(Cc2ccn(C)n2)CC(NC(c2cnc(Cl)s2)=O)C(O)C1 C1(CNC(C2CCCN2C2CC2)=O)CC2COCC2N1C(=O)COc1ccsn1 CCC(C#N)C(=O)N1CCC(N2C(=O)c3cccc(c3)C2)C1.S(C)CC C1(CNC(C(C)c2cccs2)=O)CN(C(=O)C2=NOC(C)(C)C2)CCC1(C)C C(=O)(C1CCCn2cnnc21)NCC(CNC(c1cnc(CC)s1)=O)(C)C c1(NC(C(=O)NC(CNC(C=CCC)=O)(C)C2CCC2)=O)ccc(Cl)cc1 C1(C)(NC(C(C)OCC#C)=O)CCCN(C(C2CCOC2)=O)C1 CCCC(C)(O)CC(=O)N1CC(CNC(=O)C(C)OC)CC1C.C1CO1 c1(C(=O)NCC(C)N(C(=O)Cc2cnn(CC(C)C)c2)CC)cc(OC)ccn1 N1(C(Cc2c(C)ncs2)=O)CCCN(C(=O)Cc2ccccc2Cl)CC1 N1(C(CC(C)CNC(c2cc[nH]n2)=O)=O)CCC(C)C(O)C1 CCS(=O)(=O)CC(=O)N1CCC(C(=O)NC(C)CC(F)(F)F)C12CC2 C(c1cccs1)=CC(N1CCCC1C1CCN(C(C2(O)CCSC2)=O)C1)=O c1(CNC(COC(CNC(C(C=CC)O)=O)(C)C)=O)cc(C)ccn1 c1ccccc1.C(=O)(C(=O)N1CC(NCc2ccsc2)C1)C(=O)NCCN c1(-c2n(C(CC)NCc3ccncc3)ccn2)cccc(-c2n[nH]c(CO)n2)c1 C1(NC(c2ccc(CN(CCC)C)o2)=O)CN(C(=O)C(C)S(N)(=O)=O)CC1(C)C C1(C(=O)NCC2CCN2C(=O)Cc2cc[nH]n2)(CC)CCOC1 c1(NC(C2CC(OCC3CCCCN3C(=O)CO)C2)=O)cc(C(F)F)cc(F)c1 Cc1c(C(=O)N(CCC(=O)NC(C2CCCC2)C)CCCO)cccc1O Cc1cc(-c2ocnc2C(=O)NC(CNC(c2cc(Cl)no2)=O)C2CCC2)on1 n1(CCCC)nccc1C(=O)NCCC(C)N(C(=O)C=CC(C)CC)C CCCCCC(=O)N1CC(C)(C(=O)N(C)Cc2cnn(C)c2C)C1 c1(C(N2CCN(C(c3c(CC)csc3)=O)C(COC)C2)=O)ccc2cc[nH]c2c1 c1(C(C)CCCCCC2C(CC(=O)NC(=O)CC(C)c3ccco3)C2)cnccn1 C12(NC(C3CCCC(OC)C3)=O)CCC(C1)N(C(=O)CCCN1CCCCC1)C2 c1(C(N(C2CCCC2)C(=O)Cc2ccc(Cl)cc2Cl)=O)scc2c1CCCC2 N1(C(C2C(CC)CN(C(c3ccccc3NC)=O)C2)=O)CCCC2(C=CCO2)C1 c1(CC(=O)NCC(C)N(C(=O)CC2(C(=O)OC)CC2)CC)cnc[nH]1 c1(NC(Cc2cccc(OCc3ccc(C)cc3)c2)=O)cnc(Cl)c(C)c1 c1(OCC)ccc2cc(C(=O)N(C(C)CNC(C3CCCN3C=O)=O)C)[nH]c2c1 N1(C(C(COC)OC)=O)CCC(NC(C2(CC(C)=O)CC2)=O)C(C)(C)C1 N1(C(c2ccc(CNC(C(C)CC3CCC3)=O)s2)=O)CC2C(C)C2C1 c1(OCC)cc(C(N2CCN(c3ccccc3)CC2CC)=O)ccc1C C1(C#N)(CCC=C)CCN(c2ncc(C(=O)O)cc2C(=O)O)CC1 C1(NC(CSCC(=O)NC(C)C)=O)CC(O)CN(C(=O)C(=O)NCC(F)(F)F)C1 C(=O)(C(C)C(C)C)NCC1(OC)CN(C(=O)CCC2CC2(C)C)C1 C1(NC(CC(C2CC2)NC(=O)Cn2ccccc2=O)=O)CCCC(O)C1O c1(C(=O)NC(Cc2cccs2)CC(=O)N2CCCC(CO)C2)cc2ccoc2s1 CCS(=O)(=O)CC(=O)NCC(C)NC(=O)CC(O)C1CCCC1 c1(NCc2c(N)nccc2)cc(=NCCCC2CC3CCC2C3)[nH]cn1 CC(CN1CCCC1=O)N=c1[nH]c2c(c(=NCc3nnn(C)n3)[nH]1)CSC2 c1(C(N2CCOC(C)(CO)C2)C(=O)NCCCOC)cc(C(F)(F)F)cc(C)c1 N1(C(c2ccc(OC)c(OC)c2)=O)CCN(C(=O)C(C)CF)C2CS(=O)(=O)CC12 c1(C(N2CC(NC(C(CC)NC(N)=O)=O)C(C)(C)C2)=O)c[nH]c(=N)c2[nH]ccc12 N1(C(CCN(C(=O)CC2COC(=O)C2)C)=O)CC2C(C1)C2(F)F CCC1=C(C(=O)NCC(C2CCC2)NC(C2(F)CCCN(C)C2)=O)CCCO1 N1(C(C(CC)C)=O)CC2(NC(c3cc(OC)ccc3N)=O)CCC1CC2 C(=O)(C1CCc2nccn21)N(CCCNC(=O)CC1CCC1)C1(CO)CC1 c1(NC(CN2CCC(N(C(=O)CCCN3CCCC3)C)CC2)=O)ccc(F)cc1Br CCCC(C(=O)N(C)CC1COCCN1C(c1csc(=NC)[nH]1)=O)OCC c1(NC(C2CC23CCN(Cc2cccc(F)c2Br)CC3)=O)cc(F)cc(F)c1Br c1(C(N2C(C)(CNC(C3C(=C)C3)=O)CCC2)=O)nc(C(F)(F)F)n2ccccc12 CC1(C)NC(=O)N(CCCC(N2CC3CC2(CNC(=O)C(C)(C)C)C3)=O)C1=O C1(C2CCCCC2)(C(N2CCN(C(C3C(C(C)C)C3)=O)C(C3CC3)C2)=O)CC1 c1(CC(=O)NCC(CC)NC(=O)C(C)C2CCC2)ccn(C(C)C)n1 c1(C(N2CCC(CN(C)C(C3(C)CC=CCO3)=O)CC2)=O)nccc(C#N)c1F C1(O)(CCNC(Cc2cc(C)ns2)=O)CCCN(C(C2CS(=O)(=O)C2)=O)C1 N1(C(c2ccn(C)c2)=O)CCSCC1C(=O)NC1(c2ccccc2Cl)CC1 C1(C(=O)NC(C2(O)CCN(C(=O)Cc3cnsc3)CC2)C)C2CCC3C(C2)CC13 C=CCC(C(=O)N(C(C)CN(C)C(C1CCC(=C)CC1)=O)C)C(C)C c1(C(=O)NC2CN(C(C3(Br)CCC3)=O)CC2O)c(Cl)cccc1Cl N1(C(c2ccn(C)c(=O)c2)=O)CCC2CC2(NC(c2csc3nnsc23)=O)CC1 c1(C(=O)NCC(c2ccccc2)NC(COCC(=O)OCC)=O)csc(C)c1 C=CC1(C(N2CCN(C(=O)OC)CC2)=O)CCN(C(=O)Cc2cncn2C)C1 c1(N2CC(NC(c3cnc4c[nH]nc4c3)=O)(CO)C2)nc2ncc(Cl)cc2s1 N1(C(c2ccc(C)c([N+](=O)[O-])c2)=O)CC(NC(C2(C)CC2)=O)CC12CCOCC2 c1(C(=O)NC2CC(C)(NC(c3coc(Br)c3)=O)C2)cc2nc[nH]c2cn1 C(=O)(C1CCc2ccccc21)NC(C)(C)CCC(=O)NC1CCN(C(C)(C)C)C1 CC(CCCC(=O)N1CCC(F)(F)C1)NC(=O)CN1CCC(F)CC1 C(c1ccccc1)=C(OC)C(=O)NC1CCN(C(C2CCC2C)=O)CC1 CC1(NC(=O)COC2CCC2)CCCN(C(c2cc(C3(O)COC3)on2)=O)C1 CC(C)S(=O)(=O)CC(=O)NCCN(C(=O)CN1CCS(=O)CC1)CC1CC1 N1(CCC)CC(C(=O)N(CCNC(C2CCC(CC3CC3)O2)=O)C(C)C)CC1=O C1(N(C)C(N)=O)CCC(F)(CC(=O)NCc2cn(CC)nn2)C1 CC(CF)CC(=O)NC1(CNC(c2ccc[nH]2)=O)CCOC1 Cc1c(O)nc2ccccc2c1C(=O)NC(C1CN(C(=O)CC(C)(F)F)C1)C c1(C(=O)NC2CC(CNC(CC3ON=C(CC)C3)=O)C2)ccn(C)c(=O)c1 C1(NC(C(F)=C(C)C)=O)CCN(C(=O)C(=O)Nc2ccc(Cl)cc2)CC1O N1(C(C=C(C)C)=O)CCCN(C(=O)Cc2ccccc2C(F)(F)F)CC1C(C)C N1(C(c2n(C)ccc2)=O)CCN(C(=O)CC2CCN(S(C)(=O)=O)CC2)CC1CO c1(C(N(C)CC2(O)CN(C(C3(CCOC)CCCC3)=O)C2)=O)cc(O)ccc1F C(CC(O)C(F)(F)F)NC(C1(NC(Cn2ncc(CC)c2)=O)CC(F)C1)=O c1(OC)cc(C)c([N+](=O)[O-])cc1N1CCOC(c2ccc(C)s2)C1 Cc1ccc(F)c(CC(=O)NC(Cc2ccccc2)CN)c1 c1(C(=O)NC2(CNC(C(C)C3CC3)=O)CCOC2)ccc(S(N)(=O)=O)cc1F N1(C(C(C(C)C)F)=O)CCCC(C)(C)C1C(=O)NCc1ccns1 N1(C(C=CC(CC)C)=O)CCC(C(=O)NCCC(CO)C(C)C)=C(F)C1 C1(C)(NC(C(C)CN(C)C)=O)CCN(C(C2CC2c2cccnc2)=O)CC1 Cc1c(Br)ccc(C(N2CCOC3(CC3)C2)=O)c1F.c12c[nH]nc1C(=O)N2 C1(NC(=O)CCF)CC(NC(=O)C=C2CCOCC2)C(O)C1 c1(CNC(C2(CO)CCC2)=O)cnn2c1CN(C(=O)COC1CCC1)CC2 O=C1NCC2(CC(N=c3[nH]c(N4CCOC(CF)C4)nc4ccc(Cl)cc34)C2)O1 N1(C(c2c(Br)cnc(C)n2)=O)CC2CCC(NC(c3ccc[nH]3)=O)(C2)C1 N1(C(c2nccc(CC)c2)=O)CC2CC(NC(c3ccc(F)nc3)=O)CC2C1 N1(C(C(C)N(C(C)=O)C)=O)CC2(C1)CN(C(c1csnc1C)=O)CC2CO C(=O)(CC(C)(C)CN(C)C)N(C1CCN(C(=O)C(c2ccccc2NCC)C)C1)C N1(C(c2c(CCC)onc2C)=O)CCN(C(C2(CN(C)C)CC2)=O)C(C(C)C)C1 C(CC1=CCN(C(c2ccc(F)c(Cl)n2)=O)CC1)NC(C1CC12CC2)=O N1(C(CC(c2ccc(OC)cc2)C)=O)CC(NC(c2csc(O)n2)=O)CC1(C)C C1(c2n(CC)nnn2)(Nc2cccc(C(F)F)c2C)CCOCCC1C N1(C(C(CCC)NC(=O)C=CC(=O)OCC)=O)CCCC2(C1)N=N2 N1(C(CCC(CC)OC)=O)CC2CCCC(C1)N2C(C1CCOC1=O)=O C(=O)(C(C)(Cl)Cl)N(C)CCOCCCN(C)C(C1CC1(c1ccccc1)C)=O c1(C(=O)NC2CCC(CCNC(C3(CC)CCCC3)=O)C2)ncc(N)nc1C O=C1CC(=O)CC(C(N2CCC2CNC(=O)COCC(F)(F)F)=O)C1 C1(C(N2CCC(O)(CNC(CN3C(C)CC3)=O)CC2)=O)CC2CC1CC2(F)F O=C(N=c1c(Br)c[nH]cc1Br)C1(O)CCN(Cc2ccc([N+](=O)[O-])o2)C1 c1(C(N2C(CNC(CC3C(C)CCC3)=O)CC(F)C2)=O)cc(Cl)nc(=N)[nH]1 c1(CCC)cc(C(=O)NCC(O)CNC(=O)C(C)C(F)F)c(C)o1 c1(C(=O)NC(C2CCCC2)CNC(C(C)SCC)=O)cccn2c(C)cnc12 C12(NC(CCC#C)=O)CCCN(C(c3ccnc(C)n3)=O)CC1C2 C1(C(=O)OC)CC=CCN1C(=O)Cn1nccc1C C(CCN(C(=O)CC=C(C)C)C)(C(C)C)NC(C1C(C(=O)OC)CC1)=O N1(C(C2(C)CC(C)OCC2)=O)CCCC2(C1)CN(C(=O)CSc1ccccc1)C2 CCCCC(C)(F)C(=O)NC(C1CN(C(=O)CC2CC(SC)C2)C1)C CC1(C)CCC(C(=O)NC2CC2NC(=O)C(O)CCc2ccccc2)CC1 c1(C(=O)NCC2(F)CN(C(COCC#C)=O)C2)cncc2ncccc12 c1(CN(C(C2C(=C)C2)=O)C)cnn2c1CN(Cc1ccc(OCCO)cc1)CC2 Cc1ccc(C(F)(F)C(=O)NCCCCCNC(=O)C(C)(C)n2cccn2)nc1 N1(C(CCCCCCC)=O)CCCC2C(NC(c3ocnc3CC)=O)C(C)(C)C12 c1(C(N2CCN(C(C3CC4CCCC34)=O)CC2)=O)c(F)ccc2nc[nH]c12 O=C(NNc1ncc(F)cc1F)NCc1ccnc2ccc(Cl)cc12 N1(c2cc(NC(CC=C)CC)nc(C(C)C)n2)CCn2ncc(C)c2C1 N1(C(CC2N(C)CCCC2)=O)CCC2OCCN(C(C3CCC=CCC3)=O)C2C1 c1(OCC(=O)NCC(C(C(C)C)C)NC(c2nncs2)=O)ccc2c(c1)CCC2 c1(C(=O)NC(C)CNC(=O)CC(C)(F)F)cc(S(N)(=O)=O)cc(Cl)c1F N1(C(c2c(C)coc2C(C)C)=O)C(C)CC2CN(C(=O)CNC(N)=O)CC12 C1(NC(C=CC(C)NC(C2(OC)CC2)=O)=O)C2CCCC1CC2 C(=O)(C(C(C)O)NC(=O)Cc1ccsc1C)NCc1c(CC)con1 CN1CCc2nc(C(=O)NC34CCC3CN(C(=O)C(F)n3cccn3)C4)sc2C1 CCC(CC)CC(=O)N1CCC(c2n[nH]cc2CNC(=O)C(O)C(F)(F)F)C1 CC1CCOCCN1C1CC2CN(C1=O)C2.C(C)(C)(C)OC(=O)NC1CC1 C=C(Cl)CC(C(=O)N(C1CC2CC2C1)C)NC(c1ncc(C)cc1F)=O N1(C(c2cn(CC)nn2)=O)CCCCC(C(N2CC3CCC3(C)C2)=O)C1 Cc1ccc(C(=O)NCCCCCNC(c2cc3occc3s2)=O)c2c1CCC2 C(F)(c1ccccc1)=CC(=O)N(C1CN(C(=O)C(C#N)C2CC2)CC12CC2)C C#Cc1cncc(NC(=O)C(O)CCCNC(=O)C(C)SC)c1 CC1CCN(C(=O)Cc2csc(N3CCC(O)CC3)n2)CCN1C(=O)CCCF c1(C(=O)NCC(C(C)(C)C)NC(=O)CCCn2ccnn2)cc(F)c(F)cc1F C12(CNC(C3(COC)CN(C(=O)CCNC(C)=O)C3)=O)CC(CCO1)C2 c1(CN(C2CCN(C(c3c(C(=O)OC)cco3)=O)C2)C)cccc(CN(C)C)c1 C1(C(N(CCC(=O)NC)C(C)C)=O)CCC(CO)CC1.c1(C=O)cc(C2CC2)[nH]n1 c1(SC(CC)C(N2CC(O)CC2C(=O)OC)=O)cc(F)ccc1F C1(C(N2CC(O)(CCC)C2)=O)CN(C(C2COCCN2C(C)=O)=O)CC1CC Cc1n[nH]c(C)c1CC(=O)NC1(CNC(=O)CCOCC(F)(F)F)CCOC1 C1(S(N)(=O)=O)(C(=O)NCC#CCNC(c2cn(C)cc2C(F)(F)F)=O)CCCC1 c1(C(N2CC3CC(C2)N3C(c2c[nH]c3cnccc23)=O)=O)c[nH]c2ncccc12 CC1CC(CO)N1C(c1ccc(CNC(c2csc(=N)[nH]2)=O)o1)=O c1(N2CC(CC=C)(NC(=O)CCc3ccccc3F)C2)cc(C(N)=O)nc(Cl)n1 c1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)S(C)(=O)=O)nn2cccnc2c1Cl N1(C(CC(C)NC(N)=O)=O)CCN(C(=O)C(F)(F)c2cnn(C)c2)CC1C S(=O)(=O)(c1c[nH]c(C(N2CCCC(NC(C3(F)CCS(=O)(=O)C3)=O)C2)=O)c1)NC C#CC(CNC(=O)CC(C)NC(=O)C=CC(C)CC)C(C)C Cc1cc(Cl)ccc1C(=O)N(C1CCCN(C(=O)Cn2cnc(C#N)n2)C1)C c1(C(c2cccs2)NC(C2CCO2)=O)ccccc1 c1(NC(N2CCCN3CCCC23)=O)cccc(P2(=O)CCCC2)c1 N1(CCC(F)(F)F)CCCC(N=c2ccnc(N3Cc4cccc(Cl)c4C3)[nH]2)C1 CC1CN(C(=O)C(O)(C2CC2)C2CC2)CCN1C(c1coc(Cl)c1)=O c1(-c2ccc(C)s2)cc(C)ccc1OCc1cncn1C.N1(OC)CCCC(OC)C1 C1(NC(c2ncc(OCC)nc2)=O)C(C)CN(C(=O)Cc2scnc2C)CC1C Cc1cc2sc(C(=O)NC3CCN(C(=O)Cn4ccnn4)C3(C)C)cc2s1 C1(CC(N2CC(NC(=O)CCc3ccco3)CC2C)=O)(CC)CCOCC1 C1(C(=O)NCCOC(CNC(CCSC)=O)(C)C)CCC(=O)N1C1CC1 S(=O)(=O)(c1ccc(NCCc2cc(C)no2)cc1Cl)NC(CCOC)C(C)(C)C N1(C(C2(C)C=CCCC2)=O)CCC(C(=O)N2CCC(c3cc[nH]n3)C2)=C(F)C1 N1(C(C(=O)NCC)=O)CC(C)C(NC(c2ccc(C3CC3)cn2)=O)C(C)C1 C1(NC(N(C2CCOC2)CC)=O)CCC(c2ccc(Cl)cc2)CC1 c1(CNC(c2cc[nH]n2)=O)c[nH]nc1C(=O)N(CC(F)F)CC1CC1 N1(C(C(C(C)C)CN(C)C)=O)CC(NC(=O)CC=C(Cl)Cl)C2CCCC12 c1(SCC2(C)C(NC(=O)OC(C)(C)C)CC2)cnc(O)c(CO)c1 C1(C(=O)NCCCC(C)NC(C(C)OCC)=O)CCOC(C)(C)C1 N1(CC(=O)Nc2c(C(C)=O)ncs2)CC(O)C(O)C12CCC2 N1(C(CNC(=O)C2CC2)=O)CCN(N2CCCC(c3cnco3)C2)CC1 CC1CN(C(=O)CC2C=CCC2)CCC1NC(c1ccc(Cl)c(O)c1)=O N1(C(c2cnc(C)c(C#N)c2)=O)CC2(CCN(C(=O)Cn3cnnc3O)CC2)C1 c1(CC(C(=O)NCCCCC=C)NC(=O)C(C2CCOCC2)F)cnn(C)c1O C1(NC(C2(SC)CC2)=O)C=CCN(C(=O)Cc2ccccc2F)C1 c1(C(=O)NCC(CCOC)NC(=O)C(C)CO)cncc(N2CCOCC2)c1 C1(F)(CNC(CC2ON=C(C)C2)=O)CC2CCC(C1)N2C(=O)Cc1cccnc1 c1(C(=O)NCC2CN(C(C(COC)C)=O)CC2O)cc(F)cc2cccnc12 C(=O)(C(O)CCC(C)C)NCC(C)(C1CC1)NC(C=CSC)=O Cc1ccc(C(N2CCC(NC(c3oc(Br)cc3C)=O)C(F)C2)=O)cc1Br C1(CC(=O)NC2CN(C(C(C)(C)N(C)C)=O)CC2F)CC(c2ccccc2)=NO1 C=CCC(C(=O)NC1(CN(C)C(c2cnc(OC)s2)=O)CC1)C(C)C C1(NC(=O)Cc2ccc(C3CC3)cc2)COCCN(C(=O)C(O)C2CC2)C1 CC1(C)CCC(O)(CNC(C2COCCN(C(=O)C=CCN3CCCC3)C2)=O)C1 CC1CN(C(C2C3CCC2CC3)=O)CCC1NC(C1(n2cccn2)CC1)=O c1(C(=O)NCC(c2ccc(OC)cc2)NC(=O)COC)ccc(S(C)(=O)=O)s1 C(=O)(CC(O)C(C)(C)C)N(CC(C)NC(c1ccc(OCC)cc1)=O)C CC1CN(C(C2CC(=O)NC2(C)C)=O)CCN1C(c1cc(Br)cs1)=O C1(C2CCCN(C(C3COCCO3)=O)C2)(NC(=O)Cc2cc(Cl)sc2Cl)CC1 N1(C(C2=CCCN(C(C(C(CC)O)C)=O)C2)=O)CC(C)NC(=O)C12CC2 c1(C(=O)OC)ccc(NC2CCCCN(CCCN=[N+]=[N-])C2)cc1C(=O)OC c1(C(N(CC(N2CCC2CNc2ccccn2)=O)CC)=O)cc(F)cc(F)c1O C(=O)(CCCCC(F)F)N1CC(CNC(C2(C#C)CCCC2)=O)N(C)CC1 CCCCC(F)C(=O)N(C(CNC(=O)C(C)NC(=O)CC)C1CC1)C C(CCC(C)C(=O)N(C1CCCCN(C(c2sccc2CO)=O)C1)C)OC CC1CC=CCC1C(=O)N(C1CCN(C(=O)Nc2cc(Cl)c[nH]2)CC1)CCO c1(C(N2CC(NC(c3cc(SC)oc3)=O)C(OC)C2)=O)cnc2n1CCC(C)C2 CC1(C)CC(=O)NCC1Cn1cc(C2(NC(c3cccn3CC#N)=O)CC2)nn1 C1(C(N2CC(n3cc(CNC)nn3)C(O)C2)=O)CC2(CCC2OC)C1 C1(C(=O)OC)(NCC(C)(C)[N+](=O)[O-])CCCN(Cc2ccccc2)C1 C(C(O)C(=O)NC(c1cnn(C)c1)C(=O)N(C1CCC1O)C)=CC C(=O)(C(C)C(F)(F)C(F)F)NCC=CCNC(C1(CC)CCNC1=O)=O C1(C(=O)NC2CC(C(=O)NCCNC(C3(N(C)C)CC3)=O)C2)Cc2ccccc2N1 c1(C(=O)NC2C(CNC(C(CC)C(C)C)=O)CC2)ccc2c(c1)NC(=O)CS2 CC1OCCCC1C(=O)NC1CC(CNC(=O)C=CCOc2ccccc2)C1 c1(C(C)C)ncc(Cl)c(C(=O)NC2CC23CC(NC(c2ncncc2Cl)=O)C3)n1 C1(C(N(C(C(C)C)CO)C)=O)CN(C(C2COCCO2)=O)CC1(C)C c1(C(N(C)CC2CC(OC)CN2Cc2ccco2)=O)ncc(Cl)cc1F c1(C(=O)NC2C(NC(C(C(CC)C)O)=O)CCC2)cc(F)c(F)cc1OC Cc1[nH]c(C(N2CCCC(C)CC2)=O)c(C)c1C(=O)NCc1csc(C#N)c1 C#Cc1cnc(N2CCC(CNC(C3(C)CCC(=O)NC3)=O)CC2)nc1 C1(O)(C(=O)NCC2CC(NC(C3(CCC)CC3)=O)C2)CCc2ccccc2C1 N1(C(C2C(=C)CC2)=O)CCC12CN(C(c1cccc(NS(C)(=O)=O)c1)=O)C2 C1(C(=O)NCC(C2CCCCC2)NC(C(CC)F)=O)CCN(CCO)C(=O)C1 C1(CC(=O)NC2CC(NC(=O)CSc3ccccc3)C2)CCCCC(=O)N1 C(=O)(C(C)C(C)S(C)(=O)=O)N(CCCNC(C(C(CC)(C)C)=O)=O)C C(=O)(CN1C(=O)COc2ccccc21)NCC1(C)CN(C(C(C)O)=O)C(C)(C)C1 c1(OC)ccc(CC(N2CCC(=O)CC2C(=O)O)=O)c(Cl)n1 c1(C(N(C(C)CNC(c2ccnn2CCN(C)C)=O)C)=O)ccc2nccn2n1 N1(C(c2sncc2Br)C(=O)NCCOC)CCc2c(c(CC(=O)OC)nn2C)C1 N1(C(CC=C)=O)CCC(NC(c2cc(O)n(CC)n2)=O)CC1 c1(CNC(CC2CCCN(Cc3cn(C(C)C)nc3)C2)=O)noc2ccccc12 N1(C(c2c(C)nc(C)s2)=O)CC2OCC(NC(=O)CCOCC(F)F)C2C1 c1(C(N(C)CC2N(C(c3c(CC)onc3)=O)CCC2)=O)nsc2ccccc12 Cc1cc2cc(C(=O)NCC3CC(C)(C)CN3C(=O)CCC(F)F)oc2cc1C c1(C(=O)NC(CNC(C(CCC)OC)=O)C2CCC2)c(N)ccc(Br)c1F C1(C(=O)NC(CC)COC)(CCc2ccccc2)CN(CC2CCCC2C)C1 c1(NC)cnc(Cl)cc1C(=O)NC(C1CN(C(=O)C2=C(C)OCC2)CCO1)C c1(SCC)onc(C(N2CCCC2C(C)(C)CNC(=O)C#CC2CC2)=O)c1C O=C1CC2(CN(C(c3noc(-c4ccc(F)cc4F)n3)=O)C2)C(O)CN1 N1(C(COc2cccc(C)c2)=O)CCC(C)C(NC(=O)C=CCCC(C)C)C1C CC1CC(NC(=O)CCCn2ccnc2)CN1C(=O)CCSC1CCCC1 C1(CCCNC(c2cc(O)ncn2)=O)CN(C(C2CC2c2ccccn2)=O)CCO1 c1(C(=O)NC(C)Cn2cc(CCC3CC(C)(C)CO3)nn2)cc2n(n1)CCC2 Nc1ncc(C(N2CC(F)(F)CC2CNC(=O)Cc2cnc[nH]2)=O)cc1CO C1(C(N2C(C)(C)CC(NC(c3cnn4c3CCC4)=O)C2)=O)CNC(=O)CC1(C)C CC(C(=O)NCCC1(O)CCN(C(C2(c3ccno3)CC2)=O)C1)C(F)(F)F C1(OC)(CNC(c2ccc(C)c(Cl)c2)=O)CCN(C(c2c[nH]c(=N)s2)=O)CC1 c1(NCc2cc(C)oc2Br)ccc(C)c(Br)c1 C12(C(=O)NC3CCN(C(C=CCC)=O)CC3(C)C)CC3CC(C(=O)N1)C2C3 C=CC(C)(O)CC(=O)N(C1CCN(C(=O)COCCCC)C1)CCC c1(C(=O)NC(CCCNC(CCN(CCC)C)=O)C)ncnc(C)c1OC C(N=c1[nH]c(Cl)ncc1F)C1N(C(C2(COC)C=CCC2)=O)CCCC1 CC(CSC1CC(OC(F)F)C1)C(=O)OC(C)(C)C CC1(C)CC(CNC(=O)Cc2c(Cl)cccc2Cl)N(C(=O)CC2(O)CCOC2)C1 c1(C(=O)NCC23CC2CN(C(C2CCCCO2)=O)C3)cc(O)nc(C2CC2)n1 C1(OC)CC2(C1)CC2N(C(=O)NCc1ccc(C)cn1)Cc1ccco1 N1(C(C2(OCC)CCOC2)=O)CCCN(C(c2cnc(C)o2)=O)C(C(C)C)C1 C1(N(C(C2C(C=C)C2)=O)C)CCC(NC(=O)C(c2ccc(OC)cc2)C)CC1 C1(N(C(C2C3(CC3)C23CC3)=O)CC)CCCN(C(=O)CCC2CCC2)CC1 Cc1cc(Br)cc2[nH]c(C(=O)NC3CCOC3CNC(=O)C(C)(O)C(F)F)cc12 C(c1cccnc1C)=CC(=O)NC1CCN(C(CN(C)CC)=O)C1C1CC1 Cc1ncc(C(=O)NC2CC(C)(CNC(=O)OC(C3CCC(CN)O3)=O)C2)n1C CC1(C)CCC1C(=O)NC1COCC1NC(c1nscc1Br)=O N1(C(CCCOC(C)=O)=O)CCCN(C(c2cc3n(n2)CCOC3)=O)C(C)C1 C=CCC(CO)NC(C1(C)CN(C(=O)CCN(C)C)C1)=O c1(C(=O)NC(CNC(CCc2nc(C)c(C)[nH]2)=O)C2CC2)ccc(Cl)cc1O CN=c1[nH]cc(C(N2CC(OC)C(NC(=O)C(n3ccc(C)n3)C)C2)=O)s1 C(=O)(C1=NOC(c2ccccc2)C1)N1C(C(=O)N(CCO)Cc2cc[nH]n2)CCC1 CC(C)CC(C)CC(=O)N1CCC(CO)C(NC(c2ccc(C(C)C)cn2)=O)C1 Cc1onc(C(F)(F)F)c1C(N1CCC(NC(c2nncs2)=O)C1)=O C1(C)(C(=O)NC2CC(F)(CNC(c3cn(CCC)nc3)=O)C2)CCCC1O C1(NC(c2csc(C)c2C2CC2)=O)COC2C(NC(=O)C(C)(C)N(C)C)COC12 c1(C(C)=O)nc(C(=O)N(C(C)CCNC(=O)Cn2ccc(Br)n2)C)cs1 CC1CCCCC1OCC(=O)NCC1CCN1C(c1cnc(C2CC2)[nH]1)=O c1(C(=O)NC2(C)CCN(C(c3n[nH]c(C)c3F)=O)C2)ccn2cccc2c1 C1(C(=O)NCCCN(C(C)C)C(C2COC(=O)O2)=O)CC12CCOCC2 N1(C(CCN(C)CC)=O)CCC(C(N2CCCC2C(C)O)=O)C1 C1(CNC(CCSC)=O)CC(C)N(C(=O)CNC(c2cccc(F)c2)=O)C1 C(CC(CO)NC(=O)CCN(C(=O)C(C)n1cccn1)C(C)C)SC c1(CC(=O)Nc2cc(COC)nn2C)cnc2n1CCCC2C C1(CC(=O)N(C2CCCC2)CCNC(CCOCC#C)=O)CCCC(OC)C1 C1(C)(C(=O)NCC(C)NC(c2ncoc2C2CC2)=O)CCC(=O)CC1 c1(C(N2C(C(=O)NCc3cc(OC)ns3)C(C)CC2)=O)cc2ccccc2o1 N1(c2c(C)c(NCc3nc(CO)n[nH]3)ncn2)CC(C)OC(C)(C)C1 C1(CNC(C2(O)CC(C)(C)C2)=O)CN(C(=O)CCC(CF)CF)CC12CCC2 c1(C(=O)NCC2CN(C(=O)C3=CCCCO3)CC2O)cc(Cl)cc(Cl)c1Cl N1(C(C(C(CC)O)C)=O)CC2CCOC2(C(=O)NC(c2cc(OC)ns2)C)C1 CN1C(=O)CC(C(=O)NCC2CCCN(C(=O)Cc3nn(C)cc3Cl)C2)NC1=O C1(CC)(NC(C2CCCC2CNC(C2COCC(C)O2)=O)=O)CCCCCC1 c1(C(=O)NCCN(C(=O)C(C)(F)C(=O)OC)CCC)cc(C)cc(C)c1 N1(C(=O)C(Cl)=CCl)CCOCC(NC(c2cnc(-n3cccn3)cn2)=O)C1 C1(C(=O)NCc2occ(C(=O)NCC3(CO)CCN(C)C3)n2)CCC(O)CN1C C(=O)(C1=CCC(F)(F)CC1)NCCCN(C(=O)C(Br)=C(C)C)CC CCC(C)(C)C(C(=O)N1CC2CCN(C(c3sc(C(C)C)nc3C)=O)C2C1)OC c1(CNC(=O)NC(C)Cc2ccno2)noc(-c2ccnn2C)n1 n1(CC(=O)N(C)CC2CN(C(=O)COCC(F)F)C2)cnccc1=O CC(C)(CC(=O)NCC1(C)CCCC1NC(=O)C=Cc1cocn1)C(F)F c1(C(=O)NCC(CNC(CCCC2C(C)C2)=O)F)cc[nH]c(=N)c1[N+](=O)[O-] C1(NC(c2sc(C)c(O)n2)=O)C(C)CCN(C(c2ccc(C)n2C)=O)C1C C1(N(C(CCCOC(C)C)=O)C)CCN(C(=O)CC2(C3CC3)CCC2)CC1 C(CC(C)(C)C)(C(=O)NCc1ccc(SC)o1)NC(C(CC)SC)=O c12ccc(=O)n(n1)CCO2.C(CC(CNC(C1CC1CSC)=O)NC(C)=O)OC c1(C(=O)OCC)ccc(F)cc1O.C=C1CCC12C(=O)OCC(=O)O2 C1(C(N2CCC(O)C(C)C2)=O)(CC)CCN(C(=O)CNC(C)=O)CC1 c1(OC)cnc(C(=O)NCC23CC2CN(C(=O)C2=CCCCC2)C3)c(OC)n1 Cc1ccc2c(CN3CCC(NC(c4ccc(Cl)c(C)c4)=O)C(F)C3)c[nH]c2c1 C12(NC(c3coc4c3CCCC4)=O)CCC(CN(C(=O)C(F)n3cccn3)C1)C2 C1(C(=O)NC(C)Cc2ccco2)CC(NC(=O)COCC(F)F)C(O)C1 n1(CCC#C)c(N(C)C(C)C)nnc1-c1ccc(NC(C)(C)CC)cc1 C1(C(N2C(CC(=O)OC)CCC2)=O)CN(C)CCN1C(C1CC(=O)C1)=O C1(CCNC(c2n(CC)ccn2)=O)CSCCN1C(c1cn(C2CCC2)nn1)=O CC(CC1=CCCCC1)NC(C1(N(C(=O)Cc2ccsc2)C2CC2)CC1)=O C#CCC(C(=O)NC(c1ccccc1)CNC(=O)Cc1ccccc1F)C1CC1 c1(C(N2CC(CC=C)(NC(c3oc(SC)cc3C)=O)C2)=O)c(C)ccc(C)c1C C1(CNC(C(C(C)O)(C)C)=O)CCN(C(=O)C(C2CC2)C2CC2)CCC1(F)F N1(C(COc2ccc(C#C)cc2)=O)CCC2C(C1)CN2C(c1ccoc1Cl)=O c1(-c2nc(Cc3c4cn(C)nc4ccc3)on2)cc(Br)cc([N+](=O)[O-])c1 N(C1CCc2cccnc21)C(c1c(C(=O)O)oc(Br)c1)=O Cc1nc(C2C(C(=O)NC34CC(NC(c5cn[nH]c5)=O)(C3)C4)C2(C)C)n[nH]1 N1(C(C(C)(C)CO)=O)CC2(CC(C(N3CCC(C)(C4CC4)C3)=O)CO2)C1 c1(CCN(C(C2(CC)COC2)=O)NC(=O)Cc2ccc(C)cc2)ccccc1Cl C1(C(=O)NCCNS(CC)(=O)=O)C(C2CC2)CCN1C(c1cn(C)nc1C)=O c1(C(=O)NC2CN(C(C(CSC)C)=O)CC(O)C2)ccc2nc(O)sc2c1 C1(F)(CNC(C2(C)C(C)CCC2)=O)CCN(C(=O)C=Cc2ncco2)CC1 C1(NC(C(CC(C)C)O)=O)COC2C(NC(c3cc(Cl)cnn3)=O)COC12 Cc1cc(CNC(CN(C(C)(C)C)C(=O)O)=O)ccc1CO.C(=O)(C(C)(C)C)NC(C)C Cc1[nH]nc(C(N2CCC(C(C)C(=O)N(CC(C)O)C3CC3)CC2)=O)c1O c1(C(N(CC(=O)N(C2CC2C)C)CCOC)=O)cn(C2CC2)cn1 C(=O)(CC1=NNC(=O)C1)NCC1N(C(Cc2c(C)nc(S)s2)=O)CCC1C c1(Cn2ncc(C(=O)NCCN(C(=O)CCCF)CCC)c2)ccccc1F c1(NC(CC2N(C(CCN(CC)CC)=O)CC2)=O)cccc(Cl)c1C Cc1nn(CC(N2CC3CC3(CNC(=O)C(C)CN(C)C)C2)=O)c(C)c1Br C1(C(C)C)COCCN(C(C2CCN2C(=O)C(F)=CC2CC2)=O)C1 C1(CCNC(c2c(C)nn[nH]2)=O)CN(C(=O)Cc2cncc(O)c2)CCS1(=O)=O c1(C(N2CCC(NC(C3C(COC)CC3)=O)CC2C)=O)cc(Cl)cc(Cl)c1OC c1(NC(C)=O)c(F)cncc1F.c12ccnc(c1)C(=O)N(C)C1CCN(C1)C2=O C1(C(=O)NC2CCC3CCN(C(CCCOC)=O)C32)CCc2nc(=N)[nH]cc2C1 c1(C(N2CCC(C)(CNC(c3nc(OCC)sn3)=O)C2)=O)c(F)cccc1F C1(C(N(C(CC)COC)C)=O)CCOC1CNC(c1c[nH]nc1Cl)=O c1(C(N2C(C)CC(NC(=O)CCC#N)C2)=O)cnc2[nH]cnc2c1 c1(C(=O)NCCCN(C(=O)CC(=O)NC2CC2)CC)coc2cc(F)ccc12 C1(C2CCN(C(c3cnc(C(C)(C)CF)o3)=O)C2)(NC(C(CC)SC)=O)CC1 c12cc(F)ccc1NC2.C1(c2n(CCC)nnn2)(OC(C)C)CC2COCC12 c1(C(=O)NCC(CC=C)NC(=O)C(F)(F)COC)ccc(C)c(S(N)(=O)=O)c1 c1(SC)ccc2cc(C(=O)NC3CC3NC(C3OCC4CCCC34)=O)[nH]c2c1 c1(C(N2CC(N(C(C)(C)C)C(C3C(C)C3)=O)C2)=O)nc(N)cc2ccccc12 C12(C(=O)NC(CCC(=C)C)C)C(NC(C3C=CC=CC=C3)=O)C3CC1C2C3 c1(C(=O)NCC(CC(C)C)NC(=O)COCC2CC2)ccc([N+](=O)[O-])n1C C1(C)(C(N(CCCCCCNC(c2n(C(C)C)ncc2)=O)C)=O)CCOC(C)C1 c1(SCC2N(C(C(C3CCCC3)OCC)=O)CCC2)ccnc(F)c1 c1(CNC(C2CC(CNC(C3(F)CC3)=O)C2)=O)ccc2c(c1)CC2 N1(C(c2ccc(OC)cn2)=O)CCC(C2(NC(=O)Cn3cccnc3=O)CC2)C1 C1(C(=O)NC(C)C(c2ccccc2)C)(COCC)CCCN1C(=O)CC(=O)NC C1(CNC(c2c[nH]nc2Cl)=O)CC2(CC2)CN1C(c1cc(Cl)ccn1)=O C(C)(CC(=O)N(CCNC(C1(F)CCOC1)=O)C(C)C)SC C(N=c1[nH]c(=NCCOC2CC2)c2c(F)cccc2[nH]1)c1c(C)noc1 Cc1cc(C(N2C3CN(Cc4ccc(-c5ccccn5)cc4)CC23)=O)c(C)[nH]1 N1(C(c2cc(CC)c(C)s2)=O)CCC(NC(c2cc(C)c(F)cn2)=O)C(CO)C1 Cn1cc(C(N2CCC(CO)C(NC(=O)C#CC3(C)CC3)C2)=O)c(O)nc1=O c1(C(N2CCC(NC(CC3(COC)CC3)=O)C2(C)C)=O)noc2c1CCCCC2 c1(OCC(=O)NC(C)CCCNC(=O)C(C)CC2CCCC2)ccc(CO)cc1 Cc1sc(=O)n(CCC(N2CC(NC(c3cc(C)n(C)c3)=O)C3(CC3)C2)=O)c1C c1(C(=O)NC(CCN(C(c2cccc(C(C)=O)c2)=O)C)C)ccc(N=[N+]=[N-])cc1 N1(C(CC2ON=C(CC)C2)=O)Cc2ccccc2C(NC(c2ccc(C)o2)=O)C1 C1(CC(N2C(C(C)NC(C3CC(F)(CO)C3)=O)CCC2)=O)CCC(F)(F)CC1 N1(C(CCc2onc(C)n2)=O)CCC(O)(CNC(c2ccc(N)c(F)n2)=O)CC1 C(=O)(C1=NOC(C)C1)NCC1(C(=O)NCc2c(OC)cccn2)CCC1 c1(CCC)cc(C(=O)NC(c2cn(CC3(F)CCOC3)nn2)(C)C)n[nH]1 N1(C(C=CCOCCOC)=O)CC(NC(c2cc3sccc3[nH]2)=O)CCC1C c1(C(C)CC(=O)NCC(C)(C)CN(C)C(c2cscn2)=O)ccc(F)c(F)c1 CCCC(C)(C)C(=O)N1CCCC(CCNC(=O)CCCOCC)C1 c1(C(N2CCC(N(C)C(c3snc(O)c3Cl)=O)C2)=O)nnn2c1C(=O)NCC2 C(=O)(C1CCC(=O)c2cccn21)NCC1N(C(c2cn(C)nc2)=O)CCCC1 c1(C(C)NC(=O)N(CC(O)CO)CCN)ccc(OCC(F)(F)F)cc1F C1(NC(CC2(CNC(c3ccc(C#N)cc3)=O)CC2)=O)CC2CC1C(O)C2O C1(F)(CNC(c2cn(CC=C)nn2)=O)CCCN(C(C2(C)CCCS2(=O)=O)=O)C1 N1(C(C#C)=O)CCOCC(NC(c2c(C)nn(-c3ccccc3)c2Cl)=O)C1 C1(NC(=O)CN2CCCC2=O)CN(C(C2SCCCS2)=O)C2CC12 N1(C(C(CC2CC2)OC)=O)CCOC(CC(=O)NCC(C)(O)C2CC2)C1 N1(C(C2C3CN(C(C(C)OC)=O)C2C3)=O)CCCN(C)CC1C N12Cc3ccc(cc3C1)C2=O.C1(C(C)C)(NC(=O)C(=O)c2ccco2)CCC1 Cc1ccsc1C1CC1C(=O)NCC=CCN1CC(NC(=O)C(C)N(C)C)C1 c1(CC(=O)NCC2CCN2C(c2nc(Br)c[nH]2)=O)ccc(F)cn1 CCCCCC(C)CC(=O)N1CC2(CC(CC(=O)NCCC(C)SC)C2)C1 c1(CC(=O)N(C2CC2)Cc2cccc(C(F)(F)F)c2)cc2ccccc2c(=O)o1 C1(C)(NC(C2C(CCOC)C2)=O)CC(C(=O)NOCCCN(C)C(C)C)C1 c1(CC(N2C(CNC(C3CCCO3)=O)CSCC2)=O)cc2ccccc2c(=O)o1 c1(OC)ccccc1C(C)C(=O)NCC1CCN(C(=O)C(c2ccnn2C)C)C1 c1(C(N2C(C)(CC(=O)N(C3CC(C(N)=O)C3)C)CC2)=O)cnn2ccccc12 C1(NC(CCCC=C)=O)CC2(C1)CN(C(=O)C(C)S(N)(=O)=O)C2 c1(C(=O)NCC2N(C(CC(C(C)C)O)=O)CC2)cnc2ccccc2c1 C1(CNC(c2cnn(C)n2)=O)CN(C(c2cc3ccsc3n2C)=O)C2(CCC2)C1 N(C(=NCc1cc(C(C)(C)C)on1)N1CCC(CCOC)C1)C(CC)C CCCC(C)(O)C(=O)N1CC(N(C(=O)CCSc2ccccn2)C)C(C)(C)C1 c1(CC)c(C(=O)NC2CCC(O)CN(C(=O)C(F)CC)C2)oc2ccccc12 N(C(=NCC(Cl)C(F)(F)F)NCc1sc(N2CCCC2)nc1C)Cc1cc(C)on1 C1(C)(C(N2C(CN(C(=O)CC3(NC(C)=O)CC3)C)CCC2)=O)CCC(F)(F)C1 Cc1ccc2c(C(=O)NCC3CCCN3C(=O)C(C)CC(F)F)ccnc2c1Cl N1(C(C(C=C=C)C)=O)CCC(C=C)(C(=O)NCC=Cc2ccccc2)CC1 c1(CN(C)C(C2(NC(=O)CCn3cnc(=N)[nH]3)CC2(C)C)=O)cn(C)cn1 N1(C(c2onc(C)n2)=O)CCC(CNC(=O)C(C)C(C)(F)F)C12CC2 C1(C)(NC(C(C)C2CCCO2)=O)CN(C(C2CC3CC2C3)=O)C1 C=CC(C)(CCOC)C(=O)N1CCN(CCCNC(=O)CC(C)SC)CC1 N1(C(c2c(C)nc(CC)o2)=O)CC(NC(=O)C(C)CC(N)=O)CC12CCOCC2 O=C(C1=CN2CCS(=O)(=O)N=C2C=C1)NC1CCN(C(=O)C2=CCCOCC2)C1 C=CC1OCCC1C(N1CCCCC1C1(NC(c2nn(CC)nc2C)=O)CC1)=O C1(NC(C2C(C(C)NC(C(C)OCOC)=O)C2)=O)CCn2nnnc2C1 N1(C(c2cc(C)oc2C)C(=O)NC(C(=O)OC)C)CC(C)(C)C1C1CCCO1 N1(CCOCC)CCC(N=c2[nH]c(N(C)Cc3nnnn3C)nc3cc[nH]c23)C1 N1(C(c2cccc(SC)n2)=O)CC2CC(NC(c3ncc(Cl)s3)=O)CC1C2 c1(C(=O)NCC=CCNC(=O)Cc2cccnc2)cnc(Cl)c(Cl)c1 C1(C(=O)Nc2cccc3nccn23)CC2OCCC2N(C(c2cnc(O)[nH]2)=O)C1 c1(C(=O)NC(CNC(COCCCC#C)=O)C2CC2)cn2c(n1)COCC2 C=Cc1cnn(C)c1C(=O)NCC1CCCCC1NC(=O)CCCC(=O)N(C)C CCC(CC)CCCC(=O)N1CC2OCC(NC(=O)CCc3cncn3C)C2C1 c1(C(N2CCC(CC=C)(NC(=O)C(C)C(O)CC)CC2)=O)cc2c(s1)CCSC2 C#Cc1cc(C(N2CC(NC(c3ccnn3C=C)=O)CC2C)=O)cc(Br)c1 C(=O)(CCC(=O)NN(C)C)NC(CCCNC(CN(C1CC1)CC)=O)C C(=O)(CCCCCN=[N+]=[N-])NC1CC=C(C(=O)NC(c2nc(C)[nH]n2)C)C1 Cc1ncc2n1CCN(C(=O)C(c1ccco1)NC(=O)CCOC1COC1)C2 C(CCC(C)(C)C(=O)N(CCCSC)C)NC(c1c(CC)cccc1)=O c1(CCC)ccc(C(=O)NC(C)(CNC(=O)CSC)C(C)C)cc1.C(C(F)(F)F)N N1(C(c2c(OC)cccn2)=O)CCN(C(=O)Cc2ccccc2Cl)C(CO)C1 N1(C(c2c(CNC(c3cnn(CC4CC4)c3)=O)ccs2)=O)CCOC(CF)C1 C1(CC(C)C)Oc2cc(Br)ccc2C1NCC(C)CC(F)F c1(OC)cccc2sc(C(N3CCN(C)C4CC34)=O)cc12 Cc1ccn2cnc(C(=O)NCC3CN(C(=O)C(C)C(C)C4CCC4)C3)c2c1 c1(OCC(=O)OC(CC(=O)OCC)OC)ccccc1CN C1(NC(C2CCSCC2)=O)CC12CCN(C(c1ccc(F)c(O)c1F)=O)CC2 C1(CC)(CNC(=O)C=CC(C)(C)NC(c2cc(Cl)ns2)=O)CCC(=O)N1 CCCC(CCCNC(=O)CCC(CC)OC)NC(=O)CCC1(C(=O)OC)CCC1 Cc1ccc(C(=O)NC(C2CC2C(=O)N(C)CC2CC2(F)F)C)cc1O C(=O)(C(F)CCC(C)(C)C)N1CC(C(N2C3CC(OC)CC2CC3)=O)C(C)(C)C1 N1(C(C2CCN(C)C2)=O)CCC2(CCC(CNC(=O)CC(C)(C)C)CC2)CC1 N1(C(C(C)=C2CCC2)=O)CCCC(CC(=O)NCCC2(C)N=N2)CC1 C1(NC(C2(SC)CC2)=O)CCCC(N(C)C(c2ccc(C(C)(C)C)[nH]2)=O)C1 O(NC(=O)C(c1cn(C)nn1)NC(c1ccn(CC)n1)=O)C(C=C)C C(=O)(C#CC1CCOC1)N(CC(C(=O)NC1(CC=C)CC1)C)C N1(C(C(CC#C)O)=O)CCOC(C)(CNC(=O)C=CC(C)(C)C)C1 Cc1ccc(F)cc1C(N1CC(CC(=O)N(CC(O)C2CCC2)C)CC1C)=O c1(C(N2CC(OC)(CNC(c3cc4ccsc4s3)=O)C2)=O)cccn2ncnc12 Cc1nn2cc(C(=O)NC3(C4CCN(C(=O)C(O)C5CC5)C4)CC3)nc2s1 c1(C(=O)NCC(CNC(c2c(N)cc(C)cc2F)=O)C)ccc(F)c2ccsc12 c1(C(=O)NC(C=C)CO)ccc(CNC(=O)C=CC2(C)COC2)cn1 C(=O)(C(CN=[N+]=[N-])NC(=O)Cc1ccns1)NCCC1CCC(C)(C)C1 C1(CCC)CCC(C(=O)NC2CC(NC(=O)C(N3CCC(C)C3)=O)C(O)C2)CC1 N1(C(C(CSC)C)=O)CCC(F)(C(=O)NC(CO)CCO)CC1 CCCCCC(C)(C)C(=O)NCC1CCCN1Cc1scnc1C N1(C(CCC(CC)C)=O)CC2CN(C(c3cc4c(Cl)nccc4s3)=O)CC2(C)C1 c1(C(N(CCC(=O)NCc2nncs2)C)=O)cccc[n+]1[O-] CC1CN(C(=O)COc2ccc(F)nc2)CCC1CNC(=O)CC1CCCC1 Cc1cc(Br)cc(C)c1CNC(=O)NCC(C)(C)C(C)O C(=O)(C(C)(F)C(C)(C)F)N1C(C(=O)NC2(CO)CC(OC)C2)CC(=O)C1 c1(CS(=O)(=O)CC)ccc(C(F)F)cc1.C(C(CCOC)OC(=O)C)OC c1(OC)cc(C(=O)NCC(C)CNC(=O)CC2CCOC2(C)C)sc1Cl CC#CCC(C(=O)N(CC(O)CO)C)NC(C1CCCS1)=O C(=O)(CCCC(=O)NCC1(C)CCN(C(c2ncncc2Cl)=O)C1)N(C)C C1(NC(C2(C)COC2)=O)CC2CCC1N(C(=O)C#CC1CCOC1)C2 c1(C(=O)NC2C(NC(CCCOCC)=O)CC2)cn2cc(C)ccc2n1 c1(C(N2C(CC)CN(C(C3CCC(=O)N3)=O)CC2)=O)cc2cc(C)ccc2o1 c1(CC)cc(C(=O)NC2C3CN(C(C4CC(F)C4)=O)CC23)cc(N)c1 c1(C(=O)NCC2(F)CC(NC(C(COC)C)=O)C2)c(C(F)F)n[nH]c1C C(C(=O)N1CC(N(C(=O)COc2cc(C)on2)C)C(C)(C)C1)(C(C)(C)C)SC N1(C(C(CCC)C)=O)CC2(CCN2C(c2cnc(C)c(C)c2)=O)C1 c1(C(N(CCCCNC(c2ccc(CCCCC)o2)=O)C)=O)cc(F)n(C)n1 c1(CC)cc(C(N2CCCC2CN(C(=O)C=C2CCSCC2)C)=O)no1 CCC1c2ccccc2CN1N1CC2(CC)CCCC2(F)C1 CC1(CNC(c2ccnc(CNC(=O)C(O)C3CC3)c2)=O)CCCCCC1 c1(C(=O)NC2CN(C(C3C(C#C)C3)=O)C2)ccc(I)cn1 C1(CNC(c2c(CC)onc2)=O)CN(C(C2(Cl)CC23CCC3)=O)CCO1 C(=O)(C1=CC2C=CC1C2)NC1(C(NOC(C)(C)CO)=O)CCSC1 CCC(C(=O)OC)C(=O)N(CC(N1CCCC(COC)C1)=O)C1CC1 N1(C(C(=O)NC(C)C)=O)CCCC(CNc2cc(C(C)(C)C)on2)C1 C1(CC(N2CC3CC2CS3)C(=O)Nc2ccccc2)CCCCCC1 c1(CNC(C(C)OCCN(C)C)=O)ccc(C(N2CCC(CN(C)C)C2)=O)cn1 c1(C(N2CCCN(C(Cc3cc(C)on3)=O)C(C)C2)=O)cc2ccc(Cl)cc2s1 C1(NC(C(C)SCc2ncccn2)=O)CC1C1CN(C(=O)C=CC(=O)N(C)C)C1 c1(OC)ccc(Cl)c(NC(c2ccc(I)c(F)c2F)=O)c1Cl N1(C(c2c(CC)onc2C)=O)CC2CCC2(CC(=O)NC2CCC(O)C2O)C1 c1(NC(=O)CC2CC23CC3)ccc(S(=O)(=O)Nc2ccccc2)cc1 Cc1nn2c(c1CNC(c1cnnn1C)=O)CN(C(=O)Cc1cncn1C)CC2 c1(CCC(=O)NCCN(CCC)C(c2cc(C)sn2)=O)c[nH]c2cc(C)ccc12 Cc1ccc(C(=O)NC2CCCN(CC(=O)Nc3cnc(O)o3)C2)c(F)c1F CC1=NOC(CCNC(=O)CCOCCN(C)C(C2CCS2(=O)=O)=O)C1 N1(C(C2(COC)CCCO2)=O)C(C(=O)NOCC(O)COC)CCC12CC2 Cc1ccc2[nH]nc(C(=O)NC3CN(C(C4CC(F)C(=O)N4)=O)CCC3C)c2c1 Cc1noc2nc(C(=O)N(CCC(C(C)(C)C)NC(C3CC34CC4)=O)C)ccc12 CC(C)CS(=O)(=O)NC(C1CN(Cc2cccc(NS(C)(=O)=O)c2)CCO1)=O n1(C(C)C)cc(Br)cc1C(=O)NCC1CCN1C(C1C(C)CC1C)=O C1(CN(C)C(C2(Br)CC2)=O)CCCN(C(c2occc2F)=O)C1 CC(C)CC(CNC=O)CC(=O)NC1CC(CNC(C2CCC(=O)C2)=O)C1 N1(C(C(C)C(C)NC(=O)CCc2cccnc2)=O)CC(=O)NC(=O)C1 c1(OC)cc(C(N2CCC(C)C(NC(=O)CCc3ccc(C)s3)C2)=O)ccc1F C1(C(=O)NC2(CC=C)CCN(C(C3CCC(=O)N3)=O)C2)CCC2CCCCN12 CCCCC(C)(F)C(=O)N(CCC(C(C)(C)C)NC(c1c[nH]nc1Br)=O)C c1(N2CC(C)(C)C(O)CC2)nc(NCC2=CCCCC2)c2ccsc2n1 C1(C)(CNC(C2CCN(C(C)=O)CC2)=O)COCCN(C(C2(Br)CC2)=O)C1 C(=O)(CS(=O)(=O)C1CC1)NC1C(NC(CCN(c2ccccc2)C(C)=O)=O)C1 Cc1cc(C(N2CCCC2CC(=O)NCC2(O)CSC2)=O)ns1 c1(CNC(N2CC(C)(OC(F)F)C2)=O)cc(O)n2nccc2n1 c1(C(N2C(C(=O)Nc3c(C#N)ccc(C)c3)C=CC2)=O)cccc2cn(C)nc12 N1(C(C(C(CC)O)(F)F)=O)CCN2CCN(C(c3cncc(F)c3)=O)CC2C1 c1(CC(N2CC(C)C(CNC(=O)Cc3ccns3)CC2)=O)ccc2nn[nH]c2c1 CC(C)(O)C(C(=O)NC1CCNCCC1(F)F)NC(=O)C(=O)N1CCCC1 c1(C(=O)OC)nc(=NCC(C)CNC(C23CCCN2CCC3)=O)cc[nH]1 N1(C(CSCC#C)=O)CCOC(CCNC(c2c(Cl)n[nH]c2CC)=O)C1 CCC(C)(CNC(=O)COc1ccccc1)C(=O)N(CC(C)SC)C c1(C(N(C2CCCC(NC(c3c(C)snn3)=O)C2)C)=O)cnc2c(c1)CCCO2 c1(C(=O)NCC2C(C)CN(C(=O)CN(C)C)C2)cc(Cl)c(Cl)cc1O N#CCC(C(=O)N1CCOCC1CNC(C1(C2CCC2)CC1)=O)c1ccccc1 CCC(O)C(C)C(=O)NC(C)CC(C)NC(c1ccc(-n2cnnn2)c(C)c1)=O C1(CC(=O)N(CCNC(C2C(C)(COC)C2)=O)C2CC2)CCC(C(N)=O)CC1 c1(COC(C2CC(c3ccccc3)CO2)=O)ccc(Br)c(C(F)(F)F)c1 C12(C(=O)NCC(C)(CC(C)C)NC(C(C)=CC3CC3)=O)CCOC1CC(=O)NC2 c1(C(N2C(CNC(C(CC)C#N)=O)CC(OC)C2)=O)cnc(C(F)(F)F)c(F)c1 N1(C(C=Cc2cn(C)nn2)=O)CCCC2C(NC(C3SCCS3)=O)C(C)(C)C12 c1(CC(=O)NCCNC(C(CC=C)NC(C)=O)=O)ccc(O)c([N+](=O)[O-])c1 N1(C(C(C(C)O)(F)F)=O)CC2(COC(CNC(c3cc[nH]c3C3CCC3)=O)C2)C1 C(=O)(C1CCCn2ccnc21)N(C)CC1(NC(=O)CCS(C)=O)CC1 Cc1nc2c(C(N3CCC(O)(CCNC(=O)C=CC(F)(F)F)C3)=O)cccc2o1 CC(C)CC(O)C(C)C(=O)N1CCSCC1C(N1CCC([N+](=O)[O-])CC1)=O N1(C(c2ccn(CC)c(=O)c2)=O)CC2CCCC(C1)N2C(=O)CN1CCCCC1 c1ccccc1CCN(C(=O)CS)C.N1(C)CC=CC1.CCC.C1COCCO1 CCC(O)C(C)C(=O)N1CCCCC(N(C(=O)CC2(OC)CCC2)C)C1 c1(C(=O)NC(C(=O)N(CC=C)CCC)C2CCCC2)csc(C)n1 c1(C(=O)NCc2cccc(NC(c3c(C)n(C)nc3)=O)c2)ncnc2c1CCC2 c1(CC(=O)NC2C(CNC(CCS(C)=O)=O)CC2)ccc(Cl)cc1F CC(C(=O)NCCOC1CN(C(C2CCN(c3ccccc3)C2)=O)C1)S(C)(=O)=O c1(CC#N)ccccc1C(=O)NCCC1(NC(c2ccn(C3CCC3)n2)=O)CC1 c1(C(=O)NC2C(C(N(C3C(=O)OCC3(C)C)C)=O)CCCC2)cccc(F)c1F N1(C(C2(F)CN(C(CC(CC)CN(C)C)=O)C2)=O)CC(C)(C)CCC1C c1(C(=O)OC)ccc(C(=O)NCC2CC2CNC(c2cc(C)n(C)n2)=O)cc1F c1(C(N2CCC(C)C(NC(C(=O)NCC)=O)C2C)=O)cnc(O)c2ncccc12 CC(C)CCC(=O)NC1CCC(C)(CNC(C2CC(OC3CC3)C2)=O)C1 C(=O)(C1CCc2cccnc21)NC(C(C)NC(c1cnn2c1CCC2)=O)(C)C c1(OC)cncc(C(N2CCC=CC2C(=O)Nc2conc2C(C)C)=O)c1 Cc1cc(C(F)(F)F)ncc1C(=O)NC1CCN(C(C2(C)C=CCC2)=O)CC1F CCC(F)(F)CCN=c1[nH]c(=NC(C)C2CCOC2)c2c(ncn2C)[nH]1 C#CC1(O)CC(C(=O)OC2CCCN(CC(F)F)C2)C1 CC1COc2c(C(N3CCN(C(c4ccc(O)cc4)=O)CC3C)=O)cccc21 C1(N(C(c2[nH]nc(OC)c2Cl)=O)C)CCN(C(=O)C#CC(=O)N(C)C)CC1C n1(CC=C)c(N2CCC(N(C)C(=O)OC(C)(C)C)C2)nnc1-c1coc(C)n1 Cc1cc(C)c(C(=O)N(C)CC2COCCN2C(C2CCN(CCF)CC2)=O)s1 c1(C(=O)NC2(c3cc(C)no3)CC2)ccc2c(-c3cc[nH]n3)nn(C)c2c1 Cc1oc(C(N2CC3CC2C3NC(=O)CC(C)CC(F)(F)F)=O)cc1S(N)(=O)=O N1(C(=O)NC2COCCOC2)CCCN(Cc2ccc(N3CCCC3)nc2)CC1 C=CCC(C)(CC)C(=O)N(C)CC1(CNC(C2(C)CCCO2)=O)CC1 CCC(C)C(O)C(C)C(=O)NCC(C)(C)C#CC(=O)NC1COCC1F C(=O)(CC(CC(N)=O)CC(C)C)NCC1N(C(CSCC#C)=O)CC2(CCC2)C1 N1(C(C(C)NC(CC)(C)C)=O)CCC(C)C(CNC(C2(CO)CCOCC2)=O)C1 N(C(=NCCc1cc(Br)ccc1OC)NCC1(CO)CCCC1)C(CC)C N1(C(C(CC#C)(C)NC(c2cnc(Cl)n2C)=O)=O)CCCC2(CCC2)C1 C1(CNC(C2CCCC2NC(C2CC2C2CC2)=O)=O)CCCCO1 N1(C(c2cnc(C(C)C)o2)=O)CC2C(C(=O)NC3CCN(C(C)C)C3)C2C1 C1(CC)CC(C(=O)NC2CC23CCC3)CCN1C(=O)CN(C)C(=O)C1CC1 c1(C2C(C)CCC2)nc(-c2ccc(C(F)F)cc2)nn1Cc1ccc(OC)cc1 N1(C(C2C(C)(C)C2)=O)CCCC1(C)CNC(=O)CCCn1c(O)nnc1O C(=O)(C1=CCC(C)(C)CC1)C(C(C)CNC(=O)N(C1CCCCC1N(C)C)C)=O c1(C2N(C(=O)NC3(CC(=O)OC)CS(=O)(=O)C3)CCC2)ccc(O)c(OC)c1 C1(NC(CN(CC)CC)=O)CN(C(c2ccc(OC)cc2Cl)=O)CCC1C C1(CC(N2C(Cn3cc(CCC(=O)O)nn3)CCC2)=O)CC2C=CC1O2 N1(C(c2nc(C(C)C)sc2)=O)CCC(OCCNC(=O)C(C)C2CCCC2)CC1 CC1CC=C(C(=O)NC2CCC(NC(C34CC(C)(CCO3)C4)=O)CC2)CC1 N1(C(C(c2ccccc2)NC(c2n(C)ccn2)=O)=O)CC(O)CC(O)C1 N1(C(C(C)SC)=O)CC2CN(C(C3(N=Cc4cscn4)CCOCC3)=O)CCC12 N1(C(c2ccc(C)nn2)=O)CC2CN(C(C34CCC(C)(CC3)CO4)=O)CC2C1 c1(C(N(CCN(C(CC(CCC)C)=O)C)C)=O)ccc2c(c1)NCC2 N1(C(=O)CC2(C3CC3)CC2)CC2CCC1CN2C(C1(CCF)CCOCC1)=O C1(NC(CC(=C)Br)=O)CC2CC1CN2C(c1c(OC)cccc1F)=O CCCCC(CCCC)NC(C1(C)CC(O)CN1C(c1ccc(O)nc1)=O)=O N1(C(CNC(=O)NCc2ccc(Cl)cc2)=O)CCCC(F)(F)CC1 n1(CCOC)ccc(=NC(=O)C2C3CC(O)C(C3)N2C(=O)Cc2cccnc2)[nH]1 N1(C(CN(C(=O)OCC)C)=O)CC2CC2C(CNC(c2ccccc2OC)=O)C1 N1(C(CC(=C)C)=O)CCCC(n2cc(CNC(C3CCOC3CC)=O)nn2)C1 C1(C(N(CC(c2nn[nH]n2)C)C)=O)CCN(C(c2cc(C(N)=O)[nH]n2)=O)C1C CC1C(NC(=O)CCCC(N)=O)CC2CCC1N2C(C1(CO)CC1(F)F)=O N1(CCN(C(c2c(CC)nc[nH]2)=O)C)CCN(C(=O)CC2(OC)CC2)CC1 Cc1cn2ccc(C(=O)NC3C=CCN(C(C4(C)CC(O)CN4C)=O)C3)cc2n1 c1(C(N2CCC(C)(CCNC(C3ON=C(CC)C3)=O)C2)=O)cccc2nncn12 C1(C(=O)NC2CN(C(C3CC(CC4CC4)C3)=O)C2)(OCC)CCCS1 C1(NC(C2N(CCC)CCC2)=O)CN(C(=O)C=Cc2cnn(C)c2)CC2(CC2)C1 c1(NC)ccc(Cl)c(C(=O)NCC2(NC(c3ncnc(COC)c3F)=O)CC2)c1 C1(C(=O)NCC(=O)Nc2c(F)cccc2F)CCc2ccccc2C1 c1(C(=O)NCC(O)CNC(c2cc(F)c[nH]2)=O)ccc2c(c1)OCCCO2 Cc1ccc(Nc2ncccc2C(C)C)cc1S(=O)(=O)N1CCCC1 C1(NC(C=CC=CCC)=O)CCN(C(=O)C(O)C(C)CC)C12CC2 c1(C(N2CC3N(C(C(C(=O)OC)C)=O)CC(C3)C2)=O)cc(Cl)cc2ccncc12 c1(CC(=O)NC2CCC2CNC(c2cccc(=O)o2)=O)cnc2ccccc2c1 c1(C(=O)NC2C=CC(CNC(c3cnc(OC)nc3)=O)C2)cc(C)n(C)c1C c1(OC)cc(C)nc(N2CCC(C)C(NC(=O)C=Cc3cnc(C)s3)C2)n1 CC1CCCC(CC(N2CC(CNC(=O)CCCCNC(N)=O)CC2C)=O)C1 c1(NCC2(CO)C(C=C)C2)cc(NCC2CCCOCC2)nc(C)n1 CC(CCC(C)(C)C)C(=O)N1CCC1C(=O)NC1CC12CCCC2 N1(C(c2ccc(N)c(Cl)n2)=O)CCC2CC2(NC(c2csc3nnsc23)=O)CC1 C1(NC(C(CC)(C)C)=O)CN(C(C2CCC=CCC2)=O)CCC1C C1(NC(CNC(CCC(C)C)=O)=O)CCN(C(C2(C)CCCO2)=O)CCC1(F)F Cn1nccc1CC(=O)NC1CC(CCNC(=O)CCOCc2ccccc2)C1 N1(CC(=O)NCC(C)(CO)NC(C2CC(n3cccn3)C2)=O)CCC(=O)NC1=O N1(CCCCC)CCC2(CN(C(C3CCCOC3)=O)CC(C)O2)C1 c1(C(c2n(CC)nnn2)NCCC(C)COC)ccc(F)cc1 N1(C(CCCOC)=O)CCCC1(C)CCC(=O)NCC1(C(C)C)CC1 Cc1cc(=O)c(C(=O)NCC2=CCN(C(c3cc(C)n(C)n3)=O)CC2)cn1C C1(C(=O)NC(C(=O)NC2C(C)(C)C2)c2ccoc2)CC12CCCCC2 c1(C(=O)Oc2ccc(OCC(F)F)cc2)ncn2ccccc12 C1(NC(=O)CNC(=O)C2CC2)CC2CC(NC(c3cc([N+](=O)[O-])c[nH]3)=O)CC12 c1(NCC2N(C(Cc3c(C)nccc3)=O)CCC2)ccc([N+](=O)[O-])cc1[N+](=O)[O-] N1(C(COC2(C)CCC2)=O)CCCC(NC(c2ncnn2C2CCOCC2)=O)C1 C(=O)(C(C)(C)C1=CCN(C(C2CCC(=O)N2C)=O)C1)NCC=C=C Cc1ccc(C(=O)NCCC2CCC(NC(=O)C3=COCCC3)C2)c(C)c1 C1(OCCNC(=O)CCN2CCC(F)C2)CCN(C(=O)CC2COCCOC2)CC1 N1(C(C2N(C(c3cc(C(N)=O)oc3)=O)CC(F)C2)=O)CCOCC(F)(F)C1 c1(-c2n(CCN(C)C)nc(-c3cc(F)cc(F)c3)n2)n[nH]c2c1COCC2 c1(CNC2(c3n(CCCOC)nnn3)CN(CO)CC2C)ccc2sccc2c1 c12ccc(Cl)c(c1F)CN1CCC(C1)CC2=O.N1(C)CC2CCCCC2C1.CO O=S(=O)(c1ccc(Br)cc1F)N(c1ncnc2sccc12)CC1(O)CCCNC1 c1(C(=O)NC2CC(C)N(C(c3snc(Cl)c3Cl)=O)C2)cc(F)cc(F)c1O CC1(C)CCCCC(C(=O)NCCCC2CC2(F)F)C1 C1(NC(c2c(C)oc(CO)c2)=O)CC(C(=O)N2CCCC(F)(F)C2)=CC1O CC(C)(O)CC(C)(C)NC(=O)CC(CNC(C1CCC(C)(C)C1)=O)C1CCC1 C1(NC(c2cn(CC=C)nn2)=O)CC2CN(C(c3cc(C(C)=O)on3)=O)CC12 N1(C(C(C=C)(C)C)=O)CC2CCN(C(=O)CC3CCC(C)(C)CO3)C2C1 C1(COC)CN(C(=O)C(C)(C)C(=O)N(C)C)CCN1C(C1CCN2CCC1C2)=O N1(C(COCCCCCC)=O)CCC(NC(c2cn(CCOC)nn2)=O)C(F)C1 c1(NC(C(c2cccc(Br)c2)(C)N)=O)ccc(S(F)(F)(F)(F)F)cc1 C=CCC(CNC(C1CCCN1c1nccs1)=O)NC(=O)CNS(=O)(=O)NC N1(C(c2ccc(-c3ccc(OCC)cc3)o2)=O)CCC2(CCNC2=O)C1 c1(CC(=O)NC2C(C)N(C(=O)C(C)O)CCC2)cc(F)c(F)cc1F c1(C(N(c2ncc(OCC)cn2)C2CCC(N)C2)=O)cc(C)cc(Cl)c1 CCC(C)C(C)C(=O)NCc1ccc(C(=O)NCC(C)(C)C2CCC2)o1 N1(C(c2ccnc(C)c2N)=O)CC2CCC1CC2NC(=O)CC1COCC(C)O1 N1(C(C)=O)CCCCC1C(N1CCCCC1C(N1CCCC2(CC2)C1)=O)=O c1(C(N(CCC2CCN(C(C(CC)N(C)C)=O)CC2)C)=O)cc(N)cc(O)c1C c1(OC)cc(O)c(C(N2CCC(C)C(NC(c3ccc(Cl)s3)=O)C2)=O)cc1OC C1(NC(C(C)CNC(C2(CO)CC2)=O)=O)CC(C)(C)OC1(C)C n1(CC)cccc1C(=O)NCCC(C)NC(c1ccncn1)=O N1(C(C2C(C)(COC)C2)=O)CC(OC)CC(NC(=O)CCCN(C)C(C)=O)C1 N1(C(C(Cc2ccco2)OC)=O)CC2CCCC2(NC(C2CC2(F)Cl)=O)C1 CC(C)(CC(=O)N1CC2CC2(NC(=O)Cn2cc(S(N)(=O)=O)cn2)C1)C(F)(F)F C(CSC)(CN=c1nc(N2CCCC(CO)C2)c2c([nH]1)CCOC2)OCC C1(NC(Cc2c(C)cccc2)=O)CCCCC12CCCN(C(C1C=C1C)=O)C2 C=CCC(CNC(c1cnoc1-c1ccccc1)=O)NC(C1(C)CC1)=O Cc1ccc2[nH]c3c(c2c1)CCCC3NCC1COCO1 C1(CC=C)CCCC1N=c1[nH]c(N2Cc3ccccc3C2)nc2ncn(CC)c12 c1(SC)cc(C(N2CC(C(C)NC(c3csc(Cl)c3Cl)=O)C2)=O)c(C)o1 C12(C(=O)NC(C)CN(C(=O)Cc3nc(=N)[nH][nH]3)C)CC(CC(C)O1)C2 CC1CC(C(=O)N(C2CCN(C(=O)CSC(=N)N)CC2)CC2CC2)CCO1 N1(C(CCC#C)=O)CCC(CO)(NC(=O)CCC(F)F)CC1 N1(C(CCCCCN(C)C(C2(C)CCCN(C)C2)=O)=O)CCC2(CC1)CC2CO C(=O)(C(F)(F)C(O)CCCC)NCC(CCCC)NC(=O)CCCSC(C)(C)C CC1(C)CN(C(=O)CCc2ccoc2)CC1CNC(=O)CSC1CC1 N1(C(CCCC#CC)=O)CCCC2CN(C(=O)C(C(C)(C)C)C3CCCC3)CC12 c1(NC(CC2OCCN(Cc3cccc(OCC)n3)C2)=O)c(C)cc(O)cc1O N1(C(COCCCC#C)=O)CC(CNC(=O)CSCC=C)OC2CCCC12 CN1C2CCCC1CN(C(C1CC1C1CN(C(c3coc(C4CC4)n3)=O)C1)=O)C2 c1(C(N2CC(C)(C(=O)NCc3ccc(C#N)cn3)C2)=O)cn2ccc(Cl)cc2n1 C(=O)(CC(C(F)(F)F)SC)NCC1(CC)CCCCO1.C12(CCC1)C(=O)N2 C(CCNC(=O)CSC(F)(F)F)(C(C)C)NC(C(CC)C1CCOCC1)=O C1(C(N2CC(C)OCCC2)=O)CC2CCCC2N1C(=O)CCC1(C)CC1 c1(C(=O)NC(CC(=O)N(C)CC#N)Cc2cccs2)cccc([N+](=O)[O-])c1Cl c1(CC(=O)NC2(CNC(C3(CCC)CCC3)=O)CC2)ccc(OC)c(Br)c1 c1(CN2CC(n3cc(CNC(C45CC(C4)C5)=O)nn3)C2)cc(F)cc(F)c1 c1(OCC(=O)NC2CC(O)C(F)C2)c(Cl)cc(Cl)cc1Cl C(CN=c1ccc(-c2cccc(OC)n2)c[nH]1)Nc1cc(OC)ncc1 N1(C(CC2(OCC)CC2)=O)CCCC2(CCCN2C(C2(C3CCCO3)CC2)=O)C1 Cc1ccc(-c2cn(CC3CN(C(c4ccc(C)cc4C)=O)C3)nn2)c(C)c1 C1(CC)C(C(=O)NCC2CCC2C)CCCN1C(=O)CCC1CC1(F)F c1(C(N2CC(CNC(CC(C)OC)=O)C3(C2)CC3)=O)cc2ccccc2o1 Cc1nc(CCC(=O)NC(C2CN(C(C3(C)CC3(F)F)=O)C2)C)oc1C c1(CC)ncoc1C(=O)NCCCN(C(C1CCCO1)=O)CC1CCCC1 Nc1cc(F)cc(Cl)c1C(=O)NC1CCC2CCN(C(=O)CC3CCCCC3)C12 N1(Cc2cc(C)[nH]n2)C(C(=O)Nc2cnn(CCN(C)C)c2)CC2CC12 C(=O)(C(C)CC(C)(C)C)N(CCNC(c1c(C)n(C)cc1)=O)CCOCCO C1(C(N2CC(C)(OCC(NOCC#C)=O)C2)=O)Cc2nccn2C1 C1(CN(C(C(C)OC)=O)C)CCN(C(C2CC2C(C)C)=O)CC1 n1(CC)cc(NC(=O)CC2CCCN(C(=O)C(=O)c3ccco3)C2)c(C(N)=O)n1 C1(C)(C(N2CCC(O)(CNC(c3cncc(SC)c3)=O)C2)=O)COCC1(F)F C(=O)C(C)Cc1cnc[nH]1.n12cc(nn1)C2C.N1(N2CC(CC)C2)CCOCC1 C1(NC(C(CC)NC(C)=O)=O)CC(F)CN(C(=O)C(CC)(CC)c2ccccc2)C1 CC(C(=O)N1CCCC(CCC(=O)NC2(C3CC3)CC2)C1)C(C)(C)C CCC(C)CC(C)C(=O)N(C1CCN(C(C2CC23CCCC3)=O)CC1)CC1CC1 Cc1cn2c(n1)CN(C(C1CC(=O)CN1C(C1CCOCC1)=O)=O)CC2 Cc1cc2[nH]c(C(=O)NCC3(F)CCN(C(c4cc(Cl)ccc4O)=O)C3)cc2s1 C=CC(C)(C)CC(=O)N(C)CC1(O)CCN(C(=O)C(c2c(C)noc2C)CC)C1 c1(CSc2cccc(C(=O)O)c2)c(Cl)cccc1[N+](=O)[O-] c1(C(N2CCC(O)(CNC(C34CCC(C3)C4)=O)C2)=O)ccc(Cl)cc1Cl C#Cc1c[nH]nc1C(=O)NCC1CC(NC(=O)C(C)CC=C)C1 c1(C(N(CC(=O)NCCN(C)CC)CC(C)C)=O)cc[nH]c2nccc1-2 C12(C(N3CC(C)(NC(c4nnc(C(C)(C)C)s4)=O)C3)=O)CSCC1C2(F)F Cn1cc(C(N2CC(CNC(=O)C(=O)NCC3CC3)C(F)(F)C2)=O)c(O)nc1=O C1(CNC(CC=CCC)=O)(NC(=O)Cc2ccc(Cl)cn2)CCOCC1 C1(OC)CC(C(=O)NC2CC2(C)C(F)F)N(C(=O)C(C)N2CCCC2)C1 N1(C(C=CC(C)(C)NC(CC2COCC(C)O2)=O)=O)CCC(C)(N(C)C)CC1 N1(C(C2C3(CCN(Cc4c(C)nn(C)c4C)CC3)C2)=O)CCC2CCC(C1)N2C c1(C(c2n(CCCOC)nnn2)NC(C)CCCCSC)c(F)cncc1F C1(C(=O)N(CCNC(C2(CC(F)F)CC2)=O)C2CC2)CC2CCCC2C1 N1(C(c2c(C)ccc(F)c2)=O)CCC2CC2(C(N2CC(N3CCCCC3)C2)=O)CC1 N1(C(CCOC2CN(C(C(c3cncnc3)C)=O)C2)=O)CCCCCCC1C N1(CCNC(COCCCCC)=O)CCC(NC(=O)COCC2CCC2)CC1 CCCCCCn1nnnc1C(c1cccs1)NCC1(CC(C)C)CCC1 C(=O)(CCCCC(=O)NCC1CCCN1C(C1CC1c1ccncc1)=O)NC C(=O)(C1(C)COc2ccccc21)N1CCCCC(CNC(C(C)(C)CO)=O)C1 CCC(C)C(O)CC(=O)NCCN(C)C(c1cnc2scnc2c1)=O C=Cc1cnn(C)c1C(=O)NC1CCCC1CNC(c1cnc(C)nc1CC)=O C1(NC(C(C)N(C(CC2C(C)OCC2)=O)C2CC2)=O)CCCCNC1=O c1(C(N(CC(CC)NC(=O)CCc2ccccc2O)CC)=O)cnc(O)cc1C C12(NC(c3cccnn3)=O)CCCC1N(C(c1cncc(O)c1)=O)CC2 N1(C(C(Br)=C(C)C)=O)CCN(CCCNC(=O)C(C)(C)N2CCCC2)CC1 c1(OCOC)ccc(CN2CC3C(C2)N3C(c2cnc(Br)s2)=O)cc1 C1(NC(C(c2ccc(C(F)(F)F)s2)N(C(C)COC)CCOC)=O)CC(F)(F)C1 N1(C(CC(CC)C2CCC2)=O)CC2CN(C(C3(NC(N)=O)CC3)=O)CC(C1)O2 C1(C(N2CC(C)C(C(=O)N(C)CCOCCO)C2)=O)CCC(C2CC2)C1 C(=O)(C(O)CCC(C)C)NC1CN(C(C2(CCCC)CCC2)=O)CC1F N1(C(c2cnn(C=C)c2N)=O)CC2C=CC1C(C(=O)NCC(F)F)C2 N1(C(CCNc2sc(C)c(C)c2C#N)=O)CC(N)CCc2ccccc21 c1(C(N(CCNC(C2CC2(c2ccc(Br)cc2)F)=O)CCl)=O)ccc(Cl)cc1Cl O=C1CCC2(CC1)CC2C(=O)NC1(c2ccccc2F)CC2(CC2)C1 c1(C(=O)NC(C2CCCN2C(=O)C2=CCCOC2)(C)C)cccc(P(C)(C)=O)c1 c1(CC(=O)NC23CC(NC(C4COCC(C)O4)=O)(C2)C3)ccc2c(c1)COC2 c1(C(=O)NCC2N(C(c3cc(C(C)(F)F)on3)=O)CC2)ccccc1F N1(C(COCC(=C)C)=O)CC(OCCC(=O)NCC(O)Cn2cccn2)C1 C1(CNC(CNC(=O)OC)=O)(NC(=O)COC2CCCOC2)CC1(F)F CCC(CCC(=O)N1CC(c2ccccc2)(NC(C2C=CCC2)=O)C1)OC c1(OC)ncc(C(N2CCC(C)(NC(c3cn(C)ccc3=O)=O)C2)=O)cc1Cl N1(C(CNC(=O)CCN(C2CCC2)C)=O)CCCCC1C1CCCN(C(C)=O)C1 CCC(C)CC(=O)NC1COCCC1Nc1c(NC(=O)NC(C)(C)C)nccc1 CCC(CC)C(C)C(=O)N(C1CCCN(C(=O)C(C2(O)CCCC2)F)C1)CC C(CC(C(=O)NCC1CC(F)(F)CO1)NC(c1cccnc1S)=O)SC CC1(C)C(=O)NC2CCCN(C(=O)NC3C4CCC5C(C4)C35CO)C12 C1(COC)(CNC(C2CCSCC2)=O)CCN(C(C2COCCO2)=O)C1 C1(NC(C2(C)CCCC2)=O)CC=C(C(=O)N2CC(OC(=N)O)C2)C1 c1(COC)ccc(C(=O)NC2(CCCNC(=O)C(n3ccc(C)n3)C)CC2)s1 N1(C(CCOCCC)=O)CCN(C(=O)CNC(=O)OC)CC1C1CCCC1 C1(NCCCC2N(C(CNC(=O)OC(C)(C)C)=O)CCC2)CCc2nncn2C1 c1(C(N2CCC(C)C2CNC(=O)Cc2cccc(F)c2O)=O)cc(O)ncc1F N1(C(C(C)N(C)C)=O)CC(C(N2CC3CSCC(C3)C2)=O)C(C2CC2)C1 CC1(C)OC2(C(=O)NC3COC4(CCN(C(c5cnco5)=O)C4)C3)CCC1CC2 CCC(C)CCCCC(=O)NCCC1CCCN(C(c2cnc(COC)s2)=O)C1 c1(C(=O)NC(C)CC2CN(C(C3(C(N)=O)CC3)=O)C2)nccc2cccnc12 C(CC(C)C)(C(=O)NC)N(C(C(ONC(CCCOC)=O)(C)C)=O)C c1(C(=O)NCC(C)CN(C)C(C2CC2C(N)=O)=O)cncn1C C1(NC(=O)CCc2ncc[nH]2)CCCC12CN(C(C13CCCC1CCC3)=O)C2 C1(C(N(CCOCCCNC(CC=CCCCCC)=O)C)=O)CCNC(=O)C1 O=C(N=c1[nH][nH]c2ccc(F)cc12)NC1CCCn2ccnc21 N1(C(=O)Nc2c(C)sc(C(F)(F)F)n2)CC=C(C(=O)NC2CC2)CC1 N1(C(c2n(CC)cnn2)=O)CCCN(C(=O)Cc2cnns2)C(CO)C1 Cc1ncnc(C)c1OCC(=O)NCC1CC1NC(c1ccsc1C)=O C(CC(C)C(=O)N(CCCNC(C1CC(OC)C1)=O)C)=CC c1(C(N(C2CCN(C(c3ccc(CN(C)C)[nH]3)=O)CC2)CC)=O)cc(=O)cc[nH]1 c1(C(=O)NCC(Cc2ccccc2)NC(C=C=C(C)C)=O)cnc(C)c(C)c1 C12(C(N(CCCN(C(=O)CN3CCC(N(C)C)CC3)C)C)=O)CCCC1CCC2 CC1CN(C(C2(C(F)F)CCCCC2)=O)CC1n1cc(-c2ccc(Cl)cn2)nn1 C(=O)(CCC(C)(C)C)NC1C2CN(C(c3c(CC)nccc3)=O)CC21 N1(C(C(C)NC(=O)C2CC2)=O)CCN(C(c2cscn2)=O)CC1CC(F)(F)F c1(N(CCSC)C)nc2c(c(=NC3CCN(c4cccc(Cl)c4)C3)[nH]1)SCC2 N1(C(CC)=O)CCC2(CC1)CC2C(=O)Nc1cc(O)ccc1Cl N1(C(Cc2nc(C)[nH]n2)=O)CCC2(CC2C(N2C(CO)CC2CO)=O)C1 C1(C(=O)NC(C2CN(C(C34CCCC3CCC4)=O)C2)C)(OC)CCC(F)(F)CC1 CC(C)(O)C(F)(F)C(=O)N1CC2(CCNC(=O)COC3CCC3)CCC1CC2 C1(NC(C(N2CCC(CO)CC2)C2C(C)C2)=O)CCC(F)(F)CC1 c1(C(=O)NC(COC)C(=O)N2CCCC2COC)cc(F)cc(F)c1 c1(C(=O)NCC(CCCC)NC(C2OCCN(C)C2=O)=O)ccc(C)cc1Cl Cc1ccc(C)c(C(=O)NC2CCN(Cc3ccc(Br)cc3)CC2O)n1 Cc1ccccc1CCC(=O)N(CCCN(C)C(C1CCC(C)O1)=O)C c1(CSCCC(=O)N(C)CC2(O)CN(C(C(CC)N(C)C)=O)C2)ccc(C)cc1 C(=O)(C(C)(CC)CCC)NC1C(C(N(CC#C)CC)=O)CCC1 N1(C(COCC#C)=O)CCC2CN(C(=O)C(CC)n3ccnc3)CC2C1 N1(C(c2n(CC)ccc2)=O)CCC(C(N2CC(C)(C(=O)OC)C2)=O)C1(C)C N1(C(C)=O)CCCCC1C(=O)NCCN(C(c1c(O)noc1C)=O)C1CC1 C12CCCC1N(C(C1CCC1N(C)C)=O)C2.N1(CCN(C)C)CCCC1 CC1(C)C(NC(c2nsnc2O)=O)CC1CC(=O)NC1CC2CCC1C2 CC1(C)CC2(CC(N=c3[nH]c(=NCc4c(Cl)cnn4C)[nH]c4c3COC4)C2)CO1 C#CCC(CC(=O)NCC12CCC(CC1)O2)NC(c1c[nH]nc1[N+](=O)[O-])=O C1(C(=O)NCC2CCN(CCC)C2)(CNC(c2cc(C)n(C)n2)=O)CC2(CC2)C1 O=S(=O)(c1ccc(NCC2CSCCO2)c(F)c1)NCC1CC2(C1)CC(F)(F)C2 c1(C(c2n(C(CC)C)nnn2)NCc2cccnc2)cc(C)oc1C N1(C(c2cc(CO)ccc2Cl)=O)CC2CN(C(C3CCC3(F)F)=O)CC2C1 C1(C(=O)NCC2N(C(CC(CC)CC)=O)CC3(CC3)C2)CCc2nnn(C)c2C1 N1(C(CSCCNC(CC(COC)(C)O)=O)=O)CCC12CCCSC2 N1(C(CCCS(N)(=O)=O)=O)CCC(F)(c2ccc(C(F)(F)F)cc2)CC1 C1(C(=O)NC2(CCF)CC(O)C2)(NC(C(c2ccn(C)c2)C)=O)CCCC1 n1(CCC(=O)NCC2N(C(C(C(C)(F)F)(C)C)=O)CC2)nc2ccccn2c1=O C12CCCC1NC2C(=O)NC(=O)OC(C)(C)C.C(CC(=O)N(C)C1CC1)SC c1(C(N(CCN(C(c2ccc(Cl)s2)=O)CC)CC)=O)cnc(O)c(OC)c1 C1(CC(=O)NC2(C)CN(C(C(C)CSCc3ccccc3)=O)C2)CCN(C)C1=O c1(C(=O)NCCCCN(C)C(c2ccc(CO)o2)=O)ccc(F)c2occc12 Cc1cnc(C(c2nnnn2CC(F)F)NCCn2cnnc2CC2CC2)cn1 Cc1nc(C(=O)NC2C3CN(C(=O)CCc4ccsc4Br)CC23)c(C)n1C CC1CC(NC(=O)CCC(N)=O)CN1C(=O)CCCc1ccsc1 c1(NC(C2(C)CCN2C(C2(c3cccs3)CC2)=O)=O)cnn2ccccc12 CC(C)C(O)C(=O)NCC(C)CN(C(=O)CC1CC=CCN1C)C N1(C(c2cc(C)sc2C)=O)CCC2(CC2C(=O)Nc2ccc(O)cc2)C1 C1(NC(C=C(CCC)C)=O)CCS(=O)(=O)C12CN(C(c1c[nH]nc1F)=O)C2 c1(CC)ccc(C(=O)NC(CNC(=O)CC2OCCC2C)C2CC2)c(F)c1 CC1CCC=C1C(=O)N1CCCCC1CC(=O)NCCCS(N)(=O)=O C1(CNC(CC2N(CC)CCC2)=O)CC(OC)CN1C(c1occc1C)=O CC(C(=O)NC1CN(C(=O)CN2C(=O)CCC2=O)CC1n1ccnn1)C(C)O C(=O)(C1CCc2cccc(F)c21)Nc1ccc(C(=O)NCCC)cc1 N1(C(C(C=C)(C)C)=O)CCC2CN(C(c3n[nH]cc3-c3ccccc3)=O)CC2C1 N1(C(=O)OC(C)(C)C)CC(CNC(C)CC2(O)CCC2)C(C)C1 c1(C(N2CCC(C(C)NC(=O)CNC(C3CCC3)=O)C2)=O)cccc(CC#N)c1 c1(C(=O)NC2(C)CCN(C(C3(F)CCCN(C)C3)=O)C2)cc(F)cc(F)c1O C(C(=O)N=c1ccn(C(C)(C)C)[nH]1)(C1CCC1)NC(C(C)=CCC)=O S(=O)(=O)(c1ccccc1-c1cc(Cl)cc(Cl)c1)N1CC(C(=O)NC)C2(C1)CC2 C1(NC(c2ccc(C3CC3)s2)=O)CC(F)(CNC(=O)C(F)(F)C2(O)CCCC2)C1 C=CC(C)(O)CC(=O)NCC1(C)CCN(C(c2ccncc2OC)=O)CC1 N1(C(C(S(C)(=O)=O)C2CC2)=O)CCC2OCCN(C(=O)CCn3ccnc3)C2C1 C(=O)(CCCC(=O)NC1CC(F)(CNC(c2csnc2OC)=O)C1)NCCC CC1(C)OC2CN(CCCN3CC(=O)N(Cc4ccc(Cl)cc4Cl)C3=O)CC2O1 C(=O)(C(C)(C)CCF)N1CC(C(N(C)Cc2c(C)n(C)nc2)=O)C(F)C1 C1(C(=O)NC(CNC(CC=C)=O)CC)CC(F)CN1C C1(NC(CCC(C)O)=O)CN(C(=O)CN2CCC2)CC1(C)C c1(C(=O)NC(CCOCC)C)c(CNC(=O)CC)nnn1C c1(CC)onc(C)c1C(N1CCC(OCCCNC(=O)C=CC2CC2)CC1)=O C(=O)(CCCNC(C)=O)N1C(C(N(C2CCCC2)CC#CC)=O)CC1 CC1(F)CN(C(=O)C(=CC2CCCCC2)F)CCN(C(C2CCCC2)=O)C1 C1(C)(CC)C=C(C(=O)N(C2CN(C(c3cnn4cc[nH]c34)=O)C2)C)C1 CCC(CC(C)C)C(=O)N1CCC(OCC(=O)NCc2csc(C)c2C)C1 c1(OC)ccc2c(=NCC3(C4CC4)CCCO3)c([N+](=O)[O-])c[nH]c2c1 c1(C(=O)OC(C)C)ccc(C(=O)NCCNC(=O)CCc2cccnc2F)cc1 c1(SC)cc(C(F)(F)F)ccc1CC(C)NC(C1CC(SC)C1)=O c1(C(=O)NC2C(NC(C3CC(N(C)C)C3)=O)CS(=O)(=O)C2)ccc([N+](=O)[O-])cc1 C1(C)(C(N(CCN(C(=O)CSc2nnc(S)s2)C)C)=O)CCC2(CC1)CC2 Cc1cc(CNC(=O)C=Cc2cn(C)nn2)oc1C(=O)N(C1CCC1)CCO C1(NC(CCC(C)=O)=O)COC2(CCN(Cc3cccc(O)c3)CC2)C1 c1(NCc2cn(C3CN(C(C)=O)CC34CCC4)nn2)n[nH]c2c1CC(C)CC2 C1(NC(C2(NC(C)=O)CCCCC2)=O)CN(C(=O)C(C)C)CCC1C C1(CCN(C(CC)COC)C)CCN(C(c2sncc2C)=O)CC1 C(=O)(C(C)S(C)(=O)=O)NC(C)CN(C)C.n12cc(nn1)CCNC(=O)C2(C)C C12(NC(=O)NCC3(C)CC(F)(F)C3)CCCN(CC1)C2 C12(NC(CCc3ccn(C)n3)=O)CCC1CN(C(C1CCOC(=O)N1)=O)C2 C1(c2cn(C)nc2)CN(C(C2C(F)(F)C23CC3)=O)CCN1C(c1cn(C)cn1)=O C12(CC(=O)N(C3(C(N(C4CCCCC4)C)=O)CCC3)C3CC3)CCCC1C2 C1(CNC(CC2(OC)CCC2)=O)CN(C(=O)C(N2CCOCC2)C)CCC1(F)F C12(CNC(C3N(C(CCC)=O)CSC3)=O)CC(NC(=O)C=CC3CC3)(CCO1)C2 c1(CCC(N2CCC(C)(NC(C3CCOC3)=O)C2)=O)nc2ncccn2n1 C12(C(=O)NCc3cn(C(C)C)nc3)C(NC(=O)Cc3cc[nH]n3)C3CC1C2C3 c1(C(N(C)CC=CC(=O)NCCC2NC(=O)NC2=O)=O)cc(C)nc(C)n1 C1(F)(CNC(CC(CC)O)=O)CCCN(C(c2cccc(F)c2F)=O)C1 C(=O)(CC(C(F)(F)F)NC(C1(C)CNC(=O)N1)=O)NCCC(C)N(C)C c1(C(N2CCC(CN(C)C(C3C(C)(C)C3(C)C)=O)C2)=O)c(O)ccc(Cl)c1F CCCCCCCC(=O)N1CCC(C(N2CC(NC(N)=O)C2)=O)(CC)CC1 C#Cc1ccc(C(=O)NCC2CCC(NC(c3cnnn3C(C)C)=O)C2)cn1 N#CC1CCC(CC(=O)NCCNC(c2cncc(Br)c2)=O)C1 C(CCCCC(=O)NC1(C(=O)NC2CC2F)CC1)NC(C)=O CCCC(C(=O)N1CC=CC1(C)C(=O)NCc1cc(C)[nH]n1)C(C)C N1(C(C(=O)NC2CCCN(c3cnccn3)C2)=O)CCC(O)C12CCC2 N1(C(c2cc(C)c(F)cc2)=O)CC2CCC(CNC(C3(C(C)(F)F)CC3)=O)(C2)C1 N1(C(CC(C)(C)O)=O)CCCC2CCN(C(c3ccc(Cl)s3)=O)CC12 C(=O)(CC(C(F)F)NC(c1cnc(NC)cn1)=O)NCc1c(CC)nn(C)c1 c1(CC2C(C(=O)NN(C(=O)CCCN(C)C)CC)C2)ccc(Br)c(C)n1 c12cn(C)nc1NC2=O.C(CCOC)(C(N)=O)NC(COCCOCC#C)=O c1(-c2c(SC)c(F)cc(F)c2)n[nH]c2ccc(C(=O)NCCF)cc12 CC(C)(CNC(=O)CNC(c1cnn(C2CC2)c1)=O)CO c1(C(=O)NC2CCN(C(COC(C)Cc3ccccc3)=O)C2)cccc(F)c1F CC1CCc2ccccc2N1S(=O)(=O)NC1CC12CCc1ccccc12 c1(CC(N2CCC(NC(c3cncc(NCC)c3)=O)C2)=O)ccc(F)cc1C N1(C(C2(C)CCCC2)=O)CCCC2(CCC(NC(=O)C=CC3CCCCC3)C2)C1 N1(C(C=CC(=O)N(C)C)=O)CCCCCC1CNC(C12CCC(F)(CC1)C2)=O C1(C(=O)NCC(CCCC)NC(=O)C2=NNC(=O)C2)CCC(S(N)(=O)=O)CC1 c1(CN(CCCNC(=O)CC2CCC(=O)N2)CC)ccnc(OC(C)C)c1 C1(C(=O)NCCN(C(=O)C(F)(F)CC2CCCO2)CCC)CCCCC(C)(C)C1 N1(C(c2c(C)nc(O)[nH]2)=O)CC2(C1)CN(C(=O)CCc1cnc(O)[nH]1)C2 c1(CNC(C2CC23CCN(Cc2cc[nH]n2)CC3)=O)ccc2cncnc2c1 c1(C2CCCN(C(c3c(C)n(CCN(C)C)nc3)=O)C2)ccc(F)c(Cl)c1 C12(CC(=O)NCC3C(NC(C4(C)CCCCO4)=O)C3)CC3CC(C1)CC(F)(C3)C2 c1(-c2nc(OC)sn2)ccc2cc(NC(C3(CN(C)C)CC3)=O)ncc2c1 c1(NC(CCC(C)NC(=O)CSc2nc[nH]n2)=O)ccc(F)cc1O N1(C(C(C=C=C)C)=O)CCOCC(NC(c2cc(C(F)(F)F)ccc2F)=O)C1 Cc1ncc(C(=O)NC2CN(C(=O)CCCc3cnccn3)CC2C)cn1 N1(C(CSC(=N)N)=O)CCN(C2CN(C(=O)CCC3CC3)C2)CC1 C=CCCCCCC(=O)NC1CCN(C(=O)CCc2nc(C)c(C)o2)CC1(C)C c1(C(=O)N(CCC(N2CCCCCCC2)=O)CC2CC2)c[nH]c2ccccc12 c1(C(=O)NC23CC(NC(c4c(C)ocn4)=O)C(OC2)C3)[nH]nc2ncccc12 Cc1cc(C(=O)NCC2CCN2C(C2CC=CCC2)=O)c2cnccc2c1 CC(C)C(C(=O)NCCC(C)(O)C1CC1)C(C)NC(=O)CC1CCCSC1 c1(C(=O)NC2(C)CCN(C(=O)Cn3cccn3)C2)cc(=N)[nH]c(Cl)n1 O=C1NC(=O)C(CCC(N2CC(O)(CCNC(=O)Cc3ccco3)C2)=O)N1 Cc1noc(Cl)c1CC(=O)NC1(C)CC1.N(S(=O)(=O)N(C)C)C1C2CC(C2)CNC1 c1(CC)nc2cc(F)ccc2cc1C(=O)NC1CCCN(C(C2SCCCS2)=O)C1 C1(OC)CCN(C(c2oc(CNC(c3ccsc3C#N)=O)cc2C)=O)C12CCC2 C=CC(C)C(=O)NC1CCN(C(C2CCC2C#N)=O)C1 C1(C(N2CC(CC(C)C)OCC2)=O)C2CCN(C(C3CNC(=O)O3)=O)CC12 c1(CNc2cccc(C(N3CCCC(OC)C3)=O)c2)ccc(Br)cc1I C1(NC(C2(C)C=CCN2C(=O)CN2CCCNC2=O)=O)CN2CCC1(F)CC2 C12(NC(CCNC(=O)OCC)=O)CCCC1CN(C(c1ccc(C)c(F)c1)=O)C2 CC1CC(=O)NCC1C(=O)NCCCC(=O)NCC(N1CCCC1)C N1(C(CCCC(C)NC(c2cc(=N)[nH][nH]2)=O)=O)CCC2(CCOC2=O)C1 N#CC1(NC(=O)CN2C(=O)C=CC2=O)CCN(Cc2nccs2)C1 c1(C(N2C3CN(C(c4c(C)oc(Cl)n4)=O)CC32)=O)cnc2c(c1)CNC2=O N1(C(c2cc(C#C)c(C)cc2)=O)CCC2(CCN(C(C3(C(C)C)COC3)=O)C2)C1 N1(C(C(C)OC(C)(C)C)=O)CCC(N=[N+]=[N-])(C(=O)NCCCN=[N+]=[N-])C1 C1(F)(CNC(c2nc(C)[nH]n2)=O)CCCN(C(C2CCN(C3COC3)C2)=O)C1 N1(C(Cc2nc(NC=O)sc2)=O)CC2CC1CN(C(C13CC4CC1C3C4O)=O)C2 N1(C(c2cc(Br)cc(C)c2C)=O)CCC2CCN(C(=O)C=C3CCCC3)CC12 C(C)(CC(C)(C)C)(c1n(CCC)nnn1)NCC1(P(C)(C)=O)CC1 CCC(CCC(=O)NCCNC(=O)CC1OCCC1C)NC(=O)CO c1(OC)c(C)cc(C)cc1C.C12CCC1CCNC2=O C(C)(CCC(=O)N(C1CCN(C(C2OCCCO2)=O)C1)CC1CC1)OC N1(C(C2(c3ccc(C)s3)CC2)=O)CC2CC1C2NC(C12CCCC1(C(N)=O)C2)=O C1(C2=CCOCC2)(CNC(N(C)Cc2ccccc2)=O)CCC1 C(=O)(CC1=CCN(C)CC1)NC1(C)CC(C(N2CCC(O)(CC(C)C)C2)=O)C1 C1(CNC(C(CC)C(C)C)=O)CCN(C(=O)C(=CC2CCCCC2)F)CC1(F)F C12(C(=O)NC3CC(CC#C)C3)CCC(NC(=O)C(CC3CC3)OC)(CC1)C2 C1(NC(c2nncc(CCC)c2)=O)CN(C(c2cc(C)on2)=O)C(C)(COC)C1 C1(SC)COC2(CCC2)C1.c12cc(oc1C)C(C)(C)CNC2c1nnnn1C C1(SC)C2CCN(C(N3CCOC(CNC(=O)OC(C)(C)C)C3)=O)CC12 Cc1oc([N+](=O)[O-])cc1C(N1CCN(C(C2(C)CC(C#N)C2)=O)CC1C1CC1)=O c1(C(C(=O)NC2CC2)N(C)CCOCC2CC2)ccc2c(c1)CCCC2 Cc1cc(C(N2CCN(CC#N)C(CO)C2)=O)n2nc(C(F)(F)F)cc2n1 c1(C(=O)NC2C(NC(=O)CCc3nc(O)n[nH]3)CCC2)cccc2c1CCO2 c1(C(=O)NC(C2CCOC2)CNC(CCN(S(C)(=O)=O)C(C)=O)=O)cccnn1 C(=O)(C(C)(O)C(F)(F)F)NC1C(NC(CCN(CCCCC)CC)=O)CCOC1 c1(N(CC(C)NC(c2ccc(C)s2)=O)C)nc(-c2cccs2)nc2ccccc12 CC(C(=O)NC1CCN(C(c2ncccc2O)=O)C1)P(C)(C)=O c1(C(c2nnnn2C(C2(C)CC2)C2CC2)Nc2c(C)csc2)ccc(Cl)cc1F C1(C(=O)NCC(C)N(C(=O)C(C2CCOCC2)C)C)COC2(CO)CC1C2 N1(C(c2cncc(C)n2)=O)CCC(F)(C(=O)NCc2cn(C)nn2)CC1 N(C(=NCC=CC1CC1)NCC1CCC1)CCCc1onc(C)n1 c1(NS(=O)(=O)CC2CC(CN3CCCCC3C3CCCC3)C2)ccc(O)cn1 c1(C(C)NC2CCC(C)NC2=O)cc(Br)ccc1F c1(C(=O)NCCCCCCNC(C(C)(C)SC)=O)ccc(O)c2ccccc12 C1(O)(C)CCCN(C(=O)CN2CC3CC3C2)CC1.c1(CCC(C)O)cn(CO)nn1 CC1CN(C(c2ccc(N(C)C)cc2)C(=O)Nc2ccccc2Cl)CC1C(N)=O N1(C(c2cc(OC)no2)=O)CC2(CCCCN(C(=O)C(C)NC(C)=O)C2)C1 C1(NC(CC(C)SC)=O)C(CNC(C2CN3CCN2C(C)C3)=O)CCC12CCC2 C(CCC(C)(C)NC(=O)CCc1cnc(C)o1)NC(C1(C=C)CCC1)=O C1(C)(CC)C=CCN1C(=O)CCCn1cc(Cc2cccc(N)c2)nn1 C1(C(N)=O)CCCCC1C(=O)NC1CCCC(NC(C23CC(CO)(C2)C3)=O)C1 c1(C2C(NC(c3n(C(C)(C)C)ncc3)=O)C2)cccc(F)c1F N1(C(C2(CC)CCCN2C(c2csc(CO)n2)=O)=O)CCCC(F)CC1 C12(C(=O)NCC3(C)C(C)CN(C(C)=O)C3)CC1Cc1c[nH]nc12 CCC(C(=O)N(C1CCN(CC(=O)NC(c2ccccc2)C)C1)C(C)C)C(C)C n1(CCC)nccc1C(=O)NCCC1(NC(=O)CNc2nncs2)CC1 c1(C(=O)NCC2CCN(C(c3cnc(C4CC4)[nH]3)=O)CC2)ccc(F)c(O)c1F C(=O)(C(Cn1cncn1)NC(=O)CCc1cc(C)[nH]n1)NC1(CCCC)CC1 c1(C(=O)NCC2(COC)CN(C(C3(F)CC3C)=O)C2)ccc2nc(C)cn2c1 C1(NC(CSCC)=O)CN(C(C2(Cc3ccc(OC)cc3)CC2)=O)CC1F CC1CC(=O)Nc2ccc(C(=O)NCC=CCNC(=O)C3=CCCCC3)cc2N1 S(=O)(=O)(c1ccc(C)cc1F)N(c1nc(C)cc(OCC)n1)C1C2CCC1CNC2 CCC(C)C(CC(=O)NOCCF)NC(=O)Cc1ccco1 c1(C(=O)NCC(C)NC(=O)C2=COCCC2)cc2c(s1)CCC(C)(C)C2 C(=O)(C1CCc2cc(F)ccc21)NCCNC(C=Cc1cnc(OCC)nc1)=O CCCC(C)(CCC)C(=O)NCC(O)CN(C)C(C1CCCOCC1)=O c1(CC(C(=O)NCCN(C(C(C)(C2CC2)NC(C)=O)=O)C)C)ccc(F)cc1F N=c1cc(C(N2CCC(CCCNC(c3cc(Cl)no3)=O)CC2)=O)cc[nH]1 N1(C(=O)CCCCO)CCC2(CCCN2C(C2CCCCS2(=O)=O)=O)C1 C(=O)(C1COc2ccc(Cl)cc21)N1CCC(CN(C(C(=O)NCCCC)C)C)C1 c1(C(N2CCOC(CCF)C2)C(=O)NCC)c(C)nn(C)c1Cl C1(CC=C)(C(=O)NCC(C)(O)CNC(c2ccc(CC)[nH]2)=O)CCCC1 C1(NC(C2(C)CCCC2)=O)CC2CC(NC(=O)CCN3CCOCC3=O)C2C1 Cc1ccc(O)c(C(N2CCCC2C(C)NC(=O)COCc2nnc(C)s2)=O)n1 O=C(C#CC1CCCOC1)NCC12CCC(CC1)N(C(C13CCCCC1C3)=O)C2 Cc1nnc(CCC(=O)NCC2CC2CNC(C2CC=CCC2C)=O)n1C C1(C(=O)OCC)Cc2cc(Br)ccc2N1C(c1cccc(CC#N)c1)=O N1(C(C(c2ccncc2)C)=O)CCC(N(CC(O)COc2ccccc2)C)C1 c1(C(=O)NC(CC(C)NC(c2cc(C(C)(C)C)c[nH]2)=O)C)cccnc1O c1(C(N2CCC(C)C2CNC(=O)C=Cc2ccoc2)=O)nnc(O)cc1O c1(C(=O)NCC2(CNC(C3CCC(CC)C3)=O)CC2)ccc(Br)cc1 c1(NC(C2CC3CC3N2C(=O)C=Cc2cnccn2)=O)ccc(Cl)nc1Cl C1(C(N(CCCNC(c2ccc(SC)s2)=O)C(C)C)=O)CC2CCCCCC12 CCC(C)C(O)C(=O)NCCN(C(c1ccnc(OCCOC)c1)=O)CC C1(NC(C(C=C)O)=O)CCN(C(C23CCCN2CCC3)=O)CC(C)(C)C1 Cc1ccc(C(=O)NCC2(F)CC(NC(c3nncs3)=O)C2)cc1 N1(C(CCCCC=C)=O)CCC(C)N(C(=O)C(C)NS(=O)(=O)CCCC)CC1 C=CCC(C)C(=O)NCCC1CC(NC(c2cn(C)c(O)n2)=O)C1 N1(C(c2ccc(COC)s2)=O)CCN(C)CC1CNC(C1(O)CCOC1)=O C1(NC(CCOCC#C)=O)CC(NC(c2cnco2)=O)C(O)C1 c1(OC)nc(Cl)ccc1S(=O)(=O)NCc1nc(C2CCCCC2N=[N+]=[N-])no1 N1(C(=O)C(O)C2CCC2)CCC(C(F)(F)F)n2ncc(I)c21 CC1(C)CCC1NC(=O)CCC1CCN(C(C2COCCO2)=O)C1 C1(NC(C2CC(=C)C2)=O)CCN(C(=O)CCC2C(=O)NN=C2C)CC(C)(C)C1 c1(N2CC(SC)C2)ccc(S(=O)(=O)NCc2nn(C)cc2C)cc1C#N c1(C(C)N(C(=O)C=CCNC(=O)CC2CCSC2)C)cccs1 C(CCC(C)C)(C(=O)NC1C2CCCC1CO2)NC(CCCCC#C)=O C(=O)(CC1=NN(C)C(=O)C1)NC1CN(C(CC2(OC)CCOCC2)=O)C(C)C1 C#CCC(CC(=O)NC1(CC)CCCCCC1)NC(c1ccc(O)c(F)c1)=O O(Nc1ncnc2c1ncn2C1CCC1)CCCc1ccccc1 c1(C(=O)NCC2CN(Cc3cccc(I)c3)CCO2)ccc(Br)cc1 Cc1c(C(=O)NCCC2(NC(=O)CCCC(N)=O)CCC2)sc2cccc(F)c12 Cc1cc(OCC(N2CCN(C3CCOC3)C(=O)C2)=O)cc(C)c1Br C1(CNC(C=C(C)C)=O)CC(C(=O)NC2COCC2N(C)C)=NO1 C(CC(=O)N1CC(CC2CC2)C1)(C(F)(F)F)NC(c1nc(N(C)C)oc1)=O C1(CC(=O)N(CCCN(C)Cc2cnn(C)c2)C)CC2CCC1O2 C1(C(C(=O)NC(C)C2CC2)C)CCCN(C2CCN(c3ccc(Cl)cc3)C2=O)C1 Cc1nc(CC(C)C)oc1C(=O)N(CC(C)(C)CNC(=O)CC(C)(O)C1CC1)C c1(C2N(c3cc(S(C)(=O)=O)ncn3)CCC2)ccc(S(C)(=O)=O)c(F)c1 C1(CCNC(=O)CCc2cnco2)CCC(NC(c2ccoc2Br)=O)C1 Cc1cnc(NCC2CN(C(c3csc(Cl)c3)=O)CC2C)nc1O C#Cc1cncc(C(=O)NC(C)C(C)NC(c2c(C)ccn2C)=O)c1 c1(C(C)NC(C23C(CN(S(C(C)C)(=O)=O)C2)C3)=O)cc2ccccc2cn1 C(C(=O)N=c1cc(C)o[nH]1)Oc1c(OC)ccc(CN2CCc3nocc3C2CC)c1 N1(C(c2ccc(C(Cl)Cl)cc2)C(=O)NC2CC2)CCC12CCOCC2 C1(CCNC(NOCc2cc(C)on2)=O)COCCN1C(=O)OC(C)(C)C N1(C(C2CCN(CC)C2)=O)CC(C(=O)NCCc2cocn2)C(C2CC2)C1 Cc1ccc2c(c1)CC(C(=O)N(CCCCNC(=O)C=Cc1ccsc1)C)S2 CC(Cn1cccn1)C(=O)NCC1(C(=O)NCC2CC2Cl)CC1 Cc1c(Br)c(C(=O)NC(CNC(C2COCCO2)=O)C(C)C)nn1C c1(CC)ccc(C(=O)NC2CN(C(c3ccccc3NC)=O)CC23CC3)c(C)n1 c1(CC)onc(C(=O)NCC2(F)CC(NC(=O)Cc3cncc(O)c3)C2)c1C c1(OC)ccccc1CC(C)CC(=O)NCC1CC(C)N(C(=O)COCCF)C1 C1(NC(C2CC23CC3)=O)CCN(C(c2cnn3cc[nH]c(=O)c23)=O)CC12CCC2 C1(C(=O)NC(CCCNC(C=CCC)=O)C)CCC(C)(O)CC1 c1(C(N(CC(=O)NCC(C)NC(=O)CC2CC2)C)=O)csc(=N)[nH]1 C(=O)(C1=NNC(=O)CC1)N1CCCC(C(C)NC(=O)CN2CCCC2=O)C1 C1(O)(C(C(=O)NCC(C)NC(=O)OC)F)CN(C(C2CS(=O)(=O)C2)=O)C1 CC1CC(NC(=O)C=C2CCCCC2)CCN1C(C1COC(C)O1)=O c1(C(N(C)CC2CCCN2C(C2CCNC2=O)=O)=O)cc2c(O)ncnc2cn1 C1(C(N2CC(CCNC(c3cnc(C(C)=O)s3)=O)C2)=O)CCc2nn[nH]c2C1 Cc1oc(C)c(C(=O)NCC2(NC(c3c[nH]c(C#N)c3)=O)CC2)c1Br c1(C(=O)NC(CNC(C(CC)(F)F)=O)CCOC)c(C)nc2sccn12 C1(CNC(c2cnc(C)[nH]2)=O)CN(C(c2cccnc2SC(F)F)=O)C2CC12 c1(C(=O)NC2CC(C)(CNC(C3(CCC)CCC3)=O)C2)ncn2c1CCCCC2 C12(NC(c3nc(COC)sc3)=O)CCCN(C(c3ccc(F)s3)=O)CC1C2 N1(CCN2CCOCC2)C(=O)CN(CCSCCCC)C1=O.C(C(=O)OC)S N1(C(C2C(CNC(CC)=O)C2(C)C)=O)CCC(F)(F)CC1 N1(C(c2cc(O)nc(Cl)c2)=O)CCC2CN(C(C3C4CC5C(C4)C35)=O)C2C1 c1(OC)cc(OC)nc(N2CCCC2CNC(c2cc(F)cnc2Cl)=O)n1 CC(C)CC(F)C(=O)NCCOCCNC(=O)CC1CCCCC12CC2 C(=O)(CCC(C)(C)C#N)N(CC(=O)O)Cc1cn(Cc2c(C)nc(CC)o2)nn1 N1(C(C(CSC)O)=O)CCCC2(CCN(C(C3(CC(C)C)CC3)=O)C2)C1 N1(C(CCc2onc(C(C)C)n2)=O)CC2(CCN(C(C3COC(=O)N3)=O)CC2)C1 c1(OC)c(C(=O)NCC2(O)CCN(C(C3(C(F)(F)F)CCC3)=O)C2)ncnc1C C(CC(=O)NC1CCSC1)(C(F)(F)F)NC(c1nn(C)c(=O)cc1)=O CC(CCC(=O)N1CC=CC1Cn1cc(-c2nccn2C)nn1)N(C)C C1(C(=O)NC2(C(F)(F)F)CC2)CC(F)(CN(C(=O)C=CCN2CCOCC2)C)C1 c1(C(N2CC3CN(C(c4nn(C)c(F)c4)=O)CC3C2)=O)cccc2cnccc12 C1(NC(COCCCOC)=O)C=CCCC1C(=O)NCCCCSC CC(C)CC(C(=O)NOCCOCCO)NC(C1CCC(=O)C1)=O N1(C(C2(CC(=O)OC)CCCC2)=O)CC(NC(=O)C=C(C)C(F)F)CC(F)C1 CC(C)(C)C(CNC(=O)Cn1cnc(C(N)=O)n1)NC(c1ccc(F)nc1)=O C1(NC(c2ccc(C(C)C)s2)=O)CCN(C(=O)CSCCC#N)C1(C)C C1(NC(C(C)N(C(=O)COCC(C)C)CCC)=O)CCCN1 Cc1ncnc(O)c1C(N1CCCN(C(c2cccc(C(F)F)c2)=O)CC1)=O CC(C)(C)CC(C(=O)NCCOC(=O)C1CC1)NC(C1CC=CCC1)=O C(=O)(C(CCC)S(N)(=O)=O)NCC(CC=C)NC(C1CC(n2ccnn2)C1)=O C(=O)(CC1OCCc2sccc21)NC(CNC(c1c(C)c(C(F)(F)F)n[nH]1)=O)C N1(C(CCOCC(C)C)=O)CCN(C(C2(CF)CCC2)=O)CC1 C1(C(=O)NC(C=C)CO)CN(C)CCN1C(c1cnncc1OC)=O CC1(C)C(=O)Nc2ccc(C(N3CC(NC(C4COC4)=O)CC(O)C3)=O)cc21 C(c1ccco1)=CC(=O)NC(C(=O)N(CCCn1ccnc1)C)C1CCCO1 C(=O)(CC(C)(C)N(C)C)N(C1CCN(C(=O)C(C)OC(C)=O)C1)CC Cn1cccc1-c1cc(C(N2CC(CNC(C3CC3c3ccco3)=O)C2)=O)n[nH]1 N1(C(C2N(C)C(=O)NC2)=O)CC23CCCC2(C1)CN(C(C1C=CCCC1)=O)C3 N1(C(C(COC)OC)=O)CCC(NC(=O)COC(F)(F)F)C(O)C1 c1(OC)ccc(C(C)=CC(N2CCCN(C(c3ccoc3)=O)C(C)C2)=O)cc1 N1(C(C(C)S(N)(=O)=O)=O)CCC2(C1)CN(C(=O)C(C)(C)c1cscn1)CCO2 CC1(C)CN(C(c2[nH]nnc2C2CC2)=O)CC1CNC(=O)CC#N O=C(N=c1[nH][nH]cc1Br)C1=NOC2(CCN(c3ncc(Br)c(C(F)(F)F)n3)C2)C1 N1(C(C(C2CC2)OC)C(=O)NC(C)C)CCC2(CC1)CN(C)C(=O)O2 C1(C)(C(=O)NCC2(C)CCN(C)C2)CN(C(=O)C2=NNC(=O)C2)C(C)(C)C1 CCC(CC)C(F)C(=O)NC1CC(C)(CNC(=O)COCc2nc[nH]n2)C1 CCCC(C)CC(=O)N1CCC(NC(c2cnn(-c3ccccn3)c2)=O)C1 C(=O)(C1=Cc2ccccc2C1)N(CCCCNC(C1CC2(CC2)CO1)=O)C1CC1 C1(NC(C(CC)(CO)OC)=O)CC12CCN(C(=O)CC1CCCOC1)CC2 C1(NC(=O)Cn2ccnn2)CN(C(C2CCCOCC2)=O)CC1n1cccn1 CC1(C)CCCC(C)(NC(=O)C(CCC2CCC2)NC(=O)CC(C)(C)C(F)F)C1 CC(C(=O)NC1CCN(C(c2nncs2)=O)CC1F)S(C)(=O)=O C1(C(=O)NC2C(C(=O)NC3CC(C(C)O)C3)CC2)CC(C)(C)CO1 c1(C(=O)NC2CC(C)(CNC(C3CCC(=O)N3)=O)C2)cn2cccnc2n1 C(c1ccc(O)c(O)c1)=CC(N1CC(O)(CNC(CC2(C)CC(F)(F)C2)=O)C1)=O C1(C(=O)NC(CNC(c2nc(SC)[nH]c(=N)c2)=O)C)Cc2ccccc2NC1=O c1(OC)cncc(C(=O)NC2(C3CCCN3C(=O)CN(C)C(N)=O)CC2)c1C O=C1C(=Cc2cc(Cl)ccc2OCC(=O)NC2CCNC2)Cc2cc(Cl)ccc21 c1(-c2cc(NCc3nc(C)oc3)ncc2)cc(O)c2ccoc2c1 N1(C(N(C2(c3ccc(Br)cc3)CCC2)C(c2c(C)cnnc2)=O)=O)CC2CC2C1C#N C1(C(=O)NCC2C=CCOC2)(CC)CCN(C(=O)C(O)Cn2cncn2)C1 CCCC(C)C(=O)N1CC(SC)C1.c12ccc(cc1)-c1cn(nn1)C2 C1(CN(C(C(N2CCCCCC2)C)=O)C)CCN(C(=O)CC2CC=CCC2)CC1 c1(C(COCC(N2CC(CCCCNC(C=C(C)C)=O)C2)=O)C)cccc(F)c1 c1(CCC(c2n(CC)nnn2)(C)NC2(C(=O)NC)CC2)cccc(Br)c1 C(=O)(C(F)CCC(C)C)N1CC2(N(C(c3c(C)scn3)=O)CC2)C1 C1(NC(c2c(CC)nc(C)[nH]2)=O)CCN(C(c2ncoc2Br)=O)C(C)C1 N1(C(C(C2CC2)OC)=O)CCCC(N(C)Cc2ncc(-c3ccc(C)cc3)o2)C1 c1(C(C)NC(=O)NCC(N(OCC)C)=O)ccc(C#N)cc1OC N1(C(C(CNC(C(C)CCN(C)C)=O)CC2CC2)=O)CCC2(COC(=O)N2)C1 c1(SCC)cc(Cl)ccc1C(=O)NC1CC(NC(C2(C)COC(=O)C2)=O)C1 C1(CC(=O)NC(CC#C)CC)C2CCCC2N1C(=O)CC1(C#N)CCOCC1 C(N=c1nc(C(C)C)cc(C)[nH]1)C1CC2CN(C(CCOCCOC)=O)CC1C2 C1(OC)CN(C(=O)CCc2ccsc2)CCC1CNC(=O)C(C)COC Cc1ccc2[nH]c(C(=O)NC(c3ccc(C#N)cc3)CF)cc2c1C Cc1ccc(C(=O)NCCCOCCN(C)C(C2CC(N(C)C)C2)=O)nc1O CC1(C)CCC=C1C(=O)N1CCN(C(c2ccc(C(F)F)nc2)=O)CC1C1CC1 N1(C(c2cc(C)nn2C)=O)CCC(NC(C2CC2C(N)=O)=O)C(F)C1 CC1OC2(C(=O)NC(c3cccc(Br)c3)CC3CC3)CCC1CC2 c1(C(=O)NC2C(O)CCN(CCN(C)C)C2)nnc2c(Cl)cc(C(F)(F)F)cn12 CCC(CN(C(=O)C=CC(C)(C)NC(C1CCCSC1)=O)CC)CC N1(C(CCc2n(C)cnn2)=O)CCCCC1CCNC(C1CC2CC1C2)=O C1(NC(C2N(C(C(=O)NC(C)C)=O)CCC2C)=O)CC(C)CCC1O n1(CC)cc2c(n1)CC(C(=O)NCC1CCOCC1(C)C)CC2 CC1(C)CN(C(C23CCC(CC2)C3)=O)CC(C)(C)C1NC(=O)CCC1CCOC1 C(c1ccc2ncccc2c1)=CC(=O)NC(C)CCNC(=O)Cc1ccccn1 CC1(C)CCc2cnc(N3CCC(n4ccnc4)CC3)nc21 N1(C(=O)NCCCC)CCC2(CCN(C(=O)Nc3ccc4ccccc4c3)C2)C1 c1(N2C3CC(NC(C4(CC)CCC(O)CC4)=O)C2CC3)ncnc2[nH]ccc12 N1(CC(=O)NC(CC)CNC(=O)Cc2csc(CC3CC3)n2)CC2CCC1C2 C1(C(=O)NC2CC(NC(c3cc(C(N)=O)[nH]n3)=O)C2)CCn2ncnc2C1 C1(CC)(CO)CCN(C(=O)C(C)N(C(=O)C(CC2CC2)OC)C)C1 C(=O)(C1=COCCO1)N1CCC(N(CCC)C(C2CCC2C#N)=O)CC1 Cc1nc(N(C)C)sc1C(=O)NCC1CN(C(=O)C=Cc2ccn(C)c2)C1 N(C(=NCCNS(C)(=O)=O)NCC1CCOC1)C(C#C)CCC C1(NC(c2ccc(CSC)o2)=O)CC(C)CN(C(=O)COCCN(C)C)C1 CC1CCCC(CNC(C2(NC(=O)CCc3cnn[nH]3)CC2(C)C)=O)O1 N1(C(C(CC#C)(C)C)=O)CC(NC(=O)CC=CCC)CC2(CC2)C1 CCC(C(=O)NCC(C)NC(c1cc(C(C)C)ccc1C)=O)C(C)(C)CC C1(NC(C(CCCC)(C)F)=O)CCC2(CC1)CC(NC(=O)CNC(=O)OCC)C2 Cc1ccc(C(=O)NC2CC3C=CC2O3)c(-n2cc(C(C)(C)O)nn2)c1 CC(C)(O)C(F)(F)C(=O)N1CC2C(NC(c3csc4nnsc34)=O)C2C1 C(CC(C)(C)C)(C(=O)NCC1CCN1C(C1(C#N)CC2(CC2)C1)=O)OC c1(C(=O)NC2C(NC(c3cc(C)sc3)=O)CC2)c(C)noc1C(C)C CC1(CNC(=O)C(O)C(F)(F)F)CCCN(C(=O)CNC(N2CCCC2)=O)C1 Cc1ccc2nc(C)c(C(=O)N(CCNC(C34CCC3C4)=O)C(C)C)cc2c1 C(C(C)C(=O)NC1CC1CNC(=O)C(CO)N(C)C)SC c1(CCC)nc(C(O)Cc2ccccc2F)n(-c2ccc(SC)cc2)n1 C12(CNC(C(CC=C)(C)C)=O)CN(C(c3n[nH]cc3Br)=O)CC(F)(C1)C2 c1(OC)ccc(C(=O)NC(C)CCNC(=O)Cn2c(C)ccc2C)c(F)n1 c1(C(N(C)CC2(NC(C(C)=CC3CC3)=O)CC2)=O)ccc(OC(F)(F)F)c(C)c1 C1(C(N2C3CC(NC(C4C(C)CC(C)O4)=O)C3CC2)=O)CN2CCCN1CC2 N1(C(CS(=O)(=O)NCC)=O)CCCC(CC)(NC(=O)Cc2ccccc2)C1 Cc1nccc(C(N2CCCC(CN(C(=O)CSc3n[nH]c(O)n3)C)C2)=O)n1 Cc1cc(C(=O)NC2CCC(CNC(C3(C)COCCO3)=O)C2)cc(N)c1Cl C1(C)(C(=O)NCCC(CCC)C2CC2)CN(C(=O)C(C)(F)F)CC1C C1(C(N2CC(CCNC(c3cc(OC)nc(C)c3)=O)C2)=O)CCn2nncc2C1 N1(C(C(C)CCO)=O)CC2(C1)CN(C(=O)C(c1ccccc1F)(F)F)CCO2 c1(CC(N2CC(N3C(=O)CC(NC(C=CC=CC)=O)C3)C2)=O)ccc2[nH]ccc2c1 Cc1nc(C(F)(F)F)oc1C(=O)NC(C1CCCN(C(=O)Cn2cnnn2)C1)C C1(OC)CC(CNC(c2ccc(O)cn2)=O)N(C(c2ccc(F)o2)=O)C1 c1(SC)ccc(C(=O)NCCC2(NC(=O)CC(C)C3CCCO3)CCCC2)cc1 CC1CCc2n[nH]cc2C1C(=O)NCCN(C)C(c1sccc1CN(C)C)=O c1(C(N2C(C)(C(=O)Nc3nccc(OC)c3I)CC2)=O)cnn2cccnc12 C(=O)(CC(C(C)(C)C)NC(c1cncc(CO)c1)=O)N1CCC(=C)C1 Cc1cncc(C(N2CCCC2C(C)(C)C(=O)NCc2ncc(C)s2)=O)c1 c1(C(=O)NCC(CC(C)C)NC(CCCC(C)=O)=O)c(F)ccc(C)c1Cl C1(NC(c2cc(C(C)(F)F)n[nH]2)=O)CN(C(=O)C(C)(C)C(F)F)CCC1CO Cc1nc(N(C)C)sc1C(N1CC(C)(NC(=O)CCOCC(F)F)C1)=O C(CCCC(=O)NOC(CO)C(C)C)N(C(C(CCOC)(C)O)=O)C N1(C(C(C)O)=O)CCC2CCC(C1)N2C(=O)Cc1c(F)cc(C#N)cc1Br C=CCC(C)(CC)C(=O)NC1CC=C(C(=O)N2CCSC(CC)CC2)C1 c1(C(=O)NC2CN(C(=O)CCc3ccncn3)C2)c(Cl)ccc(Cl)c1O c1(N2CCCN(C(c3c(OC)cccn3)=O)CC2)ncnc2ccc(O)cc12 C(=O)(C(F)C(C)CNC(=O)C(COC)COC)N(C1CC(=C)C1)C C1(CC(=O)NC2CCC(CNC(C34CC(C)(C3)C4)=O)C2)(OC)CCCCC1 C1(N(C(C)C)C2CC2)CC(=O)N(C(c2ccccc2O)C)C1 CC1CCCCC1(CNC(=O)CN(c1ccncc1)C)NC(=O)C#CC1CC1 Cc1c(C(=O)NC(C2CCOC2)CNC(=O)C(F)=CC2CC2)cnc2ncnn12 C(=O)(N(CC)OC)C1(CC)CC1.c12cc(on1)CNC2=O N1(C(c2sccc2C(F)F)=O)CCC2CN(C(=O)CCc3nncs3)CC2C1 c1(NC(C2N(C(CC(=O)OC)=O)CC(O)C2)=O)ccc2ncn(C)c2c1 c1(C(=O)OC)c[nH]c(=NC2CCCC(NC(=O)CC3COCCO3)C2)cn1 CCS(=O)CC(=O)N1CC(C)(CCC(=O)NCC(C)(COC)OC)C1 n1(CC)nc(C)c(C(=O)NC2C=CCN(C(C3CC3C(=O)NC)=O)C2)c1Cl c1(C(N(CC(C)(C)NC(C(C)NC(=O)OC)=O)C)=O)sccc1SC S(=O)(=O)(c1cccc(CN)c1)Nc1c(=O)cc(C(=O)OC)n(C)c1 C12(C(N(CC(=O)OC)C3CC3)=O)CC(C)(CN1C(=O)CSc1cn[nH]c1)C2 C1(CNC(C(C)C)=O)C(C)CCCN1C(c1ccnc(OCC(F)(F)F)c1F)=O C#CCCCCNC(=O)C#CCNC(c1cc(Cl)cs1)=O c1(C(=O)NC(C)CNC(=O)Cc2csc(C3CCOC3)n2)cccn2ccnc12 N1(C(Cc2ccc(C)s2)=O)CCC2CCN(C(c3cc(C(F)F)nn3C)=O)C2C1 N1(C(C2CCN(C3CCCC3)CC2)=O)CC(NCC2CCC2)CC12CCCOC2 C1(CNC(c2c(C)nncc2)=O)CN(C(C2CC2C(C)O)=O)CCN1C C1(C(=O)NC(COCC)C)CCC(CNC(c2cscc2Cl)=O)CC1 c1(-c2ccc(NC(C3=NOC(c4n(C)ncc4)C3)=O)s2)nc2cc(C)cc(C)c2s1 C(=O)(C1=C2CCN=C2NC=C1)N1C2CC(CN(C(C34CCC(C)(OC3)C4)=O)C2)C1 CC1C(NC(=O)C(Cl)=CCl)CCCN1C(C1CC1c1ccsc1)=O C1(CC(=O)NCC2CC(NC(Cc3cn(C(C)(C)C)nc3)=O)C2)CC(F)(F)C1(F)F c1(C2(C(=O)NC3CN(C(C=CC(CC)C)=O)CC3C)CC2)ccc(Cl)c(Cl)c1 C1(NC(=O)COCCc2cccs2)C=CC(CNC(C2C(C(=O)OC)C2)=O)C1 c1(C(N2C(CN(C)C)CCCC2)C(=O)NC(C)(C)C)cc(Br)cc2[nH]ncc12 C(=O)(C1CCCc2cccnc21)C(C1(N(C)C(C2CC(=O)CO2)=O)CC1)=O.CN C(=O)(C1=NOC(CNC(C2(CC3CCC3)CC2)=O)C1)N1CCCC(CC)C1 CCC(O)CC(=O)NCCC(C(=O)NC1CCN(S(C)(=O)=O)CC1)OC N1(C(C2(CO)CCN(C(C=C(C)C)=O)C2)=O)CCC2(CCN(C)C2)C1 c1(C(N2CCCC(CC)(NC(C3CC(SC)C3)=O)C2)=O)ccc(F)c(OC)c1F N1(C(c2nc(C)n(C)n2)=O)CCC(C2CC2)C1CNC(=O)C1=COCCO1 O=C(CCCn1cccn1)NC(Cn1ccnc1)C(=O)NC(CCO)C1CCC1 C1(NC(CC=CC)=O)C=CCCC1C(=O)NC(C)CCCCO C(=O)(CCCC(F)(F)F)NCC1(CNC(c2ncc(N(C)C)nc2)=O)CCCC1 C1(C(=O)OC)CC(F)(F)CC1C(N1CCC(O)(CNC(=O)CN(C)C(C)C)C1)=O CC1CC2CN(C(C3CCC4(CC4)N3C(c3cc(CO)on3)=O)=O)CC12 C(c1ccc(F)cc1)=CC(=O)NCCCNC(C(CC)C1CCOCC1)=O C(=O)(CC(C)C1CCCCC1)NCCC(C)N(C)C(C1(F)CCCC1)=O C1(CNC(C2CCC(C)CC2)=O)CCN(C(=O)C(F)n2ccnc2)CC1O C1(NC(C2(C)CCC2)=O)CC(NC(c2csc(Cl)n2)=O)C12CCC2 CCC(CC)(CCNC(C1CCN(C2CC2)S1(=O)=O)=O)NC(C1CC1F)=O C(=O)(C(C)(C)C1=CCSCC1)NCC1CN(C(C=C(C)C(C)(C)C)=O)C(C)CC1 c1(CC2C(C(=O)NCC3(O)CN(C(c4cnn[nH]4)=O)C3)C2(F)F)cccc(Cl)c1F C1(C(=O)NC(C2CCC2)C)COC2(C1)CN(C(=O)C(C)(C)F)C2 Cc1nc(CC(C)C)sc1C(=O)N(C1C2CN(C3CCSC3)CC12)C(C)(C)C CCCS(=O)(=O)CC(=O)NC1COCCN(C(=O)COCC(=O)OC)C1 C12(CNC(C(F)=CC)=O)CCCC1N(C(=O)COCP(C)(C)=O)CCC2 C(=O)(CC(C)(C)CCC)NC(CCCC)CNC(=O)C(C)S(C)(=O)=O c1(C(N2CCOCC(F)(COC)C2)=O)sc(S(N)(=O)=O)c(OC)c1OC N1(C(CCNC(C(C)(C)C)=O)=O)CC(NC(=O)C2=C(Cl)CCCC2)CC(F)(F)C1 CC1=C(C(=O)N2CC(NC(c3cc(C4CC4)n(C)n3)=O)CC2(C)C)COCC1 c1(C(=O)NC(C2CCN(Cc3nccs3)CC2)C)cc(Br)c2ccccc2n1 c1(C(=O)NC2C(C)(CN(C(CCOC)=O)C)CCC2)ccc(Cl)c(N)c1 Cc1cnnc(O)c1C(N1CC(C(=O)NCC2CCC2(F)F)CC(C)C1)=O c1(N(C(=O)CN2CC(C(F)F)C2)CCCCSCC(=O)OC)cccnc1NC.CO c1(Nc2cc(NCCCOCCCO)nc(C)n2)cc(Br)c(F)cc1C CC1(C)CC(CNC(=O)C=Cc2ccco2)N(C(C2CC=CCC2)=O)C1 N1(C(c2c(Cl)csc2Cl)=O)CC2(C1)CN(C(C1(CO)CCC1)=O)CCO2 c1(OC)c(C(=O)NC2CCN(C(C3(C)CCOC3)=O)C2)sc(C)c1Br Cc1ccc(C(C)NC(N2CCC(Nc3ncccn3)C2)=O)s1 c1(C(=O)NC2C(NC(CCn3ccc(C)n3)=O)CC2)ccnc(N(C)C)c1 Cc1cocc1CN(Cc1ccccc1)CC1CCC1 Cc1cc(F)sc1C(=O)NC1CCCC1CNC(c1csc(Cl)c1Cl)=O C1(=CC(=O)NC(C)CN(C)C(C2(C(F)(F)F)CCC2)=O)CCSCC1 N1(C(C(CC#C)(C)C)=O)CCCC2(CCC(NC(c3ccn(C)c3)=O)C2)C1 C1(NC(CCCC(C)c2ccccc2)=O)CC2(CCN(C(=O)C#CC(C)(C)C)C2)C1 C(CC)(CC(=O)NC1CCC1C(=O)OC)N(C(C(COCC)C)=O)C C(C(C)(C)CNC(=O)C(C)NC(C)=O)N(C(=O)CC1CCC2CC12)CC N1(C(C(C)CC2CC2)=O)CCCC2C1CCN2C(C12COC(CF)(C1)C2)=O c1(CCN2CCCC(C(C)N(C(=O)C(N)=O)CCO)C2)ccc([N+](=O)[O-])cc1 C(CCC(C(=O)N1CC2(CCC2)C1)NC(=O)C(F)(F)C(F)F)OC C1(NC(c2ncc[nH]c2=O)=O)CCCN(C(=O)Cn2ccc(C3CC3)n2)CC1F c1(C(N2CCC(NC(C3CC4CCC4C3)=O)C(O)C2)=O)c(Cl)cccc1[N+](=O)[O-] c1(C2C(C(=O)NC3CC(C)(NC(=O)C=Cc4nccs4)C3)C2)ccncc1F C1(CNC(C=CCN(C)CC)=O)C(CC)CCN1C(C1CC12CCCC2)=O c1(C(N(C)CC2CCCN2C(c2ccc(Cl)o2)=O)=O)cnn2c1CC(F)(F)C2 Cc1cc(C(F)F)oc1C(=O)NCC1(O)CC(NC(C2(n3cncn3)CC2)=O)C1 c1(C(=O)NC(C)(C)CCCNC(c2cn(CC3CC3)nn2)=O)ccc(Cl)cc1Cl Cc1ccc(CC(=O)NCCCCC(C)NC(c2cn(C(F)F)cn2)=O)c(C)c1 C(=O)(CC(C(F)F)n1cccn1)NC(CC)(CC)CCN C(C)(C)(CN=c1nc(SC2CC2)[nH]s1)C1CCN(C(C(C)CN(C)C)=O)CC1 CC1CN(C(c2cn(C3COC3)nn2)=O)C(C)CN1C(=O)COCC1CC1 c1(C(N(CCC(C)NC(C2(CC(C)C)CCC2)=O)C)=O)nnn2c1C(=O)NCC2 C(CC(C)(C)C)(C(=O)N1C(CC(N2CC(OC(C)C)C2)=O)C2CCCC12)OC c1(CC(=O)NC(COC)C(=O)NCc2cocn2)cncnc1O C1(C(N2C(C(C)O)CCC2)=O)CCCC(NC(C2CCN(C)C2)=O)CC1 c1(C(=O)NC(CCSC)C(=O)N(C)Cc2cc(C)cs2)cncc(F)c1C C1(c2cn(C)nc2)CN(C(C2(C(F)F)CCC2)=O)CC1NC(C1CCOC1)=O N1(C(c2cc(C)[nH]n2)=O)CC2CC(C)N(C(=O)C(C3CCCO3)C3CC3)C2C1 C1(NCc2cn(C)c(-c3ccccn3)n2)CCNCCC1CO.c1ccc(S)cc1 CCN=C(NCc1cc2cc(C(=O)OC)sc2s1)N1CCCC(CC)C1 c1(COC)nc2c([nH]1)CCN(C(C1C(=C)CN1C(=O)OC(C)(C)C)=O)C2 c1(C(N(CCCNC(c2coc(Br)n2)=O)C2CC2)=O)cc2ccccc2cn1 c1(SCC(=O)NCC(N(C(=O)C(F)n2ccnc2)C)C2CC2)cnn(C)c1 C(=O)(CCCCC(=O)NC1CN(C(=O)C(=Cc2cccs2)C)CC1N=[N+]=[N-])NC c1(C(=O)NC(CNC(Cc2c(C)n(C)nc2)=O)C(C)C)coc2c1COC2 C1(CC(=O)NC2(CO)CCC2)CCN(Cc2cnc[nH]2)C1 Cc1cc(C)n(Cc2nc(Cc3ccccc3F)nn2CC(N)=O)c(=O)n1 N1(C(CCC)=O)CCCC(CO)(NC(=O)C=C(C)C)C1.c12cccc(c1)C(=O)N2 N1(C(C2CC(SC)C2)=O)CCCN(C(c2nocc2C2CC2)=O)CC1CO N1(C(C(CSC)O)=O)CC2(C(N3CCC3CN=[N+]=[N-])=O)CCC1CC2 c1(OC)ccc(F)cc1S(=O)(=O)NC1CCN(C(C2CCCN2C(C)=O)=O)CC1 c1(CNC(c2cncc(C#N)c2)=O)ccc2cncn2c1 C(C(=O)NCC(C)(C)NC(c1occc1C)=O)(C(C)C)c1cnc(C)s1 CN1CCC(CC(=O)NCC2CC2NC(c2ccoc2Cl)=O)C1=O C(=O)(C(C)CC(N)=O)NCCC1(OC)CN(C(=O)CN2CCC2C)C1 Cn1nc(C(=O)NCc2csc(CNC(c3ncoc3C3CC3)=O)n2)cc1O c1(OC)ccccc1C(C)CC(=O)NC1CCC(NC(c2c[nH]nc2F)=O)C1 C1(NC(CN(CCC)C)=O)CN(C(=O)Cn2nnnc2C)C2CCCCC12 CC1(Cc2cccc(F)c2)CCCN1C(=O)C(=O)Nc1ncccc1Cl CN1CCC(C(=O)NC2CC3C2CCN3C(c2ccc(O)nc2)=O)S1(=O)=O C1(NC(c2cnc(C)[nH]2)=O)CC2(C1)CN(C(C1(C)CC3CCC1O3)=O)C2 N1(CC=C)CC(C(=O)OC)C2(CN(C(=O)OC(C)(C)C)C2)C1 c1(C(=O)NC(CCC)CNC(c2cc(C)sn2)=O)cnc2cccc(C)n12 C1(O)(CNC(CCCN(C)C)=O)CCN(C(c2ccc(CCF)cc2)=O)C1 C1(N(c2ccc(F)cc2)CC)CCCN(N2CCC(n3cc(C)cn3)C2)C1 CN1CCN(C(C2CCC(=O)N(C)C2)=O)C(C(=O)NOC2CCCCC2)C1 N1(C(c2n(CCOC)ncc2)=O)CCCCC(CNC(=O)C(F)=C(C)C2CC2)C1 c1(C(N2CCC(OCCNC(C=CCN(C)C)=O)C2)=O)cc[nH]c(=N)c1 CN1C(=O)CCC1CC(=O)NCC1(CNC(=O)C=Cc2ccc[nH]2)CCCC1 c1(CCC(=O)NC2C(NC(c3c(C)ncn3C)=O)CC2)ccc(F)c(F)c1F c1(SC)cc(C(N2CC3CC2C3CNC(C)=O)=O)ccc1NC(C1(O)CC1)=O Cc1cccc2c(C(=O)NC(C)CNC(c3nc(O)nc(O)c3F)=O)coc12 C(=O)(CCS(N)(=O)=O)NCC(CC)(CC)NC(c1cn(CC)nc1C(F)(F)F)=O N1(C(CC2C(C)C2(F)F)=O)CCCN(C(=O)C=CC(=O)N(C)C)CC1 c1(NC(c2c(-c3ccncc3)cncc2F)=O)cccn2nccc12 N1(C(CCc2nc(C)c(C)[nH]2)=O)CCC2CN(C(=O)CN(c3ccncc3)C)C2C1 C1(NC(c2n[nH]c(CC)c2C)=O)CCCC(C(=O)N(C)Cc2n[nH]c(C)n2)CC1 C(C)(C)(CCCCC(=O)N1CCCC(CN(C)C(c2cccc(O)n2)=O)C1)OC CC12CCC(C(N3CC4CCCC3(CNC(c3cccnc3)=O)C4)=O)(CC1)CO2 C(=O)(C(CNC(C1(C)CCCC1O)=O)CC1CCCC1)NCC1(C)CCC1 C(=O)(CC(C)C(=O)OC(C)(C)C)NCCC(=C)CNC(C1(C(C)(C)C)CCC1)=O c1(C(=O)NCCN(C(=O)CN(C2CCCC2O)C)CC)cc(C)nn1C c1(SC)cc(=NC(=O)C2CC=CC(NC(C3CC3(C)C(F)F)=O)C2)[nH]n1C C#Cc1cncc(C(N2CC(NC(=O)COc3cc(F)cc(F)c3)CC2C)=O)c1 Cc1coc(C(=O)NC2CCCC(CN(C(=O)CC(F)(F)Cl)C)C2)c1C c1(N2CC(NC(c3cc(CN(C)C)on3)=O)C(C)CC2)ncc([N+](=O)[O-])cc1Br c1(OC)nc(C)ccc1C(=O)N(CC(C)O)CCNC(=O)CCc1nccs1 c1(C(=O)NC2CC(CCNC(C3CCC(C)(CC)O3)=O)C2)ccc(OC)c(N)c1 O=C(C1Cc2c(Cl)cccc21)N1CC(C(=O)OC)OCC1=O.N12CCC(CC1=O)C2 C1(CNC(C2C(OC)CCC2)=O)CC2(CO1)CN(C(c1cc(Cl)ccc1F)=O)C2 C(CCS(N)(=O)=O)NC(C1CC(CNC(C(C2CC2)OC)=O)OC1)=O N1(C(c2ccc(C)nn2)=O)CCC(CNC(c2nnc(O)cc2O)=O)C1(C)C N1(CC(=O)NCC2(NC(CNC(=O)NC)=O)CCCC2)CCS(=O)CC1 N1(C(C2C(=C)C2)=O)CCc2c(c(CNC(=O)CCc3cccnc3)nn2C)C1 c1(C(=O)NCC2CC(NC(Cc3nc(C)sc3)=O)C2(C)C)cc(C#N)ccc1Cl c1(C(C(=O)NC)N(CCCCOC(C)(C)C)C)csc2c(Br)cccc12 N1(C(CNC(CCCCC)=O)=O)CC(NC(c2ncn(C(C)C)n2)=O)CCC1C Cc1oc(Br)c(C)c1C(=O)NCC(O)CC=Cc1ccccc1 CCCN=C(NCCc1sc(C)nc1C)NCc1ncc(C(F)(F)F)cn1 C1(CCNC(c2c(C#C)c[nH]n2)=O)CN(C(C23CC(C)(C2)C3)=O)CCS1(=O)=O N1(C(c2ccc(=N)[nH]c2Cl)=O)CC23CCCCC2(C1)CN(C(=O)C1=NOCC1)C3 CCC(C(=O)N1CC(CC(=O)NC(C)CN=[N+]=[N-])(OC)C1)n1cncn1 C(c1ccco1)=C(C)C(=O)N(CCCCCNC(C1(C)CC1F)=O)C N1(C(CC(C=C)C)=O)CCCCC(NC(=O)CCCC(C)=O)C1 c1(C(=O)NC2CCN(C(C(C(=O)OCC)OC)=O)C2CC)cccn2nccc12 C(CC(=O)NCC1(F)CCN(C(=O)COCCOC)CC1)(C(C)C)OCC c1(OC)ccc(F)cc1C(F)(F)C(=O)NC(CNC(=O)C=C(C)Cl)CC(C)C CCC(C(=O)NCCNC(=O)NC)NC(=O)C=Cc1ccsc1 c1(CC)nnc2cc(NC3CC(NC(=O)CC4CC(C)(C)CO4)C3)ncn12 C1(C(=O)NC2(C)CC=CC2)CCN(C(=O)C(O)C(F)(F)F)C(C)(C)C1 C1(C(N2CCCC2C2(NC(C3CCOCC3)=O)CC2)=O)CC2C=CC1O2 C(CC(=O)N1CC(O)(c2nn[nH]n2)C1)(C(C)(C)C)NC(C(C)OCC(C)C)=O CN(Cc1cnn(-c2ccc(Br)cc2)c1)N1CCC(CCO)(CO)C1 c1(NC(COC)C2CC2)cc(NCC(n2cccn2)C)nc(C(F)(F)F)n1 C1(OC)C2CC3CC1CC(C(=O)NCC(C(C)(C)C)NC(=O)C(F)C(C)C)(C3)C2 C(CN=c1[nH]cncc1I)C1CCC(NC(c2ccoc2Cl)=O)C1 C1(C=C)(C(N(C(C#C)C)C)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C1 c1(NC(=O)NC2CCC(CC)C2)cnc2c(c1)c(=O)n(C)c(=O)n2C N1(C(C(C)n2cccn2)=O)CCN(C(=O)C2=COCC2)CC1c1ccccc1Cl Cc1cc(C(C2CCC2)NC(=O)C(=O)NC(C)C(C)CC)c(C)o1 C1(CN(C(=O)C(F)C2CCC2)C)COCCN1C(c1ccnc(CO)c1)=O CCCCCC(CC)C(=O)NC1(C2(CC)CC(c3ccccc3)CC2)CC1 C(=O)(C(F)CC1CCCCC1)NC(CNC(C(c1cnn(C)c1)OC)=O)C1CC1 N1(C(C(CC(C)C)F)=O)C2CCC1CN(C(C1CCS(=O)(=O)CC1)=O)C2 C(=O)(CC(C)(C)CCOC)N(C(CNC(C(C(C)C)NC(=O)OC)=O)C)C c1(OC)ccc(C(CNC(=O)NC(C)Cn2cnnc2)CO)cc1OC CS(C)(=O)=NCC(=O)N1CCN(C(=O)CSCC2CCCO2)CC1c1ncc[nH]1 c1(C(=O)NCC(C)NC(=O)C2Cc3c(Cl)cccc32)nnc(O)c2ccccc12 c1(CNC(C(N2CC(SC)C2)=O)=O)ccc(S(=O)(=O)NC2=NCCO2)cc1 c1(C(=O)NC(C)(C)CNC(C2CCC3(CC3)C2)=O)csc(N=S(C)(=O)N(C)C)n1 C1(NC(COc2ccc(C)cc2Br)=O)CCCCN(C(=O)C#CC2CC2)CC1 CCCCC(C(=O)NC(C)C=CC(=O)NCCCCN(C)C)ON=C(C)C n1(CCNC(C=CC(C)C)=O)cc(C(=O)NC2(CO)CC(F)C2)nn1 C(=O)(C1=CCCCCC1)NC(CCSC)C(=O)NCCCOC(=O)N(C)C N1(C(c2n(C)ncc2C2CC2)=O)CCC(C)(C)C(NC(c2ccc(Cl)cc2)=O)C1 c1(C(=O)NCC(C)(C)COCC)c(OC)cccc1O Cc1cc(F)cc(C)c1C(N1CCN(Cc2nccn2C(F)F)CC1)=O c1(C(=O)NC(CNC(c2c(CC)n(CC)nn2)=O)C)cn(C)c(=O)n1C N1(C(C(CC(C)(C)C)O)=O)CC(NC(c2cccc(F)c2)=O)CC12CCCC2 c1(CC(=O)O)c(C)cc(C)nc1O.CCC1CN1C(C1CCCO1)=O.C1(O)CCCC1 C(=O)(CS(=O)c1cccc(OC)c1)NC1CC(NC(C=CCC)=O)C1 C(=O)(C(F)(F)C1CCOCC1)N1C(CNC(=O)CCC2CCOC2)CC1 N1(C(Cc2nnc(C)o2)=O)CCC(O)(CNC(=O)C(C)Cn2ccnc2)C1 CC(=O)CCN=C(NCc1nnc2n1CCCCC2)N1CCC(c2nncs2)C1 C#CC1CN(C(c2cnc(O)n2C)=O)CCN1C(c1ccc(C)c(C)c1)=O C12(CNC(Cc3cc(C)no3)=O)CC(NC(c3csc(C(C)C)n3)=O)(C1)C(C)O2 c1(C(=O)NC2C3CC(NC(C=Cc4cnc(C)s4)=O)CC32)cn2cnnc2cn1 C=C(C)C1OCCC1C(=O)NC1CC2(C(=O)NCC(C)SC)COC1C2 C(=O)(C(C)C(F)(F)F)NCC1CCCCN1C(c1n(CC)cc(Cl)c1)=O N1(C(C(CCC)C(=O)OC)=O)CC(NC(C2CC(O)C2)=O)CC12CCOCC2 Cc1ccc(C2CC2C(=O)NCCOC(C)(C)CNC(=O)CC2CC=CC2)s1 Cc1cc(C(=O)NC(C)CN(C)C(c2cccc(C3CC3)c2)=O)ccc1[N+](=O)[O-] C1(OC)CN(C(c2ccc(Cl)c(C)c2)=O)CCC1NC(c1cc(Br)cnc1F)=O N1(c2ncnc(CC)c2F)CC2CC(NC(c3cc(C)cc(Cl)c3)=O)CC1C2 c1(C(=O)NCCN(C)C(C2(C#N)CC2C(F)(F)F)=O)cnc2ccc(F)cc2c1 c1(CC)cccc(C(N2CCC(NC(C3CCC(C(F)(F)F)CC3)=O)C2)=O)c1N C1(F)(CNC(C(C=C)O)=O)CCC(NC(c2cnccc2C(F)F)=O)C1 C(=O)(CC(O)C(C)CC)N1CCC(C#C)(C(N2CC(N(C)CC)C2)=O)C1 c1(C(=O)NCCCC(C)NC(c2scnc2Cl)=O)ccc(=O)n(O)c1 c1(N2CC(CO)OC3(C2)CCC3)nc2c(F)c(Br)ccc2s1 C(c1cccc2ccccc12)=CC(=O)N(CCNC(C1CCOC(C)C1)=O)CC N1(C(c2ccc(COC)o2)=O)CC(NC(c2ncnc(O)c2F)=O)CC1(C)C C1(NC(c2c(C)nc(Cl)s2)=O)CN(C(c2c(F)cncc2F)=O)CC(F)(F)C1 C1(N(C(c2c(CNC(C(CC3CC3)OC)=O)ccs2)=O)C)CCC(F)(F)C1 c1(OC)nc(C)c(C(N2CCCC2C(C)NC(c2c(C)cnn2C)=O)=O)s1 N1(C(Cc2c(OCC)cccc2)=O)CCCC2CN(C(=O)CS(=O)(=O)NC)CC12 c1(C(=O)NCC2C(CC(=O)N(C(C3CCOCC3)C)C)C2)nn(C)cc1Cl N1(C(c2ccc(CC)[nH]2)=O)CC(C)C(N=c2nc(N(C)C)cc(C(F)(F)F)[nH]2)C1 C(CC(C(=O)NC(c1ccccc1F)C)NC(=O)CCCOC)=CC N1(C(c2c(C)ncnc2O)=O)CCCC(O)(CNC(=O)C(F)(F)C(F)F)CC1 CCCC(CC(C)C)C(=O)N1CC(CCNC(=O)C=CCF)C(C)C1 N1(C(C(CC)CC)=O)CCCC1C1CCCN1C(=O)COc1ccc(C)cc1 C1(C(=O)NCC(CNC(C2CCC(NC(C)=O)CC2)=O)F)CN(C)CCN(C)C1 c1(C(=O)NC2CCC(C)N(C(=O)C=C3CCC3)C2)ccc2c(Br)nn(C)c2c1 N1(C(CCc2c(C)noc2)=O)CCC(O)C1CNC(=O)CC1CCC(C)CO1 C1(C2CCN(C(C3NC(=O)CC3C)=O)C2)(NC(C2C(C)C2)=O)CC1 c1(C(=O)NC2(C)CCN(C(c3sccc3C#N)=O)C2)cc2ccc(F)cc2s1 Cc1csc(Cl)c1C(=O)NCc1cccc(NC(=O)COCCF)c1 N1(C(c2cc(CCC)[nH]n2)=O)C2CCC1C(NC(=O)C(C)CSC(F)(F)F)C2 C(=O)(C1=C(Cl)CCC1)NC(C1CCN(C(=O)CSc2ccc(F)cc2)C1)C CC(C)CCCC(=O)NC(CC1CC1)C(=O)NCC(C)(C)C(F)F C(=O)(C(C)(C)C(=O)NCCn1ccc(C(=O)NCCOc2cnn(C)c2)c1)NC C1(N(C(=O)CCN(C(=O)CCCC2CC2C)CCO)CC)CCCCC1C N1(C(c2c(C)nsc2N)=O)CCC(C)C(NC(=O)C(C2CCCCC2)O)C1 C1(NC(C=C(C)Cl)=O)CC(CO)N(C(=O)CCC=CBr)C1 N1(c2nccc(N(CC(=O)NC)C)n2)CCNC(=O)C(F)(F)C1 C1(NC(c2cc(=O)cc[nH]2)=O)CC2C1CCN2C(c1cc(C(F)(F)F)no1)=O c1(C(=O)NC2COCCN(S(=O)(=O)C3CC3)C2)cc(Br)cc([N+](=O)[O-])c1F C1(CONC(C2(C)CC(NC(COCC(=O)NC)=O)C2)=O)COCCC1(F)F CC1CCN(C(=O)C(=O)NC(CNC(=O)CCC2CC2)C2CCC2)CC1 N1(C(CC2C(C)C2)=O)CCN(C(=O)C(C)Cc2cccc(F)c2)CC1CC1CC1 C1(C(N2CCC(CN(C(c3cc(C)sc3C)=O)C)C2)=O)CCCNS1(=O)=O CCC(O)CCc1cn(CCC(=O)N(C(C)C)Cc2ccc(SC)o2)nn1 N1(C(c2n(C)ncn2)=O)CCC(NC(=O)CC(C)(C)C2CC2)C12CCC2 C(=O)(CC(O)C(C)CC)NC(CC(=C)Cl)C(=O)NCC1(CCC)CCCC1 c1(OC)cc(OC)cc(C=CC(N2CCN(C(=O)CC3(C)CC3)CC2CF)=O)c1 C1(C(=O)NCCOC2CCN(C(C=CC)=O)C2)CCS(=O)(=O)N1 N1(C(c2ccnc(C(C)C)n2)=O)CC(NC(=O)C2=NOCC2)CC2(CC2)C1 N1(C(=O)Nc2ccc(O)cc2F)CCCC2(C1)CN(C(C1COCC1O)=O)C2 C1(CCC(=O)NCc2c(CC)nco2)CCCN(C(=O)C(O)C2CC2)C1 Cc1cccc(C(C)C(=O)NC2(CNC(=O)C=CC3CCCC3)CCC2)c1 c1(C(=O)NCC(C(C)(C)C)NC(c2cnc(CC)[nH]2)=O)cc(C)c(Cl)cc1F C(=O)(CC(C(F)(F)F)NC(C1CCC(=O)N1)=O)NCCc1c(C)nn(C)c1 CC1=C(CNC(=O)C(c2cccs2)NC(=O)CC2C=CCC2)COCC1 N1(C(C(CC)CCOC)=O)CC2CCCC(C1)N2C(=O)CCC(C)O c1(C(=O)OC)cc(S(=O)(=O)NNC(=O)C(N)Cc2ccc(O)c(O)c2)ccc1Br C1(CC(N2CC(N(C)CC)C2)=O)CN(C(c2cc[nH]c2C)=O)CCC1C N1(C(C=COCC)=O)CCC(O)(C(C)NC(c2cc(-c3cnn(C)c3)on2)=O)C1 N1(C(C(=O)NCC)=O)CCN(C(c2ccnn2C)=O)CC1CCO C1(C)(CC)CCN(C(=NCCOCC(C)(C)O)NCc2ccnn2C)C1 c1(C(N2CCCC(CCNC(CC(CC)C)=O)C2)=O)cn2cc[nH]c(=O)c2n1 C1(C(N2C(CNC(c3csc(Br)c3)=O)CCCC2)=O)CC2(C1)CC21CC1 CCCCCCC(C)C(=O)NC(C1CCN(C(=O)C2=NNC(=O)CC2)CC1)(C)C c1(NCC(=O)NC(C)(CNC(=O)CCN2CCCC2)C2CC2)ccccc1Cl C1(CC(=O)NCCc2c(CNC(c3c(C)cns3)=O)nco2)CCCCC1O Cc1cc(C(=O)NC(CNC(C2(C(F)F)CCC2)=O)C2CCC2)c(O)c(C)c1 N1(C(c2c(C)ccc(C)n2)=O)CC2(C1)CN(C(C1COC(C)(C)CO1)=O)CCO2 c1(C(N(C)Cc2cc(Cl)c[nH]2)=O)cc(O)nn1C C1(O)(C(C)NC(=O)CCc2cnn(C)c2)CN(C(c2coc(CO)c2)=O)C1 C(CCCCC(=O)NCC1OCC2CCC1C2)N(C(=O)CSC(C)(C)C)C N1(C(c2c(NC)nccc2)=O)CCCN(C(=O)CC2CCCNC(=O)C2)CCC1 C12(NC(=O)C(F)F)CCOCC1CN(C(c1cc(F)ccc1C(F)F)=O)C2 O=C1NC2(CO1)CC(C(=O)NCC1(NC(C3CC4(CCC4)CO3)=O)CCOC1)C2 C(=O)(C(F)(CNC(=O)CC1CC(C)=NO1)C(C)C)NCc1ccc(CC)cn1 CCC(C)(C(=O)N1CC(NC(c2ccc(Cl)c(C)c2O)=O)C2(CC2)C1)C(N)=O N1(C(c2n(C)cc(Cl)c2)=O)CCC2(C1)CN(C(=O)CC1CCCC(=O)N1)CCO2 CCCCCC(O)C(=O)N1CCCCC1CCCNC(c1cnc(NC)cn1)=O N(C1CC2(CN(C(=O)CCc3cnccn3)C2)n2ccnc21)C(COCC#C)=O N1(C(C(C)(O)C2CCC2)=O)C2CCC1CC(NC(c1coc(Cl)c1)=O)C2 N1(C(c2n[nH]c(C)c2N)=O)CC2CC(NC(=O)C=C3CCC(C)C3)CC2C1 n1(CC)ccc(C(N2CC(NC(=O)C(N3CCCC3CO)=O)C(O)C2)=O)cc1=O Cc1c(C(=O)NCC2CN(C(=O)C(C)(C)CC3CC3)C2)cnn1CC1CCCO1 N1(C(C2C(C(=O)OC)C2)=O)CC2(C1)CN(C(=O)CCc1ccc(C)o1)CCO2 C1(NC(C(C23CCC(CC2)C3)NC(c2cc(C(C)C)[nH]n2)=O)=O)CCS(=O)(=O)C1 N1(C(C(C)Sc2ccc(OC)cc2)=O)CC(NC(=O)CC(C)(C)C)CC(F)C1 C1(C(=O)NCC2(CCC(=O)N(CC(C)(O)C3CC3)C)CCC2)CC2CCC2C1 C1(CNC(c2c(O)ncc(CC)c2)=O)CC2CCC(C1)N2C(=O)CS(C)(=O)=O C(=O)(C1=CCCCO1)N1CC(N(C(COCCCC)=O)CC2CC2)C1 c1(OC)ncc(F)cc1C(N1CCC(CC(=O)Nc2ncc(CO)cc2Br)C1)=O c1(C(N2CC(CNC(C3C(C)OC(=O)N3)=O)C(C)C2)=O)cc2cc(Cl)ncc2[nH]1 N1(C(C2C(C(=O)OC)CC2)=O)CCC2(CCN(C(c3csc4nnsc34)=O)C2)C1 c1(C(N2CCC(C)(NC(C(C(C)C)OCC)=O)C2)=O)onc2cc(C)ccc12 c1(C(=O)NC2CCC2NC(c2ncoc2C2CC2)=O)cccc(CF)c1 C(=O)(C1=CC2C=CC(C1)C2)N1C(CN(C(CCN(CCC)C)=O)CC)CCCC1 C1(C2CCCN(C(c3[nH]nnc3C3CC3)=O)C2)(NC(C(CC)C(C)O)=O)CC1 O=S(=O)(c1ccc2ccccc2c1Br)NCC1CC12CCOC2 C(C(C)(C)CC(=O)NCC1(CNC(c2ccc(N)c(N)n2)=O)CCCCC1)OC C1(NC(CCCCC#C)=O)CCN(C(c2cncc(N)c2)=O)CCC1CO c1(SC)ccc(-c2nn[nH]n2)c(NC(C2CC(c3nc(C)no3)C2)=O)c1 C1(C)(C(N(CCN(C(CS(CC)=O)=O)C)C)=O)CCC(C(=O)OC)C1(C)C C1(CN(C(=O)C(C)N2CCC2)CC)CCN(C(C2CCCOC2C)=O)CC1 CCC(CC)C(C(=O)N1CCS(=O)(=O)C(CCNC(=O)CC(C)(C)OC)C1)OC C1(NC(C2(CC)CCCN2C(=O)CCn2cncn2)=O)CNC(=O)C1(C)C c1(OC)cc(C(=O)NC(C(N2CCCC2C(=O)N(C)C)=O)C2(O)CCC2)on1 C(=O)(CCC(=O)NN(C)C)N1CCCC(CCC)(NC(=O)C(C2CCC2)OC)C1 N1(C(C(C)(C)N(C)C)=O)CCCC(CNC(=O)CC23CCCN2CCC3)CC1 O=C(C1=CC2CCCC12)NCC1CCCN1C(c1nccn2ccnc12)=O N1(C(c2c(C)nn(CC)c2C)=O)CCC(C)N(C(c2cnc(C)cn2)=O)CC1 c1(CSCC(=O)N(C2CC(NC(C(c3cccnc3)C)=O)C2)C)cccnc1 CCC(CC(C)C)C(=O)N1CCCC(C(C)Nc2cc(F)ncn2)C1 N1(C(c2cccc(C)n2)C(=O)NC2CCOC2)Cc2cncnc2C1 C12(NC(CC(C)C)=O)CCC1CN(C(c1nccnc1N)=O)C2 C12CC(C1)CCC(=O)N2.N1(C(CC2(CSC)CC2)=O)CCC1CN(C)C C(c1ccc(Cl)cc1F)=CC(N1CCN(C(CCNC(=O)NC)=O)C2C1C2)=O c1(C(N2CCCN(C(=O)C=Cc3cn[nH]c3)C(CO)C2)=O)cccc2scnc12 c1(C(=O)NC(CNC(C2C(CN(C)C)C2)=O)(C)C)ccn2cncc2c1 Cc1nc(N2CCCC(C)(CNC(c3cc(CF)on3)=O)C2)cc(C#N)n1 N1(C(c2n[nH]c(=N)s2)=O)CC2CCCC(NC(c3[nH]nc([N+](=O)[O-])c3Cl)=O)C2C1 c1(C(=O)NC2COC3(C2)CN(C(=O)CCn2ccnn2)C3)ccc2c(c1)COC2 c1(C(=O)NC(CC(C)NC(=O)CCc2n[nH]c(=N)s2)C)ncn2c1COCC2 N1(C(C(C=C)O)=O)CCN(C2CCN(C(c3cnc(C)[nH]3)=O)C2)CC1 CC(C)C(O)C(C)C(=O)NC(C1(O)CCCCC1)C(=O)NCCCOCC1CC1 N1(C(C(c2ccccc2)OC)=O)CCN(Cc2ccncc2)C2CC12 c1(OC)c(C(=O)NC2(C)CN(C(=O)C(C)C(F)F)C2)ccc2c1CCC2 c1(CCNCC2N(CC(=O)Nc3ccc(Cl)cc3)CCCC2)cccc(Br)c1 c1(CCC)ccc(C2C(=O)NCCN2CCOC)s1.C(CO)OC CCCCC(CNC(c1ccc(COC)[nH]1)=O)NC(c1cc(Cl)ccn1)=O CON(CCC(=O)N(C1CCCC1)CCF)C(=O)C1CCC2(CCC2)O1 N1(C(CC(C=C)CC)=O)CCOC2(C1)CN(C(c1[nH]c(=N)sc1C(F)(F)F)=O)C2 Cc1ccc(NCCC(=O)NCC2C(C)CCCN2C(=O)CC2=CCCC2)c(Cl)n1 S(=O)(=O)(c1cccc(N2CCOC(C)(CCO)C2)n1)N1C(C)CCCC1 Cc1c[nH]cc1C(=O)NC1(C(=O)NCCc2ccns2)CC1(C)C C1(C)(NC(Cc2ccc(CCC)cc2)=O)CCCN(C(=O)Cc2ccccn2)C1 c1(CN(C(=O)COC2CCOCC2)CCNC(CCCOC)=O)ccccc1F c1(C(N(C)CC2CCCN2C(=O)CC(C)(C)O)=O)c2c(nn1C)CCS(=O)(=O)C2 c1(C(=O)NC(CN(C(C(C)NC(C)(C)C)=O)C)C)cc(O)nn1C C1(CC(=O)N(C)CCN(C)C(c2ccn(C3CC3(F)F)n2)=O)COCCN1C c1(CC)cnc(O)c(NC(=O)NCC2(C)CCCCO2)c1 C1(C(=O)NCC2(NC(C3C(=C)C3)=O)CCOCC2)CCc2nc(C)ncc2C1 C(C(F)C(=O)NC1CC(N(C)C)C1)C(N(C(C1C(C(C)C)C1)=O)C)=O c1(-c2nnc(CC(=O)NON3CCOCC3)o2)ccc(Cl)cc1Cl C1(NC(C(c2ccc(O)cc2)C)=O)CC(C)CN(C(=O)CCC(N)=O)C1 CC1(C)CCC(CC(N2CC(NC(C3CC(=O)NC3(C)C)=O)C(O)C2)=O)CC1 CCC(O)C(CC)NC(c1cccc(-c2ccc(F)cc2)n1)=O N1(C(C(C)NC(c2cnn(C)c2N)=O)=O)CCSC2CCCC12 N1(C(c2c(C3(C)COC3)noc2)=O)CC(CNC(C2CC3CC3C2)=O)CC1(C)C N1(C(c2cc(C#C)cc(N)c2)=O)CC23CCCCC2(C1)CN(C(=O)C(C)OC)C3 C12(C(=O)NCCc3cccc(C(F)(F)F)c3)CC3CC(CC(C3)O1)C2 c1(C(C(=O)NCCCC(C)(C)NC(=O)C=CSC)OC)ccc(Br)cc1 C(=O)(C1c2c[nH]nc2CCC1C)N(CCCNC(c1n(CCC)ncc1)=O)CC Cc1cc(Cl)ccc1CC(=O)NC1CC2(C1)CC2NC(c1ccsc1C#N)=O C1(O)(CC(=O)N(C)CC2(CNC(C3(CF)CCC3)=O)CCCC2)CCCNC1 N1(C(C(C(=O)OCC)C2CC2)=O)CC(NC(C2(NC(N)=O)CC2)=O)C(C)(C)C1 N1(C(c2ccn(CC)c(=O)c2)=O)CC(C2CN(C(=O)C(C)Cc3ccco3)C2)C1 N1(C(COCCC=C)=O)CCN(C)C(C(=O)NC2(C)CCCC2(F)F)C1 C1(NC(=O)C(C2CCOCC2)O)CCN(C(=O)NC2CC2c2ccc(Cl)s2)CC1 C1(CCC)CN(C(c2cc(C(N)=O)cn2C)=O)CCN1C(=O)COCC1CC1 C1(CNC(=O)CC2CN3CCC2CC3)C(C2CC2)CCN1C(N1CCOC1=O)=O C1CCCCC(=O)NCc2cn1nn2.c1(C(C2CCOC2)C)cnn(C)c1 c1(C(N2CCC(NC(=O)NC)C2)C(=O)NC)nc(F)ccc1Br c1(C(=O)NC2CC(NC(C(CC)C#N)=O)C2)c(F)cccc1[N+](=O)[O-] O=C(CS(=O)C(F)(F)F)NC1CCC(CNC(c2ccc(C3CC3)nc2O)=O)C1 C=C(Cl)C(C)(C)C(=O)N1CC2CC(C1)C2NC(C12CC3CC1C2C3)=O C(=O)(CCC(=O)NN(C)C)NC(C(=O)NC(C(=O)NC)C)C1(O)CCC1 c1(C(N2CC(CCNC(=O)C(C)SC)(OC)C2)=O)ccc2c(c1)CCN2 Cc1nc(N(C(=O)C(=O)N(C)C(C2(O)CCC2)C)C)sc1-c1ccc(CO)s1.N(C)C CC(CC(N)=O)C(=O)N(C(C)(C)CC(=O)N1CC(O)C(F)C1)C O=C1OCCC2CN(S(=O)(=O)c3cccc(OC4CCCC4)c3)CC12 N1(C(=O)Nc2c(C(C)C)onc2)CCC(c2cn[nH]c2)CC1C C1(OC)CN(C(=O)NCc2cn(CCC(C)(C)C)nn2)C(C(=O)O)C1OC c1(C(=O)NC2C(CNC(c3ccc(C(F)F)cc3)=O)C2)cc(O)cc(F)c1 Cc1ccc(C(=O)NCC23CC2CN(C(=O)C=Cc2ccncc2C)C3)cc1C c1(C(N(C2CCN(C(=O)C(C)(C)O)C2)CC)=O)cc(F)c(OC)c(Cl)c1 N1(C(CNC(c2ncn(CC)n2)=O)=O)CCN(C(C2CC(=O)N(O)C2)=O)CC1 n1(CC)nc(C(N2CC(CNC(=O)C(C)CO)C2)=O)cc1C C(=O)(CC(C)(C)C(F)F)N1CCN(CCCNC(C2N(C)CCN(C)C2)=O)CC1 N1(C(C23CCC(C(N)=O)(C2)C3)=O)CCCCC(NC(C2CCCCO2)=O)C1 C1(NC(C(C)N(C)C(c2cc[nH]c(=N)n2)=O)=O)CCC(O)C(O)C1 C1(C(=O)NCC(=C)CCNC(=O)CC(C)n2cccn2)CC(=O)N(C(C)C)C1 C(=O)(CCCC(=O)OCCCF)NCC(c1ccccc1)N(C(=O)COC)C Cc1ncc(S(N)(=O)=O)cc1C(=O)N(C)CC1CN(C(C23CCC2C3)=O)CCO1 N1(C(COCCCCC)=O)CCC(CCCCNC(=O)CN(C)C(C)=O)CC1 N1(C(CCC(=O)N(C)C)=O)CCOC2(C1)CN(CC(=O)N(C)CC1CCOC1)C2 c1(C(C(=O)NC)N(CCN(C)C)C2CC2)ccc(CC(C)C)s1 Cc1n[nH]c(=NC2CC3CC(C2)N(C(c2cnc(C)n2C)=O)C3)s1 c1(CC)ccccc1C(N1CCC(CCNC(=O)CCc2cncn2C)CC1)=O c1(C(=O)NC2CC(NC(C3(CC=C)CC3)=O)CC2O)ccc2cnoc2c1 N1(C(c2c(C)nc(COCC)s2)=O)CCCCC(CNC(=O)C2=COCCO2)C1 C(C(C)(CO)NC(c1cc(Br)c[nH]1)=O)NC(C(c1cnccn1)C)=O CCC(COC)C(=O)NCC1CC(NC(C2(C)CCN(C)C2)=O)C1 C1(C(N2CC(C(=O)NC(c3ccsc3)C)C(C)C2)=O)CC(=O)NC(=O)C1 C1(C(C)(C)NC(c2cnn[nH]2)=O)CCN(C(=O)C(F)C2CCC2)C1 CCCC(C)C(=O)NC(C1(C(=O)N(C2CCCC2)CC)CC1)C C#CC1(C(=O)Nc2ccc(F)c(C)c2)CCN(C(=O)CN2CCC(C)C2)C1 N1(C(c2c(SCC)nccn2)=O)CC2(CCC2NC(C2CC(=O)N(OC)C2)=O)C1 c1(-c2nnc(N(C)CC3(N(CC(CBr)C4CCC4)C)CC3)o2)ccccc1Cl C1(C(=O)NC2(CC)CCN(C(CCC=C)=O)CC2)Cc2ccccc2C1C c1(C(N2CCN(C(CCc3ccc(C)nc3)=O)CC2)=O)ccc(F)c2occc12 N1(C(C2(NC(C(CCC)O)=O)CCCCC2)=O)CCCC2(C=CCO2)C1 Cc1coc(C(=O)N(C(C)CNC(c2cn(C(C)C)nn2)=O)C)c1C CC1CN(C(=O)COC(F)(F)C(F)(F)F)CCC1CNC(c1cc(Cl)no1)=O C(=O)(C(F)C(=O)NC1(C(N2CC(O)(c3nn[nH]n3)C2)=O)CCC1)OCC c1(-c2c(C(=O)NCc3ccc(OC)nn3)cccc2)c(-c2cccs2)cccc1F C1(C#N)(C(=O)NC2CC(C)N(C(=O)CSc3cccc[n+]3[O-])C2)CCOCC1 C1(NC(COCCC=C)=O)CCCCCC1NC(c1cc(O)cc(Br)c1)=O c1(C(=O)NC(C2CCOC2)CO)nc(Cl)sc1Cl C1(c2n(C(CC)(C)C)nnn2)(NCCOCC(C)C)COCC1CC1CC1 c1(CNC(C(C)NC(CC)(C)C)=O)cc(C(=O)NCC(C)(O)CN(C)C)on1 CCC(C(=O)NCCOC1CN(C(C2(CSC)CCC2)=O)C1)c1ccccc1 C1(CNC(=O)OC)C2CN(C(C3(c4ccccc4)CC3)=O)CC12.C1(C)(C)C(=O)N1 c1(C(C)C(=O)NC2CCCC2NC(c2cc[nH]c2)=O)ccccc1F Cc1c(NCCCCCC2CC2)ncnc1NC1CCSC(C)(C)C1 C12(C(=O)NCCNC(=O)NC)CC(CO1)N(C(C1CC3C(C1)C3(C)C)=O)C2 C1(OCC(=O)NC(C)Cn2cc(-c3cnn(CCF)c3)nn2)C#CCCCCC1 C(N=c1nc2sccc2c(NC2CC(C)n3ccnc32)[nH]1)c1cc(C)cc(Cl)c1 CC1NC(=O)OC12CN(C(=O)C(Cc1ccccc1Br)NC(=O)CSCCF)C2 Nc1cnnc(NNC(=O)NCC2CC3(C2)CC32CCC2)c1Cl c1(C(=O)NCCC(C)N(CCC)C)cc(CNC(C2CC2Cl)=O)on1 N1(C(Cc2c(C)cnn2C)=O)CC2(CC(NC(C3(N=[N+]=[N-])CC3)=O)CO2)C1 C1(N(CC(=O)N(c2ccccn2)CCO)CCO)CCCCCC1 C1(C(=O)OCC)CN(c2nnc(CC(C)(C)O)n2CC(C)C)C1(C)C Cc1cccc(C(=O)NCC2COCCN2C(=O)Cc2cc(F)cc(F)c2)c1Cl C1(C(=O)Nc2cnc(C)nc2)CC2(CCC2)CN1C(C1CCOC1(C)C)=O c1(C(N2CC(N(C(CCCC(C)C)=O)C)C(C)(C)C2)=O)cccc2c1CCCC2 c1(NC(C2CC(F)CN2C(c2cncs2)=O)=O)cccc(-n2cnnc2)c1 c1(NC(C2(C=C)CCC2)=O)ccc(NC(C2CC2C2CC2)=O)c(C)c1 CS(=O)(=O)C1CC(C(=O)NC2CC2CNC(c2cc(O)ccc2Cl)=O)C1 N1(C(c2cc(C)c(C)s2)C(=O)NCC(F)F)CCOC2(CCCCC2)C1 C1(C(=O)NC2(CCO)CCSC2)COc2cc(F)ccc2C1 C1(OCCCNC(c2ccc(CO)o2)=O)CCN(C(=O)CCC2CCCO2)CC1 C1(C(=O)NC(C)Cn2cnnc2)(CC)CCCN(C(=O)CC2C=NN(C)C2=O)C1 CC(CN=c1cccc(S(=O)(=O)NCCCN2CCCCC2)[nH]1)c1cnc[nH]1 c1(NCC(=O)NCC)nc(C)cc(=NCC(C)c2ccc(F)cc2)[nH]1 C(CC(C)(C)C)(c1n(CC=C)nnn1)(C1CC1)NC1C(C)CCC1C c1(C(=O)O)cccc2c1OCC2C(=O)N1CC(Cc2ccccc2)C1 C1(O)(CCNC(C(CCO)N(C)C)=O)CCCN(C(c2cscc2C#N)=O)C1 CC(=O)C(C)(C)CCC(=O)NC(C)Cn1cc(-c2ccc(C#N)nc2)nn1 C1(c2n(CCCSC)nnn2)(NC(c2cccc(Cl)c2Cl)C)CCCN(CC)C1 C=C=CCCC(=O)N1CCCC(CN2CCN(C(C3CCC3OCC)=O)CC2)C1 c1(C2(NCc3cn(C)nc3)CC2)ccc(F)cn1 O=S(=O)(c1ccc(Br)cc1N1CCC2CCC(C2)C1)NCC(Cl)(Cl)Cl C(CC1CC1)(C(=O)N(CCCN1CCCCC1)CC)NC(COC(CC)C)=O C1(C)(CNC(C2CCN(CC(C)C)C2)=O)CCCN1C(C1CCN1C)=O C1(C(=O)NCCOCCC(C)C)(NC(C2CCCSC2)=O)CC(F)(F)C1 C(=O)(C1Cc2ccccc21)N1CCCC(O)(CN(C(=O)CCOC2COC2)C)C1 C1(CNC(C(CC)(C)C)=O)CCN(C(C2(C)CC2C(F)(F)F)=O)CC1C c1(OC)ccc(NC(c2coc(C(C)NC(C3(F)CCCC3)=O)n2)=O)cn1 Cc1[nH]nc2cc(-c3ccn4ncc(C(=O)NC5CSC5)c4c3)ccc12 c1(CC)ncsc1C(=O)NC1CCCC1CNC(c1cc(C2(C)CC2)on1)=O N1(C(c2c(C)nc(CO)s2)=O)CCC(CO)C(NC(c2nnn(C)c2C)=O)C1 C1(CC(=O)NC(C(C)NC(=O)Cc2cn(C)nn2)(C)C)CCC(=O)NC1 C(=O)(C(C)(C)C(N)=O)N(CCCCCCNC(CN1C(C)CCC1)=O)C c1(C(C(=O)NC2CN(C(CC(C=C)C)=O)CC2C)(F)F)ccc([N+](=O)[O-])cc1 c1(CC(CNC(=O)NC2C3CCCCC23)CO)cc(F)c(F)c(F)c1 c1(OCC(C)C)ccccc1CN(c1cccc(N2CCC2=O)c1)C CCCCC(C)(F)C(=O)N1CCC(NC(C2CCC(C)(C)O2)=O)C(F)C1 C(CC(C)(c1nnnn1CCCOC)NCCCc1scnc1C)SC N1(Cc2c(C)c(Br)n(C)n2)CC2(CCCCC2)C1C(C)C C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(C2OCCN(C(CC(=O)OCC)=O)C2)C1 N1(C(CC(CC)(C)C)=O)C2CCC1CN(C(C13CCC1C3)=O)C2 n1(CCC(=O)NC2C(NC(C3C(CC)OCC3)=O)C2)c(C)cc(O)cc1=O N1(C(CCn2cc(CC3C(=O)NCCC3)nn2)=O)CCOC2(CCC2)CC1 CN1CCN(C(c2cc(C(F)(F)F)no2)=O)C(CNC(c2ccc(=O)oc2)=O)C1 c1(C(N2CCC(NC(CCC(=O)NC)=O)(COC)C2)=O)ccsc1S(C)(=O)=O c1(C(=O)NCC(C)CN(C)C(c2cnnn2C)=O)cnccc1N(C)C c1(N(C)C)nc2cc(NC(=O)CC3CS(=O)(=O)CCN3C)ccc2o1 C(=O)(C1Cc2ccc(F)cc21)NC1CCN(C(C(C)NC(N)=O)=O)C12CCCC2 c1(C(=O)NC2C(NC(C3(OC)CCSC3)=O)CCC2)ccc(C2CC2)cc1Cl c1(CC(N2CCCC(C)(NC(c3cnc(C)[nH]3)=O)C2)=O)cccc(S(C)(=O)=O)c1 c1(N(C)Cc2csc3ccccc23)[nH]c(=NC2CCCC(CO)C2)nc2sccc12 CCCC(C(=O)N1CCCC1C(C)NC(c1cnn(CC(F)F)n1)=O)NC(N)=O CP(C)(=O)C(O)C(=O)NCCN1CCC(NC(=O)CC2CC(F)(F)C2)CC1 c1(C(C)NC(=O)C(C)(F)c2ccccc2)ccc(Cl)cn1 c1(C(=O)NCC(CC)(CC)NC(C2CCCCCCC2)=O)cnc2[nH]cnc2c1 C1(C(=O)NCc2c(C(C)C)noc2)CN(C)CCN1C(C1C2CCC(F)(F)C12)=O c1(C(=O)NCC(C)(CNC(=O)COCc2ccncc2)OC)cccn(C)c1=O Cc1cc(C(N2CCCC(CNC(C3(C(F)F)CCC3)=O)CC2)=O)cc(F)c1 N1(C2CCCC(CC)C2)C(=O)C2Cc3ccc(F)cc3CN2C1=O c1(C(=O)NCCN(C)C(c2ccncc2C2CC2)=O)cccc(C(C)(F)F)n1 N1(C(C2N(CC)CC2)=O)CC2CC1(C(N1CCC(OCC3CC3)C1)=O)C2 c1(C(=O)NCCC2(CNC(CSSC)=O)CC2)cnc2c[nH]nc2c1 c1(C(N2C(C)CN(C(c3c(C)onc3)=O)C(C)C2)=O)cccc(P(C)(C)=O)c1 C1(CCC)(NC(=O)CC(C)(C)F)CCCN(C(c2ncccc2OC)=O)C1 N1(C(CC(=O)N(C)C)=O)CCC2(CNC(=O)C(F)C3CCOC3)CCCCC12 N1(C(C(C)(C)C23CC(C2)C3)=O)CC2CC2(c2cccc(Br)c2)C1 c1(C(N2CCC(O)(C(N3C(CCCC)CCC3)=O)C2)=O)ccc2sccc2c1O Cn1cc(NC(C2CC(C)(NC(=O)CSC(F)F)C2)=O)n(C)c1=O C1(C(=O)NCC2CCN2C(c2csc(Cl)n2)=O)CCc2ncnn2C1 C(CC(=O)NC1CC2CC(NC(=O)CCOC(=O)N(C)C)C1C2)(C(C)C)OC C1(C)(COC)CC(NC(=O)C(C)(C)C)CN1C(=O)Cc1ccc(C)nc1Cl N1(C(C(C)Cc2ccccc2F)=O)CC2CCC(C1)N2C(=O)CC1COC(=O)C1 N1(C(c2c(C)csn2)=O)CCCCCC1C(=O)N(C)Cc1ccncn1 C1(C(N2CC(N(C(C(CC)C#N)=O)C)C2)=O)CS(=O)(=O)CC12CC2 C1(CC(=O)N(CCCNC(c2ccccc2O)=O)CCO)CCCCC12CC2 Cc1ccc(Cl)c(N)c1C(N1CCC(NC(=O)C(C)N(C)C)C(F)C1)=O CC(C)C(C)(CNC(C1(CO)CC1)=O)NC(c1ccc(C(N2CCCC2)=O)o1)=O N1(C(c2c(C)nsc2C2CC2)=O)CCOC(C)(CNC(=O)OC(C)(C)C)C1 N1(C(c2c(SCC)cc(Cl)cc2)=O)CCC(N(C)C(c2ccon2)=O)C2(CC2)C1 C(=O)(C1=COCCC1)NCC1(COC)CCN(C(=O)C(C)(C)C2CCOC2)C1 CCCCCCC(C)CC(=O)NC1CCC(O)CN(C(c2ccoc2CC)=O)C1 Cc1nn(C)c(C)c1CC(N1CCSCC1CCNC(c1cncn1C)=O)=O c1(C(c2nnnn2C2COC2)NCC2(C)CCCC2(F)F)csc(S(N)(=O)=O)c1 S(=O)(=O)(c1cc(CO)ccc1N1CC2COCC2(CO)C1)N1CC=C(C)CC1 C(CC1CCCC1)(C(=O)NCCN(C(=O)CCc1cnc(C)s1)CC(C)O)OC c1(C(N(C2CCN(C(=O)C(Cl)=CCl)CC2)CC)=O)ccc2sccc2c1 N1(C(CS(CC)=O)=O)CCCC(C)(C(N2CCC(n3ccnc3)C2)=O)C1 Cc1cc(F)c(CC(N2CCC3CC3(NC(=O)CN(C)C3CC3)CC2)=O)cc1F Cc1ncc(C(=O)NCC(C)NC(=O)C(c2ccc(F)cc2F)C)cc1N Cc1ccc(C(=O)NCC(c2cccc(Cl)c2)NC(C2CC2(C)C)=O)nc1 C(C(C)(C(=O)NC1CCCCC1)NC(C1CCCO1)=O)SC Cc1ccc(C(=O)NCC2CC2NC(c2c[nH]nc2-c2cccnc2)=O)c(N)c1 C(=O)(C1Cc2c(Cl)cccc21)N1C(CNC(CCCCNC(C)=O)=O)CCCC1 C(=O)(CC(C)NC(c1cc(Br)cs1)c1nnnn1C1COC1)OCC.C1CO1 c1(CC)c(NCC2CCC2NC(=O)OC(C)(C)C)cccc1NS(C)(=O)=O N1(C(C(=O)NCCCOC)C)CCC2(CCCCN(C(c3ncccn3)=O)C2)C1 c1(CC)nc2ccc(Cl)cn2c1C(=O)NCCN(C(=O)C1=CC(C)(CC)C1)C c1(C(N2CCC(NC(CC3C(C)=NN(C)C3=O)=O)C2)=O)ccc(C)cc1[N+](=O)[O-] C=CCC(CNC(=O)C(CC)=CC)C(=O)NCC(C)(O)C(C)CC c1(COC(C)=O)ccc(C(N2CC3CC2C3C(=O)NC2CC2C)=O)cc1 CCC(=O)CCC(=O)NC(CC1CCC1)C(=O)NC1CN(C)CCC1O C1(NC(C(C2CCCC2)OC)=O)CN(C(=O)CCS(C)=O)CC1(C)C Cc1cc(C)c2onc(C(=O)NNC(=O)c3[nH]nnc3C)c2c1 N1(C(C(C(C)C)SCC)=O)CCC(NC(=O)C=CSCc2ccco2)C(CC)C1 c1(-c2scc(N(c3ccccc3)C(C)=O)n2)ccc(NC(COC)C)cc1 c1(C(N2CC(NC(c3c(CC)c[nH]c3)=O)C2)=O)cc(O)c2ccccc2c1 Cc1nccn1CCNC(=O)C(C1(C)CC1)NC(C1CCC(C)O1)=O CCC(CC)CCCNC(=O)C(C(C)(C)C)NC(c1ccccc1O)=O C1(CN(C(COCCOCC)=O)C)CCC(CC2(C(=O)NC)CC2)CC1 c1(OC)ccccc1C(=O)NCC(CO)NC(=O)CC1CCC1C c1(CC)c(C(=O)NC2CC(C(=O)OC(C)(C)C)C2(C)C)[nH]c(C)c1C(=O)OC N1(C(CC(CC=C)NC(c2nccs2)=O)=O)C2CCC1CC(CO)C2 c1(C(C(=O)NC2CCC2)N(CC)Cc2cnn(C)c2)cccc(NC(=O)NC)c1 Cc1ccc(C=CC(=O)NCCC2(CNC(=O)CCCC#N)CC2)s1 N1(C(COCC)=O)CCc2nc(C(=O)N(CCO)CCO)ccc2C1 N1(CC(=O)NCC(CN(C)C(c2cn(C3CC3)cn2)=O)(C)C)CCS(=O)(=O)CC1 C1(C(N2CCC(C)C(NC(C34CC(C3)C4)=O)C2)=O)C2CCC(C2)C1(C)C C#Cc1ccc(C(=O)NC2CN(C(C3CC(n4cnnc4)C3)=O)CC2OC)cc1 N1(C(C(C)Sc2ccc(Cl)cc2)=O)CCOCC(CNC(=O)C2=CCCS2)C1 C=C(C)C1CN(C(=O)C(C2(O)CN(C(c3cn(C)nc3C)=O)C2)F)CCO1 C1(NC(CNC(=O)NC)=O)CC(c2ccccc2)(NC(=O)CCCOC(C)C)C1 C=CC1(C(=O)N(C)CC2(COC)CCC2)CCN(C(=O)CC2CCCNC2=O)C1 C1(OC)CN(C(c2c(Br)noc2C2CC2)=O)CC1NC(c1ccoc1)=O CN1CC=C(C(=O)NC2CCC(CC(=O)NCC34CCC(CC3)O4)C2)C1 c1(-n2ncc(C(=O)NCC(CC)NC(=O)CC3CNC(=O)C3)n2)ccc(F)cc1 O=S(=O)(c1cc(Cl)cc(Cl)c1)N1CC2CN(Cc3cc(Br)ccc3Br)C2C1 c1(C(=O)NCCCCC2CN(C(CC)=O)C2)cnc(N(C)C)cn1 c1(C(=O)NC2CCN(CCNC(C(C)CC(N)=O)=O)CC2)ccc(F)c(Cl)c1N N1(C(C2N(C(=O)OC(C)(C)C)CC3C2C3(C)C)=O)CCc2ccc(C#N)cc2C1 C(=O)(C(C)(CO)OC)NC1C(C(=O)NCCSCCC=C)CC1 CCS(=O)CC(=O)NCC12CC(CN1C(c1cccc(NC(C)=O)n1)=O)C2 c1(OC)cc(C)ccc1CNC1CCC(C(=O)NC(c2ccc(Cl)cc2)C)OC1 N1(C(c2nn(CC)c(C)c2)=O)CCC(CNC(c2cc(C)c(C)o2)=O)C12CC2 c1(C(=O)NC(CC)CNC(=O)CCc2csc(=N)[nH]2)cn2ccsc2n1 CN1CC(O)CC1NC(C1(C(=O)NCC(Cc2cccc(Cl)c2)C(N)=O)CC1)=O C(c1ccccc1Cl)=C(C(=O)NC1CCN(C(C2(CC)CCOCC2)=O)CC1)C C1(C)(NC(CCC2CCC(C)O2)=O)CCCN(c2ccncn2)C1 c1(C(N2CC(C)(NC(=O)COCc3nc[nH]n3)C2)=O)cncc(N)n1 c1(C(=O)NCC2C(NC(CC=C)=O)COC2)c(-n2cccc2)sc2c1CCC2 C(CC(C(=O)NC(CC1CC1)CC(=O)NCCCC1(C)CC1)OC)OC N#Cc1cc2cc(C(=O)NCCNC(c3cnn[nH]3)=O)[nH]c2cn1 c1(OC)cccc(C2(n3cc(C4CC(C(=O)NCC5CC5(Br)Br)C4)nn3)CC2)c1 n1(C(C(=O)Nc2ccc(C)c(Br)c2)C)cnc2ccccc12 C1(CC(=O)N(C)CC2(N(C)C)CC2)N(C(c2cccs2)=O)CCC1(C)C N1(C(=O)Cc2nc[nH]n2)CCCC2C1CCCN2C(c1cc2occc2[nH]1)=O c1(CC)ccc(C(N2CCC(F)(CNC(C3CCCSC3C)=O)CC2)=O)c(F)c1 Cc1ccc(CC(=O)NC2(CCNC(=O)CN(C3CCCC3)C)CCC2)cn1 C1(NC(=O)COC(F)(F)F)C2CCC1CN(C(C1CC3CCC1NC3=O)=O)C2 C1(NC(c2cccc(OC)c2)=O)C2CC3C1C3C2C(=O)NOCC(N)=O c1(SC)ccc(N)cc1C(N1CC2CC(NC(C3(C)CCC(=O)NC3)=O)C1C2)=O C1(C)(C(N(C)CC2CCN(C)C2)=O)C=CCN1C(=O)Cc1cccnc1O C1(C(N(CCCF)C)=O)(NC(=O)C(=O)NCC2CC2)CCC(C)(C)C1 c1(C(=O)OC)ccc(C)nc1NC(C)(CNC(C1CCCN1C1CC1)=O)CC C1(C(N2C(CCNC(=O)COc3ccccc3)CCCC2)=O)CC2CC1C1CC21 N1(C(C(C=C)O)=O)CCOCC12COCCN(C(C1Cc3cccnc3C1)=O)C2 CC(C)CCCCC(=O)N(C1CCCOC1c1ccccc1)CC.C(=O)(CC(C)C(F)F)N c1(C(=O)NC2(CNC(C3CC(C#C)(O)C3)=O)CCOCC2)nccc(Cl)c1C N1(C(c2ccc(CNC(C(C(C)C)N(C)C)=O)s2)=O)CCCC2(CCC2)C1 N1(C(C(COC)COC)=O)CC2(CCOCC2)CC1CNC(=O)CCCC1CC1 c1(CC(=O)NC(CCN(C(C(=O)NCCOC)=O)C)C)ccc(C)cc1Br C=C(CC)CN=c1[nH]c(N2CCc3cccc(SC)c3C2)nc2cc(C)ccc12 C1(CC(c2n(CCCC)nnn2)(C)NCC(C)CCCCO)CCS(=O)(=O)N1C N1(C(C2OCCN(C)C2)=O)CC2CC(F)(F)CCC2(N)C1 CCC(CSC)(c1nnnn1C1CCOC1)NCC=Cc1ccco1 c1(C(=O)NCC(C)N(C(C(n2ncc(C)c2)C)=O)C)noc2c1CC(C)(C)CC2 c1(C(=O)NC(COCC)CO)c(CNC(=O)C=CC2CC2)cnn1C n1(CCC)cc(Cl)c(C(N2CC=CC(NC(=O)CCC(C)SC)C2)=O)n1 c1(C(N2CCCC(NC(C=C3CCC(C)C3)=O)C2)=O)ccc2c(c1)COC2(C)C C1(C)(NC(c2cc(C)sc2)=O)CCN(C(c2cc(C)c(-c3ccccc3)s2)=O)C1 C(=O)(C1=CCC(NC(c2c(Cl)cnn2C)=O)C1)NC(CC)C1CC1 N1(C(c2cc(OC)no2)=O)CCCC(CCNC(C2(O)CCSCC2)=O)C1 C1(NC(c2cccc(C3CC3)c2)=O)CCCCC1NC(C1(F)CCOC1)=O c1(-c2n(CC)c3c(n2)cccc3)cc(C2=CCNCC2)c2[nH]ncc2c1 CC1CCC(CC(=O)NC2CN(C(c3cnn(CC4CC4)c3)=O)CC2C)CC1C C1(O)(C(C)NC(C2C(C)C2C)=O)CCN(C(C2CCCN2C)=O)CC1 C1(C(=O)NC2(C)CN(C(=O)CC3(C)OCCO3)C2)CC2CCC1C2 C=CC1CN(C(c2cc(F)ccc2N)=O)CC1NC(=O)CCc1cn(C)nn1 c1(C(=O)NCC2CCCCN2C(=O)C=C2CCC2)cc2ncccc2[nH]1 c1(CN2CCN(Cc3cc(C(=O)O)c(O)cc3)C3C2C3)c[nH]c2cccc(O)c12 c1(C(C(=O)NCCCC2CC2)N(C(C)C)CC)cc(Br)ccc1F c1(CCC(N2CCC(C(C)NC(C3(CC#N)COC3)=O)C2)=O)ccc(F)cc1 C=CCC(CNC(C1(CC(=O)OC)CC1)=O)NC(=O)CC(C)n1cccn1 C1(CC(N2CC(C(C)NC(C3CC34CCCC4)=O)C2)=O)NC(=O)NC1=O C12CCC(C1)CCC(=O)N2.C(CCN=[N+]=[N-])NC(C1(CCOC)CC1)=O C(CCC(O)C(=O)NCc1ccc(CO)cc1)NC(C1(C)CCN(C)C1)=O C(=O)(CC(C)(C)C(F)F)N1C2CC(NC(c3c(C)noc3C(C)C)=O)C1CC2 C=CC1CN(C(=O)C(C)Cc2ccc(O)cc2)CC1NC(c1cnc(Cl)s1)=O c1(C(N2C(C)CN(C(C3COCCO3)=O)CC2)=O)ccc2nc(CO)[nH]c2c1 C1(NC(c2n(CC)ncc2)=O)CN(C(=O)Cc2nc(C)sc2C)CC(C)(C)C1 N1(C(COC)=O)CCc2ccccc2C(NC(=O)C=Cc2cccc(Cl)c2Cl)C1 c1(C(=O)NC23CCN(C(c4c(CC)cco4)=O)CC2C3)ccc2nc(O)oc2c1 C12(C(=O)NCC3C(C(=O)OC)C3)CCN(C(C3CCC3C(C)(C)C)=O)CCC1C2 c1(OCCC(N2CCC(C)(NC(CC3ON=C(C)C3)=O)C2)=O)cc(C)cc(C)c1 c1(-c2ccc(CO)cc2)csc(=Nc2cccc(Cl)n2)n1Cc1ccccc1Br CCC(CC1CCCC1)C(=O)N(CCCNC(C1CC1c1cnn(C)c1)=O)C c1(C(=O)NCC(C)CN(C)C(C2C(C)C2(F)F)=O)cccc2nc(O)n(C)c12 C1(NC(CNC=O)=O)CC(CO)C12CCC2.C12CC(C1)OCC(=O)N2 C1(NC(CC2CC(C)N(C(c3cnsc3)=O)C2)=O)CCC([N+](=O)[O-])CC1 Cc1cn2c(C(=O)NCC(C)NC(C3(C#N)CCOCC3)=O)c(Cl)nc2s1 C1(C(=O)NCCC2(NC(=O)CC3CCOCC3)CC2)CCCCC(F)(F)C1 C1(NC(CN(C(C)C)C)=O)CC2CC(NC(c3nc(Cl)c(=O)[nH]c3N)=O)CC2C1 C1(N(C(C(CC)F)=O)CCO)CCN(C(=O)Cc2ccsc2C)CC1 C1(C(=O)NCC2(COC)CCCN2C(=O)COCCC(C)C)CCCS(=O)(=O)N1 c1(C(N(CCC(C)NC(c2ccc([N+](=O)[O-])[nH]2)=O)C)=O)c[nH]nc1S(N)(=O)=O Cc1cc(NC(=O)C(C)C2(O)CCC2)ccc1NC(c1oc(C(C)C)nc1C)=O N1(C(C2CCCN(C(C3CN(C)C(=O)CC3)=O)C2)=O)CCOCC(F)(F)C1 C(=O)(C(CC(C)C1CCOCC1)N1CCN(C2CCSC2)CC1)NCCCC CCC(COC)C(=O)NCCC1CN(C(=O)Nc2cn[nH]c2)C1 NC1CCCN(C(=O)NCCC(=O)NCC2CCCCC2)C1 C1(n2c(-c3cnc(-c4ccccc4)[nH]3)nc(C(C)C3CC3)n2)CCC(F)(F)CC1 c1(OCC)c(C(=O)NCC2CCN2C(c2c(F)ccnc2F)=O)cccc1F Cc1sncc1C(=O)N(C1CN(Cc2cnc(Br)s2)C1)C C1(NC(C(C)O)=O)C=CCN(C(=O)CNC(c2cccc(Cl)c2)=O)C1 N1(C(CC(C)OC)=O)CCN(C(=O)C(=Cc2cccn2C)F)CC1C1CCCC1 N1(C(COC2(C)CCC2)=O)CC(NC(C2CC2c2ccco2)=O)C(O)C1 Cc1cc(C(N2CCN(C3CN(C(=O)C4=COCCC4)C3)CC2)=O)cc(N)c1Cl CC1(C)CCOC(C(=O)NCC2(C)CCCC2NC(C2CCS2(=O)=O)=O)C1 C1(NC(c2cc3occc3s2)=O)CCN(C(=O)CC2CCOC2)CC1F N1(C(c2c(C)ccc(O)c2)=O)CCCC2CN(C(=O)Cn3cnnc3O)CCC12 C=Cc1ccc(C(N2CC(OC)C(NC(=O)Cn3ncccc3=O)C2)=O)cc1 C1(C(=O)NC(CN(C)C(c2cnn(CC(F)(F)F)n2)=O)(C)C)CCCCS1(=O)=O c1(N2CC(C)N(Cc3cccn3C)CC2)ncnc2c1CCC2 C1(C(=O)NC2CCN(C)C2=O)CC(F)(F)CN1C(c1cccc(CO)n1)=O C(=O)(C1=CCCC1C)NC1C2CN(C(c3sc(CCC)c(CC)c3)=O)C1C2 N1(C(C(C)N(C(C2C(=C)CC2)=O)C)=O)CCCN(C(=O)NCC)CC1 C(=O)(C1CCCc2nncn21)N(CCC(C(C)C)NC(=O)C=CCF)C C12(CNC(c3ccc[nH]3)=O)CC(CN1C(=O)CSCC1CCCCO1)C2 S(=O)(=O)(c1cc(C(N2CC3CC2CCC3O)=O)n(C)c1)NC(C)C C(=O)(C1SCc2cccnc21)NC(C)CNC(c1cc(CO)ccc1Cl)=O C1(CC=C)(C(=O)NCCN(C(C)C)C(C)C)CCCN1C(C1C=CCC1)=O C1(CNC(c2n(CC)cc(Cl)c2)=O)CCCC2CN(C(=O)C#CC(C)(C)O)CC12 C#Cc1ccc(C(=O)NC2CCCC(NC(C3CC34CC4)=O)C2)c(C)c1 c1(CNC(Cc2c(OC)cccc2F)=O)ccc2c(c1Cl)OCCO2 O=C(CCCCCCNC(c1cnco1)=O)NCCC1(CO)CCC1 CCC(C)CCCC(=O)NC1COCC1NC(c1cc(C)c(C)s1)=O C12(CC(=O)NCC(C)(C)Cn3cc(CO)nn3)COC(CF)(C1)C2 c1(C(=O)NCCNC(=O)C2=NOCC2)ccc2c(=O)c3ccccc3sc2c1 C1(C(=O)NCC(CN(C(C(COC)C)=O)C)(C)C)Cc2c(F)cccc2O1 N1(N(C(=O)Cc2cccc(Cl)c2)C)CCN(C(=O)C(CO)NC(N)=O)CC1 c1(C(N(CCOC)Cc2ccccc2C)=O)coc2c1CNC2 c1(OCC)cc(C=CC(=O)NC2CCCCC2NC(=O)CC2CC2)ccc1O C(CC(C(C)C)N(C)C)NC(C1C(NC(C2CC(SC)C2)=O)CCC1)=O C1(CNC(C(CCC)(C)O)=O)CC2CCC(C1)N2C(C1CCCCC1O)=O Cc1cccc(CCNC(c2n[nH]cc2CNC(C2CC2(F)F)=O)=O)n1 c1(NC)ccc(NC(=O)C(=O)N(C)Cc2cnn(C)c2C)cc1F N1(C(c2n(C(CC)C)ncc2)=O)CCC(O)(CN(C(=O)CC23CC(C2)C3)C)CC1 CCS(=O)(=O)c1cc(F)ccc1NC(N1CCCC(CN2CCN(C)CC2)C1)=O N1(C(C2OCCC(C)(C)C2)=O)CC2CC(C1)CN(C(=O)C1=CCCCCC1)C2 C(=O)(CC1=CCN(C(=O)C(CCC)OCC)CC1)N1CC(C#C)OCC1 C(=O)(CS(=O)(=O)C(C)(C)C)NCC1N(C(C(C=C=C)C)=O)CC(F)(F)C1 N1(C(C(C)N(C(=O)CCCCC2CC2)C)=O)CCCC12CCCOC2 C1(C(N(C(C)C(=O)N(CC(O)C2CCC2)C)C2CC2)=O)CCCCNC1=O N1(C(C(c2ccoc2)NC(C=CCN(C)CC)=O)=O)CCC(SC)C1 C(C(C)(C)C(=O)NCCC1CCCCN1C(=O)CC1(C#N)CC1)OC c1(OCCCC(=O)NCc2c(C)cco2)cccc(F)c1 C(=O)(C(C)(C)CC#N)N1CCC(OCCNC(CC(C)(C2CCC2)OC)=O)C1 c1(C(=O)NC(C2CCOC2)CNC(c2cnc(CC)o2)=O)cnc(OC)c(F)c1 C1(C(=O)NC(c2ccc(Br)c(Cl)c2)C)NC(=O)C2CCC12 CC1(C)CN(C(C2C3COCC23)=O)CCC1NC(=O)C=Cc1cncnc1O Nc1c(C(=O)NCC2CCCN2C(=O)Cc2ccsn2)cc(F)cc1[N+](=O)[O-] Cc1ccc(Cl)c(C(=O)NCC2COCC2NC(c2cc(C3CC3)nn2C)=O)c1 Nc1c(Cl)c(NC(=O)CSC2NC(=S)N(c3cccc(Cl)c3)C2=O)nc(F)c1Cl N1(C(C2CCC(CC)O2)=O)CCC(C(=O)NCC2CN(C(C)C)C2)CC1(C)C C1(C)(NC(CCc2ccc(C)nc2)=O)CCCN(C(C2(C)C=CCC2)=O)C1 c1(C(=O)NCCN(C(C2(C)CCCS2)=O)C2CC2)cccc(OCC(F)F)c1 N1(C(C2(C)CCC2)=O)CCC(C2(NC(c3ccn4[nH]c(=N)nc4c3)=O)CC2)CC1 C1(N(c2cccc(F)c2)C(=O)CC2CC2)CC2CCC1N2C(C1CCC=CCC1)=O CC1(F)CN(C(C2CCCCC2)=O)CCN(C(C2CCC3(CCC3)O2)=O)C1 CCC(CNC(c1cc(C2CC2)no1)=O)(CC)C(=O)N1CCC(C)(C)CC1 Cc1cc(N)c(C(=O)NCCc2ocnc2CNC(=O)CCC2CC2)cc1C C1(C)(CNC(C2CN(CC(C)C)C2)=O)CN(C(C23CC(F)C2C3)=O)CCO1 c1(C(N2CC(NC(C3(C)C=CCC3)=O)C(O)C2)=O)cc2n(n1)CCCCC2=O C1(C(=O)NC(C)Cc2ccncc2)CC=CCN1C(c1scnc1Cl)=O N1(c2c(S(=O)(=O)N3C(CCC=C)CCC3)cccn2)CCc2cc(Br)ccc2C1 c1(CNC(C(C2CC2)OCC)=O)cccc2c1CCN(C(c1sccc1F)=O)C2 C1(O)(C(C)NC(C(C)OCCCC)=O)CCN(C(=O)C(C)=C2CCC2)CC1 c1(CN(C(C)C)CC2(C)CC2)cn(CCCO)nn1 N1(CCC)C(=O)CCC1C(=O)NCC1CCCN1C(c1cccnc1C)=O N1(C(C2C(C)(C(C)C)C2)=O)CCCC1CN(C)C(c1sccc1F)=O c1(SC)cc(C(=O)N(CCCCN(C)C(c2[nH]cnc2C#N)=O)C)oc1C C(=O)(C(C)CC(C)(C)C)NCCC1N(C(c2sc(C)c(O)n2)=O)CCCC1 c1(C(N2C(C)CC(NC(c3cccc(OC)c3)=O)C2)=O)cnccc1C#N CC1CCN(C(=O)CC2CCN(C(C3COC4CNCC4C3)=O)C2)CCC1O C1(C)(C(=O)NC(C)C(=O)NO)CC(O)CN1C(=O)CC1CC2CCC1O2 c1(NC(CSCC(=O)NCC(C)NC(C2CCC(C)(C)O2)=O)=O)ccc(F)cc1 c1(OC)ccnc(F)c1C(=O)NCC1CC(NC(C2CC(C)OC2=O)=O)C1 C(CC(=O)NCC(=O)N(C(C)CF)C(C)C)NC(C)=O c1(C(C)C)ccc(C(N2CC(NC(C3(C4CCCO4)CC3)=O)C(C)C2)=O)c(O)n1 C(CC(CNC(c1snnc1C(C)C)=O)NC(=O)CCc1cscn1)OC CC1CCC2(CO1)CN(C(C1(CNC(=O)CC3CCCC3)CC=CC1)=O)C2 N1(C(c2ccc(C3CC3)cc2)C(=O)NC(CC)(C)C)CCC2(CCN(C)C2=O)C1 c1(C(N2CC3C(CN(C(C(CC=C)CC)=O)C)C3C2)=O)c(Cl)ccc(OC)c1N Cc1ccc(C(C)(C)CC(=O)NCCC(C(=O)O)c2ccc(O)cc2)cc1 N1(C(C2(C)N(C(CN3C(C)CCC3)=O)CCC2)=O)CCc2sccc2C1 c1(C(=O)NCC2CCN(C(c3ccc(OC)s3)=O)C2)cc2c(Cl)cncc2s1 Cc1cc(C(=O)N(C2CCC(NC(=O)C(C)(F)F)C2)C)c(C)n1NC(N)=O c1(C(=O)NCC2C3CCCC2N(c2nnc(C(N)=O)s2)C3)cnc2ccnn2c1 C1(NC(C2CC(C(C)C)C2)=O)COCC1NC(c1cc(-c2ccccc2)[nH]n1)=O c1(C(=O)NC2CCCN(C(C(CC)CC3CCCC3)=O)CC2)ccccc1S(C)=O C1(NC(Cc2c(CC)cccc2)=O)CN(C(=O)CCCC(C)=O)CCC1C Cc1ncc(Br)cc1NC(C1CC1NC(c1ccc(CCC(F)F)o1)=O)=O C(=O)(CC(C)CNC(=O)CC1CCCN1C)NC(Cn1ncc(C)c1)C c1(CC)nc(C)[nH]c1C(N1CCC(C)(NC(=O)C(=O)NCC(F)F)C1)=O Cc1cncc(C(=O)NCC2CC2CNC(c2cn(CC(F)(F)F)nc2C)=O)c1 c1(C(=O)NC23CC(NC(CC4(NC(C)=O)CC4)=O)(C2)C3)nnn2c1CCCC2 c1(C(=O)NCC(C)(C)OCC(=O)NCC2(F)CC=CCC2)cccc2occc12 CC(C(O)C(F)F)NC(=O)CCOC1CN(C(C2(C)COC(=O)N2)=O)C1 C1(N(C(C(C)NC(=O)NC)=O)C)CCN(C(=O)COC)CC1 CCCC(CCCNC(c1cccc(CC)n1)=O)NC(c1cnc(C)c(N)c1)=O CC1(C(=O)NC2CCC2N2CCCC2)CCN(C(=O)C(CO)N(C)C)CC1 c1(-n2cc(C(=O)NCC(=O)OCC)nn2)cccc(OCc2ccccc2C)c1 C1(F)(COC)CCN(C(C2(c3cn(C(C=C)C(=O)OCC)nn3)CCC2)=O)C1 Nc1c(Cl)cc(C(=O)NCC2CCN2C(=O)CSC2CCCCO2)cc1Cl C(=O)(CC1NC(=O)c2ccccc21)N1CC(CNC(c2cc(F)c[nH]2)=O)C1 C1(F)(CNC(CSCC(C)C)=O)CCCN(C(=O)C(F)n2ccnc2)C1 c1(C(C)C(=O)NC(C)CCNC(=O)CC2C=CCCC2)ccccc1F c1(C2(C(N3CC(NC(C4(C)CC=CCC4)=O)C3)=O)CC2)ccc(F)c(F)c1 Cc1[nH]c(C#N)cc1C(=O)NC1CCCC1CN(C(=O)Cc1ccco1)C CCC(C)C(C(=O)N(CC(O)CO)C)N(C)C(c1cnn(C)n1)=O C(C(CC(C)C)C(=O)N1CCOC(C(C)C)C1)NC(c1cccc(C)c1N)=O c1(C(=O)NC2CN(C(C3CCC(CC)O3)=O)CC23CC3)c(F)cc(Cl)cc1F CC1OCCC1CC(=O)NCC(C(=O)N(C)CCC1CCCN1C)N(C)C c1(C2(CC(=O)NCC3CCC3NC(=O)CCC=CBr)CC2)ccc(F)cc1 N1(Cc2cnc(OC)nc2)CC2CCN(c3ncnn4cccc34)C2C1 N1(C(c2c(CC)[nH]cc2)=O)CC(C(=O)NC2CC(C)CC(C)(C)C2)C(C2CC2)C1 CCCCC(CNC(=O)CCNC(c1cccs1)=O)NC(c1cc(Cl)cnn1)=O c1(C(=O)NC2CCN(C(CC(C)(F)F)=O)C2)cnc2ccc(Cl)cn2c1=O CC(CC(F)F)C(=O)N1CC(C(=O)NCCNC(c2ccc(SC(F)(F)F)o2)=O)C1 C1(C(=O)NC(CNC(COc2c(C)occc2=O)=O)(C)C)CCc2nccn2C1 c1(CCC(=O)NCCN(CCC)C(c2cnc(O)n2CC)=O)cn(C)nc1C Cn1nc2cccc(C(=O)NC34CC(NC(c5ccc(=N)[nH]n5)=O)(C3)C4)c2n1 C1(COC)(CNC(=O)C=CC(N)=O)CCCN1C(=O)CCc1cnn(C)n1 c1(OC)cc(=NC(=O)C2(CNC(c3cc(O)ncc3F)=O)CC23CCC3)[nH]n1C c1(C(=O)NCC#CCNC(=O)C=CC2CCOCC2)c(Cl)ccc2c1OCO2 c1(-c2cn(C3C(NC(C4C5CCCC45)=O)CCC3)nn2)cccc(F)c1F N1(C(c2c(OC)cccc2)=O)CCC(N=c2[nH]nco2)(CO)CC1 C(C(=O)NCCOCC(N)=O)(C(C)C)SC.C12(CCCCO1)C(=O)NC2 CC1(CC(=O)NC2CC2CNC(=O)Cc2cnns2)CCOCC1 CC1(C)CCOC1C(=O)NC1CCCC1n1cc(CS(C)(=O)=O)nn1 Cc1nn2cc(NC(C3CCC(C)N(C4CCCCC4)C3)=O)nc2s1 C(=O)(C(C)(C)CC1CC1)NC1CCC(CCC(=O)N(CCN(C)C)C)C1 c1(CC2C(=O)O2)ccc(C)c(Cl)c1.C1(=O)CCCO1.C(CCC)OCC=C.C(C)(=O)O C1(C2CCC2)(C(=O)NCC2(O)CN(C(CSCC(C)C)=O)C2)CC1(F)F Cc1c[nH]nc1CNC(=O)C(F)C1CC(NC(C2CS(=O)C2)=O)C1 Cc1cc(C2(NC(C34CC3CN(Cc3cc(Cl)ccc3F)C4)=O)CC2)cc(C)c1 C(=O)(CC(C)(C)C(F)F)NCC1N(C(C(C(C)C)n2ccc(C)c2)=O)CC1 C1(CC)CCC(C)CN1C(C12CC1CN(C(c1ccnnc1)=O)C2)=O CCN=c1[nH]c(C(N2CCC(NC(=O)C=CC3CCOCC3)C2)=O)cs1 c1(C(=O)NC2CC(C)CN(C(c3c[nH]nc3C(F)F)=O)C2)cc2cnccc2[nH]1 c1(OC(C)C(=O)NCC2CCN2C(=O)Cc2cn(C)nc2Cl)ccc(F)cc1 c1(C(N(C2CCC(NC(=O)CCN3CCCC3=O)C2)C)=O)cnc2[nH]ccc2n1 c1(C(N(CCC)CCNC(C2CC2CC(C)(C)C)=O)=O)cc2sccc2s1 CC1OC2(C(=O)NCc3ccc(CNC(C4CCCCO4)=O)cc3)CCC1CC2 CC(C)CC(CNC(C1(C)CC2C=CC1C2)=O)C(=O)NC1CCCCCC1F c1(NC(c2ccccc2Cl)C)[nH]c(=NCC(C)CN2CCOCC2)nc2sccc12 N1(CC(=O)NC2CC(NC(C3(S(C)(=O)=O)CC3)=O)CC2O)CCS(=O)(=O)CC1 c1(OC)ncc(C(N2CC=CC(NC(c3ccc(C(C)(C)C)s3)=O)C2)=O)cc1C CC(CCC(=O)NC(c1ccc(N(C)C)cc1)CN(C)C)c1ccc(Br)cc1 c1(N(C)Cc2ccc(C)o2)nc(=NC2CSC(C)C2)[nH]c2c1CCC2 C1(NC(=O)CC2CC2)CCC(C(=O)Nc2c[nH]nc2C(N)=O)OC1 N1(C(c2c(SC)nccn2)=O)CCC(C)(C)C(CNC(c2ccccc2)=O)C1 C1(NC(c2cc(C)ns2)=O)C=CCC(C(=O)NC(c2cncnc2)C)C1 C1(C(C)NC(C2(CC#C)CCC2)=O)CCN(C(=O)CO)CC1 C1(N(C(c2c(Br)cnn2C)=O)CC)CCCN(C(=O)CS(C)(=O)=O)CC1 CC(C)CS(=O)(=O)NC(c1cc(CF)on1)=O Cc1cncc(-c2cn(CC3CCCN(C(C4CCC4)=O)C3)nn2)c1 C1(NC(CN2CC(CC)C2)=O)CCN(C(c2ccoc2C(C)C)=O)C(C)C1 CC1C(NC(c2ccc(-c3coc(O)n3)cc2)=O)CCN1C(C1C=CCC1)=O C1(=CC(=O)NC2CN(C(C(CC)(C)O)=O)CC2C(F)F)C2CC3CC(C2)CC1C3 C(=O)(C#Cc1ccccc1)N1CC(NC(=O)Cc2cccnc2)C(F)(F)C1 C1(CNC(=O)C=Cc2cn[nH]c2)CCCCN1C(=O)Cc1csc(Br)c1 N1(C(C(CNC(c2cnc(OC)s2)=O)C)=O)CCCC2(C=CCO2)C1 c1(C(N2CCCC(C)(C(F)(F)F)C2)C(=O)NC)ccc(F)c(CO)c1 C1(CCC)CN(C(c2c(SC)cnn2C)=O)CCN1C(=O)CC1C=CCCC1 CC1(C)CCc2onc(C(=O)NCC(O)CNC(=O)C(F)CC3CC3)c2C1 c1(C(=O)NCCOCCNC(C(CC)C#N)=O)c[nH]c2nccc(Br)c12 c1(C(=O)NCC(CC)NC(=O)CC2CC2C2CC2)ccc(-n2cnnn2)cc1 C1(CNC(CCN(C)CC)=O)C2CN(C(c3sc(-c4ncc[nH]4)nc3C)=O)CC12 S(=O)(=O)(c1csc(C(=O)NCC2CCN2C(c2ccc(F)cc2N)=O)c1)NC C(=O)(C1CCCc2ccccc21)NCC(c1ccc(F)cc1)NC(=O)C=CBr N1(OC(c2c(SCCCC)cnc3ccccc32)=O)CCC2(CC1)CCS2(=O)=O c1(OCC)ccc(CCCC(=O)NCCCNC(c2ocnc2C2CC2)=O)cc1 c1(CNCC2C3CCC(F)(F)C32)cnc2cc[nH]c2c1 N1(C(c2ccncc2O)=O)CC(C2CN(C(C3CC3C3CCC3)=O)C2)C1 N1(C(CC(C)F)=O)CCC(C)(NC(=O)COCC(C)(C)C)C1 N1(C(c2cc(Cl)ccn2)=O)CC2(C1)CN(C(C13CCC(F)(CC1)CC3)=O)CCO2 N1(C(CCc2ccc(C)nc2)=O)CC2CCC2(CNC(=O)C(F)=C2CCC2)C1 c1(C2(C(N(CCOCCN(C(C3C=C(C)CS3)=O)C)C)=O)CC2)cccc(Cl)c1 c1(C(N2CCC(CNC(=O)C(F)C(F)(F)F)C2)=O)nnn2c1CCCCC2 c1(C(=O)NC(CNC(c2n(CC=C)ccn2)=O)C)ccc2c(c1)COCCN2 Cn1cnc(C=C(F)C(N2CC(C(N)=O)(CNC(C3CC4CCC3O4)=O)C2)=O)c1 CC(C)CCC(=O)N1CC(CN(C)C(c2ccnc(N(C)C)c2)=O)C1 CCC(C)(F)C(=O)N1CCC(F)(CNC(c2cnn(C(F)F)c2)=O)C1 c1(C(N2CCC(CCNC(c3cc(OC)no3)=O)C2)=O)nnn(C)c1C(F)(F)F C1(Nc2nc(C)nc(SC(C)C)c2)C(C)CN(C(=O)CN2CCCC2)CC1C c1(C(=O)NC2CC(CCNC(C(C)SCC)=O)C2)cnn(CC)c1 CC1CCN(C(c2csc(Cl)c2)=O)CC1NC(C1(C(F)F)CCCC1)=O c1(C(=O)NCC(C(N2CC3(C(C(=O)OC)C3)C2)=O)N(C)C)cc(C#N)cn1C C1(CNC(C(N)=O)=O)COC(CNC(c2cn(Cc3ccccc3)nn2)=O)C1 CCCCC(CC)(c1nnnn1CCOCC)NCC1(F)COC1 c1(CNC(C2(C)CCCS2)=O)nnc2n1CCN(C(=O)C(c1ccccc1)=O)C2 N1(C(CC2(C=C)CN(C(c3cnn(C4CC4)c3)=O)C2)=O)CC(C)(C)C12CCC2 C(C(N=c1nc(-c2ccccc2)[nH]s1)C1CC1)NC(c1ccn2ccnc2c1)=O c1(CN(CCNC(=O)NC2CCCN2C)CC)ccccc1C C1(C)(C(=O)NCCC2CC(NC(C3N(CC)CC3)=O)C2)CCN(C)C1 Cc1c(Br)noc1C(=O)NCC1CCCN1C(C1CC1c1ccccn1)=O c1(-c2nc(C(C)SCC)nn2CC2CCCOC2)cnn2cc(F)cc(F)c12 C#CC1(C(N2CC(CCO)(CC)C2)=O)CN(C(=O)C(C)CO)C1 O=C1COCCN1C1(C(=O)NC2CCCCC2n2cccn2)CC1 C(c1c(Cl)nc2sccn12)=CC(N1CCC(C(C)NC(=O)COCC(F)F)C1)=O c1(CCC(=O)OCc2c(OCC#C)cccc2F)cnc2n1CCCC2 C(=O)(C#CC1(CC)CC1)N(C1CCCC(NC(c2cc(SCC)ncc2)=O)C1)C C1(C(=O)NCCCN2CCN(CC)CC2)CN(C(c2ccncc2)=O)CCN1C c1(C(=O)NC(CCNC(C2C(=C)C2)=O)C)ccnc(OC)c1 N1(CC(=O)N(C2CCN(C(c3scnc3C(C)(C)C)=O)C2)CC)CCCC1CO N1(C(c2cccc(C(C)=O)c2)=O)CCCC2CN(C(=O)CC=C(Cl)Cl)CCC12 C12(CNC(CC=C)=O)CC(NC(C3CCC3C)=O)(CO1)C2 O=C(C1=NOC2(CCN(Cc3cc(O)ccc3Br)C2)C1)NCc1ccc(F)nc1 c1(C(=O)NCC2CN(C(C(C=CC)O)=O)CC2O)cnc2c(c1)OCC(=O)N2 CC1(NC(=O)C(F)OC(F)(F)F)CCN(C(=O)CC2CC2)C1.c12cccc(c1)S2 c1(C(N2CC(NC(Cc3cc(C)[nH]n3)=O)C3C2C3)=O)cnc2cc[nH]c2c1 N1(Cc2cc(C)sc2C)CC(C2CCCN(C(c3c(F)ccc(Cl)c3F)=O)C2)C1 N1(C=O)CC(NC(=O)OC(C)(C)C)CC1(C)CO.N1(CCOC)CC(OC)CC1=O C12(C(N3CC4CCC(NC(COCCOC)=O)(C3)C4)=O)C3CCC(CC13)C2(F)F Cc1cc(CNC(C2CC3CC3N2C(c2ccc(=N)[nH]n2)=O)=O)ccn1 C#Cc1cccc(C(=O)N(C2CCCN(C(=O)CC3COC4CC3C4)C2)C)c1Cl c1(C(N2CC(CC(C)NC(C3(CC#C)CCCO3)=O)C2)=O)cc(F)c(C)cc1O C(=O)(C1Cc2ccccc21)N1CCC(C(=O)NCc2n(C)ncc2)C12CCC2 C1(C(=O)NC2CN(C(C3(CC(C)C)COC3)=O)CC(C)C2)CCc2nccn2C1 Cc1c(C(=O)NC2(CNC(=O)Cc3cnn(C(C)C)c3)CCC2)nnn1C(C)C Cc1cc(CNC(=O)C(C2(NC(=O)C=Cc3ccccc3)CCC2)C)ccc1F C(=O)(C(F)C(=O)NCC1(CC(=O)N(C)CC2CC2)CC1)OCC Cc1cc(OCCC(=O)NCC2COCC2NC(C2CNC(=O)N2)=O)c(C)c(C)c1 c1(OC)cc(C(N2CCCN(Cc3ccccc3F)CC2)=O)cc(Br)c1O C1(Nc2cc(COC)ncn2)CC(N=c2ccn3nccc3[nH]2)C1 C1(SC)CN(C(=O)CC2CCC(C#N)C2)CC1NC(=O)CCOCCN(C)C Cc1cc2cccc(CN3CCOCC3c3nn[nH]n3)c2o1 c1(N(C)C)ncnc(NC2CC3CN(C(=O)C4=CC5CCCC45)CC23)c1[N+](=O)[O-] C(=O)(C1=CC2C=CC1C2)N1CCC(CC(N2CCC(CC#C)C2)=O)C1(C)C c1(C(N2CC(C)C(CNC(C34CCCN(CC3)C4)=O)C2)=O)nccc2ccsc12 C1(CNC(c2nc(COCC)sc2)=O)C(C)CCN1C(c1cccc(N)c1)=O C1(C(N2CC(CS(C)(=N)=O)C2)=O)CC(=O)N(C2CCCCCC2)C1 N1(C(CC2CN(C(c3c(C)n[nH]c3)=O)CC2C)=O)CCCCCC1C C1(NC(c2cnc(CC)s2)=O)CCCC(NC(=O)C(C)(C)c2ccnn2C)C1 C1(CCC)(NC(=O)CNC=O)CCCN(C(=O)Cc2cnc(Cl)cc2C)C1 C(Cc1ccccc1)(CCNC(=O)C=CC1CCC1)NC(COCC(=O)OC)=O C=C(Cn1c(N(C)Cc2cc(C)c(C)cc2C)nnc1C1CC1)c1ccccc1 N1(C(C(COC)(C)C)=O)CCC(C)C(NC(=O)CN2CCCCC2=O)C1 C1(CNC(C(CC)O)=O)CC(F)(F)CN1C(c1cc(F)ccc1Cl)=O c1(COCC)nnc2n1CCN(Cc1cc(C)c(Br)cc1O)C2 c1(NC(C)C)ccc(C(=O)Nc2ncc(CC(=O)Nc3ccccc3)s2)c(Cl)c1 c1(C(=O)NCC(C)N(C(c2cnncc2C)=O)CC)ccc2c(c1)OCCCO2 c1(CN)ncnn1C.n1(CC(=O)NCC)cc(Cn2nccc2C(=O)O)nn1 c1(Nc2ccc(C(C)NCC(C)C)cn2)ccccc1CCO CCC(C)CC(C(=O)NC(CO)C1(O)CC1)NC(C1CC(=O)N(CC)C1)=O c1(-n2cc(C3(C(=O)NCC(CC(=O)OC)C)CCCC3)nn2)c(Cl)cccc1Cl c1(C(=O)NCCNC(C2CC2c2cccc(Br)c2)=O)ncnc2c1CCC2 C1(NC(c2cnccc2Cl)=O)C2CCC1N(C(C1CC1[N+](=O)[O-])=O)C2 c1(C(=O)O)ccc(S(=O)(=O)N2CCCC(C(N3CCOC(CCO)C3)=O)C2)s1 c1(C(=O)NC2CC(CNC(c3cc(C)[nH]c3C)=O)C2)ccc(F)c(S(C)(=O)=O)c1 c1(C(N(CCN(C(C(C2CC2)OC)=O)C)C)=O)c(C)cc(Cl)cc1N c1(C(=O)NC2CN(C(C3ON=C(C(C)C)C3)=O)CC23CC3)cnn2c1OCCC2 c1(C(=O)NC(C(=O)NCC(C)CC2CC2)Cn2ccnn2)ccc(O)cn1 C1(CNC(C2C(OCC)CC2)=O)(CNC(C2(CF)CCC2)=O)CCCCC1 C1(C(=O)NCC2CC(NC(c3c(N)sc(C)c3C)=O)C2)CC(C(C)(C)C)=NO1 C1(CC(=O)N(CCC(C)NC(Cn2c(C)nc(C)n2)=O)C)OCCOC1(C)C N1(C(C2CCCS2(=O)=O)=O)CCN(C(c2ccc(O)nn2)=O)C2CCCC12 CN1CCCCC1C(=O)NCc1cn(CC(=O)NOC(C)(C)C)nn1 c1(C(=O)NC(CNC(COC(c2nccn2C)C)=O)(C)CO)ccc(C#N)cc1F Cn1ncc2c(C(N3CC(NC(c4ccc[nH]4)=O)C(CO)C3)=O)cccc12 C1(NC(c2c(C)nc[nH]2)=O)CC2C(NC(C3CCC3C)=O)C2C1 CCN=c1ccc(C(=O)NC2CC2NC(c2ccsc2)=O)c[nH]1 C1(C(N(C2CC(c3cn(-c4ccncc4Cl)nn3)C2)C)=O)CCCN1C=O CC1CC2=C(C(=O)N1)C(c1c(Cl)cc(=N)[nH]c1Cl)NC(=S)N2C1CC1 c1(C(=O)NC2C=CC(CNC(c3cnccc3Cl)=O)C2)csc2c1CCCC2 N1(C(C(C)SCC)=O)CCOC2(CCS(=O)(=NC(=O)CC3OCCCO3)CC2)C1 N1(C(C2C(C)(C)C(=O)C2)=O)CC(C(N2CC3CC3C2)=O)C(F)(F)C1 c1(C(=O)NC23CC(CNC(c4cc(OC)ns4)=O)(C2)C3)cc2sccc2[nH]1 CC(CF)CC(=O)N(CCNC(=O)C(F)=CCCF)CCc1ccccc1 CC1CCS(=O)(=O)CCN1C(c1ccn(C(F)F)n1)C(=O)NC1CCC1 C12(C(=O)NCC#CCNC(Cc3cccc(OC(C)C)c3)=O)CCC(C)(C1)OC2 c1(CC(C)NC(C)=O)ccc(C(=O)NC2CC(=O)N(c3ccccc3Cl)C2)cc1 CCC(CC)CC(=O)NC1CCCCC1C(=O)NCCN1CCCC(O)C1 N1(C(C)=O)CCC2C1C(C(=O)N(CCS(N)(=O)=O)C)CCC2=O.c1(O)ccccc1 c1(C(N2C3(CNC(CN(C(C)C)C)=O)CCC2CC3)=O)cccc2c1CCOC2 Cc1nc(NC(=O)NCC2CCC(=O)NC2)sc1F C1(NC(C2CC=C(C)CC2)=O)C2CCCC1CC(NC(=O)CC(C)(C)C)C2 CC1(O)CCN(C(C2CN(C(=O)CC3CCCC4CC34)CC2F)=O)CC1O CC1CC(C(=O)NC2(CO)CN(c3nc(C(F)F)nc(=N)[nH]3)C2)CC(C)O1 c1(NC(N2C(CS(N)(=O)=O)CC(F)C2)=O)cc2c(nc1O)CCCC2 C1(C(C)N(Cc2cccnc2)CC2CC2C(=O)O)CN(C(=O)OC(C)(C)C)CCO1 N1(C(C=CC)=O)C(CNC(c2ncccc2OCC)=O)CC2CCCC12 CC1(C)CCCC(C(=O)NCC23CC2CN(C(=O)Cc2coc(C4CC4)n2)C3)C1 c1(N(C(c2nccc(C)n2)C(=O)NC2CCOCC2)C(C)C)cc(F)ccc1C N1(C(CCc2cc(C)[nH]n2)=O)CC2(C=C(C(=O)N3CCOCC(C)C3)CO2)C1 N1(C(C(C)=CC)=O)CCCC(CCC)(NC(C)=O)C1.c12ccc(cc1)s2 c1(C(N(C2CCN(C(c3cc(CC)nc(O)c3)=O)C2)C)=O)nccn2cnnc12 c1(CNc2c(C(=O)Nc3ccc(Cl)cn3)n[nH]c2)c(F)cccc1F c1(OC)ccnc(C(N2CCC(O)(CN(C)C(c3nc(C)nn3C)=O)C2)=O)c1O CCCCC(C(=O)NC1CCN(CCCCCF)C1)NC(=O)OC(C)(C)C C(=O)(C1=CC2(CCOC2)C1)NC1CN(C(c2c(C)cnnc2)=O)C(C)(C)C1 C(c1ccccc1[N+](=O)[O-])=CC(=O)NCC12C(CN(C(CN(C)C3CC3)=O)C1)C2 C(=O)(C(C#N)C(C)(C)C)NCC(C)(C)NC(c1ccc(Cc2nccs2)cc1)=O C1(C)(C(=O)NC(CC)CNC(=O)C(O)CCSC)CCCS1(=O)=O Cc1nnccc1C(=O)NC(CN(C)Cc1ccccc1)C(=O)NCCN=[N+]=[N-] C(=O)(C(C)C(O)C(C)C)NCC(CC(C)C)NC(c1ccn(C(C)C)c(=O)c1)=O C(=O)(CC(C)CC(C)C)NCCCN(C(Cc1nc(C(C)OC)sc1)=O)C c1(SCCCC(N2CC(O)(CCNC(=O)C(F)=C3CCC3)C2)=O)ccc(Cl)cc1 c1(OC)ccc2c(c1)CCC(C(=O)NC1CCCC1NC(C1CC1C(N)=O)=O)C2 Cc1nc(NCC(=O)Nc2ccc(F)cc2F)cc(=NCCOC2CCCC2)[nH]1 C1CN(N2C3CN(C)C(C3)C2)CCC1(F)F.c1(C)cc(O)ccc1Cl c1(OC)c(Cl)ccc(Cl)c1C(N1CC(O)(CCNC(=O)C(C)O)C1)=O N1(CC(=O)NC2CCC(N(C)C(C3CCNC3=O)=O)CC2)CCCNS1(=O)=O Cc1ccc(NC(=O)C(C)(C2CCC2)NC(=O)Cc2ccc(F)nc2)c(C)c1O C1(NC(c2scc(C)c2)=O)CC12CC(NC(=O)CC1C=NN(C)C1=O)C2 C(=O)(C1=CC2CCCC12)NCCC(C)N(C)C(c1ccc(N)cc1O)=O c1(NC(C=C(C)CNC(=O)C=CCF)=O)ccc(O)nc1.N1CCC1 c1(C(N2CCC(NC(C3CC34CC(F)(F)C4)=O)C2)=O)cc2c(cn1)CCCC2 N1(C(c2ccc(CC)cc2)=O)CCCC2C1CCN2C(=O)CC1CC(=O)NC1=O N1(C(C2(CC=C)CN(C(=O)CC3CCCOC3)C2)=O)CC2CC2C2CC12 C#CCCCCCCC(=O)N1CCCC1C=CC(=O)Nc1ccc(C)nc1O N1(C(C(C)SC)=O)CCCC2(CCCCC2NC(c2cn(C3CCC3)nn2)=O)C1 N1(CCC)CC(CNCC2CCCOC2)CC1=O C1(NC(C2C(OC)C2)=O)CCCC2CN(C(=O)COc3ccccc3SC)CC12 N1(C(C(CN(C(C(CCC)NC(N)=O)=O)C)(C)C)=O)CC2C(C1)C2(C)C C1(CNC(=O)C(C2CCCCCC2)O)C2CC1N(C(c1nc(Cl)cs1)=O)C2 c1(C(CCC)C)nc(-c2cc(C(C)C)nn2CCOC)n(CC(N)=O)n1 Cc1ccc(CN2CCCC(C(N3CC4CC(C3)O4)=O)CC2)c([N+](=O)[O-])c1 CC1CCn2cc(C(=O)NCc3nc(CNC(C4COC4)=O)cc(O)n3)nc2C1 Cc1nn(CCO)c(C)c1C(=O)N(C(C)CNC(=O)C(C)CO)C C1(NC(CC2CCN(C)C2)=O)CC2CC(NC(c3nc(Cl)cs3)=O)CC12 c1(C(N2C3CN(C(C4(CC)CCC4)=O)CC2C3)=O)nc(C)c(C)[nH]c1=O N1(C(c2[nH]cc(C(=O)OC)c2)=O)CC2(C1)CN(C(=O)C(C#N)C(C)(C)C)CCO2 C(=O)(C1CCN(C(=O)OC(C)(C)C)c2ccccc21)N1C(C)C(C(=O)O)CC1 C1(C2CCCCN2C(=O)C2CC2)(CNC(=O)CCc2nccs2)CCOCC1 c1(C(C)=O)cc(C(N2CCC(CO)(NC(C34CCC3C4)=O)CC2)=O)c(C)nc1C C1(CC(=O)NC(CCCC)C)N(C(=O)CSCCC(C)C)CCC1(C)C C12(NC(c3cccc(-n4ccnc4)c3)=O)CC(C1)N(C(c1cncc(O)c1)=O)C2 c1(C(CC)C)cc(C(=O)NC2CCC(NC(=O)C=CCN3CCCC3)C2)on1 C(C(C)NC(C1CC(C(=O)OC)C1)=O)(C1CC1)OCC c1(C(N(CCN(C(C(C)OC2CCCC2)=O)C)C)=O)cccc(C2CCCC2)c1 c1(OC(c2ccnn2CCOc2cscn2)=O)cccnc1NC1CCCC1 Cc1ccnc(O)c1C(=O)N(C(C)CNC(=O)C(C(C)C)n1cnnc1)C C1(CCC(=O)NCCN(C(=O)C(CO)NC(N)=O)C(C)C)CC(F)(F)C1 C1(NC(C(C)OCC)=O)CN(C(c2cc(C)c(CC)nc2O)=O)CC1N=[N+]=[N-] c1(C(=O)NCC(C)NC(=O)Cc2cnco2)ccc(C2CCC2)cc1 C#CC(C)(C)C(=O)NCC1CCN1C(C1(n2ccnn2)CC1)=O N1(C(CC(=O)NC)=O)CCOCC2(C1)CN(C(=O)CN(C1CCCC1)C)CCO2 C(CC(CC)C(=O)NCC1(CNC(c2cnc(Cl)n2C)=O)CC12CCC2)=CC C1(NC(C2OCC(C)C2)=O)CC2CCC1CN(C(c1ccccc1OC1CC1)=O)C2 C123CCCC1N(CCC2)C(=O)CCOCC(=O)NC3.C(C(C)(C)C)OC(C)C C(N=c1nc2scnc2c(N(C)CCOC)[nH]1)C1N(C(C)C)CCC1 Cc1ccc(C(N2C3CCC2CN(C(C2CCN(C)C2C)=O)C3)=O)c(N)c1Cl C(=O)(C1CN(C(=O)OC(C)(C)C)Cc2n[nH]cc21)NCCNC(CCC=C)=O c1(C(=O)NCC(COC)N)cc2c(cc1Br)OCCO2 c1(C(=O)NC2(CO)CN(C(C3(C#N)CC(C)C3)=O)C2)cnc2ccc(F)cc2c1 CN1CC2CCN(C(=O)CCN(CCCO)C(=O)CC3CCCOC3)CC2C1 CC(c1cnn(C)c1)=CC(N1CCN(C(C2CSCCS2)=O)C(C2CCC2)C1)=O c1(C(C(=O)NC(CNC(c2cnc(C)s2)=O)CC(C)C)O)ccc(Cl)c(F)c1 c1(C(=O)NCCCN(C(C2CC(C)=C(C)CC2)=O)C)ccc2n[nH]cc2n1 c1(NC(C)=O)cccc(F)c1C(N1CC(O)(CN(C)C(C2CCSC2)=O)C1)=O C1(NC(c2c(C)nco2)=O)CC2CC(NC(=O)CC3CC(=O)NC3=O)C1C2 N1(C(c2snc(O)c2Cl)=O)CCC2CCN(C(c3cc4ccccc4o3)=O)C2C1 N1(C(C2(F)CCC(C)CC2)=O)CCN2CCN(C(=O)CC3(CO)CC3)CC2C1 N1(C(c2c(C)ncnc2)=O)CCC(CNC(c2ccncc2)=O)C(C)C1 c1(N(C)C)ccc(C(=O)NC2CCCC2NC(c2c(C)nn(C)c2Cl)=O)c(F)c1 c1(OC)ccnc(F)c1C(N1CCC(O)(C(C)NC(=O)CCC(F)(F)F)C1)=O c1(C(N2CCc3scc(Br)c3C2)=O)cc(Cl)c2cn[nH]c2c1 C1(C)(CNC(CC(CC)SC)=O)CN(C(=O)CCC2(C)CC2(F)F)CC1C Cc1ccc(Cl)c(CN2CCC(OCc3cccnc3)CC2)c1 N1(C(CCC(=O)N(C)C)=O)C(CC(=O)NCCN2C(=O)CCC2=O)C2CCCC12 C12(NC(c3cn(C(F)F)cn3)=O)CCN(C(=O)CCN3C(=O)CCC3=O)CC1C2 CCC(C)(C#N)C(=O)Nc1ccc(NC(=O)C(O)C(F)(F)F)c(C)c1 C(C1CN(C(C2C(C)C2C)=O)CC1C(N1CC(=O)NCC1C(C)C)=O)=CC N1(C(c2c(CNC(=O)C=Cc3cc[nH]n3)n[nH]c2)=O)CC2(CNC(=O)N2)C1 N1(C(C(C)CCc2ccccc2F)=O)CC(c2ccccc2)CCC1C Cc1oc(S(N)(=O)=O)cc1C(=O)NC1CN(C(c2cc(F)cc(F)c2)=O)CC1C c1(NC(N(C)C)=O)cc(NC(=O)Nc2ccc(-c3ncn(C)n3)cc2)cc(Br)c1 CC1(CNC(=O)C(F)=C2CCC2)CCCN(C(=O)C(c2cccc(F)c2)O)C1 C1(CNC(c2cc(OC)no2)=O)CCCC2CN(C(=O)Cc3cncn3C)CC12 C1(O)(CN(C(=O)C(c2ccco2)NC(=O)CCC2CC2(C)C)CC)CCC1 c1(C(N2CCCC(CC(=O)Nc3ccc(C4CC4)nc3)C2)=O)cc([N+](=O)[O-])n[nH]1 CC(C)CS(=O)(=O)CCC(=O)N1CC2CC(NC(C3(SC)CCC3)=O)CC(C2)C1 c1(C(=O)NCC(C)N(C(C(C)NC(CC)(C)C)=O)C)cc2ccccc2c(O)n1 c1(C(=O)NCC(CN(C(=O)C2=CCC2)C)(C)C)cccc2c1OCCC2 C1(C(CN(C(C(C=C)C)=O)C2CCCO2)F)CCN(C(=O)C=CCCC(C)C)CC1 N1(C(C2(C#C)CCC2)=O)CCCC(CN(C)C(C2(OC)CS(=O)(=O)C2)=O)C1 c1(N(C)Cc2cncs2)nnc(C(C2(OC)CCCC2)O)n1CC(C)C(F)(F)F CCC(C(=O)NC1CN(C(=O)C(F)F)CC1(C)C)C(C)O c1(C(N(C(C(N2CCC(CCC)C2)=O)CC)C)=O)ncccc1O C1(OC(C2CC3CC2(c2ccncc2)C3)=O)CCOC2(CCC2)C1 C1(CNC(C2(C#N)C(C)C2)=O)(CNC(=O)Cc2c(Cl)cnn2C)CCCCC1 C1(NC(C2N(S(CC)(=O)=O)CCC2)=O)CCCN(C(=O)C(F)(F)CSC)CC1 N1(C(c2nc(CC)oc2C)=O)CCCCC(NC(c2csc3nnsc23)=O)C1 c1(C(=O)NC2CC(C(C(=O)N(CC(C(=O)NC)C)C)F)C2)cc(C)c(C)o1 N1(C(C2CC3(C(OC)CC3)C2)=O)CC2CCN(C(c3[nH]c(C)nc3C)=O)CC2C1 N1(C(Cc2c(C)ocn2)=O)CCCC(F)(CNC(=O)CN2CCSCC2)C1 C1(NC(Cc2c(C)scc2)=O)CN(C(=O)CC2CCN(C)C2)C2(CCC2)C1 N1(C(C2CCC(C)N(C(=O)CCc3ccsc3)C2)=O)CC2CN(C)CC2C1 C1(NC(C=C(COC)C)=O)CCN(C(=O)CN2CC(=O)N(C)C2=O)C12CC2 C1(NC(N2CCC(Nc3scc(C)n3)CC2)=O)CCc2nc(C)cn2C1 c1(N(C)C)ncc(C(=O)NCCC(O)CNC(=O)Cc2sccc2Cl)s1 N1(C(CC(C)C)=O)CCC2CN(C(=O)C(F)Cc3ccc([N+](=O)[O-])cc3)CC2C1 C12CCCC(CC1)C(=O)N2.CC1CCC(C(=O)N(NC[Si](C)(C)C)C)CC1 C#CCCCCC(=O)NCC12CC(CN1C(c1ccc(N)c(O)c1)=O)C2 C=CC1CCN(C(=O)CC2(C=C)CN(C(=O)CC3CCCC3C)C2)CC1 C(=O)(C1=C(c2cnco2)N(C2CC2C)C(=S)NC1c1cn(C)nc1CC)OCC C(CCCC(=O)N1CCCC1C(C)NC(c1cnn(C)c1C(F)F)=O)SC c1(C(=O)NC(CC)C(N)=O)cc2c(s1)CCN(C(=O)C(C)NC(C)=O)C2 c1(CC(=O)N(C)CC2(O)CN(C(c3nc(C)sc3)=O)C2)cccc(C(F)(F)F)c1 n1(CC(N2C(CC(=O)NCc3ccsc3)COCC2)=O)ccc2c(F)cccc12 C1(C(=O)NC(C2CCCN2C(=O)CC(=O)NC2CC2)C)CC(C)(C)SC(C)(C)C1 C1(C(=O)NC(C)(C)CC2CCC2)C(C2CC2)CCN1C(C1CS(=O)(=O)C1)=O C(=O)(C1CCc2cc(Br)ccc21)NCCN(C(=O)CC1CC1(Cl)Cl)C C1(C(=O)NC2C=CC(C(=O)NC)C2)(NC(=O)Cc2cncnc2O)CCCOC1 c1(CC(=O)NC2CN(C(CCCN(C(C)=O)C)=O)C(C)C2)ccc(C#N)cc1 c1(N2CC(CC(C)NC(C3CCCN(C(C)=O)C3)=O)C2)ncc(C)c(C)n1 C12(C(=O)OC)CC1CN(C(C1CN(C(c3cncc(OC)n3)=O)CCO1)=O)C2 CCCC(CC)C(=O)N(CCCNC(=O)CC12COC(C1)C2)C c1(C(=O)NC2C=CC(CNC(Cc3nc(CC)sc3)=O)C2)ccc(C#N)[nH]1 C(C(=O)N1CC(C(=O)NCCc2cc[nH]n2)C(C)C1)(C(C)C)SC c1(NC(C(CC#C)(C)NC(=O)C(C)OCC2CC2)=O)cc(C)cn(C)c1=O N1(C(C2(C)CCC(=O)N2)=O)CCN(C(c2ccc(N)c(Cl)c2O)=O)C2CCC12 CON1CC(C(=O)NCC(C)NC(=O)C(C)(C)C(=O)OCC(C)(C)C)CC1=O N1(C(c2cncnc2)=O)CCN(C(C2C3CCCOC23)=O)C2CCCC12 c1(C(=O)NCC2C(NC(C3N(C(C)C)C(=O)CC3)=O)C2)cc(=O)c(Br)c[nH]1 C1(C)(C(C2CCCN2C(N)=O)C)CC(C(=O)NCC2CCCN2C)C1 N1(C(C(c2ccccn2)C)=O)CCC(C)(CNC(=O)C=CCN2CCCC2)C1 C(CS(=O)c1ccccc1)NC(C(=O)N(C)CC1CC1c1cccnc1)=O C=C(C)CCC(=O)NCC1(CNC(c2csc(CCCCC)n2)=O)CCC1 C1(N(C)C(c2csnc2Br)=O)C2CN(C(=O)CCC3CC3(C)C)CC12 N1(C(c2nc(C)nn2C)=O)CCC2CCCC(C1)N2C(c1c(C)cncc1C)=O c1(OCC)ncc(C(=O)NCC2CN(C(=O)CSCC3CCCC3)CC2C)cn1 C(=O)(CC(C)(O)CC(=O)O)N1CC(F)CC(NC(c2c(F)ccc(C)c2F)=O)C1 N1(C(C2CC(NC(c3c[nH]c(=NC)s3)=O)C23CCC3)=O)CCCCC2(CCC2)C1 C1(NC(C(C(C)C)NC(C)=O)=O)CC2CC1CC2C(=O)NC1CCOCC1F c1(CC(N2CC(CN(C(C(CC=C)NC(C)=O)=O)C)C2)=O)c(C)nn(C)c1Cl C1(C(=O)NC(C)CSCCO)(COC)CN(C(=O)Cc2ccccc2)C1 C1(N(C(c2cc(CCNC(CCOCC(C)C)=O)on2)=O)C)CCC(=O)N(C)C1 CC(O)C(C(=O)NCC1(F)CC(NC(c2cc[nH]c2)=O)C1)NC(=O)C(F)(F)F Cc1[nH]nc2ccc(C(N3CC4(NC(c5c[nH]nc5Br)=O)CCC3C4)=O)cc12 C(=O)(CC(C)C(F)F)NCCC1(NC(c2occ(C)c2)=O)CCCC1 c1(C(C(=O)NC(C)C(C)NC(C2(n3cncn3)CC2)=O)C)ccc(F)cn1 C(=O)(C1CCc2nccn21)N1C(CC(=O)OCC)CN(C(=O)CSCCOC)CC1 c1(C(N2C(C3(NC(C4CC(=C)C4)=O)CC3)CCC2)=O)ccn(CCOC)c(=O)c1 C1(C(=O)NC2C(SC)CCC2)CCCN(C(C2(F)CCOC2)=O)CC1 c1(C(=O)NC2CCCC23CN(C(C2CC=CCC2)=O)C3)ccc2c(c1)CCOC2 C1(CC=C)(NC(C2(n3cccn3)CCC2)=O)CCN(C(=O)Cc2ncoc2C)C1 C(=O)(C(F)C(C)C(F)(F)F)OCc1cn(CCOc2c(C)nc(Cl)cc2)nn1 c1(C(=O)NC(C(C(C)C)C)CNC(c2cnns2)=O)cccc2c1CCN2 C1(C(N(C)CC2CCCN2C(=O)CCC2CC2(Cl)Cl)=O)CCCN1N=O N1(C(c2ccc(CC)o2)=O)CC(N=c2[nH]nc(C(F)F)s2)C2(CCC2)C1 c1(C(=O)NC2C(NC(C(c3cccc(OC)c3)O)=O)C2)cccc2ncsc12 Cc1ccc(C2(C(N3CCC(CF)(NC(C4C(C)C4(F)F)=O)C3)=O)CCC2)cc1 N1(C(CCN(C)CC)=O)CC(CNC(c2ccc(CNC(C)=O)cc2)=O)C2CC12 CCCC(CNC(c1c[nH]nc1C(F)F)=O)C(=O)NC(c1ccncc1)C Cc1nc(NC(C)CC(C)NC(c2ncsc2C(F)(F)F)=O)ccc1C#N N1(C(C(C)(CO)OC)=O)CC2CCC(C1)N2C(c1ccc(NC(C)(C)C)cc1)=O N1(C(c2ncc(OC)cn2)=O)CCCCC(NC(=O)C=C(F)c2ccccc2)C1 C(=O)(C1=CCCOC1)N1CCC(N(C(=O)CCc2cnccn2)CCO)CC1 C(=O)(C(C(C1CC1)C1CC1)N(C)CCc1nc(C)cs1)NCCC c1(OCC=C)ccccc1C(=O)NCC1CC(C)N(C(C2C3CC4C(C3)C24)=O)C1 C1(C(=O)NCCC(C)N(C(c2ccc(SC)o2)=O)C)CC2OC(=O)OC2C1 N1(C(c2c(C(C)C)cccc2)=O)CC2CCC2(CNC(C2(CO)CC2(F)F)=O)C1 c1(OC)cc(F)ccc1CC(N1CC(NS(C)(=O)=O)C(C#N)C1)=O N1(C(c2oc(CC)c(C)c2)=O)CCCC(C)(C)C1C(=O)NC(C)C(C)F c1(C(N2CC(Cn3cc(CCN(C)CC)nn3)C2)=O)c(C)cnc2ccccc12 c1(OC)cc(CN2CCNCC(C(=O)O)C2)ccc1C#N c1(SC)cncc(C(=O)NCCCNC(C2(F)CC2c2ccccc2)=O)c1 Cc1ccc2ncnc(N3CCC(NC(c4nccn4C)=O)C(O)C3)c2c1 c1(C(=O)NC23CC(CNC(C(C(CC)C)C)=O)(C2)C3)ccc(Cl)c([N+](=O)[O-])c1 c1(C(=O)NCCC(C)NC(C2(NC(=O)OC)CCCCC2)=O)cc2c(s1)CCC2 CCC(CC(F)F)C(=O)NC1CCN(C(c2cc(-c3ccco3)on2)=O)CC1F Cc1cc2cccc(NC(c3csc(NS(=O)(=O)c4ccccn4)n3)=O)c2cn1 c1(C(=O)NCCN(C(CCC(C)SC)=O)CC(C)O)cnc(C)c(N)c1 CC(C)C(C(=O)NC(C)CCCNC(C1(O)CC(F)(F)C1)=O)n1cnnc1 C1(CC(=O)NC)(CNC(=O)CS(=O)(=O)N2CCCCC2)CCCCC1 CC12CC(C(=O)NC3CCCCC3NC(=O)CC(=O)NC3CC3)(C1)C1(COC1)O2 C(=O)(CC(C)C(C)(C)C)N1CCCC(NC(c2c(C)n[nH]c2)=O)C1 c1(OC)c(C(N2CCC(NC(=O)CCC(C)(C)O)C(C)C2)=O)cccc1F c1(C(c2nnnn2Cc2ccccc2)NC(CC)(C)C)coc(C)n1 Cc1oc2cc(C(N3CC(C)(NC(C4CCCCS4)=O)C3)=O)[nH]c2c1C Cc1nnc(C(=O)NC2CC(F)(CNC(c3cccn3-c3ccccc3)=O)C2)s1 C(=O)(C(=O)N=S(C)(C)=O)N1CCC(O)(CN(C(C#CC(=O)N(C)C)=O)C)CC1 Cc1cc(Cl)c(F)cc1CNC1CC1C(=O)Nc1ccc(C#N)cc1C(F)(F)F C(C)(C(C)(C)C(=O)N1CCCC(O)CC1)NC(c1c(C)nncc1)=O c1(C(=O)NCCCN(C(CSCCCC)=O)C)ccc([N+](=O)[O-])c(SC)c1 C1(NC(C=C(CC)CC)=O)COCCN(C(=O)C(F)=C(C)C)C1 c1(C(N2CC3C(NC(CN(C)CC)=O)(C3)C2)=O)cn2cccnc2n1 C1(NC(c2cn(CCC)nn2)=O)CC(C(=O)N(C2CCCC2O)CC)CC1O CN1CCC2CN(C(C3(NC(=O)CC4CCC(=O)NC4)CCCC3)=O)CCC12 c1(C(N2C(CNC(C(COC)C)=O)C(C)CCC2)=O)cc2c(C)cc(F)cc2[nH]1 c1(CCC(=O)NC2(CNC(C3CC4CC3C4)=O)CCCC2)cccc(F)c1Br C(=O)(C1=C(CCCCl)N(CCC2CC2)C(=S)NC1c1cccc(Cl)c1Br)OCC C(=O)(CC(C)(CN)C(F)(F)F)Nc1cncc(-c2cccc(C)c2)c1 N1(C(C2C(C=C)C2)=O)CCC(O)(CN(C(=O)C=C(Cl)Cl)C)C1 C(CC(O)C(=O)NCc1ccc(C(N2CCC2CC2CCCC2)=O)s1)N(C)C C12CN(c3ccnn3C1)C2=O.c1(CN)nc(=O)n(C2CN(C(=O)OC(C)(C)C)C2)[nH]1 n1(C(CC)C)nc(C(=O)NCCC2CN(C(c3cscc3C(N)=O)=O)C2)cc1C O=C(N=c1cco[nH]1)C1CCCCC1NC(=O)Cc1cc(F)cc(F)c1 Cc1nc(C(N2CC(N(C)C(c3cc(Cl)cn3C)=O)C(O)C2)=O)ccc1[N+](=O)[O-] c1(C(N(C2CCCN(C(CCCNC(C)=O)=O)C2)C)=O)cnc2ccnn2c1 C1(NC(c2n(C=C)nnc2)=O)CCC12CN(C(c1ccc(OC(C)C)nc1)=O)C2 C#Cc1cnc(C(=O)N(CC(=O)NC2C(C)C2(C)C)C)c(C)c1 c1(OC)ccc(CCCCC(=O)N2CCC(CC(C)NC(=O)C(C)O)CC2)cc1 c1(C(=O)NCCNC(CCCCCC(C)O)=O)cc(Cl)cc2c1NCCC2 S(=O)(=O)(c1cc(C=CC(=O)NCC(c2ccccc2)C)ccc1OCC)NCC c1(C(N2CC(CNC(=O)C(F)OC(F)(F)F)C(O)C2)=O)cc2c(s1)CCC2 C1(CC#C)(C(=O)NCC2(F)CC(CNC(=O)C(C3CC3)N(C)C)C2)CCOCC1 c1(C(=O)NC23CC(CNC(=O)C=C4CCCCC4)(C2)C3)ccc(F)c(Br)c1 C(=O)(CCC(F)F)NC(CN(C)C(C1CCCC1(C)C)=O)(C)C C(CNC(c1cc(C2CC2)[nH]n1)=O)(CC(=O)NCCc1csnn1)OC c1(C(=O)NC2C(NC(C3CC(C)OC(C)C3)=O)COC2)c(Cl)ccc(F)c1F Cc1cc(F)ccc1NC(=O)C(c1cc(Br)c(Br)o1)N(C)Cc1ccc(F)c(Br)c1 C1(C2CCCCO2)(C(=O)NCc2cn(CCC)nc2C)CCCO1 c1(C(=O)NC(C(C)C)CNC(=O)Cc2cc(F)cc(Cl)c2)cccc2ncnn12 C(=O)(C(C)c1cc[nH]n1)NCCSCC(=O)N(CCCC)CCCO n1(CC(=O)NC2C(NC(CCCC(C)C)=O)C2)ccc2cc(Br)ccc12 c1(C2(C(=O)NC3C(CNC(Cc4nnc(C)o4)=O)C3)CC2)cccc(F)c1F N1(c2c(F)cnc(OCC)n2)CC2CN(Cc3cc4sccc4s3)CC2C1 c1(C(=O)NC2CC(C(=O)NCCSCC)C2)ccc(C(F)(F)F)c(Cl)c1 C(C(N=[N+]=[N-])C(=O)NC(CC1CC1)CC(=O)NCC1CCC2(CC2)C1)OCC CC(C)C(C(=O)N1CCCCC1CO)NC(C1(C)CC2CC2C1)=O C1(C(=O)NC(CN(C(=O)CCn2c(C)ccc2C)CC)C)COC(C)(C)CO1 Cc1sc(-c2ccco2)nc1C(=O)NCC1CC(NC(c2cc(CO)on2)=O)C1 C1(Cn2cc(C(N(CC(F)(F)F)CC)=O)nn2)CCCN(Cc2ccc(F)cc2)C1 N1(C(c2n(CCC)ncc2)=O)CC2CC1CC2NC(c1cc[nH]c1)=O C1(CC)CN(C(c2cc(C#N)c[nH]2)=O)CCC1NC(=O)CC1CC(O)C1(C)C c1(CC(=O)NC2CN(C(c3ccncc3C(F)(F)F)=O)CC2O)cccc(Cl)c1 C1(C(N2C(CN(C(c3n(C(C)C)ccc3)=O)C)CCC2)=O)Cc2cscc2C1 CCCC(C)C(=O)NC1(COC)CN(C(c2cn(CC(F)(F)F)nn2)=O)C1 N1(Cc2cnc(OC)nc2)CCC(F)(C(N2CCN(C3COC3)CC2)=O)CC1 N1(CC)CCCCC1C(=O)NCC1CC(CNC(=O)COC2CC=CC2)C1 C1(NC(COc2ccn(C)n2)=O)CC(NC(C2CC(=C3CCC3)C2)=O)C12CCC2 C(N1CC(C)CC(C#N)C1)c1onc(-c2c(Br)cc(OC)c(OC)c2)n1 C(=O)(CN=c1cc[nH]cc1)N1C(CO)CC(NC(c2c(C)snc2)=O)C1 c1(OC)cc(Cl)c(Br)cc1C(=O)NCC(CO)NC(C1(Br)CC1)=O Cc1noc(C2CC2)c1C(=O)NC1CCC1NC(=O)CC(O)CN(C)C CC1CC(=O)CCN1CC(=O)Nc1ccnn1-c1cccnc1 C1(C)(CC)C=C(C(=O)N2CC(C(C)NC(=O)C(C)C3(O)CCC3)C2)C1 N1(C(C2CC(=C)C2)=O)CC(C(=O)NCCC(C)N(C)C)C2(CC2)C1 c1(OC)cc(C(N2CC(NC(=O)C(C)(C)c3cncs3)C(O)C2)=O)cc(Cl)c1O C#CCCCCCC(=O)N(CC(C)(C)C(=O)NC1(CC=C)CCOC1)C C(C1(O)CCCc2ccccc21)N1C2(c3cn(CC(=O)O)nn3)COC(C1)C2 c1(CNC(c2ccc(C)[nH]2)=O)nccc(C)c1F.C12(CCCC1C)C(=O)N2C1CC1 CC1(C(=O)NCCOCCC(=O)NC2CCCSC2)CCC(=O)C1 Cn1nc(CC(=O)NC2(C)CCN(C(=O)Cc3cncs3)C2)cc1C(F)(F)F N1(C(CCC#C)=O)CC(NC(c2cc(O)cnc2Cl)=O)CC12CCC2 c1(CC)cccc(C(N2CCC(CN(C(=O)C(CCOC)OC)C)C2)=O)n1 C1(C(=O)NCC2N(C(C(CC)C)=O)CCCC2(C)C)CC(c2cnn(C)c2)=NO1 c1(C(=O)NC2CN(C(c3ccnc(C)n3)=O)C(C)C2)cc2ccc(Cl)c(F)c2o1 Cc1nc(Cl)nc(N2CCCC2(C)CNC(c2ccc(O)nc2)=O)c1Cl C(=O)(CCCCCN=[N+]=[N-])NC(C1CCN(C(c2cc3ncccc3[nH]2)=O)C1)C c1(CNC(CCSCCC)=O)cc(O)nc(CNC(=O)CCc2ccnn2C)n1 C(=O)(C1=Cc2cccc(OC)c2OC1)N1CCC(CNC(C(C)OCC#C)=O)C1 C1(NC(C(COCC)C)=O)CC2CCC1C(NC(c1cc3c(ccn3C)[nH]1)=O)C2 Cc1ncnc(N2CCC(C(=O)NC(c3ccc(Cl)cc3)C3CC3)C(O)C2)c1Br C(=O)(C1CSc2ccccc21)NCC1C(NC(c2csc(C)c2C)=O)COC1 Cn1c(=N)[nH]c2cc(C(=O)NC3COC4(CCCN(C(=O)CNC=O)C4)C3)ccc12 c1(C(N2CCC3(CC(NC(c4cnns4)=O)C3)C2)=O)ccnc2ccccc12 N1(C(C(C(C)C)CO)=O)CCC2(CCCN(C(C3COC4COCC34)=O)C2)C1 C1(C(=O)NCC2OCCN(CC)C2)CNCC2(CCC2)C1 C1(N(C)C(c2cocn2)=O)CCC(NC(C23CCCC2C3Br)=O)CC1 c1(C(=O)NC2CC(C)N(C(=O)Cn3cnnc3)C2)ccc2ccc(Br)cc2n1 N1(C(c2cccc(C)c2F)=O)CC(NC(C2CN3CCCC2C3)=O)C2(CCC2)C1 c1(NC(C)=O)ccc(N)c(C(=O)N(C2CCN(C(=O)C(N)=O)CC2)C)c1 C(=O)(C(C)(O)C(C)(C)C)N1CC(COC)N(C(c2ccc(F)c(SC)c2)=O)CC1 CCC(C)(C)C(O)C(=O)N1CCN(C(=O)C=C2CCC2)CC1C1CC1 CCCC(C)CC(=O)N1CCC(F)(CNC(c2ccc(CN(C)C)[nH]2)=O)C1 c1(C(N2CCC(CCCCNC(C3C(COC)C3)=O)CC2)=O)nccc(N)c1Cl N1(Cc2nc(C(=O)OCC)nn2C)CCC(=O)N(CC2CC3CC3C2)C1=O N1(C(C2CC(C)(C)C2)=O)C2CCC1CC(NC(c1cc(Cl)cc(F)c1F)=O)C2 Cc1noc(C)c1S(=O)(=O)N1CCC(O)(C(N2CCC(C#N)C2)=O)C1 C(=O)(C#CC1(C)CCCO1)NC(C(=O)NCC1CCC(C)C1)Cc1cn[nH]c1 CC1CCC(N2CCC(NC(=O)C(=O)NC(C3CCCC(C)C3)C)CC2)CC1 c1(C(N(CCCOCCN(C(C=CC)=O)C)C)=O)cc(F)c(Cl)c([N+](=O)[O-])c1 N1(C(C=CC(=O)OC)=O)CCN(N2CC(OC(=O)N(C)C)C3(CCC3)C2)CC1 N1(C(c2ncn(C)c(=O)c2)=O)CCCCCC(NC(C2CC3C=CC2O3)=O)C1 C(=O)(CC(C)C(F)(F)F)N1CC(OC)(CNC(=O)Cc2nc(C)sc2Cl)C1 C1(CCCN(C(C2C=CCCC2)=O)CC)CCCN1C(=O)C(C)N1CC(C)C1 N1(C(c2c(C)ccc(=N)[nH]2)=O)CCC2(CCCN2C(=O)CC2CCSCC2)C1 c1(C(=O)NC2(CC=C)CCN(C(c3ccnnc3)=O)C2)cnc(Br)c(OC)c1 c1(CC)cc(C(N2CC(F)CC2CNC(C2(C)CCCCO2)=O)=O)ccc1F N=c1ncc(C(=O)NC2CCCCC2NC(c2cocc2Br)=O)c[nH]1 c1(C(=O)NC2(C3N(C(CN(CCC#C)C)=O)CCC3)CC2)ccc(C(N)=O)nc1 C(=O)(CC(C)(C)C(C)=O)NC(C(=O)NC(CC)(C)CN(C)C)C(C)OC N1(C(C(CCC(C)C)NC(C2CN(CC)C(=O)C2)=O)=O)CCCC2CCCCC12 c1(C(=O)NCc2cc(C(N3CCC(CC=C)C3)=O)on2)cc2ccccn2n1 C1(NC(C2(CCC=C)CC2)=O)CCN(C(c2cnco2)=O)CC12CCC2 c1(NC2CCC(C)CC2N2CC3CCC2C(C(=O)O)C3)ccc2c(c1)CCC2 C1(C)(NC(C)=O)CCN(C(=O)C(c2ccoc2)NC(=O)C(C2CCCCC2)C)C1 C1(C(=O)NCCCCCCN(C(C(C)NC(C)=O)=O)C)NC(=O)C2CCC12 C1(CNC(c2c(C)cncn2)=O)CC2(CCC2)CN1C(=O)CSC(C)C Cc1nccc(C(=O)NC(C(=O)NCCC(=O)N(C)C2CC2)C2(O)CCC2)c1N C1(NC(c2c(C)nccn2)=O)CC=C(C(=O)NCC2(C)CCOC2)C1 N1(C(c2cc(OC)no2)=O)CC2CCN(C(c3ccn(C(C)C)n3)=O)C(C2)C1 C1(c2cn(-c3ncn(CC)n3)nn2)CCCN(C(=O)C(C(C)C)NC=O)CC1 C(CCC=C(C)C)(C(=O)N(C(C)(C)C)C(c1ccccc1)C)N(CC=C)CCC N1(C(C=C(C)c2ccccc2)=O)CCN(C(=O)C#CC2CC2)C(C)CC1C CC1(C)C2CC(CNC(C3CCC3)=O)CC12.C1(=O)C(=O)NCCN1.C12CC1C(=O)N2 c1(C(=O)NCC23C(CN(C(CCc4c(C)ncs4)=O)C2)C3)cnc(N)c(Cl)c1 C(=O)(CCCCC(=O)NC(C1CCN(C(c2ccnn(C)c2=O)=O)C1)C)NC C(=O)(C1=NOC2COCC12)NC(CC(C)NC(c1ccc(C(=O)OC)o1)=O)C c1(COc2c(CNC(C(CC)C)c3ccco3)cccc2)cccc([N+](=O)[O-])c1 C1(CC=C)(NC(=O)CC2CC=CC2)CCCN(C(C2CCN2C(C)(C)C)=O)C1 CC(C)(C)CC(O)C(=O)NC1CN(C(c2sccc2-n2cnnn2)=O)CC1O C1(NC(C2CC(SC)C2)=O)CC(O)CN(C(=O)C(F)=CCCF)C1 c1(OC)cncc(CCC(=O)N(CCCNC(c2occc2C)=O)C2CC2)c1 N#CC1CCCC1NC(=O)CC(CC1CC1)NC(=O)CC1CC(F)C1 Cc1noc(N)c1C(=O)NCCCCCN(C)C(C1CCC1n1ccnc1)=O c1(N(C)CC2CCCN2)cnc(C#N)cn1.c1(C=O)cnc(CC2CC2)s1 Cc1ccc2cc(C(N3CC4CC3CN4C(C3(O)CC(C)(C)C3)=O)=O)[nH]c2c1 C1(OC(C)C)CCOCC1.CC(=O)CN1CC(=O)OCC1=O c1(C2CCN(CC3C(C(=O)O)CC3)C2)nc2ccc(F)cn2n1 c1(CN2CCCC(Nc3ccc(C)cn3)C2)cncc(P(C)(C)=O)c1 C(=O)(C1=CC(C)(C)C1)N1C2(C(=O)NCC(C)CN3CCCC3)CC2CC1 N1(C(C2CC(=C)C2)=O)CCCCC1C1(NC(=O)C(C)NC(=O)NC)CC1 C(=O)(C1=CC2(CN(C(=O)CN=c3cc[nH]cc3)C2)OC1)NCC(C)(C)C1CC1 Cc1ncn(C)c(=O)c1C(N1CC2CC2(NC(=O)CC2CC3(CC3)CO2)C1)=O n1(CC(=O)NCC2C(NC(CC3(C=C)CCC3)=O)CCC2)cccc(O)c1=O C12(NC(C)=O)CN(C(=O)Cn3cnc4ccccc34)CC1CS(=O)(=O)C2 c1(NC(C2C=CC(NC(c3cc[n+]([O-])cc3)=O)C2)=O)cc([N+](=O)[O-])cc(Cl)c1O N1(C(c2cc(CC)oc2C)=O)CC2CN(C(=O)CC3COC(C)(C)C3)CC2C1 C(=O)(CCC(C)(C)NC(=O)C=CC(C)C)NC1(CCOC)CCC1 C1(C(C)C)CN(C(=O)CCC(C)C#N)CCCN1C(=O)C=CC(F)(F)F n1(CC(N2CCC3C(NC(CC4N(CC)CCC4)=O)C32)=O)cccc(N)c1=O N=c1[nH]c(N2CCn3c(cnc3Br)C2)nc2ccc(Br)cc12 C(=O)(CN=c1ccc(C#N)c[nH]1)NCC1C(CNC(c2c(C)cc(C)nc2)=O)C1 C1(NC(c2ccc(C#C)cn2)=O)C(CNC(=O)CC2(O)CCC2)CCC12CCC2 Cc1cc(=NCC2CCCC(F)C2)[nH]cc1S(=O)(=O)NCCCn1cccn1 Cc1cc(F)ncc1C(=O)NC(C)CC(C)NC(C1(CF)CCC1)=O Cc1cc(Br)cc2cc(C(=O)NCC(C)CNC(=O)CC(C)(C)C#N)[nH]c12 CC1Oc2ccc(C(N3CC(CN(C)Cc4ccc(Cl)cc4)C3)=O)cc2NC1=O c1(C(C(=O)NC2(CCNC(C(CC)NC(N)=O)=O)CC2)C)ccc(F)c(F)c1 N1(C(=O)N(C2CCCCC2)CCO)CCCc2c(C(F)(F)F)cccc21 c1(CC(N2CCCCC2CN2CCCC2)=O)cccc2ccncc12 N1(C(=O)Nc2c(-c3n(CC)ncn3)cccc2)CCC2(CC1)CNC(=O)NC2 c1(C(C(N2CCC(O)(CNC(CCCC#N)=O)C2)=O)(F)F)c(F)cccc1F N1(C(CCn2c(C)nc(C)n2)=O)CC(F)(F)CC1CNC(C1CCN(C)C1C)=O c1(CCC(=O)NC(C2CCCN(C(COC)=O)C2)C)cc(OC)ccc1OC C1(CNC(C2(SC)CN(C(C3CC(=C4CCC4)C3)=O)C2)=O)CCCCN1C C1(C(N2CC(c3nc(C)[nH]n3)C2)=O)CN(C(C2CCC(O)CC2)=O)CCO1 c1(C(=O)NC(c2cc(OCC)c(OC)cc2)C)cc2c(C)noc2cc1C C(=O)(C(CC(=O)OC(C)(C)C)N(C)CCNC(N)=O)NCCNC(CCSC)=O S(=O)(=O)(c1c[nH]ccc1=NC(CO)C1CC1)NC1(N(C)C)CCOCC1 c1(CC(=O)N(CC(C(=O)N(c2ccccc2)CC)C)C)ccccc1O c1(CCC(=O)NCCCN(C(c2occc2F)=O)CC)cccc([N+](=O)[O-])c1 C1(NC(C(C(C)(C)C)O)=O)C2COCC1CC(NC(=O)C#CC1CCOCC1)C2 CN1CC(C)(C(=O)NCCCC2CN(C(C3(F)CCCCC3)=O)CCO2)CC1=O C1(N(C(=O)CCc2ccsc2)CC)CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1 Cc1cccc(OCC(C)NC(=O)CNc2ccc(-c3nnc(S)o3)cc2)c1 c1(C(=O)NC2CC(N(C(C(c3cccc(C)c3)C)=O)C)C2)ccc(N)c(C)c1C C1(CNC(C(CSC)C)=O)(NC(c2cn(CCF)nn2)=O)CC2CCC1CC2 c1(C(N2CC(C)C(N(C)C(C3CCC=CCC3)=O)CC2)=O)nccc2n[nH]cc12 C1(C(=O)NC(C2CCN(C(c3nc(C)c(C)[nH]3)=O)CC2)C)CCC(N=[N+]=[N-])C1 C(=O)(C1=NOC(C)C1)NCCN1CCN(C(c2c(C)sc(O)n2)=O)CC1 N1(C(Cc2nc(C)[nH]n2)=O)CCCC(CCCCNC(=O)Cc2cnccn2)C1 C1(O)(CNC(c2n(CC)ncn2)=O)CCN(C(C2(C)CCCC2(F)F)=O)CC1 N1(C(COC(C)C)=O)CCN(C(c2ccc(C(C)(C)C)o2)=O)C(C2CC2)C1 C1(C(NOCCC)=O)CC(C)CCN1C(C1CC=C(C)CC1)=O C12(NC(C3CN4CCC3CC4)=O)CCC(Oc3ccc(OC(F)F)cc3)(CC1)CC2 C(=O)(C#CC1(CC)COC1)NC(CNC(COCCCOC)=O)CC c1(C(=O)NC2CC3CC(NC(C(C(C)C)OC)=O)CC32)ccc(F)c(C)c1C#N N1(C(Cc2scc(C)c2)=O)CCC2(CCN(c3nncs3)C2)C1 N1(C(c2nccc(SC)n2)=O)CC2CC(Nc3cc(O)nc(O)n3)CC1C2 c1(C(=O)NC2C(NC(c3cnn(CC)c3C)=O)COCC2)cc(F)ncc1OC N1(C(C(CC)CC(F)F)=O)CC(NC(=O)COCC(F)F)C2CCCCC12 C(C(=O)NCc1occc1C(N1CCN(C(C)=O)CC1)=O)(C(C)C)OCC Oc1ccnc(C2CCCN2Cc2nc(C3CC3)n[nH]2)n1 C1(NC(CCCN(C)C)=O)CCN(C(c2cnc(Cl)cc2Cl)=O)CCC1CO C1(C(=O)NCCCc2c(C)n[nH]c2)CN(C(=O)CCCC2CC2)CC12CC2 c1(CC)cccc(NC(=O)C(COC)NC(=O)C(O)CC2CCCC2)c1O C1(C(N2CCN(C(CCC3COC(C)(C)O3)=O)CC2)=O)Cc2cscc2C1 O=C(O)C(n1nccc1-c1ccccc1Cl)c1cncc(F)c1 N1(C(C(CC)(C)C)=O)CCN(C2CCN(C)CC2)C(C)C1 O=C1CC(C(N2CCCC2CNC(c2cccnc2C(F)F)=O)=O)CCN1 c1(C(=O)OCC(c2cn(C3CCCN(C(C)=O)C3)nn2)=O)cc(C)ccc1N N1(C(CN(C)CC)=O)CC2CC(NC(C34CCC3CC4)=O)C1C2 c1(C(=O)NC2CN(C(=O)C(C3(O)CCCC3)F)C2)cccc2[nH]nc(O)c12 Cc1cnc(CC(=O)NCC2CC(NC(=O)C=C3CCC(C)C3)C2)o1 c1(CC(c2ccco2)NCC(N2CC(C)C2(C)C)C)ccc(C#N)cc1 Oc1c(CN2CC(CC=CC3CC3)CC23CC3)cccc1F c1(C(=O)NCc2c(C(=O)NC3C(N(C)C)CC3)occ2)ccnnc1O Cc1cc(C(N2CCC(NC(c3ccc(O)nn3)=O)C23CC3)=O)c(O)nn1 CN=c1[nH]c(C(N2CC(N(C(=O)CCCNC(C)=O)C)C(F)C2)=O)cs1 C1(C)(C(=O)NCC2N(C(CC(CN(C)C)O)=O)CCC2)CCC(F)(F)C1 c1(C(=O)NCC2(O)CCCN(C(C(COC)N(C)C)=O)C2)ccn2ccnc2c1 c1(CC(=O)NCCC(C)NC(C2CCO2)=O)c(F)cccc1F C1(CC(=O)N(C2CC2)CC2CCCN2C(c2cc[nH]n2)=O)CCCCO1 c1(C(=O)NCC(CNC(C(CCC)OCC)=O)OC)c[nH]c(=N)c2[nH]ccc12 c1(C(C)NCC(=O)NNC(N2CC(=O)N3CCCC3C2)=O)ccc([N+](=O)[O-])c(O)c1 N1(C(C2CC=C(C)CC2)=O)CCN(C(=O)CC2C=CCC2)CC1CCO CC(C)(C)C(CO)C(=O)NC1C=CC(C(N2CC3OCC(CO)C3C2)=O)C1 CN1CCN(C)C(CNC(=O)C(CC(F)F)N(C)C(C2CCCNC2=O)=O)C1 C1(O)(CN(C)C(C2C3COCC23)=O)CN(C(=O)CC23CCCC2C3)C1 c1(C(N2CCC(N(C(CC(C)SC)=O)C)C2)=O)cc(=O)c2cc(F)ccc2o1 c1(CC)cc(C(=O)N(C(C)C(=O)NCC(C)OC(F)F)C2CC2)n(C)n1 c1(C(=O)NC2(C(N(C(C(=O)OC)C)C3CC3)=O)CC2)ccncn1 c1(OCC)ccc([N+](=O)[O-])c(C(=O)NCC23CCC(CN(C(C)=O)C2)C3)c1 c1(C=O)cc(S(=O)(=O)N2CCCC2)ccc1O.N1(C(COCC)=O)CC(NC)C1 C(=O)(C1=NOC(C)C1)NC1CN(C(C2(CC)CCNC2=O)=O)CC1C N1(C(CC2CC(CC)C2)=O)CC2CCC1CC2NC(c1cnn[nH]1)=O C(=O)(C(C)(C)CCCCC)N1CC(NC(=O)COC2CCC2)CC(OC)C1 N1(C(c2cnn(CC)c2Br)=O)CC2CC(C1)c1cccc(=O)n1C2 c1(C(N2CCC(NC(Cc3cc(C)on3)=O)(CF)C2)=O)ncnc(O)c1Br CC1CC(C(=O)N2CCC(NC(c3c(C(F)(F)F)cnn3C)=O)C2)=NO1 c1(NC(CC(CC)NC(C2COC(=O)N2C)=O)=O)ccc(C)c(O)c1C C(=O)(C1=C(C)CCCC1(C)C)NCC(C(C)(C)C)NC(CC(CC)(C)C)=O c1(C(=O)NCc2ccc(CC)cc2)cc(Br)ccc1NC(c1ccon1)=O n1(CC)nc(C)cc1C(=O)NC1CCCC(NC(C2CC(C(F)(F)F)C2)=O)C1 C1(C(=O)NC(C)CCNC(C2(C)CSC2)=O)CCc2cnn(C)c2C1 c1(CCC(=O)N(CC(CNC(C2C(CCOC)C2)=O)C)C)cccn1C N1(C(=O)CCCC(N2CCC(c3ncc[nH]3)C2)=O)CCC2(C=CCO2)CC1 C(=O)(C(F)CCC(C)C)NCC(CCOC)NC(c1ccncc1N)=O c1(NC)ccc(F)cc1C(=O)NC(C1CCN(C(=O)C(C)CSC)C1)C O(NC(=O)CCN1CCOC1=O)CC(N1CC(N(C)CCO)C1)=O Cc1cc(C(=O)N(C)CC2(O)CCN(C(C3C4COCC34)=O)C2)n(CCO)n1 CCC(COC(c1cc(C)n(-c2ccc(F)cc2)c1C)=O)CC(F)F C1(CC)C(NC(C2CCCC2C(C)C)=O)CCCN1C(=O)C(C)=C(C)C CC12CCOC(C(N3CCC(NC(c4csc(C(F)(F)F)n4)=O)C3)=O)(C1)C2 N1(C(c2cc3cccnn3n2)=O)CCC2CCN(c3ncncc3I)CC2C1 c1(C(N2CCCC(C)(C(=O)Nc3c(C)cc(Cl)nc3)C2)=O)onc2ccccc12 C(=O)(CCCC(C)(F)F)NC(CN(C(C1CC1C)=O)CC)C c1(-c2nc(-c3c(CC)nn(C)c3)on2)cccc2cnccc12 C1(OC)CC2CN(C(C3C(C)(C)C3(F)F)=O)Cc3cccnc3N2C1 C(CCC)(C(=O)N1CCC(C)(NC(c2cc(OC)no2)=O)C1)=CCC C1(O)(CN(C(Cc2c(C)noc2Cl)=O)C)CCCN(C(C2C=CCC2)=O)C1 C(=O)(C(CC(=O)OCC)OC)NC(CNC(C=COCC)=O)CCOC c1(OC)ncc(C(=O)OC)cc1NC1CCCNCC1F c1(N2CC(OC)(CNC(C3CCCC3S(C)(=O)=O)=O)C2)ccc([N+](=O)[O-])c(O)n1 CC(C)C(F)C(=O)N(C)CC1(C)CCCC1NC(=O)CSc1ccc(O)cc1 C(c1ccnn1C)=CC(=O)NC(C1CCOC1)CNC(CCc1scc(C)n1)=O N1(C(c2c(CC)cc[nH]2)=O)CC=CC1(C)C(N1CCCC(COC)C1)=O N1(C(CCCSC)=O)CCC2CCCC12CNC(c1cn(C)c(C)n1)=O c1(CNC(c2cnn(C3CCN(C)C3=O)c2)C)ccc2c(c1)CCS2(=O)=O CCC1=NOC(C(N2CC(CNC(c3ccccc3Br)=O)C2)=O)C1 N1(C(C2CC(CNC(CC(C)O)=O)OC2)=O)CC(CO)CC(C)(C)C1 C1(F)(CNC(c2c(CC)n(CC)nn2)=O)CCN(C(=O)C(F)=CC2CC2)CC1 N1(C(c2cc3nc(C)sc3[nH]2)=O)CC2CC3CC2C1C3NC(C1CCCCO1)=O N1(C(c2nc(OCC)oc2)=O)CCN(C(=O)CC2CC(OC)C2)CC1CC CC1CN(C(=O)CCN2CCN(C)CC2)CCC1NC(=O)C(C1CCC1)C1CC1 C(C)(CO)(C(=O)NC1(c2cccs2)CC1)NC(C(C)c1cc[nH]n1)=O N1(C(CC=CC=C)=O)CC2CC(C1)N(C(=O)C(CN(C)C)N(C)C)C2 N1(CCC(=O)NC(C(C)NC(c2cn(C)c(O)n2)=O)C)CCc2ccccc2C1 C1(NC(C(CN(C(CCCCSC)=O)C)C)=O)C(O)C2CCCC12 C(=O)(CCC(=O)NC1CC(NC(=O)CC(O)C2CCCC2)CC1O)OC(C)(C)C N1(C(CSC)=O)CCC2(CC1)CC2(CO)CNC(=O)Cc1sccc1Cl c1(C(=O)NCCC(C)NC(=O)CP(C)(C)=O)cccc(S(=O)(=O)N2CCCC2)c1 c1(OC)c(C)cc(C(=O)NCC#CCNC(=O)CNC=O)cc1C C1(NC(CC2C(C)CCC2)=O)CN(C(=O)CN(C2CC2)CC2CC2)CCC1(C)C c1(C(=O)OC(c2nc3ccccc3o2)C)n[nH]c2c(=O)n(C)cnc12 C1(CC(=O)NCC(C)CNC(C2CC(N(C)C)C2)=O)CCC2(CCC2)O1 c1(C(=O)NC2CCCN(C(CC3OCC(C)(C)OC3)=O)C2)ccnc2c1CCO2 c1(CN(C)Cc2cccc(C)c2)cc(Cl)c(Cl)n1C c1(N(N2CCC2c2cn(CC(=O)O)nn2)C)cnn2c1OCC(C)(C)C2.C=O Cn1cc(NC(=O)CC2CC(NC34CC(C3)C4)C2)c(OCCN(C)C)n1 C(CN=c1[nH]c2ccc(O)cc2s1)Oc1c(NC(c2cccc(=S)n2O)=O)cccc1 N1(C(=O)Nc2ccnn(CC)c2=O)CCC(C)C2(CCC2)C1 c1(C(CNC(C(C)SCCCC)=O)NC(=O)CCOC)ccccc1F C(=O)(C(C)(C)C1=CCN(C(C2CC2C(F)F)=O)C1)NCc1c(C)cn(C)n1 C1(NC(C2CC(C(C)C)C2)=O)C2CC(NC(=O)C(F)(F)CO)CC12 C1(NC(c2nc(CC)oc2)=O)CCN(C(c2cnc(C3CC3)s2)=O)C(C2CC2)C1 C1(NC(C2(CC#C)CC2)=O)CC(CNC(c2cnsc2)=O)C1 c1(C(N2CCC(C)(NC(c3cc(C)n(C(C)C)n3)=O)C2)=O)ncnc2ccsc12 C1(C)(CC)CN(C(C2CC(N(C)C(c3cncs3)=O)C2)=O)CCO1 C(=O)(CC1C(=O)Nc2ccccc21)NC(C)CNC(C1CCCS1)=O C1(C(=O)NC2(C(=O)NCC3CCN3C(C)(C)C)C(C)C2)CN(C)CCN1C Cc1oc(-c2ccccc2)nc1CC(=O)NCC1(O)CN(C(C2CC2C)=O)C1 c1(OCCOC)cncc(C(=O)NCC(C)(O)CNC(=O)CC2(C3CC3)CC2)c1 c1(CN(C(C2(OCC)CCS(=O)(=O)C2)=O)C)cnn2c1CN(c1nncs1)CC2 c1(NC(C(F)=C(C)C)=O)cccc(NC(=O)C(F)Cc2ccccc2)c1 c1(C(=O)NCC2N(C(C3C(C=C)CC3)=O)CCC(C)C2)cc(=O)c(OC)cn1C c1(C(c2n(CCCCCC)nnn2)NCc2cnoc2)c(C)nn(C(F)F)c1C N1(C(C(C)OCCOC)=O)CCC(C(C)C(=O)NC(C)C(=O)OC(C)C)CC1 c1(C(=O)NCC(CC(C)C)NC(=O)CCc2ccn(C)c2)cc(Cl)nnc1Cl c1(N(C)CC2(C)CCCC2)ccncc1S(=O)(=O)N1CCOC(C(C)(C)C)CC1 c1(C(=O)NC(C2CCCN(Cc3cccc(C#N)n3)C2)C)ccc(F)c(Cl)c1F c1(OCC(N2CCC(CCNC(COCCCC)=O)C2)=O)ccc(OC)cc1 N1(C(C(CC)OCC)=O)CC(C(=O)NCCOC(C)C)(CC)C1 c1(CC(C)NC(c2ccc(C)o2)=O)ccc(CNC(c2cnc[nH]2)=O)cc1 N1(C(C2C(NC(c3ccncc3Cl)=O)CCO2)=O)CCOC2CCCC12 C1(COC)(CNC(C2CNC(=O)N2)=O)CCCN1C(=O)CCc1ccccc1 N1(C(C(C)NS(C)(=O)=O)=O)CCOC(CNC(c2cc(CC3CCC3)c[nH]2)=O)C1 Cc1cc(F)ccc1N(C)C(=O)N(C1CC1)CC1(c2ccc(Br)cc2)CCCC1 C1(OC)COCCC1CC(=O)NCCN(C(c1coc(C2CCCC2)n1)=O)CC C1(C(=O)NC2(CCCNC(=O)CSc3nncs3)CC2)CC12CCCCC2 CC1CCN(C(C2CC(=O)CN2C(c2cnnc(O)c2)=O)=O)C1(C)C C1(CNC(c2c(C)nc(CCC)s2)=O)CN(C(C2CCCCO2)=O)CCN1C c1(OC)ccc(N)c(C(N2CC(CNC(C3(C)CC=CCO3)=O)CC2(C)C)=O)c1 C1(NC(C2(OCC)CCCC2)=O)CCN(C(c2c(C)[nH]c(C)c2C)=O)CC1CC N1(C(CCCC(=O)NCC)=O)CCC(C2(NC(c3nnc(CC)s3)=O)CC2)C1 Cc1cc(=NC(CC2CC2)C2CC2)[nH]c(=NCc2nc(C)c(C)s2)[nH]1 C1(C)(C(=O)NC(C2CC2C(=O)NCCC#CCO)C)CCCCC1C c1(OCC(=O)NCC(C)CNC(=O)CC2(C(F)F)CC2)ccc(Br)cc1 CC1(C)COC(CC(N2CC(OCCNC(c3cncc(Cl)c3)=O)C2)=O)CO1 N1(C(=O)CNc2ccccn2)CCOC(CCNC(C2CC(CF)C2)=O)C1 C1(NC(=O)C(C2CCCO2)C2CC2)CC2CN(C(=O)C=C3CCCCC3)CC12 c1(CC(C)C(=O)NCCC2CCCC(C(C)(C)C)C2)ccc(-c2nn[nH]n2)cc1 c1(C(N(CCC(=O)NC2CCC2C)CC=C)=O)cn(C)c(C)n1 C(=O)(C#CC1CCCO1)NC1CCCCN(C(Cn2ncc(CC)c2)=O)C1 N1(C(C=CCC2(NC(=O)CC3C=CCC3)CC2)=O)CCC(F)(F)C(F)C1 CN1C(=O)CCC1C(=O)NCC(C1CCCN1c1nc(C(C)(C)C)ns1)(C)C C1(SCc2cn(CC(=O)NCc3ccc(C(=O)OC)s3)nn2)CCOC(C)(C)C1 N1(C(C2C(CC)OCC2)=O)CC2(CC(CNC(c3ccc(F)cc3SC)=O)C2)C1 C1(C(=O)NC2CC(C(C)O)C2)CC2(CCN1C(c1cncc(Cl)c1)=O)CC2 c1(C(=O)OCc2cccc(SCC)c2)ccc(Cl)c(Br)c1 c1(SCC(=O)NCc2csc(CNC(C3CCC(F)C3)=O)n2)ccc(F)cc1 c1(C(=O)NC2(C)CC(NC(=O)C#CC3CC3)C2)cn(Cc2ccccc2)[nH]c1=N N1(C(c2ccc(OC)o2)=O)CCC2(CC1)CC2C(=O)NC1(CO)CC(OC)C1 C(=O)(CCCCC(=O)NC)NCC1N(C(C2(C)C(CC)CCC2)=O)CCCC1 c1(CC)ccc(C(=O)NCC23CC2CN(C(=O)CC(C)n2ccc(C)n2)C3)cn1 CC(C)C(C(C)NC(c1cccc(N2CC=CC2)c1)=O)NC(=O)COC(F)F N1(C(C(F)=CC)=O)CCN(C(=O)C=Cc2cnc(OC)nc2)C(CO)C1 c1(OC)cc(C(N2CCC(C)(NC(c3ccccc3F)=O)CC2)=O)cc(F)c1F O=C(C1=NOC(C2CCC2)C1)N1C(CNC(c2ncoc2C2CCC2)=O)CC1 c1(C(=O)OCC2CN(CC)C(=O)O2)cc(F)cc2nccnc12 c1(C(N2CCC(NC(C=C(C)C3CC3)=O)C2)=O)ccncc1-n1cccn1 c1(C(C)CC(N2CC3CC2C3NC(C2CCN(C)C2)=O)=O)ccc(F)cc1F C1(C(=O)NC2(C(=O)NCCc3cccnc3F)CCC2)Cc2nccn2C1 n1(CC(N2CCC(NC(C3CC=C(C)CC3)=O)C2)=O)cc(C)c2ccccc12 C1(CNC(CCCCOC)=O)(NC(=O)C(C)c2cccs2)CC2CCC1CC2 CC1CC(CNC(C2(F)CCOCC2)=O)CN(C(C23CC(C)(CCO2)C3)=O)C1 C(C1=CCCN(C)C1)NC(C1(CNC(C(CSC)OC)=O)CCC1)=O N1(C(c2ncc(C)cc2F)=O)CC(C(N2CCCC2C(C)(C)C)=O)CCC1(C)C CCCCC(CNC(c1csc(COC)n1)=O)NC(c1ccccc1Cl)=O N1(C(C2CC(C#C)(O)C2)=O)CC(NC(=O)C=Cc2cnn(C)c2)CCC1C CC1(C)CNCCN1C(=O)C(=O)Nc1ccccc1N1CCNC1=O N1(C(c2c(OC)c(C)sc2)=O)CC2CCN(C(=O)C(c3cnn(C)c3)O)CC2C1 N1(C(C=C(CC)C)=O)CC(CNC(=O)COc2ccc(Cl)cc2F)C2(CC2)C1 S(=O)(=O)(c1cc(C)cnc1N(CCC(=O)N(C)C)C)N(CC(CC)(C)C(C)O)C C(CC(C)(C)C(=O)NCCc1cc(C(=O)NCC2(CCO)CCC2)no1)OC c1(C(N2CC(CN(C(C3(CCC)CC3)=O)C)OCC2)=O)cc(OC)ncc1F c1(C(N2C(C3(C(=O)OCC)CC3)CCCC2)=O)cc2cc(Cl)ccc2o1 C1(C(c2cn(-c3c(SC)cccc3)nn2)O)C(O)C(O)CN1N1CCCC1 CC(C)(C)C#CC(=O)NCC1(F)CCN(C(=O)CSc2ccccc2)C1 N1(C(C(C)OCCC#C)=O)CCCC(n2cc(CNC(=O)CCC3CC3)nn2)C1 n1(CC(=O)NCC(C)CN(C(=O)CC2CCCCN2C)C)ccc(=O)n(C)c1=O N1(C(C2CC(CC)C2)C(=O)NC(C)(C)C)CCc2ncc(C)n2CC1 C1(NC(C(n2cc(Cl)cn2)C)=O)CCN(C(=O)C#CC2(C(F)(F)F)CC2)CC1C c1(CCCC(=O)NC2C(NC(C(CC)=CC)=O)COCC2)c[nH]c2ccccc12 C12(C(=O)NC(CCNC(c3cc(COC)cn3C)=O)(C)C)CC(C)(C1)OC2C c1(NC2CCCCN(C(C(C=C)(C)O)=O)C2)ncc(S(C)(=O)=O)cc1Cl N1(C(C2C(C(=O)OC)C2)=O)CCN(C(C23CCC(CO)(CC2)C3)=O)CC1C1CC1 C1(C)(CNC(c2n(C)nnc2)=O)CN(C(=O)CN2CCCCC2)C(C)(C)C1 C1(C(=O)NC(CN(C(c2cnsn2)=O)CC)C)CCCN(c2cnccn2)C1 C1(C(=O)NCC2(CNC(=O)COc3cccc(Cl)c3)CC2)Cc2ccccc2S1 Brc1ccc2nc(NCCCc3c[nH]c4cnccc34)nn2c1 C1(NC(CCC)=O)CN(C(=O)C(O)Cc2c(F)cccc2Cl)CC(C)(C)C1 c1(C(=O)NC(C)CN(C(=O)CCn2cnccc2=O)C)cc2c(s1)CCCC2 Cc1c(C(=O)NCC2CCN2C(=O)C2=CS(=O)CCC2)cccc1C#N c1(C(C(=O)NCC2CCCN2C(C2COC2)=O)O)ccc(Cl)cc1 c1(C(=O)NCC#CCNC(CC(=C)Br)=O)c(C)noc1C(F)F c1(C(=O)NCCO)cnc2n1CCCC2.c1(CN2C(C)CC2)ccc(C)cc1F C1(SC(C(=O)NCCCC)CC)CNCC1(C)C CC1(C)CC(=O)NCC1C(N1CCN(C(c2c[nH]nc2F)=O)CC1CC(F)F)=O c1(C(C)(C)C)ccc(C(=O)NC2CCC2NC(c2ccccc2)=O)[nH]1 c1(C(N(C2CC(NC(C(C(C)O)NC(N)=O)=O)C2)C)=O)ccc2cnccc2c1 CC1CC=C(C(=O)N2CC(C(=O)NC3CC(C(F)(F)F)C3)C(F)C2)CC1 c1(CCC(=O)NCC2CCN(C(COCC(=C)C)=O)C2)ccc(C(=O)OC)cc1 N1(c2ccnc(C)n2)CCN(C2CCCN(C(c3cnoc3C)=O)C2)C(=O)C1 N1(C(c2c(CC)ccc(Br)c2)=O)CCCN(C(=O)C(O)C(C)C)CCC1 N1(C(CC)=O)C(CNC(=O)C(F)(F)c2ccncc2)CC2CCCCC12 C(CC(N=c1[nH]c(Cl)nc2ccccc12)C(C)C)N(C(c1c(C)nc[nH]1)=O)C Cc1cc(CNC(=O)C(CO)NC(C2CCCN2C)=O)nn1C C1(CC)CCCC1(C)C(N1CC(C(C)NC(c2cnc(C(F)(F)F)nc2)=O)C1)=O C#CC1(C(=O)N(CC(C)C(=O)NCC2(CC)CCOC2)C)CCCC1 C1(NC(c2n(CCCC)ncc2)=O)CC(CNC(c2ccc(CC)o2)=O)C(O)C1 c1(C(=O)NCC=CCNC(Cc2nc(C)sc2C)=O)ccnc(O)c1Br C(=O)(N=c1nc(C2CC2)s[nH]1)c1ccc(CSc2cccc(C(C)(C)C)c2)o1 C1(NC(C=Cc2nc(C)sc2)=O)CCC12CCN(C(C1CC1(C)C)=O)CC2 C1(C(=O)NCC(C)(C)OCCNC(COCCCCC)=O)NC(=O)C2CC12 C1(C(N(CCN(C(C(C)=CC)=O)C)C)=O)CCN(C2CCS(=O)(=O)C2)CC1 c1(C(N2CCC(C)(NC(c3cc(Br)no3)=O)C2)=O)ccc(C2CC2)c(F)c1 N1(C(C(C)(C)OCC)=O)C2CCC1CN(C(c1oc(C)nc1CC)=O)C2 CC1(C)COCC(C(=O)NC(CNC(c2sccc2F)=O)CO)O1 c1(C(=O)NCC(C)NC(C2CS(=O)(=O)CCO2)=O)coc2ccc(Cl)cc12 C=CCCC(CC(C)C)C(=O)NC1(CNC(c2cscc2OC)=O)CC(F)(F)C1 c1(OC)ccnc(C(=O)N(C2CN(C(c3cc(C4CC4)ns3)=O)CC2F)C)c1 C1(CNC(c2[nH]c(C)c(C)c2C)=O)CC2(CCN(C(C3CCC4CC34)=O)C2)CO1 Cc1ccc(Cl)c(OC(C)C(=O)NCCCNC(c2csc(S)n2)=O)c1 C=CC1CCN(C(=O)COCCNC(C2CCCOC2)=O)CC1 N1(CC(=O)NCC2N(C(C(C)=CC3CC3)=O)CC=C2)CCCCC(O)C1=O Cc1c(C(N2CCC(NC(=O)CC3CCCC3)C3CC23)=O)cncc1Br C1(C(N2CCC(C3COC(=O)N3)CC2)C(=O)NC(C)C)CC2OC(C)(C)OC2C1 c1(C(=O)OC)cnn2c1CN(C(=O)NC1CN(c3ccc(O)cc3Cl)C1)CC2 c1(CC)[nH]ccc1C(N1CC(O)(C2CCCN2C(C2CNC(=O)C2)=O)C1)=O c1(CC(=O)NCC(CC)(C)NC(=O)C(F)C(F)(F)F)ccc(C)cc1C CN1CCN(C(=O)CC2(C(F)(F)F)CC2)C(CNC(=O)CN2CCOC2=O)C1 Cc1coc(C=CC(=O)NCC(O)CCNC(=O)CCCn2ccnn2)n1 C1(COC)(NC(c2ncccc2Cl)=O)CCN(C(c2c(C)cnn2C(C)C)=O)C1 c1(CNC(C23CC(NCc4c(C)cccc4O)(C2)C3)=O)ccc2c(c1)OCO2 CCCCCC(C(=O)NCC1CCOCC1)N(CC)Cc1ccsc1 N1(C(COCCCCC)=O)CC(NC(=O)C=CCO)CC12CCCCCC2 N1(C(C(CC(=C)C)OC)=O)CCC2(CCCC2NC(c2nc(Cl)cs2)=O)CC1 Cc1cccc2oc(C(=O)N(C3CCN(CC(C)CC(C)C)C3)C)cc12 C1(CNC(C(CC)Oc2ccccc2Cl)=O)(CO)CCCN(C(=O)CC(C)C)C1 S(=O)(=O)(c1ccccc1Br)Nc1c(C(=O)NC(C(=O)OC)C(C)O)scc1 Cc1nn(C)c(F)c1C(N1CC(NC(=O)C(C)C(F)(F)F)C(C)C1)=O C12(CNC(C(C)(C)F)=O)CN(C(=O)Cn3ccccc3=O)CC1CCO2 N1(C(c2cc(OC)ns2)=O)CCC(CF)(NC(=O)COC2CCN(C)CC2)C1 N1(C(C(C)O)=O)CC2CC(NC(=O)COc3ccc(F)cc3Br)CC(C2)C1 Cc1ccc(COC(C)C(=O)NCCN(C(c2nc(C)oc2C)=O)C2CC2)cc1 C(=O)(CC1=CCN(C(=O)CCc2ccc(C)o2)CC1)NC(CNC(=O)OC)C C1(C(N(CC(=O)NC(c2c(C)ncs2)C)CC(C)C)=O)CCCCC(=O)N1 c1(C(=O)NC(C(=O)OC)Cc2ccc(Br)cc2)cc(F)c(C(F)(F)F)cc1I S(=O)(=O)(c1cccc(=NCCn2cncn2)[nH]1)N1C(CNC(N)=O)CCC1 c1(CCC(=O)NCC(CNC(C2(O)CCOC2)=O)OC)cscc1Br CCC(O)(CNC(=O)C(C)N(C(c1cnn(C)c1OC)=O)C1CC1)CC N1(C(c2ccc(COC)o2)=O)CC(NC(=O)CC2CCOCC2)C(C)C1 c1(C(N(CCCN(c2ncnc3c2COC3)C)C)=O)cc(F)cc2nccnc12 S(=O)(=O)(c1cnccc1N1CCC2(C1)OCCO2)NCc1ncc(C)nc1 Cc1nc(CC2CC2)sc1C(=O)NCCC(C)(C)NC(=O)C(=O)NC(C)C C1(NC(C2CC(C(C)=O)C2(C)C)=O)CN(C(=O)C=C2CCN(C)C2)CC1(C)C C(=O)(C(COC(C)C)NC(=O)CN(C(=O)CC(C)n1cccn1)C)OC C1(CNC(c2scc(OC)c2)=O)CN(C(C2(C)CC2(Cl)Cl)=O)CCO1 C(C(=O)N=c1ccn(CCO)[nH]1)(C1CC=CCC1)NC(CC1CCC(=O)CC1)=O N1(C(C2OCCN(C(C(C)(C)N=[N+]=[N-])=O)C2)=O)CC2(CCCCCC2)C1 CC(C)C(CNC(=O)C(c1ccccc1)=O)NC(C1(OC(C)=O)CC1)=O c1(OCC(=O)N(CCCN(C(C2(C)C(C)CCC2)=O)C)C)cccc(C#N)c1 N1(C(c2cc(CCC)[nH]n2)=O)CCN(C)C(C(=O)NC2CC=CCC2)C1 C1(NC(C(C)c2ccco2)=O)(CF)CCN(C(=O)CC2C=CS(=O)(=O)C2)C1 C1(NC(c2cccc(C(N)=O)c2N)=O)CC2CCC1N(C(=O)CSC1CC1)C2 c1(C(=O)NCC2CCC(NC(C(C(C)C)N(C)C)=O)C2)ccc(=O)n(O)c1 C1(NC(C2C(C(C)C)OCC2)=O)CC=CCC1C(N1CCCCC1CCO)=O C(C(C)C(C)C(=O)NCC1=CCN(C(c2cc(O)nc(OC)n2)=O)CC1)OC N1(OS(c2c(C)sc(Br)n2)(=O)=O)CCC2(CC1)C(O)CC(C(=O)O)C2 C1(NC(C2(CC=C)CC2)=O)CCC(C)(NC(c2cc(C)nn2CCC)=O)CC1 Cc1ccc(N2CC(C(=O)NCC3CCN(C)C3)CCC2=O)cc1C C(=O)(C(O)CCCCC)N1CCC(=C)CC1C(N1CC(C)CC(O)C1)=O N1(C(C(F)=CCC)=O)CC(C)(C)OCC1CNC(c1cc(F)ccc1OC)=O N1(C(C(C)CC(N)=O)=O)CC(NC(=O)C(C)N2CCCC2)CC12CCCCC2 CC1CN(C(C2(F)CCN(C)CC2)=O)CCC1CO O=C(CCCC(F)C(=O)O)N1CCC(O)(c2ccccc2)C(O)C1 c1(C(N)=O)cccc2c1CN(C(C1CCN(C(C3CCC(=O)N3)=O)CC1)=O)C2 CCC(C)CC(C)C(=O)N1CCC(C)(C)C(c2cn(-c3cc(C)ccc3F)nn2)C1 C1(CNC(C(C)O)=O)CCC2(CN(C(c3ccc(F)cc3O)=O)C2)O1 C12(NC(C#CC3(C)CC3)=O)CCOCC1CN(C(c1ccns1)=O)C2 c1(C(=O)NCC(CCNC(CN(C2CC2)CC)=O)O)nc(O)nc(O)c1OC N1(C(C(N)=O)=O)CC2(CCN(C(=O)Nc3ccc(Cl)c(NS(C)(=O)=O)c3)C2)C1 N1(C(C2(C)CC2C(F)(F)F)=O)CCCC1(C)CNC(=O)CCC1CCCOC1 C1(NC(Cc2n(C(C)C)cnn2)=O)CCOC2(C1)CC(C(=O)O)C2 c1(C(=O)NC2(C)CC(NC(C(COC)OC)=O)C2)ccccc1-c1cnn(C)c1 C1(CNC(C(C)NC(C)=O)=O)CN(C(C2CC2C2(C)COC2)=O)CCC12CCC2 C1(C2(O)CCOCC2)(C(N2C3CCC(NC(CC(C(C)C)O)=O)(CC3)C2)=O)CC1 c1(CCNCc2cnn(C)c2Cl)c[nH]c2ncccc12.N12CC3CC1C3C2=O c1(COC)csc(C(=O)NCC(C)(O)CSC)c1.C1(C2CC2)C(=O)N1 c1(C(=O)NC(CNC(c2c(CC)n(C)nc2)=O)CO)ccn2c(C)ncc2c1 N1(c2nccc(N3CCC(N(C)CC)C3)n2)CCOC2(COC(C)(C)C2)C1 c1(N2CC3C(C)C3C2)cc(Br)ccc1S(=O)(=O)NCc1nc2ccc(Cl)cc2s1 CC1(C)CN(C(=O)Cc2cncnc2)CC(C)(C)C1NC(=O)CCCCC(F)F CCC(COC)C(=O)NCC(CC(=O)NC(C)(CO)CO)C1CCC1 N1(CC(CCC)=O)CCOC2(CCSCC2)CC1 CCS(=O)(=O)NC(C)C(=O)N(CC(C)(C)NC(=O)C(C)c1ccco1)C C1(NC(c2n(CC)nc(C(C)C)c2)=O)CCCN(C(=O)C2=CCCO2)CC1 CC(C)(C)CCC(F)C(=O)N1CCCC1C1(NC(=O)CCCF)CC1 c1(CC)nn(C)c(CC)c1NC(=O)Nc1cccc(-n2cc(C#N)cn2)c1 C(C1CCOc2ccc(Br)cc21)NC(c1n[nH]c(C)c1F)=O c1(C(=O)NCC(C)(CO)NC(C2CC3CC3C2)=O)nc2n(c1Cl)CCCC2 C12(CNC(C(CC)(C)C)=O)CN(C(c3sccc3S(N)(=O)=O)=O)CC1CCO2 Cc1cc(C)c(C(=O)NCC(C)C(F)C(=O)NCCCN2CCOCC2)cn1 N1(C(C(C)CSc2ccccc2)=O)CC2(CC(NC(=O)COc3ccsn3)C2)C1 C1(NC(CCCOCC)=O)CC(NC(c2cnn3c2CCC3)=O)C12CCC2 C1(N(C(C2C(=C)C2)=O)CC)CCN(C(=O)C=Cc2ncc[nH]2)CC1 N1(C(c2c(COC)cco2)=O)CCN(C(C2(CC(F)F)CCC2)=O)CC1C(C)C CC1CC(F)(F)CN1C(C1CSCCN1C(=O)C=CC(F)F)=O Cc1cc(C(=O)NCC2CN(C(C3Cc4nccn4C3)=O)CC2O)c(C)cc1Cl c1(OC)cc(C(=O)OC2CN(C(C)=O)C2)cc([N+](=O)[O-])c1OCCF C1(C(N2CCN(C(CC3C(=O)NCCC3)=O)C(CO)C2)=O)CC2CC1CC2(F)F C1(COC)(NC(=O)CCF)CCN(C(=O)CC(O)CNC(=O)OC(C)(C)C)CC1 c1(C(=O)NC(CCNC(CCC2C(C)C2)=O)c2cccs2)cc2cn[nH]c2cn1 CCC(C(=O)N1CCC(NC(=O)Cc2sc(C3CCC3)nc2C)C1)C(C)(C)CC c1(C(=O)NC2CCCC2C(N2CCS(=O)CC2)=O)cc(O)nc(O)c1 C12(CC)COC(C(=O)NCC3CCCC3NC(c3cn(C)nc3OC)=O)(C1)C2 C(=O)(CCCCCNC(C1CC2COCC2C1)=O)N(CC(COC)(C)C)C N1(C(C2C(c3ccc(C#C)cc3)C2)=O)CCN(C(=O)CSC(F)F)C2(CCC2)C1 CC(C)(F)CCC(=O)NC1CCOC(C(N2CCC3C(O)CC23)=O)C1 CC(C)CCCCC(C(=O)O)NS(=O)(=O)c1ccc(Br)cc1NC(C1CCC1)C c1(C(=O)NCC2CN(C(CCc3onc(C)n3)=O)C2)cc(F)cnc1Cl C1(N2C(C(=O)NC(C3CC3(C)C)C)CCC2)CCN(CCc2ccsc2)CC1 C1(CC)CN(C(=O)C=Cc2cccc(CO)c2)CCC1NC(c1ccc(C)[nH]1)=O C12(NC(C(CC)OC)=O)COC(CNC(c3c[nH]nc3-c3ccncc3)=O)(C1)C2 N1(C(C(CC)CO)=O)CC(NC(C2CCOC2C)=O)CC12CCOCC2 C1(C)(C(N(C(C#C)C2CCC2)C)=O)C=CCN1C(C1OCCC1(C)C)=O C1(C(=O)NC(CNC(c2cnn(CC)c2C)=O)C2CC2)CN(CP(C)(C)=O)C1 C1(NC(C2C(C(C)NC(C(C)=CC=C)=O)C2)=O)C(O)CC1O CCCCCC(=O)N1CCN(CC(C)(C)NC(C2(CCOCC)CCC2)=O)CC1 c1(CNC(CC)Cc2ccc(Cl)cc2)cnn2c1C(=O)N(C)CC2 C1(CC(=O)NC2CCC(C)(CNC(c3cnc(SC)s3)=O)C2)CCC2(CCC2)O1 C(CC(=O)NC(c1cccs1)C)N(C(=O)CN1CCCC1)CC#C C(CC(C)(C)CC(=O)NC(C(=O)Nc1cc(C)cnc1O)C1CCC1)OC Cc1cnc2[nH]cc(CNCC3(NC(=O)OC(C)(C)C)CC3)c2c1 CC1CN(C(=O)CC23CCCC2C3)CC1(C)C(=O)NCC12CC=CC(C1)OC2 C1(CC)(CC)CC(O)CN1C(=O)CC(O)CNC(=O)CCN(C)CCO Cc1cnncc1C(=O)NCCC1CSCCN1C(c1cc(Cl)ccn1)=O C1(C(=O)NC(CNC(c2c(CC)nc(C)o2)=O)CO)CC2(CO1)CC(F)(F)C2 n1(CC(=O)NCC2CN(C(c3cc(CC)no3)=O)C(C)C2)c([N+](=O)[O-])cnc1C Cc1c(C(=O)Nc2cccc(CCC(=O)Nn3cnnc3)c2)oc2cc(Cl)ccc12 c1(C(=O)NCCCCCN(C)C)ccccc1-n1cc(-c2cccc(Br)c2)nn1 C1(C)(C(=O)NCC#CC(=O)NCCCCOC(C)C)CCCOC1 C1(=O)C(CCC2CC2)N1.C1(C(=O)NCCSCC)(N(C)C)CCC1 N1(C(c2nc(OCC)sn2)=O)CCC(NC(=O)CC(C)(C)O)CC1C N1(C(CCC2C(C)C2)=O)CCC(O)(CNC(c2cnc(C3CC3)[nH]2)=O)C1 CC(F)(F)C(F)C(=O)NCC1(C)CCCN(C(=O)CCS(C)(=O)=O)C1 N1(C(C(C2CCC2)OCC)=O)CC2COCC2(C(=O)NCC)C1.C(CN(C)C)N c1(C(=O)NCCCOCCNC(c2ncc(F)cn2)=O)cc([N+](=O)[O-])cnc1O N1(C(c2c(N)ccc(C)c2)=O)CCCC2(CC(NC(C3CC(Cl)(Cl)C3)=O)CO2)C1 c1(N(C)C(=O)OC(C)(C)C)ccc(C(=O)Nc2ccn(C3CCCC3)n2)cc1I C12(NC(CC(C)C3CC3)=O)CCC(CNC(=O)Cc3cc(C4CC4)no3)(C1)OC2 C(=O)(CC(C)CC(=O)NC(C)C(C)NC(C1(NC(C)=O)CCC1)=O)OC CCC(C)C(O)CC(=O)NCC1(O)CCN(C(c2cnn(CC)c2C)=O)CC1 S(=O)(=O)(c1ccc(NC(C)C)c(C#N)c1)N1CC(C)CC(NCCC(=O)NC)C1 N1(C(C(C(CC)C)N(C)C(c2cnn(C)c2)=O)=O)CCCN(CC)C(=O)C1 Cc1cc(C(F)(F)F)nc(C(=O)NC2CCC(NC(C3CC=CCC3)=O)CC2)n1 C1(C2CN(C(C3CCCSC3)=O)C2)(Nc2cc(OCC)ncn2)CC1 N1(C(Cc2cn(C)nc2)=O)CCC12CN(C(C1(C)CCCCCC1)=O)C2 c1(C(N2CC3CC(NC(C(=O)NC4CC4)=O)C3C2)=O)cnc2c(c1)CCCC2 C1(OC)CCCN(C(=NCCC(=O)Nc2cc(O)ncn2)NC2CCCC2)C1 CC(CC(N)=O)C(=O)N(C1CCCN(C(c2ccc(N)cc2)=O)C1)CC1CC1 c1(SCC(=O)NCC2OCCCN(Cc3cn(C)nc3)C2)ccc2[nH]ccc2c1 C1(NC(c2cccc(C)n2)=O)CCN(C(C2CCC(C)C(C)C2)=O)CC1C CC(C(F)C(=O)NCCC(C)NC(=O)C1=CN=C2N=CNN2C1)C(F)(F)F c1(C(=O)NCC(N2CC(O)(C(C)NC(c3csnn3)=O)C2)=O)ccc(Cl)cc1 c1(C(N2CCC(C)C2CNC(=O)COC(F)F)=O)cc(O)cc(Br)c1 C=CCC(C(=O)N1CCC(NC(c2c(C)csc2Cl)=O)CC1C)C(C)C c1(C(=O)NC(C)C(=O)N(C2CCCN(C(N)=O)C2)CCO)cccc(O)c1F c1(C(N2CCC(N(C(C=C(CC)CC)=O)C)C2)=O)ccc(O)c(NC(C)=O)c1 N1(C(CC(C)OC)=O)CCC(C(=O)NCc2[nH]cnc2C)(C(C)C)C1 c1(CC)n[nH]cc1C(N1CC(C(C(=O)NCC(=O)NC)OC)C1)=O S(=O)(=O)(c1c(C#N)cnn1C)N1CCC(CC(C)O)CC1 c1(C(=O)NCC2N(C(C3(C=C)CC3)=O)CCCC2)ccc(Cl)c(OC)c1 C(=O)(C(C(C)CC)N(C)C(C1CCCN1C(N)=O)=O)N(CCOCC=C)C c1(CN2CCC(CC(N3C(C(=O)OCC)CCCC3)=O)CC2)ccnc(Cl)c1Br N1(C(c2ccc(CC)c(N)c2)=O)CCC(C2CC2)C1CNC(=O)C=CCOC C1(CC(=O)NCC(c2ccc(F)cc2)OC)CN(C(C2CCCC2)=O)CCO1 Cc1cc(C(=O)NCC(C2CC2)NC(=O)C(C)(F)c2ccon2)c(F)cc1N Cc1c(C(=O)NCC=CCNC(=O)C#CC(=O)N(C)C)noc1C1CC1 c1(CC(=O)NC(C(C)NC(C2(CC)CCC2)=O)C(C)C)cc(C(C)=O)ccc1N CCCC(CCC)C(=O)NCCC(C)NC(c1cc(Cl)nc(Cl)c1)=O c1(C(=O)NCC(O)COc2cccc(Br)c2)cnn2c1SCC2 CCC(C(=O)NC(C)(C)CC(=O)NC(C)C(=O)OC)C(C)C C1(C(=O)NCCc2ncc(C)o2)N(C(=O)Cc2cnoc2)CCCC1(C)C CC1CN(C(=O)C(C)C(C)O)CC(C)N(C(=O)C(=CC2CCOCC2)Br)C1 C1(C(N2CC(CC)(CC)C2)=O)CC2C=CC1N(C(=O)CCCCOC)C2 C(CNC1CCCC1)(C(C)C)N(C(=O)C(=O)Nc1ncc(CC)s1)CCC C12(CO)CCCN(C1)C(=O)OC2.C1CCCN(C)CC1.C(C)(C)(C)OC c1(C(N2CCCCC(NC(CCCC=C)=O)CC2)=O)oc2ccc(F)cc2c1C C(=O)(C1=NOC2COCC12)NC(C(C)NC(c1ncnc(OC)c1F)=O)CO c1(C(=O)NCC2C=CCN2C(=O)CCC2CC2(F)F)ccc2ccoc2c1 C1(C(=O)NCC#CCNC(c2cnc(C(=O)OC)s2)=O)Cc2nn[nH]c2C(C)C1 Cc1ccc2cc(C(=O)N(C3CCC(NC(=O)C(C(C)C)C(C)C)C3)C)[nH]c2c1 C1(C(N2CCC(C3N(C(=O)Cc4ccco4)CCC3)C2)=O)(CO)CCCCC1 C(=O)(C(=O)N=S(C)(C)=O)NC1C(SC)CN(C(=O)C2=NOC(C)C2)C1 N1(C(CCCOCCC)=O)CC(CNC(c2oc(C3CC3)nc2C)=O)CC1C CC1CC2CCC(C1)N2C(CCc1ccco1)C(=O)NC1CC(F)(F)C1 C1(C(=O)NCC2(CN(C(c3nncc(OC)c3)=O)C)CC2)CN2CCN1CC2C c1(-c2nn(C(CC)CC)c(CSc3[nH]cnc3C)n2)ccc(N(C)C)cc1F C1(C(=O)NCCCCNC(c2cnc(CC3CC3)s2)=O)CC1C1CCCCC1 Cc1cc(F)cc(C)c1C(N1CCC(CF)(NC(C2CC(=O)N(O)C2)=O)C1)=O c1(OC)ccc(Cl)cc1CC(=O)NCC12CC(CN1C(C1(C)CNC(=O)C1)=O)C2 CN1CC(C)(C)CC1C(N1CCCC1C(C)(C)NC(c1cc2c[nH]nc2s1)=O)=O C1(C(=O)NC(C(=O)NCCc2c(C)ncs2)C2CCOC2)CC12CCCC2 c1(Cc2scc(CC)n2)ccccc1CS(=O)(=O)CCc1cnccn1 CCCCCCCN1CCC(NC(=O)C(CC2CCC3CC23)NC(=O)OC)C1 c1(C(N(CC(CC)NC(=O)CNc2ncccn2)C)=O)n[nH]cc1C1CC1 C=CC1CN(C(=O)C(C)CNC(=O)CCC(C)N(C)C)CC1O C1(NC(=NCc2c(C)cn(C)n2)NC2CCOCC2)CC(C2CCC2)C1 Cc1cn2cc(CC(=O)NOCc3cn(C4COCC4O)nn3)nc2s1 C1(C(N(CC(F)F)CCC)=O)CCN(C(=O)C2CC3(CCO2)CC3)O1 CC12CN(C(=O)OC(C)(C)C)CC(Nc3nc(C4CCOC4)ns3)(C1)C2 C1(C(=O)NCC=CCNC(=O)CC(c2ccccc2)c2ncc[nH]2)CC2CC1C2 CC1(C)COC(CCC(=O)NCC2CN(C(=O)C(c3ccccc3F)(C)F)C2)C1 CC(C)CCCCN(C(=O)Cc1ccc(O)nc1)C.C12(CCCO1)C(=O)C2 c1(C(=O)NC(C=C)Cc2ccc(F)cc2)cc2n(n1)CCCCO2 N1(C(=O)CCN2CCC2)CC2CCC1CN2C(c1c(Cl)csc1Cl)=O c1(CC)cc(NC2CCCCC2CNC(C2(N(C)C)CCOCC2)=O)nc(C)n1 C1(CNC(C(CCC)C)=O)(OC)CCN(C(c2cnc(O)cc2OC)=O)CC1 CCC(C(O)C(F)F)NC(=O)Cn1ncnc1C C1(C)(CNC(C(CSC)OC)=O)CCN(C(=O)C(N2CCCCCC2)C)CC1 C1(CC(N2CC(C)(OCC)C2)=O)CN(C(C2CC2C)=O)CCO1 N1(CC(=O)N(CC(=O)Nc2ccc(C)c(C)c2)C)CCC2C(C1)NC(=O)N2C n1(CC(=O)NCC2(O)CN(C(C3C(C)CC=CC3)=O)C2)nc2c(n1)CCCC2 c1(CCC(=O)NCC2CC(NC(C(C)OCCOC)=O)C2)ccc(CC#N)cc1 C1(CC(=O)NCCC(C)NC(=O)C=CSc2ccccc2)CC(C)OC1C C1(C2CCN(C(=O)C=Cc3cccs3)C2)(NC(C2CC3CCCCC23)=O)CC1 C1(CC)CCOCCN1C(=O)CCN(C(=O)CCc1cnn[nH]1)CCO c1(SCCC(=O)NC2CN(C(CCCCSC)=O)CC2O)ncnc2[nH]cnc12 N1(C(COCCC#C)=O)CCCC(N2CCN(C(=O)CCC3CC3(F)F)CC2)C1 C#Cc1cccc(C(=O)NCC2CC2NC(=O)C2=CC(C)(C)C2)c1Cl C=CC(CC)C(=O)NCC(C1CCC1)NC(c1cnn(C)c1)=O C(=O)(CCC(CF)CF)N1CCC(C(=O)NCCC=CCCC)C1C(C)C CCC(F)(F)CC(=O)N1CCCN(CCNC(=O)CCC2CCCCO2)CC1 C1(C(=O)NCC=CC(N2CC(C(=O)OC)C2)=O)CCOCC1 C1(CC(=O)NC(c2coc(-c3ccccc3F)n2)C)CCCCC1C N1(C(c2[nH]cc(S(N)(=O)=O)c2)=O)CCC2CCC(C1)N2C(=O)CC1CCOCC1 c1(C(=O)Nc2c(C)cc(NC(C3(Cl)CCC3)=O)cc2)ccn2ccnc2n1 C(=O)(CC1OCCc2ccccc21)N1C(CNC(c2nc(C)oc2)=O)CC2CC21 Cc1nc(CNC(C2CCC2C#N)=O)oc1C(=O)NCCCCCCF CC1CC(=O)NC(C(=O)NCCCC(=O)NCC2CCC(C3CC3)O2)C1 c1(C(N2CCCC(CN(C(CC=C)=O)C)C2)=O)c(C)cc(OC)cc1F C1(CNC(c2ccc(NC)cn2)=O)COC(C)(C)CN1C(c1cccnc1S)=O C1(C(=O)NCC2(OCC)CN(C(C(CC=CC)C)=O)C2)CC2C(C1)C2(C)C c1(CC)cc(C)ccc1C(=O)NCC(CC)NC(c1cnc(Cl)c(N)c1)=O Cc1ncc(C=CCNC(C2CCCC2c2ccccc2)=O)s1 c1(C(=O)NCCC2CCN(C(c3ccc(C(C)C)o3)=O)C2)ccnc(C2CC2)c1 C1(CC(N2CC(F)(CC)C2)=O)CC(NC(=O)CN2CCNC2=O)C1(C)C C1(NC(c2cccnc2O)=O)CN(C(c2ncccc2Cl)=O)CC12CCC2 C1(C(=O)NC(C)Cn2cc(C)cn2)(CC)CCCN1C(=O)CCC(=O)NC C(=O)(C1=NOC(C)C1)N(CCCNC(c1sc(CC)c(C)c1)=O)CC1CCCC1 CN1CCCC(C(N2CCOC(CCCNC(C3CS(=O)(=O)C3)=O)C2)=O)C1 c1(C(CNCCCC)CC)noc(C)c1C(=O)O c1(-c2nn(C(CC)C)c(CCn3cnnc3C3CC3)n2)ccc(F)c(F)c1 C1(C(N2CCCC2CCO)=O)C2CC2CN1C(=O)C=Cc1ccccc1 N1(C(CC2(OC)CC2)=O)CCCC(CO)(NC(C2CCCC(C)(C)C2)=O)C1 c1(C(=O)NC(C)CCCCNC(c2nocc2C(C)(C)C)=O)cn2ccnc2s1 N1(C(CCCCCCOC)=O)CC2CCCC(C1)N(C(=O)Cc1cc[nH]c1)C2 c1(CC(N2CC(C)(NC(C3C(N(C)C)CCCC3)=O)C2)=O)ccc2c(c1)COC2 C=CCC(C(=O)NC1CCC(CCC(=O)NC(C)C(C)(C)C#N)C1)C(C)C C1(C(=O)NCC2CC(OC)CN2C(=O)C(=O)NC(C)C)Cc2ccccc2S1 C1(CNC(=O)C=CBr)COC(CNC(c2nc(C3CC3)cs2)=O)C1 N(C(=NCCC(F)(F)F)NC1CCOC(C)C1)CC.c12cccc(c1)N2C C1(CCC(C)(C)NC(CC(C)n2cccc2)=O)CCCCN1C(=O)C=CCO N1(C(C(c2ncn(C)c2)=O)=O)CCC(O)C1C(N1CC(O)(CCO)C1)=O C=CCC(C)C(=O)NC(C)Cn1cc(CNC(c2csc(CC)n2)=O)nn1 c1(C(=O)NC2C(OC)CN(C(COCC)=O)C2)ccc(Br)c(C)c1F N1(C(CSCCC)=O)CC(CNC(c2c[nH]c(=N)cc2C)=O)C(C)(C)C1 CC1(C)CC(CC(=O)NC2CC(CCF)C2)N(C(C2CC2Cl)=O)C1 c1(C(N(C)Cc2ccc(CNC(=O)CC(C)(C)F)cc2)=O)cc2n(n1)CCO2 c1(C(N(OC)Cc2ccccc2)=O)cc(S(C)(=O)=O)ccc1OC(F)(F)F N1(C(C(C)SCCCC)=O)CC(NC(c2cn(CCO)nn2)=O)C(CC)C1 N1(C(c2c(F)ccc(N)c2)=O)CC2(CCCC2NC(C2CCS2(=O)=O)=O)C1 Cc1ccnc(C(N2CCOC(CCCNC(=O)CN(C)C(N)=O)C2)=O)c1O CCC(CC(=O)NC(C)(C)COCCCNC(c1cnn(C)c1Cl)=O)C1CC1 Cc1n[nH]c(C)c1SCC(=O)NCC1C2CN(C(=O)CCCn3ccnc3)CC12 C1(CNC(=O)Nc2nccc(P(C)(C)=O)c2)CNCCC12CCOCC2 c1(C(N(C)Cn2ccnc2)=O)csc(C)c1.C(=O)(C(F)=CC1CC1)NCC1CC1C N1(C(CCN(C)C)=O)CCN(Cc2ccc(Cl)cc2C(F)(F)F)CC1C#N C1(CC(N2C(C)COCC2)=O)C2CCCC2N1C(C1CCC(=O)O1)=O CCC1=NOC(C(=O)N(CCCN(C)C(C2CCC2)=O)C)C1.c12ccccc1S2 C1(C(=O)OC)CCC(C(=O)NC(C)(C)CN(C(=O)CCOC2CC2)C)C1 C1(NC(NNC(=O)C2C(C)OCC2)=O)CC2CCC(C1F)N2C(=O)OC(C)(C)C CC1CN(C(c2c(CNC(=O)C=CCF)cnn2C)=O)CCC1O CC(C)(C)CC(C(=O)NCc1ccc(CO)o1)NC(C1CCSC1)=O CC1(C(=O)NCC2COCC2NC(=O)CNC(c2ccccc2)=O)CCOCC1 CCC(C)(O)CCNC(C1CCN(C(=O)C(C)N2CCCC2)C1C)=O N1(C(c2cn(C(C)C)nn2)=O)CC2(CC2)CC1CNC(C1(C2CCC2)CCC1)=O c1(C(=O)NC(C)C(CO)NC(c2ccc(F)c(N)c2)=O)cc2c(cn1)OCCO2 c1(CC(=O)NC(C2CCN(C(c3cc(F)c[nH]3)=O)C2)C)cc(Cl)ccc1O C1(N(CC#C)C(C2(OCC)CCOC2)=O)CCN(C(C2(F)CCOCC2)=O)CC1 c1(C(=O)NCC2(NC(c3cc(F)cc(N)c3F)=O)CC2)cc2c(=O)[nH]ccn2n1 CS(=O)(=O)C1CC(C(=O)NC2CN(C(c3cccnc3O)=O)CCC2CO)C1 c1(CC(N2CCC(N(C(=O)C(C)N3CCC3)CCC)C2)=O)cc(C)nn1C N1(C(CC=C=C)=O)CCC(C(=O)Nc2ccc3c[nH]nc3c2)CC1(C)C C1(N(C(C(C2CN(C(c3cncn3C)=O)C2)OC)=O)C)CCCCC1C C(C)(CC(C)NC(=O)CC1(C2CC2)CC1)NC(C=CC(C)C)=O C(c1cncn1C)=CC(=O)N(C1CC(NC(CCc2onc(CSC)n2)=O)C1)C C(c1cn(C)cn1)=CC(N1CCC(C(=O)NCCCn2c(C)ncc2)C1)=O c1(C(N2CCC(O)(CNC(C3C(C#C)C3)=O)C2)=O)ccc(C#C)cc1C c1(NC(N2CC(O)CC2CO)=O)cnc(C(F)(F)F)cc1Cl.N12CC3CC3(C1)C2 c1(C(=O)NCC(C)(C2CC2)NC(C(CC=C)N(C)C)=O)cc(S(N)(=O)=O)c[nH]1 N1(C(c2c(C)scc2)=O)C(C(N2CCOC(C(N)=O)C2)=O)CC2CC12 C1(NC(c2cc(SC)c(F)cc2)=O)CCC2CCN(C(=O)CC3(C)CCC3)C1C2 c1(C(=O)NC(c2n(CC)ccn2)C)cc(CNC(c2cc(C#N)c[nH]2)=O)ccn1 CC(C(=O)NCC(F)CO)(C1CCC1)NC(=O)Cc1ccsc1 c1(CCC)cc(C(N2CCC(CNC(=O)CSCC(C)C)C2)=O)c(C)o1 N1(C(=O)CSc2ccc(Cl)nc2)CCC2(CC1)CCN(C(C1(O)CCC1)=O)C2 c1(C(N2CCC3(C(C(=O)Nc4c(C)nsc4)C3)C2)=O)cc(Cl)cc([N+](=O)[O-])c1Cl C1(NC(C2(COC)CN(C(=O)CCC(C)(C)C)C2)=O)CCn2nnnc2C1 c1(CN(C(C(C)N(C(=O)Cc2ccco2)C2CC2)=O)C)ccnn1C N1(C(C(C)Sc2ccc(C#N)cc2)=O)CC2COCCC2(C(N)=O)C1 c1(OCC)cccc(OC)c1C(c1nnnn1C)NC1CC1(C)C C1(C(N(CC(O)C2CCC2)C)=O)CCCCCCN1C(=O)CCCNC(N)=O N1(C(C(CCOC)N)=O)CCCC(N=[N+]=[N-])CC1 c1(C(=O)NCC(CC(=O)NC(CCC)(C)CO)OC)coc2ccccc12 C1(NC(c2ccnc(OC)n2)=O)CC2CN(C(c3oncc3C)=O)CC12 N1(C(C2(C#C)CN(OC(=O)C3=NOC(C)C3)C2)=O)CC2C3C=CC(O3)C2C1 N1(c2ncc(OCCOC)cn2)CC2(CCCC2NC(c2nccnc2N)=O)C1 c1(NC(C2N(CC)CCC2)=O)ccccc1-c1cc(C(=O)NC2CCCC2)no1 c1(C2C(C(N(C3CSC3)CC)=O)C2)ccc(Br)cc1 c1(NC)ncccc1C(=O)NCC1CCC(C(=O)NC2CCC2C(=O)NC)CC1 C1(NC(C2(CN)CCCO2)=O)CCN(C(=O)Nc2ccncc2F)CC1 c1(CC(C)C)ncc(C(N2CC(F)(CNC(=O)CCC3CCC(=O)N3)C2)=O)s1 c1(OC)cccc(F)c1CC(N1CCC(O)C(N(C)C(C2CC2C)=O)C1)=O N1(C(C(c2ccccc2)NC(=O)NCC2CCN(CC)C2)=O)CCSC(C)(C)C1 C(=O)(C(C)CC(N)=O)NCC(CN(C(=O)CC(F)(F)Br)CC)(C)C C1(NC(c2ccc[nH]2)=O)CC=C(C(=O)N2CCC2(CO)CO)C1 CC1CN(C(=O)COc2ccc(C3CC3)cc2)CC(C)N(C(=O)COC(F)F)C1 CC(C(=O)N(C1CCN(C(C2CCC(F)CC2)=O)CC1)CCO)C(F)F c1(NCc2cc(CC)no2)ccc(S(=O)(=O)N2CCC(C)S(=O)(=O)CC2)cn1 C#CCC(C)C(=O)N1CC2C(CN(C)C(c3ccncc3F)=O)C2C1 c1(CC(=O)NCCC2CCN(C(=O)CSCC3CC3)C2)cccc(OC(F)F)n1 Cc1c(Cl)cc(C(=O)NCCCCNC(c2ccsc2)=O)cc1Br Cc1cc2cccc(CN=C(NCC3CCCO3)NCC(C3CC3)N(C)C)c2[nH]1 Nc1ncc(C(F)(F)F)cc1C(=O)NC1CC1NC(=O)C(F)CC1CCCC1 C1(CC(=O)NCCC(C)(C)NC(Cc2c(C)cco2)=O)CCCC(=O)C1 NC(=O)CCCNC(=O)CC1CN(C(=O)N(CCCCl)CCCl)C1 Cc1cc(CCC(=O)NCC=CCNC(=O)C(C)Oc2ccc(O)cc2)nn1C CC(CC(=O)NCCC1CN(C(C2(CO)CCOCC2)=O)CCO1)C(F)F c1(C(=O)NC(C2(O)CCN(C(C3CCC(C)CC3)=O)C2)C)cnc2ccsc2c1 N1(C(c2n(C(C)C)nnc2)=O)CCC(NC(=O)Cn2ncc(Br)n2)C(O)C1 C1(C)(CC)CC(NC(c2nnn(C)n2)=O)CN1C(c1ccc(N(C)C)cn1)=O c1(NC(C2N(S(CC(=O)OCC)(=O)=O)CC(F)C2)=O)cc(C)c(C)cc1Br C(CCCCC(=O)NCC=CCC(N1CCC(CN=[N+]=[N-])C1)=O)N(C)C c1(CNC(C2(C)COC2)=O)nocc1C(=O)NC1COC(C2CC2)C1 C(c1ccc(C(F)F)o1)=CC(N1C(CN(C(C(C)C2CC2)=O)C)CCC1)=O c1(C2C(C(=O)NCC(C)CNC(=O)C(C3CCOCC3)F)C2)cccnc1Cl c1(C(N2CC3C(NC(COCCCC)=O)C3C2)=O)cc2ccc(C)cc2[nH]1 Cc1nc2n(n1)CC(C(=O)N(CCCNC(c1c(C)noc1C(C)C)=O)C)CC2 Cc1cc(C#N)sc1C(N1CC(CNC(=O)C(F)(F)C2(O)CCC2)C1)=O N1(C(C(COCC)n2cc(-c3ccc(Cl)s3)nn2)=O)CC2(COC(C)C2)C1 c1(CCC)c(C(N2CC(NC(=O)C(C)O)C(C)C2)=O)cnn1-c1ccc(F)cc1 c1(SCC)nccnc1C(=O)NCCC1CCCN(C(c2cnn(C)c2C)=O)C1 C(CC(C(=O)NCCC1CC(NC(=O)CC2CS(=O)(=O)C2)C1)N(C)C)SC C(N=c1[nH]c(=N)[nH]c(=NCCCC2CC2)[nH]1)c1cccc2ncn(C)c21 C(=O)(CCCCC#N)NC(C)CN(C)C(c1ccc(C(F)F)cc1)=O Cc1ncc(CCC(=O)OCC23CC(F)C2C3)o1 C(=O)(C(F)(F)CCc1ccccc1)NC(C(C)C)CNC(=O)Cc1ccncc1 N1(C(CC(=O)OC)=O)CCC2(CCC(NC(=O)C(C)C3CCCO3)CC2)CC1 c1(C(C)=O)cc(C(=O)N(C2CCN(C(=O)CN3CCC(C)CC3)CC2)C)c(C)o1 C12(NC(c3c(CC)cno3)=O)CCCC1CN(C(c1sccc1OCC)=O)C2 Cc1cc(CNC(c2cc(CNC(=O)C(F)C3CCOC3)cs2)=O)cc(C)n1 N1(C(=O)OCC)CCC2(CC1)CC2CNC(=O)C(C)(C)C(F)c1ccccc1 N1(C(c2c(C)nc(CO)o2)=O)CCCC(C2(NC(=O)C3=CCC3)CC2)C1 C1(CC(=O)NCC(=C)CCNC(c2c[nH]c(Br)c2)=O)CCC(C)(C)C1 CC1CN(C(=O)C(C)(C)C(C)(F)F)CCC1N=c1[nH]c(C(F)F)nc(=N)[nH]1 C(=O)(N1CCCc2nccn21)C1N(C(C(CC=C)NC(C)=O)=O)CCC1 C(=O)(CC1OCCc2ccsc21)N1C(COC)(CNC(=O)C2=CCC2)CCC1 N1(C(C(CC)O)=O)CCOCC(C(=O)Nc2cn(CCF)nc2C)C1 N1(C(C)=O)CCC(C)(C(=O)NC2CCN(C(=O)CNCC3(C#N)CCC3)CC2)C1 c1(C(=O)NC2CN(C(c3c(OC)nsc3)=O)C(C)C2)ccc(F)c2cnccc12 c1(SCC)ccc(C(N2CCC(O)(COC)C2)=O)cc1 C=C=C(C)CC(=O)N(C1CCN(C(=O)CN(C2CCS(=O)(=O)C2)C)CC1)C C(CNC(=O)CCC(F)(F)F)(N=c1[nH]c(Cl)c(C#N)s1)c1c(OC)cccc1 C(C)(C(O)C(=O)NCC(C)(C)CN(C(=O)C(=O)NCCC(N)=O)C)SC N1(C(COCC#C)=O)CCC(C=C)(C(=O)NCCc2cnc(C)s2)C1 O=C1CN(C(C2CN(CCc3ccc(-n4cccn4)cc3)CCS2)=O)CCN1 c1(C(=O)NCC(C)(C)OC(=O)CNC2C(OC)(OC)CC2)cc(I)ccc1O C(=O)(C(F)(F)C(C)(C)O)NCC(CN(C(=O)Cc1ccc(C(N)=O)nc1)C)O CC(C)CC(C)(C)C(=O)N1CCOC(C(C)NC(=O)CN(C)C(C)C)C1 C12(C(N(CCCCN(C(=O)CC3CCC(=O)N3)C)C)=O)CCC(C1)C2 O=C(CCCCC1CC1)NC1CC(CNC(=O)C(C2(O)CCCCC2)(F)F)C1 c1(C(=O)NCCNC(c2c(CCC)nco2)=O)ccc(=O)n(CCF)n1 C(=O)(C(C)(F)C(=O)N(CCC(=O)NCCCOCCO)C)OC N(C)(C(=NCC1CCCCC1)NCc1nc(-c2ccncc2)n[nH]1)CCCC C12(NC(C(C=C)N(C)C)=O)CC(CO1)N(C(=O)C(C)CNC(=O)OC(C)(C)C)C2 c1(C(N2CC(C(N(CCCC=C)CC)=O)OCC2)=O)ccc(C)nc1C CC(C(=O)N1CC(C)(OCC(=O)NCc2cncn2C(C)C)C1)C(C)(C)C Cc1[nH]nc(C(N2CC(NC(c3cn(CC(F)(F)F)nn3)=O)C(C)C2)=O)c1O N1(C(CCc2cc(C)no2)=O)CCC(NC(=O)CCC#N)C(C(C)C)C1 N1(C(C2C(C)(CC)C2)=O)CCC(CCCNC(c2nnsc2C)=O)CC1 C1(COCC)(CNC(C2(OC)CCCC2)=O)CCCN1C(c1ccsc1)=O C1(CNC(CCCC#C)=O)CN(C(C23CSCC2C3)=O)CC12CC2 c1(CC)nnc(C)cc1C(N1CCN(C(=O)C#CC(C)C)C(CO)C1)=O C(=O)(CC(O)CNC(=O)COc1ccsn1)N(CC(C)C)CC(N)=O c1(C(=O)OC)coc(NC(=O)NCCC2CC(OC(C)(C)C)C2)n1 CCCC(CCCNC(=O)CCNC(C)=O)NC(c1ccc(F)c(N)c1)=O C=CC(F)(F)C(=O)N(C)CC1CCCN1C(=O)CN(C)CCOC C(c1ccccc1Cl)=CC(=O)NC1C(NC(=O)C=CC2CCOC2)CCCC1 C1(NC(c2c(F)cccc2F)=O)CC2(CCN(C(C3C4CCN3CC4)=O)CC2)C1 Cc1cc(Br)cnc1C(N1CC(CCNC(C2CC3(C2)CC(C)C3)=O)C1)=O c1(OC)cc(N2C3CCC(C3)C2C(=O)NCCCNC(C)=O)nc(S(C)(=O)=O)n1 C(=O)(C(C)(Cc1ccccc1)C(C)C)NCCC1CCN(C(C(C)CF)=O)CC1 CCCCC(CC)CCC(=O)N(C)CC1CCCC1NC(=O)CCC(CC)OC c1(C(N2CC(NC(C(C)OCC#C)=O)CC23CCC3)=O)cncc(P(C)(C)=O)c1 c1(C(=O)NC2(CN(C(c3cc(CC)c(C)o3)=O)C)CC2)ccc(Br)nc1N c1(C(N(C)CC2CN(C(=O)CCc3nnc(S)n3C)C2)=O)cc(S(N)(=O)=O)co1 C(C(=O)N1CC=CC(NC(C2CC3CC3C2)=O)C1)(C(C)C)NC(=O)OCC C1(NC(CS(=O)(=O)NC)=O)CCCC12CN(C(c1coc(CC3CC3)n1)=O)C2 CC1CN(C(C2CCN(C(=O)Cc3ccsc3)CC2)=O)CC(=O)N1 C(=O)(N1OC2C=CC1CC2)C1CC(C)N1C(c1cnc(O)c(F)c1)=O C1(CNC(CCCOCC=C)=O)CCN(C(C2(Br)CC2)=O)CC1C1CC1 CCCCCCCCC(C)C(=O)NC(C)(CNC(c1cnnn1C(C)C)=O)CC c1(OC)cccc2c(CNC34CC(C(=O)OC(C5COC(=O)C5)=O)(C3)C4)coc12 C=CCC(C(=O)N1CC(CNC(C2CNC(=O)O2)=O)C1)OC N1(C(CN(CC#C)C(c2cocc2C)=O)=O)CCC(F)(CF)C1 CN1CC(=O)N(CCCC(=O)NC2CN(C(=O)CCc3cnc(O)[nH]3)C2)C1=O Cc1ccc(C(=O)NC(CNC(c2ccc(C(O)CF)cc2)=O)CC(C)C)cc1 C1(CCNC(c2ccn(CC(C)C)c2)=O)CN(C(C2CS(=O)(=O)C2)=O)CC(C)O1 C12(C(c3nnnn3C3CCOCC3)NCC(C)OCCO)CCC(CC1)OC2 N1(Cc2cn(-c3cccc(CC(=O)OC)c3)nn2)CCCCC2(CCOCC2)C1 C1(NC(C2CCC(=C)CC2)=O)CN(C(=O)C(C)C2CCC2)Cc2nccn2C1 c1(CNC(C(=O)N(C)CC2CCCCO2)=O)sc(Cl)cc1Br N1(C(C(C)OCC)=O)CCC(C)(CNC(c2c(CC)nn(C)c2Cl)=O)CC1 N1(C(CC(=C)Br)=O)CC2C(CNC(C3(C)CS(=O)(=O)C3)=O)C2C1 C1(COC)(NC(=O)C=C2CCCCC2)CCN(C(C2(C3CCCO3)CC2)=O)CC1 N1(C(C(CCN(C)C)N(C)C)=O)CC2CCN(C(c3ccsc3Cl)=O)CC2C1 c1(CC)ccc(C(N2CC(CNC(=O)CCCN=[N+]=[N-])CC(C)C2)=O)cc1F CC(Cn1ccnc1)C(=O)NCCN(C1CCCC1)C(=O)CC1CCCO1 C1(CNC(COCCOC)=O)CC2COCC2N1C(C1CC12CC2)=O N1(C(C(C)N=[N+]=[N-])=O)CCC2C(CCCN2C(c2cccc(N(C)C)c2)=O)C1 CCC(CCOC)C(=O)NCC1(F)CC(NC(=O)Cc2ccsc2)C1 c1(OCCCN(C(=O)C=C2CCCC(C(F)(F)F)C2)C)cccc([N+](=O)[O-])c1 C(C(C(=O)NOCC1CC1)C(C)(C)C)NC(C(CC)SC)=O C1(CNC(C(CO)N(C)C)=O)CC2CCC1N(C(=O)C=Cc1cccc(O)c1)C2 c1(N2CCOCC(NC(CCn3c(C)nc(C)n3)=O)C2)ccn2c(Br)cnc2n1 C(=O)(C(C)(C)C1=CCN(C(=O)C2=C(Cl)CCCC2)C1)NC1C(O)CCN(C)C1 C12CCN(CC1)c1ccnc(n1)NCC2.C1(C(C)(C)C)COC(C(F)(F)F)C1 Cc1cc(C(N2CC(CNC(=O)Cn3c(C)ccc3C)C(C)C2)=O)c(Cl)cc1F CC(N=c1[nH]c(=NC(C)c2ccc3nc(O)[nH]c3c2)c2[nH]ccc2[nH]1)C1CCC1 C(CN=c1[nH]c(C)nc(Cl)c1CC)(C1CCCC1)NC(c1ccn(CC)n1)=O c1(N2CCC(N3C(CC(C)(C)C)CC3)C2)nccc(-c2ccccc2)n1 Cc1cc(C)c(C(N2CC(C3CN(C(c4cn(C(C)C)cn4)=O)C3)C2)=O)c(C)c1 c1(CC(=O)N(C2CCN(C(C(CCC)NC(C)=O)=O)C2)CC)c(F)cncc1Cl C=CCC(C)(CC)C(=O)NC1CC2(C(=O)NC3CCCCC3(C)O)COC1C2 CC1(C)CC(C(=O)NC2(CC(N)=O)CC2)CN1C(=O)C(=O)C1CCCC1 Cc1c(Br)ccnc1C(N1CCN(C)CC1CNC(=O)COCC(F)F)=O C1(NC(C2C=CC(NC(=O)CCCCN3CCCC3)C2)=O)CC12CCCCCC2 N1(C(C2(OC)CCSCC2)=O)CCC(C2(NC(c3csnc3C)=O)CC2)C1 N1(C(C2CC(NC(CCCCC)=O)C(O)C2)=O)CC(O)C2(CCCC2)C1 C1(C)(C(N2CCC(N(CCC)C(c3ccoc3C)=O)CC2)=O)CCC(C)(C)CC1 c1(CN2CC(C(=O)NC34CC(C(=O)OC)(C3)C4)C2)cc(OC(F)(F)F)cc(Cl)c1 Cc1nc(O)c(C(=O)NC2CN(C(C3CCCCC3)=O)CC3(CC3)C2)nc1C c1(C(=O)NC(C)CCNC(C2(CO)CCC2)=O)ccc(-c2cnn(C)c2)o1 CC(C)C(CCN(C)C(=O)Nc1cc(C2CCOCC2)no1)N(C)C c1(OC)ncc(Cl)c(=NC2CCCC23CN(c2nc(C(F)F)nc(=N)[nH]2)C3)[nH]1 C1(C(N2CCCN(C(C(C=C)(C)CC)=O)CC2)=O)COc2ccc(O)cc2O1 N1(C(Cc2ccc(C)cc2)=O)CCN(C(c2ccnnc2)=O)C2COCC12 Cc1cc(Cl)c(C(=O)NC2CC(F)(CNC(=O)C(O)Cn3cncn3)C2)cc1N N1(C(c2ncn(CCNC(C(CC)C(C)C)=O)c2)=O)CCC(C2(C)CC2)C1 C#CC1(C(N2CCN(C(C3CC(OC(F)F)C3)=O)CC2)=O)CCOCC1 c1(NCC23CC(NC(CNC(=O)OC)=O)(C2)C(C)O3)cnc2nccn2c1 N1(C(C2(NC(C3=C(C)CC3)=O)CCOCC2)=O)CC(C)CC(C)C1 C1(C(=O)NC)CCC(NC(C2CC(N)CN2C)=O)CC1 Cn1c(O)nc2cc(C(=O)NCC3CN(C(c4cnn[nH]4)=O)CCCO3)ccc12 N1(C(CC(CC)CC)=O)CCN(C(=O)CNC(=O)CN(C)C)CC(O)C1 N1(C(CC(CCSC)O)=O)CC2CC3CC2C1C3NC(c1cocn1)=O N1(C(C(C(CC)O)C)=O)CC2CCC1CN2C(c1sc(F)cc1Cl)=O CC1CC(CNC(c2ccc(C(F)(F)F)nc2)=O)CN1C(c1ccc(O)cn1)=O N1(C(CC2(C)CCN2C(=O)C=Cc2cocn2)=O)CC2C(C1)C2(F)F C1(C(N(CCC#C)CC)=O)CN(CCC2(COC)CC2)CC1C C1(CC(=O)NCc2ccn(C(C)C)n2)CCCN(C(=O)CCCF)CC1 C1(NC(C2CCCS2(=O)=O)=O)CCS(=O)(=O)C12CN(C(c1cc(C3CC3)on1)=O)C2 C(=O)(CC(C)(C)C#N)N(C(C)C(=O)NC1(C)CC(F)(F)C1)C CN=c1[nH]c(SC)ncc1CN1CC2CC1C2C(=O)Nc1cccnc1Cl c1(N2CC(CC=C)(NC(=O)C(C)SC(F)(F)F)C2)cc2nncn2cn1 C(=O)(C(O)CC(F)F)NCC(=O)NCc1cn(Cc2cccc(Cl)c2)nn1 C1(COC)(NC(C2COCC(C)(C)O2)=O)CCCN(C(c2ccco2)=O)C1 c1(CCC(=O)NC2C(NC(Cc3nc(CC)sc3)=O)CC2)cnn(C)c1C N1(C(C2CCC(NCc3c(OC)cccc3Br)CC2)=O)CCCC2(CCOC2)C1 C1(C(N2CCC(SC)C2)=O)CCCCN(Cc2ccccc2)C1 Cc1ccc(C)c(C(N2CC(CCNC(=O)CCSCC(N)=O)C(C)C2)=O)n1 N1(C(c2c(C(=O)O)sc(Br)c2)=O)CC2(CCCCC2)CC1CO C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CCN(C(CCSCC)=O)C12CC2 Cc1cccc(NC(=O)C(=O)N(CC(C)(C)CCCNC(=O)CCC=CBr)C)c1 c1(C(=O)NC2COCCN(C(C3C(C)C3)=O)C2)nn(C)c2ccccc12 C1(CNC(CC(CC)C)=O)CC12CCN(C(c1coc(C(C)(C)C)n1)=O)CC2 N1(c2nnc(CCC)s2)CCC(O)(C2(CO)CCC2)CC1 C1(NC(COC(C)=O)=O)CCCC1(C)NC(=O)CCOCC(F)F c1(OC)ccc(-c2nc(CP(C)(C)=O)n(CC3COC(C)(C)C3)n2)nc1 C1(C(N(C2CNC(=O)OC2)C)=O)N(C(c2cccc(F)c2)=O)CCC1(C)C Cc1ccc2nc(SCCC(=O)NCCC(C)NC(=O)CSCC(N)=O)[nH]c2c1 C1(NC(CCC(=O)NCC)=O)CC2CCC(C1C)N2C(c1cc(CC)nn1C)=O C1(N(C(CCC=CC(C)C)=O)C)CCCN(C(=O)C(O)C(F)F)CC1 C1(C(=O)NC(C)CCNC(=O)C=Cc2cncn2C)CCc2nccn2C1 CP(C)(=O)CCCNC(C1CC(F)CN1C(C1CN(C(N)=O)C1)=O)=O CC1CN(C(=O)CN2CC3CC3C2)CC1(C)CNC(=O)C=C1CCC(C)CC1 Cn1cc(C(F)(F)F)cc1CN(C1CCN(Cc2ccccc2)C1)C c1(OC)ccc(C(=O)NCC2CC(C)N(C(=O)CSCc3cccs3)C2)cc1Br C12(CNC(c3cc(C(C)=O)sc3)=O)CCC1CN(C(c1ccc([N+](=O)[O-])[nH]1)=O)C2 C12(NC(CCCC=C)=O)CCCCC1CN(C(c1nccc(OC)c1F)=O)C2 N1(C(C)=O)CC(COC(C)=O)C(C(F)(F)F)C1.C1(=O)CC(O)CN1 C1(C(N(CCCCC=C)C)=O)CCCCC1NC(=O)Cc1sccc1C c1(OC)cccc(CCC(=O)NCC(O)CCNC(c2sncc2C)=O)n1 c1(CC(=O)N(C(C)CNC(=O)C(C)CC2CCCC2)CC)ccn(C)n1 N1(C(COCCCC(C)C)=O)CCN(C)C(C(=O)NCCC2CCCN2C)C1 C1(C2(CC(=O)NCC3CCCCN3C(C3CC(F)(F)C3)=O)CC2)CCS(=O)(=O)C1 C12(C(=O)NC3CCC(CNC(c4c(C)cncc4)=O)C3)CCCC1CC(=O)C2 c1(CC)ncc(C(=O)NCCC2CN(C(C3CCN(C)C(C)C3)=O)C2)c(O)n1 c1(N2CCC(C)C(CO)C2)nc(=NCCc2ccn(C)n2)[nH]c2ccsc12 C1(C(=O)NCCOC2CCN(C(c3cnc(OC)nc3)=O)C2)CC(C)(C)CCO1 C#Cc1ccccc1CC(N1CCC(C)(CNC(=O)CCCn2ccnc2)C1)=O C(CCCC(=O)NCC1CCCN1C(C1(c2n[nH]c(C)n2)CC1)=O)SC C1(C(=O)NC(C)CN(C)C(c2ccc(CF)cc2)=O)CC2OC1C1CC21 N1(C(C2(c3ccccc3)CCC2)=O)CCOC(C(O)CO)C1 c1(NC(C(N(C(c2ccn(CC)n2)=O)C)C2CC2)=O)cc(C)c(C)c(C)c1 Cc1ccc(C(=O)NC2(CO)CN(C(=O)C(C(C)C)SC(C)C)C2)nc1 CC1CC(NC(c2cc(N)nc(Cl)c2)=O)CCN1C(C1CC2C=CC1CC2)=O c1(C(N2C3C(CNC(C4C(=C)C4)=O)C(C3)C2)=O)cc(Br)cc2nc[nH]c12 c1(C(N2CC(CC=C)(NC(=O)C(c3ccnn3C)C)C2)=O)c(C)nsc1NCC CC(C)(C)CC(C(=O)NCC1Cc2nccnc2C1)NC(=O)OC(C)(C)C CCC(=O)CCC(=O)N1CCCC(N(C(=O)C(C)CCOC)C)C1 c1(CN(C(C(=O)NCC(C)NC2CCCCC2)=O)n2ccnc2)ccc(F)cc1 N1(CC(=O)NCCCC2N(C(CC3C(C)C3)=O)CCC2)CCN(S(C)(=O)=O)CC1 c1(OC)cccc(Cl)c1C(N1CCCC(C)(NC(=O)C(O)CSC)C1)=O C1(NC(c2scc(OC)c2)=O)CN(C(=O)C(c2ccccc2)NC(C)=O)CC1C N1(C(C2N(C)CCC2)=O)CCCC1(C)CCC(N1CCOCC1)=O C1(C(=O)NCC(CC(C)C)NC(C2N(CC)CCOC2)=O)CNC(=O)CC1C C(C)(C(CC(=O)Nc1ccc(F)cc1C1CC1)NC(=O)C(C)=C(C)C)OC C(CCCCO)N(C)C(C1(CNC(=O)CC2C=CCC2)CCCO1)=O C1(C)(CNC(C2CCN(C(CC)=O)C2)=O)CCCN(Cc2nc(C3CC3)no2)C1 CC(C)CC(C)C(=O)N(C1CNC1)Cc1cccs1 CC(C)CCCC(C)C(=O)NC1CC(NC(c2cc(O)nc(O)n2)=O)CC1O c1(C(N2CCC(OC)(CNC(C3NC(=O)OC3C)=O)C2)=O)cc2c[nH]cnc-2n1 Cc1cc(C(=O)NC2CCC(N(C)C(c3csnc3Cl)=O)C2)c(C)s1 c1(C(=O)NCC2(CNC(c3c(CC)ocn3)=O)CCCC2)ccc(CCO)cc1 N1(C(C=CCOC)=O)CC(NC(C2(c3ccccc3C)CCCCC2)=O)C(O)C1 N1(C(C2(CCN=[N+]=[N-])CC2)=O)CCC(C(N2CCC(N3CCCC3)C2)=O)C1 c1(C(N2CCC(C)(C(=O)NCC3(C)CCCC3)C2)=O)n[nH]cc1[N+](=O)[O-] C1(CNC(c2cc(CC(=O)OC)on2)=O)C(C)CCCN1C(=O)C1=CCCSC1 c1(CC)[nH]nc(C(=O)NCC2CCCN(C(=O)C(C)(F)C(C)(C)F)C2)c1[N+](=O)[O-] C1(CNC(Cc2c(C)nsc2)=O)COCCN1C(c1csc(-c2ccoc2)n1)=O c1(C(=O)OC)cnc(NCCCOCCCNC(C2(F)CC=CC2)=O)cn1 N1(C(C(C)(CO)OC)=O)CC2CCN(C(c3cc4ncccc4s3)=O)CC2C1 c1(OC)cccc(C2(NC3CCC(OC(=O)OC4CCCC4)CC3)CCC2)n1 N1(C(C(CC#C)O)=O)CCN(C(=O)C(c2ccc(F)cc2)(C)C)CCC1C C(=O)(C1=CCCC1P(C)(C)=O)N1CCN(C(c2cc(C)cc(C)c2)=O)C(CO)C1 N1(C(c2c(C)n(C)cn2)=O)CCC(C(=O)NCC2CCCN(C)C2=O)CC1C C12=CNC(=NCC3CCN(C3)C1=O)C=C2.c1(COC(C)(C)C)cscn1 c1(OC)cc(=O)n(C)cc1C(=O)NC(C)(C)CNC(C1CCN2CCOCC12)=O CC1CCc2[nH]nc(C(=O)NCC3CN(C(=O)C4=CCCO4)CC(C)(C)O3)c2C1 Cc1cc(NC(c2ccc(F)c(-c3ccc(N(C)C)c(F)c3)n2)=O)nc(C)c1 Cn1nnc2cc(NC(N3CCCOC(CCN(C)C)C3)=O)ccc12 O=S(=O)(c1ccc(NC2CC3CCCCN3C2)cc1Br)N1CCC(CCO)C1 c1(C(=O)NCCN(C(C2CC3(CC3)CO2)=O)CC)ccc2c(c1)N(C)C(=O)CO2 c1(CCC(=O)NCCc2cc(C(=O)OC)ncc2)nnc(S)nc1O c1(CC)ncsc1C(N1CC(CCNC(=O)C(F)(F)C2CC2)C1)=O N1(C(C(CCC)N(C)C)=O)CCC(NC(c2ccc(F)c(C(C)C)c2)=O)CC1C C1(NC(=O)CCn2cccn2)C2CCC1N(C(C1CC(=O)N1)=O)C2 CCC(C)C(C)C(=O)NC12CC1CN(C(c1ccc(N(C)C)cc1)=O)C2 C12(NC(c3ccccn3)=O)CCCC1CN(C(c1cc(C(F)(F)F)no1)=O)C2 c1(C(N(CCCNC(C2C(C)C2)=O)C2CC2)=O)ccc2c(c1)SCCN2 N1(C(c2[nH]cc(C)c2C)=O)CCC(NC(=O)CC2CCC=CCC2)C(C)C1 C1(NC(c2ccc(C(C)=O)[nH]2)=O)CN(C(=O)CCc2cccnc2Cl)CC1(C)C CCC(C)(C)C(C)NCC(c1cccnc1)OC c1(CN2CC(F)CC(C(=O)NCc3cn(CCC)nc3)C2)ccc(Br)c(Cl)c1Cl C(=O)(C1CCCc2cnc(C)n21)N(CCNC(C1CNC(=O)C1)=O)CC N1(C(CCNC(C)=O)=O)CC2CC(C)N(C(=O)C#CC3CCC3)C2C1 C=C(C)C(CC(=O)NC1CCCC1CNC(=O)CN(c1ccncc1)C)OCC c1(C(N2C3C(N(C(CC(C)OC)=O)C)CC(C3)C2)=O)cc2cccc(O)c2[nH]1 c1(C(N2CCN(C(c3n(COC)ncc3)=O)C(CO)C2)=O)cccc2sccc12 C#CCCCC(=O)N(CC(=O)NCc1ncnn1C)C(C)C c1(C(N2CCC(NC(CCC)=O)C2CC)=O)ccc(S(N)(=O)=O)o1 C1(CCC=C)(C(=O)NCCC(C)c2nc[nH]n2)CN(C(=O)C(C)OCC2CC2)C1 C(C(C)CC(C)C)NC(C(COC(C)C)NC(=O)C(O)Cn1cncn1)=O N1(C(C(c2cncnc2)C)=O)CCCC(CNC(=O)CCOCC2CCC2)C1 c1(OC)c(F)ccc(CN(C)Cc2cc3c(s2)CNCC3)c1F C1(C(N(CCN(C(C(C)(C)OC)=O)C)C)=O)CN(S(C)(=O)=O)c2ccccc2O1 CCCCC(C)(F)C(=O)NCCCCC1CCN(C(C2CC2CCC)=O)CC1 C1(CNC(C2(C)CC2)=O)CCCC(NC(=O)Cc2csc(-c3cccnc3)n2)C1 C1(NC(=O)OC(C)(C)C)C2CC(C(N3CC(NC(=O)Cc4cccs4)C3)=O)CC12 c1(C(=O)NC2CN(C(CCSCC)=O)CC3(C2)CC3)c(C)c(C)c(C)c(C)c1C c1(C(=O)NC2C(N(C)C(C3C=CCCC3)=O)CCCC2)ccc([N+](=O)[O-])cc1Cl N1(C(C2(OC)CCSC2)=O)C2CCC1C(CNC(=O)CC1(C)CCCO1)C2 C1(NC(Cc2c(C)nc[nH]2)=O)CCC(NC(c2coc(C3CCC3)n2)=O)CC1 c1(CC(=O)NCC2CCCN2C(=O)CC2(O)CCCC2)ccc(Br)cc1F C(CS(=O)CC(F)(F)F)NC(=NCCCC)NCCCCF CCS(=O)(=O)CC(=O)NCC1CCCC(NC(c2ccc(C(N)=O)[nH]2)=O)C1 C1(NC(=O)C=Cc2ccc(Cl)s2)CC2CCC1(NC(=O)CCN1CCC1)C2 CC1(C)CC(CNC(C2(O)CCC2)=O)CN(C(c2cnn(CC(F)F)c2)=O)C1 n1(CC)nc(C)c(CC(N2CC(n3cc(C(N)=O)nn3)C2)=O)c1C N1(C(c2nncc(CCC)c2)=O)CC(NC(C2CNC(=O)C2)=O)CC(C)(C)C1 c1(C(N2CC(CNC(CCC(=C)Br)=O)C(C)C2)=O)cc2c(C)n[nH]c2cn1 c1(OC)ccc2c(C(=O)NC3CCCC3NC(C3CC34CCC4)=O)ccnc2c1 CC(C)C(C)(CNC(=O)Cc1cccc(C2CC2)c1)NC(C1CC2(CC2)CO1)=O c1(CC)ccc(C(=O)NC23CC(NC(=O)C(C)CN(C)C)(C2)C3)cc1[N+](=O)[O-] C(=O)(CCC(=O)NC(C(C)NC(C1COCCO1)=O)C(C)C)OC N1(C(C=CC(N)=O)=O)CCCC1CCCNC(=O)CNC(c1ccncc1)=O N1(C(CN(c2nnn(C)c2N)C(CC(C)n2ccnc2)=O)=O)CCC(CO)C(C)C1 C1(NC(C(C)CO)=O)CCN(C(=O)C(F)=C2CCCC2)C1C1CC1 C1(c2ccc(O)cc2)(C(N(CCCN(C(=O)C=C(Cl)Cl)C)C)=O)CCCCC1 C1(F)(CNC(C(C)C2CCC2)=O)CCC(NC(=O)CN2CCCOC2=O)C1 C1(CNC(CC(C)CNC(C2CC=CCC2)=O)=O)C2CCCCCC12 N1(C(c2ccc(C#C)o2)=O)CC(F)(F)CC1CCNC(=O)CCC1CCCN1C c1(CNC(CCC(C(C)(C)C)O)=O)ccc2c(c1)COCC2 c1(CCC(=O)N(C(CCNC(CCOC)=O)C)C)c[nH]c(C)c1C(=O)OC C1(CNC(C(CC#C)O)=O)CC2CCCC2N1C(=O)CCCCc1cnn[nH]1 C1(CNC(=O)C(O)C2CCC2)CCCC2(CN(C(c3cccc(Cl)c3O)=O)C2)O1 c1(C(=O)NCCCCC(C)NC(C2CC3(C2)CC3F)=O)nnc2ccccc2n1 CC1(C)CCC2(CC1)CC2C(=O)NCC1C2CC1N(C(=O)COCC1CCC1)C2 c1(C(=O)NCC2CN(C(=O)CC3CCCCO3)C2)cc2nc[nH]c2cc1[N+](=O)[O-] C(=O)(CC(C)n1cccc1)C(CONC(C1C2CCCC12)=O)=O.CC(C)NC CCC(C)CCCC(=O)NCCOCCNC(=O)CCCCCNC(N)=O N1(C(C#CC(=O)O)=O)CC2CCC(C1)N2CS(=O)(=O)Cc1ccc(F)c(C(=O)O)c1 c1(C(C)=O)ccc(S(C)(=O)=O)c(NC(c2nn(C)cc2N)=O)c1 c1(C(=O)NC(C)CN(C)C)cn2c(n1)CN(Cc1ccc(C(F)(F)F)cn1)CC2 N1(C(c2ccccn2)=O)CCC(C2CCN(C(c3cc(C(F)F)cs3)=O)C2)C1 c1(C(=O)NCC2CC(NC(CN3CCC(C)(O)C3)=O)C2)ccc2ncccc2n1 C1(NC(C(CC=C)(F)F)=O)CN(C(c2cc(C(=O)OCC)on2)=O)CC(C)(C)C1 c1(OC)cncc(C(N2CCC(F)(C(=O)N(C(C)C)Cc3cccnc3)C2)=O)c1 C1(N(C(C(CC)OCC)=O)C)CCCCN(C(=O)Cc2cc[nH]c(=N)c2)C1 C1(CNC(C2(CC)CCCO2)=O)C2CN(C(=O)C(C)NC=O)CC12 C(=O)(C(CC)N(C1CC(NC(=O)COc2ccccc2)C1)C)NCC=C Cc1cnn(CCC(=O)NC2CC(CNC(=O)CNC(c3cccnc3)=O)C2)c1 c1(C(=O)NC2CCN(C(CC=C)=O)CC2CO)c(Cl)ccc(S(C)(=O)=O)c1Cl N1(C(C2C(C)CCO2)=O)CC2CCC(C1)N2C(C1CCC2CC1CO2)=O n1(CC(=O)NCC2N(C(COCC(=C)C)=O)CCOC2)sc(=O)c2ccccc12 c1(CCC(=O)NCC(C)N(C(=O)CCC2CCCN2C)C)cccc(Br)c1 n1(CCCN(C(=O)Cc2nnnn2C2COC2)C)cc(-c2ccccc2)nn1 c1(C(N2CCC(N(C(=O)CNC(C)=O)CC)C2)=O)c(Cl)ccc(S(C)(=O)=O)c1Cl N1(Cc2cn(CCOC(C)=O)nn2)CCCN(C(C2(C3CCC3)CC2)=O)CC1 C1(CNC(=O)Nc2cc(C(C)C)nn2C)CC(N)C12CCC2 c1(C(=O)NCC(CNC(C(C)OCCCC)=O)C)ccc(N(CC)CC)cc1 C12(CNC(C(COCC)C)=O)CC(NC(c3ccsc3C(F)(F)F)=O)(C1)C(C)O2 CCC(C#N)(CC)C(=O)NCC1CN(C(c2cc(CC(C)C)c[nH]2)=O)C(C)(C)C1 C1(NC(c2c(CC)nn[nH]2)=O)(CNC(C2CCCCC2OC)=O)CCC(F)(F)CC1 C(=O)(C(CCO)N(C)C)NC(C1CCN(C(c2cccc(Cl)c2)=O)C1)C C1(C(=O)NC(C#CC)(C)C)CC=CCN1C(=O)CC(C)N(C)C N1(C(C(CN(C(CN(C)CC)=O)C)C)=O)CC2OC(=O)N(C)C2C1 N1(CCC)CCC(NC(c2ccc(CNC(C3CC3C(F)F)=O)cn2)=O)CC1 N1(c2ncc(C#N)nc2)CC(C2CCCN(C(=O)C(C3CCCCC3)O)C2)C1 N1(C(c2c(OC)ncnc2)=O)CCC2CN(C(=O)C3=NNC(=O)CC3)C(C)C12 Cc1cc(C(=O)Nc2cccc(NC(c3ccn(CC(F)F)n3)=O)c2)nc(O)n1 N1(C(C(CCCC)O)=O)CCC2(CCC(N(C)C(C3CCS3(=O)=O)=O)CC2)C1 c1(NCC)cccnc1C(N1CCCC1CN(C(C12CCCC1C2)=O)C1CC1)=O Cc1cc(CC(=O)NC(C(=O)N(C)C(C2CCCC2)C)C(C)O)n(C)n1 C(=O)(CS(=O)(=O)C1CC1)NCC1CCCC(CNC(C2C(CC)CCC2)=O)C1 C(CC(C)C)(C(=O)NCC1(F)CC(CNC(=O)CC2CCCC2(F)F)C1)OC C12(NC(c3c(C)nn(CC)c3C)=O)CCOCC1CN(C(=O)C(C)(C)C1CC1)C2 c1(C(N2CCC(F)(CNC(CN3CC(C)(C)C3)=O)C2)=O)cc(F)ccc1O N1(C(CNC(=O)OC)=O)CCCC2(NC(c3cnc(O)n3C)=O)CCCC12 n1(Cc2cc(C)no2)nnc(C(=O)NC2CC(N(C)C(C3CC3C)=O)C2)c1C Cc1n[nH]c(C)c1SCC(N1CCCCC1C(C)NC(c1cc[nH]c(=N)c1)=O)=O C12(CNC(CC(C)NC(c3nc(CC)oc3)=O)=O)CCC(CC1)CC2 C1(NC(c2ncc(OC)cc2F)=O)CCN(C(=O)CC2CC=CC2)CC12CCC2 Cc1ncccc1C(N1CC(NC(=O)C(c2ccccc2)C2CC2)C(O)C1)=O C(=O)(C(C(=O)NC(CNC(=O)Cn1nccn1)C1CCC1)C(C)C)OCC C1(C(=O)NC(CCCC=C)C)CC(C)CCN1C(=O)C(C)N1CCCC1 N1(C(c2[nH]c(=NC)sc2)=O)CCC(NC(=O)Cc2ccsn2)C(C)C1 N1(C(C2(C)ON=C(C)C2)=O)CC(NC(c2ccc(CCF)cc2)=O)CC(F)(F)C1 c1(CC(=O)NC(CCOC)CNC(=O)C(O)C2CC2)ccc(OC)c(Br)c1 c1(C(=O)NCCC(C)NC(C2(C)CCCCC2)=O)n[nH]c2c1CCC2 c1(OCC(=O)NC(C)C(C)NC(C2CC(C(F)F)C2)=O)cccc(Cl)c1 CC(CC(=O)N1CCC(Cn2cc[n+](C)c2)C1)CNC(F)F C1(CN(C2CC(=C)C2)C)CCC(OC(=O)C(CCOC)OC)CC1 CN1CCC(C)(C(=O)NC2C3CC4C2C4C3C(=O)NCC2CCCC23CC3)CC1 CCC(CC)(C(=O)NCCC1(O)CN(C(c2nnn(C)c2C(F)F)=O)C1)C(C)C c1(NCC2N=CN(C)C2)ccc(-c2ccc(C(F)(F)F)s2)cc1 c1(C(N(C2CC(NC(Cc3cn(C)nc3)=O)C2)C)=O)cc2nccnc2cc1F C1(C)(C(N(CC(C)N(C)C(c2ccco2)=O)C)=O)CCCCC1(F)F Nc1cc2ccccc2c(C(=O)NCC2CC(NC(C3CC(F)C(=O)N3)=O)C2)n1 N1(C(C2C(=C)C2)=O)CCCCC1CCN(C(=O)COCCCF)C C1(C(N2CC(C)(C)OCC2)=O)N(C(C2CC2[N+](=O)[O-])=O)CCCC1(C)C Cc1ccc(O)cc1C(=O)NC(CO)C(C)NC(=O)Cn1nc(C)c(Cl)c1C Cn1c(=O)oc2cc(-c3cc(CNC4CCc5ccccc54)c(=O)n(C)c3)ccc12 c1(C(=O)Nc2cnc(CCCC)nc2C)cc(S(N)(=O)=O)cn1C N1(C(=O)NC(c2ncc(C(F)(F)F)s2)C2CC2)CCOC(c2ccc(Br)s2)C1 CC1CCCCC1CC(=O)NC1CC(NC(=O)C(C)(F)F)C(O)C1 c1(CC(=O)NC(C2CCCN2C(c2ccc(C(=O)OC)o2)=O)C)csc(S)n1 C=C=CCC(=O)NCCCOCCNC(C1(C)CCCO1)=O N1(C(CCCOC(C)C)=O)CCCC(CN(C(=O)C=CS(C)=O)C)C1 N1(C(CCc2cc(C)on2)=O)CCN(C(c2cccn(C)c2=O)=O)C(C)C1 CC(C)CCCCC(=O)N1CCN(C(=O)CCCSc2ccccc2)CC1C c1(C(=O)NCCC(=C)CNC(C2(OC)CCSC2)=O)cc(C)c(F)cc1F N1(CC(=O)NCc2cc[nH]c2)CCN(C(=O)COc2ccc(O)cc2)CC1 C1(NC(CN(C(C)=O)C)=O)CCC(NC(=O)CCC2CC2(F)F)C1 CCCC(C)C(=O)NCCNC(=O)CCc1ccc(CO)cc1 c1(N2CC(c3ccccc3)(NC(C=CS(C)(=O)=O)=O)C2)ccc([N+](=O)[O-])cc1F C(C1CCCCc2ccccc21)NC(Cn1cc(-c2cc(C)c(F)nc2)nn1)=O c1(C(=O)NCC2CCN(C(CC)=O)CC2C)cc(SC)c(OC)cc1[N+](=O)[O-] CC1CCn2cc(C(=O)N(C3CN(C(c4cnc5nccn5c4)=O)C3)C)nc2C1 C1(Cn2cc(-c3ccc(C)s3)nn2)CCCN(C(=O)Cc2cnccc2C)C1 c1(CCC(N2CCN(CCNC3CC3)CC2)=O)c(F)cccc1F O=C(C1=COCCC1)NCC1CN(C(=O)CNC(c2ccoc2)=O)CC1(F)F c1(C(N(CCNC(C2(F)CC(C(=O)OCC)C2)=O)CC)=O)cccc(Cl)c1C c1(C2C(C(=O)Nc3cccc(C4CNC4)c3)C2)c(Cl)cccc1Cl N1(C(C(C)NC(N)=O)=O)CCOCC1CNC(=O)C(F)(F)c1cncs1 C1(C(C)C)N(C(c2cc3c(s2)CCC3)=O)CC12CCN(C(=O)CCCF)CC2 C1(C(=O)NC2(CCNC(CC3(COC)CC3)=O)CC2)COCC1C(N)=O C#CC(C)(C)C(=O)NCC1(C(=O)Nc2ncoc2-c2cccs2)CC1 c1(C(=O)NC(C)CCNC(C2CC(O)CN2C)=O)ccc2nc(O)n(C)c2c1 N1(C(CCC=CCC=C)=O)CCN(C(=O)COCC=C)C(c2ccccn2)C1 C1(C(=O)NCC2C(CNC(CCCNC(=O)OC)=O)C2)CCC(=O)N(C)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)NC1(C)CCCN(C(CSSC)=O)C1 N1(C(C(CC)OCC)=O)CCC(NC(=O)C(C)C2CCOC2)C(C)(C)C1 N1(C(CC2OCCN(C(c3c(C)snn3)=O)C2)=O)CC2CCC1C(O)C2O CC(CC(=O)NCC1CCCCN(C(=O)CS(C)(=O)=O)C1)CC(F)(F)F CC(CCCNC(=O)CNc1cn(C)nn1)NC(=O)CCC1CCCCO1 c1(CC)cc(C)ccc1C(=O)NCCCC(C)NC(=O)CSCC(=O)OC CCN=c1[nH]cc(C(N2CC(NC(=O)CCNC(C3CC3C)=O)C2)=O)s1 C(CN=C(NCC(F)=C(C)C)NCc1cc(C(F)(F)F)nn1C)CCC=C Cc1cc(Br)c(CN(Cc2ccccc2)Cc2cnn(C)c2)s1 n1(C2C(C(N(C(C(=O)OC)C)C)=O)C2(C)C)cc(CSC)nn1 N1(C(CC2(COC)CC2)=O)CC2C(NC(C3CCCOCC3)=O)CS(=O)(=O)C2C1 c1(C(=O)NC2CC(NC(C3(C(=O)O)CC(F)C3)=O)C2)cc2cc(F)c(F)cc2[nH]1 N1(c2ncc(C)cn2)CCC(C2CC2)(CN(C(=O)CC2(C)CCS(=O)(=O)N2)CC)C1 N1(C(C2C(C(=O)OC)C2)=O)CCC(C(F)C(=O)NCC2CC3(CC3)C2)C1 CCC(CC(=O)NC1CC(NC(C2CCOC2(C)C)=O)C1)c1ccccc1 C(=O)(CCCC#N)N1CCC(c2c(CNC(C3(C)C(C)(C)C3)=O)c[nH]n2)C1 N1(C(Cc2c(C)ccs2)=O)CCCC(O)(CNC(=O)CCCc2cnccn2)C1 C1(CC#C)(C(N2CCC(CCCO)C2)=O)CCCN(C(=O)OC(C)(C)C)C1 C#Cc1ccnc(C(=O)NC2CCN(C(c3nccc(OC)c3F)=O)C(C)C2)c1 C12(C(=O)Nc3c(CC)nccc3)CC(CO1)N(C(=O)Cn1cc(C#N)cn1)C2 C1(CNC(C(CCC)OC)=O)CCC(C)(C)CN1Cc1ncccc1Br c1(OC(C)C)ccc(C(N2CCC2CNC(=O)Cn2cc(N)cn2)=O)cn1 c1(CC)conc1C(=O)N(C(C)(C(=O)NCC1(CC)CCCO1)C1CC1)C C(=O)(CC(C(C)(C)C)NC(C1CCC(C)(C)CC1)=O)NCC1(COC)CCCC1 C1(NC(c2cnccc2Cl)=O)CC(CNC(=O)C(C2CC2)C2CC2)C12CCC2 C1(C(N2C(CC)(CC)CC2)=O)CCN(C(=O)C(c2ccnn2C)C)C1C C1(NC(c2nn(CC)nc2C)=O)CCN(C(=O)CO)CCC1CO C1(NC(C(C)Cc2ccccc2Cl)=O)CC2(CCN(C(=O)Cn3cccn3)C2)C1 c1(OC)cnc(Cl)cc1C(N1CCCC(C)C1CNC(c1c(C)nsc1N)=O)=O c1(C(=O)NC(CCCCNC(C2C(C)C2)=O)C)ccc(Cl)c(Cl)c1 c1(CNC(=O)CCN(CCO)C(C2CCCS2)=O)ccc(F)cc1 Cc1ccc(C(=O)NCC2CC3CCC2N3C(=O)C2=CCCCO2)c([N+](=O)[O-])c1 C=CCN=C(NCC(N1CCc2sccc2C1)C)N1CCC(C2CC2)C1 N1(C(CC)CNC(C2CCCN(C(C)=O)C2)=O)CCOC(COCC)C1 C1(C(N(C)CC2CC(F)CN2C(C2(CC(F)(F)F)CC2)=O)=O)CC(=O)NC(=O)C1 Cc1ccccc1CC(C1CCNC1)NC(c1csc(-c2ccoc2)n1)=O C12(C(=O)NC(CN(C)C(c3cn(CC4CCCO4)nn3)=O)(C)C)COC(CCO1)C2 N1(C(CCCC)=O)CCN(CCNC(=O)Cc2ccc(F)c(F)c2)C2(CCC2)C1 C1(CNC(COCCC=C)=O)CN(C(c2cc(C)oc2CC)=O)CC1C(F)(F)F CC(C)C(C)C(=O)NCCC1CCN(C(=O)C(Cc2ccsc2)N(C)C)CC1 N1(C(C(C)(C)NC(N)=O)=O)C=C(Br)CC(C(=O)COCC(F)(F)F)C1 C1(CNC(C(=Cc2cccs2)C)=O)CN(C(c2cc(Cl)n(C)n2)=O)CCN1C Cc1cc(C(c2nnnn2CCOCC2CC2)NC2COCCOC2)nc(Cl)c1Br C1(OC)CN(C(=O)CC2CC(C)(C)CO2)CC1NC(=O)C1=C(Cl)CC1 N1(C(C(OC)OC)=O)CC(CNC(=O)C(C)Cn2ccnc2)CC(C)(C)C1 CC(C)CC(C)CC(=O)NCC1CCN1C(c1ccc(CO)cn1)=O Cc1ccc(C)c(C(=O)NC2CC(F)CN(C(=O)Cn3nnnc3C(C)C)C2)c1 CCCCCCN(C)C(C1CC(C)(NC(c2nsnc2O)=O)C1)=O c1(CC(N2CCN(CCNC(C)=O)CC2)=O)cc2cccnc2nc1C N1(CCC(N2CCC(C(C)NC(C34CC3C4)=O)C2)=O)C(=O)CCC1=O C1(NC(C(C(C)C)NC(c2c(CC)[nH]cc2)=O)=O)CC(F)(F)C1(C)C C12CCC(CC1)C(=O)N2C.n1(CCCNC(=O)Cn2cccc2)ccnc1 Cc1cc(F)cnc1C(=O)NC(CC(N)=O)C(=O)Nc1cnccc1CO C(CC(C(=O)NC1CC(=O)N(C(C)C)C1)NC(c1ccon1)=O)SC c1(SC)nc(N2CC3CC(NC(=O)C(C)(F)F)C3C2)cc(C)n1 N1(C(Cc2nc(C(C)OC)sc2)=O)CC2CC1CCN2C(c1oncc1C)=O c1(OC)cc(SC)ccc1C(=O)NCC1CCC(CNC(=O)C(C)C(C)C)CC1 c1(N(C)C(c2ccc(P(C)(C)=O)s2)=O)cc2ccccn2n1 C(C(CC(=O)NCc1cccnc1)C1CCC1)NC(c1c(CCC)[nH]cc1)=O CC1(C)CCN(C(c2ccc(=O)oc2)=O)CC1NC(C1CCCSC1)=O Cc1cccc(C(F)C(N2CCC(O)(CCNC(c3ccco3)=O)C2)=O)c1 C12(C(=O)NC3CN(C(C)=O)C3)CC(CN(C(c3cnn(C)c(=O)c3)=O)C1)C2 C(c1cccc(F)c1)=C(C(=O)NCCC1(NC(C(CC)O)=O)CC1)F c1(N(C)C)ccc(C(=O)NC2CCCC(N(C(=O)C=Cc3cn[nH]c3)C)C2)cc1 CC(C)CC(C(=O)NCC(C)(C)C(=O)NCc1nc(CO)n[nH]1)C(C)C c1(C(N2CC3(OCC(NC(CC4(C)CC4)=O)C3)C2)=O)ccc2cc(O)ccc2c1 C1(C(=O)NCCC2(NC(C3CN(S(C)(=O)=O)C3)=O)CCC2)CC2C=CC1C21CC1 c1(CNC(=O)COc2ccc(Cl)nc2)ncnc(C2CC2)c1Br N1(C(c2ccc(N(C)C)cn2)=O)CCN(Cc2ccc(Cl)s2)C2CC12 C1(NC(c2ccccc2Br)=O)CCN(C(C2CCC(F)(F)CO2)=O)C12CC2 c1(C(C(=O)NCC(CC)NC(c2sc(C)nc2CC(C)C)=O)=O)ccc(C)cc1 c1(CNC(C2C(C)C2C)=O)cc(C(=O)NCC(C)N(C)C2CC2)n[nH]1 C1(C(N2CC(C)SCC2)=O)C2CCCC2CN1C(C1CC1[N+](=O)[O-])=O C(=O)(CCC(C)N(C)C)NCCCNC(CN(C(COC)=O)C)=O CC(C)(F)CCC(=O)NC1(C(N2CCC(C(F)F)CC2)=O)CC1(C)C Cc1ccn(CC(N2CCC(C(C)(C)NC(c3ccc[n+]([O-])c3)=O)C2)=O)c(=O)c1 C(=O)(C1CCCn2ccnc21)NC(CC)CNC(=O)CC1CC(OC)C1 C(c1cnc(O)nc1O)=CC(=O)NCC1(O)CCCN(C(C2CCC2)=O)C1 CC1(C)CC(NC(c2[nH]ccc2C2CC2)=O)CN(C(c2cccc(=S)n2O)=O)C1 CC1CCC(C)(NC(C2(C)CCCN2C(=O)CN2CCC(=O)CC2)=O)C1 O=C1CC(=O)CC(C(=O)NC2(C(=O)NC3COCC3N(C)C)CCCC2)C1 Cc1cc(C(C)C(=O)NC2CCC2C2CC2)c(C)o1 N1(CCC)CCCC1C(=O)NCCC1(C(=O)N(C2(O)CCOC2)C)CC1 C1(CC(N2C(C(=O)NC)C=CC2)=O)CN(C(C2C=CC2C(=O)OC)=O)CC12CC2 C1(NC(=NCC=C)NCc2cn(CC)nn2)COC2(CCOCC2)C1O C1(C(N(C2(C(N3CC(C(C)(C)C)C3)=O)CCC2)C2CC2)=O)CCOC(=O)CC1 CC1=NOC(=O)C1CCC(=O)NCC(CNC(c1n[nH]cc1Cl)=O)CO C1(CNC(C(=Cc2cn[nH]c2)C)=O)CC(C)N(C(=O)CCc2ccccc2)C1 CCC(C(=O)NC)NC(C1CCN1Cc1nc(C(C)C)cs1)=O N1(C(c2cncc(OCC)c2)=O)CCOCC(NC(c2cc(C(F)F)on2)=O)C1 C12(NC(C3CC(OC)C3)=O)COC(C1)C(NC(=O)C(C)c1ccsc1)C2 C(=O)(CCCCN(C)C)NCC(C)C(=O)NCC1CC1c1ccoc1 N1(Cc2ccc(C(=O)OC)o2)C(=O)CCN(Cc2ccnc(C(F)(F)F)c2)C1=O C12(CCNC(C3CN(c4ccc(Br)cc4)C3)=O)COC(CF)(C1)C2 C1(CC)(CC)CCN(NC(c2ccccc2)C(N2CC3C=CC2C3)=O)CC1 C#Cc1cc(C(N2C3CCC2CC(NC(C2(O)CC2)=O)C3)=O)cc(F)c1 c12ccnc(n1)N2.C1(NC(C2C(=C)C2)=O)CN(S(C)(=O)=O)C1 N1(C(C2N(C)C(C(N)=O)CC2)=O)CC(CNC(C2CC(C)(C)C2)=O)OC(C)(C)C1 C(=O)(CCCc1csc(=N)[nH]1)NC(C1CN(C(C2C(C)C2(F)F)=O)C1)C C1(SCC)CCN(C(=O)CNC(=O)CNC(C2CCCCC2)=O)C1 C1(O)(CNC(c2c(C(N)=O)coc2)=O)CCCN(C(=O)C2=CCCCO2)C1 c1(C(C(=O)NC(C)CCNC(c2cnc(C(F)F)nc2)=O)(C)C)ncccc1F CCCCC(C)C(C(=O)NCCCC)N1CCC(CN2CCCC2=O)C1 C(C)(N=c1nc2c(cnn2C)c(NCc2nccn2C)[nH]1)c1c(C)c(Cl)ccc1 c1(NC(C2CCCN2C(c2ccc(C(F)(F)F)nc2)=O)=O)cnc(Cl)c(Br)c1 c1(C(=O)NCCCN(C(C2(C)C(C)OCC2)=O)C)ccc2cc(Br)ccc2c1 c1(C(=O)NC2CC(CNC(C3(c4cccc(F)c4)CC3)=O)C2)ccn2ccsc12 c1(C(=O)NCC#CCNC(C2(n3cc(Br)cn3)CC2)=O)ncccc1O N1(C(C(CC)n2cncn2)=O)CCC(C(C)(C)C)(CNC(=O)COCC(C)C)C1 C12(C(=O)NCC(=O)N(C)C)CCCC1CCN2C(C1CCS(=O)CC1)=O C1(CC=C)(NC(=O)C(Br)=C(C)C)CCCN(C(c2cc(Cl)ncc2F)=O)C1 C1(C(=O)NCC(C)CNC(=O)CCc2cncs2)CC12CCCC2 c1(C(=O)NCCCCNC(c2cc(F)c(CO)c(F)c2)=O)cc2cn[nH]c2cn1 CC1CCC(=CC(=O)NCC(c2ccccc2)NC(c2scnc2C2CC2)=O)C1 c1(CC)conc1CC(=O)NCC1CN(C(=O)CCn2ccnc2C(C)C)C1 C1(COCCCN)CCCN(S(=O)(=O)Cc2cccc(Br)c2)C1 CC1(OCC(=O)N(c2ccccc2)CC2CC2)CN(C(=O)C=Cc2cocn2)C1 c1(C(=O)NC2C(NC(C3(C)CC=CCC3)=O)CCC2)cnnc2ccccc12 N1(C(CCCc2ncc(C)o2)=O)CCCN(C(=O)Cn2cnnn2)C(C)C1 C1(C(c2n(CCCOC)nnn2)NCc2sccc2Br)CCCCCC1 c1(C(N2CCC(NC(c3cc(C)nnc3)=O)C2)=O)ccc2c(Br)cccc2c1 c1(C(=O)NCCN(C(C(C)SCCCC)=O)CC(C)O)ncoc1CNCC Cc1ccccc1C(O)C(=O)NCc1nccn1-c1ccccn1 Cc1ccc(-c2ccccc2)c(NC(=O)C(CC(C)C)N2CCCC2=O)n1 N1(C(c2cc(CCC)on2)=O)CCC(C)(C)C(C(=O)NCC(C)(O)COC)C1 N(C1CC(C)n2ccnc21)C(CN(C(CNC(C=CC=CCC)=O)=O)C(C)C)=O Cc1nc(C(C)NC(C2OCCC2NC(=O)CC23CCCC2C3)=O)n[nH]1 N1(C(C2C(C)(Br)C2)=O)CCC2(CCN(C(=O)C(=Cc3c[nH]cn3)F)C2)C1 C(C(=O)NC1(C(N2CCCC(CC(C)C)C2)=O)CSC1)(C(C)C)OCC C(N=c1cc(NCCOC(F)(F)F)nc(C(F)(F)F)[nH]1)c1c(=N)cc[nH]c1 Cn1ncc2c(C(N3CCN(C(=O)CCC4CC4(F)F)CC34CC4)=O)ncnc12 c1(OCC)cc(C(N2CCCCC2CC(C)O)C(=O)NCc2cccs2)ccn1 Cc1cc(C(=O)N(C(CNC(C2(O)CC(F)(F)C2)=O)C2CC2)C)n2nccc2n1 c1(C(=O)NCC2C(NC(c3nc(C)sc3C)=O)CCC2)ccc(Cl)c(O)c1N c1(SC)cccc(C(N2CCCCC2CCNC(c2cnc(C)cn2)=O)=O)c1 CC1(CNC(C2CC2c2cccs2)=O)CCN(C(=O)CCN2CCOC2=O)CC1 CC(C)C(CNC(=O)C(C)(C)C)NC(c1ccnn1CC#N)=O N(C(=NCCC(=O)N(C)C)N1CC2C(C(N)=O)C2C1)CC1C(C)CCCC1 c1(C(=O)NCC(CC)(CC)NC(c2nocc2C)=O)cc2cnccc2o1 Cc1ccn2cc(CN(C)CC34CCC(CC3)C4)nc2c1 CC1CN(C(c2ccno2)=O)CC(C(N2CCOCC(C(=O)N(C)C)C2)=O)O1 n1(CC(=O)NC2CCC(NC(c3cc(C(C)C)[nH]n3)=O)C2)cc(P(C)(C)=O)cn1 C1(SC)CN(C(c2csc(-c3ncccn3)n2)=O)CC1NC(c1cnoc1C)=O c1(C(C(=O)NC2CC2)N(CC)CC2CCOC2)ccc(-c2nc(=O)o[nH]2)cc1 c1(NC(=O)CC2CCN(Cc3ccnc(Cl)c3)C2)cccc2ncccc12 CCC(C(=O)N1CCCC(COC)(NC(=O)C=C(C)C(C)(C)C)C1)C(C)C CC(C)CC(C)OCCC(=O)N(CCNC(c1cc(C2CC2)on1)=O)C1CC1 N(C(=NCCc1ccncc1)NC1CCOCC1)CCN1CC(C)C(C)C1 C1(C(=O)NC(C(=O)N(C)CC)C)CNC(=O)CN1C(=O)C=Cc1cc[nH]c1 C1(C(=O)OC)C2CC2CN1C(c1coc(CNC(=O)C(C)CSC)c1)=O C(N=c1cc[nH]cc1S(=O)(=O)NC1CCN(CC(C)C)C1)c1ccc(SC)nc1 c1(CNC(C2CC2NS(=O)(=O)c2nccs2)=O)ccc(Br)cc1F N#Cc1ccc(CN2CC3(CC(C(=O)Nc4cc(Br)cnc4O)C3)C2)cc1 NS(=O)(=O)c1ccc(Cl)c(S(=O)(=O)NC(c2cnc3c(c2)CCNC3)=O)c1 CC(CC(C)(F)F)C(=O)N1CC2(C1)CN(C(=O)CS(=O)(=O)NCC1CCCO1)C2 N1(C(C(CC)OC)=O)CCC2(CCCCC2NC(C2CCC3CC2C3(C)C)=O)C1 C(CCC(=O)NC(CN(C)C(C)=O)Cc1ccccc1)OCC.C(=O)CC c1(CN2C(C(=O)NC(c3ccc(Cl)cc3)C)C3CCC2C3)cc(Cl)cc(Br)c1F c1(OCC)ccc(C(=O)NC(C)CCCNC(=O)CC2CCC(O)C2)cc1OC CCCCC(C)C(=O)NCCCCCN(C(=O)CNc1ccc(C(N)=O)cn1)C Cc1cc(NC(=O)NCC2(C(=O)Nc3ccc(F)cc3F)CC2)cc2ccsc12 C1(C(=O)NCC2(S(N)(=O)=O)CC2)CC2(CCC2)CN1C(=O)CC1=CCCCC1 C1(NC(COc2cccc(C)c2)=O)CN(C(C2CSCC(=O)N2)=O)CC2(CC2)C1 N1(CC(c2ccc(OC)cc2)C)C(=O)NC(CCc2ccns2)C1=O C(C(CC(C)C)C(=O)NCc1cc(C(C)C)no1)NC(c1c(NC)cccc1)=O N1(Cc2ccc(C(=O)OC)nc2)CCC(C(=O)Nc2cccnc2O)C(O)C1 C(CCC(C)(C)C(=O)NC(C)C(=O)NC1CC1)NC(CCn1c(C)ncc1)=O c1(CN2CCC(C(=O)NCCCOCC(F)(F)F)C2)n[nH]c2ccc(Br)cc12 Cc1c(C(N2CCCCC2CC(N2CC3C(C2)C3(C)C)=O)=O)cccc1F C#Cc1ccc(NC(C2CC23CCN(Cc2c(F)cccc2F)CC3)=O)cc1Cl N(C(=NCCCOCc1ccc(C2CC2)cc1)NCC1CC1)CC(CC)(O)CC Cc1nc2ccc(C(N3CCC(=CCNC(C4(C)CC4(Cl)Cl)=O)CC3)=O)cc2[nH]1 O=C(CCCCC(F)F)NC1CCCN(C(c2nnn3c2CSCC3)=O)C1 C1(NC(C(C(C)C)SCC)=O)C2CC3CN(C(=O)CCN(C)CCO)C1C3C2 C1(CNC(=O)NCC(c2ccccc2Cl)N(C)C)CC2(CCOCC2)CO1 CC1(C)C2CCC1(CS(=O)(=O)NC13COC(C1)C3)C(=O)C2.N12CCC(CC1)C2=O Cc1cc(C(F)F)oc1C(=O)NCC1C(C)CCN1C(c1cnn[nH]1)=O c1(C(=O)NCC2(CNC(C(C(C)(C)C)SC)=O)CC2)cc2c(C)ccc(F)c2o1 c1(C(=O)NC(CC=C)(C)C)ccc2cc(Cl)ccc2c1 c1(C2C(C(N3CC(C)(NC(COCCCC#C)=O)C3)=O)C2)cccc(F)c1 C1(C(=O)NC2CC(CNC(CCCn3c(C)csc3=O)=O)C2)CCC2CC2CC1 S(=O)(=O)(c1ccc(Br)s1)NC1CC(NC(c2cc(C)c(Cl)cc2)=O)C1 CC1CN(C(=O)CC2CCC(C)(C)C2)CCN(C(=O)C(O)CC(F)(F)F)C1 c1(C(N(CCC(C)NC(C=CC)=O)C)=O)sc(CC(C)C)nc1C CC1=NS(=O)(=O)NC=C1C(=O)N1CCN(C(C2CC3CCCC23)=O)CCC1C c1(NC(=O)NCC(CNC(CNC(CNC(C)=O)=O)=O)C)nonc1N C1(C(=O)OC)(C(=O)OC)CCCN(C(=O)CCc2cnc(OC)c(Br)c2)C1 S(=O)(=O)(c1cccc(N(C)CC2CCN(C)C2)n1)N1CCN(CC)C(C)C1 c1(OC)ccc(C(=O)NC2CCN(C(=O)Cc3ccccc3SC)C2)cc1Cl CC(C)S(=O)(=O)c1cccc(C(=O)NCCC(O)CNC(=O)CC2(C)CCC2)c1 C1(CC)CN(CC(c2nc(-c3ccc(OC)cc3)oc2C)=O)CC(CC)O1 C(=O)(CCC[N+](=O)[O-])N(CC)CC1CCN(C(C2CC(C)(C)CO2)=O)CC1 C1(CN(C)Cc2nc(C)[nH]n2)CCCN(C(c2ccc(S)cc2)=O)C1.N(C)C CC(C)(C)C(O)C(=O)N1CCC(n2cc(CNCC3CCC(F)(F)CC3)nn2)C1 C12(NC(CCC#CC)=O)CCCN(C(c3ccc[nH]3)=O)C1C2 C(N=c1cc(NC2(C)C=CCCC2)nc[nH]1)C1(N(C)C)COC1 C1(N(C(C(C2CCCC2)OC)=O)C)CCCCN(C(c2cncc(C)c2Cl)=O)C1 C(CC1CCCC1)(C(=O)NC1CCC(C(N2CC(N(CC(C)C)C)C2)=O)C1)OC N1(C(c2c(C)cccc2F)=O)CC2CC(NC(C3(C)CC3(F)F)=O)CC(C2)C1 c1(C(N2CC(CNC(C(C)OCC3CCCO3)=O)C2)=O)cc(C(F)F)cnc1O c1(C(N2C(CNC(C3Cc4ccncc4C3)=O)C=CC2)=O)cnn2c1NCCC2 N1(C(C)=O)CCCC(NC(=O)C(C(C)C)NC(=O)C=CC2CCC2)C1 c1(C(N2C(C(N(C3CCCOC3)C)=O)CC2)=O)ccoc1CNC(=O)C1CC1 c1(NC(CN(C(C=C(C)C2CC2)=O)CC(C)C)=O)cnc(C)c(Cl)c1 C1(NC(C2CCN(C(C3CC(F)(F)C3)=O)CC2O)=O)C2CCC3C(C2)CC13 c1(C(=O)NCCN(C)CS(C)(=O)=O)ccc(OCc2ccc(C3CC3)cc2)cc1 N1(C(C(C)NC(CC)=O)=O)CCC(O)(CNC(c2cc(CC3CC3)on2)=O)CC1 CCCC(CC)CC(=O)NCCC(C)NC(=O)C#CC1(C)CC1 Cc1ncc(Cl)cc1C(N1CC(F)(F)CC1CNC(C1CCCC(=O)N1C)=O)=O C1(COC)(NC(c2cncc(C)c2Cl)=O)CCCCC1C.c12cc([nH]n1)C(=O)N2 C(=O)(C(C#N)C(C)(C)C)NC(CCCC)CNC(=O)CCSC C(=O)(C(C)CC(C)(F)F)N(CCCCCCNC(c1c(C(C)C)c[nH]n1)=O)C N(C(=NCc1cc(C(C)(C)C)on1)NCC(=O)N(C)C)CC(NOC)=O N1(C(c2cnc(CC)n2C)C(=O)NC(C)CC)CCn2c(C)nnc2C1C C1(C(N2CCC(CCCC)C2)=O)CC2(CC(NC(=O)C=C3CCC3)C2)C1 c1(C(N2CC(NC(c3nn(CC)nc3C)=O)C(C)CC2)=O)cccn2cncc12 C(=O)(CP(C)(C)=O)N(C)CCn1cc(-c2cnn(Cc3ccccc3)c2)nn1 Cc1nccc(C(=O)NC(C2CCN(C(=O)C(C)NC(=O)C3CC3)CC2)C)c1Cl c1(C2(C(c3nnnn3C(C)C)NC(C=C)C3CC3)CC2)ccc(Cl)cc1 C(CC1CC1)(CC(=O)N(C)CC1CCOC1C)NC(C1(Cl)C(C(C)=O)C1)=O n1(C(CC)C)nccc1C(=O)NC1(CNC(c2csc(Br)n2)=O)CCC1 N1(C(Cn2ccc(C)n2)=O)CC(C(=O)NC2CC=CCC2C)CC1(C)C C1(C#N)(CC)CCN(C(=O)CC(C)(C)NC(=O)CCc2csnn2)CC1 c1(C(=O)NC23C(CN(C(CCC=C=C)=O)C2)CC3)cc2ccc(OC)nc2[nH]1 c1(CC(=O)NC2CN(C(c3c(C)[nH]nc3C(C)C)=O)C2)ccc(Br)cc1C#N c1(OC)ccc(Br)c(C(=O)NC2CCCC(NC(=O)C(C)OC(C)(C)C)C2)c1 C(=O)(CC(C)(C)Cc1ccccc1)N1CCN(Cc2cnc(C)n2C(F)F)CC1 C1(O)(CNC(c2cc(CNC(C(C)N(C(C)=O)C)=O)oc2)=O)CCC(C)C1 NC1CN(C(=O)CC2COCCO2)CC2(CC2)C1 C(=O)(C(CC(C)C)C(N)=O)NCCCN1CCN(C(c2cc(C)ncc2)=O)CC1 C12(NC(CC(CC)C(F)F)=O)CCCC1(F)CN(C(C1CCCC1OC)=O)C2 c1(C(=O)NC2(C)CC(NC(CC=CC=C)=O)C2)ccc(COC)c(F)c1 CCC(C)C(O)C(C)C(=O)NCC(CC)(CC)NC(c1cc(Cl)ccn1)=O Brc1cc(I)cnc1NC1(c2ccccc2)CCCOC1 C1(C(C(=O)N(CC(CC)NC(=O)CCOC(C)=O)C)F)CCOCC1 c1(C(=O)NCC2C(NC(c3c(C)cc(=N)[nH]c3)=O)C2)cc(C)n(NC(N)=O)c1C CCC(C)C(C(=O)NC1CCC(CNC(c2ccc(N)cn2)=O)C1)OC C1(C(N2CC(C)C(NC(c3c(C#N)cnn3C)=O)C2)=O)CCC(C2CCC2)CC1 C1(C(=O)NCc2cnc(CC(C)C)[nH]2)COCCC1NC(C1CCC1)=O C1(CS(C)(=O)=O)CCCN(C(c2ccccc2F)=O)C1 c1(NCCC)ncccc1S(=O)(=O)NC(c1ccc(Br)cc1)C(C)C N1(C(C2CC(C#C)(O)C2)=O)CC(NC(C2CCN2CC)=O)Cc2ccccc21 C1(C(=O)NC2(C=C)CCCC2)COCCN(C(C2CCN(C)C2=O)=O)C1 Cc1n[nH]c(C)c1CC(=O)NC(C1CN(C(c2cc(C#N)on2)=O)C1)C c1(C(=O)NCC(C)NC(c2c(COC)n(C)nc2)=O)scc2c1OCCO2 c1(CNC(C2CCCCC2)C(=O)OCC)cccc(OCc2ccccn2)c1 c1(C(=O)NC2(CN(C(c3cc(OC)ncc3)=O)C)CC2)ccc(P(C)(C)=O)s1 Cn1cncc1C(C1CCCC1)NCC1CCCCO1 N1(C(c2c(CC)c[nH]c2)=O)CC(NC(C2CCCCC(=O)N2)=O)C(S(C)(=O)=O)C1 C(CC(C)C(=O)NCC(O)CCNC(=O)Cc1nc(C)sc1C)=CC c12cnc(nc1)[nH]2.N1(Cc2nnn(C)n2)CCC(C(=O)CN2CCCCC2)CC1 N1(C(c2nc(CNC(c3cccc(C)c3N)=O)oc2C)=O)CCOC(C)(C)CC1 CCC(CC(=O)N1CCC(COC)(NC(=O)CN(CC(C)(C)C)C)C1)C(C)C CCCC(CC)CC(=O)NC1CN(C(=O)CCC=C(C)C)CC12CC2 C(=O)(C(C(C)(C)C)NC(=O)CC1CCC(C)(C)C1)NC(CC#C)C(=O)OC N1(C(C2(NC(c3ccncc3F)=O)CCCC2)=O)CC2CCC=CC12 N1(C(C2CN(C(c3c(C)[nH]c(C#N)c3)=O)CC2F)=O)CCC2(CCOC2)C1 Cc1ccc(CCC(=O)NCCN(C(C2CCCC(F)C2)=O)C2CC2)cc1C c1(C(=O)NCCCc2cn(CC(=O)NCC)nn2)c(C)nc2cccnn12 c1(N2CCC(C)C2)ccc(C(C)NC(=O)OC2CCOC2=O)cc1 C1(CC=C)(C(N2CCCCC2CNC(c2ccncc2C)=O)=O)CCOCC1 CCC(C)CC(=O)N1CC(CC(C)NC(c2cnn(-c3ccccc3)c2Cl)=O)C1 c1(CC2(NC(=O)CCCF)CCN(C(CCC(C)SC)=O)C2)cccc(Cl)c1N c1(C(=O)Nc2cccc(C=C)c2OC)ncccc1N=c1nc[nH]cc1C#N c1(C(=O)OCc2nc(C)sc2)cccc(Cl)c1Cl.c12cn(nn1)C2C1CC(F)(F)C1 Cc1cc(C(N2CCC2CC(=O)NCC(C)C#N)=O)ccn1 c1(NC(C)=O)c(N)cc(Cl)cc1Cl.C1CCCCC(=O)NC2CN1C2 c1(N2CC(C)=C(C)CC2)[nH]c(=NCC2CC2(Cl)Cl)nc2sccc12 CC1CN(C(C2CS(=O)C2)=O)CC1CC(=O)NCc1ncnn1C1CC1 C1(OC)CCCCC1C(=O)N(C1CCN(C(c2ccc(Cl)cn2)=O)C1)CC1CC1 CC(CC(F)F)C(=O)NC1C2CC1N(C(C1C(F)(F)C13CCC3)=O)C2 c1(C(=O)NC(C2CCN(C(C(C=C)(C)C)=O)CC2)C)c(N)sc2c1CCSC2 c1(C(N2CC(CC(C)(C)CNC(=O)CN=S(C)(C)=O)C2)=O)cccc2cncn12 c1(SCCCC)cccc(CC(=O)NC(C2CCCN2C(=O)C(C)OC)C)c1 c1(C(=O)NCC(CN(C)C(C2C=CCC2)=O)(C)C)cc2cc(Cl)ccc2[nH]1 c1(NCC(CNC(c2c(SCC)cccn2)=O)O)ncnc(Cl)c1C(C)=O N1(C(=O)NC(c2onc(C)n2)c2ccccc2)CCCC2(CCN(C)C2=O)C1 N1(C(C2CC(NC(CCOC(C)=O)=O)C2)=O)CCCC(CCCO)C1 C(=O)(CCC(=O)c1ccccc1Cl)NC1(CCNC(=O)C=CC(F)(F)F)CCC1 N1(C(c2cccc(OC)c2)=O)CCCCC2C1CCCN2C(C1CC12CCC2)=O c1(CC(=O)NC2CN(C(c3ncn(CC)c3)=O)C2)cccc2cnccc12 C1(NC(c2ccnc(OC)n2)=O)CCC2CN(C(=O)CS(=O)(=O)N(C)C)CC2C1 Cc1c(-c2ccccc2C)o[nH]c1=NC(=O)c1ccc(C(N)=S)cc1 CN1CC(O)(CN(C)C(C2(CNC(=O)CC3COC(=O)C3)CCCC2)=O)C1 c1(CC2C(NC(c3cnc(OCC)s3)=O)C2(C)C)cccc(I)c1 N1(Cc2scc(C)c2)C(C(N2CCOCC2)=O)CC2CCCCC12 c1(C(N2C(C)CC(NC(=O)CCC3(C)CC3)CC2)=O)cncc2c[nH]nc12 C12(NC(c3c(C)n(C)nn3)=O)CCC(NC(c3coc(Cl)n3)=O)(CC1)C2 C12CC3(C1)CC3C(=O)N2.C(C(C)(C)C)C1C(C)C1.C1COCCO1 c1(OC)cccc(F)c1CNC(=O)NCc1ccc(-n2ccnc2C)cc1 S(=O)(=O)(c1ccc(NCc2ccnc(N(C)C)c2)nc1)NCC=C=C c1(C(=O)NC(N2CC(SC)C(N(C)C)C2)=O)ccc2c(c1)CCCO2 C1(NC(CN2CCN(C)C(=O)C2)=O)CCC2CN(C(=O)C3=CCSC3)CCC2C1 CCCCC(C(=O)NCC(C)(C)OCC(=O)Nc1ccc(F)cc1OC)C(C)C C(=O)(C(C)C(=O)NCc1ccc(C(=O)N(C)Cc2cocn2)o1)OC n1(CC(=O)NC2CC(NC(c3ncn(C)n3)=O)CC2O)cnc2ccccc12 CC1CC(CNC(C2CCCC2NC(=O)CN(C2CCC2)C)=O)=NO1 C=CCC(C)(C)CC(=O)NCCC1C(C)CCCN1C(=O)CNC(=O)OC c1(C(=O)NC2CN(C(CC(CCC)C)=O)C(C)CC2)cn(C)c(=O)nc1O N1(C(COC(C(C)NC(C2CC2(Cl)Cl)=O)=O)=O)CCc2ccccc21 N1(C(CCCOCC)=O)CC2CN(C(c3cc(Cl)ccn3)=O)CC2C1 C=CC(C)(CCOC)C(=O)NC1CCN(C(=O)C(C)CC(=O)OC)CC1CO c1(C(=O)NCC2C(C)(C)C(NC(=O)COc3ccccc3)C2)cc(F)ccc1Cl c1(CC)oc(C(=O)NC2CCOC(C(=O)N(CCO)CCN(C)C)C2)cc1C c1(C(N2CC(CNC(c3c(C)scc3)=O)OCC2)=O)ccc2c(c1)C(=O)NC2=O CN1CCCCC(C(=O)NC2CCN(CCNC(c3cnsc3)=O)CC2)C1=O N1(C(c2cccc(C)c2)=O)CCC(NC(c2c[nH]c(=O)cn2)=O)C2(CCC2)C1 C(=O)(CCS(C)(=O)=O)N(CCNC(C(C)=NOCC#N)=O)C(C)C Cc1cc(F)cnc1C(N1CCC(NC(=O)CN2CCCCCC2)C1C)=O c1(OCCC)ccc(C(=O)NCC(C)CN(C)C(c2cc(O)n(CC)n2)=O)cc1 C=CC1OCCC1CNC(c1ccc(Nc2cc(C)[nH]n2)cc1)=O C(=O)(C1=NOC(C(C)(C)C)C1)N1CC(NC(c2cc(COC)on2)=O)C(C)C1 c1(C(=O)NC(C)CNC(=O)C=Cc2nccs2)ccc(NCCC2COC2)cc1 Cc1cc(F)ccc1C(N1CCC(NC(=O)Cn2cccnc2=O)C1C1CC1)=O C1(CC=C)(C(=O)NCCN2CCCOC2=O)CCCN1C(=O)Cc1ccon1 C1(C(=O)NC(COC)COC)(NC(C2CCCSC2)=O)CCSC1 c1(C(=O)NCC(CN(C(C)=O)CC)(C)C)cccc(C#CCO)c1 n1(CCC=C)c(N(C)CC2C=CCC2)nnc1C(O)CC(C)(C)C C(=O)(C1=CCCCO1)N1C(CC(=O)NCC2CCC(C)CC2)CC(O)C1 c1(C(=O)NCCN(C(C2CC=CCO2)=O)CC)cnc(CC(C)C)s1 C12(C(=O)ON(C)C(C3CC3C(F)F)=O)CCCC1CCN2CC Cc1cccc2c(C(N3CCN(C(C4CC4(C)C)=O)CC3C(F)F)=O)cccc12 CCC(F)(F)C(C)(C)CN=c1cc(C)[nH]c(=NCCCC2CC2C)[nH]1 Cc1ccc(C(=O)NC(CNC(=O)CN(S(C)(=O)=O)C)CC(C)C)c([N+](=O)[O-])c1 Nc1ccc(C(N2CC3(CCCN(C(C4CS(=O)(=O)C4)=O)C3)C2)=O)c([N+](=O)[O-])c1 CCCC(C(=O)N1CC(O)CC1CN(C(=O)Cc1ccc(F)cc1)CC)OC c1(CC(N2CC(C)(c3cn(-c4cccc(Cl)c4Cl)nn3)C2)=O)c(Br)cccc1Br c1(OC)cc(Cl)ncc1NC(C1C(O)CCN1C(=O)CN1CCCC1)=O c1(OC)ccc(F)c(N)c1C(=O)N(C1CCCCC1N(C)C(=O)OC(C)(C)C)C Cc1c(C(=O)NCC2(CNC(c3cc(N(C)C)nc(Cl)c3)=O)CC2)cccc1N N#CCCCC(=O)N1CCCC1CNC(=O)C(F)(F)CF c1(C(N(C)C)=O)ccccc1-n1cc(-c2nc(C(=O)O)cs2)nn1 C(=O)(CC(C)C(C)(C)C)NCC(CNC(C1CC(C2CC2)C1)=O)OC C(CCC(=O)NC(C)CCCNC(=O)C=C1CCC1)=CCC=C C(=O)(C1CCCc2scnc21)NC1C2CN(C(CC3ON=C(CC)C3)=O)CC1C2 CCCC(C)(CCC)C(=O)NCC1COCC1NC(c1[nH]cc2c1CCCC2)=O C1(CNC(C=Cc2c(OC)cccc2)=O)CN(C(=O)C2=CCSC2)CCC1(C)C C1(NC(c2c(CC)nco2)=O)CCC2CC1CN2C(c1cnc(C(C)(C)C)s1)=O Cc1cc(C(=O)NC2CC(NC(=O)CC3COCCO3)C2)c(C)n1C1CCOC1 C1(C(=O)NCC(CNC(Cc2c(CC)cccc2)=O)O)CCC2(CCC2)C1 c1(CN(C(C)C(N)=O)C)ccc(C#N)cc1Br c1(C(N2CC(NC(C(CC)C(C)C)=O)C(C)C2)=O)cc(F)cc2cc[nH]c12 CC1C(NC(=O)C(C)(F)F)CC2CCC1N2C(=O)CCCC(=O)C1CC1 c1(-c2scc(C(=O)NCC#CCNC(C(CC)OCC)=O)n2)ncccc1F C1(C)(C(N2CCC(C(C)NC(c3cocc3C(N)=O)=O)C2)=O)CC=CCO1 N1(C(c2cc(C(F)F)on2)C(=O)NCC2CC2)CCC2(CCC(O)C2)C1 CN1CCCCC1C(N1CC(O)CC1CNC(=O)CCC1CC1(F)F)=O CC1CN(C(C2(C3CCC3)CC2(F)F)=O)CC(C)N(C(=O)CC(C)(C)O)C1 Cc1ccc(-c2cc(C(=O)NC3CC(C)(NC(=O)C(C)NS(C)(=O)=O)C3)n[nH]2)s1 Cc1nc(C)c(C(=O)N(CCCNC(c2cc(Br)sn2)=O)C(C)C)o1 C1(CNC(c2ccc(Br)o2)=O)CC(O)CN1C(=O)CCCc1cnccn1 C1(C2CCN(C(=O)CC3CCCOCC3)C2)(NC(C(C(C)C)CO)=O)CC1 C1(CNC(C(CC)COC)=O)CN(C(=O)CCc2cscn2)CC12CCC2 C(C(=O)NNC(=O)c1ncccc1N(C)C(C)C)Oc1c(C)cccc1 c1(CC(=O)NC2(C3CN(C(c4c[nH]c(=NC)o4)=O)C3)CC2)ccc2nsnc2c1 C=CC(O)(C(=O)N1CC(O)(CCNC(=O)CN2CCOCC2=O)C1)C(F)(F)F C(=O)(CCCN(C)N=O)N(CCCNC(C(C(CC)O)C)=O)CC1CCCC1 N1(C(C(C)Cc2cccc(Br)c2)=O)CC(NC(c2cc(Cl)n(C)n2)=O)C(C)C1 N1(C(C(C)CN(C)C)=O)CCCC(O)(CNC(=O)CSc2cccc(F)c2)CC1 CCC(CC)CC(=O)NC1CN(C(=O)C(C)(C)C2CCCCO2)CCC1C C1(CCNC(c2ccc(OC3CC3)cc2)c2n(CC)nnn2)CCC(C)(C)C1 N1(C(CCCC=C)=O)CC2(CCCC(CNC(=O)C(C)(C)N(C)C)O2)C1 C1(C)(C(=O)NCC2(O)CC(CNC(C(CC)SCC)=O)C2)CCN(C(C)=O)CC1 CCCCC(C(=O)N(CC(C)NC(c1ccnc2cc[nH]c12)=O)CC)C(C)C S(=O)(=O)(c1ccn(C)n1)N1CCOCC(NC(C(C(C)C)O)=O)C1 C1(C(N(C(C)C)C)=O)CC2CCC(C1)N2C(C1CC(O)C1)=O N1(C(C2(Br)CC2(F)F)=O)CCC(O)(C(N2CCCC2)=O)CC1 C1(CC(=O)NCC2C(NC(c3c(CSCC)cccc3)=O)C2)OCCOC1(C)C CC1CCC(NC(=O)OC(C)(C)C)N1C(=O)CONC(C1CCC2(CC2)C1)=O C1(C)(CNC(c2[nH]cc(C)c2)=O)CCN(C(c2cnn(C(C)C)c2C2CC2)=O)C1 C=CC(CC)CC(=O)NCC1CN(C(C2(C)CCSCC2)=O)CC1(C)C Cc1cc(C(=O)NCCN2CCCNC2=O)c2c(C)nn(C)c2n1 c1(CC)nocc1C(N1CCCC1CN(C(C)C(=O)NCC(C)C)C)=O Cc1ccc(O)cc1C(=O)NCCC1(O)CCN(C(=O)CCC2CC2(F)F)CC1 CC1CCc2[nH]nc(C(=O)NCC3(CNC(C4CCOC(=O)CC4)=O)CC3)c2C1 C1(C(=O)NCC(CC)NC(c2cc(C3CC3)nnc2O)=O)CCCCCCC1 C1(N(C(C2(CC(F)(F)F)CC2)=O)CC)CN(C(=O)C(C)COC(C)=O)CC1(C)C c1(C(C(=O)NCC)N(C(C)CCS(C)(=O)=O)C)nc(C(F)(F)F)n2c1CCCC2 C1(OC(C)=O)CC2(C1)CC(CNC(c1ccc[nH]1)=O)C2.C(=O)CC1CC1C(F)(F)F c1(NCC(C)CO)ncccc1S(=O)(=O)NC12CCC(CO)(CC1)C2 C=CCCCC(C)(C)C(=O)NC(C)CC(C)NC(=O)CNc1nccs1 N1(C(C(C=C)(C)CC)=O)CCc2ccc(C(N3CCOC(C)C3C)=O)nc2C1 c1(C(N(CCCNC(CC(=O)N(C)C)=O)CCO)=O)cnc2c(c1)COCC2 C12(CNC(C3CCOC3=O)=O)CC1CN(C(=O)Cc1ccccc1C(F)F)C2 c1(C(=O)NCCCCc2ccc(OC)cc2)cnc(OC)c(Cl)c1 CCC(C)(CO)C(=O)N1CCC(CNC(=O)CC2NC(=O)CNC2=O)(OC)C1 C(=O)(CC(CCC)CCC)N1C(C(=O)NCCSCC=C)C(C)C1 N1(C(C(CSC)OC)=O)CCC2(CC(NC(c3nnn(C)n3)=O)C2)C1 C1(CC(=O)NC(c2c(C(=O)NCc3n(CC)cnn3)con2)C)CCN(C)C1=O C1(CC=C)(C(=O)NCC2C=CCCC2)CCN(C(c2cn(CCC)nn2)=O)C1 C12=NC(=N)NC(=NCCCN1)N2.CC1CS(=O)(=O)CC1N(C)CCO N1(C(C=C(C)C(F)F)=O)CC(CNC(=O)CN(C)Cc2ccccc2)CC1(C)C C1(C2CCC2)(C(N2CCN(C(C(=O)NCC)=O)C(COC)C2)=O)CC1(F)F c1(C(=O)NCCCN(C(=O)CC2CCC2(C)C)C)cc2cc(Cl)ccc2n1C c1(N2CC3C(NC(C(CC)(C)C)=O)C3C2)ncc2ccsc2n1 C1(NC(=O)CCC2CCC2)CCN(C(C23CCCC(C2)OC3)=O)CC1F CN1CCC(F)(C(=O)NCCCNC(=O)C=CC(c2ccc(F)cc2)=O)CC1 N(C(=NCCOc1ccc(C(C)C)cc1)NC1CC1C(F)(F)F)CC c1(NC(C)CN(CC)CC)ncc(C)cc1S(=O)(=O)NC(CCC)C1CC1 C1(C(=O)NC2(C(N3CC(COC)C3)=O)CCN(C)C2)CCC(N=[N+]=[N-])C1 c1(C(=O)NCCCOCCNC(C(C2CCC(=O)N2)C)=O)cccc(N)c1F C(=O)(CCCC(C)(C)NC(=O)C1=NOC(C)(C)C1)NC(c1cncc(F)c1)C N1(C(CC)C(N2CCCOC(CNC(=O)CC3CC3)C2)=O)CCc2ccccc21 c1(C(=O)NCC2C(NC(C=CCC)=O)CC2)ccc(SC)o1 c1(CC)ncc(C(N2CC(CNC(C3CCOC3C)=O)C2)=O)c(C)n1 CN1CCOC(C(=O)NC2CC(CCNC(=O)CCC3CCCC3)C2)C1=O c1(C(N2CCCC(CC(=O)OC)C2)=O)ccc(-c2ccc(C)o2)c(F)c1 N1(C(CCN(C(C)=O)C)=O)CCC2C1CCCN2c1cc(C2CC2)ncn1 N1(C(COC(c2cc(CC)sc2Br)=O)=O)CCCC2(C)CCCC12 c1(C(N2CC(C)C(NC(C3CCCC(=O)N3C)=O)C2)=O)cc(O)cc(=O)o1 c1(C(=O)NCCOC)cn(CCC(=O)NC2(c3ccccn3)CCCC2)nn1 c1(C(=O)NCc2cc(C(=O)NCc3nn[nH]n3)no2)ccccc1C1CC1 CCC1=C(C(=O)N2CCC(C(C)NC(c3cnn(C)c3)=O)C2)SCCO1 C1(C(N2CC(F)(CNC(c3cnn(CC(F)(F)F)c3)=O)C2)=O)C(F)(F)C12CCC2 C1(NC(C2C(=C)CC2)=O)CC1C1CCCN(c2snc(C)c2C#N)C1 C1(CNC(C(C(C)(C)O)F)=O)C(C2CC2)CCN1C(=O)C(=O)Cc1ccccc1 c1(N2CC(NC(CN3C(C)CCC3C)=O)C(C)(C)C2)ncnc2sccc12 C1(CC=C)(NC(=O)CC2CCCO2)CCN(C(C2(C#N)CC2)=O)C1 C(=O)(CCS(=O)(=O)N(C)C)NC1CCC(N(C(CCC=CC)=O)C)C1 N1(C(CCCN(C)C)=O)CC(O)CC1CNC(C1CC1C(C)(F)F)=O CC1(C)C(NC(C2CCCC(=O)N2)=O)CCN1C(=O)Cc1cccnc1N C12(CC(=O)NCCCN(C)C(C3CN(C4CCOC4)C3)=O)CCCC1C2 c1(C(C)C)cccc(C(N2CC(CNC(=O)CCC(=O)N(C)C)C3CC23)=O)c1N N1(C(C(C)CN(C)C)=O)CC(O)(C2(CNC(=O)CC3CCC34CCC4)CC2)C1 C1(CC(=O)NCC(c2ccccc2)CNC(c2c(C)snn2)=O)CCCC(=O)N1 N1(C(c2cc(CC)sn2)=O)CCOCC1CN(C)C(c1cnc(CC)s1)=O C=CCC(CNC(C1CCSCC1)=O)C(=O)NCc1nnc(O)n1C N1(C(c2c(C)onc2C(F)(F)F)=O)CC2(C1)CN(C(C1CCCCC1O)=O)C2 CC1(CNC(C2(C)CCCO2)=O)CCCN(C(=O)C=Cc2ccncn2)C1 c1(C(=O)NC23CC(CNC(C=CSC)=O)(C2)C3)ccc(C2CCC2(C)C)cc1 C(C1(C)COC1)=CC(=O)N(CCN(C(C12CSCC1C2)=O)CC)CC(=O)NC c1(CNC(NCC2CCC(=O)N2)=NCCN2CCCC2)ccc2cccnc2c1 CCC(C)CCC(=O)N(C1CCCCN(C(=O)CCOCCOC)C1)C N1(C(CSCCC(C)C)=O)CCCCC1CCNC(=O)C=Cc1ccn(C)c1 c1(C(C)CC(=O)NC(C)(CNC(C2CCCN2C)=O)C2CC2)cccc(Br)c1 c1(C(=O)NCC(CC)NC(=O)Cc2ccno2)cc(O)cc(Cl)c1Cl C(C(C)C)(C(O)C(=O)N(CCCCCNC(=O)CN1CSCC1=O)C)OC c1(C(=O)NCCN(C(c2csc(O)n2)=O)CC)cc(F)c(F)cc1NC(N)=O CC1(C)CN(C(C2CC(C(F)F)C2)=O)CC(CNC(C2CNC(=O)N2)=O)O1 C1(OC)CCN(C(N2CC(C(CNC(C)C)NC(=O)OC(C)(C)C)(OC)C2)=O)C1 CC1(C)CC(=O)N(CC(=O)NCCCCNC(c2cc(C(C)(F)F)on2)=O)O1 N1(C(C(C)OCC(C)C)=O)CC(C)(CNC(=O)CCN(C)CCO)CC1(C)C C1(C(=O)NCC(CN(C(CC(=O)NCC)=O)CC)O)Cc2nccnc2C1 n1(CC(=O)NCC(C)CN(C)C(c2cn(C)nc2O)=O)sc2ccccc2c1=O CC(CCNC(C1(C(C)NC(C2CCCN2C)=O)CC1)=O)CCO C1(O)(CN(C(COCCCOC)=O)C)CCCN(C(=O)CCc2cnc(C)o2)C1 Cc1ccc(OC(C)C(N2CC(O)(CNC(=O)CCCSC(C)(C)C)C2)=O)cc1 C(=O)(CS(=O)(=O)C1CC1)N1CC(C)(NC(c2ccc(NC(N(C)C)=O)cc2)=O)C1 N1(C(C2(C)CN(C(c3ccc(CO)nc3)=O)C2)=O)CCCC(C(N)=O)CC1 CCC(CC)C(F)C(=O)N1CCN(C)C(NC(C2CC(OC3CC3)C2)=O)C1 C1(OC)CC(C(=O)NCCCNC(C)=O)N(C(C2CC2C)=O)C1 c1(CN(CC=C)C(C2CCN(CC3CCOC3)CC2)=O)cc(Br)ccc1F C(=O)(C1CCCc2ncnn21)NC1CN(C(c2cc(N)nc(Cl)c2)=O)CC12CC2 c1(C(=O)NC2C3(CN(C(CCC(=C)C)=O)C3)CCC2)c[nH]c2nccc(Cl)c12 CC(CC(=O)N1CCC(n2ccnc2)C1)C(C)(C)NC(c1cc(C(F)F)[nH]n1)=O C1(NC(C(C)n2cccc2)=O)CCCC(NC(=O)C=Cc2cc[nH]n2)C1 N1(C(C2(C)CC2C(F)(F)F)=O)CCN(CCNC(=O)CCc2ccccn2)CC1 N1(C(=O)CC2CCCCC2O)CCC2(C1)CN(C(=O)CC1CCCO1)C2 C(=O)(C(C(C)O)N(C)C)NC(CCNC(C(C)C#N)=O)(C)C C1(NC(c2c(C)nccn2)=O)CC2(C1)CC(C(=O)NC1CN(C(C)(C)C)C1)C2 Cc1nc(N(CCCCN(C(=O)Cc2cn[nH]c2)C)C)c2cc[nH]c2n1 C1(NC(C(=O)NCC2C(CC)CCCC2)=O)CCCCC12CC2 C(=O)(C1=CCOCC1)N(CCC(=O)NC(C1CCOCC1)C)C1CC1 C1(CNC(c2ccc(SC)o2)=O)CCCC(NC(=O)CCOc2ccccc2)C1 C1(CNC(=O)C(F)OC(F)(F)F)CC(F)CN1C(c1ccc(N2CC=CC2)cc1)=O N1(C(c2ccc(C)cc2O)=O)CC2CC(NC(=O)C=CSc3nc[nH]n3)CC2C1 N1(C(c2cc(OC)nc(Cl)c2)=O)CCC2C1CCN2C(C1CCCS1)=O N1(CC(=O)NCCNC(CN2CCC(C)C2)=O)CCC(F)(F)CC1 C1(C)(NC(C(CNC(COCC(=O)NC)=O)OC)=O)CC(C)(C)OC1=O Cc1cc(C(=O)NCC2CCOC2C)nn1CCO c1(C(=O)OC)sccc1CNC1CCC(NC(C2CC(N(C)C)C2)=O)C1 C(Cc1cnc[nH]1)(C(=O)NCC1COCC1NC(=O)Cc1cscn1)NC(C)=O N1(C(C=C(COC)C)=O)CCC(F)C(NC(=O)CN(S(C)(=O)=O)C)C1 C1(CCN(C(c2cn(CC)nc2)=O)C)CCN(C(c2ccc(OC)s2)=O)CC1 C12(NC(c3cc(OC)cc(Cl)c3)=O)CCCN(C(=O)CCOCC(C)C)CC1C2 N1(C(C(C)N2CCC2)=O)CC(NC(=O)CCc2ccc(N)cc2)C(C)(C)C1 CC(O)(CC(=O)NC12CC(CNC(c3cnnn3C3CC3)=O)(C1)C2)C1CC1 CC(C)C(C)CNC(C1(CNC(C2COCC2C(N)=O)=O)CC=CC1)=O C#Cc1ccc(C(N2CCC(CNC(c3cscn3)=O)CC2)=O)c(F)c1 c1(C(N2CC(CN(C(C3C(=C)C3)=O)C)OCC2)=O)ccn(C(C)C)c(=O)c1 c1(C(=O)NC(CNC(c2c(C)cn(C)n2)=O)C)cc2ccccc2c(=O)o1 C12(NC(Cc3scc(C)c3)=O)CC1CN(C(=O)CSc1ccccc1C)C2 S(=O)(=O)(c1ccc(F)c(Cl)c1)N(c1c(N(C)C(c2nc(O)n[nH]2)=O)cccc1)CCO N1(C(C(CCC)OC)=O)CCOCC(F)(CNC(c2cc(C)[nH]n2)=O)C1 C1(NC(CC(CNC(C2(CC)CCCO2)=O)O)=O)CCC(C2CC2)C1 c1(N(CCN(C(C2C(C)CC(=O)NC2)=O)C)C)nnc2c(c1C#N)CCCC2 c1(C(=O)NCC2CC(C)N(c3nccc(C(C)(C)C)n3)C2)cnc2n1CCCC2 C(CC(=O)NCCC1(OC)CCC1)(C(C)(C)C)NC(COCCOC)=O C(CCC(C)C)(C(=O)NC1CCN(C(=O)C2=NNC(=O)CC2)C(C)C1)NC(C)=O C1(C(=O)NC(CC(C)C)CO)CCCC12CCN(Cc1cc(I)ccc1Br)C2 C1(N(C(CC=C)=O)C)CN(C(=O)CCCn2cc(C)cn2)CCC1O c1(N(C)C)ncnc(Cl)c1CNc1cccc(-n2cc(C#N)cn2)c1 N1(C(c2onc(CC)n2)=O)CC2(CC(NC(C3(C)CC=C(C)CC3)=O)CO2)C1 c1(C(=O)NC2C(C)N(C(C3CSCCS3)=O)CCC2)ccc2c(c1)OC(C)(C)O2 c1(NC(c2c(C)ncc(C(F)(F)F)c2)=O)nc2cc(O)ccc2[nH]1.C1CO1 C(CCCCC(=O)NCc1ccc(C(=O)NCc2cnc(OC)cn2)nc1)=CC Cc1ccc(C(=O)NOCc2cn(Cc3ncoc3C(F)(F)F)nn2)cn1 Cc1cc(Br)ccc1C(=O)NCC(CNC(C1(C)CC=CCO1)=O)CO C(C)(C)(CC(=O)N(C1CCC(NC(c2ccc(C(C)C)nc2)=O)C1)C)OC c1(C(=O)NC2C(CNC(c3c(CC)n(CC)nn3)=O)C2)cc(OC)ccc1OC c1(N(CCCO)CC)ncnc2c1ncn2CC1(C(F)(F)F)CCCNCC1 CC(C)C(CCNC(c1ccc(-n2ccnc2)nn1)=O)N=c1[nH]nc(C2CC2)s1 CC12CCN(CC1)CC2NC(C1(C)CN(C(c2cnsc2)=O)C(C)(C)C1)=O c1(C(=O)NCCOCCCNC(c2cc[nH]n2)=O)ccn2c(O)nnc2c1 N1(C(CCC(=O)NCC)=O)CC(NC(=O)CC(C)C(C)(C)CC)CC2(CCC2)C1 c1(CC(N2CC(C(C)(C)O)(CNC(C3(C#C)CCC3)=O)C2)=O)sc(C)nc1C C1(CNC(C(C)N=[N+]=[N-])=O)CC(O)C(O)CC1C(=O)NCCCCOC(C)C c1(C(=O)NC2CCN(C(c3cnn(C)c3N)=O)C2)cn(CCO)c(=O)nc1O c1(C(=O)NCC(C)NC(C2CSCN2C)=O)cnc2c(c1)CCCC2 N1(C(=O)CCc2cc(F)cc(F)c2)CCC2C1CCN2C(=O)CSc1cn[nH]c1 C(CC(C(=O)N(C)C)Sc1ncc(C(=O)NC(C)(C)C)[nH]1)NC(=O)OC(C)C N1Cc2[nH][nH]c(=NC=O)c2C1.Cc1ccc(C)c(C(=O)N=c2cc[nH][nH]2)c1O Cc1occc(=O)c1OCC(N1CCC(N(C(=O)C(C)c2ccsn2)CCO)C1)=O Cc1nc(CO)ncc1C(N1CCCC(CCNC(C2CC2(C)Br)=O)C1)=O N1(C(=O)C2CC2)CCCC1.C1CC(=O)NC(C)C(=O)N1C.CS c1(OCC)ccc(NCC(=O)NC2CCCC2NC(=O)C(F)(F)COC)cn1 C(=O)(CCC(=O)NC(C)(C)CNC(C1CC(=O)N(C2CN(C)C2)C1)=O)NC(C)C C12(CNC(=O)CCc3cn[nH]c3)CCC(CN(C(C3CC3F)=O)C1)C2 C1(NC(c2c(C)occ2)=O)C2CCN(C(=O)CCOc3ccc(Cl)cc3)CCC12 c1(C(N(CCNC(CC2CC(SC)C2)=O)C2CC2)=O)cnn(CCO)c1C N1(C(c2cc(CCNC(=O)C=Cc3ccoc3)on2)=O)CCC(CO)(CN)C1 c1(N(C)CC2CN(C)C2)nc(=NCCC(C)(C)C)[nH]c2c1CCCC2 C(c1ccc2occc2c1)=CC(N1CCCC(O)(CNC(C(C)(C)CO)=O)C1)=O c1(C(N2CCN(C(CC(C(=C)C)O)=O)CC2C(C)C)=O)ncc(C#N)cc1Cl N1(C(C(C(C)C)N(C)C)=O)CC2(CCN(C(c3cnc4n3CCC4)=O)C2)C1 N1(C(C2C(C)(C)CO2)=O)CCC2(CC1)CN(C(C1CCC(F)CC1)=O)CCO2 C=CCC(CC(F)F)C(=O)N(C)CC1CCCN(C(c2ccc(N)c(N)n2)=O)C1 c1(C(N2CCCC(COC)(NC(=O)CSC)C2)=O)c(F)cc(C)cc1Br N1(C(CCCCC=CC)=O)CCN(C(=O)CCOC(C)=O)CCC1C CCC(C#N)C(=O)N1CC(C(F)(F)F)C(CNC(c2ncc(C)cn2)=O)C1 N1(C(C2(SC)CCC2)=O)CC2CCOCC2(NC(=O)CCCCCN(C)C)C1 c1(NC(C2CCN(C(c3cncc(Cl)c3)=O)CC2O)=O)ccnc(F)c1F C(=O)(CCC(C)(C)C(=O)N1C2CCC1CC(NC(C1(F)CCOC1)=O)C2)OC N1(C(C23CCC(OC)C2C3)=O)CC(C(=O)NCCS(C)(=N)=O)CCC1C c1(C(=O)NC23CCC(CNC(=O)CC(F)(F)Cl)(OC2)C3)cncc2nc[nH]c12 C1(C(N2C(C)(COC)CC2)=O)(CO)CCN(C(=O)CCOC2COC2)C1 C(CCC(C)C)(C(=O)NCCC(C)CC)NC(C(C)N(CC)CC)=O C1(N(C(C2C(=C)C2)=O)CC)CCN(C(C2(CCC)CC2)=O)C1 C(=O)(C1=CCS(=O)(=O)C1)NCC1(OC)CN(C(C2(C#N)CCOC2)=O)C1 c1(C(N2CCC(O)(C(=O)NCc3cccc(CO)c3)C2)=O)cccc(O)c1 C1(c2n(C(CC)C)nnn2)(NCc2ccn(CC(F)(F)F)n2)CC2(C1)OCCO2 CC1(C)CC1C(=O)NC(C(=O)NC1CN(C2CCC2)C1)C1CC1 C(CCCCC(=O)N1CCCCC1C(C)NC(=O)Cc1ccc(SC)cc1)OC Cc1c(C(=O)NC(C)CC(C)NC(C2CCCC23CCC3)=O)cccc1F c1(C(N(CC(=C)C)C)=O)cc(CCNC(=O)CC2CCC2)on1 Cc1cc(C)c(NC(C2CN(C(C3CCC(=O)C3)=O)CC2C)=O)c(C)n1 Cc1nc(=NC2CC3CN(C(=O)CCc4cc(Cl)cs4)CC23)s[nH]1 CC(C)C(C(=O)OCC(=O)N(C)Cc1nc(C2CC2)oc1Br)n1cnnn1 c1(OC)cc(C(N2C3CCCC2CN(C(C2(C)CC2F)=O)C3)=O)ccc1[N+](=O)[O-] C=CC1(C(=O)NCc2cccnc2Cl)CCN(C(c2oc(CC)nc2C)=O)CC1 CC(CN(C(=O)CNc1ccccn1)C1CC1)C(=O)NC(C1CCCO1)(C)C C1(C)(OCC)CCCN(C(C2CCCCCN2)=O)C1 C1(NC(c2c(N)cc(Cl)nc2)=O)CCN(C(C2COCCO2)=O)CC12CCC2 C(CC(C(C)C)NC(=O)Cc1cc[nH]c1)N(C(c1c(CC)ccs1)=O)C C#Cc1ccc(NC(=O)C(C2CCCO2)NC(c2scnc2CC)=O)cc1 C1(C(=O)NC2CCN(C(CCOC)=O)C2)CNC(=O)CC1(C)C CCCCC(O)C(=O)NC(C)(C)CCCCNC(=O)C(C1CCCCC1)O N#Cc1cn[nH]c1C(=O)NCC#CCNC(=O)C=Cc1cn[nH]c1 c1(C(=O)NCC(C2CC2)NC(C(C(C)C)F)=O)nncc2ccccc12 c1(NC(N2CCC(CN(C(C(C(C)C)NC(C)=O)=O)C)C2)=O)cnc(O)c(C)c1 N1(C(c2cc(C)sc2Br)=O)CCC2CCC12CNC(=O)CC(C)(C)C#N C(=O)(C(CO)C(F)(F)F)NC(CC(N1CC(COC)OCC1)=O)C S(=O)(=O)(c1ccc2nc(N3CCCC(CN(C)C)C3)sc2c1)NC(C)CC#N C1(C)(C(N2CCC(NC(CCSC)=O)C(F)(F)CC2)=O)COc2ccccc2O1 N1(C(CCCOCCC)=O)CC(CNC(=O)Cn2[nH]cnc2=N)C(C)C1 N1(C(COC(CC)C)=O)CCCC(CC(=O)Nc2cccc(O)c2)C1 C1(NC(C2N(CC)CCC2)=O)COC2(CCN(C(=O)COc3ccsc3)CC2)C1 c1(NC(CCCOC)C(C)C)nc(C)cc(=NCCCOCC(F)(F)F)[nH]1.C(C)(C)O C(C)(CCC(=O)N1CC(O)CCO1)NC(C(CCC)C(C)C)=O CC(C)C1=NOC(C(=O)NC2COCCC2C(N2CC3(CO)CC3(CO)C2)=O)C1 C(CC(=O)N=S(C)(=O)CCc1ccccc1)c1ccc(C(C)C)cc1 c1(C(=O)NC2CCCCN(C(c3c[nH]c(=N)s3)=O)C2)cncc2c(F)cccc12 c1(CNC(C(=O)NC(CC)C(=O)NC2CC2)=O)ccnc(OCc2ccco2)c1 C(=O)(CCCCCS(N)(=O)=O)N1C(CNC(COC)=O)CCC(C)C1 C(C)(CCCC(=O)N1CCC(C(N)=O)CC1)NC(c1cnc(C(C)C)o1)=O c1(C(=O)NC2CC(C(=O)NC3CC3Cl)C2)ccncc1Cl C12(NC(C(F)=CC)=O)CCOCC1CN(C(=O)C(C)(C)CN1CCN(C)CC1)C2 c1(C(=O)NC2(C)CCN(C(C(C)OC3CCCC3)=O)C2)ccc2c(n1)COCC2 C(=O)(C(C(C)C)NC(c1ccccc1)C(=O)OC)NC12CC(NC(CC=C)=O)C1C2 N1(C(C(CC(=C)C)C)=O)CC(NC(=O)CNC(=O)CC)CC12CCCC2 Cn1cc(C(N2CCN(C(C3(C)CC3(F)F)=O)CC2C(F)F)=O)n(C)c1=O C1(c2nc(CC)[nH]n2)CC(O)CN1C(c1csc(C)n1)=O c1(C(N2CC=CC(C(N3CC(C)SCC3)=O)C2)=O)cccc2ccnn12 S(=O)(=O)(c1cc(C(=O)O)ccc1Br)NC(Cc1c(C)cc(C)cc1C)C(=O)O S(=O)(=O)(c1cnc(N2CCCC(CC)(CO)C2)c(Cl)c1)NC(CC)CO C1(C(=O)Nc2c(C)non2)CCN(C(c2c(Cl)cnn2-c2ccccc2)=O)CC1 C1(CNC(c2ccc(SC)s2)=O)CC2CCC1N(C(=O)Cn1cc(Cl)cn1)C2 c1(C(=O)NCC(CNC(=O)CC2CCC(=O)N2)OC)cc(OC)ccc1[N+](=O)[O-] C(=O)(C(F)C(CC)CC)N1C2CC(C(N(CCN(CC=C)C)CC)=O)C1CC2 C(=O)(CS(=O)(=O)NC1CC1)NC(CC)CN(C(c1cc(C(N)=O)c[nH]1)=O)CC C1(C)(C(=O)NC(C)CCNC(c2scnc2C(F)(F)F)=O)CCS(=O)(=O)CC1 Cc1cc(C=CC(N2CCN(C(=O)C#CC3(C)CC3)CC(CO)C2)=O)ccc1F C1(NC(c2c(C(C)C)c[nH]n2)=O)CCC2CC1CN2C(c1cccc(C#N)n1)=O N1(C(c2ccc(C)c(C)n2)=O)CCC2(CCCN2C(=O)C(C)C(C)(C)O)C1 C1(CNC(Cc2ccn(CC)n2)=O)(OC)CCN(C(=O)CC2CCN(C)CC2)CC1 C1(NC(CC2C(C)CCC2)=O)CN(C(=O)CC(C)C(F)F)CC(C)(C)C1 C1(C2(NC(=O)Cc3ncccn3)CC2)CCCCN1C(=O)CN1CCOCC1 C12(C(=O)NCC3C(C)CCN3C(=O)CSS(C)(=O)=O)CCC(C)(CC1)OC2 N1(C(CCCCC(C)C)=O)CC(NC(=O)CN2C(=O)CCC2=O)CC12CCOC2 c1(SCC)ccccc1C(N1CC(CNC(c2coc(C(C)=O)c2)=O)CC1C)=O c1(OC)cc(C(O)C(=O)NCC2(CN(C)C(C3CCCS3)=O)CC2)c(F)cc1O C1(NC(=O)OC(C)(C)C)CC2COCC(C1)C2NC(c1cscn1)=O C12(CNC(C(C)CC3CCC3)=O)CCCC1N(Cc1coc(C3CC3)n1)CCC2 C1(N(C(c2nn(C(F)F)cc2Cl)=O)CC)CCCN(C(=O)CC2CCC2)C1 c1(OC)ccc(C(N2CCC(CNC(c3ncccc3Cl)=O)CC2)=O)cc1F c1(C(=O)NC2CC(CNC(CN3C(C)CCC3)=O)C2)c[nH]c2ncnc(O)c12 C1(C(N2CC(CC3CCC3)C2)=O)C=CCN1C(=O)CCCC1CCC1 C(=O)(C1=NOCC1)NCC1(NC(C(CC)N(C)C)=O)CCOC1 N1(C(C2CN(C(C)=O)C2)=O)CC=C(C(=O)NCC2CCCC2(C)C)CC1 C(=O)(C(C)(CO)NC(c1cc(OC)cs1)=O)NCC(COC)(F)F c1(CC(=O)NCC(C)NC(C2(O)CCC2)=O)coc2cc3c(cc12)CCC3 Cc1cc(Cl)c(C(=O)NC2CC2NC(C2CN3CCN2CC3)=O)cn1 c1(OC)cccc(NCCC(=O)N(C)CCN(C(=O)CC2CCOC2C)C)c1 C(CCCCCCCO)=CC(=O)N(C1CCCC(N(C(=O)CC2CCC2)C)C1)C N1(C(CCOC)=O)CCCC1(C)C(N1CCC(C(C)O)CC1)=O C=CCCC(CC(C)C)C(=O)NCC12CC(CC)(CN1C(=O)CC1CCOC1)C2 N1(C(C=C(CCC)C)=O)CCC(F)(CNC(c2cc(C3CCCC3)no2)=O)C1 C1(CNC(CN2CCC(CC(=O)OC)C(F)(F)C2)=O)CCc2cnc(C)n2C1 C(C1CN(C(=O)OC(C)(C)C)Cc2ccccc21)NC(C(C)C(F)(F)F)=O C1(F)(CCNC(=O)CCC2CC(NC(=O)C(C3CC3)C3CC3)C2)CCCC1 c1(C(=O)NC2C3(CC(NC(c4c(C)scc4)=O)C3)C2)nnn2c1CSCC2 C1(NC(=O)CN2CCCS2(=O)=O)CCN(C(c2ccnnc2O)=O)CC1O C(=O)(CC(C)C(F)(F)F)NCC(CC(C)C)NC(c1cn2c(n1)CCC2)=O CCC(C)C(C)NC(=O)C(N)c1cccs1 c1(CC)c(C(=O)NC2COCC2NC(C2CCS(=O)CC2)=O)cnn1C(C)(C)C CCC(CC(=O)NC(CNC(c1cnc(O)s1)=O)CC(F)(F)F)C(F)F C1(C(=O)NC(CC)CN(C(=O)CC(O)C(C)C)CC)CC2(CCOCC2)C1 N1(C(C2(SC)CCC2)=O)CCOC(C)(CNC(=O)C(F)(F)c2cccnc2)C1 c1(CNC(C2(CSC)CCC2)=O)ccc(CNC(=O)C(O)CN(C)C)cc1 N1(C(c2ccc(OC)cn2)=O)CCC(NC(C2(F)CCCCC2)=O)C(CO)C1 c1(C(=O)NC(CC=C)CNC(c2cncn2C)=O)ccc(C(C)C)nc1 C1(C)(C(=O)NCC(CNC(C#CC(=O)N(C)C)=O)(C)C)C(C)(C)C1(C)C CCCCC(C)C(=O)N(CCN(C(c1cc(CC)cnc1O)=O)CC)CC C1(C(N(C23CCCC2C3)CC)=O)C2CC2CN1C(=O)Cc1ncn(C)c1C C12(C(=O)NC3(CCNC(c4c[nH]cc(C)c4=O)=O)CCC3)CCOC1CCOC2 C=CCC(CC)C(=O)N1CCCC(C(=O)N(C2CCOC2)CCO)C1 c1(OCC(C)C)cc(C(C)(C)C)ccc1C(=O)NC12COC(COC(C)=O)(C1)C2 C1(NC(C(C2CCOCC2)OC)=O)CCC12CN(C(c1cc(Cl)cc(Cl)c1)=O)C2 c1(OC)cc(CC(N2CC=CC(NC(C3CC(=O)OC3(C)C)=O)C2)=O)ccc1O C1(C(=O)NCC2(C)CC(O)C2)CN(C(=O)CCC2(C#N)CCC2)CC1(F)F c1(CCC(=O)N(CCNC(C=C2CCC(C)C2)=O)C2CC2)n[nH]c2ccccc12 C(CCCC(=O)N1CCC=CC1C(=O)NC1CCOC1)OCC c1(C(C(=O)NC(C2CN(C(=O)C3=COCC3)C2)C)C)cccc(Cl)c1 C1(c2nc(CNC(C(=O)NCC)=O)[nH]n2)CCN(C(=O)C(COC)OC)CC1 CCC(C)C(C)C(=O)N1CCC12CN(C(c1snc(O)c1Cl)=O)C2 Cc1ccnc(CCCNC(=O)C(c2cccs2)NC(C2CCS(=O)(=O)C2)=O)c1 C1(n2cccn2)(CNC(CC=C=C)=O)CCN(C(=O)Cc2[nH]cnc2C)CC1 CC1=C(C(=O)NC2C=CC(C(N3CCC(C(C)C)C3)=O)C2)COCC1 N(C1CCOc2c(C)cc(C)cc21)C(CS(=O)(=O)NC)=O N1(C(C(C)OCC2CC2)=O)CCN(C)C(C(=O)NCC2CCOCC2)C1 c1(C(N2C(C(C)NC(C3=C(C)CC3)=O)CCC2)=O)cncc([N+](=O)[O-])c1 c1(C(=O)NCC(CC)NC(=O)CCn2ccc(=N)[nH]2)ccccc1F C1(NC(CCCNC(C)=O)=O)CCN(C(=O)CCC(C)(C)N(C)C)C(C)C1 c12cncc(c1)SC2c1nnnn1C1CCC1.CC1CC(COCC2CC2)CO1 C1(C2CC2)(CNC(=O)Cn2cncn2)CCN(C(c2cccc(Cl)c2)=O)C1 C(=O)(CC1CCc2ccccc21)NCC1(OC)CN(C(=O)CCn2cnnn2)C1 N1(C(C2C=CC(=O)N=N2)=O)CC2(CCN(C(c3ccc(Cl)c(F)c3)=O)CC2)C1 c1(OC)ccc(NC(c2nnnn2C(C)(C)C)c2ncco2)cc1CO C1(NC(C2CC2c2ccco2)=O)CCCCCC1C(=O)Nc1cccc(O)c1 C1(NC(C(CSC)C)=O)CCN(C(c2cnc(-c3ccccn3)nc2)=O)C(C)C1 c1(CNC(c2cc(C3CCN(C(CC)=O)CC3)no2)=O)c(Cl)sc(C)c1C C(=O)(C(O)C(C)(C)CC)N(CCN(C(c1cnc2sccn12)=O)CC)CC c12cc(OC(F)(F)F)ccc1OC2.C1(C(c2ccccc2)=O)C2CS(=O)(=O)CC12 C#CC(CNC(=O)CC1CCCN(C(=O)CN2CCCC2)C1)C(C)C CC1CN(C(=O)C(F)(F)c2ccccc2)CCC1NC(C1CCC2(C1)N=N2)=O c1(C(=O)NC(C(C)NC(=O)C=C2CCN(C)C2)(C)C)cc2nn[nH]c2cc1F C1(C(N(CCN(C)Cc2ccc(C)cc2Br)C)=O)CCc2ncnc(C)c2C1 C1(CNC(c2c(C)n(C(C)(C)C)nc2)=O)N(C(=O)C=CC2CC2)CCCC1(C)C c1(OC)ccc(C)c(C(=O)NC(C)(C)CNC(c2ccc(-c3cccs3)s2)=O)n1 C1(CNC(Cn2c(C)cnc2)=O)CC2(C1)CN(C(c1nc(Cl)sc1Cl)=O)C2 C1(CC(C)NC(CN2C(C)CC2)=O)CCN(C(c2cccn2C2CC2)=O)CC1 C(CCSC)(CN=c1cc[nH]cc1S(=O)(=O)N(C)CCOCCSC1CC1)OC c1(C(N2CCN(C(CNS(N)(=O)=O)=O)C(C(F)F)C2)=O)cc2c(F)cccc2[nH]1 C1(NC(c2scc(C)c2C)=O)CC2CC(NC(c3ncccc3O)=O)C2C1 Cc1nn2c(C)cccc2c1C(=O)NC1CC(C)(CNC(=O)C(C)CN(C)C)C1 Cc1cc([N+](=O)[O-])ncc1C(=O)NC1CCC1NC(=O)CC1CCSCC1 CC(C)(C)CCCC(=O)N1CCC(C(=O)NCCC2C=CCC2)C12CCC2 CCCCC(CNC(=O)C(C)(O)C1CCC1)NC(c1coc(Cl)c1)=O C=CCCN=C(NCC1(C)CCS(=O)(=O)N1)NCC(N1CCOCC1)C C1(C(=O)NCC2(O)CCOC2)CC12CC(NC(C1(CO)CCOC1)=O)C2 CC(C)C(CCN(C)C(c1ccco1)=O)Nc1nccc(CO)n1 C1(NC(C(Cc2ccoc2)NC(C2N(C=O)CCC2)=O)=O)CCCC(O)C1O c1(N2CCCC(COC)C2)nc(N2CCC(S(C)(=O)=O)C2)c2ncn(C)c2n1 N1(C(C(CC=C)(C)C)=O)CCC(NC(c2cnc(O)s2)=O)C2(CCC2)C1 C(=O)(C(C)CCCC(C)C)NC(CSC)(C)C(N1CC(C(N)=O)C2(CC2)C1)=O C1(CNC(C(F)=CC)=O)CN(C(=O)Cc2cccc(SC)c2)CC1C c1(C(N2CC(C(=O)Nc3nc(Cl)ccc3O)OCC2)=O)cc(Br)cc(Br)c1O c1(C(=O)NC2CCC(OC)C2)ccc(CNC(C2CC2C(C)(F)F)=O)cc1 c1(C(N2CC=CC(NC(=O)COC3CC(F)(F)C3)C2)=O)ccc2c(c1)OCCO2 C(CCC(=O)N(C)CC1(CO)CC1)OCCC.C1(c2cc[nH]n2)(C=O)CCC1 N1(C(CC2(C=C)CC2)=O)CC2(CC(C(=O)NCc3cc(OC)no3)C2)C1 c1(C(N2CCCC(NC(c3c(C)ncnc3)=O)CC2)=O)cnn2c1OCC(O)C2 C(=O)(C(C)(C)CC(C)C)N1CC(NC(C=C(C)Cl)=O)C(C)(C)C1 c1(SCC#C)cccc(C(C(=O)C=C)=O)c1.C1(N)COCC1CNC(=O)CSN c1(CC(=O)NCC(c2ccccc2)CNC(CC(=O)NCC)=O)ccncc1C CC1CCCN(C(c2cc(=N)[nH]n2C)=O)C1CNC(c1ccc(CN=[N+]=[N-])o1)=O CCCCCCC(C)CC(=O)NCC(C)NC(c1ccc(=O)n(C)n1)=O N1(C(C2(C(C)(C)OC)CC2)=O)CC2CCN(C(c3occ4c3CCOC4)=O)C2C1 N1(C(C=CCC)=O)CC(OCC)C(NC(C2CCCOC2c2cc[nH]n2)=O)C1 c1(CC(=O)NCCOCCCNC(CS(CC)=O)=O)c[nH]c2cc(Cl)ccc12 C12(CNC(C3=CC(C)CC3)=O)CCCC1CN(C(=O)CCN1CCCC1)C2 C(=O)(CS(=O)(=O)CC)NCC(C)N(C(=O)C=Cc1cncn1C)CC c1(NC(C(COCCOC)Nc2ccsc2)=O)ccc2occc2c1 N1(C(CSCCOC)=O)CCC(CN(C(=O)CCC(=O)c2cnn(C)c2)C)CC1 CC#CCCCC(=O)N1CC(CNC(=O)CC2CCOCC2(C)C)C(O)C1 C1(NCc2ccc(OC(F)F)c(Br)c2)CCc2n[nH]cc2C1 c1(-n2c(CNCC(C(F)(F)F)n3cccn3)nnn2)cc(F)ccc1N1CCCC1 N1(CC(=O)NCC2(NC(C3C(=C)C3)=O)CC(OC)C2)C(=O)CCCC1=O CCC(C(N)=O)N1CCC(CCNC(=O)C(C)SC)C1 C1(CC(=O)NCCCSCC)CCCN1C(c1ccn(C2CC2)n1)=O CCCC(CCCNC(c1sccc1CN(C)C)=O)NC(C1CNC(=O)N1)=O C1(NC(c2ccc(OC)nn2)=O)CC2CC(C1)CN(C(C1CCCC1(C)C)=O)C2 Cc1cn(C)c2nc(N3CC(C(=O)NCc4nccc5ccccc45)C3)ncc12 c1(C(N(CC=CC(=O)NCc2n(CC)cnc2)C)=O)cnc(OC)cc1C c1(N(C(C(c2cccc(C)c2)=O)=O)C2CCNC2)ccn2ncc(Br)c2n1 C(=O)(CCCCCSC)NCC(C(=O)NC(c1ccncc1)C)OC N1(C(c2sccc2Br)C(=O)NCCSC)CCCC2(CC1)CCN(C)CC2 C(=O)(C(CCC1CC1)NC(=O)CN(C)C(N)=O)NCC1C(C)OCC1 N1(C(C(CCCC)O)=O)CC2CCCC1(CNC(c1ccc3ncnn3c1)=O)C2 C1(C(=O)NC(C2(OC)CCC2)C)CNC(=O)CN1C(c1ccc(O)c(C)c1)=O c1(OC)cc(C(N2CCC(NC(c3ccc(Cl)[nH]3)=O)C2)=O)ccc1Cl C1(NC(C(CCC)NC(C)=O)=O)CN(C(c2ccc(OC)o2)=O)CCC1C N1(C(C(C)OCCN(C)C)=O)CCCC(CO)(NC(C2CCCN2C)=O)C1 c1(C(=O)NCCN(C(C=CC)=O)CCC)ccccc1CCc1ccccc1 c1(C(=O)NCC(C2CC2)NC(CC2CN(C)C2)=O)cc2ccccc2[nH]1 N1(C(c2nnn(C(C)(C)C)n2)C(=O)O)CC2(CCC2)C1 c1(C(C(C)N(C=O)Cc2cc(Cl)no2)O)ccccc1F c1(C(N(CC(C)NC(=O)C(O)C2CC2)C)=O)cc(-c2ccncc2)[nH]n1 Cc1ncc2n1CCC(C(=O)NC(C)CNC(=O)C=Cc1ccnn1C)C2 C1(C)(C(=O)NCCOCC)CC(O)CN1C(C1COCC(C)O1)=O N1(C(c2n(C=C)nnc2)=O)CC(C(=O)NC2C=CCC2)CC12CCC2 N(C1CC2(CCCC2)c2ccccc21)C(N1CCC(F)(F)C2CCCCC12)=O C(CCCCC(=O)NCC(C1CCCN1C(=O)C(C)=C1CCCC1)(C)C)=CC c1(-c2nnc(N(C(C#C)C)C)n2CC(C)C)ccc(C#N)cc1 C(CCF)(C(=O)NCCC1(O)CCCC1)NC(c1c(C)c[nH]c1)=O c1(CC(=O)N(CC(C)CNC(C2(N3CCCCC3=O)CC2)=O)C)ccc(O)cn1 c1(C(=O)NC2C(C)CN(C(C3CC(=O)NC(=O)N3)=O)CC2)ccn2c1CCCC2 Cn1cc2c(C(N3CCC3CNC(=O)Cc3ccoc3)=O)cc(F)cc2n1 N1(C(Cn2c(C)nnn2)=O)CCC2(CC1)OCCC2NC(c1ncccc1Cl)=O c1(N(CC(C)OC)C)nc(N2CCC3CCC(C3)C2)c2ncccc2n1 c1(NC(C(CN(C)C)NC(c2nc(CC)sc2)=O)=O)cnc2ccnn2c1 Cc1c(C(=O)NC(C2CCOC2)CNC(=O)COCC2CCC2)[nH]ccc1=O c1(CC(N2C(C)(C)C(CNC(=O)CC3CC3)CC2)=O)ccc2c(c1)CCCS2 N1(CC(=O)NCC23C(CN(C(C=C(C)C(F)F)=O)C2)C3)CCc2ccccc21 N1(C(C=C(CCC)C)=O)CCC2CN(C(c3ccc(C(C)(C)C)o3)=O)CC12 c1(NC(C(C)(C)O)=O)cccc(C(N2CCCC(Nc3ncccn3)C2)=O)c1 CC1CCN(C(=O)C2=COCC2)C1CNC(c1cc(-c2ccco2)[nH]n1)=O CC1CCCCC1(CNC(c1cc(C2(O)COC2)on1)=O)NC(c1cocn1)=O c1(OC)ccccc1CCC1CCN(CC(=O)NCC(c2ccccc2)O)CC1 CCC(CC(=O)NC(c1ccc(C)cn1)C)NC(c1ccc[nH]1)=O CCCC(C#N)C(=O)NCCC1(C)CCN(C(c2c(C)cccc2Cl)=O)C1 CCC(F)(F)CC(=O)NCC(C)CN(C)C(c1ccc(OCCF)cn1)=O c1(CNC(C(C(C)OC)NC(C(C=C=C)C)=O)=O)ccc(C)c(C)c1 CC(CC(=O)N1CC2(NC(=O)CN(C)S(N)(=O)=O)CCCC2(F)C1)CC(F)(F)F c1(N(C)C)cncc(C(=O)NC2CC(NC(c3cc(C4CC4)cs3)=O)CC2O)n1 c1(C(C)C)nn(C)c(NC(C2CC2NC(C2CCN(C)C2)=O)=O)c1Cl c1(-n2cc(CNC(c3cc(C(=O)OCC)c(C)s3)=O)nn2)cc(F)cnc1Cl O(NC(=O)CCOCCCNC(C1CC(O)C1)=O)C(C(=O)OC)(C)C C(C(C(=O)N1CCC(C)(F)CC1)C(C)C)NC(CC(CC)SC)=O c1(C(=O)NC2CCC(NC(C(C=CC)O)=O)CC2)ncc(F)cc1F c1(C(=O)NC(C)CCNC(=O)C(N2C(=O)CCC2=O)C)nnn2c1CCC2 N1(C(c2c(CC)con2)=O)CCN(C(c2sc(C(C)C)nc2C)=O)C(C)CC1C C1(C(=O)Nc2cnc(OC)nc2)CC(F)(F)CN1C(=O)CCC(C)N(C)C c1(-c2cccc(NC(=O)NC3CC(F)(F)C3)n2)ccc2ccccc2c1 N1(C(C(C)Cc2cnc[nH]2)=O)CCCC2(C1)CN(C(c1cn(C)ccc1=O)=O)C2 c1(C(N2CC(CC)C(NC(=O)C(C)C)CC2)=O)ccc2c(c1)nc(C)n2C1CC1 C(C1=CCN(C(=O)CC2CC3CCC2O3)CC1)NC(C(=O)NCCOC)=O c1(C(=O)OC)sc(N2CC3CC2(C(N)=O)C3)nc1C(F)(F)F C(=O)(CCCC(=O)NC(C)C)NC(CNC(C(c1scc(C)n1)C)=O)(C)C(C)C C1(N(C(CCOCC#C)=O)C)CCN(C(=O)C(C)(C)NC(=O)OCC)C1 N1(C(C(C)OCCOC)=O)CCC2(CC1)CCN(C(=O)CCC(=O)OC1CC1)C2 C(=O)(C(C)(C(C)C)NCc1cc(C)n(CCl)c1C)NC N1(C(=O)NCCNS(NC)(=O)=O)CCOCC1c1ncno1 Cc1cc(Cl)cc(N)c1C(N1CCC2(CC(NC(=O)CN(C)C(C)C)C2)C1)=O CC1CC(C(=O)NCCC(O)CNC(C23CC(CC(F)F)(C2)C3)=O)CN1C CC(CC(=O)N1CC(C(=O)NCC(Cl)C(C)(F)F)C2(CC2)C1)C(F)(F)F CCCC(C(=O)NC(C)(C)C(O)CO)NC(=O)CC(C)CN(C)C Cc1ccc(F)c(C(=O)NC2(CO)CN(C(=O)C=CS(C)=O)C2)n1 C1(CC(=O)N(CC=C)CC)CN(C(=O)C(C)c2cc[nH]n2)C(C)(C)C1 C(C(CNC(=O)C=Cc1ccco1)C(F)(F)F)NC(COC(CC)C)=O n1(COCC)nc(C)c(CC(=O)N(CC(C)NC(c2c[nH]c(=N)o2)=O)C)c1C C1(NC(=O)NC(C2C=CCCC2)C(C)C)(Cc2ncccn2)CCC(C)(C)CC1 C1(C(=O)NC(C)(C)C(N2CCCC(C(F)F)C2)=O)CC(=O)CC(=O)C1 Cn1nc(C(=O)NCC(O)C(N2CCCC(CC3CC3)C2)=O)ccc1=O N1(C(CCC(C)C)=O)CC2CC(NC(C3(c4ccc(Cl)cc4)CC3)=O)CC2C1 c1(C(=O)NCC2C(NC(COc3c(C)cccc3C)=O)CC2)ccc(C)n(C)c1=O N1(C(C2CCN(C(C(CC(C)C)O)=O)CC2O)=O)CC2OCCOC2C1 C12C3CC(CN(C3)C1=O)N2C(=O)C(C)(O)C(F)(F)F.C1(NC(=O)OCC)CC1 CS(=O)(=O)c1cccnc1C(=O)NCC1CN(C(c2ncccc2O)=O)C2CC12 c1(C(=O)NCCOCCCN(C(CC)=O)C)ccsc1CC C(=O)(C(C)C(F)(F)F)NC(CCCC)CNC(=O)CCNC(=O)OC(C)(C)C N1(C(c2nc(C(C)NC(C3CC(C(C)C)=NO3)=O)oc2)=O)CC(O)CC1(C)C C(C(C)NC(=O)CCc1cncc(F)c1)(C(C)C)NC(C(CC)=CC)=O C(=O)(CC(C(F)F)c1ccccc1)NCC1(C)CC(NC(=O)C(C)(C)C)C1 C1(C(=O)NCc2nc(CC)oc2)CCN(C(=O)Cn2nc(C)nc2C)C(C)C1 C1(CC)CNC(=O)CN1C(C1(CNC(C2CC(N(C)C)C2)=O)CCCO1)=O Cc1cc(CNC(=O)C(c2cncnc2)C)oc1C(=O)NCC1CCN(C)CC1 C1(NC(CCc2cncc(C)c2)=O)CCN(Cc2ccsc2)C(C)C1 C#CCCCCCCC(=O)NC(C1CCN(C(C2(C)CCOC2)=O)C1)(C)C N1(c2snc(CCOC)n2)CC(NC(=O)CCCc2cccc(Cl)c2)CCC1C N1(C(CCN(CC)CC)=O)C(CNC(=O)CC(O)CN(C)C)CC2CC12 CC1CCC(C(=O)N(C)CCOCCNC(c2cc[nH]n2)=O)O1 c1(C(=O)NC2C(NC(C3NC(=O)OCC3)=O)C2)cc(F)cc(Br)c1O N1(C(CC(CC(C)C)C)=O)CCCC(C2CN(C(=O)C(F)=CCCF)C2)C1 C(CC(=O)N(C1COCC1OC)C)(C(C)OC)NC(CCCOCC)=O C(CNC(=O)CC1=CCCC1)(C(C)C(C)C)NC(C=C(COC)C)=O c1(C(=O)NC(CNC(c2cnc(C)nc2C)=O)C(C)C)cc2ccc(Cl)cn2c1 C1(N(C)C)(CC)CCN(C(=O)CC(CC2CC2)NC(=O)C(C)N(C)C(C)=O)C1 N1(C(C(CC(C)C)ONC(=O)CC2CCOCC2)=O)CCC2(CCCO2)CC1 c1(C(=O)NC2CC(N(C(C3CN(C)C(=O)N3)=O)C)C2)cnc2n(c1=O)CCS2 c1(CCC(=O)N(CCNC(C2CCC(=O)N2C)=O)CC)cnc(C)nc1O C1(C(=O)NCC2C(NC(c3c(CC)cno3)=O)CCC2)CC1C1CCCC1 c1(OC)cc(C(=O)NC2CCCCN(C(=O)C(F)C3CCCC3)C2)cc(C)n1 N1(C(c2cn(CCOC)nn2)=O)C2CCCC1CC(NC(=O)CC1CC1(C)C)C2 C1(NC(n2cccc2)=O)CC2CCC(C1)N2CC(F)F C1(C(=O)NCC2(N(C)C)CC2)CN(C(C2CC(N=[N+]=[N-])C2)=O)CC(C)(C)C1 C(CO)(C(=O)NCC1(CNC(=O)CC(C)N(C)C)CCCC1)OC C1(CCC)(NC(=O)C(C2CN(C(=O)C(C)(C)NC(=O)OC)C2)OC)CCNC1=O CCCCCC(=O)NC1CC(CNC(c2nnn(C)c2CC)=O)C1 C1(NC(N2C(C(C)(C)C)CCC2)=O)CC2CCC1(C(=O)O)C2(C)C Cc1ccc2c(C(=O)NCC3CCCCN3C(=O)C(F)F)coc2c1 c1(NC(C2C(CNC(C3CCN(CC)CC3)=O)OCC2)=O)cccc2c1OCO2 CC1CN(C(C(=O)NCC2CCOC2)C2CCC2)CCN1S(C)(=O)=O c1(CCC(=O)NC(C)CN(C)C(C2(NC(N)=O)CC2)=O)cccc(Cl)c1 c1(CC(=O)NC2CN(C(C(C)NC(CC)=O)=O)CC2F)csc2nccn12 Cc1nn(C)c2sc(C(=O)NCC(O)CNC(C3CC4(CCCC4)C3)=O)cc12 C1(C(N(CCNC(c2c(C)n[nH]c2)=O)C(C)C)=O)CCC(C)CC1 CC1CN(C(=O)CC2CC(C)(C)CO2)CCC1CNC(=O)CN1CCN(C)CC1 CCCCCC(C)(C)C(=O)NCCN(C(=O)C(C)C(C)CC)CCOC c1(C(=O)NC(CC(C)NC(=O)CCCF)C)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1 c1(NC2(CNC(C(C)N3CCC3)=O)CCCCC2C)ncnc2sccc12 CC1CC(NC(=O)CCC2CCOC2)CN(C(c2cc(Cl)nnc2O)=O)C1 c1(C(=O)NC(CC)CN(C(=O)C(C2CCOCC2)F)CC)c(C)ccn1C N1(C(CSS(C)(=O)=O)=O)CCN(C(c2cccc(C3CC3)c2)=O)C(C2CCC2)C1 Cc1ccc(S(=O)(=O)NCCC(N2CCN(C(c3ccc[nH]3)=O)C3CC23)=O)cc1 CCCC(C#N)C(=O)N1CCC(C(C)(O)CNC(C2(O)CCCCCC2)=O)CC1 C=C1CC(C(F)(F)F)(C(=O)NCC(C)CNC(c2nncn2CC#N)=O)C1 N1(C(c2cc(F)cs2)=O)CCN(C(=O)Cn2cnnn2)C(CC2CC2)C1 CC(C)CC(O)CC(=O)N1CC(NC(c2ccc(C(F)F)o2)=O)C2(CCC2)C1 N1(C(C(c2ccnn2C)C)=O)CCCC(C)(CNC(C23CCC(F)(CC2)C3)=O)C1 C1(CNC(C2(COC)CC2)=O)CN(C(=O)CCSC)CC1O CC1(C)CCOC(C(N2CCC(NC(=O)CCCn3ccnn3)C(O)C2)=O)C1 CC#CC1CCN(C(=O)N(C2CN3CCC2CC3)C)C1 C1(CC(=O)NC(C)CNC(=O)C(c2ccccc2)C2CC2)CC=CCN1C C(C(C(=O)NCCCCSC)NC(=O)C(OC)OC)OC C=CCN(OC)C(=O)C1(CNC(=O)CC2(O)CCOC2)CC12CCC2 c1(C(N2C3CC(CC(NC(C)=O)C3)C2)=O)ccc2nc(S)[nH]c2c1 Cc1cccc(CNC(C2CC(F)CN2Cc2ccc(C(F)(F)F)nc2)=O)n1 C(=O)(C(CNC1CC(OC)C1)CC1CCOC1)NC c1(C2(C(=O)NC3C(OC)CN(C(C4CC5C=CC4O5)=O)C3)CC2)c(F)cccc1Cl C(=O)(C(C)(C)CCS(C)(=O)=O)NCC1(O)CN(C(C(C2CCCCC2)C)=O)C1 O=C(C1=CCCN(C(=O)Cc2cscn2)C1)NCCc1ccncn1 CCCCC(C(=O)NC(C)CN(C)C(C1(c2ccccc2C)CC1)=O)N(C)C N1(C(c2cnn(C)c2N)=O)CCN(C(C2CCOC2)=O)C(C2CCC2)C1 C1(C(=O)NC(CCCC)C(=O)NC)CCN(C(=O)CNC(=O)C(C)CC)CC1(C)C N1(C(c2c(CC)ccc(F)c2)=O)CCC2CCN(C(c3ccc[nH]3)=O)C2C1 c1(C(=O)NCC2(CNC(CC(CC)(F)F)=O)CCOCC2)nccn2nccc12 CC(N=c1[nH]c(=NCC2(C)CCC2)[nH]c2cccnc12)c1csc(Br)c1 C1(NC(c2c(F)ccc(CC)c2)=O)CCN(C(=O)CS(=O)CC)CC(O)C1 N1(C(C=CC)=O)CCC2(CCC2)C(CNC(=O)CCC(CC)OC)C1 c1(CNC(CN(C(C2CC(O)(CC#C)C2)=O)CCC)=O)cc(C)cnc1F C1(C(N2CCC(CNC(=O)CSC3CC3)(CO)CC2)=O)CCCC2(C1)CC2(F)F C12(NC(c3cc(C)oc3C)=O)CCC(CN(C(C3(Cl)CC3(C)C)=O)C1)C2 c1(C(N2CC(O)(C(C)NC(C3CC(CF)C3)=O)C2)=O)ccnc(O)c1Br C1(C(=O)NC2CC(CNC(c3cc(O)ncn3)=O)C2)CCCC2(C1)CC2(F)F Cc1nn(C)c2ncc(C(=O)NCC3CCC3NC(=O)C=CC(=O)N(C)C)cc12 c1(C(CCC(N2CCCC(OC)C2C(C)C)=O)=O)sc([N+](=O)[O-])cc1C(=O)OC CC1CCCCN1CC(=O)NC1CC(C)(C(=O)NOCCCN(C)C)C1 Nc1cnc(NCc2nc(Cl)ccc2Br)c(Cl)n1 C1(CNC(CC2CC(OCC)C2)=O)CCCC1NC(c1coc(C(C)OC)n1)=O N1(C(C=CCN(C)C(c2cc(F)n(C)n2)=O)=O)CCOCC1C1(C)CC1 c1(SCC(N2CC3C(NC(C(CSC)C)=O)C(C3)C2)=O)ccc(Cl)cc1[N+](=O)[O-] n1(CC)nc(CN2CCC(N3CCC(C)(O)C3)CC2)c(C)n1 c1(NC)cccc(C(N2CCOCC2CNC(C2CCCC2)=O)=O)n1 C(c1ccc(F)cc1)=CC(=O)NCC1(F)CCC(NC(c2c(C)scc2)=O)C1 c1(CC)ccoc1C(=O)NCC1(CCNC(C2CC(n3cccn3)C2)=O)CC1 C12(CNC(c3c(O)ccc(OC)c3)=O)CCCCC1CN(C(=O)C1=CCC1)C2 c1(N2CCOCC(NC(COc3cc(C)on3)=O)C2)cc(C)c(C#N)c(C)n1 c1(CCC(=O)NCC(CN(C(C=CCC)=O)CC)(C)C)cc(F)ccc1F N1(C(Cc2cn(CC)nc2)=O)CCCC1(C)CNC(C1CC1F)=O C(C1COc2ccccc21)N1C(=O)N(C)C(c2cc(Br)cs2)C1=O CC1CC(O)CCN(C(=O)C(=O)N(C)Cc2ccn(C)c2)C1 Cc1nc(NC(c2ccc(-c3cccc(C4(C(=O)N(C)C)CC4)c3)cc2)=O)sc1Cl Nc1c(C(N2CC3C(CNC(C4CNC(=O)C4)=O)C3C2)=O)cnn1CCO Cc1cc(C)n(CC23CC2CN(C(=O)CC(O)c2ccccc2)C3)n1 C12(C(N(CCCNC(CC3CC(OC)C3)=O)C)=O)CCC(N=[N+]=[N-])C1C2 c1(OC)cc(C(=O)NCC2(CNC(=O)CCCSC)CCC2)ccc1Cl C12(C(=O)NC3CCN(C)C3)CC1CCN2C(=O)CC(=O)NC1CC1 N1(C(CN(C(C)C)C)C)CCCC(C(=O)NCc2cnccc2N(C)C)C1 C1(SC)CN(C(c2cnn(C)c2N)=O)CC1NC(C1CC(c2ccccc2)C1)=O CC1CN(C(c2cnn[nH]2)=O)CCN1C(C12CC1COC2(C)C)=O CC1N(C(c2occc2CNC(=O)CC23CCC(CC2)C3)=O)CCOC1(C)C C(=O)(CC(CC)C(C)(C)C)N(CCC)CCNC(c1sc(C(F)(F)F)cc1C)=O CC1CCN(CC(N2CC=CC2C(=O)N(CC2=CCSC2)C)=O)C1 C1(C(N2CCC(C)(NC(=O)Cn3cccc3)CC2)=O)CCn2c(cnc2Br)C1 CCCC(C(=O)NCCN(C(=O)CCC(C)N(C)C)C1CC1)S(N)(=O)=O c1(C(=O)NC2CC(C)N(C(c3ccc4occc4n3)=O)C2)ccc2c(c1)CCN2 c1(CNC(=NC)NCCOC(C)(C)C)ccc(C#N)c(Cl)c1 CC(CCCO)N(CC(C)(C)O)C.C(C)(C)(C)OC C1(NC(c2ncc(F)cn2)=O)CCN(C(c2ncccc2Br)=O)CC1O CCC(CC)CN=c1cc(C)nc(N2CCCN3C(=O)CCC23C)[nH]1 c1(C(=O)NCCCNC(C2CC(OC)CN2C(C)=O)=O)cnn2cccc2c1 N1(CC2CCC(C)O2)CC2CC(NC(c3cnn4c3CCC4)=O)CC1C2 C1(CNC(C2CC23CCC3)=O)(CO)CCN(c2ccnc(-c3ccccc3)n2)C1 c1(CC(=O)NCC2(COC)CN(C(C(C)OCC)=O)C2)ccc2c(c1)CCC2 c1(CC(=O)NCC2CCN(C(C3(COC)CCCC3)=O)C2)cccnc1C CC1CCOC(C(=O)NC2CCCC(NC(=O)C3=CCOC3)C2)C1 c1(C(=O)NCCCCN(C)C(C2CC2C2CC2)=O)cnc(-c2ccccc2)s1 C(C)(C)(CCCNC(C1(C#N)CCCC1)=O)NC(C(C)O)=O C1(NC(C(C)C)=O)CCC2CC1CN2C(c1cc(N)c(Cl)c(O)n1)=O c1(C(=O)NC(C2CCCN(C(=O)Cc3ccsc3)C2)C)cnc(C(F)(F)F)cn1 N1(C(CC=C)=O)CCC(CN2CCN(C(=O)CCOCC3CCCO3)CC2)CC1 C1(CN(C(c2ncn(CC)c2)=O)C)CN(C(=O)Cn2cccn2)CCO1 C(C)(C(=O)N1CC2CC2(CNC(=O)C(C)=CC2CC2)C1)(C(C)C)NC(C)=O c1(C(=O)NCCCCC)cc2cc(-c3cc(F)cc(F)c3O)cnc2[nH]1 N1(C(C(C)C)=O)CC(C)C(C)(CNC(=O)COCC2CCOCC2)C1 C1(C(N(CC(CO)(CO)NC(COCCCCCC)=O)C)=O)COCCC1(F)F C=Cn1nncc1C(N1CCC(C(F)CNC(=O)CCSCC(N)=O)CC1)=O c1(OCCNC(C2N(C(C(CC)OC(C)=O)=O)CC2)=O)ccc(C(F)(F)F)cc1 c1(C(N2CC(C)C(NC(=O)CC(F)(F)Cl)C2)=O)c[nH]c2c(F)cccc12 c1(C(N2CCC(CC(C)NC(C3CCC(F)(F)C3)=O)CC2)=O)cccc(N)c1F N1(C(=O)Cn2cnnc2O)CCCN(C(c2cc3cscc3s2)=O)CC1 c1(-n2c(Cn3nc(C)cc3C)nc(C(C)OC)n2)cc(Cl)nc(Cl)c1 C1(NC(c2ccc(OCCC)cc2)=O)C2CCC1N(C(=O)C(O)C(C)C)C2 N1(C(CC2CC(OC)C2)=O)CCC2(CC1)CC2NC(=O)Cc1ccno1 C1(C(=O)NCC2CC(NC(CN(C3CC3)CC)=O)C2)CC1C1CCCCC1 C(=O)(C(C#N)C(C)(C)C)N(C(C)C(N1CCC(CO)C(C)C1)=O)C1CC1 c1(C(=O)NC(CNC(=O)CCCC2CCCC2)CO)ccc(-n2ccnc2)cn1 CC1CCCC(C)N1C(=O)Cn1cc(COc2ccc(C(F)(F)F)cc2)nn1 n1(CC)c(C)nn(CC(=O)NC(C)CNC(=O)C=Cc2c(C)coc2C)c1=O C1(C)(C(=O)OC)CCC1(C)C(=O)NCC1CC(C)N(C(c2cn(C)c(C)n2)=O)C1 C12(CC)CN3C(=O)N(CCS(=O)(=O)c4ccccc4OC)C(=O)C3(C1)C2 C#CCC(CC(F)F)NC(=O)C(CNC(c1cnncc1C)=O)CCC N1(C(C(CC)(F)F)=O)CCC2(CCC2)C(CNC(=O)C(CC)NC(C)=O)C1 c1(C(=O)NC2CC3(CCN(C(CC#N)=O)CC3)C2)cc(F)cc(F)c1[N+](=O)[O-] C1(C(C)(C)NC(CCC)=O)CCCN1C(=O)C(C)OCCC(C)C C1(C)(C(=O)NCC2C(C)(C)C2(C)C)CC(O)CN1C(=O)CN1CCNC1=O c1(C(=O)NC2C(CNC(C3(OC)CCCOC3)=O)C2)c(F)cncc1Cl C(=O)(C1=CCN(C)C1)N1C(C)(C(=O)OC)C=CC1 N1(C(CONC(c2ccc(C)nc2)=O)=O)CCCC(O)(C(N)=O)C1 N1(C(C2C(=O)CC2)=O)CCN(C(c2sncc2Br)=O)C(C2CCC2)C1 C(=O)(C(F)(F)CC(C)C)NC1C(NC(C(F)OC)=O)CCCC1 C(C(=O)OC(=O)CCC(C)c1ccccc1)(C(C)C)n1ccc(C)c1 C1(O)(CN(C)C(c2ccnn2-c2ccncc2)=O)CCCN(C(=O)CC2CC2)C1 C(N=c1ccnc(NC2(c3ccccc3F)CC2)[nH]1)C1CC(OCC)C12CCC2 C1(NC(CCOC)=O)CC2CCC1CN(C(c1ccc(Br)cc1C)=O)C2 c12nnc(N3CCCC(C)C3)n1C2.Cc1ccc(C)n1Cc1ccc(CSC)s1 C1(NC(CN(C)C)=O)CC2(C1)CC(C(=O)Nc1cccc(Cl)c1Br)C2 C1(C(N(CCCN(C)C(C2CC2C(F)F)=O)C)=O)CCn2c(cnc2Br)C1 c1(OC)ccc(C)c(C(=O)N(C2CCN(C(c3ccc(C)nc3O)=O)CC2)C)c1 c1(C(=O)NCCN(C(Cc2cn(CC)nc2)=O)C(C)C)cc(OC)cc(Cl)c1O CC(CNCC1CC1)C(=O)NC1(c2ccco2)CC1 CC1(C)CN(C(c2ccc(Cl)c(F)c2)=O)CCC1NC(c1cc(O)nc(O)n1)=O C(c1ccoc1)=CC(=O)NCCC1(CNC(C2C(C)(CC)C2)=O)CC1 C1(CC(=O)N(C2CCCC2C#N)C)CN(C(c2cncs2)=O)C(C)(C)C1 c1(OC)ccc(F)c(C(=O)NCC(CO)NC(c2ccn(C)c2)=O)c1F C1(CNC(C=Cc2ccc(C)s2)=O)CN(C(=O)CC2CC2C(F)(F)F)CCC1C c1(N2CCC(C)(COC)C2)cccc(S(=O)(=O)NCCc2ccnc(C)c2)n1 C(=O)(C(F)(F)CCn1ccnn1)NCC(CNC(=O)C(F)OC(F)(F)F)O c1(C(=O)NC2C(NC(CCc3cc(OC)no3)=O)CCC2)ccc2cnnn2c1 C1(CNC(C2C(CNC(CN3CC(C)(C)C3)=O)OCC2)=O)CC2(CCC2O)C1 CC1CCCC(C)N(C(=O)C(=O)NCCCC#N)C1 c1(C(=O)NC(CCOC)CNC(=O)C=C(C)C)cc(N)ccc1Cl C#Cc1ccc(NC(C)C(=O)NCCC(C)(C)C)cc1Cl C1(C(=O)N(CCOCCC=C)CC)C(C)CN1C(=O)CCCN(C)C N1(C(c2[nH]cc(C#N)c2)=O)C2CCC1CN(C(=O)CC(F)(F)F)C2 N1(C(c2cnc(CC)nc2)=O)CC(N(C(=O)C=Cc2cnn(C)c2)C)C(C)(C)C1 C1(NC(=O)CCc2ccco2)CS(=O)(=O)CC1NC(=O)Cc1csc(Cl)c1 C1(c2cn(C(C)C)nc2)N(C(c2ccn3ccnc3c2)=O)CC12CCOCC2 c1(C(N2CCCC(CNC(C(C)C3CCCC3)=O)C2)=O)ccc2c(c1)NCC2 C1(C(=O)NC2CCN(CCC(=O)O)C2)(C(F)F)CCN(CC)CC1 C1(NC(CCn2ccc(C)n2)=O)CC(C)CN(C(=O)CN(C)C)C1 C1(NC(COCCC=C)=O)CC(C(=O)N2CCC(O)C(C)(O)C2)=CC1O Cc1cc(C)n(-c2ccc(C(=O)NC(C)(C)CNC(C3CC(C)CO3)=O)cc2)n1 c1(C(=O)NC2CC(CNC(C3CC(C)OC3)=O)C2)cc(F)c(F)cc1F C1(N)CN(C(=O)CCn2ccnc2C)CCC1(C)C.C=CCC(CC)C1CC1Cl Cc1cc(C)n(C(C)C(=O)NC(CO)C(C)NC(=O)CSCc2ncc[nH]2)n1 N1(C(C2C(C=C)OCCC2)=O)CC(F)(F)CC1(C)CNC(=O)CC(=C)C C1(NC(C(C)NC(N)=O)=O)CCN(C(C23CCC(C#N)(CC2)CC3)=O)CC1(C)C C1(C(c2nnnn2CCC)NCC(=C)Br)CC12CCC(F)(F)CC2 c1(C(N2CCC(CN(C(=O)C3=NNC(=O)C3)C)C2)=O)ccc2oc(O)nc2c1 c1(-c2cccc(C)c2)nc(=NCC2CC2CNC(c2cccs2)=O)s[nH]1 C1(CC(N2CCC(C)(N(C(c3c(NC)nccc3)=O)CC)C2)=O)CCC(C)(C)CC1 Cc1scc(C(=O)N(CCCCNC(=O)C(O)C2CC2)C)c1Br c1(C(c2nc(C3CC3)n[nH]2)=O)cnc(C2CCC2)nc1 C(=O)(C1=C(F)CN(C(C2CC23CCCC3)=O)CC1)NC(c1ccc(F)cc1)C c1(CC(=O)NC2CCN(C(C(COCC)C)=O)C2C(C)C)c[nH]c2cccnc12 N1(C(c2ccn(C)c2)=O)CC(F)(F)CC1C(=O)Nc1ncc(F)cc1F C1(C(=O)Nc2cccc(C(=O)NCc3nn[nH]n3)c2)CCC2CCCC2O1 C(CCCCC(=O)NC1CCCCC1N(C)C(c1cc(C2CC2)ncn1)=O)=CC c1(C(N2CC(CCNC(CNC(CC)=O)=O)OCCC2)=O)nsc2ccccc12 C=C(Br)CCC(=O)N1CCC(NS(NC(C)C)(=O)=O)C1 C1(C(=O)C(C#N)c2ccncn2)(OC)CCOCC1.CSC O=C(C1CCCn2cnnc21)N1CC(C2(NCCO)CC2)C1.C12CC(=NO1)C2=O C1(NC(c2c(C)c(Cl)cnc2)=O)COC2(C1)CN(C(=O)CC(C)P(C)(C)=O)C2 CC1CCOC1CC(=O)NCC1(O)CN(C(=O)CCc2c[nH]c(=N)[nH]2)C1 C(C(C)(C(N)=O)NC(c1cnn(CCNC(=O)CCn2cc(C)cn2)c1)=O)OC c1(OC)ncc(C(=O)NC2CC(CNC(C3CCS(=O)CC3)=O)C(O)C2)cn1 C1(C(=O)NCCC(CNC(CCN(C(CC)CC)C)=O)O)CCC(C)(C)O1 N1(CC(=O)NCC(CNC(c2ncn(C(C)C)n2)=O)O)CCN(C)CC1 N1(c2nc(C#N)cc(C)n2)CC2(CCC(NC(=O)COCC(F)F)CC2)C1 c1(OCC(=O)NC2CCN(C(C3C4CNC(=O)C34)=O)C2)cc(Cl)cc(Br)c1 c1(NC(CCC#C)=O)ccc(S(=O)(=O)NC2(CN(C)C(=O)OC(C)(C)C)CC2)o1 c1(C(=O)NCC2CN(C(c3c(C)onc3)=O)C3C2C3)cccc2ncnn12 C1(C)(C(NOCC(=O)NC(C=CC)(C)C)=O)CC(=O)N(C)C1 c1(CNC(C2CC23CCN(C(c2cnc(O)[nH]2)=O)C3)=O)cc(Cl)ccc1O N1(C(c2c[nH]c(=N)s2)=O)CC2ON=C(CNC(=O)Cc3cnc(C4CC4)[nH]3)C2C1 Cc1ccc(C(=O)NC2CC(CCNC(=O)CC3COC(C)(C)C3)C2)cc1Cl Cc1cnn(CCC(=O)NCC2(CNC(=O)CCOC3COC3)CCC2)c1 C(CCCC(C)NC(=O)CS(N)(=O)=O)NC(Cc1nc(C)sc1)=O C1(CNC(C=C(C)Cl)=O)CN(C(=O)Cc2cnnn2C)CC(C)(C)O1 C1(C(N2C(CCOC)CN(C(=O)CC(C)CF)CC2)=O)Cc2nccnc2C1 CC1=CC(F)(C(=O)NCC2CCN(C(c3cnn(C)c3)=O)C2)C(F)=C1 Cc1cc([N+](=O)[O-])nn1C(C)C(=O)NCC12CC(CN1C(C1CCCO1)=O)C2 Cc1ccn(CC(=O)NC2CCC(C)N(C(c3scc(C)c3C)=O)C2)c(=O)c1 N1(C(C(CCOC)C)=O)CC2CCCN(C(C34CCCC3C4(F)F)=O)C2C1 c1(C(=O)NC2CN(C(C(C)OC)=O)CC2C)c(F)c(F)c(F)c(F)c1F Cc1ccc2sc(C(=O)NCCC(C)NC(C3CC(C)OC3C)=O)cc2c1 C(C)(CN=c1cc(Cl)nc(C2CC2)[nH]1)NC(c1cc(C)n(C2CCOCC2)n1)=O N1(C(C2C(=C)CC2)=O)CCCCC1CCNC(c1ccc(-c2cc[nH]n2)cc1)=O CC1(F)CN(C(c2cccc3c2OCO3)=O)CCN(C(C2C3CCCOC23)=O)C1 N1(Cc2cccc(C(C)(C)C)c2)CCC(F)(F)C(NC(=O)Cn2cccn2)C1 c1(CC(C)C)nc2cccc(C(=O)Nc3ccc(F)cc3C(F)F)c2[nH]1 N1(C(C(C)O)=O)CCOC2(CCN(C(=O)CC3CCN(C)C3=O)C2)C1 C1(C(=O)NC(C(=O)NC2CCC(O)CC2)C2(C)CC2)CC2CCC1CC2 C(=O)(CCCNC(=O)Nc1ccccc1)NCC(CC)NC(=O)C=CCN(C)C N1(C(c2c(CC)scc2)=O)CC(O)(C2CCN(C(c3ccsc3C)=O)CC2)C1 c1(C(N(CC(C)NC(C2CC(SC)C2)=O)C)=O)nc(C2CC2)ncc1Br CCCC(C(=O)N1CCC(C(=O)N(C2CCOC(C)(C)C2)C)O1)N(C)C N1(C(c2cc(C)[nH]c2C)=O)CC2(CC2)CC1C(=O)NCC(C)(C)N1CCCC1 C1(C(=O)NC(C#C)C2CCC2)CCCN(C(=O)CC(O)C(C)C)C1CC C1(NC(C(C(CC)C)C)=O)C(C)(C)CN(C(c2ccoc2)=O)CC1(C)C C1(C(=O)NCC(C2CCC2)NC(CSCCC)=O)CCC1C(C)(C)C C(=O)(C(C)P(C)(C)=O)NCC(CCOC)NC(c1cc(C(=O)NC)on1)=O N1(C(c2cc(C)n(CCO)n2)=O)CCC2(CC1)CC2CNC(=O)CC1CCC1 N1(C(c2cc(O)ccc2Cl)=O)CC2CCN(Cc3cc(F)c(Cl)cc3O)C2C1 c1(C(=O)NC(C)CC2CN(C(C3(C#N)CCOC3)=O)C2)ncc(F)cc1F c1(SCC)nc(C(C)C)nc(C)c1C(=O)NCC1(O)CCC(C)CC1 N1(C(c2c(C)cn(C)n2)=O)CCC2CC2(C(N2CCN(C)CC(O)C2)=O)CC1 N1(C(CN(C2CCOC2)C(C2(CC(=O)N(CC#N)CCl)CCC2)=O)=O)CCCCC1 c1(C(=O)NCC2C(C(=O)NC(C(C)O)(C)C)CCO2)cccc(O)n1 N#Cc1cc(F)c(CNC2CCCN(CCC(=O)O)C2)c(F)c1 C1(N(C(C(C2CCOC2)OC)=O)C)CCN(C(C2(C)C=CCC2)=O)CC1 C1(OC)CCCCC1C(=O)N(C)CC1CCN(C(=O)C=CC=C(Cl)Cl)CC1 C1(F)(C(=O)NC(C)Cc2nncn2C)CCCN(C(=O)C=Cc2cnn(C)c2)C1 N1(C(c2c(C)cc(C)cc2O)=O)CCN(C(=O)C(C(C)O)N(C)C)CC2(CC2)C1 C1(C(N2CC(NC(C(C)NC(=O)C3CC3)=O)C2)=O)CC2(C1)OCCO2 CCC(C)CCCCC(=O)NC1(C)CCN(C(=O)Cn2nccc2C)CC1 CN1CC(C(=O)NCC2(NC(C3CC4C=CC3C4)=O)CC2)NC1=O c1(OC)ccccc1C(CNC(c1ccc(Br)o1)=O)NC(=O)C(O)C(F)F N1(CC2(NC(C3CC3F)=O)CC2)CCN(C(C2(C3CCCCO3)CC2)=O)CC1 CC1(C(=O)NCC2CN(C(c3cnn4c3OCC4)=O)CC2(F)F)CC2CCC1O2 CC(C)CC(CNC(=O)Cc1cnn(C)n1)NC(=O)CSc1nncn1C N1(C(c2cc(F)cc(C)c2N)=O)CC2COCCC2(NC(=O)C2=CCCSC2)C1 CC(CC(C)NC(c1cc(N2CCCC2)ccn1)=O)N=c1[nH]nc(C(C)(C)C)o1 Cc1cc(C(=O)NCc2ccc(C(N3CCN(C(C)C)CC3)=O)o2)c(C)n1C C(CCC)(C(=O)NCCn1cnnc1)NC(C1C(=C)C1)=O c1(C(N(CCNC(C2(C)CC2C(F)(F)F)=O)CC)=O)nccn2c(Br)cnc12 c1(C(=O)NC(CC)CNC(c2cncc(C)c2Cl)=O)coc2c1C(=O)NCCC2 C1(CC(N2CC(C)C(NC(C3CCC(=O)N3C)=O)C2)=O)CCCC(C)(C)O1 CC(C)(C)C(CNC(=O)CC1CC(OC(C)(C)C)C1)NC(=O)CCC#N C1(CC(=O)NCC2CCC(NC(C(C=C)(C)C)=O)C2)CC2CCC1CC2 C1(C(=O)NC(c2cccnc2)CC)N(C(=O)C(CC2CC2)OC)CCCC1(C)C c1(OC)cc(OC)n2[nH]c(=NC(=O)NCc3cncnc3)nc2n1 c1(C(=O)NCC2CN(C(=O)CCn3ccnc3)CCO2)cnc2ncc(Cl)cn12 c1(CN2C(C(=O)Nc3cnc(C(C)N)nc3)CC3CC32)ccc(C)c(Cl)c1 c1(C(=O)NC2C(NC(=O)Cc3nc([N+](=O)[O-])n[nH]3)CC2)cnn2c1OCC(O)C2 c1(OC)cnc(C(=O)N(CC(C)NC(=O)CCCC2(C)N=N2)C)nc1 c1(NC(N2CCCC(c3onc(CC)n3)C2)=O)cc(C)nc(Cl)c1 Cn1c(C(N2CCC(C(O)CNC(=O)CC3CC3)CC2)=O)cnc1O N1(C(C2N(C(CC(CC)O)=O)CCCC2)=O)CCCCC(C)(C)C1 C1(Cl)(C(N(CCN(C)C(c2cnnn2Cc2ccccc2)=O)C)=O)CC1(C)C c1(CN(C)C(C2CCC(n3cc(CN4CCNC4=O)nn3)C2)=O)nc(=O)o[nH]1 c12ncc(Br)c(n1)N(CCC)C2.C(=O)(C(F)(F)F)NC1COCCO1 c1(C(=O)NCC2CN(C(CN(C)C)=O)C2)ccnc(-c2ccccc2)c1N CC(CC#N)N=c1[nH]c(=NC(CCO)c2ccccc2)c2cc(F)cc(F)c2[nH]1 C1(NC(C2C(C)C2)=O)CC12CCN(C(c1c[nH]c(C#N)c1)=O)C2 C(=O)(C1COc2ccc(Cl)cc21)NC1CC(C)(NC(c2cccn2C2CC2)=O)C1 C1(C(=O)NCC2C(OCC)CN(C(=O)CN(C)CC)C2)CCCC(F)(F)C1 c1(SCC(=O)NCC2CN(C(c3scnc3C3CC3)=O)C2)ccccc1Cl c1(CNC(c2c(C)c(F)ccc2)=O)nc2c(s1)CCN(C(=O)CC(C)(C)O)C2 c1(C(=O)NCC2C3N(c4c(OC)cnc(Cl)n4)C(CC3)C2)cnc2ccsc2c1 C1(CCC)CN(C(=O)CSCCOC)CC1C(=O)NCC1CCCC(=O)N1 CC1(C)CCOC1CNC(C1CC(NC(C2CCN2C(C)(C)C)=O)C1)=O c1(-n2cc(C(CCC)NC(=O)CC(C)(C)O)nn2)cc(Br)c(F)cc1F c1(CCC(N2CC(OC)C(NC(=O)CCCC(F)F)C2)=O)cccc(F)c1F C1(NC(CC)Cc2ccc(Cl)cc2)CCc2c(OC)cccc2C1 Cn1cnc2c1CCCC2C(=O)NCC1(F)CCN(C(=O)CCCC2(C)N=N2)C1 c1(OCCC(=O)NCc2ccccc2CSC)ccccc1OC(C(=O)NC)=O N1(C(c2ccc(CC)nc2)=O)CCC(C)(C)C1CC(=O)NC(c1ncnn1C)C N1(CC)CCC(c2nnnn2CCCOC)(Nc2cnn(C(C)(C)C)c2)C(C)C1 C(=O)(C(C(C)C)SC(C)(C)C)OCC.C(c1ccccc1)=CCNC(C)=O C1(C)(CNCC(C)=CC(=O)N(C2CCCC2)CC2CC2CCN=[N+]=[N-])CC(C)=NO1 C1(C(N2CCN(C(Cc3c(C)n(C)cn3)=O)C(CO)C2)=O)CCC([N+](=O)[O-])CC1 C(=O)(C(C)(C)CCC#N)NCc1ccc(C(N(CCC(=O)OC)CC)=O)s1 CCN=c1[nH]c(C)c(C(N2CCN(C(c3cn(C)nc3O)=O)CC2C(C)C)=O)s1 c1(CC(=O)NC2CCNCC2CO)cc(F)c(Cl)cc1Cl S(=O)(=O)(c1cccc(S(=O)(=O)N(C)C)c1)NCc1c(C)csc1 N1(C(C(n2cc(-c3ccc4nc[nH]c4c3)nn2)C)=O)CCC(=C(F)F)CC1 C1(NC(c2n(C)ncc2Br)=O)CC2(C1)CC(NC(C1COCCO1)=O)C2 c1(N(CCCNC(=O)C(=O)NC2CC2C(F)(F)F)C)cccc(O)c1 C=CC1OCCCC1C(=O)NCc1cccnc1CNC(=O)C(CC)C(C)C C1(CNC(CCN(C)CC)=O)CN(C)CCN1C(=O)CC1COC(=O)C1 C1(C(N(CCCNC(C(C)CCO)=O)CC2CCCC2)=O)CC2CC1C1CC21 n1(CC(C)C)ccc2c(NC(=O)C(=O)NC(C)C)cccc12 C=CCC(C(=O)NC(CNC(=O)C(C)=CC)CC(F)(F)F)C(C)C C1(NC(C(C(C)C)C)=O)CC2CCC1CN(C(C1C3CC4C(C3=O)C14)=O)C2 Cn1nc(C(C)(C)C)cc1C(=O)NC1COCCC1NC(=O)CC1CCCC1 N1(CC)CCOC(C(=O)N(C)CCOCCNC(=O)C(c2nc(C)cs2)C)C1 c1(C(N2C(CNC(c3n(CCC)ncc3)=O)C(C)CC2)=O)cc2n(c1)CCSC2 c1(CC)ccc(C(=O)NCC2(NC(C3(F)CC=CCC3)=O)CCC2)cc1 c1(OC)nsc(C(N2CCOCC2C2CCOC2)C(=O)NC2CCOC2)c1Cl CCC(CNC(C1CCSC(C)C1)=O)(CC)C(=O)NCCC1OCCC1(C)C C(=O)(CCC1CCc2ccccc21)N1CC(NC(Cc2cnc(C)s2)=O)C(C)C1 C1(NC(C2C(c3n(C)ccn3)C2)=O)CCCC(NC(c2ccoc2)=O)CC1 N1(C(C=CC(C)(C)NC(C(=O)NC(C)C2CC2)=O)=O)CCC(CF)CC1 C1(C(C(=O)NC2CC(CSC)C2)NC(C2CCSCC2)=O)CCCC1O CCC(C)C(C(=O)NC1CC(NC(c2nnn(C)c2C(F)F)=O)C1)NC(=O)OC c1(C(c2n(CCC)nnn2)NCC(C)(C)OCCO)nc(F)ccc1Br c1(CC)cc(C(=O)N(CCC(=O)N2CC(N3CCCC3)C2)CCCO)nn1C C1(NC(C2CC23CCC3)=O)CC2CN(C(=O)CN3CCCNC3=O)CC12 C1(CNC(c2c(C)cc[nH]2)=O)CC(C)(C)CCC1NC(c1cccn(C)c1=O)=O C1(CNC(C2CCN(CC3CC3)CC2)=O)CCN(C(C2(O)COC2)=O)CC1 C(=O)(CS(=O)(=O)NC(C)(C)C)NC(CNC(C(C)=C1CC1)=O)Cc1ccccc1 CCC(CC(F)F)C(=O)NCC1CC(CNC(c2ccc(SC3CC3)cc2)=O)C1 C(C(O)C(=O)NC(C)CCCO)NC(C1(C(=O)OCC)CC1)=O c1(C(N2CC3C(CNC(CNC(CCCCC)=O)=O)(C3)C2)=O)ccc(N)cc1F N1(C(C(=O)Nc2cnn(C(F)F)c2)=O)CCN(Cc2cccc(F)c2)C(=O)C1 c1(OC)cnc(=NNC(=O)c2c(F)ccc(I)c2Br)[nH]c1 c1(NC(=O)NC)ccc(NC(N2CCC(c3nccn3C)C2)=O)cc1 C1(C(=O)OCC)CCCN(C(c2cnnn2C(C)=S)=O)CC1 C1(NC(c2c(C)cc(F)s2)=O)C2CC3C(C2)C13C(=O)NC1(C)CCCC1C n1(C(C)(C)C)cnc(C(=O)NCC2CC(CNC(c3ccsn3)=O)CO2)n1 c1(N(C)C)cnccc1C(=O)N(C(CNC(c1ccc(C2CC2)s1)=O)C1CC1)C c1(OC)c(C(=O)NCCOC(C)(C)CNC(C2CC(F)(F)CO2)=O)c(C)nn1C N1(C(C=C(CCC)C)=O)CC2(CCC2)CCC1CNC(=O)CC1CCC(O)C1 N1(C(C2=C(CC)OCCC2)=O)CCCC2(CCN(C(c3nc(Br)c[nH]3)=O)C2)C1 C1(NC(C(C)SCc2ccccc2)=O)CC2CCC1N2 CC1CCC=C1C(=O)NCC1CC(F)(CNC(c2sc(C#N)cc2Cl)=O)C1 C(=O)(C1CC(=O)Nc2cc(F)ccc21)NC1CC(NC(c2onc(C)c2C)=O)C1 c1(C(=O)NCC(CN(C(C(CC)OC)=O)C)O)cc(N(C)C)nc2ccccc12 C(C)(C(=O)NC(C(=O)NCC1CC1OC)C1(C)CC1)OCCOCC c1(CCC(=O)NCC2CC(NC(C)=O)C2)n[nH]c(=N)s1 C1(NC(C2CCC(C)O2)=O)CCN(CCNC(=O)Cc2ccco2)CC1 CC1CCCC1C(N1CC(C(N)=O)(CNC(=O)CC2CC3CC3C2)C1)=O CCC(C)(C)C(=O)N1CCCC(CCCCNC(c2ccc(OC)nc2)=O)C1 c1(C(=O)NC2C(C(=O)NCc3cccc(OC)c3)C2)c(F)c(F)c(F)c(F)c1F c1(C(=O)Nc2cccc(CNC(C3C(=C)C3)=O)c2)nccc(Cl)c1Cl C12(C(N3CCN(C(CCCC)=O)C(C)C3C)=O)CC3CC(C1)CC(C)(C3)C2 c1(OC)ccc(F)cc1C(=O)NC1CC(CO)N(C(c2ncc(Cl)cc2F)=O)C1 c1(C(=O)OC)cc(C)n(CC(=O)NC(C)(C)C(C)NC(C2CC2F)=O)n1 C1(CCNC(C(SC)SC)=O)CCN(C(c2nnc(C(C)C)s2)=O)CC1 c1(C(N2C(CNC(C34CC(C)C3C4)=O)CC3(CC3)C2)=O)ccc(N)c2ccncc12 CC(C)C(C)(C)NC(=O)CCC1CC(NC(c2cscc2Cl)=O)C1 N1(C(c2c(SC(C)C)cccc2)=O)CCN(C(c2cc(Cl)c(Cl)n2C)=O)C(C)C1 N12CCCCC1CC2=O.N1(CCOC)CCCC1C(N1CC2CC1C2)=O n1(C(C(=O)NCC(CC)N(C)C(C2(C3CCCO3)CC2)=O)C)ccc(C)n1 Cc1ccncc1CNC(=O)C(N1CCC(O)(C(F)(F)F)C1)=O C(=O)(C1=CCS(=O)(=O)C1)NCCCCCCN(C(C1(C)CCC(C)CC1)=O)C c1(C(N2C(C)(c3ccc(Cl)cc3)CCCC2)=O)cnn2c1C(CN)CCC2 N#Cc1[nH]c(=NC2CCC3CN(C(C4Cc5cscc5C4)=O)CC3C2)sc1Cl Cc1cc(C(=O)N(C)CC2COCCN2C(C2SC3C=CC2CC3)=O)ccc1Cl C(C(CC(C)C)C(=O)NCC1(CC)CCCCC1)NC(C(CC)=CCCC)=O C1(CCOC)CN(C(=O)CCC(C)CN(C)C)CCN1C(=O)C=Cc1cnc[nH]1 CCC(C)(C(=O)NCCCNCCCOCCO)C(N)=O N1(C(C=CC(C)NC(CSCC=C)=O)=O)CCC1(C)C(=O)NC N1(C(c2ccc(CC)cn2)=O)CC2COCCC2(NC(=O)CC2SC(=N)NC2=O)C1 C(=O)(C(C(C)(C)C)SCC(N)=O)N(C1CCCC(NC(CCOC(C)C)=O)C1)C C1(NC(C2CC(=C)C2)=O)CS(=O)(=O)CC1NC(=O)COc1cc(F)ccc1F C1(CC)CCN(C(=O)CNC(c2cccs2)=O)C1CNC(=O)Cc1cnccn1 N1(C(Cn2c(C)nnn2)=O)CCC(C2CCN(C(c3cc(C(N)=O)cs3)=O)C2)C1 N1(C(C(C)Cn2ccnc2)=O)CC2CCC(N(C)C(C3(F)CCCCC3)=O)C2C1 c1(C(C(=O)NCCC2CC2)N(CCS(C)(=O)=O)C(C)(C)C)cc(F)cc(I)c1 CCCCCCC(C)(CCC)C(=O)NC1(CNC(C2(C3CC3)CC2)=O)CCC1 c1(CC)ccc(C(=O)CNC(=O)CCc2nccn2C(C)C)s1.C1(=O)CO1 c1(C(N(C2CCN(C(c3c(OC)nccc3)=O)C2)C)=O)c(F)ccc(OC)c1N CC(N=c1nc2scnc2c(N2CC3(C)COCC3(C)C2)[nH]1)c1csnn1 C1(NC(C(=O)NC(C)C)=O)C2CCN(C(c3cc(O)ncn3)=O)C12 N1(C(c2scc(CNC(C(C=C)(F)F)=O)c2)=O)CC2CCCC(O)C2C1 N1(C(c2c(CC)cco2)=O)CCOC2CN(C(C3CC3C(C)(C)C)=O)CC12 CC1CN(C(c2coc(C#N)c2)=O)CC(CCNC(c2c[nH]nc2Br)=O)O1 NS(=O)(=O)CCCC(=O)NC1CCC1NC(C1CCc2nc[nH]c2C1)=O c1(NC(N2CC(CCCCOC(CN(c3ccncc3)C)=O)C2)=O)cc(N)ccn1 c1(NC(N2CCCN(CCCOCC(F)(F)F)CC2)=O)ccc(F)c(Br)c1 C12(C(=O)NC(C3CCN(C(C4(C5CCC5)CC4)=O)C3)C)CCCC1CC(=O)CC2 C1(NC(=O)CCN(CCCO)C(c2nc[nH]n2)=O)CN2CCCC1C2 C1(NC(C2C(C(C)C)C2)=O)CCN(C(c2csc(-c3nc[nH]n3)n2)=O)C12CC2 CC(O)(C(=O)N1CCCN(C(=O)Cc2csnn2)CC1)C(F)(F)F C(=O)(CCCC(F)(F)F)NCCC1(C)CCN(C(c2cc(CC)oc2C)=O)C1 C1(CNC(=O)C=Cc2cocn2)CCC2(CN(C(c3nscc3Br)=O)C2)O1 C1(C(N(CCOC)CCNC(=O)C(C)OCC2CC2)=O)COc2ccccc2O1 CC1=NS(=O)(=O)N(C)C=C1C(=O)N1CC2CC1C2NC(=O)CC1CC=CCC1 CCC(C)(CC)C(=O)NCCC(O)C(=O)N(C)CC1CC(O)C1 C(=O)(C1CCCn2c(Br)cnc21)NCCC(C)NC(c1c(C)ccnn1)=O N1(C(c2cc(CC)[nH]n2)=O)Cc2n[nH]cc2C1C(=O)NCC(C)(C1CC1)OC C1(NC(=O)Cc2ccc(Cl)s2)CCC12CCN(C(C1(C3CC3)CCCO1)=O)CC2 c1(C(=O)NCCSC)occc1CNC(C1(n2cncn2)CC1)=O C(=O)(CCC(=O)N1CCC(O)CC1)NCC(C(C)C)NC(C1(SC)CC1)=O C1(NC(C=CC2(C)COC2)=O)(CNC(C2(C)C=CCC2)=O)CCC(F)(F)CC1 C=C(C)C(C)(C)C(=O)N1CC2(C1)CN(C(C1(C)CCCC1C)=O)C2 N1(C(C2CCCC2OC)=O)CC2CCN(C(C3(O)CN4CCC3CC4)=O)CC2C1 C1(NC(C(CC#C)C2CC2)=O)CN(C(c2cccc(Cl)c2Cl)=O)CC12CC2 CS(=O)CCC(=O)NCC(=C1CN(C(=O)CC2CCC(=O)NC2)C1)F N1(C2CCN(C(CC)C(N)=O)C2)CCN(C(=O)CC2CCS(=O)(=O)C2)CC1 c1(C(N(CC(CC)NC(c2ncncc2C)=O)C)=O)c(Cl)n[nH]c1C N1(C(c2c(C)coc2)=O)CCC(NC(c2ncsc2S(N)(=O)=O)=O)CC(C)(C)C1 N1(C(C2CCN(C)C2=O)=O)CC2CCC(C1)N2C(c1nc(=O)n(C)[nH]1)=O C1(O)(C(CNC(c2c(C)onc2)=O)C)CCN(C(=O)CN2CCCC2=O)C1 c1(CCNC(N2CC(C(=O)OCC)CC2(C)C)=O)cc2ccccc2s1 Cc1cc(Cl)ncc1C(=O)NCCN(C1CCCCCC1)C(c1nccn1C)=O c1(C(=O)NCCCCC2(NC(CC=CC=C)=O)CC2)ccnnc1O N1(CCC(=O)NCCC(C)NC(C2CC3(C2)CC3F)=O)CCCCCC1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CC(NC(=O)C(CC)C2CCOCC2)CCC1C CC1Cn2nc(C(=O)NCC3CCN3C(c3ccc(Br)o3)=O)cc2C(=O)N1 N1(C(c2cn(C)nc2O)=O)C2COCC1CC(NC(=O)CN1C(=O)CNC1=O)C2 N1(CCC)CCCN(C(C2(CO)CCN(C(c3c(C)cccc3C)=O)C2)=O)CC1 c1(NC(=O)Nc2ccc(CNC(=O)C(F)(F)F)nc2)ncnc2c1OCCO2 C12(NC(C(CCSC)NS(=O)(=O)c3cccs3)=O)CCC(C#N)(CC1)CC2 C12(CNC(C3(CC=C)CC3)=O)CC3CC(CC(C3)C1NC(=O)CCF)C2 Cc1cccc(C(N2CCC(OCCNC(c3c(C)[nH][nH]c3=N)=O)C2)=O)c1Cl C1(NC(C2C(C(=O)OC)C2)=O)CN(C(c2ccnc(OC(F)F)c2)=O)CC1(C)C c1(SCC)ccc(C(=O)NCC2C=CC(NC(=O)CN(C)CCO)C2)cn1 C(=O)(C(C)CS(C)(=O)=O)NCc1c(CCNC(c2ccc(C)cc2C)=O)ocn1 Cc1ncccc1CC(N1CCCC1CCC(=O)NC(c1cnc[nH]1)C)=O c1(C(=O)NCC2OCCC(NC(C=C(CC)C)=O)C2)c(C(F)(F)F)cccc1F C(CC(CC)C(=O)NCC=CCNC(c1cnc(O)n1CC)=O)=CC C(=O)(C1COc2ccc(Cl)cc21)NCC1C2CN(C(Cc3nnc(C)o3)=O)CC21 N1(C(C2OCC(C)C2)=O)CCc2sc(CNC(=O)Cn3cc(CO)nn3)nc2C1 C(=O)(C(C)C(F)(F)F)NC1C(SC)CN(C(=O)CC(c2cccs2)C2CCC2)C1 N1(C(C2CC(NC(C(C)CCN(C)C)=O)C2)=O)CCOCC(C)(O)C1 CC1CC(NC(=O)COC(F)F)CN(C(c2ccncc2Cl)=O)C1 Cc1cc(-c2nc(C3CCCC3O)n(-c3ccc(Cl)nc3)n2)ccc1F c1(C(C(=O)NCCOC)N(CC(C)C)C2CC2)ccc2c(c1)OC(F)(F)O2 CCCCN=C(NCC(C)(C)C)NC1CCOC(c2cccc(Cl)c2)C1 c1(C(N(C(CCNC(C2=C(C)OCC2)=O)C)C)=O)cc2c(nc1O)CCCC2O c1(C(C)(C)C)cc(NC(=O)NC2CCOC2c2ccccc2)n(CCO)n1 CN1CCCCC1CC(N1CCCC1Cn1cc(CC(C)(C)CO)nn1)=O C1(C(=O)NCc2nc(CNC(c3cnc(=N)[nH]c3)=O)sc2)CCn2nccc2C1 C(=O)(C(CC)C(=O)N1C(C(N2CC=CC2CF)=O)CCC1C)OCC CCCCC(C(=O)N1CC2CC1CN2C(=O)CCOC)NC(N)=O Cc1cccc(C(C(C)C)NC(=O)C(=O)NCc2ccc(C)s2)c1 C1(CCC(=O)NCC(=C)Cl)CCCN(C(=O)C(C)OCCCC)C1 CCC(CC(=O)N1CCC(N(C)C(c2cc(OC)cnn2)=O)C1)CC(C)C c1(CCC(=O)NCC(C)NC(CC=CCC)=O)cccc(C(=O)OC)c1 N1(C(CN2C(C)CC2)=O)CCCC(NC(c2cc(C3CC3)no2)=O)C1 C1(C(N2CCC(CNC(C(C)c3ccco3)=O)CC2)=O)CC2(CCCCC2)C1 C(=O)(C1CCc2cccnc21)N1C2C(NC(C3CC(=C)C3)=O)CC(C2)C1 c1(C(=O)NC2CCN(C(c3nc(CC)sc3)=O)CC2F)cnnc2ccccc12 C(=O)(C(C)(C1CC1)N(C)C(C1CCOC1C(C)C)=O)NCC(C1CCC1)OCC N1(C(C(c2ccncc2)C)=O)CC2(CC(NC(=O)C(F)C(F)(F)F)CO2)C1 c1(C(=O)NC(CNC(C(C)SC)=O)CO)cccc(=S)n1O C1(CNC(=O)CCC2CCCCO2)CC(F)(F)CN1C(c1cccnc1S)=O C1(NC(Cc2cn(CC)nc2)=O)CCC(CNC(C2CC(N(C)C)C2)=O)CC1 O=C1c2ccccc2-c2n[nH]c(=NCCCc3ccncc3)cc21 c1(NCc2[nH]nc(C(=O)OCC)n2)ncc2c(ncn2C)n1 C1(COC)(NC(C2CNC(=O)C2)=O)CN(C(=O)CCn2cncn2)C1 O=S(=O)(c1cccc(=NCc2cc(C3CC3)no2)[nH]1)NCCC1CCCCO1 C1(CC)CN(C(c2scnc2C)=O)CCN1C(=O)C(c1ccccc1)C1CC1 c1(OCCNC(=O)NCCC=C=C)ccc(F)c(Cl)c1 CN1CCN(C(N2CCC2(C)CCO)=O)C(COCC2CC2)C1 C1(CNC(C(CN(C)C)(C)C)=O)COCCN(C(C2CC3(CC3)C2)=O)C1 Cc1ccnc(C(N2CC(CC(=O)O)C(C)C2)=O)c1Br CC1CCCCC1(CO)NC(c1n[nH]cc1CNC(C1CNC(=O)O1)=O)=O c1(OC)c(C(N2C3CCC2C(NC(c2occc2C2CC2)=O)C3)=O)ccnc1Cl c1(NCC(c2cn(C)nc2)O)ccc(S(=O)(=O)NCC2CCOCO2)cc1Cl c1(C(N2C(C(C(=O)NCC=CC)C)CCC2)=O)ccc2occc2c1 c1(OC)cc(CN(C2CS(=O)(=O)CC2O)C)c(Br)cn1 C#CC1(O)CCN(C(=O)C(CC2CC2)NC(=O)C(C)OCCN(C)C)C1 C1(C(N(C(C(=O)NC2(CCC)CC2)C2CC2)C)=O)CCOCC1 N1(C(c2cnc(C)s2)=O)CCCC(NC(C2CCCN2C2CC2)=O)CC1 C12(NC(c3cc(O)nc(O)n3)=O)CCC(C1)N(C(c1nc(Cl)ccc1Cl)=O)C2 CCC(CC(C)C)C(=O)NC1COC2C(NC(C3(C(=O)NC)CC3)=O)COC12 c1(-c2cn(CC#N)nc2)cccn2ncc(C(N3C4CCC3CC(O)C4)=O)c12 C(CC(C)CC)(C(=O)N(C)CC=C)NC(c1cncc(C#C)c1)=O C#CCCC(O)C(=O)N1CCC(CC(C)NC(c2ccc(C3CC3)nc2)=O)CC1 C1(COC)(CNC(C2(OC)CCSC2)=O)CCCN1c1cc(C(F)F)ncn1 CCC(C(=O)NC(C)CC1CCN(C(=O)Cc2ccc(O)cc2)CC1)C(F)(F)F CC1(C)COCCN(C(C2COC(CNC(c3ccc(=N)[nH]c3)=O)C2)=O)C1 C(=O)(CCCN=c1nccc[nH]1)N1CCN(C)C(CNC(C2CC(F)C2)=O)C1 c1(C(=O)NC(C2CN(C(C3(OCC)CCC3)=O)C2)C)nc(O)nc(O)c1F C(=O)(CC(=O)N1CCCC1C1(NC(C2CC2c2cccs2)=O)CC1)OCC c1(NCC(c2ccccc2)C)sc(CC(=O)O)cc1C#N c1(OC)c(Nc2ccc(Cl)cc2)cccc1N(C(=O)CC1CC(F)CN1)C1CC1 N1(CCC)CC(C(N2CC(N(C(C3C4CC5C(C4)C35)=O)CC)C2)=O)CC1=O c1(C(=O)NCC2(CCNC(C(C)C3CCOC3)=O)CC2)ccc(P(C)(C)=O)o1 c1(C(c2ccccc2)NC(=O)NC2OCC(CC(=O)OC)C2)cccc(Br)c1 C(=O)(C(C)(C)CC(C)(C)C)NC1CC(NC(C2(COC)C=CCC2)=O)C1 N1(C(C(=Cc2ccco2)C)=O)CCC(C)(C)C(C(=O)NCC(C)(C)CC(C)O)C1 C(=O)(CC(C)C(C)C(C)C)N1CC(O)(CNC(CCSCC)=O)C1 Cc1nnc2cnc(C(=O)NC3CC4CCC(C3)N4C(C3(C#N)CC3)=O)cn12 c1(CC)cc(OC)cc(C(=O)NCC2CN(C(C3(C(N)=O)CCC3)=O)CCO2)c1 c1(C(=O)NC2C3CN(C(CCCNC(C)=O)=O)C2C3)c(F)cccc1Br C(=O)(C1=CCCCC1C)N(CC(CNC(C(n1cc(C)nc1)(C)C)=O)(C)C)C C1(C(=O)O)C(O)C(O)CCN1C(=O)NC1CCCC1F N1(C(C(COC(C)=O)C)=O)CCC2CC2(C(=O)NCCCC(C)CO)CC1 N1(C(c2c(C)ccnc2)=O)CC2CCCN(C(=O)C(F)(F)CF)C2C1 C1(NC(C(C)Cc2cccc(Br)c2)=O)CC2C1CCN2C(c1ccns1)=O N1(C(C(C(C)C)F)=O)CCC2CCC(C1)N2C1CCN(c2ccccc2)C1=O Cc1ncc(C(=O)NCC2(C)CCC(NC(C3(NC(C)C)CC3)=O)C2)c(C)n1 C1(NC(c2c(CC)onc2)=O)CCN(C(=O)C(c2ccccc2C)C)CC1CC C1(SCn2nc(C)n3c2ncn3)CC2CCCC2N1C(=O)OC(C)(C)C C1(Nc2ncc(C)cn2)CCCN(C(c2cnc(-c3ccco3)s2)=O)CC1 C1(O)(CC(=O)NCCC2(O)CCN(C(CCCC=C)=O)C2)COC(C)(C)C1 Cc1[nH]nc(C(=O)NC2CN(C(c3c[nH]nc3C3CCC3)=O)CC2C(F)F)c1Cl Cn1c(=O)ccn(CC(=O)NC2CCC(NC(c3csc4cncn34)=O)C2)c1=O c1(C(=O)NCCC(C(=O)NC2C(C(N)=O)CC2)O)n[nH]c2c1CCC2 N1(C(c2nn(CC)c(O)c2)=O)CCN(C(=O)CCCSC)C(CC2CC2)C1 c1(CC(N2C(C(=O)NC3CN(CCC)C3)CCC2)=O)ccccc1F C1(C(N2C(C(=O)NC(C(=O)NCC)C)C3CC3C2)=O)CC2(C1)CC21CC1 C1(NC(C2(C(C)(F)F)CC2)=O)CCCCC1NC(=O)C=CC(F)(F)F N1(C(=O)Cc2ccon2)CCCCC(NC(=O)C(F)(F)CC2CCCO2)C1 N1(C(c2cccc(OCC#C)c2)=O)CCN(C(C2(C#N)CC(C)C2)=O)C2(CC2)C1 C1(C(N2C(CN(C(CC(C)(F)F)=O)C3CC3)CCC2)=O)CCCC12CCC2 N1(C(c2c(CC)nc(=N)[nH]c2)=O)CC2(C1)SCCC2NC(c1cnc(C)[nH]1)=O C(C(CC(=O)N=c1cc(C2CC2)n(C)[nH]1)C1CCC1)NC(C(C(CC)O)C)=O Cc1nc(C)n(CC(=O)NC(CCC2CC2)C(=O)NC(C(C)C)c2nc[nH]n2)n1 Cc1ccc(OCC(N2CC(NC(=O)C(F)F)CC(O)C2)=O)c(Br)c1 C1(C(N2CC3CC(C)C3C2)=O)CC12CCN(C(C1COCC1(C)C)=O)CC2 c1(C(=O)NC2(CO)CN(C(Cc3ccc(C)s3)=O)C2)nc(C)sc1C C12(C(=O)NC3C(CNC(C(C)=C4CCCC4)=O)CCCC3)CCCN1CCC2 C1(C(CC)NC(=O)N(CCO)Cc2ccncc2)Cc2ccccc2C1 c1(CCOC)nc(COc2ccsc2Cl)n(-c2nccn2C)n1 c1(CCC(=O)N(CCC(C)NC(C2CCC(CCO)CC2)=O)C)ccc(F)nc1 c1(NC(C2N(C(CC3(CC)CCC3)=O)C(C)CC2)=O)ccc(CO)c(F)c1 c1(C(=O)NC(C(=O)NC(CC(=O)OC)C)CC2CCOCC2)ccc[n+]([O-])c1 C1(NC(CN2C(C)CCCC2)=O)CCN(C(C2CCOC(C)(C)C2)=O)C1(C)C c1(C(=O)NC(CC2CCN(C(C3C(OCC)C3C)=O)CC2)C)c(C)cccc1O C1(CNC(C2(C)CCOC2)=O)CCCCN1C(C1(C(F)F)CCCC1)=O c1(C(N2CCCC(CN(C(C(C)CF)=O)C)C2)=O)cc(Cl)c(F)cc1Cl C(C)(C(=O)NCC1CCC1NC(C1(CC(F)F)CCC1)=O)=CC C#Cc1ccc(C(N2CCCC(O)(CNC(c3ccnn3CC)=O)C2)=O)c(C)c1 N1(C(C(CCC)C)=O)CCN(C(c2ccc(OCCOC)cc2)=O)C2(CCC2)C1 C1(C(N(CCN(C(=O)C=CC2CC2)CC)CC)=O)CC1C(F)(F)F C1(C(=O)NCC2(O)CC(NC(c3n(CCC)nc(C)c3)=O)C2)CCCC12CCC2 N1(C(=O)CC2CC(O)CN2C(C2CC2Cl)=O)C2CCC1CC1(CC1)C2 N#Cc1ccc(F)c(F)c1NC(C1CCCCN1Cc1cc(CO)ccc1O)=O C#Cc1ccc(C2(C(=O)NC3CC(CNC(=O)CCS(C)=O)C3)CCCC2)cc1 CC(C)C(CNC(=O)Cc1cn[nH]c1)NC(=O)CNC(=O)C1CC1 CC(C)CC(C)(O)C(=O)N1CCN(C(c2ccoc2Cl)=O)C(C(C)(C)C)C1 N1(C(C=C(CCC)C)=O)CCCC12CCN(C(=O)C(O)C1=CCCCC1)C2 N1(C(c2ccc(CC)s2)=O)C2CCC1C(NC(c1ccc(C)cn1)=O)C2 C(=O)(C(C)(C)C(=O)N(C)C)N1C(CN(C(C(COC)N(C)C)=O)C)CCC1 n12nc(C)cc1C(=O)NC(=O)C2.C(c1cc[nH]n1)=CCN(CC)CC C1(NC(Cc2ccn(CC)n2)=O)CCCCN(C(c2cnnc(C)c2)=O)C1 c1(C(=O)NC(C2CCN(C(c3c(C)nns3)=O)CC2)C)cccc2c1OCCC2 N1(c2cc(OC)ncn2)CCC(C2CCN(C(c3cc4n(n3)CCC4)=O)CC2)C1 c1(OC)ccc(C(=O)NC2CCCC(N(C)C(c3occ(C)c3C)=O)C2)nc1N N1(C(c2n[nH]cc2CCC(F)(F)F)=O)CCC2(CCCN2C(C2CCCO2)=O)C1 c1(C(C)NC(C2CC2C(=O)NCCNC(N)=O)=O)ccc(F)c(F)c1 C=CC(F)(F)C(=O)N1C(C(=O)NC(c2cccnc2O)C)CC2CC12 c1(C(=O)NC2C(CC=C)C(O)C2)ncc(OCC2CC2)cc1F C=CC1CN(C(c2ccn(C3CC3)c2C)=O)CC1NC(C1COCCN1CC)=O c1(C(=O)NCC2CC(NC(C3(CCOC)CC3)=O)C2)cccc(C#N)c1 N1(C(C(CCC)=CCC)=O)CCCN(C(=O)CCNC(N)=O)CC1C(C)C c1(C(=O)NC(C)CCNC(C2(Cl)CC2)=O)nc2ccccn2n1 C1(C(=O)NCCOC)CC(O)CN1C(=O)CCC1CCCN1C c1(CC)ccc(N)c(C(=O)NC2CN(C(=O)CNS(=O)(=O)NC)CC2(C)C)c1 N1(C(c2n[nH]c(C)c2Cl)=O)CCc2ccc(C(=O)NCC3CC=CCC3)nc2C1 C(=O)(N1CCC(C(N2CCCC3(C2)N=N3)=O)O1)C1C2CN(C)CC21 Cc1cc(CN2CC(F)CC2C(N2CCC(O)C(C)C2)=O)c(F)cc1Br N1(C(Cn2c(C)ncc2)=O)CCC(C)C(NC(c2cc(C(N)=O)cc(F)c2)=O)C1 c1(C(=O)NCC(CNC(CSc2n(C)ccn2)=O)(C)C)cccc(P(C)(C)=O)c1 N1(C(CCC#CC)=O)CC(C)(C)CC1C(N1CC([N+](=O)[O-])C1)=O CC1CN(C(=O)C(C2(O)CCCCC2)(F)F)CCN1C(C1CC(C)(C)CN1C)=O C1(C(=O)NCC2CN(C(c3nc(C(C)(C)C)no3)C)C2)CCc2cncn2C1 CC1=C(C(=O)N2CC(C(O)C(=O)N(C)Cc3ccc(F)cc3)C2)CCCO1 C(=O)(C1=CCCN(C(C2CCN2CC)=O)C1)N1CCN(CC)CC1 n1(CC(=O)N(C)CC2(NC(C(CC=CC)C)=O)CC2)cc([N+](=O)[O-])ccc1=O c1(C(=O)NC(CNC(c2c(CC)n(CC)nn2)=O)(C)C)cc(C)nc(O)n1 C=CCC(CC=C)C(=O)NCCC1=CCN(C(=O)C=C(C)c2cccnc2)CC1 N1(C(COCC(=O)OC)=O)CC2(CC2)CC1CNC(c1cn(C)c(=O)cn1)=O N1(C(C=CC2CCN(C(C(CCCC)=O)=O)CC2)=O)CC(C)(C)OCC1(C)C c1(C(=O)NCCc2ccsc2)cnc2c(-c3ccc4nccn4c3)cnn2c1 N#Cc1cc(N2CCC(C3OCC3(F)F)CC2)nc(-c2ccccc2)n1 CCC(C(=O)NC1(CCNC(c2cncc(C(C)(C)C)c2)=O)CC1)C(C)O c1(SC)cn(C)nc1C(=O)NC1CN(C(=O)Cc2cnccn2)CC1O C#CC1CC2CCC1N(C(C1(NC(=O)C(N3CCOC3=O)C)CC(O)C1)=O)C2 Cc1cccc(CNC(c2ccsc2)=O)c1.C1(COCCC(=O)N2CC2)(O)CCOCC1 C1(C(N2CCC(N(C(=O)CCSC(F)(F)F)CC#C)C2)=O)CCCC(OC)C1 C12(NC(CC3C(CC)C3)=O)CCOCC1CN(C(=O)Cn1cnc(C(N)=O)n1)C2 C(=O)(CC(C)(C)CC(F)F)NCCOCCN(C)C(C1(F)CCS(=O)(=O)C1)=O CC(C)C(O)C(C)C(=O)NCC1(C)CCN(C(c2cn3ncccc3n2)=O)CC1 N1(C(C(COC)N(C)C)=O)CCC2(CC(NC(=O)CCSC3CCC3)C2)C1 c1(C(=O)NC(CNC(Cn2ncc(C)c2)=O)C)cnc2c(c1)c(C)nn2CCO C1(O)(CC)CCCN(C(=O)C(C)(CO)NC(C2COCC2C(N)=O)=O)C1 C1(OC)C(OC)CN(C(=O)CCS(C)(=O)=O)C1CNC(C1(C)CCCS1(=O)=O)=O N1(C(CCCN(C(CCC2CC(OC)C2)=O)C)=O)CC(C)(C)C12CCC2 c1(COC2CCC(C(N)CCCc3ccccc3)C2)ccc(I)cc1Br N1(C(Cc2c(C)cc(C)s2)=O)CC(NC(=O)CO)CC(O)C1 C(=O)(C(=O)NNC(=O)c1ccco1)Nc1ccc(OC)c(OC)c1 Cc1cc(C(=O)NCC2CC2NC(=O)CCOc2ccc(C)cc2C)nc(O)c1 C#CC1(C(N2CCC(C(C)(C)C)C2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 C#CCCC(O)C(=O)NCC(O)CCNC(C1CCC(C)CC1)=O N1(C(C2(C)ON=C(C)C2)=O)CC2CCN(C(=O)CCOc3cccnc3)CC12 N1(C(CCc2cn(C)nc2)=O)CCCC1(C)CNC(C1CC1OC(C)(C)C)=O C(=O)(C(C)(C)CCC(=O)N(C1CCCN(C(=O)C(O)CC(N)=O)CC1)C)OC n1(CC)nccc1CNC(=O)CCN(C(=O)CCCN(C)C(C)=O)C1CC1 c1(CSCC)cccnc1C(=O)NCC1C=CC(NC(c2c(C)noc2N)=O)C1 C1(C(N(C(C(N)=O)C2CC2)C)=O)CC(F)(F)CN1C(=O)CCOC1CC1 N1(C(=O)OCc2cc(OC(C)C)cc(Br)c2)CCC(C2CCCC23OCCO3)C1 N1(C(=O)CCCN2CCOC2=O)CCC(c2ncc[nH]2)CC1 c1(C(=O)NC(CC#C)C)cc(CNC(c2c[nH]c(=N)o2)=O)cs1 Cc1cncc(CC(=O)NCCCCC2CN(C(=O)C(C)SC(F)(F)F)C2)c1 C1(COC)(NC(=O)CC2NC(=O)NC2=O)CCN(C(=O)CC2CC(N(C)C)C2)C1 C1(O)(CCNC(C(CC)=CC)=O)CCCN(C(=O)CC(O)c2ccccc2)C1 N1(C(c2cc(COC)no2)=O)CC2CC(N(C(=O)C(C)n3ccnc3)C)C1C2 Cc1noc(C)c1C(C)C(=O)NC(C1CCN(C(=O)CCOCC(C)(C)C)C1)C CCCCCCC(=O)N1CCC(N(C(=O)C(=Cc2ccccc2)OC)C)C1 c1(C(N2CC(N(C(C(CC)C(C)(F)F)=O)C)C2)=O)cc(SC)ccc1[N+](=O)[O-] Cc1ccc(OCC(=O)NC(c2cccnc2)CNC(=O)C=CC(C)C)c(F)c1 c1(C(=O)NC2CC2CNC(c2cn(C3CCOC3)cn2)=O)cc2cccnn2c1 C(=O)(C(C)(C)S(C)(=O)=O)N(C(C)CNC(C1CC1C(F)(F)F)=O)C N1(C(C23C(CN(C(CCOC)=O)C2)COC3)=O)CCCC(N=[N+]=[N-])CC1 N1(CC2C(C#N)C2)CC2CCC(C1)C2c1nc(-c2cccnc2)no1 N1(CC(N2CCC(OC)(CNC(c3c(C)csc3Cl)=O)C2)=O)CCC(=O)NC1=O c1(C(=O)NC2(C(N(CC#C)CCOC)=O)CCC2)cc(C(C)C)no1 C1(C(N(C)CC2(O)CCCCC2)=O)Cc2ccccc2O1 C1(OC)CC2CCC1CC2C(N1CCOC(CCCNC(=O)C(C)=C(C)C)C1)=O c1(OC(=O)CCn2cccn2)ccc(-c2nc[nH]n2)nc1.C12CCN(C1)C(=O)N2C C1(C(=O)OC)C(NC(=O)Cc2cccc(C)c2Cl)C2CCCC12 c1(C(=O)NC2CCCC(NC(C3CC4(CC4)CO3)=O)C2)cc(Cl)cc(F)c1F N1(C(CC2(C)CCOCC2)=O)CC(NC(C2CCC(=O)NC2)=O)C2(CC2)C1 C=C=CCCC(=O)N1CCC(CC=C)(C(=O)NCC(C)(O)CCC)C1 c1(COC)n[nH]c(=NCC(C)(C)NC(C23CCCC2C3(F)F)=O)s1 c1(C(N2C(C)CCC(NC(=O)CCn3ccnc3)C2)=O)cnc2ccncc2c1 C12(CCNC(CCOCCCOC)=O)CCC(C1)N(C(=O)C(C(C)C)OC)C2 C1(C(N(C)Cc2cnco2)=O)CN(C(=O)C(c2cccn2C)=O)CCO1 C(CC(=O)Nn1nnc(C)c1C)C1(NC(c2c(CC)ncnc2)=O)CCC1 Cc1ncnc(N(C)CC2CCCN2C(c2ccoc2Cl)=O)c1Br CC1CCC(O)(C(=O)NC(C2CCN(C(C3CC(N=[N+]=[N-])C3)=O)C2)C)CC1 C1(C(C(=O)NC2C(C(N(C(CC)C)C)=O)CC2)C)CCCCC1 C1(C(=O)NC(c2ccccc2)C(=O)N(CC#CC)CC#C)CC=CCO1 c1(C(=O)NC2CCC(NC(=O)C(O)c3ccsc3)C2)nc(Cl)c(Cl)s1 OP(=O)(C=CCN(CC(=O)O)C1CC1)OCC.N1(CC)CCC(C2CC2)(O)C1 C1(CCNC(=O)CCc2ccccc2)CC(N=c2[nH]nc(-c3ccccc3)o2)C1 C1(CNC(c2nc(OC)oc2)=O)(CO)CC12CCN(C(=O)CSCC(N)=O)CC2 C1(C(=O)NCC(C(=O)NCC2(CC)CC2)CC2CC2)CCCCCCC1 C1(NC(c2nc(CC)sc2N)=O)CC2CC1CN(C(=O)COCC(C)(C)C)C2 C1(C(=O)NC2CC(CNC(c3sccc3Br)=O)C2)OCC2CCCC1C2 c1(CC)cc(C(=O)NC2CC3(C2)CC3NC(C2CCCCC2(C)C)=O)cc(Cl)c1 c1(C(=O)NC(C(COC(CCC(C)OC)=O)(C)C)=O)ccc2ccccc2c1 c1(C(N2CC(N(C(=O)CC3CC3C(F)(F)F)C)C(F)C2)=O)c(F)cc(F)cc1F CCCC(CC)CCC(=O)N(C)CC1(O)CCCN(C(=O)Cn2cc(C)cn2)C1 N1(C(=O)OC(C)(C)C)CCN(C(C2(F)CCOC2)=O)C(c2ccncc2)C1 CC1(C)C(NC(C2CC(=O)N2)=O)CCN1C(=O)C(C1CCCCCC1)O c1(SCC2(COC)COC2)cc(C)c(Br)cc1C CCC(C)(C)C(C)CC(=O)NCCC1CCN(C(c2cccn2C)=O)C1 C1(C(=O)NC(c2cnn(C)c2)C(=O)Nc2cn(CC#C)nc2)CC=C(C)CC1 C(=O)(C1=NNC(C(F)(F)F)C1)NC(C(C)NC(=O)CCn1cnnn1)(C)C c1(C(CC2(OC)CCC2)=O)cnn(C)c1C(=O)N(C1CN(C2CC2)C1)C.C1CO1 C1(NC(C(C2CCC2)OCC)=O)CN(C(c2ccn(CC)n2)=O)CC1CO c1(OC)cc2c(cc1C(=O)N(CC(C)NC(C1(CO)CCC1)=O)C)CCC2 C1(C(=O)OC)CCC(N(C(=O)OC(C)(C)C)CC2(c3cc(C)ccc3O)CC2)C(O)C1 Cc1ccc(C=CC(N2CC3CC3(CNC(c3sccc3C#N)=O)C2)=O)o1 N1(C(C2CC(CC)N(C(c3coc(C(N)=O)c3)=O)CC2)=O)CCNC(=O)CC1C N1(C(C(C2CCCCCC2)COC)=O)CCCCC1C1CCCN1C(C)=O N1(C(C(N2CCN(c3n(C)ccn3)CC2)=O)=O)CCC(C2CNC(=O)C2)C1 N1(C(C(C=C)(C)C)=O)CCC2(CC1)CCN(C(C1CC(CCO)C1)=O)C2 c1(NC(=O)NCC(COC)(C)OC)ccc(-c2nccn2C(F)F)cc1 c1(N(C)C)ccc(Cn2nc(-c3cc[nH]n3)nc2CC2(C(F)F)CCCC2)cc1 c1(C(=O)NC(CC(=O)OC)COC)ccn2cncc2c1.c1(C)cccc(CO)c1 CCC(O)(CC)c1cn(C2CCN(C(=O)CC3(CSC)CC3)C2)nn1 N(C1CC2(CN(C(c3csnn3)=O)C2)n2ccnc21)C(c1c(C)cno1)=O N1(CC(C(C)c2ccccc2)O)CCN(c2ccc(C(F)F)cc2)CC1 N1(C(Cc2nc(C)sc2)=O)CC(C(=O)NCC(C)(C)CCO)CC(C)C1 C1(CNC(c2sccc2Cl)=O)CCN(C(C2CCC(CN3CCOCC3)O2)=O)C1 Cc1ccc2c(c1)C(C(=O)NC(CNC(=O)Cc1cccc(F)c1)C1CCC1)C2 N1(C(c2c(CC)cc[nH]2)=O)CCC=C(C(=O)NCC(=O)N(C)C)C1 N1(C(C(C(C)C)SCC)=O)CCCC(C)(NC(c2cc(C)ccc2F)=O)C1 c1(-c2ccc(C#N)cc2)csc(=Nc2cccc(Cl)c2)n1CC1CCC(=O)N1 c1(C(=O)NC(CNC(c2cc(CC)on2)=O)CO)[nH]c(=N)ccc1Br C=Cc1cc(C(N2CCC2CO)=O)cc(F)c1.C12CCC(C1)C(=O)N2 C1(CNC(Cc2nc(C)sc2)=O)CC2CCC1N2C(=O)CCn1ccc(=N)[nH]1 N1(C(C(CC(C)C)C)=O)CCC2CCCC(C1)N2C(=O)C(F)=CC1CC1 c1(CSCC(=O)NCC2N(C(C3C(SC)C3)=O)CC(OC)C2)ccc(F)cc1F N1(C(c2cn(CC)nc2C)=O)CC(N(C(=O)CCOC2CC2)C)C(C)(C)C1 C1(C2CCN(C(c3cccnc3OCCO)=O)C2)(NC(C=CCC)=O)CC1 Cc1[nH]c(C(C)(C)C)cc1C(N1CCN(C(c2cccc(N)n2)=O)CC1)=O c1(C2C(=O)N2)scc(C)c1C.C1(CN(C(=O)OCOC(C)(C)C)CC)CC(F)(F)C1 CC1(C(=O)NC(CNC(c2cc(C3CC3)oc2C2CC2)=O)CO)CC2CCC1O2 C(=O)(C(C(C)(C)C)OC)OC.C1(=O)CC(C2CC2)CN1C1CCC1 c1(CN2CCC(N(C)C(c3cc(Br)cc(F)c3F)=O)C2)cc(F)cc(C#N)c1 C12(C(N(C3CCOC3)CC#C)=O)CCCC1N(C(c1ncn3ccccc13)=O)CC2 O=C(C(F)(F)C1=CCOCC1)NCC1CC(NC(=O)COCC(=O)OC(C)(C)C)C1 N1(C(C2(F)CCN(C(C3CCCN(C)C3)=O)CC2)=O)CCC2(CCCCO2)C1 C(=O)(CCCCCN(C)C)N1C(CNC(C(c2ccccc2)SC)=O)CC(F)C1 C#CCCC(O)C(=O)NCCN(C)C(c1cc(-c2ccncc2)on1)=O O=C(C(O)CCc1ccccc1)N1CCC(CCNC(C2(O)CCOC2)=O)CC1 CC1=NN(C)C(=O)C1CC(=O)NC1CCCN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 Cc1ccc(CN(C2CCNCC2)C(=O)CCc2ccccc2)cc1 C(=O)(CCCCCCNC(c1cnn2ccccc12)=O)NC(C#C)CC1CC1 N1(CC(C)NC(c2ccccc2)=O)CCC(=O)N(C(C2CCCCC2)(C)C)C1=O c1(CC)ccc(OCCC(N2CC(NC(C3CCCCC3)=O)C(C)C2)=O)cc1 c1(C(N(C2CCC(NC(=O)C=CS(C)=O)CC2)C)=O)ncc2c(F)cccn12 c1(C(=O)NCC(CNC(c2[nH]ccc2C2CC2)=O)O)c[nH]c2cc(F)ccc12 C=CC(C)(C)CC(=O)NCCn1cnc(C(=O)NC2(c3nc[nH]n3)CCC2)c1 C1(C(=O)NC2(CF)CCN(C(C(C#C)(C)C)=O)C2)CCC2(CCOCC2)O1 C1(NC(c2nc(SC)sc2)=O)CN(C(=O)C(C(C)C)OCC(C)C)CC1SC N1(C(C2C(CCOC)C2)=O)CC(O)CCC1C(=O)N(CC(O)CO)C c1(OCC#C)ccc(C(=O)NC(c2ccccc2F)C(F)(F)F)c(F)c1 N1(C(C(c2ccc(Cl)cc2)C)=O)CCCN(C(=O)CCc2cnn(C)n2)C(C)C1 N1(C(c2c(C)cc(C)o2)=O)CC(CC(N2CCCC3(CC3)C2)=O)C2(CC2)C1 N(C(=NCCCNC(=O)NC(C)C)NCC1CC1Cl)Cc1ccc(C)cc1 c1(NC(c2cc3ccc(SC(F)(F)F)cc3[nH]2)=O)nc2cc(F)ccc2s1 Cc1nc(O)ccc1C(=O)NC1CC=C(C(=O)NC2(CO)CCCCC2C)C1 C(CC1=CCCCC1)NC(c1cncc(NC(CN(C)C(N)=O)=O)c1)=O C(C(O)C(C)(C)C)NC(CCOCCNC(C1(CC=C)CCOC1)=O)=O c1(N2C(C(=O)NC)CCCCC2)ccc2nnc(C3CC3C)n2n1 S(=O)(=O)(c1cccnc1)NC(C(=O)N(CCC)Cc1ccnc(Br)c1)C N1(C(C2(C(C)C)CC2)=O)CC2(CCN(C(=O)CS(N)(=O)=O)CC2)C1 CC1CN(C(=O)C=CCC(C)(C)NC(=O)Cn2cnc(=N)[nH]2)CC1N(C)C C1(CC)CCN(C(=O)C=CC(C)NC(=O)CC23CCCC2C3)C1 N1(C=O)CCC2CN(C(C3(C4CC4)CC3)=O)CC12.c1(CN)ccc(C(C)(C)C)cn1 c1(OC)cc(CN2CCN(CC(=O)Nc3ccc(OC)c(Br)c3)CC2)cc(Br)c1 CC(CC(F)(F)F)C(=O)N1CCOCC1CCNC(C1(F)CCC1)=O C(=O)(C(CC(N)=O)NC(c1[nH]ccc1C)=O)NC(CC)C C1(C#N)(C(N2CCC(CN(C)CC3CC3)C2)=O)CCCC1 N1(C(c2cc(C)oc2C)=O)CCC(C(=O)NCC(c2cccs2)C)C12CC2 c1(C(=O)NC2CCC(N(C(Cc3ccn(C(C)C)n3)=O)C)C2)cc(F)ccc1N c1(C(=O)NCCOCCCNC(=O)CC2CNC(=O)C2)nnn2c1CCCC2 N1(C(=O)NC(CC)CN2CCOCC2)CC2(CCC(C(=O)NC)OC2)C1 C1(C(N2C(C(C)(C)NC(c3cc(Cl)c(Cl)[nH]3)=O)CCC2)=O)CCOC(=O)CC1 CC(C)(C)C(=O)NCC1(C(C)(C)O)CN(C(C2CC(C(F)(F)F)CO2)=O)C1 c1(C(N(c2ccccc2O)CC)=O)ccc(-c2cccc(OC(F)(F)F)c2)cc1 CC(C)CC(C(=O)N1CCN(C(=O)C(=CC2CCCCC2)F)C(C)C1)N(C)C CCCC(CCC)=CC(N1CCC(OCC(=O)NCC(C)(C)C(=O)NC)C1)=O c1(CC)nnc2c(C(=O)NC(C3CCCCN3C(c3cnns3)=O)C)cccn12 N1(CC(=O)NCC2CN(C(c3cnc(C)o3)=O)C(C)C2)CCCCCCC1=O c1(NC(COC)CCO)cc(NC(C)C(C)C)nc(C)n1 c1(C(=O)NC(C)CCc2nccs2)ccc(O)cc1 N1(C(CCC=C(C)C)=O)CC(C)OC2(CCN(c3cc(CC4CC4)ncn3)C2)C1 c1(CNC(C(C)(C)C2CC2)=O)cnn2c1CN(C(C1C3CC3C3CC13)=O)CC2 C(=O)(C1CCc2scnc21)NCC(CO)NC(c1ccc([N+](=O)[O-])s1)=O c1(NCC2CCC(C(N(C)C)=O)CC2)ccc2ccnc(Cl)c2c1 C1(C(N2CCCC(NC(c3c(C)ccc(=N)[nH]3)=O)C2)=O)Cc2ccccc2CO1 CN1CCN(C(=O)COc2cc(F)cc(Cl)c2)C(CNC(C2CCC3CC23)=O)C1 N1(C(C2(SC)CC2)=O)CC2CCN(C(=O)COCc3nccn3C)C(C2)C1 C(=O)(CC1CC(=O)c2ccccc21)N(CC(CN(C(CCCC(C)=O)=O)C)O)C c1(OC)cncc(CCC(=O)NCC(C)CNC(=O)C(C(C)C)n2cncn2)c1 C1(C(N2CCC3CCC(NC(=O)Cn4cncn4)C32)=O)CNC(=O)CC12CCC2 c1(NC(C2C(OC)CN(C(C(C(CC)C)=O)=O)C2)=O)cnc2[nH]cnc2c1 C1(C(=O)NCC2C3CN(C(c4c(C)ncs4)=O)C2C3)CCOC2(CCC2)C1 N1(C(C2C(C)CCO2)=O)CCC(NC(=O)CC23CCC(CC2)C3)C(O)C1 C(=O)(N=c1[nH]nc(Br)s1)C1C(NC(c2ccc(-c3cc(C)[nH]n3)cc2)=O)CCC1 O=C(C1=NN(c2ccccc2)C(=O)CC1)N1CC=CC1Cc1ccccc1 C(=O)(C=C1SCC(=O)N1C)N(C)CC1N(C(C2C(C)C(=O)C2)=O)CCC1 c1(OCC)cccc(C(N2CCC(C)(C(=O)NCc3cc(Cl)ccn3)C2)=O)n1 c1(OC(C)C(=O)N2CC(C(C)NC(=O)CC(O)C3CC3)C2)ccccc1 C=CCCCCCC(=O)N1CCCC(NC(=O)CC2CCN(CCF)CC2)C1 c1(C(N(C(C)CCO)C2CC2)=O)cc(Oc2ccccc2)n(C)n1 CCC(C(=O)N(CC(C)(C)CNC(=O)CCc1ccon1)C)Nc1nc(C)cs1 c1(C(=O)NC(C2CC(NC(C3(C)CCNC3=O)=O)C2)C)ccc2nccn2n1 C1(C(N2CC(NC(CC3(C)CCCO3)=O)C2)=O)C(F)(F)C12CCC2 CC1(C)CCC(C(=O)NCCCN(CCO)C(c2ccc(C(N)=O)cn2)=O)O1 c1(C(C(=O)NCCc2cn(CCCC3CCOC3)nn2)C2CC2)ccc(Br)cc1 C1(O)(CNC(COC)=O)CCN(C(=O)C=Cc2csc(Br)c2)C1 c1(C(=O)NCC(C)(CO)NC(C2CCC(C)(C)O2)=O)nc[nH]c2nccc1-2 C1(O)(CCNC(c2ncc(C)nc2)=O)CCCN(C(C2CC(F)C2)=O)C1 C1(NC(CC(CC)CC)=O)CCC2(CC1)CN(C(=O)Cc1cnn(C)c1C)C2 N1(C(C(C(C)C)OCC(C)C)=O)CC2CC(O)C1C2NC(c1cc(CO)[nH]n1)=O C1(C=O)CC2CCC(C1)N2C(C1CCC2(CCC2)O1)=O.Cc1ccc(F)cc1CCF C1(C(=O)NCCNC(=O)CC2C=CCCC2)(OC(C)C)CCOC1 c1(OCC)ccccc1C(=O)NC1CCCC(NC(c2c[nH]nc2OC)=O)C1 CCCCC(CNC(C1(OCC)CCOC1)=O)NC(=O)Cc1cccnc1 C(C(C)(C)C#CC(=O)N1CC(=O)N(C)C(C)C1)NC(C=Cc1c(C)nccc1)=O C(=O)(C(C(C)(C)C)NC(=O)Cn1cccnc1=O)NCC1OCCN(C)C1 C1(NC(C2C(C)(C)C2n2cccn2)=O)(CNC(C2CCOC2)=O)CCCCC1 C1(NC(c2cnc(CC(C)(C)C)o2)=O)CCCCC1NC(=O)CC(C)(C)C C1(O)(CC(=O)NC(C)CC(C)NC(C2(C)CC2Br)=O)COC(C)(C)C1 c1(C(=O)NC2(CN(C(=O)CN(S(C)(=O)=O)C)C)CC2)cnn2ccc(Cl)c(F)c12 Cc1cn2ccnc(C(=O)NCC(CC(C)C)NC(C3CCC(C)O3)=O)c2n1 c1(OC(C)C(=O)NC(CNC(=O)CC2CC2)C2CCC2)cccc(Br)c1 CCCC(C(=O)N1CCCC1CSC)NC(=O)CN(C)CC N1(C(C=CC=CC)=O)CCCC(O)(CCNC(=O)C(C)C(C)C)C1 N1(C(Cc2cccc(C)c2)=O)CCOCC(CNC(c2ccc([N+](=O)[O-])[nH]2)=O)C1 CC(C)CC(C)C(=O)NC1CC(NC(c2cnc(-c3ccccc3)cn2)=O)C1 C(=O)(C1SCCc2ccccc21)N1C2CC(NC(c3cncn(C)c3=O)=O)(C2)C1 C(=O)(C(CNC(c1nscc1C)=O)C(C)(C)C)NCCNC(=O)NCC C1(C(=O)NCC(C(=O)N(C2CN(C(C)C)C2)C)CN(C)C)CC2CC(=O)C1O2 N1(C(CC(C)O)=O)C(C(=O)NCCCCC2CCCO2)CCC1C1CC1 C1(C#N)(C(N(CCCCN(C)C(C2CC23CCC3)=O)C)=O)CC1(C)C CCCC(CC(C)C)C(=O)N1CCC2CN(C(=O)CCCC(C)(C)C)CC2C1 CN1CCCC(C(=O)NC(C)(CNC(c2ccnc(OC3CCC3)c2)=O)CO)C1 c1(-c2ccc(SC)s2)ncn(C)c1N(C)CCOCCO C1(C(=O)NCC2(NC(c3cc(OC)n[nH]3)=O)CCCC2)CN2CCC1CC2 N1(C(C2C3C(NC(C4C(C)CCO4)=O)C4C(C3)C42)=O)CC2CCCC1C2CO CCC(C)CC(=O)NCC1CCC(NC(C2CC2CC(C)(C)C)=O)CC1 N1(CC=C)CCC(N2CCC(N(C)C(c3cnn(C4CCCCC4)c3)=O)C2)C1=O C12(C(C)NC(=O)C(N3CCCC(C)(C#N)C3)=O)CC3CC(CC(C3)C1)C2 Cc1sc(=O)n(CC(=O)NC23CCC2CN(C(c2ccc(=O)n(C)n2)=O)C3)c1C N1(C(C(CC)CN(C)C)=O)CCCC(C)(C(=O)NCC2OCCC2C)C1 N1(C(Cn2nc(C)oc2=O)=O)CCCN(C(=O)Cc2scnc2C)C(C)C1 C1(N(C(CCCOCC=C)=O)C)CCCN(C(C2CC2c2ccc(C)s2)=O)C1 c1(C(=O)NC2CC(O)CN(C(C3CCCSC3)=O)C2)cnn2c1C(=O)NCC2 c1(C(C(=O)NCC(CC)N(C(=O)CCC(=O)NC)C)C)c(C)noc1C C1(NC(c2csnn2)=O)CC2CCC(C1)N2C(=O)CN1CSCCSC1 CS(C)(=O)=NC(=O)C(=O)N1CCC(C2(NC(c3cccc4nn[nH]c34)=O)CC2)C1 C1(CNC(=O)CC2CCSCC2)CN(C(C2(Cl)CCC2)=O)CC12CC2 CCC(CC(=O)NCC12CC1CN(C(c1cnc(S)nc1)=O)C2)C(F)F c12ccc(c(Cl)c1)OCC(=O)N2.C1(C(=O)OC)(CN)CC1S(C)(=O)=O c1(C(=O)NC2CCC3CCN(C(CCCCOC)=O)C32)cncc(P(C)(C)=O)c1 CC1OC2CCC1(NCC=CC1=CN(C(=O)OC(C)(C)C)CC1)C2 C1(COC(=O)CN2CCCCC2)CCCOCC1 N1(C(C(CC)=CCCC)=O)CCCC(N(C(=O)Cc2ccccc2)C)C1 c1(C(=O)OC)ccc(CC(=O)NC2(C)CCN(C(=O)C=C(C)C)C2)cn1 c1(OC)nc(C)ccc1C(=O)NCC1(NC(=O)CC2(C)CC2F)CCC1 N1(C(C2(C)C(C)C2)=O)C(C(=O)NC(c2ccccn2)CO)CC2CC12 C1(CNC(c2c[nH]c(=NC)o2)=O)CCCCN(C(C2CNC(=O)CC2C)=O)C1 c1(CNC(C2(CC(=O)OC)CC2)=O)nocc1C(=O)NC1CC(N(C)C)C1 C(C)(C)(C(N)C(=O)NNc1cc(Cl)ccc1Cl)OC c1(OC)ccc(C(=O)NC2(c3ccc(Cl)cc3F)CCC2)c(Cl)c1Cl c1(CCN(C(C2CCC(C)(C)C2)C(=O)NCCCSC)C)nc2ccccc2[nH]1 c1nc2c(N3CCN4CCCC4C3)[nH]c(=NCC3(OCCO)CCC3)nc2s1 C(CN=c1nc2sccc2c(N2CCC(C3CCCC3)C2)[nH]1)N1CCC(C)CC1 C1(C(=O)NCCC(CC)(C)NC(=O)Cc2cnoc2)CC2CCC1CC2 C(=O)(C(C)(C)CC#N)N(C)CC1CCN(C(C(C)Sc2ccc(C)cc2)=O)CC1 Cc1[nH]nc(Cl)c1C(N1CCC(CN(C(=O)C=CSCc2ccco2)C)CC1)=O C1(C(N2CC(NC(c3n(CC)ncc3Cl)=O)C(C)C2)=O)CC12CCOC(C)C2 N1(OC)CC(CO)CCC1C(F)(F)F.c12cccc(c1)S2 C1(C(N2CC(NC(C(CSC)C)=O)C2)=O)Cc2c[nH]cc2S1(=O)=O c1(C(N2CC(C)N(C(c3cccc(C#N)n3)=O)CC2)=O)n[nH]c2c1CCCCC2 C1(CNC(C2(C#C)CN(C(C3CCCOC3)=O)C2)=O)CCC2(CC2)CO1 C(CC(C)C)(C(=O)NC1CCN(C(c2cccc(N(C)C)n2)=O)C1(C)C)OC C12(NC(CC(CCC)O)=O)CCCC1N(C(c1cccc3[nH]ccc13)=O)CC2 Cc1cc(CC(=O)NC(CNC(c2cncn2-c2ccccc2)=O)CO)n[nH]1 N1(C(C2(COC)CCC2)=O)CCC(CO)(CNC(C2CC(S(C)(=O)=O)C2)=O)CC1 N1(C(C2CN(C(C)=O)C2)=O)CCC(C)(CNC(=O)CCCC2CCC2)C1 C(=O)(C1=CCC2CCC1N2C(C1COC(=O)N1C)=O)N1CC(C)N(C)CC1 CCC1=NOC(C(=O)NC2(C(F)F)CC(NC(=O)C(C3CC3)NC(C)=O)C2)C1 N1(C(=O)OC)CCC(C(C)NC(N2CCC3CC23c2ccccc2)=O)CC1 C1(C(=O)NC(c2nc(C)on2)C)CCN(C(=O)c2cncc(C#N)c2)O1 C1(C2CC2)(C(N2CC(c3c(C)nn[nH]3)C2)=O)CN(C(C2COCCN2C=O)=O)C1 N1(C(CN2C(=O)CCC2=O)=O)CC2CCC2(C(N2CCC(Cl)C2)=O)C1 N1(C(CCSCC)=O)CC2CCN(C(=O)COCc3cccc(C)c3)CC12 n1(CC)nccc1C(C)OC(=O)C(F)(F)OC(F)(F)F Cn1ccc(C=CC(=O)NCC2CCCCN2C(c2cnn(CCO)c2)=O)c1 C1(=CC(N2CCC(NC(Cc3cnc(C)o3)=O)C(C)C2)=O)CC2CCC(C1)N2C C(=O)(CS(=O)CCC(F)(F)F)N1C(C)(CNC(C=Cc2ncn(C)c2)=O)CCC1 C1(C(=O)NCC2CCN(C(c3n(CC#C)ccc3)=O)C2)CCC2(CCCC2)CC1 Cc1nc(C(N2CCCOC(CNC(c3ccn(C(C)C)n3)=O)C2)=O)cc(O)n1 C1(CC(=O)N(CC(CNC(C(C)OCC)=O)(C)C)C)CC(=O)NC1=O c1(C(=O)NCC2CN(C(=O)CCCc3nc(C4CC4)no3)C2)cc2oc(Cl)cc2[nH]1 C1(C(N2CC(C)(OCC)C2)=O)CC=CC(NC(c2ccnc(OC)c2)=O)C1 CC1CNc2c(C(=O)NCC3CC(NC(=O)C(C)n4cccn4)C3)cccc2C1 C1(NC(=O)C=CCN2CCCC2)CN(C(=O)Cc2cnc(Cl)s2)CC12CC2 C(=O)(C(O)CCCNC(=O)CC1CCCC(=O)C1)NC(C)C(=O)NC1CC1 c1(C(N2C(CNC(=O)C(=O)Nc3ncc[nH]3)CCC2)=O)cccc(Cl)c1C(F)F C1(NC(c2cc(C)[nH]n2)=O)COCCN(C(C2(c3cccs3)CCOCC2)=O)C1 C(CCC(C)(F)F)NC(C(N1CCC(n2cc(NS(C)(=O)=O)nn2)C1)=O)=O CC12CCN(C1)C2=O.c1(NC(=O)COc2cccnc2)cccc(C(F)(F)F)c1 C(=O)(CCCN(C)N=O)NC1CN(C(c2cc(OCC)n[nH]2)=O)CC1(C)C N1(C(C=CCN(C)CC)=O)CCC(NC(c2ncn(C)n2)=O)C(CO)C1 C=CCC(C(=O)N1CC(C)(CC)C1)NC(c1c[nH]c(C)c1)=O C(=O)(C(C)(F)C(C)(C)F)NCC(CNC(CN(C1CCSC1)C)=O)O N1(C(=O)OCC)CSCC1C(=O)NC(C1CCN(C(=O)C=C(C)C)C1)C C1(N(C(CSCCCC)=O)C)CCC2CN(C(C34CC(CC(F)F)(C3)C4)=O)CC12 C1(C(N(CCC(N)=O)CC)=O)CCN(C(=O)C(c2cncnc2)C)C(C)(C)C1 C(C)(CO)(C(=O)NCCC1(O)CCN(C(C2(CC(C)C)CC2)=O)C1)OC N1(C(c2c(C)c[nH]n2)=O)CCC(C)(CCNC(c2cscc2C#N)=O)C1 C(=O)(NN1CCc2ccc(F)cc21)C1(C(=O)NC)CC1 C12(C(=O)NCCCN(CCCNC(C(C)=CC)=O)C)CCC(CC1=O)C2(C)C C1(NC(CCCN(C(=O)C#CC2CCCC2)C)=O)CCn2ncnc2C1 C(=O)(C1COc2c(C)cccc21)NCC(CN(C(C=CC(CC)=CC)=O)C)O N1(CC(N2CCC(N(C)Cc3ccc(OC)cc3)C2)=O)CC(C)OC(C)C1 CCC(CC)C(C)C(=O)N1CCCC(CC(N2CCC(O)(CC(C)C)C2)=O)CC1 c1(C(=O)NC(C=C)C)cc2n(n1)CCCN(Cc1c(Br)cnn1C)C2 C1(CC(=O)NCCCN(C(c2cn(CCN(C)C)nn2)=O)CC)CCCC(C)C1 N12CCC(C13CC3)C2=O.C(C)(C(C1CC1)C1CC1)NC(C1CC(N(C)CC)C1)=O Cn1cc(C(N2CC(NC(=O)COc3cnn(C)c3)C(O)C2)=O)c(O)n1 N1(C(C(C2CC2)OC)=O)CC(CNC(c2ccncc2Cl)=O)CC12CCOCC2 N1(C(C(C=C)OC)=O)CCN(C(=O)C(O)COC)C(C)C1 CCC(=O)CCC(=O)N1CCC(C(C)N(C(=O)CC2(COC)CC2)C2CC2)CC1 C1(C(=O)NC(C(=O)NCC)(C)C)CN(C(C2CCSC2)=O)CC1C(C)C N1CCCC(CC(=O)N)CC1.C1(CSCCNC(=O)OC(C)(C)C)CCCO1 C(=O)(CCCC(=O)NCCC(C)(C)CNC(=O)CC1(C)CC1F)NCC c1(C(=O)NCCN(C(=O)C(O)CC2CCCCC2)C)c(F)cccc1Br Cc1cc2[nH]c(C(=O)NC3CC3CNC(c3cc(F)cc(Br)c3)=O)cc2o1 N1(C(COCCC#C)=O)CCCC1C(C)(C)CNC(c1cncn1C)=O CC(CCC(=O)NCC1(C2(NC(=O)CCCn3ccnn3)CC2)CC1)N(C)C C(=O)(CCS(=O)(=O)NC)N1CCC(N(CCC)C(C2CC2CF)=O)CC1 c1(CCNC(C(CC2CN(C(CCCOC)=O)C2)F)=O)cc(C)c(C)cc1F C(=O)(C(CCC1CC1)NC(c1cc(Cl)n(C)n1)=O)NC(c1cn(C)nc1)CO C(=O)(CCC(C(C)C)NC(c1nn(C)cc1Cl)=O)NCCC(C)N(CCC)C C1(C(N2C(C)CC(NC(c3cc(C4CC4)no3)=O)CC2)=O)CC12CCC(=O)CC2 c1(C(=O)NCCC2N(C(Cc3nc(C)sc3)=O)CCCC2)c(C)nn(C)c1F C(=O)(CC(C)C(=O)NCC1(F)CC(NC(c2[nH]nnc2C2CC2)=O)C1)OCC C12(CCNC(CNC(CC)=O)=O)CCC(CC1)N(C(c1n[nH]c(C(C)C)n1)=O)C2 N1(C(C(C)c2ccco2)=O)CCC(CCC(=O)N(C)Cc2ccnn2C)C1 c1(C(=O)NC2CN(C(c3cn(C)[nH]c3=N)=O)CC2O)ccc2cc(F)ccc2n1 c1(C(C(N2CCC(CNC(CCCOC(C)=O)=O)C2)=O)(F)F)cnc(Cl)c(C)c1 C1(C(=O)OCC)(C(=O)NCC(C)CNC(=O)CSc2cccs2)CCC1 C1(C(=O)NCC2(C)CNC(=O)O2)CN(C(c2cc[nH]c2)=O)CC1C1CC1 CCCC(C)(C)CC(=O)NC(c1c(C)[nH]c(C2CCC2)nc1=O)=O N1(C(CSCC=C)=O)CCCC1(C(=O)NCC1C2CCCOC12)C(C)C C1(CC=C)(NC(=O)CC2CC=CCC2)CCN(C(c2ccc(C)cn2)=O)C1 C1(NC(c2oc(CC)c(C)c2)=O)CC2CC1N(C(C1(CSC)CCC1)=O)C2 c1(C(=O)NCC#CCNC(c2c(C)nc(C(F)(F)F)s2)=O)ccc2c[nH]nc2c1 Cn1ccc2cc(C(=O)NC3CC3NC(=O)CCc3ccc(F)cc3)cnc12 N1(C(C2(CC)CCCO2)=O)CCC(F)(CNC(c2cc3scnc3[nH]2)=O)CC1 N1(C(c2c(C)c(F)cnc2)=O)CC(C)(C)CCC1CNC(=O)CCC(C)(C)F C1(CCNC(C(C)c2ccsc2)=O)COCCN1C(=O)CCc1ccccc1Cl c1(C(N(C(C(N2CCN(CC)CC2C)=O)CC(F)F)C)=O)ccc2cc[nH]c2c1 CC(=O)CCCC(=O)N1CCC(CNC(c2ccc(C3CC3)cc2C)=O)CC1C N1(C(c2c(C)nc(C3CC3)o2)=O)CC2CC(N(C)C(c3cnn(C)n3)=O)C1C2 Cc1ccc(F)cc1C(=O)NC1CC1CNC(C1CC(n2cnnc2)C1)=O CC(C)C(CCN(C(=O)CC1CSCCS1)C)NC(c1ccc(O)cn1)=O c1(C(=O)NC2C(C)(C)C(CNC(C3CC4(CSC4)C3)=O)C2)ccc2ncnn2c1 C=CC(CC)CC(=O)NCC1CN(C(c2cc(CC)ncn2)=O)CCO1 c1(CC)cc(C(N2CC3CC(NC(=O)C(O)CCN(C)C)C2C3)=O)cc(F)c1 N1(C(C(C=C)(C)O)=O)CCCCC(CNC(=O)CCc2ccc(OCC)cc2)C1 n1(CCC)cncc1CNC(C1CCOC1CNC(=O)CSc1cn[nH]c1)=O CC(O)(Cc1ccccc1)C(=O)NCCNC(c1coc(Br)n1)=O c1(OC(F)F)cccc(Cl)c1CNC(=NCCC1CC1)NCC1CCOC(C)(C)C1 C1(CC)C(NC(=O)CSc2ccncc2)CCCN1C(c1ccnnc1O)=O C(=O)(CCCN=[N+]=[N-])N1CC(NC(CNc2c(NC(C)=O)cccc2)=O)C(C)C1 C1(N(C(c2n(CC)ncn2)=O)C)CN(C(c2cc(C(C)(F)F)n[nH]2)=O)CC1O NC1(C(=O)NCCC2CCNCC2(F)F)CC2(CCOCC2)C1 C1(COC(C(CC)Oc2ccccc2C(C)C)=O)COC2CCCC2O1 c1(C(=O)NC23CC(CNC(c4ncc(C)cc4F)=O)(C2)C3)cc2ccncc2[nH]1 [N-]=[N+]=NC1CN(C(=O)CN2CCCCCC2)CC1NC(=O)C(O)CC1CC1 C(CC(C)C(=O)NC1CC(F)(CNC(c2ccc(N(C)C)nn2)=O)C1)OC c1(N2CCC(O)CC(C)C2)nc(=NCCCCCF)[nH]c2c1CCC2 N1(C(CCCCCC)=O)CC2CCC1C(CNC(=O)CCCC#N)C2 c1(C(N2CCN(C(c3nncc(OC)c3)=O)CC2)=O)cnc(C)cc1C CN1CCN(c2nccc(C(F)F)c2Br)CC1CS N1(C(CCSC)=O)CC2(C1)CN(C(=O)C(CCN(c1ccccc1)C)N(C)C)C2 CC(C)CC(CNC(=O)C1=CCCCC1C)C(=O)N1CC(n2ccnc2)C1 C#Cc1ccc(Cl)c(C(N2CC3CC3(CNC(C3(C)CCC(O)CC3)=O)C2)=O)c1 C1(CNC(C(C)(C)Cc2ccsc2)=O)CCCCN(C(=O)C(C)(O)C(C)(C)C)CC1 Cc1cccc(C)c1C(c1nnnn1CCCF)NCCCc1nnnn1C CCC(CNC(=O)C(=O)NCC1CSCCO1)C(=O)O C(CNC(C1CCOC(C)(C)C1)=O)(CC(F)(F)F)NC(c1c(CC)onc1C)=O N1(C(c2ccc(CC)[nH]2)=O)CC2(CCC(NC(=O)C(c3cnn(C)c3)O)CC2)C1 N1(C(C(Cc2ncn(C)c2)O)=O)CCCC(F)(CNC(c2cccc(=O)o2)=O)C1 CCC(CCCC(=O)NCCC(C)(C)CO)NC(C1CCS1(=O)=O)=O C1(C(=O)NCC2CCCN(C(=O)CCCCC3CC3)C2)CC12CCSCC2 Cc1cccc(CNc2ncc(-c3cnn(C4CCOC4)c3)s2)c1 Cc1cccnc1CCCOC(c1ccc(CSc2cccnc2)s1)=O C1(CNC(C(C)N(C)C)=O)CCCC1NC(=O)C(C)(C)C1CCCC1 N1(C(CC(=C=C)C)=O)CCCCC(CNC(c2conc2COC)=O)C1 N1(CC(N2C(C)CC(CNC(COC)=O)C2)=O)CCCc2sccc2C1=O C1(CNC(C2C(C)C2C)=O)CC2COCC2N1C(c1cn(C2COC2)nn1)=O Cc1cc(C)n(CCNC(c2cnn(CCNC(C3COC(=O)N3)=O)c2)=O)n1 C#CCCC(C(=O)NC(Cc1ccco1)CO)NC(C1CCCC(CF)C1)=O C1(NC(=O)CCc2cc[nH]n2)CCN(c2ncnc3scnc23)CC12CCC2 c1(C(=O)NC2(CC=CC(=O)NCCc3ncn(CC)c3)CCC2)nnn(C)c1N c1(OCC)ccc(CCC(=O)NCCCC(C)NC(c2sc(C)nc2C)=O)cc1 C1(NC(=O)CCn2cnnn2)CCOC2(CCC2)C1.C12CCC1C(=O)NOC2 C#CCC(CC#C)n1cc(-c2ccnn2C2CCCC2)nn1 C1(CCC)(NC(C2CC3C=CC2C3)=O)CCCN(C(=O)C=Cc2ccco2)C1 c1(C(N2CCN(C(C(F)OC)=O)C(C)C2)=O)ccc(S(=O)(=O)NC(C)(C)C)cc1 C(C(C)(C)CC(=O)N1CC2(CCC2CNC(=O)CCC2CCCOC2)C1)OC C1(O)(CNC(C(CC)NC(=O)CC2CC(C)C2)=O)CCCOC1 n1(CC)ncc(CNC(=O)C(Cn2ccnn2)NC(=O)CC2(O)CCCC2)c1C N1(C(c2cncc(C(C)(C)C)c2)=O)CC2(CCCN(C(C3CCSC3)=O)C2)C1 c1(C(=O)NCC2(NC(C(=Cc3ccco3)C)=O)CCC2)ccc2c(c1)CCCO2 CCC(Cc1ccc(Cc2ccccc2)cc1)C(=O)NC1=NCCO1 CC1CCCN(C(C2CN(C3CCOC3)C2)=O)C1CNC(C1CCCCCC1)=O N1(C(C2(CC#C)CCCC2)=O)CCC2CCN(C(c3ncc(N)cc3C)=O)C2C1 c1(CNC2(CO)CN(C(C3CC(CC)(CC)C3)=O)C2)ncc(C(C)=O)cn1 N1(C(C2C(C)(CC)C2)=O)C2CCC1CN(C(c1cc(C3CCC3)on1)=O)C2 c1(-c2nnn(CC(=O)NCCNC(c3c(CCC)n[nH]c3)=O)n2)ccc(F)cc1 c1(C(N2C(C#C)CCC2)C(=O)NCCC2(C)CC2)ccc(S(N)(=O)=O)o1 c1(C(=O)OC)ncncc1NC(=O)OC1CN(C(=O)CCOC)C1 N1(C(=O)CC2CCCC2)CCCN(C(C2COCC2n2cc(Br)cn2)=O)CC1 CCC(C)(CC)C(=O)NCC(O)CNC(c1cc(C(F)F)ccc1OC)=O N1(C(CN(C)C(N)=O)=O)CCC2CCCC12CNC(=O)CC1=CCOCC1 c1(C(=O)NC(C(C)NC(CC(=O)OC)=O)C)c(C)c2ccc(F)cc2oc1=O Cc1ccc(NCC(N2CC(c3ccccc3)(NC(=O)C(C)(Cl)Cl)C2)=O)cc1 c1(C(N2CCCC(C=C)C2)C(=O)NCCC2CC2)ccc2c(c1)COC2 c1(OC)ccncc1C(N1CCOC(C(C)NC(=O)CC2(OC)CCC2)C1)=O c1(OC)cc(CC(=O)NCC(C)NC(=O)C(CC#N)c2ccccn2)cc(Cl)c1 C(=O)(CCCC1CCC1)NCC(C1CCCN1C(=O)COC1CCOC1)(C)C C1(CCC)CCC(O)(C(=O)NCC2(F)CCCN(C(C3(C)CCC3)=O)C2)CC1 C(C)(C(C(=O)NCc1sccc1C)C(C)C)NC(c1cc(C)nnc1)=O C1(O)(CC(=O)NC2CC(CNC(C3C(C(C)O)C3)=O)C2)CCOCC1 CC1(C)C2CCC1(C)C2C(=O)NCC1CC(NC(C2CCC(C)(F)CC2)=O)C1 CCC(CC)CC(=O)NCCC1(O)CCN(C(=O)CCN2CCCC2=O)CC1 Cn1cc(C(N2CC3C(NC(C4CC45CCCC5)=O)C3C2)=O)c(C(F)F)n1 c1(CC)nc(NC(CNC(=O)CC2(N3CCCC3)CC2)C(C)C)cc(C#N)n1.OCC c1(NC)nc(C)ccc1C(=O)NCCCOCCN(C(=O)CC(C)CF)C N1(C(CC2(NC(C)=O)CC2)=O)CC2CCN(C(=O)C(n3ccnc3C)C)C2C1 c1(C(=O)NCC(C)NC(C2CCN(S(C)(=O)=O)CC2)=O)c[nH]c2c(F)cccc12 CCC(C)C(O)C(C)C(=O)NCCN(C(=O)CC1CCC(C)CO1)CCOCC c1(OCCOC)ccc(C(=O)NC(C)CNC(C2CS(=O)(=O)C2)=O)cc1 C(=O)(CS(=O)C(F)(F)F)NCC1(OC)CCN(C(C2(F)CC2C)=O)CC1 C(C(C)(C)C(=O)N1CC(CCc2cn(-c3ccccc3)nn2)C1)OC C1(C(=O)Nc2c(C(C)C)ncnc2)CN(C(C2CCC(C(N)=O)C2)=O)C2(CCC2)C1 c1(C(=O)NCCOCCNC(C2C(C)C2)=O)c(Cl)cc(Cl)c2ncccc12 N1(CCNC(C2(F)CCC2)=O)CCCN(C(=O)Cc2ccccn2)CC1 C(=O)(C1=CC2C=CC1C2)NC(CCOC)C(=O)N1CCCC(N2CCC2)C1 c1(SC)cccc(C(=O)NC2CCN(C(C3CCCO3)=O)C2)c1 Cc1cc(C)c(C(=O)NCCC(C)N(C(=O)CC2CCCOCC2)C)[nH]1 c1(NC(COCCOCC#C)=O)cccc(Cc2ccc(C)cc2)c1 CN1CCN(C(C2CCOC(=O)CC2)=O)C(CNC(=O)CCNC(N)=O)C1 N1(C(C(C(C)O)C)=O)CCCCC12CC(NC(c1cc3ccccc3o1)=O)C2 c1(C(CNC(C=CC=CCC)=O)NC(=O)CCc2cnoc2)cc(F)cc(Cl)c1 CCCCC(CC)C(=O)N1CCC(N(C(=O)Cn2ccnn2)CCC)CC1 c1(CNC(c2nnnn2C2CCOCC2)CCSC)nn(C)c(Cl)c1Br c1(CN(C)C(C2CCN(C(=O)C(COC(C)(C)C)N(C)C)C2)=O)ccc(F)cc1 N1(CC(=O)N(CCNC(CCOCC)=O)C(C)C)CCc2ccccc21 c1(CC(=O)NCCOC2CCN(C(C(CC)=CC)=O)C2)ccc2[nH]ccc2c1 CCC(C)(COC)C(=O)N1CCC(C(F)F)(CNC(c2cnc(S)[nH]2)=O)C1 C1(C(=O)NC2CC(OC)C2)(C(=O)NC(C)CC2(O)CCCC2)CCCC1 C(=O)(C1=CC2(CCN(C(C3CC3(C)C(F)F)=O)C2)C1)NC(C1CSC1)C C1(O)(C(C)CNCCC(=O)Nc2cc[nH]c2)CCN(C(=O)OC(C)(C)C)C1 CCCC(CNC(=O)CCc1ccncn1)C(=O)NC1(C)CC=CC1 c1(C(=O)OC(c2ncccc2C)C(=O)OCC)nccc2c1CNC2=O C1(NC(c2cc(C)oc2C)=O)CC(C)CN(C(c2cnnn2C2CC2)=O)C1 C1(C#N)(c2n(-c3c(C)cccc3C)nc(C(F)F)n2)CC12CCCC2 CCCCC(C(=O)NC1COCCC1NC(=O)C(CC)CC)ON=C(C)C CC(CC(F)(F)F)C(=O)NC1(CO)CCN(C(c2n[nH]c3c2CCSC3)=O)C1 c1(C(=O)NCCCC2N(C(CSCC(N)=O)=O)CCCC2)onc2ccccc12 N#Cc1cc(Cl)c(C(N2CC(F)(CNC(=O)CCN3CCC(O)CC3)C2)=O)s1 C(=O)(C1CC(=O)c2c(F)cccc21)N1C2CN(C(CC3C(C)C3)=O)C(CC2)C1 C1(CC)CCC(C(N2CC(OC)CC2CNC(=O)C(C)CF)=O)CC1 c1(N2CCCC(C)(CC)C2)nc(N2CCCN(C)CCC2)nc2c1COCC2 c1(-c2cn(CCCC)nn2)c(NC(C2CCN(C(C)=O)C2)=O)cnn1C c1(N(CC2=CCSC2)C)nc(N2CCC(C3CCCCC3)C2)c2c(n1)CCS2 c1(C(N2C(CO)CC(NC(CS(C)(=O)=O)=O)C2)=O)cc2cc(F)ccc2[nH]1 C1(C(C)C)(C(N2CCC(CCCO)C2)=O)CCCN1C(=O)CC(C)N(C)C Cc1cccn2c(C(=O)NC(C)CC(C)NC(c3cc[nH]c3)=O)cnc12 N1(C(C(C)C2CCCC2)=O)CCC(C2CC2)C1CNC(c1ccc(=O)oc1)=O Cc1cc(C(=O)NC(C)(C)COC(C)(C)C)sc1-c1ccccc1Cl N(C(=NCCCCC(F)(F)F)NCC1CSCCO1)C(c1nnc(C)s1)C C(O)(CC(=O)N1C(CO)CCC1CO)(C(F)(F)F)c1nc(C)c(C)o1 Fc1ccc2cnc(NC3CN(Cc4cc(Br)cs4)CC3(F)F)nc2c1 c1(C(N)=O)ccc2c(c1)CCC1C2OCCN1Cc1cccc(F)n1 C(=O)(C1=C(C)N(C)c2nnnn2C1)NC(CCNC(COCCC=C)=O)(C)C C1(CNC(c2ccnc(C)n2)=O)CCN(C(=O)Cc2cnc[nH]2)CC1(F)F C(C(=O)NC1CCC(CC(N2CCC(C(N)=O)CC2)=O)CC1)(C(C)C)OCC N1(C(CCC#CC)=O)CCCC(C2CCN(C(=O)C(F)(F)CC)CC2)CC1 C1(c2n(C)cnn2)CCCCC1C(=O)NC(C)CNC(=O)COc1ccon1 C1(C(=O)NCCCSCC)CCN(C(=O)C=CCNC)C12CC2 C(=O)(C1CCc2scnc21)NC(c1ccccc1F)CNC(C)=O C1(C(=O)Nc2ccc(CCO)cc2)(NC(C(C=CC)O)=O)CCCCC1 C1(C(=O)NC)CCN(C(=O)CN(C(C2CC3(CC3)C2)=O)C(C)C)C1C c1(C(=O)NCCCC(C)NC(C2C=CCC2)=O)ccc2c(c1)nc(O)n2C1CC1 C12(NC(c3c(Cl)cn(CC)n3)=O)CCN(C(c3ccc(N)c(F)c3)=O)CC1C2 C1(C(=O)OC)CC2CCC1N2C(=O)CCC(=O)NCCN1CCCC(C)C1 O=C(C1CCCc2nc[nH]c21)NC1CC(NC(=O)C2=NOC3(CCOC3)C2)C1 C1(CNC(CC2CCN(C(C(C3CCOCC3)OC)=O)C2)=O)CC(C(N)=O)=NO1 N1(C(CCOC(C)C)=O)CC2CCC(C1)N2C1CCN(C(C2CCC2C)=O)CC1 c1(C(=O)NCCCN(C(C=C2CCN(C)CC2)=O)C2CC2)csc2cccnc12 C1(CC)CN(C(C2CC(NC(C3CCC(=O)N3C3CC3)=O)C(O)C2)=O)CCO1 C1(C)(C(=O)NC2CCC(NC(c3ccc(CCC)[nH]3)=O)CC2)CCN(C)C1=O CCC(C)CC(=O)C(=O)NC1CC(NC(=O)Cc2cn(C)cn2)C12CCC2 N1(C(C2(Oc3cccc(OC)c3)CC2)=O)CCC2CCN(C(C3CCC3)=O)C2C1 N1(C(C(C(COC)C)C)=O)CCC(C2(O)CN(C(=O)CCCCSC)C2)CC1 c1(SCc2cn(CC(=O)NC(c3cncs3)C)nn2)ccccc1OC C1(OCCNC(C=C(C)Cl)=O)CCN(C(C2CCCN2C(=O)C(C)(C)C)=O)CC1 N1(C(CC)=O)C(CNC2(c3nnnn3CC(F)F)CCCC2OC)CC2CC12 C=CCCCCCC(=O)NCC1C(O)C(O)CN1C(c1cc(CC)on1)=O c1(NC(C(C2(O)CN(C(C(CC)OCC)=O)C2)F)=O)cccc(CCO)c1 c1(CNC(c2ccc(C(C)=O)[nH]2)=O)ccc(Cl)cc1F C1(NC(CCc2cc(C)on2)=O)C2CC3CN(C(c4[nH]ncc4C#N)=O)C1C3C2 Cc1cn2c(n1)C(C(=O)N1CC(CNC(C3CC(F)(F)C3)=O)C3(CC3)C1)CCC2 c1(CNC(N(C2CCN(Cc3ccccc3)CC2)C)=O)cn2c(n1)CCCC2 C12CCN(CC1)C(=O)SCCOC2C(=O)OCC.C(C(C)C)OC(C)(C)C N1(C(C=C(CCC)C)=O)Cc2nccn2CC(NC(c2ccccc2OC)=O)C1 c1(OC)nccc(I)c1C(N1CC(CC(N2CC(O)C(F)C2)=O)(OC)C1)=O O=C1CCC(C(=O)NC(C(N2CCCC2CCCO)=O)C2CCC2)C1 Cc1cc(C)nc(SCC(N2CC(NC(=O)Cc3nc(C(C)C)c(C)s3)C2)=O)n1 c1(C(=O)NCC(C)(C)NC(c2ccc(CO)cn2)=O)cncc(N)c1 N1(C(c2ccc(OC)o2)=O)CCC(C(N2CCC(C)(N(C)C)C2)=O)(C(C)C)C1 N1(C(c2c(OC)cccc2)=O)CCCCC(NC(=O)C)C1.C(CC(C)C)OC(C)=O c1(C(=O)NCC2CCN(C(C3CCC(=O)NC3)=O)CC2)ccc(F)cc1F CCC(C)C(=O)C(=O)N1CCC(C(=O)N(CC(C)CO)C)C1C(C)C C1(C(C)C(=O)N2CCC2C(=O)N(C)C)CCN(C(=O)C=Cc2ccco2)C1 Cc1cnn(Cc2cc(C(=O)NC(C)C(C)NC(=O)Cc3ccccc3)no2)c1 c1(SC)ccnc(C(=O)NCC2(CCNC(=O)C(C)N(C)C)CC2)n1 C1(C(=O)NC(C#C)C2CCC2)(CNC(C2CNC(=O)C2)=O)CC=CC1 c1(C(=O)NCC(CNC(C2CCN(C)C2=O)=O)O)cc2c([nH]1)CCCC2=O C(C)(CS(=O)(=O)CC)NC1(CCNC(c2ccccc2)=O)CCC1 C=CCC(CNC(c1cc(CO)n(C)n1)=O)C(=O)N1CC(CO)C1(C)C Cc1cccc(Br)c1C(C(=O)NC1CCNC(=O)C1)NC(C1CC1CC(C)C)=O c1(CN2CC(F)CC(C(=O)Nc3ncc(Br)cc3Cl)C2)ncc2ccccn12 c1(C)c(C)cccc1C.C1(c2ccccc2)(N2CC2)CCCC1c1c(CCCCCC)ccs1 C1(COC(C2C(C#N)CC2)=O)CCOC2(CCCC2)C1 N1(C(C(CC)NC)=O)CCC(C(=O)Nc2ccc(Cl)nc2C(F)(F)F)C(O)C1 C1(C(=O)NC2CCN(Cc3cc(C(=O)OC)[nH]c3)CC2F)Cc2ccccc2O1 CC#CCCCC(=O)N1CC(F)(F)CC1C(=O)NC1(CC)CC1 CC1CNc2c(C(=O)N(C3CCN(C(=O)C(C)C(C)(C)C)CC3)C)cnn2C1 CC1(CNC(c2sccc2C(F)F)=O)CC(F)(F)CN1C(=O)CCF CC1(N)C=C(C(=O)N(CCCNC(C2CCCC3(CC3)C2)=O)C2CC2)C=C1F C12(C(N3CCC(=CCNC(C=C4CCN(C)CC4)=O)CC3)=O)CC(C)(CCO1)C2 N1(C(C)=O)CCC2(CCCC2NC(=O)CSc2ccccc2C)C1 N1(C(CN2CCC(C)CC2)=O)CCC(C)N(C(=O)Cc2nn(C)cc2Cl)CC1 CCC(COC)C(=O)NC12CC1CN(C(C1CCN(CC3CC3)CC1)=O)C2 c1(C(=O)NC(C(COC)C)C)nc2ccccc2n1-c1ccccc1 N(C(=NCC1CCN(C)C1=O)NC(C)C)CC1(CCC)CCC1 C1(NC(=O)CNC(c2ccccc2Br)=O)CC2CN(C(=O)C=C3CC3)CC2C1 C1(NC(c2cc(C)oc2C)=O)C(CN=c2nc(C(C)(C)C)[nH]s2)CCC12CCC2 C(CCC(=O)NC1(CCNC(=O)Cn2cnnn2)CCC1)OC N1(C(c2cccc(CC)n2)=O)CC2CCC(C(N3CC4CSCC4C3)=O)(C2)C1 Cn1nc2c(c1C(N1CC3CN(C(=O)COC(C)(C)C)CC3C1)=O)CCC2 N1(C(c2cc(C)cc(C)c2)=O)CCC2CN(C(c3ncncc3F)=O)CCC12 CC(C)CC(C)(C)C(=O)NCC1CC(F)(CNC(c2cc(Cl)ccc2N)=O)C1 C1(NC(CCC(=C)Cl)=O)CC2CCC(C1C)N2C(c1cc(N)ccn1)=O S(=O)(=O)(c1ccc2c(ccn2C)c1)N1CC(C(C)OC)C1 c1(OC)cc(C(=O)NCCC(C)NC(C2CC2(Cl)Cl)=O)cnc1Br N1(C(C2CC(CC)(CC)C2)=O)CCC(F)(C(=O)N(C(C)C)Cc2ccncc2)C1 CCCC(C(=O)NCCC1(O)CN(C(=O)C=C(C)C)C1)S(N)(=O)=O C(=O)(CC1=CCCCC1)N(C1CCCN(C(c2nccc(Cl)c2F)=O)C1)C N1(C(c2ncc(C)nc2)=O)CCN(C(C2(C(C)C)CCCO2)=O)CC12CCC2 Cc1cn2cc(C(=O)NC3CC(C)(C)SC(C)(C)C3)nc2c(C)n1 C1(C(N(c2cnc(SC)s2)CC)=O)CC(=O)N(c2ccc(-c3nn[nH]n3)cc2)C1 c1(C2C(C(N3CC(N(C(=O)CC4C=CCC4)C)C3)=O)CCO2)cncc(Br)c1 c1(C(N2CCC(C)N(C(C3CC3(F)F)=O)CC2)=O)cc2nccn2c(O)n1 C(C(CC)(CC)C(=O)NCC1CNC(=O)C1)NC(CCC)=O CCC(O)(CC(=O)NCC1CCCC1NC(C1(C)CC1Br)=O)c1ccccc1 C(=O)(C(=O)C(C)(C)C)NCC(CNC(C(CC1(C)CC1)O)=O)CO N1(C(C(C)OCOC)=O)CCCN(C(=O)Cc2csc(Br)c2)CC1C C1(CNC(CC(=C)C)=O)CC2(CO1)CN(C(C1CCCC(C)(C)CC1)=O)C2 C(=O)(C1=CCCCO1)NC(C(=O)Nc1c(C(=O)OC)nsc1)(C)C1CCC1 Cc1cnc(C(=O)NCC2CC(C(=O)NC3(C(F)(F)F)CC3)C2)c(F)c1 c1(C(=O)NC23CC2CN(C(=O)CC(F)(F)F)C3)cccc2c1OCO2 c1(C(=O)NC2CCC(CNC(C3CCN(C)C3)=O)C2)ccc(=O)n(CCO)c1 C1(CC(=O)NCCCC(C)(C)NC(c2ccn(C3CC3)n2)=O)CC2CCC1CC2 c1(NC(=O)COC(C)C)ccc(C(=O)NC(C)CC(C)NC(CCSC)=O)cc1 C1(NC(CC(C)C)=O)CN(C(=O)CC(F)(F)F)CCC12CCOCC2.C(C)(C)(C)O C1(C(N2C(CNC(c3c(C(=O)OC)coc3)=O)CC2)=O)CN(C)CCO1 N1(CC)CCN(C(C2(N(C(=O)C(C)S(N)(=O)=O)C3CC3)CCC2)=O)CC1C CCCC(C(=O)N1CCN(C(=O)CCC(F)(F)F)C(CF)C1)S(N)(=O)=O c1(OCC)cccnc1C(=O)NC1COCCC1NC(=O)C(C)(C)CSC C1(C(N2CC3CC(NC(c4c[nH]ccc4=O)=O)C3C2)=O)CCc2ccccc2C1 N1(C(c2[nH]cc(CN(C)C)c2)=O)C2CCC1C(NC(=O)Cn1nccn1)C2 O=C(CCCCCF)N1CCN(C2CCN(C(C3(NSC)CC3)=O)C2)CC1 N1(C(C(C(=O)OC)OC)=O)CCOC2(CCN(C(c3cnn4cc[nH]c34)=O)C2)C1 c1(N2C(CC)CN(C(C3(c4cccs4)CC3)=O)CC2)ncnc2cnccc12 C(CC(=O)NC1CC(NCC2CC2)C1)OC N1(C(CSCC#C)=O)CCC(C)(CNC(=O)C(C)Oc2cccc(F)c2)CC1 c1(C(=O)NCCCN(C(=O)CC2CCC(=O)NC2=O)CC)ccc(O)c(F)c1 CC1(C)CC(CNC(=O)C(CCF)NC(c2ccccc2)=O)CO1 C(CC(C)C(=O)NCc1cc(C)c(C(=O)N(C)CCOC)o1)=CC C1(CCNC(c2ccoc2Cl)=O)CC2CCC(C1)N2C(=O)CN1CCCNC1=O C(=O)(CCCCC#N)NCCCN(CCCCC)C.C1(=O)CCC(=O)NCCCN1 C(=O)(CC(C)C(F)(F)F)N1CCC(NC(c2nc(C)nc(O)c2)=O)C1C(C)C c1(C(=O)NC2(C)CN(C(c3ccc(C)cc3F)=O)C2)ccc2c(C#N)c[nH]c2c1 C1(SCC(N2CCC(CC(=O)N(CC(C)C)CC)CC2)C)CCC=CCC1 c1(C(N2C(C(N3CC(C)C(CO)CC3)=O)CN(C)CC2)=O)cccc2[nH]ncc12 CC(C)C(O)C(C)(C)C(=O)N1CCOCC(C(=O)NC(c2n[nH]c(CO)n2)C)C1 N1(C(C(CCCCCC)F)=O)CCCC2(CCCN2C(=O)CNC(=O)CC)C1 C1(CCC(=O)NC2(C)CN(C(=O)COCc3nccs3)C2)CCCC(O)C1 c1(C(N(CC(=O)N(C)CC2CN(C)C2)C)=O)cscc1Cl C(CN=c1[nH]cnc(NCc2ccc(Br)c(C)c2)c1C)(c1ccsc1)OC c1(C(=O)OC)cc(C(=O)NCC2(NC(C3CC3Cl)=O)CCC2)cc(O)c1 C1(CCNC(CCS(C)=O)=O)CN(C(=O)CCN2CCC(O)CC2)CCCO1 CC(CCNC(=O)C(CNC(=O)C#CC(C)(C)O)CC1CCCC1)C(C)(C)C c1(CNc2nnc(NC(=O)NC3CC(CC(=O)OC)C3)s2)cccc(OC)c1 N1(CC)CC(C(=O)NC2CCN(C(=O)COCC3CCCO3)C2(C)C)CCC1=O N1(CC)CCCOC(CCc2ccc(Cl)nc2)C1 C1(O)(C(C(=O)N(CC#CC)CCO)F)CN(C(C2(OCC)CCOC2)=O)C1 Cc1cc(C)n(CCC(=O)NCCN(C(=O)C(C)C(C)c2ccc(F)cc2)C)n1 C1(OC)(OC)CCC1C(=O)NC(C)(C)CN(C)C(C12COCC1C2)=O C12(C(=O)NC(c3occ(C(=O)NC4CC(C(C)C)C4)n3)C)CCC(C1)OC2C c1(C(=O)NCCC2(CNC(CC=CC=C)=O)CC2)cccc(Br)c1C C1(CCNC(C=C(CC)C)=O)CN(C(C23CCC(C2)C3)=O)CC(C)O1 Cc1cn(C)nc1C(=O)NC1CCC(C)(CNC(c2cnc(C)n2C)=O)C1 N1(C(Cn2c(C(C)C)nnn2)=O)CC2CCC1CN2C(=O)Cc1ccc(Cl)cn1 C1(C)(OCC)CCN(C(C2CCN2C(C2CC3C(C2)C3(F)F)=O)=O)CC1 c1(N(C(c2cn(C)nc2)=O)C(C2C3COCC23)=O)ccc(Br)c2ccccc12 C1(NC(C2CN(C)C2)=O)CCCC(NC(c2ccc(C(F)(F)C(F)(F)F)s2)=O)C1 c12ncsc1OCC1CN(C1)C2=O.C(C(F)(F)F)OC c1(C(=O)NCC2(NC(c3ncn(CC)c3)=O)CCC2)c(Br)ccc(C)c1N C1(N(C)C(C2CC2(C)C)=O)CC2(CCN(C(C3CC3c3ccccc3)=O)CC2)C1 N1(C(C(CC)N(C)C)=O)CCC2CN(C(c3cccc(C#N)c3)=O)C2C1 C1(NC(C=C(C)C)=O)CCN(C(c2cnn(-c3nccs3)c2)=O)C(C)C1 N1(C(c2csc(Cl)c2)C(=O)Nc2c(CC)cccc2C)CC(C)OC(C)(C)C1C N(C(=NCCF)NCC(c1ccsc1)N1CCCC1)CC1CC(C(F)F)(OC)C1 N1(C(C)C)C(=O)COCC1C(N1CCC(CN(C(=O)C(=O)NCC2CC2)C)C1)=O c1(CC)ccc(C(=O)NC(C)CCNC(C2C(C#N)C2(C)C)=O)cc1Cl c1(C(N2CCN(C(C(CC)F)=O)C(C(C)C)C2)=O)cncc2c(F)cccc12 c1(OC)cc(OC)nc(C(N2CC(CNC(=O)COC(C)(C)C)C3(CC3)C2)=O)n1 C1(NC(C(=O)NC(c2cccc(OC)n2)C(C)C)=O)COc2ccccc2C1 C1(C(=O)NC2CN(C(C3ON=C(CC)C3)=O)CC2SC)CC(C)(C)CC(C)(C)C1 c1(C(N2CC3C(CNC(=O)CC4CCSCC4)(C3)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 N1(C(c2c(C)ccs2)=O)CCN(C(=O)CC2CCC3(CC2)COC3)C2CCC12 S(=O)(=O)(c1ccc(=NCCCCCCF)[nH]c1)N1CCCCC(C)(F)C1 C1(C(N(C)CCOC(C)(C)C)=O)CN(C(=O)Cc2nn(C)cc2Br)CCC1O c1(C(=O)NC(C(=O)OC)(C)C2CCCC2)cccc(S(=O)(=O)CF)c1 CCC(CC)CCCC(=O)NC(C)C(C)NC(c1occ2c1CCC2)=O N1(C(CC(CN(C)C)O)=O)CCC(NC(=O)CCOc2ccccc2F)CC1C c1(NC(C)=O)cnc(O)c(C(N2CC(N(C(=O)C=C3CCC(C)C3)C)C2)=O)c1 c1(N(C)C)ccc(C=CC(=O)NC2CCN(c3cc(O)nc(O)n3)CC2F)cc1 C(=O)(CC(C)(C)C(=O)NCCCN(C(=O)COC1CCCC(C)C1)CC)OCC N1(C(C)=O)CCCC1C(=O)NC1CC(C)(C(=O)N(C)CC2CN(C)C2)C1 N1(C(=O)OC(C)(C)C)CCCC2(CCSC2)C1.C=C1CN2C1COC2=O N1(C(C(N2CC(C)C2)C)=O)CCSCC1C(=O)NC(C)C(F)(F)F C1(CC(=O)OC)CCCC2(CN(C(=O)CC3CCn4cncc4C3)C2)O1 c1(OC)ccc(Br)c(C(=O)NCC2CCC2NC(=O)C(C)N(C)C)c1 c1(CN(C)CC2CCCCC(c3ccccc3)C2)cccn2cncc12 C1(C(N2CC(O)(CCNC(CCC(=O)N(C(C)C)C)=O)C2)=O)CCCC(C)CC1 C1(CCCC)CN(C(c2c(C)cnn2C)=O)CCN1C(=O)C(n1cc(Cl)cn1)C CC(C)(C)CCC(=O)NCCC1CN(C(C2(C)CCOC2)=O)CCO1 c1(N(CCOC)C(=O)OC(C)(C)C)ccc(NC(=O)N(C(C)C(F)(F)F)C)cc1 c1(OC)c(C)csc1C(=O)NCCN1CCN(C(=O)C(O)C(C)C)CC1 C(=O)(CC(C)(C)COC)NC1C(OC)CN(C(C2CC2CC(C)C)=O)C1 C1(CC)C2CCC(C2)N1C(=O)C(n1cc(-c2cnn3c2NCC3)nn1)C C1(C(=O)NCC(CC=C)NC(=O)CCN(CC)CC)CS(=O)(=O)CC12CC2 CC(C)C(O)CC(=O)N1CCC(F)C(NC(c2cc(C(F)(F)F)c[nH]2)=O)C1 N1(C(Cc2c(C)ncs2)=O)CCC(C)(C)CC1C(=O)NCC1CCOC1(C)C CCCC(C(O)C(=O)NCC1(C(C)(C)OC)CC1)NC(c1cccc(C)c1F)=O N1(C(C2(C)CC2F)=O)CCC(O)(CCNC(=O)C(C)(C)n2cc(Cl)cn2)CC1 C1(C(NOC(C(C)C)CO)=O)CCCN(C(=O)CN(c2ccncc2)C)C1 C1(C)(OC)CN(CC(=O)NCCOCCC(=O)N2CCC2CN=[N+]=[N-])C1 CC1=C(C(=O)NC2CCC3CC2CN3C(c2ccc(C(N)=O)[nH]2)=O)CCCO1 c1(OC)cccc(S(=O)(=O)Nc2cccc(F)c2C(=O)NC2CC2)c1Br c1(CC(=O)NCC2(O)CCN(C(C3C=CCS3)=O)C2)cncnc1O N1(C(COC(N2CCCCC2)=O)=O)CC2OCC(OCc3ccccc3)C2C1 c1(OCCCC)ccc(C(=O)NCC2(O)CCN(C(=O)CCCN(C)C)C2)cc1 Cc1nn(C)cc1C(C)C(=O)NCC12COC(CNC(c3cc[nH]c3C)=O)(C1)C2 c1(CCC)cc(C(N2CC(CNC(=O)C(C)(C)SC)CC2C)=O)nn1C c1(C(=O)NCC(C)(C)NC(CCc2cnc(C)s2)=O)cnn(C2CCCC2)c1C c1(C(=O)NC(CC)CNC2(c3ccccc3)CC2)ccnn1C(C)C C(CC(CNC(C1(CF)CC1(F)F)=O)NC(=O)CCOC)OC c1(CCC(=O)NC2C(NC(C(C)C3CC3)=O)C2)nc(-c2ccoc2)no1 c1(C(=O)NCC(C)CNC(=O)C(c2ccccc2Cl)(C)C)cccc(O)c1F N1(C(C(CC)(C)C)=O)CCN(C(C23CCOC(C)(C2)C3)=O)C(CCOC)C1 CC1=NOC2(C1)CC(C(=O)NC(C)(C)CNC(=O)CCc1ccc(F)c(F)c1)C2 C(CC(=O)NCCCCNC(c1ccccc1-n1cncn1)=O)(C(F)(F)F)OC CC(C)C(CNC(C1CCC(C)(C)C1)=O)C(=O)N1CC(=O)NC(=O)C1 c1(NCNC(C2CC3CC(NC(=O)OC(C)(C)C)C3C2)=O)cccc2ccccc12 c1(CC)noc(C)c1C(=O)NC1CC(NC(C2(CC)CCOC2)=O)C1 C1(C(N2CC(O)(CN(C(CCCOC)=O)C)C2)=O)CCC=CCC1 Cc1nc2c(cc1C(=O)NC(C)C(C)NC(=O)C1CC1)c(C)nn2C C(=O)(C1=CCCSC1)N(CCc1cn(-c2c(CN(C)C)cccc2)nn1)C CCCC(O)CC(=O)NC1CC(CNC(c2ccc(-n3cc(C)cn3)cc2)=O)C1 c12cccc(n1)NC2.C1(CC(=O)NCCC2CC(C(=O)OC)C2)CCCSC1 c1(C(N2C(CCNC(C3(C)C(C)C3)=O)CSCC2)=O)coc(S(N)(=O)=O)c1 C1(C(N2C(C#C)CC2)=O)CC2CC1CN(C(c1c[n+]([O-])c(C)cn1)=O)C2 CCC(C)(CNC(=O)CCCCCNC(c1c(F)cncc1F)=O)C(N)=O c1(C(c2cnc(CN(CCOCCCNC(C)=O)C3CC3)s2)=O)scc(C)c1Cl C1(O)(C(N(CC(CC)NC(c2ccc(-c3ccccc3)o2)=O)C)=O)CCOCC1 c1(C(=O)NCC2(F)CCCN(C(C(C)(C)OC)=O)C2)cccc2occc12 N1(CCc2c(C)cccc2)C(=O)CN(CCS(=O)(=O)Cc2ccccc2)C1=O N1(CC(C)(C)NC(C2CCCCC2O)=O)CCN(C(=O)CC2(O)CCOC2)CC1 C1(NC(C(CC)OC)=O)CC2C1CCN2C(c1cc(F)ccc1O)=O N1(C(c2ccc(N(C)C)cn2)=O)CCN(C(=O)C2=C(Cl)CCC2)C2CC12 c1(N(C)C)ccc(C2C(C(=O)NC3CCCC3NC(=O)CO)C2)cc1 C1(CCNC(C(C)NC(N)=O)=O)CSCCN1C(c1ccncc1Cl)=O C12CC3CCC1N3C2=O.c1(CNC(CN(C2CC(C)(C)C2)C)=O)ccc(Cl)s1 C1(NC(c2ccc(-c3cccs3)cc2)=O)CN(C(C2(O)CC2)=O)CCC1F C(=O)(CCCC(=O)NC(Cn1ccnn1)C(=O)NOCCCOC)OCC Cc1ncc(CC(N2CCC(CN(C(=O)CC3COC(=O)N3)C)CC2)=O)c(O)n1 c1(OC)noc(C)c1C(=O)NCC#CC(=O)N1CCC(C(C)O)C1 C(=O)(CC(O)c1ccccc1)NCC(C1CC1)NC(C1(CC)CC1)=O CC#CCCCC(=O)NCC(O)CNC(C1(C#N)CC1(C)C)=O C(=O)(C(C)CCO)NC(C1CCCCC1)CNC(C1CC(C)(C(=O)OC)C1)=O c1(CCC(N2CC(O)(CNC(c3nnn(CC)c3C)=O)C2)=O)ccc(C)c(C)c1 C1(NC(CC2C(C)(C)C2)=O)CC2CC1CC2C(=O)NC1CC(c2ncc[nH]2)C1 c1(CCC)cc(C(=O)NC2(CNC(C3(CSC)CCC3)=O)CCOC2)n(C)n1 c1(C(N(C)CC2CN(c3snc(CCC)n3)C2)=O)cnc(O)cc1OC C1(CN(C(=O)CC2CCCC2C)CC)CCN(C(c2[nH]c(C)nc2CC)=O)CC1 c1(NC(C)NC(N2CCC(c3nc(C4CC4)no3)(CO)C2)=O)cccc(Cl)c1F C1(C(=O)NC)(NC(=O)NC(c2ccc(C)cc2)CC=C)Cc2ccccc2C1 Cc1c(C(=O)NC2CC3CC2N(C(C2CC(=O)N(C)C2)=O)C3)cccc1C1CC1 C1(N(C(C2C(C)C2)=O)C)CCCC2CN(C(c3cc(O)nc(Cl)c3)=O)CC12 c1(C(=O)NCc2nc(CNC(c3cn[nH]c3)=O)nc(O)c2)cccc2c1COC2 N1(C(CC2(C)CCCC2)=O)CCC2(CCC2NC(c2cscc2Cl)=O)CC1 C(CNC(=O)CN1CCC(O)CC1)(C(C)(C)C)NC(C(C)SCc1ccccc1)=O c1(C(=O)NCCN(C(c2[nH]cnc2C)=O)CC)cc2nc(F)ccc2o1 C(=O)(C1=NOC2COCC12)NCC1CC(C)CN(C(C2(CC(N)=O)CC2)=O)C1 C12(CNC(c3n(C)ccc3)=O)CC(NC(C3CC4CC3C3CC43)=O)(C1)C(C)(C)O2 C1(N)CCCCC1C.C1(C(=O)OCC=C(C)C)(C)CC1 C(C)(CNC(=O)COCCCF)(CNC(C1(C)CC1(Cl)Cl)=O)OC N1(C(C(=O)NC(c2cccs2)C)=O)CCC2(CCC(=O)NC2)C1 C(=O)(C1=CC2CCCCCCC12)N(C1CCN(C(c2snnc2C)=O)CC1)CC c1(C(N2C3CN(C(CCSCC(C)C)=O)C(C3)C2)=O)cc2nccn2c(O)n1 N#Cc1c[nH]c(C(=O)NC(CNC(C2CCCO2)=O)C2CCC2)c1 C1(NC(=O)Cc2cnoc2)CCCN(C(=O)Cc2ccsc2Br)C1 N1(C(CC(Cn2cc(C3(C)CCCC3)nn2)C2CCC2)=O)CCC(C2CCC2)C1 C(C(CC(C)C)C(=O)N1CC(CO)C2(CC2)C1)NC(c1cc(CC)no1)=O c1(C2(C(N(CC(CN(C(=O)CSC(F)(F)F)C)O)C)=O)CCC2)ccccc1F Cc1cc(C=CC(=O)NCC2CC(NC(C3CCCC(C)(C)O3)=O)C2)c[nH]c1=N N1(C(c2cc(C)n(C)n2)=O)CCN(C(=O)CC2(O)CCCCC2)C(CC(F)F)C1 c1(OC)ccc(C)c(C(=O)NCC2CC(NC(=O)CC34CCC(CC3)OC4)C2)c1 C1(CC(=O)NCC(CC(C)C)NC(CCOC)=O)CCCC2CCCCC12 N1(C(CCn2c(C)nc(C)n2)=O)CCOC2(CCC(NC(=O)C(F)F)CC2)C1 O(N(C)C(=O)C(CNC(C1C2CCC(F)C12)=O)CC(C)C)CC(=O)OC N(C(=NC1CCC1)NC1CC1(C)C(F)F)Cc1ccc(OC(C)(C)C)nc1 c12cc(ccc1Cl)C(=O)N2.N1(CC)CCC(C(=O)O)C(O)C1 C1(Nc2ncc(C)cn2)CC2CN(C(C3C4COCC34)=O)CC12 c1(OC)cc(C)ccc1C(=O)NCCCN(C)C(C1CC1Cl)=O CC1CN(C(c2ccc(Cl)cc2N)=O)CCC1CNC(c1cc2c[nH]nc2s1)=O C(=O)(CC(C)(C)CN(C)C)N(C1CCN(C(C23CC(C(C)C)(C2)C3)=O)C1)CCO N1(C(C(C2CCN(C(Cn3ccc(C)n3)=O)C2)F)=O)CCNC(=O)C1 Cc1c(CNCC2CC(C)(C)Oc3ccccc32)ccc2c1CCC2 c1(CNC(=NCCSC)NCc2cccc(C(C)C)c2)ccc(S(C)=O)cc1 C#Cc1ccc(C(=O)NC(COC)CNC(C2(c3cc[nH]n3)CC2)=O)cc1C c1(OC)cccc(Cl)c1-n1nc(Cc2cc(F)ccc2F)nc1Cc1nccs1 c1(C(=O)NCCN(C(=O)COCCF)CC2CC2)nccc(Cl)c1O N1(C(C2(COC)CC2)=O)CCN(Cc2cc(Cl)c(Cl)cc2F)CC12CC2 N1(C(CN(c2ccccc2)C(C)=O)=O)CCCC(CO)(NC(c2cccn2C)=O)C1 CC(C)(C)C(CCc1ccc(F)cc1)NCCC1CCC1(F)F c1(NC2CC(CCNC(C(CC)C)=O)C2)ncc(Cl)c(O)n1 c1(N(CC(=O)NCCC)C)nc2cc[nH]c2c(=NC(CC)c2nccs2)[nH]1 Cn1nnc(C(=O)NC2CCCN(C(c3ccn(CC#N)n3)=O)C2)c1C(F)(F)F N1(C(C2CCC(N(C)C)C2)=O)CC2CCN(C(c3coc(O)n3)=O)CC12 Cc1nc2ccc(C(N3CCC3CNC(c3csc(CC(C)C)n3)=O)=O)cc2[nH]1 c1(OC)ncc(F)cc1C(=O)NCC1CC1CNC(=O)C1=COCCO1 c1(C(N2CCC(C)C(NC(c3cncnc3)=O)C2)=O)noc2c(F)cccc12 C1(=O)C(CC(C)C)CO1.Cc1ncc(F)cc1C(=O)OC(C)(C)C C1(NC(c2cnc3cccnn23)=O)CN(C(C2(CF)CCC2)=O)CC2(CC2)C1 C#CCC(O)C(=O)NCC(CCOC)NC(=O)C(c1ccc(O)cc1)(C)C c1(CNC(C)=O)cn(CC2CCCN2C(=O)CCC2CCOC2)nn1 C1(NC(c2cccc(O)c2)=O)CCN(N2CCN(CCn3cccn3)CC2)C1 c1(CNC(C2(C)CCN(C(C(=O)NCC=C)C)CC2)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NCC(C(=O)NC(C(=O)NCCC)CC)OC)cncnc1C CCC(C)CC(C)C(=O)NCc1ccccc1CNC(c1cnn[nH]1)=O c1(CCC(N2CC3C(NC(c4cnns4)=O)C(C3)C2)=O)cncc2ccccc12 c1(NC(=O)NC(c2ccc(Cl)cc2)c2ccccc2Cl)nc(C(F)(F)F)ccc1F C(CC(C(=O)NC1(C(=O)NC(c2ncccc2C)C)CC(F)C1)OC)OC C1(CC(=O)NCC2C(CNC(C3(OC(C)=O)CC3)=O)C2)CSCCS1 N1(C(c2n(C)cc(C#N)c2)=O)CCC2C(C1)CN2C(=O)CC1C=CCCC1 CC(O)C(C(=O)N1CCC(N(C)C(C2CCCN2C)=O)CC1)N(C)C Cc1ccc(C(=O)NCCCCC(=O)NC2(C(C)C)CCC2)cc1 n1(CC(=O)NC2(CNC(=O)CCc3ccon3)CCCC2)cc2ccccc2n1 Cc1cc(C(N2CCOC(C(N3CCS(=O)(=O)CC3)=O)C2)=O)c(F)cc1Br c1(NC(C2CCCCN2)C)cc(N2CCOC(c3nccs3)C2)ncn1 C12(CNC(c3occ(C)c3)=O)CCC(NC(=O)Cc3ccn(C)n3)(CC1)CO2 Cc1sc(N)c(C(N2CCC(C(C)NC(=O)CCOC(C)C)C2)=O)c1C c1(C(N2CCC(NC(c3cc(CC)oc3C)=O)CC2)=O)cccc2c1ncn2C C(N=c1[nH]c(=NCC2COCCO2)[nH]c2cccnc12)c1c(C)scc1 c1(C(N2CC(C)C(NC(=O)CNS(N)(=O)=O)CC2)=O)ccc2c(c1)C=CS2(=O)=O c1(C(=O)NC2CN(C(c3cncc(C)c3)=O)CC2C#N)c(Br)ccc(F)c1F c1(C(N2CC(O)(C(C)NC(C3C(CC)C3)=O)C2)=O)c(N)sc2c1CCSC2 N1(C(CCNC(=O)NC)=O)CC2C3CCC(C2C1)N(C(=O)C(C)CC(F)(F)F)C3 N#Cc1ccccc1C(N1CC(NC(=O)CNC(c2cscn2)=O)CC1CO)=O N1(C(C2N(C(C3(C)CCCC3)=O)CC(F)C2)=O)CCC(=C(F)F)CC1 c1(C(N2CC(=C(CNC(CCCCCC)=O)F)C2)=O)cc2c(=O)[nH]ccn2n1 N1(C(Cc2c(C)noc2C)=O)CC2CCOCC2(NC(c2coc(Cl)n2)=O)C1 CCC(CCO)C(C)NC(=O)NCCCCC1CCCC1 C(=O)(C1=NNC(=O)CC1)NC(C1CCCCN1C(c1cncc(CO)c1)=O)C c1(CC(=O)NC(CC)CNC(=O)CC2CC(=O)C2)cncc(Br)c1 n1(CC(=O)NCC2(F)CN(C(c3ccc(Cl)nc3O)=O)C2)cc2ccccc2n1 C(=O)(C1=C(Cl)CCC1)N(C(CNC(c1c(C)nn(CCO)c1)=O)C1CC1)C C1(C(N2CC(OCC(=O)N(C(c3ccco3)C)C)C2)=O)CN(C)CCN1C C1(C)(C(=O)NC(C2CC2NC(=O)C(c2ccc(OC)cc2)(F)F)C)CCC(=O)N1 c1(C(=O)NC(CCOC)CNC(=O)CC(C)SC)cc2cccc(Cl)c2[nH]1 C1(NC(=O)Cn2nnc(=O)[nH]2)CCCCCC1NC(c1ccoc1C(F)(F)F)=O C1(NC(c2cc(OCC)no2)=O)CCN(C(=O)C(CO)N(C)C)CC(C)(C)C1 CC12CC(NC(=O)CC3CCCOC3)(C1)C1(CN(C(=O)C(F)(F)C(F)F)C1)O2 C(=O)(C1=NOC(C)C1C)NCCOC1CCN(C(C(C)c2cc[nH]n2)=O)C1 N1(C(C(CC#C)C2CC2)=O)CCN(C(c2cc(Cl)n[nH]2)=O)C(CCCC)C1 c1(C(=O)NC2C(NC(C(C(CC)O)(C)C)=O)CCC2)ccnc2c1ncn2C N1(C(Cc2cnc(C)[nH]2)=O)CC2(CCCC2NC(=O)C=Cc2cncs2)C1 C1(CC(N2CCC(COC)(CNC(=O)CC(C)C)C2)=O)CCC(C)(C)CC1 C=CCCC(CCC=C)(c1nnnn1CCCF)NCc1cc(C(C)(C)C)no1 C(CS(=O)c1ccccc1F)NC(=O)Cc1cc(Cl)ccc1Cl Cc1n[nH]c(=NC(=O)c2csc(CN3CCCC3C(N3CCOCC3)=O)n2)o1 C(C)(C(CC(=O)NCCN(C)C(C)C)NC(=O)CCC1CC1(C)C)OC Cc1ccc(CC(=O)NNC(=O)C2OCCC2C(C)C)c(C)c1Br C1(CNC(C(C=C)(F)F)=O)CC2CCC1N2C(c1cccc(OCCC)c1)=O n1(CCOC(C2(c3c(Cl)cccc3Cl)CCC2)=O)cnc2ccccc2c1=O N1(C(C=CC(=O)NC(CC(C)C)C)=O)CCCC2CN(C(C)C(N)=O)CCC12 C(C)(C(=O)N(CCC(=O)NCCOC(=N)O)C)SC N(C(=NCCC(=O)OC)NCC(C(C)C(C)C)N(C)C)Cc1onc(COC)n1 N1(C(c2c(C)ccc(OC)c2)=O)CCCN(C(c2ncsc2Br)=O)C(C)C1 CC(C)CC(=O)C(=O)NC1CC(CC(=O)NCC2(O)CCCC2)C1 c1(OC)cc(C(=O)NC2CCN(C(C3C=CCC3)=O)C2C)sc1Br c1(OC)ccc(C(N)=O)cc1C(N1CCCC(F)(CNC(=O)C(CO)N(C)C)C1)=O N1(CC)CCC(C(=O)NCCCOC(C)C)C1.C1=CCNC1=O C=CC1CN(C(=O)C(CC(F)F)NC(c2cncnc2)=O)CC1O Cc1[nH]c(=N)sc1C(=O)NC1(CNC(C2C3CC3C3CC23)=O)CC1 CC1(C)C(=O)CC1C(N1CCC(CC(N2CC(C3CCCO3)C2)=O)C1)=O CC(C)C1=CCC(C)(C(N2CC(c3cn(CCCC(=O)O)nn3)C(O)C2)=O)CC1 Cc1scc(C(=O)N(C2CCN(C(=O)C(C)NC(=O)Cn3cnnn3)C2)C)c1C C1(NC(=O)NC2(COC)CC2)CCC(NC(=O)NCc2ccccc2)CC1 C=C(C)C(CC(=O)OCC(=O)NCCCNC)OCCN1CC(OCC)C1.SC c1(C(N2CC(CC)N(Cc3ccc(OC)cc3C)CC2)=O)ccc2ccoc2c1 c1(C(N2CC(n3cc(-c4c(Cl)ccc(OC)c4)nn3)C2)=O)nc2c(C)cccc2[nH]1 CON=Cc1ccc(C(=O)Nc2cc(Cl)c(C(=O)O)c(Cl)c2)cc1 N1(C(CC2=NNC(=O)C2)=O)CC2CN(C(c3cccc(F)c3)=O)CCC2(CO)C1 Cc1[nH]nc2cc(C(=O)NCCC(O)CNC(=O)CSCCC(F)(F)F)ccc12 c1(C(N2CCCC(CCNC(CC(=O)NCC#C)=O)C2)=O)ccc(NC)c(F)c1 C(=O)(CC(O)C(Cl)(Cl)Cl)N1CC(O)(CNC(c2sccc2C2CC2)=O)C1 CCCCC(O)CC(=O)N1CCCC(C)(C)C1C(=O)N(C)CC12CCC(CC1)C2 CC1CN(C(c2ccc(C(N)=O)cn2)=O)CC1NC(C1(O)CCSC1)=O CC(CC(=O)NC1CC2CCC1N2C(c1cc2ccccn2c1)=O)P(C)(C)=O c1(C(C)NC(c2ccc(C(N)=O)[nH]2)=O)nocc1C(=O)NC1CC1F C1(C2CCOCC2)(C(N2C(C)(C)COC2)=O)CC1(F)F c1(NC(=O)CC2N(C(C(C(=O)OC(C)(C)C)C3CC3)=O)CC2)cc(Cl)cnc1C C1(NC(C2CCC(C)(C)O2)=O)CCN(C(=O)CCC(F)F)CC1F C1(NC(c2ccc(CCC)s2)=O)CCCC(NC(=O)C=C(C)C)C1 C(=O)(CN=c1cc[nH]cc1)N1C(CCNC(c2cc(C3CCC3)on2)=O)CCC1 C1(C(=O)NCC(CC)(C)C)(COC)C=CCN1C(c1ccn(C)c1C)=O c1(C(=O)NC2CC(NC(Cc3c(C)n[nH]c3)=O)C2)cc2c(Cl)cncc2s1 S(=O)(=O)(c1cc(C(F)(F)F)ccc1Cl)N1C2CN(C(C3CCC(C)O3)=O)C(C2)C1 C(C1c2ccsc2CCN1C(c1cc(F)n[nH]1)=O)NC(c1ccc(OC)cc1)=O O=C1CC(CC(=O)NC23CCCN(c4ncc(C5CC5)cn4)CC2C3)=NN1 CC(C)CN=c1[nH]c(=NC(C)c2cccc(C#N)c2)c2c(Cl)cccc2[nH]1 C(=O)(C1Cc2ccccc21)N(C)CC1N(C(c2c(C)cc(N)c(C)n2)=O)CCC1 C=CCC(CNC(C1CC1C(C)(F)F)=O)NC(=O)C(C)=C(C)C C(CCC(C)C(=O)NC1CN(C(c2ccc(Br)nc2O)=O)CC1O)OC c1(C(=O)NC(C(C)NC(C(C)=C2CCC2)=O)CO)cc2c(nc1O)CCCCC2 C1(CC)(CO)CCCN(C(C2(C)CN(C(C3CCCC34CCC4)=O)C2)=O)C1 CC1(C)CCCC(CC(=O)NCC(C2CCCN2C(=O)CCS(N)(=O)=O)(C)C)O1 Cc1cc(CC(=O)NCc2cn(C3CN(C(C4CC(N(C)C)C4)=O)C3)nn2)n[nH]1 N1(C(c2cnc(CCOC)s2)C(=O)NCCOC)CCn2ccnc2C1 C=CCC(C(=O)N(CC(C)CC(=O)NCCCCCC)C)NC(C)=O C(CCCCCNC(C1(F)CC=CCC1)=O)NC(=O)CC1CCNC1=O C(CC(C)C(=O)NC(CNC(c1cccc(C(=O)OC)c1)=O)C1CC1)OC C(CC1CC1)(C(=O)N1CC(NC(C2CCC2C(C)(C)C)=O)C1)NC(C)=O Cc1c[nH]c2ccc(NS(=O)(=O)c3ccc(N4CCC(C(C)C)CC4)nc3)cc12 c1(OC)cc(C)c(CC(=O)NC2CC(F)CN(Cc3cccc(C)n3)C2)c(C)c1 c1(C(=O)NCC2CN(C(c3ccn(C)n3)=O)C(C)(C)C2)ccc2c[nH]nc2n1 N1(CCc2nnc(C)s2)CCC2(NC(=O)CCC3CCCN3C)CCCC12 CC(CC(=O)N1CCC(OCCNC(=O)CN(C2CCSC2)C)C1)C(F)(F)F Cc1noc(N(c2ccccc2)C(c2ccn(C3CCCC3)n2)=O)n1 C(=O)(C(O)CC(F)(F)F)NCC1CC(F)(CNC(C(C)NC(CC)=O)=O)C1 Cc1c(C(=O)NCC2C(C)CCCN2C(=O)C=C2CCSCC2)sc2cncn12 C1(CNC(C=CC=CCC)=O)(CO)CCN(C(=O)CO)CC1 CC(C(=O)NNC(=O)NC1CC2CC(C1)C2)NC1CCC(c2ccccc2)C1 C1(CNC(C2N(C(C)(C)C)CC2)=O)CC(F)(F)CN1C(=O)CCC(F)F C1(C(=O)NCC2CCCN2C(=O)CCOCC(F)F)CC2CCC(C1)S2(=O)=O Cc1ccccc1-n1ccc(C(=O)NC2CCN(S(=O)(=O)C(C)C)C2)n1 CCCC(C(=O)OC)C(=O)NCC1(F)CC(NC(C2CCCCC2O)=O)C1 Cc1cc(C)c(CC(=O)NC2CCCCC2CNC(=O)C(C)CF)s1 N1(C(CN(C2CCCC2O)C)=O)CC=C(CNC(C2(F)CCOCC2)=O)CC1 c1(-n2cc(C3(C(NOCCCC)=O)CC(F)C3)nn2)ccccc1F C12(CC(=O)O)CC(NC(=O)C=CC(=O)Nc3ccc(Br)o3)C1C2 C(=O)(C1CCc2nccn21)N1CCC(C(=O)NC2CC(C)(C)OC2=O)(CF)C1 CC1C(NC(=O)C(C)(C)C(F)F)CC2CCC1N2C(=O)CCN1CCCC1=O C(=O)(CC(C)CN=c1[nH]c(N2CCCC2CC2CCCCC2)nc(=N)[nH]1)NC C(=O)(CC(C)C(C)(C)C)N1CC(C)(NC(c2ccc(CCCCC)o2)=O)C1 Cc1ccc(C(=O)NCc2nc(CNC(=O)CCC3CC3C)cc(O)n2)c(Cl)c1 CC(C)C(O)CC(=O)N1CCN(C(=O)Cc2cncc(F)c2)CC1C(C)C C(=O)(CCCn1cc(COCC(=O)O)nn1)N1CC(CC)C1 C12(CNC(C3C=CCN(C(c4cc(C)n(C)n4)=O)C3)=O)CCC(C1)C(=O)N2 C(=O)(n1nc(CNc2nc(C)cs2)c2c1CN(Cc1cc(Br)c(Br)s1)C2)OCC C1(CCC(=O)NCC(CNC(c2oncc2Cl)=O)OC)CCCN1C CC(C)CC(CO)NC(C1C(C)CN1C(=O)C(C)N=[N+]=[N-])=O N1(C(c2ccc(C(C)=O)o2)=O)CCN(C(=O)C(C)(C)CC(F)F)CC(O)C1 C1(NC(c2sccc2C2CC2)=O)CCN(C(=O)CC2CC3CCC2C3)CC1CO C(=O)(C(C)(C)CC(=O)OC)NCC1N(C(c2c(CC)cno2)=O)CCCC1 CC(C)CCC(=O)Nc1ccccc1C1CCN(C(=O)OC(C)(C)C)CC1 c1(OC)ccc(S(=O)(=O)Oc2cc(Br)ccc2Cl)c(C)n1 C=Cn1nncc1C(N1CCCCC1CC(=O)N(C)CC1(N(C)C)CCC1)=O CN1C(=O)CCC1CC(N1CCC(Nc2cc(-c3cccc(Cl)c3)ncn2)C1)=O C1(CC(N2CC(OCC(=O)NC3C(CCCC)CCC3)C2)=O)CCC(C)(C)CC1 CC(C)C(C#N)C(=O)N(CCNC(C1CC12CC(O)C2)=O)C1CC1 c1(OC)ccc(C(=O)NC2CCC2NC(=O)Cn2cnnc2O)c2c1CCCC2 c1(C(N(CCN(C(COCC(c2ccccc2)C)=O)C)C)=O)cc2c[nH]nc2s1 C1(N(C(CC=CCC)=O)C)CCN(C(=O)C(C)=C2CC2)CC1C C1(C2CC2)(NC(c2ccccn2)=O)CCN(C(C2SCCS2)=O)C1 C1(C(N2C(C(=O)OC)CC2C)=O)CCC2CCC1N2C(c1cnns1)=O N1(C(c2cccc(OCCC)c2)=O)CCCC(NC(c2cnc(O)n2C)=O)CC1 C(=O)(C(F)CCC(C)C)NCC(CCC)C(=O)N1CCC(N2CC(O)C2)C1 CC(C)C(C)CCNC(C1OCCC1CNC(=O)C=Cc1cc[nH]c1)=O C(=O)(CC(C)(C)CC(F)(F)F)N1C(COC)CN(C(C2C=CC=CC=C2)=O)CC1 Cc1cc(C(=O)NC2CC(NC(c3[nH]nc(C(F)(F)F)c3C)=O)C2)cn(C)c1=O C(c1cc2cnn(C(C)C)c2[nH]c1=O)=CC(=O)NC(CC=C)CN c1(NCc2nc(N(C3CCC(C)(CC)O3)C(C)=O)sc2)c(F)ccc(C#N)c1F N1(C(c2c(C(C)C)n[nH]c2)=O)CC2(C(=O)NCCC3(O)CCOC3)CC1CO2 Cc1cnn(C)c1C(=O)NC(C1CCCCC1)CNC(c1ccc(Cl)cc1)=O N1(C(CSC)=O)CC2CC3CC2C1C3NC(=O)C(NC(C)=O)=Cc1cccs1 c1(Sc2c(C(N(C(C)C)C(C3CCC(C(=O)O)C3)=O)=O)n[nH]c2)cccc(F)c1 c1(C(N2CCCC(C(C)NC(C(C)NC(CC)=O)=O)C2)=O)ccc(F)c(CC)c1 C1(SC)CCN(C(=O)C(C)NC(=O)CNc2ccccn2)C1 Cc1ccc(C(N2CCCC2c2nccn2CCSC2CCOC(C)C2)=O)nn1 C1(O)(C(=O)NC2CC(CNC(c3c(F)ncc(OC)c3)=O)C2)CN2CCC1CC2 N1(C(C2C(=C)C2C(=O)OC)=O)CC(NC(=O)COCn2ccnc2C)C(C)(C)C1 C(CC(CNC(=O)C(C1CCCC1)OC)NC(c1cc(C2CC2)ns1)=O)OC C1(CNC(CCCC(N)=O)=O)CN(C(c2ccc(Cl)nc2O)=O)CC12CCC2 C(C)(C(C)C(=O)NCCCSC)NC(CC=O)=O.CCO c1(C(C)C)ncccc1NC1C=CCN1C(=O)OC(C)(C)C C1(C)(CC)CC(NC(=O)CN(C(=O)CCCN(C)C(C)=O)C2CC2)C1 Cc1c(C(N2CCCC(C)(CNC(=O)CCc3nccs3)C2)=O)cncc1Cl C12(CNC(c3n[nH]c(C)c3F)=O)CCC1CN(C(c1ccnn1C(C)(C)C)=O)C2 n1(CC)ccc(=NC(c2nnnn2Cc2ccccc2)C2(CC)CC(C)C2)[nH]1 N1(C(c2cc(C)c(C)[nH]2)=O)CCN(C(=O)CN2CCN(C(C)C)CC2)C2CC12 C12(C(N(CCCO)CCC)=O)CCN(C(c3nonc3C)=O)CCC1C2 C1(NC(c2cn3ccnc3s2)=O)CC2(CCCCN2C(=O)C2=C(Cl)CCCC2)C1 C1(NC(c2ccc(OC)nc2C)=O)CCC2(CCN(C(=O)CNC(C)=O)CC2)C1 C(=O)(C1CCCn2nccc21)N1C2CN(C(C3C(C)(C)CCCC3)=O)C(CC2)C1 CCC(CC(=O)NC1CC(O)C1)NC(=O)C(CC)n1cncn1 Cn1c(O)nc2cccc(C(N3CCCCC(NC(=O)CC4CCOC4)C3)=O)c12 N1(C(c2cnc(CC)[nH]2)=O)CC2CC(NC(=O)CSC(F)F)C1C2 N1(C(CCC(=O)NC)=O)CCC(C2(O)CC(NC(C3CC3C(N)=O)=O)C2)CC1 C1(CC)CN(C(=O)CC2CCCOC2)CCN1CC.c12scc(c1OC)NC2=O C1(C)(NC(CCOCCOC)=O)CCCCC1C(=O)Nc1cncc(C(N)=O)c1 N1(C(CC2C(C)CCC2)=O)CCN(C)C(C(N2CCC(c3ncco3)C2)=O)C1 N1(C(C(Cc2cn[nH]c2)NC(CNC(=O)NC)=O)=O)CC2CCC1C(O)C2O CC1(C)NC(=O)CC1C(=O)NC1CCC(NC(c2cccc(C3CC3)c2)=O)CC1 N1(C(C2N(C(C)=O)CCOC2)=O)CC2CCC1CN2C(=O)CC(C)(C)C1CC1 C1(NC(c2cccc(C(=O)OC)n2)=O)CN(C(=O)C(F)OC(F)(F)F)CC1(C)C C1(C(=O)NCC2C(CC(N3C(C(=O)NC(C)C)CCC3)=O)C2)CC2CCCC2C1 Cc1cc(Cl)c(Cl)cc1C(N1CC2(C1)CN(C(=O)C#CC1(C)CC1)C2)=O N1(C(c2cccc(OCCC)c2)=O)CCC(CNC(=O)CC(C)OC)C12CC2 c1(CCC)ncc(NC(C2CC(NC(=O)CN3CC(=O)NC3=O)C2(C)C)=O)cn1 c1(C(=O)NC(C(C)NC(c2cc(N)ccn2)=O)C)cc2c[nH]nc2s1 C1(C(N(C)CC2(O)CN(C(C(C=C)O)=O)C2)=O)CCCN(CC(F)(F)F)C1 c1(C(N2CC(NC(c3n(C(C)C)cnc3)=O)C(O)C2)=O)cnc(O)c([N+](=O)[O-])c1 CC1CC(C(=O)NCCCCNC(c2cncn2C(F)(F)F)=O)CO1 CC1CC(CNC(C2(CF)CC2)=O)CN1C(c1sc(Cl)cc1Cl)=O Fc1cccc2c1OCCC2NCC1CCC2(CCNCC2)CO1 C(CCCCCC(=O)O)N1CCC1=O.C=CCNC(=O)OCCCl Cc1c(CC(=O)N(CC(O)CN(C)C(C2(S(N)(=O)=O)CC2)=O)C)cnn1C C1(C(=O)NC(CCC)CO)(OC)CCN(C(c2cc(C3CC3)on2)=O)C1 C(=O)(C(F)C(C)CNC(=O)Cc1cc[nH]n1)N(CCF)CC C1(C(=O)NCCC2(OC)CN(C(=O)CCSc3n[nH]c(C)n3)C2)CC(=O)NC1=O C1(COC)CC(CNC(c2cc(O)cs2)=O)N(C(C2CNC(=O)N2)=O)C1 N1(c2ccnc(COC)n2)CCCC12CCN(C(=O)C(CC)OC1CCCC1)C2 CCCC(C(O)C(=O)NCC1(CC(C)C)CCC1)NC(=O)CCC1CCOC1 CC(C)(C)CC(=O)NCC1(NC(=O)C(F)C2CCOC2)CCCC1 C1(C(N(CCC(F)(F)F)C)=O)CC12CCN(Cc1cc3ccccc3[nH]1)CC2 CCCCCC(CC)C(=O)N1CC(CC(=O)NCC(C)(C)C(F)(F)F)C2(CC2)C1 C#CC1(C(=O)NC2(COC)CCC2)CN(C(=O)C(CCC)N(C)C)C1 C(=O)(C1=CCCSC1)NC(CC)CN(C(=O)CCC1CCCCO1)CC C(C(C)C(=O)N(OC)C(C)C)NC(CC(CCCC)O)=O c1(C(N2CCC(N(C(CC(C=C)(C)C)=O)C)C(C)C2)=O)ccc2ncncc2c1 CC1CC(c2cn(CCn3cccn3)nn2)CCN1C(C1CCC(=O)N1C)=O N1(C(c2cn(CC)nc2)=O)CCC(C(C)(C)CNC(=O)C(C)(O)COC)CC1 c1(NC(CCc2cccc(OC)c2)C)nc2c(cc1Br)CCC2O c1(C(N2CCN(C(C3ON=C(CC)C3)=O)C(C)C2)=O)nccc2n[nH]cc12 N1(C(C2CCC(C)(C)CC2)C(=O)NCCSC)CCC(C2(O)CCC2)CC1 C(C(CC(=O)N1CC[Si](C)(C)C1)NC(c1cnsn1)=O)OC C1(C(=O)NC2(CN(C(C(C)(CO)OC)=O)C)CC2)Cc2ccccc2O1 Cc1cc(C(=O)NCC2CCN(C(=O)C(C)Cc3ccco3)C2)c(N)c(F)c1 c1(C(N2CCC(CNC(=O)Cc3ccc(Cl)nc3)C2)=O)ccc2c(c1)COC2=O c1(C(N2C3CC(NC(C(=Cc4ccco4)C)=O)C2CC3)=O)ccc(Cl)c(F)c1F C(C)(C)(CCCCC(=O)N1CC(NC(=O)Cc2cc(C)no2)CC2(CC2)C1)OC C#CC1(C)CCN(C(=O)CC(C)C(C)(C)NC(=O)C(C)OCC(C)C)CC1 c1(C(=O)NCC2CN(C(CCC(=O)OCC)=O)CC2O)cnc(OC)c(C)n1 c1(C(N2CC(NC(CSCCC)=O)C(O)C2)=O)c(O)nnc2c1CCC2 c1(C(=O)NCC2(CN(C(C3C(CC(C)C)C3)=O)C)CC2)nnc(S)n1C C1(NC(C2(CSC)CC2)=O)CC2CC(NC(C3CCCCC3)=O)CC12 C=CC(C)(O)CC(=O)N1CC(=C(F)CNC(c2nn(CCC)cc2Cl)=O)C1 N1(C(C2N=C(C)SC2)=O)C2CCC1CC(NC(C1(C)CCCCO1)=O)C2 CC1CN(C(C2CCCC3CC23)=O)CCN1C(=O)Cc1ccnc(F)c1 N1(C(c2cc(C(N)=O)[nH]n2)=O)CCCC(NC(C2CCS(=O)(=O)N2)=O)C1 CCC(CC(=O)NCCCCCN(C(=O)CC(O)C1CCCC1)C)C(F)F c1(CNCCC(=O)NCC2C(C(C)C)=C2)ccccc1Cn1cncn1 C1(C(N(C2CC(O)C2(C)C)C)=O)CCC(C(=O)O)N(C(=O)OC(C)(C)C)C1 C1(C(=O)NC2CC3CC2N(C(=O)CCOCC2CC2)C3)CN2CCCN1CC2 c1(CSCC)cccc(C(=O)NC2CN(C(=O)CCc3nc(O)n[nH]3)C2)c1 C1(C(=O)NC(C2(O)CCCCC2)C)CC2(CC2)CN1C(=O)CC1=CCCC1 N1(C(C(CC)SC)=O)CCC2(C1)CN(C(C1CC(C(=O)OC)C1)=O)CCO2 N1(C(C(CC#C)(C)NC(=O)CC2CCCCC2O)=O)CCCC(C)(C#C)C1 C(C(=O)NC(c1c(C)noc1C)C)(C(C)(C)O)NC(C=CC=CC)=O C1(CC(=O)NCCN(C(=O)CCc2cnc(O)[nH]2)CC(C)O)CC2C=CC1CC2 C(=O)(C(F)(F)CN1CCCC1)N1CC(NC(C2N(CC(C)C)CCC2)=O)C1 C1(NC(c2c(OC)scc2)=O)COC2CN(C(c3cc(C)cc(C)n3)=O)CC12 C1(NC(C2CC3(CCC3)CO2)=O)CN(C(C2SCCCS2)=O)C2CCCCC12 c1(CCC(=O)NCC2(C(N3CCCC3CF)=O)CC3(CC3)C2)ncc(F)cn1 CCCCC(CNC(C1CCC(=O)N1)=O)NC(=O)Cc1cc(Cl)n(C)n1 N1(C(CC2CC(C)(C)OCC2)=O)CCC2CC1CN(C(c1ccon1)=O)C2 CCC(C(=O)NCC(CO)NC(=O)C(C)(C)OCCOC)OC(C)=O C1(C(=O)NC(CN(C(c2cc(C(=O)OC)sc2)=O)C)C)CC2(C1)CC21CC1 c1(C(N2CC(C(N3CC(C)C(=O)CC3)=O)OCC2)=O)cccc2c(O)nccc12 N1(C(C2CCCC(=O)O2)=O)CC=C(CNC(=O)C(N2CCOCC2)C2CC2)CC1 N1(C(C(CCCNC(C2CC2C2CC2)=O)O)=O)CCCC12CCOC2=O C1(C)(CNC(C(C)NC(c2cnc(C(F)(F)F)s2)=O)=O)CCCN(C(=O)C2CC2)C1 N1(C(c2cc(C)c(O)cc2)=O)CC(CNC(=O)CC2(C)CCC2)CC12CCC2 CCC(O)C(C)C(=O)NC12CC(NC(=O)Cc3cnn(-c4ccccc4)n3)(C1)C2 C1(CC)(NC(C2C3CCCOC23)=O)CCN(C(C2CCCC(C(N)=O)C2)=O)CC1 N1(C(CSC)=O)CCC2CCCC12C(N1CCC(CC2CCC2)C1)=O O(NC(=O)C(CCF)NC(C1CCC(C)(C)C1)=O)CCOCC#C c1(C(=O)NC(CC=C)CNC(c2ccc(Cl)o2)=O)c(OC)ccc2ncccc12 c1(C(N(C(C)C(=O)OC(C)(C)C)C)=O)cccn1C C#CCC(CC(=O)NCC(CC)N(C)C)NC(c1ccc(C(=O)N(C)C)cc1)=O N1(C(C(=O)NCCNC(C)=O)=O)CCC2CC2(NCCNC(C)=O)CC1 c1(C(N2CC(CN(C(C(n3ccc(C(F)(F)F)n3)C)=O)C)C2)=O)ccnc(O)c1 Cc1ncsc1COCC(=O)N(C)CCN(C(=O)Cn1nnc(C(C)(C)C)n1)C CC(C)(CCC(=O)NCCN1CCCC(O)C1)NC(c1ccsc1)=O c1(OC)c(O)cc(C(=O)NC2CC2C(N2CCN(S(=O)(=O)C(C)C)CC2)=O)cc1O C1(CN(C=O)Cc2cccc(C(F)(F)F)c2Cl)CCCC2(CCC2)O1 C1(NC(C2CCN(C(C)C)CC2)=O)CC12CCN(C(=O)CSCC(F)F)C2 c12cc(Cl)c(cc1C)[nH]c2=O.N1(C(CSC)=O)CCN(CCO)CC1C1CCC1 C1(n2cc(-c3c(C(=O)OC)n[nH]c3)nn2)CCCN(C(=O)Cc2cncc(C)n2)C1 CC1CC(NC(c2cc3c(s2)CCC3)=O)CCN1C(=O)CCc1cncnc1 c1(C(C)NC(C(=O)NCc2cn(CC(C)C)nc2)=O)csc2ccccc12 c1(NC(c2nc(-c3ccccc3)co2)=O)cccc(-c2cn[nH]c2)c1Cl N1(C(Cc2cc(C)on2)=O)CC(CNC(c2cccc(O)c2F)=O)CC12CCC2 C1(CC(=O)NC(C(C)C)CNC(=O)C(C)CSc2ccccc2)SC(=N)NC1=O c1(NCc2cnc(CC)s2)ncccc1S(=O)(=O)NC1CC1c1ccco1 c1(OC)ccc(OC)c2sc(N3CCCC3NC(C3(C)CC=CC3)=O)nc12 c1(C(CC(=O)NC2CCCC2NC(c2ccc(F)cc2)=O)O)cccc(F)c1 C1(C(=O)NCC(CNC(c2cc(Br)no2)=O)OC)(OC)CCOCC1 C1(NC(C(=O)NC)=O)CC2CCC1CN2C(=O)C(CC(C)C)n1ccnc1 c1(CCNC(=O)NCCN2CCCC(CC)C2)cc(O)nc(O)n1 C1(CNC(CCOCC#C)=O)CCCN(C(=O)C(C2CCC(O)CC2)(C)C)CC1 C=CCCC(F)(F)C(=O)N1CCCC1C(=O)N(C1(CCO)CC1)C c1(NCc2snc(CC)n2)nccc2cn(CC(=O)OC)nc12 N1(C(c2occ(C)c2)=O)C(C(=O)NCCC23CC(CO2)C3)CCC1C1CC1 N1(C(c2nc(C#C)sc2)=O)CCC(CO)(CNC(c2cn(C3CC3)nn2)=O)CC1 NS(=O)(=O)c1ccc(C(=O)NC2CCC(NC(c3ccc(F)c(O)c3)=O)CC2)s1 N1(CC(=O)Nc2cn(CCC)nc2C)CCC2CCCCC12 C(=O)(C(C)(C)CS(C)(=O)=O)NC1CCC(NC(C2(C(C)C)CCC2)=O)C1 c1(CCC(=O)NCCCCC2CN(C(C(C3CC3)OC)=O)C2)c(C)nn(C)c1C C1(C)(C(=O)NCC(CN(C(C(C)O)=O)C)C)CC2CCC1CC21OCCO1 c1(OC)ccc(S(=O)(=O)NCc2cc3sccc3s2)cn1 CCCCC(C(=O)N1CCC(CCNC(=O)C=CCCC=C2CC2)C1)C(C)C c1(CCN2CCN(C(N3CCC(O)(C(F)(F)F)CC3)=O)CC2)ccc(Cl)c(Cl)c1 c1(C(=O)NCC2(CNC(C3(C#N)CCC3)=O)CC2(F)F)cncc2nc[nH]c12 c1(C(C(=O)NC2CCCCC2)N(CCCSC)C)cc(S(N)(=O)=O)cs1 CC(c1ccccc1Cl)=CC(=O)NCC1CCC2(CN(C(=O)C(N)=O)C2)O1 C1(CC)CN(C(=O)CCCC(F)F)CCN1C(c1ccc(Cl)c(F)c1)=O C(CNC(c1cccn1CC)=O)(C(C)C(C)C)NC(c1c(CC)onc1)=O C(=O)(CC(C)C(F)F)NCCOCCNC(C(C)Oc1cccc(CO)c1)=O N1(C(C=Cc2nc(C)c(C)[nH]2)=O)CC2CCN(C(=O)CN3CCOCC3)CC12 c1(C(=O)NCC(C)(C2CC2)NC(C(C)OCC)=O)cccc(S(C)(=O)=O)c1 N1(C(Cn2c(=N)nc[nH]2)=O)CCC2CN(C(=O)Cc3ccnc(Br)c3)CCC12 CCC(CN(C)C)CC(=O)N(CCNC(C1CC1(F)F)=O)CCc1ccccc1 C1(COC)CCCN(C(=O)CNC(=O)CNC(C2(F)CCOC2C)=O)C1 CC1CCCCC1(CNC(C1(n2ccnn2)CC1)=O)NC(c1sccc1F)=O N1(C(C=C(C)C)=O)CC(NC(c2scnc2-c2ccccc2)=O)CC2(CCC2)C1 C1(C(=O)NCCN(C(=O)C(F)n2cccn2)CC)CCCC12CCC2 N1(CC(=O)NCCOCC#C)CCN(C(=O)COCCCC)CC1 c1(C(N2CCN(C(CC=CC=C)=O)CC2C)=O)cccc([N+](=O)[O-])c1O C1(NC(c2ccc(C)cc2)=O)CN(C(C2(C#N)CC2)=O)CC2(CC2)C1 c1(OC)nccnc1C(C(=O)NC1CC1)N(C)CCC1CCCCC1 Cc1c(C(=O)NCC(CNC(C2(F)CCC2)=O)C(F)(F)F)oc2ccc(F)cc12 N1(C(C(C)OC)=O)CC2CCC2(NC(=O)Cc2ncc(C)s2)C1 C1(c2ccn(C)c(=O)c2)N=C2C=CN(N2)n2nnnc21.CCCCOC Cc1cc(C(C)C)nc(=NCC2CC(CNC(c3cc(Cl)c(Cl)s3)=O)CO2)[nH]1 c1(C(=O)NC2CNCC(C)(C)C2)ccc2c(c1)NC(=O)C1CCCN21 C(=O)(C(CC)CC(C)C)NCC(CCC)C(N1CCC(=O)N(C)CC1)=O c1(OCC)ccc(CCC(=O)NCC(CC)NC(c2ccc(CC)[nH]2)=O)cc1 Cc1nn(C)c(CNCC2CN(C)CCN2C)c1S(N)(=O)=O N1(C(c2scc(C(=O)Nc3cc(Br)c(F)cc3Br)n2)=O)CCc2cccnc2C1 c1(C(=O)NC23CCC(CC2)N(C(C2CCOC2)=O)C3)[nH]cc2c1CCCC2 c1(C(c2n(CCOC)nnn2)NC2COCC2F)cc(C)cc2c1CCC2 c1(CC)ccc(NC(C2CC(=O)CN2C(=O)C(CO)OC)=O)cc1O CC(CCC(=O)N1CC(O)(c2nn[nH]n2)C1)NC(=O)COC1CCCOC1 C1(C)(C(N(CC(=O)N)C)=O)COC(=O)N1.C(CCO)(C1CC1)C(C1CC1)C1CC1 CCC(CCC(=O)NC1(C(=O)NCCC2CCCC2)CCSC1)OC CCC(C)CCCC(=O)N1CCC(O)(CN(C(=O)CSC(F)F)C)C1 C1(CC(N2CCC2)=O)(NC=O)CCSC1.C1(N2CCCC2)(C(F)F)CCC1 CN1CCC(NC(=O)C=CCC(C)(C)NC(c2n[nH]cc2[N+](=O)[O-])=O)C(C)(C)C1 c1(C(C)NC(c2cnco2)=O)cn(CC2CCCC2)nn1 C1(NC(COCCOCC)=O)COCC1NC(c1ncoc1COC)=O CC1CCC(O)(CNC(C2CSCN2C(c2cnc(N)cn2)=O)=O)CC1 C(=O)(CCCC(=O)NCC1(C)CCCN(C(=O)CC2CC3(CC3)C2)C1)OCC Cn1c(Cl)cnc1C(=O)Nc1cccc(NC(c2ncc[nH]c2=O)=O)c1 c1(CC)ccc(N)c(C(N2CCN(C(=O)C(CO)NC(N)=O)CC2C)=O)c1 N1(C(=O)NCc2c(OC)cc(Br)cn2)CC(N(C)C)C2(CCOCC2)C1 Cn1cc(C(=O)NC2CCC2NC(=O)CC2CCCC2)c(C2CCCC2)n1 c1(C(N2C3CCC(NC(=O)C(Cl)=CCl)C(C3)C2)=O)cccc2nc(O)ccc12 c1(OC)cnc(CNC(=O)CC2C=CCN2C(=O)C(C2(NC)CCCC2)=O)cn1 C1(CNC(c2ccc(CC)cc2)=O)CC2(CCC2)CN1C(C1CC1F)=O C1(OC)CC(C(=O)NCC(=O)Nc2c(C3CCC3)noc2C)N(C)C1 c1(C(=O)NC2CCN(C(C3C(C)CCC3)=O)CC2)cc(C(F)F)cc(Cl)c1 N1(C(C2C(C)(COC)C2)=O)C2CCCC1CN(C(c1ccc(Cl)c(Cl)c1O)=O)C2 C(C(C)(C)C#CC(=O)Nc1cccnc1N(C)C)NC(C(CC)n1cncn1)=O c1(C(=O)NC2(CN(C(c3scc(OC)c3)=O)C)CC2)ccc(C)nc1 O=C(CC=C(Cl)Cl)NC(c1cccnc1)C(=O)NCCOC(F)F C#CCCCCCCC(=O)NCC1COCCN1C(=O)C(C)CS(C)(=O)=O Cc1cccn2cc(C(=O)NC3CC(F)CN(C(c4c[nH]c(=O)cn4)=O)C3)cc12 C(=O)(C(CC(C)C)ONC(=O)C(C)NC(N)=O)NCc1cnc(C)[nH]1 Cc1cc(C)c(CC(N2CC(NC(=O)C(C)(C)C)C(C(F)F)C2)=O)c(C)c1 C1(O)(CNC(C2CC(C)C2)=O)CCN(C(c2csc(-c3ccoc3)n2)=O)C1 N1(C(c2n(C)ncc2)=O)CCCC12CCC(C(=O)NCC13COCC(C1)C3)CC2 c1(C(=O)NC2CC(C)N(C(C3CC(CC4CC4)C3)=O)CC2)ncsc1S(N)(=O)=O C=CCC(CNC(=O)C=Cc1ccc(C)cc1)C(=O)N(CC(O)CN(C)C)C C12(C(CNC(c3cc(C4CC4)on3)=O)NC(c3c(C)snn3)=O)CCC(CC1)C2 C1(C(N2C(C)CC2CO)=O)CCCCC1(C)NC(c1cccc(F)c1)=O c1(C(=O)NC(CCOC)CO)coc2c1CN(C(=O)CCc1cnco1)C2 C1(NC(C)=O)CCCN(C(C2C=CC(NC(=O)COCCCF)C2)=O)C1C N1(C(c2ccc(CNC(C)=O)o2)=O)CC2CCC1CN2C(=O)C(F)F c1(CN2CCC(CCC#C)C2)nc(C2CC2)n2ccccc12 C1(O)(CC(=O)NCC2CC(NC(c3cc(-c4ccco4)on3)=O)C2)CCCCC1 N1(C(C(C)(C2(C)CC2)OC)=O)CC(CNC(c2cn(C3CCC3)nn2)=O)C(O)C1 c1(C(=O)NCC(CC(C)C)(C)NC(C2CCN(C)CC2)=O)ncc2ccccn12 c1(C(=O)NCC(CC)NC(=O)CC2CCCN2C(C)C)c(C)cccc1[N+](=O)[O-] N(C(=NCCc1cccs1)N1CCS(=O)(=O)C(C)(C)C1)CC(=C)C C1(C(=O)NC2(CCC(=O)NCCN(OC)C)CCCC2)CCOC(CO)C1 N1(C(C2C(CCC)CCC2)=O)CCC2CCN(C(c3ccc(F)cc3C)=O)C2C1 c1(C(N(CC(CC)NC(=O)CC=C(C)C)C)=O)cnc(O)c2ccsc12 C(=O)(CC=C(Cl)Cl)NCC(N1CCN(C(C2(C(F)(F)F)CCC2)=O)CC1)C c1(C(=O)NCC2(O)CN(C(CCC(C)CN(C)C)=O)C2)cc(C#N)c(F)cc1F C1(C(=O)NC(c2cccnc2)CNC(=O)CO)C2CCC1(c1ccc(F)cc1)C2 Cc1ccnc(C(N2CCC(NC(=O)CC3CC3(C)C)C2)=O)c1Br CC(C)CC(C)(O)C(=O)NCc1ccc(C(=O)NC2CC(C)CC(C)(C)C2)nc1 N1(C(CC=CC=C)=O)CCN(C(c2cnc[nH]2)=O)C(CC#N)C1 c1(NC(=O)CC2CNCCN2)cc(Cl)cc2c1CCC2 Cc1ncc(F)c(NC2CC3CN(C(C4(C)CNC(=O)C4)=O)CC23)n1 n1(CCN2CCN(C(c3cccnn3)=O)CC2)cc(Br)ccc1=O N1(C(CCCC(C)=O)=O)CC(C(=O)N(C)Cc2ncnn2C)C2(CCC2)C1 N1(C(CCc2c(C)noc2C)=O)C2CC1CN(Cc1ccc(CO)cc1)C2 n1(CCC(C2(C(=O)NCCCc3ccsc3)CC2)C)cc(C(=O)NC)nn1 C(C(O)C(F)(F)F)(c1ccccc1)NC(c1c(C)nn(CC(F)F)c1)=O c1(CC(C(N2CC(C)(c3cn(-c4ncccn4)nn3)C2)=O)=O)ccc(F)cc1 C(=O)(CN=c1cc[nH]cc1)NC1CCC(NC(=O)CC(C2CC2)C2CC2)CC1 c1(CCNC(C(C2CN(C(C3COC(=O)N3C)=O)C2)OC)=O)ncccc1C N1(C(C(CC#CC)NC(C2CC=CCC2)=O)=O)CCOC(C)(C)C1C C(=O)(CC(C)CC(=O)NCC(C(C)(C)C)NC(c1cnccc1OC)=O)OC C1(C(=O)NCC2(C(N)=O)CN(C(CN3CC(C)C3)=O)C2)CCCSC1C C(=O)(C(CC(C)C)ONC(=O)CC)NC(C(=O)OCC=C)(C)C c1(-c2n[nH]c3c2CN(Cc2scc(C)c2)CC3)cccc(S(=O)(=O)N(C)C)c1 Cc1nc2cnn(C)c2cc1C(N1CC(n2cc(CN(C)CC3CC3)nn2)C1)=O CCC(C(=O)NCc1cccc(CN(C(=O)CCN(C)CC)C)c1)C(C)O c1(C(=O)NC(CC=C)CNC(C2CCOC2)=O)ccc2[nH]c(=O)cnc2c1 c1(OC)ccc(CCC(=O)NC(C2CCN(C(c3ccc(C)s3)=O)C2)C)cc1F C#Cc1ccccc1CC(=O)N(CC(C)(C)NC(C1SC2C=CC1CC2)=O)C N1(C(CC2C(C)CCC2)=O)CC2CCCC(NC(=O)C3=COCC3)C2C1 c1(C(N2CC(NC(Cc3c(C)noc3Cl)=O)C(C)C2)=O)cccc(F)c1F c1(C(=O)NC2CC(F)(Cc3ccno3)C2)nc(C(=O)NC2(COCC)CC2)cs1 C(=O)(C(CN(C)C)NC(C1CNC(=O)C1)=O)NC(c1cnc[nH]1)C C1(C(N(C2CCN(C(C3(F)CCOC3)=O)CC2)CC)=O)CCc2c[nH]nc2C1 C1(C(=O)NC2C(CNC(C3CN(C)C3)=O)C2)COCC1(C)C N1(C(C2C3N(C(CN(C4CC4)CC)=O)C(CC3)C2)=O)CCc2c(O)noc2C1 C1(NC(C#CC(C)C)=O)CCC2CC1CN2C(C1CC2(CCOC2)C1)=O C#CCC(O)C(=O)N1CC(CNC(=O)CCCSC)C(C)C1 c1(C(=O)NCC2CCCN(C(c3c(Cl)cn(CC)n3)=O)C2)cnc(N)c(CO)c1 Cc1nc(C(C)N(C)C(c2sc(N(C)Cc3ccccc3)nc2C)=O)c(C)s1 C=CCC(CC=C)C(=O)N(C(C)CNC(=O)C(C)NC(N)=O)CC N1(C(COCCCOC)=O)CC2CCC2(CNC(c2cccc(=S)n2O)=O)C1 C12(C(=O)NC(CC)CO)CCC(C(=O)NCc3cncs3)(CC1)CC2 C(CN=c1cc(NCCC2CCCC23CC3)nc[nH]1)c1cc(Br)ncc1 c1(C(=O)NC(C)CC2CN(C(=O)Cn3cc(N)cn3)C2)ccc(Cl)nc1Cl CCCCCC(CC)C(=O)N1CCC(C2(NC(c3csc(CCC)n3)=O)CC2)C1 C1(N(C(=O)CC2CC(C)(C)C2)C)CN(C(=O)COC(=O)CO)CC1F C1(NC(Cc2cc(C)[nH]n2)=O)CC12CCN(C(c1cnc3n1CCCC3)=O)CC2 c1(CC(=O)NCC(c2ccccc2)NCC2(CC)COC2)ccc2nn[nH]c2c1 c1(-c2cn(C(C)CNC(=O)CSc3ccc(Cl)cn3)nn2)cc(F)c(F)cc1F N1(C(C=CC(=O)OCC)=O)CCC2(CC1)CC2C(=O)NCC(C)(C)n1ccnc1 C1(CC(=O)NCC(c2nncn2C)C)C2CCCC2N1C(C1(Cl)CC1)=O N1(C(c2c(C)scc2)=O)CCN(C(C2OCCOC2(C)C)=O)C(CCO)C1 C=CCCC(C(=O)NCC1CCCO1)N1CCC(c2cncc(C)c2)CC1 CC(C)(C)CC(O)C(=O)NCC1CC1NC(=O)Cc1ccccc1F c1(C(N2CC(OC)C(NC(c3ccc(O)cc3F)=O)C2)=O)cc([N+](=O)[O-])c(C)s1 c1(N2CC(C)(C)c3c(ccc(F)c3)C2)nc(=NC2C=CCC2)[nH]c2c1COC2 O=C(C1CCc2ccccc21)NCC1CN(C(c2ccn3c2CCCC3)=O)C1 c1(C(=O)NC(C)(CNC(=O)C(O)Cn2cncn2)CO)ccc2c(n1)CCCC2 O=C(NNCc1nccs1)NC1C(CNCCOCCOCCOc2ncon2)C1 c1(C(N(C2CCN(C(=O)CCC3CC3(Cl)Cl)C2)CCC)=O)cn(C2CC2)nc1C N1(C(c2ncn(C)c(=O)c2)=O)CC2CCC(NC(C3COCCO3)=O)CC2C1 CC(C)CC(C(C)(C)C)NCc1ccn(Cc2ccc(F)cc2)n1 C(=O)(C(C)S(N)(=O)=O)NCC1(O)CC(C(=O)Nc2cccc(C(C)C)c2)C1 C(CCCCC(=O)NC(CC1CC1)CC(=O)OCCOc1ccccc1)C1C(C)C1 c1(N(C(=O)OC)C)cccc(NC2(C)CCOC2)c1 Cn1cc(-c2ccc(NC3CCc4c[nH]nc4C3)cc2)c2ccccc12 c1(C(N(C2CN(C(CCC)=O)C2)C)=O)cnc2n1CCC2 c1(CC)cc(OC(=O)COc2cncc(Br)c2)cc(CN(C2CCC2)CC)c1 N1(C(c2c(C)c(=O)cc[nH]2)=O)CC23CCCC2(C1)CN(C(c1cc[nH]n1)=O)C3 Cc1ccc2c(c1)CN(C(=O)CC1CCCN1C(c1cc(=N)[nH][nH]1)=O)CC2 CN(C)NC(=O)CCC(=O)NC1(C2CCCN(C(=O)CCOC3CCC3)C2)CC1 C1(NC(C2N(C)CCC2)=O)C2CN(C(c3cccc(OC(C)(C)C)c3)=O)CC12 c1(C(=O)NC2CC(C)CN(C(=O)CC3(C)CCC3)C2)ccc2cnnn2c1 C#CCC(C)(C)C(=O)NCC1(C(C)(C)C)CCN(C(C2C3CC4C(C3)C24)=O)C1 Cc1ccc(C(=O)NC2CC(C)CN(C(=O)C(c3cn(C)nc3C)O)C2)cc1F N1(C(COCC=C)=O)CC(NC(c2ccc(-c3ccc(F)cc3)s2)=O)CC(O)C1 Cc1c(C(N2CC(NC(=O)C=C3CCC3)C3(CC3)C2)=O)cccc1CO C(=O)(CS(=O)(=O)NC(C)(C)C)N1C(CNC(C2C(c3n(C)ncc3)C2)=O)CCC1 N1(C(C(C)CO)=O)CCC2(C1)CN(C(=O)CCOC1CCOC1)C2 C12(NC(c3nc(SC)sc3)=O)CCC(CC1NC(=O)CC1(N3CCCC3)CC1)C2 C(=O)(CCCCCc1nn[nH]n1)NC1(C)CCN(C(C)C)C1 C1(C(=O)NCCC(C)N(C(c2cn(C(C)C)nn2)=O)C)CCN(CCO)C(=O)C1 N1(C(C2CCC2)=O)CC(C2CC2)(C(=O)NCCc2csnn2)C1 C(=O)(C(C)C(=O)NCC(F)CNC(c1ccc(OC2CCCC2)cc1)=O)OC c1(C(N2CCC(CNC(C3CCCC(OC)C3)=O)CC2)=O)ccnc2[nH]ncc12 c1(NC(C2N(Cc3ccc(C(=O)O)cc3)CC(O)C2)=O)nc2c(s1)CCC2 O=C(C1Cc2ccccc21)N1CCCC(F)(C(=O)N(C2CCC2)C2CCC2)C1 c1(COC)nc(OC)cc(N2CC(O)(C(C)NC(c3c[nH]cc(F)c3=O)=O)C2)n1 C=C(C)C(O)CC(=O)NCc1ccc(CCNC(=O)CNC=O)cc1 c1(C(N2C(CNC(c3c(C)nc4sccn43)=O)CC2)=O)c(Cl)nc2ccccn12 c1(C(=O)NCCCC(O)C(=O)NCC2CCCS2)ncn2ccccc12 N1(C(c2c(C)cnn2C)=O)CC2CCCC(CNC(=O)C3=CCC(C)CC3)C2C1 C1(C(=O)OCC)(C(=O)NCC2(O)CN(C(=O)COCCOC)C2)CC12CC2 N1(C(CC2CC(C)C2)=O)CCN(C(c2ccnn2C(F)F)=O)CC1CF C(N=c1[nH]c(=NCC(CC)CCCC)c2sccc2[nH]1)c1c(NC)nccc1 C1(O)(CSC)CCCN(C(c2cc(Cl)cc(Cl)n2)C(=O)NCC(C)C)C1 N1(C(C(CC(C)C)C)=O)CCC2CN(C(c3cccc4c3COC4)=O)CC2CC1 N1(C(C2CCN(C)C2)=O)CC(N(C)C(c2csc(-c3ccsc3)n2)=O)C(O)C1 c1(C(=O)NC2CCN(C(=O)C(O)c3cnc[nH]3)C2)cc(Cl)cc2ccncc12 C1(CNC(C2CCC(CC)C2)=O)CN(C(C2(n3cccn3)CC2)=O)CC12CC2 N1(C(C2CCC(C(N)=O)O2)=O)CC2CC2(CNC(C2CC(F)(F)C2)=O)C1 CCC(C)(C)C(=O)NCC(C(=O)NC1CC=C(C)CC1)N(C)C C(=O)(C(C)C(C)(C)C)NCCC1CCN(c2ccnc(CC(=O)OCC)n2)C1 c1(C(N2C3CN(C(c4cc(C)oc4)=O)C(C3)C2)=O)cccc2ccnn12 Cc1cc(C(=O)NCC2(F)CCC(CNC(c3cnn(C)c3C)=O)C2)cnn1 N1(C(CC(CCC)C)=O)CCC2CCN(C(=O)Cn3ncnn3)CC12 C1(C(N2C(C(=O)N(C)Cc3n[nH]c(C)n3)(COC)C=CC2)=O)CN(C)CCN1C N1(C(CCOC2CCN(C)CC2)=O)CC2CCCC(C1)N2C(=O)C=CC=C(Cl)Cl C1(NC(C(C)Oc2cccnc2)=O)CCC2CN(C(c3cnoc3)=O)CCC2C1 C1(C(N2CCCC(NC(c3cccnc3)=O)C2)=O)(NC(C)=O)CCOCC1 c1(C(N(C2CC3CNC2C3)c2snc(C)n2)=O)cc([N+](=O)[O-])c(O)cc1O N1(C(C2(CCNC(=O)CC3CCCC3)CCCC2)=O)CC(O)(C2CCC2)C1 CN1N=C(CC(=O)N2CCOCC(CNC(c3ncn4c3CCC4)=O)C2)CC1=O c1(-c2ccc(COC)cn2)n[nH]c2c1CN(C(c1cc(F)cnc1Cl)=O)C2 c1(C(=O)NCC(C)(CO)NC(C(C=CC)O)=O)ccc2c(c1)COC2 Cc1cc(C(F)(F)F)nc(N2CC3C(NC(c4ccc(F)cc4Cl)=O)C3C2)n1 Nc1c(Cl)cc(C(N2CCCC2CCNC(c2cc(C3CC3)[nH]n2)=O)=O)cc1Cl C1(C(=O)NCC(C2CCCC2)NC(c2csc(C)n2)=O)(CC)CCCC1O Cc1noc(C(C)(C)NC(=O)CCNC(=O)C(C)Cn2cccn2)n1 c1(C(N2CC(O)(CCNC(c3cc(F)ccc3F)=O)C2)=O)cc(F)c(O)c(F)c1 C1(CC(=O)NC(CN(C(=O)C(c2ccccc2)OC(C)C)CC)C)CCC(C)CC1 C(=O)(CC(O)CC(C)C)NC1(CCOC)CCN(C(=O)C(C)=C(C)C)C1 CCN=C(NCC1CCCC(CS(C)(=O)=O)C1)N1CCC(CC(F)(F)F)C1 c1(C(C(=O)N(C2CN(C(C3(C)CC(F)(F)C3)=O)C2)C)O)ccccc1Cl C1(NC(C2C(C)(C)C2NC(=O)C=Cc2nccs2)=O)CCCCC12CCC2 CC1CC(C(=O)NC(C)(C)CNC(=O)COC2CCCCCC2)CC(C)C1 Cc1cc(Cl)c(Br)cc1C(N1CCC12CN(C(c1ccc(Cl)c(Cl)n1)=O)C2)=O C#CCCCCC(=O)NCC(=C)CCNC(=O)CCOc1cccnc1 C(CCCCC(=O)N1C(C(=O)NOCC2CC2)CCC1C)SC c1(OCC(=O)N(C(CCNC(CSCC)=O)C)C)ccc2ccc(=O)oc2c1 C1(C(=O)NC(C)(CNC(C2(CS(N)(=O)=O)COC2)=O)C2CC2)SCCCS1 C(C1=NOC2CCCC12)NCC1CCS(=O)(=O)C1 C#CCC(C)C(=O)N(CCNC(C1CCCC(C(C)(C)C)C1)=O)CCOC c1(C(N2CC(C(C)NC(=O)CC3CCC3)OCC2)=O)cc(N)c(F)cc1F C1(C(=O)NCC2CN(C(CC3CC(N(C)C)C3)=O)C2)CC2CCCCN2C1 C1(NC(C2(OC)CCCSC2)=O)CCN(C(=O)CC(C)(C)N(C)C)CC1C CC1CCC(=CC(=O)NCC2(CNC)CC2C(F)(F)F)C1 C1(C(=O)NC(c2ccc(C#N)s2)C)CCCN(Cc2noc(C3CCCO3)n2)C1 C1(NC(c2c(CC)n(C)nn2)=O)CCC(C)N(C(=O)CC(=O)NCC2CC2)C1 c1(OC)ccc(CCC(=O)NC2CC(N(C(=O)C3=CCCC3)C)C2)c(F)c1 C12(NC(CCC=C)=O)CCCC1CN(C(c1cccc(F)c1C)=O)C2 C12(CNC(c3cc(O)cs3)=O)CC1CN(C(C1CCO1)=O)C2 C1(C(=O)OC(C)(C)C)C2Cc3c(Br)cccc3C12.C12CC3CCC1(C3)CN2 C1(NC(CC2C(CC)C2(F)F)=O)CC2(CCN(C(c3csnn3)=O)CC2)C1 Cc1cccn2cc(C(=O)NCC3CCC3NC(=O)C=CCn3cncn3)cc12 CCC(C(=O)NC(CC(=O)N(C1CCCC1(C)O)C)C1CC1)C(F)(F)F C(CC(C)C(C)(C)C)NC(C#C)CCCOC(C)(C)C.C(=O)O C(=O)(C1=C(Cl)CCC1)NCc1oc(C(=O)NC(CSC)(C)CO)c(C)n1 C1(CNC(N2CC(C3CC3)C2C2CC2)=O)CCC2(CC1)NC(=O)NC2=O C1(NC(C(CCCC)NC(CC(=C=C)C)=O)=O)CCOC12CCCC2 N1(C(c2c(N)ccc(Cl)c2)=O)CC2(CCCC2NC(C2CC2F)=O)C1 CC1CC(N=c2nc3c(cnn3C)c(N(C)Cc3ccoc3)[nH]2)CCN1C C12(CNC(c3n(C(C)C)ccc3)=O)CCC(C1)N(C(=O)Cc1sc(O)nc1O)C2 Cc1cc2nc(Cl)nc(N(CC(C)NC(=O)CN3CCOCC3)C)c2s1 C1(C(=O)Nc2c(C#N)cno2)CCC2(CN(C(c3sc(Cl)nc3Cl)=O)C2)O1 C1(NC(CC(CC)(C)C)=O)CCC2(CC1)CN(C(=O)CN(S(C)(=O)=O)C)CCO2 c1(C(=O)OC)ncnc(N2CCC(C)(NC(c3ccoc3C)=O)C2)c1OC C1(C(N(C(C(=O)NC(CC)COCC2CC2)C)CC)=O)CC2CCC1O2 C1(NC(=O)CCc2ccco2)CCCCC1NC(C1CC1c1ccccc1)=O C1(C(N2CC(N(C(C(C)C#N)=O)C)C2)=O)CCC2(CCCO2)CC1 CC1(C)NC(=O)CC1C(N1CC(C(=O)NCc2cc[nH]n2)C2(CC2)C1)=O C12(CNC(C3(CC(N)=O)CC3)=O)CCC(CN(C(=O)CNC(N)=O)C1)C2 N1(C(CSCC(C)C)=O)CCC(F)(CNC(=O)C(C)NC=O)C1 CCCC1C(=O)OCC(=O)NCCN(CC)C1=O.C1(OCC)CCC(F)(F)CC1 C(=O)(C(CC)(CC)CO)NC(CCCNC(COC)=O)c1cccs1.c12ccc(o1)C2=O c1(-c2ccc(C(C)O)cc2)cc(=O)n(C)c(O)n1 N1(C(C)C(=O)NCCN(C(c2ccccc2)=O)CC2CCCO2)CCCCCC1 N1(C(c2c(NCC)scn2)=O)CC2CCC(C1)C(NC(=O)C(C)n1ccnc1)C2 CCC(CCc1ccccc1)NC1CCCCC1 Cc1ccc(NC(=O)CN2CCN(C(=O)COC3(C)CCCC3)CC2)c(O)c1 c1(C(=O)NCC2C3CN(C(C(C(C)(C)C)(C)O)=O)CC32)n[nH]c2ccc(Cl)cc12 c1(NC(c2cnc(C(C)C)nc2)c2nnnn2C(C)C)cc(Br)cc([N+](=O)[O-])c1 C1(NC(Cn2ncc(C)cc2=O)=O)CC(C2CCN(C(=O)C=CC(F)(F)F)C2)C1 O=C(CC(F)(F)F)NC1CC12CC(NC(=O)CNC(C1CCC1)=O)C2 c1(NC(C)=O)ccc(Cl)c(C(F)F)c1.C1(CC(=O)N2CC2)CCC(O)C1 c1(COC)cnc(OC)c(C(=O)NCC2CC2OC)c1.C1(=O)C(C2CC2)N1 N(C(=NCCN1CCNC1=O)NCC1(C(F)F)CCCO1)CC(=O)NC(C)C Cc1[nH]c(C(=O)NCc2cncc(Cl)n2)c(C)c1C(=O)NCC1CCCCO1 CCCC(C(=O)NC12CC(CNC(c3ccc(C(C)=O)o3)=O)(C1)OC2C)C(C)C C1(CNC(C(C=C)O)=O)(NC(c2ncc(OC(C)C)cc2F)=O)CCCCCC1 C1(NC(=O)NC(c2ccccc2OC)CC)COc2ccccc2C1O N1(C(C(CC)OC)=O)CCCCCCC1C(=O)Nc1cnc(OC)cc1C C#CCCCC(C)C(=O)N1CCC(O)(c2cn(C(C(=O)C3=CCCCO3)=O)nn2)CC1 c1(C(N2CC(CCNC(c3ccc(O)cn3)=O)(OC)C2)=O)cc(C)ccc1F CC(C)C(C)(O)C(=O)NC1CC2CN(C(=O)C(CN(C)C)N(C)C)CC12 C1(CC(=O)NC2CN(C(C(C)OC(C)(C)C)=O)C2)CSc2ccccc2O1 c1(C(=O)NCC(CNC(c2scc(OC)c2)=O)OC)cc(SC)c(C)o1 C(=O)(CC(C(F)(F)F)n1ccnc1)NC1(CO)CCN(C(c2cn(C)nn2)=O)C1 N1(C(C=C(C)C2CC2)=O)CCOC(CNC(=O)CN2CC(C)C2)C1 N1(C(CC(C(=O)OC)C)=O)CCCC(C2(NC(=O)C(F)C(F)(F)F)CC2)C1 Cc1cn(CC(=O)NC2CCCC(C(=O)NCC3COC(=O)N3)C2)c(=O)nc1O Cc1sc(C(N2CC(O)(C3CCCN3C(c3ccnn3C)=O)C2)=O)c(C)c1C CCC(C)(C)C(C)CC(=O)NC1CC(C)CN(C(C2CC3C=CC2C32CC2)=O)C1 c1(C(C)=O)cc(C(N2CC(NC(C3CN(C(=O)N(C)C)C3)=O)C(C)C2)=O)n(C)c1 c1(-c2scc(C(=O)NCCC3CCN(C(C(CC)OC)=O)C3)n2)ncccc1F N1(CC(=O)NCC2(O)CN(C(C3C(C)(C)COCC3)=O)C2)CCCCC(O)C1=O Cc1cc(N2CCC(C)(CS(C)(=O)=O)CC2)nc(NC(C)CC(C)(C)C)n1 S(=O)(=O)(c1ccc(F)c(Br)c1)N1CC2(C(C(=O)NCc3ccn(C)n3)C2)C1 c1(C(=O)NCC2CCC(NC(Cc3c(C)noc3)=O)C2)ccc(N)c(O)c1 C(=O)(C1=COc2ccccc2O1)NC(C(C(C)C)NC(CC)=O)C c1(COC)cccc(CNC(c2ccccc2)C(N)=O)c1 C12(NC(c3c(C)ncn3C)=O)CCCC1N(c1nc3ccccc3s1)CC2 C1(C)(CNC(C(C)=CC2CC2)=O)COCCN(C(C2(C)CC=CCO2)=O)C1 C1(CNC(C(CC)n2cncn2)=O)CCCN(C(=O)CCCn2cncn2)CC1 N1(C(C(OC)OC)=O)CCC(NC(C2CCCCN(C)C2=O)=O)C12CCC2 c1(C(N2CCC(O)(CCNC(c3n(C)cnc3)=O)C2)=O)ccc2cnnn2c1 C#CC(C(C)(C)C)NC(C1CC12CC(NC(C1(O)CCSCC1)=O)C2)=O C1(C(=O)NCCCC(C)NC(=O)Cc2ccon2)CC1C1CCOCC1 C#Cc1cn(C)nc1C(=O)NC1CCCN(C(=O)Cc2csc(C(C)C)n2)CC1 Cc1nn(C)cc1CC(=O)NCCN(C(=O)CCc1cnn(C)c1)C1CCCC1 C(CC(C(=O)NC1CN(C(=O)CC2COCC2O)CC1C)NC=O)SC CC1CCC(NC(C2CC(C)(F)C2)=O)CN1C(c1csc([N+](=O)[O-])c1)=O Cn1nc(C(N2CCN(C(=O)C=CC3CCCCC3)C3CC23)=O)c2ccccc12 C1(C)(CCCC(=O)N(C2CCSC2)CC2(C)C=CCCC2)NC(=O)NC1=O C1(NC(C(C)(C)n2cnnn2)=O)CC(F)(F)CC1NC(c1ncc(Cl)cc1F)=O S(=O)(=O)(c1ccc(NC2(CC)CCC(=O)N2)nc1)NC(CCCC)C C1(CC)CC(C(N2CC3(CCN3C)C2)=O)CCN1C(=O)CCC1(C)CC1 c1(C(N2CCc3ccc(O)cc3C2)C(=O)NC(C)C)cc(Br)cc([N+](=O)[O-])c1 C12(CNC(CCNC(C)=O)=O)CCC(CC1)N2C(=O)CCC(C)N(C)C Cc1coc(C)c1CN(CCN(C)C)CC.C1(C(=O)N)CCC2CC12 c1(C(=O)NC2C(C)CN(C(c3cccn3C3CC3)=O)C2)cc(N)cc(N)c1 c1(C(=O)NC(CNC(C(F)=C(C)C)=O)(C)CC(C)C)ccc2c(c1)CCC=C2 N1(C(C(CC=C)(C)N(C)C)=O)CCC2(CC1)CN(C(C1(C)COC1)=O)C2 N1(C(C(C)(C)OC)=O)CCC(N2CCC(NC(=O)COCC(C)(C)C)CC2)CC1 c1(C(N2C(CNC(C3CCCSC3)=O)CC(OC)C2)=O)cnn2cc[nH]c(=O)c12 CCC(C(=O)NC1(C)CN(C(=O)COC(C)=O)C1)n1ccnc1.c1ccsn1 C(=O)(CCC(N)=O)N1C(C2CCN(C(COCc3ncn(C)n3)=O)C2)CCC1 C(=O)(CCS(C)(=O)=O)NC1(CCNC(CNS(N(C)C)(=O)=O)=O)CCCC1 C(=O)(C(C)(C)C(=O)N(C)C)NCCN(C(C(N1C(CC)CCC1)=O)=O)CC(C)O C1(NC(C(C(C)C)C)=O)C2CC3C(C2)C13C(=O)NCC12CC(CCO1)C2 N1(CC)CCCC(C(=O)NCC2(NC(c3nc(CO)cs3)=O)CC2)C1 C(N=c1[nH]c(C)ncc1C)c1c(C)nn(COCC)c1C c1(C(N2C3CN(C(CCc4scc(C)n4)=O)CC2C3)=O)cccc2occc12 C1(CCC(=O)NCc2nc(C(C)C)cs2)CCN(C(C2CCC(CC)O2)=O)CC1 c1(C(N2C(CCC)CN(C(=O)C(C)OC)CC2)=O)cc(=O)c2cc(F)ccc2o1 N1(C(C(C2(OC)CCCCC2)(F)F)=O)CC2CC(NC(=O)CC(C)C(C)C)C1C2 c1(C(=O)NCC2C(NC(C3(CC)CCCCC3)=O)CC2)nc(C)ccc1C Cc1cnn2cc(C(=O)NCC3CCCN(C(=O)CC4OCCC4C)C3)cnc12 C1(O)(CNC(C2C(=O)NCC2)=O)CCN(C(=O)COC(F)(F)C(F)(F)F)C1 c1(C(N2CCC(OCC(C)C)C2)C(=O)NC(CC)C)ccc(S(N)(=O)=O)s1 C12(NC(C3(OC(C)=O)CC3)=O)CC(NC(=O)C=Cc3ncc[nH]3)(C1)C2 OC1Cc2ccccc2C1NCc1cnc(C(F)F)s1 CN1CCN(C(C2CCCN2C=O)=O)C(CNC(=O)Cn2nnc(C3CC3)n2)C1 CC1(C)CC2(CC(C(N3CCCN(C(C45CCC4C5)=O)CC3)=O)C2)C1 c1(C(N2CC(CC=C)(NC(COCC#C)=O)C2)=O)cc(F)cc2cccnc12 CCCCC(O)CC(=O)NC1CCC(NC(c2ccc3[nH]ccc3n2)=O)C1 N1(C(C2C(OCC)C2)=O)CCC2(CCCN(C(c3cncc(SCC)n3)=O)C2)C1 c1(CNC(C(CCC#C)O)=O)nnc2n1CCN(C(=O)CC(C)C(C)C)C2 C1(C(=O)NCCC2CCC(NC(C3(CN(C)C)CC3)=O)C2)(CC)CCCC1 N1(CCC(=O)NC(CN(C(c2nc(CC)sc2)=O)C(C)C)C)CCC(C)CC1 Cn1ncc2ncnc(N3CC4(CN(C(=O)C#CC5(C)CCCO5)C4)C3)c12 C=C(C)CCC(=O)NCCOCCCCCNC(=O)Cc1cnoc1 c1(CC)ccc(C(=O)NC2CC2NCCC(=O)NC2CCCCCC2)cc1 N1(C(CN(C(C)=O)C)=O)CCC(CCNC(c2c[nH]nc2C)=O)CC1C CONC(=O)C(=O)NC(CCN(C)C)C(=O)NCC1(O)CCCOC1 N1(C(c2cnc(CC)s2)=O)CCSCC1CCNC(C1CC(F)C1)=O CCCCCCCCC(F)C(=O)NC1CC2CC1N(C(=O)C(OC)OC)C2 c1(C(=O)NCCCNC(c2cn(C(C)(C)C)nn2)=O)c[nH]c2nccc-2c1 C12CN(CCO1)c1nnnn1CC(c1ccccc1)C2C.C1CC1.C1N=C1 C(=O)(C1=NOC(C)C1C)NC(c1ccnn1C)C(=O)NCCC#C c1(CNC(C2N(C(C(c3ccc(O)cc3)(C)C)=O)CCC2)=O)cc(Cl)ccc1F C(=O)(C1=CNS(=O)(=O)N=C1C)N1CC(NC(CC2(C=C)CCC2)=O)CC12CCC2 N1(C(CSCC=C)=O)CCN(C(c2csc(C(F)F)n2)=O)C(CCCC)C1 C(C(C)(C)C(=O)NCC(c1cnn(C)c1)C)N(C(c1n(CC)ncc1)=O)C c1(C(N2CCN(CC(F)F)CC2)C(=O)NCCCOC)ccnc(P(C)(C)=O)c1 C1(C(N(CC(C)C)CCCN2CCCCC2)=O)CCc2n[nH]cc2N1C(=O)N(C)C Cc1scc(C(N2CCN(C3CN(C(c4cnn(C5CC5)c4)=O)C3)CC2)=O)c1N C(C(O)CC(=O)NOC1CC1)NC(=O)CC1CCCO1 C(=O)(C(CCC(N)=O)=CCCCCC)N(CCCC#C)CCCCN(C(C)CCC)C.O C1(NC(C(C=C)(C)C)=O)CCC2CN(C(C3C(C)C3C)=O)CCC2C1 C1(NC(CCCCC=C)=O)CN(C(c2cc(C)c(C)o2)=O)CC1C1CC1 c1(C(=O)NCC(O)C(=O)NCc2cncn2C2CC2)ccncc1F c1(C(N2CCCC2CF)C(=O)NCC)cn(C)nc1CC1CCCOCC1 C(=O)(C(O)CC(N)=O)N1CCC(CCNC(Cc2cc(C(=O)OC)sc2)=O)CC1 Cc1ccc(NC(C2CC3CC3N2C(c2nc(C(C)C)cs2)=O)=O)cc1Br N1(C(C(CC)(C)COC)=O)CC2CCC(CNC(=O)Cc3cnn(C)c3)C2C1 C1(n2cccn2)(C(=O)NCCCN(C(CSCCOC)=O)CCO)CCC1 N1(C(c2c(C)ccs2)=O)CC(NC(c2cc(F)cc(F)c2)=O)CC12CCC2 Cc1cc(S(N)(=O)=O)sc1C(=O)N(C1C2CN(C(=O)C#CC3CCCO3)CC12)C Cc1cccc(Cn2nc(CCC(C)C)nc2CCCN(C2CCCCC2)C)c1 N1(C(C(C2CC(C(=O)NC3CC=CCC3)C2)F)=O)CC(C2CCCC2)C1 c1(C(N(CC(CNC(CC(C)C2CC2)=O)O)C)=O)ccn2c1CSCC2 C1(NC(CCN(C(C)=O)C)=O)CC(F)(F)CC1NC(=O)CCC1CCCN(C)C1 C=CC(C)(CCOC)C(=O)N1CC2(C(N3CC=C(C)CC3)=O)CC1CO2 c1(C(=O)NCCCN(C(=O)C(O)CN(C)C)CCC)nn(C)cc1C(=O)OCC c1(C(N2CCCC(CO)C2)=O)cc(-c2ccc(OC(F)F)cc2)cc2c[nH]nc12 C1(C(N(C)CC)=O)CCC(F)(CNC(=O)C(C)(C)CN(C)C)CC1 C12(CNC(C(C)O)=O)CCC(CF)(C1)OC2.c12occc1C(=O)OC2=O N1(C(CC2CCN(C(c3n(CC)ncc3)=O)C2)=O)CCSC(C)(C)C1 C12CC(CN1C(=O)C(O)(C1CC1)C1CC1)n1cc(nn1)C21CC1.c1(SCC)nccs1 C1(NC(CCOCC#C)=O)CCN(C(c2nc(C)oc2C)=O)CC1CO N1(C(CCC=C=C)=O)CCN(C)CC1CNC(c1ccnn1CCOC)=O N1(C(C(CC)OC)=O)CC2CCC(C1)C2CNC(C1CCC2(CC1)CC2)=O c1(C(=O)NC2CN(C(c3c(OC)ccs3)=O)CC2C)cc(Br)cc(F)c1O C1(NC(COC2(C)CCCC2)=O)CCCC2CN(c3nc4cccnc4s3)CC12 C(CN=c1nc2c(cnn2C)c(NCC2CCN(CCF)CC2)[nH]1)c1ccc(C)s1 c1(NCc2c(CC)cco2)nc(O)c2nc[nH]c2n1 c1(C(N2CC(NC(=O)CC(C)C)CC(OC)C2)=O)cc(O)ccc1[N+](=O)[O-] c1(C(=O)NCC2C(C)(C)CN(C(C3CCCSC3)=O)C2)csc2c(O)ccnc12 C1(F)(CNC(C(C(C)C)N(C)C)=O)COCCN(C(=O)CCc2nccs2)C1 c1(CC(=O)N(C(C)CNC(=O)C(C)n2cncn2)C)nsc2ccccc12 C(=O)(CCCCCCS(N)(=O)=O)N(C)Cc1ccccc1F Cc1cc(C(F)(F)F)sc1C(=O)NC(C1(O)CN(C(=O)Cn2cnnc2O)C1)C C#Cc1cn(C)nc1C(=O)NCCCCC1(NC(=O)CC2CCCCC2C)CC1 C(=O)(CC(O)CC(C)(C)C)N1CC2C(NC(Cc3c(C)ncc(Cl)c3)=O)C2C1 c1(C(N2CC(C(C)NC(CSCCC(C)C)=O)C2)=O)cocc1C(N)=O N1(C(C=C(CCC)C)=O)CCCC1C1CCN(C(c2c[nH]nc2C(C)C)=O)C1 C(=O)(CCCC(=O)N(C)C)N1C(CCC(N2C(C)CCCC2)=O)CCC1 c1(C(N(C(C)CCNC(c2cc3occc3[nH]2)=O)C)=O)cnc2ncnn2c1N N1(CCNC(C2NC(=O)OC2)=O)CCN(C(C2CC(CF)C2)=O)CC12CCC2 C12(CNC(C3C(C)(C)CCO3)=O)CCCC1CCN2C(c1cc2ccsc2s1)=O c1(OC)cc(C)c(C(N2CC=C(CNC(C3(CO)CC(F)(F)C3)=O)CC2)=O)cn1 c1(C(=O)NCC(CC)NC(C2(C(C)C)CCC2)=O)ccc(S(=O)(=O)NC)cc1 C1(C(=O)NC(C2(O)CCN(C(c3ccnn3C)=O)C2)C)CC=CC(O)C1 C=CCCC(C(=O)N1CC(O)(CC(C)C)C1)NC(c1c[nH]c(=NC)s1)=O C(C(CC(C)C)C(=O)N1CC2(CC(NC(C3CC(F)CN3C)=O)C2)C1)OC C12(OC)CCC(C(=O)NC3CCN(C(=O)CCCF)CC3)(CC1)C2 n1(CC(=O)NCCC2CN(C(c3c(CC)ocn3)=O)CC2C)ccc(C)cc1=O c1(C(=O)NC(CCOC)CNC(=O)CC2CCCCO2)ccc(Br)c(N)c1 C1(C(=O)NCC2C(CNC(c3csnn3)=O)C2)Cc2c[nH]cc2S1(=O)=O C#CC1(C(N2CCC3CC23)=O)CCN(C(C2CC2c2ccc(C)cc2)=O)CC1 CS(=O)c1ccc(C(c2nnnn2C2CC2)NC(c2ccc(Cl)cc2)C2CC2)cc1 Cc1nn(C)c(C)c1CNC(C1CCCN1C(=O)CCCC1CCC1)=O c1(OC)ccc(NC(=O)C(=O)N(C(C)CS(C)=O)Cc2cccc(F)c2)c(C)c1 c1(C(=O)NCC#CCNC(C2(O)CC(C)(C)C2)=O)cnc2[nH]ncc2c1 c1(C(N2C3CN(C(C4C(C#N)C4)=O)CC2CC3)=O)ccc2c(c1)CCNC2=O c1(CC(=O)NCC(C)(C)NC(C2CCC(C#N)C2)=O)cc(C(F)(F)F)c(O)nn1 N1(C(COC)=O)CCC2OCCN(C(=O)CN3CCCCC(O)C3=O)C2C1 c1(C(=O)NC(C(=O)NCC2OCCN(CC)C2)C2CCCC2)ccc(F)c(F)c1 C(=O)(CC1OCc2ccccc21)Nc1ccc(N2C(C)COCC2)cn1 C1(NC(C(CCC)(C)O)=O)CN(C(c2cscc2CC)=O)CC1C1CC1 c1(C(N2CCCC(N(C)C(c3scc(Cl)c3Cl)=O)C2)=O)c(C#N)cnn1C N1(C(C2CN(c3c(C)ccc(C)c3)C(=O)C2)=O)CCc2cccc(Br)c2C1 Cc1cc(C)c(C(=O)N(C)CC2C3CN(C(=O)C#CC(=O)N(C)C)CC23)cc1C C1(CC(=O)N(CC(C)C)Cc2cc(F)ccc2F)CCCCC(=O)N1 c1(C(=O)OC)cc(OC)c(NC(C2CC23CN(CC2CCCS2)C3)=O)cc1OC c1(OC)cc(C(N2CC(NC(=O)C=C3CCC(C)C3)C(C)(C)C2)=O)c(O)c(Cl)c1 c1(C(=O)OC)c(C(=O)N(CC(C)N(C(=O)C=C2CCC2)C2CC2)C)noc1C c1(CNC(Cn2ccc(C)n2)=O)cc(C(=O)NCCC(O)C(C)C)ccn1 C1(CNC(CCc2ncc(C)[nH]2)=O)CC2(CO1)CN(C(=O)C(N)=O)C2 C1(C)(C(N2CCC(CCNC(C(CC)N(C)C)=O)C2)=O)CCN(C)C1=O C(CCCCC(=O)NC1(CO)CCN(C(C2CCC2(OC)OC)=O)CC1)OC N1(C(C2C(C)C2)=O)CCC2(CCCN(C(=O)COc3ccccc3O)C2)C1 N1(C(CN2CC(CC)C2)=O)CC(CNC(=O)C(C)(C)CO)C(F)(F)C1 c1(C(=O)NCC2(CNC(Cn3c(C(C)C)nnn3)=O)CC2)cc2cccnn2n1 c1(C(N(C(=O)CN2CC3CCCCC3(CO)C2)CC)C)cccc2ncccc12 Cc1cc(C(N2CC(CNC(=O)C#CC3CC3)C(F)(F)C2)=O)cc(NC2CC2)n1 C(=O)(NN1CCCC1C(=O)N(C)Cc1c(C)cnn1C)C1C(CCC)C1 C1(CN(C(=O)CCc2ccc(C)cc2)CC)CCN(C(C2COC(=O)O2)=O)CC1 C(=O)(C(C)(C)CCNC(C1C2CCC(F)C12)=O)Nc1c(CC)n(C)nc1 CCC(C)(CO)C(=O)N1CC(O)(C(C)NC(c2cc([N+](=O)[O-])c[nH]2)=O)C1 N1(C(CN(C(C(CCC)F)=O)C2CCC2)=O)CCN(C(C)C)C(=O)C1 C1(N(C(C2CN(C(C)C)C(=O)C2)=O)C)CCC2CN(C(=O)CNS(C)(=O)=O)CC12 C1(C(=O)NC2CN(C(c3cc(C)no3)=O)CC2CC(C)(C)C)CN2CCC1CC2 C1(CC(=O)O)COCCN1CC(=O)Nc1ccsc1C(=O)O S(=O)(=O)(CC(=O)NCCCC(C)NC(c1csc(-c2ccccc2)n1)=O)NCC C1(C(=O)Nc2nc(C)sc2)CC12CCN(C(c1cnc(C)nc1C)=O)C2 c1(OC)cc(C(=O)Nc2sncc2C#N)c(-c2ccnc(C#N)c2)cn1 N1(C(C(C)OCC(C)C)=O)CCOCC1C(=O)NCCCCC1CC1 C1(C(=O)NCC2(CO)COCC(C)N2C)CCc2cnccc2N1 CC1CCSC1C(N1CC(F)(CNC(=O)CCc2ncc[nH]2)C1)=O c1(CC)oc(C)cc1C(=O)NCC1CCN(C(c2csc(=NC)[nH]2)=O)C1 C(=O)(C(C)(C)CNC(=O)CC1CC=CCC1)N(C(C)C)C C(=O)(C1COc2ccccc21)N(CCN(C)C(c1cncc(CO)c1)=O)C C1(S(N)(=O)=O)(c2cn(CC3N(C(C(C)C4CCOC4)=O)CC3)nn2)CCC1 N1(C(C(=O)NCCCC)C)CCC(Oc2cccnc2)C1 c1(C(=O)NCCN(C(C(C2CCCCC2)OC)=O)C2CCCC2)ccc(F)cc1F N1(c2c(Cl)ncc(C)n2)CCCC2(CCN(C(=O)C(C)(C)C)C2)C1 C=CCC(C)C(=O)N1CCCC1CC(=O)NC1COCC1N(C)C C1(OC)CC(C(=O)NC2CCC2NC(c2csnc2C)=O)N(S(C)(=O)=O)C1 O=C(CC1=CCOCC1)N1CCN(C(=O)Cc2ncc(F)cc2F)C2CC12 N1(C(C(C)NC(CC)=O)=O)CCC2C(C(=O)N(CCCO)CCO)C2C1 N1(C(c2ccc(CN(C)C)[nH]2)=O)CCC2(CCCN2C(C23CC(C2)C3)=O)CC1 N1(C(C=NOC)=O)CCC2(CCN(C(=O)Cc3c(C)cccc3C)C2)C1 C1(C(C)NC(COCCCCC)=O)CCN(C(c2cc(C(C)(C)C)no2)=O)C1 C1(N(c2snc(CCC)n2)C)CCN(C(c2oc(C3CC3)nc2C)=O)CC1 c1(C(=O)OCC(CCc2ccc(C(=O)OC)cc2)=O)cn2ccccc2n1 CN(C)NC(=O)CCC(=O)NC1C2CC1N(C(C1(C)CC3CC3C1)=O)C2 C(=O)(C(O)CC(F)(F)F)N1C2CCC(NC(C(=CC3CCC(C)CC3)C)=O)(C2)C1 c1(C(=O)NCCC)cn2c(n1)CN(C(c1cc(=O)ccn1C)=O)CC2 N1(C(c2c(CC)csc2)=O)CCCC(N(C(=O)Cn2nccc2C)CCF)C1 CCCC(CC1CCCC1)C(=O)NCC1CCC(NC(C2CCN(C)C2)=O)CC1 C1(OC(C2(CNC(=O)C(F)C3CCOC3)CC2)C)CCN(C(=O)CO)C1.C(N)(=O)N CC1(C(=O)NCc2ccccc2CNC(=O)CN2CC(=O)NC2=O)CCCCO1 N1(CC#C)CCC(CNC(=O)CC2(NC(C3CCN3CC)=O)CC2)C1.C(C)(C)(C)O C1(C(=O)NCc2nc(CC)[nH]n2)CC=CC(NC(=O)C(c2cncnc2)C)C1 C1(NC(C=CC(C)(C)SC)=O)CC(C)(CNC(=O)CC2(C3CC3)CC2)C1 Cn1cc(Br)c(CC(=O)NCc2ccc(CN3CCC(O)C3)cc2)n1 N#Cc1nc(=NCC2CC(CNC(c3cc4ccc(Cl)cc4[nH]3)=O)CO2)cc[nH]1 C(CCC(=O)NCC(CO)C(C)C)(C(C)C)NC(c1cc(C)nnc1C)=O CCC(C(=O)N1CCCCC(NC(=O)C(C)(C)N(C)C)C1)C(C)O c1(C(N2C(CNC(c3c(C)n[nH]c3)=O)C(C)CCC2)=O)cc2nc(=O)ccn2[nH]1 c1(CCC(=O)NC2CC(F)(C(F)(F)F)C2)cnc2cc(Br)ccn12 C(=O)(C1CCc2cccc(F)c21)NCCNC(c1cncc2sccc12)=O O=C(CS(=O)(=O)CC1CCCO1)NCCC1(O)CN(C(c2cnnc(O)c2)=O)C1 N1(C(c2cnn(C(C)C)c2Cl)=O)CC2CCN(C(C3CCC(=O)N3C)=O)C2C1 C1(C(C)NC(=O)NC(CS(C)(=O)=O)c2ccccc2)CC2(C1)CC21CC1 C1(NC(C2CCC(=C)CC2)=O)CCN(C(=O)Cc2cc(F)ccc2C)CC1CO C1(NCC)CCCC(N=c2[nH]c3c(c(=NCC4(C)CC4)[nH]2)CSC3)C1 c1(N(c2cn(C)nc2)CC2CC2)ncnc2c1ccn2CC#N c1(OC)ccc(C2(C(=O)NCCNC3CC(F)(F)CO3)CCCC2)cc1Cl c1(C(N2CCN(C(C(N)=O)=O)C3C2COC3)=O)cc(C2CC2)nc2ccc(Cl)cc12 c1(C(N2C3C(NC(c4cc(C5CC5)on4)=O)C(C3)C2)=O)csc2ncnc(O)c12 CC1(C)CCCC(C(=O)NCc2csc(C(=O)NC3CC(C)(C(N)=O)C3)c2)C1 C(C1CCCN1C)=CC(=O)NCC1CCC(NC(C(C)OCC2CC2)=O)C1 C(=O)(C(C)(O)C(C)C)NCC1(C(C)(C)O)CN(C(c2c(C)cc(SC)o2)=O)C1 CC1(CCNC(=O)CCC2CC(NC(c3cccnn3)=O)C2)CCOC1 Cn1ccc(C(=O)NCC(O)CNC(c2ccn(CCO)c(=O)c2)=O)c(O)c1=O n1(CC(=O)NC2(CNC(C(COC)(C)C)=O)CC2)ccc2cccnc12 c1(C(=O)NCC2CN(C(C(C=CCCC)O)=O)C2)cc(F)ccc1Cl C(=O)(C(C(C)(C)C)NC(N)=O)NCC1N(C(c2n(C)ncc2C(F)(F)F)=O)CC1 C1(C(=O)NC(C)CC2CN(C(=O)C3=CCCSC3)C2)CCn2nncc2C1 c1(C(=O)NCC(C)NC(C(C2CC2)SC)=O)ccc(Cl)c2ncccc12 c1(OCCC(=O)NCC(CNC(C2(CC#C)CC2)=O)F)ccc(C)cc1C N1(C(C2N(CC)CCOC2)=O)CCC(CNC(c2conc2C(C)C)=O)C(O)C1 C1(C(=O)NC2(CNC(C(CC)O)=O)CCOCC2)CS(=O)(=O)CC(=O)N1 N1(C(COC)=O)CCOC2(CCN(C(c3cc(C)ccc3I)=O)CC2)C1 C=CCCC(C(=O)NCC1CC12CCC2)NC(=O)CN1CCNC(=O)C1 CCCCC(CCC)CN=c1cc(C)[nH]c(=NCCCc2ccc(F)cc2)[nH]1 c1(OC)cnc(C(N2CCCC(CNC(=O)Cc3nccn3C)C2)=O)c(F)c1 C1(OC)CC2CC(COc3ccc(C(N4CCN(C)CC4)=O)cc3)CC12 N1(C(C2CCC(C)CC2)=O)CCC(CNC(C2CC2C2CCCC2)=O)C12CC2 C(CCCCOC)(c1n(CCCC)nnn1)NC(C(C)C)c1cncs1 CN1CCC(CN(C(c2sccc2Br)C(=O)NCCC2(C)CC2)C)CC1 CCCC(C#N)C(=O)N1CC(NC(c2cc(OC)nn2C)=O)C(SC)C1 CCC(C)(C)C(O)C(=O)N1CC(NC(c2cccc(C)c2N)=O)C(C)C1 Cc1cc(N)c(C(N2CCC(C)C2CNC(C2CSCC(=O)N2)=O)=O)c(F)c1 c1(C(=O)NC2CCN(C(c3cc(C)n(C4CC4)n3)=O)C2)cc(O)c2sccc2c1 c1(C(=O)NC(C)CO)coc2c1CN(C(=O)CC1(O)CCOCC1)C2 c1(SC)cccc(C(=O)NCC(C)(O)CNC(C2CCC(F)(F)C2)=O)c1[N+](=O)[O-] C1(CC=C)(NC(=O)C#CC(=O)N(C)C)CCCN(c2nnc(O)s2)C1 c1(CNC2C(C)COC2)ccnc(S(C)(=O)=O)c1 C1(NC(c2cn(CC(C)C)nc2)=O)CCCN(C(=O)Cc2csc(S)n2)C1C C12(NC(c3cc(C)on3)=O)CCCN(C(=O)C(=Cc3cccnc3)F)CC1C2 C(=O)(C(CCC)CC(C)C)NC(C(=O)N(CC#C)CCF)Cc1ccco1 CN1CCCC(N=c2nc3c(cnn3C)c(NCC3CC34CCCCC4)[nH]2)C1 C(=O)(CCC(=O)N1CCCCC1c1cn(Cc2ccncn2)nn1)NC C(=O)(CC(C(C)(C)C)NC(C1COC(=O)N1C)=O)N(CCCO)CCC c1(CC(=O)NCCCC(C)NC(CCC(=O)NC)=O)coc2ccccc12 c1(C(C)C)cccc(OC(C)C(=O)NCC(C)(C)NC(C2COC(=O)N2C)=O)c1 c1(OC)ccc2cnc(N3CCC(NC(c4cc(C)on4)=O)C(C)(C)C3)nc2c1 Cc1cc(C)c(C(=O)NCC2CCC2NC(c2n[nH]cc2C(C)C)=O)c(C)c1 C(=O)(C(C)C(C)S(C)(=O)=O)NC(CC(C)C)CNC(c1nccc2occc12)=O c1(CC)cc(NC(=O)C2=CCC(NC(C3(C)CNC(=O)C3)=O)C2)cc(C)c1 C12(CNC(c3ccnc(O)c3Br)=O)CCCC1N(C(C1COC1)=O)CCC2 c1(NCC2CCN(C(c3c(CC)ccs3)=O)CC2C)ncc(C#N)cc1C C=CCC(CC(C)C)C(=O)NCc1ncccc1C(N1CC(CO)CC1(C)C)=O C12(C(C)NC(=O)CN3CCC(S(C)(=N)=O)CC3)CC3CC(CC(C3)C1)C2 C1(CC(=O)NCC(CNC(C2(COC)COC2)=O)O)Sc2ccccc2NC1=O N1(C(C(C)SC(C)C)=O)CCN(C(C2CCCCS2)=O)CC2(C)CCCC12 C(CCCN=[N+]=[N-])NC(COC1(C)CN(C(C2CCC(N(C)C)C2)=O)C1)=O C1(C(=O)NCCOC2CCC2)(CNC(COC2(C)CCCC2)=O)CC2(CC2)C1 N(C1CCCc2c1cnn2C)C1c2c(c(C)ccc2)-n2c1nnn2.C=CCOC c1(CC(=O)NCC2CN(Cc3cnc(Cl)s3)CCO2)ccc(Br)cc1F Cc1cc(C(N2CC(O)(C(C)NC(=O)CS(=O)(=O)CCO)C2)=O)c(Cl)cc1N C(=O)(CC(C(F)F)c1ccccc1)NCC(CNC(c1c(C)nccc1)=O)(C)O N1(C(C(C)c2cccs2)=O)CCC(C2CC2)(CNC(=O)C2=CCCCC2)C1 c1(C(=O)NCC(C)(O)CNC(=O)CCN2CCCC2=O)ccc2ncsc2c1 C(=O)(C#CC1CCCCO1)NC(CCNC(c1cn(CC)nc1)=O)(C)C CC1(NC(C2COCCC2NC(c2cc(C3CC3)no2)=O)=O)CS(=O)(=O)C1 c1(C(N2CCC(NC(C3C4COCC34)=O)CC2)=O)cc2cc(Cl)cc(Cl)c2[nH]1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C(C)CC(=O)N1CC(C2CCCC2)C1)(C)C N1(C(C2(C)CCN(C(C3CCCCS3)=O)C2)=O)CCN(CCO)C(=O)C1 N1(C(CCCC)C(=O)NCCC2(C)CC2)CCC(S(=O)(=O)C(C)C)CC1 C1(OC)(CNC(=O)CC2CCOC2)CN(C(=O)C(C2CCCO2)C2CC2)C1 CC(C)CCC(=O)N1CC(C)CC1C(=O)NCC1CC(CN(C)C)C1 C1(NC(c2coc(Cl)n2)=O)CC(F)CN(C(=O)C=Cc2ccncn2)C1 c1(CC(N2CC(CCNC(=O)CN(C3CC3)CC)(OC)C2)=O)nncnc1O C(=O)(C(CCc1nn[nH]n1)NC(=O)CN(C)C)NC(CC#C)C c1(C2N(C(=O)CC3CCCN(Cc4csc(Cl)c4)C3)CCC2)ccc(F)cc1F c1(NCC(CCC)OC)cc(N2CC3CC2CN3C(C)C)nc(C(C)C)n1 CCCC(CCC)CC(=O)N1CC(O)CC1CNC(c1cc2c(s1)CCCC2)=O C1(C(=O)NCC2(COC)CCCN2C(C2CCCCCC2)=O)NC(=O)C2CCC12 C12(C(=O)NC(C)C(F)(F)F)CC(CO)(CN1C(C1CCC(N(C)C)C1)=O)C2 CC(CC(N)=O)N=c1nc(N2CC3CCC2C3)c2c([nH]1)CCCC2 C1(C(=O)NCC(C(C)(C)C)O)Cc2nccnc2CN1C(c1cccnc1Cl)=O N1(C(C2C3CN(C(CSCC)=O)CC32)=O)CCn2ncnc2C1 C(=O)(CCC(=O)NCC1CC1NC(=O)CS(=O)(=O)NC1CC1)NCC c1(C(N2C3CC(NC(COCC#C)=O)C3CC2)=O)c(C)nn2cc(C)cnc12 N1(C(C2CC(=C)C2)=O)CCC2CN(C(=O)C(O)C(F)F)CCC12 Cc1cccc(Br)c1C(C(N1C2CCC1C(CO)C2)=O)C1CCCC1 c1(C(=O)NCCC2CC(C(=O)NC(C(C)(C)OC)C)C2)cc2cccnc2[nH]1 C#CCC(CC(F)F)C(=O)NC(CC(=O)NC1(C(C)C)CC1)C(C)(C)C CC1(NC(c2ccc(F)cc2)=O)CCN(C(C2(CCC(F)(F)F)CC2)=O)C1 n1(CC)c(=O)oc2cc(S(=O)(=O)N3CCCC3c3c(C)nn(C)c3C)ccc12 c1(C(N2CC(C)CC(OC)C2)=O)ccc2c(n1)CN(C(=O)CSC)CC2 CC1CCN(C(c2ccnn2C2CCOCC2)=O)CCN1C(=O)CC(C)(C)F N1(C(C2C(C(=C)C)OCC2)=O)CC2CC(C1)CN(C(=O)C(C)OC)C2 C(=O)(CC1OC(=O)c2ccccc21)N1CCC(CNC(CSC(C)C)=O)C1 C1(C(=O)NC(CNC(CC(C)OC)=O)Cc2ccccc2)CCCC1(C)C C1(C(=O)NC(C#CCC)(C)C)CN(C(c2cc(C)nc(O)c2)=O)CC1(F)F CC1CCCC1C(=O)NCC1CCN1C(=O)C(C1CCC(=O)N1)C O=C(C1=C(CC)OCCS1)NC12CCCCC1N(C(c1cc(C3CC3)on1)=O)CC2 c1(C(=O)NC2CC(C)CN(C(c3cnns3)=O)C2)ccc2c(=O)ccoc2c1 c1(CNC2C(C(N3CCn4cccc4C3)=O)C2)c(Cl)cc(Cl)nc1Cl CC(O)(C(=O)N1CCCC1c1cn(Cc2ccc(F)c(F)c2)nn1)C(F)(F)F c1(CSC)nc(-c2cnn(C(C)C)c2Br)n(C(c2ccncc2)C)n1 C(=O)(C(C)CC(=O)NC(C1CCN(C(=O)CCNS(C)(=O)=O)C1)C)OC c1(NCc2c(CCC)cccc2)c(Cl)ccc2c(C)ccnc12 C(C)(C(C(=O)NC1CC1(c1ccccc1)C)C(C)C)OC C(=O)(CCC(=O)N1CCC(NC(=O)CCC=CC(C)C)C1C(C)C)NCCC c1(C(=O)NC2(CNC(C3CC(=C)C3)=O)CCCCC2)ccc2c(c1)CCC2(C)C c1(N(C)CC2CCN(C(C3(O)CC(C)(C)C3)=O)C2)nc2ccccc2o1 c1(C(=O)NCC(C)NC(=O)C(C)(C)CNC(=O)OC)ccc(CO)cn1 CC1CCN2N=C(C(=O)NC3(CNC(c4ccc(Cl)[nH]4)=O)CCC3)NC2=N1 C1(C(=O)NC(CNC(C2(O)COC2)=O)C2CC2)C2CCC1(c1cncs1)C2 N1(C(Cc2cn(C(C)C)nc2)=O)CC(NC(=O)CCc2ccn(C)n2)C2(CC2)C1 c1(NCC)nnccc1C(=O)NCCN(C(=O)CC1CCCN(C(C)=O)C1)C c1(C(N2C(C)CCC(NC(C3ON=C(CC)C3)=O)C2)=O)cnn2ncccc12 c1(COC)cncc(C(N2CCCCC2C(C)(C)NC(c2csc(Cl)n2)=O)=O)c1 Cc1ccc(Br)cc1CN1CC2C(C(=O)Nc3cnc(Cl)c(C)c3)C2C1 C1(CC)CCCC1(C)C(=O)NC1CC(NC(c2ccn(-c3ccncc3)n2)=O)C1 CCCCC(C)N(C(C(=O)NCC)C1CC1Cl)C CC1(O)CCN(C(C2CC(CCNC(C3C4(CC4)C34CC4)=O)C2)=O)CC1 N1(C(c2c(C(C)(C)C)cccn2)=O)CCC2(CCCN2C(C2C3COCC23)=O)C1 C1(CC)(NC(c2ccc(OC)nc2C)=O)CCN(C(=O)C(O)C(F)(F)F)CC1 C1(C(N2CC(C)N(C(C3CN(S(N)(=O)=O)C3)=O)CC2)=O)CCc2ncccc2C1 N1(C(C(C)=C2CC2)=O)CCC(OC2CCN(C(c3ccc(F)cc3)=O)CC2)CC1 C1(c2n(-c3cc(F)ncc3)nc(CSC3CCCC3)n2)CC2(CO1)CC(F)(F)C2 c1(CNC(C(C)SC(F)(F)F)=O)cnn2c1CN(CC#Cc1ccccc1)CC2 C1(C(=O)NC(C)(C)CNC(c2ccc(Br)cc2N)=O)CCc2cncn2C1 S(=O)(=O)(c1cccc(Cl)c1)N1CCC(F)(CNC(C(C(C)C)O)=O)CC1 CC1CCCN(C(c2cc(CNC(=O)CC3(C)OCCO3)cs2)=O)C1 C1(C(N(CCNC(C2(C(=O)OCC)CC23CC3)=O)C(C)C)=O)CCC=CCCC1 Cn1nc(C(N2CCC(CNC(c3nc(C4CC4)cs3)=O)C2)=O)c(C(F)(F)F)c1Cl C(C(O)C(=O)NCCC(C)NC(=O)C(C)(C)n1ccc(C)n1)=CC C1(NC(C(CC)OC)=O)CC2CCCC(C1)N2C(c1[nH]cnc1C#N)=O N1(C(c2cc(COC)on2)=O)CC2CCC1CN2C(C1OC2CCCCC2C1C)=O C1(NC(C2CC=CC2)=O)CCC2(CC1)CN(C(=O)C(O)C(F)(F)F)CCO2 c1(NC(C(N2C(C=C)COCC2)c2ccc(CC)cc2)=O)c(C)cc(C)cc1C c1(C(N(C)CC2CCN(C(C3CNC(=O)C3)=O)CC2)=O)n[nH]c2c1CCC2 c1(OC)nc(C)ncc1C(=O)NCC1(F)CCN(C(=O)C=CSC)CC1 N1(C(C2CCOC(C)C2)=O)CCN(CCCNC(C2(C(=O)NC)CC2)=O)CC1 C1(C(=O)Nc2ccc(N3CCN(C)CC3)nc2)CC12CCN(Cc1ccc[nH]1)C2 C1(CC(=O)NC2CC(C)C2)CCN(C(C23CCC(C2)C3)=O)C1(C)C N1(C(c2cnc(C#N)s2)=O)CCCC2(CCCN2C(=O)CSCc2ncc[nH]2)C1 N1(C(C(C)OCCC#C)=O)CC2(CCCN(C(C3CCCCN3C(C)=O)=O)C2)C1 c1(CC)cc(C(=O)N(C)CCC2CCN(C(c3csnc3C)=O)CC2)cc(O)n1 C1(CC(=O)NCCCN(C)C(c2ccnc(OC(F)F)c2)=O)CCOC(CF)C1 C(C(F)(C(=O)NC1CCCCC1(C)C)C(C)C)NC(c1cc(C)oc1C)=O Cc1cc(C)c(C=CC(=O)NCC2CCN2C(C2CN(C)C2)=O)cc1C c1(C(=O)NCC(CNC(c2cnc(N(C)C)s2)=O)OC)cc(Cl)c(F)c(Cl)c1 C(=O)(C1=COCCC1)N1C2C(CNC(=O)CC3CCC4CC4C3)C(C2)C1 C1(C(=O)N(C)CC2COCCO2)(NC(c2n(CC)nnc2)=O)CCCC1C C1(NC(=O)NC2C(CC)COC2)CC12CCc1cc(Br)ccc12 c1(OC)c[nH]c(C(=O)N(C2CCN(C(=O)CC3(C)CC3(Cl)Cl)C2)C)cc1=O CCC(C)CCC(=O)NC1(C)CCN(C(c2cc(OC(F)F)n(C)n2)=O)CC1 CCCC(C)CC(=O)NCC1CN(C(c2c(C)noc2C(F)F)=O)CCO1 C(=O)(C(C#N)C(C)C)N(CC(=O)Nc1cccc(CCO)c1)CCOC C1(NC(c2c(C)cns2)=O)CCN(C(=O)C(C)(C)C2CCCO2)CC1 N1(C(C(C(C)C)F)=O)CCC2(C1)CN(C(c1cnc(C(N)=O)s1)=O)CCO2 C1(CC(=O)NCc2nnnn2-c2ccccc2)CCCCC1O c1(C(C(=O)OC)NC(=O)C(c2cccc(Cl)c2)O)cc(C)cc(C)c1 C(=O)(C1=CCC(C)CC1)NCCC1CCC(NC(c2cc(C)ns2)=O)C1 c1(C(=O)NC(CCOC)CNC(c2nc(C)ccc2C)=O)snc2ccccc12 CC(CF)CC(=O)N(C)CCN(C(=O)Cc1cccc(OCC#N)c1)C N1(C(=O)NCc2nc3c([nH]2)CCCC3)c2ccncc2N2CCC1C2 CC(CC(=O)N1CCCC1CN(C)Cc1nnc(C2CC2)o1)CC(C)(C)C c1(C(N2CCC(N(C(c3cc(C)cc(C)n3)=O)CC)C2)=O)ccc(S(C)=O)cc1 c1(C(N(C)CC2CCN(C(CNS(CC)(=O)=O)=O)C2)=O)c(Cl)ccc(C)c1N CCCS(=O)(=O)C(C)C(=O)NCCC1=CCN(C(=O)CSc2nncn2C)CC1 CC1CCN(C(C2CC(F)(CO)C2)=O)CCN1C(=O)CSCc1ccccc1 c1(C(N2C(CN(C(=O)CC3CSCCS3)C)CCC2)=O)ccc(F)s1 C1(C(=O)N)C=CC(CC2(CNC(c3cnco3)=O)CC2)C1.N1(C2CCC2)CCOCC1 Cc1nn(CC(=O)NC(C)CC2CN(C(=O)CC3COCCO3)C2)c(=O)n1C Cc1ncncc1C(=O)NC1CC(C)(NC(=O)CNc2ccccc2Cl)C1 N1(C(C(COC)O)=O)CCC(CNC(c2sccc2CN(C)C)=O)C(F)(F)C1 c1(C(N2C(CCNC(c3c(Cl)cc(C)s3)=O)CSCC2)=O)cnn2ccsc12 C1(C)(N(C)CC)CCN(C(=O)CN(C(=O)CCCC2CC2C)CC)C1 N1(C(c2c(C)noc2)=O)CC(C(=O)N(C)Cc2cnn(C)c2)C(C)(C)C1 C(=O)(C1=CCCOC1)NC(C)(CNC(c1ccnc(CO)c1)=O)C1CCC1 CC(CC(F)(F)F)C(=O)NCC1CCCN(C(=O)C(C)(O)c2ccccn2)CC1 N1(C(c2cc(OC)c(O)nc2)=O)CCC(C2CC2NC(c2cocc2C)=O)CC1 C=CCC(CC)C(=O)N(C(C)(C(=O)NCCCc1cnn(C)c1)C1CC1)C C1(C(N(CCC)CCNC(c2cnc(C)cc2Cl)=O)=O)CC(C(C)=NO)C1(C)C CC1CC(C(=O)NC(C)CC(N2C3CCC2COC3)=O)=NO1 N1(C(=O)CC2CCCCO2)CC2CN(C(c3nccs3)=O)C2C1 C1(NC(=O)NCC2CCC(C)(CC)O2)CCC(C2CC2)C1 Cc1c(C(=O)NC23CCC(CC2NC(=O)Cc2csc(=N)[nH]2)C3)cccc1Cl c1(-c2cn(COC)nc2)c[nH]c2ccc(C(=O)Nc3cc(F)c(C)cn3)cc12 C1(NC(c2n(CC)cnn2)=O)CCCCCN(C(c2snnc2C)=O)C1 N1(C(C2CC(C)(F)C2)=O)CCC(CO)C(NC(c2nc(Br)c[nH]2)=O)C1 C(CCSC)(C(=O)NC1CCCC(C(C)(C)C)C1)NS(CC)(=O)=O N1(C(c2cc(SC)oc2)=O)CCOC(C(=O)N(C)Cc2nncn2C)CC1 c1(OC)cc(C(=O)NCCOCCNC(C2CCCSC2)=O)[nH]n1 C(=O)(C(CCSC)NC(c1cc(C(C)C)[nH]n1)=O)N1CC(C(=O)OC)C1 c1(C(=O)NC2C(NC(c3c(C)ccc(OC)n3)=O)CC2)cccc2ccnn12 C=Cc1ccc(C(=O)NC2COCCN(C(c3cncc(N(C)C)c3)=O)C2)cc1 CCC(C)(CO)C(=O)N1CCC(OC2CN(C(=O)CC3CCC(=O)N3C)C2)CC1 Cc1cnc(CNC(C23CC(CN2C2CC2)C3)=O)nc1 c1(N2CCN(C)C(CNC(C3CCCNS3(=O)=O)=O)C2)nc2cccc(F)c2o1 c1(C(C)NC(=O)Cc2cccs2)ccc(CNC(c2ncn(C)n2)=O)cc1 c1(C(=O)NCC(C)(C2CC2)NC(C2C(C)=C2)=O)cnc(Cl)c(C2CC2)c1 N1(C(C2CC(C)OC2)=O)CCC(Nc2ccncn2)CC1C CC(CN(C)C)CC(=O)N1CC2(NC(=O)CC3CC4C=CC3C4)CC1C2 C1(c2nc(C(C)C)on2)CCC(C)CN1C(C12CCC(CC1)CC2)=O N1(C(C(C)CF)=O)CC2CC2(CNC(c2cn(C)nc2-c2cccs2)=O)C1 c1(C2C(C(=O)NC(CC=C)CNC(=O)C(C)=C(C)C)C2)cccc(OC)c1 c1(NC(=O)OC(C)(C)C)nn2ccccc2c1SCC(N1CCCC(Br)SS1)=O c1(C(N2CC(C)(c3nn[nH]n3)OCC2)=O)ccc2c(c1)CCCNC2 C(CC(C(=O)N(C)CCN(C)C1CC1)NC(=O)CSC(F)(F)F)=CC CC(C)CC(C(=O)N(C1CC2CC2C1)C)ONC(C1C(C#N)C1(C)C)=O CC(C)C(CNC(c1cnn(CCF)c1)=O)NC(C1(C(F)F)CCCC1)=O c1(C(=O)NC2C(CO)CCN(C(CC=CCC)=O)C2)ccc2nnc(C)n2c1 N1(C(C(c2ccccc2)C)=O)CCC(C)(NC(C2CC3(CC3)C2)=O)C1 C#CC1(C)CCCN(C(C2CN(C(=O)C(CC)=Cc3cn[nH]c3)CCO2)=O)C1 C(C)(CSC)(C(=O)NCC1CCC(CO)CC1)NC(COc1ccn(C)n1)=O c1(C(=O)NC2C(NC(c3nccc(CC)c3)=O)COCC2)cc(C)n(C)c(=O)c1 Cc1cncc(C2(NC(C34CC(CO)(C3)C4)=O)CC2)c1.c12ccc(cc1)[nH]c2=O c1(C(=O)OC(C)(C)C)ccc(C2CCCN(CC3CC3(C)C)C2)cc1 C(=O)(C1CCCc2nccn21)NC1C(CNC(C(C)(C)CF)=O)C1 Cc1cc(C#N)ccc1C(N1CCC(C)(CCNC(=O)C(C)CF)C1)=O C1(C(N2CC(CNC(C(CCOC)C)=O)OCC2)=O)CN2CCN1C(C)C2 C(c1cnccn1)=CC(=O)NCC(CCNC(CC1CC(=C)C1)=O)OC C1(CNC(C(F)=C(C)C)=O)COCCN1C(=O)Cc1nnc(-c2ccccc2)o1 c1(CC)ncc(C(=O)NCC2(C(F)F)CCN(C(=O)C(C)(O)COC)C2)c(C)n1 C(N=c1ccn(-c2ncccc2F)[nH]1)(c1c(Br)n[nH]c1Br)c1n(C(C)C)nnn1 CC1CN(C(c2cn(C)cn2)=O)CC(CCNC(=O)Cc2sc(O)nc2O)O1 Cc1nc(=N)[nH]cc1C(=O)NCC1(O)CCN(C(=O)Cc2csc(NC=O)n2)C1 c1(CN2C(COC)C(C)C2)cn2cccnc2n1.C12CCCN(C1)c1nnc2s1 N1(C(C(C(C)C)CO)=O)CC(NC(C2CCC(O)CC2)=O)CC2(CCC2)C1 CCC(c1ccc(OC)cc1)=CC(=O)NC(C1CCCN1C(=O)CC(C)OC)C c1(CC)nc(C)n(C)c1C(=O)NCC(CO)NC(c1ncc(C(F)F)s1)=O C(=O)(C1=NOC2COCC12)N(C(C(=O)c1cccs1)Sc1ccsc1C#N)CC c1(CC(=O)NCC(C)NC(Cc2nc(CC)sc2)=O)cccc(OCC(C)C)c1 c1(CC(=O)Nc2c(CCN(C)C)cccc2)csc2cccc(F)c12 C1(S(N)(=O)=O)(C(N2CCC(n3cc(CCS(=O)(=O)N(C)C)nn3)C2)=O)CC1 c1(C(N2CC(NC(C(C)CN(C)C)=O)C3(C2)CC3)=O)c(N)cc(Cl)cc1Cl N1(C(CN(CCC)C)=O)CCC(O)(CN(C(=O)Cc2cc[nH]n2)C)CC1 C1(O)(CNC(c2cc(SC)ncc2)=O)CCCN(C(=O)C(F)(F)CC2CC2)C1 Cc1cc(C(=O)N(CC(C)O)CCNC(c2coc(-c3ccsc3)c2)=O)n(C)n1 c1(SC)cc(C(N2CCC2CNC(=O)Cn2nnc(=O)[nH]2)=O)c(C)o1 C(C(C(C)C)C(C)C)OC.c12ccc(c(F)c1)-n1cc(nn1)CCCNC2=O c1(C(N2CCC(C)(NC(=O)C=Cc3cccc(F)c3)C2)=O)ccc(P(C)(C)=O)o1 C(=O)(CCS(C)(=O)=O)NCCCC(C)NC(C12CC(CF)(CO1)C2)=O C1(C(=O)NC2CN(CCC)C2)CCN(C(C2CCC2C)=O)CC1C CC(C)CCCCCC(=O)N1CCC(NC(=O)C(C)CC(F)(F)F)C(F)(F)CC1 S(=O)(=O)(c1c(Br)nc(C)cc1Br)NCC(CCCC)CC CN1CCC2CCN(C(C3CC4CN(C(=O)CC5CC(F)(F)C5)CC4C3)=O)C2C1 c1(C(N2CCC(CCNC(C3CCC3(F)F)=O)C2)=O)cccc(C2(F)COC2)c1 c1(CN(C)CC2CCN(C(C3N(C(C)=O)CCC3)=O)CC2)cc2cc[nH]c2cn1 C(=O)(C1=CC2C=CC1C2)NCCC1CN(C(CCN(CC)CC)=O)CC(C)O1 N1(C(c2n(CCN(C)C)ncc2)=O)CCC(NC(=O)CCS(C)=O)C(CO)CC1 C1(CCC)(NC(=O)Cc2csc(C)c2)CCN(C(=O)CCOC(C)C)CC1 N1(CC(C)C)N=C(C(=O)NC2CCCC(NC(=O)CO)C2)CCC1=O c1(C(=O)NC(CC2CN(C(c3c(C)scn3)=O)C2)C)cc2c(C)cccn2c1 Cc1nc(CC(=O)NCC2(NC(=O)COC3CCCC3)CC2)c(Cl)s1.C1CC1 c1(C(=O)OC(C(=O)Nc2c(OC)cccc2)C)cc2n(c(=O)c1)CCS2 C12(NC(c3cc(F)c(F)c(F)c3)=O)CCC(CC1)N(C(=O)CCc1nccs1)C2 C1(CNC(C(C)=C2CCCC2)=O)CC2CC(C1)N(C(=O)C=Cc1sccc1C)C2 Cc1ccc(C(=O)NCC2(O)CC(NC(=O)C(C)n3ccnc3)C2)c(Cl)c1 C1(NC(=O)CSc2nncs2)CC2CCC1CC2NC(C1(F)CCCOC1)=O Cc1c(Br)noc1C(=O)NC1COCC1NC(c1ccnc(C2CC2)n1)=O CCC(C)C(O)C(=O)NC1(CNC(c2ccc(C(N)=O)c(Cl)c2)=O)CC1 Cc1cnc(CC(=O)NCCC(C)NC(c2c[nH]cc2C2CC2)=O)s1 C1(C(=O)NC(C(=O)NC2(C)C(C)(C)C2)C2CCCC2)C=CC=CC=C1 c1(C(N(CCC)CCNC(=O)CN2CCC(OC)C2)=O)ccc(N)c(F)n1 C1(NC(CCCCNC(C)=O)=O)CCN(C(c2ncc(C)cc2C)=O)CC1O c1(C2(C(=O)NCC3(CCNC(=O)CC4CCCOC4)CC3)CC2)cccc(Cl)c1 C1(C2CC2)(CNC(CC2(CSC)CC2)=O)CCN(C(c2ccnc(OC)c2)=O)C1 C1(C(N2C(CCC)CN(C(=O)C(F)(F)CN(C)C)CC2)=O)OCCOC12CCC2 c1(C(N2CCC(NC(C3CN(CC(F)(F)F)C3)=O)C2)=O)cn2ccnc2s1 N1(C(c2scc(CNC(C(=O)NCC3CC3)=O)c2)=O)CC2(C1)CC1(CCC1)C2 c1(-n2c(C(C3=CCSC3)NC(c3ccccc3Cl)C)nnn2)ccc(F)cc1 C=C(C)CCN=c1nc(N2CCC(OCCF)C2)c2c(ncn2CC)[nH]1 Cc1cc(C(=O)NCC(C)N(C)C(c2cc(C3CC3)[nH]n2)=O)cc(Br)c1 Cn1c(CNC(=O)C(C)(C)c2ccc(Br)s2)nc2cc(Cl)ccc12 c1(C(=O)NCC(C)(O)C(=O)O)c[nH]c2c(F)cc(F)cc2c1=O n1(CC(=O)NCCC(C)NC(CC2(NC)COC2)=O)cnc([N+](=O)[O-])c1 c1(CCNC(=O)NC(C2CCS(=O)(=O)N2)=O)nccc(O)n1 Cc1cc(CO)c(C)cc1NC1(c2nnnn2C2COC2)COCCC1C C1(CNC(=O)CC2CCC2)CN2CCCCC2CN1C(C1CC2C=CC1CC2)=O Cc1csc2ncc(C(=O)NC(C)CNC(C3CCS(=O)(=O)N3)=O)c(=O)n12 c1(C(=O)NC(c2ccc(OCC=C)cc2)(C)C)cc(C(F)(F)F)cc(OC)n1 Cn1nc(C(F)(F)F)c(I)c1CNC(C1OC2CCC1CC2)=O c12cn(nn1)CN(C(C)C)CCNC2=O.C1(NC(c2cn[nH]c2)=O)CNC(=O)O1 C1(CCNC(c2n[nH]cc2Br)=O)(NC(c2ccsn2)=O)CCCC1 N1(C(C(C(C)C)n2cnnn2)=O)CCC(C)N(C(C2CC(C)(C)CO2)=O)CC1 N1(C(c2ncc(NC)nc2)=O)CCC(NC(=O)Cn2nnc(C3CC3)n2)C(O)C1 N1(C(C2C(CNC(CCOCC#C)=O)CCCC2)=O)CC2CC3CC2C1C3 c1(C(N2C(CCNC(=O)CC3(CO)CC3)CC(F)(F)C2)=O)ccc2ncnn2c1 CC1(NC(=O)CCCc2ccccn2)CC(NC(=O)CCCN2CCCC2)C1 CC(C)(C(=O)N1C2CCC1CC(NC(C1(F)CCCC1)=O)C2)C1=CCSCC1 C1(CNC(C2CC2C(F)(F)F)=O)CN(C(=O)Cc2cscn2)CCC1C(F)(F)F c1(C(N2CC3CN(Cc4cccc(I)c4F)C3C2)=O)c(F)cc(F)cc1Cl C1(C(C)NC(c2c(C)nc[nH]2)=O)CN(C(C2CC2CN(C)C)=O)CCO1 CC1CN(C(=O)C=C2CCSCC2)CC(C)C1NC(=O)CC12CCC(CC1)C2 C#Cc1cnn(C)c1C(N1CCC(NC(c2cocn2)=O)C1)=O c1(OC)cc(CNc2cc(NC3CC(OC)CN3C)ncn2)ncn1 C1(C(=O)NC(C)Cc2ccsc2)CC2CCN(C(C)C(C)(C)O)CC12 CCC(F)(F)CC(=O)N(CCCNC(=O)CCc1cc(OC)no1)C N1(C(C)=O)CCCN(C(=O)C(C)CN(C(=O)CC23CCCC2C3)C)CC1 Cc1sc2ncc(C(=O)N(CCCCN(C(=O)C(O)C(C)C)C)C)n2c1C c1(C(C)C(=O)NC(C)(C)CNC(C2CC=CCO2)=O)ccc(Br)cc1 C(CCC(C(=O)NC1CC(CN(C)C)C1)NC(=O)Cc1cncs1)OC Cc1cc(NC(C2CC2NCc2c(F)cc(F)cc2Br)=O)c([N+](=O)[O-])cc1Br N1(C(C2CC3CC3C2)C(=O)NCC=C)CC2CC(C(=O)OC)C2C1 O=C1CN(C(C2C=CCN(C(=O)C3=CCCCCC3)C2)=O)CC2(CC2)N1 C1(CNC(c2c(C)nco2)=O)C2CN(C(C3(O)CCOC3)=O)CC12 C1(C2CC2)(C(N(C2CN(C(C(CCOCC)OC)=O)C2)C)=O)CC(CC)=NO1 C1(CNC(C2(CC(=O)OC)CC2)=O)C2CCC(C2)N1C(=O)CCC(CC)OC c1(CC(N2C(CNC(C3C(C)CCCC3)=O)CCCC2)=O)ccn2cncc2c1 C1(NC(C(C)(C)C)=O)CCCN(C(=O)C(=O)NC2CCCC2N2CCNCC2)C1 c1(C(=O)NC(C(C)(C)C)C(F)(F)F)cc([N+](=O)[O-])ccc1-n1cc(CCO)nn1 c1(C(=O)OC)[nH]c(=NC(CSc2ccccc2)C2CCOC2)[nH]c(=N)c1C#N N1(C(C(COC)OC)=O)CCC2(CC(C(=O)NCc3cc(C)ncn3)C2)C1 N1(C(C(C(CC)O)(C)C)=O)CC2(CCCN(C(c3cc(C(N)=O)c[nH]3)=O)C2)C1 c1(OCC)cccc(C)c1C(=O)NCC(C)(C)COc1ccccc1Cl N1(C(C2CC2C2(C)COC2)=O)CCC2(CNC(=O)O2)C1.C#CCC1C(=O)N1 Cn1cc(CO)c(CNC(=O)C(C)(C)NC(C2C3COCC23)=O)n1 C1(NC(C=CS(CC)(=O)=O)=O)CCC2CN(c3nc(C(C)C)nc(=N)[nH]3)CC2C1 c1(CC)ncnc(CC)c1C(=O)NC1CN(C(C23CC4CC2C3C4)=O)C1 c1(C(C)=O)ccc(C(N2CC3(CCC3NC(=O)CCc3ccsc3)C2)=O)c(C)c1 C1(C(=O)NC(CN(C(c2cc(SC)oc2C)=O)CC)C)CC2CCC(C1)O2 c1(OCCC)ccc(-c2ccc(C3CC(=O)N(C)C3=O)cc2)c(C)n1 N1(C(CCNC(=O)OC)=O)CCCCC1CNC(=O)C(C)c1cccs1 CCCC(CCCNC(c1ccn(CCC)n1)=O)NC(c1ccc(N)cc1Cl)=O c1(C(N2CC(CNC(CC#N)=O)OCCC2)=O)cc([N+](=O)[O-])ccc1OC(F)F CC(C)CC(C)CC(=O)N(C1CCCCN(C(c2cncc(F)c2Cl)=O)C1)C c1(C(N(CCC)CCNC(=O)C(O)C(C)OC)=O)c([N+](=O)[O-])ccc(C)c1C c1(C(=O)NC(C(CC)CC)C)cc(F)ccc1S(C)(=O)=O C1(CNC(C2C(C=C)C2)=O)CN(C(c2ccc(CCC=C)cc2)=O)CC12CCC2 C(=O)(C(CCC(N)=O)n1cnnn1)N(C1CCN(C(=O)C2=CCCS2)CC1)C C1(C#N)(C(=O)NCC2N(C(Cn3nnc(C)n3)=O)CC(O)C2)CC12CCOCC2 c1(C2CN(C(CCN(C(C3CN(C(C)C)C3)=O)CC3CC3)=O)C2)nncn1C N1(C(C2(C)CC=CC2)=O)CC(NC(c2cc(F)c[nH]2)=O)C(c2ccccc2F)C1 N1(C(C(c2n(CCC)ccn2)(F)F)=O)CCC2CN(C(=O)C(OC)OC)CC12 CONC(=O)C(=O)NCC(C)N(C(=O)C(O)Cc1ccccc1)C C(=O)(C(C)C(C)(F)F)N1CC(C(C)NC(c2ncc(N(C)C)cn2)=O)C1 CC1(C)OC2(C(N3CCCC(CCNC(=O)CCCN=[N+]=[N-])CC3)=O)CC1C2 Cc1cccc(CC(=O)NCCC2(C(=O)NCCC3CCC(C)O3)CC2)c1 C(=O)(C(F)CC(C)(C)NC(c1cccnc1O)=O)NCc1cc(C)ncc1 c1(OC)ccc(C(N2CCCC(F)CC2)C(=O)NCCN2CCOCC2)cc1SC C1(C(=O)NC(CO)C(C)NC(c2cocc2C)=O)(CC)CCCC1 Cc1cc(Cl)cnc1C(N1CCCC(CNC(c2ccc(F)cc2)=O)CC1)=O N1(C(C2N(C(c3c(OCC)ccc(Br)c3)=O)C3C(C2)C3)=O)CCN2CCCC2C1 C1(C(=O)NCC(C(C)C)NC(c2c(CC)n(C)cc2)=O)CCC(N=[N+]=[N-])CC1 N#Cc1cc(C(=O)NCCCCCn2cc(-c3ccc(Cl)cn3)nn2)co1 C1(C(=O)NCCC2CCCC(C)C2)CN(C(C2CCC3(CC3)C2)=O)CC1(F)F C(=O)(C1Cc2ccc(Cl)cc21)N(C)CCO c1(C2(Nc3nccc(N4CC(c5scc(C)n5)OCC4)n3)CC2)cccnc1Cl c1(C(=O)NC(C2CN(C(c3cnsc3)=O)CCO2)C)ccc2c(c1)CC2 C1(CC(=O)N(C(CC)CO)C)C(NC(c2c[nH]nc2C)=O)CC1O CC1CCN(C(=O)CCCC2(C)N=N2)CC1CNC(=O)C=Cc1c[nH]cn1 c1(CC(N2CC(O)CC(N(C(=O)C=CC3CC3)C)C2)=O)coc2cc(Cl)ccc12 N1(C(C(c2nc(C)sc2)=O)=O)CC2(CCC2NC(c2cnc3sccn23)=O)C1 CC1(C)CCCCC1C(=O)NC1CCC12CN(C(c1c(N)cccc1F)=O)C2 C1(NC(CC(C)C)=O)(CNC(c2n[nH]cc2C(C)C)=O)CC2CCC1CC2 C1(NC(C2C(C)C2C)=O)CCN(C(c2cc3n(n2)CCNC3=O)=O)CC(C)(C)C1 C(C(CC)CC)N(C(=O)CCN(C(=O)C(C)CC1CCC1)CCO)CCC S(=O)(=O)(c1cc(Br)ccc1OC)N1C(C(N(CC=C)C2CC2)=O)C2CCC1C2 N1(C2CCN(CC=C)C2=O)CC=C(CNC(c2cnoc2CC)=O)CC1 c1(C(N2CCC(n3cc(CNC(c4ccncn4)=O)nn3)C2)=O)cc(Cl)c(Cl)s1 CCC(CN(C)C)CC(=O)NC1CC(F)(CNC(=O)CSC2CCCCO2)C1 N1(C(C2=NOC(CNC(C3(CF)CC(=O)C3)=O)C2)=O)CCC2=C(CCCC2)C1 N1(C(COCC(=O)OC)=O)CCOC2(C1)CN(C(=O)CC1CCCC(C)C1)C2 S(=O)(=O)(c1cc(C(=O)NCC(C)(C2CC2)NC(=O)CCC2OCCO2)co1)NC c1(C(N(CC(CN(C(=O)Cc2nncn2C)C)O)C)=O)cccnn1 C(=O)(N=S(C)(=O)c1ccccc1C)c1c(OC)cc(C)c(OC)c1 CCC(CC(=O)N(C1CCCCC1NC(c1ccc2n[nH]cc2n1)=O)C)C(C)C C(=O)(CC(C)n1cc(Br)cn1)NCCC1CC(NC(COCCOC)=O)C1 C1(C(N2CCN(C(C(CCC)N(C)C)=O)CC2)=O)CCCN(S(N)(=O)=O)C1 N1(C(C(C2CCC2)OC)=O)CCC(CNC(=O)C(=O)N=S(C)(C)=O)C(F)(F)CC1 Cc1nocc1C(=O)NC(C1CCN(C(C2CCC(N(C)C)C2)=O)C1)(C)C c1(C(=O)NCCNC(c2c(OC)cccc2F)=O)cnc2c(C)nsc2c1 C1(NC(C2N(CC)C(=O)CC2)=O)CCN(C(c2cn(C)nc2C)=O)C12CCCC2 CCC(C)CCCC(=O)NCC(C1CC1)N(C(=O)Cc1c(C)nn(CC)c1C)C C1(C(C)C(=O)NCC(C)N(C)C)CCN(C(C2CCC2C#N)=O)CC1 C1(OC)CC(CNC(=O)C(O)Cc2ccccc2)N(C(=O)Cn2ccc(C)n2)C1 c1(C(N(CC(C)NC(=O)C(c2cnccn2)C)C)=O)ccc(OC(F)F)cc1F N1(C(c2c(OC)nn(C)c2)=O)CCC(NC(C2CCCCC2)=O)C(C)C1 C1(NC(c2c(C)cn(C)c2)=O)CC(O)CN(C(=O)CCc2ccc(F)cc2)C1 Cc1nc2[nH][nH]cc-2c(=Nc2ccc(CC(=O)NCCF)cn2)n1 C(=O)(C1CC=Cc2ccccc21)NCCC(C)NC(=O)COC1(C)CCOCC1 Cc1n[nH]c(C)c1C(C)CC(=O)NCC1CCN1C(=O)C1=CCCS1 N1(C(c2c(OC)cc(F)cc2)=O)C(C)CC2CN(C(=O)CCCCC(C)C)CC12 C1(C(N2CC(c3cn(CC(C4CC4)OC)nn3)C2)=O)CCCC12CC2 C(=O)(C(C)S(C)(=O)=O)N1CC(C)C(CNC(C2COC(=O)O2)=O)C1 N1(C(c2c(C)cc(F)s2)=O)CCC2(CNC(=O)CCc3cncs3)CCCCC12 c1(OC)ccc(C(=O)NC(C2(O)CCN(C(C3(CF)COC3)=O)C2)C)c(OC)n1 c1(OCC(N2CC(O)(CNC(c3cc(SC)oc3C)=O)C2)=O)ccc(C#N)cc1 c1(COC)cc(C(=O)NC(CNC(=O)CCN2CCOCC2)CO)n[nH]1 FC1CC(F)(F)CCC1NCc1cc2cnccc2[nH]1 C1(NC(C(C(=C)C)(C)C)=O)COC2(CCN(C(=O)CCn3cncn3)C2)C1 C1(C(=O)NC2CCCN(C(CCc3n(C)cnc3)=O)C2)Cc2cccc(F)c2O1 C1(CNC(CCCCCN(C)C)=O)CCCC2(CN(C(=O)CC3CC3(C)C)C2)O1 n1(CC(=O)NCC2C(NC(=O)C3=CCCS3)CC2)c(=O)nc(O)c2ccccc12 C1(N(C)C(C2(SC3CCC3)CC2)=O)CCCN(C(c2c(Br)cnn2C)=O)C1 c1(CC(C(=O)NCCOC)NC(C2CCC(=O)O2)=O)ccccc1Br N1(C(C(c2ccccc2)OCC)=O)CC(O)CCC1c1ccccc1 C1(C(=O)NCC2CC2C(=O)NCC(c2cn[nH]c2)C)(CC)CCC1 CC1CN(c2cc(NCCc3nnc(CO)s3)ncn2)Cc2nncn21 Cc1ccncc1CC(=O)NCC1C=CCN1C(=O)CC1(C)CCC1 Cc1nn(CC(C)C)c(C)c1CC(=O)NCC(O)CNC(=O)CC1(O)CCOC1 N1(C(C(C)N(CC)CC)=O)CC(CO)C2(C1)CN(C(C1CC3(CSC3)C1)=O)C2 N1(C(C2CC(C)(C)C2)=O)CCC2CCN(C(c3cc(F)c(O)c(Cl)c3)=O)C2C1 c1(CC)ncnc(N2CCCC(CC(=O)Nc3ccc(OC)c(Br)c3)C2)c1F c1(NC(C2C(NC(C=Cc3ccc(C)s3)=O)C2)=O)ccc2c(c1)CCCC2=O c1(OCC(=O)NC2C(NC(COCC(C)C)=O)CCC2)cccc(C(C)(C)C)c1 C1(C(=O)NCC2CCC(N(C(c3nc(C)oc3C)=O)C)CC2)COC(C)(C)CO1 c1(CC(=O)NC(CNC(CCCN(C)C)=O)C2CCC2)cc(F)ccc1Cl c1(NC(=O)NC(CC#C)COC)cc(-c2ccco2)nn1-c1ccccc1 N1(C(CCCCOCCC=C)=O)CCCC2(CCN(C(c3ncccn3)C)C2)C1 Cc1ncc(C(=O)NCCN(C(=O)CC2CCC2)CCOCCO)n1C(F)F N1(CC)C(=O)CCC1C(N1CCC(NC(c2cn(CC)cn2)=O)C1)=O CCCC(C#N)C(=O)NCCc1n[nH]cc1C(N1CCCC(CC)C1)=O N(C(=NCC1(C#N)CCCC1)NC1CCCC1)C1CC(C)OC1 c1(OC)ccc(N)c(CNC(C2(COCC(=O)NC(C)=O)CN(C(C)=O)C2)=O)c1 c1(C(=O)NCC2C3CN(C(C(CC#C)C)=O)CC32)ccc(Cl)c(Cl)c1 c1(C(=O)NC2C3(CN(C(c4c(CC)con4)=O)C3)CC2)ccc(F)c(C)c1Cl C#CC1CN(C(C)=O)CCN1C(=O)C(c1ccc(C)cc1)=O c1(C2N(C(CC3(C)CCOCC3)=O)CCCC2)cccc([N+](=O)[O-])c1 C(C(COC)CC(=O)NC(C)C(=O)NCC1(CO)CC1(C)C)OC C(CCCCC(=O)NCC1CC(NC(c2cc(C(N)=O)[nH]n2)=O)C1)OCC Cc1cc(C(=O)NCCCNC(C23CSCC2C3)=O)ncc1F c1(CNC(c2ccc(CC)[nH]2)=O)cccc(C(=O)NC2(C)CCSC2)n1 Cc1cc(C(C)C(N2CC(NC(=O)CCc3ncc[nH]3)CC(C)C2)=O)cc(F)c1 c1(C(C(=O)NCCC)N(C2CCCCC2N(C)C)C)cc(Cl)ccn1 CCS(=O)(=O)CC(=O)NC1(C(=O)NC(c2ccc(O)nc2)C)CSC1 CCC(C)C(O)C(=O)NCC1CCC(NC(=O)CC2C=CCCC2)C1 O=C1CC(C(N2CCOCC2C(=O)NCC2(CF)CCC2)=O)C2(CCC2)C1 N1(C(C(COC)(C)O)=O)CC2(CCCC(CNC(c3cc(Cl)c[nH]3)=O)O2)C1 C1(CNC(c2cnsn2)=O)CC12CCN(C(=O)CC1CCC1)CC2 Cc1cc(C)c(NC(C2CCN2C(C2CC(=O)C2(C)C)=O)=O)c(C)n1 c1(C(=O)NCC2CN(C(c3c(C)scn3)=O)C2)ccnc(CO)c1 CCC(C)(C)CCCC(=O)NC1(C)CCCN(C(c2ccc(N)c(F)n2)=O)C1 C1(CC(N2C(C(C)(C)NC(=O)Cc3ccc(Cl)s3)CCC2)=O)CC2(CCC2)CO1 C1(C(=O)NC(C(=O)OC)C(C)O)C2CC(O)C(C2)N1C(c1ccc([N+](=O)[O-])o1)=O Cc1nn(C)c(N)c1C(=O)N(C)Cc1ccccc1C(F)(F)F CC(O)CCN=c1[nH]c(N2CC34CCC3(COC4)C2)nc2c1COCC2 C1(NC(C2CC(O)(CC#C)C2)=O)CCC(O)CN(C(c2cnc(S)[nH]2)=O)C1 N1(C(=O)C(Br)Br)CCC2(CC1)CC(n1cc(-c3ncccc3Cl)nn1)CO2 CC(CC(F)(F)F)C(=O)N1CCOCC(NC(c2cc(Cl)ns2)=O)C1 C(=O)(C1CCCc2cncn21)NCC(C)N(C(C(=O)Nc1ccc(C)cc1)=O)C C1(NC(=O)C=C2CC2)CN(C(=O)Cc2cccc(F)c2)CC1C(F)(F)F c1(C(=O)NC(C)C(CO)NC(=O)C(Cl)=CCl)ccc(CCNC(N)=O)cc1 CC(C)(C)C(=O)C(=O)N1CC(CNC(=O)C(Cl)=CCl)C2CC12 C1(CC(=O)N(C2CCN(C(c3ns[nH]c3=O)=O)C2)CC#C)C=NN(C)C1=O N1(C(CCS(C)=O)=O)CCC(F)(F)C(CNC(c2cc(C(F)F)cs2)=O)C1 N1(C(c2c(C)cc(C)o2)=O)CCOC2(C1)CN(C(C13CC4CC1C3C4)=O)C2 C1(NC(c2cnc(C3CC3)o2)=O)CCN(C(C23CC(O)C2C3)=O)CC12CCC2 CCC(CCC(=O)NCC(C(C)CC)OC)NC(=O)COC1(C)CCC1 N1(C(C2CCCC(NC(c3occc3C3CC3)=O)CC2)=O)CCc2n[nH]cc2C1 C1(CNC(=NCC)NC2CCN(c3ccn(C)n3)C2)CCC(=O)N(CC)C1 C1(F)(CO)CCCN(c2nc(-c3c(Cl)cccc3Cl)cs2)C1 c1(N(C2CCN(C(=O)CC3CCCN3C)CC2)C)ncnc2ccccc12 c1(C(=O)NCC2CN(C(CS(N3CCN(C)CC3)(=O)=O)=O)C2)c(Cl)cccc1Cl c1(CC(N2C3CN(C(CC(C)C(F)F)=O)C(C3)C2)=O)c[nH]c2ccc(Cl)cc12 CC1CC(NC(=O)C=Cc2ccc(C(N)=O)o2)CCN1C(c1nc(=O)n(C)[nH]1)=O c1(OCC(=O)NC(CN(C(CC2C(C)=NNC2=O)=O)C)C)c(C)cc(Cl)cc1Cl CC(C(CO)NC(=O)Cc1csc(C2CC2)n1)NC(=O)CC1CNC(=O)C1 c1(N(CCC#N)C(=O)NCCC(F)(F)F)ccccc1OC.CO C1(C(N(CC(C)NC(C=COCC)=O)C)=O)CCN(C2CC2)S1(=O)=O C1(NC(c2c(CC)csc2)=O)(CNC(=O)C(C#N)C(C)C)CC2CCC1CC2 Cc1cc(C)c(OCC(=O)Nc2nc(-c3ccc(Cl)cc3)no2)c(Br)c1 C1(NC(C2(Br)C(C)C2C)=O)CN(C(=O)C2=NNC(=O)CC2)CC1C1CC1 CC(C(=O)N1CCC(CNC(c2coc3c2COC3)=O)C1)C(C)(F)F C1(C(CNC(COCC(C)C)=O)(C)C)CCCN1C(=O)CNS(C)(=O)=O Cc1cc(C(=O)NC2(CF)CN(C(=O)Cc3cnccc3Cl)C2)cc(C)c1N O=C1CC(CNC(=O)C(CC2CCOCC2)NC(c2cc(Cl)cs2)=O)CN1 C1(C(=O)NCC2CN(C(C)=O)CC2O)CCC(S(N)(=O)=O)CC1 N1(C(CCC(N)CC2CCCCC2)=O)CC2CCC1C1CNCC21 c1(C(=O)NCC2(CN(C(Cc3c(C)non3)=O)C)CC2)cncc2c1CCC2 c1(C(N2C(CNC(CCC(=O)NCC)=O)CCC2)=O)cc2cc(F)c(F)cc2[nH]1 C1(NC(C(C=C)(C)O)=O)CCN(C(=O)COCC(N2CCCC2)C)CCC1(F)F N1(CCOC(c2ccc(F)cc2F)=O)CCN(C(C2CCCO2)=O)C(=O)C1 N1(C(C2C(OC(C)=O)C2)=O)CCCCC(C(N2CCC(C#N)CC2)=O)C1 N1(C(CCC=C(C)C)=O)CC2CCN(C(c3cc(Br)ccc3F)=O)C2C1 N1(CCO)CCN(NC(=O)NC23CC(C(=O)OC)(C2)C3)CC1.C1C(=O)ON=C1C C1(C(C)(C)C(=O)NCC(C)(O)C2(C)CC2)CCCN(C(C2CCCS2)=O)C1 C(C(C)(C)CCOC)NC(CCN(C(C1C=CCCC1CO)=O)CC)=O C1(F)(CNC(CC(C)SC)=O)CCCN(C(c2c[nH]c(=O)cn2)=O)C1 Cc1cc(Br)c2oc(C(=O)NCC(C(C)(C)C)NC(=O)CCN(C)C)cc2c1 N1(C(c2c(CC)cco2)C(=O)NCCC#N)CCC2(CCOC2)C1 c1(C(N2CCC(CCN(C)C(C3C=CCCC3)=O)CC2)=O)cc(F)cc(F)c1 C1(CC2N(C(C(C3CC(F)(F)C3)OC)=O)CC2)COCC1C(N)=O N1(C(C2CCC(C)O2)=O)CCCC2(CCCN2C(c2cccc(O)c2F)=O)C1 N1(CC2(C(=O)OC)CCNCC2)CCOC(C(C)N)C1 CC1=C(C)CC(C(N2CCCC2(C)CCC(=O)NCCC(C)C(C)(C)C)=O)CC1 c1(SC)ncccc1C(N1CCSCC1C(=O)Nc1cccc(I)c1)=O c1(OC)ccc2c(C(N3CC4(CC(O)C4)C3)=O)n[nH]c2c1F CC(=O)C(C)CC(C)C(=O)NCC(=O)NC(C)(C)C(C)(C)CO c1(OC)c(C(=O)NCC2CC3CCC2N(C(=O)CC(C)C)C3)ccc(Cl)c1C C(CCCCCC(=O)NOC1CCOC1)NC(C(C)n1cccc1)=O CC1CN(C(C2(F)CC=CCC2)=O)CC1NCC(N1CCCC1)=O C(CCC(C)(C)C(=O)N1C(C(=O)NCC(C)(C)OC)CC1C)OC N1(c2ccnc(NCc3c(CC)con3)n2)CCC2(C)C(F)(F)C2(C)C1 c1(CCC)cc(C(=O)N(C2CCN(C(=O)C(CC)N(C)C)C2)C)[nH]n1 c1(NC)cncc(C(=O)NC(CC2CCC2)C(=O)NC(C)C(=O)N2CCCC2)c1 c1(COC)ccccc1CNC(C1CCC(C(=O)OC)C1)=O.C12(CCC1)C(=O)NC2 c1(CC(=O)NC2CC(NC(C(C3CC3)OC)=O)C2)ccc(F)cc1 C(C)(C(=O)N(C(C)CCNC(C1CCOC1)=O)C)OCCOC CCN=c1[nH]c(C)c(C(=O)NC2CN(C(=O)COc3ccc(F)cc3)CC2C)s1 c1(COC)nc(C(=O)NCC2(C(C)(C)O)CN(C(=O)CC3CC(OC)C3)C2)cs1 N1(C(CC2CC(C)C2)=O)CCCCC(NC(=O)C(c2ccnn2C)C)C1 c1(C(=O)NC(CNC(C(CC#C)O)=O)(C)C(C)C)cnc2n(c1=O)CCS2 C1(NC(C2N(CC)CCC2)=O)CC2C(NC(=O)CC3C=CS(=O)(=O)C3)C2C1 c1(C(N2C3CN(c4ncc(OC)c(C)n4)CC32)=O)c(F)ccc2c1CNCC2 C(CCS(=O)(=O)C(C)C)N1CCC(C)(NC(c2c(OCC)ccc(C)c2)=O)C1 c1(CC)cccc(C(=O)NC2CCN(C(=O)C(COC)CC)C2(C)C)c1F C(=O)(CCC(C)(C)O)NCC(C1CCCC1)NC(c1cn(CC)nc1C)=O C(=O)(C(F)C(=O)N(C)C(c1cn(Cc2cc(C)on2)nn1)C)OCC C1(C)(CNC(CN(C(CCC)=O)CC)=O)CN(C(=O)C(C)N2CCC2)C(C)(C)C1 C1(CC(=O)NCCCN(C(CCC(=O)NCC)=O)CCO)C#CCCCCC1 c1(CC(=O)N(C2CC2)CC2CCCN(C(C(CSC)O)=O)C2)ccc(F)cc1Cl n1(CC)ncnc1C(=O)NC1CC(CCNC(c2scnc2C)=O)C1 c1(CC(=O)NCC2(NC(c3ncoc3Br)=O)CC2)ccc(F)c(F)c1 C#CCC(C(=O)N1CC(O)(CNC(c2coc(C(=O)OC)n2)=O)C1)C1CC1 C1(NC(=O)CC2CC23CC3)CC2CCC(C1)N2C(C1(c2nc[nH]n2)CC1)=O N1(C(CC2C(CNC(CC3C(C)CCC3)=O)C2)=O)CCOCC1CO N1(C(C2CC(O)CN2C(c2cnn(C(F)F)c2)=O)=O)CCC(CO)C(O)C1 N1(C(c2c(CC)ncs2)=O)CC2CCCC2(NC(=O)CN2CCC(=O)NC2=O)C1 c1(CNCCN2C(C)CCC2)cc2c([nH]1)CCC2 c1(NC2CCN(c3ccccc3)C2)ccc2c(c1)OCO2 CC(C)CCCC(C)C(=O)N1CCCCC(CCC(N2CCCC2C(C)O)=O)C1 C(CC(=O)NCC(C)(C)CN(C)C)(C(F)F)NC(COCCC#C)=O c1(C(=O)NC2C3CC(NC(C(C)=C4CCC4)=O)CC32)cc(C#N)ccc1C C(C1CC1)(C1CC1)=CC(=O)N(C)CCOCCC(=O)NCCN1CC2CC2C1 C#Cc1cccc(C(=O)NC2CC(F)(CNC(=O)C(C(C)C)OC)C2)c1Cl N1(C(CC2CCN(C(=O)CC3CSCCO3)C2)=O)CCCC(F)(F)C1 c1(CC(N)C(=O)NCC2CCCN2CC(F)F)ccc(Cl)nc1 CC(C)C(C)C(CNC(=O)COC(F)(F)F)NC(c1ccccc1C(N)=O)=O c1(C(=O)NC2CCN(C(=O)CNC(c3ccncc3)=O)C2)cccnc1C1CC1 Cc1sc(O)nc1C(=O)NC(C)C(CO)NC(c1cc(Cl)c(Cl)s1)=O N1(C(CNS(CC)(=O)=O)=O)CC2CC(NC(=O)CCNC(C)=O)C2C1 c1(CC)c(C(=O)N(CCNC(=O)C(F)F)CC2CC2)cnc2cc(O)nn12 C1(COC)(NC(=O)C(C)C(F)(F)F)CCN(C(=O)Cn2cc(Br)cn2)CC1 c1(C(=O)NC2CC3(CN(C(C4N(C)CCOC4)=O)C3)C2)cc2c(cc1Cl)OCO2 c1(C(N2CC3N(C(C4C(C)C4)=O)C(CC3)C2)=O)cc(Br)c2nccnc2c1 Cc1cc(C(=O)N(C(C)CCNC(c2c[nH]c3cccnc23)=O)C)c(N)c(C)c1 Cc1ccc2[nH]cc(CCNC(=O)NCCn3cnc4ccccc34)c2c1 CC1CN2CCCC2CN1C(=O)CC1(NC(C2C(C)(C)C2(C)C)=O)CCCCC1 c1(C(=O)NCC2CC(NC(C(C=C)(C)C)=O)C2(C)C)cccc(F)c1C#N C12CCCCN1c1n[nH]c(c1Cl)NCn1cnnc1C(=O)N1CCC21.CCOC c1(C(=O)NC(C(=O)NCc2c(C)n[nH]c2C)C(C)(C)C)cncc2[nH]ccc12 C1(CNC(C(=O)Nc2c(SC(C)C)cc(Br)cc2)=O)CCC2(CCNCC2)O1 c1(OC)ncnc(C)c1C(N1C2CCC1(CNC(C1CCCC1(C)C)=O)CC2)=O CC1(C)CC(CC(=O)NCC(C)(C)Cn2cc(C(C)(C)C)nn2)CO1 c1(N2CCCC(n3ccc(C)n3)C2)c(C(F)F)cccc1[N+](=O)[O-] C1(C(=O)NC2CCN(C(CCC(=O)NCC)=O)C(C)C2)CCc2c(n[nH]c2C)C1 N1(CC)CCOC(C(=O)NCC(CNC(=O)COCc2ccncc2)CO)C1 C1(CNC(C(CC)COC)=O)CC2(CC(NC(C3CC4(CCC4O)C3)=O)C2)C1 N1(C(c2c(CC)noc2)=O)CCOC2(CCC(NC(c3cnc(Cl)[nH]3)=O)CC2)C1 c1(C(N2CC(NC(c3cc(C)n(C(C)C)n3)=O)C2)=O)cc2cc(O)ccc2[nH]1 Cc1[nH]c(=N)nc(O)c1CCC(N1CCC(C)(NC(C2C(C)C2C)=O)CC1)=O n1(CCC)nc(C)cc1C(=O)N(C(C)CN(C(=O)C(C(C)C)n1ccnc1)C)C c1(C(=O)NCC2(C)N(C(C(C)OC3CCOC3)=O)CCC2)ccc2c(c1)CCO2 c1(CC(=O)NC(c2ccc(C)s2)c2ccco2)nnc2n1CCCC2 N1(C(C2CC(OC)C2)=O)CCn2ncc(CNC(c3c(C)ncnc3C)=O)c2C1 CC1=C(C(=O)NC2CCC2NC(C2CC(CC3CC3)C2)=O)SCCO1 CC1=NNC(=O)C1CC(=O)NC1CC(N(C(=O)C=Cc2ccncn2)C)C1 C1(C(=O)OC(C)(C)C)CCC(O)(CNCc2ccc(C3OCCO3)cc2)CC1 c1(C(C(=O)NCCOCCNC(c2cc(Br)n[nH]2)=O)O)ccc(F)c(Cl)c1 C(CNC(=O)CC1CCCS1(=O)=O)(CC(F)(F)F)NC(c1c(CC)nccc1)=O c1(C(N2CCCC(NC(CCN(C)CC)=O)CC2)=O)c(C)c(C)nn(C)c1=O c1(CNC(C2C(C)(COC)C2)=O)ccc(CCNC(c2cc(C)[nH]n2)=O)cc1 C(CC(C)C)(C(=O)NCCOCCCNC(=O)CC1(C)CC1(Cl)Cl)OC CC1C2CN(C3CCN(C(=O)COc4cnc(Cl)cn4)C3=O)CC12 C1(C(=O)NC)CCC(C)(C(=O)NOC(C)C(=O)OC)C1 Cc1cnc(N2CC(NC(c3cscc3C)=O)CC2C)nc1 N1(CCCC)CCC2(CCCCN(C(=O)CC(CC)c3ccccc3)C2)C1.C(=O)(C1CCC1)N C1(NC(c2cn(C)nc2O)=O)CCC12CCN(C(=O)C1=NOC3COCC13)CC2 CC(C(C)C(=O)NOC1CCOCC1)NC(c1ccc2[nH]ccc2c1)=O c1(C(N2CCC(NC(C(C(C)C)N(C)C)=O)C(CO)C2)=O)cc2c(s1)CCOC2 N1(C(C(C)(C)NC(CNC(C2C(C)C2)=O)=O)=O)CC2C(C1)C2(C)C c1(CNC2(C#C)CN(C(=O)OC(C)(C)C)C2)cc(C(F)(F)F)c(OC)cc1C c1(CNC(c2n(CC=C)nnn2)(C2CCSC2)C)ccc(C(N)=O)c(C)c1 C1(OCC2(CNC(=O)NC(C3ON=C(C)C3)C)CC=CC2)CCCCCC1 C1(CN(C(c2cnc(C)s2)=O)C)CCN(C(=O)C(CN(C)C)N(C)C)CC1 CCC(C)CCCCC(=O)NC1CCCC1CN(C(=O)CC(C)(C)C(=O)OC)C C1(NC(C2=C(C)OCC2)=O)CC2CCC(C1C)N2C(=O)CSC(F)F N1(C(CCSCC(C)C)=O)CCC2(CC1)CC2NC(C1Cc2ccccc2S1)=O C(C(CNC(=O)C1=COCCC1)S(C)(=O)=O)NC(C(C)SC)=O N1(C(CCCC#C)=O)CC2CC3CC2C1C3NC(c1cnn(C(C)C)c1F)=O N1(C(C(CC)COC)=O)CCC(C2CN(C(c3[nH]nc([N+](=O)[O-])c3Cl)=O)C2)CC1 CC(C#N)CCC(=O)N1CCCC1CN(C)C(c1cc(-c2ccncc2)[nH]n1)=O C(CN=c1[nH]c(=NCCSCCC(F)(F)F)[nH]c2c1CSC2)n1cnc(C)c1C C1(C(=O)NC(C)CN(C)C(C2COCCN2C)=O)CCCCC1(C)C c1(C(N2C(CNC(CC3(OC)CC3)=O)CC3CC32)=O)nn(C)c2ccc(F)cc12 n1(CC(c2ccccc2)C)nc(-c2ccn(C)n2)nc1C1CC1c1ccccc1 c1(CC)cnn2c1CN(c1cc(C)[nH]c(=NCc3cc(Br)cnc3O)n1)CC2 C(CCCC)(C(=O)NCC(C)C(C)O)NC(C(CC#C)C1CC1)=O C1(C(N2CC(C#C)OCC2)=O)CC(N=[N+]=[N-])CN1C(=O)C(=O)C1CCCC1 C(C(O)CNCc1ocnc1CC)(OCC)OCC C1(C)(CC)C=C(C(=O)NCc2cn(CCCF)nn2)C1.C1CS1 C1(C(=O)OC)CCC2(CC(C(=O)O)C2)N(C(=O)Cc2c[nH]c3ccc(O)cc23)C1 S(=O)(=O)(c1ccc(Br)cc1NC(C)CCO)NCCSCC c1(OC)cncc(CCC(=O)N(CC(C)CNC(C2OCCC2C(C)C)=O)C)c1 c1(C(=O)NC2CCC(N(C(c3cc(OCC)no3)=O)C)C2)ncc(C)cc1OC C=CCC(CC)C(=O)NC1CN(C(=O)CSCCOC)CC1(C)C CCCCC(C(=O)NCC1CCN(C(=O)C(O)COC)CC1)ON=C(C)C C1(CNC(C2(CSC)CCC2)=O)CC(O)CN1C(=O)CCCCN1CCCC1 C1(C(=O)NCCNC(C2(C#N)CC3CC3C2)=O)CC(c2ccncc2)=NO1 c1(OC)cc(O)ncc1C(N1CC(N(C)C(c2ccsn2)=O)C(O)C1)=O C1(=CC(=O)NCCC2(OC)CN(C(=O)CCc3cnn(C)c3)C2)CCN(C)CC1 C1(F)(C(=O)NCC2CC(NC(CCP(C)(C)=O)=O)C2)CS(=O)(=O)CC12CCC2 C(=O)(CCC(F)(F)C(=O)N1CCN(C(=O)CC(CC)CCCC)CC1C)OCC C1(NC(c2nc(C#C)sc2)=O)CN(C(c2ccc(C)nc2O)=O)C(C)(C)C1 c1(NC(c2nc(C(F)(F)F)no2)C)ccc(S(=O)(=O)NCCC#N)cc1Cl N1(C(CC(C)OC)=O)CCCC(C2CCCN(c3cc(Cl)ncn3)C2)C1 C1(C(C=C(C)C)=O)CCCN(OC(=O)C(C)(C)C)C1=O.N12CCCC(C)(C1)C2=O N1(C(CC=C)=O)CCN2CCN(C(=O)CCC(=O)c3ccnc(SC)c3)CC2C1 C1(NC(C(CC(C)C)O)=O)CN(C(C2(C)SCCCS2)=O)CC12CCC2 C(=O)(CS(=O)c1ccc(Cl)cc1)NC1(CNC(C2N(C(C)=O)CCOC2)=O)CC1 C1(C(N(C)Cc2cc(C)on2)=O)CCOCCN1C(c1cnc(N)cn1)=O c1(C(N2CCC3(C(CNC(=O)CC(F)F)C3)CC2)=O)cc2ccc(Cl)cc2[nH]1 c1(N2CC(CC)SCC2)nc2ccccc2[nH]c1=NS(=O)(=O)c1ccc(C)cc1 c1(CN(CC2(C(=O)OC)CCCCC2)Cc2ccccc2)cccc(OC)c1Cl N1(C(C(CC)N(C)C)=O)CCC(C)(C)C1C(=O)NC(C)CN=[N+]=[N-] C(C)(C(=O)NCC1CN(C(C2(c3ccc(Cl)nc3)CC2)=O)C1)(C(C)C)OC CCCCCC(CC)C(=O)NC(CNC(c1cccc(C2(CC)CC2)c1)=O)CO C1(NC(C2CCn3c(Br)cnc3C2)=O)CN(C(=O)C2CC2)C2(CCCC2)C1 C(=O)NN1CCCC1.C=CCCCCC(=O)N1CC2(CC(=C)C2)C1 N1(C(C2(NC(=O)Cn3cncn3)CCC(C)(C)C2)=O)CCc2nncn2CC1 c1(C(=O)NC(CNC(C=C(C)Cl)=O)CO)c(Cl)cc(C(F)F)cc1Cl c1(C(=O)NC(CN(C(=O)CCC2NC(=O)NC2=O)CC)C)coc(S(N)(=O)=O)c1 C(c1cccc(C#N)c1)=CC(=O)NCCCN(C(C(C)=C1CCC1)=O)CCO CCC(O)C(F)(F)C(=O)N1CCC(C)(NC(c2ccn(C3CC3)c2C)=O)CC1 c1(C(N2CC(N(C(C3CCN(C(C)=O)CC3)=O)C)C(F)C2)=O)ccc(=O)n(C)c1 C(C1Cc2ccccc21)NC(C(CC1CCCC1)NC(c1cncc(C)n1)=O)=O N1(C(CCC=CCC=C)=O)CCCC(CC)(OC)C1.N12CC=CC1(COC)C2=O C(=O)(C1=CS(=O)CCC1)N1CCC(C)(NC(=O)CC=Cc2ccccc2)CC1 N1(C(CC(C)OC)=O)CCOCC1c1ccc(CNC(=O)N(C)C)o1 c1(C(N2C(CC)CCC2C)=O)coc2c1CN(C(C1CC3(CC3)CO1)=O)C2 CC(C(C)(C)NC(c1cnc(C2CCOC2)s1)=O)NC(c1cc(C2CC2)on1)=O c1(CN2CCC(CNC(=O)CCCc3nc[nH]n3)C2)ccc(F)cc1 C1(C(=O)OC)CCC2(CCOCC2)N1C(C1CCCN(CC(F)(F)F)C1)=O c1(CN2CC(c3ccc(C)cc3)OC(C)C2)cccc2c1OCO2 Cc1ccc2c(C(=O)NCC3(F)CC(NC(=O)C(C)C(C)O)C3)coc2c1 C1(C(C)C)CN(C(=O)Cc2cnc(C3CC3)[nH]2)CCCN1C(C1CCSC1)=O c1(NCCNC(=O)NCC)cc(N2CCCC(C)C2)nc(COC)n1 C1(OC)(CNC(C2CCN(C(C)C)CC2)=O)CCN(C(=O)CC2(O)CC2)CC1 Cc1cc(-c2cn(CC3CCN3C(=O)CN(CC(C)(C)C)C)nn2)cc(C#N)c1 c1(NC(CC)CNC(=O)C2=NOCC2)ncnc2cc(C)[nH]c12 c1(OC)c(C)ccc(C(=O)N(c2nccn2C)C)c1F CC1(CNC(=O)CN2CC3CC3C2)CCC(NC(=O)C(CO)NC(C)(C)C)CC1 CCC(CC(=O)NCC1CCCN1C(c1cn(CC)cn1)=O)C(C)C N1(C(C(C)Cc2cnco2)=O)CCCC12CCN(C(=O)Cc1csnn1)C2 N1(C(C2N(C(CC)=O)CSC2)=O)CCC(C)(NC(c2csc(CC)n2)=O)C1 N1(C(c2c(CC)n(C)nc2)=O)CC(NC(=O)Cc2ccco2)CC12CCCOC2 N1(C(Cc2cc(C)no2)=O)CCC2(CC1)CC(C)N(C(=O)C(C)C)C2 c1(C(=O)NCC(C)(CO)NC(C(CSC)O)=O)cnn(C2CC2)c1C C(=O)(C1=NOC(C)(C)C1)NCC(CNC(C1CCCC1O)=O)OC N1(C(c2nc(C(=O)OCC)sc2)=O)CCN(C(=O)CS(=O)(=O)N(C)C)CC1CC N1(C(c2c(C)c(Cl)cnc2)=O)CC(C)CN(C(=O)CCc2cnoc2)CC1C CC1CCCN(C)N1C(=O)C1CN(Cc2ccccc2)CCN1CCO N#CC1(C(N2CCC(O)(CNC(=O)C=Cc3cncc(F)c3)C2)=O)CCCCC1 C=CCCC(O)CNC(=O)C(O)CNC(C1(CO)CC(C)(C)C1)=O c1(OC)ccc(C)cc1CN1CCC(NC(C2(C3CCCO3)CC2)=O)C(C)C1 c1(C(N2CCC(CNC(CC3(C=C)CCC3)=O)C2)=O)oc(CO)nc1C CC(C)(C)C(CC(=O)N1CCC(CO)C(O)C1)NC(=O)C(c1ccccc1)F c1(C(=O)NCC2(C)CCCN2C(C2CC(F)(CO)C2)=O)cccc(=O)n1O N1(C(C2C=C(C)CS2)=O)CC(C(=O)NCC(C)(O)CN(C)C)C2(CCC2)C1 n1(CC(=O)NCC(CNC(CCN(CC)CC)=O)O)nc(C)c(Br)c1C CC(C)CC(=O)NCC(=O)NC(Cn1ccnn1)C(=O)NCC(O)CNC(N)=O c1(CN(C(c2cccc(F)c2I)C(=O)NC)C)ccc(Br)cc1OC c1(C(=O)NC2C(C)CN(C(C3CC(=O)CC34CCC4)=O)CC2)ccc2ncsc2c1 Cc1ccc(F)c(C(N2CCCC2CCCNC(C2CN(C)CCO2)=O)=O)c1O Cc1cc(F)ccc1C(O)C(=O)NC1CCN(C(=O)CSCC(N)=O)C1C1CC1 C(=O)(C(C(=O)N(CCCN(C)C(c1ccccc1C(F)F)=O)C)OC)OC CC1CCN(C(C2CCCCN2C(N)=O)=O)CC1CNc1nnccc1C#N C(=O)(C1CCCc2cccnc21)NCCC(C)NC(Cc1c(C)cc(O)cc1)=O CCC(C)(C)CCCC(=O)N1CCC(C)C(CNC(C2CCC(C)(CC)O2)=O)C1 c1(C(=O)NC(C)C(C)NC(C2(CC3CC3)CCC2)=O)cc(Br)cn2ccnc12 C#CC(CNC(c1csc(CNC(C2CCC2(F)F)=O)c1)=O)CC(C)(C)C C=CCC(F)(F)C(=O)Nc1cc(O)nc(COC(C)C)n1 c1(OC)cc(CNCc2cccc(-c3ccco3)c2)cc(N)c1OC C1(C(N(CCNC(C(C(C)C)SCc2ccccc2)=O)C)=O)CC2(CCC2)CO1 CCC(O)C(C)(C)C(=O)NCC(C)(C)CCNC(c1scc(C)c1Cl)=O Cc1cc(C)nc(SCC(N2CCN(C(C3C4COCC34)=O)C(CO)C2)=O)n1 c1(C(C(C)NCC2(COC)C=CCC2)=O)ccc2c(c1)CCC2 C1(N(C)C(c2cc(Cl)ccn2)=O)CCC2CN(C(C3CCOC3)=O)CC12 C12(NC(C(C=C)(C)O)=O)CCCC(NC(=O)C(CC)CC)(C1)C2 N1(C(c2c(OC)nccn2)=O)CC(C(=O)NCCCC2CCOC2=O)C(C)(C)C1 N1(C(c2cc(C)oc2)=O)CC(O)(C2(CNC(=O)C(C#N)C(C)C)CC2)C1 C(=O)(CCCC(CC)NC(=O)CCC1CC1C)Nc1cnc(SC)nc1 C1(NC(C2(CCOC)CC2)=O)CN(C(c2cccnc2N)=O)CC1N=[N+]=[N-] Cc1c(C(=O)NC2CC(NC(C3(Br)CC3(C)C)=O)C2)cnn1C1CC1 C(C)(C(=O)NCCN(C(=O)CCc1ccoc1)CC)=C(CC)C c1(C(=O)NC(C)C=CC(N2CCC2CC(C)(C)C)=O)cccc(Cl)c1 Cc1cc(C)c(C=CC(N2CCCC2CN(C)C(c2coc(C)c2)=O)=O)c(C)c1 C1(C(=O)NCC2C(CC)C2)CC=CCC1NC(c1ccoc1C1CC1)=O C1(NC(c2cc(C)n(-c3ccccc3)n2)=O)CN(C(=O)CC2CCC2)C(C)(C)C1 C(C(=O)N=c1ccn(CCC#N)[nH]1)=Cc1ccc(OC)cc1 C1(NC(C=C(C)C(C)(C)C)=O)CN(C(=O)CCCCC2CCC2)C2(CCOC2)C1 C(=O)(C1=CCC(NC(c2ccc(OC)o2)=O)C1)NC(C1CC1(C)C)CC c1(C(N(CCCN(C(C2CCC(C)C2)=O)C)C)=O)cc2nccnc2cc1F CC#CCCCC(=O)NCC1(NC(=O)Cc2c(F)cncc2Cl)CCC1 C(CC(CNC(c1ccsc1Br)=O)NC(=O)COc1ccsn1)OC C1(NC(c2c(CC)nns2)=O)CC(F)CN(C(C2CC(SC)C2)=O)C1 c1ccc2c(c1)OCCC(N=c1[nH]c(=NCc3ccncn3)[nH]c3c1SCC3)C2 c1(C(=O)OC)ccc(NC(=O)C(C)C)o1.C1(=O)COC(=O)CN1C C1(NC(C(=O)Nc2c(Br)c(F)cc(C(C)=O)c2Cl)=O)C2Cc3cc(F)ccc3C12 Cc1nccc(C(N2CC(N(C(=O)Cc3c(C)noc3Cl)C)C(C)(C)C2)=O)c1C N1(C(C2CN(C(c3nc(C(C)C)oc3)=O)CC(C)O2)=O)CC2OC(=O)N(C)C2C1 c1(C(=O)OCC)cc([N+](=O)[O-])ccc1N1CCC(CNC(=O)C(C)(C)C(=O)NC)C1 C(C(C)(C)CC(=O)N1CCOCC1C(=O)NCCN1CCNC(=O)C1)N(C)C C1(NC(C(N2CCSCC2)C)=O)COCCN(C(=O)CCOC2CC2)C1 C12(C(=O)Nc3cnc(Cl)nc3)CCC1CN(C(c1ncon1)=O)C2 c1(N2C(C(C)(C)NC(CC(CC)C(C)C)=O)CCC2)ncc([N+](=O)[O-])cc1F C(=O)(C(C)(C)C(F)F)NC(C1CN(C(=O)C(O)(C2CC2)C2CC2)CCO1)C c1(OCC(=O)NC2CCCN(c3nc(Cl)ncc3Cl)C2)ccc2c(c1)CCC(=O)N2 C#CC1(O)CC(C(=O)NC2CCC(NC(C3(c4ccncc4)CCC3)=O)CC2)C1 CC1CC(C(N2CC3(CCC3)C2)=O)N(C(=O)C(CN(C)C)N(C)C)C1 CCC(CC1CCCCC1)C(=O)N1CC2CC1C2NC(=O)CCC(C)N(C)C C#Cc1cncc(C(N2CC(CNC(=O)C=C(CC)CC)CC2(C)C)=O)c1 CC#CCC(C(=O)N1CCC1(C)C(=O)OC)NC(c1c[nH]cc1C)=O c1(C(=O)NCC2CCC(NC(CC(C)n3cccn3)=O)C2)ccc(F)c(C#N)c1 c1(C(=O)NC(C(=O)NCc2cn(CCC)nn2)C2CC2)ccc(OC)nc1 c1(OCOC)ccc(C(=O)NC2CCCC(C(=O)NCCn3ccnc3)C2)cc1 N1(C(Cn2ncn(C)c2=O)=O)CC=C(CCNC(C2COCCO2)=O)CC1 C=CC1(C(N2C3CCC(C3)C2C(=O)NCC2(CCOC)CCC2)=O)CCOCC1 CC(C)C1=NOC(C(=O)NCCCC(=O)NCC=CCl)C1 C(N=c1nc2c(c[nH]1)nc(N1CCC3(CCOCC3)C1)n2C)c1occc1 N1(C(C(CC)C(F)(F)F)=O)CCOC2CN(C(=O)Cn3nccc3C)CC12 C12(C(N3CCC(C(C)NC(C4(COCC)CC4)=O)C3)=O)CC3CC1C2C3O C1(NC(c2c(C)nsc2NC2CC2)=O)CCC2(CC1)CC2NC(=O)C(C)N(C)C Cc1cc[nH]c(=N)c1C(=O)NCC1(F)CC(CNC(=O)C(O)c2ccsc2)C1 c1(C(C)C(=O)N(C)CC2CCCCN2C(=O)CCC(F)F)cc2ccccc2s1 C1(O)(CNC(CN(C(=O)COC2CCOCC2)C)=O)CCOCC1 N(C(=NCCCCl)NCc1ccc(C(N)=O)o1)CC1C(C)(C)C1 C1(C(=O)NCC(CCC)OC)CCCN(C(=O)CC2CCCN2C)CC1 c1(C(=O)NCC2C(CNC(Cn3ncc(C)c3)=O)C2)ccc(C2CC2)cc1 CC1CCCN(C(=O)C(=O)NC2C3CC2N(C(=O)CSc2ccccc2)C3)C1 C1(NC(c2c(C(C)C)cco2)=O)COCCN(C(=O)C(C)n2cccn2)C1 Cc1n[nH]c(C)c1C(C)NC(=O)NCCCC(=O)NCC1CCCOC1 c1(C(=O)NCCCN(C)C(C2CCCN2C(=O)C2CC2)=O)c(F)cncc1F c1(C(=O)NC2C(C)CN(C(=O)CN3CC=CC3)C2)cccc2c(O)nncc12 Cc1ncc(C)c(=NCC(C(C)(C)C)NC(c2ccn3ccnc3n2)=O)[nH]1 N1(C(CN(C)C(C2CC(CC(=O)NC3CC3)C2)=O)=O)CCc2ncsc2C1 N1(C(C(C(C)C)SCC)=O)CC2CCCC2(CNC(=O)CN2CC(C)(C)C2)C1 N1(C(CSCCCC)=O)CCC1(C)CC(=O)NC(C)C(=O)OC(C)C c1(C(=O)NC23CC(C(=O)NCc4cncc(Cl)c4Cl)(C2)C3)ccc2ncnn2c1 C12(n3cc(-c4cnc(C)o4)nn3)CCC(C(=O)NCc3ccsn3)(CC1)C2 c1(C(=O)NCC23CC2CN(C(c2cc(Cl)no2)=O)C3)cn2cccnc2n1 C=CCCCCCCCCC(=O)N1CCC(NC(c2nonc2CC)=O)C12CC2 c1(C(N(CCNC(C(CC)N(C)C)=O)C)=O)sc(C2CCCOC2)nc1C n1(CC(N2C(C3(NC(=O)C4=CCCO4)CC3)CCC2)=O)ccc2ccccc12 Cc1csc(NC(C2COCCN2C(=O)C=Cc2ccc(Br)cc2)=O)c1C#N N1(C(C2CCCN(C(C)=O)C2)=O)CCCC(O)(CN(C(=O)CCC(C)C)CC)C1 C1(CC(=O)NC)CN(C(=O)CN(c2ncccn2)C)CCN1C(=O)CC(F)F Cc1ccc(Br)cc1CC(=O)NC1CCC1NC(C1CC(CF)C1)=O c1(C(=O)NC2CCN(C(c3nc(C)oc3)=O)C2)[nH]nc2c(=O)n(C)cnc12 C12(NC(c3cnc4sccn34)=O)CCCC1N(c1ncccn1)CC2 C=CC1(CC(=O)N(CC(c2nn[nH]n2)C)C)CN(C(=O)CC2(O)CCOC2)C1 C1(CNC(=O)Cc2cccc(Cl)c2)CN(c2ncncc2Cl)CCCO1 C(=O)(C1CCc2c[nH]nc21)N1CCC(C(C)(C)C)(CO)C1 c1(C(=O)NCC2(C(=O)NC(C)Cc3nc[nH]n3)CCCO2)cccc2c1CCC2 C#CCCCC(=O)N1CC(CNC(=O)C(C2CCCC2)OC)CC1C c1(OC)ccc(C(CNC(=O)CC2CCN(C)C2)NC(=O)CC(C)C)cc1 CC1(C(=O)NC2CCC2NC(=O)Cc2cnccc2C(F)(F)F)CCC(=O)NC1 C(c1ccccc1)=C(OC)C(=O)NCCCCNC(=O)C(C)(O)C1CCOCC1 C(C(CC(C)C)C(=O)NCc1cccnc1CNC(=O)Cc1cnc[nH]1)OC c1(C(N2CCC(N(C(=O)C=Cc3cnccn3)CC)C2)=O)cccc(N)c1F C1(CNC(c2n(CC)nnn2)(C)COC(C)C)CCSC1(C)C c1(N2CCN(C)C(c3cccs3)C2)ncccc1S(=O)(=O)NC1CCS(=O)CC1 N1(C(Cc2n[nH]c(=N)s2)=O)CC2CC(NC(c3ccn(C4CCCC4)n3)=O)C2C1 C1(CNC(C(C)C2CCC2)=O)CCCC2(CN(C(c3cccn(O)c3=O)=O)C2)O1 C(=O)(C1COc2ccc([N+](=O)[O-])cc21)N1CC(NC(c2n(CC)ncc2Cl)=O)C1 Cc1oc(C2CCOCC2)nc1C(=O)NCC(F)CNC(=O)C=C1CCN(C)C1 C1(C(=O)NC(C)C(C)NC(c2ccc(N)cc2Cl)=O)(OCC)CCC(F)(F)CC1 c1(NC(=O)CN2CCSCC2)cccc(O)c1.C12COCC1N(C(C1CC1F)=O)C2 N1(C(CN2C(C)CC2)=O)CCC2(C1)CN(C(=O)NC1CN(C3CCCCC3)C1)C2 C1(Nc2c(C(=O)OC)cccn2)CCC(C)N(C(c2scnc2C(F)F)=O)C1 CC(C)(F)CCC(=O)NCC1(C(C)(C)C)CCN(C(=O)COCP(C)(C)=O)C1 C1(CNC(c2cccnc2F)=O)CC(N=c2[nH]c(Cl)ncc2Cl)C1 C1(CNC(C(CC)(C)CC)=O)CC2CCC(C1)N2C(C1CC2C(C1)C2(C)C)=O C1(CCCCOC(=O)NCC(c2cnn(C)c2)C)CCN(C(=O)CC#N)CC1 C1(C(=O)NC23C(CN(C(=O)CC=C(Cl)Cl)C2)C3)C2C3CC4C1C1C2CC3C41 N1(C(=O)CC23CCCC2C3)CC(NC(c2cc3sccc3s2)=O)CC12CCCC2 c1(C(=O)NC2CCC(C)NC2=O)cccc2cc[nH]c12 CC1(C)CCCCC1CC(N1CCOC(CNC(C2CC=CCC2)=O)C1)=O c1(C(N(CC(CN(C(=O)Cc2ccoc2)C)O)C)=O)cc(C2CC2)on1 CCC(CNC(=O)C(CNC(c1cnn(C)n1)=O)CC1CC1)CCO CC1CC(NC(c2cnsc2)=O)CCN1C(=O)Cn1ncc(O)nc1=O C(=O)(C#CC1CCOCC1)N1C(CCN(C(C=CCOC)=O)C)CCCC1 N1(C(CCCC#C)=O)CCCC2(CCC(NC(=O)CN(CCCCCC)C)C2)C1 c1(C(C)(OC)OC)ccc(C(N2CCC(CF)(NCC(=O)C3CC3)C2)=O)cc1 CCC(C)(C)CC(=O)NCC1CN(C(c2ccc(OC(F)F)nc2)=O)CCC1C CCCCCCC(C)c1nc(C(C)SCC)nn1-c1cccnc1 C1(C(N2C(CNC(c3cc(F)c[nH]3)=O)CC(OC)C2)=O)CCCC2(CC2)C1 C1(C(=O)OC)CCCC(C(=O)NC2C=CC(CNC(=O)CSCC(F)(F)F)C2)C1 C1(NC(c2ccc(CC)[nH]2)=O)CC1C1CCCN(C(C23CC2COC3(C)C)=O)C1 c1(CNc2cc(N3CC4C(CC)(C4)C3)ncn2)ccc2c(c1)CC(C)O2 C1(C(=O)NC2CC3(CN(C(CNC(C)=O)=O)C3)C2)COc2ccc(F)cc2C1 CCN=c1[nH]c(C)c(C(=O)NC(C2CCOC2)CNC(=O)CC(F)(F)CC)s1 c1(CNC(=O)C(N2CC(O)CC2c2ccc(F)cc2)C2COC2)ccccc1Br N1(C(c2c(C#N)cn[nH]2)=O)CC2CCCC(C1)N2C(c1ncccc1Cl)=O C1(CC(=O)N(C)CCNC(c2ccc(C(F)(F)F)o2)=O)CC(O)C1(C)C C1(F)(CNC(c2nc(CCC)sc2)=O)CCC(CNC(=O)CC2CC3(CC3)C2)C1 CC(C)C(C(=O)NC1CCCC1NC(c1ncoc1C1CCC1)=O)NS(C)(=O)=O N1(CC)CCCN(C(=O)C(C2CC=CCC2)NC(c2onc(C)c2CC)=O)CC1 c1(CCC(=O)N(CC(C)N(C(c2cnc(OCC)s2)=O)C)C)cccc(F)c1F C(=O)(C(C)(C)CCCNC(=O)CC(C)C)N(CCCC)CCCO c1(C(N(C2CCCN(C(=O)C(F)OC(F)(F)F)C2)C)=O)cccc(-n2cnnn2)c1 CC(C)C(CCC(=O)NC1CN(C(C)C)CC1C)NC(c1c[nH]c2cccnc12)=O c1(C(N(CCC=C)CC(=O)OCC)=O)ccc(CCCC#N)cc1 C(CC(CC)C(=O)NCCC1CC(NC(C2CCN(C3CC3)CC2)=O)C1)=CC C1(CC)(NC(=O)CCOC)CCCN(C(=O)C(C)Sc2ccc(F)cc2)C1 c1(CC2C(C(N3C(CNC(c4c(CC)ocn4)=O)CC3)=O)C2)ccccc1CC c1(C(N2CCN(C3CCCN(C(C(F)OC)=O)C3)CC2)=O)ccc(OC)cc1Cl N1(C(Cc2cn(CC)nn2)=O)CC2C(CNC(c3nnn(C)n3)=O)C2C1 c1(CC)cccc(C(N2CCC(O)(CCNC(c3ccnc(S)c3)=O)C2)=O)c1F CCC(CNC(=O)CC1(NC(c2ccn(C3CC3)n2)=O)CC1)C(C)C C(=O)(C1=NOC2COCC12)N1C(C(N(C)Cc2cn(C)nn2)=O)C2(C1)CCCC2 C1(CC(F)(F)F)C(=O)N1.c1(NCCC)cccc(C(=O)Nc2ccccc2)c1 C1(NC(C2(COC)CC2)=O)CN(C(=O)COc2cccc(Br)c2)C2CC12 c1(CNC(C2CNCCN2Cc2ccc(F)cn2)=O)c(Cl)cccc1Cl Cc1cc(C(N2CCC(C)C(NC(c3ncccc3F)=O)C2)=O)c(O)nc1C C1(NC(C2C(=C)CC2)=O)CCN(C(c2cccc(C(C)(F)F)c2)=O)CC1F CCC(CC(=O)N1CC2(C)CC1(C(=O)NCC1CCC(CO)O1)C2)C(C)(C)C N1(C(C2CN(C(C)C)C(=O)C2)=O)CCN(C(=O)C2=NNC(=O)CC2)C(C)CC1C C(=O)(C(F)(CNC(=O)CCn1ccnc1C)C(C)C)N1C(C=C)CC1 c1(CC)[nH]nc(C(N2CCCC2CC(=O)NCC23CC(CO)(CO2)C3)=O)c1C C1(C(C)NC(Cc2nc(C)[nH]n2)=O)CCN(C(c2cn(C)nn2)=O)CC1 C(CCC(=O)NCC1C=CCN1C(=O)COC1CCOCC1)N(C)C c1(SC)cccc(C(=O)NCCC(O)CNC(=O)COc2ccsn2)c1 c1(C(=O)NCC2N(C(C(C(C)C)SC)=O)CC=C2)cn(C)c(=O)n(C)c1=O N1(C(COCC#C)=O)CCN(C(c2ccc(C)c(C)n2)=O)CC1C1CC1 c1(C(N(C)CC2(NC(C(CC)OC3CCCC3)=O)CC2)=O)cccnc1O N1(C(C2C(CC(C)C)C2)=O)CCC(C)C(CNC(c2ccc(Cl)s2)=O)C1 C(=O)(CCCS(N)(=O)=O)N1CC(C)(CNC(=O)C#CC2CC2)OCC1 C1(NCC(=O)NCCc2ccc(OC)cc2)CN2CCC1(F)CC2 c1(C(=O)NC2C(NC(c3c(OC)cncc3)=O)CC2)cc(C)nc(O)c1[N+](=O)[O-] C(=O)(C1=CCS(=O)(=O)C1)N(CCNC(CC1N(CC)CCOC1)=O)CCOC N1(C(C23OC(C)C(C2)C3)=O)CC2(CCN(C(c3cc(C4CCC4)nn3C)=O)C2)C1 c1(C(N(CC(CC)NC(=O)C(O)c2ccsc2)C)=O)c(C)ccc2nsnc12 N1(C(C(C)(C)OCC)=O)CC2C3CCC(C2C1)N(C(=O)CCc1ccccc1)C3 N1(C(C(CC)C)=O)CCOCC(C(=O)NCCCCCCCO)C1 c1(C(C)NC(=O)C(C)(C)n2cnnn2)ccc(CNC(=O)CC=CC(C)(C)C)cc1 c1(C(=O)NCC2CC3N(C(C(C)C4CC4)=O)C(CC3)C2)c(F)ccc2n[nH]cc12 N1(C(CN(C(C)=O)C)=O)CC(C(=O)NCC23CCN(CC2)CC3)CC(C)(C)C1 N1(C(c2cccn2-c2ccccc2)=O)CC2CCC1C(NC(C13CC(C1)C3)=O)C2 N1(C(CC(CNC(c2cnccn2)=O)OC)=O)CCCCC(C)(C)C1 C(=O)(CC(O)CC(C)C)N1CC(CC(N2CCC(C=C)C2)=O)OCC1 c1(C(=O)NC2CC(F)(CNC(C3C(=C)C3)=O)C2)ccc(SCCC)cc1 C1(CNC(=O)Cc2ccccn2)(NC(=O)CC2(O)CCOC2)CCCCC1 c1(C(=O)NCCNC(C(n2cc(Br)cn2)C)=O)ccc2c(c1)N(C)C(=O)CC2 c1(OCCC)ccc(C(N2CCC(C(N)=O)C2)C(=O)NC(C)C)cc1C c1(CC=C)ccccc1C(=O)NC(C(=O)NCCC(COC)OC)C(C)C C=C(C)C(C)(C)C(=O)NCC1(C(F)F)CCN(C(c2cnc(OC)nc2)=O)C1 c1(NCCCc2c(C)cccc2)nc(C)nc2sc3c(c12)CCC3 N1(C(c2c(CC)c[nH]c2)=O)CCN(C(=O)Cc2ccc(Cl)cn2)C2CCCCC12 C=CCC(CC(=O)NC1(C)CCOC1C)NC(c1cc(=O)n(C)cn1)=O c1(NCC2(CC)CC2)ccc(CCn2cc(C3C(C)(C)C3(C)C)nn2)cc1C N1(CCCC)CCCCC1C(=O)NCC(CO)NC(c1ncsc1C1CC1)=O C(CCC(C)C)(C(=O)N(C(C)CCSC)C)NC(C(C)(C)OCC)=O CN1CCC(C)(C(N2CCC(C)(CNC(c3c(Cl)cnn3C)=O)C2)=O)C1=O CCCCC(CC(=O)N1CCCCC1CF)NC(C1CCN(CC)C1C)=O C12(CC(=O)NCC3CCN(C(C4CC5CCC4C5)=O)C3)CNC(=O)C(C1)C2 C1(C(N2CCC(O)(CNC(c3cc(=O)cc[nH]3)=O)C2)=O)CCC2(CCC2)CO1 C1(NC(C=C(C)C(C)C)=O)CC(NC(c2cncc(N)c2)=O)C12CCC2 c1(C(=O)OCC(=O)N(CCCCCC)CC)cnc(C)n1C(F)F.C(CSC)O Cc1cc(Cl)cc(NC(C2CCOC2c2c(C)n[nH]c2C)=O)c1O CC1(C)CCC(CC(=O)NCC23CC2CN(C(=O)COc2cccc(F)c2)C3)O1 N1(C(CC2C(CC)C2)=O)CC2CC(C1)N(C(c1ccc(Cl)c(C(F)(F)F)c1)=O)C2 C1(COc2ccnc(OCCO)n2)CCCCC12CCC2 C1(NC(c2cc(C)n(C)c2)=O)C2CC3C(C2)C13C(=O)NC1CCC(F)CC1 CC(C)(C(=O)NCC1CCCN1C(c1cn(CC(N)=O)nn1)=O)n1cnnn1 Cc1cnc2cc(C(N3CC(=C(F)CNC(C4CCCS4)=O)C3)=O)ccn12 N1(C(C2CC(O)(CNC(C3(CC(C)=O)CC3)=O)C2)=O)CCN2CCCC2C1 c1(C(N2C(C)C(NC(=O)C(=O)NCC3CC3)CC2)=O)cc([N+](=O)[O-])c[nH]1 N1(C(c2ccc(CNC(C)=O)o2)=O)CC(C)CN(C(=O)Cn2ccnn2)CC1C c1(C(=O)NCCC2(C)CCN(C(C(CSC)C)=O)C2)ncc(F)cc1F N1(C(C(F)=CCC)=O)CCN(C(=O)CSC(C)C)C(C2CC2)C1 C1(NC(C=CC=CC)=O)CCN(C(c2ccccc2C(F)(F)F)=O)CC1(C)C.C1CC1 C1(NC(c2ccc(OC)s2)=O)CC2CC(NC(=O)Cc3cccc(C)c3)CC2C1 N1(C(CCn2ncc(C)c2)=O)CCCC(O)(CN(C)C(C2CCCC2(F)F)=O)C1 C(=O)(CCCCC(C)(C)C)N1CC(C(C(N2CCC(C#C)(O)C2)=O)O)C1 C1(C(=O)NC2C3CN(C(c4c(OC)cccc4)=O)C2C3)CCC(F)(F)CO1 c1(C(=O)NC(c2ccc(F)cc2)C)cc(-c2nn[nH]n2)cn1C c1(C(N2CC(C(O)C(=O)NCc3csc(O)n3)C2)=O)ccc(C2(NC)CC2)cn1 Nc1cc2c(cc1C(=O)NC1(CCNC(C3CCC(F)CC3)=O)CC1)OCO2 N1(C(c2ccc3cnc(C)n3c2)=O)CCC2(CC1)CN(C)C(=O)O2 C(C1CCCc2ccccc21)NC(c1c(C)sc(Br)n1)c1nnnn1CCSC N1(C2CCN(C(C(C)N(C)C)=O)C2)CCC(NC(c2ccn(C(F)F)n2)=O)CC1 CC(C)CCC(C)N(C)C(C1CN(C(c2cccc(O)n2)=O)C1)=O.NC c1(C(=O)NCC(CC=C)NC(C23COC(CF)(C2)C3)=O)ncccc1SC N1(C(CCOCC)=O)CCC(N(C(=O)C(Cc2ccccc2)C2CC2)C)C1C N1(C(C(c2c(C)noc2C)CC)=O)CCN(C(=O)C=Cc2nc[nH]n2)C(C)C1 C(=O)(C(C)(C)C(C)NC(C1CC(CF)C1)=O)NC(c1ccccc1)CC N1(C(=O)COc2ccc(F)cn2)CCC2C(CCN2C(c2cnc(Br)s2)=O)C1 N1(C(c2c(C(C)(C)C)con2)=O)CC2(CNC(C3(S(C)(=O)=O)CC3)=O)CCC1C2 Cc1cc(C#N)cnc1C(=O)NCC(O)CN(C)C(C1CCC(C)(C)CC1)=O CON(CCC(=O)NCC1CC(C)(C)CCO1)C(=O)C1CC(=O)OC1(C)C CC(O)C(C)CNC(=O)C(c1ccnn1C)NC(=O)CCc1ccsc1 Cc1csc(C(N2CC3CC2(CNC(c2nc(=O)n(C)[nH]2)=O)C3)=O)c1Br CC1(C)COCC(CC(=O)NC2CC3(C2)CC(NC(c2cnccn2)=O)C3)O1 C1(C)(C(=O)NCCCCN(C)C(C2CC(C)(C)C2C(F)(F)F)=O)CNC(=O)C1 C1(C(=O)NC(C(C)C)CN(C)C)CNC(=O)CN1C(=O)CN(C)C c1(C(N(C2CCN(C)CC2)C(c2oc(C)c(Br)c2)=O)=O)cnc2ccccc2c1 C1(CC)CCCN(C(C2CC(NC(C3(n4cccn4)CC3)=O)C(O)C2)=O)C1 c1(C(N2CCC(CNC(COc3cc(C)on3)=O)C2)=O)nccnc1C(N)=O N1(c2n(C(C(c3ccc(OC)cc3)C)C)nnn2)CCc2cccnc21 c1(COCC(=O)N(CC(C)(C)NC(c2cc(C)ncc2)=O)C)cccc(Cl)c1F C12(C(=O)NC3(C(O)C(F)(F)F)CCC3)CC(NC(C(C)(C)OC)=O)(C1)C(C)(C)O2 c1(C(N(C)CC2(O)CN(C(C(C(C)O)(F)F)=O)C2)=O)cnn2c1NCCC2 CC1=NOC(C)(C(=O)NC2CN(C(c3c[nH]nc3C3CCC3)=O)CC2O)C1 C(CN=c1nc[nH]c2[nH]c(Cl)cc12)N(C(C=CC)=O)Cc1cccc(Cl)c1 N1(C(C2CC(OC)C2)=O)CCC2(CC1)CN(C(c1nnn(C)c1C)=O)CC(C)O2 Cc1c(C(=O)NC2CCC2NC(=O)Cc2ccccc2CC(N)=O)cncc1Cl n1(CCC)cc(Cl)c(C(=O)NCCCN(C(=O)CCCc2ncc(C)o2)C)n1 C(C#CC(C)NC(=O)OCC1CC(CN(C)CC)CO1)(OCC)OC C(C(CO)(CO)NC(=O)C(O)CN(C)C)N(C(=O)C#CC(=O)N(C)C)C N1(C(COC)=O)CCN(N(C)CC2CC2)CC1.N1CC(C(C(=O)NC)OC(CC)C)C1 C1(OCCCNC(C2C(C)C2)=O)CCN(C(=O)C(c2ccccc2)C2CC2)CC1 c1(CSCc2c(OC)cc(OC(F)(F)F)cc2)cccn2ccnc12 C1(NC(C2CC(Cl)(Cl)C2)=O)C2CCN(C(c3cc(CO)[nH]n3)=O)C12 CC(C)C(C)(CNC(C1CC12CCC2)=O)NC(c1ncncc1Cl)=O N1(C(c2c(C(C)C)nco2)=O)CCC(CF)(NC(=O)C=CCN(C)C)C1 C1(OC)CN(C(c2cc(C(O)C(F)(F)F)ccn2)=O)CC1NC(=O)C=CSC N1(C(C2C(SC)CCC2)=O)CC=C(CCNC(C2C3CCC4C(C3)CC24)=O)CC1 FC1CC12CC(c1nc(-c3cccnc3)nn1C1CCCOC1)C2 c1(CN(CC)CC)ccc(C(=O)NCC2(C)CCN(C(c3cnsn3)=O)C2)cc1 C(C(C)CS(N)(=O)=O)NCC(C)(C1CC1)OC N1(Cc2c(Cl)ccc(OC)c2)CC2CCN(C(=O)C=Cc3cccnc3)C2C1 CCCS(=O)(=O)CC(=O)NC1CC(C)CN(C(=O)C(CC(C)C)NC(N)=O)C1 C1(CNC(C=C(C)c2ccco2)=O)CC(C(=O)NC2CCCCC2O)=NO1 C1(CC(=O)NCC2CC2CNC(=O)CNC(c2ccco2)=O)CCS(=O)(=O)C1 Cc1cc([N+](=O)[O-])cc(C(=O)NC2C3CN(C(=O)CC4CCC(=O)NC4)CC23)n1 c1(SC)nocc1C(=O)NC1(CCCNC(c2sccc2F)=O)CC1 CN1CCCC1C(=O)NC1CC1CNC(C1(Cc2ccnn2C)CC1)=O c1(C(=O)NC2CC(CNC(C3(C)CC3(F)F)=O)C2)cc(C(F)(F)F)ncc1Cl C(C)(CO)(C(=O)NC1CC1(C)C(F)F)NC(CC1(OCC)CC1)=O C1(CNC(C2(CC)COC2)=O)CCN(C(c2cnc(F)c(F)c2)=O)CC1C CC1CN(C(=O)Cc2csc(C3CC3)n2)CCC1CNC(C1(C2CC2)CC1)=O c1(C(=O)NCC(CNC(C2(C)COC2)=O)F)ccc2[nH]c(=N)[nH]c2c1 C(=O)(C(O)CCCNC(C1CN2CCC1C2)=O)NCc1cnc(CSC)[nH]1 c1(C(N2C3(C(N4CC(c5ncn(C)c5)C4)=O)CC3CC2)=O)cc2ncccc2[nH]1 c1(N2CC(CCCCNC(=O)NC3CC(SC)C3)C2)ncnc2c1nnn2C1CC1 Cc1cc(C(N2CCC(CCNC(C3CCCS3)=O)C2)=O)ncc1Cl N1(C(C(c2scc(C)n2)C)=O)CCN(C(=O)CCC=CC(C)C)C(CC(F)F)C1 C1(C(=O)NC(CN(C(c2ncc(OC(C)C)nc2)=O)C)C)CCCC2(CC2)C1 O=C1Cc2c(C(N3CC(O)(CCNC(=O)Cc4nc(Cl)cs4)C3)=O)cccc2N1 c1(Cc2nc(COCC)nn2-c2cccnc2)cc(Br)cn(CC)c1=O S(=O)(=O)(c1ccc(N2CCC(c3ccn(C)n3)CC2)c(Br)c1)CC(C)(OC)OC C1(NC(=O)CN2C(=O)CSC2=S)CCC2(CC1)CN(Cc1ccc(Br)cc1O)C2 c1(CCC)cc(C(=O)NC(CNC(c2cnc(Cl)s2)=O)C2CC2)ccn1 N1(C(C(OCC)OC)=O)CCC(C(=O)NOC(COC)COCC)C1C C1(CC(=O)N(C(C)C)CCNC(C2CC(=C3CC3)C2)=O)SC(=N)NC1=O S(=O)(=O)(c1cc(Cl)cc2cccnc12)N1CCN(CC)C(C)C1 N1(C(c2cc(CCC)on2)=O)CCCC12CCN(C(=O)C(O)CCC)C2 c1(C(=O)NC(C)CN(C(=O)C(=O)NC2CCCCC2)C)ccc2c(n1)CCCC2 c1(C(=O)OC(C)C(=O)Nc2ccc3c(c2)OCO3)ccc2cnoc2c1 CCCCCCC(=O)N1CCC(CN(C(=O)CC2CCOC2)CC)C1 c1(OC)ccc(Br)cc1C(=O)NCC1(F)CCCN(C(=O)Cc2cc[nH]c2)C1 S(=O)(=O)(c1ccc(N(C)Cc2cc(F)ccc2Br)cc1Br)NC1C(SC)CCC1 C(=O)(C1=C(SC)CCCC1)N1C(CN(C(CN2CCCC(CC)C2)=O)C)CCC1 CC1CN(C(C2(F)CCOCC2)=O)CC(C)C1NC(c1cc(F)cc(F)c1O)=O c1(C(C(C)NC(C2CC(C)CN2C(=O)OC(C)(C)C)=O)O)c(Cl)cccc1Cl CCC(CC(=O)N1CC2C(CC(=O)NCC(C)(O)CO)C2C1)C(F)F c1(NC2C(C)CN(C(c3ncccn3)=O)C2)ncnc2c1nnn2C c1(C(=O)NCCN(C(=O)C(O)C(C)SC)CC)cc2c(C)c(C)ccc2[nH]1 C=CCCC(=O)NCC(F)CNC(C1(NC(=O)NC)CCCC1)=O C(=O)(CC1COc2cc(OC)ccc21)Nc1cc(C(=O)OC)c(OC)cc1 Nc1c(C(=O)NC2(CO)CCN(C(C3CCCC(F)(F)C3)=O)C2)cccc1F C1(CC(=O)NC2CN(C(CCCN(C(C)C)C)=O)C2)CCN(C(N)=O)CC1 c1(OC)ccc(OC)c(CCC(=O)NCC(C)(C)NC(=O)CCC2CC2C)c1 c1(SC)ncc(C(=O)NC(C)(C)CNC(c2cc(-c3csc(C)n3)c[nH]2)=O)n1C N1(C(c2cnn(CC(F)F)c2)=O)CCC2CN(C(C3C4CCCC34)=O)CC2CC1 C#Cc1cccc(CC(N2CCC(C)C(NC(c3cc(O)nc(O)n3)=O)C2)=O)c1 C1(NC(C23C(CN(C(CCNC(COC)=O)=O)C2)C3)=O)CCN(C)CC1C Cc1cc(Br)ccc1CN(C(C1COCCN1Cc1cc(F)ccc1O)=O)CCO C(=O)(CS(=O)CC)NC(CC=C)C1CC1.O1NC(=O)C2CC2C1 c1(C(N2C(C(=O)OC(C)(C)C)CC(C)(C)C2)=O)nnn2c1CC(C)(C)C2 c1(N2CC3CC(NC(C4(C)CC4(F)Cl)=O)C3C2)nc(Cl)nc2c1CCC2 C1(C(=O)NCCC2(CNC(CSCCOC)=O)CC2)COC2(CCC2)CO1 N1(C(C)=O)CCCC(C(=O)NCCOC2CN(C(=O)C(n3ccnc3C)C)C2)C1 C1(C(=O)NCc2c(C(N(CCC(O)CO)C)=O)[nH]cc2)CC(=O)CC(=O)C1 N1(C(C23C(CN(C(CCC(=C)C)C)C2)COC3)=O)CCN2CCN(C)C(=O)C2C1 C(=O)(C(C(=O)N1CC2C(NC(c3cc(C(C)C)no3)=O)C2C1)C(C)(C)C)OCC N1(C(c2cncc(SC)c2)=O)CC(C)C(C)(CNC(=O)C=Cc2cn(C)cn2)C1 C#Cc1cc(C(=O)N(C2CCCC23CCCO3)C2CC3CNC2C3)ccc1C N1(C(C2CCCN(C(CCCC)C)CC2)=O)CCCC(O)(C(F)(F)F)CCC1 C1(C(=O)NCCC(C)O)CCCCN(C(=O)C(F)CC2CCOC2)C1 CCC(CCCO)NC(=O)N(C)CC1CC1(F)F Cc1cc(OCCC(=O)N(C(CNC(=O)C(C)O)C2CC2)C)c(C)c(C)c1 C(=O)(C(F)CC(C)(C)NC(=O)CC(O)C(C)C)N(CC(=O)NC)C C(=Cn1cccn1)NC(C1C(SC)CC1)=O c1(C(N2CC(C)C(NC(=O)COCc3ccccn3)C2)=O)c(O)ccc(Cl)c1O N1(C(Cc2c(C)noc2C)=O)CC(NC(=O)C(C)N(C)C)C2(CCC2)C1 N1(C(Cn2cc(-c3cnc(OC)s3)nn2)=O)CC2CSCC(C2)C1 CCC(O)C(=O)NCCN(C(C1CCCC1OC)=O)CC C(=O)(C(F)CCC(C)(C)C)N(CCCNC(CCc1cccc(C)c1)=O)C1CC1 C1(C(C)NC(Cc2scc(C)c2)=O)CN(C(C2CC(C(C)C)C2)=O)CCO1 N1(C(COC(CC)C)=O)CC2(CC(NC(=O)C=Cc3ccc(C(F)F)o3)CO2)C1 c1(C(N2C(C)CC(NC(C(CC(=C)C)NC(C)=O)=O)C2)=O)cnc2ccccn12 CCCC(C(=O)NC(CC)C(=O)NC1CC(C)(O)C1)NC(C)=O C=CCCCCCC(=O)N1CCCC(NC(C2CC2(C)COC)=O)C1 c1(CC)ccc(F)c(C(=O)NC2(CNC(c3ccc(C#N)cc3)=O)CCCC2)c1 c1(OC)ncnc(C(=O)NC2(C)CN(C(C3CCOC3=O)=O)C2)c1F C1(C)(COC)CCCN(C(=O)C(C(C)(C)C)NC(=O)C(C)NC(C)=O)C1 c1(N2CCN(C(CC(CC)C3CC3)=O)CC(O)C2)nc2cccc(F)c2o1 N1(C(C(C)OCCOCC)=O)CCC(CNC(c2cnc(O)o2)=O)C12CC2 C1(CNC(C(C)Cc2cnc[nH]2)=O)CC2(CCC2)CN1C(c1c[nH]c(=N)o1)=O C(C(C(=O)NCC(O)CCNC(=O)Cc1nc[nH]n1)N(C)C)N(C)C n1(CCCC(=O)NCCCC(C)NC(c2c(CC)n[nH]c2)=O)ccccc1=O C1(C(=O)NC2(C)CCN(C(c3c(C(C)C)scn3)=O)CC2)CC2(C1)CC21CCC1 c1(C(COCC(=O)NCC#CCNC(C2C(C(=O)OC)CC2)=O)C)ccccc1 CC1CN(C(c2nc(O)[nH]c(=O)n2)=O)CCN1C(=O)CCC1CC1(C)C c1(CCC)c(NC(C2CN(C(=O)CSC(C)C)CC23CC3)=O)[nH]c(C)c1C(C)=O C(CCCC(C)(C)C)N(C)C(C1CC1OCC(C)(C)C(=O)OC(C)(C)C)=O C1(CNC(C(c2nccc(C)c2)(C)C)=O)C(C)CCCN1C(=O)C(Cl)=CCl C1(CC#C)(C(=O)NCCOCC=C)CCN(C(=O)C=CCOC)C1 c1(OC)cc(Cl)c(C(=O)NC2CC(NC(c3nnc(O)cc3O)=O)C2)cc1OC CCC(F)(F)CC(=O)N1CC2CC2C1C(=O)NCC1C=CCC1 C1(n2cc(CSC)nn2)CC2CCC1(NC(=O)Cc1cncn1CC(=O)O)C2 C1(NC(C(C2CCOC2)OC)=O)CCN(C(=O)CC(C)(C)C#N)C12CCC2 C1(NC(C2(N(C)C)CCCOC2)=O)CN(C(=O)CSc2nc[nH]n2)CC2CC12 N1(CC)CCOC(C(N2CC(NC(=O)C(C)(O)c3ccccc3)CC2CO)=O)C1 CC(C)(C)CCC(C)(c1nnnn1C1CC1)NCc1ncc(Br)s1 c1(C(N2CC(NC(c3ccc(CCC)[nH]3)=O)C(C)C2)=O)nc(O)[nH]c(=O)n1 C1(C(=O)NC2CC23CC(OC)C3)(CC)CCCN1C(=O)C(C1CC1)OCC CC1C(NC(c2ncoc2C2CCC2)=O)CCCN1C(=O)COC1CCCOC1 Nc1cc(C(=O)NCC=CCNC(c2coc3c2CSC3)=O)cc(O)c1 C#CCCC(O)C(=O)NCCCCCN1CCN(C(C2(C(F)(F)F)CC2)=O)CC1 CC(C)C(CCC(=O)NCCC1CC(F)C1)NC(C12CCC(CC1)CO2)=O C1(CCC)(NC(C2CCOC(C)C2)=O)CCN(C(=O)CCCCCSC)CC1 C12C3CC4CN(C1C4C3)C2=O.Cc1nc(C(C)NC(C)(C)C)oc1C c1(NCC2N(C(c3ncc(C)c(C)c3)=O)CCC2)ncc([N+](=O)[O-])cc1Br C1(C(C(=O)NCCC(C)N(C(CCOC)=O)CC(F)(F)F)O)CCCCCC1 C(=O)(CCCC(=O)NC1CCN(C(c2nc(CO)n[nH]2)C)C1)OCC c1(C(C)NC(C2(CC)CN(C(c3cnn(C4CC4)c3)=O)C2)=O)cccnc1F c1(C(=O)NC(CCNC(c2c(C)con2)=O)C)c(S(N)(=O)=O)ncn1C C(=O)(C1=CCC2CCC1N2C(=O)CCc1cccs1)NCCCCS(C)=O N1(C(CN(S(C)(=O)=O)C)=O)C2CCC1CC(NC(=O)CC1CCOC1)C2 C1(C)(C(=O)NC(C2CCN(C(C3(CO)CCCO3)=O)C2)C)CS(=O)(=O)C1 CCC(CC(F)(F)F)C(=O)NCC12CC1CN(C(c1cc3n(n1)CCO3)=O)C2 C(=O)(C(O)CCCNC(c1occ2c1CCC2)=O)N(CC(F)(F)Cl)C CCC(CNC(=O)COCC1CCCO1)N=c1ccnc(C2CC2)[nH]1 c1(C(=O)NC2CC(O)(CNC(C(CC)N(CC)CC)=O)C2)cncc(C)c1 C(CS(=O)(=O)CC1=CCN(C(=O)Cc2nnc(-c3ccccc3)o2)CC1)OC c1(C(=O)NCCOCCN(C)C(C2SC3C=CC2CC3)=O)nc2ccccc2[nH]1 CCC(C(=O)NCC1CC(NC(=O)CCCOCCOC)C1)ON C1(OC2CN(CC(C(=O)OCC)C)C2)CCN(C2CN(C)C2)CC1.C1(=O)CO1 C(CCC(O)CO)N(C)C(C1(CNC(=O)C(=O)NCC2CC2)CC2(CC2)C1)=O NS(=O)(=O)C1CNC2(CCCC2)C1.C1(NCC2CC2)C2Cc3cc(F)ccc3C12 CC(C(=O)OC(C)(C)C)C(=O)N1CC(F)CC1CNC(c1ccccc1F)=O c1(C(=O)NCC2N(C)CCN(C(=O)CCCC(F)F)C2)c(F)c(F)cc(F)c1F c1(C(=O)NC(CC)CN(C(=O)C(C)C(CC)CC)C)cc(S(C)(=O)=O)ccc1O C1(NC(C=CCNC(c2ncc(OC)nc2)=O)=O)CCCCNC1=O CN=c1[nH]cc(C(=O)NCC(CO)NC(=O)CNC(c2ccc(OC)nc2)=O)o1 C1(CNC(C2CC(OC)C2)=O)CCC(NC(C2CCC(=O)C2)=O)CC1 C1(OC)(CNC(=O)Cc2c(C)cnn2C)CCN(C(c2cccnc2)=O)CC1 C1(C2CCN(C(=O)Cc3c[nH]nc3O)C2)(NC(C2CCCO2)=O)CC1 c1(C(N2C(CN(C(C(C=C)O)=O)C)CCC2)=O)cc(C)n(-c2ccccc2Cl)n1 CC(C)S(=O)(=O)C(C)C(=O)N1CC(NC(=O)C(C)(C)c2ccsc2)CC1CO CCC(C)(F)C(=O)NC(CNC(=O)COCc1cccc(C)c1)C1CCC1 Cc1c[nH]c(CC(N)=O)c1C(=O)N(CC(C)CNC(=O)CC1CC(C)(C)CO1)C c1(N(C(C2CCC(CNC(CSCCC)=O)CC2)=O)C)cc(C)ccc1F C1(OC)CCC(C(=O)NCc2ccc(CNC(=O)Cc3csnc3C)cc2)CC1 c1(C(=O)NCC2C3CN(C(C(CCSC)O)=O)CC32)cc(C)c(C)c(C)c1 N1(C(C(C2CC2)OCC)=O)CCCC1(CNC(C1(Cl)CC1)=O)COC N1(C(C2N(C(c3cnc(C)o3)=O)CCCC2)=O)Cc2ccc([N+](=O)[O-])cc2C1 c1(C(=O)NCC(C2CC2)NC(C(C)CF)=O)cccc(-c2cccc(Cl)c2)c1 N1(C(C2(C)C(C)CN(C(c3ccccc3)=O)C2)=O)Cc2cccc(O)c2C1 c1(C(N2CC(NC(CC(C)CF)=O)C(O)CC2)=O)ccc2nc(S)oc2c1 C1(CNC(C(CC)C)=O)CCN(C(c2c(C)nn3ncccc23)=O)CC1C1CC1 C1(NC(=O)CC2C=CCCC2)CN(C(c2nocc2Cl)=O)CC1C(F)F C1(CNC(C(=O)NCCNC(C)=O)=O)CC2CCC1N2C(C1(CO)CC1)=O c1(C(=O)NCCCNC(CN(c2ccc(Cl)cn2)C)=O)cc2sccc2s1 C1(COC)(CNC(C2CCC2C(=O)COC)=O)CN(C(=O)OC2CCCCC2)C1 CCC(CCc1ccccc1)C(=O)NC1CCN(C(C2CC(OC)C2)=O)C1 Cc1cc(=NCCC(O)CCN(C)C)[nH]c(NC(c2ccoc2)C)n1 c1(CN2CCN(CC(=O)NCCC)CC2)cc(S(C)(=O)=O)ccc1F C1(CCC)CN(C(c2c[nH]cc2C(C)C)=O)CC1NC(=O)C=CCn1cncn1 c1(NC(C(=O)NCCSCC#C)=O)ccc(C(C)O)cc1 C12(NC(C(=O)NCC)=O)CC1CN(C(C1(C)CCNC1=O)=O)C2 C1(CNC(CC(C=C)c2ccccc2)=O)CC2(CO1)CN(C(C1CCC1)=O)C2 c1(C(=O)NC(CNC(C(CCOC)(C)C)=O)C)ccc(F)c(N)c1F C1(C(C)(C)C)CCCC(NC(C2CCCN2)=O)CC1 N1(C(=O)CS(=O)(=O)NC2CC2)CCCC2(CCCN2C(c2cnc(S)nc2)=O)C1 N1(C(Cc2cc(OC)no2)=O)CCC(CNC(C2CCCN2N=O)=O)C12CCC2 C(=O)(C(CNC(c1ccccc1C)=O)C(C)C)NCc1onc(C)n1 n1(CC)cnc2c(NCC3CNC(=O)C3)[nH]c(=NC3CCCC3C(C)C)nc12 c1(N2CCC(C#N)C2)nccc(=NCCOCCCSC(F)F)[nH]1 N1(C(COC(CC)C)=O)CCCC2(C1)CN(C(c1cc(Cl)c(F)cc1Cl)=O)C2 Cc1cnc(O)c(CNC(=O)COC2CN(C(C3C=CC=CC=C3)=O)C2)c1 c1(C(=O)NCC2C(NC(C(C)CC3CC3)=O)C2)ccc2c(n1)OCC(=O)N2 c1(CC(C)NC(c2cc(C3CC3)ns2)=O)c(Cl)cccc1Cl Cc1sc(C(=O)NC2CC(Cc3nn[nH]n3)C23CCC3)cc1S(N)(=O)=O N#Cc1ccc(F)cc1C(N1CC(NS(=O)(=O)c2cn[nH]c2)C(F)(F)C1)=O N1(C(C2(C)CN(C(CC3ON=C(C)C3)=O)C2)=O)CCN(C)CC1CCO c1(CCC)cc(C(N2CCC(O)(CNC(C3(OC)CCSCC3)=O)C2)=O)nn1C N1(C(C#CC(C)(C)O)=O)CCC2(CCC(CNC(=O)CC3CC4(CC4)C3)O2)CC1 CCCCC(C)(F)C(=O)NCC1COCCN(C(=O)C(C)(C)F)C1 N1(C(c2nc(C)[nH]n2)C)CCC(C2CCN(C(c3cc(F)ccc3F)=O)CC2)C1 N1(C(C)=O)Cc2ccc(S(=O)(=O)N3CCOC4COCC34)cc2C1 O=C1Nc2cc(C(=O)NCC=CCNC(=O)C=C(Cl)Cl)ccc2C1=O S(=O)(=O)(c1cc(C(=O)OCc2cn3cc(Br)ccc3n2)ccc1F)N(C)C C12(C(=O)NCCC(C)NC(C3CC(F)(F)C3)=O)COC(CS(C)(=O)=O)(C1)C2 N1(C(c2c(C)ccn2C)=O)CCCN(C(=O)Cn2[nH]cnc2=N)C(CO)C1 c1(CCNC(c2snc(OC)c2Br)c2nnnn2CCCF)cccc(Cl)c1F CC1CN(C(C2CC(F)(F)C2)=O)CC1CNC(C1(n2cccn2)CCC1)=O c1(NC(C)=O)ncc(C(N2CCCC2CNC(C2CN(C(C)C)C2)=O)=O)s1 C1(NC(c2cc(Br)c(C(F)F)o2)=O)CC2(C1)C(C(=O)O)C2(F)F C1(N(C(C=Cc2nc(C)sc2)=O)C)CC2CC1N(C(C1CC(O)C1)=O)C2 CCCC(C(=O)NCC(Cl)Cl)NC(=O)CC1(N(C)C)CCC1 C1(C(N2CC(C)C(NC(c3cc(C(C)(C)C)on3)=O)C2)=O)CCc2ccnn2C1 C(N=c1cc(C(C)(C)C)nc(Cl)[nH]1)C1CC(NC(CN(C)CC)=O)C1 C1(N(C(=O)COc2ccsc2)C)CCC(CNC(=O)CNC(=O)C(C)(C)C)CC1 c1(NCC(CCNC(N(C)CC)=O)O)nnc(Cc2ccc(F)cc2)n1C C(c1c(Cl)nc2ccccn12)=CC(=O)NC1CN(C(C=CC(C)(C)C)=O)CC1F n1(CC(=O)N(C(C)C(=O)NC(c2noc(C)n2)C)CC)ncccc1=O c1(CCC(=O)NC2CCN(C(Cc3nc(C)[nH]n3)=O)C2)nc2cccc(Cl)c2[nH]1 CC1=CCCN(C(=O)CCC2(NC(=O)Cn3cncn3)CCCC2)C1 C(CC(C)(C)C)(C(=O)NC(CC(N)=O)C(=O)NCC(C)Cn1cccn1)OC c1(CC)nn(C)c(CNC(C(c2ccc(Br)cc2)(C)C)c2nnnn2C)c1Cl c1(CC(=O)NCC2C3CCC2CN(C(C2CC2CF)=O)C3)c[nH]c2ccccc12 C1(C(=O)NC2CCC(NC(C3(CC#C)CCCCC3)=O)CC2)CNC(=O)CC1C c1(C(N2CCCC(N(C(c3cc(SC)oc3)=O)C)C2)=O)cccc2nc(O)[nH]c12 COn1cnc(C)c1C(=O)N(C)CC1CCN(C(C2(C)COC(=O)C2)=O)C1 c1(OC)ccc(CC(=O)NCC2CCN2C(c2cc(C)no2)=O)cc1 c1(C(=O)NC(C2CCCN(C(c3c[nH]c(=NC)o3)=O)C2)C)c(C)ccc(C)c1C Cc1nc(C(C)C)ncc1C(=O)NC(CO)C(C)NC(=O)CC1C=CCCC1 C#CC(C(=O)NOC(CC(C)C)C(N1CC2CC(OCC)C(C2)C1)=O)C(C)C N1(C(C(CCC)OC)=O)CC(NC(=O)C=C(Cl)Cl)CC2(CCC2)C1 c1(C(N2CCC(NC(c3c(C)cno3)=O)C(O)C2)=O)c(F)c(F)c(F)c(F)c1F c1(OC)cc(C(=O)NCC(C)(C)CCNC(c2ccco2)=O)cc(F)c1 CC1CN(C(c2c[nH]nc2Cl)=O)CC(C)C1NC(C1Cc2ccccc2C1)=O C(C(C)C(=O)NC1CC(CCNC(=O)C(C)OCC(F)(F)F)C1)OCC c1(OCCCC(=O)NCc2ccc(OCCC)nc2C)c(Cl)cccc1[N+](=O)[O-] C(=O)(C(C)(C)CNC(=O)CC1CC(C)N(C(=O)C(C)=NOCC#N)C1)NCC C1(CC(=O)NCC2(OC)CN(C(=O)CCC#N)C2)CCCC12CC2 c1(N2CC(C)C(NC(c3c[nH]c(C(N)=O)c3)=O)CC2)ncc2c(Br)cccc2n1 c1(OC)ccc(F)c(C(=O)O)c1.c12nnc(o1)CNC(=O)C1CN(C1)C(=O)CC2 CCCCC(F)C(=O)NC(CC)CCC(=O)N1CC2CCC=CC12 CS(=O)(=O)CC(=O)N1CCC(n2cc(CC3CCC(C)(C(=O)ON)O3)nn2)C1 c1(C(N(C(C)CNC(c2ccc(O)cc2F)=O)C)=O)cc2ccc(Cl)nc2s1 CP(C)(=O)CCC(=O)NCC(CNC(=O)C(c1cccc(F)c1)O)CO N1(CCN)CC2(CCN(CN3C(=O)CSC3=S)CC2)CC1Cc1ccccc1 C1(N=[N+]=[N-])(C(=O)NCC(CC)(O)CC)CCN(C(C2CCC(F)(F)C2)=O)C1 N1(C(C(=O)NC(C)C)=O)CC2(NC(=O)CC3(C)OCCO3)CCC1C2 CCCC(CNC(=O)CCc1cncs1)C(=O)NC1CN(C)CC1(F)F N1(C(C=CCC)=O)CC(OC)C(NC(=O)COc2cccc(-n3cnnc3)c2)C1 C=CCC(F)(F)C(=O)NCCOCCC(=O)NCc1ncccc1C Cc1ccc(C(=O)N(CCCNC(C2CC(=O)N2)=O)Cc2ccccc2)cc1N N1(C(c2c(C)cns2)=O)CC(NC(C2CCOC2c2ccncc2)=O)C(C)(C)C1 Cc1cc(CCC(=O)NCC(F)CNC(c2c(C)nsc2N)=O)cc(C)c1 Cc1cc(C(=O)NCCC2CCCN2C(=O)Cc2cn[nH]c2)c(C)n1CC1CC1 CCC(CC)(CC)C(=O)N1CCC2(NC(C3CCCN3C(C)=O)=O)CCCC12 c1(C(=O)NCC(CNC(Cn2nc(C)n(CC)c2=O)=O)F)cc2ncccc2[nH]1 CS(=O)(=O)C1CCN(C(C2C3COCC23)C(=O)NCC2CCCO2)C1 Cc1ccc(Cl)cc1OCC(N1CCCC(NC(=O)CN(C2CCC2)C)C1C)=O CCC(CC(=O)N1CCC(O)(NC(C(=O)NCC=C)C)CC1)C(C)C C1(NC(Cc2cnc(C)s2)=O)CC(C(=O)N(C2CC2C2CC2)C)C1(C)C O=C1Cc2cnc(N3CCCC(CNC(c4ccc(F)cc4I)=O)C3)nc2N1 CCC(CC(=O)NC(CO)C1(C)CC1)NC(c1cc(CO)c(C)o1)=O C(=O)(C1=NOC(CNC(c2sccc2Cl)=O)C1)NC(CC)(C)C1CC1 Cc1ccc(C(=O)NC23CC(C2)N(C(C2SCCC2C)=O)C3)cc1N c1(OC)cc(NC(N2CCCC3(C)CCCCC23)=O)cc([N+](=O)[O-])c1C C12(NC(COCCC)=O)CCOCC1CN(C(=O)CN(C1CCC1)C)C2 N1(C(c2ncc(CC)cn2)=O)CCC2C(CCCN2C(C2COCCO2)=O)C1 CC1=C(C(=O)NC2CCCN(C(c3ccsc3Cl)=O)C2C)CCC1 c1(CC)nc(C)oc1C(=O)NCC(CC)(CC)NC(=O)C(C1CCCCC1)O CCC(C(=O)N1C(C)C2CC1C2NC(=O)COc1cc(C)on1)C(F)(F)F c1(OC)ccc(C(=O)NCCN(CC(C)O)C(c2ccsc2C)=O)c(OC)c1 CC(C)CC(C(=O)NC1COCCC1NC(c1cnn(CC2CC2)c1)=O)C(C)C Cc1nccc(C(C)NC(C2CCN(C(c3cncc(F)c3)=O)CC2)=O)n1 CCCC(C(O)C(=O)NCc1cn[nH]c1)NC(=O)CC(F)(F)C(F)F C=CC1(C(N2CC(CNC(C3CC(C#N)(OC)C3)=O)(COC)C2)=O)CCOCC1 c1(N(CC(C)NC(=O)C(C2CC2)C2CC2)C)nc(C#N)c(Cl)s1 c1(C(N2CCCCC(CNC(C3(CC(C)C)CC3)=O)C2)=O)ccc2occc2n1 CCCC(CC)C(C(=O)NCC1(C(=O)OCC)CC1)N1CCS(=O)(=O)CC1 C(C1CN(C(C2CCC(=O)O2)=O)Cc2ccccc21)NC(CCC=C(C)C)=O Cc1c(CC(=O)NCC=CCNC(C2CCN3CCCC3C2)=O)cccc1[N+](=O)[O-] N1(C(C(C)OC)=O)CCC(C(=O)NC2CCCCC2(F)F)C(C)C1 c1(N2CCC(C(C)(C)C)(CNC(c3ccc(F)nc3)=O)C2)c(F)cccc1[N+](=O)[O-] CN1CCC(CNC(C2CNCCN2Cc2ccnc(Br)c2)=O)CC1 N1(C(CCC#C)=O)CC(NC(c2ccc3nn[nH]c3c2)=O)CC12CCOC2 c1(CNC(CCN(C)CCO)=O)cn(CCNC(=O)CSCC(F)(F)F)nn1 C1(CCNC(C2(CCCC)CC2)=O)CN(C(c2cncn2C)=O)CC(C)O1 c1(CCC(=O)NC(CN(C(c2cc(C)c(C)s2)=O)C)C)ccc2cnccc2c1 Cc1nc(=N)[nH]c(C)c1C(N1CC(NC(C2COCC2(C)C)=O)CCC(O)C1)=O CC(C(=O)NCC1CC1NC(c1cn(C2CCOCC2)nn1)=O)C(F)(F)F CCC(CC(=O)N1CCC(NC(c2cnc3[nH]ccc3n2)=O)C(C)C1)C(C)C N1(C(C(CC(=O)OC)C)=O)CC2CC1CCC2NC(c1ccc(C2CC2)s1)=O Cc1ccc(Br)cc1CC(=O)NCCC(C)CCNC(=O)Cc1cc[nH]c1 N1(C(C(C)CC(N)=O)=O)CCCCC12CN(C(=O)C(C)(C)CO)C2 c1(C(=O)NCC2OCCN(C(c3cnc(OC)s3)=O)C2)ccc(Cl)c(F)c1N Cc1nnccc1C(=O)N(C)CC1COCCN1C(=O)CN1C(=O)CNC1=O C1(NC(=O)C=Cc2cocn2)C2CCC1N(C(C1(C3CCCO3)CCCC1)=O)C2 CCS(=O)(=O)CCNC(c1ccc(Cn2cc(CC(C)(O)CC)nn2)cc1)=O c1(-c2nc(CC)on2)cccc(C(=O)NC2CCC(CN=c3[nH]ncs3)C2)c1 Cc1ccc(C)c(C(N2CC(O)(CCNC(=O)CC3CC(C)C3)C2)=O)c1 C(=O)(C(F)C(F)(F)C(F)(F)F)N(c1ccc2c[nH]nc2c1)CC c1(CN(N2CCCC2)CCOC(=O)Nc2cn(C3CC3)nn2)c(F)cccc1Br c1(N(S(CC(C)c2ccccc2)(=O)=O)C)ccc(F)cc1Cl N1(C(C(C)C(F)(F)F)=O)CC2OCCN(C(c3cn(C)[nH]c3=N)=O)C2C1 N1(C(C2CC(NC(C(CC=CC)CC)=O)C23CCC3)=O)CCn2ncnc2C1 c1(C(=O)NCC2C3CN(C(C(CC)n4nccc4C)=O)CC32)cnc2n1CCS2 C=CCCC(C)(C)C(=O)N1CCN(C(C2CCC(=O)O2)=O)CC1CO C1(C(=O)NC(CC=CC)C(=O)NCc2nc(C)cs2)CCCC(C#N)C1 C(=O)(C(C(C)(C)C)n1ccnn1)N1C(CNC(COCCCCC)=O)CCCC1 C(=O)(C1CCCc2c[nH]nc21)NC1(COC)CCN(C(=O)C(O)C2CCC2)CC1 C1(C(=O)NCC2N(C(C3CCC(C)C3)=O)CC2)CC2CCC1O2 Cc1cn2cccc(C(=O)NC3C=CCN(C(c4cc(C)on4)=O)C3)c2n1 N1(C(c2cc(CC(=O)OC)on2)C(=O)NCC(=C)C)CCCCC1C1CCCC1 N1(C(CCCNC(=O)OC)=O)CC(C(=O)NCc2nc(C)cc(O)n2)CCC1C Cc1nc(C(=O)NCC2CCN2C(=O)Cn2cc(C)c(C(F)(F)F)n2)cc(O)n1 C1(C(N(C)CC2(OC)CCC2)=O)CCCC(NC(=O)CCCc2ncco2)C1 CC1CN(C(c2c[nH]nc2F)=O)CCN1C(c1cc(F)ccc1O)=O c1(CC(OCC)OC)ccccc1C(C)NC(=O)NC12CCCCC1C2 CCC(CC)(CC)C(=O)NC(C)CC(C)NC(=O)COCc1cccc(OC)c1 C#CCC(C(=O)N1CCOC(C2CCC2)C1)NC(=O)C(C)SCC c1(OCC(=O)NCC(C)CNC(=O)C2=CS(=O)CCC2)ccc([N+](=O)[O-])cc1Cl N1(Cc2c(OC)cncc2)C(C(=O)Nc2cc(C)ccc2C#N)CC2CCCCC12 c1(C2C(C(N3CC(C)(NC(c4c(C)cno4)=O)C3)=O)C2)ccc(Cl)cc1 N1(C(CCCSC)=O)CCCC(C2(NC(C3(C)CC3Br)=O)CC2)C1 c1(OC)ccc(N)c(C(=O)NCC2CC(NC(C3CC3(C)C(C)C)=O)C2)c1 c1(OC)cc(-c2cn(CC(C)NC(c3ccc(CS(C)(=O)=O)o3)=O)nn2)sn1 c1(C(N2CCC(NC(C(CC)C3CCOCC3)=O)C2)=O)ccc(O)cc1C c1(NC(CC(CC2CC2)NC(C2C(=C)C2)=O)=O)c(C)cc(O)cc1C C1(N(C(c2ccc(C(C)C)o2)=O)C)CN(C(C2CCCOC2)=O)CC12CC2 CC(C)(C(=O)NC1CC(CNC(=O)C(C)(C)N(C)C)C1)NC(=O)C(F)(F)F C12(C(N(CC(CNC(c3n(C(C)C)cnc3)=O)O)C)=O)CCOC1CC(=O)NC2 C=CCC(CC(C)C)C(=O)NCC(C)(F)CNC(=O)CCC(=C)Cl c1(CSC)nc(C2CC2c2ccccn2)n(-c2cncc(Br)c2)n1 C1(C)(NC(CCSC)=O)CCN(C(=O)CCCC2CCCC2)C1 CS(=O)CCC(=O)NCCC1CCN(C(=O)C=CS(C)=O)CC1 N1(C(c2c(OC)cc(F)cc2)C(=O)NC2COC2)CCN2C(=O)CCC2C1 c1(SC(C)C(N2CCC(CN(CC(=O)NCC(F)(F)F)C)C2)=O)ccccc1 C(=O)(C1=CC2C=CC(C1)C2)N1CCCCC(NC(c2ccc3occc3c2)=O)C1 C1(C#N)(C(=O)NCCC(C)(C)NC(CCCCOC)=O)CC12CCC2 Cc1nccc(C(N2CCC(C)C2CNC(c2ccnn2C)=O)=O)c1O C1(NC(CC=C)=O)CCC(NC(c2sccc2I)=O)CC1 CCC(C)(F)C(=O)N(C)CC1CCN(C(c2c(Cl)cnn2C(C)C)=O)C1 C1(C(=O)NCC2CN(C)C2)CN(C(c2cc(Br)nc(Br)c2)=O)CC(F)(F)C1 CC1C(NC(=O)CCC2CC(C)(C)CO2)CCCN1C(C1CC2(CSC2)C1)=O c1(OC)ccc(NC(c2c(-c3ccc(SC)c(F)c3)cncc2F)=O)c(C)c1C c1(C(N(C(C)CNC(c2ccc(CO)c(F)c2)=O)CC)=O)ccc(C)c(O)n1 C1(NC(c2ccc(N(C)CC)cc2)=O)CCN(C(c2cc(F)c[nH]2)=O)CC1CO CC(CN=C(NCC1CCCC2(CC2)C1)NC1CCCC1)OC(C)(C)C C(=O)(CC(C)CNC(=O)Cn1ncccc1=O)NC(C(CO)SC)C N1(C(CCCC=C)=O)CCCOC(CNC(=O)CC(OCC)OCC)C1 CC(C)CS(=O)(=O)CCC(=O)NC(CNC(c1ccccc1N(C)C)=O)C1CC1 c1(CC)ncc2c(n1)CCC(C(=O)NC1CC1NC(C1CC(OC(C)=O)C1)=O)C2 CC(CC(=O)N1CCCOC(CCNC(=O)C(C)(Cl)Cl)C1)C(F)(F)F CC(C)CCCCC(=O)NC1CCCC(NC(=O)Cn2ncccc2=O)CC1 c1(OC)nc(N2CC(O)(CCNC(c3cc(C4CC4)no3)=O)C2)nc(C)c1F Cn1cc(C(F)(F)C(=O)NCCC2(C(=O)NC3CCS(=O)(=O)CC3)CC2)ccc1=O C(=O)(C1(C)COc2ccccc21)NCC(C)NC(C=Cc1cnc(OC)nc1)=O C1(C(=O)NC(C)(C)C(F)(F)F)CN(C(C2CCCN2C=O)=O)CC12CC2 c1(NC(C2CN(c3ncc(F)cn3)C2)=O)c(O)cccc1[N+](=O)[O-] C1(C(=O)NC(C(C)NC(c2c(OC)nsc2)=O)(C)C)CCCCCCC1 CC(C)CC(CNC(C1(CO)CCCC1)=O)NC(C1(Br)CC1(F)F)=O c1(C(=O)NC2CC(NC(c3ccc(C=C)cc3)=O)C2)ccc2c(c1)C(=O)CCS2 C=C=CCCC(=O)NC1CC1CNC(C1CC(F)C1)=O c1(C(N2CCN(C(Cc3ccc(C)cc3Br)=O)CC2)=O)cc(C)nc(C)c1O C12(NC(c3cncnc3)=O)CC1CN(C(c1ccccc1)=O)C2.C1(=O)CCCO1 n1(CC(N2CCC(OCCNC(C3C(C)N(C)CC3)=O)C2)=O)nc(Cl)ccc1=O N1(C(c2c(C)ccc(C)c2)=O)CCCN(C(=O)CC2CC2(Cl)Cl)CCC1 C1(NC(C=CCC)=O)CCN(C(=O)CSc2ccc(C#N)cc2)C(C2CC2)C1 C12(NC(C(C)N3CCC3)=O)CCCN(C(=O)CN(C)Cc3ccccc3)CC1C2 C1(NC(c2c(C)cc[nH]2)=O)CN(C(C2CC=C(C(C)C)CC2)=O)CC2CCCC12 c1(OC)ccc(C(=O)N(CCCCN(C)C(c2ccoc2)=O)C)c(F)c1Cl c1(OC)ccc2c(c1)CC(NC(=O)C(=O)NCc1ccc3ccsc3c1)CCC2 CC1CCCC1(O)CNC(c1cccc(C(=O)N(C)C)n1)=O C(=O)(C(F)C1=CCCCC1)NC1(CNC(C(C)=O)=O)CCCCC1C N1(C(CSCCCC)=O)CCC2(CC1)COC(CNC(=O)C1=NOC(C)(C)C1)C2 c1(NCC(N2CCCC(C)(CNC(C3C(CC)C3)=O)C2)=O)ccccc1[N+](=O)[O-] C1(SCc2nnc(-c3cn(C)nc3)o2)CCC(O)CN1C(=O)OC(C)(C)C CCC(CC)CC(=O)N1C2CC1CN(C(C1(C(=O)OCC)CC1)=O)C2 C(=O)(C1CCCc2ccccc21)NC1(CNC(=O)CC2(O)CCOC2)CC1 C(CO)(CCCCNC(C1C2CC3C(C2)C13)=O)NC(C1(CC)CCCC1)=O c1(C(=O)NCC2(C)N(C(c3sc(C)c(O)n3)=O)CCC2)cc(F)cnc1Cl CC1(NC(c2ccncn2)=O)CCCCC1C(=O)NCC1(CO)CCC1 N1(C(C=CC(CC)C)=O)CCC(CNC(c2cnc(OC)s2)=O)(COC)CC1 CC1C(=O)N(CC(=O)NCC2(NC(c3cnn[nH]3)=O)CC2)C(=O)C1C N1(C(c2ccc(C)c(Cl)c2)=O)CC2(NC(=O)C(C)C(C)(F)F)CCC1CC2 N1(C(c2c(C)oc(CO)c2)=O)CCN(C)C(C(=O)NC(C2CCOC2)(C)C)C1 C1(C(=O)NCCC(=O)NCC(C)C)CSCCN1C(=O)Cc1cncnc1 C1(C(=O)NCC2CCC(NC(=O)COC3CCOC3)C2)C(C(F)(F)F)C1[N+](=O)[O-] CCC(C(=O)OC)C(=O)N1CC(CCCCNC(C2CS(=O)(=O)CCO2)=O)C1 C1(F)(CNC(=O)CC2CCO2)CCCN(C(=O)CCc2cn[nH]c2)CC1 N1(C(Cn2c(C)nc(C)n2)=O)CCC(NC(=O)CC2CCCOC2C)C12CCC2 Cc1cc2c(C(N3CCC4CN(C(C5CC5(C)C)=O)C4C3)=O)ccc(C)c2[nH]1 C1(C(=O)Nc2ccc(F)cc2O)CCc2nc(-c3ccc(F)cc3)sc2C1 Cc1c(O)c(=O)ccn1CC(=O)NC(C)(CNC(=O)C(F)CC1CCC1)CO N(C(=NCC(F)F)NCC1(C)CCC(C)CC1)C1C(C=C)OCC1 C=CCCCCCC(=O)N(CC(=O)NC(C)CC1CCCO1)CC1CC1 c1(CC(=O)NCC(C(C)C)NC(c2cccc(F)c2)=O)ccc(C(N)=O)cc1 c1(C(=O)NCC2(F)CCCN(C(CCCNC(N)=O)=O)C2)ccc2nn[nH]c2c1 c1(CCNC(c2nnnn2Cc2ccco2)C(C)C2CC2)ccnc(Cl)c1 c1(N2C(CNC(=O)C3=CCCOC3)CC(F)C2)ncc2scc(Br)c2n1 c1(C(=O)NCC2(CNC(C(=Cc3ccccc3)OC)=O)CC2)cc(O)cc(=O)o1 C(CN=C(NC1CCOCC1)NC1CCOC(C)C1)c1ccc(C)cn1 C(CCCCC(=O)NCC(C)(C)C(=O)Nc1ccc(C(N)=O)cc1)=CC N1(C(c2ccc(C)s2)=O)CCN(C(C2CCC(c3ccccc3)C2)=O)C(C)C1 c1(OCC(=C)C)ccccc1CN1CCCC(CCNC(c2cc(Br)n[nH]2)=O)C1 C1(N(C(=O)C=CC2CCCN2C(=O)CN2CC=CC2)C)CCCC(O)CC1 c1(CN2CCN(C(c3cccc(OC)c3)C(=O)OC)CC2)ccc(OC)cc1F C1(C(N(CC(CNC(C2(OC)CC2)=O)O)C)=O)C=C(C)CS1 C1(C(N(CC#C)Cc2ccco2)=O)CCN(C(=O)COc2ccn(C)n2)CCO1 N1(C(C2(CCCC)CC2)=O)CC2CC(NC(c3coc(Cl)n3)=O)C1C2 C1(C(=O)NCC(c2ccnc(C)c2)NC(C2C(C)=CCS2)=O)CCc2nnnn2C1 C1(CNC(CC2C=NN(C)C2=O)=O)CCCCN(C(=O)C=CC2(C)COC2)C1 CCCCC(CNC(=O)CCc1ccon1)NC(=O)CC12CC(C1)C2 C(=O)(CC(CC(C)C)NC(c1scc(C)c1C)=O)NC(CC)Cn1cncn1 C(CN=c1[nH]cnc2ccc(F)cc12)(C1CCCC1)NC(c1ccc(Cl)o1)=O Cn1cc(C(=O)NCCC(C)(C)CNC(c2cnc(O)c(F)c2)=O)ncc1=O C1(NC(=O)CC2CC(F)(F)C2)CC(F)CN(C(=O)CCSCc2ccccc2)C1 n1(CC(C)(C)C)nc(-c2cccc(CN3CCCCC3)c2)nc1C1CCOC1 C(=O)(C(C)(C)CS(C)(=O)=O)NCC(C)CNC(c1cc[nH]c(=N)c1)=O c1(C(=O)NCCCOCCC(=O)NC(c2ccc(C)o2)CC)ncncc1N Cc1nn(C)cc1C(=O)NC(CNC(c1csc(Br)c1C)=O)C1CCC1 Cn1cc(NC(c2ccc(CCO)cc2)=O)nc1C(=O)NC1CCS(=O)(=O)C1 c1(C(=O)NC(C2CN(C(C(C=C=C)C)=O)C2)C)coc2c1C(=O)NCCC2 CC1(CNC(=O)COCCCF)CCN(C(=O)CCc2cncs2)C1 N1(C(CNC(C)=O)=O)CC2(C1)CN(Cc1ccc(OCC(F)F)cc1)C2 CCCC(CC1CCCC1)C(=O)NC(CNC(=O)C=CC1CCC1)CCCC C#CCC(C(=O)NC1(CC=C)CCC1)NC(=O)COCCOC C1(NC(=O)C=Cc2cncs2)CCN(C(C2CC(F)(CF)C2)=O)CC1 c1(C(=O)NCCN(C(=O)C(C(C)C)C(C)C)CC)cc(Br)c(C)cc1O c1(C(=O)NC(CNC(C(CC)(C)OC)=O)C(C)C)c(C)nc2ccccn12 c1(C(=O)NCC(C)(CO)NC(C2CCCOCC2)=O)cnc(S(C)(=O)=O)s1 c1(CC(=O)N(CCC(C)NC(=O)CC2CCCN2C)C)ccc(F)c(Cl)c1 C1(C(=O)NC(C(=O)NC(Cn2ncc(C)c2)C)CO)CC(=O)C12CCC2 C(CN=c1[nH]c2ccccc2o1)C1CCN(C(CCc2n(C)cnc2)=O)C1 C1(CNC(C(n2ncc(C)c2)C)=O)CC(C(=O)NCCCNC(N)=O)=NO1 C=CC(CC)C(=O)NC1(COC)CN(C(C2(O)CCC2)=O)C1 C(=O)(CC(C)n1ccnc1)N(CC(CC)NC(c1cnc(C2CC2)[nH]1)=O)C C1(C(=O)Nc2ccc(F)c(F)c2)CCC2(CN(Cc3cscc3Br)C2)O1 N1(C(COCCOCC#C)=O)C2CCC(C(=O)NCC(C)(C)SC)C1CC2 c1(C(=O)Nc2cccc(NC(C3N(C)CCOC3)=O)c2)c(N)cc(Cl)cc1F N1(CCOC)CCC(N=c2[nH]c(NCc3cn(C)cn3)nc3cc(C)ccc23)C1 c1(C(=O)NCCCN(C(=O)CC2CCC(C)(C)CO2)CC)[nH]nc([N+](=O)[O-])c1Cl N1(C(C2C(C#C)C2)=O)CCOC2(C1)CN(C(=O)C(CC=C)CC(C)C)C2 Cc1nc2ncc(C(=O)NC3CCN(C(c4ccoc4)=O)CC3CO)c(=O)n2[nH]1 C#CCCC(=O)N(C1CCC1)C(C)CO.C1(N)CC1 N1(C(c2c(COC)ncs2)=O)CC(C)N(C(c2cn(C(C)C)nn2)=O)CC1C CN1CCN(C(=O)N(C2CC2)CC2C(C)(C)C2(F)F)CC1C(C)(C)C c1(C(=O)NCCC2(O)CCN(C(c3c[nH]c(=N)o3)=O)C2)csc2ccncc12 C(CC(C)C)(C(=O)NC1CCCCC1F)N(C(C(C(=O)OCC)F)=O)C C(C)(CCC(=O)NCC(c1ccccc1)NC(C1(F)CC1)=O)OC N1(C(CCCOCCOC)=O)CC(O)C(O)C1CNC(=O)CN(C)C1CC1 c1(CC)cc(C(=O)NCC(CO)NC(=O)CNC(C2CCCCC2)=O)cn(C)c1=O CCCCS(=O)(=O)CC(=O)NC1(CO)CN(C(c2cc(C)c(C#N)cn2)=O)C1 C(CCCCC(=O)NC(CNC(=O)CC(O)CC1CC1)CC(F)(F)F)SC C(=O)(CCC(C)(C)C)N1C(C(=O)NC2(C(=O)N(C)C)CC2)(COC)C=CC1 c1(C(=O)NC2C(NC(=O)CCc3nncs3)CCC2)nncc2c1CCCC2 Cc1ccnc(C(=O)NCCCC2(NC(C3CCN(CC4CC4)CC3)=O)CC2)c1 c1(C(N(C2CCN(C(c3ncnn3C)=O)C2)CCC)=O)cccnc1 C1(C(=O)NC(CCC=C(C)C)C)CC(=O)CN1C(=O)CCn1cncn1 c1(CNC(C2(CNC(C=NOC)=O)CC23CCC3)=O)cnc(O)c(F)c1 c1(NC23CCCC(C(=O)OC(C)(C)C)(C2)C3)nccc(S(C)(=O)=O)n1 N1(C(C(C)C)=O)CCN(C(C2(C(C)C)CCOCC2)=O)CC1CO C(=O)(CC(C(F)F)c1ccccc1)N1CCC(=CCNC(CCC=C)=O)CC1 N1(C(CC=CC)=O)CCC(C2CCC2)(CNC(=O)CC2CCCCC2O)CC1 C1(CNC(C2(SC)CC2)=O)CCCC12CCN(C(c1ccc(F)c(Cl)n1)=O)CC2 CCC(CC1CCCCC1)C(=O)NCC1CC(NC(c2cc(F)cs2)=O)C1 c1(CC(=O)NCC(CN(C(CC2N(CC)C(=O)CC2)=O)C)O)cc(F)ccc1F c1(CC(=O)NC2CN(C(CCOC)=O)CC2O)cc(F)cc([N+](=O)[O-])c1 Cc1cc(N(C)C(C)C)nc(NC(CC(N)=O)c2ccccc2)n1 Cc1ccsc1C(=O)NCC1CC(O)(CNC(c2cn(CCO)nn2)=O)C1 c1(-c2cc(CO)cc(OC)c2)cccc2[nH]c(C(N3CCCC3C(N)=O)=O)cc12 C1(C(C)CN(C)C)CCN(C(=O)C(C(=O)OC(C)(C)C)C2CC2)CC1 N1(C(C(C2CCN(C(c3cc(COC)no3)=O)CC2)C)=O)C2C=CCC1CCC2 c1(NC(C=C(C)C)=O)nc2ccc(-c3cc(C(F)(F)F)cc(F)c3)cc2cc1C N1(C(=O)OC)CCCC(C(N2CCC(O)(CNC(c3ncc[nH]c3=O)=O)C2)=O)C1 C12(NC(CC(C(C)C)O)=O)CCC(CC1)N(C(C1CCC(F)(F)CC1)=O)C2 c1(C(N2CCC(C(C)NC(c3ccc[nH]3)=O)CC2)=O)cc(S(N)(=O)=O)ccc1O C1(CC)CN(C(C2CC3CCC2O3)=O)CCC1CNC(=O)C1=CCCC1C c1(C(=O)NCC2CCCCN2C(=O)COC2CC=CC2)ccc(F)cc1C1CC1 c1(C(N2C3CCN(C(CCCCC)=O)CC3C2)=O)cc2c(C)c(F)ccc2[nH]1 c1(C(C)C)nc(NCc2cc(Cl)ccn2)cc(=NCc2cc(Br)c[nH]2)[nH]1 C(=O)(C(C)CC(=O)NCC1CCCCN(C(c2ccc(CO)c(F)c2)=O)C1)OC C(=O)(C(C)CC(=O)NC(C)CC1CCN(C(c2nccc(Cl)c2F)=O)CC1)OC CC1CCN(c2ncc(O)cn2)C1CNC(C1(C)CC=CC1)=O c1(N(C)CC2CCCC2)ccc(S(=O)(=O)N(C2CC(CO)C2)C)c(Cl)c1 C(=O)(C(C)CC(C)C(C)=O)N1C(CC)C(NC(c2cn(CC)nn2)=O)CCC1 CCC(CC)CCC(=O)NCC1CCC1NC(=O)Cc1cccnc1OC N1(C(c2ccc(I)cc2)C(=O)NC)CC2(C1)SCCC2C(=O)O c1(CN(CCC)C(c2ncc(SC)[nH]2)=O)cc(Cl)ccc1Cl c1(CNC(C(C2CCC2)OC)=O)ccc(C(=O)NCCOCC(F)F)s1 c1(OCC(N2CC3(CC3C(=O)Nc3cncc(Cl)c3)C2)=O)cc(Cl)ccc1Cl CC1CCC(C(=O)NC(Cn2cncn2)C(=O)Nc2ccsc2)CC1 C(CN=c1cc(F)nc[nH]1)NC(C(N1CCNCC1)C)=O C1(C)(C(=O)NCCN(CCC)C(c2cncc(-n3cccc3)c2)=O)CCCN1C C(=O)(C1CCCc2ncnn21)NCC(CC(C)C)NC(=O)C#CC1CCOCC1 c1(CC(C)C)ccc(S(=O)(=O)N(CC(C)NC(C2C3(CC3)C23CC3)=O)C)s1 C1(c2nc(-c3sc(C(=O)O)c(C(F)(F)F)n3)on2)CC12CCCOC2 CCCCC(CC(=O)N1CC(NC(C)=O)C1)NC(=O)C(O)CCN(C)C c1(CC)ccc(NC(=O)C(CNC(=O)C=C(C)C(C)C)CC2CCCC2)cn1 c1(C(N(C(C)CNC(c2ccnnc2O)=O)C)=O)ncc2cc(Cl)ccn12 C1(NC(c2cncc(F)c2)=O)CCC2(CCN(C(=O)C(O)CC(F)(F)F)C2)C1 c1(C(N2CC(C(C(N3C(C)(COCC)CC3)=O)OC)C2)=O)cn(C)nc1C N#CCCCC(C(=O)NCC1CCCO1)N1CC(CO)OC(CO)C1 CCCN=C(NCCSc1cc(C)nc(C)c1)NCC(c1cccnc1)C(C)C C#CCC(C(=O)NCCCOC1CCC1)NC(=O)CCc1cncnc1 C1(C(N2CC(CC(=O)OC)C2)=O)CN(C(=O)C(C2CCOCC2)F)CC(C)(C)C1 N1(C(CCN(CC#C)C(c2[nH]ccc2C)=O)=O)CCN(C)C2CC12 CC(CC(=O)N1CCC2(CC1)CC2CNC(C1(O)CC1)=O)C(C)(C)C N1(C(C=C(C)Cl)=O)CCN(C(=O)CC(C)C2CCCC2)CC1CO N1(C(CNC(N)=O)=O)CCCC(n2cc(CCCN3CCCC3)nn2)C1 c1(C(C)C)c(NC(=O)CCC2CCN(C(=O)C(C3CC3)C3CC3)CC2)cnn1C N1(C(COCCC)=O)CC(C)(CCC(=O)NC(C)Cn2cccn2)C1 CCC(CCC(=O)NC1(c2nc[nH]n2)CCC1)NC(c1n[nH]cc1C)=O c1(C(N2C(CNC(CC=C)=O)CCC2)=O)ccccc1OCC(=C)C c1(C(=O)NCC(C)N(C)C(c2ccc(Cl)o2)=O)cc([N+](=O)[O-])c2ccccc2c1 C1(C2CC2)(NC(CCN(C(C(C)C2CCOC2)=O)C)=O)CCCCC1 CN(C)NC(=O)CCC(=O)N(CC(O)CNC(=O)C=CCOC(C)(C)C)C N1(C(C(CC)=CCCC)=O)CC(CNC(C2(n3cccn3)CC2)=O)C(O)C1 c1(C(=O)NC2CC(NC(=O)Cc3cnccn3)C2)ccc(F)c(C(F)(F)F)c1F C(=O)(C1=C(Cl)CCC(C)C1)N(C1CCC(NC(c2ccc(C#C)nc2)=O)CC1)C N1(C(=O)CCOCC(F)F)CCC2CN(C(=O)C=CC3CCC3)CC2C1 C1(NC(CCSC)=O)CC(=O)N(C2CN(C(c3ccc(C(C)C)s3)=O)C2)C1 N1(CC(=O)NCC(C)(C)CNC(=O)CSC(F)(F)F)Cc2ccccc2C1=O CCC(CC)CC(=O)N1CC(C(=O)NCCS(N)(=O)=O)(SC)C1 CC1=C(C(=O)NC(C)CNC(=O)CCc2nc3ncccn3n2)C(=O)OC1(C)C Cc1cc(C(=O)NCCN(C)C(c2cc(C(C)C)oc2C(C)C)=O)nn1C C(CC(O)CNC(=O)C(C1CCOCC1)F)NC(CSCC=C)=O O=C1CCC(C(=O)NC(c2ccc(F)nc2)c2ncc[nH]2)c2ccccc21 CCCCC(CC(=O)NCc1cnccn1)NC(c1cn(CC)cn1)=O C1(NC(CSCC)=O)C2CCC(C2)C1C(N1CC(N(C)C)C(O)C1)=O c1(C(=O)NC(CN(C(c2c(C)nc[nH]2)=O)C)C)ccc(Oc2ccncc2)cc1 C(C(=O)NCc1ccc(C(=O)NCC(=O)N(C)O)cn1)(C(C)(C)C)OC S(=O)(=O)(c1cccc2cnccc12)N1CC(CC(N2CC(C)C(=O)CC2)=O)C1 N1(C(C(C)(C)c2cccs2)=O)CC(NC(c2nsnc2O)=O)C(O)C1 c1(OC)c(C(N2CC(NC(c3cn(C)cn3)=O)CC2C)=O)nc(O)nc1O C1(C(=O)NCC2CC3(CC3)C2)C2CCCOC12.C12(CC1)C(C)NC2=O O=C(C=Cc1cc(Cl)c2c(c1)OCCO2)NN1CC(C(=O)O)CC(C)C1 c1(C(C(=O)Nc2ccco2)N(CCOC)Cc2ccccc2)ccc(I)cc1 c1(OC)ccc(C(N2CCCCCC2CNC(c2ccc(C)o2)=O)=O)c(Br)c1 CC(C)(C(=O)NCC1CCN(C(C2(C(C)(F)F)CCC2)=O)C1)n1cc(Cl)cn1 c1(-n2ccc(C(N(CCNC(C=C(CCC)C)=O)CCC)=O)n2)ccccc1Cl c1(-c2c(C(=O)Nc3ccc(C(=O)O)c(C(F)(F)F)c3)c[nH]n2)cccc([N+](=O)[O-])c1 Cc1ccc(C=CC(=O)NC(CCNC(c2nc(Cl)sc2Cl)=O)C(C)C)cc1Cl N1(C(COc2ccc(C)c(C)c2)=O)CCN(C(C2CCCC(=O)N2)=O)CCC1C N(C1CCC(NC(c2csc(C3CC3)n2)=O)c2ccccc21)C(CCSCC)=O c1(OC)cnc(C(=O)NC(C)(CNC(=O)CC(C)C(C)C)Cn2cccn2)c(F)c1 C12(C(=O)NCC3C(NC(C4C(COC)CC4)=O)CCC3)CC1CNC2=O C12(C(N3CCC(N(C(COCCC=C)=O)CC)C3)=O)CCC(C(F)F)(CC1)CC2 CCC(C)C(O)C(=O)NC1CCN(C(c2ccc(O)cc2)=O)C1C(C)(C)C C1(CCOC)CN(C(=O)CCN2CCSC(C)(C)C2)CCN1C(=O)COC(F)F c1(C(C(=O)NC(CC)C)N(C)Cc2cc(Cl)cc(Cl)c2)cn2cc(Br)ccc2n1 N1(C(c2cnc(C(C)C)[nH]2)=O)CCC(NC(=O)C(F)(F)c2ccccn2)C(F)C1 c1(C(N(C2CCCN(C(Cc3cnc(C)o3)=O)CC2)C)=O)cc2cccnc2o1 CS(=O)(=O)c1ncccc1CNC(C1CC(c2ccncc2Cl)C1)=O C(=O)(CCCC(=O)NC(C1(CNC(c2cnn(C)c2C2CC2)=O)CC1)C)OC CCC(C)(CO)C(=O)N1CC(OCCC(=O)NCC2CC3C=CC2CC3)C1 c1(C(N(C(CNC(C(C)N2CCC2)=O)C2CC2)C)=O)cnc2n1CCCC2 N1(C(C2C(c3ccc(OC)cc3)C2)=O)CC(NC(C23CC(F)C2C3)=O)C(C)(C)C1 O=C1CCC(=O)N1CCS(=O)(=O)NCC(O)CC1OCCO1 N1(C(C2CN(C)C(=O)N2)=O)CCC(C2CC2)(CNC(c2cc3c([nH]2)CCC3)=O)C1 N1(C(c2nc(CCC)sc2)=O)CCOC(C(C)NC(C2CC2(C)CC)=O)C1 c1(N2CCC(CCOC)C2)cc(C)[nH]c(=NCCN2CCC(OC)C2)n1 CCC(F)(F)CC(=O)NCCC(O)C(=O)N1CCCC(C(F)F)C1 Cn1cc(C(N2CCCCC2CNC(=O)CSCc2ccccc2Cl)=O)c(O)n1 C1(NC(CCOCCOC)=O)CCC2CCN(C(c3ccc(Cl)c(F)c3F)=O)C12 C1(CNC(c2cc(COC)sc2)=O)CN(C(=O)Cc2ccc(Cl)s2)C2CCN1C2 C(C(=O)NCC1(C)CCCN1C(c1ccc[nH]c1=O)=O)(C(C)C)NC(C)=O C1(NC(C2CC(C)N(C)C2)=O)(CO)CCCN(C(c2coc(Br)n2)=O)C1 C1(O)(COC)CCN(C(c2ccncc2)C(=O)NC(c2cccc(OC)c2)C)C1 c1(NC)ccccc1C(N1CC(F)CC1CC(=O)NCCC1C=CCC1)=O CC(C)CCN=C(NCC12CC3CC(CC(C3)C1)C2)NCC1CCOC(C)(C)C1 C(C(C)C(=O)NC1CN(C(=O)C(Cc2cnc[nH]2)NC(=O)OC(C)(C)C)C1)OC n1(C(C)C)ncc(C(=O)NCCc2ccnc(CO)c2)c1C1CC1 N1(C(CCN(C(C(C(CC)CC)F)=O)CCO)=O)CCCC2CCCCC12 c1(C(=O)NCC(C)N(C(=O)C(C)c2cc[nH]n2)CC)cccc(C)c1Cl O=C(C1c2ccccc2CN1Cc1ccccc1C(=O)O)NC(CO)C1CCC1 c1(NC(C2(C#C)CN(C(=O)COC)C2)=O)ccncc1C=C CC1CN(C(c2cc(C3CC3)on2)=O)CCC1NC(C1CCC(=O)CC1)=O C1(CC(=O)NC(C)(CNC(c2cnco2)=O)CO)CSc2ccccc2NC1=O C(=O)(C(CC)CCCCC)N1C(CNC(C(CC#C)(C)C)=O)CC(O)C1 S(=O)(=O)(c1ccc(Br)cc1NCC1NC(=O)CC1(C)C)NC1CN(CC(C)C)C1 C1(CCNC(C(=O)NC2CC2)=O)CC(F)(F)CN1C(C1CC1F)=O N1(C(C(=O)NC(c2ccccc2-c2ccccc2)CC)=O)CC(N)CCC1C C12(NC(=O)CCOCC3CC3)CC(NC(c3occc3F)=O)(C1)C2 N1(C(c2cc(C)ncc2)=O)CCc2c(CNC(=O)C(C)O)cccc2C1 c1(OC)ncccc1C(C(=O)OC)NC(CO)(C(C)OC)c1nnnn1C1CC1 c1(N2C(CC(=O)Nc3ccc(CC#N)nc3)CCC2)ncnc2c1CCCC2 c1(NC(C(C2CC=CCC2)N(CC(c2cc(C)on2)=O)C)=O)ccccc1C N1(C(Cc2c(C)nsc2)=O)CC2CC1CCC2NC(=O)Cn1cccn1 C1(CC)CN(C(=O)C(c2cn(C)nn2)NC(c2ccc(N)cn2)=O)CCCO1 Cc1nc2cncc(C(=O)NC3CCCN(C(=O)C(F)(F)C(O)C4CC4)C3)c2[nH]1 C1(C(=O)NC(C(F)(F)CO)C2CC2)CCN(c2nccc(C(F)F)n2)C12CCC2 C12(NC(C(C3CC3)SC)=O)CC1CN(C(=O)CCCc1ccccn1)C2 Cc1cc(CNC(c2n[nH]cc2CNC(=O)CC2COCCO2)=O)c(C)s1 c1(C(=O)NC(C2CCCCN2C(=O)COC(F)F)C)ccc(OCC(F)F)nn1 C(C(O)C(=O)NCCCC1CCOC1=O)NC(C1C(C#N)C1)=O N1(C(C2CC(SC)C2)=O)CCC(C(=O)N2CC=CC(O)C2)=C(F)C1 N1(C(CC(C)F)=O)CCC(CC(N)=O)(NC(=O)C2=CCCCC2)CC1 CCCCCC(CC)C(=O)N1CC2(CC2)CC1C(=O)NCc1nc(C)cs1 C(=O)(CCC(CC)CCC)NCC(=C)CCNC(C1(C)C=CCCC1)=O c1(C(N(CCC(C)(C)NC(C2ON=C(CC)C2)=O)C)=O)cc(O)nc(O)n1 c1(OCC)nccc(C)c1C(=O)NC(C)CC(C)NC(=O)CSc1n[nH]c(O)n1 n1(C2CN(C(C(C3CN(C(=O)C(C)NC(C)=O)C3)OC)=O)C2)cc(C)cn1 C1(C(=O)NCC(C)N(C(c2nccc(C)n2)=O)C)CCc2cncn2C1 C1(NC(COCC=C)=O)CCCCN(C(=O)CC2CC(OCC)C2)C1 C(=O)(C1=NNC(=O)CC1)NCCC1C(C)CCCN1C(=O)CC(=O)NC1CC1 C1(C(=O)NCC#CCNC(Cc2c(C)nn(C)c2)=O)CCc2nc[nH]c2C1 C1(C(N2CC(Cn3cc(Cn4c(C)cc(C)n4)nn3)C2)=O)CN2CCCN1CC2 CCCCCCCC(=O)NCC=C1CCN(C(C23CCCCC2OCC3)=O)CC1 N1(C(C=CC(=O)OC)=O)CCC2(CC1)CN(C(c1cnnc(C)c1)=O)CC(C)O2 C1(C(=O)NC2CCN(C(c3c(C)c(Cl)cnc3)=O)C2C)CC2(CCCC2)CO1 c1(NC(=O)NC(c2ccnc(C)n2)CC)ccc(Br)c([N+](=O)[O-])c1 c1(CNC2CC(CCOC)(NC(C(CC)n3cncn3)=O)C2)ccc(O)c(F)c1 c1(SCC(=O)NCC2(F)CCCN(Cc3nc(Br)cs3)C2)ccc(Cl)cc1Cl N1(C(C2C(OC)COC2)=O)CC2(CNC(C3(C(=O)NC4CC4)CC3)=O)CCC1C2 CC1(NCc2ccn(C3CCCCC3)n2)CCC2(CC1)OCCO2 C1(N(C)C(c2ccco2)=O)CC2CCC(C1)N2C(=O)C(c1ccc(Cl)cc1F)O C(C(CC(=O)OC)C(F)(F)F)Sc1n(CC=C)c(-c2ccccc2)nn1 N1(C(COCC)=O)CCCC2C1CCCN2C(c1cc(O)n(CC)n1)=O N1(c2ncnc(OC)c2C)CCC2C(CCN2C(c2cc3cccnc3s2)=O)C1 N1(C(c2n(CCCC)ncc2)=O)CC(NC(c2ncccc2O)=O)CC(O)C1 N1(C(=O)COc2ccc(F)cc2Cl)CCC2CN(C(C3(O)CCOC3)=O)CC2C1 c1(NCCc2c(OCC)cccc2Cl)cc(Br)ccc1S(=O)(=O)NC1CCCO1 N1(C(C2(NC(c3c(C)nco3)=O)CCC2)=O)CCC(F)(F)CC1C N1(C(CCC=C)=O)CCC2(CN(C(C3(F)CCCNC3)=O)C2)C1C(=O)OC c1(SC)cc(C)c(C(=O)NCCC(O)CNC(=O)C(CN(C)C)N(C)C)o1 C1(NC(C(CC)=CC)=O)CC1C1CCCN(C(C2CCc3nncn3C2)=O)C1 C(C(C(C)C)N1CCOCC1)NCCCN(CC)CC Cn1cnc2sc(C(=O)NC3(C)CN(C(C4CCCCNC4=O)=O)C3)cc12 C(C(CC)(CC)NC(C1CCC1C(=O)OC)=O)NC(CN(CCCCCC)C)=O C(C(S(C)(=O)=O)c1ccccc1)NC(Cc1ccc(C)s1)C N1(C(c2c(N)ccc(Cl)c2)=O)CC2(CCCN(C(C3(CO)CCOCC3)=O)C2)C1 C1(C2CCCC2)(C(=O)NCC(C2CC2)NC(c2cc(C)nc(C)c2)=O)CCC1 c1(CNC(c2n(C)nc(-c3ccccc3)c2)=O)csc2ccccc12 C(=O)(C(c1ccoc1)NC(=O)CCOCC(C)C)N(CCCC)C1CC1 c1(C(N2CC(CCNC(CCC(C)SC)=O)OCC2)=O)cc2c(cc1O)CCC2 c1(CNC2C(C(=O)NCCc3ccc(O)cc3)C2)ccc(OC(F)(F)F)c(Br)c1 C12(CNC(C3CN(C)C3)=O)CCCC(CN(C(=O)CC3COCCO3)C1)C2 c1(OC)ccc(S(C)(=O)=O)cc1C(=O)NCCC(C)(C)CNC(C1(C)CC1F)=O c1(C(N(CCC(C(C)C)NC(C(CCCOC)C)=O)C)=O)cc2ncccc2[nH]1 C1(NC(c2c(CC)nn(C)c2)=O)CCC2(CC1)CCN(C(C1(O)CCOC1)=O)C2 N1(C(c2cc(C)oc2)=O)CC2CC(NC(=O)C(C)(C)C3CCCCO3)C1C2 C1(C(=O)NCC2(F)CN(C(=O)C(F)F)C2)CC1C1CC(F)(F)C1 CCC(C)C(C(=O)N1CCCC(C(=O)N2CCC(C(=O)NC)O2)C1C)OC N1(C(c2c(C)cc(CC)o2)=O)CCC(O)C(NC(=O)Cc2cccc(C)c2)C1 CC1=C(C(=O)NCCOCCN(C)C)Cn2nnnc2N1C CC1CCC(O)(CNC(c2cc(Cl)cs2)c2nnnn2Cc2ccco2)CC1 c1(CC)ccc(CNC(C2(CF)CC2)=O)cc1.C1C(CC)NC2C(CC2)C(=O)N1 C#Cc1cccc(C(N2CCCC(CC(=O)N(CCC3CC3)CC3CC3)C2)=O)c1C CC1(C)CC(NC(c2ccnc3ncnn23)=O)CN(C(C2CC3CCC3C2)=O)C1 c1(OC)ccc2c(C(=O)NC3(C)CCN(C(c4ccc(C)cc4)=O)C3)c[nH]c2c1 c1(OC)ccccc1CCCNCC1(O)CSC1 C1(C(=O)NCC2(O)CC=CC2)CN(C(=O)CSC2CCCO2)CC12CC2 C1(C(=O)NC2(C=C)CCOCC2)N(C(C2C(C)(C)C2(F)F)=O)CCCC1(C)C c1(C(=O)NCCCN(CCCNC(C(C2CC2)OCC)=O)C)cccc(C)c1C CC1N(C(=O)COC(N2CCC(F)(c3cccnc3)CC2)=O)CCOC1(C)C N(C(=NCC(F)F)NCC1CCC(F)(F)C1)C1CC(OCC)C1Sc1ccccc1 N1(C(c2onc(COC)n2)=O)CC2CC(NC(c3cc(C)[nH]c3C)=O)C(C2)C1 Cc1cc2[nH]c(=O)c(-c3nc(-c4ncn(C)n4)no3)cn2n1 N1(C(C#C)C)CCN(C(c2nccnc2C)C(=O)NCc2ccco2)CC1 c1(C(N(CC(=O)NCCCN=[N+]=[N-])C)=O)ccc2nccn2n1 Cc1cc(N2Cc3cccc(N)c3C2)nc(=NCCCCC(F)(F)F)[nH]1 c1(C(N2CC(NC(c3cnc(C)s3)=O)C(F)C2)=O)cccc(I)c1Cl CCCC(CCCNC(c1sccc1C(F)F)=O)NC(c1cc[nH]c1C)=O n1(-c2ccn(CC)n2)nc(-c2ccc(N)cn2)nc1C(C)CC C1(C(=O)NC(CCC)C)C=CCCN1C(c1c[nH]ccc1=O)=O N1(C(C(CC#C)C2CC2)=O)CC2CCN(C(C3CN(S(=O)(=O)CC)C3)=O)C(C2)C1 c1(C(=O)NC(CC(C)NC(=O)C2=CC3(CCOC3)C2)C)n[nH]c2ccc(O)cc12 CCCCC(C)C(=O)N(CCCNC(=O)CC1CC(C)C1)C c1(SC)ccc(C(=O)NCC2CC(NC(C3CC4(CC4)CO3)=O)C2)cc1 C1(NC(C(C(C)O)(C)C)=O)CC2CCCC(C1)N2C(C1CC2(C1)CS(=O)(=O)C2)=O N1(C(CC(C)NC(=O)CC2CC3C=CC2C3)=O)CC2CC1CS2 N1(C(=O)C=Cc2cncs2)CCC(CO)(NC(=O)Cn2cnc(C(=O)OC)c2)C1 C1(CC)(CC)CCCN(C(c2ncsc2Br)C(=O)NC2COC2)C1 CCC(C)CC(C)C(=O)N(C)Cc1ccccc1CNC(C1CC2(C1)CC2F)=O c1(N(C)C(N2CCC2c2ccccc2)=O)cccc(F)c1 C1(NC(=O)C(O)CCCNC(C23CC(CO)(C2)C3)=O)CCCC2(CCC2)C1 CC(C)(C)C(CC(=O)N1CCC(C2(NC(C3C4CCCC34)=O)CC2)C1)C(F)F O(NC(=O)C(C)(C1CCC1)NC(=O)CCCC1CCCC1)CCCC#C CC1CC(F)CN1C(C1(CNC(=O)C(C)CC2CCCC2)CCC1)=O CCC(C)C(CNC(CC1(C(N2CC(C(=O)NC)(CC)C2)=O)CC1)=O)OC n1(CCC)nc(C)c(C(=O)NCCC2CCN(C(=O)C(F)n3cccn3)C2)c1C N1(C(C2(SCC)CC2)=O)CCCC(C)(CNC(=O)CC2CC=CCN2C)C1 N1(C(CSc2n(CC)ccn2)=O)CCC2(NC(=O)C(C)CC(C)C)CCCCC12 N1(C(C(COC)(F)F)=O)CCC(NC(c2cc(C(C)C)cnc2O)=O)CC(O)C1 c1(C(=O)NCC(C)NC(c2cnn3cccnc23)=O)cnc2ccnn2c1N C12(C(=O)NCCC3(C)CCN(C(=O)CC4CCCO4)C3)CCC(CC1)OC2 C1(C(N(C)CC2N(CC)CCC2)=O)CN(C(c2cnc(C)nc2)=O)CC12CC2 C(=O)(C(C)(C)C(=O)NC1CCCCC1CNC(=O)CC1CN(C)CC1O)OC C(CCCCC(=O)N(C)CC1(O)CCN(C(=O)CC23COCC(C2)C3)C1)N(C)C N1(C(C23OCC(C)(C2)C3)=O)CCC2CC(CNC(=O)CC3CCC3)CCC2C1 C1(CC)C(C(=O)OCc2nc(C(C)C)n[nH]2)CCCN1C(=O)OC(C)(C)C N1(C(C=CC2N(C(C(C)OCC=C)=O)CCC2)=O)CCn2nc(C)cc2C1 C12(CNC(=O)CC3CC4CC4C3)CCCC(CN(C(=O)CCN3CCCC3)C1)C2 CC(C)C(C(=O)NCC(C)C(F)C(=O)NC1COCC(C)(C)C1)C(C)C CCC(C)(C)NC(=O)CC1CC(CNC(=O)CCOCC(C)C)C1 c1(C(N2CC(C(C)NC(c3nccn3C)=O)OCC2)=O)ccn2c1CSCC2 Cn1cc(C(=O)NCC2CC(NC(=O)CNC(C3CCC3)=O)C2)c2ccccc12 CCC(O)C(F)(F)C(=O)NCC(C)(C)OCCNC(=O)C=Cc1nc(C)cs1 CC(C)CC(O)C(C)C(=O)NC1(CCNC(c2cc3ccc(Cl)cc3o2)=O)CC1 C1(NC(CN(C)C(N)=O)=O)CCN(C(=O)C(O)CC2CCCCC2)CCC1(F)F C(=O)(CC1(O)CCOc2ccccc21)N1C(CNC(c2csnn2)=O)CC(O)C1 N1(C(C(C)O)=O)CC=CC1(C)C(=O)NCc1cncnc1 N1(C(C2(C)CC(=C)C2)=O)C2CCC1CN(C(=O)CCCCOC(C)=O)CC2 C(=O)(C(C(C)C)n1cc(Br)cn1)NCCN(C(C(C1CCC1)OC)=O)C c1(C(N2CC(O)CC(NC(c3c(=N)[nH]cnc3)=O)C2)=O)ccc2ccccc2n1 C1(NC(C2C(C=C)OCC2)=O)C2CC3CN(C(c4cnn5c4OCC5)=O)C1C3C2 n1(CC)cc(C(=O)NCCCN(C2CCCC2c2ccccc2)C)nn1 C(=O)(C1CCCc2nnn(C)c21)N(C1CC1)CC1N(C(CN(C)CC)=O)CCC1 C(=O)(C1=C(Cl)CCCC1)N1CCN(C(CCCC(C)c2ccccc2)=O)C(CO)C1 c1(C(N2CCOCC2CNC(=O)C(F)(F)C(F)F)=O)ccc(Cl)c2ccccc12 C(=O)(C1=CCOC1)NCC(CNC(c1n(C(CC)C)ncc1)=O)F c1(CN2CCN(c3cc(SC)nc(C)n3)C3C2C3)c(F)ccc(O)c1F CCC(CCCC(=O)NCCN1CCC(CO)C1)NC(C12CCC(C1)C2)=O C(=O)(C(F)C(F)(F)F)NC(C12CC(C1)C2)CNC(c1c(CC(C)(C)C)cccc1)=O CC1CN(C(=O)CC23CC(C2)C3)CCC1N(C(=O)Cc1csc(Br)c1)C O=C(C(F)C(F)(F)C(F)(F)F)NCC1C2CN(C(c3nccnc3SC)=O)CC12 Cc1cc(C(=O)NCC2CC3CC3N2C(=O)COc2ccccn2)c(C)cc1Cl C#Cc1ccc(F)c(C(N2CC(CC(=O)OC)C23CCC3)C(=O)NCCSC)c1 O=C1COc2nc(C(=O)NC3(CCNC(=O)C(F)(F)CO)CCC3)ccc2N1 Cc1c(CC(=O)NCC(C2CCN(C(=O)CC(O)CN(C)C)CC2)C)ncn1C C(=O)(C#CC1CCCOC1)N1CCCC(CNC(c2c(N)cccc2Cl)=O)C1 Cc1nc(C(=O)N(CCNC(c2cc(C)n(C)c2)=O)C2CC2)nn1-c1nc[nH]n1 c1(C(c2nnnn2CCC)NC(CCC)C2CCC2)cn(-c2cccnc2)nn1 Cc1scc(C(=O)NCCC2(NC(=O)CCC(C)N(C)C)CCC2)c1C C1(N(C(c2cccc(CO)n2)C(=O)NCCC2CC2)C)CCCCCCC1 O=S(=O)(c1ccc(F)cc1)N1CC2CCN(Cc3cncc(F)c3)CC2C1 c1(CC)cc(CNC(=O)C(c2cnn(C)c2)NC(=O)CCn2cc(C)cn2)n[nH]1 N1(C(c2c[nH]c(=NCC)s2)=O)CCC(C)C(NC(C2CC23CCC3)=O)C1C C12(CNC(=O)CC3COCCN3C(c3ccon3)=O)CCC(CC1)OC2 C1(C(=O)NCCOCCCC)CC12CCN(C(=O)CC(CC)CC)C2 c1(CN(C(C2CCC(NC(CC(C)C3CCCO3)=O)C2)=O)C)cccc(F)c1 c1(C(=O)NCCN2CCN(C(c3c(C)cno3)=O)CC2)cnc2ncnn2c1O c1(C(=O)NCC2(OC)CN(C(C34OCC(COC)(C3)C4)=O)C2)c(C)ccnc1C c1(OCC)cncc(C(=O)N(C)CC2CC(F)CN2C(c2ccn(C)n2)=O)c1 CCC(C)(F)C(=O)NCCCCCNC(=O)C(C)Cc1ccc(Br)cc1 Cc1cc(C(=O)N(C2CCN(C(=O)COc3cc(Cl)ccc3C)C2)C)cc(Cl)n1 Cc1cc(C)c2cc(C(=O)NCC(C)CNC(=O)CC3CCCS3(=O)=O)sc2n1 C#CCC(CC(F)F)NC(=O)C(C)(C)COC C1(C(=O)NCCN(C)C(C2CCCN2C2CCCC2)=O)CC(F)(CO)C1 c1(NC(C(=O)NCCC2CCCCN2)=O)cnn(-c2ccccc2)n1 c1(C(=O)NCCCOCCNC(C23CCCC2CC3)=O)cc2ccccc2cn1 C(=O)(C(C)(C)C(F)(F)F)N(C)CCNC(C1CC12CCC2)=O C1(CNC(C=Cc2ccc(CC)o2)=O)CCC2(CN(CCc3nc(C)cs3)C2)O1 c1(OCCOC)ccc(C(N2CCC3CC23)C(=O)NCCSC)cc1 C(=O)(C1CCCn2nccc21)NC1C(NC(C=CSC)=O)CCOC1 C=CC1COCCN1C(C1CCC1CNC(=O)C(=O)C(C)(C)C)=O C(=O)(CCCCC(C)C)N1CCC(N(C(Cn2nc(C)n(C)c2=O)=O)C)C(C)C1 c1(C(N2C(CN(C(c3c(C)ncnc3C)=O)C)CCC2)=O)cnc2[nH]cncc1-2 N1(C(C2CCCCCCN2C(C2C3CC4C(C3)C24)=O)=O)CC=C(C(=O)N)CC1.CO C1(C(=O)NC2CCN(C(C3CC(CC4CC4)C3)=O)CC2)CC12CCOCC2 Cc1c(C(=O)N(C2CN(C(=O)Cn3c(C)csc3=O)CC2F)C)cncc1Cl C(CC(C(=O)N(C)CC1COCC1O)NC(=O)CCCN1CCCC1)SC C1(CC=C)(NC(c2n[nH]cc2OC)=O)CCN(C(=O)C(c2ccncc2)C)CC1 C12(CNC(CCCn3ncc(C)c3)=O)CCC(CN(C(=O)Cc3cc[nH]n3)C1)C2 Cc1c(C(N2CCCC2(C)C(=O)Nc2cc(O)nc(Cl)n2)=O)cncc1Br c1(C(=O)NCCN(C(=O)C=C2CCCCC2)C(C)C)nocc1Br N1(C(c2c(C)scc2)=O)CC(NC(c2cnc3n2CCC3)=O)C(C)(C)C1 C1(C)(CC)CN(C(=O)CN(C2CCC2)C(c2coc(C)c2)=O)CCO1 CN1CCC(n2cc(NC(C3CC3C(=O)NC3CC3C(N)=O)=O)cn2)CC1 c12nc-1n(C)n2.CCCCSC(C)(C)F CCC1=NOC(CC(=O)NCc2ocnc2C(=O)NC(c2csnn2)C)C1 C1(N(C(=O)Cn2cnc(C(N)=O)n2)C)CCCN(C(c2cc(Cl)ns2)=O)C1 Cc1cc(O)ncc1C(=O)N(C)CCN(C(=O)C(F)n1cccn1)C CC(C)(C)C(C)(O)CNC(=O)CNC(=O)CC1CC(=O)NC1=O c1(C2(C(=O)NC3C(OC)CN(C(CN(CCC)C)=O)C3)CC2)ccc(F)c(Cl)c1 C1(CNC(CSCCC#N)=O)CCCC1CNC(c1c[nH]nc1Cl)=O C1(NC(COC)=O)CS(=O)(=O)CC1NC(c1cccc(C(C)C)c1F)=O C1(C#N)(C(=O)NC2CN(C(CCc3ccc(OC)cc3)=O)C2)CCCOC1 c1(C(=O)NCC(CNC(c2c(C)snn2)=O)C)ccnc(OC2CC2)c1 CCCC(C)(O)CC(=O)N1CCN(C(C2CCN(C)CC2)=O)C(c2cn[nH]c2)C1 C1(COC(=O)NCC)CCCCN1C(c1cnn(C)c1C)=O C1(NC(c2n(CC)nnn2)C2CN(C(=O)OC(C)(C)C)C2)CCNC(=O)CC1 c1(OC)cc(C(=O)NCCC2CCC(C(N3CCCC(C)C3)=O)C2)nn1C CSC1=C(C(=O)NC(c2cccc(C)c2)CNC(C2CCOC2)=O)CCCC1 N1(C(C)C)CCCC(C(N2CC(CNC(=O)CN3CCCNC3=O)C(O)C2)=O)C1 c1(C(C)C(=O)NCC2CCN(C(c3n[nH]cc3C3CC3)=O)C2)ccccc1F CC1(C)C(NC(=O)C=CCO)C(C)(C)C1NC(c1cc(O)ccc1Cl)=O C1(CNC(CC2(COC)CCCC2)=O)(NC(c2cnc(C)[nH]2)=O)CCCCCC1 n1(CC)nc(C(=O)NCC2(F)CCN(C(C3C=CCCC3)=O)C2)cc1C(F)(F)F c1(C(=O)NCC(=O)N(CC(C)Cc2cn[nH]c2)CC2CC2)cc(C(C)C)no1 C1(NC(CCCCOCCC=C)=O)CCCCCN(C(C2CCS2(=O)=O)=O)C1 C(=O)(C(C)CC#N)NCCN(C(Cc1cnc(C)[nH]1)=O)C(C)C C(=O)(C1CCCc2nc[nH]c21)N1CCN(C(c2c(N)c(F)ncc2)=O)CC1CO Cc1nn[nH]c1C(=O)NCC1(C(=O)NC(C)C(=O)NO)CCCO1 c1(C(=O)NC2C(C)N(C(=O)C(=O)N(C)C)CCC2)cccc2nc(S)oc12 c1(C(N(CC(CN(C(CC(C)N(C)C)=O)C)O)C)=O)ncc(C#N)cc1Cl c1(CC(N2CCC3CN(C(C=C(CCC)C)=O)CC32)=O)oc2ccccc2c1C c1(NC(C(c2ccc(Cl)s2)C)=O)ccc(OC(F)(F)F)nc1 c1(C(=O)NCCCN(C(c2n[nH]c(C)c2O)=O)CC)[nH]c(C)c(S(N)(=O)=O)c1C N1(C(c2scc(OC)c2)=O)CCOCC1CN(C(=O)C(C1CCCCC1)O)C C1(NC(=O)CCn2cc(Cl)cn2)CCN(C(C2CC(F)(F)C2)=O)CC1F c1(C(N2CC=CC(NC(CC(C)n3ccnc3)=O)C2)=O)cc2c[nH]cnc-2n1 CC1(C)Cc2ccc(C(N3CCCCC(NC(C4(F)CC4)=O)C3)=O)c(O)c2O1 Cc1nn(CC(=O)NC23CC2CN(C(=O)CC(C)C)C3)c(=O)c2ccccc12 C1(CC(=O)NCC(CNC(C2CCN(CC#C)CC2)=O)O)CC(C)CC(C)(C)C1 c1(C(=O)NC2(C)CC(NC(C(CC=C)(C)C)=O)C2)ccc2c(C)cc(Cl)nc2c1 C=Cn1nncc1C(=O)N(C1CCN(C(=O)CN2CCCC2)CC1)C C(C(=O)N(C)CCNC(c1cscc1C(F)F)=O)(C(C)C)OCC(C)C c1(C(N(CC(CNC(CC(C=C)C)=O)O)C)=O)cnc2sc(C)cn12 c1(C(C)C)ccc(OC(=O)CN(C2CC(C#N)C2)C(C2CCCCO2)=O)cc1 c1(C(N(CCCNC(=O)COC(F)(F)F)CC)=O)cc(CC2CC2)cs1 Cc1cc(C(c2ccccc2)CNC2(C(=O)OCS(C)(=O)=O)CC2)ccc1Cl c1(NCCCCC(C)NC(C=C(C)Cl)=O)cc2c(cn1)C(=O)CCC2 c1(N(C)C(N2CCOC(C3CCCCC3)C2)=O)cccc(-c2ccccn2)c1 C1(C(=O)NC(c2n(CC)ccn2)C)CC(F)(F)CN1C(c1cccc(C)c1N)=O C=CC(O)(C(=O)N1CCCN(C(C2CCN(C(C)=O)C2)=O)CC1)C(F)(F)F CC1CN(C(=O)C(c2ccccc2F)N)CCN(C2CCC2)C1 CC(C)(C)C(C(=O)N1CCC(CCNC(C2(C(C)(F)F)CC2)=O)CC1)C1CCC1 C1(C#N)(C(=O)NCC(CC)NC(C2(Cc3ccccc3)CCC2)=O)CCCO1 CC1(C)CN(C(C2CC2C#N)=O)C(CNC(=O)CN2CCS(=O)(=O)CC2)CO1 CC1=C(C(=O)N(C(C)C(=O)Nc2cncc(C(N)=O)c2)C2CC2)CCCO1 c1(CNCC2N(C(c3cc(C)[nH]n3)=O)CCC2)ccccc1Br c1(CC(=O)NCC(C)NC(C2CCN(C(=O)C3CC3)CC2)=O)cc(F)ccc1Cl C(C1c2ccccc2CCN1C(=O)C(F)=C1CCC1)NC(C(C)C1CCC1)=O C1(NC(c2ccc(CC)o2)=O)CC(C)CN(C(C23CC4CC2C3C4O)=O)C1 c1(C(N(CC(C)NC(c2cc(CC)n(CCO)n2)=O)C)=O)ccn2nccc2n1 N1(CC(=O)NCC(CNC(CC2C(CC)C2(F)F)=O)OC)CCC(F)(F)C1 Cc1ccc(C(N2CCC(NC(c3ccc(CN(C)C)[nH]3)=O)C2)=O)n1C C1(NC(c2ccc(C(N)=O)nc2)=O)CCCCCN(C(=O)CC(F)F)C1 C(c1c(Cl)nc2sccn12)=CC(N1CCC(C)C(C(F)(F)F)C1)=O c1(N(C(C)C)C(C2(CCNC(c3ccccc3)C)CC2)=O)ccc([N+](=O)[O-])cc1 N1(C(C2CCCC3CC23)=O)CCN(C(c2ccc3c(c2)CCO3)=O)C2(CCC2)C1 Cc1ccnc(N2CC=CC(NC(C3(C)CC3(F)F)=O)C2)n1 N1(C(C=CC(C)(C)C)=O)CCC(C)(C)C1C(=O)Nc1cc(F)ccc1O c1(C(=O)NC(C)(C)CCCNC(c2cccc(CO)c2)=O)cnn2ccsc12 C=C(C)CC(C(=O)N(C(CC)C1CC1)C)NC(c1oc(C)nc1C)=O c1(OC)c(Cl)nc[nH]c1=NCC1CC1NC(c1cc2c[nH]nc2s1)=O Cc1cn2cc(C(=O)NC3(C)CN(C(c4nn(C)cc4C)=O)C3)sc2n1 C1(C(=O)NC2CCN(C(CCc3[nH]c(=N)sc3)=O)C2)CC2CC1CC2O N=c1nc2ccc(C(N3CCOCC(CNC(C4CNC(=O)C4)=O)C3)=O)cn2[nH]1 Cc1cc(C(=O)C(=O)NCCC2(C(=O)NC3CCSC3)CC2)ccc1F CCC(CC(F)F)C(=O)NC1CC(CNC(c2cnc(O)n2C)=O)C(O)C1 Cc1ccc(C(=O)NC2CCC(CCNC(C3CC=CC3)=O)C2)c2cccnc12 c1(C(=O)NC(C)(C)CCNC(=O)CC2CC=CC2)ccc2c(c1)NC(=O)CC2 C(=O)(C1=C(Cl)CCOC1)N1CC(N(C)C(c2ccncc2N=[N+]=[N-])=O)C(C)(C)C1 c1(CC)cc2c(NCC3(F)CC(NC(C4C(C)OC(C)C4C)=O)C3)ncnc2s1 Cc1nc(CNC(=O)CC2(C)CCOC2)oc1C(=O)NC1CC(CCC(N)=O)C1 Cc1cc(C(=O)NCC2CCC2NC(=O)CCC2NC(=O)NC2=O)oc1Br Cc1nc(CC(=O)NCC2CCCN2C(c2ns[nH]c2=O)=O)sc1C N1(C(c2cncc(CC(C)C)c2)=O)CC2(C1)CN(C(=O)C=CCF)C2 C1(N(C)C(C2(O)COC2)=O)CCCN(C(=O)C(F)(F)c2cnn(C)c2)CC1 C1(C(=O)NC23CC(NC(C(SC)SC)=O)(C2)C3)CC(=O)N(CC2CC2)C1 N1(C(C)C(=O)NCCCC2CCCN2C(=O)CC2(C(F)F)CC2)CCC(O)CC1 N1(C(c2c(OC)nccn2)=O)CC2(C1)CN(C(c1cc(Br)ncc1F)=O)CCO2 C=CC1CCCCN1C(=O)C(CCCOC)NC(=O)Cc1cnoc1 c1(C(NN(CC=C)C(=O)OC)=O)c(P(C)(C)=O)cnn1-c1ccccc1 CCC(C)CC(=O)C(=O)N1CC2CCC(CNC(c3cc(C(C)C)[nH]n3)=O)C2C1 C=CCC(CC(F)F)C(=O)NC(CNC(C1CC(CC(F)F)C1)=O)C(C)C c1(CC(N2CC(N(C)C(C3CC(C)(O)C3)=O)C2)=O)c[nH]c2cccnc12 CN1CCN(C(=O)C(=O)Nc2ncc[nH]2)C(CNC(=O)CCc2nncn2C)C1 C1(NC(C(c2ccc(Cl)cc2)CC)=O)CCC(S(C)=O)C1 c1(C(C(=O)NCC(C2CC2)SC)NC(=O)CC2OCCC2C)c(C)cccc1Br CCC(C)(C)CCCC(=O)NCC(c1ccc(F)cc1F)NC(=O)C(C)(C)O C1(C)(C(=O)NCCN(C(c2cc(CO)n(C)n2)=O)CC)CCCS1(=O)=O C(=O)(C1=CCCN(c2ncncc2I)C1)N(c1cccc(OC(C)(C)C)c1)C Cc1cccc(CNC(C)(CCBr)c2nnnn2C2CCCC2)n1 c1(CC)cnc(O)c(C(=O)NC(C)(C)CN(C)C(c2ccnc(Cl)c2OC)=O)c1 C(=O)(CC(C)C(C)C)N1CC(CN(C(Cc2c(CC)con2)=O)CC)OCC1 c1(-c2cc(-c3ccn(C)c3)[nH]n2)nc(-c2ccnc(N3CCOCC3)c2)nn1CCCO C1(NC(Cc2cnc(C)[nH]2)=O)CN(C(=O)Cc2cccc(C)c2F)CCC1C C1(CN(C(C2C3CC4C(C3)C24)=O)CC)CCN(C(=O)Cc2csc(C)n2)CC1 C(=O)(CC(O)C(C)C)N1CC(NC(CSCC(=C)C)=O)C(Cc2ccccc2)C1 c1(C(C)NC(=O)C(=O)NC2C(C)C2C)cccc(OC(F)F)c1 N1(C(CC2C(C)(C)OCC2)=O)CCOC(C)(CNC(=O)C2=CCC2)C1 c1(C(N2CCC(NC(CCCOCCC)=O)C2C)=O)cccc2ccnn12 C12CCC(CC1)C(c1nnnn1C)N2.C1(OC)CC(CC(=O)OC)C1 CC(=O)CCCC(=O)N1CCC(NC(=O)CC2CC2)C1C c1(CNC(CC)COC)c(F)cc(Cl)cc1Br c1(OC)ccccc1C(C)NC(N1CCCC1CF)=O c1(C(C(=O)NCCCOCCN(C(C(CC)F)=O)C)O)ccc(Cl)c(Cl)c1 C=CCC(F)(F)C(=O)NCC1(CNC(=O)CCCc2cccs2)CCCCC1 CCC(F)C(=O)NCCN(CCCN(C)C)C(c1ncn(-c2ccccc2)n1)=O CC1(F)CCC(C(=O)NC2(CNC(C3CC=CCO3)=O)CCOCC2)CC1 C=CC(C)C(=O)N(CCCC(=O)N(CC(C)(C)O)C)C c1(C(=O)NC2C(CNC(CC(=C)C)=O)CCC2)cc2c(s1)CCCCCC2 c1(C(=O)NC(CNC(CCSC)=O)CC(F)(F)F)c(C(F)F)nc2ccccn12 Cc1nnc2n1CC(C(=O)NC(C)CNC(c1sccc1SC(F)F)=O)C2 c1(C(=O)NC2C(NC(c3c(C)ocn3)=O)COC2)cnccc1N1CCOCC1 C=CC1(C(=O)NCC(C)(F)C(C)C)CCN(C(C2CC3(CC3)CO2)=O)CC1 C1(CCCNC(CC2(NC(C)=O)CC2)=O)CCCCN1C(c1ccnc(C)c1)=O C1(C(C)(C)C(=O)NCCOCCNC(c2ccncc2O)=O)CCC(C#N)C1 N(S(=O)(=O)N(C)CCN1CCC(C)CC1)C(CC)C c1(CCC(N2CC(CNC(CSC)=O)C(C)CC2)=O)c[nH]c2cc(C)ccc12 CN1CC2C(C(N3CC4CC3C4C(=O)NC(C)(C)C(F)(F)F)=O)C2C1 c1(CC(N2C(CNC(CNC(N)=O)=O)CCC2)=O)c(F)cccc1F N1(C(C(CNC(CC2(OCC)CCC2)=O)(C)CC)=O)CCOC(C)(C)C1C C12(CNC(CC3(CSC)CC3)=O)CCCCC1CN(C(c1cncnc1)=O)C2 C1(NC(C(C)NC(CC)=O)=O)CN(C(C2(CCF)CCOCC2)=O)CC(C)(C)C1 c1(C(N2CCC(N(C(c3n[nH]cc3C)=O)CC)C2)=O)ccc(S(C)(=O)=O)cc1 N1(C(C2(SC)CC2)=O)CC(C2CCCCN(C(c3c([N+](=O)[O-])cnn3C)=O)C2)C1 c1(OC)nn(C)cc1C(N1CCC(C)(CNC(=O)C(N2CCNC2=O)C)C1)=O c1(NC(C)CS(C)(=O)=O)ccc(S(=O)(=O)NCC2CCCCO2)cc1Br N1(C(CC2CCCN(C)C2)=O)CC(C(=O)NC(c2ccccn2)CO)CC1(C)C CCC(CC(F)(F)F)C(=O)NCC1(F)CC(CNC(=O)C(O)C2CCC2)C1 c1(C(=O)NC(CN(C(C(c2cccc(Cl)c2)OC)=O)C)C)cc(Cl)ccc1O C1(NC(C(N2C(COCC)COCC2)CC2CC(F)(F)C2)=O)CCC(F)(F)CC1 CCC(CN(C)C)CC(=O)NCCCC(C)(C)C(=O)N(CCCC(C)(F)F)C N1(C(CCNC(COC)=O)=O)CCC(NC(c2coc(C(F)F)c2)=O)C(C)(C)C1 C(=O)(C1=NOC2(CCC2)C1)NCC1(C)N(C(C(CC)O)=O)CC(F)(F)C1 C=CC(CC)CC(=O)NCC1CCCN(C(C2CCCCNC2=O)=O)C1 C=CCCCC(C(=O)N(C)CCOC1CC1)NC(C1CCC(=O)N1)=O C1(NC(C(C2CCC2)NC(c2c(C)cccc2)=O)=O)CC2C(C1)C2(F)F Cc1cnc(C=CC(N2CCCC2CNC(c2coc(C)n2)=O)=O)[nH]1 c1(C(=O)NC2CC3(C2)CC(NC(C2CC4(C2)CC4F)=O)C3)cc[nH]c2nccc1-2 NC1C2C=CC(O2)C1C(N1CC(c2nc[nH]n2)C1)=O.c12ccoc1C2 CC1(C)C(C)(C)C1(F)C(=O)NCCC1COCCN1C(c1ccc(CO)cn1)=O c1(C(=O)NC2C(C)CN(C(=O)CC3=CCCC3)CC2)ccc2c(c1O)CCCC2 N1(C(Cn2ccc(C)n2)=O)CCCC2C1CCN2C(c1csc2c1CCCC2)=O C1(CC)CCC(NC(=O)C(c2ccccc2)NC(c2ccsc2C)=O)CC1 c1(C(C)CC(=O)NC2(CC(=O)O)CCOC2)ccc(F)c(Br)c1 Cc1c(C(=O)NCC(F)CNC(=O)C(C)(C)n2cccn2)cnn1C(C)(C)C c1(CC(=O)NCCCCN(C(C(C2CCC2)OCC)=O)C)c[nH]nc1C C1(C(N2CC(N(C(CN(CC(C)(C)C)C)=O)C)C(O)C2)=O)CC(C(C)(C)C)=NO1 N(C)(C1CN(C(=O)COC(C)C)CCc2ccccc21)C(c1c(C)cncc1)=O C1(NC(CC2N(CC)CCOC2)=O)CCN(C(c2cnc(C(C)C)[nH]2)=O)C(C)C1 CC1C(NC(c2cc(F)cnc2O)=O)C(C)CCN1C(=O)CC1CCCCC1C C1(NC(C=CCC)=O)CCN(C(=O)CC(C)C2CC2)CC1C Cc1cc(C)c(CCNC(c2ccc(Cl)cc2Cl)c2nnnn2C2CC2)c(C)c1 N1(C(C(CC)O)=O)CCC(C)(C)C(NC(C2(c3ccc(N(C)C)cc3)CC2)=O)C1 C12CC13CCN(C3)C2=O.c1(NCc2scc(C(=O)OC)c2)cncc(C)n1 C(=O)(C1=Cc2ccccc2OC1)N1C(C)CC(NC(C2CC2C)=O)CC1 c1(C(N(C2CCCN(C(C3(C#C)CCCC3)=O)C2)C)=O)cc2n(c1)CCC2 C(CC)(CCCC(=O)NC1CC(C(F)F)C1)NC(C(C=C)(F)F)=O c1(C(=O)NCC(CN(C(CC(C)C(C)(C)C)=O)C)(C)C)ccnc2[nH]c(O)nc12 C(=O)(C(C(C)(C)C)NC(=O)CC1CCCC2CC12)NCCC(CCC)F C=C(C)C(C)(C)C(=O)N(C1(C(=O)NCc2ccc(C#N)s2)CC1)C Cc1cc(CN2CCC2CNC(c2cccc(-n3cccn3)n2)=O)ccc1Cl N1(C(C2CN(C(CC)CC)C(=O)C2)=O)CC(C2CN(C(C3CCOC3)=O)C2)C1 N1(C(c2cncc(C)c2)=O)CCC(CNC(=O)Cn2cccc2)C(C)C1 C(C)(CCCCN=c1[nH]c(C(C)(C)C)nc(=N)[nH]1)NC(Cn1ncc(C)c1)=O c1(C(=O)NCC2(C)CCN(C(=O)Cc3cccc(Cl)c3)C2)nccc2[nH]ccc12 N1(C(CSCC)=O)CCC2(CCCN2C(c2cc(O)ccc2Cl)=O)C1 Cc1ccncc1CNC(=O)CC1CN(C(C2CC2(C)C)=O)CC1C C1(CNC(CS(=O)(=O)NCC)=O)CC(F)(F)CN1C(=O)CN(C)C(C)=O C(=O)(CC1=CCCCC1)N1C(C(=O)NC(C)CN2CCCC2)CC(O)CC1 C=CC1(CC(=O)NCCC2COCC2O)CN(C(c2nscc2C)=O)C1 c1(C(=O)NC2C(CNC(Cn3ccc(C)n3)=O)C2)ncc(Br)cc1F C1(CNC(=O)NCc2nc(CC)[nH]n2)CCC(=O)NC1C C(CC(C)(C)C(=O)NCCCN(C(=O)CNC(=O)NC1CCCC1)C)NC(C)=O c1(C(N2C3(CN(C(=O)CCn4cccnc4=O)C3)CC2)=O)noc2c1COCC2 Cc1nncc(C(=O)NC2CC3(C2)CC3C(=O)NCCc2ccnn2C)c1C CCCC(CC(=O)NCCN1CC(CF)C1)NC(C1CC2CCCC2C1)=O CC#CCCCC(=O)N1CCC(N(C)C(=O)C2CC2)C(C)C1.C1C(=O)N1 C1(NC(C2(F)CN(C(C34CC(CO3)C4)=O)C2)=O)C(C(=O)NC2CC2)CCC12CCC2 C1(OC)CC(C)CN(C(=O)CC2CCN(C(C3CCC4(CC4)C3)=O)CC2)C1 c1(C(N2C(C(=O)O)CC(CC(=O)O)C2)=O)c[nH]c2ccc([N+](=O)[O-])cc12 N1(C(CC)CO)CCN(C(c2csc(C(C)=O)n2)=O)CC1 c1(C(N2CC(N(C(C=C(C)C)=O)C)C2)=O)ccc(F)c(N)c1 c1(C(N(C)CC2CCN(C(C3(C#N)CCOC3)=O)CC2)=O)c[nH]c2cccnc12 CCC(CCCC(=O)NCC#CC(F)(F)F)NC(C1C2CCCC(=O)C12)=O N1(C(C2N(C)C(=O)OC2)=O)CCCC(C)(CNC(C23CCCCC2C3)=O)C1 N1(C(CCC=CC)=O)CC(C)C(C)(C(=O)NCC2(CN(C)C)CCC2)C1 c1(C(=O)NCC(C)(CO)NC(CS(CC)=O)=O)cnc2ccc(C)cn12 n1(CC)ncc(Br)c1C(=O)NCC1CC1NC(=O)C(F)=C1CCCC1 CC1(C)CC(CC(=O)NC(C2CCCO2)(C)C)N(C(=O)C=Cc2cscn2)C1 C(=O)(C1=CC2CC(C1)CC2O)NCCN(C)C(c1cc(Cl)n[nH]c1=N)=O C(=O)(CCCCC(=O)NC1(C(=O)NCCC2=CCCCC2)CCOCC1)OC c1(CNC(C(C)NS(=O)(=O)C(F)(F)F)=O)ccc(Cl)c(Cl)c1F C1(C(=O)N(CC(C)CNC(c2sccc2Cl)=O)C)(COC)CCOCC1 C(=O)(C(C(C)C)C(C)C)N(CCC(C(C)(C)C)NC(C(CO)OC)=O)C C=CCCCC(C(=O)N1CC(CC)(CO)C1)NC(=O)C=CCO c1(NC(C2OCCN(C(c3c(C)cc(O)nc3)=O)C2)C)ncc(Cl)c(C)c1C#N C(=O)(CCS(N)(=O)=O)N(C1CCCCCC1)CCNC(Cc1ccn(C)n1)=O c1(C(=O)Nc2cc3nc(C)ccc3o2)c(Cl)oc2ccccc12.CCCN1CC1 Cc1cnc2n1CCC(C(N1CCC(NC(=O)CC(C)C)C(O)C1)=O)C2 Cc1cc(C(=O)NC2CCC(Nc3ncnc(=N)[nH]3)CC2)ncn1 C(CCF)(C(=O)NCc1ccns1)NC(C=CC(=O)OCC)=O C1(NC(C2C(OC(C)=O)C2)=O)CC=C(C(=O)N2CCN(C)CC2C(N)=O)C1 O(NC(=O)C(CNC(=O)COCC=C)CC1CC1)CCC#C c1(CC2(C(=O)NC(C)CCNC(C3CC(F)(F)C3)=O)CC2)ccccc1Br C1(NC(C2N(C(CCC=CC)=O)C(C3CC3)CC2)=O)CC2(CCCCO2)C1 Cc1cc2c(NCC3CCC(C)CC3)ncc(I)n2n1 C1(C(=O)NCc2ccc(Cl)s2)CC(F)CN(Cc2ccc(C(F)(F)F)c(F)c2)C1 N1(C(C(C)(C)CF)=O)CC2(CCCN(C(c3cc4c([nH]3)CCCC4=O)=O)C2)C1 N1(C(Cc2c(C)cnn2C)=O)C2CCC1CC(NC(C1CC3(C)CC1CO3)=O)C2 c1(C(=O)NC(C)C(CO)NC(C2CC2(Cl)Cl)=O)c(F)ccc2occc12 N1(CC2CC(C)C2)CCc2ncnc(O)c2CC1 C1(C(=O)NC(CN(C)C(C2CC3(CSC3)C2)=O)(C)C)C2(CCC2)C12CCC2 C(C1CCCn2ccnc21)NCc1ccc(F)nc1 N1(C(C(C)O)=O)CC(CO)C2(CCN(C(=O)Cc3nccn3C)CC2)C1 C1(C(N2CCC(C3N(C(CCS(C)=O)=O)CCCC3)C2)=O)CCC(=O)CC1(C)C C1(CCNC(=O)C=CC2CCCO2)CC2(CCC2)C1 CN1CC(C(=O)NC2CC(CNC(=O)C(N)=O)C2)C(C(F)(F)F)C1 N1(C(C=CC(C)(C)SC)=O)CC2CCN(C(=O)C(C)NC=O)CC12 C(CNC(C1(F)CCOC1)=O)(C(=O)N(C)CC1(C#N)CC1)OC CC1=C(C(=O)N2CC(CNC(=O)Cc3conc3C)CC2C)CCS1(=O)=O C12(C(=O)NCCN(C(c3n(C)ncc3Br)=O)C3CC3)CCC(CC1)CO2 C(=O)(CCOCC1CCCO1)N(CCN(C(C)C)C(c1cnc[nH]1)=O)C C(=O)(C1=NOC(C)(C)C1)N(C1CCCN(C(c2nocc2C(C)(C)C)=O)C1)C C1(C(=O)NCC2C(NC(C(C)O)=O)CCC2)C2CCC1(c1cnco1)C2 N1(C(C2OCCN(C(CNC(C(CC)C)=O)=O)CC2)=O)CCCN(C)CCC1 C1(C)(C(N2CC3(CN(C(C4(C#C)CC4)=O)C3)OCC2)=O)COc2ccccc2O1 C1(C)(C(=O)NC2CC(C)(NC(c3ncccn3)=O)C2)Oc2ccccc2NC1=O C1(CCC)CN(C(=O)CC(C)C)CC1C(=O)NC(C)(C)CCC1CC1 Cn1c(=O)ccn(CC(=O)NC(C2CC3CCC2C3)(C)C)c1=O n1(CC(=O)NCCC2(CNC(=O)CC3CCC4CC34)CC2)nnc2ccccc12 O=C(CCCCCBr)Nc1ccc(C(=O)Nc2ccc(Cl)c(Br)c2)cn1 C(=O)(C(C)C(C)(C)C)NCC1(CNC(C(C2CCC2)OC)=O)CC1 C(=O)(CC(=O)NCCC1CCCN1C(=O)CC1(O)CCOC1)NCC#C S(=O)(=O)(c1c(Cl)cccc1Cl)N(C1CCN(c2ccccc2)C1)C c1(NC(C2CN(C(C3CCCC3)=O)CCO2)=O)c(Cl)cnnc1Cl N1(C(CCCOC)=O)CCC(NC(=O)C=C2CCCCC2)CC1C C1(CNC(C(C=C)OC)=O)CCC2(CN(C(=O)CCCC3OCCO3)C2)O1 C1(OC(c2nc(C)sc2)=O)CCC(C(=O)COc2ccccn2)CC1 N1(C(CC(C)N(C)C)=O)CCN(C(=O)CCc2csc(Br)c2)CC(O)C1 Cc1cocc1C(N1CC(F)(CNC(=O)C(C)N2CCC2)C1)=O c1(CSC)cc(C(=O)NC(CNC(c2ccc(C(N)=O)s2)=O)C2CCC2)no1 C(=O)(C(=O)C(C)C)Nc1nc(CCCC)[nH]n1 c1(OC)cc(C(=O)NC23CC(NCC4CCCC(OC)C4)(C2)C3)c(Cl)cn1 c1(C(=O)NCC(CNC(CNC(CCC)=O)=O)F)nnn(CC)c1C C=CCCC(C)(C)CNC(=O)CN(C(=O)CCCCC1CC1)C1CCC1 S(=O)(=O)(c1cccs1)N.C1(C(C2CCN(C)C2)=O)CN(Cc2ccccc2)CCO1 c1(C(=O)NC2C(C)CN(C(=O)C(=O)C3CCCC3)CC2)cc2n(n1)CCCO2 Cc1cc(OC(C)C(=O)NC2CC(CNC(c3ccnc(S)c3)=O)C2)ccc1Cl CC(Cc1ccccn1)C(=O)NCC(C)(CO)NC(=O)C=Cc1ncc[nH]1 c1(C(C(CC)C)NC(=O)C(=O)Nc2cnn(C(C)C)c2)ccc(Cl)cc1 c1(C(C=CC(=O)NCC(c2ccccc2)NC(C2C(C#C)C2)=O)=O)cnccn1 Cc1c[nH]c2ccc(-c3cnc(CC(=O)Nc4cc(F)c(F)cc4Cl)nc3)cc12 C1(CCNC(C(CC)=CCCC)=O)CCN(C(=O)CNC(=O)C2CC2)C(C)C1 N12CCC3(CN(C3)C(=O)c3ccc(s3)C1)C2.c1(C(=O)O)cccc(N2CCN(C)CC2)c1 N1(C(C(c2cnccn2)C)=O)CCN(C(C2CCOCC2)=O)C(CS(C)(=O)=O)C1 c1(C(=O)Nc2ncccc2Br)[nH]nc2c(-c3cncc(F)c3)cccc12 C1(NC(CC=C=C)=O)C2CCCC1CC(NC(c1cn(C3CCOC3)nn1)=O)C2 CCC(C)CC(=O)C(=O)NCC(C(=O)N1CC(C)(CSC)C1)N(C)C C1(C)(CNC(C2(C)CNC(=O)C2)=O)CC(F)(F)CN1C(c1ccc(Cl)c(O)c1)=O C1(C(N(CCC(C)NC(C(CC=CC)CC)=O)C)=O)CC2(CCOCC2)C1 C1(C(=O)NCC(CNC(C2CC(=C)C2)=O)OC)CC(CC)=NO1 C(=O)(C(CC(F)F)N(C)C(C1CCCN1CC)=O)NC(c1ccnn1C)CC C1(NC(C2(C#N)CCC2)=O)CCOCC1C(=O)NC1COC(C(F)F)C1 c1(C(=O)NC(CC)CNC(C23CCC(OC)C2CC3)=O)cccc2nc[nH]c12 C#CC1(O)CCCN(C(=O)CC(CC=C)NC(=O)C(C)NC(=O)CC)C1 c1(C(N(CCN(C(CN2CCC(C)C2)=O)C)C)=O)cnn2c1OCC(O)C2 CCC(CN(C)C)N=c1nc2c(ncn2CC)c(NCCCCCC2CC2)[nH]1 C1(CC=C)(C(N2CCC(F)(CF)C2)=O)CCCN1C(c1cncnc1CC)=O c1(CC)ccc(C(=O)NC2CC(C)(NC(c3cc(C4CC4)n(C)n3)=O)C2)cc1F C1(NC(N2CC=CC2)=O)CCOCCC1(F)F C1(CNC(C(CSC)OC)=O)N(C(c2cc(C#N)[nH]c2C)=O)CCCC1(C)C Cc1ncnc(C)c1C(=O)NCC(N1CCC(c2cccnn2)C1)=O C#Cc1ccc(C(=O)NC2(C)CCN(C(=O)Cc3ccc(Br)cc3)C2)nc1 CC1CN(C(c2ccc(C(O)CF)cc2)=O)CC1NC(C1(C)CCOCC1)=O c1(C(=O)NC(C)CNC(=O)C(c2cncn2C)O)cc(O)ccc1N C1(NCc2cn(CC(C(C)(C)F)(C)F)nn2)CCC2(CCNCC2)CC1 CCCCCCC(=O)NCC(C)(CC)NC(c1ccc(O)c(F)c1)=O c1(OC)ccc(SCC2CC2C(=O)NC(C2(c3cccs3)CCOCC2)=O)cc1 CCC(C(=O)N1CCC(N(C(C2CNC(=O)N2)=O)Cc2ccccc2)C1)OC C1(NC(C(C)OCCCC)=O)CC12CC(C(=O)O)C2.N12CCC(C1)CC2=O CCCCCCCC(=O)N1CCC(C(=O)NCC2(OC)CCCC2)C(C)C1 C1(NC(C2CC=CC(n3cc(CSC)nn3)C2)=O)CCN(C(C)=O)CC1(C)C c1(CNC(C(=O)NCc2n(C)ccc2)=O)ccc(CNS(C)(=O)=O)nc1 N1(C(c2cc(C)sc2N)=O)CC(C)CCC1C(=O)NC12CCCN(CC1)C2 N1(C(c2ns[nH]c2=O)=O)CCOC2(CCN(C(c3cncc4[nH]ccc34)=O)C2)C1 N1(C(c2c(CC(C)C)nc(C)s2)=O)CCCC(NC(C2CCCCC2O)=O)CC1 C1(N(C(c2n(C(CC)C)ncc2)=O)C)CN(C(C2(C(C)=O)CCCC2)=O)CC1O n1(CC)nc(C(=O)NCC(C2CC2)N(C)C(c2c(C)n[nH]c2C)=O)ccc1=O c1(C(N(CC(O)CNC(C2C3CNC(=O)C23)=O)C)=O)coc2c(F)c(Cl)ccc12 C(=O)(C(C)CS(C)(=O)=O)NCC(COC)NC(C1(CF)CC1)=O C1(C2CC2)(CNC(c2ccc3ccoc3c2)=O)CCN(C(=O)C(F)C2CCC2)C1 CC(C)(C)CCC(F)C(=O)NCC1(O)CC(C(=O)NC2(C(N)=O)CCC2)C1 CCCCCC(=O)NCC(=O)NCCCC(C)(C)NC(c1cncnc1C)=O N=C1NC(=O)C(CC(=O)NCC(O)CCNC(=O)CSCc2ccncc2)S1 c1(OC)c(C(N2CCC(NC(=O)CCCC(C)(C)C)C2)=O)cc(Br)cc1F N1(C(CCNC(C)=O)=O)CCOC(C(C)NC(=O)CNC(c2cnn(C)c2)=O)C1 c1(NC(C(CCNC(C2C(CC)OCC2)=O)O)=O)cc(C)cc(C)c1O N1(C(CS(=O)(=O)NCC)=O)CCCC(NC(c2cnc(C(C)(C)C)[nH]2)=O)CC1 c1(C(N(C)CC2COCCN2C(c2ncccc2Cl)=O)=O)nc2cccnc2s1 C#Cc1cc(Br)ccc1NC(=O)C=Cc1cc(F)cc(F)c1 c1(C(N2CCCC(NCC)C2)=O)ccc([N+](=O)[O-])s1 c1(C(C(=O)NCC(CC)NC(c2cc(CN(C)C)c[nH]2)=O)(C)C)cccc(O)c1 C#Cc1ccc(C(N2CCC(C(C)(C)NC(=O)CC(C)CC#N)C2)=O)c(OC)c1 C(CNC(=O)C(c1ccccc1)O)(CCNC(c1ccc(F)s1)=O)OC C(=O)(C#CC1CCCCO1)NC1(COC)CCN(C(=O)CSC)C1 C(CC(N)=O)(C(=O)NCCN(C(c1ncccn1)=O)C1CC1)NC(CC(C)C)=O N1(CC(c2ccc(OC)cc2)=O)CCC2(COC(CC(=O)NCC)C2)C1.C(C)(C)(C)O N1(C(C(C)O)=O)CC2(CCC(C(=O)Nc3nnccc3C(F)(F)F)O2)C1 C(=O)(C(O)C(F)(F)F)N1CC(C(C)NC(c2cc(Cl)cnn2)=O)OCC1 C1(NC(CC(CC)C2CC2)=O)CC(N=c2nc(O)c3c(ncn3C)[nH]2)C1 N1(C(c2c(OCC)ccs2)=O)CCCN(C(C2CCCC23CC3)=O)C(C)C1 c1(OC)ccccc1CC(C)CC(=O)NCC1CCN(C(=O)C2=CCC2)CC1 C(C)(C)(CC(=O)NCC1(C)CCCN1C(=O)CCCc1nncn1C)OC Cc1ccc([N+](=O)[O-])cc1C(=O)NCC1CC(C)N(C(=O)COCC(C)(C)C)C1 C(=O)(C1=CCCCCC1)NC(CC)C(=O)NOCC1(F)CCC1 C1(NC(C(CCC)OC)=O)CCCOC12CCN(C(c1nc(=O)n(C)[nH]1)=O)CC2 c1(C(=O)NCCN(C(c2ccncc2C(=O)OC)=O)CC)csc2ccccc12 CC1CN(C(c2ccc(F)cn2)=O)CCN1c1nnco1 CC1CN(C(C2CC(N(C)C)C2)=O)CCN1C(=O)CCc1ccc(C(F)F)cc1 C1(C2CCN(C(=O)C(F)C(C)(F)F)CC2)(NC(CC(C)CC(C)(C)C)=O)CCC1 N1(C(C)C)N=C(C(=O)N(CC(=O)O)C2CC2)CCC1=O c1(CC(N2CCCC(CNC(C3C(C=C)CC3)=O)CC2)=O)ccc([N+](=O)[O-])cc1 C(C)(N=c1nc(C(C)(C)C)[nH]s1)c1ccc(CNC(c2c(C)n[nH]c2)=O)cc1 c1(C(=O)NC(CN(C(C2CN(C)CCO2)=O)CC)C)cc(C)oc1C N1(C(c2cc3[nH]cc(C)c3cc2)=O)CC2(CCOCC2C(N2CC(F)(F)C2)=O)C1 C(=O)(C(C#N)C(C)C)NC(CC)(C)CNC(=O)CSc1cccc(F)c1 N1(C(c2ccn(CC)c(=O)c2)=O)CC2CCCC(NC(C3(SC)CCC3)=O)C2C1 c1(C(=O)NCC(CNC(C2CC(CC)C2)=O)O)oc2ccccc2c1COC C1(CNC(C2CCN(C(C(CC)N(CC)CC)=O)C2)=O)(CC)CCCCC1 c1ccc(SC2(c3noc(CNC4COCCO4)n3)CCCC2)cc1 CC#CCCC(=O)NCCC1CCN(C(C2CC23CCOC3)=O)CC1 C12(CNC(CC3CCC(C#N)C3)=O)CCC(F)(CC1)C2.C12CCC(C1)NC2=O C1(OC)CC(CNC(=O)C(=O)N(C)C)N(C(c2cncc(C)n2)=O)C1 c1(SC(C2(CN(C)C)CC2)=O)ccc(F)nc1 C(=O)(C1CCCn2c(C)nnc21)N1C2C(CNC(C=CC)=O)(CCC2)CC1 C(=O)(C1=CCC2CCC1N2C(C1CC=CC(O)C1)=O)NCCN(C)C c1(C(=O)NC2CCCCN(Cc3ccc(C)cc3Br)C2)cnn2c1CC(C)CC2 N1(C(C(C=C)(F)F)=O)CCC(F)(CNC(=O)Cc2cnccc2Cl)CC1 C1(NC(C(CC)OCC)=O)CC2CC(NC(c3cc(OC)ccc3Cl)=O)CC2C1 c1(C(=O)NCCC2CCN(C(Cc3cn(C)nc3)=O)CC2)cc2occc2n1C C1(n2c(C(=O)NC(CC(=O)OC)C)ccn2)CCCN(C(C)=O)C1 N1(c2nc(Cl)nc(C)c2F)CC(CNC(=O)CCC(C)N(C)C)OC2(CCC2)C1 C12(C(=O)NC3CCCC(NC(c4cc(Cl)cc(Cl)c4)=O)C3)CC3CC1C2C3O c1(C(N2C(CNC(C(C(C)(C)O)F)=O)CC(O)C2)=O)ccc([N+](=O)[O-])c(O)c1 C(=O)(C1=CC2CCCC12)N1CC(C)N(C(c2cc(C(N)=O)no2)=O)CC1 n1(C(CC)CC)nc(C(=O)NCC(C)CNC(c2csc(COC)n2)=O)cc1C c1(SCC)ccc(CN2CC(=O)NC(C)C2)c(C)c1.c12cc(ccn1)C(=O)NC2 C(CC(=O)N1CCC(C(=O)NC2CC(C)OC2=O)O1)=CC C#Cc1cc(C(N2CCC(O)C2C(=O)NC(C)CO)=O)ccc1C C1(C(NOC(CC)C)=O)CCN(C(C2COC(C)C2)=O)CC1 c1(Oc2ccccc2)ncnc2ccccc12.[O-][n+]1cnc2c(c1)N2 C(=O)(C1=CCOCC1)N1CCC(n2cc(CNC(CC(=C=C)C)=O)nn2)C1CC N1(C(c2ccc(C)nn2)=O)CCC2CN(C(=O)Cc3cc(C)ns3)CC2C1 C(=O)(CCC(=O)c1cc(C)sc1C)NCCCNC(C(C)NC(CC)=O)=O c1(C(N(CC#CC)C)=O)cc(CNC(C2CC3CC3C2)=O)no1 CC1CC(C(N2CCC(O)(CNC(c3cc(Br)no3)=O)C2)=O)CC(C)(C)C1 N1(C(c2cc(COC)on2)=O)CCCN(C(c2sccc2C(F)F)=O)CC1CO c1(C(N2C(CN(C(=O)C(O)Cc3[nH]cnc3C)CC)CCC2)=O)ccc(O)cc1 CC(CC(F)F)C(=O)NCCCOCCNC(=O)C=CC=Cc1ccccc1 C1(N(C(CCOCCOCCOC)=O)C)CCCCN(C(=O)CCC(C)SC)C1 C1(CCC)CCCC1C(=O)NC(CC1CCOCC1)C(=O)NC1C2CCCC12 C(N=c1nc(N2Cc3c[nH]nc3C2)c2sccc2[nH]1)C1(C)CCCOC1 c1(CNC(C(C)OC(C)=O)=O)cc[nH]c1C(N1CCC(F)C1)=O C1(C)(n2c(C(COC)OC)nc(-c3ccc(Cl)cc3)n2)CCS(=O)(=O)C1 c1(C(=O)NC)cc(=NCc2ccc(OC)c(OC)c2)cc[nH]1 N1(C(c2cnc(CC)nc2)=O)CC(CNC(C2CC(N(C)CC)C2)=O)C2(CC2)C1 c1(C(=O)NC2CC(NC(C3(N4CCOCC4=O)CC3)=O)C2)cnc2n1CCOC2 N1(C(c2n(CC)ncc2)=O)CCC2(CCN(Cc3ccncc3Cl)C2)C1 Cc1nccc(CCC(N2CCC(CO)(NC(=O)COCCO)C2)=O)n1 c1(CNCCC(c2ccccc2)C)nc2ccccc2n1C(C)C C(=O)(C(O)(C(F)(F)F)C1CC1)NCCN(C(c1n(C(C)C)ccn1)=O)C c1(OC)cccc(COCC(=O)NC2CCCC2NC(c2cc(C)sn2)=O)c1 CN1CCN(C(c2ccc(Cl)cc2)=O)C(C(N2CCC(CN=[N+]=[N-])C2)=O)C1 C1(C(=O)NCCCNC(c2c(N)sc3c2CCC3)=O)Cc2cc(F)cc(F)c2O1 C1(C(=O)NC(COC)CNC(c2cnc(SC)s2)=O)CCCSC1C c1(OC)cc(C(N2CC(CNC(c3coc(O)n3)=O)C(C)(C)C2)=O)cc(F)c1 O=C1NC2CN(CC(=O)NCC3CCC=CCC3)CC2N1CSc1ccccc1 N1(C(C(C)(C)N(C)C)=O)CCCC(N(C(=O)C(C)(C)C2CCCOC2)CCF)C1 N1(c2ncc(C(=O)OC)cn2)CC(NC(c2cnc(C(C)(C)C)o2)=O)C(C)(C)C1 C(=O)(C(COC)CC)NC(C(=O)NCC(CCC)C)C1CC1 N1(C(c2cc(C(F)(F)F)c[nH]2)=O)CCN(Cc2c(O)cccc2Cl)C(CO)C1 c1(NC)cncc(C(=O)NC(C)C=CC(=O)N(C(C(N)=O)C2CC2)C)c1 c1(C(=O)NC2CC3CN(C(C4(CC#C)CC4)=O)C2C3)ccc2c(c1)C(=O)NCC2 c1(C(N(CCCN(C)C(C2CC=CCC2)=O)C)=O)cnc(C(F)F)cn1 C(=O)(C#CC1CCC1)N(CCCCNC(c1c(CC)noc1C)=O)C c1(C(=O)NCC(CC=C)NC(c2csc(CO)n2)=O)cnc(Cl)c(C2CC2)c1 N1(C(C2(F)C(C)C2)=O)CC2(C)CN(C(c3cccc4c3NCCC4)=O)CC2(C)C1 C(=O)(C(F)(F)CSC)N(C)CC1(O)CN(c2ccc(C(=O)OC(C)(C)C)cn2)C1 c1(CC(C(=O)NCCCC(C)NC(c2cscn2)=O)O)cc(Cl)cc(Cl)c1 c1(CC)cc(N2CCCC(C(=O)NC(c3ccnn3C)C)C2)ncn1 C=C(CNC(=O)C1=CCC(NC(C2CCC(C)(C)CC2)=O)C1)c1ccccc1 c1(C(=O)NCC2(O)CC(NC(c3cc(C(=O)OC)sc3)=O)C2)cccc(=O)o1 c1(C(N2CC(N(C(CCC#C)=O)C)C(C)CC2)=O)cc[nH]c2nccc1-2 N1(C(C(C)CN2CCOCC2)=O)CC=C(CNC(c2cc(F)cc(Cl)c2)=O)CC1 CN1CCN2C(C1)C(=O)NCC2=O.c1(N)ccc(F)cc1.C(CC#N)CC#N C12(CC)CN(C(=O)C=C(C)C(F)F)C(CNC(=O)CC(C)c3ccco3)(C1)C2 c1(CC)noc(-n2ccnc2-c2cccc(C)c2Oc2ccccc2)c1C#N N1(C(CCOCCN(C)C)=O)CCOC2(CCN(C(C3CCC3(F)F)=O)C2)C1 C(=O)(C(C)C(=O)Nc1ccccc1)NC(CNC(C1(COC)CC(OC)C1)=O)C C=C(C)C(CC(=O)N1CCC(N(C)C(C2CC3C=CC2C3)=O)CC1)OCC C12(C(=O)NCC3(NC(C4(c5ccccc5Cl)CC4)=O)CC3)OCCCC1C2(F)F c1(-c2c(CN3CC(O)C(F)C3)cccc2)c[nH]c2ccc(Cl)cc12 c1(C(=O)NC2C(CNC(=O)CCC3NC(=O)NC3=O)CC2)cc(F)c(F)cc1O C1(CCNC(C2(C)CC(=C)C2)=O)CN(C(C2CCS2(=O)=O)=O)CCS1(=O)=O CCC(C)(C)C(C)NC(=O)C(CN(C)C)NC(c1ccc(SC)o1)=O N1(C(C(=O)NCCOC)=O)CCN(C(=O)CCn2ccnn2)CC1.C1C(=O)N1 C1(NC(c2c(C)nns2)=O)CN(C(=O)C(C2CCCCC2)O)CC1n1cccn1 Cc1cccc2c(C(=O)NC3CCN(C(C45CC(F)(CO4)C5)=O)C3)coc12 C(=O)(C1=CCCC1C)NC(CCC)C(N1CCOC(C)CC1)=O C(CC)(C(=O)NCCC1CC(NC(=O)CCc2cc(C)on2)C1)OCC C1(CC)(NC(=O)C(C)NC(=O)NC)CCCN(C(c2[nH]nc(OC)c2Cl)=O)C1 CC(CCCCNC(C1(CO)CCOCC1)=O)NC(=O)C(C)SC(F)(F)F N1(C(CN(CCOC)C)=O)CCCCCCC1C(=O)NC1CN(C)CC1(C)C c1(C(=O)NC(C2(O)CN(C(=O)CC3CC4CCC3O4)C2)C)cccc(Cl)c1F N1(C(c2c(CC)con2)=O)CC(NC(C23CCC(CC2)CC3)=O)CC(C)C1 c1(SCC)n[nH]c(=NC2CC3(CCC(C(=O)OC)CC3)C2)s1 c1(C(=O)NC(C(CO)NC(Cc2c(C)noc2)=O)C)ccc(OC(F)F)cc1 c1(OC)c(C(=O)NC2CCC(N(C(=O)CC(C)C3CC3)C)CC2)ccnc1F N1(C(CS(CCC)(=O)=O)=O)CCC2(CC1)CC(CNC(=O)Cc1cc(C)on1)C2 C1(OCC(=O)NCc2c(C(C)C)noc2)CCN(C(=O)CCC2CC2(C)C)C1 CN=c1cc(C(N2CCOC(CCNC(C3CC4CC4C3)=O)C2)=O)cc[nH]1 CC1(C)CCCC(C(=O)NC2CCCC2NC(=O)CN2CC=CC2)C1 CC1(C(=O)NCC2(NC(C3CC(=O)N(CC(F)(F)F)C3)=O)CC2)CCCC1(F)F C(c1c(F)cccc1F)=CC(=O)N(C1C2CN(C(C3(C(C)=O)CC3)=O)CC21)C N1(C(c2ccc(C)n2C)=O)CC(C2CC2)(C(N2CCC(F)(CF)C2)=O)C1 Cc1ccc(C=CC(=O)NCC2(NC(C3CC4C=CC3O4)=O)CCOC2)cc1Cl Cn1cc(Cl)cc1C(=O)NCCN(C(C1CCOC1)=O)CC1CC1 C(c1ccc(S(N)(=O)=O)cc1)=CC(=O)NCCN(C(CC=C=C)=O)CCOCCO c1(CC(=O)NC2C3(CN(C(CCNC(N)=O)=O)C3)CC2)ccc2c(c1)NC(=O)C2 N1(C(CC)=O)CCCC2(CCN(C(C3CC4(F)CC3C4)=O)C2)C1 c1(N(C(C)C)C)ccc(C(=O)NC(C)CCCNC(C2COC(=O)C2)=O)cc1 N1(C(=O)CC2CCCC2O)CC2CCN(C(=O)CCCc3ccncc3)CC12 C1(NC(C=C(C)C)=O)CN(C(c2cc(OC3CCCC3)ccn2)=O)CC12CCC2 CCCCS(=O)(=O)NCC(N1CCCCC1C(=O)NC1COCCN1C)=O N1(C(C)=O)CCN(C(=O)CCn2cc(-c3cnc(C)o3)nn2)C(C)C1 c1(C(C(=O)NC2CCC2)N(CCCCOC)C)ccc(OC)c(Br)c1 C1(C(N(CCC(=O)NC)CC)=O)CCCCN1C(=O)CCC1CCCCO1 S(=O)(=O)(c1ccc(NC(C2CCC3C(CC2)C3(F)F)=O)c(C(F)(F)F)c1)N(C)C c1(CC(C(=O)N(CC)CC2CCC2)NC(=O)C(C(C)C)SC)cnn(C)c1O c1(C(=O)NCC2CN(C(CC3(C=C)CC3)=O)CC2O)cccc2sncc12 C12(C(=O)NC3C(CNC(c4n(CCC)ccc4)=O)CCCC3)CC(C1)S(=O)(=O)C2 CCCC(C(=O)N1C(C(=O)NCCCC(C)(F)F)CCC1C1CC1)OC c1(SCC#C)ccc(C(=O)NC2CC2NC(=O)CN(C)C(=O)OC)cc1 c1(OC)[nH]c(=N)nc2sc(C(=O)NCCC(C)NC(=O)C(C)(C)O)cc12 OCC(F)(F)C(c1ccccc1)NC(c1ccc(Cl)cc1)C1CCC1 c1(CC(N2CC(CNC(=O)Cc3cccs3)C(O)C2)=O)ccc(O)c(Cl)c1 c1(C(=O)NCC(CCNC(C(CC)OC)=O)O)ccc(NC(=O)NC(C)C)cc1 c1(C(=O)OC)cc(S(=O)(=O)N2CC3(CCC(NC(=O)CO)C3)C2)ccc1C N1(C(CCCOCC=C)=O)CCCC(CNC(=O)C=CI)C1 Cn1ccc(=O)c(C(=O)NCC2CCCC(NC(c3ccc(Cl)[nH]3)=O)C2)c1 c1(C(N(CC(C)NC(=O)Cc2csc(C3CC3)n2)C)=O)ccc(C2CCC2)nc1 c1(C(N(C2CN(C(C3C(OCC)C3C)=O)C2)C)=O)ccn2c(C)cc(C)nc12 N1(C(CC(C)(C)C)=O)CCC2CN(C(C3(N4CCCC4)CCC3)=O)CCC2C1 N1(C(=O)NC2CCC=CCC2)CCC2(CCCO2)C1 c1(CCC(=O)NCCC(C)NC(C2CCN(C)C2=O)=O)cc(F)ccc1F CC(C)(O)C(F)(F)CNC(c1ccc(CNC(c2cnnn2C2CC2)=O)o1)=O Cc1cc(C(=O)NCC2CN(C(=O)C=Cc3cc[nH]n3)CCCO2)c(C)c(C)c1 N#Cc1ccc(C(N2CCC(C(N3CCN(CCCO)CC3)=O)C2)=O)c(Cl)c1 c1(C(=O)NC(CC(C)NC(C2(CC)CCC2)=O)C)ccc(C2=CCOCC2)cc1 N1(C(c2cccc(C)c2)=O)CCC(CNC(=O)CC(O)C2CC2)C(F)(F)CC1 C(=O)(C1SCCc2ccccc21)NC1CC(NC(COCCCC)=O)C1 N1(C(=O)Nc2ccc(Cl)cc2)CC2CCN(c3nccc(OC(F)F)n3)CC2C1 Cc1ccc2c(c1)CN(C(=O)COCCNC(C1CCCSC1)=O)C2 N1(C(=O)OC)CCCCC1C1CCN(CC(c2cn(C3CC3)nc2C)=O)C1 c1(NC(=O)CCC2CCCN2Cc2cc(Br)cc(Br)c2)cccc2ncsc12 C1(C2CCN(CCC3CCCCC3)C2)CCC(F)(F)CC1.O=C1CCCNC(=O)N1 C#Cc1cc(F)c(C(=O)NC23CCC(NC(c4nnc(C)s4)=O)(CC2)C3)cc1F N1(C(C(CC)(C)O)=O)CC2CC1CC2NC(c1ccccn1)=O c1(OC)ccc2c(C(N3CC4CC(NC(C5(F)CC5)=O)C4C3)=O)ccnc2c1 C1(NC(c2cc(C(C)C)no2)=O)CC2(C1)CC(NC(=O)C=CC(F)(F)F)C2 c1(C(=O)NCCCCCN(C(CSCCCC)=O)C)ccc(C2CC2)nn1 N1(C(=O)C2=COCCO2)CCC(C2CCN(C(c3c[nH]nc3C(F)F)=O)C2)C1 C(=O)(C(C)(O)CCN(C)C)N1CC(CNC(CC2ON=C(CC)C2)=O)OCC1 N1(C(C(C)NC(C2(CC)CCOC2)=O)=O)CCC(F)(COC)CC1 C(=O)(CS(=O)(=O)C1CCCC1)NC1CCCN(C(CCSCC(N)=O)=O)CC1 C(=O)(C(C)CC(F)(F)F)NC(c1ccccc1)CNC(c1c(CC)c[nH]c1)=O c1(C(N2CCC3(NC(CCSCC(C)C)=O)C(C2)C3)=O)cc([N+](=O)[O-])cn1C C1(CC(=O)NCC)COc2ccc(Br)cc2C1.c12cn(nn1)CC(C)SCC2 C1(CNC(C(CC)(C)O)=O)CC2(CC2)CN1C(=O)Cn1ncnn1 C(=O)(C(C)(O)CC(C)C)NCCCCC(=O)NC(c1c(C)ncs1)C N1(C(C2CCCOCC2)C(=O)NCCOCC)CC(O)CC(O)C1 Cc1[nH]nc2c(-c3cc(C(=O)NCC4(C)OCCO4)c4n[nH]cc4c3)cccc12 N1(C(Cc2ccc(SCC)cc2)=O)CCN(C(=O)CCN(C)C)CC1C(F)F CC1CN(C(c2ccccc2C#N)=O)C(C)CN1C(C1CCC1)=O c1(C(CNC(=O)CCC2CC2(F)F)NC(c2ccsc2)=O)ccccc1F n1(COC)nccc1C(=O)NCC1CCCC1NC(=O)C(=O)NC(C)C C1(C(=O)NC2CCN(C(c3cc(OC)n[nH]3)=O)CC2F)CCc2n[nH]cc2C1C Cc1csc2c(C(=O)N(C3CN(C(c4coc(S(C)(=O)=O)c4)=O)C3)C)ncnc12 c1(C(N2CCN(C(=O)C=Cc3cnc[nH]3)C(C(F)F)C2)=O)nnn2c1CSCC2 N1(C(C2C(C(C)(C)C)C2)=O)CCN(C(C2(Br)CC2(F)F)=O)CC2(CC2)C1 Cc1ncc([N+](=O)[O-])cc1C(=O)NC(C(C)NC(C1(CC(F)F)CC1)=O)C(C)C C1(NC(C2(C(N(C)C)=O)CC2)=O)CC2CC1N(C(C13CCC(CC1)C3)=O)C2 CCCC(C(=O)NCC(C)NC(=O)C(F)=C1CCCC1)c1ccccc1 c1(OC)ccccc1CCC(=O)NC1CC1NC(C1(c2ccccc2)CC1)=O C1(CNC(c2nc(C)sc2)=O)CCN(C(=O)C2=NOC(C)C2)CC1(F)F N1(C(C(C(C)O)C)=O)CCN(C(c2cc(CO)n(C)n2)=O)C(CO)C1 C(C(=O)NCCCCCCN(C(=O)CSC(F)F)C)(C(C)C)OC C(=O)(C#CC1CCOCC1)N(CC(O)CN(C(=O)CC1CCC(F)(F)C1)C)C c1(OC)cc(C(N2CC=CC2CNC(=O)CCc2cccc(Cl)c2)=O)ccc1Cl c1(NC(C2CCCCN2C(c2snc(Cl)c2Cl)=O)=O)cc(Cl)c(O)cc1Cl N1(C(C2CN(C(C)C)C2)=O)CC(n2cc(CCC(=O)N(C)C)nn2)C(C)C1 C1(NC(c2noc(CC)c2C)=O)CN(C(=O)C(C)(COC)CC)CC12CC2 Cc1cc(O)n2ncc(C(N3CCCC(C(=O)N(C(C)C(N)=O)C)C3)=O)c2n1 c1(C(=O)NC2CN(C(c3ccc(CCC)s3)=O)C2)ccc2cnoc2c1 C1(NC(CCCC)=O)CCC(N(C(=O)CC2OCCCO2)C)CC1 c1(N(C(=O)CN2CCC(Cc3ccccc3)CC2)C2CC2)cnc2c(c1)OCO2 N1(C(CCCSC(C)(C)C)=O)CC(CNC(=O)CCC(N)=O)N2CCC1C2 N1(C(=O)CCc2ncc[nH]2)CCN(C(c2cnc(C(F)(F)F)s2)=O)CC1 c1(OCC(=O)NCC(C)(C)N(C(C2(CC(C)C)CCC2)=O)C2CC2)ccc(Cl)cc1 C(=O)(CCCC(C)=O)N(C)CC1(O)CCN(C(C2(CCCC)CCC2)=O)C1 N1(C(c2c(CC)nn(C)c2CC)=O)CCOC2(CCSC2)CC1 N1(C(C2CCC(C)CC2)=O)CCCN(C(C2(F)CCC2)=O)CC1 N1(C(=O)CSCc2cn(C3CCOCC3)cn2)CC(C2CN(C(C)(C)C)C2)C1 N1(C(c2ccc(O)nc2Cl)=O)CC(CO)C2(C1)CN(C(C13COCC(C1)C3)=O)C2 c1(C(N2CCCCCC(NC(=O)Cc3ccon3)C2)=O)cccc2c1CCO2 N1(C(c2nc(C)oc2C)=O)C2CCC(C2)C1C(N1CCC1CO)=O Cc1nc(N2CC3CC(NC(C4CCC(=O)NC4)=O)C3C2)ccc1[N+](=O)[O-] N1(C(C(COC)(F)F)=O)CCC2(CCCN2C(=O)C=CCn2cncn2)C1 c1(C(=O)NCC2C(CNC(C3(C(C)C)C(C(C)C)C3)=O)C2)cc(C#N)c[nH]1 CCC(CC(=O)NCCC1CCCN1C(c1cccnn1)=O)C1CCC1 C1(C)(CNC(c2c(CC)n[nH]c2)=O)CCCN(C(=O)CCNC(=O)COC)C1 N1(C(CC2C(C)(C)CCCO2)=O)CC2CCC(C1)N2C(=O)C1=CCSC1 CC(=O)CCCCC(=O)NC(c1nocc1C(=O)NCC1=CCCOC1)C Cc1cn2c(C(=O)NC3CC(O)CN(C(=O)CN(CC(C)(C)C)C)C3)cnc2s1 C1(N(C(CC2N(C(c3c(C)nn(C)c3)=O)CCC2)=O)C)CCCC(C)C1C C1(CNC(Cc2c(C)scc2)=O)C(O)C(O)CN1C(C1CCCCCCC1)=O C(=O)(CC(C)(C)CC(F)(F)F)NC1(C)CCC(NC(c2cn(CC)nc2)=O)CC1 CCCCCCCC(=O)N1CC=C(CNC(C2(N(C)C)CC2)=O)CC1 CC1CN(C(c2cccc(-c3ccsc3)c2)=O)CCN1C(c1cccs1)=O CC(C)C(CCC(=O)NC1CCC(=O)NC1=O)NC(c1cc[nH]c1)=O c1(CCC(=O)NCC2N(C(C(CC)(C)CO)=O)CCCC2)nc2ccccc2s1 c1(CCC(=O)NCC(CN(C)C(C2CC23CCSCC3)=O)O)cccc(F)c1F C1(CNC(C(=O)N(CC#C)CC=C)=O)(Cc2ccc(Cl)cc2)CCN(C)CC1 N#Cc1cc(C(=O)NCC2CCCN2Cc2ccc(C(=O)OC(C)(C)C)[nH]2)cs1 c1(C(=O)NCc2cccs2)ccc2c(C(=O)Nc3cnc(Cl)nc3)n[nH]c2c1 C1(NC(C2C(c3c(C)cccc3)C2)=O)CC(C)CN(C(=O)CSC(F)F)C1 N1(C(CCC(N)=O)=O)CCC(O)(CNC(c2n[nH]c3c2CCC3)=O)CC1 C(CCCCC(=O)NCCc1ncccn1)NC(=O)CC1CC2C=CC1C2 CCC(CN(C)C)CC(=O)N(CCCCNC(c1nn(CC)nc1C)=O)C C#Cc1cc(C(=O)NC(C)(C)C(C)NC(C2COCCO2)=O)ccc1C C(C)(C)(C(F)(F)F)NC(C(C1N(C(c2c(C)nsc2)=O)CCC1)(C)C)=O N1(C(CC=CCN(C(=O)CC2CSC2)C)=O)CCOC(C2CCC2)C1 c1(NC(C2(CC)CCCN2C(c2cc(C(C)C)[nH]n2)=O)=O)cnc2ncnn2c1 C(=O)(CS(=O)(=O)CC(F)(F)F)NC1CCC(N(C(=O)COCc2nc[nH]n2)C)C1 C1(OC)CC2(C1)CC2C(=O)N(CC(O)CN(C)C(c1ccccc1F)=O)C c1(-c2cc(C(N(C3CN(C(C4CCC45CCC5)=O)C3)C)=O)n[nH]2)ccc(O)cc1 c1(OC)cc(F)c(C(=O)NCC(O)CCNC(c2cc(C)cnc2N)=O)c(F)c1 N1(C(C2=CCC(C)CC2)=O)CCCC2(CCCN2C(C2CCS(=O)(=O)CC2)=O)C1 CN1C(=O)C(F)CC1C(=O)NCC1CC(NC(c2snnc2C2CC2)=O)C1 c1(C(=O)NCCOCCN(C(Cc2ccn(C)n2)=O)C)ccnc2ccsc12 C1(C(N2CC(CCCCNC(CCc3cc(C)no3)=O)C2)=O)CCOC(=O)CC1 S(=O)(=O)(c1ccc(NCC(C)(C)CC(F)(F)F)nc1)NC(CCC)C(C)O c1(CCC(=O)NC(C2N(C(C(C)OC)=O)CCC2)C)ccncc1Br c1(NC)cnccc1C(=O)NCC(C)CN(C(=O)CC1COCCN1C(C)=O)C C1(CCC(=O)NCC(CC)C#N)CCCCN(C(C2CC(F)CN2C)=O)C1 c1(OC)ccc(Br)c(C(=O)NC2CC(C)(NC(=O)COC3CC=CC3)C2)c1 C1(CC(=O)NC(C(C)C)CNC(C2CC3(C2)CC3F)=O)CCCCC1(C)C N#Cc1ccc(C(N2CCCC(O)(CNC(c3ccccc3Cl)=O)C2)=O)cc1F N1(C(=O)NCC(C)C2CC2)CCCC2(CC1)CNC(=O)O2 C(=O)(C(F)Cc1ccccc1)NCCCN(C(c1cc(C)on1)=O)CC c1(C(=O)NCCCN(C(=O)CN2CCOCC2)C2CC2)ccc(OC(F)F)cc1 N1(C(CN(C)S(N)(=O)=O)=O)CCc2[nH]nc(CNC(C3(C)CNC(=O)C3)=O)c2C1 N1(C(c2cccc3cnccc23)C(=O)NCC=C)CCC(S(=O)(=O)C(C)C)CC1 C1(NC(=O)NC(C(C)F)C)CCCC1C CCC(CC)C(F)C(=O)N1CCCC1(C(N1CCCC(OC)CC1)=O)CC CC1CN(C(=O)Cc2cccc(Cl)c2F)CCN1C(c1cc(F)ccc1F)=O c1(-n2ccc(NC(=O)Nc3cc(C(=O)OC)[nH]n3)n2)ccccc1C CC1OC(C)C(C(=O)NCC2CN(C(C3CCCN3C(=O)C3CC3)=O)C2)C1C N1(C(CC2CC(C)OC2C)=O)CCC2(C1)CN(C(C1(C)CCC(=O)NC1)=O)C2 C(C(C(C)(C)C)NC(c1cncc(F)n1)=O)NC(C(C1CCC(=O)N1)C)=O N1(C(CCc2ccn(C)n2)=O)CCC2(C)CN(C(c3cc[nH]c3)=O)CC12 C(=O)(C1=CCCCC1C)N(CC(CC)NC(c1cnc(OC)c(OC)c1)=O)CC C1(CC(=O)N(CCOCCNC(C(CC)(C)O)=O)C)CC2(CCCC2)CO1 C1(CNC(C(C)CC2CCCO2)=O)CCC(NC(c2cc[nH]c2)=O)CC1 c1(C(N2CC(NC(COCC=C)=O)C(O)CC2)=O)cc(O)c2nc(C)n(C)c2c1 N1(C(CNC(CC)=O)=O)CC(CNC(C2(c3cc[nH]n3)CC2)=O)CCC1C C(CC(O)C(=O)NCC1(CO)CCOC1)NC(CC1(OCC)CC1)=O C1(C(=O)NC(COCC)CO)CC(CC)CCN1C(c1ccnc(O)c1)=O c1(CC(C)C(N2CC(c3ccccc3)C(O)C2)=O)ccc(C#N)cc1 Cc1ccc(-n2nc(CC3COC3)nc2Cn2cc(Br)cn2)cc1Cl c1(C(=O)NCC(CC)NC(C2CCCC2(F)F)=O)c(C(F)F)nc2ccccn12 c1(CNC(c2c(C)coc2)=O)ccc2c(c1)CCCC2NC(=O)Cc1cncs1 C(=O)(C(CCC)NC(C1(CCC)CCC1)=O)NCCSCCC=C C1(CNC(C(CC(C)C)NC)=O)CCOC2(CCOCC2)C1 c1(C(=O)NCC(C)N(C(c2cncc(N(C)C)c2)=O)CC)ccc(C)c(O)c1 N(C1CC(C)(C)Oc2ccc(F)cc21)C(C(N1CC(C)C=C(C)C1)=O)=O CC1(C)CCC=C1C(=O)NCCOC1CCN(C(C2CCOC(=O)CC2)=O)C1 O=S(=O)(c1[nH]c(=NCC2CC3CCC3C2)ccc1Br)NCc1ccccc1 C1(CCCC)CCCN1N(CCOCCOC)CCC1CC1 C(=O)(C(C)CCCC(C)=O)N1C(C(=O)NCC(C)C(=O)OC)(CC)CCC1 C(=O)(C(O)CCc1ccccc1)NC(CNC(c1nc[nH]c1CO)=O)C1CCC1 C1(C(=O)NCCN(C(=O)CC2CCCC(=O)C2)CC)CC2OC1C1CC21 C1(C2CCN(C(c3sc(C)nc3C)=O)CC2)(NC(C=CCCC)=O)CCC1 Cc1c(C(=O)NC(C)(C)CNC(=O)C(C)O)[nH]c2c(C)cccc12 N1(C(C=C(CC)C)=O)CCOCC1CN(C(=O)C(C)(C)Cc1ccccc1)C C1(C(=O)NC2CCN(C(Cc3c(C)nc(SCC)s3)=O)C2)CC(=O)OC1(C)C N1(C(C2(C(C)(C)OC)CC2)=O)CC(OC)C(NC(=O)CC2CC3CC3C2)C1 C12(NC(=O)COC3CCCCC3)CCCC1N(C(=O)CCc1ccco1)CCC2 N1(C(CC(=O)N(C)C)=O)CCC(NC(C2(C)CCN(C)C2=O)=O)C(CO)C1 N1(C(COC)=O)CCC2CCCC12CNC(c1c[nH]c(=N)o1)=O Cc1ccc(-c2cccc(NCc3ccc(C)c(Br)c3)n2)c(O)c1 CC1CC(NC(c2cc(C(C)(C)C)on2)=O)CN(C(c2cccn(C)c2=O)=O)C1 c1(N2CC(=O)NCCC2)nc(N2CCC=C(F)C2)c2ccccc2n1 N1(C(c2cccc(C)c2)=O)CCC2(CCCN(C(c3ccnn3C(C)C)=O)C2)C1 CC1CCC(NC(C23CCN(CC2)C3)=O)CN1C(C1CCN(CC(F)F)CC1)=O c1(C(=O)NC(C2CCN(C(C3C(C)C3C)=O)C2)C)cn(C2CCC2)cn1 CC1CCN(C(=O)Oc2cccc(SC(F)(F)F)c2)CC1(F)F CCS(=O)(=O)c1ccccc1CN(C(=O)C(N)=O)C Cc1cc2c(C(N3CC(CNC(c4nc(Cl)cs4)=O)CCC3C)=O)cccc2o1 C1(OC)(CNC(c2cnc(CC(C)C)s2)=O)CN(C(C2CCCN2C(C)C)=O)C1 Cc1nc(C2CCC2)oc1C(=O)NCC1CCC(NC(c2ccc[n+]([O-])c2)=O)C1 c1(C(N2CC(CCNC(C3(OC)CS(=O)(=O)C3)=O)OCC2)=O)cc(C)ncc1C C1(N(C(c2c(C)ncs2)=O)C)CCN(C(=O)CC2CC=CCC2)CC1 C(=O)(CS(=O)(=O)C(C)(C)C)N1C(CNC(CC(C)(C)C(F)F)=O)CC(F)(F)C1 c1(CSCC(=O)NCC2CCC(NC(C3(CC(F)F)CCC3)=O)C2)ccccc1 C1(CNC(=O)NCCC(CC)(F)F)CC(OC)C12CCC2 N1(C(c2nc(C)nn2C)=O)CCC(CO)(CNC(C2C3CCCCCC23)=O)CC1 CC(CN(C)C(c1cnc(S)n1C1CC1)=O)N=c1[nH]c(Cl)nc2ccc(Cl)nc12 C(=O)(C#CC1(C)CCCO1)NC1C(C)(C)CCN(C(C(C)NC(C)=O)=O)C1 C1(O)(CNC(C2CC(NS(C)(=O)=O)C2)=O)CCCN(C(C2CC23CCC3)=O)C1 Cc1cc(C(N2CCCCC2CN(C(=O)CCC2CCC(=O)NC2)C)=O)n(C)n1 C1(C(=O)NC(CCN(CC)CC)C)CC2(CC2)CN1C(c1oc(C)nc1C)=O C1(C(=O)NC(C(CO)NC(c2c(C)nn[nH]2)=O)C)Cc2cc(Br)ccc2O1 CC1(C)CC(CNC(c2cnnn2Cc2ccccc2)=O)N(C(C2CCO2)=O)C1 CC(CNC(=O)CCNC(c1ccco1)=O)CNC(=O)C(C)OC(C)(C)C C1(C(N(CCCNC(=O)Cn2ncnn2)CC)=O)CCCN1Cc1nnn(C)n1 c1(C(CC(=O)NC(CC)(C)CNC(c2csnc2C)=O)O)cccc(F)c1 [N-]=[N+]=NC1CCC(C(=O)NCC2CCCN(C(c3cnn4c3CCC4)=O)CC2)C1 C1(C)(CC)CCC(C(N2CC(COC)(NC(C3COCC3C(N)=O)=O)C2)=O)O1 C1(C(N2CC3OCCN(C(C4CCCC4F)=O)C3C2)=O)CCc2ncccc2C1 Cc1c[nH]nc1C1(C(=O)NCC2CCCC2NCC=CCc2cn[nH]c2)CC1 C(=O)(C(C)(C)CC(C)=O)NC(CNC(C(CC)SC)=O)C(C)C O(S(=O)(=O)c1ccsc1C(F)(F)F)c1ccc(-c2cn(C)nc2)cc1 C12(C(N3CC(CC(C)(C)C)C3)=O)CC(CN(C(c3cnn(C(F)F)c3)=O)C1)C2 N1(C(C2C(C)(CC)C2)=O)CCOC2(C1)CN(C(c1c[nH]c3nccc-3c1)=O)C2 C(=O)(CCCCCCNC(C1CCCOC1)=O)NCC(CC)CC N1(C(c2cnn(CC)c2C)=O)C2CCC(C2)C1CNC(C1CCCCC(=O)N1)=O CCC(C)(C(=O)Nc1cccc(C(N2CCNCC2)=O)c1)OC C1(NC(CCn2ncc(C)c2)=O)(CO)CCCN(C(C2CC(F)(CO)C2)=O)C1 N1(C(C2(SC)CN(C(=O)C(C)C3CCOC3)C2)=O)CCC(=O)N(C)CC1 N1(C(c2c(C)oc(Cl)n2)=O)CCC2(C)CN(C(=O)CN(S(C)(=O)=O)C)CC12 CC1CN(C(=O)CC2C=NN(C)C2=O)CC1C(=O)NCC1CC2(CCC2)C1 C1(C(=O)NCC(C)(C)OCC(=O)NC(c2nnc(C)s2)C)CC(=O)NC(C)C1 C(=O)(C1=C(C)C(C)(C)OC1=O)NCCCC(C)NC(CC(CC)O)=O c1(SC)ccc(C(N2CCSC(C(=O)Nc3nc(O)cs3)C2)=O)c(C)c1 c1(C(N2CC(C(=O)NCCNC(CC)=O)C2)=O)ccc(-n2c(C)ccc2C)cc1 C1(CNC(CCCCOC)=O)C(C2CC2)CCN1C(c1cc(F)c(F)cc1N)=O C1(N(C(C(CSC)O)=O)C)CCCN(C(C2(CC3CC3)CC2)=O)CC1 c1(NCC2OCC(CNC(c3cc(CC)n(CCO)n3)=O)C2)nnc(C)c(C)n1 c1(C(N(C2CCC(NC(c3ccc(F)cc3O)=O)C2)C)=O)ccn2cnnc2c1 C1(NC(c2cnc(CCC)s2)=O)CN(C(c2cc(=O)c(OC)co2)=O)CCC1C n1(C(C)C)cccc1C(=O)N(C)Cc1ccncc1 C(=O)(C(C)(F)C(C)(C)F)NCC1(NC(c2c(C)scn2)=O)CCCCCC1 C1(CNC(C2(CC)COC2)=O)C2CN(C(=O)C=Cc3ccc(C)o3)CC12 c1(C(N2CCC(=CC(=O)N(C)Cc3cccc(O)c3)CC2)=O)ccc(Br)cc1F c1(C(C)=O)c(NC(c2n[nH]cc2NCc2ccc(OC)nc2)=O)ccc2c[nH]nc12 N1(C(c2ncn(CC)c2)=O)CC2CC(O)C1C2NC(c1cc(COC)oc1C)=O C1(C(=O)NCCc2ncc(C)cn2)N(C(C2C3CCCOC23)=O)CC12CCCC2 c1(CCC(=O)NCC2(COC)CCOCC2)cccc(C(=O)OC)c1[N+](=O)[O-] c1(CC2(OC)CC2)nc(C2CCCO2)nn1-c1ccc(Cl)nc1 N1(C(C2(COC)CC2)=O)CC=C(CC(=O)NCCC2(C)CCOCC2)CC1 N1(C(C(=O)NCCN2CCOCC2)C2CCC2)CCCCC1CC1CC1 C1(N(C)CC2CCCC2c2ccccc2)CC(=O)N(C(C)(C)C)C1 C1(C(=O)OC)CCC(NC(C2CC2C2CC(F)(F)C2)=O)C(C)C1 c1(N(C(=O)OC(C)(C)C)CC)ccc(NC(C2CC2C2CC2)C)cc1C#N Cc1ccoc1C(N1CCC(C2CCCN2C(c2ccc(C(N)=O)o2)=O)C1)=O C(CC(C)C)(C(=O)NCCC1CCCN(C(=O)Cn2ccc(C)n2)C1)OC C12(NC(c3cc(C)c(C)s3)=O)CCOC(CNC(=O)CCc3ccn(C)n3)(C1)C2 N1(C(c2cnc(CC)s2)=O)CC2(COC(CNC(=O)C3=CCCOCC3)C2)C1 N1(C(C#CC(C)C)=O)CCC(C)(C)CC1C(=O)NCC(C)(O)CC(C)C Cc1cc(C)c2c(c1)CCC2NC1CCCC(N)CC1 CS(=N)(=O)C1CN(C(=O)CC2COCCN2C(c2ccc(O)cc2F)=O)C1 C=CC1CCN(C(=O)C(C2(C)CC2)NC(=O)C(C)CC(C)C)CC1 C1(C)(CNC(CCC=C=C)=O)CN(C(C2(CS(N)(=O)=O)COC2)=O)CCO1 N1(C(c2ccnc(NC3CC3)c2)=O)CC2CCC1c1ccccc12 CCCC(C)CC(C(=O)NC1(C(=O)OC)CCCC1)N1CC(CO)C(C(F)F)C1 N1(C(c2ccc(CCC)cc2)C(=O)NC2CC2)CCN(S(C)(=O)=O)CC1(C)C C1(OC)(NC2CC(c3ccccc3)C2C)CCCN(C(C2CCCN(C)C2)=O)C1 c1(C(=O)NC2CCN(C(C#CC3(CC)COC3)=O)C2)cc2c(cc1N)OCCO2 C(=O)(C1Cc2ccccc21)N1CC(C)C(NC(C2CCCCC(=O)C2)=O)C1 N1(C(CC(C)C)=O)CCN(C(C2CCC(O)CN2C)=O)C(CCO)C1 c1(C(N(CC(=O)NCC2CC(C)(C)C2)C2CC2)=O)ccccc1C1CC1 N(C(=NC1CCOCC1)NC1CCOCC1)C1CC(OC(C)(C)C)C12CCC2 C1(NC(CC(C)O)=O)CN(C(c2cc(F)n[nH]2)=O)CC12CCC2 C1(C2=CCOCC2)(CNC(c2ccc(F)cc2F)CCC=C)CC1 Cn1c(CNC(N2CCCC2(C)C(c2ccccc2)=O)=O)cnc1Br c1(OC)ccc(C(N2CC(CN3CCOCC3)C3(CCC3)C2)=O)cc1S(N)(=O)=O CN1CCC2(CCCN(C(=O)CC3CCN(Cc4ccccc4)C3)C2)C1 N1(C(c2ncc(Br)cn2)=O)CCC(C2(NC(C3(CO)CCCO3)=O)CC2)C1 n1(CC(=O)NC(C(C)NC(=O)C=C2CCOCC2)(C)C)cc(P(C)(C)=O)cn1 c1(N(C)CC2CC2(F)F)nc2ccccc2nc1N1CCN2CCOCC2C1 C12(NC(c3occ(C)c3C)=O)CCOCC1CN(C(c1cc(Cl)ccc1N)=O)C2 c1(N2CCC(NCC3(OC)CCS(=O)(=O)C3)C2)nc2c(cc1Cl)C(=O)OC2 N1(C(c2cc(C(F)F)no2)=O)CCN(C(=O)C(O)CN2CCCC2)C(CCCO)C1 C1(C(=O)Nc2nc(Cl)ccc2F)CCCC12CCN(C(c1cccnc1Cl)=O)C2 CCC(C)(CC)C(=O)N1CC(CCNC(=O)CC2CC(=O)NC2=O)C1 Cc1nc(C(=O)Nc2ccc(C#N)cc2)ccc1-c1ccc(CO)nc1 C1(NC(c2n(C)ncc2)=O)CC2CC1CN(C(=O)Cc1sccc1Cl)C2 C1(N(C(=O)CCOC2CCC2)C)CCCN(C(=O)CC2CC(F)C2)C1 C1(C(=O)NC2CC(c3ccccc3)(NC(CC=C)=O)C2)C(F)(F)C12CCC2 C1(CCNC(c2ccsc2)=O)CN(C(c2ncc3ccccn23)=O)CCS1(=O)=O C1(CNC(C2N(CC)CC2)=O)CN(C(c2cn(C(C)C)nn2)=O)C2CCCCC12 Cc1c(NC(=O)C(=O)N(C)C)cccc1N.N12CC3(CC1C3)C2=O C1(C(C)(C)NC(CC=CC)=O)CCNC(=O)C1.C12CCN(C1)C2=O N1(C(C2CC3CC2C2CC32)C(=O)NC(CC)(C)C)Cc2ccccc2C(C)(C)C1 C1(NC(c2c(CC)cno2)=O)CC2(C1)CC2NC(=O)Cn1nnc(C2CC2)n1 CC(CNC(=O)CCn1cccc1)C(F)C(=O)Nc1ccc(O)c(Cl)c1 C(=O)(CCC(F)(F)F)N1CCCC(N(C(C(CC=C)NC(C)=O)=O)CCO)C1 N1(CC(CC)C)CC(O)(CNC(c2cn(CC(c3ccccc3)O)nn2)=O)C1 n1(CC=C)cccc1C(=O)NCC1CC1NC(C1CC(C)=NO1)=O Cc1ccc(-n2cc(CO)nn2)cc1NNC(=O)c1ccnc(NC(N)=O)c1 C1(CCC(=O)NCC2N(C(CC)=O)CC2)CCCN1C C1(C(=O)NC2(c3nn[nH]n3)CN(C(C)=O)C2)CCN(C(=O)OC(C)(C)C)CC1 c1(C(N2CC3C(NC(C4CCC(C)(C)C4)=O)(C3)C2)=O)cnn2c1SCC2 C1(O)(CC)CCCN(C(=O)CC(CNC(C2(C)CCCOC2)=O)C2CCC2)C1 C(=O)(C1=CCCCC1)NCC(CN(C(CCc1c(C)cccc1)=O)C)C C(=O)(CCP(C)(C)=O)NC(C)CN(C(=O)Cc1cncs1)C c1(C(=O)NC(CC=C)CNC(=O)CNC(=O)NCC2CCCC2)cc(C)cc(C)n1 c1(NC(C(CC)(C)O)=O)ccc(NC(=O)C(n2ccc(Br)n2)C)cc1C CCC(C)(C(=O)NC1CCN(C(=O)Cc2c(Cl)c(CC)nn2C)CC1)C(N)=O C1(CC(=O)NCC(C2CCCC2)NC(c2ccc(C(C)C)s2)=O)CCNC(=O)C1 Cc1ccc(CC(=O)NCc2ccccc2CN(C)C(c2nonc2N)=O)cn1 c1(-c2scc(C)n2)cccc(C(=O)NC(Cc2ccc(Br)cc2)C(=O)O)c1 N1(C(C=C)=O)CCOC2(CCN(C(c3cn(CC(=O)N(C)C)nn3)=O)C2)C1 C(=O)(C(C(C)C)c1cccc(OC)c1)NC(C(C)NC(CSCCCC)=O)CO C1(CN(C(=O)C(C)C(C)C)CC)CCN(C(=O)CC(C)(C)SC)CC1 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)NC1CC(C)(NC(C=C(C)c2ccsc2)=O)C1 c1(C(=O)NCC(CC)NC(c2cnc(C)n2C(F)F)=O)cncc(N)c1 c1(OC)ccc(C(C)NC(=O)NC2CCCCC2CCO)cc1Br N1(c2ccnc(C(CC)C)n2)CCC(C)C(NC(=O)C(N2CCSCC2)C)C1 c1(CC2(C)CC2)nc(-c2coc(Cl)n2)n(-c2ccc(C(F)(F)F)cc2)n1 N1(C(C2C(CC)CCN2C(C2Cc3nccn3C2)=O)=O)CCC(N(C)OC)CC1 c1(CN2C(C(=O)NCc3ccc(Br)cc3)C(O)CC2)ccc(Br)c(Cl)c1 C1(NC(Cc2ncc(C(=O)OC(C)(C)C)cn2)=O)CC2CC(=O)C1O2 C(=O)(C1CCCc2cc(C#N)ccc21)NCC1(C(C)(F)F)CCC1 C=CCCC(O)CNC(c1cn(CCNC(C2CC2C(F)F)=O)nn1)=O C1(CNC(c2cc(F)n[nH]2)=O)CC12CCN(C(=O)CC1(O)CCCOC1)CC2 C1(C(=O)OC)CC(C)(NC(=O)CN2CCC2C)C1 c1(-n2cc(CO)nn2)ccc(C)cc1F.N1(C(C2(OC)CC2(C)C)=O)CCCC(C)C1 N1(C(Cc2c(C)ccnc2)=O)C(C(=O)NC2C=CCCC2)CCC12CC2 N1(C(C2CCCN(C(C(C)=CC3CC3)=O)C2)=O)CC2CC1CS2=O N1(C(C(C=CC)O)=O)CCOC(CN(C)C(c2cnncc2OC)=O)C1 C1(C)(N(C)C)CCCC1NC(c1cnc(NC(=O)CC2(n3cccn3)CC2)s1)=O N1(Cc2ccc(N(C)C)cc2)CC(NC(c2cc(F)cc(Cl)c2)=O)C(F)(F)C1 c1(C(c2n(CCC(=O)OCC)nnn2)NCc2cn(C)nn2)scc(C)c1C c1(COC(C)=O)ncc2c(n1)CCC2.c12ccc(c(Cl)c1)C(=O)N1CCCC1CN2 Cc1ccc(C(=O)NC(C)CCCNC(C2CC2F)=O)c(O)c1C c1(SCc2onc(-c3ccc(CC)cc3)n2)cc2cccc(Cl)c2cn1 c1(C(N2CCN(C(C3COC3)=O)C(CCO)C2)=O)ccc(Br)c(F)c1 N1(C(C(F)=CC)=O)CC(NC(=O)CNC(C)=O)CC(C)(C)C1 C1(CC(=O)NCCOC2CCN(C(=O)C3=CSCS3)CC2)CCS(=O)(=O)C1 C1(C(=O)NC2C(CNC(c3ncccc3F)=O)CCC2)Cc2nccnc2C1 N1(C(CSc2c(C)n[nH]c2C)=O)CCN(C(c2cc[nH]c2C)=O)CC(CO)C1 N1(C(C(C)SCC)=O)CCC(NC(c2cc3sccc3n2C)=O)C12CCC2 c1(NC(N2CCC(NCCO)C2)=O)cccc(Cn2cncn2)c1 N12CCCOC(C1)COc1nc(c(Cl)cc1)C2=O.c1(COCCO)ccccc1 c1(CNC(C=CC(CC)C)=O)ocnc1C(=O)N(CC(C)(C)O)C C1(N(C(C(C)CC2CCCC2)=O)CC2CC2)CCN(C(C2(CF)CC2)=O)CC1 c1(C(N(CC(CNC(Cc2ncc(C)s2)=O)C)C)=O)cc(Cl)cc(Cl)n1 CC1(C)CC(CNC(C2OC3CCC2CC3)=O)CN(C(c2ccc(Cl)cn2)=O)C1 c1(C(N2C3CC(NC(c4cc(C)nnc4)=O)C3CC2)=O)coc2ccc(F)cc12 O=C(C1CCCc2nn[nH]c21)NCC12CCC1CN(C(C1(F)CCOCC1)=O)C2 c1(SC)nc(C)cc(=NCC(C2CC2)NC(=O)CCN2CCCS2(=O)=O)[nH]1 C(=O)(CC(C)N=c1[nH]c(=NCC2(CCCO)CC2)c2[nH]ccc2[nH]1)NC C#CCC(C)C(=O)N(CCCCCNC(=O)C(C)C)C N1(C(c2csc(CO)n2)=O)CC2CCC(NC(C34CC(CO)(C3)C4)=O)C2C1 C12(NC(C(CSC)OC)=O)CCC(CNC(C3OCCN(C)C3=O)=O)(CC1)OC2 C(=O)(C(CC(C)C)N(C)C)NCc1ccc(CCNC(C(C)OC)=O)cc1 C1(OC)CC(C(=O)NCC2CCCC2N(C)C)N(C(=O)C=Cc2ccco2)C1 N1(C(C(CC=C)NC(C)=O)=O)CCC2CCCC12C(=O)NCC1(F)CC1 c1(COC(c2c(OC)[nH]c(=N)cc2)=O)c(F)ccc(C)c1Cl C(c1cnc2ccccc2n1)=CC(=O)NN1CC(CBr)C1.c1(C(=O)OC)ccc(F)cc1 c1(C(C(=O)NCCCC2CCCN2C(=O)CCc2cn[nH]c2)O)cccc(Cl)c1 N1(C(c2ccc(P(C)(C)=O)cc2)=O)CC2(C1)CN(C(=O)C(Cl)=CCl)CC2C(=O)O N1(C(C2CCN(CCC)CC2)=O)CC2(CC2)CC1CNC(=O)C(C)CC(F)F Cc1cc(C(=O)NCCC(O)C(=O)N(C(C)CO)C)nc(O)c1 C1(NC(c2cc(OCC)ns2)=O)CCN(C(=O)CCCOC(C)C)CC1OC CC(C)(C)C#CC(=O)N1CCC1CNC(=O)CC(=O)c1cc(Br)cs1 C1(NC(Cc2cc(C)c(CO)cc2)=O)CCC(O)CN(C(=O)C(C)N(C)C)C1 C1(NC(CCN(CC=C)C(c2cnc(O)c(C)c2)=O)=O)CNC(=O)C1(C)C N1(C(c2c(C)cn(C)c2)=O)CCOCC(CNC(=O)CC2C=CS(=O)(=O)C2)C1 N1(C(Cn2ncc(C)c2)=O)CC2COCC2(C(=O)N(C(C)CCO)C)C1 CCC(C)CCCC(=O)NCC1CC1NC(=O)COCCc1ccccc1 C(=O)(CC(C)CC(C)C)N1C(CC(=O)NC2CCC(C(C)=O)CC2)COCC1 c1(OC)cccc2cccc(C(=O)N(C3CN(C(=O)CC4OCCO4)C3)C)c12 Nc1cc(C(F)(F)F)ccc1C(N1CCC(NC(c2csnc2Cl)=O)CC1)=O c1(C(=O)NCCCCNC(C(C2CCCOC2)OCC)=O)ccc(O)c(N)n1 c1(C(=O)NCCCNC(Cc2ccc(OC(C)C)cc2)=O)cccc2nsnc12 C1(NC(c2c(N)cn(C)n2)=O)CN(C(=O)CCCN=[N+]=[N-])C2(CCCC2)C1 N1(C(C2CCOC2)=O)CCC2(CCCN(CCC3CC3(Cl)Cl)C2)C1 C1(C2CCC2)(C(=O)OC)CCN(C(=O)C(=O)NC2CCC(N)CC2)C1 C1(NCC2CC(C(=O)OC(C)(C)C)C2)CCC(C#N)C1 c1(-c2cn(CCNC(C3(C)CCCO3)=O)nn2)ccc(C2CC2)cc1 C1(C(=O)NC2(c3ccc(C)cc3)CC2)CCCN(Cc2ccc(C#N)nc2)CC1 Cc1ccc(C(=O)NC2CN(C(=O)CS(=O)(=O)N(C)C)CCC2F)cc1Cl CC1(C)CCc2c1n[nH]c2C(=O)NC1CC(NC(C2COC3(CCC3)C2)=O)C1 N1(C(C)C(=O)Nc2cnn(C)c2)CC2(COC(C)(C)OC2)C1 C1(C(=O)N(c2ccc(F)cc2)CC(F)F)NCCC12CCC(F)(F)CC2 C1(C2CCN(Cc3ccnc4ncnn34)CC2)(NC(C(CSC)C)=O)CC1 C1(N(C)C(C2CCSCC2)=O)CC2CCC(C1)N2C(=O)C(C)(C)CC1CC1 N1(C(Cc2n3cc(C)nc3sc2)=O)CCOC2CN(C(c3cnc[nH]3)=O)CC12 CN1CC(O)(CN(C)C(C2(NC(=O)COC3CCC3)CCCC2)=O)C1 CCCC(O)C(=O)NC1CC(NC(c2cccc(C)n2)=O)C(O)C1 N1(C(c2c(C)c(Cl)ccn2)C(=O)NCC2CC2)CC2CCCCC2C1C C1(NC(c2cn(CC)nc2)=O)CCN(C(=O)C2=CC(O)CCC2)CC(O)C1 N1(C(C(C=C)O)=O)CC(CC(=O)Nc2cccc(OCC)c2)C(C)C1 Cc1cc(C)c(C(=O)NCC2CC(NC(=O)CCS(N)(=O)=O)C23CCC3)c(O)n1 C1(NC(CCCOCCC)=O)CC(N=c2cc[nH]c(OC(C)=O)n2)C1(C)C CCCCC(=O)NC1CCCC1CN(C(=O)CCc1cncs1)C CN1CC(C)(C(N2CCCC(O)(CN(C(=O)CCC3CCC3)C)C2)=O)CCC1=O CCCC(C)CCCC(=O)NCC1(NC(=O)Cn2nc(C(F)F)cc2C)CCC1 N1(C(C2CCN(C(CC)=O)C2)=O)CC2(C)CN(C(=O)C#CC(C)C)CC2(C)C1 N1(CC2CN(C(C3(C)CCCO3)=O)C2)CCN(C(c2ccc(C(F)F)o2)=O)CC1 Cc1nn(C)c(C)c1CC(C)C(=O)NC(C)CN(C)C(C12CC(C)(C1)OC2C)=O C1(NC(=O)Cn2cc(Cl)cn2)COC2(CCN(C(c3cc(O)nc(O)n3)=O)C2)C1 Cc1sc(C(c2nnnn2CC(F)F)NCc2nc(C(C)(C)C)cs2)c(Br)c1C C(N=c1[nH]c(=NCC23CCCCC2C3)[nH]c2ccsc12)c1cccc(C)n1 C1(C(=O)NCCCC=C)CN(C(=O)CCc2csnn2)CC(C)O1 C(c1cocn1)=CC(N1CC(CC(C(=O)N2CC(CC(C)(C)C)C2)F)C1)=O C12(CNC(c3cnn(C)c3Cl)=O)CCCC1CN(C(C13CCC(CC1F)C3)=O)C2 N1(C(=O)Nc2ccnc(C3(C)NC(=O)NC3=O)c2F)CC2CCCC(=O)NC2C1 N1(C(N2CC3CC3(Nc3ccncn3)C2)=O)CC2CCCCC12 C12(CNC(c3cn(C)nc3Cl)=O)CCCC1CCC2 C1(CC(=O)NCC(C)(C(C)C)NC(c2c[nH]nc2F)=O)(CC)CCOCC1 Cc1cccc(Br)c1-n1cc(C(CC(N)=O)C(N2CCN(C)C(C)C2)=O)nn1 c1(C(=O)NCC(CO)NC(C(C(C)(C)C)CO)=O)cncc2c1CCNC2=O N1(C(CC(CCC)C)=O)CC(CNC(=O)CCNc2ncccn2)CC12CCC2 c1(OC)cccc(-c2nc(C3CCC=CCC3)n(-c3nc(Br)nn3C)n2)n1 C(=O)(C1CCSc2ccccc21)NCC1(C)CCN(C(C2(O)CCOCC2)=O)C1 N(C1CCCc2ccoc21)C(C(CCCNC(c1cc(CC)no1)=O)O)=O S(=O)(=O)(c1ccc(N2CCCC(c3ccno3)C2)c(Cl)c1)NCC=C Cc1c(C(N2CCC(NC(=O)CCc3ccoc3)CC2C)=O)cc(O)cc1N C(=O)(C1CCCc2c[nH]nc21)N1CC(N2C(c3ccccc3)C3NC(=O)C32)C1 C1(NC(C2CC23CCSCC3)=O)CCCN(C(c2c(F)cccc2Cl)=O)CC1 N1(c2nc(C)nc(Cl)c2)CC(C)CN(C(C2CC(F)(F)C2)=O)CC1C C(=O)(CC(C)CC(C)(C)C)NCCCCCCC(=O)N(C)Cc1snc(C)n1 c1(CC)nnsc1C(=O)NC(C)(C)C(=O)NC1CC(CCC(=O)OC)C1 c1(C(C)NC(=O)Nc2ccc(NC(=O)OC)cc2)cc(F)ccc1F C(CC(C(C)C)NC(c1n[nH]c(CC)n1)=O)N(C(C(C=C)c1ccccc1)=O)C C1(NC(C(C)NS(CC)(=O)=O)=O)CC2C1CCN2C(=O)CC1CC(F)(F)C1 Cc1c(C(=O)NC2CN(C(c3c(F)ccnc3Cl)=O)CCC2F)cccc1O N1(CC(=O)NC2CC(C)(NC(C3CC(C)(O)C3)=O)C2)CCC(CO)CC1 c1(CC(=O)N(C(C)CNC(c2ccc(C)cc2C)=O)CC)ccc(O)c(Cl)c1 c1(C(=O)NCCCN(CCCCNC(c2cn(CC)nn2)=O)C)[nH]cnc1C#N Cc1n[nH]c(C)c1CN1CC(CNC(=O)C=Cc2cc(C(=O)O)co2)C1 c1(SCC(=O)NC(CC(C)NC(C2(C(C)C)COC2)=O)C)ccc(F)cc1 c1(COC(=O)CSc2ccc(Cl)cc2)cc2c(C(F)(F)F)cc(O)nc2o1 C(=O)(C1CCCc2c[nH]nc21)N(C1C(NC(c2n[nH]c(C)c2F)=O)CCCC1)C CC1(C)OCCC1(O)C(=O)NCC1(C(N2CCC3(CCO3)C2)=O)CC1 N1(C(CCC=CC)=O)CCC(C)(C)C1C(N1CCSC(C)C1C)=O C1(NC(C(C)CC2CC2)=O)CCCN(C(=O)CSc2cccc(Cl)c2)CC1 N1(C(CC2C(C)=NOC2=O)=O)CCC2CN(C(=O)C(C)(C)C3CC3)CC2C1 C(=O)(CC(C)(C)C(F)F)N1CC(CC(C)(C)C)N(C(=O)C(=O)NCC(F)F)CC1 C1(C(=O)N(C)CC2(C)CCCO2)(COC)C=CCN1C(C1CC(OC)C1)=O c1(C(=O)NC(CCOCC)C(=O)NCCc2c(C)noc2C)nnc(O)nc1O CC1CCCCC1(CNC(=O)CCc1nc(=N)[nH][nH]1)NC(c1ccc(F)cn1)=O c1(CC)ccc(C(=O)NCC(CNC(=O)C(C)Sc2ccc(C)cc2)CO)cn1 N1(C(C=CCC2(NC(C3CC(=C)C3)=O)CCC2)=O)CCC(C(C)CC)CC1 C(=O)(C1(C)CCCc2ccccc21)NCCCCC(C)NC(C1C(C)=C1)=O C=CCC(CC)C(=O)NCCC1(C(N2CCCC(F)CC2)=O)CC1 S(=O)(=O)(c1ccc(CC(=O)N(C2CN(C(C3(C)CCCC3)=O)C2)C)s1)NC C1(C(=O)NC(C2CCCCC2)(C)C)CC2CN(C(=O)Cn3cnc(C#N)n3)CC2C1 C1(CC(=O)NCC(C(C)C)NC(=O)CS(C)(=O)=O)CSc2ccccc2NC1=O C1(CNC(c2ccc(C(=O)OC)[nH]2)=O)CC(NC(C2CCOCC2)=O)C12CCC2 Cc1ccc(C(N2CCCN(C(=O)CCC3CC3C)CCC2)=O)c(N)c1C C1(NC(C(C)NC=O)=O)CN(C(c2ccc(Cl)cc2N)=O)CC12CCC2 N1(C(COC(C)=O)=O)CCOC2(CCN(C(c3cc(Br)c(C)c(Br)c3)=O)CC2)C1 Cc1csc(C=CC(=O)NCCCN(C(=O)CC(C)NC(N)=O)CC)n1.C(C)(C)(C)O N1(C(c2c(CC)scc2)=O)CCCCC1CNC(c1scc(C)c1OC)=O c1(OC)nc(N(C2CCC(N)C2)C(C2CC(O)C2)=O)ncc1Br C1(C(F)(F)F)(C(=O)NCCN(C)Cc2cn(CCC(C)(C)C)nn2)CCCCO1 C(=O)(C(C)CC(N)=O)NC(CN1CCN(C(C(C(C)OC)N(C)C)=O)CC1)C C1(C)(C(N2CC(C)(CSC)C2)=O)CCN(C)CC1 Cc1ccc(C)c(CN2CC(F)(C(=O)Nc3cc(Br)ccc3N3CCCC3)C2)c1 C1(OC)CCCCC1C(=O)N(CC(C)CNC(c1cc(C)n(C)c1)=O)C CC1(C)CCN(C(=O)CC2CC2(Cl)Cl)C1C(=O)NCC1CC2CCC(C1)O2 C1(C)(C(N2CC3C(CNC(CCNC(=O)OC)=O)(C3)C2)=O)CC(C2CC2)=NO1 N1(C(C2(C)CC(=C)C2)=O)CCC(CCNC(=O)C(C)=C(C)C)C(F)(F)C1 c1(C(=O)NCCC2N(C(C3CC(N(C)C)C3)=O)CCC2)cncc2cnccc12 C1(OC)CN(C(=O)CC23CCCC2C3)CC1NC(=O)Cc1ccn(C)n1 C1(C(=O)NC2CN(C(CCc3onc(CC)n3)=O)C(CO)C2)CC12CCOCC2 Cc1cnc(C(=O)NCC2(CC(=O)O)CC2)s1 CCC(CCO)NC(c1ccn(CCNC(=O)CC2CC(F)(F)C2)c1)=O C1(CNC(C(c2ccccc2)OC)=O)CN(C)CCN1C(c1sccc1Cl)=O C1(c2n(CC)nnn2)(Nc2cnn(CCCCO)c2)CCC2CN(C)CC12 c1(C(=O)NC(CC(C)C)CNC(=O)CC2COCC2(C)C)c(F)cccc1Cl Fc1cc(-c2cnc(NCc3cccc(Br)n3)nc2)cc(F)c1F c1(C(=O)NCCC(=C)CNC(C2CC2(C)C)=O)ccc(CC2CCC2)cc1 N1(C(C(C)N(C(C)=O)C)=O)CCn2c(CNC(=O)C3=C(C)CCCC3)nnc2C1 c1(C(=O)NCCCC(C)NC(=O)Cn2nnnc2C2CC2)ccnc(Cl)c1Cl n1(CC(N2C(CNC(C3(C)C=CCCC3)=O)CC2)=O)cc(Br)ccc1=O N1(C(c2ccc(CCC=C)cc2)=O)CC2(COC(CNC(=O)COCCF)C2)C1 CC1CC(=O)N(Cc2ccc(F)c(F)c2)C1=O C1(NC(c2ccc(COC)o2)=O)COC2(CCN(C(c3cccc(CO)n3)=O)C2)C1 C1(NC(C2N(CC)CCC2)=O)CCC12CN(C(=O)COc1cccc(C#N)c1)C2 c1(C(=O)NC(C2CC=CCC2)C(=O)Nc2n(COC)ncc2)ccc(OC)cc1 C(=O)(C(O)CCCCC)N1CCC2C(NC(C3CC(=C)C3)=O)C2C1 c1(C(n2cc(-c3ccc(C4CCNCC4)cc3)nn2)C)cccc(F)n1 C1(S(N)(=O)=O)(C(N(C)CC2(NC(C(CN(CC)CC)F)=O)CC2)=O)CCC1 C1(NC(c2ccc(OC(C)(C)C)cc2)=O)CCC12CN(C(c1ccnnc1)=O)C2 C(C(C)(C)C(=O)NC1CC2(C1)CC2NC(c1[nH]nnc1C1CC1)=O)NC(C)=O C1(NC(=O)OC(C)(C)C)CCC(NC(CF)C(=O)OC(C)CC#N)CC1 c1(COCC=CC(=O)Nc2cncc(F)c2)cccc2ccccc12 N1(CC2CC(OC)C2)CCC(CN(C)CCOC(=O)CCC=CC(C)C)C1 c1(C(=O)NCC(C(=O)OC(CC)CO)C)ccc(OC2CC2)cc1 Cc1ccc(CN(C(c2ccc(F)c(C(F)F)c2)C(=O)NCCCF)C)cc1Cl c1(NC(C2CCN(Cc3cc(OC)cc(F)c3)CC2)=O)ccc2nccn2c1 c1(C(=O)NCC2C(NC(C3(COC)CC(=C)C3)=O)CCC2)c(C)cc(F)cc1C c1(NC2CC(NC(C3CCCS3)=O)C2)ccc(Cl)cc1[N+](=O)[O-] c1(C(N2CCC(C)(NC(C3C(C=C)C3)=O)CC2)=O)cnn2c1NCCC2 C1(CC(=O)NC2COCCC2NC(C2(CO)CCC2)=O)CCCCC12CC2 C1(NC(c2cc(C(F)(F)F)ccc2Br)=O)CS(=O)(=O)C12CCCC2 c1(OC)ccccc1C(C)(C)C(=O)NCC(C)(C1CC1)NC(=O)COC(C)(C)C Cc1cc(C(=O)NCCCC2CCCN2C(c2cocc2Br)=O)oc1C c1(C(=O)NC2CC(CNC(c3c(C)ncc(N)c3)=O)C2)cnn(C)c1S(C)(=O)=O Cc1cccc2[nH]c(=NC(C)CC(C)NC(c3oc4ccccc4c3Cl)=O)sc12 C#CCC(C)(CNC(=O)C(C)(C1CC1)N(C)C(C1CCC(=O)N(C)C1)=O)CO CC(CCC(=O)NCCC1CC(F)(F)C1)NC(C1(C)CC1(C)C)=O n1(CC(N2CCC(C)(c3cn(C4CCCC4)nn3)C2)=O)cc([N+](=O)[O-])cn1 C(=O)(C(CN(C)C)NC(=O)CCc1nncs1)NC(COC)(C)C1CC1 c1(CCCCC(=O)NCCC2CCN(C(=O)C=CBr)C2)ccc(F)c(F)c1 C#Cc1ccc(C(N2CC(CC)OC(CC)C2)=O)c(F)c1Cl c1(OC)ncc(Cl)c(C)c1C(=O)NCC1CN(C(=O)C(C)C2CC2)CCC1(F)F C=C1CCC(C(=O)NC2C=CCN(C(c3cc(C(F)(F)F)ns3)=O)C2)CC1 C(=O)(C(C)(C)C(=O)NCc1ccc(C(=O)NCc2ccco2)nc1)NC c1(CN2CCC(N(C(C(C3CCC(=O)N3)C)=O)C)CC2)ccc(F)c(F)c1 C12(C(N(CC(C)CNC(C3CC(C)N(C)C3)=O)C)=O)C3C4C1C1C2C3C41C c1(C(N2CC(NC(COCC)=O)CC3(C2)CC3)=O)ccc2nccnc2n1 C(CCCCC(=O)NCCN1CCN(C(c2cnn(CC3CC3)c2)=O)CC1)OC N1(C(CC(C)OC)=O)CC2CCC(C1)N2C(c1cc(Br)oc1C)=O c1(CCC(N2CCC(C(C)NC(C3CC(C(N)=O)C3)=O)C2)=O)ccc(O)nn1 C(=O)(C(C)(C)S(=O)(=O)c1ccccc1)NCCC(CNC(C1C(C=C)CC1)=O)O c1(CNCC2N(C(C(C(C)C)NC(C)=O)=O)CCCC2)ccc2ncnn2c1 C1(C(N(C)CC2(NC(C3CC3Cl)=O)CC2)=O)C=CC=CC=C1 c1(C(=O)NC(C2(O)CN(C(=O)Cn3cccn3)C2)C)cc2cc[nH]c(=O)c2s1 CC1(C)CC(=O)NCC1C(N1CC(OCCNC(=O)CC2CCCC2(F)F)C1)=O C(=O)(C(CC)CC(C)C)NCC1(NC(C(C)SCCCC)=O)CC1 C1(C(=O)NCC2CCN(C(=O)C=Cc3cccnc3)C2)CC2(COCCO2)C1 c1(C(C(=O)N(CC(CNC(c2ccn(C(C)C)n2)=O)C)C)C)nc(F)ccc1Cl CCC(F)(F)C(C)(C)NC(C1CN(C(C2CCCC(=O)CC2)=O)CC(C)O1)=O Cc1cc(Cl)cc(C(N2CC(CCNC(C3(C4CC4)CC3)=O)C2)=O)c1C C(N=c1ccnc(NC(C)C(C)C(c2ccccc2)OC)[nH]1)c1c(C)n(C)nc1 Cc1cc(C(=O)NCC(O)CCNC(c2cnc(C3OCCO3)s2)=O)ncc1F c1(OC)ccncc1CC(=O)NC1CCC(CNC(=O)COC(F)F)CC1 N1(C(c2occ(C)c2)=O)CCN(C(=O)Cn2cccc2)CC1c1nccn1C C1CC(O)C(=O)N1.C1(CNC(C2CC(C(C)NC(=O)C3CC3)C2)=O)C(C)C1(F)F C(=O)(C(CC(C)C)C(C)C)N(CC(CNC(C=C(CCOC)Cl)=O)C)C Cc1cccc(C(=O)NC2CCN(C(C3(c4cccs4)CC3)=O)CC2CO)c1C c1(C(N2C(C)CCC(NC(c3cncn(C)c3=O)=O)C2)=O)cc(O)cc(C#N)c1 N1(C(c2c(C#N)nc[nH]2)=O)CCCN(C(=O)CCN2CCCC2)CCC1 Cc1nc(C)n(CCC(=O)NC(C)(CNC(=O)Cc2ccsc2Cl)C2CCC2)n1 C1(CNC(C=CCOC)=O)(NC(C2CC3CC(OC)C3C2)=O)CCC(F)(F)CC1 N1(C(COCC(=C)C)=O)CCC2CCN(C(=O)C(C(C)C)n3cnnn3)CC12 C(=O)(C#CC1(C)COC1)NC12CC(C(=O)NCC(C3CCCC3)C)(C1)C2 C(CNC(=O)C1=CCCC1)(CC(F)(F)F)NC(=O)C(O)C(F)F C1(CCC(N2CCC(NC(C3CC(CN(C)C)C3)=O)C2)=O)CCCCCC1 CC1(CNC(C2CC2Cc2ccccc2)=O)CCCN(C(=O)C2=COCCC2)C1 CCCC(C#N)C(=O)NC(C)(C)CCNC(C1CCC(C(F)(F)F)CC1)=O c1(C(C)C)ncc(C(N2CCCC(N(C)C(C3C4CCC3CC4)=O)C2)=O)n1C N1(C(COc2ccc(C(C)(C)C)cc2)=O)CCCC(C2CCCC2)C1 N1(C(c2cccc(Br)c2O)=O)CC2CCC1C(O)C2 CN1CCN(CCC(=O)N(CCNC(=O)C(C2CCCCCC2)F)C2CC2)CC1 Cc1ccc(CN)c(OCC(F)(F)F)c1.C(C)(C)(CN(C)C)OC C12(C(N3CCC(C(C)C)(CO)C3)=O)CC(C)(CN1C(=O)CC1CCCOCC1)C2 c1(C(=O)NCCC2(NC(=O)CN3CCCCC3)CC2)ccc(C(=O)NC)c(Cl)c1 N1(C(C(C(C)C)C)=O)CC2(CCCC(CNC(C3CN4CCC3CC4)=O)O2)C1 C1(C(N2CCCC(NC(C(C)CCO)=O)(CO)C2)=O)CCCC(F)(F)CC1 C1(C(N2CCC(C(C(=O)NC3(CC(C)C)CC3)F)C2)=O)CN(C)CCO1 C(=O)(C(C)(O)C(C)(C)C)NCC(C)(C)OC.C1=CCOCCNC1=O C1(CC)CN(C(c2cnco2)=O)CCC1NC(c1ccc(SC(F)F)cc1)=O C(CSC)(C(=O)NCCC(C)C)OC.C1C(C)=CC(=O)N1C1CCC1 C(CCCCC(=O)NC1(C(=O)N(CCC(C)O)C)CC1)=CC Cc1nn(C)c2sc(C(=O)NCC3CN(CC(=O)NC4CC4)CCC3(C)C)cc12 C12(NC(=O)CCCF)CCCC1CN(C(c1cccc3nn[nH]c13)=O)C2 c1(C(=O)NC2CC(C)(NC(=O)CSc3cccs3)C2)cccc(C(N)=O)n1 C1(NC(COCCC=C)=O)CCCN(C(c2cc(N)ccc2O)=O)CC1 N1(CC)CCC(C)(c2nncn2C)CC1.C12CC(C1(C)C)NC(=O)NC(=O)C2 C(=O)(CCCS(C)(=O)=O)NCC(C)(CO)NC(c1cc(C(C)=O)c(C)nc1)=O Cc1ccc(C(=O)NC2(C(N3CCCOCC3)=O)CC(F)C2)nc1O c1(OC)cccc(CCC(=O)N(C)CCNC(c2cc(OC)nn2C)=O)n1 c1(C(N2C3C(NC(c4c(Cl)cn(CC)n4)=O)CC(C3)C2)=O)c(C)nc(O)nc1C C1(C)(CNC(C2CCCN(C)C2)=O)CCC(NC(=O)CC2CCCC2)CC1 C1(C(N2CC(OCCNC(C(n3c(C)ccn3)C)=O)C2)=O)CNC(=O)CC1C c1(CC(N2CC(NC(CN(C)CCO)=O)C3C2C3)=O)ccc2nc[nH]c2c1 N1(Cc2cc(CC(C)C)no2)CCC2(CCN(C(=O)Cn3ccnn3)CC2)CC1 CCCC(C)(C)CC(=O)N1CCC(CCOC)(NC(C2CCOC2C2CC2)=O)C1 c1(C(=O)NCC(CNC(c2cccc(C(N)=O)c2N)=O)O)cc(F)c(F)c(F)c1 c1(C(=O)NCC2C(C(N(C)CC3(C)CCCO3)=O)CC2)cccc(=O)o1 Cc1nc(C)c(C(=O)NC2(CCNC(c3ccc(C(F)(F)F)o3)=O)CC2)o1 c1(C(C)C)nc(N2CCC(NC(c3ccc(Cl)nc3Cl)=O)C2C)cc(Cl)n1 c1(C(N2CCC(F)(C(N3CCC(N(C)C)C3)=O)C2)=O)cc([N+](=O)[O-])cs1 C(=O)(C(C)=NOCC#N)OCC(CC#C)OC1CCN(C(C)=O)CC1 C1(C(N2C(CNC(C3CC(n4ccnn4)C3)=O)CC2)=O)NC(=O)C2CC12 N1(C(CC(=O)OCC)=O)C(CC(=O)NCC2C(CO)C2(C)C)C2CCCC12 CC(C)CCCCCNC(C1CCCCN(C(c2ccoc2)=O)C1)=O CCCC(C)(CC)C(=O)N1CC(C)(CCC(=O)NC(C)CCC(C)(C)C)C1 Cc1cccc(-c2nnc(N(C)Cc3ccns3)n2CC2CC2)n1 N1(C(COCC)=O)CCOC2(CCN(C(C3CC3C)=O)C2)C1 C1(NC(c2nc(C3CC3)cs2)=O)CN(C(=O)Cn2nnc(=O)[nH]2)CC12CC2 C(C)(C)(CCCNC(=O)CSCc1cccc(Cl)c1)NC(C1C(C)(C(C)C)C1)=O C(=O)(CC(C)=C=C)NCCOC(CNC(C(C)OCC#C)=O)(C)C c1(SCc2n(C(CC)C)ncc2)cccn1C(=O)OC(C)(C)C CC(=O)CCC(=O)N1CC(OCCC(=O)NCC2(CO)CCC2)C1 C(CCC(C)C)CCNC.N1(C(=O)NCCOC)CC(C2CCCO2)C1 C(=O)(C(C)CC(C)(C)C)NC(C(=O)NC(c1scc(C)n1)C)C(C)O Cc1c(Cl)ccnc1C(N1CCC(NC(C2(C)CC3(CCC3)C2)=O)C(CO)C1)=O C1(NC(C=C(C)Cl)=O)CCOC12CCN(C(C1CC3CCCC(C1)C3=O)=O)CC2 C1(NC(c2[nH]nc(OC)c2Cl)=O)CC2CN(C(=O)C(C)Oc3ccccc3)CC12 Cc1cc(=NC2CCC(NC(c3cncs3)=O)CC2)[nH]c(C(C)(C)C)n1 C12(CNC(C(N3CCSCC3)C)=O)CC(CO1)N(C(c1cc(O)cc(=O)o1)=O)C2 C=CC1(O)CN(C(C2CCCC2NC(=O)C(O)CSC)=O)C1 CC(C)(C(=O)N1CC2CCC(C1)N2C(=O)CCCC(=O)c1ccccc1)C(F)(F)F c1(C(N2CCOC2=O)C(N2CCC(N(C(=O)C(N)=O)C)C2)=O)cccc(Br)c1 CN(C)NC(=O)CCC(=O)N1CCCN(C(C2CCCN2C=O)=O)CC1 c1(C(N(C(CC(N)=O)C2CC2)C(CC)CC)=O)ccc(CO)o1 CC(C)C(O)C(=O)NC(C)CCCNC(=O)OC(C)(C)C C1(C(C(=O)NCCCOCCC(=O)NC(C2CCCC2)CC)O)CCCCC1 C1(N(C)CC)CCN(C(C2C(CNC(=O)C(O)C3CC3)C2(C)C)=O)C1 N1(C(C(CC)SC)=O)CCCC(NC(c2occc2F)=O)C1 Cn1nc(Br)cc1C(=O)NCC(O)CNC(=O)CCC1OCCO1 Cc1cn2cccc(C(N3CCC(C)(CNC(C4C5COCC45)=O)C3)=O)c2n1 c1(C(N2CCC(CCNC(COCC(=O)OC)=O)C2)=O)cc2nnn(C)c2s1 C1(NC(C(CCNC(CCSCC)=O)(C)C)=O)CC2CC1CC21CC1 c1(C(N(CCC2CCN(C(C(CC=C)C)=O)CC2)C)=O)nc(O)[nH]c(=O)n1 c1(C2C(C(=O)NC3CC(N(C(CNC(CN(C)C)=O)=O)C)C3)C2)nccn1C Cc1cnsc1C(=O)NCC1(C(=O)NC(C)CC2CC2)CCC1 CC1CCNCCC1N(CCSc1cccc(O)c1)C(=O)OC(C)(C)C C#Cc1cncc(C(=O)N(CC(O)CN(C)C(c2c[nH]c(Br)c2)=O)C)c1 C(=O)(CC(CNC(C1CCCCC1O)=O)C1CCC1)NCCCOC(C)C C1(NC(c2cc(C)nc(C)c2)=O)CCSC12CN(C(C1(O)CCCCC1)=O)C2 C(=O)(CCC(=O)c1cc(Br)cs1)N1CC(NC(C=CCCC)=O)C1 c1(C(N2C(CC)C(NC(c3cnn(C(F)F)c3)=O)CC2)=O)ccc(Cl)cc1F C(C(=O)NCCNC(C1CCCSC1)=O)(c1ccccc1)=CC(C)(C)C c1(-c2cnc(OC)nc2)cncc2sc(C(=O)NCC(F)(F)F)cc12 C1(C(N2CC(OCC#C)C2)=O)CC12CCN(C(C13CCCC1C3(F)F)=O)CC2 C1(NC(COCC#C)=O)CC2C(NC(c3coc(C(=O)OC)n3)=O)C2C1 CC1C2C(CCN2C(c2ccc[nH]2)=O)CN1C(c1ccc(O)nn1)=O C1(CC)C(C(=O)N(CCC(=O)NC)CC)CCCN1C(c1cnn2c1CCC2)=O c1(OC)cccc(O)c1C(=O)NC(c1ccccc1)CSCCS(C)(=O)=O C12(C(=O)NCC#CC(=O)NC(C=C)C3CC3)C(=O)C3CC1C2C3 C1(CNC(=O)C=C2CCCC2)CN(C(c2cncc(CO)c2)=O)C2CC12 CCC(CC)C(=O)NC(C1CCCCC1)CNC(C1CC(O)CN1C(C)=O)=O c1(C(=O)NC2CCN(C(C3N(CC)CC3)=O)CC2C)cnn2c1CCCN2 c1(C(=O)NCC(=C)CCNC(C2CC2(C(C)C)CC)=O)oc(C)nc1C c1(OC)cnc(Cl)nc1N1CC(=C(F)CNC(=O)C(C)OCC2CCCO2)C1 O=C(CC(C(F)F)c1ccccc1)NCC1CC(NC(=O)NC23CC(O)C2C3)C1 C(C(C)(C)CC(=O)NC1(CCO)CCCC1)NC(C(SC)SC)=O c1(C(=O)NC(C2CN(C(C(C)OCCCC)=O)C2)C)coc(C2CCCC2)n1 c1(CCN(C)CCNC(=O)CCCc2ncco2)nc(Cn2cc(Cl)cn2)cs1 C1(NC(c2ccc(C(F)F)cc2)=O)C2COCC1CN(C(c1ncccn1)=O)C2 NC1CCC=CCNS(=O)(=O)c2ccc(Cl)c(c2)C(=O)N2CC3(CC3)CC2C(C)NC1=O c1(C(N(C(CNC(C(C2CC(F)(F)C2)OC)=O)C2CC2)C)=O)coc(C(N)=O)c1 N1(C(C(CCCCC)O)=O)CC(CNC(C2(CN(C)C)CC2)=O)OC2(CCC2)C1 c1(-n2cnc(NC(C3n4cc3cn4)=O)n2)ncccc1F.c1(SCC)ccoc1 N1(C(C)=O)CCCC(C(=O)N(c2cc(F)n[nH]2)C(c2ccc(=N)[nH]c2)=O)C1 C1(COCC)CN(C(=O)OC(C)(C)C)CC1CC(=O)N(C)OCc1ccccc1 CCCC(C(O)C(=O)NC(CC)C(F)(F)F)NC(=O)COC(C)C C1CC2c3ccccc3CCN2C(=O)C(=O)NCCO1.C(C)(C(=O)ON)NC(C)=O N1(c2nc(C#N)c(Cl)s2)CCC2(COC(CNC(=O)C=CCF)C2)C1 N1(C(CCNC(COC)=O)=O)CCCN(C(C2CC3CCC3C2)=O)CCC1 N1(c2ncc(C#C)cn2)CCC2(CCCCC2NC(=O)CC2C=CS(=O)(=O)C2)C1 c1(CCC(=O)N(CCN2CCN(C(=O)COC(F)F)CC2)CO)cccnc1Cl C(=O)(C1=CC2CCCC12)NCC1CCCN(C(c2c(CC)occ2)=O)CC1 C(CC(C)C)(C(=O)NCC(C)CN(C(=O)CCn1ccnn1)C)NC(C)=O c1(CC)ccc(C(=O)NC(C)(CNC(c2cc(CSC)[nH]n2)=O)C(C)C)c(C)c1 CCCCCC(C)CC(=O)NCC1(C(=O)NC(c2nc[nH]n2)CC)CCC1 c1(N(CC(F)(F)F)C)ccc(C2CCCN2C(=O)C(C)(C)c2ccno2)nn1 N1(C(C)(C)C)CCC(N2CCSCC2CCNC(C2C=CCC2)=O)C1=O C1(C(=O)NCC2(NC(Cc3n(C)ncc3Br)=O)CC2)COCCC1(F)F c1(CN(C(c2ccc(-n3cc(CO)nn3)cc2)=O)CCO)ncccc1Cl C1(NC(c2nc(CC)oc2C)=O)C2CCN(C(c3cc(C(C)C)n(C)n3)=O)CC12 N1(C(CNC(c2ccoc2)=O)=O)CC(O)C(O)C1CNC(C1CCC=CCC1)=O CC1(C)CCN(C(C2CCC2)=O)CC1NC(=O)C=CCN1CCCC1 CC(C)(C)C1=NOC(C(=O)NC2CCN(C(C3(F)CC3)=O)CC(O)C2)C1 c1(CC)cccc(C)c1-n1nc(-c2cnn(C)c2)nc1Cn1ccccc1=O CC(C)CC(C)CC(=O)NC1CCN(C(c2nocc2Br)=O)C1C(C)C c1(CC)c(C(=O)NC(CNC(=O)CCn2cnnn2)C(C)C)nnn1C Cc1nc2ccc(C(N3CCN(C)CC3CNC(=O)C(F)(F)C(F)F)=O)cc2s1 c1(NC2CC3CN(Cc4ccn(CC)n4)CC3C2)ncnc2c1ccn2C c1(OC)ccc2c(c1)CC(C(=O)NC1CCCC1CNC(=O)Cc1cncs1)O2 C(=O)C(O)C(C)(C)C.C(=O)(C(CCSC)NCC1(CO)C2CCC12)OCC CCC(O)(CC(=O)NCC1(CNC(=O)CP(C)(C)=O)CCC1)c1ccccc1 C1(CNC(C=CC)=O)CCCC(NC(c2cccc(-c3ccsc3)c2)=O)C1 C1(C(=O)NCCC2CCN(C(c3n(C)c(S)nn3)=O)C2)CN2CCC1CC2 C1(NC(C(CCCC)C)=O)CCC2CC1CN2C(C1SC2C=CC1CC2)=O Cc1cccc(C2(CC3CCN(C(=O)C(c4ccccn4)N)C3)CC2)c1 CCC(=O)CCC(=O)NC1CC2(C1)CC2C(=O)N(CCCO)C CC1(C)CCN(C(=O)C2=COCCO2)CC1NC(c1ncc(C(F)F)s1)=O Cc1nn(CCO)c(C)c1C(=O)NC(C1CCN(C(=O)CCCCC#N)CC1)C C1(CC(=O)Nc2c(C)noc2C)CC2(C1)CN(C(=O)CC1CCC(=O)NC1)C2 C=CCC(CC)C(=O)NCC1CCCCN1C(c1cccc(OC2CC2)c1)=O CC(C(O)C(F)F)NC(C1(NC(=O)CC2CCCNC2=O)CC(O)C1)=O c1(C(=O)NC(C(=O)NCc2ncn(C)n2)c2ccco2)cccn2ccnc12 Cc1ccc2c(=O)c(C(N3CCC(C4CCCN4)C3)=O)cn(C)c2n1 C12(CNC(c3cncc(-c4c(F)ccc(CC(=O)O)c4)c3)=O)CCCC1CC(=O)N2 N1(C(C=C(COC)C)=O)CC(CNC(c2c(C)ccn2C)=O)OC2(CCC2)C1 c1(OC)ccc(CN2CCC(c3ccccc3)CC2C)c2ccccc12 CCC(CC)(CO)C(=O)NC1CC2(C1)CC2NC(=O)C(C)NC(=O)C(C)(C)C C1(NC(c2cnc(SC)s2)=O)CCSC12CN(C(c1ccc([N+](=O)[O-])o1)=O)C2 N1(C(C(C)CN(C(=O)C2=CCSC2)C)=O)CC(=O)NC(=O)C1 c1(N2C3CC(NC(C4=C(C)OCC4)=O)CC2CC3)ncc2c(ncn2C)n1 C1(NC(C2CC(C(F)(F)F)CO2)=O)CC2CCC(C1)N2Cc1nc(Cl)ccc1Cl C(C)(CCCNC(c1coc(C2CC2)n1)=O)NC(C1CN(C(C)=O)C1)=O N1(CC)C(=O)CCC1CC(=O)N(C1CCN(C(=O)C=CSCc2ccco2)C1)C C=CCCCCCC(=O)NCCCN(C(=O)CN1CCC(F)(F)C1)C(C)C c1(C(N2CCC(C(C(N3CC(CC#C)OCC3)=O)C)CC2)=O)cncn(C)c1=O O(NC(=O)CC(C)CNC(c1cc(C#N)ccc1C)=O)C(CC)CC c1(C(N2C(CC(=O)N(CCCCC=C)C)CCC2)=O)cc(C(F)(F)F)nn1C Cc1oc(-c2ccsc2)nc1CC(N1CC(NC(=O)OC(C)(C)C)CC1C)=O c1(CC)ccc(C=CC(=O)NCC2(C)CCCN2C(=O)CCSCC(C)C)cc1 c1(C(N2CCCCC(NC(C3OCC(C)C3)=O)C2)=O)cnc2ccccn12 N1(C(C(CC(C)C)ONC(C2CCOC2C2CC2)=O)=O)C2CCCC1COC2 C1(C(=O)NCC(C)(C)NC(c2ccc(SC3CC3)cc2)=O)CC12CCSCC2 C1(C(=O)NC(C(=O)N2CC(OCC(F)F)C2)C2(O)CCC2)CCCOCC1 C(=O)(C(C(C)O)NC(C1CCCC1CNC(c1cc(=O)cc[nH]1)=O)=O)OC c1(CC)nc(N2CCCC(CNC(c3cc(O)n(CC)n3)=O)C2)c(C)c(Cl)n1 CC1=C(C)CC(C(=O)N(C(C)CCNC(=O)Cc2ccsc2C)C)CC1 C(CCC)(C(O)C(=O)NCC(=O)NCCn1cccn1)NC(C(CCC)O)=O Cc1nccnc1C(=O)NCC(C(C)(C)C)NC(c1cc(Br)no1)=O C(C(CC(=O)NC(c1cccnc1)C)OC)NC(CSCC#C)=O C=C(C)CC(C(=O)N(C)CCOCCCO)NC(c1ccns1)=O C1(C2CC2)(NC(=O)C=C2CCCC2)CCN(C(C2CCCC(=O)N2)=O)C1 c1(C(=O)NCC(C2CCOC2)NC(c2c(C(C)C)nns2)=O)nccc(Cl)c1F c1(C(=O)NCC=C(C(=O)NC(C=C)C2CCC2)C)ccc(CO)s1 CC(CCC(=O)N1CCC(NC(c2ncn(C)n2)=O)C1C(C)(C)C)N(C)C c1(NC(C2C(NC(CCOC)=O)CCCC2)=O)ccc(C(=O)OC)cc1Br C1(C(=O)NC2CC(Cl)(Cl)C2)CCOC(c2cccc(F)c2)C1 CCCC(C)(CC)C(=O)NC1CC(C)CN(C(C2CCN(C(=O)NC)CC2)=O)C1 C(CCC(=O)NC1CCC1NC(C1(C)CCOC1)=O)OCC C1(CCOC)(NC(=O)C#CC(C)C)CCN(C(C2(C)CCCOC2)=O)CC1 C1(OCC)CCCC1NC(=O)C(Cc1cccnc1)OC(=O)OC C1(NC(C2C(C)OCC2)=O)(CF)CCN(C(=O)CC2COCCOC2)C1 c1(C(=O)NC(C2CCCC2)CNC(=O)C(C2CCOCC2)O)c(F)cccc1Cl C1(C(N(C(C2CCC2)C)CC)=O)CCOC1CNC(=O)CCn1ccnc1C C1(C(=O)NCC(C)NC(CN(CCC#C)C)=O)(CCN(C)C)CCC1 c1(N2C(CNC(C(c3ccc(OCC)cc3)C)=O)CCC2)ccc(C#N)c(C)n1 CC(C)CC(CNC(=O)CC1OCCCO1)NC(=O)COc1ccccc1F c1(CC)nn(C)c(CC(N2CC3C(CNC(=O)C#CC4CC4)C3C2)=O)c1Cl c1(C(=O)NCC(CCNC(=O)C(F)C2CCOC2)OC)cc(O)c(F)cc1N n1(CC)ccnc1CN(C(=O)CN(C(c1ccc(Cl)s1)=O)C1CC1)C c1(OCC)nccc(C(=O)N(CC(C)N(C)C(C2CC(F)(F)C2)=O)C)c1F C1(CC(=O)NCC2CC(O)CN2C(c2cnccn2)=O)NC(=O)CNC1=O c1(C(N2CCC(=CCNC(C3C(C)(Br)C3)=O)CC2)=O)ccc(Cl)nc1N c1(C(=O)NCC(C)(CO)NC(=O)COC2CC2(F)F)cc2c(nn1)CCCC2 C=CCCCCC(=O)NC1CCC(CC(=O)NCc2cc(C(C)C)on2)C1 Cc1c(C(N2CCOC(c3cn(CC(F)(F)F)nn3)C2)=O)cnn1CC(C)(C)O Cc1ccc(C(N2CC(NC(=O)CC(F)F)CC2C)=O)nc1C C12(CNC(C(C)SCCCC)=O)CCC(NC(=O)C(C)(C)C(F)F)(CO1)C2 c1(C(N2CC(C)(CNC(=O)CC3CCC3)OCC2)=O)c(F)cc(C#N)cc1F c1(C(=O)NCCOCCNC(=O)CO)c(Cl)cccc1Br N1(C(c2c(N)csn2)=O)CCn2ncc(CNC(C3(S(N)(=O)=O)CCC3)=O)c2C1 C1(C(=O)NC2(C(=O)NC)CCC2)C=CCN(C(C2CCCOC2)=O)C1 CC(C)(CCC(=O)NCC1(NC(C2CCCS(=O)(=O)C2)=O)CCOC1)[N+](=O)[O-] C1(CNC(=O)CCc2ccncc2)CC2CCC1N2c1ncc(Cl)cn1 c1(C(=O)NCC2CCC(C)CN2C(=O)C(F)=CCCF)c(Cl)oc2ccccc12 CN1CCCC(NC(C2CSCN2C(C2OC3CCC2C3)=O)=O)CC1 C(C(CO)(CO)NC(c1ccsn1)=O)N(C(C(c1ccc(F)cc1)CC)=O)C C1(Nc2scc(C(N(CCCC)CCO)=O)n2)CCCN(C(=O)OC(C)(C)C)C1 c1(N2CCC(O)(C(C)NC(c3c(C)cc(F)s3)=O)C2)cc2nncn2c(C)n1 C1(NC(c2c(CC)nns2)=O)CCCC12CCN(C(=O)CN1CCCC1C)CC2 C(=O)(CCC(=O)N1CCC(C(N2CCCC(OC(C)=O)C2)=O)C1)NC c1(C(N(C(C)CCNC(=O)CC2CNC(=O)C2)C)=O)cc(=O)n2ccccc2n1 c1(C(C(=O)NC2CC(F)(F)C2)N(CCC)Cc2ccc(F)cc2)ccc(C#N)o1 C(=O)(CC(C(C)OC)NC(=O)Cc1ccoc1C)NC(C=C)C c1(CN2C(C(=O)Nc3ccc(F)cc3Br)CCC2)cc(F)c(Br)cc1F c1(C(N2CCCC(C)(CNC(CC(C)OC)=O)C2)=O)ccc2c(c1)OCCC2 Cn1nc2ccccc2c1C(=O)NCC1CC(NC(=O)CN2CC=CC2)CC1O CC1COCC(C(=O)N(CC(C)N(C)C(=O)C2CC2)C)O1.C12CC(C1)CC(=O)N2 Cc1nsc(CNC(=O)C=CC(C)NC(=O)C(C)N2CCCC2)n1 c1(OC)sccc1C(=O)NCC1CC1NC(C1CCN1C1CCCC1)=O C1(CCNC)CN(C(=O)C(O)CNS(C)(=O)=O)CCN1C(=O)O.C(C)(C)(C)OC(C)=O c1(OC)cnnc(C(=O)NCCC2CCN(c3nnc(C(C)C)o3)C2)c1 CC1CN(C(C2CN(C(=O)CC3COCC3O)CC2(C)C)=O)C12CCOCC2 N1(C(CCNC(=O)NC)=O)CCC(C)C(CNC(c2cc(COC)nn2C)=O)C1 CC1CCN(C(c2ccsc2Cl)=O)CCN1c1nc2ccccc2o1 C(=O)(C(C)CC(C)C(C)=O)NC(CC)CCCC(=O)N(CC(F)F)CC1CC1 Cn1nnc2cc(C(=O)NCC34CC3CN(C(=O)OC(C)(C)C)C4)ccc12 n1(CC)cccc(NC(c2conc2CNC(=O)C(=O)C(C)CC)=O)c1=O N1(C(CCSCC(N)=O)=O)CC2CC1CN2C(c1cnc(CC2CC2)nc1O)=O C(C(C(C)(C)C)NC(=O)CNS(C)(=O)=O)NC(C(c1cncc(F)c1)C)=O N1(Cc2n(CC)ncn2)CC=C(CCNC(=O)Cc2ccc3c(c2)CCC3)CC1 c1(C(N2CC(CN(C)C(c3ccc([N+](=O)[O-])[nH]3)=O)OCC2)=O)cc2n(n1)CCC2 N1(C(CC(CC#C)NC(C2CCC(=O)N2C)=O)=O)CC2CN(CC)CC2C1 CC1(C)C(=O)CC1C(=O)NC1CCC(CNC(c2ccncn2)=O)CC1 C1(OC)CCC(CC(=O)NCCN(C(=O)C(C)(F)F)C2CCCCC2)CC1 CN1N=C(C(=O)N2CC(C3CCCCN3S(=O)(=O)c3ccncc3)C2)CCC1=O Cc1cc(N)cnc1C(=O)N(C(CC(C)C)C(=O)N(C1CCC1C)C)C CC1(C)COCC(NCC2=CCN(C(=O)OC(C)(C)C)CC2)C1 C(=O)(CCCCC(C)(C)C)N1CCC(N2CCN(C(CC(=C=C)C)=O)CC2)CC1 C1(CC=C)(C(=O)NCC2CC(=C3CC3)C2)CCCN1C(=O)C(C)OC(C)(C)C C1(C(=O)OC)CCN(C(=O)CC2(OC)CCCCC2)C2CCCCC12 c1(C(=O)NC(CNC(C(CC)c2cccnc2)=O)(C)C)ccc(N)c(SC)c1 c1(N2CCC(COC)(CNC(c3ccc[nH]3)=O)CC2)cc(C#N)ccc1[N+](=O)[O-] N#Cc1cc(C(N2CCCC2CCNC(C23CCCC2(C(N)=O)C3)=O)=O)on1 c1(COC(COC)=O)ccc(CO)c2ccccc12 N1(C(C(CCC)(C)CC)=O)CCC2(C1)CN(C(c1csc(C(C)=O)n1)=O)CCO2 C(C1=CCCN(C(=O)Cc2ncccc2C)C1)NC(CC1C(CC)C1(F)F)=O C1(CNC(CC=C)=O)CN(C(=O)CC2CC23CC3)CC1C(F)(F)F N1(C(CCN(CC)CC)=O)CC(C(=O)NC(C)(CC)CCO)CCC1(C)C CC(C)(CC(=O)NC1CN(C(C2C=CCC2)=O)CC1O)c1cccc(Br)c1 CCC(C)(C#N)C(=O)N1CC=CC(NC(=O)Cc2ccc(F)c(Br)c2)C1 c1(CNCC2CCC(C(C(=O)NC3(C)CCCCC3)O)CC2)cc(O)ccc1O C1(C(=O)NCC23CN(C(CC(CC)(F)F)=O)C(C2)CO3)CC2CCCCN2C1 C(CCCC(=O)NC1CCC1NC1(CC(=O)N(C)CC)CC1)NC(=O)OCC=C n1(CC)nnc2c(N(C3CCN(C(c4ccn(O)c(=O)c4)=O)C3)C)ncnc12 C1(NC(C2C(=C)CC2)=O)(CNC(=O)C(C)(CC)C(N)=O)Cc2ccccc2C1 C(CN=c1[nH]c2c(c(=NCc3nc4c(s3)COCC4)[nH]1)CSC2)=CCOC c1(C(=O)NCC2(O)CCN(C(C3C(=C)CC3)=O)C2)cc(=N)[nH]c(Cl)n1 C12(C(N3CC(O)(CNC(C4CC(N(C)C)C4)=O)C3)=O)CCCC(C1)OC2 c1(CNCC(CC)C2CCC2)nc(C2CCOCC2)no1 c1(C(=O)NCC(CC=C)NC(c2cc(C(C)(C)C)c[nH]2)=O)ccc2ccnn2c1 c1(OC)ccc(C(=O)NCC2(O)CCN(C(C3(C)CCC(=O)C3)=O)C2)c(F)c1Cl N#CC1CN(C(c2ccc3nonc3c2)=O)CCN1C(c1ccc(CO)nc1)=O Cc1cc(Cl)cc(C(=O)NCC(O)CNC(=O)C=Cc2ccoc2)c1N C=Cn1nccc1C(=O)NCC1CCC(NC(c2cccc(C(=O)OC)n2)=O)C1 c1(N2CCC(NC(=O)C(F)=CC3CC3)C(F)C2)ncc2c(n1)CCOC2 C1(N(C(C(COC)O)=O)C)CCC2CN(C(=O)C(C)Oc3cccc(C)c3)CC12 Cc1cc(=NC2CC(CNC(=O)C3=NNC(=O)C3)C2)[nH]c(C(C)C)n1 C(=O)(C(CN=[N+]=[N-])NC(C1OCC2CCCC12)=O)N(C)CC1CCC1 CC(C(=O)N1CCCC1C(C)NC(=O)CN1CCCC1)C(F)(F)C(F)F N1(CC(=O)C(c2csnc2Cl)=O)CC2CC2C1.C(CCNC1CC1)N CC(=O)CCC(=O)NCCCC(=O)NCCC1CCC(=O)N1 CC1COC2(C1)CN(C(=O)COC(C)(C)CNC(C1(CC3CC3)CCC1)=O)C2 c1(C(=O)OCC)no[nH]c1=NC(=O)C1(C)CCN1Cc1sc(Cl)nc1Cl c1(C(N(C)CC2CCN(C(C3CCC(C)O3)=O)CC2)=O)cnc2ccccc2c1 Cc1nc(O)nc(C)c1C(=O)NC(CNC(C1CC(C(C)(C)C)C1)=O)CC(C)C CCCC(C(=O)N(C(CO)C(C)C)C)NC(C1CC(O)C(F)C1)=O CC1CC(NC(c2cnc(F)c(F)c2)=O)CCN1C(c1ccncn1)=O C1(C(=O)NCC2C(C(=O)OC)C2)CCN(C(=O)CCC(C)(C)C)C1(C)C C12(NC(C3C(=C)CC3)=O)CC(C1)N(C(C1CCCCN1C)=O)C2 CCCC(C(=O)N1CC(C)(NC(C2CC(=O)N(C3CCCC3)C2)=O)C1)OC Cc1cc(S(=O)(=O)N2CCCN(C(=O)C(c3cccn3C)=O)CC2)c(F)cc1Cl N1(C(COC2(C#C)COC2)=O)CC2CCCC2(NC(=O)C=CSC)C1 C1(CC(=O)N(C(c2onc(C)n2)C)C)C2CN(C(c3nc(C)no3)=O)CC12 N1(c2ccc(OC)cc2)CCCC(NCCc2nc(Br)c(C)s2)C1=O Cc1ccc(CCC(N2CCC(CNC(C3OCCO3)=O)C(C)C2)=O)cc1Cl c1(CCC(C(=O)NCC)N(CCCO)CCC)nc2ccc(F)cc2s1 c1(CCC(=O)NC(CCC#N)CCO)ccc([N+](=O)[O-])cc1 C1(NC(c2nc(OCC)oc2)=O)CCN(C(c2cc(C(N)=O)n(C)n2)=O)C1(C)C C1(C(=O)NC(C(C)C)CNC(c2cccs2)=O)CCC2(CC1)CC2 c1(C(=O)NC2CN(C(=O)C=Cc3cccc(O)c3)C3CC23)scc2c1OCCO2 N1(C(CC(C)(C)c2ccccc2)=O)CC(NC(=O)C2=COCCC2)CC(F)C1 C=CC(C)CC(=O)NC(CN(C(=O)C=CC1CCCCC1)C)(CO)CO N1(C(c2cc(CO)co2)=O)CCC(NC(C2(N(C)C)CC2)=O)CC1C1CC1 N1(C(C(CC#C)(C)C)=O)CCC(C2CC2NC(=O)COc2cnc(Cl)cn2)CC1 C#CCCCCCC(=O)N1CCCC(NC(=O)Cc2cc(C)on2)C1CC c1(C(=O)NCC(CC)NC(=O)CC2CCCC(C)C2)cc(C)nn1CC N#Cc1ncc(NCCC2CCC(NC(C3CCS3(=O)=O)=O)C2)nc1C#N C(=O)(C1=C(F)CN(C(=O)COCC(F)F)CC1)N1CC(C)(C#N)C1 C(=O)(C#CC1(C)CCCO1)N1CC(N(C(=O)C=Cc2cocn2)C)C(O)C1 C#Cc1cc(C(=O)NC2C=CC(CC(=O)NCCC(C)(C)OCC)C2)ccc1C c1(C(=O)NC2CCOCC2NC(C2CCC2(F)F)=O)ccc2nc[nH]c2n1 c1(CNC(C(c2ccc(Cl)cc2)OC)C)ccc2c(c1F)OCCO2 c1(C(N2CCC3(C(NC(CN(C)C4CC4)=O)C3)C2)=O)cccc([N+](=O)[O-])c1 c1(OC)ccc2occ(C(N3CCC(C(C)NC(=O)C4=NNC(=O)C4)C3)=O)c2c1 C=CCCC(C1CC1)NC(C1CC(N(C(=O)CCC2CCCN2C)C)C1)=O C(CCC(C)CC(=O)NCC12CCC(C(=O)NC(C)C3CC3)(CC1)CO2)=C(C)C C1(CCNC(Cn2c(C)nc(C)n2)=O)CN(C(=O)C=CC2CCC2)CC(C)O1 C1(NC(C(C)Sc2nncn2C)=O)C2CCCC1CC(NC(C1CC(O)C1)=O)C2 c1(CNC(C(C)C)=O)ccc2c(c1)CCCC2NC(c1cc2n(n1)CCCO2)=O C(=O)(CN=c1[nH]c(=NCc2ccc(C)cc2Cl)[nH]c2c(F)cccc12)NC C=CCC(C)(CC)C(=O)NCC=CCNC(=O)COCCC C(=O)(C(O)C1=CCCCC1)N1CCC2C(C(=O)Nc3c(C)c(CO)ccc3)C2C1 C(=O)(C(F)CCC(C)C)NCC1(OCC)CN(C(=O)Cc2nccn2C)C1 C(C(C)(C)C(=O)NC1CN(C(=O)C(C)CSc2ccccc2)CC1O)SC N1(C(C2N(C(c3c(CC)nns3)=O)CC=C2)=O)CC2CCCC(O)C2C1 c1(OC)ccc(-c2nc(C(=O)NC(C)CN(C)C(c3n[nH]cc3C)=O)cs2)cc1 C(C)(C)(CCC(=O)NC(C)CS(C)=O)NC(CC1ON=C(C)C1)=O C(N=c1cc(Br)cc[nH]1)C1CCC(OC(C)(C)C)CC1 Cc1cccc(SCc2nc(-c3ccc(F)cc3)nn2C23CC(C2)C3)c1 c1(CNC(CC2(N(C)C)COC2)=O)cccc(NC(=O)CC2CCCN2C)c1 C1(C(=O)NCCCN(C(=O)C(C)CC2CC2)C(C)C)CN(C)C(=O)N1 c1(CN(CCNC(C(C)N(CC)CC)=O)CCOC)cnc(C)[nH]1 c1(C(C(=O)NC(CC)CN(C)C(c2cn[nH]c2)=O)O)cccc(C)c1F Cc1cn2ccc(C(=O)NC(C3CN(C(c4n[nH]c(=N)[nH]4)=O)CCO3)C)cc2n1 c1(C2(C(=O)OC)CC2)ccc(NC(C2CCCC(C(=O)O)O2)=O)c(C)c1 N1(C(C23CCC(OC)C2C3)=O)CCC(NC(=O)C=C2CCC(C)CC2)C(F)C1 CC1=CCC(C(=O)NC2CN(C(c3ccccc3NC(N)=O)=O)CC2C)CC1 C1(O)(CNC(C2C=CCS2)=O)CCN(C(c2cccs2)=O)CC1 C1(C)(C(N2CC(C(C)C)OCC2)=O)CC12CCN(C(=O)CCC(=O)N(C)C)CC2 N1(C(C(C)OCCC=C)=O)CC(C2CCCN(C(=O)CN(C)S(N)(=O)=O)C2)C1 C=CCC(CC)C(=O)N(CCC(=O)NC(CCC)CCO)CCO C(=O)(C(O)C(F)(F)F)NC1(CC)CN(C(C2CC(C)=NO2)=O)C1 N1(CCC(=O)NC(C)C)CCCSCC1c1cnn[nH]1.CN1CCCC(N)C1 CC1CN(C(=O)C=Cc2ncc[nH]2)CCCN1C(=O)C1=C(Cl)CCCC1 N1(C(C(CC)OC)=O)CCC(NC(=O)Cc2ccn(C)n2)C(CO)C1 C1(COC)(CNC(C2(F)CCOC2C)=O)CCCN1C(=O)Cc1cnsc1 CCC(O)CCCN=c1[nH]c(=NCC2CC=CCC2)[nH]c2cccnc12 Cc1scc(C(=O)NCC2CCCCC2NC(c2nsnc2O)=O)c1C N(C1CCc2cccnc21)C(C1C(NC(c2cc(C)ncc2)=O)CC1)=O C(=O)(C(F)CCCCC)NCC1N(C(C=CC=CCC)=O)CC(C)CC1 C1(C(C)NC(=O)C(C)(C)c2ccns2)CCCN(C(c2cccc(F)c2)=O)C1 c1(C(N2C(CNC(C3OCCC(C)(C)C3)=O)COCC2)=O)cc2c([nH]1)CCOC2 C1(C(=O)NC2(CF)CCN(C(=O)CCc3ccc(F)cc3)C2)CC2CCC1CC2 C1(C)(COC)CC(NC(C2(CF)CC2)=O)CN1C(c1nc(O)c(C)s1)=O c1(C(=O)NC)cncc(C=CC(=O)N(CCCNC(=O)C2=COCCO2)C)c1 CCCC(C(O)C(=O)NC1CC2CCCCC12)NC(c1cc[nH]c1C)=O c1(OC)ccc(C(C)NC(N2CC(C)(O)C2)=O)cc1OC C=CCCCC(=O)NC1CCCC1CNC(=O)Cc1ccc(O)cn1 c1(C(CC)OC(=O)COCc2nnnn2C)cccnc1 c1(C(N2CC(OC3CCN(C(c4c(SC)snn4)=O)CC3)C2)=O)cc(C)nc(C)n1 C1(NC(c2ccc(SC)cc2)=O)CCN(Cc2cc(CO)ccc2O)CC1F c1(CN2C(C(=O)OCC)C=CC2)c(OC)cccc1Br N1(C(COCCC=C)=O)CC(NC(=O)C(=Cc2ccccc2)C)CC(C)C1 C(CC(F)F)(C(=O)NC(C)Cc1cnn(C)c1)N(C(c1c(OC)nccc1)=O)C c1(C(=O)NC(CC(C)C)CNC(c2ccnn2CC2CC2)=O)ccc(Cl)cc1F CS(=O)(=O)c1ccc(C(=O)NC2CCCN(Cc3cc(F)cc(F)c3Br)C2)nc1 C=CC1OCCC1C(=O)NCC(C)(C)NC(c1cnn(C)c1COC)=O C1(N(C(=O)C=CC(F)(F)F)C)CN(C(c2ccnn2C)=O)CCC1O C(=O)(CC(C)C(C)(C)NC(=O)OC(C)(C)C)NC(C=C)C(F)(F)F CCC(C)(C(=O)NC1CCCN(C(c2cccc(F)c2)=O)CC1)C(N)=O CC1CCN(C(c2sccc2Cl)=O)C1CNC(=O)Cc1cncc(F)c1 CN(C(=NCCCC1CCOC1)NC1CCC1)CC1CCCN1C N1(C(CCCNC(=O)CO)=O)CC2(CCCC2)c2ccccc21 C1(F)(C(=O)NC(C)C(CO)NC(=O)Cc2cccc(F)c2)CCCOC1 C1(CNC(C2CC(C(C)C)C2)=O)COCCN(C(=O)CN2CCC(=O)NC2=O)C1 c1(C(N(CCNC(c2cc(C)[nH]n2)=O)CC2CC2)=O)ccc(F)c2cccnc12 C1(OCC)CCN(N2CCC(CN3CCOCC3)CC2C(N)=O)C1 N1(C(CSC)=O)CCC2(CCCN(C(c3n[nH]cc3C(F)(F)F)=O)C2)CC1 CCCC(C(=O)N1CCC(C)(C(=O)N(C)CCN2CCCC2=O)C1)NC(C)=O N1(C(c2ncoc2CNC(C23CCC(CC2F)C3)=O)=O)CCC2(CCOC2)CC1 C(CC(C(=O)NC1CCN(C2CCN(C(=O)CSC(C)C)CC2)C1)NC=O)SC C(CCC(O)C(=O)NCCN1CCOC1=O)NC(C(OCC)OCC)=O Cc1ccc(F)c(N)c1C(=O)NCC(C)CNC(=O)C(C(C)C)N1CCCCC1 c1(C(N(CCCNC(C(CC#C)C)=O)C2CC2)=O)ccc(Br)c(C)c1N N1(C(C(C)O)=O)CCCCC1CNC(=O)C(C)(C)n1cc(-c2cnccn2)nn1 Cc1nc(C)c(CNC(=O)C(=O)NC2CCOC(Cc3ccccc3)C2)[nH]1 c1(OC)cc(CN2CC(C(N3CCCCC3)=O)CC(F)C2)ccc1O.C(N)=O C1(C(N2CC(C)(NC(=O)CCc3ccc(Cl)s3)C2)=O)CC(F)C(=O)N1 Cc1nc(N2CCCCC(CNC(=O)C(F)(F)C(F)F)C2)cc(C#N)n1 C1(C(=O)NC(c2nc(C)[nH]n2)C)C2CCC(C2)C1NC(=O)CN1CCCC1 C1(CNC(C2(NC(Cc3cc(C)no3)=O)CCC2)=O)CCOC1(C)C C1(C(=O)NCC(C)CN(C)C(c2coc(C3CCOCC3)n2)=O)CCC12CCC2 Cc1cc(C(=O)NC23CCC(N=[N+]=[N-])(CC2)C3)cc(N)c1Cl N12CCN(CC1)CC2.c1(C(C)NCC(=O)NC(C)(C)C)cc(C(F)(F)F)on1 c1(CCC(N2CCC(C(C)NC(=O)CC3CC3)C2)=O)ccc2ccn(C)c2c1 N1(C(C(CCC)OC)=O)CCN(C(=O)Cn2nc(C)c(C)c2C)C(CCCC)C1 C(=O)(C(CNC(c1cncn1C1CC1)=O)CC1CC1)NCC1(CC)CCOC1 c1(C(=O)NC2(CCOC)CCN(C(C3(O)CC3)=O)C2)n[nH]c2c1CCOC2 N1(C(CC2CC(OC)C2)=O)CCCC2(CCN(C(c3cnc(Cl)[nH]3)=O)C2)C1 C1(O)(C(N2CC(C(C(=O)NCC3CCCOC3)OC)C2)=O)CCOC1(C)C N1(C(C2(F)CN(C(C(C3CC3)OCC)=O)C2)=O)CCCC(C)(CC)CC1 Cc1cc(NC(C2CCC(NC(=O)CCC3CCC3)CC2)=O)ccc1[N+](=O)[O-] N1(C(c2c(C)occ2)=O)CCC2(CC1)CC(NC(C1CCC(N=[N+]=[N-])C1)=O)C2 C1(O)(CNC(C2(CNC(CSCCC)=O)CC2)=O)CCC(C)CC1 C12(C(=O)NCC3C(NC(c4scc(C)c4C)=O)C3)CCCC1C2(F)F C1(N(C(C(C)N(C(Cn2nnc(C)n2)=O)C2CC2)=O)C)CCN(C)CC1 C1(CNC(CCOCCCOC)=O)(N(C2CCOC2=O)C(=O)C2CC2)CC(C)(C)C1 CC1CN(C(=O)COCCNC(C2CS(=O)(=O)C2)=O)CC(C2CC2)O1 N1(C(c2ccc(CO)o2)=O)CC2CC1(C(N1CCOC3CC13)=O)C2 C1(N(C(=O)CN2CC(C)(C)C2)C)CN(C(=O)C=Cc2cncs2)CCC1O Cc1c(NC(=O)C(C2CC=CCC2C)N(C)CCc2nccs2)cccc1Cl N1(C(C(c2ccc(Cl)s2)C)=O)CC2(C1)CN(C(c1cc(C#N)on1)=O)CCO2 O=C1CN(C(c2cnc(O)c(F)c2)=O)C(C(=O)NCc2cncc(Cl)c2)CN1 c1(C(C(=O)NCC=C)N(CC(C)(C)N(C)C)C)nc(Cl)cc(Cl)c1C c1(NC(CC(C)NC(C)C=CBr)=O)cccc(C(F)(F)F)c1 C1(NC(C(C2CCCC2)OC)=O)CC(N=c2[nH]c3cc(Br)cnc3s2)C1(C)C C=CCC(C(=O)NC1C2CC(NC(c3cc(O)nn3C)=O)CC12)OC c1(OC)ccc(C(=O)NCC2(Nc3nc(OC)ncc3Br)COC2)c(F)c1 S(=O)(=O)(CCC(=O)NCC1(NC(c2cc(SC)ccc2C)=O)CCCCC1)NC c1(C(=O)NC(CN(C(=O)Cc2ccoc2)CC)C)nn(C)cc1[N+](=O)[O-] c1(C(C(=O)NC)N(CC(C)C)Cc2ccc(F)cc2)nc(Cl)sc1Cl CCCC(C(=O)N1CCC1CNC(=O)CCc1nc(C)c(C)[nH]1)OCC Cc1ccc(O)cc1C(=O)Nc1cncc(NC(=O)CCN2CCOCC2)c1 c1(OC)ccc(CNC2CCCC2C(=O)Nc2cncc(C(F)(F)F)c2)c(O)c1 C12(C(=O)NC(C(C)NC(c3c(Cl)cnn3C)=O)CO)CCC(C)(C(=O)O1)C2(C)C c1(OC)ccc(-c2ocnc2C(=O)NC(C)CNC(=O)CC2CC(F)C2)cc1 C1(c2ccccc2Cl)(C(=O)NCC(CCNC(C(CC)C)=O)O)CCCCC1 C(C(C)N=c1[nH]cnc2cnn(C)c12)N(C(c1c(OCC)nccc1)=O)C c1(OC(C)C)ccc(F)cc1C(=O)N(C)CCCCNC(=O)C(C)=C1CCCC1 c1(CC)sc(C(=O)NCCCOCCN(C(=O)C(O)CC2CCCC2)C)cc1C c1(C(=O)NC2C(CNC(CCC#C)=O)CCCC2)c2c(nn1C)CCC2 CC1CCCc2c(C(=O)NC3CCCCN(C(=O)CCc4cnn[nH]4)C3)cnn21 C1(CN(C)C(c2cccc(OCCF)c2)=O)CCCCN1C(C1CCCCO1)=O C1(C(=O)NC2(C3CCCN3C(c3ccc(C4CC4)nc3)=O)CC2)C2CCCCC12 c1(C(C(=O)NCC(Cn2cc(CN(C)C)nn2)OC)C)ccc(C)s1 C1(NC(C=CC(C)C)=O)CN(C(c2cc(F)ccc2O)=O)C2CCCC12 N1(C(=O)CCc2csc(Br)c2)CCN(C(c2nn[nH]c2Cl)=O)C2CC12 N1(C(c2cc(C)nc(O)c2)=O)CCC2CN(C(=O)C(C)Cc3cnn(C)c3)CC12 Cc1oc2cc(C(=O)N(CC(C)NC(=O)C(N3CCCC3)C3CC3)C)[nH]c2c1C N1(C(COCCOCC)=O)CCN(C)C(C(=O)N(C2CC2)CC2CCC2)C1 C(COCC)(C(=O)NCCCN(C(C1(CCO)CCC1)=O)CC)OC.C(CN=[N+]=[N-])N C1(OC)CC(CNC(=O)C(C)=C2CCC2)N(C(=O)CC(C)C)C1 Cc1cc(O)nnc1C(=O)N(C1CCC(NC(c2ccncc2C)=O)C1)C C1(NC(CCCNC(c2occc2Br)=O)=O)CCCN(C(c2ccccc2)=O)C1 N1(c2c(C#N)cnc(SC)n2)CCC2CN(C(c3sccc3I)=O)CC12 c1(NC(CN(C(=O)C=CC(=O)NC2CC2)CC#C)=O)cnn2c1OCCC2 CC(C(C)(C)C(=O)NC1CC1(C)C(F)F)NC(c1c[nH]c(=S)cn1)=O N1(C(COC(CC)(C)C)=O)CCC(C(=O)NC2CCCC2CN(C)C)C(O)C1 c1(CNC(C2(CS(C)(=O)=O)CCC2)=O)cnn2c1CN(C(=O)CC1CC1)CC2 n1(CC(=C)C)nnnc1C(c1cccn1C)NCC1(C)CC1(C)C C=CC(C)(O)CC(=O)NCC1(CNC(=O)COCC2CCCCO2)CC1(F)F C(=O)(C1=CCN(C(C2COCC(C)O2)=O)C1)N(CC(CC)OC)C c1(C(N2CC(CCCNC(c3cc(C)on3)=O)OCC2)=O)cc2ncccc2s1 Cc1cccc(Br)c1C(=O)NCC1CCCN1Cc1ncc[nH]1 C1(F)(CNC(C(COC)C)=O)CCN(C(c2cnn(CC(F)(F)F)c2)=O)CC1 Cn1cccc1C=CC(=O)N(C(=O)CN(C1CCCCC1)CC(C)(C)C)CCO N1(C(CC(C)CF)=O)CCCC2CN(C(C3(CO)CC3)=O)CC12 CCCC(C(=O)Sc1ccccc1Br)c1ccccc1.C1(=O)C(C2CCC2)CO1 N1(C(CCC#C)=O)CC(O)CC1CNC(c1ccc(NC(C)C)cc1)=O CCS(=O)c1ccccc1C(=O)NCC(C)NC(=O)Cc1cccc(C#N)c1 c1(C(=O)NC(CC)CNC(C2CCN(C(C)=O)CC2)=O)ccc(S(=O)(=O)NC)o1 c1(OC)nc(C)ccc1C(=O)NCC1(CNC(=O)CCC2CCOC2)CC1 c1(N2CC(n3cc(C(C)O)nn3)C(O)C2)ccc(C(F)(F)F)cc1[N+](=O)[O-] c12ccc(cc1)NCC2N.c1(C(C)OCC(=O)O)ccccc1Br c1(CCCNC(C(=O)Nc2ccc(SC)nc2)=O)nc2ccccc2s1 C=C=CCCC(=O)NC1CC1CNC(c1ccc(COC)s1)=O N1(CC(COC(C)C)O)CCN(C(=O)NCC2CNC(=O)O2)CC1 C12(C(=O)NCC(C)(CC(C)C)NC(Cc3c(C)nc[nH]3)=O)CCC(C)(CC1)OC2 N1(C(c2ccc(CC)[nH]2)=O)CC(C2CN(C(C3CC4CCCC4C3)=O)C2)C1 C1(NC(C(F)=CCC)=O)CCN(C(c2ccc(OC)cc2F)=O)CC(C)(C)C1 c1(OC)ncc(C(c2nnnn2CCSC)Nc2cc(C)c(CO)cn2)cc1C N1(C(C2C(c3ccc(C)cc3)CCC2)=O)CCCCCC1C(=O)N1CCCO1 CCC(CC(=O)N1CC(CNC(=O)C=Cc2ccccc2C)C1)C(C)(C)C c1(C(N2C(C(=O)NC(CC=C)C)CCC2)=O)ccc(C)nn1 Cn1cnc(C(=O)N(CCC(=O)NCC(c2ccsc2)O)C2CC2)n1 c1(C(N2C(C)CCC(NC(CC(=O)OC)=O)C2)=O)nn(C)c2c1CCC2 c1(C(C(COC)C)C)nc(CO)nn1-c1cncc(Br)c1 CCCCC(O)CC(=O)N1CCOC(CNC(=O)CCF)C1 c1(CN(CCN(CC)CC)C(C2CCN(C)CC2)=O)cnc(C2CCOCC2)nc1 CC1CN(C(=O)C(C2CCOCC2)F)CCN1C(=O)C(F)OC(F)(F)F C1(C(=O)NCC2CCCC(NC(=O)CC3(O)CCCC3)C2)CC2(C1)CC(F)(F)C2 N1(C(c2csc(C)c2C2CC2)=O)CC2CCC(NC(C3CCCCCC3)=O)(C2)C1 c1(C(=O)NC(C)C(=O)NCCN2CCC3CC23)c(Cl)cnn1C N1(CC)CCOCC1CC(N1CCCC1CNC(c1cc(Br)c[nH]1)=O)=O C1(N(C(=O)CN2CCC(NCc3ccn(CC)n3)C2)CC)CCCCC1OC C#CC1CCC(NC(C2(NC(=O)Cc3cnc(C)s3)CCC2)=O)C1 c1(C(N2C(C3CCN(C(C4(SC)CCC4)=O)CC3)CCC2)=O)cc(F)ccc1F Cc1c(C(N2CC(O)CC2(C)C(=O)NCCC(C)CO)=O)cccc1O N1(CC)CCCCC1CNC(=O)C(C)CN(C(=O)Cc1cncnc1O)C C(=O)(C1=NOC2(CCOC2)C1)N(CCNC(c1c(F)ccc(C)n1)=O)CC1CC1 Cc1cc(C(C)NC(c2nc(-c3c(C)nn(C)c3C)cs2)=O)cc(C)c1 N1(c2c(C)c(NC(C)Cn3cccn3)ncn2)CCn2c(CCO)nnc2C1 CC(C)C(C(=O)N(C)CCNC(C1(C)CCCN1C(=O)OC(C)(C)C)=O)C(C)C Cc1ccncc1C=CC(N1CCCC(NC(=O)CCN2CCOCC2)C1C)=O C1(C(=O)NC(CCCNC(c2c(C)cnn2C)=O)C)CCN(CCO)C(=O)C1 C1(CC(=O)NC(CC)CCOC)(NC(C(COCC)C)=O)CCCCC1 N1(C(C2(C)COCCO2)=O)CCCCCC(NC(=O)Cc2cc(C3CC3)on2)C1 CCC(C)CCCCC(=O)NCC1(C(=O)NCC(=O)N(CC)OC)CC1 CC1CCN(C(C2CN(C(=O)CCS(N)(=O)=O)CC2F)=O)CCS1=O n1(CC(N2C(C)CN(C(c3cc(Cl)ccc3F)=O)CC2)=O)ncc2cccnc12 Cc1cc(C(N2CC3(NC(=O)C(C)SC(F)(F)F)CCC2CC3)=O)c(O)c(C)c1 c1(CNC(C(C)n2ccnn2)=O)nc2c(s1)CCN(C(c1ns[nH]c1=O)=O)C2 C12(C(N3C4(CNC(c5ccc(F)c(Cl)n5)=O)CC(C3)C4)=O)CCCC1C2(F)F c1(CN2CC(C(=O)OC)CC(CC)C2)cc2cc(Br)ccc2s1 c1(C2C(C(=O)NCC)C2C(=O)OC)ccccc1NC(C)C(C)C C1(C(=O)OC)CN(C(=O)COCCF)CC1(C)C.N1(CC(C2CCOC2)SN)CCCC1 C(=O)(C1c2ccccc2C2CC1C2)NCC1CCCN(C(C(C(C)C)SC)=O)C1 CCCC(C)CC(=O)N1CCC(C(=O)NCCF)CC1C C1(CCNC(C2CCC(F)CC2)=O)CCCCN1C(=O)COc1ccccc1Cl N#Cc1cc(C(N2CCN(Cc3cnc(Cl)s3)CC2C#N)=O)ccc1Br Cc1cccc(C)c1OCC(N1CC2CC1CN2C(c1ccncc1Cl)=O)=O N1(C(C(=O)Nc2ccccc2)=O)CCC(CO)C(NC(=O)C(O)C2CC2)C1 C12(NC(=O)C(O)CCc3ccccc3)CCCC1CN(C(c1cscc1Cl)=O)C2 C1(C(=O)Nc2cn(C)nc2)CCCN(C(=O)Nc2csc(-c3ccccc3)n2)C1 C(=O)(C1=CS(=O)CCC1)N1CC2CC(CNC(c3cc(C)ncc3C)=O)C2C1 N1(C(c2c(C)nsc2)=O)CCC(F)(C(=O)NCC=Cc2ccccc2)CC1 C1(CC(=O)NC2CC(CNC(C=Cc3n(CC)ccn3)=O)C2)CC2(CCO1)CC2 C1(C(=O)NCC2(CNC(C3C(C)(C(F)(F)F)C3)=O)CCC2)CCc2c[nH]nc2C1 N1(C(C(C)OCCC=C)=O)CC(C)C(N=c2[nH]c(Cl)nc(CC)c2F)C(C)C1 c1(C(=O)OC)cnc(=NC(CCN(C(=O)C=C2CCC2)C)C(C)C)[nH]c1 c1(OC)ccc(C=CC(N2CC(NC(C3CC(O)C3)=O)CC(C)C2)=O)cc1Cl Cn1cc(C(F)=CC(=O)NC2(CO)CN(C(C34CCC(F)(CC3)C4)=O)C2)cn1 c1(C(=O)NCC(C)(C)OCCNC(CN(C)CC)=O)cc(Br)cnc1C C=CCCCCC(=O)NCC1C=CC(NC(c2cc(Cl)ccc2NC(C)C)=O)C1 C1(CNC(c2nc(C)c(C)s2)=O)CCC(C)N(C(c2cnn[nH]2)=O)C1 CONC(=O)C(=O)NCC1CCN(C(c2ccns2)=O)CC1 N1(C(C(CC)N(C)C)=O)CCC(C)(C)C1CNC(c1ccc(F)cc1C)=O Cc1cc(Cl)cc2[nH]c(C(=O)NC3CCN(C(C4CN(C)C4)=O)CC3CO)cc12 C1(C(=O)NCCCN(C(CC2CC(OC)C2)=O)C2CC2)CCN(CC(F)(F)F)C1 N1(C(C(C2CCC2)OC)=O)CCN(C(=O)CCc2ccoc2)C(CO)C1 C1(NC(c2ncn(CC)n2)=O)CC2C(NC(C3CCC(OC)C3)=O)C2C1 N1(C(c2nnn(C)n2)C(=O)NC2CCCC2)CC2(CCCC2)C1c1ccccc1 N1(C(C2C(C=C)OCCC2)=O)CCC2CN(C(=O)CS(=O)(=O)NCC)C2C1 C1(CNC(c2cc[nH]n2)=O)CN(C(c2nc[nH]c3nccc2-3)=O)CC2(CCC2)O1 C1(NC(C2CCC(=C)CC2)=O)CCC(C)N(CC2CC2)C1 N1(C(C(C=C)C)=O)CCC(C(C)C(=O)NCC2CCC2OCC)CC1 N1(C(c2c(Cl)cc(C)s2)=O)CCCC2(CC(NC(=O)C(=O)NCC(F)F)CO2)C1 C1(C(=O)NCCCN(C(Cc2c(C)nsc2)=O)CCO)COCC1(C)C CC1c2cc(Cl)cc(Cl)c2CCN1C(C1CCCN1C=O)=O CC1CC2CC2CC1C(N1CCC(n2cc(C3(C)CC3)nn2)C1)=O n1(CC(=O)NC2C(C)CN(C(C3OCCCO3)=O)C2)ccc2ccccc2c1=O c1(CN(C(=NCCOC)NCc2ccc(COC)s2)C)c[nH]c2ccc(C)cc12 n1(CCOC)ccc(=NC(=O)CC2CN(C(=O)C(Cl)Cl)CCO2)[nH]1 C1(C2(NC(C3C(C(=O)OC)C3)=O)CC2)CCCN1C(c1c[nH]nc1SC1CC1)=O N1(C(CSC2C(=O)OCC2)=O)CCC(NC(c2cncc(Cl)c2)=O)C12CC2 C1(C(N2CCC(C3=NOCC3)C2)=O)C2C3CC4C1C1C2CC3C41 N1(C(C(C(C)O)(F)F)=O)CC(O)(C2(CNC(c3nocc3Br)=O)CC2)C1 n1(CCCC)cc(NC(C2CC(O)(Cc3ccccc3C)C2)C(C)C)c(C)n1 N1(C(=O)OC(C)(C)C)CCC2CN(C(=O)CC3CC(C(N)=O)=NO3)C2C1 C1(C(=O)NC(c2ccccc2Br)C(=O)OC)CCn2nccc2C1 Cc1c(C(=O)NCC(C)(O)CNC(C2COC2)=O)cnn1C C(N=c1cc(Cl)nc(S(C)(=O)=O)[nH]1)C1OCC(CNC(C2(OC)CC2)=O)C1 N1(C(CCC)=O)CCC(C)(C)C1CNC(=O)COCC1CCOCC1 C1(CCNC(CCN(C(C2C(C(C)C)CCC2)=O)C)=O)CC2C=CC1C2 C#CC1CCC(CNC(C2CCC(CNC(C3(C)C=CCC3)=O)O2)=O)CC1 C1(C2CCN(C(c3ncn(C(C)(C)C)n3)=O)C2)(NC(C2N(C)C(=O)CC2)=O)CC1 C1(CC)CN(C(=O)CN2CCCC2=O)CCC1NC(=O)C1=C(C)CCC1 C1(CNC(C2(C(C)C)COC2)=O)C2CC1N(C(=O)Cn1cnnn1)C2 N1(C(COCCC#C)=O)CC2CCC(C1)C(NC(c1sc(C)cc1Cl)=O)C2 C1(NC(C=Cc2c(C)ccs2)=O)CCC(C)N(C(=O)COc2ccc(F)cn2)C1 c1(C(N2CCOCC(NC(CCCCN(C)C)=O)C2)=O)cc2c(cc1O)OCO2 Cc1sc(=O)n(CC(N2CCC(F)(CNC(=O)C=CC(C)C)CC2)=O)c1C c1(C(N2CC(OCCNC(CCC=CCC=C)=O)C2)=O)cc2nccn2c(O)n1 N1(C(C(CC)(C)C#N)=O)CCCC(O)(CNC(c2cc([N+](=O)[O-])oc2C)=O)CC1 N1(C(C(C=CCCC)O)=O)CCCC1(C)CNC(=O)C(C)OCC1CC1 C(=O)(C1=COCCO1)NCC(C)(CO)NC(c1cccc(-c2nnco2)c1)=O c1(OC)cc(C#N)ccc1C(N1CC(NC(=O)C(C)CC(C)(C)C)CC1(C)C)=O Cc1[nH]c2ccccc2c1C(=O)NCC12CC1CN(C(=O)C=Cc1ccco1)C2 CC(C)(C)CCCCC(=O)NCC1CN(C(=O)CC2OC(C)(C)OC2=O)CCO1 c1(C(=O)NCC2(CNC(c3cc[n+]([O-])cc3)=O)CCC2)c(Cl)csc1Cl c1(C(N2CC(O)(C(C)NC(C=NOC)=O)C2)=O)cc2ccc(C(C)(C)C)cc2[nH]1 C1(C(N(CCCC(=O)NC)C)=O)C2CCN(C(=O)C(Cl)Cl)CC12 c1(C(=O)NCC2N(C(CC(C=C)C)=O)CCC(C)C2)c(C)ccc2nonc12 N1(C(COC)=O)CCCOC2(COCCN(C(=O)Cn3nnnc3C)C2)C1 C1(CNC(CC(CC)SC)=O)CN(C(C2(CO)CC2)=O)C2CCCCC12 C1(NC(c2ccc(CC)cn2)=O)CC2CC1N(C(=O)CCC(=O)N(C)C(C)C)C2 CC(C(CCc1ccccc1)NC(C1CN(C(N)=O)C1)=O)NC(c1cocn1)=O c1(COC)ncc(C(=O)N(CCC(C)NC(C2(C3CC3)CC2)=O)C)s1 C(=O)(C1CNC(=O)c2ccnn21)N1CC(C2(NC(C3C(C)C3)=O)CC2)C1 C1(NC(c2cscc2Br)=O)CCN(C(c2ccc(F)o2)=O)CC1O CC(C)C(C)(CO)NC(=O)CCC(C)NC(c1cnc(S)nc1)=O C1(C(C(=O)NCc2cccs2)N(CC)Cc2cn(C)nn2)CC12CCOC2 c1(C(=O)NCC(=O)NC(C)C2CC2)ncnc2scc(-c3cccs3)c12 c1(C(=O)NCC2C(NC(=O)C=CCO)CCC2)c(O)cc(O)cc1O c1(C(N2CCCCC2Cn2cc(C3(O)CSC3)nn2)=O)ccn2ccsc12 N1(C(C(CC)NC(C)=O)=O)CCN(C(=O)C=CC(=O)N(C)C)CC1COC N1(C(CCc2onc(C)n2)=O)CCN(C(=O)CC(C)O)CC1C1CC1 C1(NC(C2C(CC)CCCC2)=O)CN(C(=O)CP(C)(C)=O)CC12CCCC2 c1(Cn2c(-c3cnnc(C)c3)nc(C(CC)C)n2)cc(F)cc(Cl)c1 c1(C(=O)NCCOC2CN(C(C(C(C)(C)C)SC)=O)C2)cc(C)cc2c1OCC2 c1(C(=O)NCCC(CNC(C=Cc2cc(C)no2)=O)O)cc(N)c(F)cc1C Cc1cn2ccc(C(=O)OCc3c(F)ccc(C)c3Br)cc2n1 C1(OCCNC(C2C(C=C)C2)=O)CCN(C(C2CCOC2)=O)CC1 N1(c2nnc(C)c(C)n2)CCN(C(=O)COC(C)C)CC(O)C1 c1(CC=C)ccccc1C(=O)NCC1(F)CN(C(C2C3CCC2CC3)=O)C1 C1(NC(C(C)NC(CC)=O)=O)CCC(NC(=O)C(C)(C)n2cccn2)C1 CCCCCCC(C)C(=O)N(C)CC1CCCN1C(c1nocc1Br)=O C1(NC(c2c(C)snn2)=O)CC2CC(NC(=O)CCC3CCC(=O)NC3)CC2C1 C1(C(N(CCC(=O)N(C)Cc2cc(C)nn2C)C(C)C)=O)CCOCC1(C)C c1(NC(=O)NC2(F)CCN(C(C)=O)C2)cc(C)cc(Br)c1C Cc1nc2cccc(C(N3C4CCC3CN(C(=O)C=C(Cl)Cl)C4)=O)c2[nH]1 CC1CCn2cc(C(N3CCC(NC(c4cccc(C(F)F)n4)=O)C3)=O)nc2C1 C(=O)(C(C)C(F)(F)F)N.Cc1ccc(C(N2CCCC2CN(C(CN)=O)C)=O)s1 C=C1CCC(C(=O)NCCC2CCCCN2C(C2CC(SC)C2)=O)CC1 N1(C(c2cnco2)=O)CCCC(c2cn(Cc3cnns3)nn2)C1 C(CCC)(C(O)C(=O)NCc1ccon1)NC(C(C=C=C)C)=O CC1CCc2onc(C(=O)NCCC3(O)CCN(C(C4CC(F)C4)=O)CC3)c2C1 N1(C(C2(COC)COC2)=O)CCCC(NC(=O)CCc2conc2C)CC1 C(=O)(C=CS(C)=O)NC(C1N(C(COc2cc(C)on2)=O)CCC1)C C(CC(C(=O)NC(C)Cc1cccs1)NC(c1c[nH]nc1OC)=O)=CC C=C(C)CC(C(=O)NC1CN(C)CC1(F)F)NC(=O)C(CC1CC1)OC c1(CN2C(C(=O)NCc3nc(C)c(Br)s3)CC(F)C2)ccc2ncsc2c1 c1(C(=O)NCC2N(C(c3cnc(OCC)s3)=O)CCC2)cc(OC)cc[n+]1[O-] c1(OC)ccc(F)cc1CC(=O)NCC(C)CNC(=O)CC1NC(=O)NC1=O CCC(CC)CCCC(=O)NCC1(C(=O)NCCC2CC(C)(C)CO2)CCCC1 C(=O)(C1=CCCOC1)NCCOCCN(C(CC1C(C)OC(C)C1)=O)C Nc1cc(C(=O)NC2CN(C(c3c[nH]c(=O)cn3)=O)CC23CC3)ccc1Cl c1(C(=O)NC2CCC(CNC(C3C(C)C3C)=O)C2)cncc2ncn(C)c12 N1(C(c2cc(CC)n(C)n2)=O)CCC(C2CCN(C(c3ncccc3C)=O)C2)C1 c1(C(=O)NC2CCCCCN(C(C3C=CCC3)=O)C2)ccc2ccc(O)nc2n1 N1(C(CN(C)CC)=O)Cc2nccn2CC(NC(=O)CNS(C)(=O)=O)C1 N1(C(CC(=C)C)=O)CC(NC(=O)C=CCN(C)C)Cc2ccccc21 c1(OC)cc(Br)cc(C)c1NC(C1CC1NCc1cccc(-n2cncn2)c1)=O c1(C(N2CC3=C(CN(C(c4ccc(=N)[nH]c4)=O)C3)C2)=O)noc2cc(F)ccc12 Cc1[nH]nc2ccc(C(=O)NCCC3C(C)CCCN3C(=O)COCCO)cc12 c1(CC)nc(=NC(CNC(=O)CC(CC)C(C)C)C2CCC2)s[nH]1 c1(C(=O)NCC2(F)CN(C(c3ccc(F)cc3F)=O)C2)cc2n(n1)CC(F)C2 c1(C(N2CCCC(CN(C(=O)CCCC(C)(F)F)C)C2)=O)ccc2[nH]ccc2c1 C1(CN(C)Cc2ccccc2F)CCCCN1C(c1cc(C(F)F)cs1)=O c1(CCC(=O)NCC2C(NC(CCCC#C)=O)CCC2)cccc(F)c1Cl c1(C(N(CCCCN(C)C(C2CC(=C3CCC3)C2)=O)C)=O)cc2c(o1)CCCC2 c1(OC)cnc(Br)c(NC(C2CCN(Cc3cc(Br)cnc3F)CC2O)=O)c1 c1(C(N2CC(C)C(NC(c3ccsn3)=O)C2)=O)cc2cnn(C)c2s1 CC1=NOC(C(=O)NC2CCN(C(=O)CCc3csc(=N)[nH]3)C2)C1C c1(CC)ccccc1C(CNC(=O)Cc1cnns1)NC(c1cccs1)=O Cn1ncc2c(N3CCSC(C)(C)CC3)nc(=NC3CSC3)[nH]c12 c1(C(=O)NC2(CCNC(c3coc(Cl)n3)=O)CC2)cc2cc(Cl)ccn2n1 c1(C(=O)NC(CN(C(=O)CC2CC2)C)(C)C)cnnc(-c2cccs2)c1 N1(C(COCC(=O)NC)=O)CCC(NC(C2(F)CC2(F)F)=O)C1 c1(NC(C2CNCCN2)=O)cnc2ccc(F)cc2c1 Cc1cccc2cc(C(=O)NC(CNC(=O)CN3CCC(C)C3)C3CC3)cnc12 CC1COCCC1C(=O)NCC12CC(NC(c3cnn(CCO)c3)=O)(C1)C2 c1(C(N)=O)ccc(C(=O)NC2CCOCC2NC(=O)Cn2nnc(=O)[nH]2)cn1 c1(C(N2C(C)CCC2C)=O)cn2c(n1)CCN(Cc1ccc3cncn3c1)CC2 n1(CC)cccc1C(N1CCCC1CN(C(c1cncnc1)=O)C1CC1)=O CC12CCN(C1)C2.C1(NC(N)=O)CCCN1C=O.C12(CC1)C(=O)N2 O=C(C1=CCCC1)NC(C(=O)NCCC1CCCC2CC12)C1CC1 N1(C(C=CCCC)=O)CCCC2(CCCN2C(=O)C(N2CCCC(O)C2)C)C1 C1(N)(CN(c2ccc(Cl)cc2F)CC)CC2CCCC12 CC1CCCC(OCC(N2CC(CO)(NC(=O)C(C)(C)n3ccnn3)C2)=O)C1 N1(C(CC2CC(SC)C2)=O)CC(C2CC2C(N2CC(C)(F)C2)=O)C1 c1(N(C(C=C(C)CNC(c2cc(O)nn2C)=O)=O)C)cc(C)ccc1C C1(S(C)(=O)=O)(C(N2CCC(NC(CN(C)C(c3ccc(C(N)=O)[nH]3)=O)=O)C2)=O)CC1 C(CCCCCCCO)=CC(=O)NCC(=C)CCNC(c1occc1C)=O c1(-c2nc(CCOC)nn2-c2cc(C)nc(C)c2C)cc2c(Br)cc(C)cc2[nH]1 C(C)(C)(CCCNC(C1CC12CC2(F)F)=O)NC(CN(C)C(n1cncn1)=O)=O C(=O)(C#CC1CCCOC1)NC1CCN(C(C2(N(C)C)CCCC2)=O)CC1F C1(CNC(C(CCC2CCCC2)NC(C23CCCC2C3)=O)=O)CC2CCCC2C1 C1(C(N(CCC)CCNC(=O)CSCCC#N)=O)OC(C)(C)OC1(C)C C(=O)(C(CC=C(Cl)Cl)c1ccccc1)N1CCC(C)(NC(=O)Cn2cnnc2)C1 c1(C(=O)NC(C)CN(C(=O)CCCC(=O)N(C)C)C)cc2ccc(Cl)nc2s1 C(CC(C(=O)NC)NC(=O)COCC(=O)NCCc1scnc1C)OCC N1(C(c2c(C(=O)OCC)[nH]cc2)=O)CC=CC(NC(C2CCCN2N=O)=O)C1 c1(NC(Cn2c(C)c(O)c(=O)cc2)=O)ncnc2c1c(I)cn2C C1(NC(c2n(C)cnc2)=O)CN(Cc2ccc(Cl)c(Cl)c2F)CCC1(F)F c1(C(=O)OC)nc(=NCC(C(C)(C)C)OC)cc(COC)[nH]1 N1(C(C=CC(=O)NC2CC2)=O)CCC(F)CC1C(N1CCC(CC(F)F)C1)=O N1(C(=O)C(c2ccccc2)O)CCc2cccc3c2C(CCC3)C1 c1(CC)nc(Cl)nc(NC2(CNC(C3COC(C)C3)=O)CCC2)c1Cl c1(C(=O)NC(CC)(C)CNC(C2CC2c2ccnn2C)=O)c[nH]c2ncccc12 N1(CC)CCCC(C(=O)NCCOC2CN(C(C3(Cl)CC34CCC4)=O)C2)C1 N1(C2(CC=C(C)C)CCOC2)CC2C3C=CC(O3)C2C1 c1(NC(=O)NCCCN(C(C)=O)CCO)cccc(C(C)(C)O)c1 Cc1ccc(C)c(OC(C)C(N2CC3(CC(CO)C3)C2)=O)c1 N1(CC)CCC(CNC(=O)C(C)(C)CNC(C2C=CCC2)=O)CC1 CC1CCC(C)(C(=O)N(C2(C(=O)NCc3ncc(CO)[nH]3)CC2)C)C1 CC1(C)CN(C(c2cc(F)c[nH]2)=O)C1C1CCN(C(c2cnsc2)=O)C1 N1(C(C(C)N2CCC2)=O)CC(C(F)(F)F)C(CNC(C23CC(C#N)(C2)C3)=O)C1 C1(NC(=O)Cc2cccc(Br)c2)CCCCC12CCN(C(c1cc[nH]c1)=O)C2 Cc1nccn1CCC(=O)NC(c1cn(C)nn1)C(=O)NC(C1CCC1)C C12(CNC(CCCOC)=O)CC3CC(CC(NC(=O)CCC=C(C)C)(C3)C1)C2 C(CCSC)(C(=O)NCCCCC1CN(C(=O)CCC2CCCC(=O)N2)C1)OC CC1CCC(C)N1CC(=O)NCc1ccc(CNC(=O)C2=NOCC2)cc1 c1(CCC(=O)NCC2(OC)CN(C(=O)C(C)O)C2)cccc(C(F)(F)F)c1 N1(CC)CCOC(C(=O)NC(CC2CC2)CC(=O)NCc2ccccn2)C1 C(=O)(CCC(=O)NN(C)C)N1C2CC(NC(COCC=C)=O)C1CC2 N1(C(C(CC=C)(C)C)=O)CC(C)OC2(CCN(C(c3cc(CO)[nH]n3)=O)C2)C1 c1(C(=O)NCC2OCCN(C(C(C(C)(C)F)(C)F)=O)C2)c(Cl)oc2ccccc12 C(C(O)CC(=O)NCc1cc(CN2CCN(S(C)(=O)=O)CC2)on1)N(C)C c1(COC)ccccc1CC(N1CCCCC1C1CCN(C(=O)CC2CC2)C1)=O C#CCCN=C(NCCn1cccc1)NCc1ncn(-c2ccccc2)n1 CC(C)C(C)C(CNC(=O)Cc1csc(S)n1)NC(=O)Cc1csc(S)n1 CC(C)CCCCC(=O)NCC#CC(=O)NCCN1CCOC1=O c1(OC)ccc(I)c(C(N2CC(C)CC2C(=O)Nc2c(OC)cccc2C)=O)c1 C(c1ccc2occc2c1)=CC(N1C(CNC(C2C(=C)CC2)=O)CCC1)=O c1(OC)cc(C=CC(=O)NCCCNC(=O)CN2CC(C)(C)C2)cc(Cl)c1OC c1(CCC(=O)N(C(C)C)C(C2CNC(=O)C2)=O)c(F)cc(Br)cc1F N1(CCN(C(n2cc(C3(n4ccnn4)CC3)nn2)=O)C2CC2)C(=O)CNC1=O Cc1onc(C(N2C3CCC2C(CNC(C2(C)CC=CC2)=O)C3)=O)c1[N+](=O)[O-] C(=O)(CCCC(=O)NC1CCN(C(=O)CC2C(=O)NN=C2C)C1C(C)C)NCC C1(C(=O)NCC(C)C2CCC2)CC(C)(C)CCN1C(=O)C1=CCCCCC1 N1(C(C2CCN(Cc3c(C)nn(C)c3)C2)=O)CC(C(F)(F)F)CCC1=O c1(C(N(CCCN(C)C(c2c[nH]c(C#N)c2)=O)C)=O)ccccc1OCC(N)=O Nc1cc(C(=O)NC2CC2CNC(=O)CCC=CBr)ccc1C(F)(F)F C1(NC(COCCSC)=O)CCCCC1NC(c1ccccc1C(=O)N(C)C)=O C=C(Cl)C(C)(C)C(=O)N1CC2C(CN(C(=O)C(C(C)OC)NC(C)=O)C)C2C1 C1(NC(C(C)C(F)F)=O)CN(C(c2cnc(C(N)=O)s2)=O)CC12CCOCC2 N1(C(c2c(C)ccnc2O)=O)CC2(COC(CNC(=O)C(C)c3ncco3)C2)C1 C1(OC)CN(C(C2CCCSC2)=O)CC1NC(c1ncsc1C1CC1)=O Cc1cccc2c1CC(C(=O)NC(C)(CNC(=O)CC1CC1)C1CC1)O2 C1(NC(COCCOCC#C)=O)CN(C(=O)C=Cc2ccccn2)CC1N=[N+]=[N-] C(CCO)(C(=O)NCC1CC2CC2N1C(c1ccon1)=O)N(C)C c1(C(=O)NCCCN(C(=O)C(c2ccc(C)s2)C)CC)cncc(C)c1C C=CC(C)(O)CC(=O)NCCc1ocnc1CNC(c1cc(O)nc(CC)n1)=O N1(C(C2(C)ON=C(C)C2)=O)CC2CN(C(c3cc(CN(C)C)on3)=O)CC2C1 c1(C(N(C(C(=O)NC(c2cncnc2)C)C2CC2)C)=O)nc(=N)cc[nH]1 C(=O)(CS(=O)C(F)(F)F)N(C1CCCN(C(C#CC(=O)N(C)C)=O)C1)C CC(C)C#CC(=O)NC1CCC1CNC(=O)CCCNC(c1cccnc1)=O C1(CC(=O)NC(C(C)NC(C2(NC(C)=O)CCCC2)=O)C)SC(=N)NC1=O N#Cc1ccc(O)c(NC(C2CCCC(NC(=O)C=Cc3ccncc3)C2)=O)c1 c1(C(C)(F)F)ccnc(C(N2CCC(CCNC(=O)CC3CCOCC3)C2)=O)c1 CN=c1[nH]c(=NCCCCC#N)[nH]c(=NC2CCC(OC)C2)[nH]1 Cc1nc(NC(c2csc(-c3ccc(-c4cccnc4O)cc3)n2)=O)sc1I Cc1cccc(C(=O)NCCCC(C)NC(=O)CC2CCCCC2O)c1C c1(CC(=O)NC(C2(CNc3ccc(F)nc3)CC2)C)ccncc1Cl N1(C(c2ccc(CC)cn2)=O)CCC2(NC(c3cnc(Cl)[nH]3)=O)CCCCCC12 C1(C(=O)NCCCC)CC(F)CCN1C(=O)CC1CC2(CC2)C1 c1(C(N(CCCNC(C23CC(OC)C2C3)=O)C)=O)cnc2nccnc2c1 N1(C(C23N(C(c4sccc4F)=O)CCC2CCC3)=O)CCOC2(CCCC2)C1 c1(OC)ccc(NC(=O)CC2CN(Cc3c(C)cccc3C)C2)c(OC)c1 C12(C(N(C3CN(C(=O)CNC=O)CC3F)C)=O)C3CC(CC13)C2(F)F C1(CNC(Cc2n(C(C)C)cnn2)=O)(CO)CCN(C(=O)C(F)C(C)(F)F)CC1 CN1CCC(C(=O)NCC2CN(C(=O)Cc3csc(-c4ncccn4)n3)C2)C1 c1(C(=O)NCC(CNC(C2CC(C(F)(F)F)(OC)C2)=O)C)cccc(F)c1SC N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCN(C(c2c(C)cccc2N)=O)CC12CCC2 c1(C(N2CC(NC(c3cnc4nccn4c3)=O)C(O)C2)=O)nnn2c1CSCC2 C1(NC(c2nccc(C)c2)=O)CN(C(=O)C(C)N(C)C)CCC1C(F)(F)F C1(NC(C2CCC(OCC)CC2)=O)CN(C(=O)C(COC)OC)CCC1(C)C C1(O)(CN(C)C(C2CC2(F)Cl)=O)CN(C(c2cc(CC3CC3)on2)=O)C1 C1(NC(c2ccnnc2O)=O)CC2(C1)CN(C(=O)CCc1cccnc1)C2 c1(OC)sc(C(N2CCC2CNC(C2(C)CC3CC3C2)=O)=O)cc1Br c1(CC)ccc(CNC(=O)C(Cn2ccnn2)NC(=O)CC2CCCC2)cc1 CC1ON=C(C(=O)N2CC(O)(CN(C(=O)CC3CC(F)C3)C)C2)C1C C1(CNC(c2c(CCC)occ2)=O)CCCC(NC(c2ccoc2)=O)C1 N1(C(C(C(=O)OC)OC)=O)C2CC=C(C(=O)NC3CN(CC(F)F)C3)C1CC2 c1(C(=O)NC(c2cncnc2)C)cc(F)ncc1NC(=O)Cc1ccncc1 C=CC1(C(=O)NCC2CCN2C(c2ccc(C)c(CC)c2)=O)CCCCC1 Cc1nc(N2CCOCC(NC(=O)CCCCF)C2)c2c(C)csc2n1 C1(CC=C)(C(=O)O)CCCCN1C(c1cc(C)ns1)=O c1(C(=O)NCC(CC(C)C)NC(c2cc(CO)[nH]n2)=O)cnn2c1CCCC2 C1(C(=O)NCC2N(C(c3cnc(CC)s3)=O)CCOC2)CCc2c[nH]nc2C1 N1(C(C(C)=C2CCC2)=O)CC(NC(c2csc(-c3cnn(C)c3)n2)=O)CC(C)C1 N1(C(C(C(C)O)C)=O)CCCCC12CC(NC(=O)CCCOCc1ccccc1)C2 C1(C(=O)NCC(CN(C(=O)Cc2ccon2)C)O)CCn2c(O)nnc2C1 Cc1cc(O)c(C(=O)N(CCCN(C)C(c2cccc(C)n2)=O)C)nn1 C(=O)(C(CO)C(C)(C)C)N(CCC(C)NC(c1c(C)c(C(F)(F)F)ccc1)=O)C C(=O)(CCC(CC)OC)NC1(CC=C)CN(C(c2cc(C)nc(O)n2)=O)C1 CC1CCN(C(=O)C(c2cnccn2)C)CCN1C(C1CCCN1C)=O c1(CCC)nc2ccccc2n1CCC(N1CCCCC1c1nccn1C)=O C1(c2nnc(C)o2)CN(C(=O)NCc2ccc(F)c(C3CC3)c2)CC(C)O1 c1(C(C)=O)cn(CC(N2CC(n3ccc(Br)n3)C2)=O)nn1 C1(CNC(CC(n2c(C)cc(C)n2)C)=O)CC2(CO1)CN(C(=O)C=CCO)C2 C1(CC)CCN(C(=O)C(F)(F)c2cnccn2)C(CC)C1 CCCC(C(=O)OC)NC(=O)CC1CCN(C(=O)CNc2ccc(F)cc2)CC1 C#CCCCC(C)C(=O)N1CC2CC1CN2CCCNC(=O)C(F)(F)F O=C1CCC(C(=O)N2CCC3(CC2)CN(C(c2ccc(Cl)o2)=O)C3)n2cccc21 c1(OC)ccc(C)c(C(N2CCC(O)(C(C)NC(=O)CC(F)F)C2)=O)c1N Cc1ccc2c(c1)CC(C(=O)NCCCN(C(=O)Cc1ccoc1C)C)S2(=O)=O c1(C(N2CC(CC)N(C(c3sccc3C#N)=O)CC2)=O)ccc(F)c(F)c1C Cn1cnnc1CNC(C)(CCC1CC1(Cl)Cl)c1nnnn1-c1ccccc1 N1(C(CCC(=C)C)C(=O)NC(c2ccccc2)C)CC2(CCCCC2)C1C(C)C N1(C(Cc2ccc(C)s2)=O)CCC2CN(C(C3CC3(Cl)Cl)=O)CC2C1 S(=O)(=O)(c1cc(Br)ccc1Br)N1C(C(=O)NCCc2ccc(O)cc2)CC(=C)C1 c1(C(=O)NC(C)CCCOCc2ccccc2)cc(N)c(F)cc1F C12(NC(CN(C)CC)=O)CCC(CC1)N(C(=O)Cn1nc(C)cc1C(F)F)C2 C1(CC)CN(C(=O)CCC)CC1NC(=O)CCN(C)CCO N=c1[nH]cc(C(=O)NCC2(CNC(=O)CCC3CCCOC3)CCCC2)s1 C1(C(N(CCC2CC2)CC)=O)(OC)CCN(C(=O)CCc2conc2C)C1 c1(NC(CN(C)CC)=O)cccc(COc2ccc(CS(N)(=O)=O)cc2)c1 CCCCC(C(=O)NCC(C)N(C)C(C1CCC(=O)N1)=O)C(C)C C1(CC)CN(C(=O)C#CC(C)(C)C)CCC1CNC(C1CCCN(C(N)=O)C1)=O C#Cc1cccc(NC(=O)C(C2CCC2)NC(=O)Cn2cncn2)c1 N1(CC(=O)OC(C)(C)C)CCN(CC(=O)N(CCO)Cc2cccc(F)c2)CC1 C(=O)(CCCC(C)=O)N(CC(C)(C)CNC(c1cn(C2CCC2O)nn1)=O)CC N1(CC)CCCC(CNC(=O)C(C)(C)C2CCN(C(=O)CCc3ccco3)C2)C1 N1(C(=O)C2CC2)CCN(C(=O)C=CC2CCCO2)CC(CO)C1 CC1c2ccccc2CCN1C(c1cc2cc(Cl)ccc2s1)C(=O)NCC(F)F C1(S(C)(=O)=O)(C(=O)NCC(C)CNC(=O)C(C)(C)C2CCCO2)CCCC1 c1(C(N2CCC(OC)(CNC(c3cc(CF)on3)=O)C2)=O)cccc2nc(O)oc12 C(c1cccnc1)=CCOC(=O)C(F)n1ccnc1 C1(NC(Cc2nnc(C)s2)=O)CCC(C)N(C(C2CCCC(C)CC2)=O)C1 N1(C(CCC2CCCN(C(CCc3cc(C)no3)=O)C2)=O)CCC(F)C(F)C1 CC1(C)CN(C(c2cc(O)cc(O)n2)=O)CC1NC(=O)CC1CCCO1 CC1CCCC1(C)C(=O)NCCN(C(c1cncnc1C1CC1)=O)C1CC1 N1(C(C2CC(CCC)C2)=O)CC2(CCN(C(c3c[nH]cc3Br)=O)CC2)C1C(C)C c1(C(=O)NC2CN(C(c3ccc(NC)cc3)=O)CC23CC3)cc(F)c(Cl)cc1F CC1CN(C(c2cncc(N)n2)=O)C(C)CN1C(=O)CCc1cccnc1 c1(C(=O)NCC(CNC(=O)CC2OCCC2(C)C)OC)cnc2cc(C)nn2c1 CC(C)(CC(=O)NC1CCCCCC1NCC(=O)NC1CC1)C(F)F c1(C(N2C(CNC(C(COC)C)=O)CC(OC)C2)=O)cc2n(n1)CCO2 N1(C(C2(c3ccccc3)C(C)(C)C2)=O)CCCC(NC(C2CCCCO2)=O)CC1 Cc1csc(C(C)NC(=O)C(CO)NC(=O)Cc2cn(C)cn2)n1 C1(CNC(c2nc(CC)sc2)=O)CCCN(C(C2CC(=O)N(CC)C2)=O)C1 c1(C(N(CC(C)NC(C2(Oc3ccccc3)CC2)=O)C)=O)ncn2ccccc12 c1(C(N2CCC(NC(CC(C=C)C)=O)CC2C)=O)ccc2ncn(C)c2n1 Cc1nc(C(=O)NCC2(NC(=O)CN3CCC(C)C3)CCC2)c2n1CCCC2 Cc1nc2ccc(C(N3CC(O)C(O)C3CNC(C3CC3(F)F)=O)=O)cc2[nH]1 N1(CC(C2CCS(=O)(=O)C2)=O)CC(O)CC2(CCC2)C1 c1(C(N2CC(NC(c3c(CC)n[nH]c3)=O)C(CO)CC2)=O)ccc(Cl)c(F)c1O c1(C(=O)OCC)cc(C(=O)NC2CCN(CC(C)C)CC2)ccn1 C#Cc1cc(C(N2C(C(=O)NCC(F)C(C)(C)O)CCC2C2CC2)=O)ccc1C CCCC(C)(C)CN=c1[nH]c(C)cc(=NC2CCCN(CCO)C2)[nH]1 N1(C(C(COCC)C)=O)CC2(COC(CNC(=O)COC3CCC(C)CC3)C2)C1 C12(C(=O)NCC3C(CNC(C(CC)=CC)=O)C3)CCC(CC1)C2 c1(C(=O)NC(C2CN(C(CCCCCNC(C)=O)=O)C2)C)c(F)cc(F)cc1Cl N1(C(CC=C(C)C)=O)CC(NC(=O)CC2(C#N)CCCCC2)CC12CCOCC2 C1(CC(N2CC(N(CC=C)C)C2)=O)CCCN(C(C2(C)CCOC2)=O)CC1 CC1(C)CCCCC1C(=O)NC1(CO)CCN(C(C2CCCC(O)C2)=O)CC1 C1(C(=O)NCC(Cl)Cl)N(C(=O)CCCc2ncco2)CC12CCCC2 CN1CCCC1CC(N1CC(C)(NC(=O)CC2CCNC2=O)C1)=O c1(CSC)ccc(C(N2CCOCC2CNC(C2CC2c2nc[nH]n2)=O)=O)cc1 C=C(C)C(C)(C)C(=O)NC(C)CN(C)C(C1CSCN1C(c1cccs1)=O)=O C1(OC)CCCC(C(N2CC3CC3(CNC(=O)CC3CC(N(C)C)C3)C2)=O)C1 C1(CC(=O)NCCCCCC=C)C2CCC(C2)N1C(C1CC(C)N(C)C1)=O C1(C)(C(=O)NCC2N(C(CC=C(C)C)=O)CCC2)CC2CCC1C2 CCC(C)CCC(=O)NCCC(C)N(C(=O)CC(C)(C)O)C C1(C(=O)NCC(CNC(c2cnn(CC)c2C)=O)O)CCCC2(C1)CC2(F)F N1(C(C#CCNC(CCNC(COC)=O)=O)=O)CCC(C#N)(CC)CC1 N1(C(C)=O)CCCC(C2CCCN(S(=O)(=O)CCCN3CCCC3)C2)C1.C(CO)SCO CC(Cc1ccccc1)C(=O)NCCCC1(NC(=O)C(=O)NCC(F)F)CC1 c1(SC)ccc(C(=O)N(CCNC(=O)CCOC)CC2CC2)s1 CC(C)C(F)(CNC(=O)CC(C)C(F)F)C(=O)NCCN(C)C(=O)C1CC1 C1(NC(C2=NNC(=O)C2)=O)COC2C(NC(c3c[nH]nc3C(F)(F)F)=O)COC12 C1(C(=O)NCCCC(CO)NC(C(COC)(C)C)=O)CC2COCC2C1 S(=O)(=O)(c1cnc(NC(c2snnc2C)C)cc1C)N1CC(Br)=C(C)CC1 C=CC1(CC(N2CCC23CN(C(c2ccc(C4CC4)cn2)=O)C3)=O)CCOCC1 Cc1cc(-c2noc(CC3(C)COCCO3)n2)cc(O)c1 CC1CC(NC(C2CCC(=O)N2C)=O)CN1c1ccnc(Cc2ccccc2)n1 N=c1nc2c(c[nH]1)CC(C(=O)NC1(CNC(=O)C(O)CF)CCCCCC1)CC2 c1(C(N2CCC(CNC(C(C)NC(C)=O)=O)C2)=O)ccc(Br)c(Cl)n1 C#CCCC(O)CCNC(=O)Nc1cccc(Nc2ccc(OC)cc2)c1 Cc1nc2c(s1)CCCC2C(=O)NCC1CCC1NC(=O)CCCCC(C)(C)C CCS(=O)(=O)CC(=O)N1CCC(O)C(C(=O)Nc2ccc(OC(C)C)cn2)C1 N1(C(CC2C(C)OCC2)=O)C(C(=O)Nc2cncc(C3CC3)c2)CC2CCCC12 c1(C(=O)NC2C(NC(c3nccc(C)c3N)=O)CCC2)ccc2c(c1)C(=O)NC2 Cc1cc(-c2nc(CC3CCCCN3C)nn2C2CCOC2)nc(C(F)F)n1 C1(C)CCN(C(=O)CCNC(c2n(CC)nnn2)CC2(C)CC2)CC1.C(C)(C)S N1(C(C2C(CNC(c3cc(CO)on3)=O)CCCC2)=O)CCC12CCCOCC2 C1(NC(CCOCC#C)=O)CN(C(C2(C)CC2)=O)CC1O N1(C(COC(CC)C)=O)CCC2(CCC(NC(=O)C3CCN(C)CC3)CC2)C1 CCC(C(=O)NCC1CN(C)CCN1C(=O)C(C)C(=O)OC)C(C)O c1(N2CCC(F)(C(F)(F)F)C2)nc(NC2CC3CC4C(C3)C24)nc2ccccc12 Cc1cc(CC(=O)NCC2CC(NC(C3CCCC3(F)F)=O)C2)cc(F)c1 c1(C(=O)NCC2CC(CNC(c3cnc(S)nc3)=O)OC2)cc2c(o1)CCCC2 c1(CC)ccc(O)c(C(=O)NC2CCCC(NC(c3cc(C)nc(O)n3)=O)C2)c1 C(N=c1[nH]c2c(F)cccc2o1)C1CCCC(NC(C(c2cn(C)nc2)O)=O)C1 C(=O)(CC(C)C1CC1)N(CCC(C)NC(c1ccns1)=O)C Cc1ccccc1C(C)NC(=O)CC1C2CN(C(C3CCSC3)=O)CC12 CN1CCC(C(=O)N(C2CC(NC(=O)CS(N)(=O)=O)C2)C)CC1 N1(C(C(CC)(C)O)=O)CC2CC(NC(c3ccnc(S)c3)=O)CC(C2)C1 N1(CCNC(CN(CC#C)C(c2nnsc2C)=O)=O)CCCCCC1 c1(OC)cccc(C(=O)NCC(CNC(C2(n3nccn3)CC2)=O)OC)c1C n1(CC(=O)NC(CC)CN(C(=O)CCn2cc(Br)cn2)C)cnc(C#N)n1 O=C(NNc1cccc(Cl)c1Br)C1CCCC2(CCNCC2)O1 N1(C(c2cnc(SC)s2)=O)CCN(C(c2ccc(C)nc2N)=O)CC1CC(F)F C1(OCC)CN(C(=O)CC(=O)Nc2cncc(F)n2)CC1c1nccn1C c1(CC)ncc(Cl)c(C(=O)NCC2(NC(=O)Cc3ccnc(C)c3)CCOC2)n1 N1(C(C2C(=O)NCC2)=O)CC2(CC(C(=O)Nc3ccc4nccn4c3)CO2)C1 C1(NC(C=C(C)C2CCCCC2)=O)CCSC12CN(C(=O)C(C)(F)C(C)(C)F)C2 c1(C(=O)NC2C(CNC(C3C(C(C)C)(CC)C3)=O)CC2)cnc(C(F)(F)F)s1 n1(C(C(=O)NCC2(CNC(=O)CO)CCC2)C2CC2)nnnc1C1CC1 C1(C(N2C(CNC(c3ccc(OC(F)F)nc3)=O)CC2)=O)CCCCCS1(=O)=O C1(CC)(CC)CC(NC(=O)CCF)CN1C(=O)C(n1cc(C)cn1)C S(=O)(=O)(CC(=O)NCC1CC(CNC(=O)CCCN(C)C(C)C)C1)NC N1(C(=O)OC(C)(C)C)CCCC12CCCN(C(c1cc(=O)n3ccsc3n1)=O)C2 C1(C(=O)NC2CC(F)(CNC(c3scc(OC)c3)=O)C2)CCn2c(C)cnc2C1 c1(C(=O)NCCC2C=CCC2)coc2c1CN(C(c1cnsc1)=O)C2 C#CCCCCC(=O)N1CC(O)(C(C)NC(=O)COC(F)(F)F)C1 C=CC(C)(C)C(=O)NC1CCOC1C1CCN(C(C2CNC(=O)N2)=O)CC1 c1(CC)cnc(C(=O)NC(C)(C)CCNC(c2cc(C#N)c[nH]2)=O)cn1 Cn1cncc1C(CNC(=O)CNC)NC(C1(CSC2CCCCC2)CC1)=O C1(C(C)C)CN(C(=O)CN2CCN(C)C(=O)C2)CCN1C(=O)CN1CCCC1=O C1(C(=O)NCC2C(C)CCN(C(COC(C)C)=O)C2)CCc2nncn2CC1 C1(C)(C(N(C(C)CO)C)=O)CCCN1C(=O)Cn1cnnn1 C1(NC(C2C(CN)CN(Cc3ccccc3)C2)=O)CCC2CC2CC1 N1(c2c(Cl)cnc(OC)n2)CC(NC(c2ccc(Cl)c(F)c2)=O)CC2(CCC2)C1 c1(C(=O)NCC(CC=C)NC(=O)COC)c(F)cccc1[N+](=O)[O-] C(C(C)(C)CNC(=O)Cn1cnnn1)N(C(=O)COC)CC c1(C(N2CCCC(C)(COC)C2)C(=O)NCCC)cc(Br)ccc1OCCOC Cc1c(C(=O)NC2COCC2CNC(=O)CSC(F)(F)F)cnc2ncnn12 C(=O)(C(C)N=c1ccn(Cc2ccc(Cl)cc2Cl)[nH]1)N(CCC)CCOC c1(OC)ncc(Cl)cc1NC(c1cncc(NC(=O)CC#N)c1)=O c1(CC(=O)NCCNC(c2snc(O)c2Cl)=O)ccc2c(c1)CCC2 CC(CC#N)C(=O)N(CC(C)NC(c1ccc(C(=O)NCC2CC2)cc1)=O)C C1(N(C)C)CCC(C(=O)NCCCC2CN(C(=O)COCCF)CCO2)CC1 C#Cc1ccc(N(C)C(N2CCCC2c2ccc(C)c(Br)c2)=O)cc1 C1(C(N2CCC(O)(C(C)NC(c3csc(C)n3)=O)C2)=O)(OC)CCCCCCC1 c1(NCC(CNC(COCC)=O)NCCOCCO)nc(C(F)(F)F)ncc1Cl C(=O)(CC(C)(C)C)NCCCN(C(C)C)C(C1CC2(CSC2)C1)=O N1(C(CCCCSC)=O)CCCC(C)(NC(=O)CC2CCCOC2)C1 C(c1cc(Cl)c2c(c1)OCO2)=CC(=O)NC1C=CCN(C(C(CN(C)C)O)=O)C1 CN1C(=O)CCCC1C(N1CCN(C(=O)Cn2cc(Cl)cn2)CC1CF)=O c1(OC)c(CNC(=O)NCCCCC2(C)NC(=O)NC2=O)ccnc1Cl Cc1c2c(-c3cnc4n[nH]c(C(=O)Nc5cnoc5)c4c3)cccc2nn1C C1(CCC(=O)NCC(COC)O)CCCN(C(c2ccc(Cl)o2)=O)C1 c1(OCC)cc(C(=O)N(C(C)(C(=O)NCC(C)(C)O)C2CC2)C)on1 c1(C(=O)NCCOC2CCN(C(C3C(C)(C)C3(C)C)=O)C2)ccc2c(c1)CCO2 c1(-c2occ(C)c2)nc(COC(C)C)nn1CC1CC1C CC(=Cn1ccnn1)C(=O)NC1CCCC1CNC(c1cn(C)c(=O)nc1O)=O C(=O)(C(C)CCC(C)(C)C)NC1C(OC)CN(C(CC)=O)C1 C1(C(=O)NCCC(CC)C)N(C(=O)CN(C2CCC2)C)CCCC1(C)C C1(C(=O)NCC2N(CC)CC2)CCCN(C(c2cc(C)nn2C)=O)CC1 C1(NC(Cc2c(C)scc2)=O)COC2(C1)CN(C(c1ccc3nc[nH]c3c1)=O)C2 c1(OC)cc(C(N2CCC(C(=O)NCc3cncn3C(C)C)(CO)C2)=O)nn1C c1(C(N2CCC(n3cc(C=CC(C)C)nn3)CC2)=O)ccc2c(c1)NCC2 c1(OC)cc(C(=O)N(CC(C)(C)C(=O)NCCc2cn(C)nn2)C)ncn1 c1(C(=O)NCC(C(C)C)(C)NC(=O)Cc2cscn2)ccc(Cl)c(C#N)c1 c1(NC(C2COCCN2C(=O)CCc2ccco2)=O)cc(O)ccc1Cl C1(C(=O)NC(CC(C)NC(c2cc(C)sc2)=O)C)(C(F)F)CCOCC1 N1(C(C(CCF)NC(CC)=O)=O)CCC(C(F)(F)F)C1(C)C CC1(C)CCC(CNC(=O)CC2(C)CCN(C(C3(c4cc[nH]n4)CC3)=O)C2)CC1 C1(CC(=O)NC(CNC(C2(C)COC2)=O)(C)C2CC2)CCC(F)(F)C1 c1(C(C(=O)NC2CCOC2)N(CC)CC2CCC2)c(Br)cnn1C n1(CCNC(N2CC(OCCO)C2)=O)ncc2ccccc12 c1(CC)cccc(F)c1C(=O)NCC1(NC(c2ncccc2N)=O)CCC1 N1(C(N)=O)CCCC(C(=O)NCCCOCCNC(=O)C(O)c2ccsc2)C1 N1(C(=O)Nc2cc(SCC3CCCC3)ccn2)CCOCC1c1cccc(F)c1 c1(OC)ccccc1CCC(C)NCc1nnc(CC(C)C)n1C c1(C(N2CC(NC(c3n(C(C)C)ncc3)=O)C(O)C2)=O)ccc2c(c1)CC(C)O2 CC(=O)CCCCC(=O)N1CCC=C(C(=O)NC2CCCC2N=[N+]=[N-])C1 Cc1nccn1CCCC(=O)N1CC(CCNC(c2cn(C)cn2)=O)C1 c1(C(=O)NC2CN(C(=O)C#CC3CC3)CC23CC3)cc(F)c2c(c1)CCC2 C1(COCC(=O)NCC2(CNC(C3(C)COC3)=O)CCC2)CCCCO1 c1(CC(C)C)nnc2c(C(=O)NCCC3(NC(=O)C(C)O)CC3)cccn12 N1(CCC(=O)Nc2c[nH]c(CN3CCCC3)c2)CCNC(=O)C1 c1(OC(C)C)ccc(F)c(F)c1-c1cccc(NCc2cc(F)cc(Cl)c2)n1 c1(CC)ccccc1NC(=O)CCN(C(=O)CC1CC2(CC2)CO1)CCO N1(C(C(CCOC)NC(c2cc[nH]c(=N)n2)=O)=O)CC2CCOC2C1 C1(CNC(C2(COCC)CC2)=O)(CO)CC12CCN(C(=O)C(C)(F)F)CC2 CC(C)C(C)C(=O)N1CCC(OCCNC(c2cnc(S)n2C)=O)C1 N#Cc1cncc(CNc2nc(Cl)ccc2C(=O)NCCc2cccnc2)c1 c1(C(=O)NCC(C)(C)NC(CCC(=O)NCC)=O)ccc2nc(S)[nH]c2c1 N1(C(CC2C(C)CCO2)=O)CC(CO)C2(C1)CN(C(=O)Cc1ccno1)C2 CN1CC(CN(C2(C)CN(c3nnnn3Cc3ccco3)C2)CC(=O)O)CC1=O Cc1cnc(C(N2CCN(C(c3ccn(C4CC4)c3C)=O)C(CF)C2)=O)c(F)c1 CC1CCCN(C(=O)Cc2csc(S)n2)C1CNC(C1(CCF)CCC1)=O C1(C(=O)NCC2(F)CC(NC(C(C)n3cccc3)=O)C2)CC2CC(O)CC(C1)C2 N1(c2nccc(N(CCC)C)n2)CCn2ncc([N+](=O)[O-])c2C1 C1(C(=O)NCC2(F)CN(C(C3CC3C)=O)C2)(OC)CC(C)C1 c1(C(=O)NC2C(NC(Cc3nn(C)c(Cl)c3)=O)CCC2)nc2n(c1Cl)CCCC2 N1(C(C(C)=C(C)C)=O)CC2(CCCN(C(=O)CC3CC(O)C3(C)C)C2)C1 C1(NC(c2nnnn2C)C(C2CC2)OCC)CNCC1CO C1(CNC(=O)CC2C=CCCC2)C2CCC(C2)N1C(c1csc(C2CC2)n1)=O C1(NC(Cn2c(C)nnn2)=O)CCC2(CCCN(C(c3cn[nH]c3)=O)C2)C1 C(=O)(CCCCCCS(N)(=O)=O)NC1CN(C(C(CC=C)CC(C)C)=O)CC1C CC(C#N)C(=O)N(CCC(=O)NCCOc1ccccc1)CCCO C1(NC(C2(OCC)CCC2)=O)CN(C(C2CC(CC)C2)=O)C(C)(C)C1 C(c1ccc(F)cc1F)=CC(=O)NCC(C)N(C)C(c1n[nH]cc1[N+](=O)[O-])=O N1(C(c2c(C)cns2)=O)CC2(C)CN(C(c3coc(O)n3)=O)CC2(C)C1 C(=O)(C1COc2ccccc21)N1CCC(NC(C=COCC)=O)C2(C1)CCC2 C#Cc1cnc(C(=O)N(CCCN(C)C(c2ccc(N)cc2Cl)=O)C)c(C)c1 C1(CNC(COCCC=C)=O)CCC2(CCC2)C1NC(C1C2(CC2)C12CC2)=O c1(OCC)ccc(Cl)nc1C(N1CCC(COC(=O)CCC(C)C#N)CC1)=O N1(C(c2cnc(OCC)nc2)=O)CCC2CCCC12CNC(=O)C(C)(C)F C=CC(CC)C(=O)NC(CC(=O)OC)C1CCC1.C12CCCN1C(=O)C1CC21 C1(C(=O)NCc2scc(C)n2)C2CC3C(C2NC(=O)CN2CCSCC2)C13 C1(C)(CNC(CNC(=O)OC)=O)CCCN(C(=O)Cc2ncc[nH]c2=O)C1 Cc1onc(C(N2CCCC2C(=O)N(CCCO)C(C)C)=O)c1C c1(C(N2CCCC(C(C)NC(c3cccc(CF)c3)=O)C2)=O)ccc(Cl)nc1Cl CC1(C)CN(C(=O)C2=CCC2)CC1NC(=O)CC1CC2(CCC2)CO1 C1(C(F)(F)F)(NC(=O)NC2C(SC)CCC2)CC(F)(F)C1 c1(CN2CC(C)(C(=O)NCc3ccc(C)cc3Cl)C2)c(O)cc(Cl)cc1Cl S(=O)(=O)(c1cc([N+](=O)[O-])ccc1C#N)NCCc1nnc(C(C)C)s1 CC1(C(N2CC(N3CCNCC3)C2)=O)CCN(C(=O)C(Cl)Cl)C1 CC(C)(C(=O)N1CC2CC2(CNC(c2ccsc2C(F)F)=O)C1)S(=O)(=O)C1CC1 C1(CNC(c2n(C(C)C)ccn2)=O)(CO)CCN(C(C2CN(C3CCC3)C2)=O)C1 Cc1cc(C(=O)NC(C)C(C)C(=O)N(C)CC2CC2)cn1C C(=O)(C(CC(C)CC)NC(c1c[nH]c(C)c1)=O)Nc1cc(CC)cc(O)c1 C1(C(N2CC(C(C(=O)N(CC(O)CO)CC)O)C2)=O)CC(C)(F)C1 c1(C(C(=O)NC(C)C)N(CCC)Cc2cccnc2)nn(C)cc1I C1(C)(OCCN(C)CC)CCCN(C(=O)CCc2ccc(C3CC3C)o2)C1 c1(C(=O)NCC(CNC(C2CC(CCC)C2)=O)(C)C)cc(Br)cc(C)c1C C1(C2CCN(C(C3CC3F)=O)CC2)(NC(COC(CC)C)=O)CC1 N1(CCN(C)Cc2cn(C3CC(C(=O)O)C3)nn2)CCOC(CCC(=O)OC)C1 c1(C(=O)OC(C(=O)OCC)CCc2ccccc2)sc2nc(C)nc(C)c2c1C c1(C(N2CCC(n3cc(CNC(C(C)OC)=O)nn3)C2)=O)cccc(Cl)c1OC N1(c2cc(C(=O)OC)nc(C)n2)CCCC2(NC(=O)CC3CCCN3C)CC2C1 c1(OC)cc(C(N2C3CCC(C3)C2C(=O)Nc2cn(C)nc2C)=O)cc(Br)c1Cl N1(C(C2(NC(C3C(C(C)C)OCC3)=O)CC(F)(F)C2)=O)CCCC(C)C1C C1(NC(=O)CCCN2CCCC2)CC2(C1)CC2C(=O)NCc1ccc(Cl)s1 C(CC(C)CCNC(=O)C(C)(C)N1CCC1)NC(C=C(COC)C)=O C1(C(=O)NCc2ccc(Oc3cccnc3)c(F)c2)NCCC12CC2(F)F c1(OC)nc(C)c(C(=O)N(C2CCCC(Oc3ccccc3)C2)C(C)C)s1 Cn1cnc(Cl)c1C(c1nnnn1C(C)(C)C)NCc1nnc(C(F)F)s1 c1(C(=O)NC(C(C)(C)NC(c2cnc(OC)s2)=O)C)ccc2c(c1)CC(=O)N2 Cc1ccc(C(=O)NCC2CC2NC(=O)C(=O)Cc2ccccc2F)c(C)c1 N1(C(c2cc(O)ccc2F)=O)CCN(C(=O)C#CC2CC2)C2(CC2)C1 N1(C(C2=CCC(C)CC2)=O)CCC2C1CCCN2C(=O)CCC1(C)CC1 CC(C)C(C)C(=O)NC(CC1CCOCC1)C(N1CC=CC(O)C1)=O C(=O)(C1CCc2ccccc21)NC1CN(C(C(CSC)(C)C)=O)CC(F)(F)C1 N1(OCCSc2ccc(N(C(=O)CC3CCCO3)C(C)=O)cc2)CC(S(C)(=O)=O)C1 c1(C(=O)OC)sc(CN(C(=O)C(F)CCNC(c2ccccc2)=O)C)nc1C C(CCC(C)C)(C(=O)N1CCCC1C(=O)Nc1cccc(I)c1)NC(C)=O c1(CN=C(NCC2(OC)CCOC2)NC(C)C2CC2)cc(C)cnc1O c1(C(N2C(CNC(=O)Cn3cc(C4CCOC4)cn3)CC2)=O)ccc(F)cn1 Cc1cn2c(n1)C(C)CC(C(=O)NCCCCCCN(C(=O)C(O)C(C)C)C)C2 N1(C(C2(O)CCN(Cc3c(C)scn3)C2)=O)CC2COCC2C1 C12(CC)CCC(C(=O)NCCOC3CCN(C(C4CC4C#N)=O)C3)(CC1)CO2 C1(CN(C(=O)CCCN2CCCCC2)CC)CCCN(C(=O)C(C)C(=O)OC)C1 C1(NC(C(CC)C2CCOCC2)=O)C2CN(C(c3ccc(N(C)C)nn3)=O)CC12 C1(N(C(C2CC(C)OC2C)=O)C)CCCN(C(=O)Cn2ncc(O)nc2=O)CC1 C(C)(C(C(=O)N1CCC2(CSC2)C1)C(C)C)NC(c1c(CC)n[nH]c1)=O c1(CC(=O)NC2CN(C(c3cccnc3S)=O)C2)cnc2ccccc2c1 c1(C(=O)NCC2CC3N(C(C(C)SC)=O)C(CC3)C2)ccc2c(ccn2C)c1 N1(C(C#CC(C)C)=O)CCC(CNC(C2C3COCC23)=O)C12CCC2 C#CCC(C(=O)N1CC(O)CC1CO)NC(=O)CNC(c1ccco1)=O C=C(CNC(=O)CCN(CC(C)C(C)C)C)CCNC(=O)CN(C)C(N)=O CS(=O)(=O)CCC(=O)N1CC=CC1C(N1CCC(C(F)F)C1)=O c1(N(C)C)ccc(C(=O)NCC2CCC(NC(c3cnsn3)=O)C2)cc1F Cc1cn2c(=O)c(C(=O)NCC3CC(NC(C4COC(C)C4)=O)C3)cnc2s1 C(C(=O)OCC)(C(C)C)OCC#C.c12noc(c1C)C(=O)OCC2C N1(C(C2CC(n3cnnc3)C2)=O)CCC2CCCC(C1)N2C(C1CCCO1)=O c1(NC2(C)CN(C(C(C)(C)NC(=O)NCC(=O)OCC)=O)C2)cccc(F)c1O c1(C(=O)NCc2ccc(CCNC(=O)C(O)C3CCC3)cc2)cncc(Cl)c1Cl C1(OCC)CN(C(c2nnn(C)c2C(F)F)=O)CC1CNC(=O)CO c1(C(N2C(C)CC(CNC(C(CC)(F)F)=O)C2)=O)ccc2c(n1)CCO2 C#Cc1cnc(NCC(C)(CC(C)C)NC(c2cc(C(C)C)nc(O)c2)=O)nc1 C(C)(C(=O)N1CC(CCNC(=O)CN2CCOC2=O)C(C)C1)(C(C)C)NC(C)=O c1(C(=O)NC2CCC(CCNC(COC)=O)C2)cc(C(N)=O)ccc1N c1(NCc2cc(CC)no2)ccc(S(=O)(=O)NC(c2ncccc2Cl)C)c(Br)c1 n1(CC)nncc1C(N1CCC1CNC(c1cnn[nH]1)=O)=O N1(C(c2n(C)nc(O)c2)=O)C2CCC1C(F)C(NC(=O)CCCCC(C)(C)C)C2 N1(C(C(C)=C(CC)C)=O)CCC(C)(C)C1C(=O)NCC(C)F c1(C(=O)NC(C2(O)CN(C(c3ccc(C)n3C)=O)C2)C)cn2c(n1)CCC(C)C2 c1(C(=O)NC2CN(C(C3(OC)CCC3)=O)CC2C(F)F)sccc1S(N)(=O)=O C12(CNC(C=CC(CC)C)=O)COC(CN(C(=O)C=CC3CC3)C3CC3)(C1)C2 CC(CNC(=O)CCCC1CCCC1)CC(=O)NCC1(O)CCN(C)C1 Cc1cc(O)ccc1NC(C1CCN(C(=O)Cc2cccs2)CCO1)=O Cc1cc(C(C)C)ccc1C(=O)NC1COCCN(C(C2C(C)C2C)=O)C1 N1(C(Cc2ccc(C)o2)=O)CCC2CC(CNC(=O)CCF)CCC2C1 c1(C(=O)NCC2(n3cnnn3)CC2)cccc(CNC(C23CCCCC2C3)=O)c1 c1(C(=O)NC(C)CN(C(=O)C(F)C2CCOC2)C)ccnc(SC(C)(C)C)c1 c1(C(=O)NC(CC=C)CNC(C2CC2C(=O)OC)=O)cccc2c1OCCC2 C(=O)(CC(O)C(C)C)NC(C(=O)C(CSCCC#C)=O)CN(C)C.N Cc1cc(C(N2CC3CC2CN3C(C2(F)CC=CCC2)=O)=O)ccc1O C(=O)(C(C)n1cncn1)NCCCN(C(=O)Cn1ccnn1)CCC Cc1cc(CC(=O)NCC(C)N(C(=O)CSc2cnn(C)c2)C)cc(F)c1 c1(NC(=O)NCc2ccc(C(F)(F)F)nc2)ccc2n[nH]cc2c1 Cc1noc(C)c1CN(C)C(C1CCN1C(C1CCCS1=O)=O)=O CCC(CC)(CCC(=O)N(C)CCNC(C1CNC(=O)C1)=O)[N+](=O)[O-] C(C(F)(F)C(=O)N1CCCC(CC(=O)N(C2COCC2O)C2CC2)C1)OC C=CCCCC(C(=O)NC1(COCC)CC1)NC(c1cc(C)cc(F)c1)=O CCC1=C(C(=O)N2CCCC(NC(C3(C(C)C)CNC(=O)C3)=O)C2)SCCO1 C1(CNC(C2C=C(C)CS2)=O)CC(NC(c2cc(C)c(C)o2)=O)CCO1 N1(C(CC(CC)CC)=O)CCCC(C2CCN(C(c3csc(F)c3)=O)C2)C1 c1(C(=O)OC)cc(F)c(C(N2CC=CC(NC(C3CCCN3C)=O)C2)=O)cc1F C(C(C)(O)C(F)F)NC(CCOCCN(C)C(C1CC=CC(O)C1)=O)=O C(=O)(C1=C(Cl)CCOC1)N1CC(C)CC(C(=O)NC(C2(O)CCC2)C)C1 N1(CC(O)CC2CCCC2)CCOC2C(O)CC12 c1(CC(=O)NC(C2(CNC(C=CSC)=O)CC2)C)ccc(-n2cccn2)cc1 C(C)(CCCCNC(=O)COc1ccsc1)NC(C(C)OCCC#C)=O C1(C(=O)NC2C(CNC(C(C(CC)C)N(C)C)=O)CC2)CC2(C1)CC1(CC1)C2 CCCC(CNC(=O)C(F)CCC(=O)OC)C(=O)NCCC(=O)NC NS(=O)(=O)c1c[nH]c(C(=O)NC2CC3CC2N(C(c2ccccc2CO)=O)C3)c1 C(C(=O)NCC(O)CNC(c1cc(C2CCC2)nn1C)=O)(C(C)(C)C)N(C)C N1(C(c2cnc(CS(C)(=O)=O)s2)=O)CC2(C1)CN(C(C1(C(F)F)CC1)=O)C2 N1(C(COc2cccc(C)c2)=O)CCCC2(NC(c3nc(Cl)sc3C)=O)CC2C1 N1(C(=O)CC2CCC3CC23)CCC(C2CC2)C1CNC(=O)C(O)(C1CC1)C1CC1 C1(=CC(=O)NC2C=CCN(C(C3CC(N(C)C)C3)=O)C2)CN2CCC1CC2 N1(C(C2(NC(C)=O)CC2)=O)CCC(C)(C)C(CNC(=O)CC2(C#N)CC2)C1 CC(C)CC(F)C(=O)N1CCC(CN(C)C(c2cnn(CCO)c2N)=O)C1 C1(CC)(NC(=O)Cc2ccc(C(C)=O)s2)CCCN(C(c2ccnc(C)c2C)=O)C1 N1(C(c2sncc2C)C(=O)Nc2ccc(C(=O)OCC)cc2)CC(C)(C)CC1C C1(C(N2C(C3(O)CN(C(C=C(COC)C)=O)C3)CCC2)=O)CCC(F)CC1 CC(C)CC(C(N)=O)N(C(=O)C(C(C)(C)C)NC(=O)CC(C)n1cccc1)C N1(C(C(CC)OC)=O)CCOC(CCCNC(=O)CCc2ccoc2)C1 N1(C(CCc2cnc(C)o2)=O)CCN2CCN(C(=O)C=C3CCCCC3)CC2C1 c1(C(N2CCN(CC(=O)NCCC(C)(C)O)C(=O)C2)=O)ccc2[nH]ccc2n1 C1(CC(N2CC(NC(=O)Cc3ncc(Cl)s3)C2)=O)CCCCCC1(F)F Cc1cnncc1C(N1CCC(C2CCCN2C(=O)CCc2ccco2)C1)=O C1(C)(C(=O)NCC(CC=C)NC(=O)C=CC=CCC)CCCC1(F)F CC(O)C(C(=O)N1CCOC(CC2CC2)C1)NC(=O)C(O)CC1CCCC1 S(=O)(=O)(c1ccc(C)c(C)c1)NCC(=O)NCc1c(F)ccc(C#C)c1 CCC(CC)CCCC(=O)N1CC(CC(=O)NC2CC(C(C)O)C2)CC1C C(=O)(CC(C)(F)F)NC(CC1CN(C(CCNC(=O)NC)=O)C1)C Cc1nc(NCc2coc(C)c2)cc(=NCc2c[nH]nc2C(C)(C)C)[nH]1 c1(C(N2CCC(CNC(c3ccoc3)=O)CC2)=O)cc(Br)cnc1Br c1(C(CC)C)nc(N2CCC(NC(=O)C(F)F)C(C)C2)cc(C)n1 C1(O)(CNC(=O)C2CC2)CCN(C(C2C(c3ccccc3)C2(F)F)=O)C1 C1(CNC(C2(C)CC(C)C2)=O)CCN(C(=O)CCCn2cccc2)C(C)C1 c1(CC(=O)OCC)ccc(C(=O)NCC2CCC(C)O2)cc1.c12cn(nn1)C2 c1(NC(=O)NCC2N(CC)C(=O)CC2)cc(C)c(F)cc1I CCC(C)CCC(=O)NCCC1CC(NC(c2ncccc2C2CC2)=O)C1 c1(OC)cc(C(=O)N(C)CC2CCN(C(C3CCCC(F)C3)=O)CC2)ccc1F c1(C(=O)NCC2CC(NC(c3ncn(C)c3)=O)C2)cc2n(c1)CCC2 C(=O)(C1=NNC(=O)CC1)N1CC(NC(=O)CCCN2CCOC2=O)C(O)C1 N1(C(C2C(C)(C)C2)=O)Cc2nccn2CC(NC(C23CC2C3)=O)C1 C1(NC(c2ocnc2C(F)F)=O)CC2CC(NC(c3nncs3)=O)C1C2 CC1CC(C)N(C(c2cccc3nsnc23)=O)CCN1C(c1ccccc1Cl)=O c1(CNC(CN(C(c2cc(CC)no2)=O)CC)=O)ncc(C)cc1C N1(C(CNC(C(C=CC)O)=O)=O)CCN(C(=O)C(c2cccc(OC)c2)O)CC1 C(C(C)(C(=O)NCCCC1CN(C(C)=O)CCO1)OC)OC Cc1cccc(C(=O)NCc2ccc(C(N3CC4CCC3C4C(=O)O)=O)o2)c1F N1(C(C=C(CNC(c2c(OC)nsc2)=O)C)=O)CCC2(CC1)N=N2 C(c1cn(C)cn1)=CC(=O)NCC1(CC(=O)N(C(C)C(C)C)CC)CC1 S(=O)(=O)(c1ccccc1Cl)N1CC2C(CNC(c3cc(Br)ccc3F)=O)(C2)C1 c1(C(=O)NC2(CCC)CCN(C(C3CCC(C)O3)=O)CC2)ccn2nccc2c1 C1CCCCn2cc(nn2)CC1.N1(C(C2CC2c2cccs2)=O)CCCCC1 C(=O)(C1=CCC(C)(C)CC1)N1C(CNC(C2N(CC)CCOC2)=O)CC2CC21 c1(SC)ncc(C(=O)NC2(CO)CN(C(=O)C(C)Cc3ccccc3)C2)s1 C1(C(=O)NCC2CCC(NC(CC(C)(C)OC)=O)CC2)Cc2cccc(C)c2O1 N1(C(C2CCC(COC)C2)=O)CC2CCC2(NC(=O)CCCc2nc(C)cs2)C1 N1(C(c2c(SC)scc2)=O)CCCC(C)C1CCNC(=O)C(F)(F)C(F)F c1(C(=O)NC2(C)CC(NC(=O)CO)C2)ccccc1OOC(F)F.C1CCCO1 c1(C(=O)NC(C)CNC(c2cccc3c2COC3)=O)ccc2nc(O)cn2c1 N1(C(C2N(C(c3cnc(CC)nc3)=O)C3CCC2C3)=O)CCOc2ccccc21 c1(C(=O)NCC(CC)NC(C2CS(=O)(=O)C2)=O)c(C)ccc2nsnc12 c1(C(=O)NCCC2CCCOC2)coc2c1CN(C(c1cc(O)cc(=O)o1)=O)C2 C1(NC(Cc2c(C)noc2)=O)CC2CN(C(C3(C(F)F)CCOCC3)=O)CC12 c1(C(C)C)ccc2cc(C(=O)NC3CCCC3CNC(C3COC3)=O)ccc2c1 c1(C(N2C(C(=O)NC(c3ccn(C)n3)CC)CC2)=O)nccc2cc[nH]c12 n1(CC(=O)N(C2CCCN(C(=O)C(=O)N(C)C)C2)COC)ncc(C)cc1=O c1(SC)c(C(N2CCC(NC(=O)C(C)SC)C2C)=O)ccc2c1OC(F)(F)O2 c1(C(N2C(CS(CCOCC)(=O)=O)CC(OC)C2)=O)cc2n(c1)CCOC2 C1(NC(C2CCC(C)N(C(C3CC(=O)C3)=O)C2)=O)CCC(=O)N(C)C1=O N1(C(C2C(C)(C)C2(F)F)=O)CCOCC(C(N2CCC(n3ccnc3)C2)=O)C1 C(=O)(C(C1=NOC2CC12)N1CCN(CCO)C(C)(C)C1)NCCCC c1(NCc2c(Br)cn(CC)n2)ccc(S(=O)(=O)NC2(CO)CCOCC2)cc1Br c1(C(c2nnnn2CCCF)NC2(C=C)CCC2)cccc(OC)c1Cl N1(C(c2cc(CC)nn2C)=O)C2CCC1CC(NC(c1ccnn1C(F)F)=O)C2 C#CCC(C(=O)NC)NC(=O)CN(CCC)C(C1CCCCS1)=O c1(CC(N2CC3C(NC(C(N4C(=O)CCC4=O)C)=O)(C3)C2)=O)cc(F)ccc1F c1(C(=O)O)ccc2[nH]cc(CNC(c3ccc(C4NC(=O)NC4=O)cc3)=O)c2c1 C1(C(=O)NC2C(CNC(C(C)(C)NC(=O)NCCC)=O)CCC2)CCN(C)C1=O N1(C(CNC(N)=O)=O)CCC2(NC(c3ccc(F)c(CO)c3)=O)CCCCC12 C(CCC(=O)NCC(F)CNC(=O)C(c1ccccc1)N(C)C)N(C(=O)OC)C Cc1ccc(CC(=O)NC(C)CN(C(=O)CCCc2cccs2)C)cc1O N1(C(CCn2ncn(C)c2=O)=O)CCC2CCC12CNC(=O)C#CC(C)(C)C C1(NC(c2cnc(S)n2-c2ccccc2)=O)CN(C(=O)C2CC2)C2(CCC2)C1 C(CO)(CC(F)(F)F)NC(CCC)C(c1nnnn1C1CCCCC1)OCC c1(CCC(=O)N(C2CCN(C(C(CC=C)C)=O)C2)C)ccc(Cl)c(OC)c1 Cc1cc(C(N2CCCC(C(C)C(=O)NCC3(O)CC(C)(C)C3)C2)=O)cnn1 c1(NC)nc(C)ccc1C(N1CCCCC1CNC(=O)Cc1nncs1)=O Cc1cc(C(=O)NCC2(NC(c3ccns3)=O)CCOCC2)[nH]c1C c1(CC(C)C(=O)NCC(C2CC2)NC(C2CCOC2C)=O)ccc([N+](=O)[O-])cc1 c1(C(N2CCC(CN(C(CCOC(C)=O)=O)C)C2)=O)ccc2c(c1)CCCO2 c1(SC)ccc(O)c(C(N2CC3C(CNC(=O)CCc4cccnc4)C3C2)=O)c1 N1(C(c2cn(C3CC3)cn2)C(=O)NCC(C)C)CCC(NC(C)=O)CC1 c1(C(N2CC(C)N(C(c3sccc3C(F)F)=O)CC2)=O)cnc2ncc(Cl)cn12 N1(C(C2(CO)CC(C)(C)C2)=O)CC(NC(=O)C2=COCCO2)CC(F)C1 C1(C2CCC2)(C(N2C(CCNC(CCc3nc(C)sc3)=O)CSCC2)=O)CCC1 c1(N(CCCNC(C(C)OCc2cccc(C)c2)=O)C)cc(Cl)c(O)nn1 N1(C(C(C(C)C)C)=O)CC2CC3CC2C1C3NC(c1nnc2ccccn12)=O C1(O)(C(C)(C)C)CCN(C(=O)C(=O)NCCCOC2CCC2)CC1 C1(COC)(CNC(C2(C)CCOC2)=O)CCCN1C(=O)Cc1ccccc1Cl CC1CCN(C(c2cc(=O)cc[nH]2)=O)C(CNC(=O)C(C)n2ccnn2)C1 CC1CC(C(N2CCCC(N(C)C(C3CCS(=O)CC3)=O)CC2)=O)CC(C)(C)C1 C1(NC(c2c(COC)nn[nH]2)=O)CC(C2CCN(C(C3SCCCS3)=O)C2)C1 CCCCCC(C)(CC)C(=O)NCC(CC)(CC)NC(=O)CC(O)CCSC CC(C)(CC(=O)N1CCC(CC(F)F)C1)n1cccc1 O=C(C1=NN2CCN=C2N1)NC1CN(C(C2CCC([N+](=O)[O-])CC2)=O)C1 C(C1CCOCC1)=CC(=O)N(C(CCC=C)=O)C(C1(c2ccsc2)COC1)=O C1(NC(C(F)=CCC)=O)CCN(C2CCN(C(=O)CCC(C)SC)CC2)CC1 C1(NC(C2CS(=O)(=O)C2)=O)CC1C1CCN(C(c2ccn3ccnc3n2)=O)CC1 N1(C(CC2(C)CCOC2)=O)CCC2(CCN(C(c3occ4c3CCC4)=O)C2)C1 c1(CN(CC(=O)NC(C(=O)N(C)C2CC2)C2CCCO2)C)ccc(F)cc1 c1(CC(N2CCC3CN(C(=O)Cn4nccn4)C3C2)=O)cccc([N+](=O)[O-])c1 C1(C(=O)NCCC(C)N(C(CCC(C)OC)=O)C)CC12CCc1ccccc12 c1(C(=O)NCCc2c[nH]c3ccc(Br)cc23)ccncc1C1=COCCC1 C(C(C)(C(C)C)NC(c1cn(CC)cn1)=O)NC(C1(CC#C)CCC1)=O N1(C(c2cc(COC)on2)=O)CC(NC(C2CCOC2)=O)C2CCCC12 N1(C(c2ccnc(OC3CCC3)c2)C(=O)NCCOC)CC2CCCC(O)C2C1 C1(NC(=O)CSc2ccccn2)CC(O)CN(C(=O)C=Cc2cncnc2O)C1 c1(C(=O)NC2CC(NC(c3csc(CO)n3)=O)C23CCC3)cnn2cnnc2c1 C1(NC(c2cccc(N)c2)=O)CN(C(=O)COc2ccccc2)C2(CCOC2)C1 C1(CN(C(CCNC(=O)NC)=O)C)CCCC1NC(=O)CC(Cl)Cl CC1CCn2cc(C(N3CCOC(CNC(=O)CN4CCOCC4)C3)=O)nc2C1 Cn1cc(Cl)c(C(=O)NCC2CCC(CNC(=O)CC3CC4COCC34)CC2)n1 C1(NC(C(C=CC)O)=O)CC(CNC(=O)CC(F)F)CC1O N1(C(CCC=CC)=O)CCC(C)(C)C(C(=O)NC(C)CC(C)(C)OC)C1 Cc1noc(C)c1C(C)C(=O)NCCOCCN(C)C(C1CCS(=O)(=O)C1)=O c1(CN(CC(F)(F)F)C(CC2CCN(CC(=O)NCC)C2)=O)ccccc1NC N1(C(=O)OC(C)(C)C)C2CCC(NCS(=O)(=O)c3ccco3)C1CC2 CC1C(NC(c2ccc(O)nn2)=O)CCN1C(=O)Cc1cnccn1 N1(C(Cn2cnc(=N)[nH]2)=O)CC(=O)CC1C(=O)NC(CO)C1CC1 CC(C)CC(F)C(=O)N(C)CC1COCCN1C(c1ccc(F)cc1Cl)=O N1(C(c2cnc(C)[nH]2)=O)CC2CC1CN2C(c1c(O)cccc1O)=O c1(C(=O)NC2CCC(Nc3nc(C)nc(Cl)c3)CC2)ccc2cncn2c1 C(=O)(C(CN=C(NCc1cnnn1C)NC(C)C1CC1)C(C)(C)C)OC C1(CC)C(NC(=O)CN(C)Cc2ccccc2)CCN1C(c1cc(C#N)c[nH]1)=O C1(CNC(C(C)(c2cccs2)NC(=O)C(C2CCCCC2)F)=O)CC[Si](C)(C)C1 c1(C(=O)NCCC(C)N(C)C(c2cncc(F)c2)=O)cc(S(C)(=O)=O)co1 N1(C(c2c(Cl)cn(CC)n2)=O)CCC(C)C(NC(c2ncncc2C)=O)C1 c1(C(=O)NC(C)(C)CO)c(NC(c2ccc(C3CC3)nc2)=O)sc2c1CCC2 C(=O)(CCC(=O)NCCC)NCC1C(C(=O)NCC(=C)Cl)CCC1 C1(C(N2CCC(C(C)(C)NC(C3CC34CCC4)=O)CC2)=O)CN2CCN1CC2 CC(C)(C)C1CCNc2c(C(=O)NCCNC(=O)CCC3CC(F)(F)C3)cnn21 C1(NC(c2c(C)c[nH]n2)=O)CCN(C(=O)C(Cc2ccsc2)NC=O)C12CC2 CCCCC#CC(C)(C)NC(c1cc(CNC(c2ccc(C)c(F)c2)=O)[nH]n1)=O c1(C(=O)NCCCOCCN(C(CC(C)SC)=O)C)cn(C)nc1C C1(C(=O)NC(CN(C(Cc2ccc(C)o2)=O)C)(CO)CO)CCc2nnnn2C1 c1(C(N2CC3(CC(NC(C(C(C)(C)C)SC)=O)C3)C2)=O)cc2n(c1)CCCC2 O=C(CC1OCc2cc(Cl)ccc21)NCC1CCC(CNC(C2(O)CC2)=O)CC1 N1(C(C(C)(C)O)=O)CCCC(C2CC2NC(=O)CCCc2ccsc2)C1 C1(=O)C(F)(CC)C(=O)NC2(CF)CCN1C2.C(=O)(CC(=O)N(C)C1CC1)NCC c1(C(=O)OC)cc(C#N)ccc1NC(C1CCN(Cc2cc(Br)c(Br)s2)CC1)=O C12(CNC(=O)Cc3ccnnc3O)CCCC1N(C(=O)CCN1CCC1)CCC2 C(C(O)C(=O)N(CC(C)C(=O)N1C(CO)CC1C)C)SC C1(CNC(CCCC#N)=O)C2CCC(C2)N1C(=O)CCOCc1ccccc1 C1(COC)CC2(CCN2C(=O)Nc2ccc(C(=O)N(C)C)c(Cl)c2)C1 N(C1CCCn2nncc21)C(C(=O)NC(C)Cc1ccccc1F)=O C1(C(=O)NCC=CC)CCCCN(C(c2c[nH]c(C)c2)=O)C1 c1(C(=O)NCC(O)CNC(c2ccnc(Cl)c2F)=O)cc2ccc(O)nc2s1 C1(NC(C(C(CC)CC)C)=O)CN(C(C2CC(C3CC3)=NO2)=O)C2CCCCC12 c1(C(N2CC(C(C)NC(CC(CC)O)=O)C2)=O)cc([N+](=O)[O-])ccc1OC c1(C(=O)NCCCCNC(c2c(CC)cno2)=O)cnc(OC)cc1OC C(=O)(CC1=C(C)NS(=O)(=O)N=C1C)NC1C=CC(CNC(C(C=C=C)C)=O)C1 C1(N(C(C=CC(C)C)=O)C)CCC(NC(=O)CC(C)N(C)C)CC1 C(=O)(C(CCOCCO)NC(C1CCCNC1=O)=O)NCCNC(C)=O CC(N(C)N1CC(Cc2ccccc2)CC1C)c1cccc([N+](=O)[O-])c1 C1(=O)C(CC(F)F)N1.C(=O)(CC(C)(O)C=CC)N(CCCC)CC(=O)OC c1(OC)ccc(C(N)=O)cc1C(=O)NC1CCC1NC(=O)CN1CCC(C)C1 c1(CC(C)NC2(C(=O)N(C)C)CCC(C)C2)cc2ccccc2s1 n1(CC)nc(C(c2nnnn2CCOC)NCC2CC(F)(F)C2)c(Br)n1 C1(NC(C(C(C)C)OCC(C)C)=O)CCN(C(c2csc(=N)[nH]2)=O)CC(C)(C)C1 N1(C(COC)=O)CCC(O)C(C(N2CC3CCC2CO3)=O)C1 Cc1ncnc(O)c1CCCc1nc(CCCCN(C)C)nn1CC(C)(C)C N1(C(c2c(CC)n[nH]c2)=O)CCCC(NC(=O)C=Cc2nc(C)c(C)[nH]2)CCC1 N1(CC(N2C(CCOC(C)C)COCC2)=O)CCc2ccccc2C1=O c1(OC)cc2c(cc1OC)C1(CC1)CN(C(C1(C)CC3(CC3)C1)=O)C2 Cc1ncnc2c1CC(C(=O)NCC1(NC(=O)CSC(C)C)CCOCC1)CC2 N1(C(=O)Cc2cnns2)CC2CCN(C(c3cccc(F)c3F)=O)C(C2)C1 C1(NC(C2(C)CC=CC2)=O)CC2(CCCN(C(=O)CCn3cccn3)C2)C1 c1(COC(C)C)ccc(C(N2CC(NC(=O)CN(C)C3CC3)CC2C)=O)cc1 C1(CC)(CC)CC(NC(=O)CC(C)N(C)C)CN1C(=O)CC(C)(F)F CCCC(C(=O)N1CC(O)(C(F)C(=O)NCc2ccc(=O)n(C)c2)C1)C(C)C C(=O)(CCS(=O)(=O)Cc1ccccc1)NCCN(CCC)C(C1CC(C#N)C1)=O C1(CNC(C2(CCOC)CCC2)=O)CC2(CCN(C(=O)CCC(C)(F)F)C2)CO1 C1(NC(c2csc(-c3ccccn3)n2)=O)CCN(C(C2(F)CC=CC2)=O)CC1F N1(C(COCC)=O)CCOCC1CN(C)C(c1cnc(CC(C)(C)C)s1)=O C1(CCN(C)C(C2CSCCS2)=O)CCCCN1C(C1(C2CCC2)CC1)=O c1(C(N2CC(C(C)NC(=O)CC3CC(F)C3)C2)=O)cc2ccccc2n1C Cc1cc(C)c(C(=O)NCC2CN(C(c3nnn(C(C)(C)C)n3)=O)C2)c(Cl)n1 Cc1ccnnc1C(=O)NC12CC(NC(=O)CNC(c3ccoc3C)=O)(C1)C2 c1(CC)cc(Cl)ccc1C(=O)N(C1CCCN(C(=O)CCCC#N)C1)CC CC(C)(C)C(CNC(c1csc(CCP(C)(C)=O)n1)=O)NC(C1CCCOC1)=O N1(C(CNC(C(CC)C)=O)=O)CC2CCN(C(=O)CC3CC(C)=NO3)CC12 c1(C(=O)NC(C2CCOC2)C)csc2c1CCN(C(c1cnnc(Cl)c1)=O)C2 c1(C(=O)NCCN(C(COC(CC)C)=O)CC(C)O)cccc2c1CCOC2.O c1(C(=O)NC2C(NC(=O)Cc3cnsc3)CCC2)ccc(Cl)cc1O c1(CNC(c2c(OC)ccc(F)c2)c2nnnn2C)csc2cccc(F)c12 C(C(C)C(=O)NC(C)CNC(=O)C(C)(C)c1ccnn1C)OCC Cc1cnc(Br)c(NC(C2CCC(NCc3c(Cl)cncc3Cl)C2)=O)c1 C1(NC(C=CC=CC)=O)CCN(C(=O)Cc2cccc(C)c2)C1CC C1(C(N(C2CCCN(C(CCC(C)C)=O)C2)C)=O)CCCC12CCC2 C1(C(C)C)CN(C(C2CC(F)(F)CS2)=O)CCN1C(=O)COCC1CCCO1 c1(NC(C(c2cccc(C)c2)NC)=O)ccc(C2CCCCC2)cc1F C1(C(=O)NC2(C3N(C(CCc4c(C)ncs4)=O)CCC3)CC2)CC2(C1)CC(O)C2 C12(CC(=O)NC3C(NC(c4cnc(C(C)OC)s4)=O)C3)CCC(CC1)OC2 O=C(C(C1=CCSC1)N1CCOCC1c1cnc(Cl)c(Cl)c1)NCCC1CC1 c1(OC)ccc2c(c1)NC(=O)C2CC(=O)Nc1c(-n2cccc2)sc2c1CCC2 c1(C(N(C(c2cn(-c3cc[nH]c(=N)c3)nn2)C)C)=O)ccc(Cl)c(C(F)(F)F)c1 N1(C(C2(NC(=O)CNS(N)(=O)=O)CCN(C)C2)=O)CCC(C2CCCC2)C1 c1(OCCCN)cccc(C(=O)NC(CC(=O)O)C2CC2)c1 c1(C(N2C(CNC(c3c(C)ccnc3)=O)CC(C)(C)C2)=O)ccc2occc2n1 N1(C(c2c(CC)nn(C)c2)=O)CC2CC(C1)C2NC(=O)C(C(C)CC)NC(C)=O C12(CNC(c3cccc(-c4nc[nH]n4)c3)=O)CC1CN(C(=O)CC1C=CCC1)C2 c1(CCCC)nc(CNC(=O)C(=O)NC2CCCC(C(F)(F)F)C2)c(Cl)[nH]1 C=CCC(CNC(C1CCCN1C)=O)NC(c1cc(C(F)(F)F)no1)=O C(CC(F)F)(C(=O)NOCCc1ccccc1)NC(c1c(C)cc(F)cc1)=O C(=O)(C(CCC1CC1)NC(c1sccc1CO)=O)NCCN1CCC(C)C1 C1(NC(C2(CCCC)CC2)=O)CC2CC(C1)N(C(c1c(Cl)n[nH]c1C1CC1)=O)C2 c1(C(=O)NC2(CNC(CN3C(C)CC3)=O)CCOCC2)cc(F)c(CO)c(F)c1 C(C(=O)N1CC(NC(=O)CC(=O)NCC(F)(F)F)C1)(C(C)(C)C)N(C)C N1(C(CCC#CC)=O)CCC2(CC1)COC(CNC(=O)C(C)CN(C)C)C2 C12(CNC(=O)CCC3CC3)CCCN(C(c3ccc(SC(F)F)cc3)=O)C1C2 N1(C(CC(COC)NC(C2CCCCCN2C)=O)=O)CCOCC2(CC2)C1 C1(NC(C(CC#C)C2CC2)=O)CN(C(c2cccc3cncn23)=O)CC2(CC2)C1 Cc1cccc(C)c1NC(=O)C(c1cnc(Cl)s1)N(CC(N1CCCC1)=O)C1CC1 CN1CCN(C(=O)CNC(c2cccs2)=O)C(CNC(C2(C)COCCO2)=O)C1 C1(NC(c2cscc2Cl)=O)Cc2ccccc2C1NC(c1cc(F)n[nH]1)=O c1(C2(C)CCO2)cccc(C(=O)N(C(c2cccs2)=O)CC2CCCO2)c1 CN1Cc2ccccc2CC1C(N1CCC1C(=O)NC1CC(CO)C(O)C1O)=O C1(NC(c2cccc3ncccc23)=O)CCC2(CCN(C(=O)CO)C2)C1 C1(NC(CCC=C)=O)CC1C1CCCN(C(C2(CF)CC3(CCC3)C2)=O)C1 C1(CC(=O)N(CC(C)NC(c2[nH]ccc2C2CC2)=O)CC)CCCCC1(F)F C1(CNC(C2N(CCC)CCCC2)=O)CN(C(=O)C=C(C)C)CC2(CCC2)O1 C(C(=O)N1CC(N(C)C(=O)C2CC2)C(C(F)F)C1)(C(C)(C)C)NC(C)=O C1(CNC(COCC=C)=O)CN(C(C23CCCC2C3Br)=O)CCC1(C)C C1(CNC(=O)Cc2cn[nH]c2)CC(NC(C2(Cl)CC2(F)F)=O)CC1O O=C(C1CCc2ccc(Cl)nc21)NC1CN(C(=O)CCc2cscn2)CC1O N1(c2snc(SC)n2)CCOC(C)(CNC(c2ccnc(Cl)c2)=O)C1 C12(CNC(c3cc(CC)no3)=O)CC(CF)(CO1)C2.C12COC(C1)NC(=O)C2 C1(C(=O)NCC(CC)(C)O)(NC(=O)CCc2cncn2C)CCCCC1 C1(n2cc(-c3cn(CCC)nc3)nn2)CC2CCC1(NC(c1cnc(C)s1)=O)C2 C1(NCc2cn(CCCC(=O)NCc3[nH]cc(C)c3)nn2)CC2CCC1CC2 Cc1ncc(C(=O)NC2CCN(C(c3c[nH]c(=N)cc3C)=O)CC2C)c(O)n1 C(C)(CS(C)(=O)=O)N(Cc1n(CC)ccc1)CC c1(C(=O)NC2C(NC(CCCSC(C)(C)C)=O)CC2)cc(Cl)cc(C(F)(F)F)n1 C(CC(CC)C(=O)N1CCCC(C)(NC(=O)CCc2cnc(C)o2)C1)=CC CCCCS(=O)(=O)CC(=O)NC1CN(C(C2CC2C#N)=O)CC1OC N1(C(C(CC)(C)C)=O)CCC(C2CCN(C(c3cncn3C)=O)CC2)C1 N1(C(C(C(C)C)C)=O)CCN(C(C2(COC(F)(F)F)CC2)=O)CC(C)(F)C1 N1(C(C2CCCN(c3nccc(OC)n3)C2)=O)CC(=O)N(C)CC1C C1(CC)CCCCCCN1C(C1OCCC1NC(=O)CC12CCCC1C2)=O c1(C(=O)NCCCC(C)NC(=O)C(C)(C)C(N)=O)ccc([N+](=O)[O-])s1 c1(CN(c2nnc(-c3ccco3)n2CC(F)(F)F)C)cn(C)nc1Br c1(C(=O)NCC2(O)CCCN(C(CN(C(C)C)C)=O)C2)cc2ccnn2cn1 C1(C(=O)OC)(Cc2ccccc2)CCCN1C(=O)CNC1COC(C2CC2)C1 c1(C(=O)NCC(CC)NC(=O)Cc2cccc(OC)c2OC)cccc(F)c1O CC(CN(C)C)CC(=O)NCC(C1CCN(C(=O)CC2CCCN2C)CC1)(C)C c1(C(=O)NC2C(CNC(=O)CCOC3CCOC3)CC2)cccc2c1C(=O)CC2 O=C(CS(=O)(=O)Cc1cccs1)NC1CCC1NC(C1CCOC1)=O C1(C(N2CCC(CC(C)C)C2)=O)CN(C(c2ccn(C(F)F)n2)=O)CC1F C1(C(=O)NC(CCOC)COC)(CF)CCNC1=O c1(OCC)cccc(-c2nc(-c3c[nH]c(C)c3)n(C(CC3CCC3)C(C)C)n2)n1 Cc1ccnc(COC(c2ccsc2C)=O)n1 C1(C(=O)NC(C(=O)NC(COC)(C)C2CC2)C)CC2CC(=O)C1O2 C1(C(N(CCCN(C(c2c(N)ccc(C)c2)=O)C)C)=O)CCC(=C(F)F)CC1 NS(=O)(=O)c1csc(C(=O)NC2CC(CNC(c3cc4ncccc4[nH]3)=O)C2)c1 c1(OC)[nH]c(=N)nc2sc(C(=O)NC(C)CC(C)NC(c3cn(C)nn3)=O)cc12 C(C)(C(=O)N1CCCC(C)(NC(=O)C=C(C)C(C)C)C1)(C(C)C)OC CC1CN(N(C)C2CN(C)C(C(F)(F)F)C2)CCN1C CN1CC(=O)Nc2cc(C(N3CC4CCC3CN4C(=O)C3=NOCC3)=O)cnc21 C1(NC(=O)Nc2c(Nc3c(OC)c(C)ccc3)cccc2)CCC2(CC1)COC2 CC12CCCOC1CN(C(=O)NCc1cn(C3CCOC3)nn1)C2 C1(CC(=O)NCC(CN(C)C)O)C2CCC(C2)N1C(=O)CC1CCCN1C c12ccc(cc1O)C1(CC1)C(=O)N(CC1CC1)C1CCN2C1.c1(S)csnc1C.CO Cn1c(C(=O)NC2CC(CNC(C3(Cl)CC34CCC4)=O)C2)cccc1=O N1(C(CCC(c2ccc(C)cc2)=O)=O)CC2CC3CC2C1C3NC(C1CCC1)=O c1(CC)sc(C(=O)NCC2CCCCC2NC(=O)CCCF)cc1Br C(=O)(C(C(=O)OC)OC)NCC(CN(C(CN(CCC#C)C)=O)C)(C)C C(N(C1CC1)N1CC(O)C(O)C1CO)c1ccc(N(C)C)cc1 Cc1cc(C)c2nc(N3CCC(C)C(NC(c4cnc(C)s4)=O)C3C)sc2c1 Cc1nccc(C(N2CC3CC(NC(=O)CCSc4nnnn4C)C2C3)=O)c1C c1(C(N2C(C(C)NC(C(CC)N(CC)CC)=O)CCC2)=O)cc(C(F)F)n(C)n1 c1(C(=O)NCC(c2cccc(C)c2)NC(C(C=C)(C)O)=O)ccc([N+](=O)[O-])s1 C1(CC)(NC(C2CCC3(CC2)CC3)=O)CCCN(C(c2cn(C)nc2OC)=O)C1 c1(CNC(C(C)OCC#C)=O)c[nH]nc1C(=O)NC(C1CCCCC1)(C)C c1(C(N2CC(CCNC(c3c(OCC)n[nH]c3)=O)C2)=O)cccc2nc(C)[nH]c12 C1(NC(c2c(C)cno2)=O)CN(C(C2CN(C)CCO2)=O)C2(CCC2)C1 C1(CCF)(NC(=O)CCn2cc(CCNS(C)(=O)=O)nn2)CCN(CC)CC1 N1(C(C(CO)NC(C(C)C)=O)=O)CCC2CN(C(=O)C=Cc3nccs3)CC2C1 C1(C)(C(=O)NCC23CC(NC(C(c4cnccn4)C)=O)(C2)C3)CC(C)(C)C1 c1(C(=O)NCCC2CC(NC(C3CC3C(F)(F)F)=O)C2)ncncc1Cl C1(C(=O)NCCn2cc(C(=O)NC(c3ccccn3)C)nn2)Cc2nccn2C1 CCCC(C(N)=O)OC(C1CCN(c2cc(C)n(C)n2)C1=O)=O C1(NC(C2CCC2)=O)C2CCC(C2)C1C(=O)Nc1cc(Cl)ccc1O Cc1ccc(Cl)c(C(=O)NC2CCN(C(=O)C(C(C)C)N3CCN(C)CC3)C2)c1 c1(CCN(C)C)ccccc1C(=O)NCC1CCCN1C(=O)C(C)(F)F N1(C(c2n(C(C)C)ncc2Cl)=O)CCC(C)C(CNC(=O)CCc2nncs2)C1 C1(NC(C(CN(C(C(C)(C)OCCC)=O)C(C)C)C)=O)CN2CCC1(F)CC2 N#Cc1ccc(CNC(=O)C(=O)NCC2=NOC3CC23)cn1 S(=O)(=O)(c1ccc(Br)cc1N1CC(O)C(C2CC2)C1)N(CCC#N)CCC C(=O)(C(O)CC(F)(F)F)NCC1(CO)CCN(C(C2N(CC)CCOC2)=O)CC1 c1(C(=O)NCC2N(C(CCN(CCC)C)=O)CCCC2C)cc2scc(C)c2[nH]1 c1(SC)nc(N2CCCC(NC(=O)C=Cc3ccco3)CC2)cc(C(F)F)n1 N1(C(C(C)SC(C)C)=O)CCC(=O)N2CCCC12 CC1(C)CCCOC1C(=O)NC1CC(O)C1CC(=O)NCc1cncnc1 c1(C(=O)NC2CCCN(C(C(CCC=C)(F)F)=O)CC2)c[nH]c2ccc(O)cc12 c1(C(CC)=O)cc(C(=O)NC2CCC(NC(c3cn(C)nc3O)=O)CC2)ccc1F C1(C(=O)OCC)COCCN1Cc1cc(C)on1 c1(C(=O)NCCCCC(C)NC(COCCCC#C)=O)ccn2nccc2n1 C1(C2CCCN(C(c3cnc(C(C)C)n3C)=O)C2)(NC(CC(CC)C)=O)CC1 c1(C(=O)NC2CC(NC(CCc3nc(C)sc3)=O)C2)ccc(F)cc1Cl C(=O)(C1=NOC(C)C1)NC1(CC)CN(C(C2CCCC2C)=O)C1 C(=O)(C(C)S(=O)Cc1ccc(OC)nc1C)NC(CC)C C1(NC(c2cccc(C)c2Cl)=O)C(C)CN(C(=O)CCc2cccs2)CC1C c1(CC(=O)NCC2(F)CN(C(C(CC)c3cccnc3)=O)C2)cc(C)cc(F)c1 c1(NC(NC2C(C)CCCC2)=S)ccc2sncc2c1 C(CC)(C(=O)N1CC(C(=O)NCC(C)CC2CCC2)(SC)C1)OCC N1(CCC(C(=O)OCC)F)C(=O)CCN(Cc2nnc(COC(C)(C)C)s2)C1=O c1(C(=O)Nc2cnc(OCC)nc2)cc(Cl)ncc1NC(c1coc(Cl)n1)=O c1(CC(N2CCC(NC(CCC3C(C)(C)C3)=O)C23CC3)=O)c(F)cccc1C#N CC1(C(N2CC(OCC(=O)NCCn3ncccc3=O)C2)=O)CCOCC1 N1(C(C2(C#C)CCC2)=O)CCCC2CCN(C(c3cnn(C(C)C)c3C)=O)CC12 N(C(=NCCCF)N1CCC2CCCCC2C1)Cc1cc(C)oc1C c1(CC)[nH]nc(C(=O)NCC2CCC(C(=O)NCc3cn[nH]c3)CC2)c1F C(=O)(C(CC(C)C)c1ccccc1)N1CC(N(C(c2cc(C)oc2)=O)C)C(O)C1 C1(NC(c2ncc[nH]c2=O)=O)C2CCC1N(C(=O)C(O)C1CCC1)C2 CCC1=NOC(C(=O)NC2CCCC2NC(=O)C(=O)NCCOC)C1 C12CN(CC(F)(F)C1)C2=O.c1(NC(CN(C)C)=O)cnccn1 C1(C(N2CCC(C)C2CNC(=O)C(F)=C2CCC2)=O)Cc2nccnc2C1 CC(C(=O)N1CCC2(C1)CN(C(=O)CN1CC(=O)N(C)C1=O)C2)C(C)C(C)(C)C c1(C(=O)NC2C(NC(C3(C)CC(C)(C)C3)=O)COC2)ncc(F)cc1N c1(C(N2CCC(OC)C2)=O)cc(CN(C)C)c(C)s1.C12CN(C1)C2=O c1(C(=O)NCC(C)C(=O)NC(CO)C(F)(F)F)c[nH]c2ncccc12 C(=O)(CC(C)(C)O)N(C)CC1CCCN1C(=O)COCC1CC=CC1 c1(C(=O)NCC2CCC(F)(CNC(C(CCC)C)=O)C2)ccc(P(C)(C)=O)o1 C1(C(N2C(CNC(c3cc(F)cc(F)c3)=O)CC3(CC3)C2)=O)CCCC(F)(F)C1 c1(N(C)C(C2CC(n3ccnn3)C2)=O)ccc2cc(Cl)cnc2n1 C1(CC)(CC)CC(O)C(O)CN1C(=O)Nc1cc(C)nc(O)c1 CC1(C)CC(N(C)C)CN(C(C2(N3CCCC3)CCC2)=O)C1 c1(C(N2CC(CNC(C3(Br)CC34CCC4)=O)C2)=O)cnc2ccoc2c1 N1(C(C(c2cnccn2)C)=O)CC2CC(NC(=O)Cn3nnc(C4CC4)n3)C1C2 N1(C(C2(OC)CCSCC2)=O)CCC2(CCCN2C(c2cc3cscc3s2)=O)C1 C(=O)(CCCC(C)(C)C)NCC12CC(NC(Cc3nc(C)[nH]n3)=O)(C1)C(C)O2 c1(C(N(CCCN(C(C(CC(C)C)(F)F)=O)C)C)=O)cccc2cc(O)ccc12 C=C(C)C(CC(=O)N1CCC(CF)(NC(=O)CSCCCC)C1)OCC C#CCCCCC(=O)NCC1CC(NC(=O)CN(C(C)=O)Cc2ccccc2)C1 C(=O)(C1CCc2cccc(F)c21)N1CCC(CNC(CCc2n(C)ccn2)=O)C1 N1(C(C(C(C)C)SCC)=O)CCN(C(=O)CCSCC(N)=O)CC1CCO c1(NC(=O)NCC2C(C(=O)OC)CCC2)ccc(S(C)(=O)=O)nc1 c1(C(N2CC3C(CNC(CC(C)O)=O)(C3)C2)=O)csc2nnsc12 c1(C(=O)NCCNC(C(c2ccc(Br)cc2)(C)C)=O)ncc[nH]c1=O N1(C(C(C=C)(F)F)=O)CCOC2(CCCN(C(c3cccnc3O)=O)C2)C1 c1(CNCCNC(C23C(C)OC(C)(C2)C3)=O)cc(Br)c(Cl)c(Br)c1O C(=O)(C(C)(C)C1CCCN1C(c1cc(C)on1)=O)NC(C1CCCC1)CC C1(CNC(C2C(C)C2)=O)CC2CCC1N2C(C1CCC(CO)CC1)=O n1(CC=C)cc(CNC(=O)CCc2ccon2)nn1 c1(C(N2CCSc3ncccc32)=O)cc(Cl)cc2ccccc12 CCN=c1[nH]c(C(=O)NCC2(F)CC(CNC(C3CCCC(C)O3)=O)C2)cs1 C1(CNC(CC2C(C)C2(F)F)=O)(NC(C2CCC(C)(C)C2)=O)CCOCC1 c1(NC(C(C2CC=CC2)N(C(C)C(=O)OC)CC)=O)ccc(Cl)cc1 Cc1cn2c(n1)CCC(C(N1CC=CC(NC(=O)Cn3ncccc3=O)C1)=O)C2 C1(CC)CN(C(c2cc(F)n[nH]2)=O)CCN1C(=O)C1=NOCC1 c1(C(=O)NC(C(C)C)CNC(C2(C(=O)OC(C)(C)C)CCC2)=O)cc2n(n1)CCO2 CON(CCO)C(=O)c1cncc(CNC(=O)C=Cc2cc[nH]c2)c1 C1(NC(c2c(OC)c(Cl)ccc2)=O)CCC(O)CN(C(c2cnccn2)=O)C1 c1(C(=O)NC(C)C(C)NC(=O)CSC2CC2)cc(C2CC2)nc2ccnn12 c1(NC(C23CCC(CC2)N3)=O)cc(Cl)nc(C2CCCO2)n1 N1(C(c2cc(C)cc(Cl)n2)=O)CCC(CNC(C2CC(C)CO2)=O)C(F)(F)CC1 c1(C2N3CCC(C3)NC2=O)cc(OC)n(C)n1.C1(OC)CC(NS(N)(=O)=O)C1 C(CCC(=O)N(CC(N1CC(COC(C)=O)C1)=O)C(C)C)OCCOC C1(C)(C(N(C(C)CN(C(=O)COCC2CCC2)C)C)=O)CCOCC1 c1(C(=O)OC2CC(OCC(=C)C)C2)n[nH]c2ccc(Cl)cc12 N1(C(c2c(OC)cnnc2)=O)CCOC2CN(C(=O)C(C3CC3)SC)CC12 C(c1nc(C)cs1)=CC(=O)OCC1(OC)CC(OC)C1 CC1CN(C(=O)CCNC(=O)Cc2ccccc2)CCC1NC(=O)CP(C)(C)=O C(CCCCC(=O)NCC1CCC1NC(c1cc(F)ccc1O)=O)OCC CCC(C)C(O)CNC(=O)CC1(NC(C2CCOCC2)=O)CCC1 c1(CC(N2CCOCC(CNC(C(C)CC(F)F)=O)C2)=O)nnc2n1CCCC2 N1(C(C2CC(=C)CN2C(c2ccncc2Br)=O)=O)CCC(O)C(C)C1 C1(C(=O)NCCCOCCN(C)C(c2ncn3c2CCC3)=O)CC2CCCC2C1 N1(C(c2ncc(OC)cn2)=O)C2CCC1CN(C(c1ccc(C)c(Cl)c1Cl)=O)C2 C1(NC(Cc2ccn(C(C)C)n2)=O)CC2(C1)CN(C(C1(C(F)F)CC1(F)F)=O)C2 Cc1cc(=O)n(C)nc1C(=O)NCC1(CNC(=O)C=Cc2ccsc2)CCCC1 CC1(C)OCCC1C(=O)NCC(C)(F)CNC(C1(C2CCCCO2)CC1)=O C(=O)(C1CCc2cccc(O)c21)NCCCNC(COCCC(C)C)=O c1(C(C)C)ccc(F)cc1NC(=O)NCC1CCOC1 C(=O)(C(C)(C)CNC(N)=O)NC1C(NC(c2c(C)coc2)=O)CCC1 N1(C(C(C)C)=O)CC2CCC(C1)C(NC(C1CC1c1ccc(Br)cc1)=O)C2 C1(C(=O)NCc2ccc(C(N(C(C3CCCO3)C)C)=O)s2)CCS(=O)CC1 N1(C(C(n2c(C)ncc2)C)=O)CCC(C=CC(=O)NCC(C)N(C)C)CC1 CCC(C)CCCCC(=O)NC(C)CN(C)C(c1[nH][nH]c(=N)c1Br)=O C(N=c1nc(N2CCOCC2)[nH]c(=NC2CCCCC2C#N)[nH]1)c1cc(C)oc1 C(=O)(C1CCCc2nn[nH]c21)N(C)CC1CCCCN1C(=O)C(F)=C1CCCC1 n1(CC)cc(C(=O)NCCC(O)C(=O)NCCCCNC(N)=O)c(C)n1 CCC(C)(CNC(=O)C=CC(C)(C)SC)NC(C1CC1CC(=O)OC)=O c1(C(=O)OCC(C)CN(C)C)ccc2c(ccn2C)c1 N1(C(Cc2ccn(C(C)C)n2)=O)CCc2[nH]nc(CNC(C3(C)CCC3)=O)c2C1 N1(C(C(C)n2cccn2)=O)CCCC1(C)CNC(=O)Cc1cc(C(C)(C)C)no1 O=C1CCC(C(=O)NC2CCCCN(C(=O)CSc3cccs3)C2)n2cccc21 C(CCCCC(=O)NC1(C(=O)NCCC2NC(=O)NC2=O)CC1C)OCC c1(C(=O)NCC2(C)CC(NC(C(C)=C3CCC3)=O)C2)ccccc1SC(F)(F)F C1(C(=O)NCC(C2CCC2)NC(c2cc[nH]n2)=O)CCC2(CCCC2)C1 C1(C)(CCC(=O)NCCC(C)(C)NC(C=CC(=O)N(C)C)=O)CCC(=O)N1 C(=O)(C(CNC(C)C(=O)Nc1cc(C)co1)N(C)C)NC(CC)(C)C N1(C(C(C)NC(C)=O)=O)CCC(C(=O)N(C(C)C)CC2CCCO2)CC1 c1(C(=O)NCC(C)(C)CNC(=O)CC2CC3CCC2O3)c[nH]c2c(Cl)cccc12 c1(C(=O)NCC(=C)CCNC(=O)C(C2CCC(=O)N2)C)ccc(OC)cc1 N1(C(C2(CC=C)CCC2)=O)CC(Nc2nc(C)cc(C)n2)C(C)(C)C1 C(C#Cc1cccnc1)NC(CC(C)N(C(C(C)N=[N+]=[N-])=O)C)=O c1(C(C)NC(C2(NC(C(C)N3CCCC3)=O)CC2)=O)ccncc1 n1(COC)ccc(C(=O)NCC(C)N(C(=O)CCCn2cncn2)C)n1 c1(C(N2CCCC(NC(C3(C4CCCCO4)CC3)=O)C2)=O)ccnc2ccnn12 N1(C(CCn2c(C)csc2=O)=O)CCCCC1C1CCCN1c1ncncc1Cl c1(C(N(C2CN(C(C(CC(C)C)O)=O)C2)C)=O)ccc([N+](=O)[O-])cc1 CC1C(C(=O)NC2(c3ccsc3)CC2)CCCN1C(=O)CC1CN(C)C1 c1(C(=O)NC2(C)CCN(C(CCC3C(C)C3)=O)C2)cc(F)c(F)c(F)c1F C(=O)(C1=CCCC1(C)C)NC1C2CN(C(C(CC(C)C)N(C)C)=O)CC21 C1(NC(c2cccc(C3CC3)n2)=O)CCCCN(C(c2n[nH]cc2Cl)=O)CC1 c1(C(=O)NC(C(C)C)CCNC(=O)C=CCN2CCOCC2)nccc(Cl)c1F CC1(C)CCCC1C(=O)NCCC1CCN(C(C2(C(N)=O)CC2)=O)C1 N1(C(=O)C2=CCCOCC2)CCCC12CCN(C(C13CCCN(CCC1)C3)=O)C2 C1(CN(C(=O)C(F)C2CCOC2)C)CCC(CNC(C23CC2CNC3=O)=O)CC1 C(=O)(CC(C)CC(=O)OC)N1CCC(=C)CC1C(=O)NCCc1nccc(C)n1 c1(C(N(CCCNC(c2cc(C3CCOCC3)no2)=O)C)=O)nc2ccccc2o1 N1(C(c2cc(OC)nn2C)=O)CC(O)CCC1C(N1CCC(c2cnco2)C1)=O CCC(CC(=O)NC1(CCCNC(c2cc(CC(C)C)[nH]n2)=O)CC1)C(F)F N1(C(C(C(=O)OC)C)=O)CCN(C(CC(C)C)=O)C2CC12.C1CC(=O)N1 C1(CNC(C(C)NS(C)(=O)=O)=O)CCN(C(c2c(Cl)cnn2C)=O)C12CC2 C1(NC(Cc2cccc(C(C)(C)C)c2)=O)CCCCN(c2ncnc(=N)[nH]2)C1 O=C1CCC(S(=O)(=O)NC2(CNC(=O)Cc3ccsc3)CCCC2)CC1 c1(NC(CC(C)(C)NC(C(C=C)OC)=O)=O)c(C)cccc1C c1(C(=O)NC(C(=O)OC)C)cc(Br)c(OC)cc1OC.N12CCOC(C1)C2=O c1(C(=O)OC)c[nH][nH]c1=NC(=O)C1CN(C(=O)CCc2ccoc2)CCN1 C=CC1(CC(=O)NCCCCCN(C)C(c2conc2C)=O)CCC1 Cc1[nH]c(C)c(C(N2CC(C(=O)NCc3ncccn3)C(F)(F)C2)=O)c1C C1(C(N(C(CNC(C(C)c2ccco2)=O)C2CC2)C)=O)CCc2ccnn2C1 N1(C(CC)=O)CCSCC1CCNC(c1cccc(NC(N)=O)c1)=O C1(CNC(C2C(C#C)C2)=O)CC(O)CN1C(=O)Cc1csc(NC=O)n1 N1(C(C2(C)CN(C(=O)CSCC(F)F)C2)=O)CCCCC1CCCO C1(CC(N2CCC(CCCNC(CCCOC)=O)CC2)=O)CCCCC1(C)C c1(C(=O)NC(CC#C)C(=O)NCC2(CO)CC2(C)C)cc(C)cc(C#N)c1 C1(C(=O)NCC(C)NC(=O)Cc2cc(C3CC3)on2)CCCCC1O N1(C(CC(C)OC)=O)CCC2(CC1)CC(N=c1nc(C(F)(F)F)[nH]s1)CCO2 c1(C(N2CC(C)C(C(=O)O)CC2)=O)cncc2c1CCC2 C(=O)(CCCC(OC)OC)NCC(C(=O)N(C1CC1)CC)CC1CC1 N1(C(CCCOCC=C)=O)CC(NC(=O)Cn2cc(Cl)c(C)n2)CC1(C)C C=CC(C)(CC)C(=O)NC(C)CC1CN(C(c2ccc(-c3ccncc3)s2)=O)C1 CC(C)C(C(=O)NCC[Si](C)(C)C)NC(=O)CN1CCCCC1C N1(C(C(CC(C)C)ONC(C2(n3cnnn3)CC2)=O)=O)CC(=O)N(C)CC1C Cc1cc(C(=O)NC2(CNC(c3ncccc3N(C)C)=O)CCOC2)[nH]c1C c1(C(N2CC(CNC(=O)C=CC3CCC3)OCCC2)=O)cnn2c1OCC(F)C2 C1(NC(C23C(CN(C(c4cnc(C)o4)=O)C2)C3)=O)CCCOC12CCC2 CCC(C)CCC(=O)N1CCC(NC(c2ccc(F)cc2F)=O)C(OC)C1 CCCCC(F)C(=O)NCC1C(C(=O)NC2(C3CCCO3)CC2)C1(C)C N1(C(CSC)=O)CC2CCC(C1)C2CC(=O)Nc1ccc(-c2ncno2)cc1 CC1(C)CCC(C(=O)NCCN2CCN(C(c3coc(Br)c3)=O)CC2)OC1 Cc1ncc(NC(C2(O)CCN(C(c3sccc3Br)=O)C2)=O)nc1C c1(C(=O)NC2(CO)CCCN(C(=O)C(F)=C3CCC3)C2)cc(F)c2[nH]nnc2c1 N1(C(C(C)=C(C)C)=O)CC(C)(C)CCC1CNC(=O)Cc1cccc(C(N)=O)c1 c1(N2CC(C)(CNc3c(C(=O)OC(C)=O)scc3)C2)ncnc2c1ncn2C Cc1cc(C(=O)NC(C2(O)CN(C(=O)Cc3ccon3)C2)C)ccc1Cl Cc1cc(C(=O)NCC2CCN2C(C2CC(C)C2)=O)n(CC(F)F)n1 c1(N2CC(C(=O)NC)OCC2)nc2c(c(=NCC3C(C)(C)C3(C)C)[nH]1)CSC2 C1(C(=O)NCC2N(C(C3=C(C)OCCS3)=O)CC2)COc2ccc(Br)cc2O1 c1(Cn2c(N3CC(CC)SCC3)nnn2)cc(OC)c(OC)c(Cl)c1 CC1CCCCC1(CNC(=O)C(C1CCOCC1)O)NC(=O)CCS(C)(=O)=O c1(C(N2CC(C(=O)Nc3cnn(-c4ccccn4)c3)C2)=O)ccc([N+](=O)[O-])o1 C(CCC#C)(C(=O)OC)NC(C(CC#C)C)=O CCCC(CCCNC(c1csc(Br)n1)=O)NC(=O)C(O)CC(C)C Cc1nc(O)[nH]c1C(=O)NCCC1CCCCN1C(C1C(C)C1(F)F)=O c1(NC(C2CCCN(c3nc(OC)cc(OC)n3)C2)=O)cc(C)c(C)cc1Br C(=O)(CCC(=O)NC(COC)CNC(=O)C(C)OCCN(C)C)NC C1(NC(c2c(OC)nccc2)=O)CN(Cc2ccc[nH]2)CC1C#N C(=O)(N=c1cc(C(N)=O)n(C)[nH]1)C1C2(CCN(C(c3ccc(CSC)o3)=O)C2)C1 c1(OC)ccc(C(N2CCC(C(=O)NCC3(CO)CC(C)C3)C2C(C)C)=O)cc1 C1(C(=O)NCC(C2CCN(C(c3n[nH]cc3C)=O)CC2)C)(CC)CC(C)(C)C1 N1(C(c2c(OC)cnc(Cl)c2)=O)CCC(C2CC2NC(C2CC2F)=O)CC1 C1(CN2C(=O)CC2)C(CN2CCCC2C2CC2)CCN1.c1(C=O)cccnc1 N1(C(C(C)CC(F)F)=O)CCC2(CC(C(N3CCC(c4nn[nH]n4)C3)=O)C2)C1 N1(C(c2c(C)cccn2)=O)CCC(C)CC1C(=O)O N1(c2ncc(F)c3c2[nH]cn3)CCCC(C2CCNCC2)C1 N1(C(c2c(CC)occ2)=O)CC2CC(C(=O)NCCCN(C)C(C)=O)(C2)C1 FC1(F)CCCCC1CNCc1sc(I)cc1Cl c1(C(=O)NC(C(C)NC(c2cc(C(C)C)sn2)=O)C)cncn(C)c1=O CC1=C(C(=O)NC2CC(c3ccccc3)(NC(c3ccc(C)s3)=O)C2)CCO1 CC1CCCC(C(=O)NCC(C)(C)NC(c2cccc(SC(F)(F)F)n2)=O)O1 C1(C)(C(=O)NCC(CNC(C2(COC)CCOC2)=O)OC)CCCCC1 c1(NC(C2(C)N(C(CC=CC)=O)CC2)=O)cc(C)cc(C)c1O C1(C(=O)OC)C(C)CC(C)CN1C(=O)OC(C)(C)C.C12CCCN(C1)CC2=O Cc1nc(C)c(CNC(=O)CC2COCCN2C(=O)C(C)O)s1 c1(N(C2CNC2)C(c2csc([N+](=O)[O-])c2)=O)ccn2ncc(I)c2n1 CC1CCC(NC(=O)COC2(C)CCC2)CN1C(=O)CCN(CC(F)(F)F)C c1(C(N2CC(C)N(C(C3CC(C4CC4)C3)=O)CC2)=O)c[nH]c2ncccc12 N(C(=NCCF)NCC1CCN1C1CCCC1)Cc1ccc(C)cn1 C1(CC(=O)NCC2CC(OC)CN2C(c2ccsn2)=O)CC2(CC(OC)C2)C1 Cc1[nH]c2ncccc2c1C(=O)NC1CCC1NC(=O)C(CC(F)F)C1CCC1 CC(F)(F)CCC(=O)N1CCCCC(C(=O)NCC2CC2Cl)C1 N1(C(C(C)N(C)C)=O)CC(NC(c2cccc(N)c2O)=O)CC(C)(C)C1 C1(C(N2CCC(CSC)C2)=O)CN(C(=O)CC2(N(C)C)CC2)CC1CO C(C)(N=c1[nH]c2c(c(=NCCN(CC(F)F)C)[nH]1)SCC2)c1ccc(C)cc1 C1(NC(C(C=CC)O)=O)CCN(C(c2cscc2Cl)=O)C1c1ccccc1 C(=O)(C1CCCn2cnnc21)NC1CC(NC(=O)COCc2nc(C3CC3)no2)C1 c1(NC(c2ccn(CCNC(CC3CC(SC)C3)=O)c2)=O)cn(C)c(=O)nc1O C1(C(N2CCC(NC(c3c(C)nn(C)c3Cl)=O)C(O)C2)=O)C2CCC1(C)C2(C)C c1(C(N2CCC(COC)(NC(=O)C=CC(C)(C)SC)C2)=O)cn2ccccc2n1 C1(CN(C(CCN(C)CC)=O)C)CCCN(C(=O)C(O)c2ccsc2)C1 C(=O)(C1=CC2CCC(C1)C2)NCC1CN(C(C2CCOC2)=O)CC(C)(C)O1 CCC(CC(=O)NCC(=O)NCC(=O)N(C(CF)CF)C)C(C)(C)C c1(C(N(CC(N2CCN(C(CCC(C)C)=O)CC2)=O)C)=O)c(N)ccc(F)c1F CCCC(CNC(=O)Cn1cncn1)NC(c1cccs1)=O C=CCC(C)(CC)C(=O)NCC(O)CCNC(c1ccnc(Cl)c1O)=O C#CCC(C)(C(=O)NCc1cc(F)ccc1C)NC(C1CC2CCCC2C1)=O C(=O)(C(C)C(C)(C)C)N1CC(CNC(CCC#C)=O)(COC)C1 C1(SC)CN(C(=O)COc2cc(C)on2)CC1NC(c1sc(F)cc1C)=O C1(C(=O)NCCC2CC(NC(C(c3ccccc3)C)=O)C2)CCCCCC1(F)F Cc1nc2cncc(C(=O)NC(CNC(=O)C(F)C(C)(C)O)C3CC3)c2[nH]1 c1(C(C)(C)C)ccc(C(=O)NCC(C)(O)CNC(=O)C(O)C2CC2)cc1Cl C1(NC(c2ccoc2)=O)CC(O)C1CNC(=O)C(F)CC1CCOC1.C1CC1 c1(C(=O)NC(CC=C)CNC(C2C(C(F)F)C2(C)C)=O)ccn(C(C)C)c1C C(C)(C)(CCC(=O)N1CCCC(O)C1C)NC(CC=CC)=O Cc1nn(C)c(C(F)F)c1C(=O)NCCC(C)(C)NC(=O)C=CC1CCCN1C c1(OC)cc(CN2CCCC2(C)C(=O)Nc2cnn(C(C)C)c2)ccc1C#N c1(OC)cc(CC(=O)NCCC2CCN(C(=O)CN3CCC(O)CC3)C2)ccn1 C(=O)(C(C)CC(F)F)N(C(CN(C(c1c(C)oc(-c2ccccc2)c1)=O)C)C)C N1(C(C=CC=CCC)=O)CCC(CNC(c2ccn(CCOC)n2)=O)C12CC2 C1(CC(=O)NCC(CO)NC(C2CCOCC2)=O)Cn2ccnc2NC1=O c1(C(N(CCCNC(C(CC=C)NC(C)=O)=O)C(C)C)=O)cccc2sccc12 C1(O)(CN(C)C(c2cc(Cl)nn2C)=O)CCN(C(C2(C)COC(=O)N2)=O)C1 N1(CCCCCC(=O)OCC)CC2(C(=O)OC(C)(C)C)CCC2(CO)C1 Cc1ccc(-c2nc(C(F)F)nn2C2CCOC(C)(C)C2)c(O)n1 C1(C2CCCN(C(=O)CN(C)CCO)C2)(NC(c2ccc(CC)nc2C)=O)CC1 n1(COC)cc(CN(C(C)C(C)(C)C)C(=O)CC2(C)N=N2)c(O)nc1=O c1(N2CCCC(OCC)C2)nc2c(c(=NCCS(=O)CC(F)(F)F)[nH]1)COCC2 c1(NC(c2n(CC)nnn2)c2occc2C)ccc(-c2ccccc2)cc1C N1(C(C=C(C)C)=O)CC(CNC(c2nnc(C)s2)=O)C(C)(C)C1 N1(C(CS(CC)(=O)=O)=O)CCC(C)(C)C(C(=O)NC2C=CC(C)(C)CC2)C1 N1(C(=O)NC(c2n(C)ccn2)C2CC2)CCC2(CC1)C(F)(F)C21CCC1 O=C(CCCCC(F)(F)F)NCC1CN(C(C2CCC(F)(F)C2)=O)C1 CC(CC(C)(F)F)C(=O)N1CCN(C(=O)CC(C)(F)F)CCC1C C1(NC(c2cc(Br)cn2C)c2n(CCSC)nnn2)CCC=CCCC1 c1(-c2cn(CC(=O)NCc3ccccc3)nc2)cncc(OC2CCCCO2)c1 c1(SC)cscc1C(=O)NCC1(CN(C(=O)CC2CCC(C)C2)C)CC1 c1(NC(C2CC(F)CN2C(c2cc(C(F)(F)F)c[nH]2)=O)=O)cc(F)c(Cl)c(Cl)c1 C1(C(=O)NCCC2(OC)CN(C(C3CCNC3=O)=O)C2)CCCN(S(N)(=O)=O)C1 c1(OC)ccccc1NCCC(=O)NC(c1cc(C)n(-c2nn[nH]n2)n1)C N1(C(Cn2nnc(C)n2)=O)CCC(CNC(C2(CCF)CCOCC2)=O)C(C)C1 C12(NC(Cc3cc(C(N)=O)sc3)=O)CCCC1(F)CN(C(C1CCCCO1)=O)C2 C(=O)(C(C)C(C)COC)NCC(COC)NC(C(CC=CCC)C)=O C(=O)(C(CC(C)C)N(C(=O)CCCNC(C)=O)C)NCC(=O)OCC N1(CCCNC(COCCCC)=O)CCC(NC(=O)C(C2CCOCC2)F)C1 c1(C2C(NC(c3c(C)nc[nH]3)c3nnnn3C)CCC2)ccc(F)cc1 C(C)(C(N=c1ccnc(COC)[nH]1)C(C)C)NC(c1c(CC)nco1)=O C=CCC(F)(F)CNC(=O)C(C(C)C)NC(C1COC(=O)N1)=O N1(C(C2(CCC)CC2)=O)CC(NC(C2CCC(F)(F)C2)=O)C(C(F)F)C1 c1(C(C(=O)NC2CC2)N(CC(C)C)C(c2ccncc2)C)ccc(C#N)c(F)c1 Cc1c(C(=O)NC(=O)CNC(C)(CO)CC(C)C)cccc1CS(C)(=O)=O C1(C(=O)NC(C(=O)OC)C2CC2)C2CCC(C2)N1C(C1C2C=CSC12)=O C(=O)(C(CC(=O)OC)N1CCCCC1)N(CCNC(C1(COC)CC1)=O)C Cc1cc(C(=O)N(C(CNC(c2sc(=N)[nH]c2C2CC2)=O)C2CC2)C)nc(C)c1 Cc1nccc(C(=O)NCCC2(C)CCN(C(=O)C(CC(C)C)N(C)C)C2)c1O C1(CC(=O)NCC2CC(F)(F)CN2C(c2cc(O)cs2)=O)CCCCCC1(F)F c1(CC(C)C)nccc(C(=O)NCC(C)CNC(=O)CC2COCCO2)n1 CC(=O)CCC(=O)N(C1CC(C(N2CC3CC3C2)=O)C1)C N1(C(C2C(C(C)C)CCC2)=O)CC2(CCN(C(c3ccn(C)c3)=O)CC2)C1 c1(CNC(CCCN(C(C(C=C)(C)O)=O)C)=O)c(O)cccc1F c1(C(=O)NC2CCCN(C(c3c(C(C)(F)F)n[nH]c3)=O)C2)cccc(O)c1Cl C1(CC)CN(C(=O)NCC2CCCOC2C(C)(C)C)CCN(C)C1 CC1c2nccn2CCN1CC(=O)Nc1cccc(C2(C)CC2)c1 Cc1cn2ccnc(C(N3CCN(C)C4(CC4)C3)=O)c2n1 C12(NC(c3nc(CC)sc3N)=O)CCCC1CN(C(=O)C(O)c1ccco1)C2 CCC(CC)CC(F)C(=O)N1CCC(F)(C(=O)NCC2CN(C3CC3)C2)C1 N1(C(CN(C(COC)=O)C)=O)CC(C(=O)NCC2(O)CC3CCC2O3)CCC1C C1(C(N2CC(C(N)=O)(CNC(c3ccc(CC)cn3)=O)C2)=O)CC2C(C1)C2(C)C CC(CCCCO)NC(=O)CC1CC(NC(=O)CNC=O)C1 c1(NCCN(C(C2C(CCC)CCC2)=O)C)ccc(Br)c(C)c1[N+](=O)[O-] c1(C(C)=O)c(Cl)nc[nH]c1=NCC=CCNC(c1cc(C2CC2)nc(O)c1)=O c1(C(C)C)ncc(C(=O)NC2COCCC2NC(C2CCCOC2)=O)cn1 c1(CC)oc(C(N2CC(C)C2C(=O)NOC2CCC(O)C2O)=O)cc1C C(N=c1nc2c(cnn2C)c(NCc2coc(C)c2)[nH]1)C1C(C(=C)C)OCC1 C1(F)(CNC(C(CCO)N(C)C)=O)CCCN(C(=O)CC2CCCCC2)C1 N1(CCNC(N(C(c2ccccc2)CC)CC(C)C)=O)CCN(C)C(=O)C1 C(=O)(C1CCCc2cncn21)NC(C(C)C)CNC(=O)CCOC1CCOCC1 Cc1cnc(C(=O)NCCC2(NC(c3cccc(F)c3)=O)CCC2)c(Br)c1 S(=O)(=O)(c1cccnc1N1CC2(C)COCC2(C)C1)N(CC)Cc1ccncc1 C(CCCCCCC(=O)N1CCC1CNC(=O)C(c1ccc(Cl)cn1)(F)F)SC c1(C(=O)NCCC2CCC(NC(c3c(C)nc(C)o3)=O)C2)ccc(F)c(N)c1 N1(c2nc(OCC)c(Cl)cn2)C2CCCC1CN(C(=O)C(C)(C)CC(F)F)C2 C1(NC(N(C(C)CSc2ccns2)CC)=O)C2CCC(C2)C1N(C)C C1(C(N(CCNC(C2(OCC)CCSCC2)=O)C2CC2)=O)Cc2nccn2C1 O=S(=O)(c1ccc(N2Cc3cccnc3C2)c(Br)c1)NCCCn1cncn1 n1(CC)cc(CC(=O)NC(C2CCOC2)C)c(C)n1 N(C(=NCCC(=O)OC(C)(C)C)N1CCCC(C)CC1)C1CC2(CC(OC)C2)C1 c1(N(CC(C)(C)C)CCC#C)[nH]c(=NCCC(C)c2ccccc2)nc2scnc12 CC1CC(NC(c2cc(O)cc(Cl)c2)=O)CCN1C(C1C2CCC12)=O c1(C(=O)NCCN(C)C(c2ccc(O)c([N+](=O)[O-])c2)=O)cc2n(n1)CCNC2=O C#CCCN=C(NCCS(=O)(=O)CC)NCC1COCCO1 C12(NCC=CCC(C)(C)NC(c3c(C)ccnc3)n3cncn3)CCCC1CCO2 C(=O)(CC(C)(C)C#N)N1CCCC(CN(C(=O)COCc2nnc(C)s2)CC)C1 c1(CC(C(=O)NC(C)CCNC(=O)Cn2ncnn2)C)ccc(Cl)cc1 c1(C(=O)NCC23CC(NC(C(C(C)(C)C)=O)=O)(C2)C3)ccnc2ccsc12 C1(NC(=O)CC2(C(F)(F)F)CC2)CC(NC(C2CCCCC2)=O)C12CCOCC2 C(c1ccccc1OC)=C(C(=O)N(C(CC)CNC(C1CC1C(C)(C)C)=O)C)C C(=O)(C1CCc2ccccc21)N1C(C)CC(NC(C2CN(CC(F)(F)F)C2)=O)C1 c1(CC)cc(F)ccc1CC(N1CCCCC1CN(C)C(C1CCCCO1)=O)=O c1(C(=O)NCC(CC)NC(C2(OC)CCC2)=O)cn(-c2ccn(C)n2)cn1 c1(C(=O)NCCOCCNC(c2c(C)oc(Cl)n2)=O)cc2c([nH]1)CCOC2 C1(NC(c2cnc(CC3CC3)s2)=O)CN(C(=O)C2=COCC2)C2CCCCC12 c1(CC)cc(F)ccc1NC(C1(CO)CC1)=O.c12cccc(c1)C(=O)N2 C1(C(N2CCCC(CNC(C3(C)CCOCC3)=O)C2)=O)CCCC2(CCC2)C1 C1(NC(c2c(CCC)onc2C)=O)COCCN(C(=O)C(CC)N(C)C)C1 Cc1cc2cc(CN3CCNC(=O)C3C(N)=O)ccc2s1 c1(OC)ccc(-c2cc(C(=O)N(C(C)C)Cc3ccnc(Cl)c3)on2)cc1 c1(CN2CC(NC(c3cnc(C(C)(C)C)nc3)=O)C2)c(O)ccc2ccccc12 C(=O)(C1=C(Cl)CCOC1)NCC1C(C)CN(C(c2cc(Cl)cn2C)=O)C1 S(=O)(=O)(C1CN(CCSc2ccccc2)C1)N(C)CCn1cnnc1 C(=O)(C1=C(C)CCCC1)NC1CCN(c2cc(C(C)=O)nc(C)n2)C(C)C1 c1(CCCNC(=O)NCC2(CCCOC)CCCC2)ccc(F)cc1 N1(C(C(CCC)NC(N)=O)=O)CCC(C(=O)N(CCF)CCOC)C(C)(C)C1 CC(C)C(C)(CNC1(N2CCOCC2)CCSC1)NC(=O)OC(C)(C)C c1(OC)cccc(SCC(=O)NCC(CO)NC(c2scnc2C2CC2)=O)c1 C1(NC(C=CC)=O)CCN(C(C23CCC(C(F)(F)F)(CC2)CC3)=O)C12CCC2 CCC(C)(O)C(=O)NC1CC(C(=O)NCC(=O)NCC(F)F)C1 C(c1ccc2occc2c1)=CC(N1CCC(C(C)NC(c2ccns2)=O)CC1)=O c1(CN2CCC3(C(C(=O)Nc4nc(C(F)(F)F)cs4)C3)C2)cc(Br)c(F)cc1O n1(C(C)C)ccc2ccc(C(=O)NC(C)CCNC(C3CC3C#N)=O)cc12 c1(C(=O)NCC2CN(C(CCC(=C)Br)=O)C(C)C2)ccc(N(C)C)cc1F C1(CNC(=O)CCN2CCCC2=O)CN(C(c2cnc(C(F)F)cn2)=O)CCO1 C1(N(C(C(CC)C)=O)CC)CCN(C(C2(Cl)CCC2)=O)CC1 c1(CN2CCCC(C(=O)NC3CCC(CO)CC3)C2)cc(F)cc(Cl)c1 c1(OC)cc(CC(=O)NCC(C)N(C(=O)C(c2ccccn2)O)C)on1 CS(=O)C1CN(C(C2CCOCC2NC(c2cnncc2O)=O)=O)C1 c1(C(=O)NCC2CCCN(C(C3N(C)C(=O)NC3)=O)C2)ccc(C(F)F)c(F)c1 CC(C)CC(=O)C(=O)N1CCC(C)(NC(C2CC2(C)Br)=O)CC1 CP(C)(=O)C1CCCCC1C(N1CCC(NC(=O)CC2COC3CC2C3)C1)=O C(CCO)(C(=O)NCCCn1cc(CCCC(C)O)nn1)N(C)C C(CC(C)(C)C)(C(=O)N(C1CCN(C(c2nc(C)nn2C)=O)CC1)C)OC N1(C(CCN(C(=O)C(C(=O)OC)OC)CC)=O)CCCC12CCCC2 C1(CN(C(c2cc(COC)on2)=O)C)COCCN1C(C1CCOC1=O)=O CC12CC1CCN2C(=O)NCc1ncccc1C(F)(F)F c1(C(N(C2CCCN(C(C3CCCOC3C)=O)C2)CC)=O)cc(OC)cc(F)c1 c1(OC)ccc(Cl)c(C(N2CCCCC2CNC(c2ccc(C)c(F)c2)=O)=O)n1 C1(C(=O)NC(CNC(c2cnn3c2OCC3)=O)C2CC2)CCc2ccccc2O1 C1(C)(CNC(c2c(CC)n(C)nn2)=O)CC(OC)CN1C(=O)Cn1cncc1C N1(C(c2ccc(CCC)s2)=O)CCC(C(F)F)(CNC(c2c[nH]c(=N)o2)=O)C1 CC1COCCC1N(C(C1CCOC(c2cccc(F)c2)C1)C(=O)NC1CC1)C C1(C(C)NC(C(C)(C)SC)=O)CCCN(C(=O)CCOC2CCC2)C1 C(CC(C)(C)C)N(C(=O)C=CCC(C)(C)NC(=O)C(C)OCOC)C c1(C(C(=O)N(CC(C)NC(C(C2CCCCC2)NC(C)=O)=O)C)O)ccncc1 C12(CC(=O)NCCC3CN(C(C4C(c5n(C)ncc5)C4)=O)C3)CCC(CC1)OC2 c1(N2CC(F)(C(=O)NC(c3ccc(Cl)cc3Cl)C)C2)ccn2ncc(Br)c2n1 C(=O)(CCS(=O)c1ccc2c(c1)OCCO2)NC(c1nnc2n1CCCCC2)C C1(NC(C2CCOCC2)=O)CN(C(c2ccccc2CC2CCCO2)=O)CC1O CC1CN(C(c2ccc(C(N)=O)[nH]2)=O)CC1(C)CNC(=O)C(F)OC(F)(F)F c1(-c2nc(C(=O)NCC(COCCOC)O)sc2)ccc(F)c(Cl)c1 CC(C)(C)CC(=O)NCC1CN(C(c2c[nH]nc2-c2ccccc2Cl)=O)CCO1 C(=O)(C(C(C)C)NC(C)=O)N(CC(=O)OCC(F)(F)F)CCC c1(C(=O)NCC(C)(O)CNC(=O)C=CBr)cc2cscc2s1 N1(C(c2c(C)ncc(Cl)c2)=O)CC2COCCC2(NC(=O)CN(S(C)(=O)=O)C)C1 N1(C(CC(CN(C)C)O)=O)CCC(NC(=O)CCc2ccnn2C)C(O)C1 CCCCC(O)C(=O)NCC#CCNC(C1COCCN1C)=O N1(C(C(CSC)O)=O)CCCC2(C1)CN(C(c1cc(C)n(C3CC3)c1C)=O)C2 c1(N(C)CC)nc(-c2ccc(Cl)cc2)nn1C(C1(C)CC1)C N1(C(=O)OC)CCC2CN(C(=O)CSc3ccc(C(=O)OC)cc3C(C)C)CC12 Cc1nc2cccc(C(=O)Nc3cccc(N4CCCNC4=O)c3C)n2n1 N1(C(c2c(C)cc(C)s2)=O)CCCC(C)(C)C1CNC(C12CCCC(CO1)C2)=O N1(C(C2(C)CC2)=O)CCN(C(C2CC2Sc2ccccc2)=O)CC(O)C1 c1(C(=O)NC(C2CCCN2C(C2CC=CC2)=O)C)cc2cc(Cl)ccc2o1 c1(NCCCOCCC=C)ccc(S(=O)(=O)NCC2CC2(C)C)cc1Cl C(C(N)CS(C)(=O)=O)NC(c1n(C)nc(C2CC2)c1)=O CCCCC(C(=O)NCC(C)NC(c1cscc1F)=O)N(C)C C(CCC(C)C(=O)NCC1CC2(CC2)CN1C(c1nccnc1C)=O)OC c1(C(=O)NC(CNC(CCCCN(C)C)=O)(C)C)nn2cccnc2c1Cl c1(N2CC=C(CNC(C3C(C)(Br)C3)=O)CC2)ncc2ncnc-2[nH]1 CC1=NOC2(CCN(C(C3CCCN(C(C4CCCNC4)=O)C3)=O)CC2)C1 Cc1ccc2cc(C(N3CC=CC(NC(C4(P(C)(C)=O)CC4)=O)C3)=O)cnc2c1 c1(C(N2C(CNC(CCCCC=C)=O)C(C)CC2)=O)cc2c(cnn2C)nc1O N1(C(c2cc(COC)[nH]n2)=O)CCC(N(CCO)C(C2(OC)CCCCC2)=O)CC1 CC1CCC(CNC(=O)CCOc2cccc(F)c2)N(C(=O)CC2CC2)C1 c1(C(=O)NCC(C)(C)NC(C23CCC(CC2)CO3)=O)cnc(O)c(Br)c1 N1(C(c2[nH]cc(C(C)=O)c2)=O)CC=CC(C(=O)NC2C3CCCCC23)C1 CCC(N=c1ccnc(N)[nH]1)c1cnccn1.N1CCC(Oc2ccccc2)C1 C=CC1(C(=O)NCC2(CNC(=O)CC3CCOC(C)(C)C3)CCC2)CCOCC1 c1(OCC(=O)NC(C2CN(C(=O)CCC(=O)N3CCOCC3)C2)C)ccccc1O N1(C(CC(C(=O)OC)C)=O)CCCC12CCN(C(C1CN3CCCN1CC3)=O)C2 c1(C(N(C)CCc2cn(CCOC3CCOC3)nn2)=O)c[nH]c2cccc(F)c12 N1(C(CN2CCC(C)C2)=O)CCC(C(=O)NCC2=CCCOC2)C(O)C1 C(=O)(C(C)(CO)NC(=O)COC1CCCCC1)NC(C(=O)NC(C)C)C c1(OC)cccc([N+](=O)[O-])c1C(N1CC(NC(C2CN(C)C2)=O)C2(COC2)C1)=O Cc1cc(CN(CC(C)C)C(=O)NCC2CC23CC3)n(C)n1 S(=O)(=O)(c1c(F)cccc1F)N1CCC(F)(C(=O)Nc2c(I)ccc(C#N)c2)C1 C1(NC(CN(C)C)=O)CN(C(c2sccc2F)=O)CC2(CC2)C1 c1(C(=O)NC2CC(NC(C3C(c4nc(C)[nH]n4)C3(C)C)=O)C2)cnccc1C c1(NCC(=O)NC(C)CN(C)C(c2csc(O)n2)=O)ccc(C(F)(F)F)cn1 c1(CC(=O)N(CCN(C(COCC(=O)OC)=O)C)C)cnc2n1CCCC2C C1(NC(c2ccc(C(F)F)cn2)=O)CCN(C(C2CCCCS2)=O)C12CCCC2 N1(C(CC(CC)C)=O)CCC(F)C(NC(=O)CCNC(=O)Cc2ccccc2)C1 N1(C(C(N2CCCCC2)C)=O)C(CNC(=O)CCCCc2cnc[nH]2)CC2CC12 C1(O)(CN(C(C(COC)(C)OC)=O)C)CCCN(C(=O)C(=Cc2cnc[nH]2)C)C1 N1(C(C=NOC)=O)CC(=O)NC2CN(C(c3cnn(C(F)(F)F)c3)=O)CCC12 c1(C(N2C(CCNC(C3CC(=C)C3)=O)COCC2)=O)cc(O)c2ccoc2c1 CCCCCCC(C)CC(=O)N1CCN(C(=O)CNC(=O)OC)CC1CC C(=O)(C1=CC(C)(COC)C1)NC(C(=O)NC1(COC)CC1)C1CCC1 Cn1nc(CNC(C23CCC(C2)C3)=O)cc1C(=O)NC(CO)CCC1CC1 c1(OC)ccccc1OCCC(=O)N(CCC)C(c1cnc(C(=O)OC)s1)C N1(C(c2cc(CNC(Cc3cc(C)sc3)=O)no2)=O)CCCC(NC(N)=O)C1 C1(NC(CSCC(C)C)=O)COC2(CCN(C(c3cc(Cl)cc(F)c3N)=O)C2)C1 C1(C#N)(NCCCC(N2CCCC(c3onc(C)n3)C2C)=O)CCS(=O)(=O)CC1 Cc1nc2c(C)cc(C(=O)N(C(C)CCNC(=O)C(O)c3cnc[nH]3)C)cn2n1 c1(OC)cc(OC)c(CSCC(=O)OC(c2ccc([N+](=O)[O-])cc2)=O)c(OC)c1 N=c1ccc(C(=O)NCc2ncc(Br)cn2)n[nH]1.C12CCCN(C1)C(=O)c1cn2nn1 c1(N(C(CC)C(=O)N2CCCCC2)C(=O)OC(C)(C)C)ccc(F)c(Cl)c1C#N c1(NC(C(C2(O)CCC2)NC(Cc2ccc(C)nc2)=O)=O)cnc(C)nc1C C(CCCCC(=O)NCC1CCCOCC1)N(C)C(c1cc(O)cs1)=O c1(CC)cc(CC(N2CC(C(C)NC(=O)CC3CC3C)C2)=O)ccn1 c1(C(=O)NC2CC(F)(CNC(c3cnco3)=O)C2)c[nH]c2nc(Cl)ccc12 CC(C)C(CCN(C)C(C1CCC(F)(F)C1)=O)NC(C1CCCN1C=O)=O C1(CCC(=O)N(CC(C)NC(CN2CC(C)C2)=O)C)CCCN(C)C1 c1(NCc2c(OC)nsc2OC)[nH]c(=NCC(C2CC2)C2CC2)nc2sccc12 C1(C(=O)NC2CC3CN(C(C(C)OCCC(C)C)=O)CC32)CCS(=O)(=O)C(C)C1 C1(C(=O)NC2(CNC(C3CCS(=O)(=O)C3)=O)CCOCC2)CN2CCC1CC2 C1(C(=O)O)CCc2n[nH]cc2C1.c1(CC(=O)NC(CN(CC)CC)C)c(C)n[nH]c1C N1(C(C2CC(C)(F)C2)=O)CCCC(F)(CNC(C2CCC3CCC2O3)=O)C1 C12(NC(c3c(Br)c(C)n(C)n3)=O)CCCC1CS(=O)(=O)C2 C(C)(CCCCCO)NC(C(Cn1ccnn1)NC(CSCCOC)=O)=O N1(C(C=CC2N(C(CCCN=[N+]=[N-])=O)CCC2)=O)CC2CCCC2(CO)C1 C#Cc1ccc(CC(=O)N(C(C)CCNC(=O)CC2CCC(C)(C)O2)C)cc1 CCCC(C)(C)CC(=O)N(CC(C)(C)CNC(c1cncc(OC)n1)=O)CC c1(CC(=O)NCC(C)NC(C(CCC)C#N)=O)cc(Cl)c2c(c1)OCCCO2 c1(C(=O)NC2CC(NC(c3cc(Cl)c(Cl)c(Cl)c3)=O)C2)ccc(F)c(F)c1F c1(NC(N2CC(O)CC2C2CCC2)=O)nc2c(s1)CSCC2 c1(C(N2CCC(Cn3cc(C=CC)nn3)C2)=O)cc(OC(F)F)cc(Br)c1 c1(C(=O)NC(CCCC)CNC(=O)C(C2CCCCC2)O)cc2cn[nH]c2cn1 C1(CCC)CN(C(=O)CCC2CCCC2)CC1NC(C1(n2cnnn2)CC1)=O O=C1NCCN(C(=O)Nc2n[nH]cc2Br)C1c1ccccc1OC(F)(F)F CC(CC(=O)N1CCC(CNC(=O)Cc2cccnc2O)CC1)C(C)(C)C C(C(O)C(=O)N1CC(O)(CN(C)C(C2(F)CCOC2)=O)C1)SC C12(CNC(c3c(C)occ3)=O)CCC(C1)N(C(=O)CCN(C1CCCCC1)C)C2 N1(C(c2c(C)cc(C)o2)=O)CC(CNC(=O)C(C)Cn2ccnc2)C(F)(F)C1 n1(CC(=O)NC(C)CN(C(=O)CCC2CCOC2)C)cc(C#N)c(O)nc1=O N1(C(C(CC)O)=O)CCN(C(c2cccc(C)c2Br)=O)CC1CC(F)F CC1CCC(CC(=O)NC2(C)CC(C(=O)NCC(CO)C3CCC3)C2)O1 c1(CC(=O)NC23C(CN(C(c4c(OC)scc4)=O)C2)C3)cccc2c1OCCO2 Cn1nccc(C(=O)NC2(CO)CCN(C(=O)Cn3nnc(=N)[nH]3)CC2)c1=O CC(C)C(F)(CNC(C1C(C)(C)C1(F)F)=O)C(=O)N1CCCCCC1 c1(CC(=O)NCCC2(CNC(C3CCCN(C)C3)=O)CC2)cc(F)cc(Br)c1 c1(OC)ncc(F)cc1C(N1CCOCC1CNC(=O)CCc1ccc(Cl)s1)=O C1(C2CC2)(CNC(C2CC(C)SCC2)=O)CCN(C(=O)C(F)(F)C(F)(F)F)C1 C1(CC=C)(NC(=O)COc2cnn(C)c2)CCCN(C(=O)C(C)c2ccsc2)C1 N1(Cc2sc(C)c(Br)c2)CC2C(C1C(N1CCOCC1CO)=O)C2(C)C C1(NC(CC(C=C)CC)=O)CN(c2ncnc(Cl)c2CO)CCC12CCC2 S(=O)(=O)(c1cc(C)ccc1-c1ccccc1)N1C(CCCC)CCCC1 c1(C(N2CC(NC(=O)Nc3ccc(Cl)cc3)C(O)C2)=O)ccc(O)c(F)c1F c1(OC)cc(F)c2c(C(=O)NCCCC(C)NC(C3CCC(=O)C3)=O)n[nH]c2c1 C(CS(=O)(=O)CC(F)(F)F)NC(NC(CC)C)=NCCNc1ccc(F)cc1F S(=O)(=O)(c1ccc(C(N2CCCC2(C)CNC(=O)C2=CCCC2)=O)o1)N(C)C c1(NC)ccc(C(=O)NCC2(CCNC(=O)COCc3scnc3C)CC2)nc1 CC1CCC(C)N(C(CS)C2CC2)C1.c1(C2CN(CC3CC3)C2)cc(O)n[nH]1 Cc1ccc(C(N2CCCC(C)(C(=O)NCc3ccco3)C2)=O)cc1S(C)(=O)=O C1(C(N2CCC(F)(c3cn(CC(=O)O)nn3)C2)=O)COc2ccc(Br)cc2C1 c1(C(=O)NC2CC(NC(COC3(C#C)COC3)=O)C2)cnc2ncccc2c1 c1(OC)nc(C)ncc1C(=O)NCC(C1CCOC1)NC(C1OCCCO1)=O c1(OC)ncc(Cl)c(=NCC2CN(C(=O)C(C)(C)CN(C)C)CCCO2)[nH]1 C1(CNC(COCCSC)=O)CC12CCN(C(c1cc(C)nn1C)=O)CC2 c1(C(=O)NCCNC(c2c(CCC)onc2C)=O)cc(F)c2c(c1)CCC2 C#CCC(O)C(=O)NC1COCC1CNC(c1sc(C)nc1C)=O C1(NC(CC=C(C)C)=O)CN(C(c2cc(Br)c(C)o2)=O)CC1(C)C c1(C(=O)NCC2(O)CN(C(CCSCCCC)=O)C2)ccc2cc(O)ccc2c1 S(=O)(=O)(c1ccc(=NCCc2cccnc2)[nH]c1)N1CCC(C)CC1C CCCCCCCNC(=O)C(COCC)NC(C1C2CCC(F)C12)=O c1(SC)nccc(=NC2CC(C(=O)NCc3cc(Br)ncc3Br)C2)[nH]1 C(=O)(C1=CCCOC1)NCC(=O)N(c1ccc(O)cc1O)C(=O)C(Cl)Cl.CO C1(NC(C2CC(O)CN2Cc2ccc(OCCBr)cc2)=O)CCC(F)(F)C1 Cc1cc(=NC2CCCC(C(F)F)CC2)[nH]c(NCc2nccn2C(F)F)n1 C1(CCC(=O)O)(NC(=O)CSC(F)F)CCOC1 N1(C(CC2C=NN(C)C2=O)=O)CCC2CCN(C(=O)COCc3nc[nH]n3)CC12 C(C)(CCC(=O)NC(C1CN(C(=O)CN2CCC(=O)CC2)C1)C)SC c1(C(=O)Nc2ccc(NCc3c(OC)cccn3)nc2)sc2nccnc2c1N c1(C(=O)NCC(C)(C2CC2)NC(C(CC(C)C)F)=O)occ2c1CCOC2 c1(NC(C2(C(=O)OCC)CC23CC3)=O)cccc(SC(CC)C(=O)N(C)C)c1 C1(C)(C(=O)NCC(C)(C)C(F)F)CCN(C(C2CC(O)C2)=O)CC1 N1(C(C2CC(=O)NC2)=O)CCCC(N2CCOCC2)C1.c12ccc(cn1)[nH]2 c1(C(=O)NCCN(C(CC(C)OC)=O)CCc2ccccc2)c(C)[nH][nH]c1=N C(c1ccc([N+](=O)[O-])s1)=CC(N1C(C)CC(NC(=O)CCC(N)=O)CC1)=O c1(C(c2n(CC)nnn2)NC2(c3ccc(Br)cc3)CC2)nc(OC)ccc1F CC(C)C(CC(=O)N=c1cc2c(Br)cccn2[nH]1)c1ccon1 C1(CNC(c2cc(Cl)ns2)=O)CN(C(=O)Cn2cccnc2=O)CC2(CCC2)O1 CCCCS(=O)(=O)NC(C(=O)N(C)CCNC(=O)C=C(CC)CC)C(C)C CC(CCC(C)(C)C)C(=O)NC1CC(CN=c2[nH]nco2)C1 C(=O)(CCCCC1CC1)NC(c1ccccc1OC)CNC(COCCCC)=O c1(C(C)OC)nc(C(=O)NCC2CC(NC(C3CC3(F)Cl)=O)C2)cs1 C1(C)(NC(C(C2CCCCC2)C)=O)CC(NC(C2CCC2(C)C)=O)C1 c1(C(=O)NC(C2CCN(C(=O)C=CSC)C2)CC)cc(-c2ccccc2)[nH]n1 c1(OC)cccc(C(C)CC(N2CC(CNC(c3cc(C)c[nH]3)=O)C3CC23)=O)c1 C1(C(N(C2CCN(C(c3ccc(C)c(O)n3)=O)C2)CCC)=O)CCCCNC1=O Cc1ccc(NC(=O)C(C)OC2COC2)c2nccn12 C=CC(C)N=c1[nH]c(N(CC(C)COCCOC)C)nc2c1CCCC2 c1(C(c2n(CCOC)nnn2)NCCC(F)(F)F)ncc(C)n1C c1(NC(CNC(CN(c2ccnc(C(N)=O)n2)CC)=O)=O)ccc(OC)cc1 c12ccc(Cl)cc1CN1CCN(CC1)C2.c1(C(=O)NCCCOCC)cccs1 C1(C(=O)NCC=CCCOC)CN(C(C2C3CC(=O)CC23)=O)C(C)(C)C1 c1(C(CC)=O)ccc(OCC(=O)NCCCCNC(=O)C(CO)N(C)C)cc1 Cc1sc(C)c(C(=O)NCC(C)(C)NC(=O)CCc2ccc(C#N)cc2)c1C N1(c2cc(N3CCC(CCNC(C)=O)CC3)ncn2)CCC(C)(C2CC2)C1 N1(C(c2c(C)nccn2)=O)C2CCC1CC(CNC(C1(C)C=CCCC1)=O)C2 C1(N(C(C)=O)C)CCN(C(=O)Cn2cnc(NS(=O)(=O)N(C)C)n2)CC1C n1(Cn2c(C)cc(C)n2)c(CC2CCC2)nnc1N(C)OC1CCCC1 CCC(CC)(CCNC(=O)C(C1CCCO1)C1CC1)NC(=O)CCCN(C)C C1(C)(NC(C(CC=C)CNC(c2ccccc2CC#N)=O)=O)CCC(=O)NC1=O c1(C(N(CC(C)N(C(c2c(C)nc(CO)o2)=O)C)C)=O)ccc2occ(C)c2c1 n1(CCCC)cc(C(N2CC(CNC(c3ccn(C)c3)=O)C(O)C2)=O)c(C)n1 n1(CC)nnc2c1C(C(=O)NC1CC(F)C1)CN(C(=O)CN1CCNC1=O)C2 C(=O)(C1=CC2(CN(C(c3cnnn3C3CC3)=O)C2)OC1)NCC(CC(C)C)OC CCCCCCC(=O)NCCCC(O)C(=O)NC1CN(C)CCCC1 Cc1cc(F)c(CNC(=O)C(=O)NCC2C(C)CCC(=O)N2C)c(F)c1 c1(SC)ccc(C)c(C(=O)NCC2CC2CNC(C2CCC(C)C2)=O)c1 CC1=C(C(=O)NC2CCCC2NC(c2cc(C)sn2)=O)C(C)(C)CCC1 N1(C(C2N(C)C(=O)OC2)=O)CC(O)C(O)C1CNC(c1ccnc(C(F)F)c1)=O c1(C(=O)NC(C(C(C)C)NC(c2cn(CC(N)=O)nn2)=O)C)c[nH]cc(Cl)c1=O C1(CNC(Cc2c(C)cnn2C)=O)CN(C(C2(C(=O)OC)CC2)=O)CCN1C C1(C(=O)NCC(C)CN(C)C)CC(NC(c2ccn(C)n2)=O)CCO1 c1(NC(=O)CC2CCCC3CC23)cccc(CNC(c2cncc(Cl)c2)=O)c1 C1(C(=O)NC(C)(CNC(c2c(F)cccc2Cl)=O)C2CC2)CC(C2CCCC2)C1 N1(Cc2scc(OC)c2Cl)CCCC2(CC2C(=O)O)C1 CCC(C)(C(=O)NCC1CN(C(c2[nH]c(C)c(C(C)=O)c2C)=O)CC1C)C(N)=O C#Cc1cc(C(=O)NC2CC(CNC(C3CC3c3ccc(F)cc3)=O)C2)cc(N)c1 C1(C(C)NC(CC(=O)NCC)=O)CN(C(=O)C(c2ccc(Cl)cc2)C)CCO1 Cc1csc(Cl)c1C(=O)NCC(C)(CO)NC(=O)Cn1cc(C2CCOC2)cn1 c1(OC)ccccc1CN1CC(NCCCN2CCCC2=O)C1 Cc1cc(C(=O)NCCC(C)NC(C2COCCN2C)=O)nn1CCO S(=O)(=O)(CC(=O)N(CCCN(C)C)CCNC(=O)C(C)n1cccn1)NC C#CC1(O)CCN(C(=O)C(C2CCC2)NC(=O)CSC(C)(C)C)C1 c1(N2CCC(CNC(C3C(=C)C3)=O)C2(C)C)nc(Cl)nc2[nH]c(O)nc12 C=CCN=C(NCc1ccc(CO)cc1)N1CCN(Cc2ccccc2)C(C)C1 C1(C(N2CC(CNC(COCCCCC)=O)C(C)(C)C2)=O)CC2(COCCO2)C1 N1(C(C(C)(C)SC)=O)CCC2CCN(C(C3(C)CC4CCC(C3)S4)=O)CC2C1 N1(C(Cn2ncc(C(C)=O)c2)=O)CCN(C(c2cnc3sccn23)=O)CCC1C C(N=c1nc2c(ncn2C(C)C)c(N2CCNC(=O)C2)[nH]1)C1C(C)CCC1 Cn1ccc(S(=O)(=O)NC2CCCCC2C(=O)Nc2ncc(Br)cc2O)n1 CCCCCCCCOCC(=O)NCCCN(C(C1ON=C(C)C1C)=O)C1CC1 N1(C(COC)=O)CCCC(NC(=O)CSc2cn[nH]c2)C1 C1(C(=O)NCc2c(C(=O)NC(C)Cc3ccoc3)con2)CC2CCC(C1)C2 C1(NC(C=NOC)=O)CC1C1CCN(C(C2CC(c3cnn(C)c3)=NO2)=O)CC1 CCC(O)C(C)(C)C(=O)NCCCN1CCN(C(=O)CC23CCCC2C3)CC1 C#CCC(CC(F)F)C(=O)C(C)=O.c12cccc(c1)C(=O)N2.C(CCCO)O N1(CC(=O)NC2CN(C(=O)C=CCF)CC3(CC3)C2)CCc2ccccc2C1=O Cc1oc([N+](=O)[O-])cc1C(N1CCC(C)(NC(=O)C(N2CCCC2)C2CC2)C1)=O c1(C(N2CC(CNC(=O)CC3(N4CCCC4)COC3)C2)=O)cncc(F)c1 Nc1ccc(NC(=O)NC2(Cc3cn(CCO)nn3)CCCCC2)c(F)c1F c1(OC)ccc(F)cc1C(N1CC(NC(C2CCS(=O)(=O)N2)=O)C2(CC2)C1)=O C1(OC)COCCC1NC(=O)C(C)(C)CN(C)C(c1csc(C)n1)=O C1(NC(=O)NCC2CC(OCC)C23CCC3)C2C3CC4C5CC(C1C35)C24 N1(CC(=O)NCCCN(C(C(=O)NC(C)C)=O)CCO)CCCCC(O)C1=O C1(C(=O)NCCN(CCOC)C)COCCC1NC(c1ccnc(OC)c1)=O N1(C(CCC#C)=O)CCC(c2cc(CNC(=O)Cc3ccn(C)n3)on2)CC1 N1(C(CC2CCC(=O)N2)=O)CC(C(F)(F)F)CCC1C(=O)O C(=O)(CCCCCc1ccccc1)N1CCCC(NC(C(C)O)=O)C1 C(N=c1[nH]cncc1I)C1CCCN(C(c2ccn(CC(F)(F)F)n2)=O)C1 C#CC1(C(=O)NC2CCCC2NC(=O)CNC(=O)NCC(F)(F)F)CCC1 c1(C(N(C)CCNC(C2(CF)CCC2)=O)=O)cc(-c2ccccn2)cc(F)c1 C1(NC(=O)C2CC2)CN(C(=O)CCCc2cccc(Br)c2)C2(CCOCC2)C1 C1(C(C)NC(C2CS(=O)(=O)C2)=O)CCN(C(=O)CCOC2CCC2)CC1 n1(CC)cnc2c(N3CCC4(CC(OC)C4)C3)nc(=NCC(C)CSC)[nH]c12 C1(NC(C2(C=C)CCCCC2)=O)CN(C(=O)C=CCC)CC12CCC2 Nc1cc(F)cc(C(N2CCC(NC(c3ccnc(S)c3)=O)C(O)C2)=O)c1F C12(C(N(CC=C)C)=O)CCC(NC(=O)C(C)CCC)(CC1)C2 C(=O)(C1COc2ccccc21)NC(CC=C)CNC(C1CCC(C)CC1)=O C=C(C)CC(C)C(=O)N1CCCCC(CNC(=O)CC(C)(C2CCC2)N(C)C)C1 N1(C(c2n(C)ncc2)C(=O)NCc2ccccc2Br)CCSCC1(C)C c1(NC)cnc(C(N2CCOCC2CNC(c2ncsc2C(C)C)=O)=O)cn1 c1(C2(C(N(C3CCN(C(c4cc(C5CC5)ns4)=O)C3)CC)=O)CC2)ccccc1 Cc1cc(C(c2nnnn2CCCF)NCCCC(C)(C)OC(C)C)c(C)s1 Cc1cccc(C)c1C(O)C(=O)NC1CCN(C(c2c(C)noc2C)=O)CC1O c1(OC)ccncc1CC(=O)N(C1CN(C(=O)CC(=O)NC2CC2)C1)C C(C(O)C(=O)N1CC=CC1CNC(=O)CC1CC1)OC C1(C(N(CC(CC)C)C)=O)CCCN1NC(=O)CC1(C#N)CC1 C1(C(N2C(C)(c3ccccc3)CC(O)C2)=O)COC2C(O)COC12 CCC(F)(F)C(=O)NCCC(C(=O)N1CCCC(C(C)(C)C)C1)OC C1(N(C(=O)C#CC(=O)N(C)C)C)CC2CCC(C1)N2C(=O)CCC(F)(F)F N1(C(c2[nH]c(=N)sc2)=O)CC2(NC(c3cccc(SCC#N)c3)=O)CC1C2 C1(C(=O)NC(C(C)NC(c2ncoc2C2CCC2)=O)CO)CCCN(C(N)=O)C1 c1(C(C)NCc2c[nH]nc2C(F)(F)F)cccc2nc(-c3cccnc3)[nH]c12 C(=O)(C1=CCCN(C(c2ccc(Cl)s2)=O)C1)N1CCC(O)(C(N)=O)C1 c1(C(N2CCN(C(c3cnn[nH]3)=O)CC2CO)=O)cncc2cc(Cl)ccc12 N1(C(C(c2cccc(F)c2)C)=O)CCC(C)(C)C(CNC(=O)C(C)N(C)C)C1 C12(C(N3CCCC(N(C(c4cncc(C=C)c4)=O)C)C3)=O)CCC(=O)N1CCS2 N1(C(=O)CC2(c3ccccc3)CC2)CCC(C2CCN(C(=O)C=C(Cl)Cl)C2)C1 c1(C(=O)NC(C(C)NC(=O)C2=NNC(=O)CC2)C)ccc2c(c1)CCCCN2 c1(OCC)nnc(CN(C)CC2CCN(C(=O)C(C3CCC(=O)N3)C)C2)s1 c1(C(=O)NCC(CC=C)NC(c2cccc(OC)c2)=O)cc(C)n(C(C)C)c1 C(C)(CCC(=O)N1CC(CF)(NC(=O)C=CC2CCCC2)C1)OC C1(CNC(c2sc(CC)c(C)c2)=O)(NC(=O)CCCCC#N)CCC(F)(F)CC1 N1(C(C2CC(CNC(C(CC)(C)C)=O)C2)=O)CCCC2(CCOC2)C1 c1(CC)cccc2c(CC(N3CCCC3CC(=O)NCC3CC3F)=O)c[nH]c12 c1(C(N2CCC(N(C(c3c(CC)occ3)=O)CC)C2)=O)coc([SH](=O)=O)c1 CN1CCC(C2(C(N3CCC(C)(NC(C4CCS(=O)(=O)C4)=O)CC3)=O)CC2)CC1 C(CCC(C)(C)C(=O)NCC#CC(=O)N(CC(F)Cl)C)OC C12CC(C(O)C1)NC(=O)c1coc(n1)C(=O)NC2.C1(COC)CC1C(=O)OCC c1(OC)cnc2[nH]c(C(=O)NCC3CCN(C(C4(NC(N)=O)CC4)=O)C3)cc2c1 CCC(C)(CO)C(=O)NCC1CCN(C(=O)Cn2ccnc2C)C1(C)C O=C1CC(=O)CC(C(N2CCC(O)(Cn3cc(CC(O)C4CC4)nn3)C2)=O)C1 N1(C(C=CCCC)=O)CC(C(=O)Nc2cccc(OC)c2CO)C(C)(C)C1 N#Cc1cnc(N2CCC3(CN(C(=O)Cc4cnoc4)CCO3)C2)c2sccc12 c1(OC)nc(Br)ccc1C(N1CCC(O)C1C(=O)NCc1nn[nH]n1)=O c1(CCNC(=O)N(c2cnn(CC3CCOC3)c2)C2CC2)c[nH]c2c(Br)cccc12 N1(C(c2ccc(OCC)nc2)=O)CCCC(OC)(NC(c2ccnnc2)=O)C1 Cc1ccc(F)c(C(N2CC(C)(CNC(C3(C)CCOCC3)=O)C2)=O)c1Br Cc1cncc(NC(=O)CNC(=O)CN(C)C)c1.N12CC=CC(C1)C2=O Cc1cc(NC(c2cnn3c2OCC3)=O)ccc1NC(=O)Cc1ccsc1Cl c1(C(=O)NC2CCC2CNC(c2c(F)cc(F)cc2F)=O)scc2c1OCCO2 c1(C(N2CCC(C)C2CNC(C2(O)CC2)=O)=O)ccc2nccnc2n1 c1(CC)cc(C(=O)N(CC(C)NC(C2CC23CCC3)=O)C)c(C)nn1 N1(C(C=C(C)c2ccco2)=O)CCC2(CCC(NC(=O)CO)CC2)CC1 C(=O)(CCS(=O)(=O)C1CCCC1)N1CC(C)C(CNC(=O)CCCCC2CC2)C1 c1(OC)nc(C)ncc1C(N1CCCC1C(C)NC(c1sccc1C)=O)=O CONC(=O)C(=O)N(CC(=O)N(CC(C)C)CCO)C N1(C(c2cccc(SCCC)c2)=O)CC(NC(=O)C=CC(C)C)CC(C)C1 C1(C(=O)NCC2CCN(C(c3cc(C4CCC4)no3)=O)C2)CCCCS1(=O)=O C=CC1(C(=O)N(CC(O)CNC(c2nn(C(F)F)cc2Cl)=O)C)CCCCC1 O(NC(=O)C(CO)NC(=O)C(c1cnn(C)c1)=O)CC(=C)Cl C1(CNC(CN(C(=O)C(C)CN(C)C)C(C)C)=O)COCC1O CC1(CNC(=O)C(O)CC2CCCCC2)CN(C(=O)CCCC(N)=O)CCO1 C(=O)(C#CC1(C)CCCO1)N1CCN(C(C(CC)NC(N)=O)=O)CC1C C1(C(=O)NCc2c(C(N(CC(CC)OC)C)=O)[nH]cc2)CC(=O)N(CC)C1 c1(OC)ccc2cc(NS(=O)(=O)C=Cc3ccccc3)ccc2c1 c1(CC)n[nH]c2c1CN(Cc1ccc(OC)cc1OCC(F)(F)F)C2 N#CC1(C(N2CC3(CCN3C(C3(O)CCC3)=O)C2)=O)CC12CCC2 c1(OC)ccc(C=CC(=O)NC(CO)C(C)NC(C2CC2C(N)=O)=O)cc1F N1(C(C(CC=C)OC)=O)CCC(C2CCN(C(=O)CCCC3CCC3)CC2)C1 Cc1c(C(N2CC(F)(C(=O)NOC(CO)C(C)C)C2)=O)ncn1C C1(CC(=O)N(CC(C)N(C(=O)CCc2nc(CC3CC3)no2)C)C)CC2CC2C1 Cc1cc(C(=O)N(C)CC2(O)CCN(C(=O)C(C)(C)N(C)C)CC2)cnc1C c1(C(N2CC(CC=C)(NC(C3CC3F)=O)C2)=O)ccc(Cl)c(O)c1 Cc1cnn(C)c1CC(=O)NC(C1CCCN(C(c2cc[nH]c2C(C)C)=O)C1)C N1(C(CCC(C)=O)=O)CC2CCC1C(CNC(c1ccoc1C)=O)C2 c1(C(=O)NCC2CC(OC)CN2C(c2cc(O)ncn2)=O)cc(F)cc(F)c1O c12cc(n(C(F)F)n1)NC2=O.N1(C(C(N)=O)=O)CCC(NCc2ccccc2)C1 C12(C(N3CCC(O)(CC)C3)=O)CC(C)(CN1C(C1CCCCO1)=O)C2 C12(C(N3CCCC(CN(C(=O)C(F)C4CCCC4)C)C3)=O)CCCN(CC1)C2 CC#CC1CCN(C(C2C=CCN2C(c2ccc(OC)s2)=O)=O)C1 Cc1cc(C(=O)NC(C)CCN(C)C(c2ccnn2C)=O)c(C)cc1Cl Cc1ccc(C(=O)NCCC2CSCCN2C(=O)C(F)C2CCCC2)cc1C N1(C(C(C)Cc2cnc[nH]2)=O)CCCC(N(C(=O)C(C)n2cnnn2)C)C1 N1(C(c2c(CC)n(C)cc2)=O)CC(NC(c2ccc(CO)c(F)c2)=O)C(C)(C)C1 Cc1ccc(F)c(C(=O)NC(C)(C)CCC(=O)NCC2CC(N(C)C)C2)c1 C12(NC(C(C3CCC(=O)N3)C)=O)CCC(CC1)N(C(=O)C(C)(F)F)C2 N1(CC)CCN(CC(N2CCCC(N(C)C(C3(C4CCCO4)CC3)=O)C2)=O)CC1 c1(CNC(=O)NC2CCC(C)C2)ccc(Cl)nc1 C1(CNC(C)=O)CN(C(C2CC(C)CO2)=O)CC1C Cc1cn2c(n1)C(CC(N1CC(C)N(C(=O)OC(C)(C)C)CC1C)=O)CCC2 N1(C(=O)CCn2cc(-c3ccc(Cl)cn3)nn2)CCCC(C2CC2(F)F)C1 c1(OC(COC)=O)cc(C)ccc1CN=C(NCC1CCC(C)O1)NC1CC1 c1(N(C)CCc2cccs2)ncccc1S(=O)(=O)N1CCC(C)(CCO)C1 C1(O)(C(=O)NC(C(=O)NCCOCCOC)Cc2cn[nH]c2)CCSCC1 C1(=CC(=O)NC(C2CCN(C(=O)Cc3ccno3)C2)C)CCOCC1 c1(C(=O)NC(c2ccnn2C)C(=O)NCC2CCC(C)C2)cc(O)nc(O)n1 C1(C(=O)NC(C)CNC(c2ccc(CC#N)cc2)=O)Cc2nnsc2S1 C1(C(N(C(C)COC)CC=C)=O)CCCC1CNC(=O)C(C1(O)CCCC1)F c1(C(=O)NCC(C)(CNC(C2CC23CCOC3)=O)OC)c(C)[nH]c2ccccc12 N1(C(C(C(C)C)NC=O)=O)C2CCC1CN(C(=O)C1=CC3CCCC13)CC2 c1(OC)cc(C)cnc1C(=O)NC(C)(C)CCCNC(C1(O)CCSC1)=O Cc1cc(C(=O)NC2CCCCC2NC(=O)CCC2CC2C)nnc1C c1(C(N2C(CN(C)C(C3CC34CCOC4)=O)CCC2)=O)cccc(C#CCO)c1 N1(C(C(OC)OC)=O)CC2(C1)CN(C(=O)CC1CCN(C)C1=O)CC2CO C(=O)(C(C)(CSC)NC(=O)C(CC)C1CC1)N(CC#C)CCOC c1(C(=O)NC(CCCC)CNC(=O)COCCOC)cc(C)c(Cl)cc1OC c1(C(N(C)CC2(CNC(C3CCCC(O)C3)=O)CC2)=O)cc2c(F)cccc2[nH]1 C1(C)(C(N(CC(CN(C(=O)CN(c2ccccc2)C)C)O)C)=O)C=CCCC1 c1(C(=O)NC2C(CNC(c3c[nH]nc3C(F)(F)F)=O)C2)cccc2cnsc12 C12(CNC(c3c(C)nc(C)s3)=O)CC(NC(=O)CN3CC(=O)NC3=O)(CCO1)C2 N1(n2cc(C)nn2)CCN(C(=O)Oc2ccccc2C)C(CO)C1.Cc1nnco1 C12(C(=O)NCCC(C)CCNC(=O)C(C)(C)F)CCC(C(F)(F)F)(CC1)C2 N1(C(C(C)=C2CCCC2)=O)CC(CNC(=O)C(C)Cc2cnc[nH]2)OC(C)(C)C1 c1(CCOC)cc(C(=O)N(C)CC2(CNC(C3C4CCCC34)=O)CC2)no1 C1(C(=O)NCc2occ(C(=O)NCc3cc(C)ns3)c2)CCC2(CC1)CC2 C=C(C)C(C)(C)C(=O)NCC(C1CCN(C(C2(C#N)CCOC2)=O)CC1)(C)O c1(OC)ccc([N+](=O)[O-])c(CC(=O)NCC(C)NC(C2C=CS(=O)(=O)C2)=O)c1F c12ccc(c(Cl)c1)S(=O)(=O)N2.C(CC(C)N1CCCC1)NC1C(CC)C1 C1(CC)CCN(C(=O)CCN(C(C2CC3(CCCO3)C2)=O)C(C)C)CCO1 N1(C(C(C)=C(CC)C)=O)CC(C(=O)NCC2(CCO)CC2)C(F)(F)C1 N1(C(C(c2cccnc2)NC(=O)C=CCN2CCC2)=O)CCCc2occc2C1 N1(C(C(=O)N(C(C)CS(C)(=O)=O)CC)=O)CCC(C(c2ccccc2)C)CC1 CC1CCC(CNC(c2cc(N)ccc2F)=O)N(C(c2cc(Cl)cnn2)=O)C1 N1(C(c2c(C)ocn2)=O)CCC2C(NC(c3ccnc4[nH]cnc34)=O)C2CC1 C(N=c1[nH]c(=NC2CC3(CCC3)C2OC)c2sccc2[nH]1)C1(COC)CC1 C(CNC(c1nc(C)oc1C)=O)(C(C)C(C)C)NC(C1(NC(C)=O)CC1)=O c1(NC(=O)C=CCN2CCCC2)nccc(=NCCC2CCS(=O)(=O)C2)[nH]1 C1(N(C(COCCCC#C)=O)C)CN(C(=O)Cc2cnc(C)nc2O)CC12CC2 C(=O)(C(COC)(CC)CC)NCC1C(C(N(CCCC(CC)CC)C)=O)C1 Cn1c(C(=O)NCC2(NC(=O)CCC3CCC(=O)NC3)CCOCC2)nnc1S N1(C(CCCS(N)(=O)=O)=O)CCC2(CC1)OCCC2NC(c1occc1Cl)=O C(=O)(C1=NOC2(CCOC2)C1)N1C2C(NC(=O)Cc3c(F)cccc3F)C(C2)C1 C1(NC(c2n(C)nc(C(F)F)c2)=O)COC2(C1)CN(C(C1(F)CCOCC1)=O)C2 C12(C(N3CC(C)C(NC(=O)C(C)C(C)(F)F)C3)=O)C3CC(CC13)C2(F)F C=C(C)C(C)(C)C(=O)N1CC(NC(c2cc(Cl)c[nH]2)=O)CC(O)C1 c1(CNC2CC(C(N3CCOCC3)=O)C2)cc(Cl)cc(Br)c1 C1(CC(=O)OC)COCCN1C(C1(O)CCN(S(=O)(=O)CCCCl)C1)=O c1(C(N(CC(CNC(C(Cc2ccc(C)cc2)C)=O)O)C)=O)ccc([N+](=O)[O-])[nH]1 N1(C(c2cnn(CC)n2)=O)CC2CC1CN2Cc1ccc(C)cc1 n1(CC(N2C(C(C)(C)CNC(=O)C(F)=CCCF)CCC2)=O)cccc(N)c1=O C12(C(=O)NC3CC(CNC(C(F)=CC)=O)CC3O)CC3CC(CC(C3)C1)C2 Cc1ccc2oc(C(=O)NCC(C)(C3CCC3)NC(C3CCCS3)=O)cc2c1 Cc1ccc(C)c(OCC(N2CCN(C(=O)CC3CCCSC3)C(CO)C2)=O)c1 CC1CCc2nc(N3CCCCC(C)C3)[nH]c(=NCCS(=O)(=O)N(C)C)c2C1 c1(C(=O)NC2CC(C)OC2)cccc(-n2cc(CN3CCCC3C(=O)O)nn2)c1 CC(C)S(=O)(=O)CC(=O)N1CC2(CCN(C(=O)CC(c3ccccc3F)C)C2)C1 c1(C(COC(C(C2CC2)OC)=O)O)ccc(C)cc1 C1(C2CC2)(CNC(C(COC)(C)C)=O)CCN(C(c2c(C)cccc2C)=O)C1 O=C(C1Cc2ccccc21)NCC1CCN(C(C2CC3(CCC3)CO2)=O)CC1O CCC(C)C(C(=O)N1CCCC(C#N)C1)N1CCOCC1 Cc1nn(CC(=O)NCc2cc(C(=O)NCC3(CO)CCCC3)on2)c(=O)o1 c1(C(N(C2CCN(C(CSCC(C)C)=O)C2)C)=O)cc(O)nn1C c1(CNC(C2C(OC)C2)=O)ccc(C(C)NC(c2cn(C(C)C)cc2C)=O)cc1 S(=O)(=O)(c1ccc(C)cc1)CC(=O)NC(CN1CCN(C(C(CC)F)=O)CC1)C C(=O)(C(C)C(O)C(C)C)NCC1CCC(NC(C2(OC)CCCOC2)=O)CC1 c1(OC)cc(C(C)NCC(c2ccc(Br)cc2)O)c(O)c(Br)c1 c1(C(=O)NCC2C(NC(c3nccc(N)c3)=O)CCC2)cc2cnc(Cl)cc2s1 N1(C(C(C(C)C)n2cnnc2)=O)CCCCC(CNC(c2cccc(CO)n2)=O)C1 N1(C(C(C)SCCCC)=O)CCCC(C)(NC(c2cnn(C)c2F)=O)C1 c1(CNCC(COc2c(SC)cccc2)O)c(Br)nc(C)n1C N1(C(CCC#CC)=O)CCCC(C)C1CNC(C1(NC(N)=O)CC1)=O C(=O)(CC(C)(C)NC(=O)C(F)OC(F)(F)F)NC(c1nc(C)[nH]n1)CO c1(OC)ncccc1C(N1CCOCC1CC(N1CCC(C(F)F)C1)=O)=O CCCC(F)C(=O)N1CCSCC1C(=O)NC1CC2CC2C1 N1(C(c2cc(C)nc(C(F)F)n2)=O)CC(C)Cc2cc(Br)cnc21 C(CC1CCOCC1)(C(=O)N(C)CC1CCCO1)NC(C=CC(=O)OCC)=O N1(C(C(C(C)C)n2cccc2)=O)CCC(C2CC2)C1C(=O)NC1CC(C(=O)NC)C1 C[S+](C)CCC(O)C(=O)N1CCCC(C)(CNC(=O)CC2CCOCC2)C1 C1(Nc2ccc(OC(CCC(=O)O)=O)cc2)CC2(C1)CC(c1nn[nH]n1)C2 c1(C(N2CCC(NC(c3cc4c(s3)CSC4)=O)C(F)C2)=O)cc(F)c(F)cc1Cl C1(C(=O)NC2CN(C(c3ncc(OCC)nc3)=O)CC2O)CC(C)(C)OC1(C)C N1(C(=O)NCC2CC3(CC(C)(C)C3)C2)CC(CCO)c2ccccc21 n1(CCC#C)c(N2CCOC(c3nnc(C)o3)C2)nnc1-c1cccc(Br)c1 Cc1ccc(CN(C2CC2)Cc2ccc(C#N)nc2)cc1C N1(C(CC2(N(C(C(C)C#N)=O)C)CC2)=O)CC(O)CC1(C)CO C(CCN=c1[nH]c2ccc(F)cc2s1)N(C(CC1(C(=C)F)CCC1)=O)C(C)C c1(CNC(N2CCCC(c3cnc(CC)o3)C2)=O)cnc(OC)cc1C C12(C(=O)NC3C4CN(C(c5cn(CC)nc5)=O)CC43)CC(C1)C(C)(C)O2 C1(NC(C2C(=C)C2)=O)CCN(C(c2cc(-c3ccc(OC)cc3)oc2C)=O)C(C)C1 C(C(C)(C)CCCNC(c1nnnn1-c1ccc(C#N)cc1)CCC1CC1)OC C1(NC(C(C)CS(C)=O)=O)CC2CCC(C1)N2C(=O)CC1CCC2(CC1)COC2 c12c(C)nn3c1CN(CC3)C2=O.c1(C(=O)NC(C)=O)cccnc1C(N)=O Cc1cccc(F)c1CC(N1CCC(CF)(NC(=O)CCNC(N)=O)C1)=O N1(C(CSC)=O)CCC(C)CC1C(=O)NCC=Cc1ccccc1 C=CCCC(C)(C)CNC(C1C=CCCN1C(=O)Cn1nnc(C)n1)=O c1(C(=O)NCCC(C)NC(CCc2cc(C)nc(C)c2)=O)ccn2c1CCCC2 c1(CC)ncncc1C(=O)NC1CN(C(=O)C(C)(C)c2cc[nH]n2)CC1OC Cc1oc([N+](=O)[O-])cc1C(=O)NCC(O)CNC(=O)C(C(C)C)N(C)C C(C(C(=O)N1CCCCC(C)C1)C(C)C)NC(C)=O c1(OC(C)C)cc(NC(C(=O)NOCCF)C2(C)CC2)ncn1 c1(SCC(=O)NCC(Cc2ccccc2)N(C(CC=C)=O)CC)ccccc1O Cc1nsc(C(N2CC(O)(C(C)NC(c3n[nH]cc3F)=O)C2)=O)c1N c1(CC)cc(C(N2CCN(c3nncs3)CC2)C(=O)NC(C)C(=O)OC)ccn1 C1(OC)CCCC1C(=O)N(CCCc1cn(CCCCF)nn1)C1CC1 Cc1cc(C(N2CC3CC(NC(c4cnc5n4CCS5)=O)C2C3)=O)cn(C)c1=O c1(C(N(CCC(C)NC(C(F)=C(C)C)=O)C)=O)c(C)ccc2c1CCCN2 N1(C(CCC=CC)=O)CC(NC(c2cc(OC)n(C)n2)=O)C(CCC)C1 Cc1cncc(C(=O)NCC2CN(C(c3ccc(CO)cn3)=O)CC2O)n1 C1(C(N2C(C)C(NC(C3CN4CCC3CC4)=O)CC2)=O)Cc2nn[nH]c2C(C)C1 C(CC(=O)N1CCC(O)(C(C)NC(C2COC(C)(C)C2)=O)CC1)(C(F)(F)F)OC c1(C(=O)NC2C(CNC(CCc3cc(C)no3)=O)C2)c(C)ccn1C c1(C(N2CC3(CC(NC(CCC(C)SC)=O)C3)C2)=O)nccc2cccnc12 N1(C(C(S(CCC)(=O)=O)C)=O)CCOC2(CCN(C(c3conc3CC)=O)C2)C1 CCCCCS(=O)(=O)CC(=O)NC1CCCN(C(c2cc(=O)n(C)o2)=O)CC1 c1(C(=O)NCCCN(C(C2CCC(C)O2)=O)C2CC2)cc(=O)c2ccncc2o1 c1(OC)cc(C(N2CC(CCNC(c3cnc(Cl)[nH]3)=O)OC(C)C2)=O)ccc1Cl C1(C(=O)NC(c2nccn2C)CC)CC12CCN(C(=O)CSC(F)F)C2 C1(CC)CCOC1C(=O)NC1(C)CN(C(C2CN(CC(C)C)C2)=O)C1 C#CC1CC2(CC2)CN1C(c1ccc(Cl)cc1C(F)F)=O c1(C(=O)OC)ccc(O)nc1N1CCC(CF)(NC(=O)CCCCCO)C1 c1(CCC)nc(C(=O)NCC2(NC(C3CCC(F)C3)=O)CCCC2)co1 C(C1CCC(C2CC2)CC1)=CC(N1C2CCC1CNC2)=O C=CC1(C(=O)Nc2ccc(CO)c(F)c2)CCN(C(=O)CCc2nccs2)CC1 C1(C(C)(C)C)CCN(C(C2CCCCC2NC(c2cn(C3CC3)cn2)=O)=O)CC1 c1(CCC(=O)N(C2CCN(C(=O)COCC3CCC3)C2)CCC)ccc(C)cc1 N1(C(CC(CCC)O)=O)CCC2(CC1)CC(NC(c1n[nH]c(C)c1C)=O)CCO2 C1(CNC(c2c(C(C)C)occ2)=O)CC(C(=O)NC(CN(C)C)CCO)=NO1 N1(C(c2cc(SC)oc2C)=O)CCN(C(c2cnc(Cl)s2)=O)CC1CF C(=O)(CC1=NNC(=O)C1)N1CCC(OC)(CNC(=O)C(C)c2cccs2)CC1 c1(C(=O)NCCC2OCCN(C(C=Cc3ncn(C)c3)=O)C2)cn2c(n1)CCC2 C(=O)(C1=C(C)OCCS1)N1CCC(CNC(CC(C(=C)C)OCC)=O)C1 n1(CC(=O)NCC(C2CCC2)NC(C2(C)CCCO2)=O)ccc2ccc(F)cc12 N1(C(CCCOC)=O)CCC(C)(C)C1CNC(c1cc(C(F)(F)F)nn1CC)=O CC1CC(NC(=O)CC2OCCC2C)CN1C(=O)Cn1cc(CO)nn1 C=C(C)CC(C(=O)NC1CCN(C(c2ccc(C3CC3)o2)=O)C1CC)OC c1(-c2ccc(C(C)NCc3ncc(C4CCOCC4)o3)cc2)ccc([N+](=O)[O-])cc1 N1(C(c2cc(OC)cc(Cl)c2)=O)C2CCC1CN(C(=O)C(C)OCC(C)C)C2 c1(C(=O)NC(C)CCNC(=O)CC2CCC(O)C2)cccc(C(N)=O)c1 c1(C(N(C(CNC(c2occ(C)c2)=O)C)C)=O)ccc(N)c2cnccc12 N1(C(C(CC)CC(F)F)=O)CCN(C(c2ncoc2C(F)(F)F)=O)CC(C)(C)C1 CCC1=NOC(C(=O)NC2CC(NC(=O)C(c3cnn(C)c3)C)C(O)C2)C1 c1(CN2CC(NC(CCC(=O)OC)=O)C(C#N)C2)cc(Cl)c(C)c(Cl)c1 CC1CCc2ccccc2N1CCN=C(NCC1CCCN1C)NCC(F)F C1(C(N(C(c2ccccc2)CNC(Cc2c(C)non2)=O)C)=O)CC(F)C(=O)N1 C=C(C)CCCC(=O)N1CCC(C2CCCN2C(=O)CCCNS(C)(=O)=O)C1 c1(C(=O)NC(C(C)NC(c2cn(CC=C)nc2)=O)CO)cc2ccccc2nn1 c1(C(=O)OCC)ccc(C(C(=O)NC)N(C)CC2CCN(CC3CC3)C2)o1 CC1(C(N2CCCC(CCNC(c3cc(N)cc(F)c3)=O)C2)=O)CCC2CC2C1 C1(C)(CNC(C(C)Oc2cccnc2)=O)COCCN(C(c2cccn2C)=O)C1 C(=O)(C(C)(O)C(C)(C)C)NCC(C(C)(C)C)NC(c1nc(C(F)(F)F)cs1)=O C1(NC(c2nc(C(C)(C)C)sc2)=O)CCCCC1NC(=O)C(F)C1CC1 CCC(C)C(C)CNC(C1COCCN1C(=O)CC(C)OC)=O c1(NC(CCCC=C)(CC)c2nnnn2C2CCCC2)ccc2oc(O)nc2c1 C1(O)(CNC(c2cscc2C2CC2)=O)CCN(C(c2ncsc2C2CC2)=O)C1 c1(N(C)C)ccc2c(c1)OCCN2C(c1ccnc(OC(F)(F)F)c1)=O C1(NC(CCN(S(C)(=O)=O)C)=O)CCCCC1NC(=O)C=CS(C)=O Cc1cc(=NC(=O)CC(C)c2ccc3c(c2)OCO3)[nH]n1C1CCCCC1 C1(NC(c2c(C)ccnc2)=O)CCN(C(=O)Cn2cncc2C)CCC1(F)F c1(NC)ncnc(NC(CNC(=O)CCC(=O)N(C)C)C(C)(C)C)c1[N+](=O)[O-] CCC(c1cccc(Cl)c1)=CC(=O)NC1CC(N(C)C(c2[nH]cnc2C)=O)C1 C(=O)(C(CC)SC)NCCCNC(C1C(C=C)C1)=O C=CCCCC(C(=O)N1CC(OCCO)C1)NC(=O)C(C1CCC1)OCC c1(CC)ccc(C=CC(=O)NC2CN(C(=O)Cc3cncn3C3CC3)C2)cc1 N1(C(COCC#C)=O)CC=CC(C(=O)N(C2CCC2)CC2CCC2)C1 Clc1c(NC2CCNC3CC23)cccc1I c1(OC(C)C)ccc(C(C)NC(=O)N(CCS(C)(=O)=O)C(C)C)cc1 c1(OC)cc(C(N2CC3CC2C3NC(=O)C(C)OCCC(C)C)=O)cc(Cl)c1 c1(NC(COC)C2CC2)nc(=NCC2CCCOCC2)[nH]c2c1CCC2 C(=O)(C1=NOC2(CCC2)C1)NCCCCC(C)NC(c1n(CCC)ncc1)=O Cc1cc(C(=O)NCC(c2ccccc2)CNC(=O)C(=O)NC2CC2)c(C)cn1 C1(NC(CC2CC(=C)C2)=O)CN(C(c2cnc[nH]2)=O)CC2CCCC12 C(=O)(C(F)(F)c1cccnc1)N(C(C#C)C1CCC1)C C(=O)(CCC(=O)NCC1CCCN1C(=O)CC1CCNC1=O)NC CCCN=C(NCCCC1CCOC1)NCCc1nccnc1C CCCC(C)(O)CNC(=O)CC1CCCN(C(C2(Cl)CC2(F)F)=O)C1 C1(C(N2C(C)CC(NC(=O)C(C)(O)C3CCC3)C2)=O)CCCC(C)(C)C1 C1(NC(C(C=C=C)C)=O)CN(C(C2CC(C)(C)C2)=O)C2CCCC12 c1(N2CCN(c3cc(NCC4CCCC(C)CC4)ncn3)C2)cncc2c1CCC2 C(CCCCC(=O)NC1CN(C)CC1C)OC c1(SC)cn(C)nc1C(=O)NC1CCCN(C(=O)CCc2cn(C(C)C)nn2)C1 c1(C(=O)NCCC(C)(C)NC(C(C)OCCOCC)=O)cn(C(C)(C)C)nc1C c1(NC(=O)N(C2CS(=O)(=O)C2)Cc2ccc(F)cc2Br)cccc([N+](=O)[O-])c1 N1(C(CSCC=C)=O)CC(C2(NC(c3cc(O)cc(Cl)c3)=O)CC2)C1 C1(C2(O)CCN(C(c3cccc(N)n3)=O)CC2)(NC(C(C)C2CCC2)=O)CC1 CC1CN(c2cc(N3CCC(Cc4ccccn4)C3)ncn2)CCC1(F)F N1(C(c2c(C)n[nH]c2)=O)C(C(=O)NCC2(O)CCN(C)C2)CCC1C1CC1 C1(C2OCCO2)CCN(NCC)CC1.C1(C)CC(=O)N(C2CCCC2)C1 CCCCC(C(=O)Nc1cccc(Cl)c1)N(C1CC1)Cc1ccc(C)o1 c1(CNS(c2ccc(CSC)s2)(=O)=O)nc2ccccc2nc1C c1(CN(C(C2CCOCC2)C)C)cn(C)c(=O)c2ccccc12 C1(NC(C2OCCN(C(C(C)CC(N)=O)=O)C2)=O)CC2CC1CC21CC1 c1(C(=O)NCC(CNC(C=CCC)=O)CO)nc(Cl)ccc1OCCOCC c1(NCC(=C)C)nccc(N2CCC(C)(c3cccc(F)c3)C2)n1 N1(C(c2scc(C)c2)=O)CC2COCC2(C(=O)NCC(C)S(C)(=O)=O)C1 CC1(OC2CC(C(=O)OCC3(NC(=O)CCc4ccco4)CCC3)C2)CCCC1 c1(CC(N2CC(CNC(C(CC=C)CC)=O)C3(C2)CC3)=O)c(C)cc(C)nc1O c1(CC)ccc(C=CC(=O)NCCC(C)NC(c2ncc[nH]c2=O)=O)o1 C1(C(N2CC(SC)C(NC(C3(C(=O)NC4CC4)CC3)=O)C2)=O)CCC2CC1CO2 N1(C(c2c(N)sc(C)c2C)=O)CCN(C(C2CCCC2O)=O)C2(CCC2)C1 N1(Cc2cn(CC(N3CCC(OCc4ccsc4)C3)=O)nn2)CCCCCC1=O N1(C(CC=CCC)=O)CC2CC1C2NC(C1CC1C(C)(C)C)=O C1(NC(C(CCSC)OC)=O)CCC2(CC1)CC2NC(c1ccnn(C)c1=O)=O CN=c1[nH]ccc(C(N2CC(C(N)=O)(CNC(=O)C(F)OC(F)(F)F)C2)=O)c1N c1(C(N2C(CNC(c3cn(CC)nn3)=O)CC2)=O)ccc2c(c1)NC(=O)C(C)O2 N#Cc1cc(F)ccc1CN1CCOCC(NC(c2ccccc2Cl)=O)C1 C1(C2CN(C(=O)CN(C)CCOC)C2)(NC(C2CC(CCC)OCC2)=O)CC1 C1(NC2(CNC(=O)OC(C)(C)C)CC2)CC2CCC1N2C1CCc2ncccc21 CCCC(C(=O)NCCC(O)C(=O)NCc1coc(CC)n1)OCC c1(C(=O)NC2CC(F)CN(C(=O)C=Cc3cocn3)C2)ccc2nccn2n1 N1(C(c2n(C)ncc2Cl)=O)CCC(CO)C(NC(=O)C(c2ccc(Cl)cc2)O)C1 C(CC(C)(C)CC(=O)N1CCN(C(c2cccc(CC(C)C)c2)=O)C2CC12)OC C1(SCC(N2CCC(N(C(=O)CC3(CO)CC3)CC)C2)=O)CCCCO1 C1(C(=O)NCC2(OCC)CC2)CC12CCN(C(C1CC(C)(O)C1)=O)CC2 C=C(Cl)CCC(=O)NC(C)CCN(C)C(c1cc(C)n(-c2ccc(F)cc2)n1)=O Cc1cc(C(=O)NC2CC2NC(=O)C(C)(O)Cn2c(C)cccc2=O)cnc1O c1(CC(N2CCC(COC)(NC(C3CC3C3CC3)=O)C2)=O)cccc(F)c1F C1(C(=O)NCCC#C)CN(C(=O)C(C)Cc2ccc(OC)cc2)CCO1 c1(CNC(C2(CC)CC2)=O)ccc(C(=O)NCC(C)(C)OC)nc1 N1(C(CCN(C(=O)CC2CCCC23CC3)CC2CC2)=O)CC2C3C=CC(C3)C2C1 C12(NC(c3cncnc3)=O)CCN(C(=O)CC3CCC4(CC3)CC4)CC1C2 c1(C(=O)OC)nc(N(C(C)CNC(c2cnc(Cl)s2)=O)C)ncc1Cl c1(N(C)CC2CC2(F)F)cc(S(=O)(=O)NC2CC2C(C)(C)C)ccc1C#N C(=O)(C1CCCn2cnnc21)NC1CCN(C(c2nc(C)n(C)c2C)=O)C1 C1(CC)CN(C)C(=O)CN1C(=O)C(C1CN(C(c2ccccc2OC)=O)C1)OC C(=O)(CC(C)CCc1ccccc1)N1CC2C(NC(CCOC)=O)C2C1 c1(C(N2CC(NC(CC(C=C)C)=O)C(F)CC2)=O)cc(C)nc2c(O)cccc12 C=C(C)CCCC(=O)NC1CN(C(=O)CC2CC3CCC2CC3)CC1OC c1(C(=O)NC2CC(C)(C)N(C(c3cccnc3O)=O)C2)ccc2c(c1)OCO2 c1(C(=O)NCCC(=O)N(C(CC)CN(C(=O)COC)C)C)cccc(OCC)n1 c1(C(N(CC=CC(=O)NC2(CCOC)CCC2)C)=O)cc(C(N)=O)[nH]n1 N1(C(C2C(C)(C)C(NC(c3n[nH]cc3Cl)=O)C2)=O)CCC2(CC1)CSC2 C1(NC(CNC(=O)OC)=O)CCCC1NC(=O)COC1CCCOC1 N1(C(C)=O)c2ccccc2CC1C(=O)NC1CC1CNC(c1ccc(C#N)s1)=O Cc1cccc(C)c1C(O)C(=O)N1CC(CCNC(C2CCCC(O)C2)=O)C1 N1(C(C(C)C)=O)CC2(C1)C(C(=O)NCC1CC1(C)C)CCS2(=O)=O N1(Cc2nnc(-c3occc3)s2)CCN(CCc2cn[nH]c2)CC1 c1(C(=O)NCC(=C2CN(C(C3(CC#C)CCCO3)=O)C2)F)ccccc1C N1(C(C(C)(C)C)=O)CCC2CN(c3ncncc3F)CCC12 c1(C(=O)NC(CN(C(C2CC3CCC3C2)=O)CC)C)ccc2c(c1)CN(C)CC2 c1(CC)ccc(C(=O)N(C)CC2(O)CN(C(=O)C3=CCCCC3)C2)c(Cl)c1 CCCC(CCCNC(c1[nH]nnc1C)=O)NC(=O)CCc1c(Cl)cccc1Cl c1(CNC(=O)NC(c2cccc(F)c2F)CO)nc2cccc(Br)c2[nH]1 O=C1CCCC(C(N2CCOCC2CNC(C2(CC(F)F)CC2)=O)=O)O1 C(=O)(CC(C)(C(F)F)N(C)C)N1CCCC(O)(CN(C(CC)=O)C)C1 C1(NC(c2c(CSC)nccc2)=O)CC(=O)NC(=O)C1.C1=CCNC1=O C1(CC(=O)N(C2CCN(C(c3c(C)scc3)=O)C2)C)CCNC(=O)C1 c1(NC(=O)NCCC)cc(OC)cnc1Cl Cc1cc(C(N2CC(NC(C3(C4CCCCO4)CC3)=O)CC(C)C2)=O)cc(N)c1 Cc1csc(C(C)NC(=O)C(CC2CC2)NC(C2C=CCCC2)=O)n1 c1(C(=O)NCCCN(c2ncc(C#N)cc2F)CC)cccn2nncc12 C1(NS(CC(C)c2ccc(F)cc2)(=O)=O)CCCc2ccccc2C1 Cc1nn(C)c2c(NC3CC4C=CC3C4)nc(=NCC(=O)NC3CCC3)[nH]c12 N1(C(CC2CCN(C)C2=O)=O)CC2(CCCC2)C1C(=O)NCC1(F)CCN(C)C1 CC1(O)CC2CC1CN2C(=O)NC(c1ccccc1Cl)CO CC(C)CN=C(NCC1(O)CCS(=O)(=O)C1)NCC(N1CCOCC1)C Clc1cc[nH]c(=NCCCc2cccc(Cl)c2Br)c1Cl C1(C(N(CCN(C(C(CC)O)=O)C)C)=O)CCN(c2nc(C)cs2)CC1 c1(CN(CC)CC)ccc(C(=O)NCC2CN(C(=O)C(C)(C)CO)CC2C)cc1 C1(CNC(c2ccc(C)c(F)c2F)=O)CN(C(c2cccs2)=O)CC2(CCC2)O1 C1(C(=O)NCCCCC(C)(F)F)C2CCCC2CN1C(C1CCO1)=O N1(C(C(C(C)C)NC=O)=O)CCC(CO)(NC(c2cc3[nH]ccc3s2)=O)CC1 C1(CNC(CCn2c(C)ncc2)=O)CN(C(=O)C(F)C(F)(F)F)CC(C)(C)C1 C(CC(C(=O)NCCN1C(=O)CCC1=O)NC(C1CC(C)=NO1)=O)SC n1(CC(=O)NCCOCCNC(Cc2c(C)nn(C)c2C)=O)nnc2c1CCCC2 C(=O)(C1CCc2c[nH]nc21)OC(C1CC(=O)N(c2ccccn2)C1)=O C(=O)(C1=NN(C)C(=O)CC1)NCCCC(C)NC(c1ccc(C)c(C)c1Cl)=O C1(NC(c2cn(CC=C)nn2)=O)CCCC12CN(C(c1ccc(C)c(N)c1)=O)C2 C1(CNC(C2C(CNC(c3c(CC)nn(C)c3)=O)CC2)=O)Cc2nccn2C1 c1(C(N2C(CN(C(C3(C)ON=C(C)C3)=O)C)COCC2)=O)cc2n(c1)CCC2 N1(C(C2(NC(c3c(CC)occ3)=O)CCCC2C)=O)CCC12CC(C)(CO)C2 CC(C)CC(C(=O)NCC1=CCCN(C)C1)ONC(C1CCCOCC1)=O C(=O)(C(C1CN(C(=O)COCCCF)C1)OC)NCC1(OCC)CC1 N1(C(c2ccccc2Cl)C(=O)NCCCSC)CCOC2CCN(C)CC12 N1(C(C(C)(C)C2CC2)=O)CCCC(F)(CNC(C2CS(=O)(=O)CCO2)=O)C1 CN1CCC(NC(=O)C=CI)C12CCCN(C(c1ccc(-c3cc[nH]n3)s1)=O)C2 c1(COC(C2(C)CC(C)=C(C)CC2)=O)cc(=O)oc2cc(C)c(C)cc12 C1(F)(C(=O)NCC(=O)NCc2ncn(CC)n2)CC=CCC1 CN1CCCC(C(=O)NCC2(O)CN(C(C3(C(F)F)CCCO3)=O)C2)C1 C1(C(N2CCCC(C3N(C(C(CC)(C)C)=O)CCC3)C2)=O)Cc2cccnc2C1 c1(OC(C)C)ccc(C(=O)NC2CN(C(=O)Cc3cccn3C)C3CC23)cn1 CCCCC(C)C(=O)N1CCCC1CN(C)C(C1CC12CCCC2)=O C(C(=O)N1CCCC1(C)CCCO)(C(C)(C)C)NC(CN1C(C)CCCC1)=O C(=O)(CCC(=O)N1CCOCC1CCNC(c1ccc(C(C)N)cc1)=O)NCC c1(C(N2CC(NC(c3c(C)c(Br)cnc3)=O)(CO)C2)=O)cc2c(ncn2C)[nH]1 C(=O)(CC(C)(C)N(C)C)NCC(CNC(c1cc(OCC)no1)=O)(C)O N1(C(C(=O)NC(C)C)=O)CCC2(CO)CN(C(c3scnc3Cl)=O)CC2C1 Cc1cnnc(C(=O)NC2CC(C)N(C(c3csc(C(F)(F)F)n3)=O)C2)c1 C1(NC(c2c(CNC(C3C(C)OCCO3)=O)noc2)=O)(CO)CCCCC1C N1(C(c2cccc(C#C)c2)=O)CCN(C(c2cn(CCC)nc2C)=O)C(C)C1C C(=O)(C(O)C(F)(F)F)N1C(CCCNC(Cn2c(CCC)ncc2)=O)CCC1 c1(C2C(C(N(CCNC(C(C3CC3)SC)=O)C)=O)C2)ccc(S(N)(=O)=O)cc1 CCC(CC)C(C)C(=O)NCCNC(=O)Cn1cc(C(C)O)nn1 c1(CC(=O)NCC(C)NC(c2c(NC(C)=O)cncc2)=O)ccccc1S(C)=O C1(NC(Cc2nc(NC(=O)CCCc3ccc(F)cc3)sc2)=O)CCC(=O)NC1=O c1(CC(=O)NCC(CCC)NC(c2ccc(C#N)[nH]2)=O)cccc(C)c1F S(=O)(=O)(c1ccc([N+](=O)[O-])c(Cl)c1)Nc1c(C(N2C(C)CCC2)=O)c(F)ccc1 CC1CC2CCC(C1)N2C(C1C2CCC(C2)C1NC(C1(F)CCC1)=O)=O N1(C(c2c(OC)nsc2)=O)CC2(CC(C(N3CCC(O)C3(C)C)=O)CO2)C1 CC1(C#N)CCN(C(C2CC3CC3N2Cc2ccc(O)cc2)=O)CC1 c1(C(N(C2CCC(NC(c3c(Cl)nc(OC)s3)=O)CC2)C)=O)cc(Cl)nc(=N)[nH]1 C#CCCCC(=O)N1CC(C(=O)NC(c2ccnn2C)C)(COC)C1 C1(NC(C2C=CCC2)=O)COC2(C1)CN(C(c1nocc1-c1ccccc1)=O)C2 C=C1CCC(C(=O)NCC2CC(C(=O)NCCC3(O)CCOC3)C2)CC1 C(C(CC(C)C)C(=O)N(CC(=O)NC1CC1)C)NC(c1c(C#C)c[nH]n1)=O C12(NC(C3CCCC(OC)C3)=O)CCCCC1N(C(=O)OC(C)(C)C)CCC2 C1(C(=O)NCCCNC(=O)Cc2cn3c(n2)CCCC3)CC12CCS(=O)(=O)CC2 CN1CC(C)(C(N2CC(N(C(=O)CSc3ccc(Cl)s3)C)C2)=O)CCC1=O C(=O)(CCCCC(F)(F)F)N1C(CN(C(C23OC(C)C(C2)C3)=O)C)CCC1 c1(C(C)NC(=O)OCC(N)=O)cccc(-n2ccnc2)c1 N1(C(CC2C(C)OCC2)=O)CCCC2(C1)CN(C(C13CC(C)(CCO1)C3)=O)C2 C1(CC)C(C(=O)NCCC(C)F)CCN1C(=O)Cc1cscn1 Cc1nccc(Cl)c1C(=O)NC1CC(CO)N(C(c2ccnc(Cl)c2N)=O)C1 N1(Cc2c(C)cc(OC)nc2)CCC2CN(C(=O)CCN3CCOCC3)CC2C1 c1(SC)cccc(CC(=O)NCC(C)CN(C)C(c2cnc(C)s2)=O)c1 c1(C(N2CCCC(NC(c3c(C)cncc3)=O)CC2)=O)cc2cc(N)ccc2o1 c1(C(=O)NCCC(CC)(C)NC(=O)C2=C(Cl)CCC2)ncc(Cl)cc1F c1(NC2C(F)(F)CCN(C(c3cc(CO)on3)=O)C2)ncnc2ccc(Br)cc12 N1(C(Cc2ccc(C)o2)=O)CC2CCCC(NC(=O)CSc3nnnn3C)(C2)C1 C1(C(=O)NCC(CCCC)NC(c2ncsc2C(C)C)=O)CC2CCCC(C1)C2 CC(CC=Cc1ccccc1)C(=O)N(C1CCCN(C(c2ccccc2)=O)C1)C n1(CC)cnnc1SCC(=O)NCC(c1ccccc1)NC(C1CCN1CC)=O c1(C(C(=O)NC2CC2)N(CCC)CCOC)nc(C)ccc1F C(=O)(C(CO)C(F)(F)F)NCCC1(O)CCN(C(c2c(C)n(C)nc2)=O)CC1 C1(OC)CCCC(NC(C2(NC(C3COCCC3C)=O)CC2(C)C)=O)C1 c1(OC)cccc(N(C(=O)C=CCNC(C2CCC(C)(C)C2)=O)C)c1 c1(CC)c(NC2CCN(C(C3CC4CCCCN4C3)=O)C2)nc(C)nc1Cl C1(C(=O)NCCc2c(C)n[nH]c2)(NC(=O)CC2CC(=O)C2)CCOCC1 N1(C(C(c2n(C)cnn2)(C)C)=O)CCC(O)(CCNC(c2csc(Cl)c2)=O)C1 C1(C(=O)NCC2N(C(c3c(C)n(C)nn3)=O)CCCC2)CCC(=O)C(C)C1 CCC(F)(F)C(C)(C)C(=O)NC1C=CC(C(=O)NCC(C(F)(F)F)OC)C1 c1(C(N2CC3CCN(Cc4c(Br)ccc(NC)c4)C3C2)=O)cccc2[nH]ccc12 n1(CCC(=O)NCC23CC2CN(C(=O)CC2CCOC2)C3)cc[nH]c(=O)c1=O N1(C(c2c(OC)cccc2OC)=O)CCC2(CC1)COC(C)C2 C#CCCCCCC(=O)NC(C)C=CC(=O)NC1CCc2nn[nH]c2C1 CCC(C)CC(C)N(C)C(c1sccc1CNC(c1ccccc1OC)=O)=O c1(CNCC)c(OC)cccc1C(=O)NC1CC(NC)C12CCC2 CC(C)C(=O)C(=O)NC(C(=O)NCC1(F)CCOCC1)C1CCCO1 CON(C(=O)C1=NOC(Cc2nn[nH]n2)C1)C1CCN(CC(C)(C)O)CC1 c1(NCC2(C(=O)OC)CC2)ncnc2c1ncn2CC(O)C(C)(C)CO CCCC(CC)C(=O)NCCC1(O)CCCN(C(c2cnc(=N)[nH]c2)=O)C1 Cc1ccc(O)c(CC(=O)NC(C)CN(C)C(c2ccncc2C)=O)c1 Cc1cccc(Br)c1C(C(=O)NCC(O)C(N)=O)NC(=O)C(F)C(C)(C)O CC1CC(C)(C(=O)NCC=C2CCN(C(=O)C(=O)NCC3CC3)CC2)CCO1 c1(CN2CCC(NC(c3ccc(CO)o3)=O)CC2)cc2n(n1)CCSC2 CC(C)CC(O)C(C)C(=O)N1CCC(F)(C(=O)NC(c2nccs2)C)CC1 N1(C(c2c(C)c(Cl)ccn2)=O)CCC(CNC(=O)C(O)C(C)(C)C)C12CCC2 CCC1=C(C(=O)NOCC(N2CC(O)(C(F)(F)F)C2)=O)CCCO1 C(=O)(CC(O)CC(C)C)N1CCC(C(=O)NC(C(=O)OCC#C)C)C1 Cc1ncn(O)c1C(=O)NC1CCCC(N(C)C(c2cnsc2C)=O)C1 CCC(C)C(O)CC(=O)NC1CC2(C1)CN(C(C13CCCC(CO1)C3)=O)C2 Cn1nnc(C=CC(N2CCN(CCCCCNC(=O)CCC3CC3)CC2)=O)n1 C(=O)(C(CCC1CC1)NC(=O)Cc1cc(C)on1)NC(c1ncnn1C)CC C(C)(C)(CC(C)NC(=O)CC1CCN1C(c1cc(CO)oc1C)=O)OC c1(C(C)NC(C2(NC(=O)CC3CCCC3)CC(F)C2)=O)nnc(O)n1C CC(F)(F)CCC(=O)NC1CCCC1NC(=O)CN1CCS(=O)CC1 C1(N(C)C)(C(=O)NC2CCC(CNC(c3cc(Br)n[nH]3)=O)C2)CCCCC1 c1(CC(=O)NCC2N(C(C3(COC)CCC3)=O)CC2)cc(F)ccc1O N1(C(C2(NC(Cn3ccc(C)n3)=O)CCCCC2)=O)CCOCCC1C c1(C(=O)NC2CC3(C(NC(=O)Cn4cnnn4)C3)C2)cccc2c1OCO2 C1(C(C)C)(COC(C2CCCC(CO)CC2)=O)CN(C(C)(C)C)C(=O)C1 C1(C(=O)NCCN(C(=O)C(c2ccccc2)C)CCOC)CCC(OC)C1 CCCC(CCC)CC(=O)NC1COC2(CCN(C(c3cccnc3N)=O)C2)C1 C(=O)(C1=CC2(CCOCC2)C1)NCC(C)CN(C)C(C1CCCC12OCCO2)=O C1(NC(CC(C)C2CCCO2)=O)CN(C(c2sccc2C(F)F)=O)CC1(C)C n1(CC)cc(C(=O)NCCN(C(=O)C(O)CC(N)=O)C(C)C)c2ccccc12 c1(C(=O)NCC2CCN(C(CCC)=O)C2)cc2c(Cl)cccc2nc1C C(=O)(C1=CCCOC1)N1CCCC(N(C2CC2F)C(=O)OC(C)(C)C)C1 C(CC(=O)NCC1(F)CCC(NC(c2cscc2OC)=O)C1)(C(F)(F)F)OC C1(CNC(C2NC(=O)CC(=O)C2)=O)CC(C(=O)N2CCCc3nncn32)=NO1 C(=O)(CCC(=O)N(C1CC(NC(=O)C(c2cccc(Cl)c2)N(C)C)C1)C)OC C1=COC(c2noc(-c3cn(Cc4ccccc4)nn3)n2)CC1 c1(CC(=O)NC(C)CCNC(=O)CN(C)C2CC2)cc(Cl)c(Br)cc1F C12(CNC(COC(CC)C)=O)CCC(CNC(c3[nH]ccc3CC)=O)(CC1)CO2 Cc1nc(CNC(=O)C(CNC(=O)CNCC(C)(C)C)CC2CCCC2)sc1C Cc1ccc(CNC(C2CC(C)CN2C(C2CC2[N+](=O)[O-])=O)=O)nc1 Cn1cnc(C(=O)NC2CC(NC(=O)CC3CCC(C4CC4)O3)C2)n1 N1(C(c2cnc(C)cn2)C(=O)NCCOC)CCCC2(C)CCCC12 c1(C(N(CCNC(C(C)=C(CC)C)=O)C)=O)nn(CC)c(=O)c2ccccc12 N1(C(CC2(C=C)CN(C(=O)Cc3ccoc3)C2)=O)Cc2cccnc2C1 c1(CC(=O)N(C2CCN(C(c3cc(-c4cccs4)on3)=O)C2)C)ccc(O)cc1 N1(C(C(C)C(=O)N(C(C2(C(F)(F)F)CC2)=O)CC2CC2)=O)CC(O)(c2cc[nH]n2)C1 C1(NC(CC(=O)N(C)C)=O)C2CCC1N(C(=O)Cn1cnc(Br)n1)C2 c1(C(=O)NC2C(NC(Cn3c(=N)nc[nH]3)=O)CC2)ccc(S(N)(=O)=O)o1 Cc1cc(S(=O)(=O)N2CC3(CC3C(N3CCCC3C)=O)C2)c(C)cc1Cl C1(C(=O)NCC(C(C)C)(C)NC(c2cccs2)=O)CN(CP(C)(C)=O)C1 N1(C(C(COC)COC)=O)CCN(C(c2ccc(O)nc2C)=O)C2CCCCC12 c1(C2(C(=O)NCC(CC)(CC)NC(=O)C(=O)N(C)C)CCC2)ccc(C#N)cc1 c1(C(N(CCNC(C2CC3(OC)CC2C3)=O)C)=O)cccc(S(C)=O)c1 c1(OC)cc(F)cc(C=CC(N2CCN(Cc3cnc(Cl)nc3)CC23CC3)=O)c1 CN1CCN(C(=O)CCc2ccncc2)CC1c1cn(Cc2ccncn2)nn1 Cc1cnc(N(C2C3CCC2CNC3)C(=O)CNC(=O)C(C)(C)C)cc1Cl N1(C(Cc2c(C)cccc2)=O)C(C)CC2CN(C(=O)Cc3csc(=N)[nH]3)CC12 N1(C(N2CC(C)S(=O)CC2)=O)CCn2ncc(Cc3cn(CC4CCOC4)nn3)c2C1 N1(CCN(C(C(Cc2ccccc2)N(C)C2CC2)=O)C)CSCCSC1 c1(N2CCC(O)(C(=O)Nc3cc(C(=O)OC)no3)C2)ncc2c(ccn2C)n1 c1(CCCC)ncc(C(=O)NCC(C2CC2)NC(=O)C=CCN(C)CC)s1 N1(C(Cc2scc(CC)n2)=O)CCCC2CN(C(c3ccnc(Cl)c3)=O)CC12 C(=O)(CS(=O)C(F)(F)F)N1CCC(NC(c2ccc(C(=O)OC)cn2)=O)(CO)C1 c1(C(=O)NCC=CCNC(C2(C)CCC(=O)C2)=O)c(F)ccc2n[nH]cc12 C(CCN=c1[nH]c(=NCCc2ccn(C)n2)c2[nH]ccc2[nH]1)N(C(C)C)C CC1(C)CCN(C(C2C3CCC2(C)C3(C)C)=O)CC1NC(=O)Cc1cc[nH]n1 Cc1c(C(=O)N(C2CC2)Cc2ccncc2-c2nn[nH]n2)cnn1C1CCCC1 c1(-c2ncc(C(=O)NC3CC(C)(NC(C(C)CO)=O)C3)s2)c(F)cccc1Cl C1(C(N2CC(OC)(CNC(=O)Cn3cc(C(F)(F)F)nn3)C2)=O)CC1C1CCC1 C1(NC(C2CCC(CC)O2)=O)CCC12CCCN(C(C1CC(CC3CC3)C1)=O)C2 C1(CC(=O)NC2C(C)CN(C(C3CC(=O)CO3)=O)C2)CCC(C)(C)CO1 c1(C(=O)NCC(CNC(C2CN(C(N(C)C)=O)C2)=O)O)cn2cc(Cl)cnc2n1 c1(C(N2CCC(NC(C(CC)(C)COC)=O)C2)=O)c[nH]c2cccc(Cl)c12 C(=O)(C1=CCCCO1)NCCC1(C)CCN(C(=O)CCN2CCCC2=O)C1 c1(OC)cc(Br)cc(C(=O)NCC(C)S(C)=O)c1N Cc1ccc(C(N2CC3CN(C(=O)C=CBr)CC3(C)C2)=O)c2c1CCC2 N1(C(Cc2ncc(C)o2)=O)CCC2(CCC(NC(c3csc(O)n3)=O)C2)CC1 c1(C(=O)NCCCC2CCCC2O)cc(O)nc2c1CCCN2 c1(C(N(C(C)C(=O)NCCc2noc(=O)n2C)CC)=O)ccc(Cl)cc1 CCC(CS(=O)(=O)c1ccccc1)NC(=NCCCC(F)F)NC1CCCCC1 N1(C(c2ccc(C(=O)OC)s2)C(=O)NCc2cccs2)CC(=O)NC2(CC2)C1 c1(CC)ncnc(N2CCN(C)C(CNC(=O)CNc3nccs3)C2)c1OC C1(C(=O)NC(CN(C(C(CCC)OCC)=O)C)(CO)CO)CCCCN1N=O CCCC(O)C(=O)NC(C)CN1CCN(C(c2cc(C)c(C)o2)=O)CC1 c1(C(N2CC(C(=O)Nc3nnco3)NCC2)=O)c(Cl)cccc1[N+](=O)[O-] Cc1noc(N)c1C(=O)NCCOCCCNC(c1cncc(C2CC2)c1)=O CC(C)C(O)C(C)(C)C(=O)NCC1CCC(C(=O)NCCC#CCO)O1 c1(-n2c(C(CCC=C)NCCOc3cccc(Br)n3)nnn2)ccc(C)c(F)c1F C1(C(N2C(C=CC(=O)NCc3c(C)n(C)nn3)CCC2)=O)CNC(=O)CC1C c1(N(C2CNCCC2(F)F)Cc2c(F)ccc(Br)c2)cc2ncnn2cn1 n1(CCCNC(=O)CC2COC(C)(C)C2)ccnc1C=CC(N1CC(C)(OC)C1)=O N1(C(c2c(F)cccc2Cl)=O)CCC2CCCN(C(=O)C3=CCCS3)C2C1 N1(C(C(C)CO)=O)CC(C2CCN(C(C3CCC4(CC3)CC4)=O)CC2)C1 c1(C(=O)NCCCOCCNC(C2(C#C)CCC2)=O)cc(C)n(C(C)CC)n1 C1(CNC(c2ncnc(C)c2Br)=O)(CO)COCC2CCCCN12 Cc1cc(C(=O)NCC(O)CN(C)C(c2cccc(C3CC3)c2)=O)n(C)n1 C1(CNC(C2C(OC)CC2)=O)CCN(C(c2ccc(C)nc2O)=O)CC1(F)F C1(C(=O)NCC2C(NC(CSCc3c(C)cccc3)=O)CC2)CC2(CCC2)CO1 C(=O)(C(C)(C)CCC(=O)NCC(O)CN(C)C(C1CC=CC1)=O)OC c1(C(C(=O)NCCCN(C(C)C)C(c2cc(C(F)(F)F)cs2)=O)O)cncn1C C1(NC(c2occ(C)c2C)=O)CC2CN(C(c3ccnc(C(N)=O)c3)=O)CC2C1 C(=O)(CC1=CCOCC1)N1CC(NC(c2n(C)c(S)nc2)=O)C(C(F)F)C1 N1(C(C)C)CC(C(F)(F)F)C(S(=O)(=O)Cn2nc(C(F)(F)F)c3ccccc23)C1 c1(C(=O)O)ccccc1-n1cc(C(C2CCOC2=O)N2CCSCC2)nn1 C1(CC)CN(C(=O)CO)CCC1NC(=O)CCC(=O)Nc1sccc1C(=O)OC C1(CC=C)(NC(c2nc(C(=O)OC)sc2C)=O)CCN(C(=O)C(CC)SC)CC1 N1(C(c2cn(C)nc2)=O)C(C(=O)N(CC(F)F)CCO)CCC12CC2 c1(OC)ncc(C(=O)NC2(C3CCCCN3C(=O)CSCC(F)F)CC2)cn1 C1(CNC(C2(CC)CC2)=O)CCCCN1C(C1CCCN1c1ncccn1)=O C1(C(C)C(=O)N2CC(N(C)C)C2)CCN(C(=O)CN2CCNC2=O)C1 c1(C(=O)NCC2CC(NC(c3cccc(=O)o3)=O)C2)cc(Cl)cc2cccnc12 Cc1c(C(=O)N(CC(=O)NCc2cnn[nH]2)C2CCC2)cccc1F c1(SC)ccc(NC(=O)CC2(N(C)C(c3ccnn3C)=O)CC2)cn1 Cc1ncc(C(=O)NCC(C)NC(=O)C(C2CCC(=O)CC2)F)c(C)n1 c1(CNC2CC(C(=O)Nc3nc(Br)ccc3O)C2)cc(F)c(Cl)c(F)c1 N1(C(C2(CC#C)CC2)=O)CCN2CCN(C(=O)COC(C)C)CC2C1 N1(C(c2cc(CCC)ncc2)=O)CCC(CNC(c2nccn2CC)=O)C(C)C1 C1(CNC(C(c2ccc(C#N)cc2)(C)C)=O)CCCN(C(C2CSC2)=O)CC1 C1(CNC(c2ccc(SCC)nc2)=O)CN(C(=O)C=Cc2ccco2)CCCO1 N1(C(c2cc(CCC)nn2C)=O)CC2CC1CCC2NC(=O)CNC=O C(CCC(=O)NC1CC(CC(=O)N(C(C)CC(C)C)C)C1)=CCC=C c1(CNC(N2CCCC2CSC2CC2)=O)cncc2[nH]ccc12 c1(C(=O)NCCCCCNC(c2c(CC)nn[nH]2)=O)cnc(N)c(CO)c1 C(=O)(C1=C(C)CCCC1(C)C)N1CC(CC)C(NC(c2ccnnc2)=O)CC1 C1(NC(c2ncn(CC)c2)=O)CN(C(=O)CCc2cccnc2Br)CCC1O N1(c2n(CCOCC=C)c(C3(OC)CCOC3)nn2)CC(CCO)OCC1(C)C Cc1ccc2c(c1)SC(C(N1CC3CN(C(=O)C(C)c4ccsc4)CC3C1)=O)C2 N1(C(CCC=C(C)C)=O)CCCN(C(c2cc(C(F)F)cs2)=O)C(C)C1 C1(C(C)NCCOCCSC)CCSCC1 C1(C(=O)NC2(CC=C)CCOC2)CCN(C(=O)C=Cc2ccc[nH]2)O1 N1(C(C(C(C)C)n2cnnc2)=O)CCCOC(CNC(=O)CC2CCOC2)C1 C(=O)(CCS(=O)(=O)C1CCCC1)NC12C(CN(C(CCC(=O)NC)=O)C1)CCC2 c1(NCCOCCNC(C2CC(C)SCC2)=O)ncnc2sc3ccccc3c12 C1(C(C)C)CN(C(c2cnc[nH]2)=O)CCN1C(C1CC(OC(F)F)C1)=O c1(C(N(CC(N2CCC(O)(CC#C)CC2)=O)CC(C)C)=O)ccc2cc[nH]c2n1 C1(CNC(c2cc(CC)oc2C)=O)CN(C(c2ccnc(CC)n2)=O)CCN1C C1(C(N2CC(CNC(C3=NNC(=O)CC3)=O)C(O)C2)=O)CCc2nncn2CC1 c1(NC(=O)Cc2cnn(-c3ccccc3)n2)ccc(N2CCOCC2)c(Cl)c1 C1(NC(c2c(CC)ncs2)=O)CCN(C(=O)C(F)C2CCCC2)CC(C)(C)C1 C(C(=O)NCC1CCC1NC(c1nn(C)cc1C(C)=O)=O)(C(C)(C)C)NC(C)=O c1(CN(CC2=C(C#N)CCC2)CC)ccc(Cl)cc1Cl c1(C(N2CC(C)(CC(N3CCCCC3C3CC3)=O)C2)=O)c(O)cccc1[N+](=O)[O-] N1(C(C2CN(C(c3ncnc(C)c3C)=O)CC23CC3)=O)CCc2n[nH]cc2C1 c1(CC(=O)NC2(CNC(=O)CC34CCCC3C4)CCC2)c(O)ncnc1O c1(NC(c2c(C)nns2)C)cccc(CN2CCN(C)CC2)c1 C12(C(=O)NC3CN(C(C(C)=CC)=O)C3)CCC(OC)C1C2 CCCCCC(O)CC(=O)N1CCN(CC(N2CCCC(CCCC)C2)=O)CC1 CCCCC(C)(F)C(=O)N1CC=C(C(=O)NCC(C)(C)CCO)CC1 CC(=O)CCCC(=O)N1CCC(CO)(CNC(c2nccc(Cl)c2F)=O)C1 CCC(C)(CNC(=O)CC1CCCCC1)C(=O)NC1CC(CO)C12CCC2 C#Cc1cc(C(=O)N(c2cn(C3CC3)nc2C(=O)O)C)cc(I)c1 C12(C(N3CCC(O)C3c3ccccc3Cl)=O)CC(CC1C(=O)O)C2 N1(C(CCC=C(C)C)=O)CC2CC(C1)N(C(=O)C=Cc1cscn1)C2 C(=O)(C#CC1CCOC1)NC(C(C(=O)Nc1c(OC)ccc(O)c1)C)C Cc1nc(CNC(=O)C(O)CCN(C)C)oc1C(=O)NOCCCN(C)C N1(CCN(C(C(CC)O)=O)C)CCN(C(C2(C(C)(F)F)CC2)=O)CC1 CC(C)CS(=O)(=O)CC(=O)N1CC2CCCC(NC(=O)Cc3ccccc3)C2C1 N1(C(C2CN(CC)C(=O)C2)=O)CC=C(C(C)(C)C(=O)NC(C)CN2CCCC2)C1 c1(OC)cc(C(N2C3CN(C(=O)CC4COCCO4)CC23)=O)cc(O)c1O C1(NCCCC)CCN(C(C2CC(C)(C)C2)=O)CC1C C1(CC(=O)NC2CC3CCC(C2)N3C(c2cn[nH]c2)=O)COc2ccccc2O1 CCC(C)C(C(=O)NCCc1ccccc1)N(C(=O)Cc1coc(C)c1)C CCCC(O)CC(=O)N1CC(NC(c2ccn(CCO)c(=O)c2)=O)CCC1C CCCCCCCCCC=CC(N1CC(NC(=O)C(C)C2CCCC2)C(F)C1)=O C1(CNC(CC(C)CF)=O)CN(C(c2ccc3c(c2)CCC3)=O)C2COCC2O1 C1(CC=C)(NC(=O)CCNC(=O)COC)CCN(C(C2(F)CCOC2C)=O)CC1 C(CC(C)(C)C(=O)NC(CNC(=O)CCN1CCC1)CC(C)C)OC N1(C(c2c(C)nsc2)=O)CCC2(CC1)CC2C(=O)NCc1sccc1Cl N1(C(c2ccn(C)c2)C(=O)NCC=C)CCC(c2cccc(C(=O)OC)c2)CC1 N1(C(c2ncccn2)=O)CCCC2(CCCN2C(=O)CC2CCCC2)C1 c1(OCCC(=O)N(C2CN(C(C3C(SC)CCC3)=O)C2)C)ccc(C)cc1C C1(CC(C)NC(C(C)C#N)=O)CCN(C(=O)CCCn2c(O)nnc2O)CC1 C1(CC(=O)NCn2cc(C(C)(C)C)nn2)CCN(C(=O)Nc2ccccc2)C1 N1(C(c2ccc(CC)cc2)=O)CCC(NC(=O)COC)C(CO)C1 C1(NCC(C(C)C)CO)CN(C(=O)CSC(F)(F)F)CC1C1CC1 C1(C(=O)NCCCN(C(C(N2CCCCC2=O)C)=O)C2CC2)CC2(C1)CC2F C(=O)(CC1=CCCCC1)N(C)CC1CCN(C(c2c(CC)c[nH]n2)=O)C1 C12(CNC(CCCCCSC)=O)CCCC1CN(C(=O)CCCCSC)C2 C1(C)(C(=O)NCCCn2c(C)nnc2)C=CCN1C(=O)C(C(C)C)C1CCC1 c1(OCC(=O)NC2CN(C(CS(N)(=O)=O)=O)CC2O)ccc(Br)cc1F C1(CC(=O)NCC2CC(COC)C2)COCCN1C(=O)Cc1ccsc1 Cc1cc(NC(=O)Cn2cc(CC(O)C(C)(C)C)nn2)c(C)n1CO.c1ccnn1C Cc1ccc(CC(=O)N(C)CC2(O)CCCN(C(=O)CC(C)(C)O)C2)cc1Cl Cc1ccc(F)cc1C(=O)NCC1CN(C(=O)CCC=CC(C)C)CCC1C c1(CC(=O)NCC2(C(C)NC(c3cnsn3)=O)CC2)c[nH]c2ccc(F)cc12 C1(C(N2CC(F)(CNC(C3(C)ON=C(C)C3)=O)C2)=O)CCc2cncn2C1 N1(C(c2cc(CNC(C3(C=C)CCC3)=O)nn2C)=O)CC2(C1)CC(C)(O)C2 C(=O)(CC(C)CCC(=O)NC1CC(C)CN(C(c2ncc(C)cc2C)=O)C1)OC C12(C(=O)NCC(C)(C)NC(C(CC#C)CC#C)=O)CCC(CC1)C(C)(C)O2 c1(CC(=O)NCC(CC)NC(C2(COC)CC2)=O)ccc(OC(C)C)cc1 C1(C)(CC)CC(NC(=O)C(CC(F)F)NC(=O)C(C)CC(N)=O)CCO1 c1(C(N2CC3C(CNC(C4C(C(=O)OC)C4)=O)(C3)C2)=O)c(OC)ccnc1OC C1(CNC(c2nn(C)c(C(N)=O)c2)=O)CCC(C)(C)CN1C(c1cc(O)cs1)=O N1(C(C2CC(=O)CN2C(=O)CCc2cn[nH]c2)=O)CC2C=CCC(C2)C1 c1(NC)cnc(Cl)cc1C(=O)NCCCC1CN(C(c2cnc(Cl)[nH]2)=O)CCO1 c1nnccc1C(F)(F)F.C1(SC)CCC(NC)C1 C1(CNC(c2cscn2)=O)CCCN(C(=O)CC2(CSc3ccccc3)CC2)C1 C1(=CCNC(C2(CC(C)C)CC2)=O)CCN(C(=O)C(O)Cc2ccccn2)CC1 C(=O)(C(O)CC(F)(F)F)NC1C(n2cc(CC(C)(C)OC)nn2)CCC1 C1(C)(CNC(C=C(CCC)C)=O)CCN(C(c2cc(N(C)C)nc(Cl)c2)=O)CC1 N1(C(C2C(c3ccc(C)o3)C2)=O)CC(C2CN(C(c3ccc(Br)cc3)=O)C2)C1 C1(C(N(C2CCN(C(C3CN(C(C)=O)C3)=O)CC2)CC)=O)OC2CCC1CC2 n1(C2C(C)CCCC2)c(C2CCC(F)(F)CC2)csc1=Nc1cnn(C)c1 c1(CC(=O)NCC(C)N(C(=O)CCc2cn(C)cn2)C)cncnc1O C(=O)(CCCCCO)Nc1cccc(NC(CC(C)(F)F)=O)c1 Cc1csc(C(=O)NC(CC2C(C3(c4ncccn4)CC3)CC2O)=O)c1 C1(c2cn(-c3cc(C)c(N)cc3)nn2)CC(C)N(C)CC1C CC(CCNC(=O)C(CO)NC(N)=O)CCNC(c1cnc(CC(C)(C)C)s1)=O C1(C(N(C(C)C(F)(F)F)CC)=O)CC12CCN(C(C)C(C1CCCCC1)=O)CC2 CC(C)C(C)(O)CNC(=O)C(CO)NC(=O)CC1CCOCC1 N1(C(C2C(C)(COC)C2)=O)CCN(C(=O)C(c2ccccn2)O)CC(O)C1 N1(C(CC(COC)NC(=O)C=CCN2CCC2)=O)CCCC2(CCOC2)C1 N1(C(C2C(OCC)CC2)=O)CCCC2(CCN(C(=O)C(O)CC(C)C)CC2)C1 C1(NC(c2ccc(CNC(COCCOC)=O)o2)=O)CC2CCC2C1 c1(C2C(C(N(C3CCC(O)CC3)C)=O)C2)cc(F)cc(Cl)c1 CC(O)C(C)(C)C(=O)NCC1(NC(c2cc(CCO)on2)=O)CCCC1 C(C(F)(F)F)(C1CCC1)C(=O)NC(c1ccccc1)C(=O)NC1CC(C)C1 CN1CCCC(F)(C(=O)NCC2CN(C(c3c[nH]c(=S)cn3)=O)C2)C1 c1(NC)ncc(C(=O)NCC2CCN(C(=O)CC3CCCS(=O)(=O)C3)C2)cc1Cl c1(C(=O)NC2CCC(N(C(CN(C(C)=O)C)=O)C)CC2)c(O)ncc2c1CCC2 c1(CC(N2C(C(=O)NC(C(C3CC3)OC)C)CC2)=O)ccsc1C N1(C(C2CCc3ccnn3C2)=O)CCC2(CC1)CCN(C(C1C=CCS1)=O)CC2 c1(OCC2(C(N)=S)CC2)nc2cc(OCCC(=O)O)ccc2o1 c1(N2CCC(NC(c3c(C)n(C(C)C)nc3)=O)C2C)cc(S(C)(=O)=O)ncn1 C1(C(=O)NC(CC)C(=O)NC)C2CCCC2CN1C(=O)C(C#N)C(C)(C)C CC(C)(C)S(=O)(=O)CC(=O)N1CCN(C(=O)CCC2CC2(Cl)Cl)CC(C)(F)C1 C=C1CCN(C(=O)CCC=C(C)C)C(C(=O)N(CC(O)COCC)C)C1 Cc1ccc(NC(=O)CC2(NC(=O)C#CC3CC3)CC2)cc1C C(=O)(C(C)(O)C(C)C)N1CC(NC(C(n2c(C)ccn2)C)=O)C(O)C1 C(=O)(CN=S(C)(C)=O)NCC(C)CNC(c1ccc(C2CCCC(=O)N2)cc1)=O C1(N(C(c2cnc(C(C)C)o2)=O)C)CCCN(C(=O)C(C)CN(C)C)CC1 c1(C(=O)N(CC(N2CCC(N3CC(O)C3)C2)=O)CC2CC2)ccc2c(c1)OCO2 O=C1CCc2ccc(CNC(=O)CNS(C)(=O)=O)nc2C1.C1(O)CCCC1N c1(SCC2(CO)CN(C(C3N(C(C(C)C)=O)CSC3)=O)C2)cccc(F)c1 N1(C(C2=CC(O)C(NC(=O)C=Cc3ccncc3)C2)=O)Cc2n[nH]cc2C1CO C=CCCCCCCC(=O)N1CCCC(F)(C(=O)NC(C)(C)CCCO)C1 C1(NC(CN(C(COC)=O)C)=O)CCN(C(=O)C(n2ccnc2C)C)C1C C(CCC(C(=O)NCC=CCOC)NC(c1ccc(C)cc1O)=O)OC C(C1c2ccccc2CN1C(c1cc(Cl)ncc1N)=O)NC(C(CCC)OC)=O C12(NC(c3ccc(CC)s3)=O)CCOC(CNC(C34CC(C)C3C4)=O)(C1)C2 CC(C)(C(=O)NCC(C)(O)CNC(c1c[nH]nc1-c1ccsc1)=O)C1CC1 C1(CC(=O)NCc2cc(C)oc2)CCCCC1NC(c1nccnc1N)=O c1(C(N2CC(O)(CN(C)C(C3CCC3)=O)C2)=O)cc(Br)n2c1CCC2 C1(C)(CNC(C(C)(C)c2ccno2)=O)CCN(C(c2ccccc2C2CC2)=O)C1 C1(c2n(CC)nnn2)(NCC(F)C2CCC2)CCCC1N(C)Cc1ccccc1 Cc1cc(CC(N2CCCC2C(C)(C)NC(=O)CC23CC(C2)C3)=O)n[nH]1 C1(NC(C(C=C)O)=O)CN(C(=O)CC2CCCN2C)CC1CO c1(C(=O)NC2CCC2NC(C2(F)CCC2)=O)csc(-c2cn[nH]c2)n1 c1(CCC(C)NC(C2C(OC)CCC2)=O)ccccc1O C1(CNC(COCCN(C)C)=O)CCCC1NC(c1ncoc1-c1ccon1)=O CCC(O)C(C)(C)C(=O)NCc1cc[nH]c1C(=O)N(C1CC(F)(F)C1)C Cc1nc(C)c(C(=O)NC23CCCC2N(C(=O)C=CC(C)(C)C)CC3)nc1C C(=O)(C(C)CC(N)=O)NC(CNC(C1(c2ccc(C)nc2)CC1)=O)(C)C1CCC1 CN1CCCC2(CCN(Cc3conc3C3CC3)C2)C1=O C1(NC(C23CC(C(=O)OC)(C2)C3)=O)C2CN(C(=O)Cc3cccc(OC)c3)CC12 CC(CN=c1[nH]n(C)cc1[N+](=O)[O-])NC(=O)CC1CCCCO1 C(=O)(C(O)C(C(C)C)NCCCC(=O)NC1(c2cc[nH]n2)CC1)OC C1(NC(C(N2CCCN(C(C)=O)C(C)C2)=O)=O)CS(=O)(=O)C12CCCCC2 Cc1ccc(-c2cc(C(=O)Nc3cc(F)c(F)c(Br)c3)n[nH]2)c(C)c1F c1(C(=O)NC2CC(C)(CC)N(C(=O)COCCOC)C2)cc([N+](=O)[O-])c(C)s1 Cc1c(NC(c2conc2C(C)NC(=O)CCC(=O)C2CC2)=O)cnn1C(C)C C(=O)(C(F)CCC(C)(C)C)NC(CNC(COC(C)C)=O)CO CC1(C)CCc2sc(NC(=O)NC34CC3CS(=O)(=O)C4)nc21 C=CC(C(=O)N(CCC(=O)N(C)CCC1CCCN1C)CCO)OC C(C(CC(=O)NC(CC1CC1)CO)NC(c1cnc(N)cn1)=O)OC CC1(NC(c2cncc(F)c2)=O)CCCN(C(=O)C2=CCSC2)C1 c1(C(=O)NCC(CNC(c2[nH]ccc2C2CC2)=O)CO)ccn2cnnc2c1 C=CC1OCCC1C(=O)NCC1(F)CC(NC(c2cnc(C(C)OCC)s2)=O)C1 c1(CCNC(=O)NCC2CC(OCC(F)(F)F)C2)ccc(OCF)cc1 Cc1ccc(F)cc1CC(=O)NCC1(NC(C23CC(C2)C3)=O)CCCCC1C c1(C(=O)NCCC2CCN(C(CC(C=C)CC)=O)C2)c(Cl)ccc2c1OCO2 c1(C(=O)NCCC(=O)NCCc2cn(C)nc2)cc(F)cc(F)c1 C12(C(=O)NC3CCCC(NC(=O)COc4cn[nH]c4)C3)CC3CC(C(=O)N1)C2C3 CCC(C(=O)N1CCCCC(CCC(=O)NC(C)(CSC)CO)C1)C(C)C C1(NC(c2ccn(C)n2)=O)CN(C(c2n[nH]cc2F)=O)CC1c1cnn(C)c1 C1(NC(CC=CC=C)=O)CN(C(=O)Cc2ccc(NC(N)=O)cc2)CC(C)(C)C1 C(CNC(=O)C(C)(C1CC1)OC)(CC(C)C)NC(CC1(NC(C)=O)CC1)=O n1(CC(N2CC(C(=O)OC)(OC)C2)=O)ncc(C#N)c1I C(=O)(C(O)CC[S+](C)C)N(C1CCN(C(c2c(COC)cccn2)=O)C1)C Cc1nn(C)c(Cl)c1C=CC(N1CC(NC(=O)C=Cc2cnccn2)C1)=O Cc1ccccc1OCCCC(=O)NC1CC(F)(CNC(=O)C=CC(C)C)C1 c1(C(N2CC(C)(NC(CC3C(CC)C3(F)F)=O)C2)=O)cc(OC)ncn1 C1(c2n(C)ncc2)CN(C(=O)C(C)(C)C2CC2)CCN1C(c1ccns1)=O N1(C(COC(C)=O)=O)CC2(CCCC(CNC(C3CC(C)=NO3)=O)O2)C1 c1(C(N2CC(C)(C(=O)Nc3c(C)n[nH]c3)C2)=O)cccc(C2CC2)c1 C12(NC(CCC3OCC(C)(C)C3)=O)CCC(NC(=O)CC3CC3(Cl)Cl)(CC1)C2 c1(OC)cc(C)c(NC(C2CC2C2CN(C(c3cncs3)=O)C2)=O)cn1 C1(C(=O)NCC2(CC)CCC(=O)N2)CCCN1NC(=O)C1C=CC=CC=C1 c1(C(N(C(CNC(C(CSC)C)=O)C)C)=O)cc(C)n(-c2cnn(C)c2)c1C C1(c2cn(Cc3cccc(C)c3)nn2)CN(C(=O)Cn2nccc2C)CCN1C Cc1ccc(F)cc1N(C(=O)C(N1CCN(c2nc(C(C)C)no2)CC1)C)C C1(CNC(c2ccns2)=O)CCCN(C(C2CCCN2CC(F)(F)F)=O)CC1 C(=O)(C1=NNC(=O)CC1)N1C(CNC(C(CC=C)NC(C)=O)=O)C(C)CCC1 N1(C(CCOCCOC)=O)CCC(CF)(NC(=O)C(C)NC(N)=O)C1.C(C)(C)C Cc1cc(CC(=O)NC2CC3CC2N(C(c2csc(C(F)F)c2)=O)C3)cc(C)c1 C1(CC(=O)OCCC=C)CCN(C(C)COC)CC1 N1(C(C2(C#C)CC2)=O)CCC(C(C)CNC(c2onnc2CC)=O)CC1 c1(C=O)cc(C#N)c(F)cc1[N+](=O)[O-].N1(CC)CCc2nc(-c3ccc(=N)[nH]c3)sc2C1 C1(C)(C(=O)NC2CCN(CC)C(C)C2)CN(C(c2ccoc2)=O)C(C)(C)C1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CCC(O)(C(C)CNC(c2ccsc2C)=O)C1 c1(C(C(=O)NC2CC(NC(=O)C=CCN3CCCC3)C2)=O)c[nH]c2ccccc12 C1(C2CC2)(NC(C2CC(NC(C3CC4C=CC3O4)=O)CCO2)=O)CCC1 C#CCCN=C(NCCC1(O)CCCC1)N1CC2CCN(C)C2C1 c1(C(N2C(CCNC(=O)CC34CC(C3)C4)CCC2)=O)cnc2[nH]cncc1-2 c1(CC(=O)NC2(C)CCN(C(CCCCC)=O)CC2)cccc2occc12 C12(C(N3CC(OC)C3)=O)CC(CCO1)N(C(C1CC(=O)CCO1)=O)C2 N1(C(CN(C)C)=O)CCCC(O)(CN(C)C(C23CC(C)(CO2)C3)=O)C1 c1(CC(=O)NC(C2CN(C(=O)C(=O)NCC(F)(F)F)C2)C)ccnc(F)c1F c1(CNC(C(c2nc(Cl)cs2)N(c2ccccc2)CC)=O)ccccc1OC C1(Nc2c(C(=O)OCC)cncc2)CCC2(CC1)CN(C(=O)C(C)(O)C(C)C)C2 N1(C(C2CC(CC)C2)=O)CCN(C(c2occc2C2CC2)=O)CCC1C C(C(C)CN=c1cc[nH]c(-c2nccs2)n1)NC(C(CC)CSC)=O N1(C(c2cnc(OC)s2)=O)CCCC(C2CN(C(=O)C=C3CCC3)C2)C1 N1(C(C2CC(SC)C2)=O)CCC=CC1C(=O)N(C(C)C(C)(C)O)C CCC(C)CCC(O)CC(=O)N1CC(C)CN(C(c2ccc(Br)o2)=O)C(C)C1 c1(C(N2CCN(Cc3c(C(C)(C)C)[nH]cn3)C(CO)C2)=O)cccc2ccoc12 C1(C(=O)NCC2N(C(CC(C)(C)C3CC3)=O)CC(F)C2)CCOCC12CCC2 C=C=CC(C)C(=O)NCCC1COCCN1C(c1cc(C(=O)OC)co1)=O c1(CC(C(=O)N(C)CC2CCOC2)NC(c2c[nH]nc2CCl)=O)cnn(C)c1O c1(C(=O)NCC2CN(C(C3(C)CCCCO3)=O)C2)cc(C(F)(F)F)c(Cl)cn1 C1(NC(c2ccc(CC)cc2)=O)CC12CCC(NC(c1ncccc1C)=O)CC2 CN1CCN(CCC(N2CCOC(CNC(c3cc(CO)ccn3)=O)C2)=O)CC1 CC1CN2CCN1CC2C(N1CCC(CCNC(=O)CSc2ccncc2)C1)=O C1(C(N2CCC(C(C(=O)NC3CC(CSC)C3)C)C2)=O)C2CCC(C2)C1C C1(CN(C)C)COCC1NC(=O)CC1(NC(C2CNC(=O)C2)=O)CCC1 CC(C)CC(O)C(=O)N1CC2(CC2C(=O)Nc2c(Cl)cnn2C)C1 C1(NC(c2ccc(-c3nc(C)sc3)s2)=O)CCCN(C(=O)Nc2nccn2C)C1 N1(C(C2N(CC)CCCC2)=O)CC2CC(NC(C3CC(=O)N(C(C)C)C3)=O)C2C1 C1(C(C#C)NC(C(F)(F)F)C2CCCCC2)CCC(F)(F)CC1 c1(CCCn2c(N(CC(=C)C)C)nnc2-c2nccs2)ccc(F)c(Br)c1 c1(-c2ccc(C)cc2C#N)cc(C(=O)Nc2ncc[nH]2)c2cc[nH]c2c1 C(C(=O)N=c1cc[nH]cc1-c1ccccc1)N(C)Cc1cccc(C#N)c1 C1(N2CCCC2)(C(C)NC(C(C)NC)=O)CCCC1.c12ccc(o1)CN2.OC C=Cn1ncc(C(N2CC(O)(C(F)C(=O)NCC3(C#N)CC3)C2)=O)c1N C(=O)(C(C)(C)CC(C)C)N1CC(C)CC(CNC(CCN(CCC)C)=O)C1 CC1(C)Cc2ccccc2C1NCc1n[nH]cc1Br CC1CN(C(c2csc(C(F)(F)F)n2)=O)C(C)CN1C(=O)COCCCN=[N+]=[N-] c1(C(=O)NCC(C)(C2CCC2)NC(=O)C2=CCCCC2)nccc2ccsc12 c1(CN(C(C2(CC)CCOC2)=O)CCNC(c2ncoc2C)=O)ccc(Cl)nc1 C(CCC(C)C(=O)N1CCCC(c2ccccc2)(CO)C1)OC C(=O)(CC1OCc2ccccc21)N(CCCOCCN(C(C(COC)O)=O)C)C C(c1nccs1)=CC(=O)NC1CC(CCNC(C2(CO)COC2)=O)C1 CCCC(C)CN=c1cc[nH]cc1S(=O)(=O)N1CCC23CCCCC2(C1)C3(F)F N1(CC)CC2CN(C(=O)CC3CCCN(C(=O)CCCF)CC3)CC2C1 N1(C(C(C)(C)SC)=O)CC(C(=O)NCCc2cnc(C)s2)CC(C)(C)C1 c1(C(=O)NC(C)CC(C)NC(=O)C(C)(C)N(C)C)c(F)ccc2c1OCO2 c1(C(=O)NC2CCN(CCNC(=O)OC(C)(C)C)C2)ccnc(C2(C)CC2)n1 c1(C(N2CC(C)C(CNC(=O)CCOCC(F)F)CC2)=O)cccc2cnsc12 c1(OC)c(C(=O)NCCCCN(C)C(C2CC23CC3)=O)occc1=O C1(C(=O)Nc2c(C)cc(F)cc2)(CN)COCC2CCCN12 CCCCC(O)CNC(=O)C(c1cnn(C)c1)NC(c1ncoc1C)=O C1(NC(C(C)SC(F)(F)F)=O)CC(C)N(C(=O)COCC2CCCO2)C1 S(=O)(=O)(c1cccc(NCC2CC2)c1)NC(c1cccc(SC)c1)=O C(C(=O)NC1CCC(F)(CNC(c2nc(O)c(C)s2)=O)C1)(C(C)C)SC C1(O)(CNC(C2(N(C(c3cnn(C)n3)=O)C3CC3)CCC2)=O)CCOCC1 C(=O)(C(C)S(N)(=O)=O)NCCOC1CCN(C(C2OCCN(C(C)=O)C2)=O)C1 Cn1ncc(C(=O)NCCNC(c2cc(-c3ccccn3)no2)=O)c1N N1(C(c2ccccc2S)=O)CCC2CN(Cc3ccc(Br)cc3Br)CC12 c1(CC)cccc(C)c1C(=O)NCC1(COC)CN(C(C2CCOC2)=O)C1 N1(C(CC(=O)NCC)=O)CCOC(C(C)NC(C2(C)CS(=O)(=O)C2)=O)C1 C1(NC(=O)CCNc2ccccn2)CCCN(C(=O)C=CSc2nc[nH]n2)C1 c1(CN2CCCC(NC(c3ccc(Cl)c(O)c3)=O)C2)c[nH]c2ncccc12 c1(C(=O)NC(C)(C)CNC(=O)CC2CC(C)(C)CO2)cc(Cl)cc(Br)c1 CC1=C(C(=O)N2CC3(CCCC3NC(=O)C(C)C(C)O)C2)Cn2nnnc2N1C Cc1nc(C(=O)NCC(C)NC2CC23CCOC(C)C3)c2ccnc-2[nH]1 CC1CCCN(C(C2NC(=O)CC2C)=O)C1CNC(c1nc(=O)cc(N)[nH]1)=O c1(SCC(=O)NCc2cccc(CNC(C(CC)(C)O)=O)c2)nc(C)cc(C)n1 Cc1nc(NCC2C(=O)NCCC2C)cc(=NCc2ncccn2)[nH]1 Cc1nc(C(N2CCCN(CCNC(C3CCC3F)=O)CC2)=O)c2ccccn12 Cc1c(NC(=O)N(C)C)cccc1C(N1CCC(Cc2ccccc2)C1)=O c1(N2CC(C(C)NC(C(CN(CC)CC)F)=O)OCC2)ncnc2cnn(C)c12 N1(C(C(C)C2(O)CCC2)=O)CCC(C)(C(=O)NCC(O)Cn2cccn2)CC1 CC(C)(O)C#CC(=O)NC1CC2(NC(c3coc(C(C)(C)C)n3)=O)COC1C2 N1(C(c2cc(Cl)ccc2Cl)C(N)=O)CCOC2(CCCC2)C1 C(=O)(CC1=NNC(=O)C1)N1CC(CC(C)NC(=O)C(CN(C)C)N(C)C)C1 c1(C(=O)Nc2ccccc2C(N2CCCCCC2)=O)c(F)cc(O)cc1F c1(C(C2(C)CC2)NC(c2n(CC=C)nnn2)C(C)CC)cccc(Cl)c1 c1(CCC(N2CC(CNC(CN(CCC)C)=O)C(O)C2)=O)cccc(OC)c1F n1(CC)cnnc1CN(CCNC(C1(c2ccc(C)s2)CC1)=O)C1CC1 N1(C(c2c(C#C)cccc2)=O)CCc2ccc(C(N3CC(OCC)C3)=O)cc2C1 c1(CC(=O)NC2C3CCN(C(c4c(C#N)scc4)=O)C3C2)csc2ccccc12 N1(C(c2cnc(C)nc2)=O)CCCCC(CNC(C2CC(C(C)C)C2)=O)C1 N1(CC(=O)NCC=CCC(N2C(COC)C=CC2)=O)CC(=O)NC1=O N1(C(C2C(C)(C)CO2)=O)CCC2(CCCN(c3cc4c(cn3)C(=O)CCC4)C2)C1 C1(NC(C=CCOC)=O)CCC12CN(C(=O)C(c1ccc(OC)nc1)(F)F)C2 CC1(C(=O)NCCN2CCC(NC(=O)CCC3CC3(F)F)CC2)CCCS1(=O)=O c1(CN(C)CC2CCCN(C(C)=O)C2)cc(I)c(Br)c(F)c1F N1(C(COCC(=C)C)=O)CCN(C(c2ccc(C(C)(C)C)o2)=O)C2CC12 C1(C)(C(=O)NCCCC2CCN(C(C(C)C(F)(F)F)=O)CC2)CCCCCCC1 C(=O)(C(C)P(C)(C)=O)NC1C(C)CN(C(=O)CCCCSc2ccccc2)C1 c1(OC)ccc(CN)cc1C(=O)NCCN1CCOCC1 Cc1ccc(NC(C2C(C)CCN2C(=O)CC(C)(C)O)=O)c(CO)c1 O=C1CCC(CCC(=O)NCC2CCN(C(=O)Cc3ccccc3)C2)C1 Cc1cnc(NCc2ccsc2)c(S(=O)(=O)N2CCC(Cc3ccco3)CC2)c1 c1(C(N2CCCN(C(C(CCC)OC)=O)C(CO)C2)=O)ccc2nc(C)[nH]c2c1 C1(NCC(CC)C)COCCN1C(=O)C(=O)N(C1CCN(S(C)(=O)=O)CC1)C CCC(CNC(=O)C(Cc1cc[nH]n1)NC(c1ccnnc1C)=O)(CC)C(N)=O N1(C(C2(CCNC(CC3(C#N)CC3)=O)CCC2)=O)CC2CCCC(C2)C1 Cc1c(N)ccc(C(=O)NC2CCCC(NC(=O)Cn3ncnn3)C2)c1C C(CS(=O)(=O)CC(=O)N(C(CC(F)F)C(=O)N(C(C)CO)CC1CCC1)C)OC N1(C(c2cc(-c3ccco3)on2)C(=O)NCC=C)CCCC(N=[N+]=[N-])CC1 O=C(CCCO)NNC(=O)C(=O)SC.c12ccc(F)c(c1)N1CC(=O)N2C1=O N1(C(c2c(CC=C)cccc2)=O)CCC2(CCN(C(C3CC3C)=O)C2)C1 CC1(C)CCC(NCc2cc(OC(F)F)ccc2OC(F)F)c2ccc(F)cc21 C1(NC(CC2CC(NC(c3nc(OCC)oc3)=O)C2)=O)CCC(C)(C)C(C)C1 c1(OC)c(F)cc(F)c(CN2CC3(CC3)CC2C(=O)N=c2[nH][nH]cc2I)c1F N1(C(c2cccc(OC)c2)=O)CC(CNC(=O)C(F)(F)C(O)C2CC2)CC1(C)C C=CCCCCCCC(=O)NC1CN(C(c2nccnc2C(=O)OC)=O)C1 C1(C)(CNC(COc2cc(C)on2)=O)COCCN(C(=O)Cc2cnn(C)c2)C1 C12(C(N(C3CCN(C(C4(C(C)(F)F)CC4)=O)CC3)CC)=O)CCCCC1C2(F)F N1(C(C=CCN(C(C(C)CC#N)=O)C)=O)CC2(CCC2(C)C)C1 Cn1c(CNC(c2csc(Cc3ccccc3)n2)=O)nnc1C1CCC1 C1(CNC(C(C)C(C)O)=O)CCC2(CCN(C(C3(N4CCCC4)CC3)=O)CC2)O1 Cc1nnc2ccc(C(=O)N(C(C)CNC(=O)C(F)CC(C)C)C)cc2c1C C1(C(=O)NCC(CN(C(=O)CNC(=O)C(F)(F)F)CC)(C)C)CC(=O)OC1(C)C c1(C(N(CCOCCNC(c2c(C(C)C)[nH]cc2)=O)C)=O)cc2cnn(C)c2s1 c1(C(=O)NCC2C(C(=O)NC3(CC4CC4)CCC3)C2)snnc1C1CCC1 N1(CC(=O)NCC2CC(CNC(=O)CCN3CCOC3=O)OC2)CC(=O)NC1=O CCCC(CCNC(=O)C(c1cnn(C)c1)NC(c1nocc1C)=O)CCC c1(C(=O)NC2C(NC(C3(C)CCCC3)=O)CS(=O)(=O)C2)cc2n(c1)CCCC2 N1(C(c2cnc(C(C)C)nc2)=O)CCN(C(C2CCCCO2)=O)C(C(C)(C)C)C1 c1(C(=O)NCCN(C(C(C)n2cncn2)=O)CCc2ccccc2)cc(Cl)no1 c1(C(=O)OC)ccc(C)c(CNC(=O)NCc2cccc(C)c2F)c1 N1(C(c2cnc(S)[nH]2)=O)CCOC(C(=O)NC2CCC(COCC)C2)C1 Cc1noc(C)c1CN(C)C(C1(NC(C23COCC2C3)=O)CCSC1)=O CCC(CC(=O)NC(C1CCCN1C(=O)C(c1ccc(F)cc1)C)C)C1CC1 N1(C(C(C)(C(C)C)OC)=O)CC2CCC1C1CN(C(=O)CCC(C)C)CC21 c1(C(N2C(C(C)NC(C3(C)CC3(F)F)=O)CCC2)=O)ccc2c(c1)CCC2(F)F N1(C(CCc2cc(OC)no2)=O)CCC(N(C(=O)C(CCO)N(C)C)CC)CC1 C1(C(=O)NCCOC2CCC2)C2CC(O)C(C2)N1C(=O)C1=CCCC1 C1(C(=O)OC)CC(C)CN(CC(N2CCCC(C(=O)N(C)C(C)C)C2)=O)C1 c1(CC(=O)NCC(C)N(C(CC(OC)OCC)=O)C)ccc(F)c(COC)c1 N1(C(C2(OC)CCC(C)C2)=O)CCC(NC(C2CCC2)=O)C(C(=O)O)C1 c1(OCC)cc(Cl)ccc1C(=O)NC1(F)CCN(C(=O)COCCOC)C1 CC(N=c1nc2c(cnn2C)c(NCCCC#N)[nH]1)C1CCN(C)C1 c1(C(=O)NC(CN(C(CCN(C(CCC)C)C)=O)C)CC)nccc(C)n1 c1(C(N2C(C(=O)NCC(C)CN(C)C)CC(C)C2)=O)nccc2[nH]ccc12 C1(NC(C2CCCC2)=O)CCSC12CN(C(c1csc(O)n1)=O)C2 CC1CCC(CC(=O)NCC2(F)CC(CNC(c3cn(C4CC4)nn3)=O)C2)O1 C1(CNC(CN(C(COC)=O)C)=O)(NC(C2CC2(F)Cl)=O)CC2CCC1CC2 c1(C(C)C)cc(NC(C)C(C2CCCCC2)NC(C2CN(C)CCO2)=O)ncn1 N1(C(C=C2CCC(C)C2)=O)Cc2ccccc2C(NC(=O)CN(S(C)(=O)=O)C)C1 c1(C(N2CCC(CNC(CSC)=O)C2)=O)ccnnc1C Cc1ccc(C(=O)NC2CC(C(=O)OC(C)(C)C)C2(C)C)c(N)c1C C1(OC)(CNC(C2CCN2C(C)(C)C)=O)CCN(C(=O)C(F)(F)C2CCCC2)C1 c1(CC(N2CCC(OC)(CNC(C3CC3C)=O)CC2)=O)cc(F)c(F)c(F)c1 CC(=NO)c1cc(C(=O)NC2CC2NC(c2cccc(N(C)C)n2)=O)cnc1O C1(C(N(C(C)C(=O)NCC23CC(F)(C2)C3)C)=O)CC2OC1C1CC21 C1(CNC(C(c2cncnc2)C)=O)CC2(CC2)CN1C(=O)C=CCO C1(NC(c2c(CC)nc[nH]2)=O)CN(C(=O)C(OC)OC)CCC1CO Cn1nc(CNC(=O)CC(C2CCC(O)CC2)N)cc1-c1cccnc1 CCC(CC)C(C)NC(C12CC(CN1C(=O)CN1CSCC1=O)C2)=O c1(C(=O)NC(=O)C(C)SCC)cc(C(N2CCCC2COC)=O)ns1 C1(NC(c2c(C(C)C)csc2)=O)CC2(CCN(C(=O)CC3(C)CC3)C2)C1 Fc1cccc2nc(NC3C4CCCCC34)nc(N3CC=CCC3)c12 N1(C(C(=O)NCc2cc(C(C)(F)F)ncc2)=O)CC(O)C2(CCOCC2)C1 C1(NC(C2C(C)(CC)C2)=O)COC2(C1)CN(C(c1ccc(C(=O)OC)cc1)=O)C2 c1(CN(c2ccc(Cl)cc2)CCN(C)C)c[nH]c(=O)c2ccnn12 C(CCC(C(=O)NCCC1CC(C)(C)C1)NC(c1c[nH][nH]c1=N)=O)OC C1(C(=O)NCC(C)(C)NC(C=CC(C)(C)SC)=O)CC2(CCCCC2)CO1 C1(CNC(C2CCCCC2O)=O)CCCC(NC(=O)C(c2cccnc2)O)C1 c1(C(=O)NC2(C)CCN(C(=O)CC3CCC(=O)N3)CC2)csc2ccncc12 C1(CCNC(C(COC)N(C)C)=O)CCN(C(C2(N(C)C)CCCSC2)=O)CC1 N1(C(C(CC=C)OC)=O)CCN(C(=O)C(C(C)OC)N(C)C)CC2(C)CCCC12 CCCCCC(F)C(=O)N1CCC1C1CCCN(C(c2ccoc2Cl)=O)C1 c1(C(N(CC(C)CNC(C2CSCCS2)=O)C)=O)cc2ccccc2[nH]1 C1(O)(C(C(=O)NCC(CNC(Cc2c(C)noc2)=O)O)F)CCCCC1 C1(NC(C2(OC)CCOC2)=O)CCC(NC(C2CC2c2cnc[nH]2)=O)CC1 CS(=O)C1CCC(NC2(c3nnnn3C)CCCSCC2)C1 c1(-c2cn(CC(N3CCC(N4CCOCC4)C3)=O)nn2)ccc(F)c(C(=O)O)c1 N1(C(C(C2CCOC2)OC)=O)CCCC(NC(=O)CC2CN3CCN2CC3)C1C c1(COCC)nc(C)c(C(=O)NC2CCCC(NC(C3CC3F)=O)C2)s1 CC1=C(C(=O)NC2CCCC2C(=O)NCC2CCC(=O)N2)CCC1 C(CC)(CCC(F)(F)F)(c1n(CC=C)nnn1)NC(c1ccc(OC)cc1)C C1(C)(CNC(=O)OC(C)(C)C)CCC(C(=O)Nc2nccc(-c3ccccc3)n2)C1 C1(C(C)C)CN(C(=O)C(C(C)(C)C)N(C)C)CCCN1C(=O)CS(=O)(=O)N(C)C N1(C(C(CSCC)NC(C2CCCC2C(C)C)=O)=O)CCC(N(C)OC)CC1 N1(C(C#CC(=O)N(C)C)=O)CCC(NC(=O)C=CC(C)(C)SC)C(F)C1 N1(C(c2c(C)csn2)=O)CCC(O)C(N(C)C(C2CCCC2(F)F)=O)C1 c1nc(C)c(C(C)C)o1.C12(COC)CC1C(=O)NCCCN(C)C(=O)C2.COC C1(NC(NC)=O)COC(=O)N1C.CCC(C(=O)N1CCC(c2nn[nH]n2)C1)SC c1(C(C)C)ncc(Br)c(C(=O)N(C)CC2COCCN2C(=O)C=CCO)n1 N1(C(C(C)(C)C2CCOCC2)=O)CCCC(CCNC(=O)CN2CCOC2=O)C1 Cc1cc(C)c(CNC(C2(C(C)C)CCN(C(C3CN(C(N)=O)C3)=O)C2)=O)cn1 c1(C(N2CCC(NC(C3(C(F)F)CCCO3)=O)C(O)C2)=O)cccc2c1OCO2 C(=O)(C(CO)NC(C1CC(N(C)C)C1)=O)N(CCN(C)C)C C1(CNC(C2CCSCC2)=O)CC2CCC(C1)N2C(=O)CC1CCCNC1=O c1(C(N(C2CCC(NC(CC=CCC)=O)C2)C)=O)ccc(C(=O)NC)c(F)c1 c1(CN(C)C(C2(N(C)C)CC2)=O)ccc(CNC(c2nscc2Br)=O)cc1 c1(C(=O)NCC(CN(C(C(C)CC(F)(F)F)=O)C)C)ccc2c(O)nccc2n1 N1(C(CN(CC)CC)=O)CCC(NC(=O)C(C)Oc2ccccn2)C1(C)C C1(N(C(COCCOCCOCC#C)=O)C)CC(NS(C)(=O)=O)C1 c1(CC(N2CCC(NC(c3sccc3C3CC3)=O)C2)=O)cc2cc(Cl)ccc2[nH]1 C1(NC(C2CCC2c2nc[nH]n2)=O)(CO)CCCN(C(=O)Cn2cncn2)C1 Cc1ccc(Br)cc1CC(=O)NC1CC1CNC(=O)C(C1CC1)C1CC1 C1(CCOCC)(C(=O)NCCCCNC(=O)C(C)N(CC(F)(F)F)C)CCCC1 C(CC(C(C)C)NC(C1(C2CCCCO2)CCC1)=O)N(C(c1cc(C)sc1)=O)C c1(OC(C(=O)NC(C2OCCN(C(C(C)OC)=O)C2)C)(C)C)ccc(F)c(F)c1 C1(CNC(COC(CC)C)=O)CCCCN(C(=O)C(F)(F)Nc2ccccc2)C1 N1(C(C(CC)F)=O)CC2CC2(NC(=O)CCc2c(C)noc2C)C1 C1(C(=O)NC)(NC(=O)CCC23CC2CCN3)CCCCC1 c1(C(=O)NC(C2COCCO2)C)cnc2c(c1)CNC2=O CCCCS(=O)(=O)CC(=O)NC1CCOCC1NC(=O)Cc1sc(O)nc1O C1(C)(CNC(C(CC(=C)C)OC)=O)CN(C(C2CCC2C(=O)OC)=O)C(C)(C)C1 C(=O)(C(C)CC(=O)NCCCOCCC(=O)N(c1ccc(O)cc1)C)OC c1(NC(C2CCCN(Cc3cc[nH]n3)C2)=O)c(O)cccc1F C1(CC(n2cc(Cn3ccc(C(=O)OCC)n3)nn2)C)CCN(C)CC1 N1(C(C(F)=CC)=O)CC(NC(=O)Cc2coc(C(F)F)n2)C(n2ccnn2)C1 c1(C(=O)NCC2OCC(CNC(c3c(CC)nc(C)[nH]3)=O)C2)cc(Cl)ccc1O N1(C(C2(S(C)(=O)=O)CC2)=O)CCCC(NC(=O)C(=Cc2cccc(F)c2)F)CC1 c1(C(=O)NCCNC(C23OCC(CC)(C2)C3)=O)ccc(N)c(F)c1 C=C=CC(C)C(=O)NCCCCN(CCCNC(=O)CCCCN(C)C(C)C)C C(=O)(CCCC(C)(C)NC(c1cccnc1O)=O)NC(C)CCN(C)C c1(C(N2CC(C)C(NC(C3CCOC3)=O)C2)=O)csc2nnsc12 C1(CC(=O)N(CC(N2CCC(OCC=C)C2)=O)CC(C)C)CCCOCC1 C(=O)(C(F)(F)C(F)F)NCC(c1cn(C)nn1)NC(CS(=O)(=O)NCC)=O c1(C(C)NC(c2c(C(CC)(C)C)cccc2)=O)cccc(F)c1F N1(C(c2c(F)ccc(C#C)c2)=O)CCOC2(CCN(C(c3c[nH]nc3C)=O)C2)C1 c1(C(N(C)CC2(O)CCCN(C(C(CCSC)O)=O)C2)=O)cccc2c1OCC2 N1(C(C(C)(C)O)=O)CCC2(CC1)CN(S(=O)(=O)CC#N)CCO2 Nc1c(C(=O)NCC2(NC(=O)CC3CCC(O)C3)CCOCC2)cc(F)cc1Cl c1(SC)ncc(C(N2CCC(F)(CF)C2)C(=O)Nc2ccccc2)n1C c1(OC)ccc(CC(C)C(=O)NC2CCC2NC(=O)CN2CC3CC3C2)cc1 Cc1csc2ncnc(NC3CCC3C(C)C)c12 c1(NC2CC3CN(C(CC4CCC(=O)NC4)=O)CC32)ncc2scc(Br)c2n1 c1(C(=O)OC)coc(C(=O)NC23CC(NC(c4ccc(C(C)C)[nH]4)=O)(C2)C3)c1 c1(C(N2CCN(C(C(CC)C)=O)CC3(C2)CC3)=O)ccc2nnc(C)c(C)c2c1 c1(C(N2CCCC(N(C(C(C=C)(C)O)=O)C)CC2)=O)[nH]c2c(c1C)C(=O)CCC2 Cc1cccc2c(C(=O)NCC3CC3NC(C3(N(C)C)CCCCC3)=O)coc12 N1(C(CNS(CC)(=O)=O)=O)CCC(CO)(CNC(C2(O)CCCCCC2)=O)CC1 C1(NC(C2(C)CC(=C)C2)=O)(CF)CCN(C(=O)C(c2ccccn2)O)C1 CC1C(OC(c2ncoc2C2CCOCC2)=O)CC(=O)N1C c1(C(=O)NC2C=CC(CNC(CCn3c(C)cc(C)n3)=O)C2)c(F)cccc1Cl c1(CNC(COCCC)=O)nc(C)c(C(=O)NCc2ccn(C(C)C)n2)o1 C1(C)(C(N2C(CN(C(=O)CC34COC(CF)(C3)C4)CC)CCC2)=O)CCSCC1 C(CC(F)F)(C(=O)NCCc1cn(CC)cn1)N(C(c1c(CC)n[nH]c1)=O)C C1(NC(CN(C2CC2)CC)=O)(CC)CCN(C(=O)C(C)CSC2CC2)CC1 c1(CN(C)S(N)(=O)=O)ccc2n[nH]cc2c1.N12CCCCC1Cn1cc(nn1)C2 c1(C(=O)NC2CN(C(c3scc(C)n3)=O)CC2C)ccc2ncn(C)c2c1 c1(-n2cc(CN(C(CN3CCC(OCC)C3)=O)C)nn2)cc2cccc(C)c2[nH]1 C1(CCOC)(NC(=O)CCCC(C)O)CCN(C(c2ccncn2)=O)CC1 C1(OC)CC(C(=O)OC(C)(C)C)CN(C(=O)C(N2CC3CC2(C)C3)=O)C1 C12(C(=O)NC3C4CN(C(C5(c6ccccc6)CCC5)=O)CC34)CC3CC1C2C3O N1(NC(C2CC(CC3(NC(C4CC(CC)C4)=O)CCOC3)C2)=O)CCCS1(=O)=O c1(C(=O)NCC(C)(C)NC(CC(COC)C)=O)cccc2c[nH]nc12 N1(C(C23CC(C)(C2)C3)=O)CCOC(CNC(c2sc(Br)cc2Cl)=O)C1 Cc1nc2c(o1)CCCC2CC(=O)N1CC2CC2(NC(=O)CC=C(Cl)Cl)C1 C(CCCC(=O)NC(C(=O)N1CC(c2cccs2)C1)c1ccco1)OC Cc1ccc(C(N2CCC(C)(C)C2CNC(C2CCCCO2)=O)=O)nc1O C1(C(=O)NCC2(OC)CCCC2)CCOCCN1C(=O)C(C)C1CCC1 C12(C(N3C(CN(C(C4C(C)OCC4)=O)C)CCC3)=O)CCCC1C2(F)F C1(NC(c2c(CC)[nH]cc2)=O)CC(CNC(c2cnc(CC3CC3)s2)=O)C1(C)C C1(NC(CNC(=O)OCC)=O)CN(C(c2ccccc2NC)=O)CC2(CCC2)C1 CC(CCCCNC(=O)C(=Cc1cccnc1)F)NC(=O)CC1CCCO1 C12(CNC(CN(CC)CC)=O)CCCC1CCN2C(=O)C=Cc1ccncn1 N1(C(C(C(C)C)SCC)=O)CCC(NC(=O)CCCc2cncs2)CC(C)(C)C1 C1(CNC(C2(CC)CCOC2)=O)CCN(C(c2cncs2)=O)CC1CC c1(C(=O)NC2CN(C(Cn3c(C)cc(C)n3)=O)C(C)C2)ccc(CCCC)c(C)c1 c1(CC(=O)NC2CC(C)(CNC(c3nc(C)sc3)=O)C2)cnccc1C C1(O)(C(=O)NCC(C)CN(C(=O)COc2ccon2)C)CCSCC1 c1(NC(CN(CCOc2ccc(CN)nc2)CC)=O)cccc(CCCCC)c1.OC c1(C(=O)NCCCN(C(CC2CC(C)C2)=O)C(C)C)ccc(F)cc1F N1(C(C2(CSC)CC2)=O)CCC(CCNC(=O)CCc2ccc(O)cc2)CC1 Cc1cnn(C)c1C(=O)NC(C1CCCN(C(C2CCN(C(C)C)CC2)=O)C1)C N1(C(Cn2c(C)cnc2)=O)CCC2(CCCN(Cc3ccc(F)cc3)C2)C1 c1(CNC(CC=C(C)C)=O)ccc(C(=O)Nc2cccc(C3CC3)c2)cn1 C1(NC(C2CCCC2)=O)CN(C(c2cn3ccccc3n2)=O)C2(CCCC2)C1 CC(C)(C)C(CNC(c1cnn(C(C)(C)C)c1Br)=O)NC(C1CCC2CC12)=O c1(C(=O)NCCC2CC3CCC(C2)N3)nc2ccccn2c1Br CC1CCC(NC(=O)CC(C)(C)c2cccs2)CN1C(=O)CC1(O)CCCOC1 N1(C(C(OC)OC)=O)CCN(C(=O)CCc2ccc(C)nc2)C(CF)C1 CCC(CC)C(=O)NCC(=O)NCC1CCCCN1C(C12CC(CC)(CO1)C2)=O Cc1ccc(C(C)(CNC(=O)NCc2cc(C)c(C)o2)CO)cc1 C(=O)(CCCCCF)N1CCC(F)(CNC(=O)CCc2ccccc2)C1 C1(NC(C2CCCC2)=O)CCCC1CC(=O)N(C(C)C(=O)OCC)CCC C(=O)(C(C(C)C)N(C)C)N(CCCNC(=O)C(C1CC1)SC)CCC CC1CCCCC1(CNC(=O)C(C)(C)C(N)=O)NC(=O)C=C1CCCCC1 N1(C(c2ccc(SC)o2)=O)C2CCC1(CNC(C1(C)CCNC(=O)C1)=O)CC2 n1(CC)nc2c(c1C(=O)NC1CN(C(C3(C(N)=O)CC3)=O)CCC1F)CCCC2 N1(C(c2cc(CCCCC)[nH]n2)=O)CCOCC(NC(=O)CSc2cn[nH]c2)C1 c1(C(N2CC3C(NC(Cc4cnn(C)n4)=O)C3C2)=O)c[nH]c2cccnc2c1=O c1(CC(=O)NCC(N(C)C(c2ccn(C)n2)=O)C2CC2)cnc2cccnn12 c1(C(=O)OC)cc(C)n(CC(=O)NCCNC(c2nccc(C)n2)C)c1C C(=O)(CC1CCc2cc(Br)ccc21)NCCCNC(C(CC#C)C1CC1)=O Cc1csc(=NCC(=O)NC2(C)CN(C(c3cnn(C(C)C(C)C)c3C)=O)C2)[nH]1 C1(NC(C2(CCCC)CCC2)=O)(COC)CCN(C(c2ccncn2)=O)C1 C(=O)(CC(C)(C)C)NCC1C(NC(C(CC2CC2)OC)=O)CC1 C12(C(N(C)Cc3c(CNC(C4C(=C)C4)=O)cccc3)=O)CCC(OC)(CC1)CC2 C(=O)(C(C)(C)C#C)N(CCC(=O)N(C)CCC1CC1)CC#C N1(C(C2CC=CC2)=O)CCC(CC2COCCN2C(C2CC=CCC2)=O)CC1 c1(C(N2CCC(C(=O)NC(CC)C)CC2)=O)ccc2ncccn12 N1(C(C(C(=O)OC)C)=O)CCCC12CCN(C(c1nccnc1C)=O)C2 N1(C(c2n(CC=C)ccc2)=O)CC2CCN(C(=O)C=CCOC)C2C1 O=C(C#CC1CC1)N1CC=CC(C(=O)NCCC2CC(F)C2)C1 CCCCC(C(=O)N1CC=CC(NC(C2CCC(C)=C(C)C2)=O)C1)N(C)C CS(=O)(=O)c1ccccc1C(N1CC(NC(C23CCCC(CCC2)C3)=O)C1)=O c1(C(N2CCCC(CCC(=O)NC3CC3C3CCC3)C2)=O)cc([N+](=O)[O-])n[nH]1 c1(O)ccc2cc(C(=O)NCCNC(C3CCCS3)=O)ncc2c1.C1(OC)(C)CC1 C=CCCCCC(C(=O)Nc1cccc(OC)c1)N1CCOC(CN(C)C)C1 C(=O)(CS(=O)(=O)CC(C)C)NC1C(NC(c2c(C)oc(Cl)n2)=O)COCC1 N1(C(c2n(C)nc(Br)c2)=O)CC2CCN(C(=O)CC3COC(=O)C3)CC2C1 CC1(CNC(=O)CC(F)F)CCCN(C(=O)C(c2ccc(F)cc2)C2CC2)C1 C1(COC)CN(C(=O)C(C)(C)CF)CCN1C(=O)Cc1c(C)noc1Cl C#Cc1cccc(C(=O)NC(C(=O)NCC2NC(=O)NC2=O)c2ccoc2)c1C C1(C(=O)NC(C)C(CO)NC(c2ccc(N)c(Cl)c2O)=O)CCc2cncn2C1 C(=O)(C1=Cc2ccccc2C1O)NCCOCCCNC(c1c(C)noc1C)=O n1(CCOC)cc(CNC(=O)C(Cc2ccccn2)NC(=O)CC(C)O)nn1 c1(-c2cn(CC3N(C(C4(COC)COC4)=O)CCCC3)nn2)cccc(Cl)c1F c1(CC)ccc(C(=O)NC2(CNC(=O)C(C)=C3CCCC3)CCCC2)o1 N1(C(C2(C#C)CN(C(c3cnn(CCO)c3)=O)C2)=O)CCn2ccnc2C1C C1(NC(c2ccc(OC)nn2)=O)CCN(C(c2c[nH]c(=N)nc2C)=O)CC(O)C1 C1(CC(=O)NCC)CCC2(CC1)CCN(C(=O)C(N1CCC(C)C1OC)=O)CC2 CC1CCCC1C(=O)NCC1(F)CC(NC(=O)COC2CCOCC2)C1 N1(C(c2cc(C)c(C)o2)=O)CC2CN(C(=O)C(C)c3ncco3)CC2(C)C1 c1(C(=O)NCC2N(C(CCSCCCC)=O)CC2)cncc2ccccc12 C(=O)(C(CC(C)C)OC)NCC(CC)NC(c1cccc(CO)n1)=O c1(C(=O)NC2C=CCN(C(C3CC3(Cl)Cl)=O)C2)cc([N+](=O)[O-])cc2ccccc12 C(=O)(C(C(C)C(C)(C)C)N1CCOC(c2n[nH]c(CO)n2)C1)NC(CC)C C=CC1(CC(=O)NC2(COC)CN(C(c3cnc(C4CCCO4)s3)=O)C2)CCC1 c1(C(N2CC(NC(C(C)=C(C)C)=O)C(C(F)F)C2)=O)ccc(Cl)c(F)c1 C(=O)(C(F)C(C)(F)F)N(CCC(=O)NC1CC12CC2(F)F)CC#C c1(C2(C(N(CC(CC)NC(=O)CCCNC(C)=O)C)=O)CC2)cccc(C#N)c1 c1(SC)cccc(F)c1C(=O)NC1CC(N(C)C(C2CCCN(C)C2)=O)C1 c1(C(=O)NCC(CC)N(C)C(C2(C)COC2)=O)ccnnc1O CC1CCN(C(=O)CC2CCOCC2)C1C(=O)NOC1CCC1 C12(C(=O)NCC(CC)NC(c3ccc(COC)s3)=O)CC3CC(C1)CC(O)(C3)C2 C1(N(C(=O)C(=O)NCc2ccccn2)C)C2CCOC2C1(C)C.c12nccn1C2 Cc1c(C(=O)N(C)CCN(C)C(C2CC2[N+](=O)[O-])=O)sc2nccn12 c1(-c2cn(-c3ccn(C(CC)CC)n3)nn2)ccnc(F)c1.C1C(=O)NCCO1 Cc1nc2ncccn2c1C(=O)N(C1CC2CC1CN2)c1cc(C(C)(C)C)no1 C(=O)(C(O)CC(C)C)NCC1(O)CCN(C(c2ncn(CC)c2)=O)C1 O=S(=O)(c1ccc(Br)cc1NCCCC1CC1(Cl)Cl)NCCN1CCC2(CC1)CC2 c1(CNC(c2ccccc2C(F)(F)F)=O)ccc(F)nc1Br C1(CNC(CCC)=O)CN(C(c2nc(Br)c[nH]2)=O)CC12CCC2 N1(C(C2CC(OC)C2)=O)CC(C(=O)NCC(=O)NCC(F)F)CCC1(C)C c1(C(N(CCNC(C2CC(=O)N(O)C2)=O)CC)=O)ccc2c(c1)OC(F)(F)O2 c12ccc(nc1)c(=O)n2C.C1(C(=O)OC(C)(C)C)CCN(Cc2ncccn2)CC1 CC1CCN(C(=O)C(F)C2CC2)C(CNC(=O)C(c2cccnc2)(C)C)C1 c1(C2(C(=O)NC3(C)CC(C)C3)CCC2)ccc(-c2nn[nH]n2)cc1F C1(CCC(=O)NCCOC2CN(C(c3csc(-c4cccs4)n3)=O)C2)CCCOC1 c1(CNC(c2ccc(Oc3ccccc3)c(Cl)c2)=O)ccc2c(Br)cccc2c1 c1(C(N(C2CCCC(NC(=O)C3CC3)C2)C)=O)ccc([N+](=O)[O-])cc1[N+](=O)[O-] C1(C)(CN(C)C(C2CC2CNC(c2csc(Cl)c2)=O)=O)CCCC1 C(=O)(CC1=CCN(C(=O)C(C)n2cccc2)CC1)N(C1C(C)CN(CC)CC1)C S(=O)(=O)(c1cnc(NC(c2ccc(C)s2)C)c(Cl)c1)NCC(CC)(C)COC C#CCCN=C(NCc1cn(CCC)c2ccccc12)NCC(C)(C)CC(C)O C1(OC)(CNC(c2c[nH]nc2C2CCCO2)=O)CN(C(c2cccs2)=O)C1 CC(CC(F)F)C(=O)N1CCC(O)(CCNC(=O)COc2ccc(F)c(F)c2)C1 c1(COC)nc(CNC(=O)C(C2CCOC2)NC(C2CC(C)(C)C2)=O)no1 c12cnn(c1C)CCCC2.C1(N(CCC#C)CC=C)CCN(C(=O)C2CC2)CC1 C1(C(N2CC(COC)(CNC(=O)C=CC(C)C)C2)=O)CCc2ncc(C)n2C1 N1(C(C2CCCN(c3ccn(C)n3)C2=O)=O)CCC2(CC(NC(=O)CO)CO2)C1 Cc1nn(C)c(C)c1C(N1CCOC(C(N2CCC(O)(C(N)=O)C2)=O)C1)=O n1(CC)nc(C(C)C)cc1C(N1CC2CC1C2CNC(=O)CCC1CCCO1)=O C1(NC(C(CCCC)C)=O)CCC2(CC1)CN(C(C1C3CCCC13)=O)C2 c1(C(=O)NC2CC(N(C(c3c(CC)cco3)=O)C)C2)ccc(N(C)C)c(C#N)c1 C(=O)(CS(=O)(=O)CC)NCCOCCNC(c1cc(CC)no1)=O C1(CNC(C(CC)n2cccn2)=O)CCN(C(c2ccc(Cl)cc2)=O)CC1O N1(C(C2(COC)CC=CC2)=O)CCC2CN(C(C3CCc4ccnn4C3)=O)C2C1 C1(NC(C2C(=C)CC2)=O)CC12CCC(NC(c1cc(S(N)(=O)=O)c[nH]1)=O)CC2 C=CC1(NC(=O)CC2(NC(=O)CC(C)OCC)CCC2)CCOCC1 C1(NC(C(CNC(C2CCCOC2)=O)O)=O)CC2(CCC2)C1O C1(C(C)NC(C2(C3CC3)CCCO2)=O)CCN(c2ccnc(CN(C)C)n2)CC1 c1(NC(C(=O)NCC(C)(C)C(F)(F)F)=O)ccc(C#N)c(Cl)c1 C12(NC(Cc3ccc(CCCC)cc3)=O)CC(CNC(=O)C(C)SC)(C1)OC2C C=CCCCCC(=O)N1CC(CNC(C2CC2c2cccs2)=O)C(O)C1 C(CC(CO)NC(=O)CCCNC(=O)C(CO)OC)=CC N1(C(C)=O)CCC(C2CC2)(C(=O)OC(C)(C)C)C1.N12CCCC13CN(C3)C2=O c1(C(=O)OC)ccc(N2CCC(CNC(=O)C(=Cc3cccs3)C)C2)nc1C c1(C(N2CCC(CN(C(C(C)CC3CC3)=O)C)C2)=O)cc(Br)ccc1O C1(CC(=O)N(CC(C2CC2)OC)C)CC(C)N(C(=O)OC(C)(C)C)C1 c1(C(N2CC(NC(CCc3n(C)ccn3)=O)C(C(F)F)C2)=O)n[nH]cc1[N+](=O)[O-] C1(CNC(C(Br)=C(C)C)=O)CC2COCC2N1C(c1coc(C(N)=O)c1)=O C1(C(=O)NCC2(C(=O)N(C)CC3CC3(C)C)CC(=C)C2)CCC(CC)CC1 C(=O)(C1Cc2ccccc21)NC1CCN(C(c2ccn(C)c2)=O)C1C1CC1 C1(C(=O)NCCCCNC(CC(=O)N(CC#C)C)=O)C=CC=CC=C1 CCC(C(=O)N1CC(C)CCC1CNC(c1ccc(NC=O)cc1)=O)C(C)C CC(C)C(C)C(CNC(=O)CCc1ccc(F)cc1)NC(=O)C(F)=CCCF Cc1ncc(CC(=O)NCCOCCCNC(C2(C(F)(F)F)CC2)=O)[nH]1 Cc1nc(C(=O)N)cn1C.N1(C(C(C)CC=CC=CC2CCCC2)=O)CC2(CCC2)C1 c1(C(=O)NC2(CCNC(Cc3nnc(C)o3)=O)CC2)cnc(C)c(C)c1 Cn1ccnc1CC(=O)NCCCN1CCC(NC(=O)CCn2cc(Cl)cn2)C1 N1(C(COCCC=C)=O)CCOC(CCCNC(=O)CC2CC=CCC2)C1 Nc1ccc(NC(C2CN(C(=O)CNS(=O)(=O)C3CC3)C2)=O)cc1[N+](=O)[O-] c1(CCC(N2CCN(C(=O)C(F)OC(F)(F)F)C(CO)C2)=O)ccc(F)c(F)c1 c1(-c2c(C(C)NCC(F)(F)F)cccn2)ccc(C)c(F)c1F C1(C(=O)NC(CCCC=C)C)CN(C(c2ncnc(C)c2C)=O)CC1(C)C C1(C)(C(N2C(CN(C(c3cc(C)no3)=O)C)CCC2)=O)CC(C#N)C1 c1(C(N2CC3C(C(N4CC(OCC)C4)=O)C3C2)=O)ccc2c(c1)CC2 C(=O)(C(O)C(C)(C)CC)NCc1cccc(NC(c2nncc(CCC)c2)=O)c1 c1(N(C(c2ccc(C)o2)C(=O)NC(=O)NCCCSCC)C)ccc(F)cc1Br C1(NC(C(CC)F)=O)CN(C(c2cncc(OC)c2)=O)CC1CC CC1CN(C(=O)CNC(=O)Cc2ccccc2)CCN1C(=O)COCCF CC(C)CC(C)(O)CNC(C1CCCC(NC(c2cc(Cl)cs2)=O)C1)=O N1(CCOC)C2CCC1CC(N(S(=O)(=O)CC(=O)Nc1ccccc1)C)C2 Cc1cnc(N(C(=O)CCCCCl)CC2(F)CCCNC2)nc1C c1(CCC(=O)NCC2CCN2C(=O)C=CC2CCC2)ccc(Cl)nc1 Cc1ccccc1CCC(=O)NC1CCC(CNC(c2ccccc2Br)=O)CC1 c1(C(N2CCOC3COCC23)C(=O)NCCOC)cc(C)c2occc2c1 CC1CN(C(=O)C=C2CCOCC2)CC1CNC(c1cnc(C2CC2)nc1)=O c1(OCC)ccc(-c2cnc(OC)c(C(N3CCOC(CC)C3)=O)c2)cc1F C#Cc1cccc(C(=O)NC(C)(CSC)C(=O)NCCCC(=O)OC)c1 Cc1nn2cc(NC(C3CC(CNC(=O)C(C)Sc4ccccn4)C3)=O)nc2s1 C(=O)(CC(O)C(C)(C)C)NCCN(C(C)C)C(C1CCc2nc[nH]c2C1)=O N1(Cc2ccc(C)cc2)CCC(NC(c2ccc(C(C)C)s2)=O)CC1C c1(C(=O)NC(C2CC2(Cl)Cl)C)ccc(OCC2CC2)c(F)c1 Cc1sc(C(=O)NCC(C)(CO)NC(=O)Cc2ccc(O)cc2)nc1Br CC(CCS(C)(=O)=O)NC(=NCCSC)NCc1ncnn1-c1ccccc1 n1(CC)nc(C(=O)NC23CCC2CN(C(c2csc(Cl)c2OC)=O)C3)ccc1=O c1(N(CC(C)CNC(c2ccc(N3CCCC3=O)cc2)=O)C)snc(Cl)c1C#N N(C1CCc2cccc(Cl)c21)C(CNC(c1ccc(C)cc1)c1nnnn1C)=O CC1(C)C=C(C(=O)N2CCC(C(C)(C)C(=O)NC3(C)CCCCC3)C2)C1 N1(C(c2cn(CC)nc2C2CC2)=O)CCC(NC(=O)Cn2cncn2)C12CC2 c1(NCC(CC)(CC)NC(=O)CC2CC3CCC2C3)cc(C)nc2c(C)cnn12 c1(C(C)=O)cnc(Cl)[nH]c1=NCC1CCC(NC(=O)C=C(C)I)C1 C1(F)(C(=O)NC2CCC(C(N)=O)C2)CCN(C(=O)CCC2CC2)CC1 N1(c2nc(C)cc(OC)n2)CC2CCN(C(C3CC3c3ccc(F)cc3)=O)C2C1 c1(NC(C)=O)nc(C(=O)NCC(C)N(C(=O)Cc2cnn(C(C)(C)C)c2)C)cs1 CC(CCCCO)NC(c1ccc(CNC(C2CCC2(F)F)=O)cn1)=O C(=O)(CC(O)CNC(=O)CC(C)n1cccn1)NC(C1CCCC1)C#C C1(C(N(C(CNC(C(C)CS(C)(=O)=O)=O)C2CC2)C)=O)CCC2C(CC1)C2(F)F n1(CC(=O)NC(CC(C)C)CNC(=O)Cc2ccns2)nc(Cl)ccc1=O C1(CC=C)(NC(c2ccc(=O)n(C)c2)=O)CCCN(C(c2cnnc(Cl)c2)=O)C1 c1(CCC)ccc(-n2nc(C(C)O)nc2CCCn2ccnc2)cc1 O=C(CC(C(F)F)C1CCCC1)N1CC(O)(c2cscc2)C1 O=S(=O)(c1cncc(Br)c1)NC1CN(C(c2cc(Br)ccn2)=O)CC(F)(F)C1 O=C(CCCCCNC(C1COC(=O)N1)=O)NCC1(O)CCOC1 N1(C(CC2CC(OC)C2)=O)CCC(CNC(=O)C(C)CN(C)C)C(O)C1 c1(CN2CCC(CCCNC(C3CC3F)=O)C2)ccc2ccoc2c1 C(C(C)(C)CC(=O)NC(C)(CNC(=O)C=Cc1scnc1C)C1CC1)OC CCCCCC(C)N=c1ccc2[nH]c(-c3ccco3)cc2[nH]1 c1(C(=O)NCC2(NC(CN(C)CC)=O)CCOC2)ccn(CC(F)(F)F)c(=O)c1 CN1CCCC(CCC(=O)N(C(CNC(C2(C#N)CCC2)=O)C2CC2)C)C1 N1(C(=O)NCc2ncc(C#C)cn2)CCC2CCCCC12 N1(C(COC(C)=O)=O)CC(NC(=O)C(C)C2CCC2)Cc2ccccc21 C1(CNC(c2cn(C)nc2Cl)=O)CCCCN(C(C2CN3CCC2CC3)=O)C1 Cc1nc2c(N3CC4(CN(C(=O)C(C)(C)F)C4)C3)ncnc2[nH]1 c1(C(=O)NCCC2CCN(C(C3(O)COC3)=O)CC2)cncc2c(Cl)cccc12 Cc1nn(C)c(C(=O)Nc2ccccc2OCc2ccc(Br)c(F)c2)c1Cl CC1CCN(C(=O)CC23CCC(CC2)C3)CC1NC(c1ccsc1Cl)=O Cc1[nH]nc(C(=O)NC(C)(C)CNC(C2CC2c2ccnn2C)=O)c1O c1(CNC(=NC)NCC(O)COCC(C)C)ccc(N2CCOCC2)cc1 N1(C(C23N(C(c4cc(C)[nH]c4)=O)CC(C2)C3)=O)CC2CC1CN2C(C)C CC1CC(C)(C)CCC1NC(=O)NCCc1cccs1 N1(C(c2c(F)ncc(-c3cc(C)c(F)cc3)c2)=O)CCC2(CC1)OCCO2 C=C=CC(C)C(=O)NCC(C1CC1)N(C(=O)CCc1cccnc1Br)C CC1CCCN(C(C2CCCCCCC2)=O)C1CNC(C1CCC1)=O N1(C(c2c(SC)ccs2)=O)CCC(NC(C2CCCC(C(F)(F)F)C2)=O)C1C C1(C(=O)NCCC(=O)N(C2CCCCC2)C)CN(Cc2nnnn2C)CCO1 CC(CC(=O)NCCCN(C)C(C1CC(C)(C)OC1(C)C)=O)C(C)(C)C CC(c1ccccc1Cl)=CC(=O)NCCOC1CN(C(C2CC23CC3)=O)C1 c1(C(=O)NC2CC(N(C(=O)CCc3n[nH]c(=N)s3)C)C2)nnc2ccccc2n1 C1(NC(CNS(CC)(=O)=O)=O)CCCC(NC(=O)C=C2CCCCC2)C1 CC1(CNC(C2CCCN2C=O)=O)CCN(C(c2cccc(C#N)c2)=O)CC1 Cc1cc(CC(=O)NC2CC(CCNC(=O)Cc3ccoc3C)C2)no1 Cc1nn(C)c(C)c1-c1cn(CC2C=CCN2C(c2occc2Br)=O)nn1 C1(NC(C2(CNC(CC(C)OC)=O)CCC2)=O)CCCC(O)C1O c1(OC)ncc(F)cc1C(=O)NC(C1CCCN1C(C1CSCC(=O)N1)=O)C c1(C(N2CC(O)(C(C)NC(CC(C)SC)=O)C2)=O)cnc(C(F)F)nc1 N1(C(C(c2cncn2C)N(C)C)=O)CCC2CN(Cc3ccccc3)C2C1 c1(C(N2CC(C)C(NC(c3cccs3)=O)C2)=O)cc(Br)c(F)cc1N c1(NC(CC)C(C)O)ccc(S(=O)(=O)N(CCCCN(C)C)C)c(Br)c1 c1(C(=O)NC(C2N(C(C=C(C)C)=O)CCCC2)C)cnc(C2CCC2)nc1O CC(C(=O)NC1CC(F)C1)C(C)NC(=O)CC1(C)CC1 N1(C(c2c(CC)cccc2)=O)CCCC(NC(c2ccc([N+](=O)[O-])[nH]2)=O)C1C Cc1cc2ncc(C(=O)NCC=CCNC(c3ccnnc3C)=O)cc2[nH]1 CC1(C(=O)NCC2CC(F)CN2C(=O)C=Cc2cnc[nH]2)CCCOC1 C(=O)(CC(C)P(C)(C)=O)c1c(OC)cccc1.C1(=O)NNC(=O)C2CCN1CC2 C1(NC(c2c(SC)ccs2)=O)CC(C2CCN(C(=O)CNC=O)C2)C1 C=CC(CCC)CC(=O)N1CCCC(C(=O)NC(c2ccsc2)C)C1CC Cc1cc(=O)c(C(N2CCCC2(C)CNC(c2cccc(C3CC3)n2)=O)=O)c[nH]1 c1(CNC(C(C2(O)CCC2)NC(CC2C(C)C2)=O)=O)cnn(CCF)c1 c1(CNC(C2CC(F)CN(C(c3ccnc(F)c3)=O)C2)=O)cc(O)nc(O)n1 CN1CCN(C(=O)C=C(Cl)Cl)C(CNC(c2cn(C)nc2Cl)=O)C1 c1(C(=O)NC2C(NC(C(CC)O)=O)CC2)cc(F)ccc1OC(C)C N1(C(Cc2cn(C(C)C)nc2)=O)CCCC(NC(C23CCC2C3)=O)C1 C12(NC(CS(=O)(=O)NCC)=O)CCCC1CN(C(=O)CC1CN3CCC1CC3)C2 FC1(CNC(c2ncsc2Br)c2nnnn2C2CCCC2)CCCCC1 C1(CN(C(=O)CCc2cnccn2)C)CCCN(C(C2COCCO2)=O)C1 c1(CC(=O)OC)cc[nH]c(=NCCC2(CNC(=O)C(C(C)C)NC(N)=O)CC2)n1 Cc1[nH]c(C#N)cc1C(=O)N(C)CC1CCCC(NC(c2cnnc(C)c2)=O)C1 N1(C(C(CCCC)(C)F)=O)CC2CCCC(C1)N2C(=O)C(CC)CC(F)F c1(C(N2CC(OC)C(NC(=O)C(O)C(C)C)C2)=O)c(Cl)ccc2ncccc12 CCCCCC(C)CC(=O)NCc1cc[nH]c1C(=O)NCCN(C)C(C)C c1(C(=O)NC2(CNC(c3[nH]cc(C(C)=O)c3)=O)CCC2)cc(O)ncn1 C=CCC(C)(CNC(c1conc1C(C)NC(=O)CN(C)C)=O)CO c1(C(N2CC(CCC)C(NC(=O)Cc3c[nH]nc3C)C2)=O)cc2cn[nH]c2cn1 c1(OC)cccc(C(C)(C)NC(=O)CCC(=O)c2cccnc2)c1C C1(NC(C2CC3(C2)CC3F)=O)CN(C(c2c[nH]c3nccc-3c2)=O)CC12CCC2 c1(C=O)c(O)cccc1Br.N1(C(C)=O)CC(OC(C2CC2C(C)N)=O)C1 c1(SC)ccc(C(=O)NCC2(Nc3ccncn3)COC2)cc1Br C1(C(C)(C)CNC(C2CCCC2F)=O)CCCN1C(C1(C2CCCO2)CC1)=O CCC(C)(CNC(=O)CN1CCOCC1)C(=O)N1CCC(N(C)CC2CC2)CC1 c1(C(N(CC(C)NC(c2ccnc(NC)c2)=O)CC)=O)ccc(C)c2c1CCC2 N1(C(C2CN(C(C)=O)C2)=O)CCC(C(C)NC(=O)CSC(F)(F)F)C1 Cc1ccncc1CCNC(C12CC1CN(C(c1ccc(CO)o1)=O)C2)=O c1(CNC(CC2C3CN(C(C)=O)CC2CC3)=O)nccc2ccccc12 C1(C(C)C)CN(C(C2CCS(=O)(=O)C2)=O)CCCN1C(=O)C1=NNC(=O)CC1 C1(NC(C2C(=C)CC2)=O)CC2(C1)CC(CNC(C1CC3CCC(C1)C3)=O)C2 C(=O)(CCCCC(C)C)NCC1CCC(CNC(c2c(C)ccnc2Cl)=O)CC1 N=c1[nH]cnc2cc(C(=O)NCC3CCC3NC(=O)CCF)ccc12 CCC(C)C(C(=O)N(C)CCC1CCCC1)N(C)C(c1ccc(O)nc1C)=O c1(OCC)ccc(Br)c(CN2CC3CC2CN3C(C2CCCS2(=O)=O)=O)c1 C1(C(=O)NC2C(NC(c3ccccc3Br)=O)CC2)CCc2nncn2CC1 CC1OC(C)C(C(N2CCCC(N(c3cc(Cl)nc(C4(C)CC4)n3)C)C2)=O)C1C C(=O)(C(F)(F)C(O)C(C)C)NC1CC(NC(C2N(C(C)=O)CCOC2)=O)C1 CCC(CC(=O)N1CC(F)CC1CNC(c1cnn(CC(C)C)c1C)=O)C1CC1 N1(C(c2c(C)con2)=O)CCC(NC(c2ccn(CCF)n2)=O)C(O)C1 C1(CC(=O)NC2C3CCN(C(c4cncc(C)n4)=O)C32)OCCCC1(C)C N1(CC(=O)NCCC(=O)N(CC(C)O)C)C(=O)CCCC1=O C=CCC(C(=O)NCCCCCC(=O)N(CC(CC)OC)C)C(C)C CCCCCC(=O)N(C)CC1COCCN1C(C1CC1(C(C)C)CC)=O c1(NC(=O)NC2CC(C(C)(C)C)C2)cccnc1 CC1(C(N2CCC(c3cccs3)CC2)=O)CCCCCCC1 N1(C(C(c2cccc(C)c2)O)=O)CC(C2CCN(C(c3ccc(=N)[nH]n3)=O)C2)C1 C1(NC(COCCC=C)=O)CN(C(c2ncsc2C2CC2)=O)CC2(CC2)C1 C=C1Cn2c(C(=O)NC3CC(C)CN(C(c4cnc(Cl)s4)=O)C3)nnc2S1 Cc1cc(C(=O)NC(CNC(=O)C=C2CC2)C(C)C)n[nH]1 c1(C(=O)NC2(F)CC(NC(c3ccc(CN(CC)CC)o3)=O)C2)cc(CO)n(C)n1 CN1CCC(C(=O)NCCC2(C(=O)NCC3(CO)CCCO3)CCC2)C1=O CC(CC(=O)NC1(CNC(c2conc2C2CCC2)=O)CCOC1)n1ccnc1 N1(C(c2c(C)scn2)=O)CC(NC(=O)CC2C=CS(=O)(=O)C2)C(C)(C)C1 N1(C(C=CCOC)=O)CC(N(C(=O)CN(C)S(N)(=O)=O)C)C(F)C1 C(=O)(CS(=O)(=O)CCO)N(C1CCN(C(C(F)SC)=O)CC1)CCO N1(C(C(C2(C)CC2)NC(CCOCCCOC)=O)=O)CCC(F)CC1 N1(CC(=O)NCC(CC(C)C)NC(c2ccc(C)s2)=O)C(=O)C(=O)N(C)C1=O N1(C(c2nnc(C)s2)=O)CCC(NC(c2cncn2C)=O)C(C)C1 N1(CC)CCc2nc[nH]c2C1c1ccncc1CC(=O)OC(C)(C)C c1(NC(N2CCC(F)(C(=O)Nc3ccc(N(C)C)nc3)C2)=O)cc(F)cnc1Cl N1(C(COCCOC)=O)CCCC(CNC(=O)CCn2cnnn2)CC1 C1(CNC(C(=Cc2ccco2)C)=O)CC(O)CN1C(=O)C(=O)NCC(F)F c1(C(=O)NCCNC(=O)C=CCn2cncn2)cccc2occc12 Cc1nc2nccc(N3CCOC(C)(CNC(=O)C(F)(F)c4cncs4)C3)n2n1 C=CCN=C(NCC1CCCC1(F)F)NCC(C)(C1CC1)OC N1(C(C2C(C)(C)COC2)=O)CCOC2CCN(C(=O)CCCN=[N+]=[N-])CC12 N1(C(c2nc(C)[nH]n2)=O)CCOC(CNC(C2CCC23CCC3)=O)C1 c1(-c2c(C)cccc2)ccc(Cl)c(NC(=O)C(c2cccc(F)c2F)N)c1 c1(OCC)cccc2c1CCCN2C(c1nnn(-c2ccccc2)c1C(C)C)=O N1(C(CNC(C)=O)=O)C(CC(=O)NCC(O)CC(C)C)C2CCCC12 c1(C(=O)NC2CC(n3cccn3)C2)ccc2cc[nH]c2c1F c1(C(N2CC(NC(c3cnc(S)[nH]3)=O)C(C(F)F)C2)=O)c(Cl)ccc2c[nH]nc12 N1(C(C(C=C)C)=O)CCC(C)(C)C1CC(=O)NCC1CC1CC(C)(C)C C1(CCNC(CN(C)CCO)=O)CCN(C(=O)COC2CCCOC2)C1 C(=O)(C1=NNC(=O)C1)NCc1cn(CCNC(c2cc(C)nn2C)=O)nn1 C1(NC(C(CC)F)=O)CCCC12CN(C(=O)C1=C(C)CCCC1)C2 Cc1cc(C)c(C(N2CCCC(C)(NC(C3CCC(C)(F)CC3)=O)C2)=O)c(S)n1 CC(C)C(CC(=O)NC1CC(CCNC(c2cnn(C)c2)=O)C1)c1ccccc1 C1(C2(NC(c3c(SC)ccs3)=O)CC2)CCCCN1C(=O)Cc1cnc[nH]1 C1(C(C)C)CC(O)CN1C(c1nc(N(C)C(C)C)sc1Cl)=O c1(C(N2CC(C(N3CCC(C(=O)OCC)CC3)=O)C2)=O)cccc(C)c1I CC(C)(C)CCC(=O)N1CCCC(CO)(NC(C2CC3CC2C2CC32)=O)C1 c1(C(N(CC(CC)NC(=O)COC2CCOC2)C)=O)cccn1C1CCCC1 c1(C(N2C(C(=O)Nc3cc(O)ccc3Cl)CC(F)(F)C2)=O)nc2ccccc2[nH]1 C(=O)(CCCC(C)c1ccccc1)NC1CCN(C(C2CC(=C)C2)=O)CC1 C12(C(N(CCN(C(C(n3ccc(C)n3)C)=O)C)C)=O)CC3CC(C1)CC(C)(C3)C2 Cc1ccc(NNC(=O)C2CC(=O)N(C(C)(C)C)C2)cc1C Cc1ccc(S(=O)(=O)NCCC(=O)NC(C)CCCCNC(=O)C2=CCC2)cc1 C#Cc1cccc(C(=O)NCC2(C(N3CC=CC3)=O)CC23CCC3)c1 N1(C(CNC(CC)=O)=O)CC(C)CCC1C(=O)N(C1CCCC1C)C C(=O)(CC(C)C(F)(F)F)N1CCCC(CC)C1C(=O)N(C1CCOC(C)(C)C1)C N1(C(CCC#C)=O)CC2CS(=O)(=O)CC2(CNC(c2cnn3c2OCC3)=O)C1 N1(c2cc(NCC3CCCC(=O)N3)nc(C(C)C)n2)CCC2(CCNC2=O)CC1 C=CC1(C(=O)NC(CC)CC(=O)OC)CCN(C(c2cc(F)c[nH]2)=O)C1 C1(C(N2C(C)(C(=O)Nc3c(OC)nc(Cl)cn3)CC2)=O)CCc2ccccc2C1 C12(NC(C3CN(C)C3)=O)CC1CN(C(=O)CSc1nccn1C)C2 CCC(O)CC(=O)N1CCC(C2CCCCN2C(=O)CCc2cncn2C)CC1 c1(OC)ccc(CN2CCCC2)cc1NC(N1CCC(C)(c2nn[nH]n2)CC1)=O c1(C(=O)NC(C(CO)NC(C=C(CCC)CCC)=O)C)cc2ccsc2n1C N1(C(c2[nH]c(=NCC)sc2)=O)CCC2C(CCCN2C(=O)C=Cc2cnc[nH]2)C1 Cn1ccc(CC(=O)NCCC2CCN(C(=O)CCCc3ccsc3)C2)n1 C(=O)(CC(C)C(F)F)NCCOCC(=O)NCC(CC(=O)OC)O CC(C)C(C)C(=O)N1CC2(NC(c3ccc(NCC(N)=O)cc3)=O)CC1C2 N1(C(CSCC(C)C)=O)CCC(=CCN(CC)CC)CC1.C(=O)(CCC)NCC=C n1(CC(N2CC(C(C(=O)NCC(COC)(F)F)OC)C2)=O)cccnc1=O C12(C(N(C)Cc3cc(C)no3)=O)CCC(CC1NC(=O)COc1ccccc1)C2 c1(OC)ncc(C(N2CC(OC)CC2CCNC(c2ccnnc2S)=O)=O)cn1 c1(C(N2CC(C(C)NC(=O)C3=CCCS3)C2)=O)c(F)c(F)c(F)c(F)c1F c1(C(=O)NCCC(=O)OC)ccc2c(C)c(C(=O)Nc3ncccc3Cl)[nH]c2c1 N12CCCCC1C(=O)NC1(CCC1)C2=O.C1(SC)CCCN1C(=O)CNC(C)=O C#Cc1ccc(C(N2CC(NC(c3ccc(OC)s3)=O)CC2C)=O)c(F)c1 Cc1[nH]c(C#N)cc1C(=O)NCC(C1CCCC1)NC(c1ncc(Cl)nc1Cl)=O CC1c2nncn2CCN1C(=O)NCC1CCc2nnc(C(F)F)n2C1 C1(C(=O)NC2C(C)CN(C(C3CC(C(F)(F)F)C3)=O)C2)Cc2ccccc2O1 CN1CCN(C(=O)C(C2CC2)NC(c2cccc(Cl)c2)=O)C(CO)C1 c1(CC)nc(=N)[nH]cc1C(=O)NCC(CNC(=O)C(F)C(F)(F)F)CO Cc1cc(Cl)c(C(N2CCN(C(c3ccsn3)=O)CC(C)C2)=O)cc1[N+](=O)[O-] N1(C(c2c(Cl)cc(C)s2)=O)CCC2CN(C(=O)C(C)Cn3ccnc3)CC12 CC1(C)COCCC1CC(=O)NCCOC1CN(C(=O)C=CCn2cncn2)C1 C1(NC(C2CCC(=O)N2)=O)CC(F)CN(C(=O)CSC2CCS(=O)(=O)C2)C1 C(=O)(CCC(=O)NCC1(NC(c2ccc(C)nc2)=O)CCC1)NCC C(=O)(C(C)(C)C(C)(F)F)NCC1CC(C)(C)N(C(=O)CC23CC(C2)C3)C1 c1(C(=O)NCCN(C(C(CC)n2cccn2)=O)C2CC2)cc(C(F)F)ncn1 c1(OC)ccc(CN(C)CC2CCC2(F)F)cc1 c1(OCC)ccc(C(=O)NCCN(C(=O)CC2CC(C)(C)CO2)C)cn1 C(=O)(C1=NOC(C)C1)NCCC1(O)CN(C(c2c(C)ncnc2)=O)C1 CC(CS(C)(=O)=O)NC(=O)C=CC(C)NC(C1COCCC1C)=O C1(C(N2CCCC(CCC(=O)NCC3C4COCC34)C2)=O)(OC)CCCOC1 C1(C(N2C(CNC(c3ccc(CC)o3)=O)CCC2)=O)(OC)CCS(=O)(=O)C1 c1(C(N2CCC(NC(C3(c4ccccc4)CC3)=O)C2)=O)cc(F)c(O)c(F)c1 c1(C(=O)NCC2(CCNC(CCc3cnc(C)o3)=O)CC2)cc(N)c(O)c(F)c1 N1(CC(=O)OC(C)(C)C)CCOCC1.C12CC(C1)N(C(=O)Cc1cccs1)C2=O CC1CC(CNC(=O)C(C2CCN(C)C2)NC(=O)OC(C)(C)C)CCC1(C)C C1(NC(C=CC)=O)CN(C(C2CCSC2)=O)CC1O C(=O)(CCCCNC(=O)OC(C)(C)C)NCCCNC(CCSCCCC)=O C1(CC)CN(C(C2CN(C(=O)C(C)n3ccnn3)CC2OC)=O)CC1O CC1(C(=O)NCC2(O)CC(CO)C2)CCN(C(=O)CCOCC2CCC2)CC1 N1(Cc2c(OCC)n[nH]c2)CC2(CC2C(=O)OC)C1.N1(C=O)CCN(C=O)CC1 C1(CNC(CCC2(C)N=N2)=O)CC2COCC2N1C(c1cccnc1C1CC1)=O C1(C(=O)NCCCN(C(C2CCSC2)=O)C2CC2)CC1C1CC(F)(F)C1 c1(NCC2CN(C)C(=O)C2)nccc(=NCC2(CO)COCCN2C)[nH]1 C1(N(C(COC)=O)C)CN(C(=O)CC(c2cccs2)NC(C)=O)CC1F C1(C)(CC(=O)N(CCC)CC)CCN(C(=O)CCn2ccc(C)n2)C1 N1(C(C2(CC=C)CCCN2C(=O)CC2CC(C)C2)=O)C2CCC(C2)C1CO Cc1nn(C)c(C)c1CCC(=O)N(C1CC2CC1N(C(=O)Cc1cnc[nH]1)C2)C C(C(O)CC(=O)N=c1ccn(CCO)[nH]1)NC(c1nc(C)oc1C)=O S(=O)(=O)(c1ccc(NC2CCOC(C(C)C)C2)c(Br)c1)N(CCSC)CC c1(C(N2CCC(O)(CCNC(C(CN(C)C)O)=O)C2)=O)cc2cccc(Cl)c2[nH]1 C1(NC(=O)OC(C)(C)C)CN(N2CCCCCCNC(=O)CC2)CC1C(F)(F)F c1(OCC(=O)Oc2ccc(Cl)cc2Cl)cc(Cl)ccc1F CC1CCCCC1CC(=O)NCCCC(C)(C)NC(=O)CCn1ncn(C)c1=O C1(c2cn(C3CN(C(C4(C)CC4(Br)Br)=O)C3)nn2)(N(C)C)CCOC1 c1(C(=O)NCC(CNC(CCOCC#C)=O)OC)ccc2c(c1)COCO2 c1(OC)cc(-c2cncc(C(N3CCN(C)C(C)C3)=O)n2)cc(C)c1 N1(C(C(C)=CC2CC2)=O)CC(C(=O)NC2CCOCC2F)C2(CCC2)C1 C(=O)(C1CCCCc2ccccc21)NC(C)(C)CNC(C1CC2C=CC1CC2)=O C1(NC(c2nnc(CC)s2)=O)COC2(C1)CN(C(c1ccc(C)cc1O)=O)C2 Cc1ncc2c(n1)CC1CCC2N1C(c1ccc(I)s1)=O Cc1cccc2[nH]c(=NCC(C3CCCCC3)NC(c3cnns3)=O)oc12 c1(NC2C(CC(C)C)CCCC2)ncc(Br)cc1S(C)(=O)=O N#CC1CCCC(C(=O)NCC2COCC2NC(c2cc(C(F)F)cs2)=O)C1 Cc1coc(C(=O)NCC2CCCC2C(N2CC(O)(CCO)C2)=O)c1 N1(C(CC2CC(C)C2)=O)CCC(CC(=O)N(CC(C)(C)CO)C)CC1 C12(C(=O)NCCC3(O)CCN(C(CC(C=C)C)=O)C3)CCC(CC1F)C2 N1(C(c2ncn(CC)n2)=O)CCOC(C(N2CC(F)(C#N)C2)=O)CC1 C(=O)(C(C(C)(C)C)NC(C)=O)NCc1scc(C(N2C(COC)CCCC2)=O)c1 c1(N2C(=O)NC(C(C)COC3CCCO3)C2=O)cncc2nnnn12 N1(C(C(CC)=CC)=O)CCC(C(F)CNC(=O)CN2CCCCCC2)CC1 C12(C(=O)NC3CN(C(C(C)OCCOC)=O)C(C)(C)C3)CCC(N=[N+]=[N-])C1C2 N1(C(CC(CC)C2CCC2)=O)CC2CN(C(=O)CNC(N)=O)CC2(C)C1 CC1(C)CCC(NC(=O)C=Cc2cocn2)C(CNC(c2cnn(C3CC3)c2)=O)C1 N1(C(=O)NCCC(C(C)C)N(C)C)CCc2ncccc2C1 C1(C(N2CC(O)(C(C(=O)N(CC(C)C)CC)F)C2)=O)COCCN1C O=C(C1c2ccccc2CN1C(c1ccc(=O)oc1)=O)Nc1cc(Br)[nH]n1 C1(C)(C(=O)NCC(C2CCCCC2)NC(C2CCN(CC)C2)=O)CC2CC2C1 c1(C(=O)NCCCCC2CN(C(CCOCCOC)=O)C2)occc1Br Cc1nc(C(=O)NCCCC2(NC(=O)CCCc3ccncc3)CC2)cc(O)n1 C1(NS(CC(C2CCCC2)OC)(=O)=O)CC2(C1)CC(N)C2 Cc1cccc(COCC(=O)NCCCN(C(=O)CC2CC=CCN2C)C)c1 N#CC1(C(=O)NCC2CCCN2C(C2CC3(CCC3)C2)=O)CC2(CCC2)C1 c1(CN2C(C)(C(=O)Nc3cc(OC)nnc3)CCC2)ncc(Br)cc1C C(=O)(CCS(=O)(=O)N(C)C)N(C1CCC(NC(=O)C(c2ccc(Cl)s2)=O)CC1)C C1(CC(C)NC(CCCC#CC)=O)CC2CCC(C1)N2C(C1(C)CCCC1C)=O C(=O)(CCCC(F)(F)F)NC1C2(CC(NC(C(C(C)O)N(C)C)=O)C2)C1 C(=O)(C(CC1CCCC1)C(C)C)NCC(C1CC1)NC(Cn1c(C)nc(C)n1)=O Cc1cnc(N2CC3C(CNN(C)C)C3C2)nc1NC(=O)C1=CC(C)(C)C1 C(=O)(C1=CC2CCCCCC12)N1C2CN(C(c3c(C)cnnc3O)=O)CC1CC2 c1(C(N2C(CNC(c3nccc(CC)c3)=O)CC(O)C2)=O)cccc2c1COC2 c1(C(N2CC(NC(c3ccc(C)nn3)=O)CC2(C)C)=O)cccc2ccn(C)c12 C1(C)(CNC(CSCC=C)=O)CCCN(C(=O)CCCCCOCC)C1 C1(NC(COCC(C)(C)C)=O)CN(C(c2c[nH]c(Br)c2)=O)C2(CCCC2)C1 c1(C(N(CC(OC)OC)CC2CC2)=O)ccc(=O)n(CCF)n1 N1(C(c2cnn(C)n2)=O)CCCC(O)(CNC(C2CCC(C(N)=O)C2)=O)CC1 C12(CNC(C=C(C)Cl)=O)CCCC1CCN2C(=O)C1=COCCO1 S(=O)(=O)(c1cnc(NC(=O)Nc2nnc(O)nc2O)s1)NC c1(C(C(=O)NCCCOCC2CC2)N(CC(C(C)C)C)C)ccc(C2CC2)cc1 N1(C(CCCC)=O)CCN(C(=O)C=C2CCC2)CC1c1cccc(Cl)c1 C1(CNC(C2(F)CCN(C)CC2)=O)CCCC12CCN(C(=O)C=C1CCC1)CC2 C(C(=O)N1CC(OCCC(=O)N(CC(C)O)C2CCC2)C1)(C1CC1)SC CC1CCC(NC(=O)C(F)C2CC2)CN1C(=O)CCc1ccccc1Cl CCC(C)(C)C(O)C(=O)N1CCCC(C(=O)N(C(C)(C)C)CC2CCOC2C)C1 C(CCN=c1nc(N(CCCN(C)C)C)cc[nH]1)c1c(OC)c(F)ccc1 c1(C(N2CC(O)(C(C)NC(C3CCCOC3)=O)C2)=O)ccc2ncc(Br)n2c1 N1(C(C(CSC)C)=O)CC(C2CN(C(C3(C(C)C)CC3)=O)C2)C1 c1(C(=O)NC2CN(C(=O)Cc3ccnnc3O)C2)cc2c(nn1)CCC2 C#CCC(O)CC(=O)NC1(C)CCN(C(c2cncc(N3CCCC3)n2)=O)CC1 C(=O)(C1=C(C(C)=O)C(c2ncc(Cl)cc2Br)NC(=O)N1CC(=O)O)OCC C=CCCCC(C(=O)NC1CC1)N1CCC(CO)(Cc2ccccc2)CC1 c1(OC)ncc(C(N2CCC(NC(c3cscc3OC)=O)C(CO)C2)=O)cc1Cl c1(NCC)ncc(C(=O)NCC(C)N(C(=O)C(C(C)C)NS(N)(=O)=O)C)cc1Cl N1(C(CNC(CNC(CC(CC)C)=O)=O)=O)CC2(C1)CC(C)(C)C2 Nc1c(F)cc(C(=O)NCC2CN(C(=O)C=CBr)CC2C(F)(F)F)cc1F CCCCC(C(=O)N1CC(N(C)C(c2nc(C)oc2OC)=O)C1)N(C)C N1(C(C(CC#C)O)=O)CCC2CN(C(=O)CCCc3ccccn3)CC12 C1(CNC(C2(CCNC(C(CSC)C)=O)CC2)=O)CCCN(C)C1=O C=CCCC(O)CN(C)C(C1(CNC(c2cc(C(F)F)[nH]n2)=O)CC1)=O C1(CNC(C(CC#C)NC(c2snc(C)c2N)=O)=O)CCCCC1(C)C C1(N(C(c2cccc(CC)c2)=O)C)CN(C(c2c[nH]nc2OC)=O)CCC1O Nc1cc(C(N2CC(F)(F)CC2CCNC(=O)Cc2cc[nH]n2)=O)cc(F)c1 C1(C(=O)NCCC2CC(NC(c3nc(CCC)sc3)=O)C2)C2(CC2)C12CC2 C1(C(=O)NC(C)(CNC(C2CCC(C)CC2)=O)CO)Cc2nccnc2C1 C#CC1CC2(CC2)CN1C(C1CC(NC(=O)CC2CC2CC)CCO1)=O c1(CC)ccc(C(N2CCC(NC(c3cc(CC(C)C)c[nH]3)=O)CC2)=O)cc1 S(=O)(=O)(c1ccc(NC(C)CN2CCCC2=O)c(F)c1)N1CCC(OC)(CO)C1 c1(C(=O)NC(CC)CN(C)C(c2ccccn2)=O)cccc(CC2CC2)c1 N1(C(C2(C)CCOC2)=O)CC(NC(=O)CSc2ccccn2)CC(F)C1 c1(N2C(C(N(CC)CC)=O)CCC2)cc(C)nc(-c2ccccc2Cl)n1 N1(C(C2CC(SC)C2)=O)CCC2C(C(N3CCC(N(C)C)(CO)C3)=O)C2C1 C1(N(C(c2c(C)nsc2)=O)CCF)CCCN(C(=O)CC2CCCC23CC3)C1 N1(C(c2nc(C)sc2C)=O)CCCC12CN(C(=O)CN1CCNC1=N)C2 C(=O)(C1CCCc2sccc21)N(CCNC(=O)C(C)(c1cccs1)N(C)C)CC c1(OC)nccc(C(=O)N(C)CC2CCCN(C(=O)COC3CCC3)C2)n1 N12CC(C3(CC3)C1)C2=O.C1(COCCOC2CN(C(=O)NC)C2)CCC(C)(C)O1 C12(NC(c3ccc(OC)cc3)=O)CCC(CC1)N(C(C1CC=CCO1)=O)C2 N1(C(C(C2(C)CC2)NC(CCNC(=O)OCC)=O)=O)CC2(C1)OC(=O)NC2C CC(C)(C)CC(=O)N1CCCCC1C(N1CCC1C(N)=O)=O CC1(C)CCCC1CNC(C1CCC(CNC(=O)C(=O)C2CCCC2)C1)=O c1(OC)cc(CNC(N2CCC(C)(C)C(SC(C)(C)C)C2)=O)cc([N+](=O)[O-])c1 N1(C(c2ncc(C)nc2)=O)CCCC2(CNC(=O)C(C)(C)C(N)=O)CCCC12 CC(C)C(C#N)C(=O)NC(C(=O)N(C1CC2CC2C1)C)C(C)(C)O Cc1c(C(=O)NC2CN(C(=O)CC3CCS(=O)(=O)C3)CC2C)ccc2cncn12 c1(C(=O)NC2C(NC(C(CC)Sc3ccccc3)=O)CC2O)nnn(CC)c1C c1(C(=O)NC2(CNC(CC(C)(C)C)=O)CC(F)(F)C2)cccc2ccncc12 C(=O)(C1CCOc2ccc(F)cc21)NCC1(NC(CN(C)C)=O)CCOCC1 C1(NC(CC(CC)CN(C)C)=O)CC2CC(C1)N(C(C1CCOCC1)=O)C2 C(=O)(CCCC(F)F)N1CCN(C2CCC(NC(CCC(C)N(C)C)=O)CC2)CC1 C(CCCC(=O)NC(C1CCOC1)CO)NC(COCCCC(C)C)=O CC1C(C(=O)NCC2CC3CCC(C2)C3)CCCN1C(=O)CN(C1CCCC1)C C=C(C)CCCC(=O)NCC1(OC)CCCN(C(=O)C(c2cncc(F)c2)C)C1 c1(CC)c(-c2nc(CCO)nn2CC(F)(F)F)cnn1C(C)(C)C C1(CC(N2CCC(CN(C(c3cnc(C)nc3)=O)C)C2)=O)CCCCC1(F)F c1(C(N(CCC)CCNC(C2CCC(=O)N(C)C2)=O)=O)c(F)cc(C#N)cc1F c1(NC)ccc(OCc2cn(C(C)C(=O)N(C)Cc3ncccc3C)nn2)cc1 C1(NC(CC2C(C)(C)N(C(C3CC4CCCC4C3)=O)CC2)=O)CC2COCC(C1)C2 c1(C(N2CC(NC(C3C(OC)CCCC3)=O)C2)=O)ccc(C)c2c1NCCC2 C(C(C(=O)NC1CCOCC1)NC(C1CC(n2cc(CSC)nn2)C1)=O)OC c1(C(C)NC(=O)C(=O)N(C)C(c2nccn2C)C2CCOCC2)cnnn1C n1(C(CC)C)ncc(NC(=O)OCC(=O)N(CC(C)(C)C)CC)c1C.C(C)(C)C N1(C(c2cc(CSCC)on2)=O)CC2CN(C(=O)C(c3scnc3C)O)CC2C1 c1(OC)c(CN(C(=O)C(C)Cc2cnco2)C)cccc1F N1(C(C=COCC)=O)CCC2CN(C(c3c(CC)nn(C)c3CC)=O)CCC2C1 N1(C(=O)OC(C)(C)C)CCC2(CCC2)C(CNC2CC3C(C2)C3(F)F)C1 c1(C(N(C)CC2(O)CCN(C(C=CCCOC)=O)C2)=O)c(F)ccc(OC)c1F c1(C(N2C(COC)COCC2)C(=O)NCc2cn(C)nc2C)ccc(C)cc1Cl c1(C(=O)NC2CC(C)N(C(c3ccc(CN(C)C)o3)=O)C2)c(N)cc(F)cc1Cl C1(C#N)(C(=O)NCC2N(C(c3cc(OC)n[nH]3)=O)CC2)CCOCC1 C=CCC(C)C(=O)NC1CCC(NC(c2ccnc(OC(F)(F)F)c2)=O)CC1 Cc1[nH]c(=NCc2ccc(F)nc2)sc1C(=O)Nc1sccc1C(N)=O N1(C(C(C)C2CCC2)=O)CC(NC(=O)C(=Cc2c[nH]cn2)F)C(C)(C)C1 N1(C(C(=O)NCc2c(OC)cccc2)CC(F)F)CCCC2(CCC2)C1 C(CCC(=O)NCC(C)(C1CCC1)NC(=O)CC1COCCO1)OCCN(C)C c1(C(=O)NC(C)(CNC(=O)COC2CCOC2)C2CC2)c(F)cccc1Cl c1(OC)nc(Cl)c(C(N2CC(=C(F)CNC(=O)CC(C)C3CCCO3)C2)=O)s1 c1(CC(=O)N(CCCCNC(CSCC(=O)OC)=O)C)ccn(C(C)C)n1 c1(C(=O)NCC(C)N(C)C(C2C(C)C2(F)F)=O)coc(C2CCOCC2)n1 C(=O)(NNc1ncc(F)cc1F)N1CCC(C)(C)c2c1cccc2 S(=O)(=O)(c1ccc(=NCc2cn(C3CC3)nn2)[nH]c1)NC(CC)CSC CC1(C)CC2(CO1)CN(C(=O)C(C1CCN(C(=O)CSC(F)F)C1)F)C2 C1(CCNC(C=CSC)=O)CN(C(=O)C(C)NC(c2cccs2)=O)CCO1 C(=O)(C(O)(C(F)(F)F)c1ccccc1)NC1CC(N(C)C(c2cc(Cl)c[nH]2)=O)C1 C(CCSC)(C(=O)NC1CCCC1NC(=O)C(c1ccccc1)N(C)C)SC c1(N2CC(OC)C3(C2)CC3)nc2c(c(=NCCCC3CCCCC3)[nH]1)CSC2 C(=O)(C(C)(C(C)C)OC)N1CCCC(N(C(c2ccc(OC)cn2)=O)C)C1 C12(C(=O)NCC3(NC(C=CCC)=O)CCCCC3C)CCCC1CC(=O)C2 N1(C(C)=O)CC(N=c2cc(NCC3CC(N(C)C)C3)nc(C(F)(F)F)[nH]2)C1 Cc1nn(C)c2c(NC3CCn4cnnc4C3)nc(N3CCOC(C)(C)C3)nc12 C1(C)(CC)CC(N(CCCCC)C)CN1C(=O)CCN(C)C1CC1.C1(=O)CO1 CCCCC(C)CCC(=O)N1CCCC(CCNC(c2cc(C)c[nH]2)=O)C1 C1(OC)CCN(C(=O)C(C)NC(c2occc2C)=O)CC1(C)C c1(C(=O)NCCC2CCN(C(C(CCC)C)=O)CC2)ccc2ccccc2c1C Cc1nc(NC(C2CCN(C(C3CCC(C)CC3)=O)C2)C)c(Cl)cc1C#N CC1C(NC(c2cnco2)=O)CCCN1C(c1ccc(C(N)=O)cn1)=O c1(NC(C(CNC(C(CC)(F)F)=O)CC2CC2)=O)cc(C)c(F)cc1O C12CC(F)(C1)CS(=O)(=O)NC2=O.C(CC(C)N(C)CC)NC(C)=O c1(C(N2CCC(COC)(NC(=O)Cn3nnc(=O)[nH]3)C2)=O)cc2n(n1)CCCN2 N1(C(C(C)NC(C2CCC2)=O)=O)CCOC(CN(C)C(c2cccc(N)n2)=O)C1 C1(N(C)C(C2CC2CF)=O)CCC(NC(=O)C=Cc2ccc[nH]2)CC1 c1(CCCC(=O)N(C2CCC(NC(c3c(C)nc[nH]3)=O)C2)C)ccc(F)c(F)c1 C(C(F)(F)C(=O)NCC(O)CN(C)C(C1CN(C2CCOCC2)C1)=O)OC O=C1CCCCC(C(N2CC=CC(NC(=O)CCCc3ccc(F)cc3)C2)=O)C1 c1(CC(=O)NCC(C)(O)CNC(C2CCC3CC23)=O)cccc(Cl)c1F C1(C(=O)NCCn2ncc(CNC(C3(F)CCN(C)C3)=O)c2)CCCC12CCC2 c1(N(CC=C)C)ccc(S(=O)(=O)NC(COCC2CC2)COC)cc1Br c1(C(=O)NC2CCCN(C(C(CC)NC(C)=O)=O)CC2)ccc(Cl)c([N+](=O)[O-])c1 c1(CC)cc(F)c(NCc2ccc(C3CC3)o2)cc1F N1(C(c2cc(CC)[nH]n2)=O)CCC(C(C)(C)C)(CNC(=O)COC2CCOC2)C1 C1(C)(C(N2CCCN(C(C)=O)CC2)=O)CC(O)CN1C(C1CS(=O)(=O)C1)=O c1(C(=O)NCCCCNC(C2(CC)CCC2)=O)nn(C)c(Cl)c1Cl C1(=CCNC(=O)CC2COCC2O)CCN(C(C2COC(=O)O2)=O)CC1 N1(CC(N2C3CN(Cc4ccc(C)cc4C)C(C3)C2)=O)C(=O)OC(C)(C)C1=O c1(C(C)=O)cc(C(=O)NCCC2CN(C(=O)CN3CC4CC4C3)CCO2)n(C)c1 C(C(C)(C)CN(C(=O)C(F)(F)c1ccccn1)C)NC(C(C1CCCO1)OC)=O N1(C(C2(CF)CCN(C(c3cc(OC)n(C)n3)=O)C2)=O)CCCC(O)C1C C(=O)(CCCC(C)(C)C)N1CCC(C(=O)NCCN(C(C)C)C(C)C)(CC)C1 C(=O)(CCC(C)CCCC)N1CC(NC(c2c(C=C)cnn2C)=O)CC1(C)C CN1CCCC1(C)C(=O)NC1COCC1CNC(=O)CSCc1ncc[nH]1 n1(CC(C2CC2)OC)c(N(C)CS(C)(=O)=O)nnc1C(c1ccc(Cl)cc1)O C1(C(N2CC(C(C=O)O)C2)=O)CC12CCCC2.C12CN(C1)NC2=O.C(=O)C1CC1 N1(C(Cn2c(C)nc(C)n2)=O)CCC(C=CC(=O)NCCC2=CCCCC2)CC1 c1(C(C(=O)NCCC2(C)CC2)N(CCOC)CCF)ccc(SC)s1 CCCCC(CNC(CCc1ccccc1F)C(=O)NCCCSCC)CC c1(OC)ccc(CC(N2CCN(CC(C)NC(=O)C(C)C#N)CC2)=O)c(F)c1 C(=O)(C(C(C)CC)N(C(=O)CC1CCC(O)C1)C)NCc1nc(CC)oc1 N1(C(CSCCC(C)C)=O)CCCC1(C)CNC(=O)COCP(C)(C)=O c1(N(C2CN(C(C3CC3(Cl)Cl)=O)C2)C)nc(Cl)nc2c1ncn2C CC1(C)C(NC(=O)CCOc2cccc(C#N)c2)CCN1C(=O)COCCCF c1(C(=O)NC2CC(O)(CNC(CCCC)=O)C2)ccc(-n2cccc2)cc1O C1(C(=O)NCC(C)(CNC(c2csnn2)=O)OC)CCCN2CCCC12 c1(CCC(=O)NC(c2csc(Br)c2)C)nnc(C2CCCC2)o1 C1(NC(c2c(C)nccn2)=O)CC(O)CN(C(C2C3CCC2CC3)=O)C1 C12(CNC(c3cc(OC)ncc3)=O)CCCC1CN(C(=O)Cc1ccn(C)n1)C2 C1(n2cnnn2)(CC(=O)NCC(CNC(c2c(CC)ncs2)=O)O)CCSCC1 C1(CNC(C2CC(SC)C2)=O)CN(C(=O)CN2CCC(C)(O)C2)CCN1C C=CCC(C(=O)N1CCC(N(C(=O)C(COC)CC)CCC)CC1)C(C)C CC1CN(C(=O)C(c2ccnn2C)O)CC1N=c1cc(Cl)nc(C2CCC2)[nH]1 C(C(C)(C)CC(=O)N=c1ccn(C)[nH]1)NC(C1(C)CN(C)C(=O)C1)=O c1(N(C(=O)C(C)NC(=O)C(C)(C)C)CC2N(CC)CC2)[nH]cnc1C#N Cc1ccc2nc(CNC(=NCCCC#N)NC3CCOCC3)cn2c1 c1(C(C(=O)N2CC(NC(=O)CSc3cscn3)C2)OC)ccccc1Br C=CC1(CC(N2CCCC2CN(C(c2scnc2Cl)=O)C2CC2)=O)CCC1 C1(C(N2C(CNC(c3c(C)cc(C)s3)=O)CCC2)=O)CC(S(C)(=O)=O)C1 c1(CN2C(C(N(CC=C)CC=C)=O)CC(F)C2)c(O)ccc(F)c1F c1(C(=O)NCC(CNC(C2(C)ON=C(C)C2)=O)F)cc(Cl)c2cc(Cl)ccc2n1 CCC(C)C(O)CC(=O)NCC1CCCCC1C(N1CC(CC(N)=O)C1)=O n1(C(C(=O)OC)C)nnnc1C(c1cnn[nH]1)NCCCOCCOC C(C)(C)(C(C)c1ccccc1)OC(CN(CC(F)(F)F)CC)=O c1(C(=O)NCC(CC=C)NC(C2CC(F)C(=O)N2)=O)cc(Cl)c(OC)c(Cl)n1 C1(C(N(C(CCNC(Cc2c(C)n(C)nc2)=O)C)C)=O)CCCNS1(=O)=O S(=O)(=O)(c1ccc(C(=O)NCC(C)(CO)NC(C2(c3cc[nH]n3)CC2)=O)o1)NC Cc1cn(C)nc1C(=O)NC1CCOCC1C(=O)N(C)CC1(N(C)C)CCOCC1 C(CC(=O)N1CCC(NC(=O)C(C(C)C)N(C)C)C(C)(C)C1)(C(F)(F)F)OC N1(C(CC(COC)(C)C)=O)CCC2(CCCN(C(C3(F)CCOC3)=O)C2)CC1 CC1CC(=O)NC(C(N2CCC(C)C2C(=O)NC2CCC(N(C)C)C2)=O)C1 c1(CN(C(=O)C(N2CCCC(CCN)C2)=O)C)c(F)cccc1Br N1(C(CC=C=C)=O)CC2CC(NC(C3CCN(Cc4ccccc4)C3)=O)CC1C2 C12(C(=O)Nn3nc(Cl)ccc3=O)CCOC(COC(C3(C)CC3)=O)(C1)C2 C1(NC(C2CCS(=O)(=O)N2)=O)CCN(C(c2cc(C3(O)COC3)on2)=O)CC1O C(=O)(C(C)CC(=O)NCCC(C)N(C(=O)C1=COCC1)C)OC c1(C(=O)NCC(CCNC(C2ON=C(CC)C2)=O)OC)cn(C)ccc1=O N1(C(C(C)(C)c2cccs2)=O)CCCC2(CC(NC(=O)Cc3cnns3)CO2)C1 c1(OC)ccc(C(=O)NC(C)C(C)NC(=O)CC23COC(C)(C2)C3)cc1Cl c1(OC)cc2c(cc1F)CN(N1CCC13CCOC(C)(C)C3)CC2 N1(C(CC2CC(OCC)C2)=O)CCCC1C1(C(=O)NCC(C)(C)n2cccn2)CC1 C1(C(=O)Nc2cc(C)nc(Cl)c2)CCC2(CN(C(c3ccc(Br)cc3I)=O)C2)O1 c1(C(=O)NC2(C(=O)NCCC#C)CCCC2C)cnn(C)c1C#N c1(C(N2CC(NC(CC3(CSC)CC3)=O)C2)=O)ccnc(OCC(F)F)c1 N1(C(CC)=O)CCC(C(F)C(=O)N(C)C)C1 CCCC(C)(O)CC(=O)N1CC(OC)C(NC(c2csnc2C2CC2)=O)C1 C1(NC(C2(COC)COC2)=O)CC2CC(NC(=O)CC3CCOC3)C1C2 c1(C(=O)NC(CCCNC(CCOCC#C)=O)C)ccc(-c2cscn2)cc1 N1(C(C2CCC(N(C)C)C2)=O)CC2CC1C2CNC(c1ccc(C(N)=O)o1)=O C#CCCC(C(=O)N(CCC#C)CCC)NC(=O)C(C)SCC=C Cc1cc(C(=O)N(C2CCN(C(=O)C(C)NC(=O)C3CC3)C2)C)cc(C)c1N C1(CC(=O)N(CCC)CCN(C)C)CCCC(NC(C2CC(F)C(=O)N2)=O)C1 C1(C(=O)NC2CN(C(C(CC=C)CC)=O)CC2C)CCC2(CCCC2)CC1 C(N=c1nc2scnc2c(NCCN2CCc3ccccc3C2)[nH]1)C1CC(=C)C1 N#CCS(=O)(=O)c1ccc(C(=O)NCCCNC(c2cnc(S)[nH]2)=O)cc1 c1(C(N2CCCC(C(C)NC(=O)C(F)=CC3CC3)C2)=O)cc(N)cc(O)c1 c1(C(=O)NCC(CO)NC(C2CCC2(F)F)=O)cccc(CN2CCOCC2)c1 C1(OCC)CC(C(=O)NCCn2cc(-c3cc(F)ccc3N)nn2)C12CCC2 C(=O)(C1=Cc2ccc(Cl)cc2OC1)NC(CN(C(C(C=C)(C)CCOC)=O)C)C CCC(CC(=O)N1CC(OC)CC1CNC(=O)CCc1ccc(OC)nc1)SC C=CC(C)(C)CC(=O)NC1(COC)CCN(C(c2cc(F)cs2)=O)C1 c1(C(=O)NC2CCCC(NC(=O)C=Cc3nccs3)CC2)ccc2cc[nH]c2n1 CC1CN(C(c2cncc(C(F)F)c2)=O)CC1CCNC(c1cc(CO)[nH]n1)=O C1(C)(C(=O)NCC(CC)NC(=O)C=Cc2cc[nH]c2)CCCCCC1 c1(C(CNC(C2(N)C(C)CC2)=O)(F)F)ccc(C(=O)O)cc1 C1(NC(C=CCCC)=O)CCC2CCN(C(c3ccoc3Cl)=O)C12 c1(C(N2C(CNC(c3csnn3)=O)CC2)=O)cnn(CC2CC2)c1 O=S(=O)(c1ccc(NC2C=CCC2)cc1Cl)N1CC2(C1)CC2(F)Br c1(C(=O)NC2C=CC(CNC(C3(CC#C)CCOC3)=O)C2)cc(Cl)c(N)cc1F CC(C)CC(F)C(=O)N(CCCNC(=O)CCC(C)c1ccccc1)C1CC1 CC1(C)CCC(O)(C(=O)NCC2CCCCC2NC(c2cccc(O)n2)=O)CC1 N1(N2C(=O)NCCC2)CCN(C(C2CC(C(F)(F)F)C2)=O)C(=O)C1 CCC(C)C(O)C(=O)NCC(C)(C(C)C)NC(C1(O)CCCCCC1)=O c1(C(=O)NCC2(CNC(C(CCC)C)=O)CCCCC2)cncc2c[nH]nc12 C1(=CC(=O)NCC(c2c(F)cccc2F)NC(CC)=O)CCCCC1(C)C c1(CC)nc(C(N2CCCN(C(C3CC3(F)F)=O)C(C)C2)=O)c2ccccn12 c1(OC)nc(C(=O)NC2(CNC(=O)CC3CC(SC)C3)CCCCC2)sc1C C(C)(CNC(=O)CCc1cnc(C)s1)(CC)NC(C1C(OC)C1)=O C1(CNC(CC(CC)C)=O)CN(C(=O)COCCCF)CCN1C c1(C(N2C(CCNC(CS(CC)=O)=O)CCC2)=O)cnc(O)c2cncn12 N1(C(=O)CCc2cncnc2)CC2CCC(C1)C2NC(C1(C2CC2)CC1)=O S(=O)(=O)(c1cc(Br)ccc1Cl)N1CC2CN(C(c3cnn4ccccc34)=O)CC21 c1(C(=O)NCC2N(C(C(C=C)O)=O)CC(O)C2)cccc(F)c1OC(F)(F)F C1(NC(C2ON=C(CC)C2)=O)CN(C(c2c(Br)n[nH]c2C)=O)CCC1O c1(COC(C)C(=O)NCCN(c2nnnn2-c2ccccc2)C)ccncc1 N1(C(C(C#N)=CC(C)C)=O)CCCC(NC(=O)CC2NC(=O)NC2=O)CC1 Cc1cc(O)ccc1C(=O)NCC1(C)CCN(CCNS(C)(=O)=O)CC1 C(=O)(CCC(=O)c1ccc[nH]1)N(C1CCCN(C(=O)CCc2cnn(C)n2)C1)C C(=O)(C#CC1CC(F)(F)C1)NCC=CCNC(c1c(C)ncc(Br)c1)=O N1(C(C2(CNC(C(C(C)C)F)=O)CCCO2)=O)CC23CCC2(COC3)C1 C(=O)(C(CCF)NC(=O)Cn1cncn1)NCCN(CC)CC CON(C)CCCNC(=O)C(c1ccoc1)NC(C1CC=CCC1)=O c1(-c2nnc(C)o2)ccc(C(=O)NCC2CC2NC(C2CC2C)=O)cc1 N1(C(c2c[nH]c(=N)o2)=O)CC(CNC(=O)C=CC(F)(F)F)OC2(CCC2)C1 c1(OC)ccc(Cl)c(C(=O)NC2CCN(C(=O)C(N3CCCCCC3)C)C2)c1 N1(C(c2c(C)ccs2)=O)CCCC(CNC(c2coc(C(N)=O)c2)=O)C1 c1(-c2ccc(C)nc2)ccc(N2CCCC2c2nc(N(C)C)no2)nc1C C(C(=O)NC(C)CCCCNC(c1cc(C(C)C)no1)=O)(C(C)C)OC c1(CC(N2CC(NC(C(C)SCC)=O)C3(C2)CCC3)=O)cccc2c1SCCC2 c1(C(N2C(CC)CCC2)=O)cc(NC(=O)OC)cc(C(=O)OC)c1 N1(C(C(CCC)C)=O)C2CCC1CC(C(=O)NCc1c(Cl)cccc1Cl)C2 N1(C(c2c(CC)noc2C)=O)CC2CC(NC(c3cn(CCO)nc3C)=O)C2C1 C12(NC(C(C)OCC(C)C)=O)CC(C1)N(C(=O)C=Cc1cscn1)C2 CC1CN(C(c2cccn2C)=O)CC(C)N1C(=O)C1=C(Cl)CCCC1 c1(C(=O)NCC(C)(C)NC(C2CC(C)=C(C)CC2)=O)cc(C)c(C)c(F)c1 C(=O)(C(CNC(c1nccnc1OC)=O)C(C)(C)C)NC1CC(=C)C1 Cc1cc(F)c(S(=O)(=O)N2CCN(C3CC3)c3cc(F)ccc32)c(F)c1 Cc1cc(N)n2ncc(C(=O)NC3CCCC3CNC(=O)CN=S(C)(C)=O)c2n1 CC(C#N)C(=O)N1CCC(CCNC(=O)C(=O)Nc2ncc[nH]2)C1 CC(C)CC(CNC(=O)C(C)C#N)NC(=O)CCN(CCC(C)(C)C)C N1(C(c2ccc(C)nc2C)=O)CCC(N=[N+]=[N-])(C(=O)NCC(C)CN(C)C)C1 N1(C(C(CCC#C)O)=O)CCCN(C(c2nn(C(F)F)cc2Cl)=O)CC1C c1(C(=O)NCC2CC(COC)CN2C(=O)CC2CCOCC2)cccc(C)c1O C1(NC(=O)C(=Cc2c[nH]cn2)F)COCCN(C(=O)CC2CC(O)C23CCC3)C1 N(C1CCc2ccc(Br)cc21)C(C1(C)CCN1C(c1cc(F)cc(Br)c1Cl)=O)=O C1(C(=O)NC(c2n(C)ncc2)C(=O)N2CC(c3ncc[nH]3)C2)C2CC3C(C2=O)C13 c1(C(=O)NC2CC(F)(C(=O)OC)C2)ccc(C2CCNCC2)nc1 c1(COC(C)C(=O)N(C)CC2(O)CCN(C(=O)CC(F)F)C2)ccc(F)cc1 Cc1nc(Cl)[nH]c(=NC(C)CNC(c2ccc3c(c2)CN(C)C3)=O)c1Cl C(=O)(C(C)C(C)NC(=O)Cn1cc(C)cn1)NCCC(C)(C)OC C1(C(N2CC3C(CNC(c4cc(CC)no4)=O)C3C2)=O)CN(CP(C)(C)=O)C1 CCC(O)C(C)C(=O)NCC(C(C)(C)C)NC(C1C(C)C1C)=O O=C(C1=NNC(C(F)(F)F)C1)NC1CN(C(c2ncccn2)=O)CCC1F C1(NC(c2cn(CC)nc2)=O)CC2CC1N(C(c1nnn(C)c1N)=O)C2 C12CCN(CC1)C(=O)CCC1CC(C1)N2C(c1[nH]cc(CC)n1)=O.C1(CO)CC1 C(c1ccc(F)cc1F)=CN1CCN(C(CSc2ccc(C)cc2)=O)C2C1C2 N1(C(C(C)O)=O)CCCC(O)(CNC(=O)C(O)c2ccco2)C1 c1(NCC2N(CCNC(=O)OC(C)(C)C)CCOC2)cnn2cccc(Cl)c12 c1(OC(C(N2CC(CNC(c3cc(C)sn3)=O)OCC2)=O)C)ccc(F)c(F)c1 C1(C(=O)NC2CCC(CCNC(c3ccn(C(C)C)n3)=O)C2)CC2C(C1)C2(F)F Cc1oc(C#N)cc1C(=O)NCC1CC1NC(C1(c2cccnc2)CC1)=O C1(C(N(C2CCC3(CC2)CC3)C)=O)CC1C1CN(C(=O)Cn2cc(Cl)cn2)C1 n1(COCC)nc(C)c(CC(=O)NC(C)CNC(C23CCC(CC2O)C3)=O)c1C CCC1=C(C(=O)NCC2(F)CN(C(c3ncnc(C)c3C)=O)C2)SCCO1 C1(NC(C2CSc3cn2nn3)=O)CCC(C#N)CC1.N1(CC)CC2C(CO)C2C1 CC1(C(=O)OCCC2CC2(Cl)Cl)CCC(=O)NC1 C1(CC=C)(NC(=O)Cc2cc(F)cc(Cl)c2)CCN(C(C2CCCCO2)=O)CC1 C(=O)(C(C(C)C)NC(c1ccc(CNC(=O)C(C)(C)C)cc1)=O)NC(COC)C C12(C(N3CCC(C(N(C(C)C(N)=O)C)=O)CC3)=O)CCC(C1)OC2C C(c1ccc(OC)cc1C)=CC(=O)NCC1CCN(C(C(CCOC)C)=O)C1 c1(NC(=O)NC(c2ccc(OC)cc2)CO)nc2cc(Cl)ccc2o1 N1(C(c2c(CC)nns2)=O)CC(C(=O)NC(c2ccoc2)C)C(C)(C)C1 C#CC(C)(C)C(=O)NCCCOCCCNC(=O)CC1CCCN1C c1(C(=O)NC2C=CCN(C(Cn3c(C)nnn3)=O)C2)ccc2ccccc2c1F c1(C(N2CCC(O)(CN(C(c3nc(C)c(C)s3)=O)C)C2)=O)ccc(Cl)nc1O CC(C)CC(C(=O)N(CCC(=O)NC1CCC(C2CC2)C1)CCCO)C1CC1 c1(C(=O)NC(C)CNC(c2ccc(F)cc2N)=O)sc([N+](=O)[O-])cc1Cl c1(C(N2CCC(CC=C)(NC(=O)C(C3CC3)OCC)C2)=O)cc(N)cc(F)c1 CC(F)(F)C(F)C(=O)N1CC2CC2(C(=O)NCCCC2CCC2)C1 c1(C(=O)NCC2=CCN(C(c3cc(C)ns3)=O)CC2)nc[nH]c2nccc1-2 C(C)(CCC(C)(C)C)NC(C1(CCNC(C(C=C=C)C)=O)CCC1)=O N1(C(CC2C(C)(C)CC2)=O)CC2(C1)CN(C(c1ncc(Br)cn1)=O)C2 N1(C(C(C2CC2)OC)=O)CCC2CCCC12C(=O)NC1CC2C(C1)C2(F)F C1(N(C(=O)Cc2n[nH]c(=N)s2)CCC)CCN(C(=O)CCNC(=O)CC)CC1 c1(C(N(C2CCN(C(=O)CC3(O)COC(C)(C)C3)C2)C)=O)cccc(=O)n1C c1(NC(CC(C)C(=O)O)(C)C)cncc(S(C)(=O)=O)c1 NS(=O)(=O)c1cnn(CC(=O)NC2CCCCC2NC(=O)C(F)(F)CO)c1 C1(C(=O)NCCC#C)C2CCCC1CN(C(=O)Nc1ccc(C#N)cc1)C2 CC1OCCC1C(=O)N(C)CCN(C(=O)CC1(O)CN(C(=O)OC(C)(C)C)C1)C c1(C(N(CC(CNC(C(N2C(CC)CCC2)=O)=O)O)C)=O)ccc(C(C)C)cn1 C(CC(=O)N(C)Cc1ccccn1)(C(C)(C)C)NC(C1C(CC(C)C)C1)=O C1(C(=O)NCC(C)O)CC(F)CN1C(=O)C(c1cccc(Br)c1)O C1(CC(=O)NC2(c3cn(C)nn3)CC2)C2CCCC2N1C(=O)Cc1ccccn1 C1(NC(c2cccs2)=O)CC2CCC(C1)N2C(=O)CCc1cc(F)ccc1F N1(C(C(C)OCCC=C)=O)C2CCC1C(C(=O)NCC1CCCOC1)C2 C1(C(C(=O)N(C2(C#C)CC2)C)NC(=O)CSCCC#N)CC=CCC1 C1(NC(c2c(C)nc(C(C)C)o2)=O)CN(C(=O)CC(C)CN(C)C)C(C)(C)C1 c1(OC)cccc(CC(=O)NC2CCN(C(C3(F)CCOC3)=O)C2)c1Cl C(=O)(C1=CCc2ccccc21)N1CCC(NC(C2(C3CCCCO3)CC2)=O)CC1 CS(=O)(=O)c1ccc(C(N2CCC(CO)(NC(C3CCCOCC3)=O)CC2)=O)[nH]1 N1(C(c2cncc(C#C)c2)=O)CCC(C(=O)NC(C)CCN(CC)CC)C12CCC2 Cc1c(C)c(=NC(C)C2CCN2C(=O)OC(C)(C)C)[nH][nH]c1=N n1(CC(=O)NCC(C(C)C)NC(C(CC)F)=O)c(C(F)(F)F)nc2ccccc12 C1(NC(c2ccc(C)cn2)=O)CC(NC(=O)CCCSC(C)(C)C)C12CCC2 C(=O)(C(C)C(=O)NC(C1CCCCC1)C(=O)NC1(C)CNC(=O)O1)OC CN1CCC(C)(C(=O)NCC2CCCN2C(=O)Cn2ncc(C#N)c2N)CC1 O=C(C1CC(O)c2ccccc21)NC1CC(O)(CO)C1 c1(CC(=O)NCC(CC)NC(c2coc(C)n2)=O)sccc1C CC1(CO)CCN(C(c2sccc2NC=O)=O)CC1O.c1(C=O)ccc(Br)nc1F C1(CN2C(CC(=O)OCC)COC3(CCC3)C2)CC2(CCOCC2)C(=O)O1 C#Cc1ccc(C2CCCC2NC(=O)C(=O)NCCOc2cccc(C)c2)cc1 C1(CC(=O)N(CC(=O)NCC)C)CC(C)N(C(=O)Cn2cccc2)C1 c1(C(N2C(CNC(C3=CC(C)(C)C3)=O)CC3(CC3)C2)=O)cccc2c1COC2 c1(C(N2CCC(CNC(CCC3N(C)CCC3)=O)CC2)=O)ccc(N)cc1O c1(CCC(N2CC(C(N3CC(N)C3)=O)C3(CC3)C2)=O)cnc2ccccn12.OC CON(C)C(=O)Cn1cc(-c2cccc(C(F)F)c2)nn1 n1(CC(=O)NC(CNC(C(=Cc2cnc[nH]2)C)=O)C2CC2)cc(Br)ccc1=O N1(C(C(C)O)=O)CCOC(CCNC(c2cscc2C(F)(F)F)=O)C1 C(=O)(CCCCC(F)F)N1CC(N(C(=O)CC2CC3(CC3)CO2)C)C(C)(C)C1 N1(C(C=CC(C)NC(C2CCCCN2C)=O)=O)CC2(CCOCC2)C1 C(c1ccccc1)=CC(=O)NC(C(c1ccccc1)OC)C(C)C.C(=O)(C=CCO)N C=CC(C)(C)CCN=C(NC1CCCC1)N1CCC(O)C(CO)C1 C1(CNC(C(c2n(C)ncc2)(F)F)=O)CC2CCC(C1)N2C(=O)CC1CCCC1 c1(C(=O)OC)ccc(C(N2CCCC2Cc2ccccc2F)=O)n1C C#CCC(O)C(=O)N1CC=CC1CNC(=O)Cc1cccc(CC(=O)OCC)c1 CC(=O)CCCC(=O)NC(C(=O)N(C(C)CC(F)(F)F)C)C1CCCC1 c1(OC)cc(C(=O)NC(C)C(C)NC(c2ccc(CO)c(Cl)c2)=O)cc(Cl)n1 C(c1cncc(F)c1)=CC(=O)NCCC(C)N(C(=O)CCC(=O)N(C)C)C C12(NC(=O)CCn3cnccc3=O)CCC(CN(C(c3cnc(Cl)s3)=O)C1)C2 c1(C(=O)NCC(C2CCC2)NC(CC(=O)NCC)=O)cc2c(s1)CCC(C)C2 CC1OC(C)CC1C(N1CC2CC1(CNC(C1(CO)CCC1)=O)C2)=O N1(C(c2cc(COC)oc2C)=O)CC2CCOC2(CNC(c2cc(C)[nH]n2)=O)C1 Cc1ncc(C(N2CCOCC(CNC(c3csnc3Cl)=O)C2)=O)cc1N CCCC(C)(C)CC(=O)NC1CC(CCNC(C2(C)CCNC(=O)C2)=O)C1 c1(-c2ccon2)cn(CCNC=O)nn1.CS(=O)(=O)NCCNCC1(C(N)=O)CC1 C(c1ccc(F)cc1)=CCNC(CCCNC(C(C)NC(C)=O)=O)=O C=C(Cl)C(C)(C)C(=O)NC(C)CN1CCN(C(=O)C(C)(C)N2CCOCC2)CC1 c1(C(C(=O)NC2CCCCC2)N(C(C=C)C2CC2)C)cc(F)cc(I)c1 c12ccc([N+](=O)[O-])cc1C2.c1(OC)cccc(C(CO)NS(C)(=O)=O)c1 CCCCC(C)(F)C(=O)N1CCC2(CC(NC(=O)CSc3ccncc3)C2)C1 C1(NC(C(Cc2c(C)noc2C)C)=O)COCCN(C(C2CC3(C2)CC3F)=O)C1 c1(C(N2C(CCNC(c3ccc(SC)o3)=O)CSCC2)=O)cc(N)nc(Cl)c1 N1(C(c2cncn(C)c2=O)=O)CC2(C1)CN(C(C1C3CCCCC13)=O)CC2CO C12(NC(c3c(CC)occ3)=O)CCCC1CN(C(C1(CF)CCC1)=O)C2 N1(CCC)CCCCC1C(=O)NC(C)C(CO)NC(=O)C(C)(C)N(C)C N1(C(C2(F)CN(C(CC(C)n3cccn3)=O)C2)=O)CCC2(CCC(O)C2)C1 c1(C(=O)NCC(C)(CO)NC(=O)CC2CSC2)cn2ccnc2s1 C1(NC(C2CC3CC2C2CC32)=O)CC2(CCN(c3ccc([N+](=O)[O-])cn3)CC2)C1 c1(CC(=O)N(CCCNC(C(=O)NCCC(C)C)=O)CCO)ccc2c[nH]nc2c1 C1(C(N(CC#N)Cc2ccccc2)=O)CCc2ccccc2C1 C1(CNC(=O)CCCC2CCCO2)CCCN(C(C2CC3CCC2CC3)=O)CC1 C1(SCC)CCC(C(=O)N(C2CCC(NC(=O)C3=COCC3)CC2)C)CC1 N1(C(CCC#CC)=O)Cc2ccccc2C(NC(=O)C(C)CS(C)(=O)=O)C1 C1(NC(c2c(C)oc(C#N)c2)=O)CC12CCC(NC(=O)CC(C)N(C)C)CC2 N1(C(c2c(C)nn(C)c2)=O)CCCC(C)(C)C1CNC(=O)CSC1CCOC1=O C1(C2CC2)(C(N2CCC(C=C)C2)=O)CN(C(=O)C(C)CC2CC2)C1 c1(N2C(C(C)(C)C)CCC2)cncc(C#N)n1.N12CC(CC1=O)C(=O)NCC2 c1(NC(COCC)C2CC2)ncccc1S(=O)(=O)N1CCCC1c1ccc(C)s1 C(=O)(C1OCCc2ccccc21)NC1C(C)CN(C(=O)CCCCCC#N)CC1 c1(-n2c(-c3cc(O)n(C)n3)nc(-c3ccc(C)cc3)n2)cc(Cl)cc(Cl)c1 c1(C(N(CC(=O)NCCC(C(C)C)OC)CCC)=O)cccn2nccc12 N1(C(CN(C)C)=O)C2CCC1C(C(=O)NCCC(O)C1CCC1)C2 C(=O)(C1CCCc2c(OC(F)(F)F)cccc21)NCCCCC(=O)OC(C)(C)C C1(c2n(CCCOC)nnn2)(NCCCS(C)=O)CCC2(CCC(CBr)O2)CC1 C1(CNC(C(C)(C)CF)=O)CC12CCN(C(c1cc3cccnc3o1)=O)CC2 C(=O)(C(F)CC(C)(C)C)NCC(CCOC)NC(C(CC)(C)COC)=O C1(NC(=O)CC2C=CCC2)CCN(C(c2nnc3ccccn23)=O)C12CCC2 c1(C(N2CC(O)(CNC(C34CC(c5ccccc5)C3C4)=O)C2)=O)cccc(F)c1 N1(C(C2C3(CCN(C(c4sc(Cl)nc4Cl)=O)C3)C2)=O)Cc2ccccc2C1 C1(OC)C(OC)CN(C(c2cnc(C)o2)=O)C1CNC(C1CCOC1C(C)C)=O Cc1cc(C(=O)NC2CN(C(=O)OC(C)(C)C)C2)nc(O)c1.C12CC(C1)N2C C1(N(C(N2C(C(CC)OCc3ccccc3)CCC2)=O)C2CC2)C=CC(C)(C)CC1 CC(C)C(C)(CNC(=O)C(C)NC(c1ccoc1)=O)NC(c1ccc(Cl)cn1)=O C(=O)(C1=CC2C=CC1C2)N1C(CNC(c2cccc(CC)c2O)=O)CC2(CC2)C1 CN1CCN(CC(=O)NC2C3CN(C(=O)CC4CC(O)C45CCC5)CC23)CC1=O N1(C(C2N(C(C)=O)C(=O)CC2)=O)CCN(C(c2sc(O)nc2C)=O)C2(CC2)C1 N1(C(c2ccnnc2)=O)CCC2CCC(C1)N2C(C1CCc2ccnn2C1)=O C12(NC(CCOc3ccc(C)cc3)=O)CCC(CC1NC(=O)C1=COCC1)C2 c1(Sc2ccc(OC)cc2)nc(NC(C2(C)CC=C(C)CC2)=O)cc(C)n1 CC1(C)CCN(C(C2Cc3nccn3C2)=O)CC1C(=O)NC1C2CCC(F)(F)C12 c1(C(N2C(CNC(Cn3c(C(C)C)ncc3)=O)CC(O)C2)=O)c[nH]cc(Cl)c1=O c1(C(N(C)CC2CCCN(C(c3cnsn3)=O)C2)=O)ccc(F)cc1NC(N)=O c1(C(=O)NCC2OCCN(C(C(CC)C)=O)C2)ccc(N)c(C)c1F N1(Cc2n(CC)ncn2)CCC(NC(C2CCc3nncn3C2)=O)CC(C)(C)C1 CCC1=NOC(C(N2CCCC2(C)CCC(=O)N(C)Cc2ccnn2CC)=O)C1 N1(C(c2c(C)scc2)=O)CC2CCCC(C(N3CC4CC4C3)=O)C2C1 c1(C(N2CC(CC(=O)NCc3cocn3)OCC2)=O)nc[nH]c1[N+](=O)[O-] C1(N(C(c2c(C)nco2)=O)C)CCC2CN(C(=O)C(F)C(C)(F)F)CC12 N1(C(CSCC(c2ccncc2)C)=O)CCC(NC(c2c[nH]cc2C2CC2)=O)C1 C1(N(C(CC(C)(C)OC)=O)C)CCCN(C(C2CC2Cc2ccccn2)=O)CC1 C(CCN=c1[nH]nc(C(F)F)o1)N(C(=O)C=C1CCCCC1)C C(=O)(C(CC(F)F)c1ccccc1)NCC(CC)NC(c1cccnc1NC)=O CCC(CC(=O)NC1CC2CCC1(C(=O)NCC(C)(O)C(C)C)C2)CC(C)C C1(CNC(=O)CC2C=CCC2)COCCN1C(C1CC=CCO1)=O N1(c2cc(C)ncn2)Cc2ccccc2CC1C(=O)Nc1nc2c(s1)COCC2 Cc1cc([N+](=O)[O-])c(Cl)cc1NC(C1CN(C(=O)CCN(C)C)CCO1)=O C1(C(=O)NCC2CC(CC)C2)C(C)CCN1C(c1ccc(N)cn1)=O C(C(C)C(=O)N1CCCC1CN(C)C(c1cnc(C2CCC2)s1)=O)OC C(=O)(C(C)(O)C(F)(F)F)N1CC(OC)C(NC(c2cc(C)nc(O)c2)=O)C1 C(N=c1cc(C)[nH]c(=NCC2CC(F)(F)CO2)[nH]1)c1cc(OCC)c(C)cc1 c1(C2C(C(N(S(=O)(=O)CC3CC(F)(F)C3)C)=O)C2)cccc(F)c1 Cc1nc(C)c(C(N2CCCC(NC(=O)C(C)ONC(=O)OC(C)(C)C)C2)=O)s1 Cc1ccc(F)c(C(=O)NCC#CC(=O)N2CC(C(C)(C)C#N)C2)c1 N1(C(c2c(C)csc2)=O)CCC(C2CC2)C1C(N1CCC(CO)CC1)=O c1(C(=O)NC2C(CNC(c3cc(C)sn3)=O)CCC2)cc2ccsc2s1 c1(CN(C(CCN(CCCCC)CC)=O)C)nnc(O)o1 c1(N2CCCC(C(C)NC(Cc3cn(CC)nn3)=O)C2)cc2nncn2cn1 N1(C(c2nc(CC)oc2C)=O)CC(CNC(=O)Cc2ccsc2)OC2(CCC2)C1 N1(C(c2cn(CC)nc2)=O)CC(NC(C2(C)C=CCC2)=O)C(O)C1 C(=O)(CC(C)(C)CNC(c1cccc(O)n1)=O)N1C(C)(CC(C)C)CCC1 C12(C(=O)NC(CNC(CN=S(C)(C)=O)=O)CO)CCCN1S(=O)(=O)CC2 C1(NC(CC2CC(CC)C2)=O)CC(C(=O)NCC2(Cl)CC2(F)F)=CC1O c1(C(N2CC3(N(C(c4cccc(C)c4)=O)CC3)C2)=O)ccc2c(c1)OCCO2 N1(C2CCN(C(=O)C=Cc3cc[nH]c3)C2)CCN(C(c2cccnc2)=O)CC1 CCCCCCCCNC(C1(C)CCN(C(=O)C(C)(C)O)C1)=O c1(C(CCO)NC(=O)NCC23CC(CC2CO)C3)ccc(F)cc1F c1(NC2CCCN(C(CC(C)(O)C3CCCCC3)=O)CC2)ncc2ccsc2n1 C(=O)(C(CCCOC)NC(=O)OC(C)(C)C)N1CCN(CC(=O)OC)CC1 C#CC1CC2(CC2)CN1C(C1CC(C)(C)CN1C(=O)Cn1nnnc1C)=O N1(C(C=CCN(C)CC)=O)CCC(O)(CNC(C2CCC23CCCO3)=O)CC1 O=C(C1=CCOCC1)NCC(CO)NC(c1cc(C2CCCCC2)[nH]n1)=O N1(C(C(C(C)SC)O)=O)CCc2[nH]nc(CNC(=O)COCC(C)(C)C)c2C1 C(c1ccc(F)c(F)c1)=C(C)C(=O)NCC1CN(C)CCN1C(c1cnsc1C)=O C(=O)(N=c1[nH]oc2ncccc12)C1C(NC(C(c2ccccc2)OC)=O)CCC1 c1(OC)cc(C(=O)NC2CC(C)(NC(=O)C=Cc3ncc[nH]3)C2)c(F)c(Cl)c1 N1(C(CC(=C=C)C)=O)CCN(C(=O)C(c2ccc(Br)c(C)c2)C)CC1CO C1(OC)CC(NC(c2cn(C)c(=O)n2C)=O)CN(C(C2(C)CCNC(=O)C2)=O)C1 Cc1nc(C2CCCN(c3cccc(C(N)=O)n3)C2)n(-c2cccnc2C)n1 C1(NC(c2ccc(NC)cn2)=O)CCC(C)N(C(=O)CSc2ccc(F)cc2)C1 CC(CC(=O)NCCC1CN(C(C2CCn3ccnc3C2)=O)C1)CC(C)(C)C c1(OC)ccc(OC)c(CC(=O)NCC(C)CNC(=O)CC(C)F)c1 c1(C(N2CC(OCc3cn(CCC)nn3)C2)=O)cc(-c2ccccc2)nc(O)c1 Cc1cc(N)cnc1C(=O)NCc1cccc(C(=O)NC(C)CC2CCCO2)n1 C(N=C(NC1CCC1)N1CCC2(CCOCC2)CC1)C1(C(C)(F)F)CCOCC1 CN1CCCCCC1C(=O)NCC(C)(F)CNC(=O)CC(O)c1ccccc1 c1(OC)nccc(I)c1C(N1CCSC(C(=O)Nc2ccc(Br)c(C)n2)C1)=O O=[N+]([O-])c1cc(Cl)c(NCC2COC(C(F)(F)F)CN2)cc1Cl c1(C(N2C(C(C)C)CN(C(=O)CN3CC(C)(C)C3)CC2)=O)ccc(F)cc1C#N Cc1nsc(C)c1C(=O)OC1CCS(=O)(=O)C1 C(C(CC)(CC)CO)NC(C(C)N(C(=O)CC1CC(C)=NO1)CC)=O c1(C(=O)NCC2CCC(NC(CN(CC)CC)=O)C2)ccc2c(c1)C(=O)CCS2 N1(C(C=CCNC(C2(CCC)CCC2)=O)=O)CCC2(CCCCO2)C1 c1(C(C(=O)NCC)N(CCCCC)C(C)C)ccc([N+](=O)[O-])cc1OC C1(CNC(Cc2c(C)n[nH]c2)=O)CC(C)N(C(c2ccnc(CC(C)C)n2)=O)C1 C1(CC(=O)NCC(C)CNC(=O)CCOCC(C)(C)C)CCCCC12CC2 C(=O)(C(C)(C)CNC(=O)CC1(C)CCN(C(c2ccc(CC)nc2)=O)C1)NCC c1(C(N2CC(NC(C(C)C(C)(F)F)=O)C(C)(C)C2)=O)ccc([N+](=O)[O-])c(C#N)c1 c1(CNC(C(=O)NC2CCCC(OC)C2)=O)cc(Cl)cnc1Cl C1(NC(Cc2c(Cl)cn(C)n2)=O)CCN(C(=O)CCc2ccccc2)CC1F c1(C(N2CC=CC(NC(C(C)C3CCCO3)=O)C2)=O)cccc2c1CCCC2 c1(OC(C)C(=O)NC2CN(C(c3cnns3)=O)CC2F)cccc(CO)c1 CC(CC(C)(C)CO)NC(=O)COC1CC(NC(c2ccc(Cl)cc2)=O)C1 c1(CC)nc(C)n(C)c1C(=O)NCC1CC(NC(c2ccc(OC)cc2O)=O)C1 N1(C(c2c(CNC(CN3CCC(C)C3)=O)c[nH]n2)=O)CCC(C#N)C1 C1(C(=O)NCC2(CCNC(c3cccs3)=O)CC2)CC12CC2 C1(C(C)NC(C2CC(Cl)(Cl)C2)=O)CCN(C(c2cnoc2C2CCC2)=O)CC1 C#CCC(C)(C)C(=O)NC1CN(C(=O)C(c2ccc(OC)c(F)c2)C)CCC1C C1(C(=O)NCCNC(C(c2ccc(C)cc2)(C)C)=O)C(C)(C)C1(F)F.C(C)(C)C C1(C(=O)NCCOCCOCC)CCOCC1NC(=O)C(C)(O)CC c1(N2CCCC2)cccc(Cl)c1.C1(COC)(CNC=O)CCC1 N1(C(c2ccc(O)nc2)=O)CC2OCCN(C(=O)CCOCC(F)(F)F)C2C1 N1(C(CC2C(C)(C)C2(C)C)=O)CC(C(=O)Nc2c[nH]ccc2=O)C2(CC2)C1 C1(CN)CCC2CN(Cc3c(NC(c4ccc(CC)c(C)c4)C)noc3C)CC12 c1(CNC(C(C)OCC)=O)nc2c(s1)CCN(C(C1(F)CC=CC1)=O)C2 c1(CN2CCCC(COC)C2)ccc2cc(F)c(F)cc2n1 CC1CN(C(=O)C(CNC(=O)CC2CCN(C)C2=O)N(C)C)CC(=O)N1C c1(CC)ccnc(C(N2CCC(OCCNC(c3nc(Cl)sc3C)=O)C2)=O)c1 c1(C(N(C2CCCC2)CCC)=O)ccc2c(N(C)C(C)=O)ncnc2c1 CC(F)(F)C(F)C(=O)NCC1(F)CCCN(C(=O)C(=C2CCCCC2)F)C1 CC1CCC(C)C1NC(=O)C(Cc1ccoc1)NC(=O)C(=O)NC1CC1 C1(NC(CC(CC)C)=O)CCCN(C(C2CCN(C(C)C)CC2)=O)CC1 C=C(C)CC(C(=O)NC1CC(C2CC2)C1)NC(=O)CCN1CCCCC1 Cc1[nH]cc(C(N2CC(NC(c3nn(C)cc3Cl)=O)C(N=[N+]=[N-])C2)=O)c(=O)c1Cl N1(C(c2n(CC)ncc2C)=O)CCC=C(C(=O)NC2CCOC23CCCC3)C1 c1(CC)cc(C(N2CC3(CCC3NC(=O)CC(C)C3CCCC3)C2)=O)ccc1C S(=O)(=O)(c1ccc(F)cc1F)NC(c1ccccc1)C(=O)O c1(CNCc2cncc(OCC)n2)cccn(Cc2ccccc2)c1=O C1(CNC(CSc2nc(C)[nH]n2)=O)CN(C(=O)C(c2ccccc2)F)C(C)(C)C1 N=c1cc(C(N2CCC(NC(c3ccc(Cl)o3)=O)C2C2CC2)=O)nc(Cl)[nH]1 C1(CNC(CC(=O)OC)=O)CCN(C(c2cn(C)nc2SCC(C)C)=O)CC1 C1(Cc2cn(C3(C(N(C)OCC)=O)CC3)nn2)CNC(=O)C12CC2 CC(CCN(C)C)C(=O)N1CC2CC2C1C(=O)NCC1=CCCC1 CC1(C)CCN(C(C2CCC(C)CC2)=O)CC1CNC(=O)C(O)C1CC1 C1(C(=O)NC2(CCC)CCC2)CN(C(C2CCCCN2C(=O)C2CC2)=O)CCO1 c1(OC)ccncc1C(=O)NCC1CCN1C(=O)C(CCO)N(C)C C1(NC(C2N(CCC)CCCC2)=O)CCN(C(C2(C#N)CCCCC2)=O)CC1O c1(OC)c(NC2CC(C)N(C(=O)Cc3ccn(C)n3)C2)ncnc1Cl C12(NC(C(CCC)OC)=O)CCC(C1)N(C(c1ccc(O)c(N)n1)=O)C2 Cc1ccc2c(c1Br)CCCN2C(c1ccc(F)cc1F)C(=O)NC1CCCC1 Cn1ccc(=O)c(C(N2CCC=CC2C(=O)NC2(CO)CCC2)=O)c1 CC(C)(C)CC(O)C(=O)NC1CN(C(c2ccnc3ccnn23)=O)CC1(C)C c1(C(=O)NCC23C(CN(C(C(CN(CC)CC)F)=O)C2)C3)cnc(O)cc1C C1(C(=O)NCC2(C=C)CCC2)CC(C#N)C1.C=CCC(=O)OCC c1(COC)ccc(C(=O)N(C2CCN(C(=O)CCC3CC3(Cl)Cl)C2)CCO)cc1 c1(C(=O)NC(CNC(C2OCCN(CC)C2)=O)CC(C)C)ccc(O)c(O)c1 c1(C(=O)NCC2CCN(C(CC(=O)NCC#C)=O)CC2)cc2nc(=O)ccn2[nH]1 CC(c1ccccc1)=CC(N1CCC(N(C)C(C2(C)CC(O)CN2C)=O)CC1)=O c1(NC(C2N(C(c3cn(C)cc3C(F)(F)F)=O)CC=C2)=O)ccc(C#N)cc1Cl C(C1=NOC2CN(C(c3c(C)nn(CC)c3C)=O)CC12)NC(C=CC=CCC)=O N12CCOCC3(C1)CN(CCO3)C(=O)Cn1cc(nn1)C2=O.CC(C)(C)C1CC1 C#Cc1ccc(C(=O)NCCN(C(=O)C(F)OC(F)(F)F)C2CC2)cc1F C1(C2CCN(C(COC(C)(C)C)=O)C2)CCCCN1C(=O)Cc1ccc(Cl)s1 c1(C(=O)NCCCN(C(CSCC=C)=O)C)ncncc1OCC c1(OCCCC(=O)NCC23C(CN(C(C4C(C=C)C4)=O)C2)C3)c(C)cccc1C C1(OC)CC2(C1)CN(C(=O)C(O)CNC(=O)C(C)C(F)(F)F)C2 N1(C(C(C)CN2CCCCC2)=O)CCCC2(CCN(C(=O)Cc3ccoc3)C2)C1 C(=O)(CCCS(C)(=O)=O)NCC1C(C)(C)CN(C(=O)Cn2cc([N+](=O)[O-])cn2)C1 N1(C(C=CCC)=O)CC2(C1)SCCC2NC(C1CC12CCCC2)=O C1(C(=O)NC(CC(C)C)(C)CNC(C2COC(C)C2)=O)CN2CCCN1CC2 C(=O)(C(C)C(C)C(C)(C)C)N1CC2(CN(C(c3c(C)ccn3C)=O)C2)C1 C1(C(=O)NC2(C)CCCN(c3nccn4nnnc34)C2)CCCCC1C1CC1 CC(Cc1ccccn1)C(=O)NCC1CC(F)(CNC(=O)CC2(C(F)F)CC2)C1 c1(CNC(c2ccc(CNC(C(COC)(C)C)=O)o2)=O)cc(C)c(C)nn1 c1(C(=O)NC2C(Cn3cc(C(CC)O)nn3)CCC2)cnc2cc(C)nn2c1 N1(C(C(n2cc(-c3c(C(=O)OC)cc(F)cc3)nn2)C)=O)CCC2(CC1)CSC2 c1(C(=O)NC2CCC(CNC(C34CC(CO3)C4)=O)C2)cc2cccc(Cl)c2s1 C1(NC(CS(=O)(=O)N(C2(S(C)(=O)=O)CCC2)C)=O)C2CCC(C2)N1C(=O)OC(C)(C)C C#Cc1cccc(C(=O)NC(CNC(c2cc(C(C)(C)C)no2)=O)C(C)C)c1F C1(NC(C2C(C)CCCC2)=O)CN(C(c2ccn(C)n2)=O)CC(C)(C)C1 C1(C(=O)NCCC(=C)CNC(=O)CCc2cccnc2Cl)CCCN1N=O c1(N(CC(=O)N(C2CC(NC(=O)CNS(C)(=O)=O)C2)C2CC2(F)F)C)ccccc1 C(C)(C(C(C)C)NC(c1ccc(C(F)F)cn1)=O)NC(COCCCCCC)=O c1(CN2CCC(=CC(=O)NCCC3N(C)CCC3)CC2)cccc2[nH]ncc12 CCC(C)CCCCC(=O)N(CCCNC(=O)C=Cc1cnccc1C)C c1(C(N2CC3(CCN(C(C(CC=C)C(C)C)=O)C3)C2)=O)coc2c(C)cccc12 C(=O)(C(C)(O)C(C)(C)C)Nc1c(SCC)cc(C(=O)O)cc1 Cc1nc(NC2CC(CNC(c3cnn(C)c3C3CC3)=O)C2)c(F)c(C)n1 CCCC(O)CC(=O)NC1CN(C(c2cncc(F)c2)=O)CC1c1cnn(C)c1 Cc1cc(C=CCN2CCCC(O)C2CCO)ccc1OC(F)F NC(=O)C(CCC(=O)O)OC(=O)CCSc1ccc(Cc2cc(F)ccc2F)cc1 Cc1cc2c(Br)ccc(C(=O)NCC(C)CN(C(=O)C(C)CF)C)c2o1 N(C(=NCC1CC1)NCc1ccco1)CC1C(CF)C1 c1(C(=O)NCC2CN(CC(=O)OC(C)(C)C)C2)cc2cc(Br)cc(Br)c2o1 C1(C(=O)NCCC(=C)CNC(c2ccc(CC)s2)=O)CC(=O)NC(CC)C1 CCC(CC(=O)N(CC(C)CO)C)N(C(=O)CC1(C)OCCO1)C CC1C(C(=O)NCCS(N)(=O)=O)CCN1C(C1CC=CC1)=O C1(C(=O)NC2CCC(N(C(C3CCCCO3)=O)CC)CC2)CC(C)CC(C)C1 CCC1=NOC(C(=O)NC(Cc2cccs2)CC(=O)Nc2cc(OC)ccn2)C1 c1(C(=O)NC2C(NC(C3C(CC)OCC3)=O)CCC2)cnn2c1NCCC2 N1(C(C2(NC(C(C)C#N)=O)CC(F)C2)=O)CC(O)C2(CCCC2)C1 N1(C(C2CC(OC)C2)=O)CCCCC1CCCNC(C1CCCN(C(C)=O)C1)=O Cc1cnc(F)cc1C(=O)NCCCCC(C)NC(=O)C(c1cncn1C)O CC1(C)CCOC(C(=O)NCC2CCCCC2NC(c2coc(CO)c2)=O)C1 Cc1cc(C(N2CCC(C)(C)C2CNC(C2CCCCC2)=O)=O)cc(N)c1 CC1C(NC(=O)CN2CC3CC3C2)CCCN1C(c1ccc(CC2CC2)cc1)=O c1(CC(N2CCC(CNC(C(CC)C#N)=O)(OC)C2)=O)ccc2n[nH]cc2c1 C=CCCC(C(=O)NCC12CCC(CC1)C2)NC(=O)Cn1[nH]cnc1=N C1(CNCC2(c3c(Br)cccc3)CCCCC2)CCC2COCCC2C1 S(=O)(=O)(c1ccc(NCC2CCS(=O)(=O)N2C)c(F)c1)NC(C1CCN(C)C1)C C1(F)(CNC(CC(C)C)=O)COCCN(C(C2CCC(C(F)(F)F)CC2)=O)C1 c1(C(N2C(CCNC(c3c(COC)noc3)=O)CCCC2)=O)[nH]c(=N)ccc1C c1(C(N2CCC(OCCNC(CN(C(C)=O)C)=O)C2)=O)csc2cncn12 N1(C(C(F)=CCC)=O)CC(N(C(=O)C(C)C(C)O)C)C(O)C1 N1(c2c(C)cncn2)CCN(C(c2cnc3ccccn23)=O)CC1C#N C1(c2n(CCSC)nnn2)(NC(C)(C)CNS(C)(=O)=O)CCCC1(C)C c1(C(N2CCC(NC(C3CC(C#N)(OC)C3)=O)C2)=O)cn2nc(C)cc2[nH]c1=O c1(CC)cc(Cl)ccc1C(N1CC(NC(c2c[nH]nc2OC)=O)C(C)(C)C1)=O C(CCCCC(=O)N1CCCC(C)(NC(=O)Cc2nnc(O)s2)C1)N(C)C C(=O)(C(F)CC(C)C)N(CCN(C(CN(CCC#C)C)=O)CC)CC C1(c2cccc(F)c2)(NC(=O)C=CC2CCCO2)CCN(C(=O)C=CC2CC2)C1 N1(C(CCOCC)=O)CCCN(C(c2cc(C)n(C)c2C)=O)CC1CO c1(C(=O)NC(C)CCCNC(=O)C#CC2(C)CC2)coc(S(N)(=O)=O)c1 C1(NC(c2c(C)nco2)=O)CN(C(c2cnn3c2OCC3)=O)CCC1CO N1(C(C2C(C)C2)=O)CCC2CCN(C(=O)Cc3ccc(O)nc3)CC2C1 CC(C)C(C(=O)N1CCCC(NC(c2cc(-c3ccccc3)co2)=O)C1)NC=O N1(C(CC(CC)N(C)C(C2CC2CC(C)C)=O)=O)CCC(=O)N(C)CC1 C(=O)(CC(=O)NCC(O)CCNC(C1CCCN1C)=O)NCC#C c1(C(=O)NC(C(C(C)C)NC(c2cnc(OC)nc2)=O)C)ccc(OC)c(Cl)c1 CCC(C)(CCNC(=O)C(=Cc1cnn(C)c1)C)NC(=O)CC1CC(C2CC2)C1 C(=O)(C1=CCCCC1)N1C(CCNC(Cc2cc(C)ns2)=O)CCCC1 N1(C(C2C=CC(NC(CN(C(COC)=O)C)=O)C2)=O)CCCCC1=O n1(CC(=O)N(C)CC2CN(C(=O)C(O)CC(F)(F)F)C2)c(O)nc2ccccc12 c1(C(=O)NCC(C(C)C)NC(C(CC)OC)=O)cccc(-n2cnnn2)c1 Cc1cc(Cl)ncc1CC(N1CC2C(CN(C(=O)C(C)(C)N(C)C)C)C2C1)=O N1(C(c2ccc(CC)cc2C)=O)CC2CC(C)N(C(c3cc(C)ncn3)=O)C2C1 C1(NC(C=CCCC)=O)CCC(C)(CNC(c2cnc(N(C)C)o2)=O)C1 C=CCC(C)C(=O)N(C)CCOCCNC(=O)CC1CC2CCC1O2 Cc1csc(C(=O)NCCc2n[nH]cc2C(=O)NCCC2CCC3CC23)c1C c1(C(N2CCC(C(C)NC(C3C(=C)CC3)=O)CC2)=O)csc2cccnc12 CCC(C(=O)NCCN(CCOC)C(C1CSCN1C(C)=O)=O)n1ccnc1 C(=O)(C1=CNC2=NCCC2=C1)NCC(CNC(c1onc(C)c1C)=O)C C1(C(=O)NCc2cccc(CN(C(C(CC)(C)O)=O)C)c2)CCc2c[nH]nc2C1 C#CCCCC(C)C(=O)NCC12CC(NC(=O)CCC(=O)OCC)(C1)C2 c1(C(C)C)nc2[nH]ccc2c(=NC(C)C2CCN(C(=O)C(C)(C)C(C)(F)F)C2)[nH]1 c1(C(=O)NC2(COC)CCN(C(=O)Cc3cn[nH]c3)C2)cc2ccccc2o1 C1(CCCNC(C(C)(C)C)=O)CCCCN1C(=O)CCCOc1ccccc1Cl O=C1CC(C(=O)NCC2(NC(c3ccc(Br)c(O)n3)=O)CCOCC2)=NN1 C(CCCCCN(C)C(c1cnoc1C1CCOCC1)=O)NC(CC=C)=O C(C)(C)(CC(F)C(=O)N1CC2CCCCC12)NC(C1C(CC)CCC1)=O C(C(C)(CC(C)C)NC(=O)C(C)OCCN(C)C)NC(Cn1nc(C)oc1=O)=O N#Cc1cnc(NC(=O)CC2CCCN2Cc2cc(O)ccc2O)c(I)c1 C12(C(=O)OCC)CCC(=O)C(NCC(c3cccn3C)=O)C1C2 C1(NC(CC2(OC)CN(C(CCC(C)OC)=O)C2)=O)COCCC1(F)F N1(C(C(CC)N(C(CC(C(CC)C)O)=O)C)=O)CC2CCCC(O)C2C1 C1(C)(C(=O)NCC2CN(C(C3(CC#C)CC3)=O)CC2C)C(C)(C)C1(C)C C1(C(=O)NC2C3CCCOC23)(CC)CCN(C(c2nonc2N)=O)CC1 C(=O)(CCS(=O)(=O)C1CCCC1)N1CCCC(NC(CC2C(C)(C)C2)=O)C1 c1(C(N2C(CCc3cn(CCC=C)nn3)CCC2)=O)cncc(-n2cccn2)n1 Cc1nc2cc(C(=O)NC3CN(C(=O)C(=O)NCC(F)F)CCC3CO)[nH]c2s1 C1(CCC(=O)N(C2CCCCC2)C)CCCN(C(C23COCC2C3)=O)C1 Cc1c(C(N2CC(O)CC2CNC(=O)C(C)CC2CC2)=O)ccc2c1CCC2 N1(C(C2C(CC)OCC2)=O)CC(C)CN(C(C2CC2C2CCCCC2)=O)C(C)C1 C1(C)(C(=O)NCC2CN(C(c3c(OC)scc3)=O)C(C)C2)CC2(CCC2)C1 C(C)(C(=O)NCCn1cnc(C(=O)N(C(C)C(=O)OC)C)c1)(C1CC1)OC N1(Cc2cc(C#N)c(F)cc2)CCC2(CCCN(C(=O)CC3COCCO3)C2)C1 C(=O)(C(F)CC(C)(C)NC(=O)Cc1ccns1)NCc1c(C)nn[nH]1 Cc1ccc(NC(C2CCCN2C(=O)Cc2cccc(Cl)c2)=O)c(C)n1 C1(C(N(CC(C)(C)NC(=O)CC2CC(NS(C)(=O)=O)C2)C)=O)CC(F)C(=O)N1 N1(S(CC)(=O)=O)CCC(C(=O)NC2CN(C(=O)C(c3cccc(F)c3)O)C2)CC1 C(=O)(CC(C)C(C)C)N1CC(CC(=O)NCCSCC#C)C(C)C1 C(N=c1nc2sccc2c(NCc2ccccc2)[nH]1)C1C(=O)C2C1CCCCC2 CCCCCCCCCCC(=O)NCC1COCC1NC(c1sccc1SC)=O c1(CNC(C(C)N(C)C)=O)ncc2ccccc2n1.c1(C2CN2)ccccc1F c1(C(=O)OCC)nnc(SC)nc1N1CCC(NC(c2ccon2)=O)C(F)C1 N1(C(c2cnc(C)o2)=O)CCC(C(=O)NC(C)Cc2nc[nH]n2)CC1C C1(CNC(C(CCSC)O)=O)CCCCCN1C(=O)Cn1cccc(C)c1=O C1(C(=O)NCCC2(OC)CN(C(C(COC)(C)C)=O)C2)CC1C1CCCC1 c1(-c2ccc(C(=O)NC(c3cc(C)ccc3C)CC)o2)ccc(CNC)c(F)c1 c1(-c2cn(C)nc2)ccc2cc(C(=O)NCC3CCO3)n(C)c2c1 Cc1nc(N2CCC3(C2)NC(=O)N(C)C3=O)c2c(C)c(C)sc2n1 c1(N2CC(C#N)C3(C2)CCC3)[nH]c(=NCc2nn[nH]c2C2CC2)nc2sccc12 CCN=c1[nH]cc(C(=O)NCCCCC(C)NC(c2cnn(C3CCC3)c2)=O)s1 C(=O)(CCC(=O)NCC1(CCNC(c2[nH]c(C)nc2C)=O)CC1)NC c1(C(N(C2CCN(C(Cc3nccc(OC)n3)=O)C2)C)=O)cncc2nc[nH]c12 CCC(C)C(CC(=O)NC(CO)CCOC)NC(=O)CC1(O)CCCOC1 N1(C(C2CC(C)(F)C2)=O)CCC2(NC(=O)CCCCC(N)=O)CCCC12 Cn1nc(C(F)(F)F)cc1CC(N1CC(O)(CNC(C2CCS(=O)CC2)=O)C1)=O C1(C(=O)NC2CC(CCNC(CC(c3ccccc3F)C)=O)C2)CCN(C)C1=O C1(NC(c2cccc(C(F)F)c2)=O)CN(C(=O)CCC2CC2(F)F)C2CC12 c1(C(C)C)c(C(=O)N(C)CCNC(=O)CC2(O)CCCC2)nc2n1CCCC2 c1(NC(C2CN(C(c3c(NC)cccc3)=O)CC(C)C2)=O)cccn2ncnc12 c1(OC)ncc(Cl)c(C)c1C(=O)NC1CC2CCC(C1)N2 C1(NC(c2nc(C)[nH]n2)=O)CCN(C(c2ccnc(F)c2)=O)C12CCC2 c1(C(=O)NCC23C(CN(C(C(CC)OC)=O)C2)CCC3)cc(F)c(F)c(N)c1Cl C#CC1(C(=O)NC2CCCCC2NC(c2cc[nH]c(=N)c2)=O)CCCC1 c1(CNC(C2CC(CNC(Cc3cc(C)on3)=O)OC2)=O)nn(C)c(=O)n1C c1(C(=O)NCC(CC=C)NC(=O)CCCc2ccc(Br)s2)ncccc1C C1(CC)(NC(c2nc(OC)ccc2F)=O)CCN(C(C2COCC(C)O2)=O)CC1 N1(C(C(C)OCC=C)=O)CC(CC(=O)NCC23CCC(F)(CC2)C3)C2(CC2)C1 N1(C(CC2N(C(c3ccc(C)cc3)=O)CCC2)=O)CC2CC2C1C#N Cc1ncc(Br)cc1C(=O)NCC1(O)CCCN(C(=O)CC2(CO)CC2)C1 C(CC)(CC)(CCNC(C1CC2C=CC1C2)=O)NC(c1n[nH]c(CC)c1Cl)=O C(C(C)(C)CNC(=O)Cn1cnnc1O)N(C)C(C1CN(c2nncs2)C1)=O C1(C(N2C(CN(C)C(c3cc(=O)cc[nH]3)=O)CCC2)=O)Cc2ccc(F)cc2O1 C(=O)(C#CC(C)(C)CNC(C1CC1(C)C(C)C)=O)Nc1c(C)ccc(O)c1C c1(C2C(C)CC2C)nc(-c2ccc(COCC(F)(F)F)cc2)nn1C1CC1 C1(CNC(c2c(C)ccn2C)=O)CN(C(=O)CC2CCS(=O)(=O)C2)C2(CCC2)C1 C12(CNC(C(C)N(C)C)=O)CN(C(c3cc(C(F)(F)F)cs3)=O)CC(F)(C1)C2 N1(C(C2ON=C(C)C2)=O)CC(C2CC2C(=O)NCCn2ncnn2)C1 C=C=CCC(=O)NCC(O)CNC(=O)CCC1CCOC1 N(C1C(=O)Nc2cccc(Cl)c21)C(c1cc(F)ccc1F)=O c1(NC2CC(NC(c3cnc(C)n3C)=O)C2(C)C)nc2ccc(O)cc2s1 N1(C(CCNC(C)=O)=O)CC2CCC(C1)N(C(c1cc([N+](=O)[O-])cs1)=O)C2 N=c1ccc(C(=O)NC(C2CCOC2)CNC(=O)C=Cc2ccsc2Br)c[nH]1 CC1COCCN1CCNC(=O)CC(C1CC1)NC(=O)CC1CSCCO1 C(C)(C(=O)N(CCC(=O)N1CC(CN(C)C)C1)C)(C1CC1)OC N1(CCOC)CCC(NC(CC2CCCC2)C(=O)O)C1 c1(C(=O)NCCC2(NC(COCC)=O)CCC2)cc(F)ccc1-n1ccnc1 Cc1c(C(=O)NCCN(C(=O)CSC(F)F)CCOCCO)ccn1CCO C1(C(=O)NCC(=C)CCNC(=O)CCc2ccccc2)CC2(CO1)CC(F)(F)C2 C12(NC(c3c(C)noc3C)=O)COCCC1CN(C(c1cncc(Cl)c1)=O)C2 c1(C(N2CCC2C(N2CCc3cccnc3C2)=O)=O)ccc(I)c([N+](=O)[O-])c1 C1(C(=O)NCC(CNC(=O)COc2ccc(Cl)cc2)OC)CCCCC(C)(C)C1 N1(C(c2c(CNCc3cncc(NCC)c3)cccc2)=O)CCC(=O)C(C)C1 C1(C(=O)NCCCCC(=O)NC)CN(C(c2cccc(=O)o2)=O)CC1(F)F Cc1nccc(CNC(C2CC2C(=O)Nc2cccc(O)n2)=O)n1 O=C(C#CC1CCCCC1)N1CC2CCCC(C1)N2C(C1CC2(CCC2O)C1)=O C1(CNC(CCCn2c(C)ncc2)=O)C(O)C(O)CN1C(=O)C(C)n1cccn1 C12(NC(CCC)=O)CCCC1CN(C(c1cc(-c3ccccc3Cl)[nH]n1)=O)C2 C1(CC)CC(C(=O)NCC2CN(C(=O)CSc3cn[nH]c3)CCN2C)CC(=O)N1 C(=O)(C1=NN2CCCN=C2N1)NCC(C(C)(C)C)NC(C1N(C)C(=O)NC1)=O N1(C(C2CCCN(c3ncccn3)CC2)=O)CCOCC(F)(F)C1 N1(C(C(c2c(C)nn(C)c2)O)=O)CC2CCCC(C1)N2C(=O)C(F)C(C)(C)O C=CC1CN(C(=O)Cc2csc(CO)n2)CC1.C(=O)(C(F)(F)CC)NCCN(C)C Cn1[nH]c(=NC(=O)Cc2ccc(-c3cnccn3)cn2)cc1Cl S(=O)(=O)(C1CC1c1ccccc1)N(CC(C)C)CC(N)=O CCCC(CCC)C(=O)NCCCCCC(=O)NCc1ccc(F)cc1O C(=O)(C1=CC2CC=CCC12)NC1CC(NC(c2c(O)ccc(C(C)(C)C)c2)=O)C1 c1(C(N2C3CN(C(C(=O)NCC(C)C)C)C(CC3)C2)=O)cccc2c1CCOC2 N1(C(C(COC)O)=O)CCN(C(c2cc(O)nc(Br)c2)=O)C(CO)C1 N(C(=NCCF)NCC1CCOC1)CC1(COC)CCOCC1 Cn1cncc1C=CC(=O)NC1CCCC1CNC(=O)Cc1coc(C(F)F)n1 C1(C(N(C(CCNC(C2N=C(C)SC2)=O)C)C)=O)CC2(CCC2)C1 c1(CCC)cc(C(=O)NC2CC2NC(C2CN(CC(C)C)C2)=O)no1 C1(C(=O)NC2CCN(C(c3cn(C)nc3Br)=O)C2)CCn2c(O)nnc2C1 c1(C(N(c2cnsc2)C)=O)[nH]ccc1CNC(=O)C(C)(F)c1ccon1 N1(C(COCC(=O)NC)=O)CCC(C(=O)NCC2(C)CC2(C)C)C(O)C1 N1(C(=O)CC(F)(F)C(F)F)CCC(C2CCCN(C(c3cc(Cl)c(Cl)s3)=O)C2)C1 CC1CCN(C(=O)COCC2CCCO2)CC1NC(C1(C(N)=O)CC1)=O N1(C(C(C)CC2CCCC2)=O)CC(F)(F)CC1(C)CNC(c1cnn(C)c1)=O CC1(C)CC(CNC(c2cc(C3CC3)on2)c2nnnn2C(C)(C)C)CNC1=O C12(NC(C3N(CCC)CCCC3)=O)CCCC(CN(C(=O)C=CC(F)(F)F)C1)C2 c1(C(=O)NCC(CN(C)C(c2cnoc2-c2cccs2)=O)O)nc(=O)n(C)[nH]1 C1(C(N2CCC(CN(C(=O)CC3CC3(C)C)CC)CC2)=O)(COC)CCOCC1 c1(C(N2CC3CCCC(OC)C3C2)=O)oc2ccc(I)cc2c1C CC1CCc2nc(CNC(=O)CC(C)NC(=O)OC(C)(C)C)sc2C1 Nc1cccc(F)c1C(N1CCC1CNC(c1ccc(F)cc1F)=O)=O c1cc(-n2cc(C3CCOC3)nn2)c2c(c1)COCC2 c1(CC)ccc(C(=O)NC2C=CCN(c3ncc4c(n3)COC4)C2)cc1[N+](=O)[O-] CCC(C)CCC(=O)N1CCCCC1CNC(c1cnn(CCC(C)C)c1C)=O CC1COC(C)(C)CN1C(=O)C(=O)NC1CC(=O)N(CC2CC2)C1 Cc1cc(C(=O)NC(C(=O)NCCc2ncoc2C)c2ccoc2)co1 CCC(CC(=O)N1CCCC1(C)C(=O)NCCCC1CC1)SC C1(C(=O)NCc2c(C(=O)NCc3nnc(CC)o3)nco2)CCC(O)CN1C N1(C(C=C(C)C(C)C)=O)CCCN(C(c2ncncc2Cl)=O)CCC1 Cc1cc(CC(=O)N(C2CCN(C(c3cnn(C)c3C(C)C)=O)C2)C)nn1C C1(Sc2nc(C(C)OCC)on2)CCS(=O)(=O)C1 C1(COC)(NC(c2scc(C)c2Cl)=O)CCN(C(C2(SC)CC2)=O)CC1 c1(C(N(CC(CN(C(c2ccc(C#C)o2)=O)C)O)C)=O)cnc2sccc2c1 c1(C(N2CC(C)(NC(C3CC(CC)C3)=O)C2)=O)cc(Br)ccc1N Cc1ccnc(CNC(=O)C(C)N(C(c2ccncn2)=O)C2CC2)n1 C1(NC(C2(CC)CC(C)(C)C2)=O)CC(C)CN(C(=O)C=CCN(CC)CC)C1 CCC(CC(=O)N1CCOC(CC(=O)NOCCCN(C)C)C1)OC c1(OCC)nc(N2CC(C(=O)Nc3ccc(C)nc3C)C2)ncc1OC CC(C)C(C)(CNC(N1CC(O)C2(CCC2)C1)=O)C(C)C C1(c2cn(CCC(C(=O)N(CC(c3ccccc3)C)C)C)nn2)CCC(=O)CC1 O=C(NNc1c(F)cccc1F)c1ccc2nc(O)oc2c1 c1(C(=O)NCC2CCC(NC(CCCC(=C)C)=O)C2)cc2cc(OC)ccc2[nH]1 C(=O)(CCN(OC)C(=O)CC1CCCO1)NC(CCN(CC)CC)C c1(C(N2CCC(F)(CNC(CC(CCC)O)=O)CC2)=O)nnc2ccccc2n1 c1(-c2ccc(CCCCN(C(=O)OCC)C(C)C)o2)ccccc1Cl N1(CC#CCO[Si](C(C)(C)C)(C)C)CCc2c(OCC(F)(F)F)cccc2C1 C(CNC(C1(Cl)CC1(F)F)=O)(C(=O)N(C)Cc1cccs1)OC CC1=C(C(=O)N2CCC(N(C(=O)C=Cc3cscn3)C)C(C)C2)CCO1 c1(OC)cccn2ncc(C(=O)Nc3ccc4nc(CC5CCCO5)oc4c3)c12 C1(CN(C)C(c2coc(C#N)c2)=O)CCN(C(c2occc2F)=O)CC1 c1(C(=O)NCC2CCC(CNC(C3(C(=O)OCC)CC3)=O)C2)cc(C)ccc1O C1(OC)CC(C(N2CC(N(C(=O)CCSc3ccc(C)cc3)C)C2)=O)CC1OC c1(C(=O)NCC2CCCC2NC(c2cocn2)=O)ccc(F)c(C2CC2)c1 C1(C(=O)NC2(CC#C)CCC2)(CC=C)CCN(C(=O)COCCCN=[N+]=[N-])C1 Nc1ncc(Br)nc1C(=O)NC1(CNC(=O)CC2CC=CCC2)CC1 C1(C(=O)NCCN(C(C2CCC(C)(C)C2)=O)CC)OCCCC1(C)C c1(C(N2CCN(C(CC(C)c3ccccc3)=O)CC2C)=O)ccc2c(n1)NCC2 CCCC(C)(CC)C(=O)N1CC(CNC(C2(C#N)CC2(C)C)=O)C(C)C1 Cc1ccc2cc(C(N3CC4CCC4(CCNC(=O)C(F)(F)CO)C3)=O)oc2c1 C(=O)(C1=CCCOC1)NCC(C(=O)N(C(C(C)C)CO)C)CC1CCCC1 n1(CC)nccc1C(=O)NCC(CNC(=O)CCCC1CCCC1)OC c1(C(=O)NC2C(CNC(CN3CC(CC)C3)=O)C2)ccc2oc(S)nc2c1 C1(NC(C2CCN(C(C)=O)CC2)=O)CN(C(c2csnn2)=O)C(C)(C)C1 c1(C(=O)NCC2C(NC(CSC(C)(C)C)=O)CCC2)cnc2sccn12 C1(NC(C2(CCC)CC2)=O)CCCN(c2cc(Cl)c(O)nn2)C1C c1(OC(C)C)ncccc1C(=O)NC1CN(C(C2CCC(F)(F)C2)=O)CC2CC12 CC1(C)CCCN(C(=O)CCNC(N)=O)C1CNC(c1cncc(Cl)n1)=O c1(CN(CC(=O)N(CC(Cl)Cl)C)Cc2cn(-c3ccsc3C(=O)O)nn2)ccccc1 N1(C(C2(CC)CC2)=O)CCC2(CCC3ON=C(C(=O)NC4COC(=O)C4)C23)CC1 C1(OC)CC2CCC1(NC(C1CC3CC1CC3NC(=O)OC(C)(C)C)=O)C2(C)C C(=O)(C1=CCCN(C(C2CCOC2C=C)=O)C1)NCC(CC=C)(C)C C1(C(C)(C)C)(CNC(c2cc(CCCO)on2)=O)CCN(C(c2cc[nH]n2)=O)C1 C1(CNC(C(CC)O)=O)N(C(c2nccc3[nH]ccc23)=O)CCCC1(C)C C(CC(C)C(=O)NCC1CCN(C(c2c(Br)nnn2C)=O)C1)OC C1(NC(CC2(C(=C)F)CCC2)=O)COC2(C1)CN(C(=O)CCCOC(C)(C)C)C2 c1(N2CCCC(OC(C)C)C2)nc2ccccc2c(=NC(C)C2CCC2)[nH]1.C1CC1 C1(NC(c2cc(CCC)n(C)n2)=O)COC2(CNC(C3CC3C(C)C)=O)CC1C2 C(=O)(CCCC(F)(F)CO)N(CCCCCCNC(c1ccnc(Cl)c1O)=O)C c1(OC)cc(N)ccc1C(=O)NCC1C2CN(C(C34COC(CCO3)C4)=O)CC12 Cc1cc(=NC2CC(C(N)=O)C2)[nH]c(N2CCOC(C)C2)n1.N(C)C CC(C(C)C(=O)NCCc1cn(-c2c(Cl)ccnc2Cl)nn1)S(C)(=O)=O C1(CNC(c2c(CC)ncs2)=O)CN(C(=O)C(C)(CC)OC)CCC1(C)C Cc1nncc(C(N2CCCC2CN(C(=O)C=C(Cl)Cl)C2CC2)=O)c1C N1(C2CCN(C(CC(C)c3ccccc3)=O)C2=O)CCC2(CC=CCO2)CC1 N1(C(C2(OC)CCOC2)=O)CC(CNC(=O)C(C)Oc2ccccn2)C(O)C1 c1(OC)ccc(CC(C)C(=O)N2CC(n3cccn3)(CO)C2)cc1F C(=O)(C1=CCCC1C)NC(CSCC)C(=O)N(CCCN(C)C)C C1(CNC(CCC=C)=O)CN(C(=O)C(C)SCCCC)CCC12CCC2 c1(CNC(C2CCCCO2)CO)cc(OC(F)(F)F)ccc1F CCCCC(C(=O)NCC(CC)CC)NC(C1CCN(CC)C1)=O c1(OC)ncccc1C(=O)N(C)CC1CN(C(=O)CC(C)(C)C)CCO1 C1(C(=O)NCCCNC(C(F)=C(C)C)=O)CC(C)N1C(=O)OC(C)(C)C Cc1cc(C(=O)NC(C2CCCN(C(=O)C=CBr)C2)C)c(C)c(C)c1 c1(SC)nc(N2CCCCC2CNC(=O)CCC(C)N(C)C)cc(O)n1 C(=O)(CC(CNC(C1(C)CCCCO1)=O)C1CCC1)NC(c1ccc(F)cc1)C c1(CC)cccnc1C(N1CCN(CCNC(c2cc(OC)ncn2)=O)CC1)=O C1(N(C(C(C)OCCC=C)=O)C)CN(C(c2cn(C(C)C)nc2C)=O)CC1(C)C Cc1ccc(C(=O)NCCCN(C(=O)C(F)(F)C2CCCC2)C2CC2)c(F)c1C C=C=CCCC(=O)NCc1noc(C(C)(C)C)n1 C1(C(N2C(CN(C)C(C3CC4CCC4C3)=O)CCC2)=O)CCc2nncn2C1 C(=O)(C1=CS(=O)(=O)CCC1)N1C(CNC(c2c(OC)c[nH]n2)=O)COCC1 c1(C(=O)NC(C(=O)NCCNC(N)=O)CC(F)F)cc2cccnc2[nH]1 c1(CNC(C2N(C(c3n(CCC)ccc3)=O)CC=C2)=O)cnc(C)c(C)c1 C(=O)(C1COc2ccc(Cl)cc21)NC1C2(CC(NC(CC=CC)=O)C2)C1 C1(C(=O)OCC)CN(C(=O)C2=NOC(C3(O)COC3)C2)CC12CCN2 c1(COC)c(C(N2CCOCC(CNC(=O)C=CCO)C2)=O)sc2cccc(F)c12 c1(N(C)C)ccncc1CNC(=O)C(N1CCC(NC(c2ccccc2)=O)C1)=O c1(NC(C(c2cccc(OC)c2)C)=O)cc(C(=O)O)c(C)c(C)c1 c1(N2CCC(C)C2)nc(=NC2CC3(CCC3)C2)[nH]c2c1CCC2 C1(NC(C=CC(C)NC(c2n(C(C)C)ccc2)=O)=O)CCCOC12CCC2 c1(C(=O)NCC=C2CCN(C(C(CC)C#N)=O)CC2)cnn2cc(Br)cnc12 C(=O)(C1=CNC2=NCCCN12)N1CCC(CNC(C(C)(O)C2CC2)=O)C1 C1(CNC(C2(CC#C)CCCO2)=O)CCN(C(=O)CCC2CC2(C)C)CC1O c1(-n2cc(CC(C)C)nn2)ccccc1CCC(=O)NC(C)C(C)(F)F c1(C(N2CC(CC(=O)NCc3cc(C)nn3C)OCC2)=O)cc(Cl)c(Cl)cc1C C(=O)(C1COc2ccccc21)NC1C(C)(CN(C(C=CC=CC)=O)C)CCC1 C1(C(=O)NCC(N2CCN(C(C(=O)NCC)=O)CC2)=O)C2C(=O)OCC12Br C(C(C)(C)CC(=O)N1CCC(O)C1C(=O)NCCC1CC1C)OC c1(CC)cn2c(n1)CC(C(N1CCC(C(F)(F)F)C(NC(=O)C(N)=O)C1)=O)CC2 C12(NC(C(CCC)OC)=O)CCC(C(=O)NCCc3ccncn3)(CC1)C2 c1(C(=O)OC)ccc(C)cn1.C12(C)CCN1C(=O)CCC1CCN(C1)C2 N1(C(CC(=C=C)C)=O)CC(F)(F)CC1CCNC(c1c(C)ccn1C)=O c1(SC)cccc(OCC(=O)NCCN(C(=O)C(O)CCSC)C2CC2)c1 CCC(CCC(=O)N1CC(CNC(c2ccnn2CC(C)C)=O)(COC)C1)OC CC(C)CC(C)C(=O)NC(CN=[N+]=[N-])C(=O)NCc1cncc(C#N)c1 c1(NC(C2CC(C)(NC(=O)CC3(C(F)(F)F)CC3)C2)=O)cnc(SCCO)nc1 Cc1cnc(C)c(NC(C2CCCC(NC(c3c(C)n[nH]c3C)=O)C2)=O)n1 n1(C(C)(C)C)cc(C(=O)NCC2C=CC(NC(=O)C(F)=CC3CC3)C2)cn1 N1(C(c2c(C)cncn2)=O)CCC2C(CCCN2C(=O)CNC=O)C1 c1(CC)occ(C)c1C(N1CC(c2cn(C3CC3)nn2)C1)=O.c12ocnc1C(=O)N2 C(CC(C)C)(C(=O)NCCCN(C1(O)CC1)C(c1ccncc1)=O)NC(C)=O N1(CC(N2CCC(NC(Cc3ccc(C)s3)=O)C2)=O)CCCCCCC1=O C(F)(F)(C(F)(F)F)C1(C(=O)NC(CN(C(=O)CC2(C3CC3)CC2)CC)C)CCC1 C1(C(C(C)C)NC(CCn2ncc(C)c2)=O)CCN(C(=O)CCCC2CC2)CC1 c1(C(C(=O)NCCCCCN(C(=O)Cn2ncn(C)c2=O)C)O)ccc(F)cc1 C1(CN(C(CN(CC)CC)=O)CC)CCCN(C(=O)CCC(=O)NC)C1 c1(OCCCC(=O)NC2CC(CC(=O)N(c3ccn(C)n3)C)C2)cccc(Cl)c1 C1(C(=O)N(C(C)COCC)CC)(NC(CCN(CCC)C)=O)CCOCC1 C1(C)(CNC(C(C=C)(C)O)=O)CC(F)(F)CN1C(c1ncccc1OCC)=O S(=O)(=O)(c1cc(C(=O)NC2CC3CC(NC(=O)CSC(F)F)C2C3)co1)NC CC1CN(C(=O)CCc2c(Cl)cncc2Cl)CCCN1C(=O)CC1CC(F)C1 Nc1cccc(CC(N2CC=CC(NC(=O)C=Cc3ccc(Cl)cc3)C2)=O)c1N c1(C(=O)NCC2(O)CC(OC)C2(C)C)cc(Br)cc2nn[nH]c12 Cc1cc(C(=O)NCC(C)NC(=O)CN(C)C(N)=O)nn1-c1cccc(Br)c1 c1(N(CCCOC)C)ncccc1S(=O)(=O)NC(C)C(C)CO N1(C(c2c(COC)nn[nH]2)=O)CCC(C2CC2)C1CNC(=O)CC1(COC)CC1 C1(C(=O)NCC2(C(C)(C)O)CN(C(CCC#C)=O)C2)CC(O)CN1C(C)=O N1(C(CCCOCC)=O)CCCN(C(c2cnn3c2SCC3)=O)CC1 C(=O)(CC(C)CC(=O)N1CC(C(=O)NCCC(=O)N2CCCC2)C(CC)C1)OC CCCCC(F)C(=O)N1CCCC(N(C(=O)Cc2coc(C)n2)CC)C1 C1(C(N(C2(CC(=O)NC3(CCO)CCC3)CC2)C)=O)(NC(N)=O)CCC(C)(C)C1 CS(=O)(=O)CCC(=O)NC1CCC1CNC(c1cnc(C2CC2)nc1)=O C1(C(=O)NOCc2ccc(F)cc2)C=CCCN1C(c1cnn[nH]1)=O c1(-c2n(C)c(N3CCOC(c4ccccc4)(CO)C3)nn2)cn2ccsc2n1 Cc1ccnc(C)c1C(N1CCCN(C(=O)CCn2cncn2)CC1)=O C(=O)(CC(O)CN(C)C)N(CCN(C(c1cnc(C(C)OC)s1)=O)CC)CC c1(C(N(CC(COC)(C)C)C)=O)ccnc(CNC(=O)C(C2CCOCC2)F)c1 C(=O)(C(O)C(C)C)NCCC1CCN(C(C2C(C(=O)OC)C2)=O)C1 Cc1nc(C)c(C(N2CC(NC(c3sccc3CC#N)=O)C(C)C2)=O)[nH]1 Cc1ccc(C(C)CC(=O)N2CC(NC(=O)CCCc3ccc(C)cc3)C2)cc1 C(CN=[N+]=[N-])(C(=O)NCCN1CC=CCC1)NC(C1CCN(CC)C1)=O c1(C(N2CCC(O)(CCNC(C(c3cnn(C)c3)C)=O)C2)=O)cnc(O)c(Cl)c1 c1(NC(C(=O)N(C(CO)CO)C)C(=O)NS(C)(=O)=O)cc(Cl)cc(Cl)c1 c1(CC(=O)NCC2C3CN(C(C(C)C4CCCO4)=O)CC32)ccc([N+](=O)[O-])cc1 C1(NC(c2ccn(CC)n2)=O)CN(C(=O)C(C)(C)Oc2ccc(F)cc2)CC1C C(=O)(C1=Cc2ccc(Cl)cc2OC1)NC1C2CC(NC(CC)=O)CC1CCC2 N1(S(CC(C)C)(=O)=O)CCC2(CCCC2C(N2CCN(C3CCCC3)CC2)=O)C1 C(C(O)CC(=O)NCC1(F)CCC(NC(c2csc(Cl)c2)=O)C1)N(C)C C1(N(CC)CC)CCN(C(=O)NCCC2(C)CCO2)CC1 C1(C2CCCN(C(=O)Cc3sc(C)cc3C)C2)(NC(CCCC(=C)C)=O)CC1 CN1CCCC(C(=O)NCCn2cc(C(=O)N(C3CCN(C)C3)C)nn2)C1 c1(C(=O)NC2CCC(NC(C3CCCC34CC4)=O)C2)ccc(O)c(Cl)n1 n1(C(CC)CC)nc(C(=O)N(C(C)CNC(C2CC(O)C2)=O)C)cc1C C1(NC(Cc2n(C(C)C)cnn2)=O)CC2CC(NC(=O)Cc3cc[nH]n3)CC12 O=C(CC1=CCOCC1)NCC1CCC(NC(c2ccc[nH]2)=O)C1 C1(NC(c2cc(OC)no2)=O)CC(N=c2ccnc(SC)[nH]2)C12CCOCC2 C(CC(C)(C)C)(c1n(CC)nnn1)NCc1c(Cl)cnn1C CCC(CN(C)C)CC(=O)N1CCCCC(NC(c2cnc(O)n2C)=O)C1 n1(CC)cnc2c(NC(CC(c3ccccc3)C)=O)nc(N(C)CCF)nc12 c1(OC)ccc(C(CNC(=O)CC2CC2(C)C)NC(=O)CSC(F)F)cc1 Cc1ccc2c(c1)N(C(C1CCCN(C(=O)C(n3nccc3C)C)CC1)=O)CC2 C(=O)(C1CCCc2ccccc21)NC1CC(CNC(CC2(C#N)CC2)=O)CC1O c1(CCC(=O)NC2CN(C(c3c(C)cc[nH]3)=O)C3C2C3)cccc(Cl)c1Cl N1(C(c2c(N)nccn2)=O)CCC2CN(C(=O)CC3CC(=O)NC(=O)C3)C2C1 c1(C(=O)NC(CNC(C(CC(C)C)OC)=O)CC(F)(F)F)occ2c1CCOC2 C1(NC(c2ccc(Cl)cc2I)=O)CCNC2(CCC2)C1 N=c1[nH]c(-c2c[nH]c(C(=O)NCCC3(O)CN(C(C4CC4F)=O)C3)c2)cs1 Cc1cnc2cc(C(N3CC(N(C(=O)Cc4ccc(CO)cc4)C)C3)=O)ccn12 C1(OC)(CNC(=O)C=Cc2cnn(C)c2)CCN(C(=O)C(C2CC2)NC(C)=O)C1 Cc1ncnc(C(=O)NC2CC(C(C)NC(=O)Cn3ccnn3)C2)c1C C(=O)(C(CNC(c1[nH]nnc1C)=O)C(C)C)NC(CC(=O)OC)(C)C CC1CN(C(C2CCC(C)C2)=O)CC1NC(=O)C(c1ccccn1)O Cc1cccc(-n2cc(C(N3CC(CNC(=O)OC(C)(C)C)CC3C)=O)nn2)c1 C(=O)(C1=CCC(F)(F)CC1)NCCOCCN(C)C(C1CCOCC12CCCC2)=O C(c1ccc(Cl)cc1)=CC(=O)Nc1ccnnc1Nc1cccnc1 c1(OC)cccc2cccc(C(=O)NC3(CNC(=O)CC4COCC4O)CC3)c12 N1(C(C(=O)NC(c2onc(C)n2)C)=O)CCc2cc(Br)ccc2C1 CC1=NN(C)C(=O)C1CC(=O)NC(C)CNC(=O)Cc1cc(O)nnc1O c1(C(N2CC(N(C(C3C(C)OCC3)=O)C)C(C)(C)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C=CC(C)(C)CC(=O)NC1CC(CNC(c2nc(Cl)sc2Cl)=O)C(O)C1 c1(OCC(C)(N)CO)ccc(S(=O)CCC#N)cc1 c1(C(=O)NC(CN(C(c2ccc(OC)s2)=O)C)C)cc2c(F)cc(F)cc2o1 c1(C(=O)NCC2C(NC(CC3N(CC)C(=O)CC3)=O)CC2)nccc2ccsc12 Cn1ccc2cc(C(N3CCC4(COC(CNC(=O)CCCF)C4)C3)=O)cnc12 c1(OC)ccc(C)cc1C(C)NC(=O)C(c1ccc(Br)cc1)C c1(CC)c(C(=O)NC2CN(C(=O)C(C)S(C)(=O)=O)CCC2F)[nH]c(C)c1C(N)=O C(=O)(C(C)CC(C)C(C)=O)NCC1(C(N2CCC(N(CC)CC)C2)=O)CCC1.OCCCC n1(CC)cnnc1C(=O)NCCCCN(C(=O)C(O)Cn1cncn1)C C(c1cncs1)=CC(=O)NC(C1(C(=O)NC(c2nncn2C)C)CC1)C CCCC(C(=O)N(CCC)CCNC(c1coc(C(F)F)c1)=O)C(C)C CC(C)CC(C)(C)C(=O)NC1CCN(C(=O)C(C)(C)Br)CCC1CO c1(OC)ccccc1C(C)(C)C(=O)NC1CC(CNC(=O)C2=CCOC2)C1 C1(CC)CN(N(CCF)C(C)C2CCC2)CC1c1ccccc1 c1(C(=O)NCC(CNC(C2C(C)(C)C2(C)C)=O)OC)cc(Cl)cc(C)c1O N1(C(CC(C)NC(N)=O)=O)CC2(COC(CNC(c3cc4n(c3)CCC4)=O)C2)C1 c1(COC)ccc(C(N2CSCC2C(=O)NOCC2CCCO2)=O)o1 C1(NC(CC(C)N(C)C)=O)C2CCC1CN(C(c1cc3c([nH]1)CCCC3)=O)C2 O=C(CCCc1cnccn1)NCc1nnc(-c2ccccc2)s1 C1(C(N(CCC(=O)NC)C)=O)CCCC1CNC(=O)CCCn1ccnc1 c1(CCC(N2CC(C)C(CNC(=O)C3=CCCC3)C2)=O)ccc2c(c1)COCC2 N1(C(C(CC#C)(C)CC)=O)CCC(C2CC2NC(c2nncn2C2CC2)=O)CC1 C(=O)(C(F)C(=O)NC(CCSC)C(=O)N(C(C)CCO)C)OCC C(CC1=CCCCC1)N(C)C(C1CC(C(=O)NCC2CC(=O)NC(C)C2)C1)=O c1(C(N2CCC(NC(C34CC(CCC)(C3)C4)=O)C(O)C2)=O)cc(O)c(F)cc1N C1(C(N(CCF)CC)=O)(SC)CN(C(=O)C=Cc2cncs2)C1 C=CC1(CN2CCCN(c3nc(-c4c(F)cccc4F)ns3)CC2)CCOCC1 N1(C(CN(CC(C)(C)C)C)=O)CCN(C(c2ncsc2C(F)(F)F)=O)CC(O)C1 N1(C(c2nc(C(C)OC)sc2)=O)CC2C(NC(=O)Cc3cc(C)sc3C)C2C1 c1(C(N2CCC(C)C(NC(C3C(F)(F)C34CCC4)=O)C2)=O)coc(S(N)(=O)=O)c1 c1(C(=O)NC(C2N(C(c3ccc(C(C)=O)s3)=O)CCC2)C)ccc2nncn2c1 N1(C(C2CCNCC2)C)CCN(Cc2ncccn2)CC1 C=CC(CCC)CC(=O)NC1COC2(CNC(c3csc(Cl)c3)=O)CC1C2 Cc1sccc1CC(=O)NCCOCCN(C(=O)CC1CCOC1C)C c1(NC(=O)OC(C)(C)C)nc(CNC2CCCO2)cs1.c12ccc(o1)[nH]c2=O Cc1ccc(F)c(C(=O)N(CC(C)(C)CNC(=O)CC(C)C(C)C)CC)c1 C(=O)(C#CC(C)(C)C)N1CC(n2cc(CNC(c3ccc(CC)[nH]3)=O)nn2)C1 N1(C(c2n(CC)c(O)nc2)=O)CCC2(CCN(C(=O)Cc3ccccc3Cl)C2)C1 N1(C(c2cnc(C(C)C)s2)=O)CCCN(C(=O)CC2(O)CCOC2)C(C(C)C)C1 C=CCN=c1[nH]cc(C(=O)N(C)CCC2CCN(C(c3cscn3)=O)CC2)s1 C1(OC2CC2)CCN(C(=O)CC2CC(OCCNC(C(C)(O)CN(C)C)=O)C2)C1 C1(C(=O)NC(C)(CNC(=O)CCc2ccc(Cl)nc2)C2CC2)CC2(CCCC2)C1 c1(C(=O)NC(CCC)C2CCCC2)sccc1CNC(=O)Cc1ccc(C)s1 c1(C(N(C)CC2N(C(C(C)S(N)(=O)=O)=O)CCC2)=O)n[nH]c2c1COCC2 CC1CCN(C(=O)CCC#N)C1CNC(c1cc(C(F)(F)F)ncn1)=O C(=O)(CC(F)(F)C(C)(F)F)NCCOCCN(C(C=CCN(CC)CC)=O)C C1(C(=O)Nc2nc[nH]n2)CCN(C(=O)Nc2ccc(-n3ccnn3)cc2)CC1O CC(F)(F)CCC(=O)NC1CC1CNC(c1ccc(Cl)cc1)=O N(C(=NCCc1nc2c(s1)COCC2)N1CCC(OCC2CC2)C1)CC(F)F C(C(C)C(=O)NC(CN1CCCC1)C(=O)NC(C)(C)CCOC)OCC Cc1oc(C)c(C(=O)NC2CN(C(=O)CC(C)C3CC3)CC2C)c1C Cn1cnc2c(N3CCCCC3CNC(c3nc[nH]c4nccc3-4)=O)ncnc12 c1(NC(c2ccc(C(=O)O)cc2)=O)cc(C(F)(F)F)ncc1F C1(CC)CCC(C(N2CCOCC2CC(=O)N(CCCO)CCCO)=O)CC1 CCCCCCC(=O)NCC(C)(CC)C(=O)NCc1ccccc1C c1(CC(=O)NCC(CNC(C(CC)(F)F)=O)C)c[nH]c2cccnc12 c1(NC(CCc2n3cc(C)nc3sc2)=O)nc2c(s1)C(C)OC(C)C2 C(N=c1nc2sccc2c(NCC2CC23CCOC3)[nH]1)C1(C(N)=O)CCCCC1 c1(C(N(CC(CC)NC(c2cocc2C)=O)C)=O)n[nH]c2c1CC(C(C)C)CC2 c1(OC)cccc(CN2CCN(C(c3ccncc3O)=O)C(CC#N)C2)c1Br C1(C)(C(N2CC(CNC(CCC=CCC=C)=O)C(C)C2)=O)CCN(C)CC1 c1(C(=O)NC(C(C)NC(c2nn(CC)c(C)c2)=O)C)cnc2c(Br)cccn12 c1(OC)cccc(C(F)(F)C(=O)NC2CC(C)N(C(c3ncncc3F)=O)C2)c1 c1(N(C(C2CCCCC2)=O)CCN2CCNCC2)ccccc1CO C1(CNC(C2(CC=C)CCOCC2)=O)(OC)CCN(C(=O)COCC)CC1 O=C(CC1CCCN1)N1CC(CSc2ccccn2)C(O)C1 C1(C(=O)NCCCN(C(=O)CC2OCCOC2(C)C)C(C)C)CCC(=O)N(C)C1 c1(CC(=O)NCCC(C)(C)NC(c2ncncc2F)=O)ccc([N+](=O)[O-])cc1F C12(NC(c3c[nH]c(=O)cn3)=O)CCC1CN(C(=O)CCC1CC1)C2 C12(NC(C3(COC)CCN(C(COC(CC)CC)=O)C3)=O)CCCN(CC1)C2 c1(C(=O)O)ccc(C(=O)NC2CC2C(N2CCCOCC2)=O)cc1 Cc1ccc(C(N2CC=CC(NC(C3CC(CCO)C3)=O)C2)=O)c(F)c1F c1(C(=O)O)ccc2cc3ccc(-c4cccc5cc[nH]c45)cc3nc2c1 C(=O)(C(O)C(F)(F)F)NCCC1CC(OC)CN1C(c1ccc(C#N)o1)=O c1(CNC(=O)NC(C)C(=O)NC2CC2NC(=O)C2CC2)ccccc1Cl C1(C(N2C(CN(C(Cn3nnc(C)n3)=O)C)COCC2)=O)CCCCC(=O)C1 C1(C)(C(=O)NCC(c2cccc(C)c2)NC(c2cc[nH]n2)=O)CCCCC1(F)F C1(CN(C)CCF)COC(C(F)F)C1 N1(C(C2(C(N)=O)CCC2)=O)CCN(C(=O)CN2CCCCC2)C(CCO)C1 C(=O)(CCC(=O)N1CCCC(CN(C)C(C)C)C1)N(CC)CC c1(CNC(C=C2CCC(C)C2)=O)ccc(CNC(C2(F)CC=CCC2)=O)c(F)c1 N1(C(C(C(CNC(c2cc(C)oc2)=O)C)F)=O)CCC2CN(C)CCC12 C1(CC(=O)NCCCC2CC(C)C2)CCN(C(C2(Cl)CC2(F)F)=O)C1 Cc1cn(C(C)C)cc1C(=O)NCC1(F)CCC(CNC(c2coc(Cl)n2)=O)C1 C1(NC(c2c(CCC)nco2)=O)CC(C2CCN(C(C3CCC(C)O3)=O)CC2)C1 CC(Cc1ccnn1C)C(=O)NCC(O)CCNC(=O)C=C1CCCCC1 c1(C(=O)NCC2C(C)CCN(C(COCC#C)=O)C2)ncnc2ccsc12 C#CCC(C)C(=O)NCC1C(C)CCN1C(C12CC3CC1C2C3)=O c1(C(N2CC(C(C)NC(=O)CC(C)(C)F)OCC2)=O)coc2c(F)cc(Cl)cc12 CC(C)S(=O)(=O)CCc1cccc(-n2c(C(c3n[nH]cc3Br)N)nnn2)c1.OC CC1CN(C(=O)C(=O)NCC(c2ccccc2)N2CCOCC2)CC(=O)N1 N1(C(C2(C)CC(C)C2)=O)CCOCC(NC(=O)Cc2cncc(O)c2)C1 N1(CC(C)C)CCC(C(=O)N(CCCCNC(=O)C(C)c2ccsn2)C)C1 c1(C(CC)OCC)nc(CN2CCCC2)nn1-c1ccc(C2CC2)cc1 CC(C)C(C)C(CNC(C1CN(C2CCCCC2)C1)=O)NC(c1cnsn1)=O c1(CN2C(C)CCCCCC2)c[nH]c2c(Br)c(C)ccc12 N1(C(C(C)SC(C)C)=O)CC(C)C1C(=O)NCC1CCCSC1 N1(C(C(COC)COC)=O)CC2CCN(C(c3c(F)cc(F)cc3Cl)=O)CC12 Cc1[nH]nc2c1CC(C(=O)NC1CCC(CNC(=O)C=CC(C)C)CC1)CC2 c1(CCC(=O)NCC2C(NC(C3(C)C(C)(C)C3)=O)CCC2)cc(Cl)cc(Cl)c1 C1(NC(C2(COC)CCCC2)=O)CCC2CCN(C(C3(Cl)CC3)=O)C1C2 C(=O)(CC(c1ccccc1)NC1CC1F)OC(C)(C)C C1(OCC(=O)NCC2(CNC(C(CC)F)=O)CC2)CCN(C)CC1 c1(C(c2n(CCCSC)nnn2)NCCCS(C)=O)nc(C)n(C)n1 c1(N2CCN(C(=O)NCC3CCCN(C)C3)CC2)nc2ccc(Br)cc2o1 C1(OC)(CNC(c2ocnc2C)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC1 C1(OC)CN(C(=O)CCCC2CCCO2)CC1NC(=O)CC1(OC)CCC1 c1(C(=O)NCC(CC)NC(=O)Cc2nncn2C)cn(C)nc1C O=C1CN(C(=O)CN2CCCC2CC2CC3CCC2C3)CCN1 Cc1ccc(CNCC2(C(=O)Nc3ccccc3N3CCCC3)CC2)c(Br)c1 Cc1c(N)c(C(N2CCC(CF)(NC(c3nccc(Cl)c3F)=O)C2)=O)nn1C c1(C(C)OC(CNc2scc(-c3ccc(CCC)cc3)n2)=O)ccc(C)cc1C C(=O)(C(F)C(C)(C)O)N1CCN(CC2CCN(C(C3(C(C)(F)F)CC3)=O)CC2)CC1 N1(C(c2c(CC)cco2)=O)CCN(C(=O)C(c2cc(C)oc2C)C)CC1CC C1(C(N(CCN(C(C2CN(C(=O)NC)C2)=O)C)C)=O)CC(C)(C(C)(C)C)C1 CN1CCOc2c(C(=O)NCC3(NC(=O)CC(C)(C)O)CCOCC3)cccc21 c1(C(N2CC(CCC=C)(C(=O)N(CCCO)CC)C2)=O)c[n+]([O-])c(C)cn1 CC(CC1CCCCC1)C(=O)N1CCC(CNC(=O)CC2CC(C)(C)C2)C1 c1(OC)ccnc(F)c1C(=O)NC(C)CCCNC(C1CCCC1CF)=O C(CO)(CCCCNC(c1n[nH]c(C2CC2)c1Cl)=O)NC(C1C(C)(C)CCC1)=O n1(CC(C)NCC2(O)CCC2)ccc(C(F)(F)F)n1 CC(C)(C)C(C)(C)C(=O)N1CCC(CNC(=O)C2=COCC2)CC1 C(=O)(C1OC(=O)c2ccccc21)N1C(C)CC2CN(C(c3ccccc3)=O)CC21 c1(C(=O)NCc2c(C)ccs2)ccc(NC(=O)C(C)OCC(F)(F)F)cc1F N1(C(=O)OC)CCCN(Cc2c(Cl)cccc2I)CC1 c1(C(CNC(=O)CCOCC(F)(F)F)NC(CC2(C#N)CC2)=O)ccccc1 c1(C(=O)NC2C(NC(C=Cc3c(C)coc3C)=O)C2)cc2c(C)ccc(F)c2o1 N1(C(CCC(=O)OCC)=O)CCCC(C2CCCN(C(C3CCN(C)C3)=O)C2)C1 C(=O)(C(CC(C)C)NC(=O)COCC(F)(F)C(F)(F)F)OC(CC)(C)C CC1CCC(Cl)=C(C(=O)N(CCNC(C2CCC(F)CC2)=O)C2CC2)C1 n1(CC)ccc(C(N2CCC(C)(NC(=O)C3=CCCC3)C2)=O)cc1=O c1(C(=O)NCC2(F)CC(CC(=O)OC)C2)cc(C)n(C(C)(C)C)n1 c1(C(=O)OCC)noc(Nc2ccc(-n3nccc3C)cc2)c1C CC1(C)CCC(CC(=O)NCCC2CN(C(=O)C(F)(F)CO)CCO2)C1 N1(C(c2c(C)coc2)=O)CCC(N(C)C(C2Cc3ccccc3O2)=O)C2(CC2)C1 C1(CC(=O)NCC(C(C)C)NC(C(CC)Sc2ccccc2)=O)CC2CCC1O2 N1(C(CC)=O)CC2CC(NC(c3ccc(NC(C)=O)[nH]3)=O)CC2C1 C1(C(=O)NC(C2(O)CCCCC2)C(N2C(CCC)CCC2)=O)CC2(C1)CC(O)C2 c1(C(C(=O)NC(c2cn(CCO)nn2)C)O)cc(F)cc(F)c1 c1(C(N2CCC(C(=O)NCC(F)Br)(CC)C2)=O)cc2ncccc2[nH]1 CCC(C(O)C(F)(F)F)NC(=O)NCC1(O)CCC(CC)C1 c1(C(C)=O)ccc(C(=O)N(CCCCN(C(=O)CCCOC(C)C)C)C)nn1 c1(OC)cc2c(cc1OC)C(NC(c1ncccc1C)C)CC2 N1(C(C2CCCCC2)C)CC2COCC2(C(N2CCC3(C2)CC3(F)F)=O)C1 C12(NC(Cc3ncc(C)s3)=O)CCCCCC1N(C(c1cnc[nH]1)=O)CC2 c1(C(N2CC(CC)C(NC(=O)C(C)=C(C)C)C2)=O)c(C(F)F)cccc1SC C1(C(N2CC(C)C(CN=c3cc(Cl)nc[nH]3)C2)=O)CCc2nncn2CC1 C1(CN(c2nnc(C3CC3)o2)C)CCN(C(=O)Cc2ccc(Cl)cc2)CC1 N1(C(c2cc(CO)on2)=O)CCCC2C1CCN2Cc1cc([N+](=O)[O-])ccc1Cl n1(CC)ccc(C(N2CCC(O)(CN(C(=O)COCC(F)F)C)CC2)=O)cc1=O Cc1nc(C)c(C(=O)NCCC(O)CNC(c2c[nH]cc2-c2ccccc2)=O)s1 C1(NC(c2c(OC)nccc2)=O)CC(N=c2[nH]c3c(cc2C#N)COCC3)C1 N1(C(c2c(C)sc(O)n2)=O)CCC2CN(C(C3Cc4nnc(C)n4C3)=O)CC12 c1(C(N2CCCN(C(Cn3c(C)ccn3)=O)CC2C)=O)c[nH]c2c(F)cccc12 c1(C(N2C(C(=O)Nc3c(C)ccnc3Br)CC(F)C2)=O)c(Cl)ccc(Br)c1Cl C1(NC(=O)Nc2c(C(=O)OC(C)(C)C)c(F)ccc2)C2CCC3(COC(=O)C13)O2 N1(C(C=Cc2ccc(SC)s2)=O)CC2(C1)SCCC2NC(c1ccncc1)=O c1(C(=O)NC2CCC(CC(=O)N(C(C)C(=O)OC)CC)C2)ccc2cc[nH]c2n1 C1(NC(CC2CC(=C)C2)=O)CC2CCC1N2C(c1n[nH]c(C(C)(C)C)n1)=O CCCC(C)(C)C(=O)NC(CNC(C1(Br)CC12CCC2)=O)C1CCC1 c1(C(C#C)NC(=O)C=CC=C(Cl)Cl)ccc(OCCOCC)cc1 CC1CN(C(=O)C2=CCC2)CCCN1C(=O)CC(C)(C)Cc1ccc(Cl)cc1 c1(C(=O)NCCC(C)N(C(CCCCCNC(C)=O)=O)C)ccc(S(C)(=O)=O)o1 N1(C(CCCCOCC)=O)CCC(NC(c2cc(C#N)oc2C)=O)C2(CCC2)C1 c1(C(N2CCOC3CCN(C(C4CSC4)=O)CC32)=O)cnc2ccc(F)cc2c1 CCCC(CNC(c1cc(OC)ncn1)=O)C(=O)NCC(CC)n1cccn1 c1(C(=O)NCCC2CN(C(C(c3c(C)cccc3)C)=O)C2)ccc2cc[nH]c2n1 C1(CNC(CC2CC(=C)C2)=O)(OC)CCN(C(=O)C(C)(C)C2CCOC2)CC1 C1(F)(CNC(C(C=C)OC)=O)CCCN(C(=O)C(O)Cc2cnn(C)c2)C1 c1(OC)ccc(CN2CC3CN(C(c4cccc(I)c4C)=O)CC3C2)c(F)c1F C(N=c1nc2scnc2c(NCc2nncn2CC)[nH]1)c1cc(CC)on1 C1(OC)CC(C(=O)NCC2(CNC(C3(C)CC3(C)C)=O)CCC2)N(C(C)=O)C1 O=C(N=c1ncn(Cc2cc(C(F)(F)F)on2)[nH]1)NC(c1cc(F)ccc1F)CO C(CO)(CCCCNC(C1CNC(=O)N1)=O)NC(CC(C)F)=O C1(C(N2CCC(C(C)NC(C3CN(C)C3)=O)C2)=O)CCC(=O)N1C N1(CCC(CC)O)C(=O)NC(Cc2ccccc2)C1=O N1(C(CCn2c(C)ncc2)=O)CC(F)(F)CC1(C)CNC(=O)C(C)NC(N)=O C1(C(C)C)CCOC1C(N1CC(N(C(=O)C(C)CC2CCCCC2)C)C1)=O c1(C(N2CCN(C(=O)C3=CCCCO3)C(C(F)F)C2)=O)cc2ccsc2s1 c1(C(=O)NCC(C)(C2CC2)NC(CC(CC)O)=O)n[nH]c2c1CCCC2 c1(NC(C2N(C(c3n(C)cnc3)=O)CCC2)=O)ccc(CNn2cccn2)nc1 c1(C(=O)NC2(C(=O)OC(C)(C)C)CCCOC2)n[nH]c2cc(F)ccc12 C(N=c1[nH]c(C)ncc1C)C1CCC(NC(C(CCC)OC)=O)CC1 N1(C(c2c(CC)nco2)=O)CCC(O)(CNC(=O)CCc2ccc(O)cc2)CC1 c1(C(N2CCCC2C2CC2)=O)cc2cccc(-c3c(F)cc(CO)cc3F)c2[nH]1 c1(C(=O)NC2C(C(N(C(C#C)(C)C)C3CC3)=O)CCC2)ccc(C)nn1 C1(N(C(c2snc(SC)n2)=O)C(c2ccc(F)cc2)C)CCCCCC1 c1(C(C)(F)F)ccnc(C(=O)NC2C3CN(C(C4CCCN4C=O)=O)CC23)c1 Cc1ccc(-c2nc(C(=O)NCCC3CN(C(C4(CF)CCC4)=O)C3)cs2)cn1 CC1=C(C(=O)N2CC=CC(NC(C3CCOC(C)C3)=O)C2)Cn2ncnc2N1C c1(OC)cccc2c1C(C(=O)NC1CCOC3(CCOC3)C1)CC2=O C(CCCC(=O)NC1CC(F)(CNC(c2ccc(C(C)(F)F)cc2)=O)C1)OC C1(C(=O)NC(CNC(Cc2ccn(C)c2)=O)C2CC2)CCC(F)(F)C1 C1(C#N)(CNC(c2c(C)nc(CNC(=O)C=Cc3ccoc3)o2)=O)CC(C)(C)C1 N1(C(C2CC(C)(C)C2)=O)CC(NC(C2(C)CCC(=O)N2)=O)C(C(F)F)C1 C12(NC(c3nc(C)c(C)s3)=O)CC(C)(C1)OC21CN(C(=O)CCC(C)N(C)C)C1 C1(C(=O)NCC(c2ccsc2)C)CCC(C2CC2)N1C(=O)COCC(F)F C1(O)(CNC(c2ccnc(C3CC3)n2)=O)CCN(C(C2CC3CC3C2)=O)C1 C(=O)(C(CC(N)=O)NC(=O)CCCCN(C)C)NCC(C=C)O CCC(CC(=O)N(CCCNC(c1ccc(OC)s1)=O)C)OC C1(NC(c2c(C)occ2)=O)CCCCN(C(c2cn(C)nc2C(F)(F)F)=O)C1 C1(CNC(C2CC(=C)C2)=O)N(C(=O)C(F)OC)CCCC1(C)C N1(C(Cc2c(C)n[nH]c2)=O)CCCN(C(=O)C(C)(F)F)C(C)C1 C1(CNC(C(CC#C)(C)C)=O)CN(C(C2CCC2(F)F)=O)CC(C)(C)C1 Cc1cncc(CN2CC(NC(c3sccc3Br)=O)C(F)C2)c1 c1(C(=O)OC)c(NC(=O)C2=NOCC2)oc2ccccc12 CCCCC(CNC(=O)C(F)(F)c1nccs1)NC(=O)CCCCF C1(C2CCC2)(C(=O)NCC(CC=C)NC(c2ccccc2SC(C)C(N)=O)=O)CC1 O=C(CN1C(=O)Cc2cc(Cl)ccc21)NCC1(NC(c2ccncc2Cl)=O)CC1 CCCC(C)C(C)N=c1nc2c(cnn2C(C)C)c(N(C)CC)[nH]1 C(=O)(C(C)(C)C(=O)NC(C)CNC(c1cccc(-c2ccc(F)cc2)n1)=O)OC C12(NC(c3ccnc(C)c3C)=O)CCCCCC1N(C(=O)COC(F)(F)F)CC2 C1(N=[N+]=[N-])(C(=O)NC(C)CC(C)(C)O)CCN(C(=O)CCn2cccc2)C1 C(=O)(C1CCCc2nncn21)N1CCC(CCNC(C(C)SC(F)(F)F)=O)CC1 c1(C(N2CC(OC)C(NC(C3CCC4(CCC4)C3)=O)C2)=O)cc2cn[nH]c2cn1 Cc1c[nH]nc1C(=O)NC(C)C=CC(=O)NCC(c1ccnn1C)O c1(C(=O)NCC2(O)CCN(C(c3c(CC)csc3)=O)C2)ccc2c(c1)NCCC2 Cc1cc(CNC(C2CN(C(=O)CCSC(F)(F)F)CC2C)=O)cc(O)c1 n1(CC)c(C)nc([N+](=O)[O-])c1NC(C)C(=O)NC C(=O)(C1=NOC2(CCC2)C1)N1C(c2cn(Cc3cncc(C)c3)nn2)C(C)CC1 C1(C(=O)NC2CC(OCC(=O)NCc3cn(CC)nc3)C2)CCN(C)C1C N(C(=NCCCCl)NCCNC1OCCC1C)Cc1cnc(CCC)o1 N1(C(C2C(=C)C2)=O)CCCC(C(=O)NCCC2COCCO2)CC1 N1(C(CCC=C)=O)CCOC2(CCN(C(=O)C(C)(F)C(=O)OC(C)(C)C)C2)C1 N1(C(COC)=O)CC2(CCN2C(=O)CCCC2CCCCC2)C1 c1(C(=O)OC)cncn1CC(=O)N(CCCNC(=O)CC1CCC(C)C1)CCO C(=O)(NN1CCCC1C(=O)NCC12CCN(CC1)CC2)C1C(C)C1C C1(CN(c2ccc(C(=O)OC)cc2)CCC)(NCCC#N)COC(C)(C)OC1 c1(N2CCC(C)(CNC(c3ccnc(CO)c3)=O)C2)snc(Cl)c1C#N C(=O)(CCCCC(C)CC)NC1CCC(C(N(OCC)CC)=O)C1 C1(N(S(=O)(=O)CC2CCC2C(=O)O)CCC)CC(OCC)C12CCCC2 N1(Cc2cn(C(C)(C)CCNC(=O)Cn3cnnn3)nn2)CC(=O)CCC1=O c12ccc(cn1)[nH]c2=O.C1(CCOC)CCCC1.C1(NC=O)CC(CN(C)C)C1 C12(CNC(c3c(COC)cc[nH]3)=O)CC1CN(C(=O)Cc1c(Cl)cnn1C)C2 CC(N=c1nc2scnc2c(N2CCCC2)[nH]1)c1nc(=N)[nH][nH]1 N1(C(C=CC(C)(C)NC(=O)C=CC2CCC2)=O)CCC2CCC(C2)C1 C(=O)(CCC(C)OC(C)(C)C)NC(CC)CNC(C1CC1C(F)(F)F)=O Cc1oc(C#N)cc1C(=O)NC1CCN(C(C2(C3CCCO3)CCC2)=O)C1C c1(N(CCC(=O)NC(C2(C)CC2)(C)C)SC(F)(F)F)ccccc1 N(C1COc2cc(F)ccc21)c1nccc(=NC(C)c2n(CC)ccn2)[nH]1 N1(C(CCN(CC#C)C(C2CCCC(CC)CC2)=O)=O)CCCC(C)(C)CC1 N1(C(CCN(C(c2c(OCC)nn(C)c2)=O)C)=O)CCC(O)(CO)CC1 c1(Nc2cccc(OCC(N3CCCC(O)C3)C)c2)c(Br)cc(Br)cc1Br C1(NC(C(c2ccccc2F)C)=O)CN(C(=O)CSc2ccccn2)CCC1C C(=O)(C(F)(F)C(F)F)NC1(C)CC(NC(CC(C)NC(C2CCCCC2)=O)=O)C1 n1(CCC)nccc1C(N1CCC1(C)CC(=O)N(C1CC1(C)C)C)=O C(c1cnc(C)nc1O)=CC(=O)NC(CC(C)NC(c1ccc(C)nc1)=O)C CN1CC(C)(C)CC1C(=O)NCC12CC(CO1)N(C(C1CC(C3CC3)=NO1)=O)C2 N1(C(COCCC)=O)CC2CC2(NC(c2ccccc2C2CCCC2)=O)C1 N1(CC(N2CC(CC(N3CC(C(=O)OC)C3)=O)C2)=O)CCCCC1=O C12(C(=O)NC(C)CNC(c3cccnc3N(C)C)=O)CCCC1OCC2 N1(C(c2c(C)n(C)nc2)=O)CCCC(C)(C)C1C(=O)NC1CC(C)CC(C)(C)C1 O=Cc1cncc(C(=O)NCc2nc(-c3ccccc3)n[nH]2)c1 C1(NC(Cc2cc(C(C)(C)C)on2)=O)CC(C(=O)Nc2ccsc2)C1(C)C c1(C(=O)NCC2C(C)CCN2C(c2cnc(C#N)s2)=O)ccn(CCO)c(=O)c1 C1(C(N2CC(CNC(=O)COc3ccc(C(N)=O)cc3)C2)=O)(CC)CCNC1=O N1(C(C(C)CCN(C)C)=O)CCC(C2(NC(=O)CC(C)SC(F)(F)F)CC2)C1 c1(C(=O)NCCN(CCOC)C(c2cc(F)n(C)n2)=O)ccc2nc(C)oc2c1 c1(C(=O)NC2CC(CNC(C3ON=C(C)C3)=O)C2)[nH]cc2c1CCC2 c1(C(=O)NC2CC(C(C)NC(C(CC)O)=O)C2)cc(O)ccc1Cl C(C)(CNC(c1cnc(S)n1C)=O)(CC(C)C)NC(CCN(C(CCC)C)C)=O C(=O)(C1=C(C#N)CCC1)N(CCCNC(c1cc(C(F)F)cs1)=O)C(C)C c1(C(N(C)CCN(C)C(C2(F)CC=CCC2)=O)=O)ccnc2c(F)cccc12 C#CC1(O)CC(C(=O)NC2CC2CN(C(C2(O)CC2)=O)CC)C1 C1(OCC)CC2(C1)CC2C(=O)NCCC1(CNC(c2nocc2C2CC2)=O)CC1 C12(C(N(CCCC(N3CCC(O)(CO)C3)=O)C(C)C)=O)CCC(CC1)C2(C)C N1(C(c2n(C=C)ncc2)=O)CC2CCCC(N=c3ccnc(C(C)C)[nH]3)C2C1 c1(C(C(N2CC(CN(C)C(C3C4COCC34)=O)C2)=O)=O)cnn(C)c1 C(=O)(C1=CCN(C(=O)Cc2ccc[nH]2)CC1)N1CC(C)C(N(C)C)C1 N1(C(C(C)(C)CCCO)=O)CCCC(C2CCCN(C(=O)CCC[N+](=O)[O-])C2)C1 C1(NCc2nnc(C)o2)CC(NC(c2cc(Br)c[nH]2)=O)C12CCC2 C=CCC(C)(C)CC(=O)NCC(C)C(F)C(=O)NCc1nnc(C2CC2)o1 C(=O)(CCCC(C)(F)F)NC1CN(C(c2cnn(CCCC)c2C)=O)CC1C C(=O)(C1=C(C)CCOC1)NCC1(C)CCCN(C(COC(C)=O)=O)C1 C1(NC(=O)CC2(C(F)F)CC2)CCCN(C(c2nnc(O)cc2O)=O)CC1 C1(C(=O)Nc2cc(OC)cc(O)c2)CCN(C(=O)C(C)=C(C)C)CC1(C)C C1(NC(CNS(C)(=O)=O)=O)CCC(NC(=O)CCCC2CCC2)C1 c1(CC(=O)NC2CC(F)(CNC(C=C(CC)C)=O)C2)coc2c(C)c(Cl)ccc12 C1(c2ncco2)(C(=O)NC(CNC(C2CC23CC3)=O)C2CCC2)CCC1 C(=O)(C1=CCCOCC1)NCC(C)N(C)C(C12CC(C1)C2)=O c1(-c2n(CC)c(N3CCCC3SC3CCCCC3)nn2)cn2ccc(C)cc2n1 N1(C(CCC(C)(C)C)=O)CC(C2CCCN(C(C3OCC4CCCC34)=O)C2)C1 C(=O)(C1=CCCC1C)NCc1c(C(=O)NCC(CC)C(C)C)c[nH]n1 C1(C(=O)NCC2CC(F)CN2C(=O)C=Cc2ccoc2)CC12CCOCC2 CC1(C)CN(S(=O)(=O)c2ccc([N+](=O)[O-])cc2F)Cc2cc(Cl)ccc21 C(c1cncc(C)c1)=CC(=O)N(CC(C)NC(C(CC#C)O)=O)CC CC1=C(C(=O)NC(C2CCN(c3nc(C(C)(C)C)nc(=N)[nH]3)C2)C)CCS1(=O)=O C1(C)(C(N(C)CC2C(C)C2)=O)CC(O)CN1C(=O)COCC(F)F CC1(CNC(c2ccc(NC(N)=O)nc2)=O)CCC(NC(=O)Cc2ccon2)C1 S(=O)(=O)(c1ccc(C#N)cc1)N1CCC(C(=O)OCc2cc(CCC)no2)CC1 N1(C(CCOCCC)=O)CCC(CNC(c2ccc(C)c(O)n2)=O)C(C)C1 C=C(C)CC(C(=O)NCCCCc1cn(CCCOC2CCC2)nn1)OC C1(CC(=O)NC(c2cn(C)nn2)C(=O)NC(C)C(=O)NC2CC2)CCN(C)CC1 O=C1C2C3CC4C2C2(C(N5CCC(NC(=O)C(F)(F)C(F)(F)F)C5)=O)C1C3C42 C1(NC(c2nccc(C)n2)=O)CCN(C(c2ccncc2Cl)=O)C12CCC2 CC(CCC(=O)NC1CCN(C(=O)C#CC2CC2)C1C)c1ccccc1 N1(C(c2ccc(OC)cc2)=O)CC2CN(Cc3cc(C)nc(O)c3)C2C1 C1(CNC(C(CC)OC)=O)C(OC)C(OC)CN1C(=O)CC12CC(C1)C2 c1(OC(CC)C)cc(C)ccc1CNC(C1CCCCC(=O)C1)=O C12(C(=O)NC(C(C)C)(C)CNC(=O)C=CC3CCCO3)CCC(F)(CC1)CC2 N1(C(CC(C=C)CC)=O)CCC(C=C)(C(N2CCC(CC)CC2)=O)CC1 C1(NC(CCOCCOCC)=O)CCSC12CN(C(c1ccsc1SC)=O)C2 c1(C(N2CC3C(C(N4CCC(F)C4)=O)C3C2)=O)cc(Br)cc2cn[nH]c12 C1(C(CCCC)c2ccccc2)=CCC(N=[N+]=[N-])C1.NCC N1(C(C2(C)CCN(C(C(CC)OCC)=O)C2)=O)CCCC(C)C1CO C(=O)(CC(F)(F)C(F)(F)F)N1CCCC(NC(c2cc(C(C)C)n(C)n2)=O)CC1 c1(C(N(CCCN(C(c2c(COC)ccs2)=O)C)C)=O)cccc(F)c1SC C1(C(=O)NCC2N(C(CCOCCOC)=O)CC2)Cc2ccccc2O1 N1(C(CCOC(C)=O)=O)CCC(C2CCCCN2C(C2CCN(C)C2=O)=O)CC1 CCC(CC)CC(=O)NC1CCCCN(C(c2cnccc2F)=O)C1 c1(C(=O)Nc2c(C3C(CSCC)C3)occ2)c(C)nn(-c2ccccc2)c1Cl C1(O)(C(=O)NCCc2ccncc2)CCN(Cc2ccc(-c3ccc(Br)s3)s2)C1 Cc1nn(C)c(C(F)(F)F)c1C(=O)Nc1ccccc1CN1CCOCC1 Cn1ccc(C(=O)NCC(C)(C)CNC(=O)Cc2ccns2)c1C1CCC1 C(=O)(CC(O)CC(C)(C)C)NC(C)C=CC(N1CC2COCC2(CO)C1)=O Cn1cnc2sc(C(=O)NCC(C(C)(C)C)NC(=O)Cn3ccccc3=O)cc12 C(C(=O)NC(C)CNC(c1cc(C2CCOC2)[nH]n1)=O)(C(C)C)NC(COC)=O N1(C(CCOCC#C)=O)CCC(C2CC2)C1C(=O)OC.C12CC(C)(C1)CNC2=O c1(C(=O)NC2CCC(NC(CC3(C)CC3)=O)CC2)ccc(Cl)cc1N c1(NC(C)=O)cc(C(=O)NCC(C)(C(C)C)NC(=O)C(C)C(F)(F)F)ccc1F C(=O)(C1=NOC(C)C1)NC1C(NC(c2ccn(CC)n2)=O)CC1 C1(C(N2CC(CC(=O)NCC(C(=O)NC)C)(OC)C2)=O)CN2CCN1CC2 c1(C(=O)NC(C(C)C)CNC(C2(c3cccnc3)CC2)=O)ccnc2c1CCO2 N1(C(CC(=C)Br)=O)CCCCC1CCNC(=O)COCC1CCCOC1 C1(CC(=O)NCCc2cnn[nH]2)CCN(C(=O)C=CCN2CCC2)C1 CC(N=c1[nH]c2c(c(=NCC3CC3(C)C)[nH]1)SCC2)c1snnc1C1CC1 N1(CC(C)(C)NC(C2C(C)(CC)C2)=O)CCN(C(c2ccccc2SC)=O)CC1 N1(C(C2CC(C)(CC)C2)=O)CC(F)CC1CN(C)C(c1ccnc(N(C)C)c1)=O c1(OC)ccc(C(=O)N(CCC(C)NC(c2cc(Cl)ns2)=O)C)c(Cl)c1 c1(NC2CCC(C)(C)CC2)ccc(S(=O)(=O)N2CC3C4C=CC(O4)C3C2)cc1F c1(C(=O)NCC(CCNC(C(CCC)C#N)=O)O)noc2c1CN(C(C)C)CC2 N1(CCS(Cc2ccc([N+](=O)[O-])nc2)=O)CCc2ccccc2C1 c1(OC)ccc(NC(C2CCN(C(c3ccc(O)nc3C)=O)CC2)=O)cc1C c1(C(C)NC(C(N2C(C(=O)OC)CC(F)(F)C2)=O)=O)ccc(Cl)c(Cl)c1Cl C1(CNC(=O)COc2ccccc2)CCN(C(c2ccc(Cl)c(Cl)n2)=O)CC1(F)F c1(C(=O)NC2COCC2NC(C2CC2CF)=O)cc2cc(C(F)(F)F)ccc2s1 C1(CNC(CC=CC=C)=O)CCN(C(c2ccnn2CC(F)(F)F)=O)C12CC2 C1(COCC)CCN(C(C2(NC(c3c[nH]c(C)c3)=O)CCCC2C)=O)CC1 C(=O)(C(F)(F)C(C)O)N(C(c1cn(-c2cccc(Br)c2)nn1)C)C CCC(CC)C(=O)NC(C)C(C(C)C)NC(c1cnn(C(C)C)c1Br)=O c1(C(N2CC(CCNC(C(C3CCC(=O)N3)C)=O)C2)=O)cnn2cccc(Cl)c12 CC(CC(=O)N1CC(N(C)C(c2cnn(C3COC3)c2)=O)C(C)(C)C1)C(F)(F)F CC1COCCN(C(C2CC(NC(=O)C(C)n3cccc3)C2)=O)C1 N1(C(CC23C(CN(C(COCCSC)=O)C2)CC3)=O)Cc2cccc(F)c2C1 c1(C(C(=O)NCCCC#C)N(CCC)CC)cnc(-c2ccco2)s1 C12(C(=O)NCC3CCN(C(c4cncc(OC)n4)=O)CC3)CCC(N=[N+]=[N-])C1C2 C=CC1CN(C(C2CC3CCCC3C2)=O)CC1NC(c1csc(C)c1)=O CCC(CCCO)NC(=O)CSCCNC(=O)CC=C(C)C c1(OC)cc(C(=O)NS(=O)(=O)c2cccc(F)c2OC(F)F)cc([N+](=O)[O-])c1Cl c1(C(=O)NCC2N(C(C(C=C)O)=O)CC=C2)cccc(C)c1[N+](=O)[O-] CC1CCN(c2ncc(C(N3CC(O)(CN(C(=O)C(C)CF)C)C3)=O)s2)CC1 n1(CCCCNC(C2CC(O)(Cc3ccccc3)C2)=O)cc(C(O)C2CC2)nn1 CN1CCC2CCN(C(C3CCN(C(C4(O)CCOCC4)=O)C(C)(C)C3)=O)C2C1 N(C1CCc2cccnc21)C(CC(C)C(C)(C)NC(=O)Cc1cccnc1)=O C(=O)(C(C)(O)CCN(C)C)NC(C(=O)NC1(C(C)O)CC1)C1CCC1 c1(OC)cnc(Cl)[nH]c1=NCC1(NC(c2ccnc3ccnn23)=O)COC1 C(=O)(C(F)CCC(C)C)NC(CC)CN(C(c1n[nH]c(=N)[nH]1)=O)CC C(=O)(CCC(=O)N1CCCC(NC(=O)CN(C(=O)C(C)C)C)C1)NCCCOC N1(C(=O)CSc2cccc(F)c2)CCC(C(F)(F)F)(Cc2ccc(F)cc2)C1 c1(CN2CCCC(C(=O)NCc3cncc(Br)c3)C2)cc(Br)ncc1Br C1(C(=O)NCC(C2CC2)NC(C2(C)CCNC2=O)=O)Cc2n[nH]cc2C(=O)N1 C=CC(C)(C)CC(=O)N1CCCCC1C(=O)NC(C)C(O)C(F)F C1(C(C)C)N(C(=O)N(C)C)CC12CCN(N1CCC(C(C3CC3)=O)CC1)CC2 N1(C(CCC(C)OCC)=O)CCOC2CN(C(C3CN(C(=O)N(C)C)C3)=O)CC12 N1(C(c2n(CC)nc(C)c2)=O)CC(C(N2CCC(C3CCC3)C2)=O)C2(CCC2)C1 C1(NC(CC(C)O)=O)COC2(CNC(=O)C(c3ccccc3F)(F)F)CC1C2 c1(OC)ccc2cc(C(=O)NCC(C)CN(C)C(C3CCCO3)=O)ncc2c1 Nc1ncccc1C(=O)NC1(C(N2C(CSc3ccc(O)nn3)CC2)=O)CC1 c1(C(N2C(CNC(C(C)N(CC)CC)=O)CCCC2)=O)cc2ccccc2nn1 C1(C(=O)NCC(CNC(=O)CCNC(C2CCCO2)=O)O)C(F)(F)C12CC2 c1(N(CC(C)NCc2cccc(F)c2C#N)C)cccc(C(N)=O)c1[N+](=O)[O-] N1(C(c2c(C)coc2)=O)CCN(C(c2ccc(F)c(Br)c2)=O)CC(CO)C1 CN1CCN(C(c2cc(F)cnc2O)=O)C(C(=O)NCC2(C)NC(=O)NC2=O)C1 N1(C(CC2CC(=O)NC2=O)=O)CCCC2(CCN(c3ccnc4ncnn34)C2)C1 c12ccc(cc1)c(=O)n2C.C1(C)CN(C(=O)CC2CC3CC3C2)CCO1.CC(=O)N CCC(C(=O)NCC(C)(CC)NC(=O)Cc1n[nH]c(C)n1)OC.C(C)(COC)N CC(C)(C(=O)NCC1(F)CN(C(=O)CCc2ccoc2)C1)c1cnc[nH]1 C(C)(CNC(=O)Cn1cncc1C)(CC1CCCO1)N(C(c1cnn[nH]1)=O)CC C1(NC(C(C)n2ccnc2)=O)CCN(C(C2(C(C)(F)F)CC2)=O)CC1F Cc1ccc(F)c(C(=O)N(C(CC(F)F)C(=O)Nc2cccc(N(C)C)c2)C)n1 Cc1nc(O)ccc1C(=O)NCC(C)CNC(c1ccnc(-n2cccc2)c1)=O Cc1c(C(N2CC=CCC2C(N2CC(C)(C#N)C2)=O)=O)nnn1C c1(C(=O)NC(C2CCCCC2)CNC(C2CC2[N+](=O)[O-])=O)ccnc(O)c1 C1(F)(CNC(=O)CSc2nncs2)CCCN(C(C2CCCCC23CC3)=O)C1 N1(C(CCC=CC)=O)CCN(CC(C)NC(c2csc(COC(C)=O)n2)=O)CC1 N1(C(c2cccc(C)c2)=O)CC2C=CC1C(C(=O)NC(C)(C)C(C)C)C2 C(C(F)(F)CC(O)CO)C(c1ccc(C)s1)C(=O)NCCCC1CC1.CCO c1(C(=O)NCC(CNC(C2(CCC)CCC2)=O)O)cc(OC)c(C)c([N+](=O)[O-])c1 CC(CC(=O)N1CC(CCCCNC(=O)CC2COC(C(F)(F)F)C2)C1)NC(N)=O N1(C(C2CCC(CCCC)CC2)=O)CCN(C(=O)CC2(CSC)CC2)CC1C Nc1cccc(CC(=O)NC(C)(CNC(=O)CC2CCCCO2)C2CC2)c1N N1(C(C(C)OCC#C)=O)CC2(CCCC2NC(=O)Cc2cc(Cl)n(C)n2)C1 N1(C(C(Br)=C(C)C)=O)CCOC2(CCN(C(c3ccc(Cl)nc3O)=O)C2)C1 C1(C(CNC(Cc2nc(CC)sc2)=O)F)CCN(C(c2csc(C)c2)=O)CC1 c1(C(=O)NC2CC(C)(C(=O)OC(C)(C)C)C2(C)C)cc(Br)c(C)c([N+](=O)[O-])c1 N1(C(c2cc(C)on2)=O)CCC(NC(=O)Cc2ccc(O)cn2)C(C)(C)C1 c1(CNC(CCCOCC)=O)ncccc1CNC(=O)C(C1CCCO1)OCC C(CC(C(=O)N1CCC(C(=O)NCC)C1)NC(C12CC(F)(C1)C2)=O)=CC C12(C(N3C4C(CNC(C(N5CCCCCC5)C)=O)C(C4)C3)=O)CCCN1CCC2 Cc1cc(C)cc(C=CC(=O)NCC(C)N(C)C(c2cccn3nccc23)=O)c1 C1(CNC(=O)Cc2ccnc(O)c2)CC2CC1CN2C(C1(F)CC1)=O n1(CC)ncc(C(N2CCC(N(C(=O)C(O)C3CC3)CC(C)C)CC2)=O)c1Cl C(=O)(C1=COCC1)N1CC(CNC(=O)C(c2ccccc2)O)C1 c1(OC)cc(C#N)ccc1C(=O)Nc1ccc(C(N2CC(=O)NC(C)C2)=O)nc1 CC1(C)CCN(C(c2cn(C3CC3)cn2)=O)CC1NC(=O)Cc1cccnc1O c1(C(N(CC(C)O)CCNC(C(CC(=C)C)C)=O)=O)cc2ccnc(Cl)c2s1 CCCCCCCCCC(=O)NCC1CC(NC(=O)CC2CCCOC2)C1 N1(C(CCCc2c(C)ccs2)=O)C2CCC1C(C)C(NC(=O)Cc1ccon1)C2 c1(OC)cccc(CC(N2CC3C(C(=O)NCCc4ccccc4Cl)C3C2)=O)c1 C=C(Cl)C(C)(C)C(=O)NC1CCC(CNC(=O)COc2cc(C)ccc2F)C1 Cc1ccc(Cl)c(C(=O)NC2CC(F)CN(C(=O)C=Cc3ccc(Cl)cc3)C2)c1 c1(CN2C(CNc3cnc(OC)c(Br)c3)CCC2)ccc(O)c(C#N)c1 C1(CC#C)(NC(C2(NC(C3CCC3(OC)OC)=O)CC(F)C2)=O)CCCOC1 c1(C(=O)NCCN(CCC)C(C2(C)CCCC2C)=O)nc2ncc(C)cn2n1 C1(C(N2CC(CCNC(c3cccc4sncc34)=O)C2)=O)CCCCC1C1CC1 C#CC1(C(N2CCOCC(C(=O)NCC3(C)CNC(=O)O3)C2)=O)CCCCC1 C(=O)(C1=CCCOC1)NC1(C2N(C(c3cccc(CC)c3)=O)CCC2)CC1 C#CCC(CC#C)C(=O)N1CC(N(C(=O)CSc2ccc(C)cc2)C)C(C)(C)C1 c1(CC)cc(C(=O)NC(CNC(=O)CSc2cn[nH]c2)CO)ccc1F C1(NC(=O)Cn2cnnn2)CCCN(C(c2cccc(-n3cnnn3)c2)=O)C1 CC(C)C(CNC(c1cc(C#N)n(C)n1)=O)C(=O)NC1CN(C)NC1=O C(=O)(CC(C1CC1)NC(=O)C(CC1CCC1)NC(=O)C=CCCC(C)C)OC N1(C(CCC=C)=O)CCC2(CC(NC(=O)CCc3cnc4n3CCCC4)CO2)C1 c1(CC(=O)NCC(CC)NC(=O)CCCOC)cc(C)on1 N1(C(c2ccnc(OC)n2)C(=O)NCCCCCC)CC(CO)C2(CCC2)C1 Cc1cc(-c2cnccc2C(N2CC(F)CC2CO)=O)ccc1F C1(C)(CNC(C2C(CNC(C3(CC)CCC3)=O)CC2)=O)CCN(C)CC1 C#CC1CCCN(C(=O)C(C)(C)CNC(C2CCC(C(=O)OC)C2)=O)C1 N1(C(=O)CN2CCN(C(C3CCS(=O)CC3)=O)CC2)CCC(CC2CC2)CC1 N1(C(COc2cn(C)nc2)=O)CC2CCC(CNC(=O)Cc3ccns3)C2C1 c1(CCCC(=O)NCCCCn2cc(C(=O)OC)nn2)ccc(Br)cc1 C1(C(=O)NC(c2nocc2C(=O)NCCCC2CCCCC2)C)COCOC1 c1(COCCCNC(c2nnnn2CC(F)F)(C)C2CC2)ncc(Cl)cc1Cl.NC C(CCCCCOC(=O)C(C)CC=Cc1ccccc1)SCc1cc(C)no1 C1(NC(CCC=C(C)C)=O)CCCN(C(C2CC2c2ccc(F)nc2)=O)C1 c1(-c2cn(CC3CC(CNC(CC(CC)C)=O)C3)nn2)ccc2c(c1)CCC2 c1(N2CC3C(CSCC)C3C2)cc(C)[nH]c(=NCC(=O)NCc2ccccc2)n1 N1(C(C=COCC)=O)CCN(CCN(C(=O)CSCc2ccc(F)cc2)C)CC1 CC1COc2c(C(N3CC4CCC(C3)N4C(=O)C(C)O)=O)cccc21 C1(CCOC)CN(C(C2C3(CC3)C23CC3)=O)CCN1C(C1SCCCS1)=O C#Cc1ccc(C(N2C3CCC(C3)C2C(=O)N(CC(C(C)C)OC)C)=O)cc1C N1(C(C(CC)OCC)=O)CCCC(CCNC(c2n[nH]c(C3CC3)c2Br)=O)C1 CC1CCN(C(=O)CCc2cnn(C)c2)CC1CNC(c1ccc(Cl)c(F)c1)=O CN1CCCC(C(=O)NC2(C(F)C(=O)NOCC3CCOCC3)CCCC2)C1 C1(C(=O)NC(c2nnc(C)s2)C)C=CCCN1C(c1ncoc1C)=O CC(C(=O)NCC1(O)CCN(C(c2ncoc2C(F)(F)F)=O)C1)C(C)(F)F C(C(=O)NCC(C)(C)CC1CN(C(=O)Cn2nnc(C)n2)C1)(C(C)(C)C)OC C1(NC(COCc2ccc(C)s2)=O)CN(C(=O)C2=CCCSC2)CC1C1CC1 c1(C(=O)NC2CN(C(CN(C)C)=O)CC2(F)F)ccc(F)c(F)c1Cl c1(C(=O)NCCCN2CCN(Cc3ccc(C)s3)CC2)ccn2cncc2c1 c1(OC)ccc(C(=O)NCC2CCC(NC(c3cc(F)c[nH]3)=O)C2)c(C)c1OC C(=O)(CCCCCCCCCNC(=O)C(C)(C)CC1CNC1)OC N1(C(CCC(C)(C)F)=O)CCC2(C1)CN(C(c1c[nH]nc1Cl)=O)CCO2 C(=O)(C(C)(C)C(C)(F)F)N(CC(CN(c1cc(OC(C)C)ncn1)C)O)C C1(C(N2CCC(F)(CNC(CC)=O)CC2)=O)CCC2CCC(=O)N12 C1(CCC)CN(C(=O)Cc2cscn2)CCN1C(=O)C(O)Cc1cccc(Cl)c1 c1(NC(C=C(C)C)=O)ccc(-c2cn(C3C=CCCC3)nn2)cc1 Nc1ccnc2c(C(=O)NC3CCN(C(C45CC(CN4C4CC4)C5)=O)CC3)cnn12 N1(C(CSCCC)=O)CCCC1(C)CNC(=O)COc1ccccc1 N1(C(CC(CC)SC)=O)CCC(NC(c2cnc(C(N)=O)cn2)=O)C(O)C1 C1(NC(CCn2c(C)nc(C)n2)=O)CN(C(C2SCCCS2)=O)CC(F)(F)C1 N1(C(C=CC=CCC)=O)CCN(C(c2cc(C3CC3)[nH]n2)=O)C(C)CC1C C1(CC)CC(C(=O)NCC(O)C(C)(C)C)CCN1C(=O)CC1CCCN1C CC(C)(C)C(C(=O)NCC1=CCCOC1)NC(=O)CCC1CCC(=O)C1 C1(NC(C=CC)=O)CCC(NC(C2CCCN(C(=O)OC(C)(C)C)C2)=O)CC1 c1(NCCNC(C)C)nccc(=NCC(F)(F)C(F)(F)C(F)(F)F)[nH]1 c1(CNC(C2(CCC)CC2)=O)ccc(C(C)NC(=O)CCOC2CC2)cc1 N1(C(C2(CCCC)CCC2)=O)CCOC(CCCNC(=O)C(C)CN(C)C)C1 c1(C(N2C3CN(CC(=O)N(C)C)C(CC3)C2)=O)ccc2cc(N)ccc2n1 c1(C(=O)NCC2CN(C(C(CN(C)C)O)=O)CC2O)cnn2c1S(=O)(=O)NCC2 Cc1ccc(C(=O)NC2C3CC4C2C4C3c2nc(CN(C)C)no2)cc1O C(=O)(C1=CCCC1C)N.C1(C(=O)OC)(N(C(=O)C=CC)C)CC1 Cc1nccc(C(=O)NC2CCCC(NC(=O)CN3CCCC3=O)C2)n1 N1(C(C2C(C)(C)C2)=O)CCCC(NC(c2cccc(Oc3ccccc3)n2)=O)C1 CC(C)C(CCN(C)C(c1cccc(C(F)F)c1)=O)NC(C1CC2(CSC2)C1)=O C1(C(=O)NC2CC(CNC(C=CC=CC)=O)C2)COCCN1C=O c1(NC(C2CC(=C)CN2C(=O)C2=CC=NC(=O)C2)=O)cc(Cl)nc2ccccc12 c1(CNC(=O)NC2CC(C)OC2)ccnnc1O N1(C(C(C)N(CC)CC)=O)CCC(C(=O)NC(c2nnc(C)s2)C)(CC)C1 c1(C(=O)NC2(CC=C)CN(C(C3CC(C(C)C)=NO3)=O)C2)c(C)nc(O)nc1S c1(OC)ccc(C(C(=O)NC(C)(C)C)N2CCC2C2CCC2)cc1C n1(CC(=O)NC2CCC(CNC(Cc3c(C)nsc3)=O)C2)ccccc1=O c1(C(=O)NCC(CO)NC(=O)CNC(=O)C2CC2)cccc(C2CCOC2)c1 C(=O)(CS(=O)(=O)CC)NCC(CC)NC(=O)CC1CCCS1(=O)=O CCCC(C(=O)NCC1CCOC1=O)NC(c1ccccc1O)=O N1(C(CC(C)C)=O)CCC(NC(c2sccc2OC(F)F)=O)CC1C1CC1 c1(C(N(CC(CC)NC(=O)CCc2cnoc2)C)=O)ccc(N(C)C(C)=O)cc1 C#CCC(C(=O)NC(c1cn(C)nn1)C)NC(c1cc(OCC)ns1)=O N1(C(c2c(OC)nsc2OC)=O)CCC2CC2(NC(=O)C=CSC)CC1 C(=O)(CC(C)P(C)(C)=O)N1CCC(C)(CNC(c2cc(C)sc2C)=O)C1 C=CC1(CC(=O)NCC2CCCC(C)O2)CN(C(c2ccc(C)n2C)=O)C1 C1(COC)(NC(c2cncc(Cl)c2C)=O)CCN(C(C2(O)CCC2)=O)CC1 c1(C(N2CCCC(C(C)NC(c3c(C)sc(O)n3)=O)C2)=O)c(F)ccnc1Cl Cc1cc(C(=O)NCC2(c3ccncc3)CNC2)c(F)c(Br)c1 CCC(CC)(C(=O)NCCOC1CCN(C(=O)C(C)CO)C1)c1cccc(Cl)c1 c1(OC)ccnc(OC)c1C(=O)NCC(O)CNC(=O)CC1CCCCC1(F)F C1(NC(C2N(CC)CC2)=O)CN(C(=O)Cn2ccc(C3CC3)n2)CC1O c1(C(N2CC(C(N)=O)C(NC(C3(C)CCOC3)=O)CC2)=O)ccnc2ccnn12 CC(C)(CNC(=O)C(=O)NC1(C(c2csc(C(C)(F)F)n2)=O)CC1)CCN CCC(C)(C(=O)N1CCc2ccsc2C1)C(F)F CCC(C)C(CC(=O)N(CCN(C)C)C(C)C)NC(C1CC12CC2)=O C1(NC(C2(CC)CCC2)=O)C2CCN(C(=O)CCCC(C)(C)C)CCC12 N1(C(COCCC=C)=O)CCN(C(=O)C2=CCOC2)C(CC2CC2)C1 N1(C(c2c(CC)n(C)nc2)=O)CC2CCC2(CCNC(C2(C#N)CC2)=O)C1 c1(C(=O)NCC(O)CCNC(C2(C(F)F)CCCO2)=O)ccccc1OCCF N1(C(C(CC)OCC)=O)CCC(=O)NC2CN(C(c3nc(=N)cc[nH]3)=O)CCC12 Cc1nc(O)nc(C)c1C(=O)NCC1CN(C(=O)C(C)(Cl)Cl)CCC1C Cn1cc(NC(=O)C(F)C2(CNC(=O)OC(C)(C)C)CC2)c(C2CCC2)n1 c1(-c2c(C)nn(C)c2)cccc2[nH]nc(C(=O)Nc3ncc(I)cc3Br)c12 c1(NC(CCSCC)C)ccc(S(=O)(=O)N2CC3OCOC3C2)c(Cl)c1 C=CC1CN(C(C2CC(CF)C2)=O)CC1NC(c1cc(Cl)cnc1C)=O C1(NC(C(=O)NCC(C(=O)OCC)C(C)C)=O)CCCc2ccccc2C1 N1(C(CC=C=C)=O)CCC(C(=O)N(CC(O)COC)C)(C(C)C)C1 C12(CCNC(CSCCN(CC)CC)=O)CCC1CN(C(=O)C(C)S(C)(=O)=O)C2 C1(NC(C2C(CC)C2)=O)CCC2CN(C(=O)C(c3cscn3)N(C)C)CC2C1 c1(C(N2CC(C(C)NC(=O)C(C)N(C)C)OCC2)=O)cc(S(N)(=O)=O)co1 c1(OC(C)C)ccc(C(=O)NCC2(C)CCCN2C(C2CC2C)=O)c(Cl)c1 C(C)(C)(CN=c1cc(C(F)(F)F)nc[nH]1)c1cn2c(n1)CC(C)CC2 c1(CC(=O)NCCCOCCNC(CC2C(C)CCCC2)=O)ccc(Cl)cc1Cl C1(NCc2cn(Cc3ccccc3)nn2)CCN(CC(C2CC2(C)C)OC)C1 c1(C(=O)NCc2c(C(=O)NC(CCCC)CC)occ2)ccc(C)nc1O c1(CCC(N2CC(CN3CCN(C(C(C)O)=O)CC3)C2)=O)nc2ncccn2n1 c1(C(N2CC(NC(C(C(CC)C)NS(C)(=O)=O)=O)C2)=O)cc(Cl)cc(F)c1N N1(C(c2cc(OCC)c(C)cc2)=O)CCC2(CCC2NC(C2CC2(F)F)=O)CC1 N1(C(C(C)OC2CCOC2)=O)CC2CC1C2NC(=O)C(C)c1ccco1 N1(C(C(=O)NCCC(=O)OCC)c2cn[nH]c2)CC(CC)C2(CCCCC2)C1 c1(CCCSCC)nc(-c2ccnc(C(F)(F)F)n2)n(-c2ccnc(Cl)c2)n1 CN1N=CC(CC(N2CCC(C(=O)NC(C)(C)C(C)(C)C)CC2)=O)C1=O CC1(C)C(CC(=O)NCC2C3COCC23)CCN1C(=O)CSC(F)F C1(CN(C)C(c2c[nH]c(=N)s2)=O)CC(F)CN1C(C1CCCN1C=O)=O c1(C(N2CCCC(N(C(c3cc(C)sc3C)=O)CCF)C2)=O)ncn2c1CCC2 C1(NCc2cn(C)nn2)CC(NC(C2(C)CCCCCC2)=O)C12CCC2 Cc1nn(C)cc1-c1cn(C(C)C(=O)NCCC2COC(C)(C)C2)nn1 N1(C(C(CCC)OC)=O)CC(CNC(c2c[nH]cc(Cl)c2=O)=O)CC1(C)C c1(C(=O)NCCc2c(CNC(CCC(=C)C)=O)nco2)cn(C)c2ncccc12 N1(C(C2(OC)CCC2)=O)CC2CCC2(C(=O)NCC(O)CC2CCCC2)C1 c1(CCC)c(C(=O)NCC2CN(C(c3cccn3C)=O)CC2O)cnn1C C12(C(N3CCC(CC(N4CC(C)C(F)C4)=O)CC3)=O)CCC(N(C)C)(CC1)CC2 c1(OC)ccc(NCCC(=O)NCCCc2cccnc2)cc1 C1(NC(c2scc(C)c2Cl)=O)CC2(CCN(C(C34CCCC3CC(=O)C4)=O)C2)C1 N1(C(CCN(CC)CC)=O)CC2CC(NC(=O)Cc3ccc(Cl)c(Cl)c3)C2C1 N1(C(C=CCN(CC#C)CC)=O)CCC(CO)(CNC(C2CC(F)(CO)C2)=O)C1 CC(CN(C)C(c1cnn(-c2ccncc2)c1)=O)N=c1[nH]nc(O)s1 c1(CSCC)ccccc1C(=O)NCC1CC1NC(C12CC3CC1C2C3)=O C1(CNC(c2cc(C(F)F)nnc2O)=O)CCCCCN1C(=O)CC1CCCO1 CC(CS(C)(=O)=O)C(=O)NC12CC(NC(=O)CCn3ncc4c3CCCC4)(C1)C2 c1(CC=C)cccc(C(=O)NC2(C(=O)NC(c3ccc(C)cc3)C)CC2(C)C)c1 c1(C(=O)NC2CCC(NC(c3ncc[nH]c3=O)=O)C2)cc(F)ccc1C(F)F O=C(CC1=CCCC1)N1CC2C(C(=O)NCCCF)C2C1 N#CC1(C(N2CC3(CCN3C(=O)CN3CCN(C4CC4)CC3)C2)=O)CCCOC1 NS(=O)(=O)c1ccc(C(=O)NCC2CC(NC(c3cscc3F)=O)C2)cc1 C(=O)(C(C)C(C)S(C)(=O)=O)NCC1(F)CN(C(c2c(C)cnn2C)=O)C1 c1(C(N2CC(CNC(c3n(CC)ccn3)=O)C(F)(F)C2)=O)cnn2c1OCCC2 Cn1nc(C(F)(F)F)cc1C(c1nnnn1CCCF)NC1CC(C2CC2)C1 CN1CCOC(C(=O)NC2(C(=O)N(C3CC(F)(F)C3)C)CCOCC2)C1 C1(C(=O)NC(C2Cc3ccccc3O2)(C)C)Cc2cccnc2NC1=O N1(C(CCCNC(C)=O)=O)CC2CCC1CC2NC(c1nccc2cc[nH]c12)=O CC(C(C)(C)C(=O)N1CCN(CCO)C(=O)C1)NC(=O)CCC1CC1(C)C C12(CC(=O)NC3CC(C)(NC(C(C)Cc4ccccc4)=O)C3)COC(CF)(C1)C2 C1(CC)CCN(C(c2ccon2)=O)C1CNC(=O)C(CCO)N(C)C C#Cc1ccc(CC(=O)NC2CC2NC(=O)C(CC)n2ccnc2)c(F)c1 N1(C(c2c(C)nc(C(C)C)s2)=O)CC2=C(C1)CN(C(c1nn(C)cc1N)=O)C2 C=C(C)C(CC(=O)N(CC(C)O)CCNC(c1cc2occc2s1)=O)OCC C1(C(N2CCN(C(CCC)=O)CC2)=O)CC12CCN(Cc1nc(Cl)ccc1F)C2 C(=O)(CC(C(F)(F)F)NC(=O)C=CC1CCCCC1)N(C1CCNC1=O)CC C1(C(N2CC3(COC3)C2)=O)C2CCCC2CN1Cc1ccccc1 c1(C(N2CC(F)(CNC(=O)CC3(O)CCCOC3)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 C1(CC(=O)N(C)Cc2cc(=N)[nH][nH]2)C2CN(C(c3cc(CO)[nH]n3)=O)CC12 C1(NC(c2c(OCCOC)cccc2)=O)CCCN(c2ncncc2I)CC1 CC1CCC(NC(=O)Cn2ccc(C(F)(F)F)n2)CN1C(=O)CCc1nccs1 C1(C(C)NC(C)C(=O)NC2(c3cnn(CC(=O)O)c3)CC2)COc2ccccc2O1 C1(NC(=O)CC2CCN(C(=O)CO)C2)CCC(NC(=O)C(F)n2ccnc2)CC1 N1(C(C(C)CSC(F)(F)F)=O)CCN(C(c2cn(C)nn2)=O)C(c2cn[nH]c2)C1 O=C(C1=CCCCO1)Nc1ccc(C2CCN(Cc3ccc(Br)c(Br)c3)C2)cc1 Cc1ncn2ccc(C(N3CC4C(NC(c5nn[nH]c5Cl)=O)C4C3)=O)cc12 C1(C(=O)NCc2c(CNC(C3CN(C)C3)=O)cccn2)CCc2nn(C)cc2C1 C1(CC(=O)NCC(CN(C)Cc2cc(C)sc2)(C)C)CCCCCC1 N1(C(=O)C(F)C2CCOC2)CCC2(C1)CN(C(c1ccnc(Cl)c1F)=O)C2 c1(N2CC(C#N)OCC2)nc(=NCc2ccccc2Br)[nH]c2c1SCC2 C(=O)(CC(C)(C)CC(F)(F)F)N(CCCNC(c1ncc(F)cn1)=O)C N1(C(c2cnn(CCCC)c2C)=O)CCC(CNC(c2cc(Cl)on2)=O)C12CC2 N1(C(C2(C(C)C)N(C(c3ccc(CC)nc3)=O)CCC2)=O)CC(OC)CCC1C c1(C(=O)NC2CCN(C(C3C(C)(C)CO3)=O)C2(C)C)cn2c(n1)CCCC2 N(C(=NCC(=O)Nc1cccnc1)NC1CCCC1)C(C1CCCC1)C#C C1(O)(CNC(c2cccc(OC)n2)=O)CCN(C(c2ccc(=O)n(C)n2)=O)CC1 N1(C(c2c(CC)con2)=O)CC2(C1)SCCC2NC(=O)Cc1cc(F)ccc1F N1(C(Cn2c(C)ccn2)=O)CCC2(CC(C(=O)N(C)CCC3CN(C)C3)C2)C1 N1(C(CCS(N)(=O)=O)=O)CCCCCC(NC(c2cc3cc(Cl)sc3[nH]2)=O)C1 N1(C(CCN(C(C)=O)C)=O)CCCCC1CNC(C1(C(F)(F)F)CCCCO1)=O CC(C)CC(CC(=O)O)NC(C1CCCN(Cc2cncc(N(C)C)c2)CC1)=O c1(OC)ccc(C=CC(=O)NCC(CNC(=O)CC2CC2)CO)cc1 C=C1CC2(C1)CC(C(=O)NCC(c1ccccc1)CNC(=O)CCC(F)(F)F)C2 c1(C(=O)OC)c[nH]c(=NCCCCC(C)NC(=O)C(C)C(C)C)cc1C N1(C(C=C(C)Cl)=O)CCCCC(CNC(=O)C(C)Sc2ccccc2Cl)C1 c1(C2(CN(C)C)CC2)cn(CCNC(=O)CONC(=O)OC(C)(C)C)nn1 C(C1CCS(=O)(=O)c2ccccc21)NC(=O)NC1CC(C(CC)CC)OCC1 Cc1cc(C(N2CCC2CC(=O)NCC2CCC2N(C)C)=O)cnc1C O(P(=O)(CCCNC(Cn1cccn1)CC)OCC)CC C1(C(C)C)C(NC(=O)Cn2cncn2)CCN1C(c1cc(C2CC2)nn1C)=O c1(CNc2nccc(N3CC(C)C(C)C3)n2)c(F)cccc1F O=C1CC2CC(C(N3CCN(C(=O)CCc4ncco4)CC3)=O)C1C2 C(c1cc(F)cc(F)c1)=CC(=O)N(C1C2CN(C(C3(CCF)CCC3)=O)CC12)C N(C(=NCC1CCOC1)N1CCC(C2CCC2)C1)Cc1cc(C(F)(F)F)no1 Cc1cccc(F)c1C(=O)NC1CCC(CC(=O)NCC2CCCNC2=O)C1 c1(N2CCC(C(C)NC(C(c3c(C)cccc3)C)=O)CC2)ccccc1[N+](=O)[O-] C12(NC(C3N(C(C(C4CCN(C(C)C)C4)F)=O)CCC3)=O)CCC(C1)C(O)C2O c1(C=O)[nH]c(O)nc1C.c1(C)cn(CC2(CN(OC)CC3CCCC3)CC2)nn1 c1(CC(=O)N(C(C)CN(C(=O)CC2CCOC2)C)C)cncc2ccccc12 N1(C(CNC=O)=O)CCC(C(F)(F)F)CC1CNC(c1cc(C(N)=O)[nH]n1)=O c1(C(=O)NCC(CO)NC(C2(C(C)C)CCCO2)=O)ccc2cccnc2c1 C#Cc1cc(NCCCCCNC2(c3nnnn3C)CCOC(CC)C2)ccc1Cl c1(C(=O)NC(CNC(CC(C=C)C)=O)C2CC2)ccc(OC)c(OC)c1C N1(C(C(CN(C)C)NC(C(C)OCC)=O)=O)CC(C)(C)CC1C CC1(NC(=O)Nc2cccc(-c3ncc[nH]3)c2)CCOC1C1CC1 CC1CCN(C(=O)C(C)Cc2ccccc2F)C1CNC(=O)C=Cc1cnc[nH]1 N1(C(=O)Cc2csc(Cl)n2)CCC(C2CCN(C(=O)C3=CCCC3)CC2)C1 N1(C(CCC2CCCN(C(c3n(C=C)ncc3)=O)C2)=O)CC(O)C(C)(C)C1 c1(C(C)OCC)ncc(C(N2CC(O)(CNC(C3(COC)CCOC3)=O)C2)=O)s1 C1(NC(C2CN(C(C)C)C2)=O)CC2(C1)CC(NC(c1cc(C3CC3)on1)=O)C2 CCC(C)C(=O)C(=O)N(CC(=O)NC(c1nn(C)cc1O)C)C c1(C(=O)NC(CCNC(CCCOCCOC)=O)C)cc2c(C)ccc(C)c2[nH]1 C=CCC(C)(C)C(=O)N1CCCCC(N(C(=O)C=CCOCCOC)C)C1 C1(CCNC(CC)=O)CC(F)(F)CN1C(=O)C(C)CN1CCOCC1 N1(Cc2c(F)ccc(OC)n2)CC2CCCCC2C1.c12cc(ncn1)N2 C1(NC(=O)C(Cl)(Cl)Cl)CCC2(C1)CN(C(=O)NCc1cc(F)c(C(=O)O)cc1F)C2 C1(C(N2CCC(CC(=O)NC(C)(C)C=CCl)C2)=O)CCCCC(=O)N1 CCCC(CCC)C(=O)NC1CCC(NC(c2cc(C3CCC3)no2)=O)C1 c1(C(=O)NCCN(CCC)C(C2CCCC23CC3)=O)cc2c(C)cc(F)cc2[nH]1 C(c1c(F)cccc1F)=CC(=O)NC1CCCC(NC(CCC(C)(F)F)=O)C1 CCCCC(C)CCC(=O)N1CC(NC(=O)C(C)(C)c2ccno2)CC(C)C1 S1(=O)(=O)c2ccc(c(C#N)c2)N1.C12(CN3CC(CC)OCC3)CCCC1C2(F)F C(=O)(C(C)C=C=C)NCC(CC=C)NC(c1ccc(N2CC=CC2)cc1)=O CCC(C(=O)N1CC(C(=O)NCCc2cn(C)nn2)C2(CC2)C1)C(C)C C1(C(=O)NCC2(NC(=O)CCc3cncc(F)c3)CCOC2)(CC)CCOCC1 N(C(=S)c1cccc(Br)c1)(CCC#N)Cc1ccc(CCC)cc1 C=Cn1nccc1C(=O)N(C(C)CNC(c1sc(-c2ncc[nH]2)nc1C)=O)C c1(C(=O)NCC(CN(C(c2nc(C(C)C)oc2)=O)C)O)cccc(C2COC2)c1 N1(C(CN(S(C)(=O)=O)C)=O)CCCCC1C1CCCN1Cc1ccc(F)cc1Cl C=CCC(CC=C)C(=O)NC1CC2CC(NC(=O)C(COC)COC)CC12 c1(OCC#C)cccc(C(N2CCCCC2CC(=O)O)=O)c1 c1(C(=O)NCC(=O)NC(CC(C)NC(C2(CC)CCC2)=O)C)cncc(Br)c1 N1(C(c2cnc[nH]2)=O)CCC2(CCCN(C(C3CC34CCCCC4)=O)C2)C1 CC(C)C(CCC(=O)N1CCN(C2CC2)C(C)C1)NC(=O)CCC(N)=O C1(CNC(=O)OCC(c2ccccc2)N2CCC2)CCC(C(F)(F)F)CC1 C1(NC(C(C)(C)OCC)=O)CCC(NC(=O)CCC2CCCC2)CC1 C(=O)(CC1c2ccccc2C(=O)N1C)NCC=CCNC(Cc1nnc(C)o1)=O N1(C(C(C)=C(CC)C)=O)CC(CNC(=O)CN(C(=O)COC)C)CC1(C)C C1(C(=O)NC(C)C(CO)NC(=O)COC2CCCC2)CCS(=O)(=O)N1C N1(C(CSC)=O)CCC2(COCC(CNC(c3cccnc3C(F)F)=O)O2)C1 CCCC(C)CC(=O)N1CC=CC(NC(c2ccn(CC3CC3)c2C)=O)C1 C1(O)(C(=O)NC2C(CC)C2)CCN(S(=O)(=O)Cc2ccc(Br)cc2)CC1 n1(CC(=O)NCCC2CCN(C(=O)CC3CC=CCC3)C2)nc2c(n1)CCCC2 N1(C(CN(C(C)=O)C)=O)CCCC(C)(C(=O)Nc2cnc(Cl)nc2)C1 c1(C(=O)NCC(C2CCOC2)NC(c2c(C)[nH]nc2Cl)=O)csc2c1CCCC2 C1(C(=O)NCCC2CCC2)COCCC1NC(C1(CO)COC1)=O C1(C(N(C)Cc2nccn2C)=O)CCCN1C(=O)COC1CCC1 c1(C(=O)NC(CNC(c2ccc(F)c(F)c2F)=O)CO)ccc(F)c2c1OCC2 C1(NC(CNC(CC)=O)=O)CCCC12CCN(C(=O)COCCF)C2 C(=O)(C1=CCC2CCC1N2C(=O)Cn1cccn1)N(C1COCC1O)CC C1(CC)(NC(=O)CC2CC(F)C2)CCN(C(C2CCCCC2(C)C)=O)CC1 Cc1cccc(F)c1CNC(=O)Cc1csc(=NCc2ccc(N(C)C)cc2)[nH]1 Cc1ccc(C(=O)NC(C)CC(C)NC(C2(F)CC=CCC2)=O)c(O)c1 C(c1cocn1)=CC(=O)NC1CCC(NC(=O)COCc2cccnc2)C1 C(=O)(C(C(C)NC(C1CC2CC(=O)C1O2)=O)C(C)C)NCC=CCCC N1(C(C2CCCN(CCC)C2)=O)CCC2(CCCN(c3ncccc3C#N)C2)C1 c1(NC(C2C(CNC(C(C(COC)C)C)=O)CCCC2)=O)ccc2nncn2c1 c1(C(N(CC(=O)NC(C(C)(C)O)C2CC2)CC)=O)ccnc(C)c1C CS(=O)(=O)c1ccc(C(=O)NC2CN(C(C3CC3C#N)=O)C3(CCC3)C2)s1 C1(c2ccc(F)cc2)(C(=O)OC)CCN(C(=O)C(C(C)O)N(C)C)C1 C(=O)(CCCC(F)(F)F)N1CC(SC)C(NC(=O)C(c2cc(F)cc(F)c2)O)C1 N1(C(c2coc(CS(C)(=O)=O)n2)C)CCN(C(=O)CS(N)(=O)=O)CC1CF N1(C(C2C(OC)CCC2)=O)CCN(C(c2cc(Cl)c(Cl)n2C)=O)CC1CO N1(C(C(C(=O)OC)C)=O)CC2(C1)CN(C(C1(n3nccn3)CC1)=O)C2 c1(C(N(CCCNC(C2CCCO2)=O)CC)=O)cccc(C(F)F)c1F c1(C(=O)NC2CC3C(NC(C4C(C)=CCS4)=O)C3C2)n[nH]c(C)c1[N+](=O)[O-] C1(C2CC2)(NC(CCC(=O)NCC)=O)CCN(C(=O)CN2CCS(=O)(=O)CC2)C1 c1(C(=O)NC2C(C(N(CC=C)C3CC3)=O)COCC2)cc(C)ccc1F c1(C(C)(C(F)(F)F)NC(C(C2CCNCC2)C)=O)ccc(C#N)cc1 C1(C(=O)NCc2cc(C(N(CC(COC)(C)C)C)=O)n(C)n2)CCCC2(CC2)C1 C(CCC(O)C(=O)NCCC1CCCC(C)C1)NC(CC=CC)=O n1(CCCC)cc(C2(C(=O)OC)CN(C(=O)C(n3cc(Br)cn3)C)C2)nn1 c1(C(N2CCCC(CCNC(CC)=O)C2)=O)cc(O)cc(O)n1 C1(NC(CC(COC)(C)C)=O)CCN(C(C2CCCC3(CCC3)O2)=O)CC1(C)C C12(C(N3CC(CCCCNC(=O)Cc4ccno4)C3)=O)CC3CC(CC(C3)C1)C2 CC1CCC(=CC(=O)NCC2CC2NC(c2n[nH]cc2-c2ccncc2)=O)CC1 C(=O)(CC(C)P(C)(C)=O)N1C(CO)CC(NC(c2c(CC)ocn2)=O)C1 N1(C(C2(CC(C)C)CC2)=O)CC(NC(C2CC(=C3CC3)C2)=O)C(O)C1 C(C(=O)N1CC(N(C(=O)CC2OCCCO2)C)C1)(C(C)C)NC(C(C)OC)=O N1(C(c2c(CC)nn(C)c2)=O)CC2(CCC2NC(=O)C(C)SC(C)C)C1 N1(C(C2(NC(C)=O)CCC2)=O)CCCN(C(C2CCC(=O)NC2)=O)C(C)C1 c1(CNC(COC2CN(C(CC(CC)OC)=O)C2)=O)cnc(F)c(C)c1 c1(N(C(=O)CC2CCCC(=O)N2)CC)ccc(F)cc1.C1C(F)(F)CN1 C1(CC)C(C(=O)NOCC(=O)OC(C)C)CCCN1C(c1ncc(N)cc1C)=O c1(C(=O)NC(C2CCCCC2)C(=O)NCc2cc(Cl)no2)cc2sccc2[nH]1 C(=O)(C1=CC(C)(C)C1)N(C1(CC(=O)NCC2CCCOCC2)CC1)C c1(CC(N2C(CCCNC(C3C(C)OCC3)=O)CCC2)=O)ccc(O)cc1 CCC(C)C(C(=O)NC(C)(C)CCCNC(c1cccc(Cl)c1OC)=O)OC N1(CC(=O)NNC(=O)c2ccccc2)CC(O)CC2(CC2)C1 C12(C)CCN(C1)C(=O)CCN(C)C(=O)C1CCC1OO2.N(C)(CC)CC CC1(C)CN(C(=O)CCCC(=O)C2CC2)CCC1NC(=O)Cc1ccc(F)cc1 C=C(C)CC(C(=O)N1CCSC(C)C1)NC(=O)CC1CC2CCC1O2 Nc1c(C(=O)NC2CC(NC(c3ccco3)=O)C2)ccc(F)c1F c1(NC(C(=O)NCc2cc(C)c(I)cc2)=O)ccc2c(c1)CC(N)C2 C1(O)(C(=O)NCCSCC(=O)NCC2(C(C)(C)O)CC2)CCCC1 c1(CCC)nc(C)c(C(=O)NCC2(C)CCN(C(c3cnoc3C3CC3)=O)C2)o1 C#CCCCC(=O)NC12CC1CN(C(=O)C(C)(F)c1ccccc1)C2 c1(C(N2C(CNC(C3N(CC)CC3)=O)C=CC2)=O)ccc(C(F)(F)F)c(F)c1C N1(C(N2CCC(C)CC2)=O)CCc2c(F)ccc(C#N)c2C1 c1(CC(=O)NC2CCN(C(C(CC#C)C)=O)C23CC3)cc(Cl)cc2c1OCC2 C1(C(=O)NCCc2cc(CC)no2)CCCCC1NC(C1(CO)CCC1)=O c1(C(=O)NCC2N(C(Cc3c(C)con3)=O)CCC2C)ccc(F)cc1[N+](=O)[O-] c1(C(N2CC(N(C)C(c3ccsc3)=O)C(O)CC2)=O)cnn2ccn(C)c12 CC1CN(C(=O)CO)CC1n1cc(-c2ccsc2)nn1 C=CC(C)(CCOC)C(=O)N1CCN(CC(C)(C)NC(C2(C)CCCO2)=O)CC1 C1(CNC(C(C)C(C)(F)F)=O)CC(C)(C)OC1(C)C C(=O)(CC(=O)NC1CC1)N(CC(CNC(CC=C)=O)O)C n1(CCCn2cc(C(C)OC)nn2)ncc2ccccc12 C(C(CC1CCCC1)C(=O)NCc1ncc(C)[nH]1)NC(CC(C)SC)=O N1(C(C=CC(c2ncccc2F)(C)C)=O)CC(NC(=O)CC(=O)NCC2CC2)C(F)C1 N1(C(C(=O)NCCSC)C2CCSC2)CCOCC1c1c(C)n[nH]c1C C1(NC(c2cccc(F)c2C(F)(F)F)=O)CC2CC1CN(C(c1cnsc1)=O)C2 c1(C(N2CCC(COC)(NC(=O)Cc3ncccc3C)C2)=O)cc(F)ccc1Cl N#Cc1ccccc1OCCS(=O)(=O)NC1(c2cccc(F)c2)CCCC1 c1(C(=O)NCCOCCCN(C(=O)CCN2CCOC2=O)C)ccc(Cl)c(F)c1 CCCC(C)CC(=O)N1CCC(CCC(=O)NC23CC2CN(C)C3)C1 C1(O)(C(C(=O)N(CCC(N)=O)CC)F)CN(C(c2coc(N(C)C)n2)=O)C1 C1(NC2C(C#N)Cc3c[nH]nc3C2)COC2(CCN(C(C3CCCC3)=O)CC2)C1 CCC(CC(=O)N1CCC(C)(C)C1C(=O)N(C)Cc1sccc1C)CC(C)C C1(C)(CNC(C(C2CCN(C(=O)OC(C)(C)C)C2)C)=O)CC(O)C1 C(=O)(CCCC(C)(C)C#N)NC1C(C(N(CC(CC)O)CC)=O)CC1 C#CC1(C(=O)NCC(O)CC(=O)NCC(C)C(C)C)CCCCC1 CCCCCC(O)CC(=O)N(C(C)C(N1CC(C)(C)CC1C)=O)CC CCS(=O)c1ccccc1C(=O)NC1(CNC(C2CC2(Cl)Cl)=O)CCCCC1 N1(C(C2(CC=C)CCC2)=O)CC(NC(=O)C(C)(C)CF)C(F)C1 Cc1cncc(C(=O)NC(C(=O)NCC(C)C(F)F)C(C)C)n1 Cc1cc(=O)ccn1CC(N1CCC1CNC(c1cn(C2CCOC2)cn1)=O)=O c1(C(=O)NC2CC(CNC(=O)C(c3ncccc3F)(F)F)C2)ccc(Cl)cc1Cl Cc1cc(C(N2CCCC2)=O)ncc1-c1ccccc1CN(CC(=O)O)C Cc1csc(C(C)C(=O)N(CCNC(C2CCC(=O)N2)=O)C2CC2)n1 N1(C(C(CSC)OC)=O)CCCCC1C1(NC(c2csc(C)c2)=O)CC1 c1(C(N(CCCN(C(C(C)Oc2cccc(F)c2)=O)C)C)=O)cncc(F)c1Cl CCC(C)(CCNC(c1cnn[nH]1)=O)NC(=O)CCCOC(C)C N1(C(C(F)=CCC)=O)CC(C(=O)Nc2ccc(N(C)C)nc2)CC(C)(C)C1 c1(NC(N2CC(NCCC3CC4CCC3C4)C2)=O)cccc(N2CCOCC2)c1 C1(CNC(c2ccn(C3CC3)n2)=O)(CNC(C2(Cl)CC2)=O)CC1(F)F N1(C(C(=O)NC2CC2)=O)CCC2CN(C(=O)CC3OCCCO3)CC12 c1(CC)nnc2n1CCCC2C(=O)NCCCc1cn(C2COCC2O)nn1 c1(C(N(CCCNC(CNC(CCC)=O)=O)CCC)=O)sc(O)nc1C C1(NC(C2CN(C)CC(C)O2)=O)CC2(CCN(C(=O)CC(C)(C)C)C2)C1 c1(SC)ccccc1CC(=O)N(CCCCNC(C1CC1(F)Cl)=O)C c1(C(=O)NCC2C(CNC(c3c(C(C)C)ocn3)=O)C2)nccn2nccc12 c1(C(N2C(C(=O)NCC3N(CC)CCCC3)CC3CC32)=O)occ2c1CCC2 N1(C(C2CCCC(OC)C2)=O)CCOC2CN(C(=O)C(N)=O)CC12 Cc1cc2ncn(CC(=O)NC3CC(O)CN(C(C4CCCC4)=O)C3)c2cc1C c1(C(=O)NCc2c(OC)n(C)nc2)cc(F)ccc1CN C=C1CC2(C1)CC(C(N1CCC(NC(=O)Cn3ncnn3)C1C)=O)C2 c1(C(=O)NC(C(C)NC(CCc2cc(C)no2)=O)C)ccc(-c2ccsc2)cc1 N1(C(CCc2ncc(C)[nH]2)=O)CC2CCCC1(CNC(C1CCCCC1O)=O)C2 c1(C(N(C2CCN(C(=O)COCC(F)F)C2)CC)=O)cccc2nc[nH]c12 CC1CN(C(=O)CCc2ccn(C)c2)CCC1N(C(=O)C=CC1CCC1)C c1(C(=O)OC)ccc(S(C)(=O)=NC(=O)CC(C)(C2CCCCCC2)OC)cc1 C1(C(N(C)CCOCCNC(c2cc(F)ccc2Cl)=O)=O)CCc2cncn2C1 N1(C(C(C(C)C)C)=O)CCN(C(C2CCC(C)(C)C2)=O)CCC1C c1(C(N(CC(C)NC(c2c(C)ccc(OC)n2)=O)C)=O)ccc2c(C)[nH]nc2c1 N1(C(C(Cc2cn[nH]c2)NC(=O)CC=C(Cl)Cl)=O)CCC(C2CCC2)C1 C1(CNC(CCSCC(C)C)=O)CN(C(=O)C(F)(F)Sc2cnn(C)c2)CC1C C1(NC(C23CC(C)C2C3)=O)CCC2(CC1)CN(C(C1CCC(C(=O)OC)O1)=O)C2 c1(C(=O)NC23C(CN(C(c4ccc(C)o4)=O)C2)C3)cc2sc(C)cc2s1 C(=O)(C1=C(C)OCCS1)N1CCC(C=C)(C(N2CCOCCC2CC)=O)C1 c1(C(N2CCCC(NC(C3CCS(=O)(=O)C3)=O)C2)=O)cc(Cl)ccc1Cl C(=O)(CCCCCCN=[N+]=[N-])N1C(CNC(=O)C(C)C2CC2)CC(OC)C1 c12ccc(c(C#N)c1)[nH]2.c1(C(N2C(C)CCC2)=O)ccnc(-c2ncc[nH]2)c1 c1(CNC(=O)Nc2c(C)n(CC(C)C)nc2)ccc(=O)n(C2CC2)c1 Cn1cc([N+](=O)[O-])c(C(=O)NC2CCCN(C(=O)Cc3ccns3)CC2)n1 C(=O)(CCCN=[N+]=[N-])NC1C(NC(C2C(C)(C)CCC2)=O)CCCC1 Cc1ccc2c(ccn2CC(N2CC3CCC2CC3O)=O)c1 c1(C2CCN(C(c3nc(C(=O)O)nn3C)C)CC2)ccc(Cl)cc1Cl N1(C(CCc2cc(C)[nH]n2)=O)CCOC(CC(=O)NCCn2cnnn2)C1 N1(C(CC2N(C(CC3CC(=C)C3)=O)CC2)=O)CC(F)(F)CC1C c1(C(N2CC(C)C(CNC(=O)C(N)=O)C2)=O)ccc(O)cc1F CC1(C)CC(CNC(=O)CCOCC(F)(F)C(F)F)CN(C(c2csnn2)=O)C1 C(=O)(C(C)C(O)CCCC)N1CC(CC(CCC)(C)C)C1.C12(CNC(=O)C1)C(=O)N2 N1(C(c2n(CC=C)ccn2)=O)CC2C(CNC(=O)CCC(C)C)C2C1 C1(CNC(c2ccc(F)cc2Cl)=O)C(O)C(O)CN1C(C1CC2C=CC1O2)=O S(=O)(=O)(c1ccc(NC2CCC(N(C)C)C2)cc1Br)NC(CC(=O)NC)C C(=O)(CC(CC(C)C)NC(=O)Cc1cn(C)cn1)NC(CC=C)(C)CC=C C1(O)(C(C(=O)OCC)(F)F)CCN(C(CCCNC=O)C(=O)NC)CC1 O=C(CC1=CCCCC1)NCCC12CCC1CN(C(C1CN(C3CCC3)C1)=O)C2 CCCCC(C(=O)NC(CNC(c1occ2c1CCOC2)=O)C1CC1)C(C)C C1(NC(c2c(SCC)nccn2)=O)CN(C(=O)CCOCC(F)(F)F)CC1(C)C C12(NC(C3C(SC)CCC3)=O)CC(C1)N(C(=O)COCc1cc(C)on1)C2 c1(CC)cc(C(=O)NCc2ccoc2C(=O)NOC2CCC2)c(C)o1 c1(CC(=O)NCC2(C)CC(NC(C3C=CCC3)=O)C2)c(Cl)cccc1Cl C1(NC(c2c(CNC(CC3(C)CCCCC3)=O)cc[nH]2)=O)C(=O)OCC1(C)C C(=O)(C(O)C(F)(F)c1ccccc1)Nc1ccc(N2CC(C)OCC2)nc1 N1(C(COCC)=O)CC2CN(C(=O)C(C(C)C)n3cc(C)cn3)CC2(C)C1 C(C(CC(C)C)C(=O)NOC(C)(C)CO)NC(c1ccnc(C)c1C)=O N1(CC)CC(CNC(=O)C(CC2CCCC2)NC(=O)CC(Cl)Cl)CC1=O c1(C(N2CCC(NC(C=CCOC)=O)(CO)CC2)=O)c[nH]c2ncccc12 c1(C(N(C)CC2N(C(C(C=C)C)=O)CCC2)=O)cc2cccc(C)c2[nH]1 C(=O)(CC(C)C(C)C(C)C)N1C(CCNC(C(CC=C)C)=O)CCC1 N1(C(CCC=CC)=O)C2CCCC1CN(C(=O)CCCCNC(C)=O)CC2 c1(C(N(CCNC(c2cncnc2C)=O)CC)=O)cccc2c3c([nH]c12)CCC3 Cc1nn(CC(N2CCC(NC(c3ncccc3F)=O)C(F)C2)=O)cc1[N+](=O)[O-] c1(C(=O)NC2CC(NC(c3c(OCC)ccs3)=O)C2)c(OC)ccnc1F CC1c2ccc(Br)c(Cl)c2CCN1CC1(c2cccc(F)c2)CCC1 C1(NC(C(CCC)(C)CC)=O)CC1C1CCCN(C(=O)CCCOC(C)C)C1 CN1CCCCCC1C(N1CCC(C(F)C(N2CCCC2CN=[N+]=[N-])=O)C1)=O c1(C(=O)NC(CCC)CC(=O)NCCN2CC3CCC2C3)ccc2n[nH]cc2c1 c1(COC)ccccc1C(=O)N(CCC(C(C)C)NC(=O)CC1(O)CC1)C C1(C(=O)NCCCC2(O)CCC2)(CNC(CCCNC(=O)OC)=O)CC(C)(C)C1 C1(C(N2CCN(C(c3c(C)n(CC4CC4)cc3)=O)CC2)=O)CCCC1S(C)(=O)=O c1(CC)nc(C)oc1C(=O)N(CC(C)NC(=O)C(C)SCc1ccccc1)C c1(OC(C)CNS(CCO)(=O)=O)ccc(I)cc1.c1(C)cc(-c2ccccc2)no1 N1(C(C2C(C)(C)CC2)=O)CC(CO)C2(C1)CN(C(c1cc3n(n1)CCC3)=O)C2 C1(CNC(c2cnc(CC)s2)=O)CN(C(=O)CN2CCC2C)C2(CCOCC2)C1 N12CC3COCC3(C1)C2=O.CCC(CN(C)C)C(=O)N1CC(O)CC1CC c1(Cn2cc(C(N3CC(CN)C3)=O)nn2)oc2ccccc2c1Br c1(NCCC(=O)NC2CCCN(C(=O)CN3CCCC3)CC2)cccc(F)c1F CCCCCC(CC)C(=O)NC1CC(C(F)C(=O)NCCCCF)C1 C1(CNC(C(C)=CC)=O)CC2CCC1N2C(C1CCCN(S(C)(=O)=O)C1)=O C1(C(=O)OC)CC(C)N(C(c2scc(C(C)=O)c2Cl)C(=O)NCCC2CC2)C1 C(C)(C(=O)NCCCC)NC(=O)OC(C)CCC.C(C)C c1(C(=O)NCC=CCNC(C2(CC(C)C)CC2)=O)cc(F)c(Br)c(F)c1N c1(C(=O)NC(C(C)NC(=O)CCc2ccoc2)CO)ccc(O)c([N+](=O)[O-])c1 c1(OC)c(Br)cc(C(=O)O)cc1S(=O)(=O)NCCC(O)C(=O)O CCC(CC(=O)N1CCN(CC2CCN(C(c3ccccc3)=O)CC2)CC1)OC C1(C(N(CC(C)NC(C2CC(=O)N(C3CC3)C2)=O)C)=O)CCCN1N=O N1(C(CC(C)O)=O)CC(N(C)C)C(CNC(c2csc(Cl)c2)=O)C1 c1(C(=O)NCCNC(c2cc(Cl)cnn2)=O)cc(F)c(F)cc1O CCCCCC(C)(C)C(=O)NCC(=O)NCCC1CCCS1 C(=O)(C#CC(C)(C)C)N1C(C(=O)NC2(c3ncc(C)o3)CC2)(COC)C=CC1 N1(C(C2(OCC)CCCC2)=O)CCOC(CNC(=O)Cc2ccsc2C)C1 C1(NC(c2ccc(-c3cscn3)nc2)=O)CC2CC(NC(c3cccs3)=O)C1C2 Cc1cccc2c(C(=O)NC3CCCC3NC(=O)CC=C(Cl)Cl)n[nH]c12 Cc1[nH]ccc(=NC(=O)CNC2CC2C(=O)NC2CCN(C)C2)c1F C1(CNC(c2c(C)nsc2)=O)CC2CN(C(=O)CCc3ccc[nH]3)CC12 C12(CN(C(=O)Cc3ccn(CC)n3)C1)C(=O)NC2.C(C(C)(C)O)OC=C Fc1ccc(Cl)c(Br)c1CNC12CCC1CNC2 CC1NC(=O)CCC1CNC(C1(NC(c2ccccn2)=O)CC(O)C1)=O C1(NC(CC(=C)Br)=O)CCC(CNC(=O)CN2CCCC2=O)CC1 C1(C(=O)NC(C(=O)NCC2CCCN(C)C2)Cn2ccnn2)CC12CCCCC2 CC1=CCC(C(N2CC=CC(NC(=O)CN3CCCC3=O)C2)=O)CC1 c12ccc(cc1O)NC(=O)C2.C1(SC(C=CC(=O)OC)(C)C)CN(C)CCO1 c1(CNC(=O)NC(C)C(c2cccc(Cl)c2)O)cc(Br)ccc1F c1(CC(C(=O)OC(C(C)O)(C)C)NC(=O)OCC(C)(C)C)cc(F)cc(F)c1 C(=O)(CCC1=NNC(=O)CC1)NCCCC(C)NC(=O)CSCc1cccs1 C=C(Cl)CC(C(=O)NC(CO)C(=O)OC)NC(=O)CCCCOC.O(C)CC C1(NC(CC2ON=C(CC)C2)=O)CN(C(=O)C(C)(C)c2cc[nH]n2)CCC1CO CC(O)CCCCCC(=O)N1CCC2CN(C(=O)COC3CCCC3)CC2C1 c1(C(=O)NCC2N(c3c(F)cnc(C)n3)CCC2)cccc2c1ccn2C c1(CC)ccc(C(N2CC(O)(C(C)NC(c3oc(C)cc3C)=O)C2)=O)cc1CC CC(C)CC(CNC(C1CCOCC1)=O)NC(c1n[nH]cc1-c1ccccc1)=O c1(C(N2CC(SCC(=O)N(C)CC)C3(C2)CC3)=O)ccc2nnn(C)c2n1 N1(C(C)C)CCCC1C(N1CCCC1C(C)NC(c1cnnn1C1CC1)=O)=O N1(C(CC(=O)NC2CC2)=O)CC(NC(c2ccc(-c3nccs3)cc2)=O)C(O)C1 c12cc(ccc1OC)C(=O)NCC1CCCN(C1)C(=O)C2.C1(CC)CC1C(C)C N1(C(C(C)N(CC)CC)=O)CC(C)(C(=O)NCC(C)(C)C(C)(F)F)CC1(C)C N1(C(c2n[nH]c(=N)[nH]2)=O)CC2(CC2)CC1CNC(c1cnoc1C1CC1)=O c1(C(N2C(CNC(C(C(C)C)F)=O)CCC(C)(C)C2)=O)cc(F)c(N)cc1F c1(OC(CC)C(=O)N2CCC2Cn2cc(C3CCC3)nn2)ccccc1CO N1(C(c2cc(C)nc(Cl)c2N)=O)CCC2(CC1)OCCC2NC(C1CCSC1)=O c1(C(=O)NCCCOCCNC(c2c(N)sc(C)c2C)=O)cn2ncccc2n1 c1(N2CCC(C3N(C(c4cn(CC)nn4)=O)CCC3)C2)cc(C)c(C#N)c(C)n1 C1(OC)CC(CNC(=O)CC2CC(OC)C2)(NC(=O)C=C2CCOCC2)C1 N1(c2ccnc(C(C)C)n2)CC2CC(NC(C3CCCC4C3C4(F)F)=O)CC1C2 O=C1CS(=O)(=O)CC(C(N2CCC(CF)(NC(=O)Cc3nncs3)C2)=O)N1 C(=O)(CS(=O)(=O)CCO)N1CC2C(NC(CCC(=O)NCCNC(C)=O)=O)C2C1 N1(C(CC)=O)C2CCC1C(CNC(=O)C(c1cccc(C)c1F)O)C2 C1(C(N2CC(NC(C3CC3(F)F)=O)C(O)CC2)=O)CSC(c2ccccc2)=N1 C(c1ccc(OC(F)F)cc1)=CC(=O)OC(=O)C(F)=CCCC(=O)OC c1(C(=O)NCC2(NC(C(C)N(C)C)=O)CCOCC2)cc(Cl)ccc1O c1(OC)cccc(C(C)=CC(=O)NC23CCCN(C(=O)C(O)C4CC4)CC2C3)c1 CC1(C)C(C)(C(N2CCCCC(NC(C3CC(Cl)(Cl)C3)=O)C2)=O)C1(C)C c1(C(N2CC(NC(C(F)OC)=O)C2)=O)ccc(C(C)F)cc1 C=CCC(C)(C)CC(=O)NCCC(C)N(C(=O)CC1CCC(=O)N1)C CC(F)(F)CCC(=O)NN1CCCC1C(=O)NC12CC=CC(C1)OC2 C12(NC(c3cscc3F)=O)CCC(CC1NC(C1(c3ccc(F)cc3)CC1)=O)C2 c1(C(N(C(C(=O)NCc2ccc(CC)cn2)C)CC)=O)cc(C)c(C)cn1 N1(C(c2nn(C)c(Cl)c2Cl)=O)CCOc2ccc(Cl)cc2C1 C1(CCC(=O)NC2CC(CCF)C2)CCCCN(C(C2CCCC2C2CC2)=O)C1 S(=O)(=O)(c1ccc(COC(C)(C)C)c(F)c1)N(C)CC.C12CCCC(C1)CCN2 C1(n2cc(C=CC)nn2)CC2CCC1(NC(c1cnc(C(F)(F)F)cn1)=O)C2 S(=O)(=O)(c1cccc(Br)c1C#N)N(c1ccc(C(N2CC(C)OCC2)=O)cc1)C1CC1 C(=O)(CC(C)(C)CC(F)F)N1CCC(CN=c2[nH]nc(C(C)C)o2)(C)C1 C(C(CC(=O)N1CCC(N(C)C)C1C)C1CCC1)NC(CCc1onc(C)n1)=O C1(N(C(C(C)NC(CC)=O)=O)CCC(=O)N2CCCC2)CCC(C)(C)C1 C1(=CC(=O)NC(C(CO)NC(C(C(C)C)OC)=O)C)C2CC3CC(C2)CC1C3 CC1(NC(=O)CCc2cnco2)CCCN(C(C2COC(=O)N2)=O)C1 N1(C(C(C)OCC2CC2)=O)C(C(=O)N(C)CCC2CCOCC2)CCC12CC2 C(CC(CC)C(=O)NCC1(O)CN(C(C2CCC=CCCC2)=O)C1)=CC c1(NC(=O)NC(c2ccccc2NS(C)(=O)=O)C)c(F)ccc(Br)c1F C1(C(N2CCCC(CCNC(CC3CC(C)C3)=O)C2)=O)CCc2ccccc2O1 C=CC1OCCC1C(N1CC(C)(OCC(=O)NC2CCCC2(F)F)C1)=O Cc1cccc(C)c1C(O)C(=O)NC(CC(C)(C)C)c1cccnc1 C1(C(=O)NCCOC(CC)(C)C)CCCCN1C(C1(C)CCCS1)=O N1(CC)CCC1C(=O)N(C(C)CN(C(=O)C(C)N(C)C(C)=O)C)C Cc1nc(C)c(CC(=O)NC(CNC(c2cc(-c3ccccn3)ns2)=O)CO)s1 Cc1ccc(C(=O)NC(C)CNC(=O)C(F)(F)c2nccs2)cc1N C1(NC(c2c(CC)non2)=O)CCCC12CCN(C(c1cc(Cl)ccn1)=O)CC2 C=CCCCCCCC(=O)N1CCSCC1CCNC(c1cnc(O)n1C)=O n1(CC)c(C(=O)NCC2CC2NC(C2CC3(CC3)CO2)=O)cnc1O c1(C(=O)NC2(C3N(C(CC(CC)O)=O)CCCC3)CC2)c(Cl)ccc(F)c1C c1(C(C(=O)NC(CC)CN(C)C(C2(CF)CC2)=O)=O)cnn(C)c1 C#Cc1ccc(C(=O)NCCCN(C(c2cc(C)c(CO)cn2)=O)C2CC2)nc1 C1(CC)CN(C(c2cncc(C)n2)=O)CCN1C(c1ccc(C(C)(F)F)nc1)=O N1(C(c2cc(COC)[nH]n2)=O)CCCC(CCO)CC1.C1C(O)CC(=O)N1 C1(NC(C(C)S(N)(=O)=O)=O)CN(C(c2c(N)cc(F)cc2F)=O)CC2(CCC2)C1 c1(OCC)ccc(OCC(=O)NC2CN(C(=O)CC3CC34CC4)C2)cc1 c1(-c2ccccc2)c[nH]c2ccc(F)cc12.CCN=C(NCCCC1(C#N)CC1)N c1(Cc2cn(CC(CCNC(CCCCC)=O)F)nn2)cc(NC)ncc1Cl CCC(C)(CNC(C1COCCO1)=O)NC(=O)Cn1ccc(C(F)(F)F)n1 C#Cc1cc(C(N2CC(C)(CCC(N3CCC(OC)C3(C)C)=O)C2)=O)ccc1C N1(C(C(CC)Sc2ccccc2)=O)CC2(CCC(NC(=O)COCCF)CC2)C1 C1(CC)CN(C(=O)C(C)(CSC)NC(c2cnn(C(F)F)c2)=O)CCO1 c1(C(N2CC(CC(C)NC(=O)CCCC3CC3)C2)=O)ccsc1S(N)(=O)=O C(=O)(C1=COCCC1)N1C(C(=O)NCCC(C)O)CCC1C c1(C(N(C2CCN(C(=O)CC3(CSC)CC3)CC2)CC)=O)sc(C#N)cc1C CCC(O)C(F)(F)C(=O)NC(c1nccc(C)n1)C1CC1 C1(NC(=O)CN2CCCCC2)CC2CC1CN(C(c1ncc[nH]c1=O)=O)C2 O=C1CC(CN(CCCc2nn[nH]n2)C2CC2)C2(CCOCC2)C1 c1(C(C)NC(c2c(Br)ncc(C)c2)c2nnnn2C)cc2cnccc2o1 C1(O)(CN(C(C(CC)C)=O)C)CCN(C(c2ccccc2-n2cccn2)=O)CC1 c1(C(N2CC(C)C(CNC(=O)C=CBr)CC2)=O)ccc2nc(O)oc2c1 N1(C(c2cnc(C)o2)=O)CC(C(=O)NCCC(F)(F)CO)CC(C)(C)C1 c1(C(=O)NC2CCC(NC(c3nc(C)n(C)c3)=O)CC2)cccc(N)c1C(F)F Cc1[nH]c(-c2ccccc2)c(C)c1CN1CCC(CC(N2CCCC2)=O)C1 c1(OC)cc(C(N2CCCC2C(C)NC(=O)C(C)CF)=O)ncc1Br c1(CC(=O)NC2(C)CN(C(=O)CCCCC3CC3)C2)ccc2n[nH]cc2c1 C1(CN(C(c2ccc(C)n2C)=O)C)CN(C(c2ncsc2C2CC2)=O)CC12CC2 c1(C(N2CCCC(n3cc(C4(O)CCOC4)nn3)C2)=O)ccc2cncn2c1 c1(OC)nc(C(=O)NC23CC(C2)N(C(c2ccnn2CCF)=O)C3)cc(O)n1 C(=O)(N=c1ccn(CCF)[nH]1)C(N1CCN(CCCCC(=O)OC)CC1)=O C(=O)(CC(O)CC1CC1)NCC1C(NC(CCc2cn(C)nc2)=O)C1 C(=O)(C1CCc2nccn21)N1C(CCNC(C=CC(=O)N(C)C)=O)COCC1 CC1CCOCC1C(=O)NC(C1(O)CCCCC1)C(=O)NCCc1ncon1 CCCC(C(=O)OC)C(=O)N(CCCNC(c1cccc(C(C)(C)C)n1)=O)C(C)C C(=O)(C(C)CS(C)(=O)=O)NC(C(C)C)CCN(C(=O)CS(=O)(=O)NC(C)(C)C)C c1(OC)ccc(C=CC(N2CCCN(C(C3CCN(C)C3)=O)CC2)=O)cc1F CC(C)CCCC(=O)NC1CCN(C(=O)CCc2cnn(C)n2)C(C)C1 C1(C(=O)NC2CCCN(c3nc(C)c(C#N)cc3)C2C)CCCC2(C1)CC2(F)F c1(N(C)C)cncc(C(N2CCOC(CNC(=O)COCCF)C2)=O)n1 c1(NC(CC(C)O)C)ccncc1S(=O)(=O)NCC(C1CCCCC1)(C)C C1(NC(c2cc(Br)co2)=O)C=CCN(C(=O)Cn2cc(CO)nn2)C1 C=CCCCCCCCCC(=O)NC1CS(=O)(=O)CC1NC(C1CC(O)C1)=O c1(CNC(C(C)N(C)C(C2(C)COCCO2)=O)=O)cnc(O)c(F)c1 c1(C(N2CC(C)(NC(CCC(C)SC)=O)C2)=O)[nH]c2c(F)cc(F)cc2c1C S(=O)(=O)(c1ccc(C(C)(C)C(=O)NCCn2cc(C3(C)COC3)nn2)cc1)NC c1(OC)ccc(C(N2CC(N(C(=O)CCOC3CCC3)C)C(O)C2)=O)c(N)c1F Cc1cc2c(C(=O)NCCC3CCCCN3C(=O)C(C)N3CCC3)cccc2o1 CC1=C(C(=O)NCC2C(CNC(c3oc(CO)nc3C)=O)C2(F)F)SCCO1 c1(OC)ccccc1CC(=O)N(CCNC(c1cnn(C)c1C1CC1)=O)C(C)C c1(CC)nn(C)c(C(=O)NOCCCn2cnnc2C2CC2)c1Cl S(=O)(=O)(c1ccc(C(=O)NCCCNC(=O)C(C#N)C(C)C)o1)NC N1(C(CCC(C)C)=O)CCCC12CCCN(C(=O)CC1=NNC(=O)C1)C2 CC(C)C(O)CC(=O)N1CCN(C(c2ccc(C(F)F)cn2)=O)C(CCO)C1 Cc1cc2[nH]c(=O)c(C(N3CCN(C(C4SCCCS4)=O)CC3CF)=O)cn2n1 c1(OC)ccccc1SCC(C)CNC(=O)C(O)CCn1nc(C)cc1C CCC(CO)(C(=O)N(C(C)C(=O)NCC1CCCSC1)C1CC1)OC C1(NC(CN(CCC)C)=O)CC2CN(C(c3ccc(C)cc3SC)=O)CC12.CN C1(C(=O)NCc2c(C)snn2)CC(O)CN1C(=O)Cc1cn(C(C)(C)C)nn1 C1(NC(C2C(C)C2C)=O)(CF)CCN(C(=O)C(Cc2ccccc2F)N(C)C)C1 C(=O)(CC(C)(C)NC)NCC(CNC(C=CCOC)=O)OC.CC=C N1(C(CCCC(C)NC(C(COC)(C)O)=O)=O)Cc2cccc(O)c2C1 C(CCCCC(=O)NCC(N1CC=CC1)=O)n1cc(CC(C(C)(C)C)O)nn1 c1(NC(C)=O)sc(Cl)cc1C(=O)NC1CCC1NC(c1cncnc1C)=O C(CC1CC1)(C(=O)N1OC2CCC1CC2)NC(c1ccc2nccn2c1)=O c1(NC(C2(C)N(C(=O)OC(C)(C)C)CC2)=O)ccc(NC2(C)CC2)c(F)c1 C1(F)(CNC(Cc2c(CC)cccc2)=O)CCCN(C(=O)Cc2cnc(C)[nH]2)C1 C1(C(N2CCC(F)(C(=O)NC)C2)=O)CC2CN(C(=O)CC(=O)NC3CC3)CC2C1 C1CC(C(C)C)N1.C12CC(C)N(C1)C(=O)NC2.CC(C)CC(=O)OC(C)(C)C C12(C(N3CC(C)C(C(=O)NCC(C)(C)C4CC4)C3)=O)CCC(CC1F)C2 N1(C(COC)=O)CCC(C2CCCN(C(=O)CC(C)CC(C)(C)C)C2)CC1 c1(N(C2CCS(=O)(=O)C2)Cc2cccc(C)n2)ccnc2c1cnn2C C12(CNC(Cn3ncc(C)c3)=O)CCC1CCN2C(=O)CCn1cccnc1=O C1(O)(C(C)NC(c2c(C)noc2C)=O)CCN(C(=O)C(C(C)C)C2CCC2)CC1 C(=O)(C1=CCC(C)(C)CC1)NC(CNC(C(C(C)C)OCC(C)C)=O)C c1(C(N2CC(NC(C3(C)CC=CCO3)=O)C(O)C2)=O)cncc(N)n1 N1(C(C2(C(N)=O)CC2)=O)CCC(C(O)CNC(c2cscn2)=O)CC1 Cc1cc(C(=O)NCCCN(C)C(c2ccn(C)n2)=O)[nH]c1C#N c1(C(C(N2C(CNCc3c(C)cccc3)COCC2)=O)=O)ccc(F)c(C)c1 c1(C(=O)NC)ccc(C(=O)NC2CN(C(c3ccnc(S)c3)=O)CC2C)cc1F c1(C(C)=O)cc(C(=O)N(C2CC(NC(=O)CC3CC4CC4C3)C2)C)c(C)o1 C1(NC(C2C(C)CN2C(C2CCCC2F)=O)=O)CCn2nnnc2C1 c1(CC(N2CCC(C(C)(C)NC(c3cc(C)no3)=O)C2)=O)cncc(Br)c1 C1(C(=O)OC)CCCCCCN1C(=O)C(C)(C)C N1(C(C2(COC)CCOC2)=O)CCCC(CN(C)C(c2[nH]ccc2C)=O)C1 c1(C(=O)Nc2ncc(Br)c(C)c2I)cc2c(F)c(F)ccc2s1 CC#CCC(C(=O)NCC(C)(O)CC)NC(c1cc(C(C)=O)c[nH]1)=O N1(C(C(COCC)NC(=O)C=NOC)=O)CCN(C)CC1CO O=C1CC(=O)CC(C(=O)NC(C(=O)NC2CCN(CCCO)C2)c2ccoc2)C1 c1(C(N2CCC(O)(CNC(CC=C=C)=O)C2)=O)cc(C)c(C#N)c(C)c1 C1(CCNC(C2C(C)N(C)CC2)=O)CN(C(=O)C#CC(C)(C)C)CCS1(=O)=O c1(OC)ccc([N+](=O)[O-])c(C(N2CCCC(NC(=O)C(C)C(C)C)C(F)C2)=O)c1 c1(CNC(c2c(C)cc(C)o2)=O)nc(CNC(=O)C(C)N2CCC2)cc(O)n1 c1(N(C2CCN(C(CCc3cnn(C)n3)=O)C2)CCO)ncnc(Cl)c1F O=C(N=c1nc(-c2cccc(Cl)c2)[nH]s1)NC(C(F)F)C(F)F C(=O)(CCCN=c1ccc(S(=O)(=O)N2CCCC(CC3CC3)C2)c[nH]1)NC N1(C(Cc2nnc(C)o2)=O)CCC(CF)(NC(c2cc(CN(C)C)on2)=O)C1 c1(C(=O)NCC(CO)NC(C(C)c2cccs2)=O)cc(Cl)ccc1N CC1CC(C(N2CC=CC(NC(=O)C(C(C)(C)C)C3CCC3)C2)=O)CC(C)O1 Cn1ncc2ncnc(N3CCCC34CN(C(c3ncsc3Br)=O)C4)c12 C(C(=O)N1CCCC1CNC(c1cnc(-c2cnccn2)s1)=O)(C(C)(C)C)SC N1(C(C(CCC)F)=O)CC=C(C(=O)N2CCC(C)(C(=O)OC)CC2)C1 C12(C(=O)NCC)CCC(NC(c3cc(Br)ccc3F)=O)(CC1)CC2 c1(N2CCC(c3cc(C)[nH]n3)C2)nc(NCc2scnc2C)c2ncn(C)c2n1 c1(NC(C2CC(O)CN2C(C2(F)CCC2)=O)=O)cccnc1C(F)(F)F c1(CNC(C(C)(C)OC)=O)cccc(CN(C)Cc2nncs2)c1 c1(C(=O)NCC2N(C(c3nccc(COC)c3)=O)CC2)cc(SC)ccc1C C(=O)(CCS(=O)(=O)Nc1cccc(CO)c1)N(C1CC(NC(CC(C)O)=O)C1)C N1(C(c2nc(C(=O)OC)oc2)=O)CC(CNC(c2ccnc(O)c2)=O)C(O)C1 CC(CNC(C1CCS1(=O)=O)=O)CC(=O)NCC1(C)CC(F)(F)C1 C(=O)(CC1=CCN(C(c2ccc(C)cc2F)=O)CC1)N1CC(OCC#C)C1 n1(CC(=O)N(CCCNC(=O)C(C)CCOC)CC)cccc(N)c1=O C1(CCOC)(NC(c2cn(CCC)nc2)=O)CCN(C(c2cccs2)=O)C1 c1(N2C(C)CC(C(C)(C)C)CC2)nc(Cl)nc2cccc(F)c12 N1(C(CCC(C)O)=O)CC2CC1CN(C(c1n[nH]c(C(C)(C)C)n1)=O)C2 c1(C(=O)NC2CN(C(=O)CC3(O)CCC3)CCC2F)c(F)cccc1[N+](=O)[O-] N1(C(CCc2cccc(OCC)c2)=O)CC2(C1)CN(C(c1cncc(C)c1)=O)C2 N1(C(CC)CC)CC(C(N2CC3CC3(NC(C3NC(=O)C4CC34)=O)C2)=O)CC1=O CCC(C)(C)C(O)C(=O)NCC(C(N1CC(CO)CC(C)(C)C1)=O)OC CC1CC(C(=O)NCC2(C(N)=O)CN(C(=O)CP(C)(C)=O)C2)CCN1C c1(CC)oc2ccccc2c1C(=O)NC1CC2CN(C(=O)C=C(C)C)CC12 c1(C(=O)NC2CCC(CNC(C=CC=CC)=O)C2)cc2ncccc2o1 N1(C(C2CCC(CCCC)C2)C(=O)NCC=C)CC2OCCN(C)C2C1 c1(CCN=C(NCC(C)(CO)N2CCC2)NCC2CCC2)nnc2c(=O)[nH]ccn12 C1(C(=O)NCC(CN(C(=O)C(C)C(C)C)CC)(C)C)CCCC(C#N)C1 C(=O)(CCCC(=O)N(CCNC(=O)C(C)C1(O)CCC1)C(C)C)NCCC N1(C(CC(COC)C)=O)CCOCC(CNC(c2cnoc2)=O)C1 N1(C(c2[nH]cc(C)c2C)=O)CCC2(CC2)CC1C(=O)NCCOCCF c1(C(N2CCC(C)(NC(C(Br)=C(C)C)=O)CC2)=O)cc(Cl)c(F)cc1O C1(CNC(C2CC(=O)N2)=O)CC2COCC2N1C(=O)CCCCF N1(C(C(CC(C)C)C)=O)CC2CCC1C(CNC(C1C(F)(F)C13CCC3)=O)C2 C1(CCC#C)CCCN(C(=O)CCC(C)NC(=O)CCN(C)C)C1 C1(OCCNC(COCCC=C)=O)CC12CCN(C(=O)C=CCOC)CC2 C1(C(=O)NC(C(C)NC(CC2CCN(C(C)C)CC2)=O)(C)C)CC2(CCCC2)C1 C#Cc1ccc(CNC2CCN(C(c3c(O)cccc3Br)=O)C2)cc1 CC1(C(N2CC3CCC3(CNC(c3cccnn3)=O)C2)=O)CCCS1(=O)=O N1(C(CCOCC(C)C)=O)CC2CC1CC2NC(c1ccc(Cl)s1)=O Cc1c(Br)ccc(N(CCCCN(C)C(c2cnn3ncccc23)=O)C)c1[N+](=O)[O-] C1(CC=C)(C(=O)NC2(C(C)O)CC2)CCN(C(C2CC2C(C)C)=O)C1 C1(COC)(CNC(=O)CSC(F)F)CCCN1c1ncccn1 c1(C(=O)NCCN(C(C2C(=C)CC2)=O)CCC)cccc2c(C)cccc12 N1(C(=O)Nc2ccc(C)c(C(=O)NC3CC3)c2)CCC2(CCCN2C)C1 c1(CC(C)C(=O)NC2(C)CCN(C(C3(O)CCSC3)=O)C2)ccc(O)c(O)c1 N1(C(c2n(C)nnc2)=O)CC2CC1CCC2NC(C1CCS(=O)(=O)N1)=O C(CC(O)C(=O)NCC1(n2cc(C3(C4CC4)CC3)nn2)CC1)SC C1(C(=O)NCCc2c(C)ccnc2)CC(C)CN(C(C2CCS(=O)CC2)=O)C1 CCC(CC(=O)NCC1(CNC(c2conc2C(C)(C)C)=O)CCCC1)C(C)C n1(C(C)C)nc(C(=O)N(C)CCn2ccnn2)c(Br)n1 C1=C(CN=c2[nH]c3c(c(=NCc4cc(C5CC5)no4)[nH]2)CCC3)CCCCC1 N1(C(=O)CCC2(NC(C34CCC(C3)C4)=O)CCC2)CCC12CCSCC2 CC1(C(=O)NCC(O)C(=O)NCC2CC23CCCCC3)CCC2CC2C1 c1(N2CCC(CCNC(C3CC(=C)C3)=O)C2)nc2cc(F)ccc2o1 c1(CCCC(=O)NCCC2(O)CN(C(C3CCCC34CC4)=O)C2)ccc(Cl)cc1 C12(CNC(c3c(C)scc3)=O)COC(CNC(=O)CCOC(C)CC(C)C)(C1)C2 C1(C(C(=O)NCC2CCCO2)N(CCCC#C)C2CC2)CC2C=CC1C2 CCC(C)(C)CC(=O)N(CC(N1CCC(O)(C(N)=O)C1)=O)CC(C)C N1(C(COCCCC)=O)CC(NC(=O)C2=NOCC2)C(C(F)(F)F)C1 c1(C(N2CC3(C(NC(C4C(CCC)C4)=O)CC3)C2)=O)cc(F)c2cn[nH]c2c1 c1(C(N(C(CNC(c2cc(C)c(N)cc2)=O)C2CC2)C)=O)cc2ccccc2o1 c1(C(=O)NC(CNC(C(C(C)C)NC(=O)OCC)=O)C)cc([N+](=O)[O-])c(C)s1 C1(C2CCOCC2)(C(N2CCCC(N(C(=O)CSCC(N)=O)C)C2)=O)CC1 [N-]=[N+]=NC1CCC(C(=O)NC2CC(F)CN(C(c3cccc[n+]3[O-])=O)C2)CC1 C(=O)(C1=NOC(C)C1)N(CCN(C(C(CCC)c1ccccc1)=O)CC)CC Cc1ncnc(C)c1C(N1CCC(NC(=O)C(c2ccc(Cl)cc2)CO)C1)=O C1(F)(C(=O)NCCCC(C)NC(CN(S(CC)(=O)=O)C)=O)CCCOC1 c1(C(C(=O)NC(C)(C)C)N(C2CCOC2)C)cc(Cl)cs1 CC(CC(=O)N1CCN(C(=O)COC2CC2)CC1C1CCC1)C(C)(C)C C(C1c2ccsc2CCN1C(c1sc(=N)[nH]c1C)=O)NC(CCC=C=C)=O C1(NC(=O)COC(F)F)CC12CCN(C(c1cccc(F)c1Br)=O)CC2 CCCCCC(O)C(=O)N1CC2CCC1CN2C(=O)CC1CC2CC2C1 Cc1ccc2nc(CSC3N(C(C4C5CCC4CNC5)=O)CC(C)(C)CC3)cn2c1 N1(C(c2n(CCC)ccc2)=O)CCOC(CNC(C2CCCC(C(N)=O)C2)=O)C1 c1(C(N2CC(NC(COC3C(CC)CCCC3)=O)(CO)C2)=O)cc(O)nc(O)c1 c1(C(=O)NC2C(CNC(CN(C)CC)=O)C2)ccc(Cl)c(Br)c1F C(=O)(C1=CCCCO1)NCC1CN(C(c2ccc(NC)cn2)=O)CC1O C1(NC(C(C)CC2CCC2)=O)CCCCN(C(c2ccccc2C(C)(F)F)=O)C1 C1(C(C)C)COCCN(C(=O)N(c2ccc(Oc3ccc(Cl)cc3)cc2)C2CC2)C1 N1(Cc2c(NS(C)(=O)=O)cccc2)CCOC2(CCCNC2)C1 C(C(C(=O)N1CCCC1CCNC(=O)C(C)(F)c1ccon1)OC)OC C(CN=c1nc(N2CCC(SC(F)F)C2)c2c([nH]1)CCOC2)N(CCCOC)C S(=O)(=O)(c1cc(NC(C2(CF)CC23CCOCC3)=O)ccc1OC)NC N1(C(C2CN(C(=O)NC)C2)=O)CC2(CC2)CC1CO.C12(C(=O)N)CC=CC(C1)OC2 c1(CCCCC(N2CC=CC(NC(=O)COC3CCC3)C2)=O)ccc(O)c(F)c1 C(=O)(C1=COCCO1)NCC1OCCN(C(CCNC(N)=O)=O)C1 C1(C(N2C(CO)CC(N(C)C)C2)=O)CCN(C(C2(N3CCCC3)CC2)=O)CCO1 C(=O)(C(C)(C)CC(F)F)N1CCC(N(C(=O)CC#N)CCC)C1 c1(COCC(CNC(=O)CN2CSCC2=O)O)ccccc1 c1(C(C(=O)NC(CN(C(COCCOCC)=O)CC)C)C)c(C)n[nH]c1C c1(C(N2CCC23CCC3)C(=O)NC(CC)(C)C)ccc(F)c2c1CCC2 N1(C(C(N2CCOCC2CCc2ccc(O)cc2)=O)=O)CCNCC1CF c1(OCC)nc(Cl)ccc1C(=O)NC1CCCN(C(=O)C=C(Cl)Cl)C1C c1(NC(=O)CCC2CC2(Cl)Cl)cccc(CNC(C2CNC(=O)N2)=O)c1 CC1(CO)CCN1C(C1(CNC(=O)C(C)(C)N2CCCC2)CC1)=O c1(C(=O)NC2C3(CNC(CS(C)(=O)=O)=O)CCC(C2)C3)ccc([N+](=O)[O-])cc1 N1(C(C(Cc2ccoc2)NC(C2CCC(F)(F)C2)=O)=O)CCCCCCC1 c1(OC(C)C)cccnc1C(=O)NCC(O)CCNC(c1ocnc1C1CC1)=O C(C(=O)N1CCCC1C1(NC(c2ccccc2NC(N)=O)=O)CC1)(C(C)C)OC Cc1ncc(C(N2CC(NC(C3CCC34CCC4)=O)CC2CO)=O)c(=N)[nH]1 C(C)(CCCCNC(=O)Cc1cccc(C(F)F)c1)NC(C(C)OCC#C)=O Cc1cc(C(N2CCCCC(NC(C3C(C)C3C)=O)C2)=O)cc(C)c1OC(F)F C=C(C)CC(C(=O)NCCC1(C)CC1(F)F)NC(=O)CCn1cncn1 c1(CCC(=O)NC(CC=C)CNC(=O)CC)ccc(S(=O)(=O)CC)cc1 N1(C(Cc2c(C)cccc2C)=O)CCCN(C(C2COCCC2(F)F)=O)CC1C CN1CCOCC1C(=O)NCC1CCC(NC(C2CCCC3CC23)=O)C1 C1(F)(C(=O)NCc2cc(C(N(CC)Cc3ccoc3)=O)sc2)C(C)(C)C1(C)C N1(C(C(C)(C)N(C)C)=O)CCC(C2CC(NC(c3nn(C)c(Cl)c3Cl)=O)C2)C1 Cc1ccc(C)c(OCC(N2CCCCC2COC(c2ccccn2)=O)=O)c1 C=CC(C(F)(F)F)NC(=O)C(c1ccccc1)NC(c1c(C)n[nH]c1C)=O C(=O)(CN=S(C)(C)=O)N1CCC(C(C)(C)NC(C2N(C)CCOC2)=O)C1 c1(SC)ccc([N+](=O)[O-])cc1C(=O)NC1CCOCC1NC(=O)C(F)CC1CC1 C1(CC(=O)N(C2(C(=O)NC(C)Cc3cnn(C)c3)CC2)C)CC(C)(C)CO1 c1(OC)cccc(C(O)C(N2CCC(Cc3cccc(C)c3)CC2)=O)c1 N(C(=NCCC1CCCCO1)NCC1(c2ccc(F)cc2)CC1)CCC(C)(C)O Cc1nn(C)c(C(F)(F)F)c1C(=O)NC(C)CC(C)NC(=O)CC(=O)NC1CC1 CC(CC(=O)NC1(C)CN(C(c2ccc(O)o2)=O)C1)C1CCCO1 N1(CCCc2onc(C)n2)Cc2ccccc2CC1CNC(C1CCS(=O)(=O)N1)=O c1(C(N(C2CN(C(C=CC(C)(C)SC)=O)C2)C)=O)cc(F)c2[nH]nnc2c1 C#Cc1ccc(C(=O)NCC2CC3CC3N2C(c2ccc(Br)cc2N)=O)nc1 Cc1nn(CC(=O)NCCC(C)(C)CNC(=O)C(C)(C)CO)cc1[N+](=O)[O-] c1(C(N2CC(NC(C(C)(C)CC#N)=O)C(C)(C)C2)=O)nccc2cccnc12 C(=O)(C1CCCc2nn(C)cc21)N1CC2CC(CN(C(C(CCC)C#N)=O)C2)C1 c1(C(=O)NCCN(C(=O)C(F)C2CCCC2)CC)cc(-c2cccnc2)no1 C(=O)(C#CC(C)(C)C(F)F)N1C(C)C(c2ccccc2)CCC1 c1(C(N(CC(C)NC(c2cnn(CC(F)F)c2)=O)C)=O)cc([N+](=O)[O-])n[nH]1 c1(CNC(=O)Cc2ccoc2)ccsc1C(=O)NCCn1cnnn1 C1(CCCCNC(C23CC(C)(C2)C3)=O)CCCN(C(=O)CCn2ccnc2)C1 C1(OC2CCN(C(C(=O)NCCOC(C)C)=O)C2)CCCC1(F)F c1(SC)ccsc1C(=O)NC1CC(N(C(=O)C=Cc2ccsc2)C)C1 N1(C(c2cc(OC)ns2)=O)CCN(C(c2ccc3cccnn23)=O)CC2(CC2)C1 C1(C(NOCC=CC)=O)CN(C(=O)C(OCC)OCC)CCN1C c1(C(C)NC(=O)CCCCNC(=O)COCCN(C)C)ncc(F)cc1F N1(C(CC(=O)OC)=O)CCc2cc(CC(=O)Nc3ccc(O)cn3)ccc2C1 N1(C(c2c(CC)n(Cc3ccccc3)nc2)=O)CCN(C(=O)C(C)O)C(C)C1 N1(C(C(C)C(C)(F)F)=O)C2CCC1C(C)C(NC(=O)COCCc1cccs1)C2 CC(F)(F)CC(=O)N1CCOCC1CC(=O)NCC1CCCOCC1 c1(C(N2C3CC(NC(CCC)=O)CC2CC3)=O)cc2cc(O)ccc2nc1C c1(C(=O)NC2(c3c(C)cccc3)COC2)cc(F)cc2ccoc12 C(=O)(CCCC(=O)NC1COCC1NC(=O)Cc1cscc1Br)N(C)C C1(NC(C(C)SCCCC)=O)CCN(C(c2scc(C)c2C)=O)C1C c1(NC(N(C)CC2CCN(c3cc(CC)ncn3)CC2)=O)ccc(OC)c(C)c1 c1(CC(=O)N(C(C)(C)CN)CC)c(C)nc2nc(=N)[nH]n2c1C N1(S(CCOC)(=O)=O)CCN(C(c2cc(Cl)cc(Cl)c2)=O)C2(CC2)C1 CC(CCCC(=O)N(C1CC2CC2C1)C)NC(C1CC1(C)C(F)F)=O N1(C(Cc2c(C)con2)=O)CC(CNC(n2nc(C)oc2=O)=O)OC2(CCC2)C1 c1(CN(C(C(C)OCCC(C)C)=O)CCNC(=O)C=CCO)ccccc1 C1(C2CCCN(C(C34CCC(CC3)C4)=O)C2)(NC(C(CCC)N(C)C)=O)CC1 C1(CNC(C(C2CCOCC2)OC)=O)CC2CN(C(=O)C(C)(C)C(N)=O)CC12 c1(C(N(CCCCCNC(c2c(CC)csc2)=O)C)=O)c[nH]c2ccc(Cl)cc12 C1(C(=O)NC(C2CCCCC2)CNC(C=C(CCC)C)=O)CCCN1CCOC Cc1cc(C(=O)NCC(F)CNC(=O)CNC(=O)C=Cc2ccco2)ncc1Cl C1(C)(CNC(C2(CC)CCC2)=O)CCCN1C(=O)CCOCC1CCCO1 N1(C(c2ccc(F)cn2)C(=O)NCCCSCC)CCc2cc(Cl)ccc21 C1(CCCC(=O)NCC2(F)CC(CNC(C(C)OCC=C)=O)C2)CCCC(=O)N1 C(C(O)CC(=O)NCC12CCC(CC1)O2)NC(CC(C)N(C)C)=O C1(C(N(CCC=C)CC(=C)C)=O)CN(C(c2cc(C3CC3)ccn2)=O)CCC1(C)C c1(C(=O)NC(C2(O)CN(C(C3(C#N)CCC3)=O)C2)C)[nH]nc([N+](=O)[O-])c1Cl N1(C(CCCC2(C)N=N2)=O)CCC(O)C(NC(=O)CCC2CCC2)C1 C1(CC(=O)NC(CNC(c2cc3ccsc3s2)=O)C2CCC2)CC2(CCC2)CO1 c1(O)cnc2c(c1)CCCC2.n1(CCC)ncc(C)c1NC(c1ccc(C(C)C)cc1)=O n1(CC(=O)N(CCCCN(C(C2CCCC(C)C2)=O)C)C)ccc([N+](=O)[O-])n1 N1(C(C(n2cc(C3(c4ccccc4)CC3)nn2)C)=O)CCCC2(C=CCO2)C1 Cc1nnc2n1C(C(=O)NCC(C)NC(C1(n3cnnn3)CCCCC1)=O)CC2 C(=O)(C1CCc2c[nH]nc21)N1CCN(C(=O)Cn2cncn2)CC1C1CC1 C1(CNC(c2cc(-c3nc(C)sc3)oc2)=O)CC(F)CN1C(=O)COC1CC1 N1(C(C(CC)N(C)C)=O)CCC(CNC(c2ncn(C)n2)=O)(COC)C1 c1(C(N(CCNC(CC(=O)NCC#C)=O)CCOC)=O)nc(Cl)c(CC)[nH]1 c1(OC)sc(C(=O)NC2(CNC(c3ncccc3N)=O)CCC2)cc1Br C1(NC(C(CC#C)NC(=O)CC2CCC(=O)CC2)=O)CCC12CCCC2 c1(C(=O)NC(c2cnn(C)c2)C(=O)NCc2cnc(C(C)C)[nH]2)c(Cl)cnn1C C(CC(C)C)(C(=O)NCC1CCCCC1C(N1CC(F)CC1CO)=O)OC c1(C(N(CCCCCNC(C(CC)(C)C)=O)C)=O)cnc2sc(C)c(C)n2c1=O C1(NC(c2c(C(C)(C)OC)[nH]cc2)=O)CCC(n2cc(C(C)(C)O)nn2)CC1 C1(CNC(c2ccoc2Cl)=O)CCCN(C(=O)C=Cc2ccc[nH]2)C1 N1(C(C2N(C)CC2)=O)CCN(C(C2(CC(F)F)CC2)=O)CC1C1CC1 CCCCC(C(=O)N1CC(F)(CNC(C2CCCSC2)=O)C1)C(C)C N1(C(CCNS(CC)(=O)=O)=O)CCC(CNC(=O)C(=CC2CCCCC2)F)CC1 C1(C(=O)NCC2C(NC(CN(CCOC)C)=O)CC2)(N(C)C)CCCC1 Cc1cn2cc(C(=O)NCC3CN(C(=O)CCC4CCOC4)C(C)(C)C3)sc2n1 C(=O)(CN=c1cc[nH]cc1)NCc1nccc(C(N2CCOCC(C)C2)=O)c1 CC1=CCCN(C(=NCCC2CCN(C)CC2)NCC2CCCCO2)C1 N1(C(CC2N(CC)C(=O)CC2)=O)CCC2(C1)CN(C(=O)Cc1cn(C)cn1)C2 N1(C(c2c(C)noc2)=O)CCCC2(CCCN(Cc3cc(F)ccc3F)C2)C1 C12(C(=O)NC(CN(C(CSCCOC)=O)C)C)CC(CC(C)O1)C2 C(C#CCN=c1nc(N2CCCC(C(=O)N(C)C)C2)c2c(ncn2CC)[nH]1)OC c1(CC)nn(C)c(CC)c1C(=O)NC(C)CN(C)C(c1ccn(C)c1)=O N1(C(C(CC)OC)=O)CCC(CCOC)(C(=O)NC2CCCC(OCF)C2)CC1 C1(C(=O)NC(CC(=O)NC)(C)C)CN(C(=O)C(C2CCCCC2)=O)CC1(F)F C1(C)(C(N(C2CCN(C(C(C)OCC#C)=O)CC2)CC)=O)COC(C)(C)CO1 N1(C(Cc2nc(NC(c3c(N(C)C)cccc3)=O)sc2)=O)CC2C(C1)C2(F)F Cc1ncsc1CC(=O)N(CCCNC(c1cnsn1)=O)Cc1ccccc1 C=CCC(CNC(=O)CCN(C(=O)C(C)NC(C)=O)CC)CC(C)C c1(CN(S(=O)(=O)CC2CCCOC2)C)cccc(OC2CCCC2)c1 N1(C(Cc2cc(OC)no2)=O)CC2CCC1C1CN(C(c3ccccc3O)=O)CC21 c1(C(=O)NCC(C)(CNC(=O)CCCNC(N)=O)OC)nccc2ncccc12 C1(CCC(=O)NC(C(=O)OC)(C)C2CC2)CCN(C(=O)C(C(C)C)NC=O)CC1 N1(C(CSCCNC(COCC(=C)C)=O)=O)CCC12CCOCC2 N1(C(COC(CC)CC)=O)CCOC2CN(C(C3COCC3(C)C)=O)CC12 N1(C(COCCCCC)=O)CC(O)(CNC(c2ncnn2C)=O)C1 CN1CCC(NC(=O)C=C2CCSCC2)C12CCCN(C(c1cnns1)=O)C2 N1(C(c2sc(CC)c(C)c2)C(=O)NC2COC2)CC2CCC1CN(C(C)=O)C2 C#CCC(C)(C)C(=O)NCC(C1CC1)N(C)C(c1cc2sccc2s1)=O N1(C(c2c(CC)nco2)=O)CC(N(C)C(c2cc(COC)no2)=O)C(O)C1 c1(C(N2CC3C(CNC(C(C(CC)O)C)=O)C3C2)=O)c(F)ccc(O)c1O c1(CC)ccnc(C(=O)NC(CC2CCCC2)C(=O)NC(C)Cc2cnc[nH]2)c1 C#CC1(C(=O)N(CC(CC)NC(=O)CCCNC(c2ccco2)=O)C)CCCC1 C(=O)(C1Cc2ccccc21)N1CC=C(CNC(c2c(CC)onc2)=O)CC1 Cc1nn(CC(=O)N(C)CCN(C(=O)COCC2CC2)C)c(=O)o1 N1(C(C2CCC(=O)NC2)=O)CC2(CCC2)CC1C(=O)NCCC(Cl)Cl C1(NC(=O)CCN2CCCCC2)CC(F)CN(C(C2Cc3cscc3C2)=O)C1 Cc1cc(Cl)c(C(=O)NC2(C)CCN(C(c3ncccc3F)=O)CC2)cc1C C1(CNC(C(C2CC2)SC)=O)CCN(C(=O)CNC(=O)CN(C)C)C12CC2 C1(NC(C(C2CCC(C)CC2)CC)=O)CN(C(=O)Cc2ccc(C)o2)CC12CC2 N1(C(c2c(CC)con2)=O)CCN(C(C2CC2Cl)=O)CC12CCC2 CC1=NOC(C)(CNC(=O)C(C)N(C(=O)Cc2ccon2)C)C1 Cn1nc(C(=O)Nc2ccc(I)cc2-c2nn[nH]n2)c(Cl)c1Cl C1(NC(COCC(=O)NC)=O)COCCC1NC(=O)C(F)CC1CCC1 C1(CNC(CCS(C)=O)=O)CN(C(=O)C#CC2CC2)C2COCC2O1 CCC(C)(C(=O)N(C1(C(=O)NCC(C)C#N)CC1)C)OC CCCCC(O)CC(=O)N(CCNC(C)=O)Cc1ccncc1OC C1(CNC(c2cc(CNC(C3C(C)CCO3)=O)sc2)=O)CCC(=O)NC1 S(=O)(=O)(c1ccc(C(=O)NC(c2nnc(O)n2C)C)cc1)NCC(C)O c1(OCC)nc(Cl)ccc1C(N1CC=CC1CNC(C1CCC(O)CC1)=O)=O Nc1cccc(Cl)c1CNCC(O)Cn1ccnn1 CCC(C(=O)Nc1ccc(NC(c2ccc(NC)cn2)=O)cc1C)C(C)C N1(C(CCOCCOC)=O)CC2C3CCC(C(NC(=O)C(O)P(C)(C)=O)C3)C2C1 Cc1cccnc1C=CC(=O)NCC1C(C)CCCN1C(c1coc(O)n1)=O N1(C(C(C)OCCC(C)C)=O)CC(C)(C(=O)NCC2(CF)CC2)CC1(C)C CC(C)(C)C(O)C(=O)N1CC(O)C(O)C1CNC(=O)C=C1CCC1 C1(N(C(c2c(C)snn2)=O)C)CCC2CN(C(C3CC(O)C3)=O)CC12 C(=O)(C(CCNC(C)=O)C(C)(C)C)OCC(CCCC)CC C=CC(CC)CC(=O)NC1CCOC(C(N2CC(OC(C)C)C2)=O)C1 CC1(C)Cc2cc(CN(c3cccc(-c4ccncc4)c3)C=O)ccc2O1 C1(N(C(C(F)=C(C)C)=O)C)CCCN(C(c2ccc(C3CCCO3)[nH]2)=O)C1 C1(C(N2CCC(C(C)(C)NC(C3COC(=O)C3)=O)C2)=O)CCN(S(N)(=O)=O)CC1 C(=O)(C(C)Cn1ccc(C)n1)NCCCN(C(CCC)=O)CC N1(OC(C2(NC(C=CCCC)=O)CC2)=O)CCCCCCC1C C1(NC(C2(C)CC2)=O)CCN(C2CCN(C(C3CC34CCCC4)=O)C2)CC1 N1(C(C2(C#N)CC2)=O)CCCN(C(c2cn3ccnc3s2)=O)CCC1 c1(COC)ccc(C(N2CC(CNC(=O)Cc3ccco3)C(C)C2)=O)cc1 c1(C(N(c2nnc(C3CN(C)C(=O)C3)n2CO)CC2CC2)=O)ccc(Br)c(F)c1F N1(C(c2c(C)n(C)nc2)=O)CC(NC(C2CCCC3(CC3)C2)=O)C2(CCCC2)C1 c1(C(=O)NCCC(C)NC(c2conc2C2(C)COC2)=O)ccc(C(F)F)cn1 C1(NC(C(c2ccc(F)cc2)C)=O)CCCN(CC2CC3CCC2O3)CC1 N#Cc1cc(C(=O)NCC2CCCN2C(=O)CCCn2cccn2)ccn1 C1(C(=O)NCC(C)C(=O)NC)(NC(COCCC=C)=O)CCOCC1 C1(CNC(C2ON=C(CC)C2)=O)COCCN(C(=O)CCc2cncc(O)c2)C1 c1(C(=O)NCC2CC(NC(C3C4CCCOC34)=O)CC2O)cc(Cl)nnc1O N1(C(C(C)O)=O)CC(O)(C2CCN(C(C3(C(F)F)CCCC3)=O)CC2)C1 Cc1onc(Cl)c1C(=O)NC(C)CCCNC(c1cc(C2(C)COC2)no1)=O C1(OC)CC2(C(=O)NC3CC3NC(=O)C(c3cncn3C)N(C)C)CC12 Cc1cccc(C(=O)NCCCCC2CN(C(C3CCCC34CC4)=O)C2)c1N CC(C)C(CO)CCNC(C1CC(F)CN1C(=O)C(c1ccnn1C)C)=O C1(C)(CNC(CS(CC)=O)=O)CC(F)(F)CN1C(=O)CCN(C)CCO C1(NC(c2c(C)nncc2)=O)CCC2(CCCN(C(c3ccc(Cl)cn3)=O)C2)C1 O=C(C#CC1CCCO1)NCCCOCCCNC(=O)C(c1cccc(F)c1)O N1(CCNC(C(CC)O)=O)CCC(NC(=O)CC2(C#N)CCC2)CC1 c1(C(C)C(=O)NC2CCN(C(=O)CSC(F)F)CC2)cc(F)cc(F)c1 C12(C(=O)NCC3CCCC(NC(=O)CCCN4CCCC4)C3)CCC(CO)(CC1)C2 c1(C(=O)NCCCCNC(C2N(CC)C(=O)CC2)=O)ccc(C)cc1C C#CC(CNC(=O)C(C1CCCO1)NC(=O)CC1CCN(C)CC1)C(C)C c1(OC)sccc1C(=O)NC1CCCC1NC(=O)CCN(S(C)(=O)=O)C c1(NC(C2CN(C(=O)CSC(F)F)CCO2)C)c(F)cccc1[N+](=O)[O-] c1(C(=O)NC2CC(CNC(c3c(C)coc3)=O)C2)cc(O)cc(F)c1F C(=O)(C1=CC2C=CC(C1)C2)NC1CCC(NC(c2cc(C)c(=O)n(C)c2)=O)CC1 CCC(CC)C(C(=O)NC(c1ccccc1)C)N1CC(CC)CC(C)C1 C=CC1OCCCC1C(=O)N(CCC(C)NC(c1cc(Br)cnc1C)=O)C C1(NC(C2CCC(NC(c3n(C)nc(O)c3)=O)CC2)=O)CCCC(O)CC1 Cc1cc(Cl)c(C(=O)N(CC(C)O)CCNC(c2cnc(S)[nH]2)=O)cc1F CCC(Cc1cn(-c2cccc(CC(N3CC=CCC3)=O)n2)nn1)C(=O)O Cc1ncccc1C(=O)NCC1CCN(C(=O)CSc2ccccc2)C1 c1(CCC=O)c[nH]c2cc(Cl)ccc12.C12(C(N(CCCN)C)=O)CC3CC1C2C3 N1(C(CNC(C(CC)C)=O)=O)CC(CNC(c2cnnc(C)c2)=O)C(F)(F)C1 c12ccc(cc1)OCC(=O)NC2.C(CCCn1cnnc1)N(C)CCO.C1CCO1 c1(COC)nc(C)ncc1C(=O)NCc1cn(C(C)C(=O)NC(C)(C)C)nn1 c1(C(=O)NCC2(CCNC(CCCC(C)C)=O)CC2)cc2n(n1)CC(C)NC2=O c1(C(=O)NCC(CNC(C(CC)CC)=O)(C)O)ccnc2cc(F)cnc12 C=CCC(C)(CC)C(=O)N1CC2(C1)CN(C(c1cnc(C3OCCO3)s1)=O)C2 C1(N(C(=O)C(=O)C(C)(C)C)C)CC2CCC(C1)N2C(=O)C=Cc1ccnn1C Cc1ccc(F)cc1C(N1CCCC(CC(=O)NCc2ncc(CO)[nH]2)C1)=O CN1CC(NC(=O)CCNC(=O)CC(C)(F)F)C(F)(F)C1 C1(NC(C(CC=CC)NC(C2CN(C)CCO2)=O)=O)CCCCC1(C)C C1(NC(C2CC2CNC(c2c(C)coc2C2CC2)=O)=O)CCC(C#N)CC1 N1(C(C2OCCN(C)C2=O)=O)CC(NC(C2(S(N)(=O)=O)CC2)=O)CC(C)(C)C1 N1(C(C(=O)NCC(=C)CCNC(C2(NC(C)=O)CC2)=O)=O)CCCC(C)C1 CCCCC(C)(F)C(=O)NCC1C2CC1N(C(=O)CCc1cnco1)C2 C(=O)(CCS(C)(=O)=O)NC(C(C)NC(C1(c2cccc(OC)c2)CCCC1)=O)C C12(NC(c3cc(OC)no3)=O)CCCC1CN(C(=O)C1=COCCC1)C2 S(=O)(=O)(c1ccc(NCC2CCCC(F)C2)c(F)c1)NCc1c(C)nns1 C1(CCNC(C2C(C)=CCS2)=O)CN(C(=O)CNC(=O)CN(C)C)CC(C)O1 c1(CC(=O)NCCNC(=O)CC2=CCCCC2)ccc(F)cc1[N+](=O)[O-] CC1(C)C(OCC(N2CCCC(C)(CN=c3[nH]nc(C(F)F)s3)C2)=O)CC1(F)F CCC(C)C(CC(=O)N(C)CC1CC1(F)F)NC(=O)C(O)C(C)(C)C C(CN=c1[nH]c2c(c(=NCC3(Br)CC3(F)F)[nH]1)CCCC2)c1cc(C)c(F)cc1 CC(C)(C)C1=NOC(C(=O)NCC2CCN(C(=O)Cn3cncn3)C2(C)C)C1 S(=O)(=O)(c1cnccc1N(C)Cc1ccco1)N(CC(C(C)C)OC)C c1(OC)cc(NC(c2ccc(CN3CCC(CO)C(O)C3)s2)=O)c(Br)cn1 c1(C(=O)NC2C(NC(C(CC)Oc3ccccc3)=O)C2)cc(C)c(C)cc1C N1(C(c2ccnc(C)c2O)=O)CCC(C2(NC(=O)CS(N)(=O)=O)CC2)C1 c1(C(=O)NC2C3CC(NC(CCC(CC)OC)=O)CC32)ccc2c(c1)OCO2 N1(C(C(C(C)C)O)=O)CCC2(COC(CNC(=O)Cc3csnn3)C2)C1 CCC(C)CC(C(=O)N(C)Cc1scnc1C)NC(=O)CCCC1CC1 c1(CC(=O)N(CCNC(C2(OC)CCCC2)=O)C2CC2)cc(F)ccc1F c1(SC(=O)OC2(c3cccnc3)CC2)ncnc2c1cnn2-c1ccccc1F c1(C(=O)NC(CC)CNC(=O)C(c2ccc(F)c(Cl)c2)C)cccc2c1OCC2 c1(C(=O)NC(C(C)NC(c2c(C)ccc(F)c2)=O)C)c(F)ccc2ccncc12 Cc1cc2cccc(C(N3CCN(CCF)CC3)C(=O)NCCSC3CC3)c2o1 S(=O)(=O)(c1cc(C)c(-c2ccno2)cc1C)N1CC(COC)OCC1 c1(C(N2CC3CN(C(c4nc(C)nn4C)=O)C3CC2)=O)cc2cc(F)ccc2o1 C=C=CCCC(=O)NOC(CC(C)C)C(=O)N(C)CC1CCCO1 C1(CNCc2c(C(=O)OC)[nH]cc2)COCCN(C(C2CN3CCC2CC3)=O)C1 S(=O)(=O)(c1ccc(C#N)c(NC2CCC(=O)NC2)c1)N1CCCC(CCC)C1 C1(NC(COCCOC)=O)CC2(C1)CC(NC(C1CCCOCC1)=O)C2 N1(C(CC(C)C)=O)CCCC1(C)CNC(=O)CCNC(=O)CC1CCCCC1O c1(C(N2CC(F)CC(NC(C(C)=C3CC3)=O)C2)=O)cccc(C2=CCOCC2)c1 C(=O)(C(C)S(C)(=O)=O)NC1(CO)CN(C(C(CC=CC)NC(C)=O)=O)C1 C1(NC(CC2CC(SC)C2)=O)CCCC1CN(C(=O)C(C)Cc1cnc[nH]1)C1CC1 c1(C(=O)OC)ccnc(C(=O)NC2CCC(NC(=O)CC3COCC3O)CC2)c1 Cc1cn2c(C(=O)NC3CN(C(=O)C(C)OCCC(C)C)C3)c(Cl)nc2s1 C12(C(N(C(CC)CC)C3CC3)=O)CC(C)(CN1C(c1ccc(Cl)cn1)=O)C2 CC1(CNC(C2CC(=C3CC3)C2)=O)CCCN1C(=O)CC1(C2CC2)CC1 C1(C#N)(C(=O)NCC2(CO)CCN(C(c3ccc(CC)s3)=O)C2)CC12CCCC2 N1(C(c2c(C)c(N)cnc2)=O)CCC(NC(=O)CC2C=NN(C)C2=O)C(C)(C)C1 N1(C(C(n2ccc(C)n2)C)=O)CCC2(CCN(C(c3conc3C)=O)CC2)C1 N(C1CN(c2ccncn2)Cc2ccccc21)C(C1CCc2nnc(O)n2C1)=O c1(C(=O)NC(C(=O)OC)CC2CCCCC2)cccc(-c2cn[nH]c2)n1 S(=O)(=O)(c1cccc(N(C)C)c1)N(CCC(C)C)Cc1ccc(Br)cc1 N1(C(COCCCC)=O)CCCC(C)(NC(=O)CC(C)(C)C#N)C1 Cc1ccc(C=CC(=O)N(CC(C)NC(C2(C)CCCS2(=O)=O)=O)C)nc1 C1(CNC(CN(C)C(N)=O)=O)CC(O)CN1C(c1cn(CC2CCCC2)cn1)=O Cc1c(NCC2CCC3(CC3)C2)ncnc1N1CCC(OCc2ccccc2)C1 C#CCCCCC(=O)NCC1CCCN(C(C2CC3(CC3)CO2)=O)CC1 c1(CC(=O)NC(CNC(c2cn(CC)nc2C)=O)C2CC2)c(N)nc(C)nc1O CC(CC(=O)NCC1(F)CCCN(C(C2CC(F)(F)CS2)=O)CC1)CC(C)(C)C C12CCCN(C1)C(=O)C(C(=O)OC)N2C(C1(c2cccnc2)CC1)=O.CC.OC Cc1nc2c(s1)CCCC2CN(C)C(=O)NCc1nc2cc(Cl)ccc2s1 C(=O)(CC(C)N(C(=O)CCc1cc(C)on1)C)NC(C#C)CC1CC1 N1(C(c2n(CC)nnc2C)=O)CC(C)C(NC(c2cc(F)c[nH]2)=O)C(C)C1 c1(C(N2CC3CC(C(=O)NC4CCC(C)(C)C4)(C2)C3)=O)ccc2cc[nH]c2n1 N1(C(C=CC(C)(C)SC)=O)CCCCC1C(=O)N(CC(C)(O)C1CC1)C C(CCCC(=O)N1CCC(c2nnc(S)o2)CC1)NC(N)=O C1(NC(CCC(CC)C)=O)CC2CCC1CC2NC(c1c(C(F)F)cccc1N)=O N1(C(C(C)(C)OCC)=O)CCC2(CCC(NC(c3ccc(C)n3C)=O)C2)CC1 C(=O)(C#CC1CCC1)N1CC(NC(CCCSc2ccc(CC)cc2)=O)C(C)C1 N1(C(C(CC)=CC)=O)CC2CCC2(NC(c2cc(C#N)c[nH]2)=O)C1 c1(NC(C2CCCN(C(c3cc(O)ncn3)=O)C2)=O)cnncc1Br C#CCCCCC(=O)N1CC(F)CC1CNC(C1OCCOC1C)=O c1(C(N2CCC(CCCCNC(CC(=O)NCC)=O)CC2)=O)c(F)cccc1Cl C=CCCC(C)C(C(=O)NCc1cccc(F)c1)N(C1CC2CC3C(C2)C13)C c1(C(N2C(CNC(c3conc3C3CCC3)=O)CC2)=O)cccc2c[nH]nc12 N1(C(C2N(C(C(C)CCN(C)C)=O)CC(=O)NC2)=O)CC(C)(C)OC(C)(C)C1 C1(C)(CNC(COCCCCCCCC)=O)CN(C(=O)CCOCC)C(C)(C)C1 C(=O)(C1OC(=O)c2ccccc21)NCC(CC)NC(=O)C(C)(C)OC(C)C C12(NC(=O)CCn3ccnn3)CCOCC1CN(C(=O)CCC1CC(F)(F)C1)C2 N1(C(C(N)=O)=O)CC23CCCCC2(C1)CN(C(c1cc(Cl)cc(Cl)n1)=O)C3 C1(C#N)(C(=O)NC2CCC(N(C(C(=O)NC(C)C)=O)C)CC2)CC12CCCC2 C1(OCC(C)C)CCN(C(N2CC(C)(C(C)C)C2)=O)C1 C1(C(N2CCCC(CC(=O)NC(c3ncccn3)CC)C2)=O)CC2(C1)CC(O)C2 C1(NC(C(c2ccc(-c3nn[nH]n3)cc2)C)=O)CCCC(C(C)(C)C)C1 C1(CC(=O)NC2(CCNC(C3C(C)C3)=O)CCCC2)CCCC(C)(C)O1 c1(COC)cc(Br)c(C(N2CCOCC2C2CC2)C(=O)NC2(C)CC2)s1 N1(C(C(CCC)C)=O)CCC(CC(N)=O)(NC(C2CC(F)C2)=O)CC1 c1(C(=O)OC)ccc2c(CNCc3cccc(NC4CCCO4)c3)csc2c1 C=C(Cl)C(C)(C)C(=O)NC1CN(C(C2(F)CC2c2ccccc2)=O)CC1C C1(CNC(c2n(CCCC)ncc2)=O)CN(C(c2ccnc(O)c2)=O)C(C)(C)C1 c1(C(N2CCS(=N)(=O)C(C)C2)C(=O)NCCC)cc(OC)c(OC)cc1Br c1(C(=O)NCC2CC(F)CN2C(C2CC23CCC3)=O)nccn2nccc12 N1(C(CSCC(C)C)=O)CCC2CN(C(=O)Cn3nnnc3C3CC3)CC2C1 c1(OCC(=O)NC2CCCC2CNC(C23CC(F)(C2)C3)=O)cccc([N+](=O)[O-])c1 N1(C(CCOCCOCC)=O)CC(OC)CC(NC(=O)CCN2CCCC2=O)C1 c1(C(N2CCC(NC(Cc3ncc(C)s3)=O)CC2C)=O)occ2c1CCOC2 CC(CCC(=O)NOC(N1CCN(C)CC1)c1cn(C2CC(O)C2)nn1)C(=O)O c1(CNCC23C(CN(C(=O)Cn4ccccc4=O)C2)C3)cc(F)cc(I)c1 C#Cc1ccc(C(N2CC(NC(c3ccc(Cl)nc3N)=O)CCC2C)=O)cc1 c1(C(=O)NCC2CN(C(C(C)C#N)=O)CC2C(F)(F)F)ccn(C)c(=O)c1 N1(C(C2(C=O)CC2)=O)CCCC(CN2CCN(C(=O)CP(C)(C)=O)CC2)C1.CO C(=O)(C(C(C)(C)C)OC)N(C(CN(C(c1nncc(OC)c1)=O)C)C)C C=C(Cl)CC(C(=O)NCc1cc(C2CC2)no1)NC(C1CCC1CC(C)(C)C)=O C#Cc1ccc(F)c(C(=O)NCC(CC(F)(F)F)NC(C2CC(C(F)F)C2)=O)c1 C1(NC(C(C)(C)S(C)(=O)=O)=O)CCN(C(c2cscn2)=O)CCC1(F)F CCCCCC(CNC(=O)Cc1ncc(C)s1)NC(=O)CN1CCCC1=O C(c1cccc(F)c1Cl)=CC(N1C2C(NC(C(C)C3CCCO3)=O)C(C2)C1)=O c1(C(N(CC(=O)NCCCC2C=NNC2=O)CC)=O)cnc(O)c(C)c1 C(=O)(CCCCOCC1CCCC(C)O1)OC N1(C(C2CC(OC)CN2C(c2cc(C#N)cs2)=O)=O)CCCC(C)(O)C1 C1(NC(C(C)O)=O)CC2CCC1CN(C(c1ccnc(N(C)CC3CC3)c1)=O)C2 C1(O)(CC(=O)NCCN(c2ncc(Cl)c(O)n2)CCC)CCCN(C)C1 c1(-n2ncc(C(N3CC(NC(=O)CN4CC5CC5C4)C3)=O)n2)cccc(Br)c1 c1(C(=O)NCC23CC2CN(C(c2cc(Cl)cnn2)=O)C3)cc(F)c(CO)c(F)c1 Cc1cc(CC(=O)NCC2CC(F)(CNC(=O)C(C3CCCCC3)O)C2)no1 N1(C(C2(CC)CC2(F)F)=O)CC2(C1)CN(C(c1cccnc1C1CC1)=O)CCO2 c1(CN(C(C)C(=O)NC2CCCCC2)CC)ccccc1[N+](=O)[O-].C1CC(=O)O1 c1(CC)nncn1NC(=O)C1CC(NC(c2ccc(C)cc2O)=O)C1(C)C O=C(C1=C(Cl)CCCC1)NC1CC(O)CN(C(c2cc(F)n[nH]2)=O)C1 c1(OC)ccc(Cl)cc1C(=O)NCC1(O)CN(C(c2cc(O)nc(O)n2)=O)C1 C(=O)(C1=CC2CCC=CCCC12)N(C(C)CCNC(=O)CCc1ncccn1)C CCC(CC(C)C)C(=O)NCc1nc(C(=O)N(C2CSC2)C)c(C)o1 C1(NC(C(CCCC)O)=O)CC2(CCCN(C(C3CCS(=O)(=O)C3(C)C)=O)C2)C1 c1(C(=O)NC2C(F)CCN(C(CC3C(=O)NC(=O)N3)=O)C2)ccc2nc[nH]c2c1 c1(C(=O)NC2CCCN(C(CCc3n(C)ccc3)=O)C2)scc2c1OCCO2 CC1CN(C(=O)CCC2CC2(C)C)CCC1NC(C1CCC(N(C)C)CC1)=O N1(C(C(C(C)C)(C)C)=O)CC2(NC(c3cccc(O)c3Cl)=O)CCCC2(F)C1 c1(C(=O)NC2CC(S(N)(=O)=O)C2)cc2cc(Cl)c(Cl)cc2[nH]1 c1(C(=O)NCC(C(C)(C)C)NC(=O)CCF)cc(N)cc2c1OCCO2 C(CNC(=NCC1CC1)NCC1CN(C2CC2)C1)(C(F)(F)F)OC c1(CCC)cc(C(=O)NCC2CCCN2c2nc(COC)ns2)nn1C N1(C(c2c(CNC(CN3CCC(OC)C3)=O)cc[nH]2)=O)CC(N(C)C)C(C)(C)C1 c1(NCC(N2CCN(C(C=CSC)=O)C3C2C3)=O)ccccc1[N+](=O)[O-] C1(NC(C2(CC=C)CC=CC2)=O)CC(C)CN(C(C2CC(=O)NC(=O)N2)=O)C1 C1(CC=C)(NC(C2SCCCS2)=O)CCN(C(c2csc(C#N)c2)=O)C1 c1(NC(c2nc(C(=O)N(c3cccc(F)c3)CCO)cs2)=O)cccc(Br)c1F N1(C(Cc2c(C)noc2C)=O)CC2COCC2(C(=O)NCC2CC23CC3(F)F)C1 C1(NC(C(C(C)O)C)=O)CCOC12CCN(C(C1CNC(=O)CC1C)=O)CC2 CC(C)C(C(=O)NC(C1CCCN1C(c1cc[nH]n1)=O)(C)C)n1ccnc1 c1(N2C(NC(=O)OC(C)(C)C)C3CCC2C3)nc2ccc(O)cc2s1 C1(CC(=O)N(C)Cc2cc(OC)no2)CCCCN1C(c1cn(C2CC2)cn1)=O C1(N(C(CCSCC(C)C)=O)C)CCCC(NC(c2cc(CO)[nH]n2)=O)C1 N1(C(C(CSC)C)=O)C(C(=O)NCCCc2ncn(C)n2)CCC12CC2 C1(CNC(CC(CC)O)=O)C2CCCC1N(C(c1ccc(F)s1)=O)C2 N1(C(C=Cc2c(C)ncs2)=O)C2CCC1CC(CNC(=O)CCc1nc[nH]n1)C2 C(=O)(CCCCCCN=[N+]=[N-])NC1C(C)CN(C(c2c(Cl)cccc2Cl)=O)CC1 O=C(C#CC1CCCCC1)NC1(CNC(=O)CCC2CCC(=O)N2)CCOC1 Cc1nc2ccccn2c1C(=O)NC(C1CCCN1C(=O)C(F)CC1CC1)C c1(OC(C)C)ccc(NC(=O)NC(c2ccc(Cl)cc2)CC2CC2)cc1 C1(F)(C(N2C(C(=O)NC)CCC2)=O)CCCN(C(=O)C=CC(C)(C)SC)C1 C1(NC(c2cn(CC=C)nc2)=O)CN(C(c2ccc(C)n2C)=O)CC1C1CC1 c1(OC)cc(C(N2CCCC2C(C)NC(=O)C(n2nc(C)cc2C)C)=O)ncn1 N1(C(c2ccc(CCC)[nH]2)=O)CC2CCN(C(c3cc(C(N)=O)co3)=O)CC2C1 c1(C(=O)NC(C)C=CC(=O)NCC(F)(F)CO)ncncc1Cl c1(C(N2C(CCc3cn(CC(=O)NCC)nn3)CCC2)=O)ccc(O)c(CC)c1 c1(CC)ccc(C(=O)NCCOC2CCN(C(=O)C=CCO)C2)cc1 CCC1=NOC(C(=O)NC2CCC(CNC(C3(C)CCOC3)=O)CC2)C1 C(=O)(C1=C(C#N)CCC1)N1CC(C)(CCC(=O)N2CC(N3CCC3)C2)C1 C1(C)(NC(CC2CCCC(C)C2)=O)CCN(C(c2cc(C3CC3)ccn2)=O)CC1 c1(CCOC)cccc(C(=O)NC(c2ncc[nH]2)CN2CCCCCC2)c1 C#CCCC(C(=O)NCC1(CCN(C)C)CC1)NC(c1ccc(C)o1)=O C1(OC)CC(NC(C2CC3CCC(C2)O3)=O)CN(C(c2n[nH]c3c2COC3)=O)C1 c1(C(N(C)CC2(NC(CC(CC=C)(C)C)=O)CC2)=O)cc2n(n1)CCNS2(=O)=O C1(CNC(CC(C)(C)OC)=O)CN(C(=O)C2=COCCC2)CCC1C(F)(F)F C(C1=CCN(C(=O)CC(c2ccccc2)C2CC2)CC1)OCC(=O)N(C)C Cc1nn(C)cc1CN(C)C(C1CCCN(C(=O)CCC2CC2C)C1)=O CC(C)(C(=O)NCC(c1ccccc1)NC(=O)CNc1ccccc1)C1CC1 N1(C(CCSc2n(C)ccn2)=O)CCC2CN(C(c3cc(=O)n(C)cn3)=O)CC12 C(=O)(CCC(C(C)C)NC(c1cccc2occc12)=O)N(c1c(C)cccc1)C C1(C(=O)NCCC2ON=C(C)C2)CCN(C(=O)C(C)c2ccsc2)CC1C CC1CCCC(CNC(C2(NC(c3nccnc3N)=O)CSC2)=O)O1 C1(COC)(CNC(c2nc(Cl)sc2C)=O)CCCN1C(=O)C#CC(=O)N(C)C O=C1Cc2c(-c3ccc(CNC(c4cnccc4[N+](=O)[O-])=O)nc3)cccc2N1 c1(CNC(C23CC(CCC)(C2)C3)=O)ccc(N=c2cc[nH]cc2)cc1 C1(NC(C(C)NS(CC)(=O)=O)=O)CN(C(=O)Cc2c(C)noc2C)CC1C(F)F C1(CC(N2C(CCCNC(C3(COC)CC=CC3)=O)CCC2)=O)C=NN(C)C1=O C#CCCC(C(=O)NC(CC(=C)C)C(=O)OC)NC(=O)CC1CC(SC)C1 O=C1NC(=O)C2(CCCC23CN(Cc2c[nH]c4ncc(Br)cc24)C3)N1 Cc1ccc(N)cc1C(N1CC(N(C(=O)CCn2cnnn2)C)C(F)C1)=O C(=O)(CCCS(N)(=O)=O)NCC1C(CNC(c2c(N)cc(F)cn2)=O)C1 CN1CCCC1C=CC(=O)NCC1CC1NC(c1coc(C(F)F)c1)=O c1(CC(=O)N(CCNC(c2n(CC)ncc2C)=O)C)cc(F)c(F)cc1F C1(O)(C(=O)NCCC)CCN(C(C)Cc2ccccc2OC)CC1 c1(C(N(C2CCCC(N(C(CC(=O)OC)=O)C)C2)C)=O)ncn2c1CCCC2 N1(C(C(C)(F)F)=O)CCCCC1c1n[nH]cc1C(=O)NCC(Cl)=CCl C(=O)(C#CC1CCCOC1)NCC1(C)CCN(C(c2c(C)cc(N)cc2)=O)C1 CCCCCCC(=O)N1CCCC(C)(CNC(C2CN(C)CCO2)=O)C1 n1(CCC(=O)NC2CCCN(C(c3cc(OC)ns3)=O)C2)ccc2cccnc12 c1(C(N2CCN(C(=O)C3=C(Cl)CCC3)C(C(F)F)C2)=O)ccc2nc[nH]c2n1 N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCC(C)C(NC(=O)C2=CCCSC2)C1 c1(C(c2nnnn2C2CCOC2)NCCNC(=O)OC)csc(Cl)c1Cl C12(CNC(C3(S(N)(=O)=O)CCC3)=O)CCCC1CN(C(=O)Cc1ccoc1)C2 c1(C(=O)NCCN(C(=O)CSc2ccccc2)C)cc(F)c(F)cc1N N1(CC(=O)NC(c2cccnc2)C(=O)NCC2CC23CC3)CC2CC2C1 C(=O)(C(CC)C(C)(C)CC)NCC(=C)CCNC(=O)Cc1nc[nH]n1 c1(OCC(=O)NC2C3(CC(NC(c4c(C#C)c[nH]n4)=O)C3)C2)c(C)cccc1C C12(NC(=O)CCN3CCCC3)CCCCC1N(C(c1cnc3sccn13)=O)CC2 CN1CCN(C(=O)CSc2cn[nH]c2)C(C(N2CC(F)(C#N)C2)=O)C1 N1(C(c2cn(C(C)C)nc2)=O)CCCCCC1CNC(C12CCCC(CO1)C2)=O N1(C(c2cnn(C)c2N)=O)CCS(=O)(=O)C(CCNC(C2CC=CCC2)=O)C1 c1(NC(=O)NCC(N2CCC(C)CC2)C(C)C)ccc(=O)n(CC(F)(F)F)c1 C=CCC(CNC(C1OC2CCC1C2)=O)C(=O)NC1CN(C)NC1=O C1(C)(CNC(=O)NC(c2c(C)noc2C)CC)CC2CC2C1 Cc1c(C(N2CCC(NC(C3C(C)C3(F)F)=O)C2)=O)csc1Br c1(CC)cccc(NC(C2(CNC(=O)CN3CCC(C)(C)C3)CC=CC2)=O)c1 C1(C(N2C(CC)CN(C(c3cc(C)ns3)=O)CC2)=O)CN2CCC1(C)CC2 C1(C(=O)NCC(CN(C(=O)CCCn2cccn2)C)(C)C)CCC(N(C)C)CC1 c1(C(=O)OCC)nc(C(=O)N(C)CCNC(c2cnc(C(C)(F)F)s2)=O)c(C)s1 C1(C)(C(=O)NCCC(=O)NCC(CSC)OC)Cc2ccc(C)cc2C(=O)O1 c1(C(=O)NCCOCCOCCNC(C=CCC)=O)cnn(C)c1C c1(C(=O)NCC(C)N(C(=O)C2=COCCC2)C)ccc2nc[nH]c2c1F C(=O)(C(CC(N)=O)NC(=O)C=Cc1cc[nH]c1)N(C)CCN1CCCC1 c1(-c2ccc(OC)c(C)c2)cc(C(N2CC3CNC(=O)C3C2)=O)cc2[nH]ncc12 CCC(CC)CC(F)C(=O)N1CC(OC)C(C(=O)NC(C)(C)C(=O)NC)C1 N1(C(=O)C=Cc2ccncc2)CCC=C(C(=O)N2CCC3CC23)C1 C(=O)(C(=O)N=c1[nH]n(C(C)(C)C)cc1C)c1ccc(CCCC)cc1 C1(CC(=O)NC(C(N2CC(=C)C2)=O)C2(O)CCC2)CCCOCC1 C(=O)(CCCCC(N)=O)N1CCC(C)C(CC(=O)NCCOCCCO)C1 c1(C(N2CCC(N(C(c3cncc(COC)c3)=O)C)C2)=O)cnc(Cl)cc1N C1(C(=O)NC2CCS(=O)(=O)C2)CC2(CCN(C(c3ccc(F)cn3)=O)CC2)CO1 CCCC(C(=O)N(CCCNC(C1(CO)CCOC1)=O)C1CC1)OC c1(C(=O)NCCN(C(C2(C#N)CC3CC3C2)=O)CC)ccc2sc(O)nc2c1 c1(N2C(C)CCN(C(CC(CC)C)=O)CC2)ncnc2sc([N+](=O)[O-])cc12 N1(C(C(C)N(C)CC)=O)CCC2CN(C(c3cn4ccsc4n3)=O)CC2C1 c1(C(C)C)nc(C(=O)NCC2CCC2C(F)(F)F)cs1 C1(NC(c2ccc(OC)nc2Cl)=O)CC2CC(C1)CN(C(c1cscn1)=O)C2 c1(C(=O)NC23CC2CN(C(c2cc(F)n[nH]2)=O)C3)c[nH]c2cccc(Br)c12 C1(CNC(C2CC(C)(F)C2)=O)C(C2CC2)CCN1C(=O)C(F)C1CCC1 C(=O)(C(CNC(c1cnncc1OC)=O)C(C)C)NCC1CCCC(CC)C1 CC1(C#CC(=O)NCC2CC(F)CN2C(c2nc(C3CC3)cs2)=O)CCCO1 C(CC1=CCN(C(C2CCS(=O)(=O)C2)=O)CC1)NC(C(n1cc(Cl)cn1)C)=O C12(C(=O)NCC(C)N(C)C(c3cc(-c4ccco4)on3)=O)CC(C1)C(C)(C)O2 C(=O)(CCCS(N)(=O)=O)NC(CC)(CNC(c1cc(O)cc(O)n1)=O)CC N1(C(CC(C)F)=O)CC2C(CN(C(=O)Cn3nnnc3-c3ccccc3)C)C2C1 c1(C(N2CC(c3ccccc3)(NC(CC=CC)=O)C2)=O)ccc(=O)oc1 C(=O)(C1=NOC(C)C1)N1C(C)(CC(=O)NCC(=O)OCC=C)CC1 C(CCCC(CO)NC(=O)Cc1ccnc(O)c1)NC(CCC=CCC=C)=O N1(C(CC(CC)OC)=O)CC2(CCCC2)C1C(=O)NCc1snnc1C C=CC1(C(=O)NC(C)CCO)CCN(C(C2CC(F)CN2C)=O)C1 C1(NC(C2CCCO2)=O)CN(C(c2cc(Cl)no2)=O)CC2(CCC2)C1 c1(C(N2C(C)(C(=O)Nc3cnc(C)nc3)CCC2)=O)cc(F)c(Br)c(F)c1 c1(-c2c(C(=O)NCCC(C)NC(C3C(C(=O)OC)C3)=O)c[nH]n2)cccc(Cl)c1 n1(CC(=O)NC2C=CCN(C(C(CC)NC(N)=O)=O)C2)nc(C)c([N+](=O)[O-])c1C C1(O)(CCNC(C(C)=CC)=O)CCCN(C(c2ncc(C(F)(F)F)cc2O)=O)C1 C(=O)(C1CCCc2nc[nH]c21)N1CC(NC(c2nc(CC)sc2)=O)C(C)C1 N(C1c2ccccc2CC1NC(C1(F)CCOC1)=O)C(CCC1(C)CC1)=O c1(CC)ccc(C(=O)NC(=O)C(COC)N(CC)CC)cc1.C12(CCC1)CN2 c1(C(=O)NCC2(F)CC(NC(c3nc(CCC)oc3)=O)C2)cccc(O)n1 C1(CCC)CN(C(=O)C(C)(C)C(C)O)CCN1C(c1cn(C)c(O)n1)=O N1(C(C2(CSC)CC2)=O)CC2(COC(CNC(=O)C3=C(Cl)CC3)C2)C1 c1(CC(=O)NCC2C(C)CCCN2C(C2CCOC2)=O)ccc2nonc2c1 c1(OC2COCCN(C(CC)=O)C2)ccc(F)c(C(=O)OC)c1 n1(CC2(COC)CC2)ncc(N(C(=O)C(C)OCC(C)C)C)c1COC C(CC1CCC1)(C(=O)OCCOCCCC1CCOC1=O)NC(=O)CC1CCC1 N1(C(C(CC)OCC)=O)CC=C(CCNC(=O)C2=NOC(C)C2C)CC1 C1(NC(CC(C)NC(N)=O)=O)CCCN(C(c2cccc(NS(N)(=O)=O)n2)=O)C1C C1(C(=O)NCCC(CNC(c2cccc(OC)n2)=O)O)CCOC(C)(C)C1 C1(C(=O)NCC2(N(C)C)CCCC2)CC2(CCN1C(c1cccc(O)n1)=O)CC2 N1(C(C(N2CCN(C3(C)CCCCCC3)CC2)=O)=O)CCC2(CO)CCCC12 C#Cc1cnc(N(C)CC2CCN(C(=O)C(C)OCC(C)C)C2)nc1 C1(C(=O)NC2CC(CC(=O)NCC3CCC=CCC3)C2)(OC)CCCOC1 c1(-c2nc(OC)sn2)cccc2nc(C(N3CCC(N(C)C)CC3)=O)cn12 c1(CC(=O)NCC2CCN(C(COCCC(C)C)=O)C2)ccc2nsnc2c1 c1(C(=O)NC2C3CN(C(c4c(CC)occ4)=O)CC32)cc2n(n1)C(C)CCC2 CC1CCCCC1NC(=O)CN(C)C(c1nn(C)cc1Cl)=O c1(C(C)NC(N(C(C(=O)OC)COC(C)C)C)=O)c(Cl)ccc(F)c1Cl c1(CC)nn(C)cc1CNC(=O)C(c1cccc(Cl)n1)N c1(C(N(C2CCN(C(CC(C)(C)O)=O)C2)CC2CC2)=O)cc2n(n1)CCO2 c1(C(=O)NC(CC2CN(C(CC(C)OC)=O)C2)C)cccc(OC)c1 C1(=O)C(CF)NC(=O)OC(C2CCC2)C(=O)NCCCN1C.C(C)(C)(C)OCC c1(CCNC(CN(C(COCCCC(C)C)=O)C2CC2)=O)cc(O)ncn1 C1(N(C(=O)CN2CC3CC3C2)CC#C)CCN(C(C2CCCOC2)=O)CC1 Cc1ccc(C(C(=O)NC2CCOC2)N(CCC(C)C)C)cc1OC(F)F C1(C(N)=O)CN(C(C2CCC=CO2)=O)CCC1NC(c1cc(Cl)nc(Cl)c1)=O N1(C(c2c(C)nc(C)o2)=O)CCN(C(=O)CNC(=O)Cc2ccccc2)C2CC12 Cc1ccc(Cl)cc1NC(C12CC(NC(c3cccc(Cl)c3F)=O)(C1)C2)=O N1(C(C(CCSC)N(C)C)=O)CC2CC(NC(=O)CN(C)C(=O)C3CC3)CC1C2 c12noc(n1)C1CCC(C1)C(=O)NC2.c1(CC)cscc1C1OCCO1.C1CN1 C1(CNC(C(F)=CC)=O)C(C)CCCN1C(=O)CNC(c1ccsc1)=O C1(C)(NC(COCC=C)=O)CCCCC1C(=O)NCCCSCC c1(C(N(C)CC2CCCC(NC(C=C(C)C)=O)C2)=O)ccc([N+](=O)[O-])c(N)n1 N1(C(C(=O)NC)=O)CC(NC(=O)COc2ccccc2C(C)(C)C)CC1C C(C)(C)(CCC(=O)NCC1(O)CCN(C(=O)C(F)C(C)(C)O)C1)OC C1(CC(N2CCC(NC(CC(CC)(F)F)=O)C(C)C2)=O)COC2(CCC2)CO1 C=CC(C)(C)C(=O)NC(c1ccc(C)cc1)CNC(c1c(C)n[nH]c1C)=O C1(C(C)CNC(=O)CCC2CCCO2)CCN(C(=O)CCc2cn(C)nn2)CC1 C(=O)(C1=COCCC1)N(C1CCCN(C(c2nnn(COCC)c2N)=O)C1)C C(=O)(CCC(C)(C)C#N)N(C(C(CC)C)C(=O)NCCC(Cl)Cl)C C(C)(CO)(C(=O)N(C(C)CNC(=O)Cc1ccc(C(N)=O)nc1)C)NC(C)=O CC(C)CCC(=O)NC1CCOCC1C(=O)Nc1cnn(C)c1Cl C12(CN3C(=O)CN(CCc4nnc(C)s4)C3=O)COCCN1C(=O)OC2 C#CC(CNC(c1ccc(CNC(=O)Cc2nocc2CC)o1)=O)CC1CC1 c1(C(=O)NC2C(CNC(C(C3CC3)SC)=O)COC2)cc2sccc2[nH]1 N1(C(c2c(CC)nn(C)c2)=O)CCC(CO)C(NC(c2c(C)noc2CC)=O)C1 C(=O)(C1=NOC(C)C1)N(C(C)CNC(c1nocc1Cl)=O)C C=CC(CC)CC(=O)NCCNC(=O)CC(C(C)C)c1ccon1 C=CC1COCC1NC(=O)C(O)C1CN(C(=O)C(CC)CC)C1 c1(C2CN(C(C3Cc4nccn4C3)=O)C2)cc2ccccc2s1 C(=O)(C1=CCCC(C)(C)C1)N1CC(O)(C(C)NC(c2cn(CCC=C)nn2)=O)C1 Cc1nc2c(C(=O)NCCNC(C3CN(C(=O)N(C)C)C3)=O)cccc2o1 C1(O)(CNC(CC(C)SC)=O)CCCN(C(=O)CCc2cccc(O)c2)CC1 C1(C(=O)NC2CCCN(C(C3(CC(F)F)CC3)=O)CC2)Cc2cccc(F)c2O1 N1(C(C(C)NC(C)=O)=O)CC2(CCC(C(=O)NC(CC(C)C)C(N)=O)O2)C1 C(=O)(C#CC(C)(C)C)NC(C)CCNC(c1sccc1Cl)=O C(=O)(C1=NOC2COCC12)NCCCCC(C)NC(c1[nH]cc(C)c1)=O N1(C(C=C(C)C(C)(C)C)=O)CC(C(=O)N(C)Cc2nnc(C)s2)CCC1(C)C c1(CC(C)C)cccc(OCC(=O)NC(=O)NC2CCCC2)c1 N1(C(C(C)CF)=O)CC2(C1)CN(C(=O)CC1(CO)CCOCC1)C2 c1(C(=O)OCC)cc(OC)cc(NCP(C)(C)=O)c1Cl C(=O)(C(CC(F)F)NC(c1ncccc1N)=O)N1CC(CCC)OCC1 C#Cc1cc(C(N2CC(CCNC(c3ccccc3C)=O)(OC)C2)=O)ccc1C C1(CN2CCC(C(C)(C)F)CC2)CC2(CCOCC2)C(=O)N1 C1(NC(C(C)C2CCCC2)=O)CCN(C(C2CC(NS(C)(=O)=O)C2)=O)CC1 Cc1cc(C(N2CC(N(C)C(c3ccccc3Cl)=O)C(C)(C)C2)=O)ncc1C#N N1(C(c2cc(CC(C)C)[nH]n2)=O)CC2(C1)CN(C(c1sccc1Cl)=O)CCO2 CCCC(F)C(=O)NCCC1(O)CN(C(C2CCN(C)CC2)=O)C1 C(=O)(CC(C)C(F)F)N1CCC(C(CNC(COCC#C)=O)(C)O)CC1 Cc1c(C(N2CC(CNC(C3CC34CC(C)(C)C4)=O)C(O)C2)=O)cncc1N c1(C(=O)NC(COC)CNC(=O)C(C)C2CCCC2)ccnc(C)n1 N1(C(CCCOCC=C)=O)CCN(C(c2cnn(CC(C)C)c2)=O)C(CF)C1 N1(C(C(=O)NCC)=O)CCCC2(C1)CN(C(=O)C(C)CN1CCCC1)C2 C(CC(C)(C)C)(C(=O)NC1COC(C(F)F)C1)NC(C(c1ccncc1)C)=O C(c1nc(C)cs1)=CC(=O)N(CC(CC)NC(=O)CCC(=O)N1CCCC1)C CC(C)C(C(=O)N(CC(C)NC(C1(CSc2ccccc2)CCC1)=O)C)N(C)C c1(C(=O)NC(CNC(CC(=O)OC)=O)C2CC2)cc(NC2CC2)nc(C)c1 c1(C(N2C(CC(=O)NOCCN3CCOCC3)CCC2)=O)cccc(F)c1 Cn1cc(CNC(C23CC(F)C2C3)=O)c(C(F)F)n1 N#Cc1ccc(-c2ccc(OC(C34CCCC3CCC4)=O)cc2)nc1 C1(CNC(C(C)SCCCC)=O)(CO)CCCN(C(C2CCCC(O)C2)=O)C1 n1(C(C)C(=O)N(C(C)CN(C)C(c2cnco2)=O)C)cnc2ccccc12 C1(CNC(C(c2ccccc2)OCC)=O)COCC1NC(=O)CSCC(N)=O C(C)(CO)(C(=O)NCCC(=O)NC(N)=O)NC(C1CCN(CC)C1)=O C1(NC(C2CC(NC(C=CC(C)(C)SC)=O)C2(C)C)=O)CN(C)C(=O)C12CC2 C12(NC(CCCCC=C)=O)CCCCC1N(C(=O)C=Cc1ccnn1C)CC2 C(=O)(C(O)CCCNC(C1CCC2(CC1)CC2)=O)NC1C(c2n(C)ncc2)C1 Cc1nc(Cl)nc(N2CC3CC2CCC3NC(C2(C)CCS(=O)(=O)CC2)=O)c1F N1(C(C(CCC)C)=O)CCC(NC(=O)CCC2CCCN2C)C(CO)CC1 CCC(CC(=O)NC(C(=O)NCc1nc[nH]n1)C1CCC1)C(F)F C(=O)(CCCOc1ccccc1)NCCC(C)NC(=O)Cc1cc[nH]c1 C(=O)(C(CC(C)C)C(C)C)NCCC1CCCN(C(C2(SC)CCC2)=O)C1 c1(C(=O)NCC(CNC(C(CC=C)(C)CC)=O)OC)cc(C)c2occc2c1 c1(OC)nsc(OC)c1C(N1CCOC(CNC(c2cc(C(N)=O)[nH]n2)=O)C1)=O N1(C(C2CC(CC(=O)OC)C2)=O)CCC(C(N2CCC3(CC2)N=N3)=O)CC1C c1(C(N2CC(O)(CC(N3CCC(NC)CC3)=O)C2)=O)cc(F)c(OC)c(F)c1 c1(C(=O)NCC(CC=C)NC(CC=C=C)=O)cc(F)c(Br)c(F)c1N c12cc(ncc1Cl)OCCn1nc(Cc3ccc(OC)cc3)nc1-2.CC=CC c1(-n2cc(CCCCSCC(=O)Nc3ccc(C(=O)O)o3)nn2)cncc(Br)c1 C(=O)(C(C(C)(C)C)OC)NCC(C)(Cn1cccn1)NC(CCCCOC)=O C1(NC(C2CCN(CC)C2)=O)CC2CCC(C1)N2C(c1cc(C)c(F)cc1N)=O C(C(C)(C)CC(=O)N1CCC(NC(=O)COC(C)C)C2CC12)OC c1(OC)ccc(Br)cc1CCN=C(NCCF)NC1CCS(=O)(=O)C1 c1(OC)nc(Cl)c(C)cc1N=c1ccnc(CO)[nH]1 N1(CCOC(C)=O)CCN(CC2CC2OC(C)C)CC1 Cc1nn(C)cc1C(N1CC(F)CC1C(=O)Nc1cn(C)nc1C(F)(F)F)=O Cn1ncc2c(NC3CC(F)C3)nc(N3CCC4(CC3)NC(=O)CC4=O)nc12 c1(C(=O)NCC(C2CCN(C(C3(CF)CC3)=O)CC2)C)nn2cccnc2c1Cl C1(CC)CN(C(=O)C(C)Oc2ccc(C)cc2)CCN1C(c1cc(F)c[nH]1)=O c1(OC)ccc(OCC(N2CCC=CC2CNC(=O)C=CC(F)(F)F)=O)cc1 N1(C(COC(C)C)=O)CC2CC1CC2NC(c1cc(F)cnc1O)=O C1(CNC(C(F)=C(C)C)=O)C(C)CCN1C(c1oc(Br)cc1C)=O C1(NC(=O)Cc2cccc(Br)c2)COCCN(C(C2(C3CC3)CCC2)=O)C1 c1(OC)cc(C(=O)N(CC(O)CN(C(=O)C(C)O)C)C)c2ccccc2c1 N1(C(CCN(C(C)=O)C)=O)CC(NC(=O)CCC(N)=O)C2CC12 N1(C(c2c(CC)nccn2)=O)CC(NC(=O)C=Cc2ccccc2)C2(CCC2)C1 c1(CN(CCOC)CCN2CC2)cc(C(=O)OC)cs1 c1(C(N(C(c2ccc(Br)s2)C(=O)OC)C)C)nc2ccccc2s1 O=C1CCCc2cc(C(N3CCCC4(C3)CN(C(=O)C=CCF)C4)=O)ccc21 N1(C(c2c[nH]c(=N)o2)=O)CCc2ccc(C(F)(F)F)cc2C1 c1(-c2nc(N(C=O)CC3C=CS(=O)(=O)C3)sc2)cc(Br)c2c(c1)OCCO2 C1(CC(=O)NC2CC(CCC)C2)C2CCCC2N1C(=O)C(C)(C)C(=O)OCC c1(NCc2ccc(C)cc2C)cc(=NCCc2ccc(S(C)(=O)=O)s2)[nH]c(C)n1 C1(NC(CCC=CC)=O)CCN(C(C2(COC)CCOCC2)=O)CC1C C(=O)(C1=CS(=O)CCC1)N(CC(CC)NC(c1ccn(CCC)n1)=O)C C(=O)(C(C)(F)C(C)(C)F)N1CCC(C(C(=O)N(CCCF)CC)F)C1 CC(CC(=O)N1CCC1C(=O)N(C)CC1(C)CN(C)C1)c1ccco1 C1(C(C(=O)NC2C(CCCC)CCC2)C)CCN(C(c2cc[nH]n2)=O)CC1 C=CC(CCC)CC(=O)NCCCOCCNC(=O)CCC(=O)c1cnn(C)c1 C12(NC(c3n(C=C)ncc3)=O)CC(CNC(C3CC4CCC3CC4)=O)(C1)OC2C c1(-c2cn(C(C)C)nc2)ncc(Cl)cc1C(=O)NCC1CCC1 C(=O)(CCC(C)CC)NC(c1c(C)cccc1Br)C(=O)N(CC=C)CC C1(C(=O)NCCC(CNC(c2ccc(C(F)(F)F)cc2)=O)O)CC2(CCC2O)C1 CCC(CNC(=O)CCc1cccc(Cl)c1)(CC)NC(c1ccnc(S)c1)=O C1(C(=O)NC2CCC(C(=O)Nc3ncccc3Br)C2)CCCC2CCCCC12 N1(C(C2CCN(c3n(C)ccn3)C2)=O)CC2CC(NC(=O)C(C)(C)CF)C(C2)C1 c1(OC)ccc([N+](=O)[O-])c(CN2CC(C(N3CCCC(C)(O)CC3)=O)C2)c1 C1(C(=O)NC(CC=CC)C(=O)NC2(CO)CC3(CCC3)C2)CCC2(CCC2)O1 C(C)(CN=c1cccc(S(=O)(=O)NC(C)Cc2nccn2C)[nH]1)OCC=C N1(C(CCC=C=C)=O)CC2CCCC1CN(C(=O)C=CC(C)(C)C)C2 N1(C(C(CC)C2CCOCC2)=O)CCC(NC(=O)Cc2cnsc2)CC1C C1(CNC(CC(CC)C)=O)CN(C(c2ccnc(C)c2)=O)CCC12CCC2 CC1(C)NC(=O)CCC1NCC(N1CCS(=O)(=O)CC1c1ccccc1)=O O=C1CCC(CC(=O)NC2C3CCN(C(c4ccsc4Cl)=O)C23)CN1 C1(C)(NC(C2N(C(C(C)=C3CCC3)=O)CC2C)=O)CCC(=O)N(C)C1 C1(CCNC(=O)Nc2ncc(-c3ccccc3)s2)CCCCCC1 c1(OC)ccc(C(=O)NC(C(C)NC(c2cnn(CC(F)F)c2)=O)C(C)C)nc1 CC(C)C(C#N)C(=O)N1CCC(C(N2CC(OC(F)F)C2)=O)C1(C)C c1(CC)ncoc1C(=O)NC(C(N1CCC(CN(C)C)C1)=O)n1cncn1 c1(C(=O)OC)ccc(C)c(C(=O)NC(CNC(C2CCCS2(=O)=O)=O)C2CC2)c1 N#Cc1c(-c2ccccc2)nn(CC(N)=O)c1N C12(CNC(C3CC=CCC3)=O)CCCC1N(C(c1cc(F)n[nH]1)=O)CC2 CC(c1ccccc1F)=CC(=O)NCC#CCNC(C1CC1[N+](=O)[O-])=O C(C)(C(=O)NNC(=O)c1cccc(OC(F)(F)F)c1)Nc1ccc(C)s1 [N-]=[N+]=NC1CN(C(C2CC23CC(O)C3)=O)CC1NC(c1cc(CCCO)on1)=O c1(C(=O)NCC2CCN(C(C3CCCO3)=O)C2)sc(Br)cc1Cl c1(C(N(C2CC(NC(CC=C(C)C)=O)C2)C)=O)ccc(Br)cc1C#N C(=O)(CCCCCCCCCCCBr)N1CC(C(N2CCC(OC)C(F)C2)=O)C1 CN1CC(NC(C2CCCNC2)=O)CC1=O C1(C(=O)NC2CC3(CC(NC(c4cnsn4)=O)C3)C2)CCn2cnnc2C1 C1(C(=O)N(CC(C)NC(=O)CC(C)N2CCCC2=O)C)(COC)CCCCC1 Cc1cccc(C(N2CC(NC(c3ccccc3C(C)C)=O)C3CC23)=O)n1 c1(CCC(N2C(CNC(c3cc(CC)ncn3)=O)CCC2)=O)ccc(C)c(C)c1 C(C1CN(C(=O)CCC2CCC(=O)N2)Cc2ccccc21)NC(COCC)=O c1(CNC(C(C=CC)O)=O)cc(C(=O)NC2CC2CN(C)C)n(C)n1 c1(C(=O)NC2CCCN(C(C3CC(C)(O)C3)=O)C2)c(F)cccc1Cl c1(OC(C)C)ccc(C(=O)NC2CN(C(=O)C(C)C(F)F)CC2C(F)F)cc1N N1(C(C)=O)CCC(C)(C(=O)NCC(C2CC2)N(C)C(C2CC2C(N)=O)=O)CC1 c1(OC)cc(C(=O)NCC2CCN2C(C23CCC(CC2)C3)=O)c2c(c1)CCCC2 C1(NC(CCc2ccc(C)s2)=O)CN(Cc2ccc(C#N)cc2O)CCC1(F)F c1(C(N(CC(C)NC(c2ccc(Cl)o2)=O)C)=O)csc(C(F)F)n1 CCCCCCC(C)CC(=O)NCC1CN(c2ncncc2Cl)CCN1C Cc1cc(C)c(C(=O)NC2CC2CNC(c2ccc(C(F)(F)F)o2)=O)[nH]1 c1(C(N2C(C)(C)C(NC(C3CCC4CC4C3)=O)CC2)=O)nc2cccnc2s1 Cc1noc(C)c1C(C)(C)C(=O)NCC1(F)CN(C(=O)CCC#N)C1 CCCCC(C(=O)NCC1CCC(C)N1C)NC(c1cnc(N)cn1)=O CC(C)(C#N)CC(=O)NCCC1(C)CCN(C(=O)CC2CC(C)(C)C(=O)N2)C1 C1(O)(C(=O)NC2(CCOC)CCN(C(C3(F)CC=CC3)=O)C2)CCC(C)(C)CC1 C12(C(=O)NC(CC)(CNC(C3CC3(C)C(F)F)=O)CC)CCCN1CCC2 n1(CC)ncc(Cl)c1C(=O)N(C)CCNCc1ccncc1Cl.n12cc(nn1)C2 CN1CC(C(=O)NC2(CNC(C3CCS3(=O)=O)=O)CCCC2)OCCC1=O C1(C(F)(F)F)(CNC(C)(Cc2ccccc2)C(F)(F)F)CC2CCC1CC2 C1(C(=O)NC(CC)CNC(=O)C(c2ccc(F)cc2)CO)Cc2ccccc2N1 N1(C(c2ccc(C#C)cn2)=O)CCC2(CCCN2C(c2nccnc2Cl)=O)C1 c1(C(N(C2(C(=O)NC(C)CCN3CCCC3)CC2)C)=O)cc(F)c[nH]1 C12(C(N3C4CCC3CC4)=O)CC(C)(C1)OC2C.c1(C(=O)NC)cc(Cl)ncc1F C12(C(N3CC4C(NC(=O)C=C5CCOCC5)C4C3)=O)CCC(CC1O)C2 C(CCC(O)C(=O)NCCCc1nncs1)NC(c1c(C)ocn1)=O C1(NC(C(C)Oc2cccnc2)=O)CCC12CCN(C(C13CC(F)(C1)C3)=O)CC2 CC(C)C(C#N)C(=O)NC1CC(CC(=O)NC2CCC3CC3CC2)C1 CC(C)(O)CC(=O)NCC(O)CCNC(c1cc(C2CCOC2)[nH]n1)=O N1(C(C(c2ccccn2)C)=O)CCOCC(NC(c2sccc2C2CC2)=O)C1 C=CC(C)(CC)C(=O)NC1(C2CN(C(c3ccc(CO)cc3)=O)C2)CC1 c1(OCC)cncc(CCC(N2CCCC2CNC(=O)C(Cl)=CCl)=O)c1 C1(N(C(CCCC)=O)C)CN(C(C2COC(=O)C2)=O)CC1(C)C C1(C#N)(OC)CC(C(=O)N(CC(O)CN(C)C(c2cc(C(N)=O)[nH]n2)=O)C)C1 N1(C(CCNC(C)=O)=O)CC2CCC1C2NC(c1ccc(CNS(C)(=O)=O)o1)=O N1(C(c2cnn(CC)c2C(F)(F)F)=O)CCOC(C)(CNC(=O)C(F)OC)C1 c1(N(C(Cc2c(C)nc[nH]2)=O)C)cccc(F)c1 c1(C(N2CCC(NC(c3cc(OCC)n[nH]3)=O)C(O)C2)=O)cnc2occc2c1 c1(C(=O)NCCCCN(C(C2(C)CCN(C)CC2)=O)C)cc2cccnn2c1 c1(CC)ncc2c(n1)CCC(C(N1CCOCC1CNC(=O)C(=O)N(C)C)=O)C2 c1(C(=O)NC2(C)CCN(C(=O)CSC3CCCCO3)C2)ccc2c(n1)CCCC2 Cc1nccc(C(=O)NC(CCN(C(=O)CC(O)c2ccccc2)C)C(C)C)n1 C1(C)(NC(C2C(c3n(C)c(S)nn3)CC2)=O)CCN(C(c2ccoc2Cl)=O)CC1 C1(CNC(N(c2ccc(C)cc2)c2ccccc2)=O)CCC(C2CC2)C1 C(C(CC)(CC)NC(c1cncn1C)=O)NC(C1C(CC)OCC1)=O C12(NC(CCC=CC)=O)CCCCC1CN(C(C13CCCC(C)(C1)OC3)=O)C2 C1(CNC(C2(C(F)F)CC(=C)C2)=O)CN(C(c2cc(C)n(C3CC3)n2)=O)CCO1 c1(NC(C2CCN(C(c3cc(OCC)no3)=O)C2)C)nccc(-n2ccnc2)n1 c1(OC)cnc(SC)[nH]c1=Nc1cnn(C(C)(C)C)c1.c12ccccc1CC(=O)N2 C(=O)(C(C)(C)C(F)F)N1CC(CC2(NC(CC(C=C)C)=O)CCOCC2)(SC)C1 C12(NC(=O)OC(C)(C)C)CCC(COC)(C1)OC2.C(=O)(C1C(=O)N1)NCC N1(C(c2c(C)noc2)=O)CCCCC(C(=O)NC2CCN(C)CC2C)C1 CCC(O)C(C)C(=O)N(C1CCCC1)CCNC(c1cc(C2CC2)cs1)=O N1(C(C(c2ccco2)NC(Cc2c(C)cccc2)=O)=O)CC(O)CC(O)C1 N1(C(c2ccc(N(CCC)CC)cc2)=O)CCN(C(=O)CCCOC)C(C)C1 C1(NC(C2N(C)CCC2)=O)CC2CC(NC(c3sccc3CN(C)C)=O)C1C2 CC(C(=O)NOCCOCCO)N(C(=O)Cc1ccsc1)C N1(C(CCC=C)=O)CCC2(COC(CCNC(=O)CS(=O)(=O)NC3CC3)C2)C1 C12CC(CNC(=O)CSc3nncs3)N(C1)C2=O.c1(C(=O)OC)cc(C(N)=O)co1 Cn1nccc1C1(C(N2CC(O)(c3cc[nH]n3)C2)=O)CCC1 C(CC(C)(C)CNC(=O)CC(CC1CC1)NC(C1(CO)CCCCO1)=O)OC N1(C(c2csc(S)n2)=O)CCN(C(=O)C(O)C2CCC2)CC(O)C1 N1(C(C2C(C=C)C2)=O)CCOC(CCNC(=O)CCC(C)N(C)C)C1 c1(CC(=O)NCC(CO)NC(CCOC)=O)csc(SCCN(C)C)n1 C(Cn1cncn1)(C(=O)NC1COC(=O)C1)NC(C(C)=C(C)C)=O c1(C(N(CCCOC(c2cn(CC3(C)COC3)nn2)=O)C)=O)ncnc2c1CCC2 c1(SC)cc(C(N2CC3C(CN(C)C(c4cccn4C)=O)C3C2)=O)c(C)o1 C1(CCC(=O)NCCN(C)C)CCCN(C(=O)Cn2cnnn2)C1 CCCCCC(O)CC(=O)N1CC(NC(=O)Cc2cccc(OC)c2)C(F)C1 c1(-c2nc(C=C(CC)CCC(=O)OC(C)(C)C)on2)cn(C)c(=O)n(C)c1=O C(=O)(CCC(C)C(C(=O)NCCCSC)N1CCCC1C(=O)N(C)C)OC c1(C(N(c2nc(SC)c(Br)cn2)CC2(C)CNC2)=O)cc2c(cc1Br)OCCO2 Cc1nc(C(=O)NCC23CC2CN(C(C2C(C(F)F)C2(C)C)=O)C3)c(C)n1C c1(OC)cc(N)ccc1C(=O)NCC#CCNC(c1sccc1F)=O N1(C(c2cc(CC)on2)=O)CCC(C(C)C(=O)N(C(C)C(C)(C)O)C)CC1 [N-]=[N+]=NC1CCC(NC(c2cnn(-c3ccccc3Br)c2)=O)CC1 CC1CCC(Cl)=C(C(=O)NCC2CC2NC(c2ccc(-c3ccccn3)s2)=O)C1 C1(C(C(=O)NC(c2cn(-c3ccccc3)nn2)C)O)CCOCC1 C1(C(=O)NCC=CCNC(C2CCC(=O)O2)=O)CS(=O)(=O)CC12CCC2 C1(C(=O)NCc2c(C(N(C3C(C)CC3)C)=O)occ2)CC2(CC(=O)C2)C1 c1(N2CC(C)C(F)(F)C2)nc2ccc(Cl)cc2c(=NC2CC(CCO)C2)[nH]1 C1(NC(C(CC(=C)C)NC(=O)CC(C)F)=O)C2CCN(CC2)C1C c1(C2(C(=O)NCC(CNC(=O)CC3C=CS(=O)(=O)C3)OC)CC2)cc(F)ccc1C CC1(CNC(c2cnccc2Cl)=O)CCCN(C(C2CCC3CC23)=O)C1 Cc1cc(CNC(C(c2ccc(F)cc2)(C)C)c2nnnn2C)nnc1C c1(C(N2C(CNC(C(C)OCC)=O)CC3CC32)=O)ncc2c(F)cccn12 CCCCC(CC)CCC(=O)N1CCCC1(C)CNC(=O)Cn1cc(CO)nn1 C1(NC(c2c(C)ccnc2)=O)CN(C(=O)CCS(C)(=O)=O)CC2(CCC2)C1 N1(C(CC2(NC(C)=O)CC2)=O)CCC(C)C1C(=O)N(C)Cc1cnc[nH]1 c1(C(N2C(C(=O)OC)CC(F)(F)CC2)=O)cc(S(N)(=O)=O)cn1C c1(COC)nc(C)ncc1C(N1CCCC(SC)CC1)=O.C12(CC1)C(=O)N(C)C2 C#CCC(C(=O)N=c1ccn(CCCO)[nH]1)NC(=O)CCN(C)CC N1(C(C=CCN(C)CC)=O)CCN(C)CC1C(=O)NC1CCCC(C)C1 c1(C(N2C3C(NC(=O)C=C4CCC4)CC(C3)C2)=O)ccn2c1CSCC2 C#Cc1cc(C(=O)NC(C)CC(C)NC(=O)CC2(OC)CCOCC2)ccc1Cl c1(OC(C)=O)ccc(C)c(CC(=O)NCc2ccn(C(C)C)c2)c1 C1(C)(CNC(COC(CC)(C)C)=O)CN(C(C2CCCC(=O)N2C)=O)CC1C CCCC(O)C(=O)N1CCN(C2CCN(C(=O)CC3CCC3)C2)CC1 c1(CC)nnc(C)cc1C(N1CCC(C)C(NC(=O)CS(=O)(=O)NC)C1)=O c1(C(=O)NC(C(C)NC(c2onc(CC)c2C)=O)C)n[nH]c2cc(Cl)ccc12 C(=O)(C(C)(C)S(C)(=O)=O)N1C(CNC(CC2C(C)=NOC2=O)=O)CC1 c1(C(=O)NC(CC)CN(C(=O)CNC(c2cccs2)=O)C)cc(Cl)cnc1OC C(c1ccc(F)cc1F)=CC(N1CCCC(CNC(=O)CC2CC(F)C2)CC1)=O C(=O)(CC(C(C)(C)C)NC(=O)C=Cc1ccc[nH]1)NCc1ccc(C#C)cc1 N1(C(CSCc2c(C)nc[nH]2)=O)CCC12CCN(C(C1CC1(F)F)=O)CC2 C(=O)(C1=CCC(C)(C)CC1)N1CCN(C(C(CSC)O)=O)C(C(C)(C)C)C1 c1(CC(=O)NC2CCC(NC(CCOCCC)=O)C2)coc2ccccc12 c1(C(=O)NCCC(=C)CNC(C)=O)cncc(OCCC)c1.OCC c1(C(N)=O)ccc(NNC(=O)C2CCNC3(CCCCC3)C2)nc1 Nc1ccc(Cl)nc1C(=O)NCC1CC1CNC(c1ccns1)=O C1(C(N(CC(CC)NC(=O)C(c2ccc(F)cc2)O)C)=O)CC2C=CC1C21CC1 C1(NC(C=NOC)=O)CN(C(c2cnn(-c3ccccc3)c2C2CC2)=O)CC2CC12 c1(C(N2CC(C(C(=O)NCCCCN=[N+]=[N-])O)C2)=O)cc(F)ccc1F C(=O)(CCCCCS(N)(=O)=O)N(CCCCNC(C(C)Oc1cccnc1)=O)C Cc1ccc(OCC(=O)NC2CCC(F)(CNC(=O)C=Cc3cscn3)C2)cc1 C(=O)(C(F)(F)COC)N(CCNC(C1C(C)C1C)=O)CC c1(CNC2(CC(=O)Nc3ccc(C)c(O)c3Cl)CCC2)c(F)ccc2occc12 CCCC(C)C(=O)NCc1cc(C(=O)N(C)C(C2CCCCC2)C)on1 CC1Oc2c(C(=O)NC(C(F)(F)F)P(C)(C)=O)cccc2C1C c1(C(=O)OC)cc(NC(N2CCCC(C(F)(F)F)CC2)=O)cc(Cl)c1 N1(C(c2c(C)[nH]nc2CO)=O)Cc2occ(C(=O)NCc3ncc(F)cc3F)c2C1 C1(C(=O)NCc2cc[nH]c2C(=O)NCc2ccc(C)o2)(CC)CCCO1 C1(NCC(=O)NC(c2ccccc2)C(C)C)CNC2(CCCOC2)C1 C1(C(=O)NC(C(C)C)CNC(c2nnc(C(C)(C)C)s2)=O)(CO)CCCCC1 Cc1ccc(OC(C)C)cc1-c1nc(C2C(c3ccccc3)C2(C)C)no1 N1(C(CCCCCC#C)=O)CC2C3CCC(C2C1)N(C(=O)C1=CCC(C)CC1)C3 C1(=O)C2=CC3(CCN(C3)N1C(C1(C)CC3C=CC1C3)=O)C2.CC1CC1NC.C1CC1 C1(C(=O)NC2CN(C(c3ccn4ccsc34)=O)C2)Cc2ccccc2CO1 c1(OCC)cc(C)nc(Nc2ccc(NC(c3cc(Br)ccc3NC)=O)cc2)n1 Nc1ccc(CCC(=O)NCCNC(c2cccc(N(C)C)n2)=O)cc1F c1(C(N2CCN(C(C(CC(CC)C)C)=O)CC2)=O)cc2ccc(O)cc2[nH]1 c1(OC)ccnc(N2CC(NC(c3ccn(CCN(C)C)n3)=O)CC2C)n1 c1(C(N2CCCC(c3cn(CCCOC)nn3)C2)=O)cc(S(C)(=O)=O)ccc1F c1(CN2C3C(C(=O)NC(c4ccc(Br)s4)C)C(C3)C2)nccc2ccccc12 c1(C(N2CC(CC(=O)NCC(=C)C(F)(F)F)C(C)C2)=O)ccc2c(c1)CC2 C1(O)(C(=O)OC)CCN(C(=O)CCCN2CCCC2)C1.C12CCN(C1)C2=O N1(C(CCN(C)C(C2CCOC2=O)=O)=O)CC(=O)NCC1C(N1CCCC1)=O Cc1cc(Br)cnc1C(=O)NCC(C)(C)CN(C)C(c1nc(=O)n(C)[nH]1)=O Cc1cc(C2CC2NC(N2CCN(CCO)CC2C)=O)cc(O)c1 c1(C(=O)NC(C)CCN(C(=O)C(O)C(C)(C)C)C)cc2n(c1)CCOC2 Cc1ccc(C(=O)NCC(O)CNC(=O)C(C)(C)CN2CCN(C)CC2)c(C)n1 c1(SCCCNC(C2CCCC2(F)F)=O)cn(C2CCc3c(Cl)cccc32)nn1 O=C(C(F)C(F)(F)F)NC1CC(F)CN(C(c2cnccc2Cl)=O)C1 Cc1nc2ccccc2cc1C(=O)N(C1CCCN(C(C2(C(C)C)CC2)=O)C1)C c1(C(=O)NC2CCCN(C(Cc3cn(CC)nn3)=O)C2)cn2c(n1)COCC2 Cn1ccc2cc(NC(C34CC(NCc5cc(Br)c(F)cc5Cl)(C3)C4)=O)ccc12 C1(CC(=O)NC2CCCC(NC(=O)CC3(C)CC(F)(F)C3)C2)(OC)CCCCC1 c1(OC)ccc(F)cc1C(=O)C(=O)N(CCCNC(c1cocn1)=O)C C1(C(=O)NC2CCC(C3CC3)C2)(CC)CCN(C(c2cn[nH]c2)=O)CC1 C1(C)(CNC(C2CCC(CC)C2)=O)CCN(C(=O)CSCc2c(C)noc2C)C1 N1(C(c2cc(C)c(Br)s2)=O)CCN(C(=O)CN(C)C)CC12CC2 C=Cn1nncc1C(N1CCC(C)(CNC(=O)C(C2CCOCC2)OCC)C1)=O O=S(=O)(c1ccc(NCCc2ccns2)c(F)c1)N1Cc2ccc(CO)cc2C1 N#CC1=C(C(=O)NCCN2CCN(C(c3onc4c3CCCC4)=O)CC2)CCC1 c1(CN2CCC(c3noc(C)n3)(NC(C)=O)C2)cccc(Cl)c1O C1(F)(CNC(c2c(C)oc(C3CC3)n2)=O)CCCN(C(c2cn(C)c(O)n2)=O)C1 CC1(C#CC(=O)N2CCN(C(=O)CCc3cc[nH]n3)CC2C2CCC2)CCCO1 CC1(C(N2CC(CO)(NC(c3cnc(C(C)(C)C)[nH]3)=O)C2)=O)CC2(CC2)C1 CC1CCCN(C(=O)C(=O)NC2(C)CC(NC(=O)C(=O)NC3CC3)C2)C1 C1(NC(c2cnn(C)c2Cl)=O)CCCCN(C(=O)CN2CC3C=CC2C3)C1 C12CCC3CCN(C1C3)C(=O)c1ncc(cc1C)C1CN2C1.C(C(C)(C)C)=[SH]C Cc1cc(CCC(=O)N(C2CC2)CC2CCCN(C(c3ccon3)=O)C2)c(C)s1 c1(N(C)C)ccc2cc(C(=O)NCC3C=CCN3C(=O)C3=CCOC3)ccc2n1 c1(C(=O)NC(C(CO)SC)C)cc(Br)cc([N+](=O)[O-])c1N CC(C)(C)C(CC(=O)N1CCC(C(N)=O)C1)NC(C1(CO)CCCCC1)=O c1(C(=O)NC(CC)CN(C(=O)C(C)OCCOCC)C)cccc(C)n1 C(C)(C(O)C(=O)N(CCCN(C(=O)CCc1cccc(OC)c1)C)C)OC CCCC(CCO)N=c1[nH]c2c(c(=NCCOC(F)(F)F)[nH]1)SCC2 c1(C(C)=O)ccc2c(c1)CCN(c1nnc(C3CCSCC3)n1CC(C)C)C2 CCCCC(C)(CO)NC(=O)C(O)C1CN(C(=O)CCCC(C)C)C1 C1(C(=O)NCc2noc(C)n2)(SC)CN(C(=O)Cc2n[nH]c(C)n2)C1 c1(CC(=O)NCCC2(C(=O)NC3COCC3CO)CC2)ccc(O)cc1 N1(C(CCCCC#C)=O)CCCCC2(CCN(C(C3(O)CC3)=O)C2)C1 C(C)(CNC(=O)C=Cc1ccc[nH]1)(CNC(=O)C(C)(C)c1cnn(C)c1)OC c1(C(=O)NC(CCC)CC(=O)N2CCC=C(Cl)C2)ccc2ccoc2c1 c1(N(CCOC)CC)ccc(S(=O)(=O)N2CC(NC(C)=O)CO2)c(C)c1 N1(C(c2cccc(C3CC3)c2)=O)CC2CCC(C1)N2C(C12CCC(CC1F)C2)=O CC(C)S(=O)(=O)c1ccc(Cl)c(C(=O)Nc2c(Cl)cccc2C#N)c1 N1(CC)CC(NC(=O)C(C2CCN(C(c3cnns3)=O)CC2)C)CCC1=O c1(C(=O)NC(C(N2C(CC=C)CCCC2)=O)C2CCCC2)ccc2n[nH]cc2c1 N1(C(c2c(CCC)occ2)=O)CC(NC(C2CN(C(C)C)C2)=O)C(C)C1 c1(NC(c2csc(-c3cnc(C4CCCN4)[nH]3)c2)=O)ccc(-c2cncnc2)cc1 Cc1ccccc1C(=O)NCC(C1(O)CN(C(=O)C(F)CC2CC2)C1)(C)C c1(C(N2CCC(N(C(c3cn(CCC)nc3)=O)CC)C2)C)ccc(C#N)cc1 C(=O)(C(=O)C(C)C)NC(c1cn(C)nn1)C(=O)NC(c1c(C)ncs1)C C1(C(=O)NC(C)C(C)(C)NC(c2cccc(C3CC3)c2)=O)COCCC1(F)F c1(C(N2CC3CN(C(CCCCC=C)=O)C3C2)=O)cc2cccc(Cl)c2o1 C1(C2(CC(C(C)C)O)CC2)CCCCCC1.c12cn(nn1)C1(CC1)C(=O)N(C)C2 c1(NC(c2c(C)cccc2Br)=O)n[nH]c2c1CN(Cc1cccc3cc[nH]c13)C2 c1(C(=O)NCCCCCCNC(C2CC(F)C2)=O)cn2ncccc2n1 N1(Cc2nc(CCOC)on2)CCCCC(NC(=O)CCc2cnc[nH]2)C1 C(=O)(C(F)(F)CC=C)N1C2(CNC(CCNC(c3nc(CC)[nH]n3)=O)=O)CC(C1)C2 c1(-n2c(C3CN4CCN3CC4)nc(CCCCC)n2)ccc2c(c1)OCCO2 CC(F)(F)CCC(=O)NCC1(O)CCN(C(C2(c3ccc(Cl)cc3F)CC2)=O)C1 N1(C(C2C(=C)CC2)=O)CC2C3CCC(C2C1)N(C(=O)C1CCCc2cncn21)C3 c1(NC(C2CC(=C)CN2S(=O)(=O)C2CCC(=O)CC2)=O)nc(Cl)c2ccnc-2[nH]1 N1(C(Cc2c(C)ccnc2)=O)CCC2CC1CN2C(c1[nH]ncc1C#N)=O CC(Cc1cnn(C)c1)C(=O)NCCOCCCNC(C1(F)CC1)=O Cc1cccc(OC(C)C(=O)NC(C2C(NC(C3CC=CC3)=O)CCOC2)=O)c1 N1(C(CC2C(C)(C)C2)=O)CCCC1C(C)(C)CNC(c1ccoc1C1CC1)=O C(=O)(CCCS(C)(=O)=O)NCC1CC(F)(CNC(c2c(C)nc(C3CC3)o2)=O)C1 Cc1cccc(CCC(N2CCC(NC(c3cnoc3C)=O)C(C)C2)=O)c1Br CC1(O)CCN(C(C2(NC(=O)C=CC3CCOC3)CCC2)=O)C1 c1(C(=O)NC2(CC)CN(C(C3(n4ccnn4)CC3)=O)C2)cccc2c(C)[nH]nc12 c1(C(N(CCc2ccc(C)cc2)C)=O)cccc2c1C(C#N)C2 N1(C(c2cn(CC=C)nn2)=O)CCCC(O)(CNC(C2CCCCC2CC)=O)C1 c1(C(=O)NCC(CC=C)NC(c2ccc(C=C)cc2)=O)cc(F)ccc1C(C)C c1(CNC(C2CC(OC)(OC)C2)=O)cc(C)c(C(=O)NCCc2cnnn2C)o1 c1(NC(C23C(CN(C(c4ccccc4I)=O)C2)C3)=O)cc(O)cc(F)c1 CC(C)CCC(C)N(C)C(C1CCC(C)N1C(c1coc(N(C)C)n1)=O)=O C(=O)(C(C)(C)CCC#N)NCC1C2CN(C(C(C)n3ccnn3)=O)CC21 C1(CNC(CC(C(C)C)O)=O)N(C(C23CCOC(C)(C2)C3)=O)CCCC1(C)C N1(C(C2C(C)(C)COC2)=O)CCC(C)(C)C(NC(=O)CC2=NNC(=O)C2)C1 N1(C(Cc2nnc(C)o2)=O)CCC(CNC(c2cnc(C3CC3)o2)=O)C(C)C1 N1(CC(=O)N(CC(C)C)C(=O)COc2cc(C)on2)CCC(N)CC1.C(C)(C)(C)NC S(=O)(=O)(c1ccc(C#N)c(NCc2cc(F)ccc2Cl)c1)N(C(C)CS(C)=O)C N1(C(CCC=C)=O)CCCC(C(=O)NC2CCN(S(=O)(=O)CCCOCC)C2)C1 N1(C(CCC=C)=O)CCCCC1CCCNC(C1CC1OCC)=O N1(C(CC(C)(C)N(C(C=C(COC)C)=O)C)=O)CC2CC(C)C2C1 c1(CC)c(C(=O)NC2CC2CNC(c2ccc(C(F)(F)F)nc2)=O)nnn1C.COC N1(C(C2(C#C)CC2)=O)CCCCCC1CNC(=O)C(CC(C)C)NC(=O)NC c1(C2C(NC(N(CC(CC)C)CC)=O)C2)c(Cl)cccc1Cl CC(C)(C)CC(F)C(=O)NCC(c1ccccc1)NC(c1ccnc(CO)c1)=O CC1=NN(c2ccccc2)C(=O)C1NC(c1ccnc(-n2cccc2)c1)=O C1(C(N2CC3C(NC(c4c(OC)scc4)=O)(C3)C2)=O)CCCC(F)(F)CC1 C1(C(=O)NCCCN(C(=O)CCC2CC2(Cl)Cl)C)CCCCO1 c1(NCCCNC(c2c(C)nc(CCC)o2)=O)c([N+](=O)[O-])c(C)nn1C(C)C CC1CC(c2cn(C3CCC3)nn2)CCN1NC(=O)CS(=O)(=O)Cc1cccs1 C1(NC(C(C)CN(C)C)=O)CN(C(c2ccc(OC(F)(F)F)cc2)=O)CC12CC2 C1(C(N2CCCC(NCC(F)F)C2)=O)CCCC12CCOCC2 c1(OCCOC)cncc(C(=O)NCC(C2CCOC2)NC(C2(CF)CC2)=O)c1 c1(NCCC(C)OC)nc(=NCc2cc(C)ncn2)[nH]c2c(C)nn(C)c12 C12(C(=O)Nc3ncn(C)n3)CCC1CN(S(=O)(=O)Cc1ccccc1)C2 CC(C(=O)NC1CCCCC1NC(=O)Cc1cscn1)P(C)(C)=O N1(C(c2cc(CC)no2)=O)C2CCC1C(NC(=O)CC(C)(C)c1ccccc1)C2 N1(C(C2(CC=C)CCC2)=O)CC2(C1)CN(C(=O)C=Cc1ccc(OC)cc1)C2 C(=O)(C1=CC(O)CCC1)NC1COCCN(C(C2(CC)CC(C)(C)C2)=O)C1 FC1(CN=C(NC2CCCCC2)NC2CCN(CC(F)F)CC2)COCCOC1 N1(C(C2C(C)CC(=O)N2)=O)CCCC2CN(c3ccnc(CO)n3)CCC12 N1(CCC(=O)NCC(CCCC)NC(c2cc[nH]n2)=O)Cc2ccccc2C1=O c1(C(N(C(C)CN(C(=O)Cc2ccc(C#N)cc2)C)C)=O)ccc2nsnc2c1 CC1(C(=O)NC2CCN(C(c3c[nH]cc(Cl)c3=O)=O)CCC2)CCNC(=O)C1 C1(C#N)(CC(=O)NCC(C(C)(C)C)NC(CCc2cnn(C)n2)=O)CCOCC1 N1(CC)CCC(NC(=O)CC(C)(C)CNC(C2(C)COC2)=O)C(C)C1 C1(C(N2CCC(F)(CO)C2)=O)C(O)CCN1C(=O)C(c1cccc(Br)c1)O CC1C(NC(c2cccc[n+]2[O-])=O)CCCN1CCCOc1ccccc1 c1(NC(C)Cc2ccccc2)ccc(S(=O)(=O)NCC2(C)CCOC2)cc1C#N CC1(C)CCC(C(N2CC(CC(F)F)C2)=O)(NC(=O)CN2CCNC2=O)C1 C(=O)(C1OC(=O)c2ccccc21)N1CCC2(OCCN(C(C(C)(C)SC)=O)C2)C1 c1(N(C(c2ccc(-c3ccsc3)cc2)C(=O)NC2COC2)C)ccnc(Br)c1 CC1CCCn2ncc(C(=O)NC3C=CC(CNC(C4CC(O)C4)=O)C3)c21 N1(C(CN(CCC)C)=O)C2CCC1CN(C(c1cccc(C)c1O)=O)C2 C1(C(=O)OC(CC)C(=O)N2CCCCC2)(C(=O)OC)CC(C)=C(C)C1 C(=O)(CS(=O)(=O)C(C)(C)C)N(CCCCCCNC(C1CCCC(CF)C1)=O)C C1(C(=O)NCC(CC)(C)CC)CC(C)(C)CN1C(=O)CC(CC)OC C12(NC(c3c(Cl)cc(C)c(C)c3)=O)COCCC1CN(C(c1cccnn1)=O)C2 c1(C(N2C3CN(c4nccc(Br)n4)CC23)=O)cn2ccc(Cl)cc2n1 C#Cc1ccc(Cl)c(C(N2CC3CCN(C(c4cc(C)oc4C)=O)C3C2)=O)c1 Cc1cc(NC2CCN(C3CCC3)C2)nc(NC2CC2c2ccccc2Br)n1 CCCCCC(O)CC(=O)N1CCC(CNC(=O)C(C)CC2CCCC2)CC1 CCCCCCCCC(F)C(=O)NCCCN(C(=O)C(O)C(C)C)C1CCCC1 N1(C(CNC(C2CCCSC2)=O)C(F)F)CCN(C(=O)Cc2ccsc2)CC1 c1(OC)c(C(N2CCC(NC(=O)C=CC(F)(F)F)CC2)=O)c(C)nn1C C=C1CCC(C(=O)NC(C)CCCCNC(c2ccncc2C(F)(F)F)=O)CC1 CC(C)CCCC(=O)N1CCC12CN(C(=O)CC1(O)CCC1)C2 c1(C(=O)NC(C(C)C)CCN(C)C(C2CC23CC3)=O)ccc2[nH]ccc2c1F S(=O)(=O)(c1nc(N2CCOC(C3CCC3)C2)ccc1Br)NCC1(CC)CCCO1 N1(C2CCN(C3CCN(C)C3=O)CC2)CC(=O)Nc2ccccc21.C12CCCC1S2 c1(COC)nc(C(=O)N(C(C(=O)NC(C)Cc2nccn2C)C2CC2)C)co1 c1(N(CCc2n(C(CC)C)nc(-c3ccc(Cl)cc3)n2)C)cc(C)ccc1C C1(C)(C(=O)Nc2c(OC)cccc2)CCN(C(=O)Cc2ccc(Br)nc2)CC1 C(=O)(C(C(=O)NCC(O)CNC(c1cc2cnn(C)c2s1)=O)C(C)(C)C)OCC CCCC(O)C(=O)N(CCCCCNC(=O)CC1COC(C)(C)C1)C Cc1c(F)ccc(C(=O)NC2CC(CCNC(=O)CCCC(C)(C)C)C2)c1Cl N1(C(c2c(Cl)n[nH]c2C2CC2)=O)CCC2CCCN(Cc3ccccc3)C2C1 c1(C(N2CC(O)(CN(C(CC(n3ccc(C)n3)C)=O)C)C2)=O)c[nH]ccc1=N N1(C(CCN(C)CC)=O)CC2(CC(CNC(=O)CCc3cc(C)nc(C)c3)C2)C1 CCC(CC(=O)NCCn1ccnc1)N(C)C(C1CC(OC(C)(C)C)C1)=O C(=O)(CCC(C)S(C)(=O)=O)N(C1CCN(C(=O)CNC=O)CC1)CCC N1(C(c2cn(C)nc2C2CCCC2)=O)CC2CCCC(C1)N(C(=O)C=C(Cl)Cl)C2 CC(C)C(C#N)C(=O)NCc1nnn(C)c1C(=O)NCC1CCCOC1 C1(CC)CN(C(=O)CCS(C)=O)CCN1C(C1C2CCC1(c1cscn1)C2)=O c1(C(N2CCN(C(CC(=O)NCC)=O)C3C2C3)=O)ccc2c(c1)ncn2C c1(CS(N2CCN(CC(=O)N(C)C)CC2)(=O)=O)cccc(C#N)c1 c1(C(=O)NCC2CN(C(CC3CC(OC)C3)=O)CC2(C)C)cn2ccnc2cn1 C(CCCCCNC(=O)CN(C)CCO)N(C(c1c(C)n[nH]c1)=O)C CCCCC(C(=O)NC1CC2(C1)CC2NC(C1CC(C)C1)=O)NC(N)=O C1(C(=O)NCC2CCN(C(C3ON=C(CC)C3)=O)C2(C)C)CC2(CCCC2)CO1 CC1CN(C(=O)Cc2ccn(C)n2)CCS1(=O)=O N1(C(CC2=NNC(=O)C2)=O)CC(C2CCCCN(C(c3scnc3Cl)=O)C2)C1 C(=O)(C#CC(C)(C)C)NC1C=CC(CC(N2CCC(C(C)CO)CC2)=O)C1 C1(CNC(Cc2c(C)scc2)=O)CCCCC1NC(c1cnn(C)c1F)=O C#Cc1cccc(CNC(=O)CCCN(C(=O)C(=O)NC2CC(OC)C2)C)c1 C1(C(N(C2CCCC2)CCNC(CC(=O)OC)=O)=O)CCn2cc(C)nc2C1 C(c1ccccc1F)=CC(N1CC(C(C)NC(C2CC2c2cccs2)=O)C1)=O C12(CNC(CCCC)=O)CCCC1N(C(=O)Cc1cc(F)ccc1Br)CC2 c1(C(N2C(CNC(C3CN(C)C(=O)N3)=O)CCC2)=O)coc2c(Cl)cccc12 CC1CN(C(=O)Cn2cnc(C#N)n2)CCC1NC(=O)C(=O)NCC1CC1 C1(CNC(C(c2ccc(Cl)cc2)(C)C)=O)CN(C(C2(C)CC2(F)F)=O)CCO1 N1(C(c2ccc(C)o2)=O)CC2CCC1C1CN(C(C3CC(n4cnnc4)C3)=O)CC21 c1(COC)ncc(C(=O)N(CC(C)(C)CNC(=O)Cc2cccs2)C)c(O)n1 C1(NC(c2c(C)ncs2)=O)CN(Cc2ccc(O)cc2OC(F)(F)F)CC1C#N CC(C)CC(C)CC(=O)NCCn1cc(C(=O)NC(C)CCC(C)(C)C)nn1 c1(C(N2CC(CNC(C(C)n3cccc3)=O)C2)=O)ccnc(N2CCC(C)C2)c1 N1(C(CNC(=O)OC)=O)C2CCCC1CN(C(C1(C#N)CCOCC1)=O)CC2 C(CC(O)C(=O)NC12CC(NC(c3ccc(C4(O)COC4)cc3)=O)(C1)C2)N(C)C c1(C(=O)NC2CCN(C(=O)C(c3ccccc3Cl)O)C2)cccc(C(F)(F)F)n1 O=C(C1=NOCC1)N1CCC(c2ccccc2)CC1.c12nocc1C(=O)NOC2 C1(CNC(CN(S(C)(=O)=O)C)=O)(CO)CCN(C(C2OCCC2C)=O)CC1 C1(C(N(C)CCNC(=O)CN2CCOCC2)=O)CCCC1S(C)(=O)=O n1(CC(=O)N(C2C(C)CCN(C(C3(CO)COC3)=O)C2)C)cnc2ccccc12 CC1(C#CC(=O)N2CCCCC2CCCNC(C2CCC3CC23)=O)CC1 N1(C(CC2(CC)CC2)=O)CCCC(C(=O)OC)C1.C1=CC(=O)Nc2ccc1o2 c1(C(N2CC(C(C)NC(C=Cc3c(C)nccc3)=O)C2)=O)ccn2nnnc2c1 N1(C(c2n(C)cc(Cl)c2)=O)CCCN(C(C2CC3C=CC2C3)=O)CC1 Cc1[nH]nc2ccc(C(=O)N(C)CCOCCCN(C)C(c3cc[nH]c3)=O)cc12 c1(NC(C2(SC)CN(C(=O)Cc3cscn3)C2)=O)c[nH]ccc1=O C1(c2cccnn2)(N(C)CC2(CO)COC2)CCC(P(C)(C)=O)C1 c1(C(N2CCN(c3c(F)cnc(C)n3)C(CC#N)C2)=O)cnc2[nH]ncc2c1 c1(C(=O)NCC(C)(C2CC2)NC(C(CC=CC)CC)=O)ccc2nn[nH]c2n1 CC1(C)CCC(CNC(C2(C)CC2(C)C)=O)N(C(c2cnc(S)nc2)=O)C1 C(CCC(=O)NCC(CNC(=O)C(c1cnn(C)c1)OC)CO)N(C(=O)OC)C C(c1ccccc1)=CC(=O)NC(C1CCCCC1)CO c1(NC(c2cn(CCN(C)C)nc2)=O)ccccc1C1CCCCC1 C(=O)(CCCC(C)(C)C)NC1CC1CN(C)C(C1(COC)CCC1)=O C#CCC(C)(C(=O)NCC1CC12CC2(F)F)NC(c1cn(C)nc1OC)=O C1(C2CCC2)(C(=O)NCC(CNC(C2(C(F)(F)F)CC=CCO2)=O)OC)CCC1 c1(C(=O)NCC(CNC(C(C)(c2cccs2)N(C)C)=O)(C)O)ccc(F)cc1F N1(C(CCCOCCOC)=O)CCC(C)C(CNC(=O)CC2=CCCC2)C1 c1(C(=O)OC)ccc(-c2ccc(CNCCN3CCN(C)CC3)cc2)nc1N Cc1cc(C(N2CC(F)CC2CNC(=O)C(C)(C)Cc2cnn[nH]2)=O)ccn1 c1(N(C)C)cccc(C2(C(=O)NCC3CC3NC(=O)CC3CCCC3)CC2)c1 N1(C(c2cn(C(C)C)c(=O)cc2)=O)CC(NC(=O)CCC2CCC2)C(C2CC2)C1 C1(C(=O)NCC(CN(C(C2C(CC)C2)=O)C)C)C(C(F)(F)F)C1[N+](=O)[O-] c1(C(C(=O)NCC(C)(C)NC(CC(C)SC)=O)O)cc(F)c(F)c(F)c1 N1(C(C2CCC(C)CC2)=O)CCC(CNC(=O)CCc2cccs2)C(O)C1 c1(CCCC(=O)NCC2C(NC(C3(C(C)(F)F)CC3)=O)C2)ccc(Br)cn1 C1(NC(C(C)NC(CC)=O)=O)CN(C(C2CC(N3CCOCC3)C2)=O)CC1F N1(C(C2N(C(C(C=C)(F)F)=O)CC3CCCC32)=O)CC2CCC1C(O)C2O Cc1cnc(C(N2CCN(C(C3CC(=O)N(c4ccccn4)C3)=O)CC2)=O)cn1 N1(C(=O)OC(C)(C)C)CCSC(CNC(=O)Cc2cnccc2Cl)C1 c1(C(=O)OC)ncc(C)cc1C.c12ncccc1NC(=O)N1CCN2CC1 c1(OC)cc(NC(c2nnnn2-c2ccc(Cl)cc2F)c2cocn2)cnc1Br N1(C(C(CC(C)C)NC(C)=O)=O)CCCC(C2CN(Cc3cc(Cl)ccc3O)C2)C1 N1(C(CNC(CNC(C2CN(C)C2)=O)=O)=O)CCCC(CN(C)C)CC1 C1(NC(Cn2ccc(C)n2)=O)CN(C(=O)CCCCC(C)C)C2CCCC12 C1(NC(C(CSC)C)=O)CN(C(=O)CSC(C)C)CCC1c1ccc(F)c(F)c1 c1(-n2cc(CN3CCN(C(C(CC)CO)=O)CC3)nn2)cc(Cl)ccc1CO N1(C(C=C(CCC)C)=O)CC2(CCCCN2C(c2cc(C)co2)=O)C1 C1(CNC(Cc2cc(C)nn2C)=O)CN(C(C2CCC(=O)N2C)=O)CC(C)(C)C1 C1(CCNC(=O)CC2CCCC2)CN(C(c2ccsc2Cl)=O)CCCO1 C#Cc1ccc(C(=O)NC2(CCCC(=O)NCC(C)CC)CCC2)nc1 CC1(C)CCCC(C(=O)NCC2CCC(C(N3Cc4ncsc4C3)=O)O2)C1 c1(C(=O)NCCC(C)NC(CC2(CC=C)CCCC2)=O)n[nH]c2ccc(O)cc12 C1(CC(=O)NCCN(C(C)C)CC)CC(O)CN1C(=O)CCc1ccco1 c1(C(C)=O)ncnc(NC2CC(F)(CNC(=O)COCc3ccccc3Cl)C2)n1 c1(C(C)C)ccsc1C(=O)NCC1COCC1NC(C1COCCO1)=O C1(C(=O)NCC2C(CNC(c3ccc4nn[nH]c4n3)=O)C2)CCc2nn[nH]c2C1 C1(C)(C(N(C2CCCC2)C)=O)CCCN(C(=O)Cc2c(Cl)cccc2Cl)C1 C1(NC(CC(n2c(C)cc(C)n2)C)=O)CCN(C(c2n[nH]cc2F)=O)C(C)C1 CCC(C)(C#N)C(=O)NCC1CN(C(=O)C(C2CCCCC2)O)CCO1 n1(CC(C(=O)Nc2cccc(C(CC)C)c2)(C)O)c(C)cccc1=O C1(CCNC(c2ccc(F)s2)=O)CC(F)(F)CN1C(=O)COc1ccc(O)cc1 Cc1c(C(N2CC(N(C)C(C3CC(F)C(=O)N3)=O)C2)=O)[nH]c2cc(F)cc(F)c12 Cc1cccc(C(N2CCCC(C3CCCN3C(=O)CC(C)(C)C#N)C2)=O)c1C S(=O)(=O)(CCC(F)(F)F)NCCc1cccnc1.n12ccc(nc1=O)NC(=O)C2 C1(NC(c2cn3ccnc3s2)c2n(C(CC)C)nnn2)Cc2ccccc2C1 C1(C(N(CC(=O)NCC(C)F)CC)=O)C2(CC2)C12CC2 c1(C(N2CC3(CC(CNC(COCC#C)=O)OC3)C2)=O)cn2ccc(C)cc2n1 c1(NCc2ccc(C)o2)nc[nH]c(=NCC2(C)CC2(C)C)c1C CC(C)CCC(F)C(=O)NCC(O)CC(N1CC(CO)C(C)(C)C1)=O Cc1oc2cc(C(=O)NCC3CCCN(C(C4(CO)CCCO4)=O)C3)[nH]c2c1C c1(NC2(c3n(CCCC)nnn3)CCCC(C)C2)ccc2cc[nH]c2c1 C123CCC(CO1)(C2)NS(=O)(=O)C3.c1(C(=O)OCC)sc(C(=O)OC)cc1N C1(CC(C)NC(c2scc(COC)c2)=O)CCN(C(C2(C#N)CC=CC2)=O)CC1 N1(C(C(C)N(CCC)C(c2cn(C)ccc2=O)=O)=O)CC(C2=NOC(C)C2)C1 N1(C(C(C)CC(F)F)=O)CCN(C(=O)C(C)(C)COC2CCCC2)C2(CC2)C1 c1(CN(C)CCc2ccc(F)cc2)nccc(C)n1.Cc1nnc(N)s1 N1(C(CCCCC)=O)CC(C(=O)NCc2ccccc2CO)C2(CC2)C1 Cc1coc2ccc(CC(N3CCCC3(C)CNC(=O)C(F)(F)C(F)F)=O)cc12 c1(C(N(C2CC2)CC2CCN(C(C=CC)=O)CC2)=O)cnc2n1CCCCC2 N1(C(CCCN(C)C)=O)CCC2CC2(NC(=O)CSc2nncs2)CC1 C1(CNC(C(CSC)OC)=O)CCN(C(C2(c3ccncc3)CC2)=O)CC1C C1(NC(c2cccc(C(N)=O)c2)=O)CN(C(=O)Cc2csnn2)CC12CC2 CCCCCCCC(=O)NC1CC(NC(c2cnn(C(C)C)c2N)=O)C1 c1(C2C(NC(CN3C(C)CC3)=O)C2)ccccc1C(F)(F)F c1(C(=O)NC2C=CCN(C(C3(F)CCCCC3)=O)C2)c[nH]c2nc(F)ccc12 Cc1ccc2c(c1)CNCCN2S(=O)(=O)CC(C)C(F)F C1(NC(C(C)(C)c2ccccn2)=O)CC(O)CN(C(C2CCC(C#N)CC2)=O)C1 c1(C(N2C(CN(C(CS(CC)=O)=O)C)CCCC2)=O)cnc2c(=O)[nH]ccc2c1 c1(CC(=O)NC(C(C)C)Cn2ccnc2)cc(C(F)(F)F)nn1C C1(N(C(c2cc(OC)n(C)n2)=O)C)CN(C(c2cc(C)ccc2C)=O)CC1(C)C c1(C(=O)NCC(CNC(C(C(CC)C)NC(=O)OC)=O)O)cc2n(n1)CCOC2 N1(C(CCc2c(C)noc2C)=O)CCCC(F)(CNC(C2CC(F)CN2C)=O)C1 C(C#Cc1cn(-c2ccc(Cl)cc2)nn1)NC(C1CCCC1C1CC1)=O C(=O)(C(CC)C(=O)NCCOCC(=O)N(C(C)C)Cc1cccs1)OC C(=O)(C(C(=O)N1CC(CNC(c2coc(C(N)=O)c2)=O)C1)OC)OC C=CC1(C(=O)Nc2cccc(C)c2)CCN(C(=O)C(F)CC(C)(C)C)CC1 C1(C(=O)NCCOCCN(C)C(c2ccnn2CC2CC2)=O)C2(CC2)C12CC2 c1(C(=O)NC(CCCNC(CC2ON=C(CC)C2)=O)C)nnc2n1CCCCC2 C1(C(=O)NCCC(C(C)C)NC(C23CCC(F)(CC2)C3)=O)CCCCC(=O)CC1 c1(C(N2CCC(C)C(NC(c3ccnn3C3CC3)=O)C2)=O)ccc2nn[nH]c2c1 C#Cc1cc(NC(C23CC(C)(CN2C(c2cc(C#N)[nH]c2C)=O)C3)=O)ccc1C C=CCCCCCCCC(=O)NC(CN(C(=O)C(C)=C(C)C)CC)CC N1(C(CCCC=C)=O)CCCC1C1CCCN1C(c1ccc(C#N)c(O)c1)=O C1(C(=O)NC(C2CCN(C(=O)OC(C)(C)C)C2)C)CCCN1CCC1CC1 C12CN(CC1(C)C)C(CCCC1CCC1)C(=O)N2.CC(C)(C)OC(C)(C)C c1(C(=O)NCCC(C)NC(=O)C=CC2CCCO2)ccc2nnn(O)c2c1 CCC1=NOC(C(=O)N(CCC(=O)NCCOC)CCO)C1.C1(CC)CCC1 Cc1cc(F)c(C(=O)NC(CNC(c2cnc(-c3ccco3)s2)=O)CO)c(Cl)c1 C(=O)(CC(C)C(=O)OC)NCCOC1CCN(C(CNC(=O)OC)=O)C1 C#Cc1cnc(C(N2CCC(N(C)C(C34COCC3C4(F)F)=O)C2)=O)c(C)c1 C(=O)(C1CCCc2c[nH]nc21)N1CC(NC(C(CCC)C)=O)(CC)C1 N1(C(CCOC)=O)CCCC2(CCCCC2NC(=O)CCC=CBr)C1 CC(C)(C#N)CCC(=O)NC1CC2CC(NC(C3(C)CCCCO3)=O)CC2C1 C#CCC(CC(=O)Nn1cnnc1)NC(=O)C(N1CCOC1=O)C CCCCCCC(C)(C)C(=O)NCC1CC(C(F)(F)F)CN1C(=O)CC(F)F C(=O)(C(C)CCC(C)(C)C)N(CCCCC(=O)NCc1cc(C)sc1)C c1(C(=O)OC)cccnc1C(=O)NCC1(CNC(C2CC(C)(C)CO2)=O)CC1 c1(NC(N2CC(C)(C(=O)OCC)OCC2)=O)coc2ccc(OC)cc12 N1(C(COC(CC)CC)=O)CCCC(NC(C2(Br)CC2)=O)C1C N1(C(C=C(CNC(COCCCC)=O)C)=O)CCCC(N(C)CC)C1 C(=O)(C(F)(F)C(F)F)NCC(C)(CNC(c1cncn1C1CC1)=O)OC C12(C(N(CC(N3CCN(C(C(CC)(F)F)=O)CC3)=O)C)=O)C3CC(CC13)C2(F)F C(=O)(CC(F)(F)Cl)NCC(C)(O)CNC(=O)Cc1ccc(OC(F)F)cc1 C1(C(=O)NC(COC)C(=O)OC)C(C2CC2)CCN1C(=O)CCC(CF)CF C12(NC(CC(=C)C)=O)CCCCCC1N(C(=O)CCCN(C)C(=O)OC)CC2 C1(CC(=O)NC(CNC(C(C2CCCCC2)C)=O)CO)C=NN(C)C1=O C1(C(N(C(C)C(=O)NCc2cccnc2)CC)=O)CCCSC1C C1(C(=O)NC2CC3(C(NC(C=C4CCC(C)CC4)=O)C3)C2)CCCCN(C)C1=O C(=O)(C1=C(C2CCOC2)N(C2CC2)C(=O)NC1c1nc(Br)cs1)OC N1(C(c2c(C)cc(C#N)cc2)=O)CCC2OCCN(C(C3CCCOC3)=O)C2C1 c1(C(C(=O)NC(CC)CNC(=O)C(C)n2ccnc2)C)cncnc1 N1(C(C(C)c2ccco2)=O)CCCC(CCC(=O)N(C2(C)CC2)C)C1 C1(n2cc(C(C3CC3)OC)nn2)CC2CCC1(NC(=O)Cc1cccc(Cl)c1F)C2 c1(C(=O)NCC(CC)NC(c2cn(C3CCC3O)nn2)=O)cc(C)c(F)cc1Cl C(=O)(C(C)(C)CF)N1CC(OCCNC(C=COCC)=O)C1 c1(OC)cc(C(=O)NCC(C)NC(c2n[nH]c(C3CC3)c2Cl)=O)cc(Cl)c1 C1(C(=O)NCCC(C(C)C)OC)CCCCCCN1C(c1cccc(F)c1C)=O C1(=CC(=O)NC2CC3CN(C(C(C(CC)C)C)=O)CC32)C2CC3CC(C2)CC1C3 Cc1cc(O)c(C(N2CCC(NC(C3CC(C)CO3)=O)C2(C)C)=O)nn1 C1(NC(C2CC(C)CN2C(=O)CC2CCC(=O)N2)=O)CC(C)(C)C12CC2 C(CCC(=O)N(C)CCOCCN(C(=O)C(C)N(CC)CC)C)OCC c1(C(=O)NCCc2c(CNC(C3ON=C(C)C3)=O)nco2)cnn(C)c1Cl C1(C(=O)NC(C(C)SC)C)CC(C)(NC(C2CCC2C#N)=O)C1 N1(C(CN(C)C(C2CC3CCC2O3)=O)=O)CCN(C(=O)C(F)CC2CCC2)CC1 C(CN(CC1CC=CCC1)N(C)Cc1cnn(C)c1)OC N1(C(c2scc(OC)c2)=O)CCCC(C(=O)NCCN2CC=CC2)C1C N1(C(C2CN(C(C)C3CC3)C(=O)C2)=O)CCC(C)N(C(=O)Cc2ccoc2)CC1 [N-]=[N+]=NCCCCC(=O)NCC1CCCC1NC(c1ccc(C(F)(F)F)[nH]1)=O CON1CCC(CC(=O)NC(CO)C(C)NC(c2cc(CN(C)C)on2)=O)CC1 c1(CC)nc(C)c(C(=O)NCCC2CCCN2C(=O)CCc2ccnn2C)s1 c1(C(N2CC(C)(NC(C=CC(CC)=CC)=O)C2)=O)ncn2ccccc12 c1(C(=O)OC)ncccc1C(=O)NC(C1CCN(C(c2cc(F)c[nH]2)=O)C1)C C(=O)(C(C)(O)CC(C)C)N1CCN(C(CNC(CC2C(C)=NNC2=O)=O)=O)CC1 c1(OC)cc(C#N)ccc1NC(=O)C(C)OC(=O)C(F)C1CCC1 c1(C(N2CC(NC(C3C4COCC34)=O)C(F)CC2)=O)cccc2nc[nH]c12 Cc1ccn(CC(C)C(=O)NC(CNC(c2sncc2Br)=O)CO)n1 C1(NC(c2nccc(OC)c2F)=O)CN(C(=O)CC2(CO)CCC2)CC12CCC2 CN(C)S(=O)(=O)N(C)CC(=O)NC1CC1NC(c1cc2c(s1)CCC2)=O CC(C)CC(O)C(=O)N1CCCCC(CNC(c2cnc(Cl)n2C)=O)C1 CC(C)C(C(=O)NCCN(C(=O)CCCC#N)C1CCCCC1)NC(N)=O C(CCCC(=O)NC(C1CCCC1)CNC(C1(Cl)CC1C(C)=O)=O)N(C(C)=O)C C1(C)(C(=O)NCCCCN(CCCNC(=O)CCc2ccon2)C)CCCS1 N1(C(C2(C)N(C(CS(CC)(=O)=O)=O)CC(O)C2)=O)CC2CCCC(O)C2C1 C(CNC(C1CC2CCC1CC2)=O)(CC(F)(F)F)NC(C(C(C)C)SC)=O N1(C(COCC#C)=O)CCC2(CCCN2C(c2coc(COC)n2)=O)CC1 c1(C(=O)NCc2c(C(=O)NCCC[Si](C)(C)C)occ2)ccsc1C#N N1(C(COCCCCCC)=O)CCC(C(=O)NCCCc2cccs2)CC1 CCC(C)CCCC(=O)NCC1(C)CCCN1C(c1cc(C(C)C)oc1C)=O CCC1=C(C(=O)NCCCNC(c2nccc(OC)c2N)=O)SCCO1 CCS(=O)CC(=O)NCC1CN(C(c2ccnc(F)c2)=O)C1 CC1(C)C(CC(N2CCC(N(C(=O)CO)Cc3ccncc3)CC2)=O)CC1O N1(C(c2c(C)ncn2O)=O)CCC(NC(c2ccsc2Cl)=O)C(F)(F)CC1 n1(CC(N2CCN(C(C(CC)C)=O)CC2COC)=O)cc([N+](=O)[O-])c(C)n1 c1(CC(N2CCC(O)(CF)C(O)C2)=O)ccc2c(c1)CN(C1CCNC1=O)CC2 Cc1cc(Br)ccc1C(=O)NC1CCN(C(C2CC2F)=O)CC1O c1(C(=O)NCC2C(CNC(=O)CSCc3ccccc3Cl)C2)cc2cccn2cn1 N1(C(CC(C=C)C)=O)CCC2C(CCN2C(c2csc(C(C)(F)F)n2)=O)C1 C12(C(=O)NC3CC(NC(Cc4c(C)nc(C5CC5)s4)=O)C3)CC=CC(C1)OC2 C(C(C(=O)NCCn1cc(CO)nn1)NC(=O)C(O)CC1CCCC1)SC N1(C(C(C)N(C)C)=O)CC2CC(C1)N(C(=O)Cn1cc(Br)cn1)C2 N1(NC(C2CC(N(C)CC)C2)=O)CCN(C)CC1CO.c12cncc(c1)C(=O)C2 C1(OC)CCCC1C(=O)NC1(n2cncn2)CC1.N12CCCC1CNCC2=O CC1CN(C(C2C(CNC(c3cnsn3)=O)C2(C)C)=O)CC(C)(C)C1 C(CC(C)(C)CC(=O)NCCC1(NC(C2SCC=C2C)=O)CCCC1)OC CCCS(=O)(=O)NC(C)C(=O)N(C1CC(NC(=O)COCC)C1)C c1(C(=O)NC2CN(C(C(CC)C#N)=O)CC2C)cnc2ncnn2c1O C1(NC(C2CCC(O)CC2)=O)CC2CCC(C1)N2C(c1ccns1)=O c1(NC(C2(C(C)NC(=O)CC3CCCCO3)CC2)=O)cncc2ccccc12 CCC(CC)(C(C)C)NC(C1CCCC1NC(c1sccc1C)=O)=O C1(CNC(C2(COC)CC=CC2)=O)C(C)CCCN1C(=O)CCC1CC1(C)C CCC(C)C(CC(=O)NC1CN(C)CC1C)NC(=O)C(C1CCC1)OC S(=O)(=O)(CC(=O)NC(C(=O)NCC1(C)CCCOC1)C1(O)CCC1)NC N#CC1(C(N2CCC(O)(CNC(=O)Cc3ccco3)C2)=O)CC2CCC1CC2 c1(C(N2CCC(OCCNC(CS(C)(=O)=O)=O)C2)=O)ccc2c(c1)COCO2 c1(CC(=O)NCC(C)N(C(c2nc(C(C)OC)sc2)=O)C)cccc(C#N)c1 c1(N2CCC(C(C)C)CC2)nc2ccc(Cl)cc2c(=NC2CCCCCC2C)[nH]1 c1(C(N2CCC(NC(CC=C=C)=O)CC2C2CC2)=O)cncc2c[nH]nc12 C#CCCC(C(=O)NC1CCN(C)C1(C)C)NC(=O)C(CC)OCC C12(CC)CN(C(=O)C(c3cc(F)cc(F)c3)O)C(CNC(=O)C(C)COC)(C1)C2 C1(NCC2CCC(C)N(C(=O)OC(C)(C)C)C2)CCCC(F)(F)CC1 C(=O)(CCC(F)F)N(C1CCN(C(=O)C(c2ccc(Cl)cc2)CO)C1)C c1(C(=O)NCC2C3CN(C(=O)CC4OCCCO4)CC23)occ2c1CCC2 N1(C(=O)C=Cc2cc[nH]c2)CCN(C(C23CCCC2C3(F)F)=O)CC1CCO c1(CC2CCS(=O)C2)nc(-c2ccc(N3CCCC3)nc2)nn1-c1cccs1 C1(OC)(CNC(C2(C)CCSCC2)=O)CCN(C(=O)Cn2nc(C)nc2C)C1 CC1CC2(CC(C(N3CC(O)CCC3C(=O)NCC3CC(C)(C)C3)=O)C2)C1 N1(C(C2(CCC)CC2)=O)CC2(CC(NC(=O)C(C)OCc3cccc(C)c3)C2)C1 C(CCCCCNC(=O)Cn1ccnn1)N(C(=O)C=CC(c1ccc(F)cc1)=O)C N1(C(c2c(C)coc2)=O)CCN(C(=O)C(C)NC(=O)C(C)(C)C)CCC1C C1(C)(C(=O)NC(c2ccncc2)C)CCN1Cc1cnc(-c2ccccc2)[nH]1 c1(CC)nc(C)c(CC(N2CCC(C)(CNC(=O)C(C)CC)CC2)=O)c(C)n1 C1(C(F)(F)F)(CC)CN(C(c2cn(C)nn2)C(=O)NCC2CCOC2)CCO1 c1(OCCOC)ccc(CC(=O)NCCC(O)CNC(c2cccs2)=O)cc1 C=CCC(C)C(=O)NCC(C1CC1)NC(c1oc(-c2cnn(C)c2)nc1C)=O c1(CC)noc(C)c1C(N1CC(CNC(c2ccncc2OC)=O)C(O)C1)=O C1(CNC(C(F)=C(C)C)=O)CN(C(c2csc(C)c2N)=O)CCC12CCC2 c1(C(N2CC(NC(CN3CC(C)C3)=O)C(F)C2)=O)cccc([N+](=O)[O-])c1Br c1(C(C=CCNCCC)NC(=O)C(C)C)ccccc1 C(N=c1[nH]c2cc(Cl)cc(Cl)c2o1)C1C(C)CN(C(c2cnn(C)c2N)=O)CC1 C(=O)(CCCC(=O)NCC1(OC)CN(C(c2cccnc2Cl)=O)C1)NC C1(NC(CC=C=C)=O)CCN(C(C2CC(C3CCC3)C2)=O)CC1(C)C C1(F)(C(=O)Nc2ccc(Cl)cc2)CCOCC1.n12cc(nn1)C(=O)N1CC2C1 C=CC1CN(C(=O)C(C)P(C)(C)=O)CC1NC(=O)CC(C)(C)COC C(=O)(CCCCCCn1cc(CCCCO)nn1)Nc1c(C)cc(O)cc1 N1(C(c2cc(CC)no2)=O)CC(OC)CC1(C)CNC(=O)CN1CCCC(CC)C1 C1(NC(c2scc(C)c2)=O)CCC2(C1)CN(S(=O)(=O)C(F)(F)F)C2 C1(F)(CNC(c2cccc(F)c2Cl)=O)CCCN(C(c2cscn2)=O)C1 C(C)(N=c1[nH]c(=NC2CCCC2)[nH]c2cc[nH]c12)c1c(C)nc(C)[nH]1 C1(NC(C(C(C)C)C)=O)CCN(C(C2CCC3(C2)N=N3)=O)C12CCCC2 c1(OC)n[nH]cc1C(=O)NC(C(=O)NC(CO)CCF)C1CCCO1 C1(CNC(c2ccc(CSC)o2)=O)CN(C(c2cnc(Cl)[nH]2)=O)CC1C(F)(F)F c1(CCC(=O)NC(CNC(c2cccc(F)c2)=O)CO)cccnc1F c1(COC)nc(NCCCOC(C)C)cc(=NC2CCOC(C)(C)C2)[nH]1 C1(CC)(CNC(C2COCCC2NC(=O)Cc2cn(C)cn2)=O)CCCCC1 C#CCCCCCCC(=O)NC1(CF)CCN(C(c2ncnc3c2CCC3)=O)C1 Cn1cnc2ccc(-c3cccs3)cc12.C12CN(CCO1)C(=O)C(=O)N1CC2C1 c1(C(CNC(c2sncc2C)=O)NC(C(C)(C)NS(C)(=O)=O)=O)cccc(C)c1 C(=O)(CC1C(=O)Nc2ccccc21)N(C)CC1CCN(C(C=CC=CC)=O)C1 c1(C(=O)NC2(CN(C)C(C3CC4C=CC3C4)=O)CC2)ccc2c(c1O)CCCC2 Cc1nn(CC(=O)NCCCC(C)NC(C2CC23CCOC3)=O)c(=O)o1 CS(=O)(=O)CC(=O)NC12CC(CNC(=O)CCNC(c3ccco3)=O)(C1)C2 N#CC1CN(Cc2ccccc2OCc2ccccc2)CC12CCC2 c1(CC(N2CC(C)C(NC(=O)CC3CCCC34CC4)C2)=O)c(O)ncnc1O N1(C(C(=O)NC(CC)(C)C)c2cn[nH]c2)CCOC2(CCC(C)(C)C2)C1 N1(CC)CC2CN(C(C3CN(C(=O)CC(O)CC(C)C)CC3F)=O)CC2C1 C(=O)(C1=C(C)OCCS1)N(C1CCCN(C(C2CSCN2C(C)=O)=O)C1)CC c1(C(=O)NC2CC3C(NC(c4c(C)ccc(O)c4)=O)C3C2)cc2n(c1)CCCC2 C1(CNC(c2cscn2)=O)COCCN1C(=O)C(C1(O)CCCC1)F c1(C(=O)NC(CNC(C(C)OCCC#C)=O)CO)cnc(O)s1 C1(CNC(CC(=C)C)=O)CN(C(c2cc(C(CC)CC)no2)=O)CC12CC2 CC(C)(C(=O)N1CC(CNC(=O)CNc2ccccc2)C1)C(F)(F)F C1(C(C)NC(C2CCOCC2)=O)CCN(C(c2cnc(C(C)(C)CF)o2)=O)CC1 CC(=O)CCC(=O)N(CC(=O)NCCC1OCCC1(C)C)C(C)C C=CCCCCC(C(=O)NCC1CC1(F)F)N1CCCC(N(C)CC=C)C1 C(=O)(C1CCCn2nccc21)N1C(CNC(C2N(CC(C)C)CCC2)=O)CC1 N1(C(C2C(COC)CC2)=O)CC=CC(C(N2C(CO)CC2C)=O)C1 N1(C(CC(=C=C)C)=O)CCC2CN(Cc3c(OC)ccc(F)c3Br)CC12 c1(-c2cc(C(N(CC(CC)NC(=O)C(C)COC)CC)=O)on2)ccc(Cl)cc1 C1(C(N(C(C#C)C)C2CC2)=O)CC(NC(=O)CCSCCCC)C(O)C1 CC(C)C1=CCC(NC(=O)CCC2CCCN2C(C23CCN(CC2)CC3)=O)CC1 N1(C(c2cn(CC(C)C)nc2)=O)CC(N(C)C(C2CC2C(N)=O)=O)C2(CC2)C1 N(C(=NCCCCl)NCC(c1ccccc1)(C)C)CC1(SC)CCOCC1 c1(C(=O)OC)cc(C(=O)NCC=CCNC(=O)COCC(C)C)cnc1C C1(NC(C(C(C)C)c2cnn(C)c2)=O)CC2CCC1CN2C(c1cncn1C)=O C1(NC(C)=O)CCC(=O)NC1.N1(C=O)CCCC1.C12CC(C1)C(=O)N2C N1(C(C2(CC=C)COC2)=O)CC(NC(c2coc(C3CC3)n2)=O)CC(C)C1 c1(OCCOC)cccnc1CN(C1COC(C)(C)C1)C=O c1(C(=O)NC(C)CCNC(=O)C(C(C)O)N(C)C)ccc2cnsc2c1 CC(CC(C)(C)C)C(=O)N1CCN(C(c2ccnc(C3CC3)n2)=O)CC1CO C#CC1CCCN(C(=O)C(C(C)(C)O)NC(=O)CCNC(=O)NC)CC1 c1(C(C(=O)OC)NC(C2CCCN2c2nnc(CC(C)C)s2)=O)ccccc1Cl C(C)(C(=O)N(CC(C)NC(c1cc2sccc2[nH]1)=O)C)(C(C)C)NC(C)=O Cc1ccc(C(=O)NCC(F)CNC(=O)C(O)C(C)(C)C)c(Br)c1 c1(C(N2C(C)(CNC(C(C(C)C)C)=O)CCC2)=O)nc(Cl)cc(N)c1Cl N1(C(CN(CCOC)C)=O)CCC(NC(=O)CC2(NC(C)=O)CC2)CC1C c1(CC)cc(Cl)ccc1NC(C1CCN(C(c2cnc(CO)nc2C)=O)C1)=O C1(CN(CCN(C)C)CC2CCCCC2)CC2OC(C)(C)OC2C1 Cc1nc(C)c(C(=O)NCC2CCCC2C(N2CCCCC2CF)=O)s1 N1(C(c2c(C)ccs2)=O)CCN(C(C2CCN(C)C2)=O)CC1 c1(C2(C(=O)NC(C)CN(C)C(c3ccc(Cl)cc3)=O)CCC2)ccc(Cl)c(F)c1 Cc1occc(=O)c1OCC(=O)NCCCC1(NC(=O)CCC2CCC2)CC1 C(c1cncc(F)c1)=CC(N1C(C(CNC(CCOCC)=O)(C)C)CCC1)=O N1(C(C=C(C)Cl)=O)CCC2CN(C(=O)COc3ccc(O)nn3)CCC12 CC1CC2(CO1)CN(C(=O)CCCCCN(C(=O)CC1CC3CCC1O3)C)C2 C(=O)(C(O)Cc1cnc[nH]1)NCC1(CNC(=O)C(O)C2CC2)CCC1 N1(C(CCOCC)=O)CCC2(CC1)CN(C(C13CC(C1)C3)=O)CC2CO CC(C)CC(C(=O)NC1CCC1CNC(c1cnc(N)cn1)=O)C(C)C N1(C(c2c(C(C)C)nco2)=O)CC2CC(C(=O)NC3CCCSCC3)(C2)C1 C(CC(C)(C)C(=O)N1CCN(C(=O)C(O)C(F)F)C(c2ccccc2)C1)OC Cc1nc(C)c(C(C)NC(C2(NC(=O)CC3CCCN3C)CSC2)=O)[nH]1 c1(OC)cc(C)c(CN2C(C(=O)Nc3cccc(OC)c3F)CC3CC23)c(C)c1 C=C(C)C1CCC(C)=CC1CC(=O)N(CCNC(=O)CC)Cc1ccn(C)c1 c1(CCC)ccc(C(N2CC3CC3(NC(=O)C(C)(O)CC)C2)=O)cc1 C(=O)(C1=C(Cl)CCCC1)NCC(CCNC(C=Cc1ccc(CC)cc1)=O)O c1(CCC)onc(C)c1C(=O)NCCNC(=O)C(c1ccc(F)cc1)(C)O Cc1ccc(C(=O)NCc2ccc(Br)c(C)c2)c(-n2cc(CCN(C)C)nn2)c1 C(=O)(C(CCCC)ON=C(C)C)NCC1(NC(CCC(=C)Cl)=O)CC1 C(c1ncccc1C)=CC(=O)N(C1CCN(C(c2cnc(CCC)s2)=O)C1)C c1(C(C)C)[nH]nc(C(=O)NCCC(C)NC(C2(C#N)CCCO2)=O)c1Br N1(C(C(F)=C(C)C)=O)CCC2(CC2)CC1C(=O)NCCS(C)(=N)=O c1(C(N(CCn2cc(C34COC(C3)C(O)C4)nn2)CC)=O)nnn2c1CCC2 C(CC)(C(=O)NCC(C)(CO)NC(=O)COCc1scnc1C)=CC C(=O)(C1COc2ccccc21)N(C(C)CNC(=O)COC1CC(F)(F)C1)CC C1(C(=O)NCCN(CCCN(C)C)C(c2n(C=C)ncc2)=O)CC2CCCN(C1)C2 c1(C(=O)NCC(C)NC(c2nccc(C(F)(F)F)n2)=O)ccc(Br)nc1O c1(N(C(C(C)SCC)=O)C)nc(C(C)(C)C)no1 c1(COC(=O)CCC2CC2(Cl)Cl)cc(Cl)c(Cl)s1 N1(C(C2C(NC(C3(CC)COC3)=O)CCOC2)=O)CC2(CCOC2=O)C1 c1(N2C3CCN(C)CC2CC3)nc(=NCCC=CBr)[nH]c2cc[nH]c12 c1(C(=O)NCC2(NC(C3CC(SC)C3)=O)CCOC2)cc(F)ccc1C(C)C c1(C(=O)NC(C2CCN(C(c3cc(F)n[nH]3)=O)C2)C)cc(Cl)c(Cl)c(Cl)c1 CC1CC(CNC(C2CC2C)=O)CCN1C(=O)CNC(c1ccsc1)=O C(C(CC(C)C)NC(c1csc(C)n1)=O)NC(COCCC#C)=O N1(C(Cc2cn(C)nc2)=O)CCN(C(c2cn(C)cn2)=O)CC1c1cccnc1 C(CCCCCCC)NC(C1(CC#C)CCN(C(C2CCC(C(N)=O)C2)=O)C1)=O C(=O)(CCC(C(=O)NCC(C(C)(C)C)NC(=O)Cc1csc(C)c1)N(C)C)OC c1(OCC(=O)NC(CNC(c2nc(OC)oc2)=O)(C)C2CC2)ccc(Cl)cc1Cl N1(CC(=O)NCC2CC(F)CN2C(c2cccc(O)c2Cl)=O)C(=O)CCCC1=O C1(NC(CC(C2CC2)NC(C2(C)CCCCO2)=O)=O)CC2CCCCCC12 N1(C(c2cc(OCC)no2)=O)CC2CC(C1)N(C(c1ccc(CC)nc1C)=O)C2 CCCC(C(C)(C)C)NC(=O)C(Cn1cccn1)NC(=O)CCC(C)(F)F c1(OC)ccc(OC)c(C(=O)NCCN(C(=O)CC2CC(O)C2(C)C)C(C)C)c1 N1(C(c2scc(COC)c2)=O)CCC(CC(=O)NCC23CC(CN2C)C3)C1(C)C CN1C(=O)CSC1=CC(=O)NC1CN(C(c2ncccc2Cl)=O)CCC12CCC2 C1(CNC(c2cnn(C(F)F)c2)=O)C2CCC(C2)N1C(=O)C(F)F c1(C(N2CCC(N(C(=O)C(OC)OC)CC#C)CC2)=O)cccc(=O)n1C C(=O)(C(O)CCCNC(c1cc(C(F)F)[nH]n1)=O)NCCC(=O)NO C(=O)(CC(C)C(=O)NCCC1(C(N2CC3CCC3(C)C2)=O)CCCC1)OC c1(C(N(CC(=O)NCC2(C(N)=O)CCCC2)CC#C)=O)ccc(C#N)cn1 N1(C(c2ccc(NC)cn2)=O)CCCN(C(=O)CCC2NC(=O)NC2=O)CC1 S(=O)(=O)(c1cccnc1)NCC(N1CCC(NC(c2cnccn2)=O)C(O)C1)=O Cc1cc(=O)n(CCC(=O)N(C(C)CNC(C2CCN(C3CC3)CC2)=O)C)cn1 c1(C(=O)NCC(CNC(C2(CC)CC2)=O)C)ccc2c(c1)CCCC2 C(CNC(=O)C=Cc1ccncc1)(CC(=O)NC(C(C)(C)O)C1CC1)OC c1(SCCOC(C2C(C(=O)OC(C)(C)C)C2)=O)ccn(C2CCCC2)n1 c1(C(=O)NCC2(NC(CSCCC#N)=O)CCC2)cccn2cnnc12 N1(C(C23CCC(CO2)C3)=O)CC2CCC(C1)N2C(C12CCCC(C1)OC2)=O C=CC1(NC(c2ccccn2)c2nnnn2CCCCCC)COC1 N1(C(c2cn(C)nn2)=O)CCC(C(N2CCCC(CCF)C2)=O)C1(C)C Cc1ccc(N(C)C(C2CCN(C(=O)C(=O)N(C(C)C)CC)CC2F)=O)c(Cl)n1 c1(CC)cc(C(N2CCN(C(c3ccc(Cl)cc3)=O)C(CO)C2)=O)ccc1O c1(OC)cnc(C(=O)N(CC(C)N(C(=O)CC2C=CS(=O)(=O)C2)C)C)c(F)c1 C(=O)(CCC(C)S(C)(=O)=O)N1C(C(C)C)CN(C(=O)C(C)(C)C2CC2)CC1 C(CCF)(C(=O)N1CC(O)(C(C)C)C1)NC(C(C)NC(=O)C1CC1)=O COn1cnc(C)c1C(N1CCC(C(C)NC(=O)CCc2ccc(C)s2)C1)=O c1(CNC(C(CC)OC)=O)ccc(C(N2CCCC2(C)CO)=O)cn1 CN1CCN(C(C2(c3cnn(C)c3)CCCO2)=O)CC1CNC(=O)CCC1CC1 CN1CCN(c2ncc(Br)cn2)C(CNC(C2(C)CC(C)(C)C2)=O)C1 N1(C(c2n[nH]cc2Br)=O)CCN(C(c2ncc(F)cc2F)=O)C(C(F)F)C1 C(N=c1[nH]c(=NCCOCC2CC2)c2ccccc2[nH]1)C1CCS(=O)(=O)CC1 C#CCCCCCC(=O)N1CCCC(C(C)(O)CNC(=O)C(=O)C(C)(C)C)C1 C1(CC(=O)NCCCN(C(=O)CC2CC2C)C2CC2)(CC)CCC1 C(=O)(C1=CC(C)(C)C1)N(C1CCN(C(c2c(CC)nco2)=O)C1)CC1CC1 C(=O)(C1c2ccccc2C2CC1C2)NCCOCCNC(c1cnc[nH]1)=O c1(CC)ccc(-c2nc(C)c(C(=O)NCCC3CCCN(C)C3)s2)cc1 N1(C(C(COC)(F)F)=O)CCN(C(c2cnoc2C)=O)C(CC(F)F)C1 c1(C(CC(C)C)CC(c2nnnn2CC)(C)NC(C(CC)C)=O)ccc(Cl)cc1 N1(CC(C)NC(CSCCC)=O)CCN(C(c2ncncc2F)=O)CC1 C1(CC(=O)NCCC2(CNC(COCCCCC)=O)CC2)COCCN1CC N(C(=NCCC(=O)N(C)C)NC1CC=CCC1)CC1CCC(CCCC)CC1 c1(OC(C)C)cnc(N(C(C)CNC(=O)C(O)Cc2cnc[nH]2)C)nc1 CCC(CNC(=O)CCC1CC1(Cl)Cl)NC(=O)CCOCC1CC1 C=C(C)CC(C(=O)N(C)Cc1ncnn1C)NC(c1ccc(C#N)cc1)=O C(=O)(CCCCCN(C)C)NCC1N(C(C(C(C)C)OCC)=O)CC=C1 CC1CN(C(C2CC2c2ccc(Cl)cc2)=O)CC1CNC(c1c[nH]ccc1=N)=O C1(C(=O)NCC(CC)CO)CC2(CCN1C(=O)C(c1ccn(C)c1)C)CC2 N1(C(c2ccc(OC)nn2)=O)CCC(C)CC1CNC(=O)CCc1cnn(C)n1 C1(C(=O)NCCN(CCO)CC)CCC(C)N(C(=O)Cc2cnsc2)C1 c1(C(N2CCC(CNC(C=CC=CCC)=O)C(C)C2)=O)ccc2c(c1)CC(C)O2 c1(C(=O)NC23C(CN(C(CC(=C)C)=O)C2)COCC3)cccc(S(=O)(=O)CC)c1 C1(CC(=O)NC(C(C)C)(C)CNC(C2CC=CC2)=O)Cc2cc(F)ccc2O1 c1(NC(C2C(C(=O)Nc3c(OC)ncnc3Cl)C2)=O)nc(C)c(Cl)cc1Cl N1(C(C=CC2N(C)CCC2)=O)CC2CC1CN(C(c1cccnc1C(F)F)=O)C2 c1(OC)cc(C(=O)NCC(F)CNC(C23CC(C)(C2)OC3C)=O)cc(Cl)n1 c1(CC)ccc(C(=O)NCC2CC(C)N(C(=O)CC3(COC)CC3)C2)cn1 CC(C)CC(C(=O)NC1CC12CCC2)ONC(c1cccc(=O)n1C)=O Cc1cc2c(N3CCC(NC(=O)C(N)c4cscn4)CC3)ncnc2s1 CC(C)C(N)CC(=O)NCC1(C(=O)O)COCC1(C)C c1(OC)cccc2c1N(Cc1cn(CC(c3cccc(C)c3)O)nn1)CC2 Cc1cccc(C(C)(C)C(=O)NCC(C)NC(=O)C(c2cn(C)nc2C)C)c1 C(N=c1[nH]cnc(Cl)c1C#N)C1(C)CCC(NC(C=C(C)Cl)=O)CC1 N1(C(C2N(C)C(=O)CC2)=O)CC2CC1CN(C(C1CC1c1cccc(O)c1)=O)C2 c1(OC)ccc(C=CC(=O)NCC(CO)NC(=O)Cc2ccc(C)cc2)cc1 C#CCCCCC(C(=O)NCc1ccc(OC)cc1)N(C)CC1CCCN1C N1(C(Cn2c(C(C)C)nnn2)=O)CC2CC(CNC(=O)C3=NNC(=O)C3)C2C1 C1(CNC(c2nc(CC)oc2)=O)CCCCN1C(C1CC=CC1)=O C12(NC(c3c(CC)n(C)nc3)=O)CCCC1N(C(c1ccc(F)c(C)c1)=O)CC2 N1(C(C2CC(F)CN2Cc2cccnc2Cl)=O)CCN2C(=O)CCC2C1 c1(OC)ccc(C(N2CCC(NC(C3(F)CCOC3)=O)CC2)=O)cc1OCCO Cc1ccoc1CNC(=O)Cn1cc(C(C)(C)C2CC2)nn1 N1(C(CCNC(N)=O)=O)C(CNC(c2cccc(-n3cnnn3)c2)=O)CC2CC12 C1(CNC(C(CO)OC)=O)CC(C)N(C(c2nnn(C(C)(C)C)n2)=O)C1 C12(C(N3C4CN(C(C5CC6CCC(C5)S6)=O)C(C4)C3)=O)CC3CC(CC1C3)C2 C#CC1(O)CC(C(=O)NC(C(C)NC(c2cccc(COC)c2)=O)C(C)C)C1 C1(SCC)CN(C(=O)CC2(COC)CC2)CCN1C(=O)Cc1n[nH]c(C)n1 c1(-c2cn(CC3OCCN(C(c4ncc(C)o4)=O)C3)nn2)ccnc(Cl)c1N c1(CC(=O)NC(CCNC(C2(C(CC)(F)F)CC2)=O)C(C)C)ccc(Cl)c(Cl)c1 N1(C(c2onc(CC)c2C)=O)CC2CC1CC2CNC(=O)CC1CC1 c1(CN2CCC(NC(c3cc(C)c(F)nc3)=O)C(O)C2)ccc(C#N)cc1C c1(CC(N2CC(C(C)NC(CCC)=O)C2)=O)c[nH]c2cccc(F)c12 N1(C(c2ccc(CSC)cc2)=O)CC2CC1CN2C(=O)C(F)OC(F)(F)F N1(CC(N2CCCC2)C)CC(=O)N(CC(COC)(C(F)(F)F)c2ccccc2)C1=O CC1CCC(CNC(=O)CCF)CN1C(=O)CNc1ccc(O)cc1 C1(OC)(CNC(=O)C(O)CC(C)C)CCN(C(c2c(Cl)sc(C)c2C)=O)CC1 n1(CC)nnc(C(N2CCN(CC(=O)NCCc3ncnn3C)CC2)=O)c1C N1(C(c2nc(NC(C)=O)sc2)=O)CCOC2(CCN(C(=O)CC(F)F)C2)C1 N#Cc1cccc(CNC(=O)C(N2CC3CC(F)(C3)C2)=O)c1Br c1(C(C)NCC(C)(C)NC(C2CCS(=O)(=O)C2)=O)cccc2ccccc12 C(CC(C)C(=O)N1CCC(CCOC)(NC(=O)CCCN(C)C)C1)=CCC C1(C)(NC(CC(=C)C)=O)CCCN(C(=O)Cc2ccnc(Cl)c2F)C1 c1(NC2C(CC)CCCC2)ccc(S(=O)(=O)N2CCc3c[nH]nc3C2)cn1 c1(OC)nscc1C(=O)NCC(C1CC1)NC(c1cc(-c2ccc(C)o2)[nH]n1)=O CN1CCOC(CNC(C2C(NC(=O)C=Cc3ccsc3)C2(C)C)=O)C1 CC(C)(O)C#CC(=O)NC(C(=O)NCCC1(C)CCCC1)C1CCCO1 c1(CCC(=O)NC(CC=C)CNC(c2ccsc2C)=O)cc(C)nc(C)c1 C(C)(CC(=O)N1CCCC(O)(CCNC(c2cnsn2)=O)C1)(C(F)F)N(C)C C(CC(C)(C)CNC(c1ccc(NC(=O)CCSC)cc1)=O)NC(C(C)=CC)=O C(=O)(CC1CCc2ccccc21)NCC(C)(C1CCC1)NC(CCCN(C)C)=O C(=O)(C(CC=CCl)c1ccccc1)NC(C)CCNC(c1[nH]ccc1C1CC1)=O CC1C2CC(C(=O)NC3CN4CC3(C)C4)(C2)N1C(=O)OC(C)(C)C c1(CN2CCC(CC(=O)Nc3nc(Br)cs3)C2)cc(Br)cc(F)c1F C(=O)(C(=O)CC(C)CC)NC(CC#C)C(=O)N1CCCCC1CC C1(C(=O)NC(C(C)O)(C)C)CC(NC(=O)CN(C2CCCC2)C)C(O)C1 CC(C)C(C(=O)N1CCC(O)CO1)c1ccn(C)n1 c1(C(=O)NC(CC(=O)NCC(CC)(C)O)COC)cccc(O)c1F c1(C(=O)NCCCC(C)NC(=O)CCS(=O)(=O)N(C)C)ccc(N=NC(N)=O)cc1 c1(CN(C(=O)NC(c2cccc(C(F)(F)F)n2)C)C)ccc(C(F)(F)F)c(F)c1 N1(C(c2ccc(CO)c(Cl)c2)=O)CCC2CN(C(c3ccc(O)cn3)=O)CC12 N1(C(c2c(N)cccn2)=O)CCCC(NC(c2coc(C(F)F)n2)=O)CC1 Cc1nnc2n1CCC(C(N1CC(NC(=O)CC3CN4CCN3CC4)C1)=O)C2 CCC(CC)CCC(=O)NC(C)CCN(C)C(c1ncoc1CCC(F)(F)F)=O CC1(C)CC(CNC(=O)COc2ccccc2Cl)N(C(=O)CP(C)(C)=O)C1 CC1CN(C(c2c[nH]c(Br)c2)=O)CCC1NC(=O)CCC1CCCCC1 C1(C(N2C3CC(NC(C4(C)COC4)=O)CC2CC3)=O)CCc2ccccc2C1O CC1(C)CN(C(=O)CC(O)CNC(c2coc3c2COC3)=O)CCS1 N1(C(c2nc(OC)oc2)=O)CC(C)N(C(=O)Cc2ccc(Cl)cc2Cl)CC1C N1(C(C(CCc2ccc(CC)cc2)C)=O)CC2CCN(C3CCN(C)C3=O)C2C1 c1(C(=O)NCC2CCN(C(CCC=CC)=O)C2)ccc(C2(C)CC2)cc1 CC(CC(=O)NCCOCCN(C)C(c1cc(O)nn1C)=O)CC(C)(C)C c1(C(=O)NC2CCC(NC(C3(CCC=C)CC3)=O)CC2)c(C)cncc1C c1(C(N2CCCC(NC(CCC(C)OCC)=O)C2)=O)cc2c(o1)CCCC2 N1(C(C(CC)C)=O)CC(NC(c2cnsc2)=O)CC2(CCOCC2)C1 c1(CCC(=O)NC2(CC=C)CN(C(C3CCN(C)C3)=O)C2)cnc(C)nc1O C(CCC(O)C(=O)NCC1CCC2(CC2)CO1)NC(C(CCC)F)=O c1(OC)cc(C)ccc1OCC(=O)NC1CCC(NC(c2nnsc2C)=O)CC1 C(=O)(CCS(=O)(=O)c1ccccc1)NCC(CC=C)NC(c1ccccn1)=O C1(c2ccccc2)CC(C(=O)OC)CCN1C(=O)NCC1C(CO)C1(F)F Cc1cc(Br)c(S(=O)(=O)NC2CCN(CC(F)F)C2)cc1Br O=C(CCC(F)(F)F)NCC1CCCC1NC(=O)CC1CCCC1 CC(C)(C)C(C(=O)NC1CCCC1CO)NC(=O)COC1CCCCC1 Nc1ccc(CCC(=O)N(CCCNC(C2CCCCC2O)=O)C2CC2)cc1F CCC(C)(C#N)C(=O)N1CC(NC(c2cnn(-c3ccccc3)n2)=O)C(O)C1 N1(C(COC(C)(C)C)=O)CC(C(=O)NC2CC(P(C)(C)=O)CN2)CC12CCC2 C1(OC)CC(CCNC(c2ccc(F)cc2)=O)N(C(=O)CCc2cnco2)C1 c1(C(=O)NC2C(NC(C3C(C)C3C)=O)COC2)cncc(-c2ccccc2F)c1 CC(CCC(=O)NC1CCCC(CNC(=O)CNS(C)(=O)=O)C1)N(C)C c1(CC(=O)NCCN(C(C2C(c3n(CC)cnn3)C2)=O)C)ccc(Br)cc1 c1(C(=O)NC2CN(C(C(CC)=CC)=O)C2)cc(Cl)ccc1SC1CCCC1 c1(CC)ccnc(C(=O)NC(CCNC(=O)C(F)n2cccn2)C(C)C)c1 C(=O)(C1CCc2ccccc21)NC(C1CCCN1C(=O)COCCOCCO)C C1(NC(CCC(C)C)=O)CN(C(=O)CCCNC(c2cccs2)=O)CC(F)(F)C1 N1(C(C(COC)N(C)C)=O)CCC(C(F)CNC(=O)CSC(C)(C)C)CC1 c1(OC)c(C(=O)NCC2CC2NC(c2ccc(C3(O)COC3)cc2)=O)cnn1C C1(=CC(N2CCC(C(C)(C)NC(=O)C(C#N)C3CC3)C2)=O)CCC(C)(C)CC1 C(=O)(CCC1C(=O)Nc2ccccc21)NC1CN(C(CCC#CC)=O)CC1C N1(C(c2ccc(C)cc2Cl)C(=O)NCC=C)CCCCCCC1CC n1(C(C)C)ccnc1C(=O)NCC(C)(C)CC1CN(C(=O)COCC2CC2)C1 Cn1cnn(CC(=O)NC2CCCC2C(N2C(CO)CC2CO)=O)c1=O N1(C(c2cc(=N)[nH]cc2)=O)CCC(NC(C2CCCS(=O)(=O)C2)=O)CC(O)C1 C1(NC(Cc2nc(C)[nH]n2)=O)CCN(C(=O)Cc2c(F)cccc2F)CC1O CC(=Cn1ccnn1)C(=O)NCC1COCC1NC(c1cc(C2CCC2)on1)=O c1(OC)ccc(F)c(C(=O)NC2CC(CNC(C3(OC)CCSC3)=O)C2)n1 c1(NC(=O)C(N2CC(CO)OC(CO)C2)=O)cccc2c1OCC2 c1(C(N2C(CN(C(=O)C(C)(C)CF)C)CCC2)=O)cc(Cl)ccc1-n1cncn1 S(=O)(=O)(c1ccc(Cl)c(C(=O)O)c1)N1C(C)(C(=O)NCC(C)C)CC1 c1(CC)cc(C(=O)NCC2(F)CCN(C(c3oncc3C)=O)C2)ncn1 n1(CC)cc(Br)c(C(=O)NCC2CC(NC(=O)C(O)c3ccsc3)C2)n1 N(C1CC2(CN(C(c3ccsc3C#N)=O)C2)n2ccnc21)C(C1CCC(C)O1)=O n1(CC(=O)NC2C(CNC(C3(S(C)(=O)=O)CC3)=O)COC2)cc2ccccc2n1 c1(C(=O)NC2CCN(C(C3C(=C)CC3)=O)C2C2CC2)ncc(C)cc1F c1(C(=O)NCc2cn(CC(C)NC(CCC(=C)C)=O)nn2)cc([N+](=O)[O-])n[nH]1 N1(C(C(=O)NCC)COc2ccccc2)CC(CC(F)(F)F)OC(C)C1 C1(CN(C(c2c(C)c(I)nn2C)C(=O)NCCC#N)CC)COC(C)(C)OC1 c1(C(N2CCC(C3CCCO3)C2)C(=O)NCCCF)ccc(Cl)c(Cl)c1 C(CCNC(c1ccc(=O)oc1)=O)(C(C)C)NC(C1N(C(CCC)=O)CSC1)=O c1(C(=O)NC2CN(C(C(C)n3cccc3)=O)CC(O)C2)cc2cccnc2[nH]1 N1(C(C=C(CCC)CCC)=O)CC2CC(C1)N(C(=O)C=CCF)C2 N1(C(C=Cc2nnn(C)n2)=O)C2CCC1C(F)C(NC(=O)CC1C=CCC1)C2 Cc1nc(C(=O)NCCCCCC2CCN(C(c3nccs3)=O)CC2)c(C)o1 C(=O)(CC(C(C)C)NC(=O)CCCNC(=O)OC)N(CCCC=C)C c1(CC(=O)N(CC(O)C(F)(F)F)C)c(F)cc(F)c(Br)c1F C1(C2(C=C)CCC2)(C(=O)NC2CC(NC(C(C=C=C)C)=O)C2)CCC1 c1(C(N(C2CCC(NC(=O)C(C)(F)F)C2)C)=O)cccc(Cl)c1O C1(CC(N2CC(CNC(c3n(C)ccn3)=O)C(C(F)(F)F)C2)=O)OC(C)(C)OC1=O C(=O)(CC(C)(C)C(F)(F)F)NCC12CC(NC(CCC(=O)NC)=O)(C1)C2 c1(CC(C)N(C(c2cn(CCN)nn2)=O)CC)ccc(OC)cc1 CC(C)CC(CNC(c1nn(C)cc1N)=O)NC(c1ccnn1CCF)=O c1(C(N(CC(C)O)CCNC(c2n(C)nc(C)c2Cl)=O)=O)cc2ccncc2s1 Cc1nn(C)c(C)c1OCC(N1CCN(C(=O)CSC2CC2)C(C2CCC2)C1)=O c1(NCC)cccnc1C(N1CC(CCNC(=O)CCOC2CCOCC2)C1)=O c1(C(=O)NCC2(CC(=O)NCC(C)C#N)CC2)c[nH]c(=S)cn1 c1(C(=O)NC(CNC(c2c(OCC)nccc2)=O)CC)sc2ccccc2c1C C12(c3n(CC)c(N(CC(C)C(=O)NC)C)nn3)CCCCC=C1OCC2 c1(C(N2CCN(C(CSCC=C)=O)CC2CC)=O)ccc(Br)c(C)c1F N1(C(CCCS(C)(=O)=O)=O)CC(CO)C2(C1)CN(C(=O)CCc1nc(=N)[nH][nH]1)C2 N1(CCNC(CSC)=O)CCN(C(c2cc(-c3ccccc3)ns2)=O)CC1 c1(C(N2CCC(OCCNC(C=CC(N)=O)=O)C2)=O)ccc(F)cc1F c1(C(N2C(CNC(c3[nH]cc(C#N)c3)=O)CC2)=O)cc2ccccc2nc1O Cc1cc(C(=O)NC2CC(C)N(C(=O)C3=CCCS3)C2)ncc1C(N)=O N1(CC(=O)N(C(C)C)C(C)C)CC(NC(c2cccn2C2CCCC2)=O)CC(C)C1 c1(CC)ccc(C(=O)N(CC(C)N(C(=O)CN2CCC(C)C2)C)C)c(O)c1 c1(OC)ccc(F)cc1C(F)(F)C(=O)N(CC(C)NC(=O)CCCC1CC1)C C1(CNC(C2C(=C)C2)=O)(CO)CC12CCN(C(c1cncc(OC)n1)=O)CC2 C(=O)(C1CCCc2n[nH]cc21)NC1C2CC(NC(C3CC(C)(F)C3)=O)C(CC2)C1 c1(N(CC(=C)Br)C)nc(=NCc2ccc(OC(F)F)nc2)[nH]c2c1CC(C)CC2 Cn1nc(C(=O)NC2CCN(Cc3coc(-c4ccccc4)n3)C2)ccc1=O N1(C(CC2(COC)CC2)=O)CCCC(N(C)C(c2coc(Cl)n2)=O)CC1 Cc1ccc(C(=O)NC(C2(CNC(=O)CCCC(F)F)CC2)C)c(N)c1 N1(C(c2n(C)ncc2Br)=O)CC2(CC2)CC1C(N1C2CCC1CC2)=O c1(C(N2CC(c3cn(C)nc3)OCC2)=O)cc(F)c(F)cc1N N1(C(C(C)O)=O)CC(O)C(O)C1CNC(c1ccc(Cn2cncn2)cc1)=O C1(C(=O)Nc2cn(CC)nc2C)CC(NC(=O)C(C)CC2CCC2)C12CCC2 c1(C(N(CCCF)CC)=O)cc(CCNC(=O)CC2CCCCO2)on1 C1(C)(C(N2CC(C)(CCC(=O)NCC(C(C)C)O)C2)=O)CCCOC1 CCC(C)CCC(=O)N1CC(NC(=O)CS(=O)(=O)NC(C)(C)C)CC1COC CCCCC(C)CCC(=O)NC1(C(N2CC(O)C(O)C2)=O)CCC(C)(C)C1 C12(C(N3C(CNC(c4c(CCC)cccc4)=O)C=CC3)=O)CCC(C)(C1)OC2 c1(C(=O)NC(CNC(CCC#C)=O)C(C)C)cnc2ccc(Br)cn12 c1(OC)ccc(SC(=O)NCCOCC(=O)OC(C)(C)C)c(OCCF)c1 CCC(C)C(O)CC(=O)N(CC(=O)NCC(C)Cc1cn[nH]c1)CC c1(N2CC(NC(c3c(C(=O)C(C)C)cc(C)s3)=O)C(O)C2)nc(C)cc(C)n1 C12(CNC(C(CC)C)=O)CC(NC(=O)CC3NC(=O)NC3=O)(C1)C1(CCC1)O2 c1(C(=O)NCC2(F)CCN(C(C3(C)CCOCC3)=O)C2)cnc2ncccn12 N1(C(c2c(C)nsc2C)=O)CC2CCN(C(C3(C)CCCN3C)=O)CC2C1 C(=O)(CC(C(C)C)c1ccon1)N1C(CNC(C(C)c2ccsc2)=O)C(C)CC1 N1(Cc2scc(C)n2)CCN(C(c2cnc(Br)o2)=O)C(C#N)C1 N1(C(Cc2nc(C)oc2)=O)CCC(C)CC1CNC(=O)C(C)S(C)(=O)=O N1(C(CCCN(C)C)=O)CC2(CCN(C(c3ccc(O)c(F)c3)=O)CC2)C1 C1(NC(c2nccc(C(F)(F)F)n2)=O)CN(C(c2cc(F)c[nH]2)=O)CCC1O CC(C)CC(Cn1cc(C2CCCO2)nn1)NC(=O)CCN1CCOC1=O N1(C(CCS(C)(=O)=O)=O)CCCC2(CCCN2C(=O)Cc2ccc(Cl)s2)C1 Cc1ccc2c(C(=O)Nc3cc(O)c(Br)cc3C)csc2c1 N1(C(=O)Nc2nccc(COC)n2)CCC2C(CCN2C)C1 c1(NC(C2(CC#C)CCCC2)=O)cc(F)c(C#N)c(Br)c1 C(=O)(CC(O)CNC(C1CCCN1CC)=O)N(C)Cc1ccn(CC)n1 C=CCC(C)(C)CC(=O)N1CC(O)CCC1C(N1CC(S(N)(=O)=O)C1)=O c1(C(=O)NC2CC(CNC(C(CCSC)OC)=O)C2)cc2ccccc2[nH]1 C1(NC(=O)C=Cc2ccsc2)CC2CCC1N(C(=O)CCc1ccnc(Cl)c1)C2 c1(CC)nc2ccccc2n1CCOC(=O)CC1CC(SC)C1 CC(C)CS(=O)(=O)CC(=O)NC12CC1CN(C(c1cc(F)ccc1O)=O)C2 c1(C(=O)NC2CC(CC(N3CCCC(CC)C3)=O)C2)ccc2[nH]ccc2c1 CC(=O)C(C)CC(C)C(=O)NC(C1(C(=O)N(C)Cc2cc(C)on2)CC1)C Cc1cccc(C(=O)NC2CC2C2CCCC2)c1I c1(OC)cccc(SC(c2ccccc2Cl)C)n1.C1C(=O)O1 CCC(C)CCCC(=O)NCCOCCOCCNC(=O)Cc1ccsn1 C=C(Cl)C(C)(C)C(=O)N1CCC(N(C)C(c2cn(CC3CCCOC3)nn2)=O)C1 c1(C(=O)NC(CC)CNC(=O)C(C)NS(=O)(=O)CCC)ccc(C(C)=O)c(F)c1 C1(NC(CCNC(CCn2c(C)ncc2)=O)=O)C(C)(C)C1(C)C CC(C(=O)NC12CC(C1)N(C(=O)CNC(N1CCCC1)=O)C2)S(C)(=O)=O CC(CCNC(=O)Cc1csc(C(F)(F)F)n1)CCNC(=O)CS(N)(=O)=O C1(C(=O)NCC(F)CNC(C2(F)CC2)=O)CCN(c2ccccc2)C1 C1(CNC(c2cn(CC)nc2)=O)CN(C(=O)C=CCOC)C2CCCCC12 c1(C(=O)NC2CCC(N(C(c3c(C)ncn3C)=O)C)CC2)cc(Cl)ccc1F C1(C(=O)NC2CCC(CNC(C=CC(=O)N(C)C)=O)O2)CCC2(CCC2)C1 N#Cc1ccc(S(=O)(=O)NC2CC3CCCCN3C2)cc1NCCC(=O)N1CCCC1 c1(CC)nccn1C(C)CC(=O)NCC1CCN1C(=O)C=C1CCC(C)C1 C12(CNC(C)=O)CCC(CC1)N2C(c1scnc1-c1ccc(Cl)cc1)=O Cc1c(NC2(c3nnnn3C3CC3)CCOC(CCN(C)C)C2)cccc1Cl c1(C(N(CC(C)NC(=O)COC(C)(C)CC)CC)=O)ccc(NC(C)=O)cc1 c1(Sc2c(C(NNC(c3n(C)cc(Br)c3)=O)=O)cccc2)ccc2c(c1)COCC2 CC(C)(C(=O)NCC=CBr)C1=CCN(C(c2ncccc2F)=O)C1 c1(C(N(CC(CNC(C(CC2CCCC2)OC)=O)C)C)=O)ccc(C)cc1O C1(NC(c2ccc(C(=O)OC)o2)=O)CS(=O)(=O)CC1NC(=O)CCCF CCCCC(C)C(=O)NCCN(C(=O)CCc1cnn(C)n1)Cc1cccnc1 C(=O)(C(F)(F)CCn1ccnn1)N1CC2C(CNC(c3ccsn3)=O)(C2)C1 C1(O)(CN(C(C(C)c2cccs2)=O)C)CCN(C(c2sccc2Cl)=O)C1 C1(CC)CN(C(=O)C(C)N2CC(C)C2)CCC1CNC(=O)Cc1cccc(F)c1 N1(C(C(C)(C)CF)=O)CCC(NC(c2cc(O)cc(Cl)c2Cl)=O)C(F)(F)CC1 N1(C(=O)CC2CCCOC2)CC2(CCN2C(c2cn3ccnc3s2)=O)C1 Cc1nccnc1C(N1CCCC(c2cc[nH]c(=N)n2)C1)=O N1(C(CN2CC(C)C2)=O)CCC2(CC1)CC2NC(=O)C(c1cc(F)ccc1F)=O N1(C(=O)C2CC2)CC2(CCC2)CCC1CNC(c1cnc(OC)c(C)c1)=O C1(NC(c2cc(C(CC)C)no2)=O)CCOCC1NC(c1ccc(CF)cc1)=O c1(CCCC)ccc(CC(=O)NCC(C)(O)CNC(C2(CCC)CCC2)=O)cc1 C12(CNC(C3C(C)OCCC3)=O)CCC(CC1)N2C(C1(CC2CC2)CCC1)=O Cc1ccccc1C1CCCN(C(=O)Nc2ncc(Cc3ccccc3Cl)s2)C1 C1(CNC(C(C)OCC)=O)CCC2CN(C(c3ncccc3N)=O)CC12 Cn1ncc(C(=O)NC(C2CCN(C(=O)C=Cc3ncc[nH]3)C2)(C)C)c1F N1(C(C2CC=CC(NC(=O)C=CCO)C2)=O)CC2COCC(C2)C1 C(=O)(CCCCCCCO)N1C(CC(=O)Nc2cc(C)no2)CCC1 Cc1nc2nccc(C(=O)NCC3CCN3C(c3csc4cccnc34)=O)n2n1 Cc1ccc(C)c(C(=O)NC2CC(CNC(=O)CS(N)(=O)=O)C23CCC3)c1 C1(CC(=O)NC2CN(C(c3c(C)cnnc3)=O)C2)CCCC(F)(F)C1 N1(C(C2CCCSC2)=O)CCC2CCCC12C(N1CC2CC=CC1C2)=O C(=O)(C1=CC2(CCOCC2)C1)NC(C1CCN(C(c2c(SC)cn(C)n2)=O)C1)C CCS(=O)(=O)C=CC(=O)NC1CC(C)N(C(=O)CCc2nnc(C(C)C)o2)C1 C(CC(O)C(=O)NCP(C)(C)=O)NC(C1(C)CCCC1)=O N1(C(C2C3N(C(c4nc(C)n(C)c4)=O)C(CC3)C2)=O)CC2(CNC(=O)OC2)C1 C1(CNC(c2c(C(C)C)scn2)=O)CC(C)(C)CN1C(c1ccncc1O)=O FC1(F)C(CN=c2[nH]cnc(NC3CC(n4ccnc4)C3)c2Cl)C12CCOCC2 C1(CNC(C=C(COC)C)=O)COCC2(CCN(C(C3(C4CC4)CC3)=O)C2)O1 C=C(Cl)CC(C(=O)N1CCC(O)(CN(C)C)C1)NC(C1C=CCCC1)=O C1(C(N2CCC(C)(F)C2)=O)CCC2(CC2)N1C(C1CC2CCC(C1)O2)=O C1(NC(C2(S(C)(=O)=O)CC2)=O)CC2CCC1CC2NC(C1CC=CCC1)=O c1(N2CC3CC(NC(c4c(SC)nccn4)=O)C3C2)c(C)c(C)nc2ncnn12 C(=O)(C1=CCC(NC(=O)CC2C=CCC2)C1)N(C(C#C)C)C N1(C(CCNC(C)=O)=O)CC(C)(C)CC1CC(=O)NC(C)(C)C(O)CO c1(CC(C)C)nc(C2CCC(C(=O)OC(C)C)O2)n(Cc2cccc(F)c2)n1 CC(C)CC(O)C(C)C(=O)NCC1(CC(N2CC(N=[N+]=[N-])C2)=O)CC1 c1(CC(N2C(C)CC(NC(C34CC(C3)C4)=O)C2)=O)ccc2c(c1)CCC2 N1(C(c2cc(C)sn2)=O)C2CCC1CN(C(c1c(O)nnc(C)c1C)=O)CC2 c1(OC)ccc(CNC(=O)C(=O)NCC2(C)CCC2)c(OC)c1 C1(C(C)NC(NOCC=CC)=O)CCCN1C(=O)OC(C)(C)C Cc1nn(-c2ccccc2F)c(C)c1NC(C1C(C)C1(F)F)=O c1(C(=O)NC2(C)CN(C(=O)Cn3ccc(C4CC4)n3)C2)ccc(Cl)cc1Cl N1(C(c2c(NC)scn2)=O)CCC(C=CC(=O)NC2CCC23CCCC3)CC1 n1(CC(=O)NCC2(CNC(C3SC4C=CC3C4)=O)CCC2)cc2ccccc2n1 C(c1c(F)cccc1F)=C.c1(CNc2cccc(OCCF)c2)nccc2[nH]ccc12 c1(OC)ccc(CC(=O)NCC(C)(CC(C)C)NC(c2cc(C)c[nH]2)=O)cc1Cl CON(CCC(=O)NCC1CCC(O)CC1)C(=O)c1cnc(=N)[nH]c1 N1(C(C)=O)CCCC1(C)CC(=O)NCC1CN(C(c2csc(NC(C)=O)n2)=O)C1 c1(CCC(=O)NCC(CC)NC(c2cn(CCCF)nn2)=O)ccncc1 N1(C(=O)NC(c2ncc(C(F)(F)F)[nH]2)C)CCC=CCC1 C1(NC(=O)CCCN2CCCCC2)CCN(C(=O)CC2COCC2O)CC1O Cc1cncc(CC(=O)NC(C)(CNC(c2cnccc2N(C)C)=O)CO)c1 S(=O)(=O)(c1ccc(C#N)cc1Cl)N1C2CN(C(Cc3c(C)ccc(Br)c3)=O)CC21 N1(C(C2(C)CCOCC2)=O)CC(C(=O)NC(CO)CCCO)C2(CC2)C1 C1(CC#C)(C(N2CCC(CN(C)C)CC2)=O)CCN(C(C23CC(CO)(C2)C3)=O)C1 Cc1nc(C)c(C(=O)NC(C)(CNC(C2CCOC2(C)C)=O)C2CC2)s1 c1(C(N2C(C(C)(C)NC(=O)COc3ccsc3)CCC2)=O)ccc2nn[nH]c2n1 C1(CNC(C(CC#C)C)=O)CCC2(CN(C(=O)CC34COCC(C3)C4)C2)O1 C12(CNC(CCOCC(C)C)=O)CN(C(=O)C(=O)N(C)C)CC1CS(=O)(=O)C2 N1(C(c2sc(C(=O)OC)c(N)c2)=O)CCC(F)C(NC(c2ccnc(S)c2)=O)C1 C1(CNC(c2c(NC)cccc2)=O)CCN(C(C2CN(C3COC3)C2)=O)C1(C)C Cc1cccc2c1OC(C(N1CCN(C(C3(O)COC3)=O)CC13CCC3)=O)C2 C(=O)(C(C)(C)C(=C)Cl)N1C(C(N2C(CN(CC=C)C)CCC2)=O)CSC1 C=CCCCC(=O)N(CCC(=O)NC(C)(C)CCN)OC C1(CC(=O)NCC(C2CCN(C(C(C)NC(C)=O)=O)CC2)O)CCCC(F)(F)C1 CCCCCCCC(=O)N(CCCNC(=O)CCS(N)(=O)=O)CC Cc1noc(C)c1C(=O)NC1CN(C(=O)CCOC2COC2)CC1n1ccnn1 C1(CCOC)(NC(C(CCC)N(C)C)=O)CCN(C(C2NC(=O)OC2C)=O)CC1 CCCCC(COC)NC(=O)C(F)CN(C(=O)CCN(C)CCO)C C(CC(O)C(=O)NC(C)C(=O)NO)NC(C(=O)NC)=O C1(C(=O)NCCCCN(C)C(C23CC4CC2C3C4)=O)CCC(=C(F)F)CC1 C(=O)(CC(C)(O)C=C)N(C1CC1C1CCC1)C(CCCC=C)=O C1(C)(NC(CN2CCCC(CC)C2)=O)CCCN(C(=O)Cc2cnnn2C)C1 N1(C(C2(CC=C)CCOCC2)=O)CCC(CNC(c2nnc(C)s2)=O)C(F)(F)C1 CC(C)(F)C(C)(F)C(=O)NCC1(F)CCCN(C(c2ccc(C#N)s2)=O)C1 O=C(C(O)c1ccsc1)NCCNC(=O)CCNC(c1ccoc1)=O C(=O)(CC(=O)N(C)C)N(C1CCN(C(C2C(C(=O)OC)C2(C)C)=O)C1)CC C(=O)(C(C)CCOC)N(CC(CNC(C1(CC#C)CCC1)=O)C)C C(CCC(C(=O)NCC1CCC(C)(C)CO1)NC(=O)CS(C)(=O)=O)OC CN1CCCC1(C)NC(C1CN(C(c2cn[nH]c2)=O)CC12CC2)=O N1(C(C2CC(F)(F)C2)=O)CC2OCCN(C(c3cc(O)n[nH]3)=O)C2C1 CCC1=C(C(=O)NC(CC(=O)N2CCC(O)CC2C2CC2)C(F)F)CCCO1 c1(C(N2CCC(C)C(NC(=O)CC3=NNC(=O)C3)C2)=O)cc2ccccn2c1 CC1C(NC(=O)C=Cc2cocn2)CC2CCC1N2C(c1cccc(N)c1F)=O Cc1c(F)ccc(CN(C)CC2CN(C(=O)CCc3cn(C)nn3)C2)c1Cl Cc1cc(N2CCOC(C)(C)C2)ncc1S(=O)(=O)NCC1CCC=CCCC1 N1(C(C#CC(C)C)=O)C2CCC1C(CNC(c1cccc(Cl)c1O)=O)C2 N1(C(c2n(C=C)nnc2)=O)CC2(CO)CC1(C(=O)NCCN1CCOCC1)C2 CCN=C(NCc1coc(CC)n1)NCC1CCC(C)O1 C(=O)(C1=NNC(C(F)(F)F)C1)NCC1C(C)CN(C(c2ccsc2Cl)=O)C1 CCC(C)(C(=O)NC1CCCCC1NC(=O)C(C)(C)c1cncs1)C(N)=O C1(NC(C(C(C)O)C)=O)CC2CN(C(c3cnn(CC4CC4)c3)=O)CC12 C#Cc1cnn(C)c1C(=O)NC1CCC1NC(c1cccc(Cl)c1Br)=O C1(CNC(c2nccc(OC)c2)=O)CC(F)(F)CN1C(=O)C(C1CCOC1)OC c1(N2CCC(C(C)NC(C(C(C)C)O)=O)CC2)ccc(S(=O)(=O)NC2CC2)cn1 c1(C(N2CCN(C(C3(CC#C)CCC3)=O)CC2CC)=O)cccc([N+](=O)[O-])c1N C1(COC)CCCC(C)C1.c12ncccc1C(NC(=O)OC(C)(C)C)C(=O)NC2 C(=O)(C(C)(C)C1CCC1)N(CCCOCCNC(CCOC(C)=O)=O)C C=CC1OCCC1C(=O)NCC(CCC)NC(c1ccc(CO)cn1)=O N1(CCOCC)CCN(C(c2cc(C3CCCC3)no2)=O)CC1 C(=O)(C=CS(C)=O)NCCCN(C1CCCC1)C(c1c(C(C)=O)ccs1)=O CC1CN(C(=O)Cn2ccc([N+](=O)[O-])n2)CC(C)CN1C(C12CC(F)(C1)C2)=O CCCC(CCCO)C(=O)N1CCC(CNC(c2cc(O)n(CC)n2)=O)C(C)C1 c1(C(N(CCNC(C2(F)CC2C)=O)CC)=O)scc(Cl)c1Cl C1(OC)COCC1NC(=O)CCNC(c1ccns1)=O CC(CC(N)=O)C(=O)NCCCCCNC(C1(C)COCCO1)=O C(=O)(C1=CCCCC1C)NCC1(O)CCN(C(c2cnc(CC)nc2)=O)C1 N1(C(c2cc(CC)on2)=O)CCN(C)C(CNC(=O)Cc2cnns2)C1 c1(C(N2CCC(C=CC(=O)N(C(C3(C)CC3)C)C)CC2)=O)ccc2c(c1)CCC2 Cc1cc(C(=O)N(C)C)ncn1.C(=O)(C(C)C(C)NC(C1(CF)CC1)=O)NC S(=O)(=O)(c1ccc(C)c(C(N2CCN(C(=O)C(C)C(C)O)CC2)=O)c1)NCC C1(CNC(CC=C)=O)CCN(C(C2CC2C(=O)NCCO)=O)C12CC2 CC1CN(C(=O)C2=CSCS2)CC1CNC(c1ccc(Cl)cc1)=O C1(CNC(C2N(C(C)=O)CCC2)=O)C(C)CCN1C(=O)Cc1cnoc1 N1(C(C=C2CCC(C)C2)=O)CCCC2(C1)CN(C(=O)COCC(C)(C)C)CCO2 C12(C(N3CCN(C)C(CO)C3)=O)CCC(CC1)N(C(C1CC1C#N)=O)C2 O=C(C1=CCCCC1)NC1(C2CCCN2C(=O)C=Cc2cncs2)CC1 C1(C(=O)NC2(C)CCN(C(CNS(CC)(=O)=O)=O)C2)CC(=O)N(C)C(=O)N1 Cc1cc(=NCCC#CCO)[nH]c(N2CCCN(CC(C)O)CC2)n1 CC1OC2(C)CC1(C(=O)NC1CCCN(C(=O)Cn3nnnc3C3CC3)C1C)C2 C1(C(=O)NCC(C2CCC2)NC(c2c(C)noc2C2CC2)=O)CC12CCSCC2 N1(C(CCCC)=O)CC(C(F)(F)F)CC1CNC(c1ccnc(C(F)(F)F)n1)=O O(NS(=O)(=O)c1cc(Br)ccc1C#N)CCCOCC c1(NC(CSC)C)ncc(C(=O)O)cn1.c12nc(co1)C(=O)NC2 c1(C(N2CC3C(NC(C=C(C)C(F)(F)F)=O)(C3)C2)=O)ccnc2ccc(O)cc12 n1(Cc2ccncc2F)ncc(C(=O)NC2(C(C)(C)C)CC2)c1C1CC1 c1(C(N(C2CCN(C(CCC(C)OC)=O)C2)C)=O)cccn2c(C)nnc12 CC1CCC(NC(c2nnc(S)n2C)=O)CN1C(c1ccc(N)cc1Cl)=O N1(C(CCCSC)=O)CCC2(CC1)C(N(C)C(c1n[nH]cc1Cl)=O)CS2(=O)=O N1(C(C23N(C(=O)C(O)C4CC4)CCC2CCC3)=O)Cc2n[nH]cc2C1CO C12(SC)CCC(CN(C(C)(C)CNC(C3(C)CC(C)C3)=O)C1)C2.c12nnnn1C2 C1(C(N2CCC(CC(=O)N(CC=C)CC3CC3)C2)=O)CN(C)C(=O)N1 c1(C(=O)NC2CC3CC2N(C(C2(Cl)CCC2)=O)C3)cc2cnccc2o1 C=CCC(C)(C)C(=O)N1CCC(Cc2nn[nH]n2)(NC2CCCN(C)C2C)CC1 c1(OC)ccccc1CC(=O)NC1CC(CNC(=O)C(O)C(C)SC)C1 S(=O)(=O)(C1CS(=O)(=O)c2ccccc21)N(CC(F)F)CC C12(C(N(CC)CC3CCCCN3C(=O)CC3CCC3)=O)CCC(F)C1CC2 C=C(Cl)CC(C(=O)N(CCC(=O)NC1CC1)C)NC(=O)CCc1ccoc1 C=CC(C)(CC)C(=O)NCC(=O)NCC(N1CCC(CSC)CC1)=O N1(C(CN2CCC(C)C2)=O)CCC2(CC1)CC2NC(=O)C=CC1CCCCCC1 C(=O)(CCCC(C)(F)F)N1CC2(CC(NC(C(N3CCN(C)CC3)C)=O)C2)C1 c1(C(N(CC(CC)NC(=O)C(O)CN(C)C)CC)=O)ncnc(O)c1Cl C1(N(C(=O)CC2CCCOC2)CC#C)CCN(C(=O)CCCOCC=C)CC1 c1(C(CC(=O)N(C)CC2CC(F)CN2C(=O)CC(C)(C)C)O)cc(Cl)cc(Cl)c1 c1(C(N2CCC3C(C(=O)NCC(CC)(C)O)C3C2)=O)cnn2ccc(Cl)c(F)c12 c1(C(=O)NC2C(NC(CCSCc3c(C)noc3C)=O)C2)ccc(F)c(F)c1N N1(C(C(C)CN(C)C)=O)CCC2(CC1)CCN(C(C1Cc3cccnc3C1)=O)C2 c1(N(CC(c2ccccc2)O)CC(C)O)ncccc1CC(=O)OC N(C1CS(=O)(=O)c2ccccc21)C(c1n(C(C)(C)C)nnn1)c1cncnc1 CC(C)C(C(C)NC(C12CCC(C1)C2)=O)NC(c1nn(C(C)(C)C)cc1Cl)=O c1(CC(=O)NC(CC=CC(=O)NCC(CC)O)(C)C)cn(C)nc1C CC(C)(C)C(C(=O)NC1(CNC(=O)C(C)(C)C2CCC2)CC1)n1ccnn1 N1(C(C(C)NC(C)=O)=O)CC(CO)C2(CCN(C(=O)C(C)C(C)(F)F)CC2)C1 N1(C(C(C)(C)OC)=O)CCCC(C(=O)NCC(c2ccccc2)O)C1 CC1(C)Cc2cc(S(=O)(=O)N3CCOC(Cc4ccc(F)cc4)C3)ccc2O1 C1(NC(c2ccon2)=O)CN(C(=O)COCC2CCOC2)C2(CCC2)C1 c1(C(=O)NC(C2CCCCC2)C(C)NC(=O)C=C(Cl)Cl)cnc2scnc2c1 c1(OC)ccc2nc(N3CCC(CF)C3)[nH]c(=NCCC3CCC3)c2c1 c1(CNC(C(=O)NCCCSCC2CCCO2)=O)cc(-c2ccccc2)cs1 c1(NCc2ccnc(C)n2)nc(N2CCC(=NO)CC2)nc2c1ncn2C c1(C(=O)NC2CC(CNC(C3C(C(C)(C)C)CC3)=O)C2)cccc2c1C(=O)NC2 C1(CNC(C2C(SC)CCC2)=O)(NC(=O)C(C2CCCCCC2)F)CCCCC1 C(CCCC(C)NC(c1cncn1C)=O)NC(C1(C=C)CCC1)=O c1(C(N2CC(C(C)NC(c3c(C(C)C)ccs3)=O)C2)=O)c(F)cccc1[N+](=O)[O-] CC1CN(C(=O)CCS(C)(=O)=O)CCCN1C(c1c(N)cc(Cl)nc1Cl)=O N1(C(c2c(C(C)(C)C)cccc2)=O)CC2CCN(C(c3cc(F)c[nH]3)=O)C2C1 c1(OCCNC(C(C)(N(C(C(C)OCCOC)=O)C)C2CC2)=O)cccc(C)c1 N1(C(c2ccccc2C)C(=O)NCC(=C)C)CC(C)N(CC)C(C)C1 C1(NC(C(C)NC(=O)C(C)(C)C)=O)CCCCN(C(=O)Cc2c[nH]nc2O)CC1 CCC(CC)(CC)C(=O)N1CCCC2(NC(=O)Cc3ccc(O)nc3)CC2C1 Cc1[nH]c2ccccc2c1C(N1CCC(NC(c2cc[nH]c2C)=O)C(C)C1)=O c1(C(=O)NCC2(CNC(c3cnco3)=O)CC2)n[nH]cc1C(F)(F)F Cc1nc2ccccc2nc1C(=O)NC1CCC2CC1CN2C(c1cocn1)=O Cc1nc(C2CC2)[nH]c1C(=O)NC(C)(C)C(C)NC(=O)CSC(C)(C)C C1(NC(C2CN(C(C)=O)C2)=O)CCCC12CN(C(=O)CNC(C1CCC1)=O)C2 c1(N2CCC(OC)CC2)ccc(S(=O)(=O)NC(c2ccncc2Cl)C)cc1Cl C1(CCNC(C2(C=C)CCCCC2)=O)CN(C(=O)C(C)(C)COC)CCS1(=O)=O Cc1ncnc(C)c1CC(=O)NC1CCC1NC(=O)C(c1ncccc1F)(F)F CCCN=C(NCC1(C)CCCOC1)NC1CC(OCCN(C)C)C1(C)C N1(C(=O)OC(C)(C)C)CCCC2C1CCCN2C(c1cncc(F)c1C(=O)O)=O Cc1noc(C)c1CC(N1CCC1CNC(=O)CC1CCC(=O)N1C)=O CC1OC2(C(N3CCCC(CN(C)C(C4CC4C(N)=O)=O)C3)=O)CC1C2 C(=O)(C1CCCc2ccnn21)NCC1CC(NC(c2cnc(C)[nH]2)=O)C1(C)C C(=O)(CCCS(N)(=O)=O)NC1(C)CC(NC(C(F)(F)C2(OC)CCC2)=O)C1 C1(CC)CC(C)CN(C(=O)CC2C3CCC(C3)N2C(c2cc(CO)ccn2)=O)C1 C1(CNC(CNC(CNC(C)=O)=O)=O)CCN(C(=O)Cc2csnn2)C1(C)C CC(CC(N)=O)C(=O)NC1C=CCN(C(=O)CC2COC(C)(C)C2)C1 c1(C(=O)NCCN(C(=O)CCc2cscn2)CCOC)cc(C(C)C)[nH]n1 C=CC1(C(=O)NCC2(OC)CCC(C)C2)CCN(C(=O)C(C)SCCC)C1 CCC(CCC(=O)NCC1(F)CCCN(C(c2cccc(OC)c2O)=O)C1)OC CCCCCC(O)CC(=O)N1CC(C)CN(C(C2COCCN2CC)=O)C(C)C1 CC1(C)CC(CC(=O)NC2CCC3CCC23)N(C(c2cncc(Cl)c2)=O)C1 c1(CC)nn[nH]c1C(=O)N(C(C)CCNC(C1CCCC1C)=O)C c1(C(=O)NCCN(C)C(c2nc(Cl)cc(N)c2Cl)=O)cc(Cl)c(F)cc1F Cc1cc(CNC(=O)C(=O)C(C)C)oc1C(=O)NC1(C)CC1 N1(CCCOC)C(=O)CCN(CC2CCC(C)CN2C(=O)OC(C)(C)C)C1=O c1(C(N2CCC=C(CNC(C3(C)CCCC3O)=O)C2)=O)ccc2cnoc2c1 N1(C(CC2C(C)(C)CCC2)=O)CCCc2nc(O)ccc2C1 c1(C(C(=O)NCCCF)N(C(C)COC)CC)ccc2nc[nH]c2c1 C1(NC(c2nc(CCC)sc2)=O)CCCC(N(C)C(c2nocc2C)=O)C1 C1(NC(C2(CCC)CCC2)=O)CN(C(=O)CCS(=O)(=O)NC)CCC1(C)C C(CC1=CCN(C(c2ccnnc2C)=O)CC1)NC(c1cc(OC)ncc1Cl)=O CC(=O)CC(C)(C)C(=O)N1CCC(C)N(C(=O)C#CC(C)C)CC1 N1(C(c2n(C)nc(CNC(C3CC=CCO3)=O)c2)=O)CC(O)C(C)(C)C1 Cc1ncc(CNC(C2(C)CC(NC(=O)C(c3cncnc3)C)C2)=O)o1 c1(CC)onc(C)c1C(=O)NCC1(C(=O)N(CC)Cc2cccs2)CC1 c1(OC)cccc(-c2noc(C)c2C(=O)NCC2CC2NC(=O)CS(C)(=O)=O)c1 Cn1cc(NCC2CCC(C(=O)Nc3cnc(C4CC4)nc3)CC2)c(C(F)F)n1 c1(C(=O)OCC2CCN(C(C)=O)C2)cnccc1-c1cccc(F)c1 CCC(CNC(=O)CCCOC(C)(C)C)(CC)N(C(=O)C(COC)NC(C)=O)C N(C(=NCC(C)C)NCC1(Sc2cccc(F)c2)CC1)Cc1c(OC)nsc1OC C1(NC(CCC(C)OCC)=O)CCN(C(c2ccc(CO)c(F)c2)=O)C12CC2 C(=O)(CC1OCCc2ccsc21)NC(C)(CNC(c1cnc(Cl)s1)=O)C1CC1 C(=O)(CCCC(F)F)NCC1CN(C(CP(C)(C)=O)=O)CC1O C#CCC(C)(CNc1ncccc1OC(=O)CCCc1cn(C2CC2)nn1)CO N1(C(Cc2n(C)ccc2)=O)CCCC1C1CCCN1C(=O)C1=CC(C)(C)C1 C1(CC(=O)NCC(C)N(C(C2CCCN2C2CCCC2)=O)CC)CCC=CCC1 CC1(C)CCC(C)(C(=O)NC2CC(CNC(=O)CCOCC3CCC3)C2)CC1 C1(C(=O)NC2C=CC(CNC(C(C)=CC)=O)C2)CCc2nc(C(F)(F)F)cn2C1 CCC(CC)C(=O)N(C1CN(C(C2CCOC2)=O)C1)C Cc1cc(C(=O)NCC2CCC2NC(C2CCOC2(C)C)=O)ncc1N C1(NCCNC(c2cn(CCC)nc2)=O)CNCC(C)C1 c1(SC(C(=O)NC(c2cn(C(C(C)O)C)nn2)(C)C)C)ccc(F)cc1 C(CCCC(=O)NC1CCC(n2cc(C(=O)O)nn2)C1)(C1CCCCC1)OC c1(CNC(CN(C(CC2C(C)=NNC2=O)=O)C2CC2)=O)ccc(F)c(O)c1 Cc1ccccc1OCC(=O)NCC1CCN1C(=O)C(F)C1CCOC1 N1(C(Cc2c(C)noc2Cl)=O)CCCN(C(=O)Cc2ccsc2C)C(CO)C1 C(C)(C(O)C(=O)N1CC(C(N)=O)(CNC(=O)COC2CCCCC2)C1)SC N1(C(C2CC(C)OC2)=O)CC2CCCN(C(c3cnc4c(c3)nnn4C)=O)C2C1 C1(S(N)(=O)=O)(C(N2CCC(CCNC(C(C)NC(N)=O)=O)C2)=O)CCC1 c1(C(N2CCC(N(C(C=CC)=O)CCO)C2)=O)nc(Br)n2c1COCC2 N1(C(C(CC=C)CC)=O)CC(CO)C2(C1)CN(C(=O)CCSC)C2 C(=O)(C(C(C)C)n1cnnn1)NCC1CCN(C(CCC=CCC=C)=O)C1 c1(C(N2CC(OC)C(NC(=O)Cc3ccns3)C2)=O)c[nH]c2ccc(F)cc12 c1(SCC(=O)NC2(C)CCN(C(C(C)c3cccs3)=O)C2)ccc(F)c(F)c1 C#CC1CCC(CNC(=O)C=C(C)CNC(=O)Cn2ccnc2C)CC1 c1(C(N2CC(O)(CNC(c3cc4cc[nH]c4cn3)=O)C2)=O)ccc2c(c1)OCC2 c1(N(C2C(C)CCNCC2)C(c2cccc([N+](=O)[O-])c2)=O)csc2c(Br)ncn12 c1(C(=O)NCCCCOC)ccc(CNC(C2COC(C)C2)=O)s1 Cc1cc(C(=O)NC2CCCN(C(c3ccc(OC(C)(C)C)nc3)=O)C2)ccn1 C1(SCC)CCC(=O)N1C.C1(=O)CCOC(OCC)CN1 c1(C(N2CCC(CN(C(C3CCSC3)=O)C3CC3)CC2)=O)ccnnc1O c1(C(N2CCC(CC(F)F)CC2)C(=O)NC(C)(C)C)ccc(Cl)c(Cl)c1 C1(C(N(C)CC2(O)CN(C(c3cc(C#N)cs3)=O)C2)=O)CCCCC12CCC2 c1(C(C(N2CC(N(C)C(c3csc(O)n3)=O)C2)=O)O)ccc(F)c(F)c1 c1(NC(C)=O)cc(C(=O)NC2CN(C(=O)CC(C)c3cccnc3)C2)cc(F)c1 N1(C(=O)Cc2cccc(F)c2)CCN(C(=O)CNS(=O)(=O)c2cccs2)C2CC12 N1(C(C=CC)=O)CCC2(C1)c1[nH]cnc1CCN2C(C1(c2cncn2C)CC1)=O C1(C(=O)NCCC2CC(NC(=O)C(OC)OC)C2)(OCC)CCCCCC1 N1(C(C)=O)CCOCC1C(=O)NCCCN(C)C(c1sccc1C)=O c1(OC)nc(Nc2ccc(NC(=O)Cn3nc(C)c(Cl)c3C)cc2)ncc1Br C(=O)(CCP(C)(C)=O)N(C)Cc1ccccc1CNC(=O)Cc1c(Cl)cnn1C N1(C(C(C)NC(=O)NC)=O)CC(NC(=O)CCS(C)(=O)=O)CC12CCC2 C(=O)(CC1=CCN(C)CC1)N(CCCNC(c1c(CC)cccc1F)=O)C C(C(CC)n1cccn1)NC(=O)NCCCN(CCC#C)C N1(C(CCC(=O)OCC)C)CCOCC(C(=O)N(C2CCNC2=O)CC)C1 C(=O)(CC1COc2ccccc21)N1CCCN(C(Cc2c(C)cccc2)=O)CC1 C(=O)(C1=CCOCC1)N(C(CCCNC(C(CC)OC1CCCC1)=O)C)CCOC n1(CC)cc(Cl)c(C(C(=O)NC2CC2)N(C)C)n1.C1(CC(=O)NC)CC1 c1(C(N2C(CCNC(C(COC)(C)O)=O)CCCC2)=O)cc(C2CC2)cnc1Cl c1(CNC2C(C(=O)Nc3cncc(C(F)(F)F)n3)C2)cc(I)ccc1Br N1(C(CCCC(=O)OC)=O)CCC2(NC(=O)Cn3cc(C4CC4)cn3)CCCC12 c1(C(N2CC(C(=O)O)C(CCO)C2)=O)cccc(O)c1OC(F)(F)F C=CCCC(C(=O)NC1CC(C)(C)OC1=O)NC(=O)CC1CCC(=O)C1C C(=O)(C(CO)C(C)(C)C)NCC1(COC)CN(C(=O)C=C2CCN(C)C2)C1 C1(CN(C(=O)OC(C)(C)C)CC)CCCN1CC(CSC)CC1CCC1 S(=O)(=O)(c1ccc(N2CCCC(N3CC(O)C3)C2)c(Cl)c1)N(CC=CC)CC c1(OCC)ccc2cc(C(N3CCC4CC4(NC(C4CCC4)=O)CC3)=O)[nH]c2c1 N1(C(c2c(OC)ccs2)=O)CC2CCN(C(c3cnn(-c4nccs4)c3)=O)CC12 N1(C(C2=CC(C)(C)C2)=O)Cc2n[nH]cc2C1C(=O)NC1CC(C2CC2)C1 C(=O)(CC(C)C(=O)N1C(CC(N2CCCC2CC(C)O)=O)C2CCCC12)OC c1(-c2ccc(C#C)cc2)c(C)sc2nc(SCC(=O)OC)nc(O)c12 Cn1c(=N)[nH]c2cc(C(=O)NC3CC4(C3)CC(NC(C3CC3F)=O)C4)ccc12 C1(C(N2CCN(C(c3cnc(S)nc3)=O)CC2)=O)CS(=O)(=O)CC12CCC2 c1(C(N2CC(C(C)NC(c3c(C)cnn3C)=O)OCC2)=O)ccc2snnc2c1 C1(COC)CCCCN(C(=O)CCC2CCCCN2C(c2cccc(=O)o2)=O)C1 C(=O)(C1COc2ccc(Cl)cc21)NC(CC=C)CNC(C1CCCCCCC1)=O c1(C(N2CCC(NC(c3nccc(C#C)c3)=O)(CF)C2)=O)ccc(C#N)c(F)c1 N(C(=NCCC(=O)N1CCN(CC)CC1)NC1CC2CCC1O2)C(CC)C CC1CN(C(c2cc(C(C)(F)F)on2)=O)CCC1NC(=O)COCc1nc[nH]n1 c1(C(=O)NC2C(NC(C(C(C)(C)C)NC(N)=O)=O)COC2)ccc2nonc2c1 C1(NC(CSc2nc(C)[nH]n2)=O)COCCN(C(=O)C(C)NC2CC2)C1 c1(C(=O)NC2CN(C(CC(CC)O)=O)C(C)C2)cccc2cnnn12 C1(NC(c2cccc(C#C)c2)=O)CCC12CCN(C(=O)CC1C=CCC1)CC2 C(=O)(C(C)N=c1cc[nH]cc1)NC1CC(O)(CNC(C(C)OCC)=O)C1 C(=O)(CCCCC(=O)NC(C1CCN(C(C)C)CC1)CC(=O)O)OCC c1(C(=O)NCC)cc(OC)ccc1-c1csc(NC(c2ncsc2NC)=O)n1 C1(NC(C=C2CCC(C)CC2)=O)CN(C(C2(C#N)CC(C)C2)=O)CC1(C)C c1(C(N2CCN(CCNC(C3C(OC)CCC3)=O)CC2)=O)coc2c1CCCC2 c1(CNC(CSCCCC)=O)cn(C2CCN(C(=O)C(C)CF)C2)nn1 N1(C(Cn2c(C)nnn2)=O)CCN(CC(C)NC(=O)CC2(C)CCCO2)CC1 C1(C(=O)NCC(c2ccncc2)C)(CNC(=O)Cn2cnc(=N)[nH]2)CC12CCC2 C12(NC(C(C)OCCN(C)C)=O)CCC(NC(C3CC(Cl)(Cl)C3)=O)(CC1)C2 N1(C(C2(CC=C)CCCN2C(c2cccc(C)c2O)=O)=O)CC2(CNC(=O)C2)C1 Cc1cc(F)cnc1C(=O)NCc1nc(C(=O)NC2C(O)CC2O)co1 c1(C(=O)NCC2N(C(C(C)OCCOC)=O)CCCC2)cncc(C)c1Cl C1(NC(c2c(CC)con2)=O)CN(C(=O)CNC(=O)OC)CC2(CCC2)C1 N1(C(C(C)OC2COC2)=O)CCC(CF)(NC(c2cnc(S)n2C)=O)C1 C(=O)(C(C)CC(C)(C)C)NCC(C(N1C(CC)(CO)CCC1)=O)C C1(C(=O)NC(CNC(c2c(CC)scc2)=O)C2CCC2)Cc2ccccc2O1 C1(C(N2CCCC(NC(c3cnnc(O)c3)=O)C2)=O)CC(C2CC2)=NO1 c1(SCCC(N2CC(CC=C)(NC(=O)CC(C)C)C2)=O)ccc(C)c(C)c1 N1(CC(=O)NCCC(C)C)CC(NC(=O)C(C)n2cccn2)CCC1C C(=O)(CC1=NNC(=O)C1)N1CCC(C)(CNC(CC(CC)C2CC2)=O)CC1 CC1CC(C(=O)Nc2ccccc2)CCN1C(C1CCCCCCC1)=O C1(NC(c2cc(CC3CCC3)c[nH]2)=O)CCN(c2nc(C3CC3)ns2)CC1O N1(C(c2ccn(CCC)n2)=O)CC(NC(=O)C(C)CCO)C(C)(C)C1 N12CCC(CC1)OCC2.C1(C(=O)O)C=CCN1CCO C1(NC(CC(=O)NCC#C)=O)CC(CNC(c2sc(CO)nc2C)=O)C12CCC2 C1(O)(CC(=O)N(C(CNC(c2c(C)oc(CO)c2)=O)C)C)CCCCCC1 C1(C(=O)NCCC(=C)CNC(=O)C(F)(F)c2nccn2C)CCCC(O)C1 Cc1cccc2c(C(=O)NC3C4CC3N(C(C3(C(F)(F)F)CC3)=O)C4)cccc12 c1(OC)cc(C(N2CCC(C(C)NC(c3cc(C)nn3C)=O)CC2)=O)cc(F)n1 C(=O)(C1=CCSC1)NC(CNC(=O)CC1(C(F)(F)F)CC1)CO c1(C(N(CCN(C(CCNC(=O)NC)=O)C)C)=O)c(F)cc(OC)cc1Cl c1(C(=O)NC(CCCNC(c2cc(CC)cc(Cl)c2)=O)C)cc(N)c(C)cc1Cl C1(CC=C)CCCCN1c1cc(N2CCC(C(F)(F)F)(CO)C2)ncn1 CC1CCCC(CC(=O)NC2(CF)CCN(C(=O)CCn3cccn3)C2)O1 Cc1cc(Br)ccc1C(=O)N(C1CCN(C(=O)C(C)C(C)O)CC1)C C1(C(=O)NC2(C(N(CC)Cc3ccoc3)=O)CCCC2)C(C)(C)C1(C)C C1(NC(c2cc(CNC(c3cnc(C)s3)=O)no2)=O)CCC(=O)N(C)C1 Cc1ncc(C(=O)NC2CCC2CNC(=O)CCC2OCCO2)c(C(C)C)n1 Cc1ncc(C(=O)NCCC(C)N(C(=O)CC2COCCO2)C)cc1N C=C1C(C(=O)NCCOCCCNC(=O)CCC2CC2(Cl)Cl)C1C(=O)OC c1(CC(=O)NCC(C)CNC(c2cc(C(C)(C)C)n[nH]2)=O)cnc(C(=O)O)nc1 Cc1cc(NCCN(CC(=O)N(C(C)(C)C)C(C)C)C)cnc1-n1cccn1 C1(C(=O)NC(CC(=O)OCC)C)C(C)OCCN1C(=O)C=NOC Cc1cc(C(N2CCCC2(C)CNC(=O)C(C)OCC2CC2)=O)c2n[nH]cc2c1 c1(Cn2c(-c3nc(C)oc3)nc(C3CSC3)n2)ccc(Cl)cc1Cl Cc1c(C(=O)N(C2CN(C(c3cn(C4CCOC4)cn3)=O)C2)C)cccc1C#N N1(C(C(=O)NC(C)C)=O)CCC(F)(CNC(C2CCN2C2CCCC2)=O)C1 CCC(F)(C(=O)OC)C(=O)N(CC(C)NC(=O)CCN1CCC1)C C1(NC(CCCNC(CC(C)(C)C)=O)=O)CC2CN(c3ncccn3)CC2C1 C(=O)(CCCN=[N+]=[N-])NC(C(=O)N(CCC(O)CO)C)Cc1cc[nH]n1 C12(C(=O)NC3CCCCC3NC(C3CC34CCC4)=O)CC3CC(C1)CC(O)(C3)C2 N1(C(COC(CC)(C)C)=O)CCN(C(c2nocc2C)=O)CC1C C1(NC(C(CC)N(C)C)=O)(CO)CCCN(C(c2cncc(Cl)c2C)=O)C1 c1(SCC(=O)NC2C3CN(C(c4c(C)cco4)=O)C2C3)ccc(F)cc1F c1(C(=O)NCC2N(C(c3nc(C)nc(O)c3)=O)CC(F)C2)ccc2c(c1)OCC2 c1(C(N2CCC(C)(NC(C3CCC(C)(C)O3)=O)CC2)=O)cncc2ccccc12 N1(C(C(C)N(C)C)=O)CC(C)(C)CC1CNC(c1coc(N(C)C)n1)=O CC1(C)CC(=O)C=C(c2cccc3nc(C(N4CCCCC(C)(F)C4)=O)sc23)C1 CC(C)(C)C(O)C(=O)N1CCC(OCCNC(c2ccn(C(F)F)n2)=O)C1 N1(C(=O)NCCc2cc(O)cc(F)c2)CCOc2cc(F)ccc2C1 N1(C(c2scc(OC)c2OC)=O)CCCC(NC(c2cc(N)ccc2O)=O)C1C C1(NC(CCOC)=O)CCC2(CC1)CN(C(c1ccc(F)o1)=O)CCO2 C(=O)(NN1CCS(=O)(=O)CC1)C1(C(=O)OC(C)(C)C)CCN(C(=O)OC(C)(C)C)C1 c1(-n2cc(C3N(C(c4c(C)nsc4C)=O)CCC3)nn2)ccc2occc2c1 C1(CC(=O)N(C(C)CNC(=O)CCc2cn(C)nc2C)CC)CC(C)(C)OC1=O C1(NC(CNC(=O)OC)=O)CCN(C(c2ccc(-c3ccncc3)o2)=O)CC1C C1(C(=O)NCc2ccc(Br)nc2)CC(F)(F)CN1C(c1cc(C2CC2)on1)=O Cc1cnc(C(C2CC2)NC(=O)NCC(C(C)C)c2ccnn2C)[nH]1 n1(CC2CN(C(C(=O)NCC)=O)C2)cc(CCNC)nn1 c1(C(N2C3(CNC(CCc4ncn(C)c4)=O)CC(C2)C3)=O)csc2nccn12 N1(C(c2c(C)nnn2C)=O)CCC2(CCOCC2)C(CNC(C2CC(F)C2)=O)C1 c1(NC(N(C(C)C)Cc2cnn(C)n2)=O)ccc(C2CCC(=O)N2)cc1 C(c1ccc(Cl)nc1)=CC(=O)NC1(CNC(C2(CO)CCCC2)=O)CCC1 C1(NCC(c2cccc(Cl)c2)N(CC(=C)C)C)CCC(F)(F)CC1 CCCCCC(F)C(=O)N(C)CC1CCC(NC(C2(CC)CCCO2)=O)CC1 N1(C(c2ccc(OCC)cc2)=O)CC2CC(C1)N(C(=O)CN(C)S(N)(=O)=O)C2 Cc1nc2cc(C(N3CCCC(C)(NC(=O)CSc4cccs4)C3)=O)ccc2o1 N1(C(CCc2ccnc(C)n2)=O)CCC(C)C(NC(=O)Cc2sc(O)nc2O)C1 Cc1cc(N)c(C(N2C3CCC2C(NC(=O)CCCc2cccs2)C3)=O)cc1F C(=O)(CCC(=O)N1CCC(C(C)NC(=O)CN2CCC(OC)C2)CC1)NC N1(C(c2cn(CC)nn2)=O)CCC(N(C(=O)C(C)n2cccn2)CCO)CC1 C1(NC(C(C2(O)CCCCC2)CC)=O)CN(C(=O)Cn2nnnc2C)C(C)(C)C1 CC(CCc1ccc(F)cc1)C(=O)NC1CC(CNC(C2CCC(O)C2)=O)C1 c1(OCC)cc(C)nc(N2CCNCC2C(=O)NC(c2cc(F)cc(Cl)c2)C)n1 N1(C(C(COC)OC)=O)CCCC(O)(CN(C)C(c2cnn3c2OCC3)=O)C1 C1(NC(c2ccn(C3CCCC3)n2)=O)CC(O)CN(C(C2(F)CCCCC2)=O)C1 Cc1cc([N+](=O)[O-])ccc1C(N1CCCC(NC(C)=O)CC1)=O C1(CNC(C2CCC(C3CC3)N2C(=O)C=Cc2cscn2)=O)C2CCCCCC12 C1(N(C(c2c(CC)occ2)=O)C)CCN(C(c2cc(CC)c(C)s2)=O)CC1C c1(C(N(C2CCN(C(C(C3CCC3)OCC)=O)C2)C)=O)csc2c(F)cccc12 C1(CC=C)(NC(c2nc(CC)cs2)=O)CCCN(C(=O)C(O)C(F)F)C1 C1(F)(CNC(c2cccc3cnsc23)=O)CC(N=c2[nH]nc(C3CC3)s2)C1 N1(C(C(=O)C2CC2)=O)CCC2CC2(C(N2CC3C(CO)C3C2)=O)CC1 Cc1ccc(NC(c2cccc(NC(=O)Cc3ccc(Cl)c(F)c3)c2)=O)cc1I c1(C(=O)NCCCCCCNC(C(CC#C)C2CC2)=O)ccn2c(C)cnc2c1 c1(NC(C2C(C)CN(C(C3C=CCC3)=O)C2)=O)ccc(O)c(CO)c1 C(=O)(CC(C(C)(C)C)NC(c1ncc(CC)cn1)=O)N(CCCO)CC#C c1(C(N2C(C)CN(C(CCCCC)=O)C(C)C2)=O)[nH]c2ccc(Cl)cc2c1Cl C1(CNC(C2(CNC(CCC(=O)NCC)=O)CC(C)(C)C2)=O)NC(=O)OC1(C)C C1(C(=O)NCC2C(C)(C)OC(=O)N2)CCN(C(C2(CO)CC2)=O)C(C)(C)C1 O=S(=O)(c1cc(F)cc(F)c1O)N1CCn2c(C3CC3)nnc2C1 CC1CC(CNC(=O)C(O)CN(C)C)CN(C(c2ccc(C3CC3)nc2)=O)C1 c1(C(N2CCC(CNC(CCNC(COC)=O)=O)C2)=O)c(F)ccc2occc12 C1(OCC)CCCC(NC(=O)CCC2(C)CN(C(C3CCSC3)=O)C2)C1 CCCCCC(C)NC(c1cccnc1CNC(c1ccncc1F)=O)=O N1(C(C2C3CN(C(C=Cc4n(C)ncc4)=O)C2C3)=O)CCCC2CCCCC12 c1(C(N2C3CN(C(CCCNC(=O)OC)=O)C(C3)C2)=O)nn(C)cc1S(N)(=O)=O Cc1cc2nc(n1)NCc1c(n[nH]c1C)C(=O)N1C3CN2C(C3)C1.C1(CO)CC1 C=CCC(CNC(c1cnnc(C)c1)=O)C(=O)NC(CC1CC1)C1CC1 N1(C(C2CCN(C(C)=O)CC2)=O)CC(NC(c2cn[nH]c2)=O)CC12CCCC2 C1(c2cc(C)no2)COCCC1NC1CC(n2ccnn2)C1 C(=O)(C(O)CCCNC(c1ccc(O)c(F)c1)=O)NCC(C1CC1)SC c1(C(=O)NC(CNC(CCOCCC)=O)C(C)C(C)C)cccc2c1CNC2=O c1(C(=O)NC2CC2C(=O)Nc2ccncn2)cc([N+](=O)[O-])c(Cl)c([N+](=O)[O-])c1 C(=O)(CCCCCN(C)C(c1cc[nH]c1CC)=O)N1CC(C(=O)OCC)C1 c1(C(=O)NCC(C(=O)NC(COCC)C)N(C)C)ccn(C)c(=O)c1 c1(CC)c(NCCN2CC(C)OC(C)C2)nc(Cl)nc1Cl N1(C(C2(CC=C)CCN(C(C)=O)C2)=O)CC2COC(=O)C2C1 c1(C(N(CCC(C(C)C)NC(C2C(=C)C2)=O)C)=O)cn2cnnc2cn1 C(CCC(C)CC(=O)OCCCN1CCCC1)=C(C)C C[S+](C)CCC(O)C(=O)NCC1CCC1NC(c1ccc(C(F)(F)F)nn1)=O C12CCC(CC1)C(=O)N1CCN(CC1)C(=O)O2.Cc1cc(CC(=O)N(C)C)on1 N1(C(Cc2cnc(C)s2)=O)CCOCC1CC(N1CC(F)C(F)C1)=O C1(C(N2CC(CC(C(=O)N(C)Cc3c(C)ccs3)F)C2)=O)CCC=CCC1 c1(C(=O)NC2CN(C(c3cncc(OCC)c3)=O)CC2C)cc(Cl)ccc1F c1(C(=O)NC(CNC(C(CC(C)C)F)=O)(C)C)cc([N+](=O)[O-])ccc1Br C#Cc1cc(C(=O)N(C(C)CNC(c2cncc3c2CCC3)=O)CC)cc(N)c1 c1(N2CC(C)N(C(c3ccnn4cccc34)=O)CC2)ncnc2c(F)cccc12 c1(C(N2CC3(CN(C(c4c(CC)cco4)=O)C3)C2)=O)ccc([N+](=O)[O-])c(O)c1 c1(OC)ccc(C(=O)NC(CNC(c2cc(C)n(C(F)F)n2)=O)CO)c(F)c1Cl C(=O)(C#CC1CCCO1)N(C1CCN(C(=O)C(C(C)C)NS(C)(=O)=O)C1)CCC c1(C(=O)NC2(CO)CN(Cc3cccc(C(F)(F)F)n3)C2)c(F)cccc1F Cc1cc(Cl)ccc1C(=O)NCC(O)CNC(=O)C(C)(C)C12CC(C1)C2 S(=O)(=O)(CCC(=O)NCC1CCCCN(C(=O)C(F)=C(C)C2CC2)C1)NC C1(NC(C(=CC2CCCC2)C)=O)CC(O)CN(C(=O)Cc2n[nH]cc2Br)C1 C1(NC(=O)C(c2ccccc2)=O)C2CCN(C(=O)C(F)=C3CCC3)CCC12 N1(c2ccc(CC)cc2)C(=S)NC(c2cccc3nccn23)C2=C1C(C)NC2=O c1(OC)ncnc(NC2CCC(C(=O)NCc3ccc(C#N)nc3)C2)c1C N1(C(C(C=C=C)C)=O)CCCC(NC(c2ncn(C)n2)=O)CC1 O(NC(=O)C(c1ccc(C)cc1)C(=O)OC(C)(C)C)CCCC#C Cc1[nH]c(C(=O)NCC2CCN(C(c3ccc(C(C)C)s3)=O)C2(C)C)c(C)c1C N1(C(CCSc2cn(CC(CC)CC)nn2)=O)CCC12CC(C(=O)O)C2 Cc1cnc2nc(C(=O)NC3CC(CNC(c4sccc4CC#N)=O)C3)nn2c1 Cc1c[nH]c(C(=O)OCC(=O)C(=O)NC2(c3cccs3)CC2C)c1 NS(=O)(=O)c1ccc(C(=O)Nc2ncc(-c3c(F)cc(O)cc3F)cc2O)cc1 C1(C(=O)NCC2(NC(C3SCCS3)=O)C(C)C2)CCC=CO1 C1(C)(CC(C)C)CC(=O)N(CN2CCOC(c3ccc(F)cc3)C2)C1=O C1(C(N2C(CC)CN(C(c3coc(C(N)=O)c3)=O)CC2)=O)Cc2nnc(C)n2C1 CCCC(C(=O)N1CC=CC1C(N1CCC(CCC)C1)=O)N(C)C Cc1ccc(F)c(-c2ccc(NC(c3ccn(-c4ccccc4)n3)=O)cn2)n1 Cc1scc(C(=O)N(CCC(C(C)C)NC(=O)C(C)N(C)C)C)c1Br CCCCCCC(F)C(=O)N1CCN(C(=O)C=CCF)C(CCOC)C1 C(N=c1cc(C)nc(C)[nH]1)C1OCCCN(C(CCCSC)=O)C1 S(=O)(=O)(c1csc(C2OCCO2)c1)CNC(CN(C)C)CCO c1(C(=O)Nc2c(OC)ccc(C)n2)cnc2c(C3=CCNCC3)cnn2c1 N1(C(c2c(OC)nccn2)=O)CC(O)CC1(C)C(N1CC(C)OCC1C)=O C1(CCNC(c2cnn(CC)c2Br)=O)CCCN(C(=O)CSC(C)C)CC1 N1(C(C(CC=C)CNC(c2[nH]cc(C)c2C)=O)=O)CCC(C)(O)C(O)C1 Cc1nn2cccnc2c1C(=O)NCC1CN(C(=O)COC2CCOC2)CC1C N1(C(C(C)(C)C2CC2)=O)C(CNC(C2(F)CCOC2)=O)CC2CC12 Cc1ccc2[nH]c(C(N3CCOCC(NC(=O)C(CO)N(C)C)C3)=O)cc2c1C c1(SCCNCC(CSC)(C)C)nnc2n1CCNC2 N1(C(=O)NCC(c2cccnc2)C2CC2)CCCC(Cc2cccc(CO)c2)C1 c1(CN2CC(NC(c3ncccc3Cl)=O)C(F)(F)C2)cc(Cl)c(O)c(Cl)c1 C(=O)(CC(C)(C)n1cc(CNC2CCNCC2)nn1)N1CC(C(N)=O)(OC)C1 N1(CC(C)C)N=C(C(=O)N2CC3CC2CN3C(c2ccccc2Cl)=O)CCC1=O C(C(C(F)(F)F)OC)NC(c1cncc(CC)c1)c1n(CCOCC)nnn1 c1(C(=O)NCC2CC3(CCC(CN)OC3)C2)cccc2cc(F)ccc12 c1(C(=O)NC2CCC(N(C(=O)CCN3CCCCC3)C)CC2)cnc2[nH]nnc2c1 N1(C(CC(COC)C)=O)CCCN(C(=O)CCc2ccco2)CCC1 c1(-n2cc(C3(O)CN(C(C4CCCS4(=O)=O)=O)C3)nn2)cc(Cl)nc(Cl)c1 Cc1nc(C2CCCO2)sc1NC(C1CCN(CC2CC2)CC1)=O C1(C(N2CC(NC(=O)C=NOC)C3(CC3)C2)=O)(NC(CC)C)Cc2ccccc2C1 Cc1cccc(C(C(F)(F)F)NC(C2CCN2C(=O)OC(C)(C)C)=O)c1 c1(C(N2CC(SC)C(NC(C3CC(Cl)(Cl)C3)=O)C2)=O)cccc(O)c1C Cn1ccc2nc(N3C4CC3CN(C(C3CC3(C)C)=O)C4)nc(Cl)c12 c1(C(=O)NCC2CCN2C(=O)CCc2ncco2)cc2c(cc1Br)CCN2 c1(COC)ncc(C(N2CC3CC3(NC(=O)CC3CCCOC3)C2)=O)c(O)n1 C(=O)(CCCCC(N)=O)NC1CN(C(CCCOC(C)C)=O)CC1CO c1(C(=O)NCCC2(CNC(=O)C#CC3CC3)CC2)ccc([N+](=O)[O-])cc1Br Cc1cn2c(n1)CN(C(=O)CCCNC(c1cc(C)sc1C)=O)CC2 c1(CNC(Cn2ncc(OCC)c2)=O)ccccc1NC(=O)OCCCOC N1(C(C(=O)N(C(C)C)C)C)CCCOC(CNC(=O)CC(C)(C)C)C1 C(C(CC(F)(F)F)NC(=O)C(c1ccccc1)=O)NC(C=Cc1ccc(C)s1)=O CCCCCCC(=O)NCCN(C(=O)Cc1scnc1-c1cccs1)CCOC NS(=O)(=O)c1ccc(C(=O)NCC2C3CN(C(=O)Cc4cnsc4)CC23)c(Cl)c1 N1(C(C(=O)NCCCOC)C(C)C)C2CCCC1CC2 c1(C(C)(C)C)cc(C(N2CCC(NC(C3CCOCC3)=O)C2)=O)cs1 C(=O)(CC(COC)NC(=O)Cc1ccc(F)cc1)N(CCC)CCO C1(C(=O)NCC(C(C)C)NC(=O)C=C(Cl)Cl)CN(C(N)=O)CCO1 C12(NCC3CCN(C4CCCCC4)C3)CCC(C(=O)OC)(CO1)C2 C1(CC(N2CC(CC(C(=O)N(C3CCCC3)C)F)C2)=O)CC(C)(C)CO1 c1(Cn2c(C(C)C)nc(C3CC3)n2)cc2ccccc2o1.N12CC(CC1=O)C2 N1(C(CC(C)(C)N(C)C(C2CC3CCC(C2)O3)=O)=O)CCC2(COC(=O)N2)C1 CC1=C(C(=O)NC2CCN(C(=O)C=Cc3nccs3)CC2F)CCS1(=O)=O C1(C(N(C2CCN(C(=O)C(O)Cn3cncn3)CC2)C)=O)CC(C)(C)CN1C N1(C(C2CC=CC(NC(CC3C(C)(C)C3)=O)C2)=O)CC2(CO)CC2(CO)C1 c1(C(N2CCC(N(C(C3SCCS3)=O)CC)C2)=O)ncccc1N C1(NC(=O)NC(c2cccc(OC)c2)C(=O)OC)CCCCC12CCC2 c1(CCC)ncc(N(C(C(=O)NCCN(CC)CC)C2CCCC2)C)s1 N1(CC)CCCC1CC(=O)OCC1CC(CC2CCC2)CO1.c1(CN)cn[nH]c1 CC1=C(C)CC(C(=O)N(C2CC(C(=O)NCC3CCSCC3)C2)C)CC1 c1(C(N(CCCOCCN(C(C2(COC)CCC2)=O)C)C)=O)cc(C)ccc1C N1(C(Cc2c(C)nsc2)=O)CCN(C(C2CCOC2C)=O)CC1CC(C)(C)C c1(-c2c(C)c(Cl)ccc2)csc(=Nc2ccnc(Cl)c2)n1C1CCC1(C)C(F)F N1(C(Cc2cn(CC)nc2C)=O)CC(NC(=O)CN(C)C(C)=O)C(C2CC2)C1 C=CC(F)(F)C(=O)N(C(C)(C)CC(=O)NC1CCCCC1OC)C CC(C)C(C)C(=O)NC(C)CCC(=O)NC1(CCF)CC1 C1(CNC(=O)CCc2ccoc2)CCCCN1C(=O)COC1CC1 N1(C(c2n(C)ccn2)=O)CCCC(O)(CNC(c2cccc(F)c2Cl)=O)C1 C1(C(N2CC3(CN(C(CCCOC(C)(C)C)=O)C3)C2)=O)COc2ccccc2O1 c1(OC)ccc(S(=O)(=O)N(c2ccc(Br)cc2)CCN2C3CNC(=O)C2CC3)cc1 c1(C(=O)NC2C(CNC(C(C=C)O)=O)C2)ccc(Br)c2c1OCCC2 CS(=O)(Cc1ccc(Br)cc1)=NS(=O)(=O)c1ccc(C(=O)N=S(C)(C)=O)cc1 c1(N(CCCC=C)C)nc(=NCC2(C)CCS2)[nH]c2c(C)nn(C)c12 C1(NC(Cc2cn(CC)nn2)=O)CN(C(c2cc(Cl)ncc2NC)=O)C(C)(C)C1 CC(F)CC(=O)N1CC(CNC(C2(C)CCCO2)=O)C1 c1(C(N2CCC(O)(C(C)NC(C(C)=CC)=O)C2)=O)cc(C)cc([N+](=O)[O-])c1 CCC(C)(C(F)F)NC(=O)C(CCC)n1cc(-c2ccccc2F)nn1 C(=O)(CC1=NN(C)C(=O)C1)N(C1CCC(NC(c2cccc3c2COC3)=O)C1)C CC(N=c1cc[nH]cc1S(=O)(=O)N1CCCN2CCCC12)C1CSC1 CCC1=C(C(=O)NC(C2CCN(C(=O)CC(COC)COC)C2)C)CCCO1 CC1C(NC(=O)C(F)C(F)(F)F)CC2CCC1N2C(=O)CC1C=CS(=O)(=O)C1 c1(C(=O)NC(C)C(C)NC(c2cc(Cl)ccc2Cl)=O)ccc2sncc2c1 C1(C(C(=O)NCC)N(C(C)C)CC2CC2)CCOC1(C)C C1(C(=O)O)(NCC(=O)N(C2C(C)C2)C)CCN(C(C2CC2(C)C)=O)C1 N1(C(c2ccon2)=O)CC2=C(C1)CN(C(c1ccnn1C1CC1(F)F)=O)C2 c1(CCCCC)ccc(NC(C2CCC(NC(=O)Nc3nccs3)CC2)=O)cc1 C1(C(=O)NCC(CC)O)CC2CCN(C(c3cccc(F)c3N)=O)CC12 N1(C(Cn2cc(C(=O)N(C3CCCCC3)CCO)nn2)=O)CC2COCC(C2)C1 CCC(CC)C(F)C(=O)NC1CCCC(C(N2CC([N+](=O)[O-])C2)=O)CC1 N1(C(CC)=O)CC2CCC(C1)N2C(C1CCN(Cc2ccccc2)CC1(F)F)=O N1(C(c2ccn(CC)c2C)=O)C2CCC(C2)C1CNC(=O)Cc1cnn(C)c1C C1(C(N(CCOC)C)=O)CN(Cc2ccc(Cl)cc2)CC1C(F)(F)F C1(N(C(C2CCC(C(F)(F)F)CC2)=O)Cc2cccs2)CC2CCC1C2 C1(C(C(=O)NC2(C)CC2)N(C)Cc2ccc(Cl)o2)CC2C(C1)C2(F)F CC1CCN(C(=O)C(C)(C)c2cncnc2)CC1NC(=O)Cc1nccs1 n1(CC)cc(NC(c2cccc(CNC(=O)CC(C)OC)n2)=O)c(C#N)n1 C(CNC(=O)C(O)CCN(C)C)(CC(F)(F)F)NC(c1n(C=C)ncc1)=O C1(CC(N2CC(CCNC(=O)Cn3nnc(C)n3)C(C)C2)=O)(OC)CCOCC1 C(=O)(C1=NN(C2CC2)C(=O)CC1)N1CC=CC(NC(CCc2onc(C)n2)=O)C1 Oc1nc2cc(CNC3CCC(CCCCCBr)C3)ccc2o1 C1(NC(CNC=O)=O)CCCC(CNC(C23COCC2C3)=O)C1 c1(C(=O)NC(CC=C)CNC(C2CCCCO2)=O)c(C)nnn1C N1(C(=O)Cc2ccsc2Cl)CCC2CN(C(C3CCN(C4CC4)C3=O)=O)C2C1 C(=O)(C1=CCN(C)C1)N1C(C(=O)NCC2(CC)CCOC2)CCCC1 Cc1noc(CCCNC(=O)C=CC(C)NC(c2cc(Cl)c[nH]2)=O)n1 c1(C(N2CCN(C(=O)Cc3cnoc3)CC2CF)=O)sc2sccc2c1Cl CC1(CNC(C2CCN2CC2C3COCC23)=O)CCOCC1 C1(NC(c2cccc(C)c2Cl)=O)CCN(C(=O)C=Cc2cccs2)CC1(C)C CN1CCN(C(=O)C=Cc2cncn2C)C(C(=O)NCC(c2ccccn2)O)C1 c1(C(N2CC3CN(C(c4nn(C)c(F)c4)=O)CC3C2)=O)cccc2c1nnn2C N1(C(=O)C=C2CCOCC2)CCCC(C(C)(O)CNC(=O)CCn2cnnn2)C1 CCC(C(C)(C)O)NC(C1(C)CN(C(c2sccc2C#N)=O)C1)=O N1(C(c2cc(C)nnc2O)=O)CCC2CN(C(=O)CCC3CCCOC3)CC12 c1(CC(C(=O)OC)CNCC2(CSC3CC3)CC2)ccc(C)cc1F C(=O)(C(CC1CCCO1)NC(=O)Cc1nccn1C)OCC c1(C(=O)NC2CC3CN(C(CN(C)CCO)=O)C2C3)cc2cccn2c(O)n1 N1(CCNC2S(=O)(=O)N3C(C)(CCC3)C2)Cc2ccccc2OCC1=O CCCC(F)C(=O)NCC1(C)CCC(NC(c2ccncc2OC)=O)C1 C1(CCOC)CN(C(C2CN(C3CCC3)C2)=O)CCN1C(=O)C1=NOCC1 Cn1c(=O)nc(O)c2cc(C(=O)OCc3ccc[nH]3)cnc12 C1(OC)CC(CC(=O)NCC2(C(=O)NCC(=O)N(C)C)CC2)C1 N1(C(C(C)CF)=O)CCC2(CCC2)C(NC(C2C=CC=CC=C2)=O)C1 c1(OC)cccc(CCC(=O)NC2CC2NC(=O)C=Cc2cn(C)cn2)c1F C1(C(CO)NC(=O)CC(Cl)Cl)CCN(C(C2CC2F)=O)CC1 C1(C(=O)NC(C2(O)CCCCC2)C(=O)NCCSCCOC)CCN(C)C1=O c1(C(N(CCC(C)NC(C2CCC(O)C2)=O)C)=O)ccc2ccnn2c1 C(=O)(CCCCCCn1cc(C(C)NC)nn1)N(C(C)CC)CC=CC C(CC(=O)NCc1ccccc1CO)(C(F)F)NC(C12CCCC1C2)=O c1(N2CCOCC(CNC(c3c(OC)ccc(C)c3)=O)C2)ncnc2c1CCO2 CC1CCC(C)N1CC(N1CC(O)(CCNC(=O)CCc2cncs2)C1)=O N1(C(C2C(CC)C2)=O)CCC2CN(C(c3c4c(nn3C)CCOC4)=O)CC2CC1 CC1(NC(C2CCCC2O)=O)CC(NC(=O)Cc2nc[nH]n2)C1 C1(C(N(CCC(=O)NC(C)C(C)CO)CC=C)=O)CC2(CSC2)C1 C(C)(C(C(=O)NCC1(C)CSC1)NC(=O)COCC(F)F)OC c1(CC)cc(C(N2CCC(CNC(=O)CCNC(N)=O)C(O)C2)=O)ccc1O C=C1CSCC(=O)NCC1.c1(C(=O)NC)cnoc1-c1ccc(C)o1 C1(C)(NC(C(c2scc(C)n2)C)=O)CCN(C(C2CCC(C(N)=O)CC2)=O)C1 c1(C(=O)NCC2N(C(CS(=O)(=O)NC)=O)CCC2)cc(C2CC2)cnc1Cl c1(-c2nn(CC(C)(C)C)c(-c3cc(-c4ccco4)[nH]n3)n2)ccc(F)c(Cl)c1 C1(C2(O)CCOC2)(C(=O)OCC(C)CC2CCCCC2)CC1 C1(C)(NC(CCn2cc(C(CCC=C(C)C)(C)O)nn2)=O)CCCC1O N1(C(c2cc(Br)cc(F)c2F)C(=O)NC(C)C)CCOCC12COCCN(C)C2 c1(C(=O)OC)ccccc1CNC(C1CC1(OCC)CCCC)=O.COC C1(C2CN(C(C3(C)CCN(C)C3)=O)C2)(NC(C2C(C#C)C2)=O)CC1 C1(O)(CNC(c2c(C)nc(C)[nH]2)=O)CCN(C(=O)C=Cc2nc(C)c(C)[nH]2)CC1 C1(C2(NC(CCN(C)CCO)=O)CC2)CCCCN1C(c1cc(F)c[nH]1)=O C1(C(=O)NC(c2cn(C)nc2)C(=O)NCCN2CCC(C)(O)C2)OCCCC1(C)C N1(C(c2cc(C)cc(C)n2)=O)CC(NC(=O)C(C)(C)CO)CC12CCCOC2 Cc1ncc2ccc(C(=O)N(C(C)CCNC(C3OCC3(C)C)=O)C)cn12 C1(C(=O)OC)CCN(C(=O)NCC2(C)CC2(Cl)Cl)C1SC(C)(C)C CS(=O)(=O)C(C(=O)NCC#CCNC(C12CC(CN1C1CC1)C2)=O)C1CC1 c1(NC)nc(C)ccc1C(N1CCCC1CN(C(=O)C(=Cc1c[nH]cn1)F)C)=O C(=O)(CN=c1cc[nH]cc1)N(C)CC1CCCN1C(C1CCN2CCCC2C1)=O C1(C(=O)NC(C(=O)OCC)C)CCN(C(C2CC23CCC3)=O)C1(C)C N1(C(CCCOC)=O)CCC2(CCCC2NC(C2CC(C(C)(C)C)=NO2)=O)CC1 c1(C(C(=O)NCC2CCOC2)N(C)Cc2c(C)ccs2)cc(F)cc(I)c1 C(=O)(C(C)(C)CC(=O)N(CCNC(c1c(Cl)c(C)nn1C)=O)CC)OCC c1(CN(CCC(=O)NC2CCC(CC)C2)CCCO)cc2c([nH]1)CCCC2=O c1(C(=O)NC2CCCN(C(CCCNC(C)=O)=O)CC2)cncc2ncn(C)c12 N1(C(C=CC(CC)=CC)=O)CCN(C(c2cnc(N(C)C)cn2)=O)CC1CCC C1(NC(C(CC(C)C)O)=O)CC12CCN(C(=O)CC1(C)CCCCC1)CC2 C1(NC(C(CC=C)C)=O)CCCCC12CCCN(C(=O)CC1CCCC1(F)F)C2 N1(C(C(CC2CC2)OC)=O)CCCCC(C(=O)Nc2ccc[n+]([O-])c2)C1 c1(C(N2CCC(N(C(=O)C(C)O)CC)CC2)=O)ccc(F)c2ccsc12 CC(C)C#CC(=O)NC(C1(O)CCN(C(=O)CC2CCOC2=O)C1)C C1(CCNC(C(C)CN2CCOCC2)=O)CSCCN1C(c1coc(Br)n1)=O c1(OCC)ncc(C(=O)NCC2(F)CCCN(C(=O)CCC(C)CC)C2)cc1Cl C1(CC(=O)NCC2(C)CCCN2C(c2cc(O)cs2)=O)CC(O)C12CCC2 N1(C(C(COC(C)=O)C)=O)CCCC(C)(C(=O)NCCCCCN(C)C)C1 c1(C(=O)NC2CCCN(C(c3nccc(CC)c3)=O)C2)c(C)cc(C)cc1N c1(CC(C)C)ccccc1NC(=O)C(F)C1CCCC1 C1(CNC(C(C)=CC)=O)CCCN(C(c2c[nH]cc(Br)c2=N)=O)CC1 N1(C(CCCOCC)=O)CCC(O)C1C(N1CCC(N2CC(O)C2)C1)=O N1(C(CC(C)(C)NC(C(CC#C)C2CC2)=O)=O)CCC12CCN(C)C2 C(=O)(C(O)CCNC(c1nccnc1C)=O)N(C(CCCC)C)C C(=O)(CN1C(=O)COc2ccc(Cl)cc21)N(C)CC1CN(C(C)=O)CC12CC2 C(=O)(C1CCc2cc(F)ccc21)NC(CC)CNC(c1cc(C(F)F)on1)=O C1(CC)C(NC(=O)CCCCN(C)C)CCN1C(=O)CCC(=O)c1ccccn1 CC1CCN(CC(=O)N(C)CCN2CCN(C(=O)C(C)(C)C3CCC3)CC2)CC1 c1(C(N(CC(CC)NC(c2c(Cl)cnn2C(C)C)=O)C)=O)cccc(C(C)C)c1 N1(C(c2ccc(SC)o2)=O)CCC(C(N2CCC(CC3CCC3)C2)=O)C1C(C)C n1(CC)cc(Cl)c(C(=O)N(CC(CO)(CO)NC(C2CC2(F)F)=O)C)n1 c1(NC(C(C)Cn2cccn2)=O)cccc(CNC(C2COCC2(C)C)=O)c1 C1(C(=O)NCCCN(C(=O)CCc2nnc(C3CC3)o2)CCO)C2CC2C2CC12 c1(COC)ccc(C(=O)NCCCOCCNC(=O)C(C)N2CC(C)C2)cc1F CCN=C(NCc1cccc(N(C(=O)CNC)C)c1)NCC(C)(C)C(=O)OC O=C(CCC1=CCCCC1)NC1CCN(C(=O)Cc2ccnc(C(F)(F)F)c2)C1 c1(C(=O)NCC2N(C(c3c(COC)cco3)=O)CCC2C)c(C)cc(O)nc1C N1(C(C(n2cc(Br)cn2)C)=O)CCC2(CCC(NC(=O)CC3CC3)C2)CC1 Cc1ccc(C(=O)NCCC(O)CNC(=O)CC2(O)CCCCCC2)cc1N N1(Cc2n(CCC)ncn2)CCCC(CO)(NC(c2ccc(Cl)nc2OC)=O)C1 CCC(CC)CCC(=O)N(C)CC1CCCN1C(C1CC2(CCO1)CC2)=O C1(NC(c2cnc(Cl)s2)=O)CC2CN(C(=O)COCC3CC3)CCN2C1=O N1(C(c2ccc(OC)nc2Cl)=O)CCN(C(C2OCCCO2)=O)C(C)C1C N1(C(c2cscc2F)=O)CCC2CN(C(=O)CSc3ccc([N+](=O)[O-])cc3)C2C1 c1(C(=O)NCC23CCC(CC2)N3C(=O)C=Cc2nccs2)ccn2nncc2c1 c1(-c2cc(C)[nH]n2)ccc2c(C(N3CCNC(=O)CC3)CC3(C)OCCO3)c[nH]c2c1 c1(CC(=O)N2C3CCN(C3)C(=O)CC2C2CC2)ccc(F)c(F)c1.C=CCC1CC1 CC(CO)(CO)NC(C1(CCNC(C2CCOCC2)=O)CC1)=O C(=O)(C(C)CC(=O)OC)N1CCC(C2N(C(C3CC(CC)C3)=O)CCC2)CC1 C1(OC)CC(NC(=O)CCNC(C)=O)CN(C(=O)C(C)OC)C1 C1(C(N2CCC(NC(C(OC)OC)=O)CC2C)=O)CC2(C1)CC1(CC1)C2 c1(C(C)OCC)nc(CC(N2CC(O)(CNC(=O)Cc3n[nH]c(C)n3)C2)=O)cs1 C1(CC)CN(C(=O)CN(c2ccccc2)CC(C)C)CCN1C(=O)CNC(C)=O C(N=c1c(Br)c[nH]cc1[N+](=O)[O-])C1N(C(=O)Cc2cccc(F)c2)CCC1 C1(C(N2CCCC(CC(=O)NCc3c[nH]nc3C(F)F)C2)=O)CCCCC(=O)N1 c1(C(=O)NCC#CCNC(c2c(C)ccnc2C)=O)nccc2c1NCCC2 N1(C(CCCC(OC)OCC)=O)CC2CCCC2C1C(=O)NCCOCCNC c1(N(C(C2N(C(C)=O)CC2)=O)CC2(c3cccs3)CC2C)ncc(C(F)(F)F)s1 c1(C(N2CCCN(C(CCN(CCC)C)=O)C(C)C2)=O)ccc2cnc(C)n2c1 C1(C(=O)NCc2c(C(N(CCCOC)CCO)=O)occ2)CCCCC1C c1(CC(=O)NC2(CNC(c3cnn(CC4CC4)c3)=O)CC2)ccc(F)cc1F C=CC(C)(CCOC)C(=O)NCC1CCCCN1C(=O)Cc1cccnc1 C(=O)(C1=CCCCC1C)N1C(C)CCC(C(N(CC(CCC)C)C)=O)C1 c1(C(C)NC(c2cc(C)n(C)n2)c2nnnn2C2COC2)cc2ccccc2o1 Cc1nc(N2CCC(NC(C3CCCC3c3ccccc3)=O)C2)c(C)c(C)n1 c1(CC)cn2c(n1)CC(C(N1CC(CNC(C3(CC)CCNC3=O)=O)C1)=O)CC2 C(=O)(C1CCc2nccn21)NC(CNC(c1cc(CCC)[nH]n1)=O)CC(F)(F)F C1(CC)CN(C(=O)OC(C)(C)C)CC1C(N1CC(N(C)C)C(O)C1)=O c1(CC)cc(C(=O)NC(C)CCCCNC(=O)C=CC2CCOC2)ccc1C C1(F)(C(N2CC3C(NC(c4ccc(C)nc4C)=O)C3C2)=O)CCCCC1(F)F c1(COCC(=O)NCCC2CC(NC(C3(CC)CC3)=O)C2)nnc(S)n1C c1(C(=O)NC23CC(NC(c4ncncc4Br)=O)(C2)C3)cccn2nccc12 N1(C(CSC)=O)CC(NC(=O)CC(C)c2ccccc2)C(F)C1 c1(OC)c(C(=O)NCc2csc(CNC(C3CCCC3SC)=O)n2)cccc1F C1(CNC(c2cccc(SCCOC)c2)=O)CCN(CC2CCC2C)CC1 C(=O)(CCS(C)(=O)=O)NCC1CCN(C(C(C=C)O)=O)C1 C1(C(=O)NCCCC2CCCN2C(C2CCCO2)=O)CC(=O)N(C2CCCC2)C1 CC1CC(CCC=CC(=O)OC)CN1C(=O)C(F)=CC1CC1 C(C(C)(C)CS(=O)(=O)CC)NC(c1n(CCC)nnn1)(C)C1CC1 N1(C(Cc2n[nH]c(=N)o2)=O)CC(NS(C)(=O)=O)Cc2ccccc21 C(=O)(CC(C)(C)C(C)(F)F)NC(C1(O)CN(C(=O)Cn2cc(Br)cn2)C1)C Fc1cc(CN2CCOC(C3CC4CCC3C4)C2)c2c(c1)CCC2 CC(C)C1=NOC(C(N2CCCC2CN(C)C(c2conc2C2CC2)=O)=O)C1 c1(NC(CCCC=C)C)ncc(S(=O)(=O)N2CCCC2COC)cc1Cl CCC(C)CCCCC(=O)NCCC1CC(C(N2CC3(CCC(=O)O3)C2)=O)C1 c1(C(NOC(C(=O)NCC23CCC(OC)C2C3)CC(C)C)=O)cccc(C#N)c1C C1(F)(C(=O)NC2CC2NC(C2CCOC2)=O)CCCCC1 C(=O)(C1=CNC2=NCCC2=C1)N(C1CCN(C(=O)C(C)CCCOC)CC1)CC N1(C(C2C(OCC)C2C)=O)CCCCC1C1(NC(c2nccc(C)n2)=O)CC1 Cc1cc(C(=O)NC2CCCC2CC(=O)NC(C)C2CC2)cc(O)n1 c1(C(=O)Nc2nc(C(=O)OCC)c(CC)s2)ccc(O)c(CO)c1 N1(C(=O)C=C2CCCC2)CCC2(CC1)CN(C(C13COCC1C3)=O)C2 C1(n2c(N3CC=C(C)CC3)nnn2)CCCN(C2(c3cccc(Cl)c3)CC2)C1C CCC(O)C(C)(C)C(=O)N1CCCC(N(C(=O)Cc2cncc(C)c2)C)CC1 C(CCCC(CO)NC(=O)Cc1csc(C)c1)NC(C(C(C)C)OC)=O C#Cc1cnn(C)c1C(N1CC2CC1C2NC(C1CCN(C(N)=O)CC1)=O)=O O=C(C1=COc2ccccc2O1)NCCC1CCCN(C(=O)C(F)C2CCC2)C1 N1(C(C2CCCN(C(C=C(C)C)=O)C2)=O)CCOC(C2CC2)CC1 c1(C(=O)NC(C(=O)N(C)C)(C)C)coc(C2CCCN2C(=O)OC(C)(C)C)c1 c1(NC(C2CC23CN(C(c2cncc(F)c2)=O)C3)=O)nccc2cccnc12 Cc1cccc(C)c1CC(=O)NCC(C(C)C)NC(C1(CON)CC1(F)F)=O N1(C(c2cc(CC)nn2C)=O)CCN(C(=O)CCC=C(C)C)C2CS(=O)(=O)CC12 C1(C(=O)NC(CCC)C)CCCC12CCN(C(=O)Cc1cccn1C)C2 c1(C(=O)NCC2(C)N(C(c3c(C)sc(O)n3)=O)CCC2)cc2c[nH]nc2s1 N1(C(c2oc(CC)c(C)c2)=O)CC2(CNC(=O)C(C)=C(C)C)CC1CO2 c1(C(=O)NCC2CCCN2C(=O)COC2CCOC2)cc(O)nc2c1CCCC2 c1(N2CCC(NC(c3cnc(OC)nc3)=O)C(O)C2)ncnc2c1COC2 Cc1cc(C(N2CC(NC(=O)C3=CCSC3)CC23CCCC3)=O)cc2nc[nH]c12 C=C(C)C1CN(C(=O)CCN(C)C(C2CCC2COC)=O)CCO1 N1(C(c2cc(Cl)cs2)=O)CCCC(N(CCO)C(c2cc(CCO)on2)=O)C1 C12(C(N3CCN(CC(=O)N(C)CC4CCSC4)CC3)=O)CCN(CC1)CC2 c1(C(=O)NCC2OCCN(C(CN3C(C)CC3)=O)C2)ncc(F)cc1F c1(C(CNC(C(C)C23CC(C2)C3)=O)(F)F)nnc2ccccn12 C=CC1(CC(=O)N(CC(C)N(C)C(c2c(C)coc2C)=O)C)CCCCC1 CCCCCC(F)C(=O)N1CCN(C(C2(CC3CC3)CCC2)=O)CC(O)C1 c1(N(C(C(CC2CCCC2)NC(C(C2CC2)OC)=O)=O)C)cc(C)cc(C)c1 C(CNC(=O)CCCC1CCCCC1)(C(C)C(C)C)NC(C(C)(C)OC)=O C1(C(=O)NCC2N(C(c3n[nH]c(C)c3Cl)=O)C3C(C2)C3)CCC(C)(C)CC1 c1(NC(C2CCN(Cc3cnc(C)s3)CC2)=O)ccc2nccnc2c1 C1(CNC(c2nc(CC)sc2)=O)CC(NC(c2ccncc2)=O)C1(C)C C1(C(=O)NCCCN(C(=O)COc2ccccc2Cl)C)Cc2ccccc2S1 c1(OC)cc(Br)c(O)cc1C.c1(C(C2CC2)=O)ccc(C2CCC2)cn1 CC(O)C(C)C(=O)N(C)CCOCCCN(C(=O)C(C)(C)c1ccns1)C C1(NC(c2n(CC(C)C)ncc2)=O)CC(C)N(C(=O)COc2ccccc2Cl)C1 C1(C(N2C(CN(C(=O)CC(C)(C)CC)CC)CCC2)=O)CC(C(C)C)=NO1 C=CCCCCCC(=O)NC(CNC(=O)CC1C=CS(=O)(=O)C1)C1CCC1 C1(CNC(C(CC)OC)=O)(CO)CCCN(C(=O)CCC2(C)CC2)C1 N1(C(C(C)N(C)C)=O)CC2CCC(C1)C(NC(=O)Cc1cc(Br)cs1)C2 N1(C(C(C)C(C)O)=O)CC2(CCN(C(C3SCCS3)=O)CC2)CC1C C1(NC(CN(C(C)=O)C)=O)CC2CN(C(=O)CC3C=CCCC3)CC12 N(C1CC2(CN(C(=O)Cc3cccnc3)C2)n2ccnc21)C(CCC(C)(C)F)=O CC1=C(C(=O)NC2CC2NC(=O)C=Cc2cscn2)Cn2nnnc2N1C N1(C(c2ncc(C)nc2)=O)CC2CC1CN2C(C1CCC1Cc1ccccc1)=O C12CCCCN1N(C)CCC2.c1(C=O)ncc[nH]c1=O.C1(C=O)(N(C)C)CC1 C1(C(N(CC(C)NC(=O)CC2(C#N)CCC2)CC)=O)CC(C(C)C)=NO1 c1(NC(CNC(=O)CCN(CCCN(CCNC(N)=O)C)C)=O)ccc(F)cn1 c1(OCCC)ccc(C)cc1-c1cnc(NC(=O)Cc2ccc(Br)cn2)c(C)c1 c1(C(=O)OCC2CCC(F)(F)C2)ccc2c(n1)OCCO2 c1(NC(N(C2CCC(C)(C)CC2)CCC)=O)nc2ccc(OC)cc2s1 C1(CCC(=O)N(C)CCn2cncn2)CCCN1C(=O)CCc1cscn1 CCC(C)(CC)C(=O)NCC1CCCC(CNC(c2ncc(OC)cn2)=O)C1 C1(C(=O)NC2C(NC(C3C(OCC)CC3)=O)COC2)CN2CCN1C(C)C2 S1(=O)(=O)c2ccc(C#N)c(c2)NCCCN1.c1(OC)cccc(NC2CC2)n1 C(=O)(C(C)CC(F)(F)F)NCC1(O)CCN(C(COC2(C#C)COC2)=O)C1 CCCC(CC)C(=O)N1CCN(C(=O)CCN2CCSC(C)(C)C2)CC1C(C)C C1(CCC)CN(C(c2ccc(CC)c(Cl)c2)=O)CCN1C(=O)CCn1cccn1 Cc1ccc(S(=O)(=O)N2CC=CC2C(=O)Nc2cncnc2I)cc1C C1(C(N2CC(OCC#C)C2)=O)CC(C)CN(C(=O)C(C(C)C)NC(C)=O)C1 Cc1nc(N2CCC(C(C)(C)C#N)CC2)cc(-c2ccc(F)cc2)n1 C(CN=c1nn[nH]n1C)C1CCN(C(c2c(C)snc2)=O)C1 C1(CCNC(Cc2cc(C)no2)=O)COCCN1C(=O)C(O)CN1CCOCC1 C1(NC(C(C2CCOCC2)C)=O)CCN(C(c2ccnc(Cl)c2N)=O)C1(C)C N1(C(CC2(CNC(c3cc(COC)[nH]n3)=O)CC2)=O)CCC2CCNC(=O)C12 CC1CCN(C(C2CSC2)=O)C(C(=O)NCC(F)(F)Cl)C1 c1(CCC(=O)NC2CCCC2NC(C2CCCC2O)=O)cnc2n1CCCC2 C(=O)(C(C)CCC(C)(C)C)N1CCC(COC)(NC(=O)C(CO)C(C)(C)C)CC1 N1(C(=O)NCc2ccc(C#N)s2)CCN2C3CCC(C3)C2C1 N1(C(C(CCOC)NC(Cc2c(CC)con2)=O)=O)CCC(F)(CF)CC1 C(=O)(CCCCCCCCC1CC1)N1C(C)(CNC(=O)CC(O)C2CC2)CCC1 CC1(C)CCC(C(=O)NC2CCC(C#N)CC2)CN1C(C1(C)COCCO1)=O N1(C(C23C(C)OC(CC2)C3)=O)CCC2(CC1)CCN(C(C1CC1(F)F)=O)CC2 C1(CNC(c2cccc(C)c2Br)=O)CC2(CO1)CN(C(C1CCCC1)=O)C2 C1(CN(C(=O)COCCSC)C)CC(F)CN1C(C1CCC1c1ccccc1)=O C1(C(=O)NC2(CF)CCC2)(NC(C(COC(C)=O)C)=O)CCN(C)C1 c1(C(c2nnnn2C(C)C)NC(C(C(C)C)SC)=O)cn(C)c2cccc(C)c12 c1(C(C(=O)N(CC(CC)NC(c2sccc2SC)=O)C)O)cncn1C C#Cc1cn(C)nc1C(=O)NCCCCN(C)C(C1CCC(OC)C1)=O C1(C)(CNC(C2CC(OCC)C2)=O)CCCN(C(C2(C)CCC3CC3C2)=O)C1 C1(NC(=O)NCC(C(F)(F)F)c2ccccc2)CCCS(=O)(=O)C1 c1(C(C)OC(c2ccsc2Cl)=O)ccc(Nc2ccccc2)cc1 C1(CCNC(c2c(C(C)C)c[nH]n2)=O)CCN(C(=O)C(F)CC2CC2)CC1 C1(NC(C=C(C)c2ccco2)=O)COCCN(C(=O)C=Cc2cncn2C)C1 N#CCS(=O)(=O)c1ccc(C(N2CCN(C(c3nc(Cl)cs3)=O)CC2)=O)cc1 Cc1ncccc1-c1cn(C2CN(C(c3ccccc3CC(C)(C)C)=O)C2)nn1 CC(O)C(C)(C)C(=O)N1CC(C(N)=O)(CNC(c2cc(C(F)(F)F)cc(O)n2)=O)C1 C1(NC(c2c(C)cns2)=O)CCN(C(=O)CC(O)C2CC2)CC1F C1(N(C(=O)C2=CCOC2)C)CCCCN(C(C2CC2c2ccccc2)=O)C1 c1(C(=O)NCC(C)CNC(=O)CCCCC(F)F)cc(P(C)(C)=O)ccn1 CC(C)C(F)(CNC(=O)CCC(C)N(C)C)C(=O)NCCn1cnccc1=O c1(C(=O)NC2CC3CC(NC(c4ccc(CC)[nH]4)=O)C3C2)c2c(nn1C)CCC2 O=C1Nc2ccc(-c3nnc(CN(C4CC4)CC4CC4)o3)cc2C12CC2 N1(C(c2[nH]cc(C(N)=O)c2)=O)CC2CC(NC(=O)Cc3cnns3)C(C2)C1 C(=O)(CC(C)CC(C)(C)C)N1C(NCc2ccc(CCCC)cc2)COCC1 C1(C)(C(N(CC(C)N(C(c2c(CC)c[nH]c2)=O)C)C)=O)CCCCNC1=O c1(C(=O)NCCC(=C)CNC(C2CCCCN2C)=O)cncc(N)n1 c1(C(=O)OCCCN2C(=O)CNC2=O)nn(-c2ccccc2F)c2c1CCC2 C(=O)(CC(O)CC(C)(C)C)N1CC(CC)C(C(=O)NC(CO)CCO)C1 C1(NC(C(C)CO)=O)CC2C1CCN2C(c1cn(C(C)(C)C)nn1)=O C(=O)(C(O)C(C)(C)C)NCC1(C(C)(C)O)CN(C(=O)CC23CC(C2)C3)C1 C1(C(=O)NCC2CCCN2C(c2ccnnc2)=O)CCC2(CCOCC2)O1 C(C1C(C)C1(Cl)Cl)=CC(=O)NCC(CNC(c1ccc(CN(C)C)o1)=O)OC C1(NC(CCN(C(COCCCCC)=O)C)=O)C(=O)OCC1(C)C C=C(Cl)C(C)(C)C(=O)N1C2CCC1C(CNC(=O)CNc1ccccc1Cl)C2 CCCC(CC)C(=O)N1CCC(N(CCC)C(c2c(C)cnnc2O)=O)C1 c1(CNC(C2CCN(Cc3ccc(Cl)s3)CC2)=O)cccc(Cl)c1F C1(CNC(C2(C)CCN(C(c3nn(CC)nc3C)=O)C2)=O)CC(=O)N(C)C1=O C1(CC)CCC1(c1nnnn1C1CCOCC1)NCc1ccsc1Cl N#Cc1cc(F)c(NC(=O)CC2CCCN2C(=O)CCN2CCCC2)cc1Cl c1(C(=O)NC2C(CNC(C(C)C)=O)CCC2)cc2scc(Br)c2[nH]1 C(=O)(CC1=NN(C)C(=O)C1)N1C(CNC(C2C(OCC)C2)=O)COC(C)(C)C1 N1(C(C(CCC)N(C)C)=O)CCCC12CCN(C(c1cc(C3(C)CC3)on1)=O)C2 N1(CC(=O)OC)CC(C(=O)N(CC(C)CNC(C2CN(C(C)=O)C2)=O)C)CC1=O c1(C(=O)NCCOC(CNC(C(CC)N(C)C)=O)(C)C)ncccc1F Cc1cc(C(N2CCC(c3ccnn3C)C2)C(=O)NCCC2(C)CC2)sc1Cl C=CCC(C(=O)NCCN(C(=O)C(C)n1cncn1)C1CC1)C(C)C N1(c2cc(C(=O)OC)ncn2)CCCC(NC(=O)Cc2cc(C)no2)C1C C(C(=O)N1CCC(C(C)NC(C2(c3ccccc3F)CCC2)=O)C1)(C(C)C)OC C1(CNC(C2(COC)COC2)=O)CN(C(=O)C=CCCC(C)C)CC1C N1(C(c2c(C)cc(C)o2)=O)CCC2CCC(C1)N2C(c1cc(C2CC2)nnc1O)=O C1(NC(=O)Cc2cncnc2)CCCCC1C(N1CC(C(=O)N(C)C)C1)=O CC1(CO)CCCN(C(C2(F)CN(C(=O)CC3CC3)C2)=O)C1 C1(CNC(CC2OCC(C)(C)C2)=O)CCN(C(c2cnnn2C2CC2)=O)C1(C)C N1(C(C(C)S(N)(=O)=O)=O)CCC2(CCN(C(C3(O)CCSCC3)=O)C2)C1 C(c1cn(C)cn1)=CC(=O)NC(CC)CN(C(=O)C(C)NC(C)=O)C c1(C(N2CCC(NC(c3scc(OC)c3)=O)C2C)=O)cn(C)c(=O)cc1C N1(CC(=C)Br)CCC(N(C)C(c2ccc(Cn3cc(Cl)cn3)s2)=O)CC1 c1(CNCC2N(C(C#CC(C)C)=O)CCC2C)oc2ccccc2c1CO C(c1cccnc1)=CC(=O)NCCC1CC(NC(C2CN(c3nncs3)C2)=O)C1 Nc1nc(Br)ccc1C(=O)NC1CC(F)CN(C(=O)Cn2ncnn2)C1 C1(NC(c2c(Cl)ncc(C)c2)=O)CCN(C(c2c[nH]c(=N)o2)=O)C12CCCC2 c1(N2CC(CNC(CN(C)CC)=O)N(C)CC2)ncnc2c1CCC2 Cc1cccc(C(O)C(=O)NC2CCCCN(C(c3cc(N)ccn3)=O)C2)c1F c1(NC(C)C)nccc(=NC(C)c2nccc(=N)[nH]2)[nH]1.C12CCCN(C1)C2 C1(CNC(C2CC(N(C)C)C2)=O)CCC12CN(C(=O)Cc1ccc(F)c(F)c1)C2 c1(N(CC(=O)NC(CC)CNC(c2cnn[nH]2)=O)CC)ccc(C(F)(F)F)cc1 N1(C(C2C(CC)C2)=O)CCN(C(c2cc(C)ccc2Br)=O)CC1C(C)C CCCCC(C)C(=O)N1CCN(C2CN(C(c3cc(OC)nc(C)c3)=O)C2)CC1 C1(CNC(C2(OC)CCSC2)=O)CN(C(C2(CC(C)C)COC2)=O)CC(C)(C)C1 c1(C(=O)NC2(CNC(c3cc4sccc4s3)=O)CC2)cc2ccccc2[nH]1 N1(C(c2cn(C3CC3)nn2)=O)CCNC(=O)C1.c12n[nH]cc1CC1N(CC1)C2=O CC1CCN(C(=O)COC2CC2)C1CNC(=O)Cc1csc(C2CCCCC2)n1 C1(NC2CC(c3ccccc3)(NC(C3C(C)CC=CC3)=O)C2)CCCC(=O)N1C C12(C(=O)NC(c3ccc(OCC)cc3)C)CCC(CC1)N2Cc1ccccc1 C1(C(C)C(=O)NCCCc2cncnc2)CCN(C(C23CSCC2C3)=O)CC1 C(=O)(CS(C)(=O)=O)NC(CC=C)CNC(=O)CCc1csc(C)n1 C1(CN(C(C)C)C)CCN(C(C2CCCC(C3CC3)O2)=O)CC1 c1(C(c2nc(-c3ccco3)nn2Cc2ccc(C)cc2)CC)ccc(F)cc1 C1(NC(C(C)NC(c2ccc(C3CC3)cc2)=O)=O)CCCC(C)(C)CC1 CCCC(C(=O)N(CC)Cc1cccs1)NC(=O)Cc1ccccc1O C(C1Cc2ccccc21)NC(C1C(C)(C)C1C(=O)O)=O CCCCC(O)CCC(=O)N1CC(NC(c2cc(Cl)ncc2N)=O)C(C)(C)C1 C1(O)(C(N2CC(CNC(c3cc(CC)on3)=O)OCC2)=O)CCC(C)CC1 C(=O)(C1=C(C)CCCC1(C)C)N1CC(F)CC(NC(CC2CC(OCC)C2)=O)C1 N1(C(C(CC)NC(N)=O)=O)CCCC(C)(C(N2CCC(O)C(C)C2)=O)C1 C1(C2CCOCC2)(CNC(CCCOC)=O)CCN(C(C2CCN(C)C2C)=O)C1 C1(CNC(CC=CC=C)=O)CC(F)CN1C(=O)COc1ccc(C(F)(F)F)nc1 c1(C(=O)NCC(CC=C)NC(=O)C2=C(C)OCCS2)n[nH]c2c1CCOC2 c1(C(N2CCC(NC(=O)CCOc3ccc(F)cc3)C2)=O)ncc2n1CCCC2 C(=O)(C(O)C(C)(C)CC)NC1CC(NC(c2cncc(C(=O)OC)c2)=O)C1 c1(-n2cc(CCC(C)(C)O)nn2)ccc(-n2cc(Br)cn2)cc1 CC(C)(C)CC(O)CNC(C1(CCNC(=O)CCc2cccnc2)CC1)=O Cn1[nH]nnc1=NCC1CCCC1NC(C1CN2CCN1CC2)=O c1(CC)cc(C(N2CCN(CC(=O)N(C)C)CC2)C(=O)NC2CC2)cc(F)c1 N1(CCNC2CCCC(C#C)C2)CCN(C(=O)OC(C)(C)C)CC12CCC2 C1(NC(C(C)Cc2cnc[nH]2)=O)CN(C(=O)Cc2cccc(Cl)c2Cl)CCC1C c1(CNC(c2ccc(NCc3cc[nH]n3)nc2)=O)cccc(F)c1 N1(C(C2CC2CC)=O)CCOC2(C1)CN(C(=O)Cc1ccccc1C1CC1)C2 Cc1cc(F)c(F)cc1NC(C1CCCN1C(=O)Nc1ccc(Cl)cc1C)=O O=C(C1=CC2CCC=CCCC12)NCC1CC(NC(C2(CO)COC2)=O)C1 C1(N(C(CCOC(C)=O)=O)C)CCCC(NC(=O)Cc2cccc(Cl)c2)C1 C12(NC(c3c(CC)occ3)=O)CC3CCC(C1C2)N3C(c1nocc1C1CC1)=O c1(OC)cccc(C(=O)NCC(=O)NCC#CCNC(=O)C=CC(C)(C)C)c1 N1(C(CCCCOC)=O)CCCC12CCC(NC(=O)C(C)Cn1ccnc1)CC2 C1(C(=O)NC(Cc2cc(C)no2)C)CCCC12CN(C(c1cc(C)n(C)n1)=O)C2 c1(C(N2C(CNC(c3cc(Cl)ccn3)=O)CCCC2)=O)occ2c1CCCC2 N1(C(CCOCC(C)C)=O)CCN(C(=O)CCP(C)(C)=O)C(C)C1 C1(CC)CN(C(=O)C(O)C(C)C)CCC1CNC(=O)CCCC1CCC1 CC1Oc2ccc(C(N3CC4C(CNC(=O)CC(C)N(C)C)C4C3)=O)cc2C1C c1(C(N(C2CN(C(C(C)C#N)=O)CC23CC3)C)=O)n[nH]c2ccccc12 C1(CC(=O)OC)CCN(S(=O)(=NC(=O)C(C)Sc2ccccc2)N(C)C)CC1 c1(NCCC2CCCC(C)C2)ccc(S(=O)(=O)N2CCC(C)(C)CC2)cc1Cl N1(Cc2cnc(C)o2)CCC2(CCCN(C(C3CCCCCC3)=O)C2)C1 c1(C(=O)NC(CNC(C(CC)n2cncn2)=O)C(C)C)nc(C(F)(F)F)oc1C c1(OCC)ccc2cc(C(N3CCC(C(=O)O)C(O)C3)=O)[nH]c2c1 N1(C(C)=O)CCOCC1C(=O)NCCCCN(C(=O)CCc1cccc(O)n1)C C#CC1(NC(=O)CC(C(C)(C)C)NC(=O)C(C)CO)CCCCCC1 C1(NC(c2c(Cl)nc(N(C)C)s2)=O)CC2CCC1N2C(=O)CC1CCC(=O)N1C c1(C(N(C(CNC(c2n[nH]c(C)c2O)=O)C2CC2)C)=O)cc2ccc(Cl)nc2s1 c1(N(CC(CCC)C)C)nc(N2CCC(F)(F)C(C)C2)c2ncsc2n1 O=C(CCCCC(F)(F)F)NCCCCCCNC(C1CCC2(CCC2)C1)=O N1(C(C2CN(C(C)=O)C2)=O)CCC(C)N(C(=O)COCCOc2cc(C)on2)CC1 CC(C)C(CN=c1nc(NCC(C)C#N)c2c([nH]1)CSC2)OCCO C=C=CCCC(=O)N1CCCC1C(C)(C)NC(=O)C(O)Cc1ccc(F)cc1 C1(O)(C(=O)NC2CCCC(NC(=O)CC3(CO)CC3)CC2)CN2CCC1CC2 c1(CCC(=O)NCCC(C)NC(=O)C(O)CN2CCCC2)cc(Cl)cs1 Cn1cnc(C(=O)NCC(C)=CC(N2CC(C(C)(C)C#N)C2)=O)c1 N1(C(c2n(C)c(C#N)cc2)=O)CC2OCCN(C(=O)C=C(Cl)Cl)C2C1 C1(C(N2CC(NC(C(C)N(C)Cc3ccccc3)=O)C2)=O)CCN(C)C1=O CCCCCCC(=O)NCCc1cc(C(=O)NCC2CCC(C)N2C)no1 O=C(N=c1[nH]oc2c(Br)cccc12)C1CCCC1C1CCNCC1 Cc1nccc2c([N+](=O)[O-])ccc(N3CCN(c4ncc(C(=O)O)s4)CC3)c12 N1(C(C(CC)NC(C)=O)=O)CCOC2CN(C(c3ccnnc3C)=O)CC12 Cc1ccc(F)c(CNC(=O)C(c2cn(C)nn2)NC(C2CC(F)(F)C2)=O)c1 c1(CC)ccc(C(=O)N(C)CCN(C)C(C2(c3ccccc3)CC2)=O)s1 N1(C(C(C)(C)C2CC2)=O)Cc2ccccc2OC2(C1)CN(C(=O)CC1CCC1)C2 CC(C)(CCCC(=O)NCCC1(C)CC1)NC(C1CC(C2CC2)=NO1)=O c1(C(=O)NCC2CCC(NC(c3cn(CC(N)=O)nn3)=O)C2)ccc(O)nn1 c1(C(=O)NC2CC(CCNC(c3cc(O)nc(Cl)c3)=O)C2)cncc2sccc12 Cc1nn(C)c(Cl)c1CC(N1CC(NC(c2cnnc(O)c2)=O)CC1C)=O N1(C(C2(C)C(C)(C)C2)=O)CC2CN(C(c3cc(O)c(F)cc3N)=O)CC2C1 O=C(CCS(=O)(=O)c1cccc(Br)c1)N1CCCCC(O)CC1 c1(C(N2C(C)CC(NC(C3CCS3(=O)=O)=O)CC2)=O)ccc2c(O)nncc2c1 C(C(C)(C)CNC(C1C2COCC12)=O)NC(CCNC(C1C(C)C1)=O)=O N1(C(c2c(C)[nH]cc2)=O)CCC(O)(C(C)CNC(c2ccnc(C(N)=O)c2)=O)C1 c1(C(c2n(CCCSC)nnn2)NCc2csc(C)n2)cc(C(C)C)ccc1F c1(C(=O)NCC2(CNC(CC3OCC(C)(C)C3)=O)CCC2)cccc2cncn12 C1(CC(=O)OC)C(=O)NCCN1C(=O)C(N1CCN(c2cnccn2)CC1)C CCC(O)C(C)C(=O)NCCN(C(c1nc(F)ccc1Cl)=O)Cc1cccc(Cl)c1 Cc1cc([N+](=O)[O-])ccc1C(=O)NC1CC1C(=O)Nc1c(F)cc(Br)cc1Cl N1(C(CCN(C(C)=O)C)=O)CCC(N(C)C(c2cc(-c3ccco3)cs2)=O)C1 N1(C(c2ccc(COC)s2)=O)CC2(C1)SCCC2NC(c1csc(C)c1)=O c1(OCC(=O)NC2(C(F)F)CC(NC(C=C(COC)C)=O)C2)cccc(C)c1 N1(C(c2c(C)ccc(Cl)c2)=O)Cc2ccc(C(=O)Nc3cnn(C)c3)cc2C1 C(=O)(C(C)(COC)OC)NC1(CO)CN(C(c2ccc(COC)o2)=O)C1 O=C1C(NC(c2nnnn2CCCF)c2cnsc2)CCN1O N1(C(c2cc(Br)n[nH]2)=O)CCN(C(c2cnccc2Cl)=O)C2CCC12 Cc1ccc(C(N2CCN(C(=O)Cc3cc(Cl)sc3Cl)C(C)C2)=O)c(C(C)C)n1 c1(C(=O)NC(C(C)C)CO)nc(NC(c2ccc(OCF)cc2)=O)cn1C CCC#CCCNC(=O)CCSCC.C1(=O)N(C)O1 c1(Oc2c(CNC(C3C(N(C)C)CC3)=O)cccc2)ccc(F)cc1F N1(C(C(n2cc(C(C)(C)F)nn2)C)=O)CCOCC2(CCC2)C1 CC(CCC(C)(C)C)C(=O)NCC1(CC(=O)N(C2CC2)Cc2ccco2)CC1 S(=O)(=O)(c1ccc(N(C)CC2CCCO2)nc1)NC1C2(CC(OCC)C2)C1 C1(NC(C(n2ncc(C)c2)C)=O)CCC(NC(C2CC2CF)=O)CC1 O=C(C1=CC2CC=CCC12)NCC1=CCN(c2nccc(-n3ccnc3)n2)CC1 c1(C(C)C(=O)NCC#CCNC(=O)CN(C)C(=O)C2CC2)ccc(Br)cc1 C(=O)(C1CCCn2ccnc21)NC1(CNC(C2(C)CC(F)(F)C2)=O)CCC1 C1(CCNC(C=CC=CC)=O)CSCCN1C(c1ccc(O)nn1)=O Cc1nc(N(C)C(=O)NCC2CCN(C(C)C)C2)sc1C N1(C(C2=CC(C)(CC)C2)=O)CCN(C(c2c(O)cccc2F)=O)C2(CCC2)C1 Cn1cncc1C=CC(N1CCCC(CCC(=O)NCC2=CCCC2)C1)=O C(CCC)(CC(=O)N1CCN(C)C(=O)C1)NC(C(CC=C)OC)=O N(C1CS(=O)(=O)Cc2ccccc21)C(C1(C)CNC(=O)C1)=O C=C1CCN(C(=O)C(C(C)C)OC)C(C(N2CCCOCC2C)=O)C1 Cc1noc(C)c1CC(C)C(=O)N(C)CCN(C(=O)COC1CCOCC1)C CCC(O)C(C)(C)C(=O)N1CCC(C=CC(=O)NC2CCOCC2(C)C)CC1 Cc1c(C(N2CC(CNC(C3CCC4(CCC4)C3)=O)C2)=O)[nH]c2ccccc12 N1(CC(=O)OCC)CCC2NC(=O)OCC2C1 CCC(C)(CNC(c1c(CNC(=O)C(O)C(C)(C)C)cnn1C)=O)C(N)=O N1(C(CCC(=O)OC)=O)CCN(C(c2nc(C)n(C)c2C)=O)C(C)C1C n1(CC)c(CNC(=O)CCC2CCC(NC(=O)C=Cc3ccco3)C2)nnc1O C1(CN(C(COCc2nnc(C)s2)=O)C)CCC(NC(=O)C(C)(C)CO)CC1 N1(C(C(C)CNC(c2cc([N+](=O)[O-])n[nH]2)=O)=O)CCC(C2=NOCC2)C1 C(C(CO)C(C)CC)NC(C1(NC(CCC#C)=O)CCOCC1)=O N1(c2cccc(CC#N)n2)CCC(F)(F)C(C(F)(F)F)C1 C(=O)(C1CCc2ccccc21)NCCC(CC)(CC)NC(c1ccncc1F)=O N1(C(C(C)C(C)NC(=O)C(C2CCCCC2)C)=O)CCOC2CCC12 C1(C)(C(N2CCC(N(C)C(c3c[nH]c(=N)o3)=O)CC2)=O)CCCCNC1=O CC1(C)COCCC1C(=O)NC1(CNC(=O)CC2CCSCC2)CCCC1 c1(C(=O)NCC(C)NC(c2cn(C(C)(C)C)cn2)=O)ccc(O)cc1[N+](=O)[O-] Cc1cc(C#N)ccc1C(=O)NCC1(CNC(=O)C(C)(C)CC(F)F)CC1 c1(C(N(CCN(C(CN(C)CCO)=O)C)C)=O)cc(C(F)F)cc(F)c1 c1(C(=O)NCCCN(C(c2cc3scc(C)c3[nH]2)=O)C)coc2c1C(=O)NCC2 C1(NC(C(C)=C(C)C)=O)CCC(NC(c2ccsn2)=O)CC1 N1(C(C(C)OC)=O)CCC(CCC2CCCN(C(c3cn(CC)cn3)=O)C2)CC1 n1(C(C)(C)C)cc(NC(=O)C(=O)NC2(C)CC2c2ccccc2)nn1 c1(NCC2CCCN(CC(F)(F)F)C2)c(Cl)ccnc1Br Cc1ccc2c(=NC3CCC(C)C3)[nH]c(=NCc3ccn(C(C)C)n3)[nH]c2c1 C1(C)(CNC(C(CC)C2CCC(=O)N2)=O)CCCN1C(C1CC(F)(CF)C1)=O N1(C(C(CC)=CCCC)=O)CCN(C(=O)C(N2CCOCC2=O)C)CC1CF C1(C2CC2)(NC(CC2(C=C)CC2)=O)CCN(C(=O)C(C)OCc2ccccc2)C1 C1(CNC(CCCC(C)O)=O)C(C2CC2)CCN1C(=O)CCc1ccncc1 O=[N+]([O-])c1ccc(Cl)cc1CNc1ccc(-c2cnc[nH]2)cc1 Cc1ccc(Br)c(C2CCCN2C(=O)Nc2cnc(Cl)c(N(C)C)c2)c1 c1(C(N2CCCSC2)=O)c(F)c(F)c(F)c(F)c1F Cc1ccc(C(=O)NCC2(O)CN(C(c3sccc3Br)=O)C2)c(C)c1Br CC1(C)C2CCC1(C)C2C(=O)NCCC1CCC(NC(c2ccncc2N)=O)C1 Cc1cc(C(=O)NC2CC(NC(=O)C(O)C3CC3)CC2O)nn1C(C)C O=C1CN(CC(=O)NCC23COC(CNS(=O)(=O)CC4CCCO4)(C2)C3)CCN1 C1(C(=O)NC(C)C(=O)NCC2(Cl)CCC2)CCCN1C1CC1 N1(C(C2(CC#C)CCCO2)=O)CCC(NC(C2CCN2C(C)(C)C)=O)C(C)C1 C(=O)(CCC(CF)CF)N1C(C)(C(=O)NOCCCN(C)C)CCC1 C12(CCCCCC1)C(=O)N2.C1(C(=O)NCC2C(COC(C)C)C2)CCC2(CCC2)O1 c1(OCC(=O)NCC(=O)SCCCC)ccccc1.C1(CO)CNC(=O)CN1 c1(NC(C2CC(O)C2)=O)ccccc1.c12cc(n[nH]1)C(=O)NC(=O)CCS2 CCC(CC(=O)N1CCN(C(=O)C2=NOC3(CCC3)C2)CC1CCO)CC(C)C C1(OC)CN(CCCNc2cc(C(F)(F)F)cc(N)c2)CCC1C C1(C(N2CCCCC(CO)C2)=O)CN(C(c2csc(Cl)c2)=O)CC12CCC2 N1(C(CCc2ccc(C)o2)=O)CCC(C)C(CC(=O)NC(C)(C)C(=O)N(C)C)C1 O=C(C1CCc2nccn21)NC1CCN(CCNC(=O)CCc2ccccn2)C1 C#CCCCCC(=O)N1CCN(C(c2cc(OC)ns2)=O)C(CO)C1 C#CCC(C)(C(=O)N1CC(O)(CCO)C1)NC(=O)CCC1(C)CC1 C(C)(C(=O)N(CCCOCCN(C(=O)C(=O)NCC(F)(F)F)C)C)OC C1(F)(CNC(c2c(C)onc2)=O)CCC(NC(C2CCC(C)(C)C2)=O)C1 c1(C(N2CC(CC=C)(NC(=O)C(C)S(C)(=O)=O)C2)=O)cnc2c(c1)CCOC2 C1(CC)(NC(c2cc(C3CC3)nn2C)=O)CCCN(C(=O)CC2CC2)C1 c1(C(=O)OC)cc(OC)cc(CN2CC(C(=O)O)C(C)C2)c1 c1(N(C)Cc2n(CC)ccn2)nc(N2CC(CO)OC(C)C2)c2c(n1)COC2 c1(C(N(C(CNC(CC(CC)c2ccccc2)=O)C)C)=O)cn2nc(C)sc2n1 C1(C(=O)Nc2c(CC)ccnc2)CCCCN(C(=O)CN2CCCCC2)C1 CN1CCN(C)C(C(=O)NCC2CCC(NC(=O)CC3CC34CC4)CC2)C1 Cc1nc(CNC2CCCC2(C)c2ccc(C(F)(F)F)cc2)sc1Br Cn1cc(CNC2CC3(C2)CC(NC(=O)C2=COCCC2)C3)c2cccnc12 N1(C(C(CC)SC)=O)CCn2nc(CNC(c3nc(O)sc3C)=O)cc2C1 CC(c1ccccc1C)=CC(=O)N(C1CCC(NC(=O)C(O)CC(C)C)CC1)C N1(C(CS(=O)(=O)NCC)=O)CC(NC(=O)Cn2cc(C)cn2)CC12CCOCC2 c1(C(=O)Nc2scc(-c3cn(C(C)(C)C)nc3)n2)ccc(Br)c(Cl)c1 C12(C(N3C(C(N4CCCOCC4)=O)CC4CC43)=O)CC3CC(C1)CC(O)(C3)C2 C1(N(C(CCN(C)CCNCC2CC2)=O)C)C=CCCCC1 N1(CCC(N2CCN(Cc3cccc(C)c3C)CC2)=O)Cc2ccccc2C1 N1(c2cc(CC)ncn2)CCC2(CCCN(C(=O)COC(C)(C)CC)C2)C1 c1(C(C(=O)NC2CCOC2)N(CCC=C)CC)cccc(-c2ccncc2)c1 c1(C(=O)N)cccc(F)c1C(F)F.CC(C)(C)CC(=O)C(C1(CN)CC1)=O C(C(O)CC(=O)NC1(CC#C)CCCC1)NC(C1(CO)CCCC1)=O C1(NC(Cc2c(C)cnn2C)=O)CC2CC1N(C(=O)CCSc1ccccn1)C2 C=CC1(C(N2C(C(=O)NOCC(C)CC)CCC23CC3)=O)CCCCC1 C(=O)(CCC(CC)CCC)NC(CC#C)(C)C(=O)N(CC(=O)NC(C)(C)C)C c1(CS(=O)(=O)NCC(=O)NC(c2cccnc2)C2CC2)ccc(Cl)cc1[N+](=O)[O-] c1(OC)cnc(F)cc1C(N1CCC(CNC(c2cn(C3CC3)nn2)=O)C1)=O C1(C(N(CCCC(=O)NCC2(F)C(C)(C)C2(C)C)C)=O)CCCCC1(C)C c1(C(=O)NCCN(C(c2c(CC)nnc(C)c2)=O)C(C)C)ccc(C#N)cc1O CCS(=O)(=O)c1cccnc1C(=O)NCC1CC(NC(C2C3CCC2CC3)=O)C1 N1(C(COCCOCC)=O)CCN(C(=O)Cc2cc(Cl)cs2)CC2CCCCC12 c1(C(N2C(CN(C)C)CC(O)C2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 C1(C(N(C2CN(C(c3cc(C(C)C)n(C)n3)=O)C2)C)=O)CC(C)OC(C)C1 c1(OC)ccc(F)c(C(N2CCNC(C(=O)NCc3cnccc3OC)C2)=O)c1 Cc1c(NC(C2COCCN2C(c2cc(O)ccc2F)=O)=O)cccc1Br O=C(CC(Cl)Cl)NCCCC1(CNC(C2CC(CN(C)C)C2)=O)CCCC1 N1(C(Cc2n(C)ccn2)=O)CCC(C)(CC(=O)Nc2ccc(Cl)cc2)C1 c1(C(N2CCC(N(C(=O)C(O)C3CC3)CC)C2)=O)ccn2cc(C(=O)O)nc2c1 Cc1n[nH]c(C)c1CC(=O)NCCN1CCN(C(=O)CC2CCCS2(=O)=O)CC1 C1(OCCCC(=O)NCC(CNC(C2CC(CC)C2)=O)(C)C)CCC(C)CC1 FC1(F)CC(N2CCC(Nc3nccnc3I)CC2)CC1 C1(NC(C(C2CC(F)(F)C2)OCC)=O)(COC)CN(C(C2CC2C)=O)C1 C#Cc1ccc(C(=O)NCCCN(C(c2c[nH]c(=NC)s2)=O)C(C)C)c(OC)c1 CCCC(O)C(=O)N1CC=CC1(C)C(=O)NCCN(CCC)C(C)C C#Cc1nc(C(N2CCC(CNC(c3cnn(CCC4CC4)c3C)=O)C2)=O)cs1 c1(C(=O)NC(CC(C)NC(Cn2c(C)c(Cl)cn2)=O)C)n[nH]c2c1COC2 c1(NC(C2(CNCc3ccc(O)nc3)CC2)=O)cccc2c1OCO2 CC1CN(C(=O)C(=O)NC2(c3ocnc3C(F)(F)F)CC2)CCC1N1CCCC1 C1(NC(C(CC=C)OC)=O)CCN(C(=O)CCc2cccnc2C)C12CC2 C1(O)(C(C(=O)NC2CC(C(=O)OC)C2)NC(C2SCCS2)=O)CCCCC1 c1(C(=O)OC(C)(C)C#N)ccc(NC2CCS(=O)(=O)C2)c(N)c1 c1(C(N2CC(OCCNC(C3CC(C)OC3)=O)C2)=O)nc(Cl)c(Cl)s1 c1(C(=O)NC(C)(CNC(C2CC3C=CC2O3)=O)CO)cncc2cnccc12 Cc1cn(C(C)(C)C(=O)NC2CC(NC(=O)CC3CC3(Cl)Cl)C2)cn1 c1(C(N2CCC(N(C)C(c3ncn4c3CCC4)=O)C2)=O)c(Cl)cc(Cl)nc1N C1(CNC(C(C)SCCCC)=O)CC(C)(C)CN1C(C1CCN(CC(C)C)C1)=O CC#CC1CCN(C(C2CN(C(C3CCC3(OC)OC)=O)CCO2)=O)C1 c1(OCC)c(C(=O)NCC2CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)cccc1F C12(CNC(C(C)=C(CC)C)=O)CC(NC(c3cccn3C(C)C)=O)(CO1)C2 C1(C(=O)NCC2CC(F)(CNC(C3N(N=O)CCC3)=O)C2)CCCC1C1CC1 CCCCC(C)C(=O)NCCc1n[nH]cc1C(=O)NCC1CCC(O)C1 c1(NC23CCN(C(C(C)NS(CC)(=O)=O)=O)C2CCC3)cc(C)nc2ncnn12 C1(C(=O)NC(CSCCC)C(=O)OC)CN(C(=O)OC(C)(C)C)CCS(=O)(=O)C1 c1(C(=O)NCCOCCOC)oc(CNC(c2cnc(C)n2C)=O)nc1C Cc1c(C(=O)NCCC(N2CCC(C)C(CO)C2)=O)cncc1F c1(C(=O)NC2C3(CC(NC(c4cnccn4)=O)C3)C2)ccc(Br)cc1F c1(NC)cncc(C(=O)NCCC2CN(C(C3CCCN3S(C)(=O)=O)=O)C2)c1 CC1CCCCC1n1nc(CC2CCCC2)nc1C1CC(=O)N(CCN(C)C)C1 C1(C(N(CC(C)SC)C)=O)CCC2(CC2)N1C(=O)CC(C1CC1)C1CC1 CCC(O)C(C)(C)C(=O)N1CC(CNC(C2CC2C(C)(C)C)=O)C(F)(CO)C1 CC1CN(C(C2CCN(C)C2)=O)CC1(C)CNC(C1CC2(CSC2)C1)=O C(CCC(C)C(=O)NC(C)CCCNC(=O)Cc1cncn1C1CC1)OC N1(C(Cc2cc(C)on2)=O)CCCC(C2CCCCN2C(=O)CN(C)C(N)=O)C1 c1(OC)ccc(OC(F)(F)F)c(C(=O)NC2CCC2NC(=O)CCSC(C)C)c1 N1(C(CC2(OC)CCCC2)=O)CC(NC(=O)CSc2n[nH]c(O)n2)C(F)C1 c1(CCNC(NC(C(=O)NC)(C)C)=NC)c[nH]c2cc(Cl)cc(Cl)c12 CC1CCC=C1C(=O)N1CCN(C(=O)Cc2ccc(O)c(Cl)c2)CC1CF C1(NC(C(C)CS(C)=O)=O)CC2(CCN(C(c3cnc(N(C)C)s3)=O)C2)C1 c1(C(=O)NC(C2C(C(N(C3CCC3)CC#C)=O)C2)C)cc(C2CC2)on1 c1(OC)nccnc1C(=O)NC1CN(C(=O)CCc2csc(=N)[nH]2)CC1OC Cc1ccsc1CC(=O)NCC=CCNC(C1CCN(Cc2ccccc2)C1)=O C(=O)(CCCC(C)(C)NC(=O)CC1CCC(C)O1)NCc1ccc(C)cc1F C(=O)(CC(F)(F)C(F)(F)F)NC1C(NC(C2CCN(C)C(=O)C2)=O)COCC1 C(=O)(CC(C)CC(=O)NC1CCC(CCNC(=O)C2=CCOC2)C1)OC C#CC1(C(=O)NCCS(C)(=O)=O)CCN(C(c2ccsc2Cl)=O)C1 Cc1nn2c(c1C(N1C3CCC1CN(C(C14COCC1C4)=O)C3)=O)CCCC2 C(C1CCc2ncnn21)NC1C(C)CCCCC1 C1(NC(C)=O)COCCN(C(c2c(CCc3ccccc3)noc2C)=O)C1 c1(C(N(C2CCN(C(C(C3CC3)OCC)=O)C2)CCO)=O)cnc2cc[nH]c2c1 N1(C(C(=O)NC2CC2)=O)CCCCC1CCNC(C1(F)CCCOC1)=O N1(C(C2C(C=C)C2)=O)CCC2(C1)CN(C(=O)C(C1CC1)SC)C2 Cc1nc(CCC(=O)OCc2nc(C(F)(F)F)n(C)n2)[nH]c1C CC(CC(N)=O)C(=O)NC(CNC(c1cnc(C2CC2)[nH]c1=N)=O)C(C)(C)C C1(CNC(c2c(C)nco2)=O)CN(C(=O)Cn2c(C)c(C)sc2=O)CCN1C c1(C(=O)NC2C(CNC(C(C)OCC3CC3)=O)CC2)cnc(S)[nH]1 c1(-n2cc(C(=O)NC3CC(SC)C3)nn2)ccc(N)cc1 C(=O)(C(C)CS(C)(=O)=O)NC1C=CCN(C(=O)Nc2cnc(C)nc2C)C1 C12(CNC(Cc3n(C)ncc3)=O)CC1CN(C(=O)Cc1csc(Br)c1)C2 c1(C(=O)OCC(N2CCCC(c3nnc(C)o3)C2)=O)nncc2ccccc12 c1(NCC(C(=O)OC)(C)NC(=O)OC(C)(C)C)cc(OC)ncc1Cl CC(=O)CCCC(=O)N1CCCC1C=CC(N1CCOC(C)(C)C1)=O c1(NC(=O)CC2CC(NC(=O)Cn3cnnc3O)C2)cccc(Cl)n1 C(=O)(CCCCC(=O)NC)NCCCN(C(=O)CCC(C)(C)C#N)CC Cc1nn(C)c(C)c1C1CCCN1C(C1CCC(CNC(C)(C)C)CC1)=O c1(SC)ccc(O)c(C(N2CCC(NC(c3ocnc3C(F)F)=O)C(F)C2)=O)c1 N1(C(C2(CC=C)CC=CC2)=O)CC(C2CC2)C(F)(C(=O)O)C1 C(=O)(C=C1SCC(=O)N1C)NC1CCN(C(CN2CCN(C)CC2)=O)C12CCC2 CCC(CNC(=O)CC1CCC(=O)N1C)(CC)C(=O)N1CC(C)(C(F)(F)F)C1 C1(NC(c2c(CC)nns2)=O)COC2(C1)CN(C(C1CCC1(C)C)=O)C2 CC1(C(=O)NCC2(CNC(=O)CNC(=O)C(F)(F)F)CC2(F)F)CCOC1 N1(C(C)=O)CCCC1(C)C(=O)N(C1CCC(C(=O)CC)CC1)C(C)C CC(C(C)(C)C(=O)N(C)CCC1CC1)NC(C1C2CCCCC12)=O CC1CCC(=CC(N2CCC(NC(=O)C(c3ccc(Cl)nc3)(F)F)C2C)=O)CC1 c1(Nc2cccc(C(N3CCC(C)(F)C3)=O)c2)ncc([N+](=O)[O-])cc1Cl C1(C(N2CCC(C(C)CO)CC2)=O)CN(C(c2ccsc2C#N)=O)CC1(F)F CC1CN(C(C2CC(N)C2)=O)CC(C)N(C2CC2)C1 C1(C(=O)NCCCOCCOC)CC2CCN(C(=O)C(C)(O)C(F)(F)F)CC12 N1(C(=O)NCCCCC2C(C)C2)CCOC(C2CC(F)(F)C2)C1 c1(C(=O)NCC#CCNC(CNC(C)=O)=O)ccc(C2CCOC2)cc1 C1(O)(C(N(C)CCOCCC(=O)NC(C(C)(C)O)C2CC2)=O)CCOCC1 N1(C(C(C)C2CC2)=O)CCCC2(C1)CN(C(C1CC3CCC1C31CC1)=O)CCO2 c1(NCC)cnccc1C(N1CCC1CNC(c1ccnc(OC)c1)=O)=O CC(CCCCNC(=O)C(C)c1cccs1)NC(=O)Cn1cnnc1O CC(C1CCCCC1)=CC(=O)NC(c1ccccc1)CNC(c1[nH]ccc1C)=O C1(NC(c2cc(CC)no2)=O)CCCC(NC(c2cn(C3CCC3)nc2C)=O)C1 C=CCCCC(C(=O)NC(C1CCCC1)C)NC(C1CCOC1)=O C(c1ccsc1)=CC(=O)NCCC1CC(NC(=O)CCOC2CCC2)C1 C1(CCC)CN(C(C2(C)CCCOC2)=O)CCN1C(c1ccc(F)c(CC)n1)=O C(=O)(C(O)(C(C)C)C(F)(F)F)NC1(CNC(c2c(C)snn2)=O)CCCCC1C C(=O)(C(F)(F)CC1CC1)NCCN(C(c1nc(Cl)cs1)=O)CC c1(C(=O)NC2CC(CCNC(c3ncc(C(F)F)s3)=O)C2)cccc2ccnn12 C1(CNC(C2CCC=CCC2)=O)CC12CCN(C(C1CC3(CCCC3)C1)=O)CC2 Cc1cccc(CNC(C2CSCN2C(C2CC3CC3C2)=O)=O)c1O CCCC(CNC(C1(OC)CCN(C(c2cc(C)nn2CC)=O)C1)=O)CCO Nc1cc(Cl)ccc1C(=O)NCCCCNC(=O)CCCC1CCOCC1 C1(CC=C)CCN(C(C2C=CCN(C(=O)C(C)NC(=O)NC)C2)=O)CC1 C1(C(=O)NC2CC(=C3CC3)C2)(CC)CCN(C(c2cncc(C)n2)=O)C1 C(=O)(C1CCCc2ccnn21)NCC1(F)CC(NC(C(C)(C2CC2)OC)=O)C1 CC1C2CC(C2NC(=O)COc2cc(F)cc(Cl)c2)N1C(=O)Cn1ccnn1 C1(NC(C(C)S)=O)CN(c2nccc(C(F)F)n2)CC1F Cc1ccc(C=CC(=O)NCc2cn(CC(N3CCC(O)CC3)=O)nn2)o1 N(C(=NCC1(CO)CCC1)NCCC1CCOC1)CC(=O)NC(C)C N1(C(CCC=CCC=C)=O)CCN(C(=O)Cc2ccnn2C)CC1CC(=O)NC C(=O)(CC(C)CC(F)(F)F)NC12CCN(C(CCCC(=O)OCC)=O)C1CCC2 N1(C(COC(CC)C)=O)CCCC1CCCNC(c1n[nH]cc1C(F)(F)F)=O c1(C(=O)OC)cscc1-c1c[nH]cc1C c1(C(N(C(c2c(C)cccc2)c2ccc(Cl)cc2)C)=O)nn2ccccc2c1Br C1(NC(CC(CC)C)=O)CCCN(C(C2CCC(=O)O2)=O)CC1 C(=O)(C(O)CC(F)(F)F)NC(C(=O)NCc1cnn(CCF)c1)Cn1cncn1 C=C1CCN(C(c2ccc[nH]2)=O)C(C(=O)NCC(C)N=[N+]=[N-])C1 C1(C(N2C(CC=O)CC2)=O)(CO)CCCCCC1.c1(CN)csc(Cl)n1 CC1C(NC(=O)Cc2ncsc2Cl)CCN1C(=O)CC1CC(F)C1 C1(C)(NC(CC2(N(C)C)CCC2)=O)CC(NC(C2CCC(O)C2)=O)C1 C1(N=c2[nH]nc(-c3ccccc3)o2)(CNC(C2C(C)(C)CC2)=O)CCOCC1 Cc1ccc(=O)n(CC(=O)NCC2CN(C(C3CCCN(C)C3)=O)CC23CC3)n1 CCCC(CCC)C(=O)N1CCCC(NC(c2ccc(C)o2)=O)CC1 c1(Sc2ccc([N+](=O)[O-])c(Cl)c2)c(F)c(F)c(F)c(F)c1F c1(C(=O)NCCN(C(=O)C(C2CC2)OC)CC)cc(Cl)cc(Br)c1N n1(CC(=O)N(C(CNC(c2c(C)ncnc2O)=O)C)C)sc(=O)c2ccccc12 C1(C(=O)NCCN2CC3CC3C2)CN(C(=O)CC2CC2(Cl)Cl)C2(CCC2)C1 C1(NC(c2ccc(C)c(CO)c2)=O)CCN(C(C2CCC2C)=O)CC(C)(C)C1 C12(NC(C3C(C)C3)=O)CC3CC(C1)CC(CNC(=O)CNc1nccs1)(C3)C2 N#CC1CCC(C(=O)NC2CCC(NC(c3ccc(N4CCC4)nc3)=O)CC2)C1 c1(C2(NCC3NCC(C)(C)C3)CC2)cc(Br)ccc1F C1(CCNC(C(COC)(C)C)=O)CCCN(C(C2(C)C=CCCC2)=O)CC1 C1(CNC(C(CC=CC)NC(c2ccc(CSC)o2)=O)=O)CCC(=O)NC1C N1(C(CCCNC(C)=O)=O)CC(CNC(C2CC(C)(O)C2)=O)C(C)(C)C1 C1(C(N(C2CCN(C(c3n(COC)ncc3)=O)C2)C)=O)CC(F)(F)CCC1(C)C C1(C(=O)NCC2(CC(C)C)CCC2)(NC(C2CCCO2)=O)CCN(C)C1 c1(C(N2CC(CC)C(NC(=O)CC(CC)CC)CC2)=O)ccc(C)c([N+](=O)[O-])c1 c1(C(N2CCC(CNC(C(F)OC)=O)C2)=O)cc(C#N)c(C)cn1 c1(C(=O)NCCCNC(c2c(C(C)(C)C)noc2)=O)ccnc2ccc(F)nc12 C1(F)(C(N(CCCNC(=O)CCc2nncn2C)CC)=O)CCOC1C c1(C(=O)NCC2CC(NC(C3(NC(C)C)CC3)=O)C(O)C2)cc2ncccc2s1 c1(C(=O)NCCC2CC(NC(C3CCC(F)C3)=O)C2)nccc2ccsc12 c1(OC)ncnc(N2CCCC(NC(=O)CC3OCCCC3(C)C)C2)c1OC N1(C(CC(C)SC)=O)CC(C)(C)CCC1CNC(=O)CC1CCC(C)(O)CC1 O=C(N1CC(O)C(O)CO1)c1nn2c(c1Br)OCCC2 c1(NCC)cccc(-c2cn(CCNC(C3C(C)C3(F)F)=O)nn2)c1 c1(OC)cc(-c2ccc(C(N3CCCC3C3(O)CC3)=O)cc2)sc1S(N)(=O)=O C1(C#CC(=O)NCCCCNC(=O)CCc2cccnc2Br)(CC)CC1 Cc1ccc(C(N2CCN(C(=O)CSC(C)(C)C)CC2CF)=O)c(N)c1C Cc1cc(NC(=O)C2CC2)sc1C(N1CC(SCCNC(=O)CC(F)(F)F)C1)=O O=C(CCCNC1CCOC(c2ccc(F)cc2)C1)c1ccccc1 Cc1cccc(=O)n1CC(C)(O)C(=O)N(CCC(C)NC(=O)Cc1nc[nH]n1)C CCCCC(C)(F)C(=O)N1CC(CC(=O)NCCCC(=O)NO)(OC)C1 c1(CN2CC(CC(=O)Nc3cnccc3Br)OCC2)cc2ccccc2[nH]1 c1(OC)cc(F)c(F)cc1NC(=O)NCc1cc(F)c(F)c(F)c1 c1(C(N(CCCNC(C2(SC)CCCC2)=O)CC)=O)ncc(SC)cn1 c1(NCc2ccc(C)cc2F)cc(C)c(S(=O)(=O)NC2CCCS(=O)(=O)C2)cn1 C=Cc1cnn(C)c1C(=O)NC1COCCC1NC(C1CN(C(N)=O)C1)=O c1(C(=O)NCC(C(C)(C)C)NC(=O)CC2(C)CC2(F)Cl)cc2cccc(F)c2o1 C(=O)(C#CC1CCOCC1)N1CC2(CNC(CCC(=O)N(C)C)=O)C(C1)CCO2 N1(C(c2c(C)c[nH]n2)=O)CCN(C(=O)CCc2nc(C(F)(F)F)n[nH]2)C2CCC12 CCCCCC(O)CC(=O)N1CCC(CNC(c2coc(CO)c2)=O)(OC)CC1 C(c1cncc(O)c1)=CC(N1C(C2CCN(C(CCCC)=O)CC2)C(C)(C)C1)=O c1(C(N(C2CC2)CC2N(C(c3nc(C(C)C)sc3)=O)CCC2)=O)nc(=O)n(C)[nH]1 C(CC)(C(=O)NC(C)CCCNC(c1ccc(Cn2cc(Cl)cn2)o1)=O)OCC c1(OC)ccc(Cl)cc1N1CCC(NC(=O)NCc2ccc(C)s2)C1 N1(C(CCCC=C)=O)CCC(O)C(NC(c2cc(Cl)cnc2OC)=O)C1 N1(C(C(n2cc(Cl)cn2)C)=O)CC=C(CCNC(c2nocc2C2CC2)=O)CC1 c1(C(=O)NC(CC(C)NC(=O)CNC(N)=O)C)cccc(C2(C#N)CC2)c1 C1(C)(NC(c2cc(C)sn2)=O)CCCN(C(c2ccncc2C2CC2)=O)C1 c1(OC)c(C(N2CCCC(CN(C(=O)Cn3cncn3)C)C2)=O)csc1C c1(C(=O)NCC(CC)NC(c2nc[nH]c2C(C)(C)C)=O)ccc2c(c1)CCO2 CCC(C#N)C(=O)N1CCN(C(=O)C(n2cc(-c3ccccc3)nn2)C)CC1 C12(C(N(C3CC(O)C3(C)C)C)=O)CCCC1CN(C(c1ccnn1C)=O)C2 c1(CC(=O)NCCCCC(C)NC(Cc2ncc(C)s2)=O)ccccc1S(C)=O n1(CCC(=O)NC2CC3CCC2(C(=O)O)C3)c(=O)oc2cc(Cl)ccc12 c1ccn2ncc(CN3CCC4(c5cccnc5)CC4C3)c2c1 Cc1cnc(C(C)NC(C2(F)CN(C(=O)C(F)F)C2)=O)s1 C1(C(=O)NC2C(NC(c3n(CC#C)ccc3)=O)CC2)CCC2CC1C2(C)C c1(NC(C2CN(C(c3ccc(OC)nn3)=O)C2)=O)ncnc(OC)c1[N+](=O)[O-] Cc1c(C(N2CCC(C)C(NC(=O)C=Cc3cccnc3)C2)=O)nn(C)c1N Cc1cccc(C(C)C(N2CCC(O)(CCNc3nccc(CO)n3)C2)=O)c1 C(C)(C)(CC(F)C(=O)N(CCCO)C(C)C)NC(c1cccc(C)c1C)=O c1(C(=O)NC(CN(C(C2CC2CN(C)C)=O)CC)C)cnc(O)cc1C c1(C(=O)NCC2N(C(c3c(C)cc(Cl)cn3)=O)CCC2)ccc2c(C)c[nH]c2c1 c1(C(=O)NC2C(CC)N(C(C3CCSCC3)=O)CC2)ccc(S(C)=O)cc1 CCC(C)(C(=O)NCC1CC1NC(c1nc(C)ccc1O)=O)C(N)=O c1(C(N(C2CN(C(CC3CCCN(C)C3)=O)C2)C)=O)cccc(P(C)(C)=O)n1 Cc1cc(F)ccc1C(=O)NCC1CCCN(C(C2CCCCS2(=O)=O)=O)CC1 C1(NC(CN(C)C(N)=O)=O)CC2(C1)CC2NC(c1c[nH]cc1C1CC1)=O c1(C(N2CCN(C(C(C)CC(F)F)=O)CC2)=O)coc(C#Cc2ccccc2)c1 c1(NC(C(N2CCN(CCOCC)C(=O)C2)=O)=O)ccc2c(c1)CCC(O)C2 C12(NC(C(C)=C(CC)C)=O)CCCC1N(C(c1c(C)cnn1C)=O)CC2 C(=O)(C1OCCc2c(O)cccc21)NCC1C(C)CN(C(C2(Cl)CC2)=O)C1 C1(NC(C(CC=CC)NC(=O)C2=C(C)CC2)=O)CC2C=CCC(C1)C2 N1(C(CC(=C)Br)=O)CC(C)C(NC(=O)CN2C(=O)NC(C)(C)C2=O)C(C)C1 C(C(C)(C)C(=O)NC1CCN(c2nncs2)C1)OC(C)(C)C c1(C(=O)NC(C)Cc2ccc(O)c(O)c2)cc(Cl)c2[nH]c(O)nc2c1 N1(Cc2ccc(COCC)o2)CC2(CCC(C(=O)NCCC3CCCC3)O2)C1 c1(C(=O)NCC2CC(Cn3cc(CO)nn3)C2)ccc(Br)cc1Cl C1(C(=O)NC2CC(CCNC(=O)CC3CC3C3CC3)C2)CC2(CCC2)C1 n1(CCCC)nc(C)c(CNC2(c3nnnn3CC)CCC2C2CC2)c1Cl c1(C(=O)NC(C2CCCC2)CNC(CC(C)F)=O)nnn2c1CCCC2 C=CCC(CNC(=O)CNC=O)NC(=O)CC1CS(=O)(=O)C1 c1(C(N(CCCNC(=O)CC2(C)CC2(F)Cl)CC)=O)ccc2cc(O)ccc2c1 N1(C(CCC(=C)Cl)=O)CC2CCC2(NC(=O)C=Cc2nc(C)co2)C1 N1(C(C2(C)CC2(F)Cl)=O)CC2CC(C1)C2NC(=O)CC1CC1 C(=O)(CCCOCCNC(C1C(C(=O)O)C1(C)C)=O)N(C1CSC1)C C12(CCN(CCC(=O)NC3CC3)CC1)C(=O)N2.C1(COC)CC12CCSCC2 C1(C2(O)CCC2)(C(=O)NC(C2CCN(C(c3cn(CC=C)nc3)=O)C2)C)CC1 N12CCCN(CC1)CCC1CCC3(CC13)C2=O.CC(C)(C)OC(=O)NC(C)(C)C c1(OC(C)C)nc(N2CCC(NCc3cnc(O)c(Cl)c3)C(O)C2)ncc1Br CC(CC(F)(F)F)C(=O)NC1CC(CNC(=O)COc2ccccc2F)C1 N1(C(=O)NCc2c(C)ocn2)CCC12CCCCC2 c1(C(N(C)CCN(C)CC2CCN(Cc3ccccc3)CC2)=O)cccc(I)n1 Cc1ccc2oc(C(N3CC4CCC4(NC(c4ccc(Cl)cn4)=O)C3)=O)cc2n1 C12(CNC(CCSCC(=O)OC)=O)CCC(NC(C3CCC(=O)NC3)=O)(CO1)C2 C(=O)(C#CC(C)(C)CNC(C1CCSC1)=O)N1CC(N(C)C)C1 C1(C(=O)NCCOCC(F)(F)F)CC12CCN(C(=O)CCC1CCCC1)C2 c1(-c2ccc(Nc3nc(-c4cc(O)ncc4)sc3)cc2)c[nH]c2nccc-2c1 N1(C(=O)NCCCCOCC)CCC2(CC1)CN(C)C(=O)O2 N1(C(c2cccc(C#C)c2)C(=O)NC(C)C(=O)OC)CCc2ccc(O)cc2C1 N1(C(C(C2CCC2)OCC)=O)CC2CCC2(C(=O)NCC2(C)CC(F)(F)C2)C1 c1(CNC(c2csc(C3CCCN3C(c3cc[nH]c3)=O)n2)=O)ccc(F)cc1Cl CC(C)(C)CC(C)(C)C(=O)NCC1(NC(=O)Cc2ccccc2Br)CC1 C1(NC(c2ccnc3cc[nH]c23)=O)C2CCN(C(c3cscn3)=O)CCC12 c1(CC(N2CC(NC(CN(C3CC3)CC)=O)C(O)C2)=O)cc(Cl)ccc1OC c1(C(N(C2CCC(NC(=O)CCC3CC3(F)F)C2)C)=O)cc(C(N)=O)no1 c1(C(=O)NCC2CCCCN(C)C2=O)cc(F)c(F)c(F)c1O CC1(C)CCN(CC2CCC(NC(=O)OC(C)(C)C)CC2)C1C1CC1 Cn1cnc(C(=O)NC(C)(CNC(C2CC(C3CC3)=NO2)=O)CO)cc1=O C1(CC(=O)NCC2(CO)CCN(C(CN(C)C3CC3)=O)C2)CCC2(CC2)CO1 Cc1cn2c(n1)CCC(C(=O)NCC1CC(=O)NC(C3CC3)C1)C2 C12(C(N(C3CN(C(C=Cc4c(C)n[nH]c4)=O)C3)C)=O)CCC(C(=O)O)(CC1)CC2 C1(NC(C(C)(C)n2cncn2)=O)CCOCC1C(=O)N(C1CCC1)CCO C1(NC(C(F)=CC)=O)CC(O)CN(C(C2(c3cccc(Br)c3F)CC2)=O)C1 C1(CCC(=O)NCCC(C(=O)OC)C)CCCCN(C(c2c[nH]c(=O)cn2)=O)C1 CCCC(C)(C)CC(=O)NCC1C(C)CCN1C(c1ncccn1)=O N1(C(N(CC)CC)=O)CCC2(C(N3CCC3(C)C(=O)OC(C)(C)C)=O)CC2C1 O=[N+]([O-])c1ccc(CSCCC2CCC3CC23)c([N+](=O)[O-])c1 c12cccc(F)c1C(=O)N2.Cc1ncc(CN2C3CCC2CC3)cn1 c1(C(N2CC(NC(c3cc(C)on3)=O)(CO)C2)=O)cccc2c1nnn2C C(CS(=O)(=O)C1CCCC1)N1CC2C(C(N3CCCCC3CO)=O)(COC2)C1 N#Cc1c[nH]c(=NC2CCC(C(N3CC4CC4C3)=O)OC2)c2sccc12 N1(C(c2c(Cl)cc(C)s2)=O)CCC(F)(CNC(=O)CSC2CC2)CC1 O=C(CCC(=O)c1cc(Cl)sc1Cl)NCc1ccc(OC(F)F)nc1 c1(C(=O)NC(C(CO)NC(C(CC)C)=O)C)cccc(N2CCCC2)c1 C1(C(=O)NC(CC)C(=O)OC)CC2(CCN(C(=O)Cc3cc(C)on3)C2)CO1 c1(OC)cc(C(N2CC3CC2CN3S(=O)(=O)CC2CCC2)=O)cnc1Cl C1(NC(C2CCOCC2)=O)CC2CN(C(c3ccnc(Cl)c3F)=O)CC12 CS(=O)c1nc2ccc(NC3CC(CO)C3)cc2[nH]1 C(C(CC(F)(F)F)NC(C1CCCS1)=O)NC(CCN(C(C)=O)C)=O c1(C(=O)NCC2C(NC(c3ccc(OC)cc3N)=O)C2)ccc2nc(Cl)nn2c1 c1(C(=O)NC2CCC(NC(C(CCCC)C)=O)C2)cnn2ccnc(N)c12 CC1CCN(CC(=O)N(C2CN(C(=O)CN(C3CCC3)C)C2)C)C1 CCC(CC(C)C)C(=O)NC1(COC)CCN(C(c2cccc3nn[nH]c23)=O)C1 c1(CC)conc1CNCCNC1COCC1F CC1CN(C(=O)COC2CCOC2)CC1NC(c1cncc(N(C)C)c1)=O c1(OC)cc(NC(=O)C(c2cccs2)NC(=O)C(F)CC(C)C)cc(O)c1 C1(C(N2CC(N(C(C=CC=CCC)=O)C)C2)=O)CC12CCCOC2 C1(CN(C(C(CC)C(C)C)=O)CC)CC2CCC(C1)N2C(=O)C1=C(C)OCCS1 C1(C(=O)NC(c2c(C)ncs2)C)CCC2(CC2)N1C(=O)C(C)CO c1(C(COCCOCCOC)NC(=O)NC2CCN(C3CC3)C2)ccc(F)cc1 c1(OC)cccc(C(CNC(C2CC23CCCC3)=O)NC(c2cccnc2)=O)c1 c1(OC)ccc(-c2nc(Cc3ccc(=O)n(C)n3)n(C3CCOC3C)n2)cc1F C(=O)(C#CC1CCOC1)NC1CC2(C(NC(=O)CCNC(C3CCC3)=O)C2)C1 C(N=c1nc(C)nc2[nH][nH]cc1-2)C1(OC)CN(C(c2nnn(C(C)C)c2C)=O)C1 c1(SC)nccc(=NC2CN(C(=O)Cc3ccccn3)CC23CCC3)[nH]1 N1(C(CN(C(C(CC(=O)OC)C)=O)C2CC2)=O)CCN2CC(C)CC2C1 Cc1cc(C(N)=O)cs1.c12nnnn1C1CC(CC2(C)N)C1.C(C)C N1(C(CC2(CC)CCOCC2)=O)C2CCC1(CNC(c1csc(C)n1)=O)CC2 N1(C(c2c(C)cno2)=O)CCN(CCN(C(=O)C(N2CCCC(O)C2)C)C)CC1 C1(C(=O)NCCc2n(C)ncn2)CCN(C(c2ccc(C(N)=O)[nH]2)=O)CCO1 N1(C(C(c2c(C)noc2C)C)=O)CC(NC(c2ccc(F)s2)=O)CC2(CC2)C1 c1(C2C(N(C(=O)NCCC(C3CCCC3)OC)C)C2)ccncc1 c1(C(N(CCC)CCNC(=O)C(C)Oc2ccccn2)=O)ccc(C(F)(F)F)s1 Cc1ccc2c(c1C(N1CC(C3CN(C(C4CC(F)C4)=O)C3)C1)=O)CCCN2 N1(Cc2cn(C3CN(C(=O)OC)C3)nn2)CCN(C(c2cc[nH]n2)=O)C(CO)C1 c1(C(N2CC(O)(CC(=O)N(C(C)(C)C)CC3(C)CCC3)C2)=O)ccccn1 c1(C2(C(N(CCNC(C3CCC3C)=O)CC)=O)CC2)ccccc1Cl CCCC(CC)CCC(=O)NCC1CN(C(c2cc(Cl)ncc2O)=O)CCCO1 CCC(C)CC(C(=O)NC(C)C(=O)N(C)CC)NC(=O)Cc1ccco1 CC(C)C(C(=O)NCC(C)Cn1cccn1)N1CCCS1(=O)=O N1(Cc2c(OCCC#C)cccc2)CCCC(C(=O)N(CCCCCC)C)CC1 Cc1cnccc1CCNC(=O)NC(c1nncs1)C1CC1 C1(C)(NC(C(C)SCCCC)=O)CCCN(C(C23CC4CC2C3C4)=O)C1 c1(C(N(C(C)C(=O)NC(c2ncsc2C)C)CC)=O)cnn(CCF)c1 N1(C(C2(CC(=O)OC)CC2)=O)CC2CCC(CNC(C3CC(C)(C)CO3)=O)(C2)C1 C1(CN(C(=O)CC2(O)CCC2)C)CN(C(=O)C(N2CCCC2)C2CC2)CCO1 C(C(C)C)(C(O)C(=O)N1CCSCC1C(=O)NCC1(O)CCN(C)C1)OC C12(CNC(C=C(CCC)C)=O)CCC(NC(=O)C(O)CSC)(CO1)C2 c1(C(=O)NCC(CNC(C2C(OC)CCCC2)=O)(C)C)c(Cl)ccc(Cl)c1O C1(N(C(=O)COc2ccon2)C)CCC(NC(=O)C(F)C2CCC2)C1 C1(C(=O)NCC2CCCC(NC(=O)CCc3cncnc3)C2)(OC)CCOCC1 c1(-n2cc(C3CCN(C(=O)CC4CC=CCC4)CC3)nn2)cccc(Br)c1 N1(C2C(=O)NCC2)CCC(NC(c2cc3sccc3s2)=O)C(O)C1 N1(C(c2n(CC=C)ccn2)=O)CCC(O)(CNC(=O)C(C)(C)C)CC1 N1(C(c2nn(CC)c(O)c2)=O)CCCOC(CCNC(=O)CC2CC=CCC2)C1 C#CCCCCCC(=O)NCC(C)CC(=O)N(C)CC1CC1 c1(NC(N2CCN(C(C(CC)C)=O)CC2)=O)c(I)cc(Br)cc1[N+](=O)[O-] c1(C(N2CC3C(NC(C4CC(C)C4)=O)(C3)C2)=O)ccc(O)c([N+](=O)[O-])c1 Cc1nn(C)cc1CC(=O)NCC(CC(C)C)NC(c1nc(=N)cc[nH]1)=O c1(CC)cccc(C(N2CCC(C(N3CCC3(C)C)=O)C2C)=O)c1 N1(c2ncc(C)s2)CC2C(C(=O)NC(c3cccc(C(C)C)c3)C)C2C1 CC(CCC(F)F)NC(=O)NCC(c1cnn(C)c1)C Cc1nccc(C(=O)NC2CCC(CNC(c3c(C)noc3C(F)F)=O)C2)c1C C1(NC(=O)CC(F)F)COC2(CCN(C(=O)CN3CCOCC3)C2)C1 N1(C(CC(=O)OCC)=O)CCC(O)C(NC(c2cncc(SC)c2)=O)C1 C(=O)(C(C(C)C)n1cc(Br)cn1)NCC(C)NC(COCCCC#C)=O C1(C2C(=O)N2)CCC(C(=O)O)CC1.C1(N(CCCC(C)O)C)CCC(CO)CC1 N1(C(CC2C(C)(C)C2(C)C)=O)CC2CCC1C(NC(c1cnn(C(F)F)c1)=O)C2 N1(C(CCCC)=O)CC2CCC1C1CN(C(=O)Cn3cc(C(F)(F)F)cn3)CC21 C=CCCC(F)(F)C(=O)N1CCC(F)(CNC(c2cncc(F)c2Cl)=O)CC1 N1(C(C(COC)C)=O)Cc2ccccc2CC1CNC(=O)CCc1scnc1C C1(NC(=O)C=CSc2nc[nH]n2)CC2CN(C(c3ccc(O)nn3)=O)CC2C1 C(=O)(C1=CCOC1)NC1CCC(CCNC(C2(C)CCOC2)=O)C1 C1(CNC(c2cc(CC)[nH]n2)=O)CCC12CCN(C(c1cncnc1)=O)CC2 c1(CSC)cc(C(=O)NCC2(NC(=O)CCC(F)F)CCCCC2)ccc1F c1(C(=O)NCC(C)NC(C(CCSC)O)=O)cc(F)cc2ccoc12 CCCC(C(N)=O)NC(c1ccoc1CNC(c1ccccn1)=O)=O c1(OC)ccc(OC)c(CC(=O)NC(C2CN(C(=O)CCc3ccon3)C2)C)c1 N1(C(CN(C(Cn2c(C)ncc2)=O)C)=O)CC2CC2(CNC(c2ccoc2)=O)C1 c1(COCC(=O)NC(C)CNC(=O)CSc2ccccc2)ccnc(O)c1 C12(CNC(CCCOCC=C)=O)CC(CN1C(=O)C(C)(C)F)C2 C1(C(=O)NC2C=CCCC2)CCCN(C(=O)COc2ccc(O)cc2)CC1 c1(C(=O)NC2CN(C(C3COCCN3)=O)C2)cc2cc(F)ccc2[nH]1 c1(C(N(C2CCCN(C(C3(C4CC4)CC3)=O)C2)C)=O)cccc2c1NCC2 C1(C(=O)NCc2c(OC)cccc2)CN(C(=O)OC(C)(C)C)CC1(F)C(=O)O c1(OC)cc(N)c(F)cc1C(=O)NC1(C)CC(NC(=O)Cc2ccoc2)C1 C(C)(C)(CC(=O)NCC1CN(C(c2cnns2)=O)CC1C)OC S(=O)(=O)(c1ccc(Br)cc1NCC1(C)CCC(=O)N1)N(C)CCn1cc(Br)cn1 c1(OC)cc(C)ccc1C(=O)NC1CCCC1NC(=O)CC1CC1C(F)(F)F C1(NC(Cc2ccc(-c3cn(C(C)C(=O)O)nn3)cc2)=O)COC2COCC12 c1(C(=O)NCC2C(CC)CCN2C(=O)Cc2ccsc2C)cc(C)c(F)c(C)c1 C1(C)(C(=O)NC2CC(CCNC(c3[nH]cc(C)c3)=O)C2)CCCNC1=O C1(C)(CC)CCC(C(=O)NC2(CNC(=O)C(=Cc3ccccc3)C)CCCC2)O1 c1(C(CNC(CN(C(=O)CC2CC3C=CC2C3)CCC)=O)=O)cccc(C)c1 CC1CN(C2CC2)CC1NC(C1(CCNC(=O)CC2CC2)CC1)=O N1(C(c2cccc(NC(C)=O)n2)=O)CCC2(CCN(Cc3cc[nH]n3)CC2)C1 CC(C)CC(=O)NCCCC(=O)NC1CC(NS(C)(=O)=O)C1.C1(=O)CCN1C C1(C(=O)OC)CCCCC1C(=O)NCCCCNC(=O)C=Cc1cscn1 c1(C(N2CCN(C(=O)CSc3ccccc3)C3CC23)=O)cc2c(cn1)OCCO2 CC1CC(=O)NCCN1C(C1(CNC(c2cc(O)ncc2F)=O)CC=CC1)=O c1(N2C(C(=O)Nc3ncc(F)cc3F)CC2)ncnc2ccc(Br)cc12 N1(C(C2CCC(C)CC2)=O)Cc2occ(C(=O)NCCC3CC3C)c2C1 C(N=c1[nH]cncc1Cl)C1CC(NC(c2ccc(OC)c(Cl)n2)=O)C1 C1(OC)CN(C(C2C(C#N)C2(C)C)=O)CC1NC(=O)C(F)(F)c1cnccn1 c1(C(N(CC)CC2CCCN2C(C2CC23CC3)=O)=O)cccc2ncc(C)cc12 CC(C(=O)NCCN(C(=O)COCC(F)(F)F)C1CC1)=CC1CC1 N1(C(CC(C)O)=O)CCCC12CCN(C(c1cc(Cl)ccc1F)=O)C2 CC1CCCC(CNC(c2cc(CNC(=O)CSc3nc[nH]n3)cs2)=O)O1 C1(CC(N2CCC(N(C(C3CC=CC3)=O)CC)C2)=O)CC(C)(C)OC1=O c1(CCCC(=O)N2CCCC2Cn2cc(-c3ccns3)nn2)ccc(Cl)cc1 C(=O)(C(F)CC(CC)CC)NC(CCCC)CNC(c1cc(C)ncn1)=O CN=c1cc(C(N2CC(C(=O)NC(C)(C)C(=O)NC)C(C(F)(F)F)C2)=O)cc[nH]1 c1(NC(CCC(CC)OC)=O)nc2cc(Cl)c(Br)cc2n1C C1(C)(C(N2CC(O)(CNC(CN3CC(C)C3)=O)C2)=O)CCCCC1(F)F N1(C(=O)C#CC2CCCCO2)CCCC2(C1)CN(C(=O)C(F)(F)C1CC1)CCO2 N1(C(N2CCCC(c3c(NC(C)=O)c[nH]n3)C2)=O)CCCC2CCNCC12 C1(=CC(=O)NC2C3(CC(NC(c4cc(C)oc4C)=O)C3)C2)CN2CCC1CC2 c1(C(C)C)cccc(C(N2CC(C(N)=O)(CNC(C3CC(F)(F)C3)=O)C2)=O)n1 C1(C(=O)NCC2(NC(=O)C(c3ccc(F)cc3)=O)CC2)CCC2(CC1)CC2(F)F C1(N(C(=O)C(F)OC)CCCC)CCN(C(=O)Cn2cncn2)CC1 c1(OCCc2nn(C)c(-c3ccco3)n2)cc(Cl)cc(Br)c1 C1(N(C(C(COCC)NC(=O)C=CCO)=O)C)CCC(=O)N(C)C1 CC(C)CC(C(=O)NCC1CCN1C(C1CCC(C)(O)CC1)=O)NC(=O)C(C)(C)C C12(C(=O)NCC3C(NC(c4c(CC)ccs4)=O)C3)COC(CC3CC3)(C1)C2 c1(C(N(CC(CNC(c2n(CC)ccn2)=O)O)C)=O)ccc(Br)c(OC)c1 C1(NC(C2CC(CC)(CC)C2)=O)CC2CC(C1)N(C(c1ccc(Cl)c(O)c1)=O)C2 C=CCCCC(=O)NCCCCC(C)NC(c1ccc(C(F)F)s1)=O c1(N(CCCOC)C)nc(=N)[nH]c(=NC(C)CC2CCCO2)[nH]1 C1(C(N2C(C)(CO)CCC2)=O)CCN(C(=O)C2CCOC(=O)CC2)O1 c1(C2CCN(C(C(C)CC3CCC3)C(=O)NC3COC3)C2)ccc(Br)c(F)c1F CC1CCCC=C1C(=O)N1CC(O)CC1(C)C(N1CC(=O)NC(=O)C1C)=O c1(SC)ccc(Cl)cc1C(=O)NCC1(CNC(CNC(=O)OCC)=O)CCCC1 C1(NC(C2(C=C)CCC2)=O)CC2CC1N(C(C1CCC(F)(F)C1)=O)C2 N1(C(C(C)(C)C#N)=O)CCC2(CCCCC2NC(c2cccc(Cl)n2)=O)CC1 C1(F)(CNC(C2N(C)CCOC2)=O)CCN(C(=O)COCC2CCOC2)CC1 Cc1c(C(=O)NCC2CC(NC(=O)C(C3CCOCC3)C)C2)sc2ccccc12 c1(OC)ccc(OC(C)C(=O)N(CC(C)CNC(=O)CSCC(C)C)C)cc1 N1(C(c2ncc(F)cn2)=O)CC(C2CCCCN(C(c3cnco3)=O)C2)C1 CC1CN(C(C2CCCNS2(=O)=O)=O)CCN1C(C1CC2CC2C1)=O C1(C(=O)NCC2CC(CC)(CC)C2)C(CC)CCCN1C(=O)C1=CC(C)(C)C1 C1(NC(CC2ON=C(CC)C2)=O)CCC(O)CN(C(=O)C=C2CCC2)C1 C1(CNC(C2(CC)CC(C)(C)C2)=O)COC(C)(C)CN1C(C1CCC1(C)C)=O N1(C(c2c(C)nn[nH]2)=O)CC(NC(=O)CC(C)(C)N(C)C)C2CCCC12 CC(C)(CC(=O)N1CCCC2C1CCN2C(=O)CCCC1CC1)CC(F)(F)F C12(C(=O)NCc3ccco3)COCC1CN(Cc1nsc(-c3ccco3)n1)C2 N1(C(Cc2nc(C)c(C)[nH]2)=O)CCC(NC(=O)CCNC(=O)CC(C)C)C(F)C1 N1(CC)CCCC(ONC(=O)C(C)N(C(=O)C(C)N2CCCC2)C2CC2)C1 CC1CC(NC(c2cnccn2)=O)CCN1Cc1nccs1 C1(NC(=O)COC(F)F)CCC2CN(C(c3cnc4[nH]cncc3-4)=O)CCC2C1 N1(C(CC2C(NC(C(N)=O)=O)CCCC2)=O)CCC(O)CC12CC2 C1(CCOC)(NC(=O)CSc2ccccn2)CCN(C(C2(C#N)CC2)=O)C1 C1(C(N2C(CC)C(O)CC2)=O)CC(NC(=O)C(C)c2cc[nH]n2)C12CCC2 C(=O)(CS(=O)(=O)N(C)C)NCC1C(NC(C2CC(C(=O)OC)C2)=O)CCC1 C(=O)(C(F)(F)c1nccs1)NC1(CN(C)C(C2(C)CC2(F)F)=O)CC1 CC(C(F)C(=O)NCCOCCCNC(=O)COc1ccc(Cl)c(F)c1)C(F)(F)F C1(N(C(C(CC)OC)=O)C)CCCN(C(=O)C(F)(F)c2ccccc2)C1 C1(CCNC(C(C)OCCC=C)=O)(OC)CN(C(c2ncsc2C2CC2)=O)C1 N1(c2ncnc(NC3CCC(C)(NCC)C3)c2C)CCc2c(Cl)cccc2C1 C1(C(N(CC(C)(C)NC(C2CCS(=O)(=O)C2)=O)C)=O)CCc2cc(F)ccc2O1 N1(C(C2(CN(C)C)CC2)=O)CCC2CN(C(c3cc(Cl)ns3)=O)CCC2C1 C1(NC(c2c(CC)cco2)=O)CC2CC1CC2C(=O)N(C)CC1CCN(C)C1 c1(C(N2CCN(C)CC2CNC(=O)CC2CCC2)=O)ccc2[nH]ccc2c1F C(=O)(CCCS(N)(=O)=O)NCC1CC(C(C)(C)C)CN(C(C(COC)(C)C)=O)C1 C1(NC(CCCCCNC(C)=O)=O)CC2CC(C1)N(C(c1cnn(C)c1C)=O)C2 CCCCCCCC(=O)NCC(F)(C(=O)NC1CC1(C)CCOC)C(C)C N1(CC(=O)N(C)CC2N(C(C3C(C)C3)=O)CCC2)CCCNS1(=O)=O C1(CC)CN(C(C2CCN2C(=O)CSc2ccc(C)cc2)=O)CCO1 C1(NC(c2c(OC)cccc2F)=O)COC2(CCN(C(c3cc(O)cs3)=O)C2)C1 N1(C(C23CC(C#N)(C2)C3)=O)CC2CCC(NC(c3cnc4ccsc4c3)=O)(C2)C1 CCCC(C(=O)OC)C(=O)N1CC=CC1(C)C(=O)NCC1=NOC(C)C1 c1(CNC(COCCC(C)C)=O)cc(O)nc(CNC(C2COC(C)(C)C2)=O)n1 CC1(C)C(NC(c2ccn(C3CC3)n2)=O)CC1CNC(c1cc(F)cs1)=O C(=O)(C(CO)C(C)(C)C)NC1CC2CN(C(c3c(C)c(Cl)ccn3)=O)C1C2 c1(C(N(C)CCNC(=O)Cc2csc(C3CC3)n2)=O)ccn2cccc2c1 c1(C(N2C(CCCNC(c3cnn(CC)n3)=O)CCC2)=O)ccc(=O)n(CC)n1 C1(CC(=O)NCCCNC(C2CC2c2ccccc2Br)=O)CCCC12CC2 C(=O)(C1=CC2(CCOC2)C1)NCC1C2N(C(C3CC(SC)C3)=O)CC(CC2)C1 Cc1ccc(CN2CCC(C(=O)Nc3ccc(C#N)cc3F)C2)c2ccccc12 C1(CC(N2C(CNC(c3c(C)cc(CC)o3)=O)CC2)=O)COc2ccccc2O1 CC1=C(C)CC(C(N2CC(F)CC2CC(=O)NCCc2cccs2)=O)CC1 c1(C(=O)NCC2CC(F)(CNC(=O)CO)C2)cnc2n(c1=O)CCS2 c1(NCC2CN(C(c3n(CC)ncc3[N+](=O)[O-])=O)C2)cc(S(C)(=O)=O)ncn1 C1(CCNC(=O)CC2CC23CC3)CN(C(=O)CCC2CCC2)CCO1 C(=O)(C(N=[N+]=[N-])C(C)C)NC(CC#C)CC(=O)Nc1ccc(Cl)nc1 c1(C(=O)NCCCNC(c2c(C)ccnn2)=O)nc2ncc(CCO)cn2n1 C=CCC(C(=O)N1CCC1CNC(c1cn(CCN(C)C)nn1)=O)N(C)C CS(=O)(=O)C(CNC(c1cc2sccc2[nH]1)=O)CNC(C12CC(F)C1C2)=O Cc1ccc2c(c1)CC(C(N1CC=CC(NC(=O)CNC(=O)C(C)(C)C)C1)=O)S2 n1(CC(N2CCC(NC(Cc3nc(C)sc3Cl)=O)C2C)=O)nc(C)c(C)c1C N1(c2cc(OC(C)C)ncn2)CCC(NC(C2(F)CCOC2)=O)C2(CCC2)C1 CC1(CNC(=NCCOC(F)(F)F)NCC(F)F)CCC(F)(F)C1 c1(CC(=O)N(C(C)CCNC(C2CCC(=O)NC2=O)=O)C)ccc2c(c1)CCC2 c1(C(=O)OCC)nsc(=NCCCNC(=O)COC2CCCOC2)[nH]1 C1(NC(CN(CCC)C)=O)CCC(C)(C)CC1CNC(c1ncnn1CC)=O CC(C)C(CNC(=O)C(C)C1CCOC1)NC(c1cn(CCN(C)C)nn1)=O Cc1nc(S)sc1CC(=O)N(C(C)CCNC(=O)C(C)OC1CCCC1)C C(=O)(C(CN(C)C)c1ccccc1)NCCN(C(CC=CC=C)=O)CCOC C1(c2c(Br)c(C)n(C)n2)NC(=O)N(CC(=O)O)C2=C1C(=O)N(C)CC2 c1(NC2C(C(N3C(C)COCC3)=O)C2)ncnc2c1ccn2C S(=O)(=O)(c1ccc2c(c1)CC(C)(C)O2)NC(C1CCCCO1)C#C c1(CNC(C2(OC)CCC2)=O)nc(CNC(C2C=CCC2)=O)cc(O)n1 Cc1cc(N(CCCN(C(=O)CC(C)(C)O)C)C)nc(-c2cccs2)n1 N1(c2nc(CC)cc(CC)n2)CCOCC12COCCN(C(=O)CNC(=O)NC)C2 CC#CCCCC(=O)N1CCC(CC(C)NC(C2CCC2OCC)=O)CC1 C(CCCCCC(=O)N1CCCC1CCCNC(C1(C(C)C)CC1)=O)SC O=C1NCN(C(c2csc(Cl)c2)=O)CN1 O=C(CCCc1nc(C2CC2)no1)NCC1(CNC(C2OCCO2)=O)CCC1 C(=O)(C(CCc1ccccc1)NC(=O)OC(C)(C)C)N(C(CC#C)C)C c1(N(C)C(c2ccc(Cl)cc2)c2ccccc2Cl)nc(Cl)cc2c(Br)cccc12 C1(C(N2CCC(CNC(c3occc3CC)=O)C(C)C2)=O)(OC)CCCCCC1 c1(C(=O)NCC(CC(=O)N2CCC(OCC)C2=O)C2CC2)cn2ccccc2n1 C1(CC(=O)Nc2ccc(F)nc2)CC2(C1)CN(C(=O)C=CC1CCOCC1)C2 N1(C(C2(CC)CCCC2)=O)CC2CCCC2(CNC(c2ccc(F)cc2F)=O)C1 N1(C(c2c(C)scn2)=O)CC(NC(=O)CCC2CC2(Cl)Cl)C(N=[N+]=[N-])C1 c1(C(N2C3CCN(C(C(COC)C)=O)C3CC2)=O)c[nH]c2cc(Cl)ccc12 c1(C(N2CC(OCC)C(CNC(=O)CCC(N)=O)C2)=O)n[nH]c2c1NCCC2 C1(C(C)C)CN(C(=O)CC2CCC(O)C2)CCC1NC(=O)CCNC(N)=O c1(OC)ccccc1CC(=O)NC1CCC1NC(C1CCC(CC2CC2)CC1)=O C1(NC(c2cc(C3CCC3)no2)=O)CN(C(C2SCCCS2)=O)CCC1O N(C(=NCCF)NCC1(C)CC1(F)F)CC(C)C C1(C(=O)NC(C)C(N)=O)CC12CCN(C(C1CC1c1cncn1C)=O)CC2 N1(C(C(C2CCC2)OC)=O)CC2CC(NC(C3CCCN3C)=O)C2C1 C1(C(=O)NCC(CC(C)C)NC(=O)CCC=CBr)CCC2CC1C2(C)C N1(C(C2CC2Cl)=O)CCCCC1C1CCC1 c1(C(N2CCCCC(N(C(CCC#C)=O)C)C2)=O)cncc2ncn(C)c12 c12ncn(C)c1NC2=O.N1(CC)CCCC(CC(=O)NCC2CC(=O)N(C)C2)C1 C1(C)(CC)CC(NC(=O)C=Cc2cnc[nH]2)CN1C(=O)CC1CCSCC1 c1(OCC)cccc(C(=O)NC2COCC2NC(=O)C(C(C)C)n2cnnn2)c1 N1(C(C=CSC)=O)CC(CNC(C2(CO)CC(C)(C)C2)=O)C2(CCC2)C1 N1(C(C(CC)F)=O)CC2CN(C(c3ccc(C)cc3O)=O)CC2(C)C1 C=C1CN2C(=O)CCC2(C(=O)NCCOC2CN(C(=O)C(C)(C)C3CC3)C2)C1 CC(C)CCC(O)C(=O)N1CCC(CN(C(=O)CC2(N(C)C)COC2)C)C1 Cc1c(F)ccc(-c2ccccc2CN(C)Cc2ccccn2)c1O N1(C(c2n(C)ccn2)=O)CCCCC2(CCN(C(=O)Cn3cnccc3=O)C2)C1 C1(C)(NC(C)=O)CCN(C(C2CC(F)CN2C(C2CSCC(=O)N2)=O)=O)C1 c1(-c2n(-c3cccc(OCC)c3)nc(CC(C)OC)n2)cnc2[nH]cnc2c1 N1(C(CSC)=O)CCN(CCNC(c2nnsc2C2OCCO2)=O)CC1 C1(C(N2CC(F)(CNC(COC3(C)CCOCC3)=O)C2)=O)CCC2(CCC2)O1 CC(C)(CC(=O)N1CC2C(NC(c3csc(C4CC4)n3)=O)C2C1)C1CCCCC1 c1(NCC(COCC)C)cc(=NCc2ccc(SC)cc2F)[nH]c(COC)n1 c1(OCC=C)cccnc1C(N1CCCCC1CNC(=O)C(C(C)C)OC)=O CC=C=CCCN=C(NCCC1CCC1)NCC1CCS(=O)(=O)CC1 c1(C(=O)NCCCOCCNC(c2ccc(OC)nn2)=O)ccc(N)c(C)c1F N1(C(CC(CCC(=O)OC)C)=O)CCCC2(C1)CN(C(=O)CNC=O)CCO2 N1(C(C(F)OC)=O)CC(CNC(=O)CCC2CCCC2)C(n2ccnn2)C1 CC1(CNC(=O)CCn2ccnc2)CN(C(=O)CC2CCCSC2)CCO1 N1(C(Cc2c(C)n[nH]c2C)=O)CC(C)(C)OC2(CC3CCC2C3)C1 N1(C(C2CCN(C(C3C(C)CCO3)=O)C23CC3)=O)CC2(C)CC1CCO2 c1(C(N2CC(NC(CCS(N)(=O)=O)=O)C(O)C2)=O)ccc2c(c1)CCC2 c1(CC(N2CC(COCC)C2)=O)ccc(OC(C)C(=O)OC(C)C)cc1 C1(CCNC(C2CCSC2)=O)CCN(C(c2cc(-c3ccco3)[nH]n2)=O)CC1 C(c1cccnc1)=C(C(=O)NCC(C)NC(=O)C(C)(O)C1CC1)F C1(CNC(C=C(C)C)=O)COCCN(C(C2CCC(C)(O)CC2)=O)C1 c1(C(=O)NCCC2N(c3snc(C(=O)OC)n3)CCC2)ccc2nsnc2c1 Cc1cc(C(=O)NCC(C2CCCCC2)NC(C2COC(C)C2)=O)c[nH]1 C(C(=O)NCc1ccc(C(=O)NCCc2cocn2)s1)(C(C)C)SCC c1(CC(=O)NC(CNC(C(C=CC)O)=O)C(C)C)ccc(Cl)cn1 c1(OC)ccccc1OC(C)CNC(N1CCN(C2(CO)CC(O)C2)CC1)=O C(=O)(CC(=O)N(CC)CC1(F)CN(C(=O)C(O)Cc2cnc[nH]2)C1)NCC#C N1(C(C2(F)CCN(C(CCN=[N+]=[N-])=O)C2)=O)CCN2CC(F)CC2C1 C1(CC(N2CCCC(CN3CCC(N)CC3)C2)=O)CC2(CCOCC2)C1 N1(C(CC)=O)CCCCC1CCN(C)C(c1cn(C)nc1Cl)=O C(c1cnccc1C)=CC(=O)NCC1(CNC(CCC(C)SC)=O)CCCC1 CCC(CC)CC(F)C(=O)NC1CCN(C(=O)CC2CCC(=O)C2C)CC(O)C1 S(=O)(=O)(c1cn(C)cn1)NCC(N1CCC(N(C(C(F)=C(C)C)=O)C)C(C)C1)=O c1(CN2CC3(C(C(N4CCn5nccc5C4)=O)C3)C2)cc2cc(F)ccc2o1 C1(CCSC)CCN(Cc2cnn3c2CN(C(=O)C(N)=O)CC3)CCC1(F)F C1(NC(Cn2ncc(C#C)c2)=O)(CNC(=O)COCC2CC2)CCC(F)(F)CC1 C1(NC(C2CCC(=C)CC2)=O)COCCN(C(c2cc(C(N)=O)[nH]n2)=O)C1 c1(CCC)ccc(CSCC(=O)NCC(C)(C)NC(C2CCC(O)C2)=O)cc1 C=CCC(C(=O)Nc1ccc(CC)cc1)NC(=O)C(=Cc1cn[nH]c1)C N1(C(C2N(C(N)=O)CCCC2)=O)CCOCC(NC(c2ccc(O)cc2Cl)=O)C1 C1(C(N2C(C3(NC(c4c(C#C)c[nH]n4)=O)CC3)CCC2)=O)CC2CCC(C1)N2C Cc1cc(C)c(C(=O)NCC2CC(NC(C3(C)CCC(=O)NC3)=O)C2)cn1 C1(O)(CN(C(=O)C(c2ccccc2)O)C)CCN(C(=O)CN(C2CCCC2)C)C1 c1(C(=O)NCCC(C)NC(=O)Cc2ccc(F)cn2)ccc(O)cc1F CC1(C)CN(Cc2ccc(O)c(Cl)c2)CCC1NC(c1ccncc1O)=O CC(C)(CO)CCNC(=O)C(CCC1CC1)NC(=O)CCc1cnccn1 Cn1cc(C(=O)NC2CN(C(c3cnn(CCO)c3)=O)C3CC23)c(C(F)F)n1 C(=O)(C1=CC(C)(C)C1)NCCC(CNC(c1ncc(OC)nc1)=O)O C1(CCC(=O)NC2(C3N(C(CCC4C(C)(C)C4)=O)CCC3)CC2)CCCCCC1 c1(CNC(C2CC(C)CN2C(=O)Cc2ccc(O)cc2)=O)ccc2c(c1)OCO2 C1(O)(CC(=O)NCC2N(C(CCNC(C)=O)=O)CCC2C)CCCN(C)C1 CC1CN(C(=O)CC2(n3cccn3)CC2)C(C)CN1C(=O)CC(C)C(F)(F)F N1(C(c2ccc(C(C)=O)o2)=O)CCC(CNC(=O)C(C)OCC2CC2)C(F)(F)C1 N1(C(=O)NCCc2nc(C)c(-c3ccccc3)s2)CCC(O)(C(F)(F)F)C(O)C1 N#Cc1ccsc1C(=O)NCC1CCOC1C(N1CCCC(CF)C1)=O c1(SC)cc(C(=O)Nc2c(Cl)cc(C)cc2Cl)cc(SC)c1 Cc1ccc(C(N2CC(C(=O)NCC3CC(C)(C)CO3)C(C(C)C)C2)=O)cc1 c1(C(N(C(C)C(=O)NC(C)(C)COC(F)F)C)=O)ccc2[nH]nc(Cl)c2c1 N1(C(CCCOCCC)=O)CCC(C)(C(=O)NCc2coc(C)c2)C1 C=CCCC(=O)NCC1CC(C(=O)NC2CCN(CC(=O)OCC)C2)C1 CCCCS(=O)(=O)CC(=O)NCC(O)CNC(c1cnc2[nH]nnc2c1)=O c1(C(=O)NCC(CC=C)NC(C2CC(CC3CC3)C2)=O)cc(N)cc([N+](=O)[O-])c1 c1(C(N2CCC(NC(C(C(=O)OCC)F)=O)CC2C)=O)c[nH]c2cccc(C)c12 C1(CC(=O)NCC(CCCC)O)CN(C(=O)CC=C(C)C)CC12CC2 N1(C(C=CC(CC)=CC)=O)CC(NC(c2c[nH]nc2CC)=O)CC12CCOC2 C1(NC(C(Br)=C(C)C)=O)CCC2CN(C(=O)CN3CCS(=O)(=O)CC3)CCC2C1 Cc1ccc(C(=O)NCC(C)(C2CC2)NC(=O)C(F)(F)c2cncs2)c(CO)c1 c1(C(=O)NCC(CC)NC(C2(CCF)CCOCC2)=O)cc(C)oc1C C(=O)(C(C)(C)CC(F)F)N1CCC(CNC(CNC(c2cc(C)nn2C)=O)=O)C1 N1(C(C(F)=CCC)=O)CC(NC(c2cc(C(N)=O)cs2)=O)CCC1C C1(NC(=O)COCCO)CCN(C(C2CC3(CCOCC3)CO2)=O)C12CCCC2 c1(OC)ccc(C(C)=CC(=O)NCCN(C2CCCC2)C(=O)COC)cc1 C1(NC(CCC(C)SC)=O)COCCN(C(=O)CSc2ccc(O)cc2)C1 c1(C(=O)NC(COCC)C(N2CCC(CC3CC3)CC2)=O)scc(C)c1OC c1(C(=O)NC23CCN(C(Cc4ccn(C)n4)=O)CC2C3)ccc2nc(S)oc2c1 C1(C)(C(=O)NCC(Cn2cc(-c3ccnn3C(C)C)nn2)OC)CCCC1O c1(C(=O)NCCC(C)NC(=O)C(C(C)(C)C)n2ccnn2)cc2ccncc2[nH]1 C(CNC(c1cc(C2(C)COC2)no1)=O)(C(C)C)NC(C(C)OCCC#C)=O C(=O)(C(C(C)C1CCCC1)N(C(c1ccc(Cl)cc1)CN(C)C)C)NC(CC)C Cc1ccnc(O)c1C(N1CC(c2ccccc2)CCC1=O)=O Cn1ccc2ccnc(C(=O)NC(CNC(=O)C#CC3(C)COC3)C(C)(C)C)c12 N1(C(C(F)=CCC)=O)CC2CCCC(NC(=O)C=CC(=O)N(C)C)(C2)C1 O=S1(=O)c2ccc(Br)cc2NC2CCCN1C2.C1(CCOC(F)F)CC1(Cl)Cl C(=O)(CC(O)CNC(c1nccn1CC)=O)NCCN(C(CC)C)C CC(C)C(O)CC(=O)N1CC2(CCN2C(c2ccoc2C(F)(F)F)=O)C1 c1(CC)ncccc1C(=O)NC1CCCN(C(=O)CC2C=CCCC2)C1 c1(OCC(N2CCCC(CCNC(C(CCC)O)=O)C2)=O)ccc(Cl)cc1Cl c1(NC)cnccc1C(=O)NC1CC(CNC(=O)CCCc2ccsc2)C1 N1(CC(=O)NCCC2(O)CCCN(C(CC(C)C)=O)C2)CCCCCCC1=O CC(C)C(F)C(=O)N1CCCC1(C)CNC(=O)C=Cc1cc[nH]n1 CC1CCC(C)(C(=O)NCCOCCOCCCNC(c2nonc2N)=O)C1 C1(C(=O)NCC(C)N(C(c2nc(C)sc2)=O)C)Cc2nn(C)cc2C(=O)N1 CC1CN(C(c2cc(C(N)=O)c[nH]2)=O)C1C(=O)N(C)CCC1CN(C)C1 CC1CCN(C(C2(Cc3ccc(O)cc3)CC2)=O)CCN1C(C1CC1F)=O CN1C(=O)N(C2CCCC2)C(=O)C1c1ccc(C(F)(F)F)cc1 C1(C(=O)OC)CC(c2nc(C3CC3)no2)N(C(=O)C(c2ccccc2)SC)C1 Cc1c(C(=O)NCC2CCCCN(C)C2)cccc1-n1cnnc1 C1(C)(CNC(CC(=C)C)=O)CCN(C(C2(NC(C)=O)CCCC2)=O)C1 C=CCC(C)(CNC(=O)C(C1(C)CC1)NC(=O)C(CO)OC)CO N1(C(C2CC(SC)C2)=O)CC(NC(=O)C(n2ccnc2C)C)C(F)C1 N1(C(c2cccc(OC)c2)C(=O)NC2(C)CC2)CC2CC3CC(C2)CC1C3 CCC(C)(O)Cc1cn(CC2CCCN2C(=O)C(C)(F)c2ccon2)nn1 N1(C(C(CC)NC2CN(C(=O)OC(C)(C)C)CCO2)=O)CCC(OC)CC1 N1(C(c2cncc(SC)c2)=O)CCCC(C)(CNC(C2CCC(=O)NC2)=O)C1 c1(C(=O)NCC2C(NC(Cc3n(C)cnc3)=O)CC2)cccc2c[nH]nc12 N1(C(=O)COc2ccc(Cl)c(Br)c2)CC2(CC=CC2)C1c1ccccc1 C1(C(=O)NCC2CN3CCC2C3)CN(C(=O)C2=COCC2)CC1C1CC1 c1(OC)ccc(CCC(N2CCC(NC(c3ncccc3OC)=O)C2C)=O)cn1 C(=O)(C1CCCc2nc[nH]c21)NCC1N(C(Cc2cn(CC)nc2)=O)CC(O)C1 N1(C(C(C)n2cccn2)=O)CCC(C)(C)C1CC(N1CCC2CCCC12)=O C1(C(C)NC(C(SC)SC)=O)CCCN(C(C2(CF)CCOCC2)=O)C1 c1(C(=O)NCC(C)NC(C2CC(SC)C2)=O)cccc(Br)c1 C1(NC(C(C)P(C)(C)=O)=O)C(C)(C)CN(C(C2(C)CC=CCC2)=O)CC1(C)C CC1CN(C(c2[nH]nnc2-c2ccnn2C)=O)CCC1NC(c1cc(Cl)c[nH]1)=O CCC(C)CC(C)C(=O)N1CC(F)(CNC(C2(CC3CCC3)CC2)=O)C1 c1(OC)cccc(S(=O)(=O)NCCCN(c2ccc(Cl)c(Cl)c2)C)n1 CC(=O)CCCC(=O)NCC1CCCN(C(=O)C(c2cccnc2)C)CC1 C(C1c2ccsc2CCN1C(c1sccc1F)=O)NC(C(C)(C)C1CC1)=O C(=O)(C1=NOC(C)(C)C1)NC1C=CC(C(=O)Nc2cc(C)c(C)nc2)C1 c1(C(=O)NCC2OCC(CNC(C(C3CC3)OCC)=O)C2)nnc2n1CCOC2 C12(C(=O)NCCCC(=O)NC)CC(CN(C(=O)CCC(C)CN(C)C)C1)C2 N1(C(C)=O)CC(O)CC1C(=O)NCC(C)CNC(c1cc(-c2ccns2)on1)=O N1(C(CSCCCC)=O)Cc2[nH]nc(C(N3CC(S(C)(=O)=O)C3)=O)c2C1 Cc1cc(C(=O)C(=O)NCC2CCCN(C(=O)CSCCC(C)C)C2)ccc1F c1(C(=O)NCC(CC)N(C(=O)C(C)C2CCC2)C)cccc2c1ccn2C c1(C(=O)NCCN(CC(C)O)C(=O)CC2(C)CCC2)cnc(N)c(Cl)c1 N1(C(C)=O)CCC2(CCCC2NC(=O)NC2CCC(C3CCC3)CC2)CC1 n1(CC)nc(C)c(C(=O)NC2CN(C(=O)C(C)(O)C(C)C)CC2C(F)(F)F)c1C C1(C(=O)NCC(CC)N(C)C)CCC(C)(C)N(C(C2(OC)CCC(C)C2)=O)C1 CC1(C)COCC(CC(=O)NCC2CCCN2C(C2(O)COC2)=O)O1 N#CC1(C(N2CC3CC3(NC(=O)C=Cc3cccs3)C2)=O)CCOCC1 CC1CN(C(c2ccccc2CC(C)(C)C)=O)CC1NC(=O)C=CCN(C)C n1(CC)nc(C(=O)NCCC2CC(NC(C3(C)CC3F)=O)C2)c(C)n1 c1(CNC(c2c(CCNC(c3n(CC)nnc3)=O)n[nH]c2)=O)cc(O)ccc1F N1(C(C(C2CC2)NC(C(C)N(C)C)=O)=O)CC(=O)N2CCCC2C1 C(CCCCC(=O)NCC(C)(C)OCCNC(C1CCCCS1(=O)=O)=O)=CC CCC(C(=O)NCCC1CCCN1C(=O)C(c1cccnc1)C)NC(N)=O c1(C(=O)NCC(C)(C2CC2)NC(C2(CC)CCCCC2)=O)cc(C)n(C)c1C N1(C(CC)=O)CCCC(C(N2CCN(C(=O)N(CC(C)C)C)CC2)=O)C1 C1(NC(c2cc(C)oc2C)=O)C2CC(O)C1N(C(c1cnc(C3CC3)o1)=O)C2 N1(C(C(CC2CC2)OC)=O)CC(C)C(C)(CNC(C2(C)SCCCS2)=O)C1 C1(NC(C(Cc2cnn(C)c2O)NC(C2CN(C)C2)=O)=O)CCn2ccnc2C1 C(c1ccco1)=CC(=O)NCC1C=CCN1C(=O)COCC(F)F C(=O)(CCCS(C)(=O)=O)NCC(CNC(=O)C=CC(C)(C)SC)OC c1(-c2nc(CCCC)nn2CCN2CCCN(C)C(=O)C2)ncc2cc(Cl)ccn12 C1(NC(C2C(C)C2)=O)CCCCC1.C1(C)C(=O)N(CCOCCO)CCN1 C1(NC(C(C=C)(C)C)=O)CC2CC(C1)N(C(=O)Cc1ccc(Cl)nc1C)C2 C=CC1(CC(=O)NCCN(CC(C)O)C(C2CCC(N(C)C)C2)=O)CCC1 c1(COC)ccc(C(=O)NC(CNC(=O)COCc2ncnn2C)CO)s1 c1(C(C(=O)NC(C)CC)N(CC#CC)C)cc(-c2ccccc2)on1 CCC(CC)CCCC(=O)NC1(C(=O)NOCC(=O)OCC)CCSC1 C1(NC(C2(CCCC)CC2)=O)CC(C)(CNC(=O)Cc2cnc(C)s2)C1 C1(NC(CSCCOC)=O)COC2(C1)CN(C(c1scnc1Cl)=O)C2 c1(C(=O)NC2CCN(C(c3c(COC)nn[nH]3)=O)C2)ccc(C(F)(F)F)nc1 C(c1cccc(C#N)c1)=CC(=O)NCCC(C)NC(CCc1c(C)cccn1)=O C1(CCNC(C(C)O)=O)CCN(C(c2cnccc2C2OCCO2)=O)CC1(F)F c1(C(=O)OC)ccc2cccc(CNC(c3ccc(N(C)C)cc3)=O)c2c1 Cc1[nH]nc(C(N2CC3CC2C3C(=O)N(CC(C)(CO)N(C)C)C)=O)c1O N1(CC(c2c(C)sc3ccccc23)C)C(C)CC2CN(CC)CC12 c1(CC(=O)N(C2CN(C(=O)CSC(F)(F)F)C2)C)cnc[nH]1 c1(CCC(=O)NC2C(NC(CSC)=O)CCCC2)ccc2c(c1)OCO2 C1(CC)(NC(=O)C=C2CCC(C)CC2)CCCN(C(C2CCCC2F)=O)C1 c1(N2CCC(=C)C2)nc(N2CC(C(N)=O)CC(C)C2)nc2c1CCCC2 C1(C(=O)NCCCCNC(=O)C(F)CC2CCC2)CCC2C(C1)C2(F)F c1(OC)ccc(F)c(C(=O)NCC2CCCCCN2C(c2ccc(OC)o2)=O)n1 c1(C2C(C(=O)NC3(OC)CCNC3)CC2)ccc2c(c1)OCO2 N=c1cc[nH]c(C(N2CCN(C(=O)C(F)n3cccn3)CC2)=O)n1.C(=O)CNC C1(N(C(=O)CC2(C(F)F)CC2)CC)CCN(C(=O)CN(C2CC2)CC)C1 C#Cc1ccc(CC(N)C(=O)NC2CC(NC(N)=O)C2)cc1 C1(NC(=O)CC(C2CC2)C2CC2)COC2CN(C(C3CC(F)(F)C3)=O)CC12 CCCCCC(O)CC(=O)N1CC=C(C(N2CCNC(=O)CC2C)=O)C1 C(=O)(CS(=O)(=O)Cc1ccccn1)N(C)CC1(NC(c2cn(C)cn2)=O)CC1 c1(-c2ccc(SCCCC)o2)nc(C(F)F)nn1CCc1ccccc1 C1(CN(C)CCc2nc(=O)o[nH]2)CCN(C(C2CC3CCC2C3)=O)CC1 C(CCNC(c1ccc[nH]1)=O)(C(=O)NCCn1cnnc1)OC c1(C(C)(C)C)cc2n(n1)CCN(C(C1CCN(CC3CCCC3)C1)=O)C2 c1(OC)c(C)csc1C(=O)NCC1CCC(NC(=O)CCn2c(C)ccc2C)C1 C1(C(N2CCN(C(=O)CC34CCCC3C4)CC2)=O)CC(=C(F)F)C1 C(=O)(CCCC(C)O)Nc1cccc(NC(C(C)NC(=O)NC)=O)c1 c1(C(N(CC(=O)NC(c2ncc(C)[nH]2)CC)C2CC2)=O)cn(C)nn1 O=C(CCC(F)(F)F)NC1CC2CC1CN2C(C1(c2ccccc2)CCC1)=O N1(C(C=CC)=O)CC(C(=O)NCC2OCCC2(C)C)CC12CCC2 c1(C(C)=O)ccc2c(c1)CCC(C(=O)NC1COC(C)(C)O1)C2.c12cccn1c2=O C1(CNC(c2nnn(CC)c2C)=O)COC(C)(C)CN1C(C1CC1CC(C)C)=O Cc1cc(Cl)cc(N)c1C(=O)NC(CCN(C(=O)C=Cc1cnc[nH]1)C)C(C)C C=CC(CC)CC(=O)N(CCCOCCN(C)C(C1CCCCS1)=O)C N1(C(C=COCC)=O)CCCCC1CNc1ncc(C(=O)OC)cn1 c1(COC(CCCNC(=O)NC2CCOC2)=O)cc(F)cc([N+](=O)[O-])c1 C(=O)(CCC(C)(C)NC(=O)C1=C(Cl)CC1)NC12C(CN(C)C1)C2 c1(C(N2CC3CN(C(Cc4c(C#N)cccc4)=O)C3C2)=O)ccc2ocnc2c1 C=C(C)CC(C(=O)N1CCC(n2cc(-c3ccccc3CO)nn2)CC1)OC c1(C(=O)NC2C3CN(C(CN4C(=O)CN(C)C4=O)=O)CC32)cc(O)cc(N)c1Cl c1(CC(=O)NC(C(C)NC(C2CCS(=O)(=O)C2)=O)CO)ccc2c(c1)CCOC2 C1(F)(C(=O)NCCCCCCO)CCN(Cc2ccc(Cl)cc2)CC1 C(C(=O)NCc1cnn(C)c1C(=O)NCC(C)(COC)CC)(C(C)C)OCC c1(OC)ncc(Br)cc1NC1CCN(C(=O)CCC(=O)NC)CC1 C(=O)(C1CCCc2nc[nH]c21)NCC1(C)CC(NC(c2cn3ccsc3n2)=O)C1 C12(CNC(=O)C=CCO)CCCC1N(C(C1CC1c1ccoc1)=O)CCC2 N1(C(C(CCCC)O)=O)CCCC2(CNC(c3cnc(Cl)cc3Cl)=O)CCCC12 c1(-n2cc(CN3C(C(=O)O)C=CC3)nn2)ccccc1NC(c1nc(Cl)cs1)=O N1(C(CCC2CC(OC)C2)=O)CCC(C2CC2)C1C(=O)NCC1CCC(C)(C)C1 N1(C(c2cnns2)=O)CCC2(CC1)CN(C(C1CCC=CCCC1)=O)C2 c1(C(=O)NC2C(O)CCN(C(c3c(C)ccc(N)c3)=O)C2)n[nH]c2c1CCSC2 C1(C(=O)NCCC2CCN(C(c3nc(C)n(C)c3C)=O)C2)CN(CP(C)(C)=O)C1 N1(C(C(CC)OC)=O)CC23CCCC2(C1)CN(C(C1CCC2(CCOC2)O1)=O)C3 c1(C(N2CCC(OC)(CNC(=O)CC3CCCCO3)C2)=O)ccc(C)c(C)c1Cl c1(CC)ccc(CCC(N2CCC(CNC(=O)C(F)(F)CC3CC3)CC2)=O)cc1 C(C(C)(C)C(=O)NCCc1cc(C(=O)N(C)Cc2cscn2)no1)SC c1(NC(C(CC)C)=O)cccc(C(N2CCCC(c3ccccc3)C2)=O)c1 O=C(CC1=CCCC1)NCC(CNC(C12CCC(CO)(CC1)C2)=O)CO N1(C(C=CC(CC)C)=O)CCC(CCOC)(NC(=O)Cc2sccc2C)C1 C(=O)(CCCC(=O)C1CC1)N1CCC(O)(C(C)CNC(=O)Cc2ccn(C)n2)C1 C1(NC(c2cc(C)sc2C)=O)CCCC2CN(C(C3CCC(C(N)=O)O3)=O)CC12 N1(C(C2(C)CCOCC2)=O)CCCCC(C(=O)NCC2(F)CC(CO)C2)C1 CCCC(C)(C)CC(=O)NC1COC2C(NC(=O)C(F)(F)CC)COC12 C(=O)(CCC1=NNC(=O)CC1)NCC1CCC(CNC(C2C(C(C)C)C2)=O)CC1 c1(C(N2CCN(C(CCC=C(C)C)=O)CC2C(F)F)=O)ccn2ccnc2n1 C1(NC(C(C)N(C(=O)C(F)C(C)(C)O)C)=O)CN(C)CC1(F)F Cc1cccc2cc(C(N3CCCN(C(c4cc(Cl)cn4C)=O)CC3)=O)nn12 Cc1nc(C(=O)NC2CC(C)N(C(=O)CCc3cnc[nH]3)C2)c2ccccn12 C(=O)(C(C)C(C)(C)C)NCC(CCNC(C(C)(C)OC(C)=O)=O)O c1(NC(C2N(C(COC)=O)CC(O)C2)=O)c(F)ccc(Br)c1F c1(C(N2C(C)(CCC(=O)NCC(F)C3CCC3)CCC2)=O)c[nH]c2ncccc12 C(C(C)(C)C#CC(=O)NC1CCC12CCCC2)NC(CC1(CC)CCC1)=O N1(C(C(c2n(C)cnc2)O)=O)CC2(CC(NC(=O)CC3CCC(O)CC3)CO2)C1 c1(COCC(CN(CCOCCN(c2ncc[nH]2)C)CC)O)ccc(F)cc1 C1(NC(C2CCN(C3CC3)CC2)=O)CC2(C1)CN(C(=O)CC1(O)CCOC1)C2 N1(C(CC2(OC)CN(C(C3C=CCCC3)=O)C2)=O)CCC(C(N)=O)CC1 c1(CNCC2CCCCN2C(C2C(C(N)=O)C2)=O)ccc(Cl)cc1Br C1(C)(C(=O)NCCC(C)NC(=O)CCNC(=O)C=CCl)CCNC(=O)C1 C1(CNC(C=CC(C)(C)NC(c2c(C)cco2)=O)=O)(CO)CC2CC2C1 C1(NC(CCC=C)=O)CN(C(c2cc(C)c(C)nn2)=O)C(CC)(CC)C1 C(=O)(C(CCC1CC1)NC(=O)Cc1cn(C)cn1)NCC1CC(C(=O)OC)C1 CC(C)C(C)C(=O)NCCC1CC(NC(=O)C(C(C)C)c2cccc(Cl)c2)C1 C1(NC(c2n(C)c(O)nc2)=O)C2CC(O)C1N(C(c1ccc(O)nc1Cl)=O)C2 CC1=NOC(C)(CNC(=O)C#CCNC(C2CCCN2C(C)C)=O)C1 N1(C(c2[nH]cc(C#N)c2)=O)CCC2CCC12CNC(=O)CCN1CCCC1=O N1(c2nccc(C)n2)CCCC(C)(CNC(c2ccc(C(N)=O)s2)=O)C1 N1(C(Cc2nc(C)sc2Cl)=O)CCC(CNC(=O)C(=O)N(C)C)C(C)C1 CCC(CC(=O)NC(C1CCCCC1)CNC(c1cnc(Cl)s1)=O)SC Cc1cccc(F)c1C(=O)NCC1CC(NC(C2OCCN(C)C2=O)=O)CCO1 CC(C(C)(O)C(=O)NC1CC(NC(c2cc(O)cc(Cl)c2)=O)C1)c1ccccc1 CCC(C)(CCC(C)C)C(=O)N1CCC2CN(C(c3cccnc3S)=O)CC2C1 O=S(=O)(c1ccncc1Br)NC1CC2(CCC2)C1O c1(OC)ccc(C(=O)NC2CCN(Cc3nc(C)cs3)C2)cc1 N1(C(C2CCN(CC)C2)=O)CCN(C(c2cc(OC)nc(C)c2)=O)CC1CSC C1(C)(CNC(C(C)(F)F)=O)CN(C(C2CCCOCC2)=O)C(C)(C)C1 C(CC1CC1)(C(=O)N1CC(O)(C(C)NC(=O)CCCn2ccnn2)C1)OC C(CC(C)C)(C(=O)N1CCCCCO1)ONC(c1ccc(C)c(Cl)c1)=O N1(C(c2[nH]cc(C)c2)=O)CCC(NC(C2(c3ccccc3)CCCO2)=O)C1(C)C C1(C(=O)NC2CCCN(C(C)C)C2)(COC)C=CCN1C(c1csnc1Cl)=O C12(C(N(CCC)CCN(C)C)=O)CCN(C(c3cc(C#N)cs3)=O)CCC1C2 C12(CNC(c3c(C#N)csc3)=O)CCC1CN(C(=O)CC1CCC13CCC3)C2 CCCC(C)(O)CC(=O)NC(C1CCN(C(c2c(Cl)cncc2Cl)=O)CC1)C c1(C(=O)NCC2(NC(c3c(C)ocn3)=O)CCOCC2)n[nH]c2c1CCCCC2 CCC(C(=O)NCC(C)NC(=O)C(C)(O)c1ccccn1)OC c1(C(C)=O)ccc(C(N2CCN(C(C3CCC(C)O3)=O)CC2)=O)cc1 C1(NC(COCCC)=O)C=CC(CNC(=O)Cn2cnnn2)C1 C12(C(=O)OCc3cccc(OCCC#C)c3)CCN(C(=O)OC(C)(C)C)CC1C2 C1(C2(O)CCOC2)(C(=O)NCC2CCN(C(c3c(C)[nH]nc3CO)=O)CC2)CC1 C=C(C)C(C)(C)C(=O)N1CCC(O)C(NC(c2ccc(C(C)(C)C)[nH]2)=O)C1 c1(C(=O)NC2CCC(NC(CNS(N)(=O)=O)=O)C2)coc2c1CS(=O)(=O)C2 CCC1C(=O)Nc2ccc(C(=O)NCC(C3CC3)NC(=O)C3=CCCS3)cc21 N1(C(CCCC)=O)C2CCC1C1CC1(NC(C1CCc3nncn3CC1)=O)C2 c1(C(N(C2CCN(C(C3(CC)CCCC3)=O)C2)CC)=O)ccc(CO)cc1 c1(C(=O)NC2C(NC(=O)C=CC3CCCO3)CCCCC2)cc2cccnc2s1 CCC(C)C(=O)C(=O)N1CCN(C(c2ccc(CO)nc2)=O)C(C)C1 C(C(CNC(C1(Cc2ccc(F)cc2)CCC1)=O)C(F)(F)F)NC(=O)CCCF N1(C(C(C)(C2CC2)OC)=O)CC2CCCCC2(CN=c2nn[nH]n2C)C1 c1(C2C(C(N(CCCCN(C)C(c3cc(F)n[nH]3)=O)C)=O)C2)cc(F)ccc1F C(COC)(CCCC)(c1n(CCOC)nnn1)NCCOC1CCCCC1 c1(CCCC)nn(C)c(-c2nc(CCC)nn2CCOc2ccccc2)c1Cl N=c1ncn(CCC(N2CC(F)(C(=O)NCC3CC(=C4CC4)C3)C2)=O)[nH]1 C1(C)(C(=O)NCC(C(C)C)NC(C2CCCN2C(=O)C2CC2)=O)CCC(F)(F)CC1 N1(C(c2cc(OCC)no2)=O)CCN(C(=O)CN(C)C(=O)C2CC2)C(C)C1 N1(C(C=CC(C)(C)SC)=O)CC(C)CN(C(=O)Cc2csc(N)n2)CC1C C1(CC(C)NC(C2CCCCS2)=O)CCN(C(c2cncn2C)=O)CC1 C(C1CCC(C)CC1)=C(C)C(N1CC(NC(=O)COCCCN(C)C)C(F)C1)=O C(CN=C(NCC12CCC(CC1)C2(C)C)N1CCC(OC)C1)N(C(=O)OCC)C N1(C(c2ccc(C(C)(C)C)cc2)C(=O)NC(C)C)CCCC(C)(O)C1 c1(C(N(CCCNC(=O)CC2CC2(Cl)Cl)CC)=O)ccncc1-n1cccn1 Cc1cc(F)cc(C)c1C(=O)NC1CC(CNC(=O)CC2(N(C)C)CCC2)C1 N1(C(c2ccc(CC)cn2)=O)CCC(CNC(c2cc(C)sc2C)=O)C1(C)C N1(C(c2c(NC(c3c(C#C)cccc3)=O)ccs2)=O)CC2CN(C)CC2C1 O=C(C1=CC2C=CC1C2)NCC1CCN(C(=O)CC2CCCO2)C12CCC2 N1(C(CCCC#N)=O)CCC2(CC1)OCCCC2NC(c1ncc(Cl)cc1F)=O C(CN=c1ccc2c([nH]1)CCCC2=O)(N(C(C(CCC)CC(C)C)=O)C)C1CC1 C1(O)(CNC(C2(C)CCC2)=O)CCCN(C(=O)CCNC(=O)C=CCl)C1 N1(C(c2c(CC)nn[nH]2)=O)Cc2n[nH]cc2C1C(=O)NCC1(CCO)CC1 N1(C(C2(OC)CCN(C(=O)CCCC(C)=O)C2)=O)Cc2cncnc2C1 Cn1cc(-c2oncc2C(=O)NCCC2CC(NC(=O)OC(C)(C)C)C2)cn1 C1(CNC(c2ccccc2)=O)(CO)CC(F)(F)C1.C1CCC(=O)N2CC=CC2CO1 c1(CN(C(C(CCC)O)=O)C)cnn2c1CN(C(C1CCCS1(=O)=O)=O)CC2 Cc1c(C(N2CCCC2CN(C(=O)C=C2CCCC2)C)=O)[nH]c2c(C)cccc12 CC1=C(C(=O)N2CC(NC(C3CC(C)CCO3)=O)C(F)C2)C(=O)OC1(C)C C1(NC(C(c2ccccc2)OC(C)C)=O)CCCC1NC(=O)Cc1cocn1 C1(C(C)C(=O)NCC2CCCN2C(=O)CNC(c2ccoc2)=O)CCCCCC1 Cc1nc(C2CC2)nc(O)c1C(=O)NCCOCCNC(C1CC(C)(F)C1)=O c1(COC)nc(NCc2cccc(N)c2F)cc(=NC2CCCc3occc32)[nH]1 c1(C(=O)NC2CCC(NC(C3(CCC)CC3)=O)C2)nnn(-c2ccccc2)c1C c1(C(=O)NC(C(C)NC(c2c(C)cc(F)c(Cl)c2)=O)C)cccc2c1CCC2=O CC1COCC(C(N2CC(C(=O)NC(C)(C)C(C)(C)O)C(C)C2)=O)O1 c1(CC)nnsc1C(=O)NCC(C(=O)NC(Cc1ccco1)CO)N(C)C C(=O)(N=c1cc[nH]cc1O)c1nccc(Cc2c(-c3n(CC)ncc3)csc2)c1 N1(C(c2cc(F)c[nH]2)=O)CCC(C2CCN(C(c3ccc(F)cc3Br)=O)C2)C1 c1(CC)ccc(C)c(NC(=O)CC2CC(NC(=O)C=CC(=O)N(C)C)C2(C)C)c1 C1(CNC(c2c(C)ccnc2)=O)C2CCC1CN(C(c1cc(Cl)ccc1C)=O)C2 c1(C(=O)NC2CC(NC(C34OC(C)C(CC3)CC4)=O)C2)cc([N+](=O)[O-])ccc1N c1(N2C(C)(C)C(CNC(=O)C(F)CC3CC3)CC2)nc2cccnc2s1 C(=O)(C(C)(CC)C(N)=O)N(CC(CO)(CO)NC(c1[nH]cc(CC)c1)=O)C c1(-c2c(C)nn(C)c2C)ccc2c(c1C(N1CCCC(C#N)C1)=O)OCO2 C1(C(=O)NC2CC(O)(CNC(C3(C=C)CCC3)=O)C2)CC2CC1CC2O c1(NC(=O)CN2CCOCC2)ncc2scc(Br)c2n1.N12CCCC(NC)(C1)C2 c1(CC(=O)NC(CC=C)CNC(c2ccn(C3CCC3)n2)=O)ccc(F)cc1Cl c1(C(=O)NC(CNC(C(C=C)(C)CC)=O)(CC)CC)ccc2snnc2c1 N1(C(COC2(C#C)COC2)=O)CCCCCC1C(=O)NCCN(C(C)C)CC CCC(C(=O)N1CC(O)(CCc2cn(-c3cccc(F)c3OC)nn2)C1)C(C)O c1(CN(C(=O)C(C)CO)CCNC(COCCCC#C)=O)ccccc1 N1(C(c2cccc(C)c2)=O)CC(NC(=O)CC2CCC(=O)O2)CC(C)C1 C=C(C)CC(C(=O)NC(CC(=O)NCc1nccc(C)n1)C(C)C)OC C1(NC(C(C)N(CC)CC)=O)CN(C(=O)CCCN2CCCC2)C(CC)(CC)C1 CC1CN(C(C2CCC(NC(c3ccc(Br)cc3I)=O)CO2)=O)CC(C)O1 N1(C(c2nc(CC)sc2)=O)CCOC(CCNC(=O)C(C2CCOCC2)O)C1 CCCCC(O)C(C)C(=O)NOCC(=O)NC(C)C1CC1 Cc1nsc(C)c1C(=O)NCC(O)C(=O)NCCn1nncc1C CON(C)C(=O)CC1(C)CCN(C(=O)CCc2ccc(C)o2)C1 N1(C(c2n(CC#C)ccn2)C(=O)NC(C)(C)CC)CCCN(C)CCC1 c1(OC(=O)Nc2n(CC)nc(C)c2)ccc(OC(C)(C)C)cc1I c1(C(N(CCC)CCNC(=O)C(c2c(C)n[nH]c2C)C)=O)cnc([N+](=O)[O-])n1C N1(C(C2C3(CC(NC(C4(COCC)CCC4)=O)C3)C2)=O)CCC2CCN(C)CC12 N1(C(c2cc3nnn(C)c3s2)=O)CC2CCC(C1)C(NC(C1CSC1)=O)C2 c1(CC)cnc(OC)c(C(=O)NCCN(CC(C)O)C(C2CCCN2C(C)=O)=O)c1 c12cc(Br)cc(c1Cl)C(=O)N2.CCCCCC=CC(=O)NC1CC1C(=O)OC C(=O)(C1=C2CCCN=C2NN1)NCCCN(C)C(C12CCC1C2)=O C1(C(N(C2C(C)CCN(C(=O)CSC(C)(C)C)C2)C)=O)CCOCC12CCC2 CC1CCCCC1(C)n1cc(CN(C(=O)C(C)Cc2ccc(F)cc2)C)nn1 N1(C(CN(CC)CC)=O)CCCCC1C(=O)N(CC(C1CCCCC1)O)C1CC1 CCC(C)C(C(=O)N1CC=CC1C(=O)OC)NC(=O)CCn1cccn1 C1(OCC)CCN(CCc2cn(CC(=O)Nc3sccc3CCC#N)nn2)CC1 c1(SC)cncc(C(=O)NCC2CC(NC(=O)C(C)C)C2)c1 CCCC(CCC)C(CC)NC(c1nnnn1C)C1CC=CCC1 c1(NC(C(C2CC2Cl)OCC)=O)cc([N+](=O)[O-])ccc1C CCC(C(=O)NCC(CNC(=O)C(C)(C)CF)OC)C(C)C c1(C(N(CC(C)NC(=O)C(C)OC2CCCCC2)C)=O)cccc(F)c1 C1(C(=O)NCC(C)(C(C)C)NC(c2c(C)onc2)=O)CC2CCC(C1)O2 N1(C(C2C(C)CCO2)=O)CCC(C(C)(C)CNC(=O)CCN2CCC2)CC1 C1(C(=O)NCC(C)NC(c2csc(Cl)n2)=O)CC(=O)CC(=O)N1 c1(C(=O)NCCN(C(C(C)NC(N)=O)=O)CC2CCC2)cc(CC2CC2)c[nH]1 c1(C(N2CC(C)CCC2CO)C(=O)NCCCSC)ccc2c(ccn2C)c1 C1(C(N(CC(CNC(c2ccc(SC)s2)=O)(C)C)C)=O)CN2CCN1C(C)C2 c1(OC)ccc2c(c1NC(=O)C(N1CCCC1c1noc(C3CC3)n1)=O)CCC2 C(CC(CC)CO)NC(C(Cc1cc[nH]n1)NC(CCN(CC)CC)=O)=O C1(C(C)NC(=O)C=CC2CCC2)CN(C(C2C3CC4C(C3)C24)=O)CCO1 N1(C(CN(C2CCCC2)C)=O)CC(O)C(F)C1.C12CCC(C1)C(=O)N2 C1(CC(=O)NCC2(C)CC2(F)F)CCCCN(C(=O)CC2(O)CCCOC2)C1 C1(SC)CC(c2nnnn2C2CC(F)(F)C2)(NCC2CC(SC)C2)C1 C1(C(N2CCC(C)C(NC(=O)CCCCCF)C2)=O)CC1C1CCCCC1 CC(C)CC(=O)NCCOCCN(C(=O)C(CO)N(C)C)C N1(C(c2nc(C)oc2)=O)CCCC(C)C1CNC(=O)NCCNC1CCCCC1 c1(C(=O)NC2C3CN(Cc4c(OCC=C)cccc4)CC32)cc(F)c2cn[nH]c2c1 N1(C(CC(CC)C(C)C)=O)CCCC2(CNC(=O)Cc3ccc(Cl)s3)CCCC12 c1(C(=O)NCCCC(C)(C)NC(C2CC=CCO2)=O)[nH]nc2ncccc12 c1(CCC)cc(=NCC2(C3CC3)CCN(C(=O)CC(O)C3CC3)C2)[nH]c(Cl)n1 C1(COC)CC(CNC(=O)Cc2cnoc2)N(C(c2nocc2C(C)C)=O)C1 Cn1cnc2cc(C(N3CC4(CC(CC(=O)NCC(C)(F)F)C4)C3)=O)ccc12 Cc1cc(C(=O)NC(C2(O)CN(C(C3(F)CCCOC3)=O)C2)C)cn1C N1(C(C=CC(C)(C)N)=O)CC(C#N)(c2ccccn2)C1 C1(C(N2CC3C(NC(C(COC)COC)=O)C3C2)=O)CN2CCN1C(C)C2 N1(C(Cn2ncc(C#N)c2)=O)C2CCC1C(CNC(=O)CN1CCNC(=O)C1)C2 c1(C(N2C(CC=C)(C(=O)NC3CCCC3C(C)C)CCC2)=O)cc(O)nc(O)n1 c1(C2C(N(C(c3cc(C4CC4)nc(O)c3)=O)CCO)C2)ccc2ccccc2c1 c1(C(=O)NC(CC#CC)C(=O)O)ncnc2sc(-c3ccc(CC)cc3)cc12 C(c1cccc(Br)c1)=CC(=O)NCC1CCC(NC(C23CC(CO2)C3)=O)C1 Cc1ccc(NC(=O)C(N2CC3CCC(C2)N3CC(C)(C)O)=O)cc1C#N c1(C(c2n(C)ccn2)NC(c2cn(C)nc2-c2ccc(Cl)s2)=O)ccccc1O C1(Nc2cn(CCC(=O)N(C)C)nc2)CCC(F)(F)CC1 N1(C(C2=C(C)OCC2)=O)CCC2(CCCC2NC(=O)CCN(C)C(C)=O)C1 Cc1ccc2c(CC(=O)NCC3C(C)CCN3C(=O)Cc3ccsn3)c[nH]c2c1 c1(CCC)nnsc1C(N1CCC(OCCNC(=O)CCC2CCN2CC)C1)=O CCCCCCCCC(=O)NC(C)(C)CNC(c1cnn(C2CCCC2)c1)=O Cc1ncc(C(N2CC3CC(NC(c4ccc(N(C)C)nc4)=O)C3C2)=O)c(=N)[nH]1 C1(C2CCOCC2)(C(=O)NC2CCN(C(C=CS(C)=O)=O)CC2)CCOCC1 c1(CC)c(C(N2CCN(C(c3nnnn3C)C)CC2)=O)nnn1CC c1(C(C(C)C)=O)c[nH]c(C(=O)NC2CN(C(=O)CSC(F)(F)F)C2)c1 c1(C(N(CCOC)CCNC(C)=O)=O)cccc(N)c1C C(N=c1[nH]c(=NCCCOC(=O)N(C)C)[nH]c2ccsc12)C1C(C)C1(F)F C1(O)(C(N(CCC(=O)NCC2CCOC2)CCO)=O)CCSC1 C(=O)(CCCCCC(C)C)N(CCCC)C(c1ccc(OC)cc1)C N1(C(C2C(CCC)CCC2)=O)CCC2CN(C(c3cnn(C)c3C)=O)CC2CC1 c1(OC)cc(NC(C2CC3C=CC2CC3)=O)ccc1NS(C)(=O)=O C(N=c1[nH]c(=NCCCCCCOC2CC2)[nH]c2c1CSC2)c1c(C)ocn1 C1(C(=O)NCC(C2CCC2)OC)CC(CCNC(=O)C(C)n2ccnc2)C1 Cc1ccc(-n2cc(C3(N4CCCC4C4NC(=O)NC4=O)COC3)nn2)cc1Br C(=O)(C(C)(CC)C(=O)N1CC(CNC(c2cn(C)nc2O)=O)C2(CC2)C1)OCC CCC(O)C(C)C(=O)N1CCC(NC(=O)CC(C2CCC2)C2CCC2)C1C c1(C(=O)Nc2c(C(=O)OCC)onc2C)ccc(F)c(-c2cncc(CO)c2)c1 C(CCC(=O)N(C(C)C(N1CCCC1CC1CC1)=O)C1CC1)OCCC N1(C(C(CCC=C)(C)C)=O)CCOC2(CCCN(C(=O)CNC(=O)C(C)C)C2)C1 N1(C(C=C(C)C(F)F)=O)CCCC(C2CCN(C(=O)CCc3nnnn3C)C2)C1 S(=O)(=O)(c1ccc(NC(CCO)C2CCC2)c(Br)c1)N(CC(O)CC(F)(F)F)C c1(OC)c(C)cc(C(=O)N(CC(C)NC(C2CCCCC(=O)N2)=O)C)cc1Cl O=C(O)C(CCOCc1ccc(-c2ccccn2)cc1)Oc1ccccc1 C1(O)(C(N(CCC(C)NC(c2csc(-c3cnccn3)n2)=O)C)=O)CC(C)(C)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1C(C)N(C(c2cc(Cl)cc(F)c2F)=O)CC1 C1(NC(c2csc(O)n2)=O)CN(C(=O)C=Cc2cnccn2)CC1C1CC1 N1(C(Cc2c(C)occ2)=O)CCC2(C=C(C(=O)N3OC4CCC3C4)C2)C1 C#Cc1ccc(NC(=O)C(CC(C)C)ONC(C2(SC)CC(=O)C2)=O)cc1 N1(C(c2c(C)ccs2)=O)CC(C)(C)OCC1CNC(=O)CCS(C)(=O)=O c1(C(=O)NCCC2CC(NC(c3snnc3C3CC3)=O)C2)cc(O)cs1 C1(CC)(NC(=O)C(C)CCOC)CCN(C(C2NC(=O)OC2C)=O)CC1 N1(C(C2(CCC=C)CC2)=O)CC2CS(=O)(=O)CC2(NC(=O)C#CC(C)(C)C)C1 N1(CC2CC(CSCCC3(CS(C)(=O)=O)CC3)C2)CCCNC1=O Cc1ccnc(C)c1NC(C1(C)CCCN(C(=O)C(C)Oc2ccccn2)C1)=O C1(NC(COCCC=C)=O)CCC12CCN(C(C1CC1OCC)=O)CC2 c1(OCCCC(=O)NCCC(C)NC(=O)Cc2cnsc2)ccc(C(C)C)cc1 C1(O)(C(=O)NC(CC(C)NC(CC2(CC)CCC2)=O)C)CCCCC1 c1(C(N(CCNC(C2CCCCC2C2CC2)=O)CC)=O)cc2ccc(Cl)cc2[nH]1 CC(CC(=O)NC1CN(C(C2CNC(=O)C2)=O)C1)NC(C1CCCC1)=O c1(C(=O)NCCC(=C)CNC(c2n[nH]cc2C(C)C)=O)ccc(C(C)=O)c(F)c1 C1(CC(=O)NCC(C)N(C(=O)CN2CC3CC3C2)CC)COCC(C)(C)O1 C1(NC(C(CC)=CCCC)=O)CN(C(=O)CC(O)CN(C)C)CC2(CCC2)C1 C1(C(N2C(C(C)NC(c3cnn(C4CC4)c3Cl)=O)CCC2)=O)CCCC2(CC2)C1 C1(N2CCC(Oc3ccc(Cl)cn3)CC2)Cc2ccccc2O1 N1(C(C)C)CCC(CN(CC(F)(F)CO)C)CC1.c12n[nH]c(n1)CNC(=O)CC2 C1(C(N(c2cccc(C)c2)C)=O)CN(C(c2ccc(C3CC3)o2)=O)CC(C)(C)C1 c1(C(N(CCCNC(C(C)N(C(C)=O)C)=O)CCO)=O)ccn2ccnc2c1 Cc1cccc2c(C(=O)NCCCCC3CN(C(=O)C(C)(C)C4CC4)C3)coc12 C12(C(C(=O)OC(CC(=O)OC)C)C)CC3CC(CC(C3)C1)C2 Cn1ncc2ccc(-c3noc(-c4cccn(C(F)F)c4=O)n3)cc12 C(=O)(C1=CCC(F)(F)CC1)N(C1CN(C(C2CC(C)C2(C)C)=O)C1)C CC1CN(C)CCCN1C(C1CCOC1CNC(c1cc2cccn2cn1)=O)=O C1(C(N2CCC(CCOC)(NC(=O)CCC=C(C)C)C2)=O)OCC2CCCCC12 c1(C(N2C(CCNC(C(C)(C)C(N)=O)=O)CCCC2)=O)cccc2c1NCC2 c1(C(=O)OC)ccnc(N2CCC(NC(c3cc(Br)co3)=O)C2)c1[N+](=O)[O-] N1(C(c2n[nH]c(C)c2C)=O)CC(NC(c2nn(C)cc2Cl)=O)CC(C)(C)C1 C1(C(=O)NC2C=CCN(C(C(C)c3ccco3)=O)C2)CCCCC12CCC2 C(=O)(C(O)C(F)(F)F)NC1CN(C(c2ccc(COC)s2)=O)C1 C1(C(=O)NC2C(C)CCC2C)C2CCCC2CN1C(C1CC2CC2C1)=O n1(CC(=O)NCCN(C(C2(C)CCC2)=O)C2CC2)nnc2ccccc2c1=O N1(C(=O)NC(C)CCC#N)CCC12CC1CCC2C1 C(=O)(C(C)(C)CC(F)(F)F)N1CC(CCC)N(C(=O)CC2CCCCN2C)CC1 Cc1cc2ncnc(N3CCC(NC(=O)C(F)(F)CO)C3C)c2[nH]1 C1(NC(CCCNC(N)=O)=O)CCC2CN(CCOCC(F)F)CC2C1 C1(C(N2CC(C)(C(=O)NCC(C)OCCO)C2)=O)CCCCC1F C1(NC(C(CC2CN(C(CNC(C)=O)=O)C2)F)=O)CCC(F)CC1 c1(N2C(CCNC(c3ccc(Cl)s3)=O)CCCC2)[nH]cnc2nc(Cl)cc1-2 Cc1ncoc1C(=O)NCC=CCC(=O)NCCCCc1cnc[nH]1 c1(C(N2CCC(COC)(NC(=O)C(C)CSC)C2)=O)ccc2cc(C)ccc2n1 c1(CC)c(C(=O)NCC(CO)NC(=O)Cc2ccns2)cnn1CC c1(C(=O)NCC(C(C)(C)C)NC(C2C(C)C2C)=O)cnn2cc(C(N)=O)cnc12 C(=O)(C1=CC2(CCOCC2)C1)NC1N(S(C)(=O)=O)CCCC1 c1(OC)ccc(N)c(C(N2CCC(O)(C(C)NC(=O)CC(=O)NC3CC3)C2)=O)c1 N1(C(CCC2CCC(=O)C2)=O)CCC2CCN(C(=O)Cn3cccn3)CC12 CC1CN(C(=O)COCC2CCCC2)CCC1NC(=O)C=CC1CC1 c1(C(C(=O)NCCC2N(C(COC)=O)CCCC2)C)cc(F)ccc1Br C1(C(N2CC(C(N(CC(=C)C)CC(=C)C)=O)(COC)C2)=O)CC=C(C)CC1 C1(C(N2C(C)CCC(CNC(c3csc(CO)n3)=O)C2)=O)CCc2nncn2C1 c1(CNC(c2n(CCOCC)nnn2)c2ccns2)n[nH]c2ccc(C)cc12 CCC1=C(C(=O)N2CCC(NC(=O)Cc3cscn3)CC2C2CC2)SCCO1 N1(C(C2(CC)CCOC2)=O)CC(CO)C2(C1)CN(C(=O)C(SC)SC)C2 C(=O)(C(F)(F)C(C)(C)O)N1CC(CN(C(C(CCC)NC(N)=O)=O)C)OCC1 CC1(C(N2CC(OC3CCN(C(c4cccs4)=O)CC3)C2)=O)CCCOC1 C12(NC(C3CNC(=O)O3)=O)CCC(CN(C(c3cccc(C4CC4)n3)=O)C1)C2 c1(C(N2CC(NC(C(=O)NC(C)C)=O)C3C2C3)=O)cc(C#N)ccc1O Cc1nc(C(=O)NC2(C3CCCN3C(=O)CC(C)C(F)F)CC2)c2ccccn12 CC(CF)CC(=O)N(C)CC1CC(F)CN1C(c1cnn(C2CCC2)c1)=O N1(C(C2C(=C)C2)=O)CCC(CCOC)(NC(=O)CCCN2C(=O)CNC2=O)CC1 n1(CC)c(CN2CCN(CCc3ccccc3)CC2)nnc1-c1cnn(C)c1 N1(C(C(C)OCc2cccs2)=O)CC(F)(F)CC1(C)CNC(C1CNC(=O)C1)=O c1(C(=O)NC(c2cn(C)nn2)C(=O)NCCCOC)c[nH]c(C)c1 c1(OCC)cccc(CN2CC(C)(C(=O)NCc3cscn3)C2)c1 C(=O)(CCS(=O)(=O)NCC1CN(C(c2ccc(Br)cn2)=O)CCO1)OC c1(C(N(CCNC(C(C2CCOCC2)OCC)=O)C)=O)nnn(C(C)(C)C)n1 C1(C2CC2)(CNC(C(CN(C)C)N(C)C)=O)CCN(C(C2(C)COC2)=O)C1 C1(C(CNC(c2cc(I)ccc2Cl)=O)=O)CC12CCOCC2 C1(NC(C(CCC)NC(N)=O)=O)CC2CN(C(=O)C=C(C)Cl)CC2C1 c1(C(=O)NC(C2OCCN(C(c3c(C)csc3C)=O)C2)C)ncc2[nH]ncc2n1 C12(C(=O)NCCC3(NC(c4c(N)cncc4)=O)CC3)CC=CC(C1)OC2 N(C1CCc2ccc(Br)cc21)C(C1CC(=C)CN1C(=O)CNS(C)(=O)=O)=O C1(OCC(=O)NC(CC)CNC(=O)C(=Cc2ccco2)C)CCCCC1C N1(C(C2(COC)CCC2)=O)CC(NC(C23COCC2C3)=O)CCC(O)C1 N1(C(C(CCC)C)=O)CC2CCN(C(C3(CCF)CC3)=O)C(C2)C1 C1(CNC(c2cnc(C)o2)=O)CN(C(=O)C=Cc2nc(C)c(C)[nH]2)CC1(C)C C12(C(N3C(CC)C(NC(=O)CSC(F)F)CC3)=O)CCCC1CC(=O)C2 c1(N(C(C(C)(C)C(F)F)=O)CC(=O)NC2CCC2(F)F)ncnc2c1CCO2 N1(C(C=C2CCC(C)C2)=O)CCCC(N(C)C(c2cnn(C)c2N)=O)CC1 C1(NCCC)CCC(n2cc(C(C)(C)CC3CC3)nn2)CC1 C12(CCNC(C=Cc3occ(C)n3)=O)CCC(C1)N(C(=O)CCCNC(N)=O)C2 C1(CC=C)(C(N2CCC(n3cccn3)C2)=O)CCN(C(=O)C(C)N2CC(C)C2)C1 c1(OC)cc(C(=O)N(C(C)(C(=O)OC(C)(C)C)C2CC2)C)nc(C)c1 c1(C(=O)NCC2(NC(c3cccc(C)c3)=O)CCOC2)cc(F)ccc1O c1(OC)nc(Cl)ccc1C(=O)NC1CCN(S(=O)(=O)Cc2ccc(C)c(C)c2)C1 N1(C(C=NOC)=O)CC(CNC(C2(Cc3cnn[nH]3)CCC2)=O)C2CC12 CC(C)C(C(=O)NCc1ncccn1)C(C)NC(=O)CC1OCCCO1 c1(CC(=O)NCC2(CC(=O)NC3(COC)CCCC3)CC2)cn(C)nc1C C1(C(=O)NCC2(NC(c3cc(SC)nn3C)=O)CCCC2)CN(C)CC(C)O1 N1(C(C=C2CCC(C)CC2)=O)C2CCC(C2)C1C(N1CCOCC(CO)C1)=O N1(C(CC(=O)NCC(CC)NC(C2CC3CC2C3)=O)C)CCCCC1=O c1(CC)cc(C(=O)NC2(CN(C(=O)CN3CCCCC3C)C)CC2)c(C)nn1 CCC(O)C(C)C(=O)N(C1CCN(C(c2ncoc2C2CCCCC2)=O)C1)CC C1(NC(C(N2CCOCC2)C)=O)CC2(CCN(CC(N3CCCCC3)=O)C2)C1 C(C(C(=O)NCCC(O)C1CCCC1)NC(c1ccnn1C)=O)SCC C#CCC(C)(C)C(=O)N1CCN(C(C2SC3C=CC2CC3)=O)C(CO)C1 C(CCCCC(=O)N1CC2CC2(NC(=O)C=CCCC=C(C)C)C1)NC(C)=O C1(NC(c2cc(CCC)on2)=O)CCCN(C(=O)C(CC)CCC)CC1 C1(C(=O)NCCc2c(C)ocn2)CCC(CNC(C2CC(C)(C)CO2)=O)CC1 c1(-c2scc(C(=O)OC)n2)cccc(-c2nccn2CC2CCOC2)c1 c1(OC)noc(C)c1C(=O)NC(C)CN(C(=O)C(C)NC(c1cccs1)=O)C C1(NC(C(C(C)C)SC)=O)CCN(C(c2ccc(Br)nc2O)=O)CC1F C1(C(=O)NCc2scc(CNC(C3(C)CC4CC4C3)=O)n2)C2CC3C(C2=O)C13 CCCC(C)(C)CC(=O)NC1CN(C(c2sc(Cl)cc2Cl)=O)CCC1C C1(C(N(CC(CC)NC(c2ccccc2Cl)=O)C)=O)CC2C=CC1CCC2 c1(CC)ccc(NC(C23CC2CN(S(=O)(=O)CC(=O)OC(C)(C)C)C3)=O)cc1Cl CCC(CCOC)C(=O)N1CC(O)CC1C(=O)NCC(n1cccn1)C C(CC(C)(C)C(=O)NCC1CCCN1C(C12CC(C(F)(F)F)(CO1)C2)=O)SC C1(NC(CC(COC)C)=O)CC2CCC(C1)N2C(C1(C)CCCO1)=O c1(N(C(C(=O)NCC2CCCO2)C2COC2)CC)ccccc1 Cc1cc(=O)n(C)nc1C(=O)NC(CNC(=O)CCc1cc(F)ccc1F)CO C1(CN(C(=O)CCC2(C)CC2(F)F)C)COCCN1C(C1COC(=O)N1C)=O CC1CC(NC(c2cccc(COCC(F)(F)F)c2)=O)CN1C(=O)C(C)(F)F C12(NC(=O)C=Cc3ccc(Cl)cc3)CCCN(C(=O)CC3CC=CCC3)CC1C2 c1(CC(=O)NC(C2CCCN(C(=O)COCP(C)(C)=O)C2)C)cnn2c1CCCC2 C(=O)(C1CCc2cc(F)ccc21)N(C(C)CNC(=O)C(C)(C)n1cncn1)CC c1(CC(=O)NCC(C(C)(C)C)NC(c2cncc(F)c2Cl)=O)c(F)cccc1F c1(CNC2(CC(=O)NCC3CSCCN3)CCC2)cnc(Cl)cc1Br c1(C(N2CC(N(C(CCN(CC)CC)=O)C)C2)=O)cncc2c1CCC2 C(CC(C)N=c1[nH]c(N2CCOC(C(C)C)C2)nc(=NC)[nH]1)N(C)CC C1(NC(C(CNC(CC(=O)NCC)=O)N(C)C)=O)CCN(C)CC1 N1(C(C2N(S(CCC)(=O)=O)CCC2)=O)CCN(C(=O)CC2(C3CC3)CC2)C(C)C1 c1(C(N(C2CCC(C(=O)NCC(C)(C)C3CC3)C2)C)=O)cnc(N)cn1 N1(CCC(=O)NC(C)CNC(c2nn[nH]c2Cl)=O)CCC(O)CC1 N1(C(C2CCCCC2)=O)CCOC(CC(=O)NCC(C)(C)CC2CCOCC2)C1 C(CC(C)(C)C)(C(=O)N1CCOC(CNC(=O)CCC(C)(C)N(C)C)C1)OC C(=O)(CCCCCC(C)C)NC1(C(=O)NC(c2c(C)ccnc2)C)CC(F)(F)C1 N=c1[nH]ccc(C(=O)NCCC2CN(C(=O)C(F)(F)C3CC3)CCO2)c1[N+](=O)[O-] Cc1nccnc1CNC(C1C2CC1N(C(=O)C(N1CCOC1=O)C)C2)=O N1(C(C(C)n2ccnn2)=O)CCCC12CCN(C(=O)CC1CN(C3CC3)C1)CC2 C1(OCC)CCN(C(=O)CC(CNC(=O)Cc2cccn2C)OC)CC1 C1(N(C(=O)CCc2cn(C)cn2)C)CC2CCC(C1)N2C(C1CCCCO1)=O c1(C(=O)NC(C)CNC(C2CCC3(CCC3)O2)=O)cnn2ccn(C)c12 O=CN1CCN(C(C2CC(F)CN(Cc3cccc(Br)c3O)C2)=O)CC1 CCCC(O)C(=O)N(C)CC=CC(=O)NCC1(CCO)CCCC1 CCC(CC)C(=O)N(C)CCNc1nccc(Br)n1 C1(CNC(C(c2ccco2)NC(C2CCCCO2)=O)=O)(CO)CC2CC2C1 N1(C(c2ccc(CC)s2)=O)CC(NC(=O)CC2CN3CCN2CC3)C(C2CC2)C1 C1(C)(CNC(C(C2(O)CCC2)NC(C(CC=CCC)C)=O)=O)CCCCCC1 CC1CN(C(c2sccc2-n2cccc2)=O)CC1NC(c1cc(C(F)F)on1)=O C(C(C)(O)CNC(c1nnc(C(C)(C)C)s1)=O)NC(C(C)=C1CCCC1)=O C(C)(C(=O)NCC1CCN(C(C2CC(SC)C2)=O)CC1)(C(C)C)OC C(C(C(=O)NCc1coc(C)n1)NC(=O)CCNC(=O)CO)SCC N1(Cc2nc(C(C)OCC)sc2)CCN(C(=O)C(C)n2cccn2)CC1C N1(C(C(CC(C)C)O)=O)CC(NC(C2(F)CCOC2)=O)CCC(O)C1 C1(C(=O)NCC(C)(C)OCCNC(C2C(C)C2)=O)COCCO1 N1(C(C(CSC)OC)=O)CCN(C(=O)Cc2ccc(F)cc2)CC(C)(F)C1 C(=O)(C(C)(C)CC(C)(C)C)NCC1(NC(C(C)Cc2ccccc2)=O)CCCC1 CCCCC(C(=O)N1CC2(C(N3CCCC4(CC4)C3)=O)CC1CO2)N(C)C CC(CC(C)(F)F)C(=O)N1CC(CCCCNC(c2cc(CN(C)C)on2)=O)C1 c1(C(=O)NC2C(NC(c3cncn3C3CC3)=O)CC2)[nH]ccc1C1CC1 C1(C(N2C3C(NC(=O)Cc4cc(C5CC5)on4)C(C3)C2)=O)CC12CCCOC2 c1(NC(C)=O)cnccc1C(=O)NC1CC(O)(CNC(c2sccc2F)=O)C1 N1(C(C2c3c(nc(C)[nH]3)CCC2)=O)CCC2(CC1)OCc1ccccc12 n1(CC)ncc2cc(C(=O)N(CC(C)NC(=O)Cc3ccc(C)s3)C)cnc12 c1(COC)cccc(C(=O)N(C2CCC(NC(=O)C(=O)NC3CC3)C2)C)c1C CC1(C)OCCC1CC(=O)N(C1CCC(C(C)(C)C)CC1)CC(=O)O CCCCC(CC)C(=O)NC1CN(C(c2cc(C)ccc2Cl)=O)CC1OC c1(C(=O)NCC2(NC(c3c(C)cco3)=O)CCCCC2)occ2c1CCOC2 Cn1ncc2ccc(NC(=O)CC3CC(NC(c4ccc(Br)nc4)=O)C3)cc12 C=CC(C)(CC)C(=O)NC1C2CCC(C2)C1C(=O)NCCCC(=O)N(C)C Cc1cc(NC(CC2(CNCCCc3scnc3C)CC2)=O)ccn1 c1(C(N2CC(NC(CC3N(C)CC=CC3)=O)C2)=O)cc([N+](=O)[O-])c2nsnc2c1 N1(c2n(CCOC)c(-c3cc(N)ccc3F)nn2)CCCC2CCCC12 Cc1cncc(C(N2CCC2CNC(=O)C(c2ccn(C)n2)C)=O)c1 c1(N2CC(C(N)=O)(CNC(CS(CC)(=O)=O)=O)C2)cccc(F)c1C#N Cc1cn2c(C(=O)NCC(C)NC(=O)Cc3cnc4n3CCOC4)c(Cl)nc2s1 C(=O)(C#CC(=O)N(C1CCC1)C)N(C1CCN(C(c2cc(C)oc2)=O)C1)C N1(C(c2cnc(C)nc2C)=O)CC2(CCCC2NC(=O)CCN2CCCC2=O)C1 CC(CN(C(=O)CCN1CCCCC1)C)C(=O)N(C)CCc1cnn(C)c1 C1(C)(C(=O)NC2C(C)(C)OCC2)CCCN(C(=O)C(=O)C2CCCC2)C1 c1(C(=O)NCC(C2CCCCC2)NC(C(CC)F)=O)nccn2nc(C)cc12 CC1CCN(C(C2(C)CCOC2)=O)CCN1C(c1nc(Cl)sc1Cl)=O CCCC(O)CC(=O)NCC(O)CNC(=O)C(c1ccc(Br)s1)=O C1(O)(C(C)NC(=O)Cn2cccc2)CCN(C(=O)C(C2CCCCC2)O)CC1 C(=O)(C(C)(C)C#N)N.c1(C2CC(=O)N(C)CC(=O)N2)cccc(Cl)c1.C1(O)CC=CC1 Cc1ccc(CN2CCC(F)(C(=O)NC(c3ccccc3)C3CC3)C2)c(Cl)n1 N1(C(Cc2cn(Cc3ccn(CC)n3)nn2)=O)Cc2ccccc2CC1CCO C1(CNC(C2N(CC)CC2)=O)CN(C)CCN1C(=O)CCN(C1CCCOC1)C N1(C(CCNS(CC)(=O)=O)=O)C(C)C2CC1C2NC(c1nn(C)cc1C)=O C1(NC(c2ccc(CCC)cc2)=O)CCN(C(C2CS(=O)(=O)CCO2)=O)CC1O c1(C(=O)NC2C(CNC(CCS(C)(=O)=O)=O)C2)cc(N)c(O)c(F)c1 N1(C(c2cc(CC)nn2C)=O)CCC2(CCCC2C(=O)NCc2cncnc2)C1 Nc1ncnc2c1ncn2CCCC(=O)Nc1nc(-c2cc3c(s2)CCSC3)cs1 C(C(C)C)(C(O)C(=O)NCC(C1CCC1)NC(c1ncn2c1CCC2)=O)OC N1(C(c2cc(CC)ncc2)=O)CC2CCC(C1)N(C(=O)CN(CC(C)(C)C)C)C2 C12(COC)CN(C(c3cnc[nH]3)=O)C(CNC(C3CN4CCC3CC4)=O)(C1)C2 C1(CC)(CC)CC(NC(c2cc(C)nn2C2CC2)=O)CN1C(=O)CC(C)(C)C c1(C(=O)NCC2CC(CC(=O)NCC3COC(=O)C3)C2)ccc(C2CC2)cc1 c1(C(=O)NC2C=CCN(C(C(COC)OC)=O)C2)[nH]c2cc(F)cc(F)c2c1C C(CC(C)C)(C(=O)NC1CN(C(=O)CN2CCSCC2)CCC1F)OC n1(CCC)nc(C)cc1C(=O)NC1CCC1CNC(=O)CCc1cnc[nH]1 C(=O)(C(CNC(C1CCC(C)(C)OC1)=O)C(C)(C)C)N(C)C(C1CC1)C1CC1 CCC(CC)(CC(=O)OC)C(=O)NC1CCN(C(=O)C(N2CCCC(C)C2)=O)C1 C=CC1(C(N2CCCC(CF)C2)=O)CCN(C(C2CC(=O)N(OC)C2)=O)C1 CC1CN(C(C2CCC2(C)C)=O)CC1NC(c1ccc(N(C)C)nc1)=O c1(OCC)cnc(N)cn1.C1(NC(=O)C=COC)C2CC1N(C(=O)C(C)(C)OC)C2 C=C(C)CN=C(NCc1ccc(OCC)nc1C)N1CCc2c(nnn2CC)C1 N1(C(C(CC)CC)=O)CC2CCC(CNC(=O)Cc3ccccc3CO)CC2C1 c1(C(=O)NCC(CNC(c2c(C)ncnc2O)=O)C)c(F)ccc2c1OCO2 C=CCC(CC)C(=O)N(CCCNC(C1CC(F)C(=O)N1)=O)C(C)C C12(NC(c3ccc(CSC)o3)=O)COC(C1)C(NC(=O)CCc1ccn(C)c1)C2 N1(C(Cc2ccnc(C)n2)=O)CCCC(O)(CCNC(=O)CNC(=O)C2CC2)C1 c1(C(=O)NCC(n2cc(C3C4COCC34)nn2)C)cc(Cl)ccc1Br C1(C(=O)NC2CC(O)(C(F)(F)F)C2)(COC)C=CCN1C(=O)NC(C)C c1(C(=O)NC(C)CC(C)NC(c2sccc2OC(F)F)=O)cccc2ncsc12 N1(C(CCC2(C)CCCN2C(=O)CSc2nc[nH]n2)=O)CC2CCC(C1)O2 C=CCCCC(=O)N1CCC(CCOC)(NC(c2[nH]nnc2C(=O)OC)=O)C1 C1(C2CCN(C(c3cc(C#N)ccc3Cl)=O)C2)(NC(CC(C)CF)=O)CC1 c1(C(=O)NCC2CCC(C(=O)NCC)CC2)cccc2c(Br)cccc12 n1(CC)cnc2c(NCC(c3c(F)cccc3F)C)[nH]c(=NCC(F)(F)Br)nc12 C=CCC(C)(CC)C(=O)N(C)CCN(C(=O)C(F)(F)C(C)O)C C1(CNC(COC)=O)CCCCN(C(C2(Cc3cccnc3)CC2)=O)C1 C(=O)(CCCCC(C)(C)C)NC(c1ccccc1)C(=O)N(C)CC1(OC)CCC1 c1(C(N(C2CCCN(C(=O)C(C)(O)C3CC3)C2)CC)=O)cc(O)nc(N(C)C)n1 CC(CNC(=O)CCN(C)CCO)C(=O)NCC(CC1CC1)CO c1(C(=O)NC2CCC(N(C)C(c3cc(O)nc(Cl)c3)=O)C2)cccn2nccc12 C(=O)(CC(C)(C)Cc1ccc(Cl)cc1)NCC1(NC(CC2C(C)C2)=O)CCCC1 Cc1nc(Cl)[nH]c(=NCC2CCCC2NC(C2(CO)CCC2)=O)c1Cl C(CCCCC(=O)N1CC(NC(=O)C(C)C(O)CC)C(CO)C1)=CC C1(NC(C(F)=CC)=O)CN(C(=O)C(C)c2ccco2)CCC1c1cccc(F)c1 c1(CC(=O)NCCNC(C2C(C(=O)OC)CC2)=O)cccc(F)c1F C1(NC(C(C)C(C)(F)F)=O)CCN(C(C2CN3CCCN2CC3)=O)CC12CCC2 C12(C(N(CCNC(C(C)(C)OC)=O)C3CC3)=O)CCCC(=O)N1CCC2 CC(C)CC(C)(O)C(=O)N(CC(=O)NCC(C)(C)CCCO)C(C)C C(c1ccncc1)=CC(=O)N(C)CC1(CNC(=O)C=CC(F)F)CC1 c1(C(=O)OC)ccc2c(c1)OC(F)(F)CN2C(=O)NC(C1CCCCC1)(C)CO CCC(CC(=O)N1CC(O)(C(C)NC(c2cc(CC(C)C)c[nH]2)=O)C1)OC c1(C(C)C)nc(NCCCCS(C)=O)cc(=NCC2(C)CCC(F)(F)CC2)[nH]1 c1(NC(C)=O)cnc(C(=O)NC2CC(NC(=O)C(O)Cn3cncn3)C2)c(Cl)c1 C1(C(NOC(C2CCOCC2)CC)=O)CN(C(c2csnc2C)=O)CCO1 N1(C(CN(C(C)=O)C)=O)CC(C)C(NC(=O)Cc2ccn(C(F)F)n2)C(C)C1 Cc1cc(C(=O)NCC2CCC(NC(=O)CC3CCCOC3)CC2)cc(C)c1Br c1(C(=O)NC2C(NC(C(CC)O)=O)CCC2)oc(CC(C)C)nc1C c1(C(=O)NCCN(C(C2CCNC2=O)=O)C2CC2)cc(Cl)nc(Cl)c1 N1(C(N2CCCCC(OC(C)(C)C)C2)=O)C2CCC1CN(C(=O)N(C)C)C2 C12(CNC(C3CN(C)C3)=O)CC(NC(=O)C3=CCCSC3)(C1)C(C)(C)O2 C(C(=O)NCC(C)(C)OCC(=O)NCC1CC(CO)CO1)(C(C)C)SCC c1(CC(N2C(CCNC(C(CC=C)CC)=O)CCCC2)=O)c[nH]c2ccccc12 c1(CC(=O)N(CC(C)N(C(C2CC(CCC)C2)=O)C)C)c(C)nn(C(C)C)c1C N1(C(CN(CCC)C)=O)CCC(CC(=O)NC(c2ccncn2)C)C1 C1(C(=O)NOCCOCCF)CC(C)(C)CN1C(=O)Cc1cccc(F)c1 C(=O)(C#CC1CCC1)NC(c1ccccc1F)CNC(c1c(C)onc1)=O CC1CCc2n(C3CCCS(=O)(=O)C3)ccc2C1 c1(C(=O)NCC2N(C(CC3C(C)(C)C3(C)C)=O)CC2)cc(S(N)(=O)=O)cs1 N1(C(C2(c3ccc(F)cc3)CCC2)=O)CCC(NC(=O)C(F)C(C)(C)O)C(F)C1 c1(CN2CC(C(=O)Nc3c(OC)ccc(OC)c3)SCC2)cc(F)c(Br)cc1Cl Cc1cnc(C)c(C(N(C2CCN(C(=O)CCS(C)=O)C2)CCO)=O)c1 CCCC(CN)OC.C(=O)(C(Cn1cccn1)NCC)C(C1CN(C(C)C)C1)=O c1(CN(CCNC(=O)Cc2ccc(F)cc2Cl)CC)cccc2nn(C)cc12 c1(C(N2CCN(C(CCCC(OC)OC)=O)CC2)=O)cc2c(Cl)cc(F)cc2[nH]1 C1(CN(C(c2scc(C)c2)=O)C)CCC(NC(c2noc(C3CC3)c2C)=O)CC1 c1(C(=O)NC(C2CC(NC(C3CC=CCC3)=O)C2)C)ccnc2cc[nH]c12 c1(C(=O)NC(CC=C)CNC(C2OCCO2)=O)ccc(F)c(I)c1 c1(C(=O)NC(CC)CNC(C2CC2COC)=O)cc2c(OC)c(Cl)ccc2[nH]1 C1(NCC=CC)CCC(CC(=O)OC)C1(C)C C1(NC(C(CC#C)(C)CC)=O)CCC2(CCN(C(=O)C(C)CC3CCC3)C2)C1 C1(C)(C(=O)NCCC2(NC(C=CC(C)C)=O)CCC2)C2CCC(C2)C1(C)C c1(C(N(C2CCN(C(=O)CC3CCCCCO3)C2)CC)=O)sc(CO)nc1C C(=O)(C1c2ccccc2CN1C(c1ccc(Cl)nc1Sc1c[nH]c(=N)s1)=O)OC C12(NC(=O)C3CC3)CCCC1CN(C(=O)Cc1scnc1-c1ccccc1)C2 C(=O)(C(F)(F)CCn1cccn1)NCC1(NC(C2CCCCC2O)=O)CCCC1 N1(C(CSCCCC)=O)CCCC(C)(C)C1C(=O)Nc1cccc(OC)c1C C(=O)(C(C)(C)C(=O)NC1CCCN(C(=O)CCc2cc(C)[nH]n2)CC1)NC CCC(CO)C(=O)NCc1ccc(CNC(=O)CCOC2CC2)cc1 C(=O)(C1=CCCOCC1)NC1C(C(N2C(C)(C(C)C)CC2)=O)C2CCC1C2 C(C(C(F)(F)F)N1CCOCC1)NC(=O)COCC(=O)NC1CC1 C1(COC)CCC(C(N2CCCC2CNC(=O)Cc2cc(C)ns2)=O)C1 C12(CNC(=O)C=C3CCCC3)CCC(C1)N(C(c1cc(O)ccc1F)=O)C2 N1(C(C2N(C)CCC2)=O)CC=C(CNC(=O)Cc2cnsc2)CC1 c1(OC)ccc(C(=O)NCCCNC(=O)CC(C)F)c(OC2CC2(F)F)c1 C(=O)(CC(C)(C(F)F)N(C)C)N(CCNC(c1cn(CCC)nn1)=O)C CCC(CC(F)(F)F)C(=O)NC(CN(C)C(c1ccc(NC(N)=O)cc1)=O)CC c1(C(N2C3(C(N4C(C)CC5(CC5)C4)=O)CC3CC2)=O)ncc2ccccn12 C(C1=NOC2CN(C(=O)CCCCCF)CC12)NC(c1c(C)nn(CC)c1Cl)=O C1(C(=O)NC(C)CN(C)C)CC2CC2N1C(c1cc(Br)ccn1)=O C(N=c1[nH]c(=NC(C)CC)[nH]c2cccnc12)c1ccc(C(C)C)nc1 N1(C(CCc2nc(C)c(C)o2)=O)CCC2(C1)CN(C(C1CC(C)N(C)C1)=O)C2 CC1CN(C2CC2)CC1NCCNS(=O)(=O)N(C)C C1(C(N(C2CCN(C(=O)COc3ccccn3)C2)CC)=O)CC(=O)NC(=O)N1 C(=O)(C(O)C(C(C)C)OC)NC(C(=O)N(CC)CC1CC1)CCSC C1(C(N2CC(C(=O)NCC34CCC(CC3)O4)C(F)C2)=O)CCC2(CCC2)O1 C(CN=c1[nH]cc2ccnc-2[nH]1)OC1CCN(C(=O)C(c2ccc(Cl)cc2)O)C1 N1(C(CCN(C(c2cn(C)nc2)=O)C2CC2)=O)CCCC2(C=CCO2)C1 c1(C(N(CC(CNC(c2scc(C)c2)=O)C)C)=O)cc2ccncc2[nH]1 c1(C(N(C2CC3(CNC3)C2)C(C(=O)OCC)Cc2cnc[nH]2)=O)cccc(F)c1 N1(C(C2N(CC)CCCC2)=O)CC2CCC(N(C)C(C3CN(C)CCO3)=O)C2C1 C1(C(N2CCC(C(C#C)C)CC2)=O)CC(C)CCN1C(C1CCCSC1C)=O N1(C(C(C(C)(F)F)F)=O)Cc2c[nH]c(=N)nc2C1 Cc1nc(C2CC2)nc(C)c1C(=O)NCC(C)CNC(c1nc(C2CC2)no1)=O c1(NC(c2ccc(CCCCC)o2)=O)cccc(NC(C2CCCSC2)=O)c1 C12(NC(CN(C)C)=O)CCC(CN(C(C3CCSCC3)=O)C1)C2 N1(C(C(=O)Nc2cscc2Cl)=O)CCCC2(CCCN2)C1 C1(C(=O)NCC(C(C)C)NC(c2ccc(C)n2C)=O)CCC(F)(F)CC1(C)C N1(C(C(CCC)O)=O)CCCC(O)(CNC(c2ccc(CNS(C)(=O)=O)o2)=O)C1 Cc1nc(C)c(C(=O)NC(CNC(c2cn(CC(F)(F)F)nn2)=O)CO)c(C)n1 C1(C(=O)NCC#CCNC(C2(C)CCN(C(C)=O)C2)=O)CCc2cnnn2C1 Cc1cc(NC(c2ccc(O)nn2)=O)ccc1NC(c1n[nH]c(C)c1O)=O c1(OC)n[nH]c(C(=O)N(CC(C)NC(=O)C(c2cccnc2)O)C)c1Cl N1(C(CCC)=O)CCC(C(F)(F)F)C(CNC(C2CCN(C)CC2)=O)C1 C12CCN(CC1)C(=O)CNC2.N1(CC)CCC(NC(C2CCCN2)=O)C1 CCC(C(=O)NCC1(OC)CCN(C(c2c(C)n[nH]c2C)=O)CC1)C(C)(F)F CC(C)CC(C)C(=O)N(CCCCN(C)C(C1(c2cccnc2)CC1)=O)C N1(CCNC(C2(COC)CCCC2)=O)CCC(NC(c2cc(OC)no2)=O)CC1 N1(C(CNS(C)(=O)=O)=O)CCOC(CNC(c2cccc(CC(F)(F)F)c2)=O)C1 C1(C(C)NC(c2cn(CC=C)nn2)=O)CCN(C(=O)CC2CC=CCN2C)CC1 c1(CC)cc(C(=O)NC2CCCC(NC(c3cncnc3C)=O)C2)cn(C)c1=O c1(C(c2nnnn2C2CC2)NC(C2CC(F)(F)C2)C)cc(CO)ccn1 CC1(C)CN(C(=O)C2=COCC2)CC(C)(C)C1NC(=O)CCn1cccn1 C1(NC(C(CC)=CC)=O)CCN(C(c2cc(C3CC3)[nH]n2)=O)C12CCCC2 c1(C(N2C(C)CCC(NC(C(COC)(F)F)=O)C2)=O)cc(Cl)cc(Cl)c1F N1(C(C2CC3(CCC3)C2)=O)CCC2CN(C(C3CCCOC3)=O)CC2C1 c1(C(C(=O)NCCSC)N(CCC2CC2)CC2CC2)cccc2c1CC(C)(C)O2 N1(C(C2CCC(CC)O2)=O)CC(O)CC1C(N1CCC(C(C)OC)CC1)=O C1(COC)(NC(c2cc(-c3ccncc3)no2)=O)CN(C(C2SCCC2C)=O)C1 C1(C)(CNC(=O)CC2(OC)CN(C(=O)COC3CCCC3)C2)CCCOC1 CCCCC(O)CC(=O)NC1CC1CNC(=O)C(c1cccc(O)c1)(C)C c1(SC)cc(C)ccc1C(N1CCC(OCCN(C(=O)C2=CCCS2)C2CC2)C1)=O C1(NC(c2ccc(F)cc2)=O)CCCCCN(C(C2CC3CC2C3)=O)C1 C1(N(C(CN(C)CC)=O)C)CCCN(C(=O)C(=O)NOC)CC1 c1(C(=O)NC(CN(C(C(C)OCC)=O)CC)C)ccc(S(=O)(=O)CC(N)=O)cc1 c1(NC(C2CN(C(c3cccc4c3OCCO4)=O)C2)=O)ccc([N+](=O)[O-])cc1F c1(CC(=O)NCC2(NC(CCCC3C(C)C3)=O)CCOC2)ccc(C(N)=O)nc1 c1(C(=O)NC(CNC(c2c(C)occ2)=O)(C)C)cc(C(C)(C)C)oc1C N1(C(CN2C(C)CC2)=O)CC2CS(=O)(=O)CC2(NC(=O)CNS(=O)(=O)C2CC2)C1 Cc1cc(C=CC(=O)NC2CC(=O)N(C3CN(C(=O)C(C)N(C)C)C3)C2)on1 C(=O)(CCC(=O)NC1CN(C(=O)Cc2ccns2)C2CC12)NCCNC(C)=O c1(C(=O)NCC(C)(CO)NC(=O)C(c2ccc(Cl)cc2O)=O)cn2c(n1)CCC2 c1(NCC2(NC(c3[nH]nc(OC)c3Cl)=O)COC2)nc2c(cc1Cl)C(=O)OC2 C1(C(N(C(CC)CNC(c2cnc(N(C)C)nc2)=O)C)=O)CCC=CCCC1 c1(OC)ccc(C=NOCC(N2CC(c3ccc([N+](=O)[O-])cc3)C2)=O)cc1 C(=O)(CCCCCC(C)C)NCCCCC1CN(C(c2cc(C)cc(F)c2)=O)C1 C(=O)(CC(C)NC(N)=O)NCC1CN(C(C(c2ccn(C)c2)C)=O)C1 C(=O)(C1CNc2ccccc21)NC(C)CNC(C1CC2(C1)CC2F)=O C1(COC)CN(C(=O)C=C(C)CNC(=O)Cn2cc(Cl)cn2)C1(C)C C(=O)(C1=NOC(C(=O)NC2CC(CO)N(C(c3cccnc3S)=O)C2)C1)OC N1(C(C2C(OCC)C2)=O)CC2CCCC2C1C(=O)NC(C)COC(=O)NC C1(O)(C(=O)OC)CCN(C(C(=O)Nc2ccccc2Cl)c2cnc[nH]2)C1 C12(NC(C(F)=CC)=O)CCC(CN(C(c3cnc(OCC)cn3)=O)C1)C2 c1(N2C(=O)CC(C(=O)NCC(CC)NC(=O)CN3CC=CC3)C2)c(C)nn(C)c1C N1(C(c2c(C)cc(C)c(C)c2)C(=O)NCC(F)F)CCC2(CC1)CN(C)C(=O)O2 O(NC(=O)C(CNC(=O)C=NOC)N(C)C)CC#C C1(NC(c2c(OC)c[nH]n2)=O)CN(C(c2csc(CC(C)C)n2)=O)C2(CCC2)C1 N1(C(C(CC)OCC)=O)CC=C(C(=O)NC2(C)CC(O)C2)C1 C12(CNC3(N4CCCC4)CC3)CN(C(C3(CS(N)(=O)=O)COC3)=O)CC1CCO2 C(=O)(C1=NOC(C)C1C)Nc1c(C)cc(NC(c2cncn2C)=O)cc1 C1(C)(C(=O)NC(C2CN(C(C(CC)SC)=O)C2)C)CCC(F)(F)CC1 Cc1c(C(F)F)cccc1C(N1CCOC(C(C)(C)C)C1)C(=O)NCCSC c1(C(=O)NCCOC2CCN(c3cncc(C(=O)OC)n3)C2)ccc(C)c(F)c1 c1(C(=O)NCC2(F)CCC(NC(C3(SC)CC3)=O)C2)nccc2ccncc12 c1(C(=O)NC2C(CNC(=O)CCSC3CCCC3)C2)ccc2cncn2c1 c1(CCC)n[nH]cc1C(N1CCCC1CN(C)C(C1CC1c1ccoc1)=O)=O C12(C(=O)NCCC3CCC3)COC(C(=O)O)(C1)C2 C1(CN(C(c2cc(OCC)c(OC)cc2)=O)CC)CCc2ccccc2C1 C=CC(C)(O)C(=O)NC1CC1NC(c1cc(Br)ccn1)=O Cc1cc(Cl)c(C(N2CCCCC2CC2(O)CCCCC2)=O)s1 N1(C(=O)CCCCC(F)F)CCCC2(C1)CN(C(=O)CC1CCS(=O)(=O)CC1)C2 N1(C(C(CO)NC(=O)CN2CC=CC2)=O)CCCc2ccccc21 c12ccccc1CCn1cc(nn1)CC(=O)N(CCF)C2=O.c1(C)nc[nH]n1.CO C(=O)(C1CCc2c[nH]nc21)NC1CC(NC(C(C(=O)OC)C)=O)C1 C1(NC(c2n(C)nc(CNC(=O)CCNC(=O)CO)c2)=O)CCC=CCCC1 c1(C(=O)NC(CN(C(c2cc(CSCC)on2)=O)C)CC)cccc(Cl)c1C c1(C(N2CCC(C(C)NC(c3c(OCC)ccs3)=O)C2)=O)nnn(C)c1N CCCCCS(=O)(=O)CC(=O)N(C)CCOCCN(C)C(c1c[nH]c(C#N)c1)=O CC(C)CC(CNC(C1CCOC1(C)C)=O)C(=O)NCc1ncc(CO)[nH]1 C(=O)(C1(CC)CCCc2ccccc21)N1CCC2(CN(C(C(CC)OC)=O)C2)C1 c1(CNC(C2C(COC)CC2)=O)cc[nH]c1C(=O)NCCC1CCC2CC12 n1(CCCC)ncc(C(=O)N(C(C)CNC(c2cnc(O)s2)=O)C)c1C C(C(C)C)(C(O)C(=O)N1CCN(CC(N2CCN(C(C)=O)CC2)=O)CC1)OC c1(C(N(CCCCCCNC(C(CC)(C)C#N)=O)C)=O)c[nH]nc1S(N)(=O)=O n1(CC(=O)NCC(C)(C(C)C)NC(COCC#C)=O)cc(C#N)c(O)nc1=O c1(CC(=O)N(CCNC(=O)C=C2CCOCC2)CC)cc(N2CCCC2)ccn1 N1(CCC(=O)NC2C=CCN(C(C=C(C)Cl)=O)C2)C(=O)c2ccccc2S1(=O)=O c1(C(N2CCC(CNC(C(C)C3CC3)=O)CC2)=O)nnn2c1C(=O)NCC2 CC(C)(C#N)CCCC(=O)NCCCC(O)C(=O)NCC1(C)CCCC1 c1(NC(C2(C)CCN(C(C(C)NC(C)=O)=O)CC2)=O)ccc2nsnc2c1 CCC(C#N)(CC)C(=O)N1CCC(C(=O)NCC2(O)CCCCC2)CC1 c1(C(N(C)CCOCCCN(C(=O)C(F)n2ccnc2)C)=O)ccc2c(c1)CC2 C1(C)(C(=O)NC(C2CCN(C(c3cncnc3)=O)C2)C)CC=CC1 Cc1ccc(O)c(CC(=O)NCCC2CN(C(c3n[nH]c(C)c3Br)=O)C2)c1 C1(C(C)(C)C)CCCC(NC(=O)NC(CNc2cnsn2)C2CCC2)C1 c1(CN2C(CC(=O)Nc3ccc(O)cc3Br)COCC2)cccc2cccnc12 N1(C(C2N(C(CC)=O)CSC2)=O)C2CCC1(CNC(=O)Cn1cnnn1)CC2 C12(CC)CC(C(=O)NCCC3COCCN3C(=O)C(F)F)(CO1)C2 N1(C(C=Cc2ccc(CC)o2)=O)CC(NC(C2CSCCS2)=O)CC1(C)C CC(C)C1=CCC(NC(C2N(C(=O)CC(O)CN(C)C)CCC2(C)C)=O)CC1 c1(CC(=O)NCC(C(C)C)(C)NC(=O)Cc2sc(O)nc2O)ccc(Cl)c(F)c1 CC(C)C(O)CC(=O)NC(C1CN(C(=O)C(c2ccc(F)cc2F)(F)F)C1)C c1(C(=O)NC2CCN(Cc3c(OC)ccc(Br)c3)C2)ccc2nc(C)oc2c1 C=CCC(CC(=O)N=c1cc(OC)n(C)[nH]1)NC(=O)CCC(C)OC C1(N(C(C(C)C2CCOC2)=O)C2CC2)CCN(C(=O)OC(C)(C)C)CC1 c1(C(=O)NC2(CCNC(C3(C)CCC(OC)CC3)=O)CC2)cc(C#N)ccc1N C1(C2CCN(C(=O)C3=NOCC3)CC2)(NC(CCCCN(C(C)C)C)=O)CCC1 c1(OC)ccc2c(C(=O)NCC3(C)CCCN3C(C3CCC3(C)C)=O)c[nH]c2c1 c1(CC)ccc(C(=O)NCC(C(C)(C)C)NC(=O)CN2CCOCC2)cn1 Cc1nn[nH]c1CNC1CC1c1cncs1.N1CCCC1COC CC1CC(NC(c2ccc[nH]2)=O)CN(c2nnc(-c3cccn3C)n2C2CC2)C1 N1(CC)C2CCC1CN(C(=O)CCC(C)NC(=O)CC(C)c1ccco1)C2 c1(C(=O)NCCC2OCCN(C(C(CC)(C)CO)=O)C2)ccc(S(N)(=O)=O)nc1 N1(CCC2(CCC=C)N=N2)CCC2CCN(C)CC12 C1(N(C(C(CC)CC)=O)C)CCN(C(c2cncc3c2CCC3)=O)CC12CC2 Cc1c(O)nc2ccccc2c1C(=O)NC1CC1NC(=O)C(CN(C)C)C(C)C C1(N(C(c2nc(C)no2)=O)CC)CCCN(C(=O)CC2CCCCC2C)C1 C1(NC(Cn2ccc(C)n2)=O)CC12CCN(C(C1CCC(C(N)=O)O1)=O)CC2 C12(C(N3C(C)(CCO)CC3)=O)CC1CN(C(c1ccc(C3CC3)o1)=O)C2 C=C=CC(C)C(=O)NCc1ccc(C(N2CC(CC)C(O)C2)=O)nc1 N1(CC(=O)NC2C(CNC(c3c(C)nncc3)=O)CCCC2)CC(=O)N(C)C1=O N1(C(c2c(OC)c[nH]n2)=O)CC(NC(=O)C(C(C)C)NC(C)=O)CC(F)C1 C1(O)(CNC(C(C)=CC)=O)CC2CCC(C1)N2C(c1cc(CC)n(CCO)n1)=O c1(C(N2CCN(CCNC(C(CCSC)O)=O)CC2)=O)nccc(C)c1F S(=O)(=O)(c1ccc(N2CCOC(CCO)C2)c(Cl)c1)N1CCCCC(C)(F)C1 C(=O)(C1Cc2c(Cl)cccc21)NC1C(NC(CC(=O)OCC)=O)CC1 N1(C(C2C(C)OC(=O)N2)=O)CCC(C)(C)C(CNC(c2cc([N+](=O)[O-])c[nH]2)=O)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCCC(N(C)C(c2cc[nH]n2)=O)CC1 CN1C(=O)NCC1C(=O)NCCC1CN(C(=O)CCSCc2ccccn2)C1 C(=O)(CCCC(C)(C)C#N)N1C(C(=O)NC(c2c[nH]ccc2=O)C)CCCCC1 N1(C(C(CC(=O)OC)C)=O)CCCC2(NC(=O)CCCn3ccnc3)CCCC12 C(=O)(C(CCC1CC1)NC(C12CCC(OC)C1C2)=O)N(CC#C)CCO Cc1cnc(F)c(C(N2CCC(C)C(CNC(=O)CCC3CCCCC3)C2)=O)c1 N1(C(C2C(CNC(CC(COC)COC)=O)OCC2)=O)CCOCC(F)(F)C1 C12(C(=O)NCCN(CCC)C(c3cncs3)=O)CC(C)(C1)OC2C C1(CNC(c2nn(C)c(O)c2)=O)CCN(C(=O)COC2CCCOC2)C12CC2 C1(CCO)(NC(C2CC(O)CN2C(c2cc[nH]c2)=O)=O)CCCCC1 C12(CNC(c3sccc3C(F)F)=O)CC(CN1C(=O)C=CI)C2 c1(C(N2CC3C(NC(C(CCOC)OC)=O)C3C2)=O)cc(SC)cc(Cl)c1 CC(C)CC(CC(C)C)C(=O)NC1CN(C(C2CS(=O)(=O)CC(=O)N2)=O)CC1F N1(C(CCSCC)=O)CCC2(CCCC2NC(c2cc([N+](=O)[O-])cn2C)=O)CC1 C1(NC(C(N2CCOCC2)C)=O)CC2(C1)CC2NC(=O)C(O)CC1CCCC1 C1(C2CC2)(NC(C2C(C)C2)=O)CCN(C(=O)C(C)(C)N2CCCCC2)C1 N1(C(CC(=C)C)=O)CCC(N2CCC(NC(c3ccc(CO)cc3)=O)CC2)CC1 CCCCC(C(=O)N(CCCNC(c1ccnc(COC)c1)=O)C1CC1)N(C)C Cc1nccc(CCC(N2CCC(C)(NC(C3CC3(C)C)=O)C2)=O)n1 C=C(C)CCCC(=O)N1CCC(N(CCO)C(c2c[nH]c(C#N)c2)=O)C1 c1(C(=O)NCC2CC(F)(CNC(=O)CC3CCOCC3)C2)cncnc1C1CC1 Cn1ccn2c(CCNC(=O)NC3CC4CCC3CC4(C)C)nnc2c1=O c1(C(N(CC(C)N(C)C(c2cscc2Br)=O)C)=O)ccc2cc[nH]c2n1 C(C)(C)(C(=O)NC1CC(CC(=O)N(C2CN(OC)C2)C)C1)NC(=O)NCCC Cn1nc(Br)cc1CC(=O)NC(CNC(=O)CNC(=O)NC1CC1)C1CC1 c1(-n2ncc(C(N(C)CCN(C)C(C3CCC(C)(C)O3)=O)=O)n2)ccc(Cl)cc1 C1(NC(=O)C(C2CCN(C(c3ccon3)=O)C2)F)CC2CCC1O2 C1(C(N2CC(O)(CNC(CCC=CC)=O)C2)=O)Cc2ccc(F)cc2O1 CC(C)CC(F)C(=O)NCC(C)CNC(=O)C=CC(=O)NC1CC1 N1(C(c2cnc(CC)nc2O)=O)CCC2C(C1)CN2C(c1cscc1C)=O C1(CNC(C(CC#C)C2CC2)=O)COCCN(C(c2cc(C)c[nH]2)=O)C1 CC1CCC(=CC(=O)NC(C2CCCN(c3nc(CC4CC4)ns3)C2)C)CC1 C(=O)(C(Cn1cncn1)NC(c1nnsc1C)=O)NC(CC)C1CCC1 N1(C(C(C2CN(C(=O)C(C(C)C)NC(C)C)C2)OC)=O)CC2CCCC2C1 C12(CNC(C(CC)(C)C)=O)CCC1CCN2C(=O)CCCc1cccs1 N1(C(c2c(C)c[nH]n2)=O)CCN(C(=O)Cc2ccnc(F)c2)C(CCO)C1 c1(CC(N2C(C3(O)CN(C(C(CC)SC)=O)C3)CCC2)=O)cc(Cl)ccc1Cl n1(CC#C)c(C)cc(C(=O)NC(C2CCOC2)CNC(c2cn(C)nn2)=O)c1C Cc1ccc(CS(=O)(=O)NCC2CCN(CC34CC(CCO3)C4)C2)c(F)c1 C1(C(N2CC3(CCC3)C2)=O)CC1C1CN(C(C2(F)CC=CC2)=O)C1 c1(C(=O)NC2CCN(C(CCCN(C)C)=O)CC2O)cc2cc[nH]c(=O)c2s1 c1(C(=O)OCC)cnc2c(C)cc(C)cc2c1NC.N12CCCC(C1)C2=O c1(NCc2c(C(=O)OCC)scc2)ccc(-c2ncn(C)n2)cc1 c1(N2CCN(C(=O)Nc3cccs3)CC2)nc(Cl)nnc1Cl C=CCC(C(=O)N1CC2CC2(C(=O)NCC2CCCC2(C)C)C1)NC(C)=O C(=O)(C1=NNC(=O)CC1)NCC1CCN(c2ccnc(C(CC)C)n2)C1 N1(C(c2c(C)nc(CO)s2)=O)CCC(NC(=O)C2=CCCCO2)C(C)C1 C(=O)(C1=CCOCC1)N1CCC(C(N(CCC=C)CC)=O)C1C(C)C C#Cc1cc(C(=O)NC2CCOCC2C)cc(I)c1 N1(C(c2c(CC)nco2)=O)CC(CNC(=O)C=Cc2ccc(C)o2)OC(C)(C)C1 c1(NC(N2CCC(N(c3ccc(Cl)cc3Cl)C)CC2)=O)ccc([N+](=O)[O-])cc1Br C(=O)(C(C)(CNC(=O)CNC(c1ccc(OC)c(OC)c1)=O)S(C)(=O)=O)OC C1(C(=O)NCC2(CCNC(C=C(C)C)=O)CC2)CC2CC(C1)CC(F)(F)C2 C1(C(=O)NC2(C(N(CC(=O)N(CC)CC)C)=O)CC2(C)C)CCCC12CCC2 C#CC1(O)CCN(C(=O)C(C)NC(=O)C(CC(C)C)NC(C)=O)C1 c1(C(N(C(C)C)CCNC(=O)C#CC(C)(C)C)=O)cc([N+](=O)[O-])ccn1 C(=O)(CCN(OC)C(=O)C(CNC(C1(C)CC(C)C1)=O)OC)OC C(=O)(C(C(C)(C)C)NC(N)=O)NCC(CNC(Cc1n(C)ncc1)=O)CO N1(C(c2cnc(CC)s2)=O)CCC(C(C)C(=O)NCC2(C(F)(F)F)CC2)CC1 N1(C(CCn2c(C)ccc2C)=O)CCC(CNC(=O)C2=C(Cl)CC2)CC1C C1(C(=O)NCC2CN(C(Cn3ccc(C)n3)=O)CC2C)CCc2nnn(C)c2C1 C(=O)(C(C)(O)CC(C)C)NC(CC(C)NC(C(CC=C)N(C)C)=O)C C1(CC)CN(c2ccccc2CC(=O)NC(=O)NC)CCN1Cc1ccccc1 N1(C(c2c(C)nc(COC)s2)=O)CC2CC(NC(C3CC4CCC3O4)=O)CC1C2 C(CC(F)(F)F)(c1ccccc1)NC(c1noc(C2CCC2)n1)C N1(C(C(CC)(F)F)=O)CCN(C(c2cn(CC3CCOC3)nn2)=O)C2(CCC2)C1 c1(C(=O)NC2C3CN(C(C(F)=CC)=O)C2C3)ccc([N+](=O)[O-])c(C)c1 CCCC(C(F)(F)F)NC(=O)C(CNC(=O)C(C)(COC)CC)C(C)C C1(NC(C2N(C(CCN(C)CCO)=O)C(CO)C2)=O)CC(O)CC(C)(C)C1 C1(NC(c2c(COC)nn[nH]2)=O)CN(C(C2CC(C)(C)CCO2)=O)C(C)(COC)C1 c1(SC)ccc(-c2ccc(CN3CCCC3Cc3cccc(C)n3)nn2)c(C)n1 c1(C(=O)NCCCC(C)NC(C2CCSC2)=O)ccccc1F Cc1cn2c(CC(N3CCCC(C)(C(=O)N(C4CCN(C)C4)C)C3)=O)csc2n1 c1(C(N(C2CCN(C(C3CNC(=O)C3)=O)C2)CCC)=O)coc2c1CCCC2 N1(C(C(c2n(C)ccc2)=O)=O)CC2CC1CN2S(=O)(=O)Cc1ccc(F)cc1F C1(C(=O)NCC#CCNC(Cn2c(C)cc(C(F)F)n2)=O)CCCC(=O)N1C C1(NC(c2c(CC)oc(C)c2)=O)CN(C(C2CC(=O)N(C3CC3)C2)=O)CCC1F c1(N2CC(C)C(N(C)C)CC2)nc(N2CCCC(C)CC2)nc2c1COCC2 C1(NC(=O)NC(c2cccc(OCC#N)c2)C)CC(N)C(O)C1 NS(=O)(=O)CCC(=O)NCC1CC2CC2N1C(=O)CCc1ccc(C(F)F)cc1 C1(CCCNC(C(C)(F)F)=O)CCN(C(c2cc(Cl)no2)=O)CC1 c1(OCC(=O)NCC(C(C)C)NC(C2COC(C)(C)C2)=O)ccc(C(N)=O)cc1 CN=S(C)(=O)CCNC(C1CSCN1C(C1CCC1)=O)=O C1(S(C)(=O)=O)(C(=O)NC2CCCN(C(C3(OC)CC(C)C3)=O)C2)CCOCC1 C(=O)(CCCS(N)(=O)=O)NCC1C(NC(c2ccc(CC)c(OC)c2)=O)C1 Cc1nnc2n1CCC(CNC(NC1CCc3sc(Br)cc31)=O)C2 C1(C#N)(C(N(CCCC(=O)NCCC2ON=C(C)C2)C)=O)CC1(C)C CN1CC(C(=O)NCC2CC2NC(=O)Cc2nn(C)cc2Cl)CC1=O C(=O)(C(=O)NNC(=O)c1ncccn1)Nc1c(CC)ccc(C(=O)OC)c1 C1(NC(C2C3(CCN(C(C4(C#N)CCC4)=O)CC3)C2)=O)CCOC2(CCOCC2)C1 C=CCC(C)(C)CC(=O)N1CCN(C(=O)CC2SC(=N)NC2=O)C(C2CC2)C1 C=CCC(C)(C)C(=O)NC1CCC(C(=O)NCc2ccccc2CO)C1 C1(NC(CC=C)=O)CCCN(C(=O)C(c2ccccc2OC)OCC(F)(F)F)C1 c1(C(N(CCCNC(C2(CCCC)CC2)=O)C)=O)cnc2n1CC(C)CC2 c1(C(N2CCC(C(=O)NCCCOC(=N)O)(OC)C2)=O)cnc(O)cc1C C1(CNC(=O)CCF)CCCCN1C(c1csc(Cc2ccccc2)c1)=O C1(CCN(C(=O)C(C#N)C2CC2)C)CCCCN1C(c1cnns1)=O c1(C(N(CC(C)NC(c2onc3ccccc23)=O)C)=O)c(Cl)ccc2c[nH]nc12 c1(CCCC)nc(C(=O)NCC=CCNC(C23CC(C2)C3)=O)cs1 C(CC)(C(=O)NCCN(C(C)CC)C)NC(CN(CCC)CC)=O C1(CCNC(c2c(CC)nns2)=O)CCCN(C(=O)CS(=O)CC)CC1 c1(C(N2C(CNC(Cn3ncc(C)c3)=O)CC2)=O)c(C)ccc(C)c1C c1(CNC(C(=O)N(C)C)=O)cnc(CCNC(=O)COC2CCOC2)[nH]1 c1(NC(N2C(c3n(CC)ncc3)C(C)(C)CCC2)=O)nc2ccc(O)nc2s1 C(=O)(C(F)C(C)(C)O)NC(CCOC)CNC(c1cccc(CC(C)C)c1)=O CC1(C)CCN(C(c2cccc(Cl)c2)=O)CC1NC(=O)C1=CCOC1 N1(CCCNC(CN(C(C)C)C)=O)CCC(NC(=O)Cc2cnns2)C1 Cc1cnc(N)c(C(=O)NC2CC3(C2)CN(C(C2CCCCNC2=O)=O)C3)c1 c1(C(N(C2CCCCC2)C)=O)ccc(NC)cc1.N12CC3CC1(C3)C2 c1(C(=O)NC2(c3cn(Cc4cc(C)on4)nn3)CCC2)c(C)c(C)nn(C)c1=O N1(CC(N2C(CNC(C3(C=C)CC3)=O)CC2)=O)CCN(C2CC2)C1=O c1(N2CC(C)CS(=O)CC2)nc(NCCCc2ncco2)c2ncn(C)c2n1 c1(N(C)C)nc(C(=O)NCC2(NC(=O)CNS(N)(=O)=O)CCC2)cc(O)n1 C1(CN(C(=O)CCC2CCCC2)C)CCN(C(c2c[nH]nc2C2CCC2)=O)C1 c1(C(N(C2CCCN(C(=O)Cc3ccc(Cl)cc3)C2)CC)=O)cncc(CO)c1 C#Cc1ccc(CC(=O)NC2C3CCN(C(c4ccn(CC)n4)=O)CCC23)cc1 CN1CCCCC1CC(=O)NCC1CC(C(=O)NCCC2CC(F)(F)C2)C1 c1(C(N2CCC(C)C(N(C(=O)CC3(C)CC3)C)C2)=O)cccc2c1CCOC2 c1(CC(=O)NCC(CNC(c2nn(C(F)(F)F)cc2Cl)=O)CO)cccc(O)c1 C1(NC(COC(CC)C)=O)CCSC12CN(C(c1cc(O)n(C)n1)=O)C2 C(CCCOC)(C(=O)N1CCOCC(O)C1)NC(C(F)=CCC)=O C#Cc1cccc(NC(=O)CC2CC(NC(=O)NCc3cc(Br)cnc3C)C2)c1 CC(C)CC(CNC(c1cccnc1C(F)(F)F)=O)NC(C1CC(C)(C)C1)=O C=C=CC(C)C(=O)NC(C)(C)C=CC(=O)N(C)CC1(N(C)C)CCC1 c1(C(N2CCN(C)C(CNC(C3CC3CF)=O)C2)=O)nn(C)c2c1CCCC2 C1(C(=O)NCC(O)Cn2cccn2)(NC(C=CC(CC)C)=O)CCOCC1 c1(C(N(CC(C)C)OCC)C)nc(C(C)C)cc(Cl)n1.C1(C)(C)CC1 N1(C(C(CC)C)=O)CCC2CCN(C(c3ccc(-n4ccnc4)cc3C)=O)C2C1 c1(C(=O)NC(C(C)C)CCN(C(=O)C(F)=C2CCCC2)C)ccc(Cl)c(C#N)n1 C1(CC(=O)NCC(C)NC(c2c(C(=O)OC)coc2)=O)CCCS(=O)(=O)C1 c1(C(C(=O)NCCC2CCCN2C(=O)CCN2CCOCC2)O)ccccc1Cl C1(O)(CNC(C(C2CCC2)OCC)=O)CCN(C(C2CN(C3COC3)C2)=O)CC1 C1(CC#C)(C(=O)OCC)CCCN(C(c2ncccc2-c2nncn2C)=O)C1 C12(C(=O)NCC(CC)NC(=O)CSc3ccccc3Cl)CCCC1OCC2 CCCC(CCC)CC(=O)NC1COCC1CNC(=O)CC(C)c1ccccc1 C(C(=O)N=c1cc[nH]cc1)NC(=NCCc1nc(C)sc1)NC1CC1C c1(C(N(CC(C)CNC(=O)C=Cc2ccncc2)C)=O)ccc(N(C)C)c(F)c1 c1(C(N2CC(N(C(CCOC(C)C)=O)C)C3(C2)CC3)=O)c(Cl)cccc1[N+](=O)[O-] C(=O)(C1=CC2C=CC1C2)N(CC1N(C(Cc2cc(C(N)=O)sc2)=O)CCCC1)CCl c1(C(C(=O)NCCC(=O)OCC)N(C2CCNC2=O)C)ncc(Cl)cc1F N1(CC)CCCCC1C(=O)NCC(C)CC(=O)NCC(CO)N(C)C c1(OC)c(C(=O)NC2CC(CNC(=O)CN(C)C)CC2O)c(C)nn1C N1(C(C(CC)(C)OC)=O)CC(C)C(C)(CNC(=O)CCCCSC)C1 C1(CN(C)C(c2ccoc2C2CC2)=O)CN(C(c2cccc[n+]2[O-])=O)CC12CC2 N1(CC(=O)NCC2(CNC(c3cc(C(N)=O)oc3)=O)CC2)CCCCCC1 n1(CCN(C(C2(CC)CCC2)=O)C)cc(CC(O)C(=O)N(C)CC)nn1 C1(NC(C(CC)n2cncn2)=O)CC(C)CN(C(=O)CNC(c2ccoc2C)=O)C1 c1(CCC(N2CC(N(C)C(c3csnc3Cl)=O)C2)=O)nnc(S)nc1O c1(C(=O)NC2CC(CNC(C3(O)CCCCC3)=O)C2)ccnc2[nH]ncc12 c1(OC)ccc(N2CCN(C(c3cc(OC)ccn3)C)CC2)cc1 C1(CC(=O)NCc2occ(C(=O)NC3(c4nc(C)[nH]n4)CC3)n2)CCN(C)C1=O c1(CCC(=O)NC2(COC)CN(C(C3(O)CCOC3)=O)C2)c(Cl)cccc1Cl c1(C(C(=O)N(CCNC(C2CCN(C)C2C)=O)CC)(F)F)cc(Cl)ccc1OC Cc1cncc(CC(=O)N(C)CC2CN(C(c3cnc(N(C)C)s3)=O)C2)c1 C1(CC)CN(C(C2(CCF)CCOCC2)=O)CCN1C(=O)CC(C)c1ccco1 C1(CC(N2C3CN(C(C4C(COC)C4)=O)C(C3)C2)=O)CCC2(CCC2)CO1 C(CO)(CN=c1nc(N2CCC(SC(F)F)C2)c2c([nH]1)COC2)OC S(=O)(=O)(c1c[nH]c(C(=O)NCCCNC(C2COC(C)(C)CO2)=O)c1)N(C)C c1(C(=O)NC(C)CC2CCN(C(C3CC3C#N)=O)CC2)cc2ccncc2[nH]1 CC1CN(C(c2cnn(C)c2-c2ccc(F)cc2F)=O)CC(C)C1(F)F Cn1cc(Cl)c(CC(=O)N(CC(F)F)CC2CC2)n1 N1(c2ncc(C)cn2)CC2COCC2(C(=O)N(C2CC2)Cc2ccncc2)C1 Cc1cc(C(=O)NCc2cc(C(=O)NC(c3ccnn3C)CO)n[nH]2)c(N)s1 N1(C(C=CCC)=O)CCN(C(=O)CC(C)C(F)F)C(c2ccnn2C)C1 Cc1cc(Cl)ccc1Sc1ccc(NC(=O)NCC(N2CCOCC2)(C)C)cc1 C1(NC(C2CCC=CO2)=O)CN(C(C2CCCNS2(=O)=O)=O)C2(CCOCC2)C1 CC1CC(NC(c2ncoc2Br)=O)CN(C(=O)CC2CC3(CCC3)C2)C1 N1(C(C2CCN(CC)C2)=O)CCC(C(=O)NCC2CC3CCCC3C2)=C(F)C1 N1(C(C(CCC)O)=O)CCC2(C1)CN(C(=O)C(C)N1CCCC1)CCO2 CCC(CC)CC(F)C(=O)N1CC(C)N(C(=O)CC23CCCN2CCC3)CC1C C(=O)(C1=NOCC1)N1CCC(C(C)C(N2CC=CCC2)=O)C1 CC(C)(C)CC(O)CC(=O)NCCCCC(=O)N1CCC(n2ccnn2)C1 c1(C(=O)Nc2c(CC)cccc2OC)ccc(O)c(C=O)c1 N1(C(c2cc(CNC(C3(OC)CCC(C)C3)=O)oc2)=O)CCC(O)C(C)(C)C1 N1(C(CC2(C)CNC(=O)C2)=O)CCOCC(C(=O)O)C1 C1(C(N2C(C3(C(N(C)Cc4c(C)n[nH]c4)=O)CC3)CCC2)=O)OCCCC1(C)C CC1Cc2cc(C(N3CCNCC(CO)C3)=O)ccc2N1 Cc1nnc2n1CCCC2C(=O)NC1C2CC1N(C(c1ccc(F)c(O)c1)=O)C2 Cc1nccc(C(=O)NCCCCC(C)NC(C2C3CCCOC23)=O)n1 c1(C(=O)NCCC2CCCCN2c2cc(C(F)F)ncn2)ccnc2[nH]cnc12 N1(C(CCc2ncc(C)[nH]2)=O)CC2CC(C1)N(C(C13CCN(CC1)C3)=O)C2 c1(OC)ccc(C(=O)NC2CC23CC(NC(=O)Cc2cncn2C)C3)c(O)c1F C12(C(N3C(CC)CC(O)C3)=O)CCN(C(c3ncc(F)cc3F)=O)CCC1C2 C=C(Cl)CCC(=O)NC(C1(O)CCCCC1)C(=O)NCC1CC1(C)C Cc1nc(CCC(=O)NCC2CCCN2C(c2ccc(C3CC3)cc2)=O)[nH]c1C C12(C)CCN(CC1)C2=O.c1(SCC=C)cccc(CCc2ccccc2)c1 CC1C2CC(C2NC(=O)CCC2(C)CC2)N1C(C1CC(=O)NC1(C)C)=O N1(C(C2CCN(C(c3c(C)cncn3)=O)CC2O)=O)CC2(CCOC2=O)C1 c1(N(C(CC)C)Cc2ccco2)ncnc2c1ncn2C(C)CO c1(OCC(=O)NC2CC(CCNC(=O)C(F)=C3CCCC3)C2)cccc(Cl)c1 C(=O)(C1CCCc2n[nH]cc21)N1CC(CNC(c2c(C)nns2)=O)C(C)CC1 CC(C)(C)C(O)CC(=O)N1CCCC(NC(=O)C(C)(O)C(F)(F)F)C1 CC1NC(=O)C2=C1N(C1CCCC1)C(=O)NC2c1ccnn1C1CCC1 N1(C(N(C(C)(C)C)CC(=O)Oc2ccccc2)=O)CC(O)(N2CCC2)C1 c1(C(=O)NC(CNC(c2c(OC(C)C)cccn2)=O)C)ccc2cccnc2c1 N1(C(C(C)C2CCC2)=O)CCS(=O)(=O)C(CCNC(c2cccc(O)n2)=O)C1 C1(C(N(CCC(=O)NCCc2cc(C)no2)CC)=O)CCCOCC1 N1(C(C(C)O)=O)CC(C)(C)OCC1CNC(=O)Cc1csc(Cl)c1 Cc1cncnc1C(N1CC(CNC(C2(C)CS(=O)(=O)C2)=O)C(O)C1)=O c1(C(=O)OC)cc(C#N)cnc1NCC(O)CNC1(F)CCOC1C c1(C(N(CC(C)NC(c2ccn(C3CC3)n2)=O)CC)=O)cnn2c1OCC(F)C2 C1(C(C(=O)N(C)CC2C3CN(C(c4c(C)scn4)=O)CC32)O)CCS(=O)(=O)CC1 C1(C)(CNC(C2C(C)CCO2)=O)CCC(NC(C2CC(F)(F)C2)=O)CC1 c1(C(=O)NCC2(CNC(C3C(C)(CC)C3)=O)CCCC2)c(Cl)ccc2c[nH]nc12 c1(CNC(C(C)N(CCC)C(c2ncc(F)cn2)=O)=O)cc(O)ncn1 CC1CC(=O)NCCN1C(C1CN(C(=O)C(C)C(F)F)CCO1)=O C1(C(=O)NC2(CNC(C(C)(F)F)=O)CCOC2)C2CCCCC12 Cc1c(C(NC=CC(=O)C(F)(F)F)=O)[nH]c2cc(C(=O)O)ccc12.C(C)(CC#N)N C12(CC(=O)N(CC)Cc3cccs3)CCC1CN(C(=O)CC1CCCN1C)C2 O=C(C(C(F)(F)F)C(F)(F)F)NCCn1cc(-c2ccc(Cl)cc2)nn1 N1(C(c2cc(COC)on2)=O)CC2(CCN(C(C34CC(F)(C3)C4)=O)C2)C1 C(=O)(C1=CCC(C)(C)CC1)NCC(CNC(C(C)(C)N(C)C)=O)O C1(C(=O)NC2C(CNC(Cc3nc(C)[nH]n3)=O)COC2)CC2CCC1CC2(F)F N1(CCC)CCCC1C(=O)NCC1CCCN1C(=O)C(=O)Cc1cccs1 C(C(F)(C(=O)N1CCC(O)CC(C)C1)C(C)C)NC(C1C(C)CC1)=O CC1(C)CCCCC1=CC(=O)NC1CCCC1NC(=O)COCP(C)(C)=O C1(CC(=O)NCc2ccc(Br)s2)COCCN1Cc1ccco1 N(C(=NCCCOC)NCc1ccsc1)CCC1(O)CC1C(F)(F)F.N1CCCC1 N1(C(CC2(CSC)CC2)=O)CCN(C(=O)CC2CCC(C)(C)CO2)CC1C c1(C(N2CC=CC(NC(C3CCCN3C3CC3)=O)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 CC(C)C(O)CC(=O)NCC1CN(C(c2cncc(C(F)F)c2)=O)C1 c1(-c2cnc(Nc3cncc(-c4cc(C(C)=O)ncc4)c3)s2)ccc(F)c(C)c1 C(CC(C)C)(C(=O)NCC1CC1NC(c1cnc(S)n1C)=O)NC(C)=O C(=O)(C1=C(C)CCOC1)N(C(C(N1CC(OC)(CO)C1)=O)C)C1CC1 CC1CC(C(=O)NCC2CCN(C(c3cnc(C(F)(F)F)cn3)=O)C2)CC(=O)N1 c1(C(=O)NC2CC(CNC(C34C(C)(C)OCC3C4)=O)C2)ccnc2ncccc12 c1(CC)c(C(=O)NC2(C)CN(C(=O)C(CO)NC(N)=O)C2)nnn1C C1(C2CC2)(C(=O)NCc2c(C(C)C)con2)CN(C(=O)CCCCN(C)C)C1 c1(C(N2CCC(CNC(C(C)OCOC)=O)C2)=O)ccc(Cl)nc1OC c1(NC(CC2N(C(C(C)OCC#C)=O)CCOC2)=O)cnc(OC)c(C)c1 CCC(C)C(C(=O)N1CCC(NC2CC2)CC1)N(C(=O)CS(=O)(=O)NC)C C(CC)(CCC(=O)NC1(CN(C)C)CC1)NC(C(CC)NC(C)=O)=O N1(C(C(C)CO)=O)CC(NC(c2cnc(C3CC3)[nH]2)=O)CC(F)(F)C1 C1(CNC(C(C)(C)NC(=O)NCC)=O)CCCCN1C(=O)Cc1cnc(C)s1 C(=O)(CC(CC)CCCC)N(CCC(=O)N(CC=C)CCO)CC1CC1 c1(CC)ncc(C(=O)NCCC(CNC(=O)CC2C(C)C2(F)F)OC)s1 Cc1cc(COC)oc1-c1nc(CCN(C)C2CC2)nn1C(C1CCC1)C C1(NC(CC2(C(F)(F)F)CC(=O)NC2)=O)CN(C(C2CCC2)=O)CCC1CO N1(C(CC2(C)CCCCC2)=O)CCC(NC(=O)COC2CCOCC2)C(CO)C1 c1(CC(=O)NCC(CNC(=O)C(C)NC(C)=O)OC)ccnc(F)c1F c1(OC)ccc(Cl)c(CC(N2CCC(F)C(NC(C3(CO)CCC3)=O)C2)=O)c1 C1(NC(=O)OC)CN(C(=O)C(=O)Nc2nc(-c3cccc(I)c3)cs2)CC1C C1(C2CCN(c3cc(C(C)C)ncn3)C2)(NC(C(CC)NC(C)=O)=O)CC1 C1(C#CC(=O)NC2CC(CNC(=O)CNC(c3cccs3)=O)C2)(CC)CC1 CCC(C)(F)C(=O)NCC1C=CCN1C(c1ccc(C2(C)CC2)cc1)=O N1(C(C=COCC)=O)CCN(C(c2ccc(Br)nc2N)=O)CC1C(C)C Cc1oc2ccccc2c1C(=O)NCC1(F)CC(CNC(=O)CC(C)C(F)F)C1 N1(c2cncc(C(=O)OCC)n2)CCCC(C)(C(=O)OC)C1 CCC(CC(=O)N1CCN(C)C(CNC(c2cccc(C)c2)=O)C1)C(C)C c1(NCC2(C(N(CC(=O)N(C)C)C)=O)CCNCC2)ccc(F)cc1 c1(C(N2CC(C)(C(=O)Nc3cc(Br)ncc3F)C2)=O)cc(F)c(Cl)c(C#N)c1Cl n1(CC)nnc2c(NC3CC(CNC(C4(C(=O)OC)CC4)=O)C3)ncnc12 N1(C(C2OCC(C)OC2)=O)CC2CCCN(C(=O)C(F)F)C2C1 C1(CNC(c2c(CC)nc(C)o2)=O)CCCCN(C(=O)CC(F)(F)F)C1 N1(C(=O)Nc2c(SC)cccc2)CC(NC(c2ccnc(CO)c2)=O)C2(CC2)C1 C#CCC(C)C(=O)NCC1CCN1C(=O)CCCNC(c1ccco1)=O C(CCC(=O)NOCC(=O)NCCC1CCC(C)(C)O1)OCC c1(NC(C2(COC)CC2)=O)cnc(F)cc1C(=O)Nc1nc(C)cs1 C1(CC(=O)NCC(C(CC)C)O)C2CCCC2N1C(C1(C(F)(F)F)CC1)=O c1(NC(CC(C)NC(c2coc(C(F)F)n2)=O)C)nc(C(C)(C)C)ccc1C#N CC(c1ccsc1)=CC(=O)NC(C)CN(C)C(c1cc(C)on1)=O C(c1csnn1)=CC(=O)NC(C1CC1C(=O)NCC1C2COCC12)C c1(C(N(C2CNCC(F)(F)C2)c2nccc(C(C)C)n2)=O)cc(O)ccc1F c1(CSCC(=O)NC(CN(C)C(c2cnn[nH]2)=O)(C)C)ccccn1 Cc1nn(C)c(C)c1C(=O)N(C1(C(=O)NCCN2CCCC(O)C2)CC1)C C1(O)(C(=O)NC(C(=O)OCC)C(F)(F)F)CCN(C(=O)COCC(C)(C)C)CC1 Cc1ccc(NC(N2CCC(O)(Cc3cccnc3)CC2)=O)cc1Cl C1(c2n(CC3(C)CCC3)nc(-c3ccoc3)n2)CCc2nc[nH]c2C1 CC#CCC(C(=O)NCC(C)C1CC1)NC(=O)C=CC1CCCN1C CC1(NC(c2n[nH]cc2Cl)=O)CCCCC1C(=O)NCC(O)CO c1(C(=O)NC2CC(C)(CNC(Cc3n(C)ncc3Cl)=O)C2)cc(Cl)c(F)cc1N O(NC(=O)CCCCC(=O)NC1CN(C(c2cocn2)=O)CC1F)C(C)(C)C C1(OC)CCCC1C(N1CC(CNC(C2(CC3CC3)CC2)=O)C1)=O c1(C(N(CCC)CCNC(c2nn(C)c(C)c2Cl)=O)=O)c(C)cc(C)cc1C N(C(=NCCc1cccs1)NC(C)C1CC1)CC1(c2ccc(OC)cc2)CCC1 N(C1CCCc2n[nH]cc21)C(C(C1CN(C(C2(C)CCCS2)=O)C1)OC)=O c12cc(cc(F)c1Cl)S(=O)(=O)NCc1cn-2nn1.c1(C(C)C)ccnc(CO)c1 CCCC(C)C(=O)NCCCNC(c1cc(C(=O)OC(C)(C)C)n[nH]1)=O C(=O)(C(CNC(=O)CC(C)(C)C(C)=O)C(C)(C)C)N1CCC(OCC)C1 Cc1n[nH]c(C)c1CC(=O)NC1(C(=O)NCCC(=O)N(C)C)CC(CO)C1 C1(C(N2CCN(C(c3cc(CC)ncn3)=O)C(CC)C2)=O)OC(C)(C)OC1(C)C C=CC1(C(=O)NCc2ccc(CNC(C3OCCC3C)=O)cc2F)CCCCC1 N1(C(CN(C(c2cc[nH]c2)=O)CC)=O)CCC12CCCSC2 C1(CCC)CN(C(=O)C(F)=C(C)C)CCN1C(=O)C(C1(O)CCCC1)F c1(C(N2C(C)(CNC(C(C(C)C)(C)O)=O)CCC2)=O)ccc2c(c1)N(C)CC2 N1(C(CCc2c(N(C3CCC3)C)cccc2)=O)CC(C)CN(c2nncs2)C(C)C1 N1(C(C(C2CCCC2)OCC)C(=O)NC2COC2)CCC(F)(COC)CC1 N1(C(C)C)CC(NC(=O)CCCc2cccnc2)CCC1=O c1(C(N(CCCNC(C2(C)CCCNC2=O)=O)C)=O)cn(CCO)c(=O)nc1O C1(COC)CC(CNC(c2cnccn2)=O)N(C(c2coc(C(C)C)n2)=O)C1 C(=O)(C(C)(C)CCNC(c1ccc(OC)nn1)=O)NC1(C#C)CC1 C1(CCC(N2C(C)CCC2)=O)CCCN(C(c2nnsc2N)=O)C1 N1(CCC(=O)NC2CC(CNC(C=C(CC)C)=O)C2)CCC(F)C1 C(N=c1[nH]c2ncc(Br)cc2s1)C1(SC)CC1 CC(CNC(C1CCCN(C(C2COC(=O)N2)=O)C1)=O)(CO)CO c1(C(=O)NC2C(NC(C3C(c4n(C)ncc4)C3)=O)COCC2)cccc(Cl)c1N n1(CC)cc(C(=O)OC)c(C(F)F)n1.C12(CCOC1)c1nc(no1)C(=O)N2C C1(C(=O)NC(CC=C)(C)C)CCCN(C(=O)CC(C)(C)OC)CC1 C(CN=c1[nH]c(=N)[nH]c(=NC2c3ccccc3CC2C)[nH]1)N1CCCC(C)C1 c1(CCC(=O)NC(c2c(F)cccc2I)C)ccc(Cl)c(Br)c1 CC1(C)CN(C(C(=O)NCSc2ccccc2)C2COC2)C12CCC2 c1(OC)ccc(C(=O)NC2CCCN(C(C3CC3CC(C)(C)C)=O)C2C)cc1C CCC(CCOC)C(=O)NCC1C=CCN1C(=O)COc1c(C)ncnc1C C(C(CCOC)NC(c1ccc(Cl)o1)=O)N(C(c1coc(CN(C)C)c1)=O)CC C(=O)(CCc1ncc[nH]1)NCCCN(CCC)C(C1CC1(C)CC)=O N1(C(CC(CC)C(C)C)=O)CCC2C(CCCN2C(C2CC2n2cccc2)=O)C1 C1(C(N(CC(O)CO)CC)=O)CCN(C(=O)CC2(COC)CC2)C1 C1(NC(C(C)NC(CC)=O)=O)(CF)CCN(C(c2cc(C3CC3)ns2)=O)C1 c1(CC(=O)NC(C)CNC(C2(CCF)CCOCC2)=O)n[nH]c2ccccc12 Cc1cccc(NC(=O)C(=O)NCC(F)CNC(c2cnncc2C)=O)c1 C1(CCNC(C(C)(C)OCC)=O)CCN(C(C2CC(C)C2(C)C)=O)CC1 CCCC(C)CC(=O)N1CC(F)CC1C(=O)N(C)CCC1CCCCC1 CC(C(=O)N1CCCC(CCNC(C2CCCN2C(=O)C(F)(F)F)=O)C1)C(C)O C1(C)(C(=O)NCCN(C(c2c(C(=O)OC)cco2)=O)C2CC2)CC2CCC(C1)S2 N1(C(C2OCCC(NC(C(F)=C(C)C)=O)C2)=O)CC2CCCC(O)C2C1 c1(C(C)C(=O)NC(CO)C(C)NC(=O)C2=CCCC2)ccc(Cl)c(Cl)c1 C1(OC(c2cccc3cncn23)=O)CCC2(CCCOC2)C1 c1(-c2cncc(CC)c2)ccc2c(C(=O)Nc3cc(Cl)nn3C)cnn2c1 N1(CCNC(N(C2CCCC2F)CCC)=O)CCCOCC1 c1(OC)cccnc1C(=O)NCC1(CNC(=O)C=CC(c2cc(C)on2)=O)CC1 c1(NC(c2ccccc2CN(C)C)=O)cccc(CC(F)C(=O)OC)c1 C1(C(N2CC(C(C)NC(CCSCC)=O)C2)=O)CC2(CCC2OC)C1 n1(C(C)C)ccc(C(N2CC3(C2)CN(C(=O)CS(=O)(=O)N(C)C)C3)=O)cc1=O C1(NC(C(C(C)C)F)=O)CCN(C(c2ccc(O)cc2)=O)CC1CO C=C(C)CCC(=O)N1CCCC(N(C(=O)Cc2csc(-c3ccc(C)o3)n2)C)C1 c1(C(=O)NCC=CCNC(C2(C)CCCS2(=O)=O)=O)cc2c(s1)CCOC2 CCCCC(C)CC(=O)NC(c1ccc(OC)cc1)CNC(=O)COCC CC(c1ccccc1)=CC(=O)N(CCCOCCNC(=O)C1=CCC1)C Cc1nc(C(=O)NCC2(NC(=O)C=CC3CCOC3)CCC2)c(C)s1 CC(CCC(=O)N1CC2CC2(NC(=O)C(CCC)OC(C)(C)C)C1)N(C)C C1(NC(CCOCCCOC)=O)CCCCN(C(c2n[nH]c(=N)s2)=O)C1 Cc1nccc(C(=O)NC2CC(C(=O)NC3CCCN(C(N)=O)C3)C2)n1.CC(C)C N#Cc1cn[nH]c1C(=O)NCC1(C(N)=O)CN(C(=O)Cc2ccccn2)C1 Cn1cc(C2=NOC(C(=O)NC3CCN(C(c4cn5c(n4)SCC5)=O)C3)C2)cn1 CC1(C)CC(=O)N(CC(=O)NC2CCC(NC(c3ncccn3)=O)C2)C1=O N1(C(C(C2CCOCC2)OCC)=O)CC2C(CNC(=O)C(Cl)=CCl)C2C1 c1(C(N2CCCC(C(=O)O)C2)=O)cnn2c1OCCC2.c12ccc(cc1)[nH]c2=O C1(F)(CNC(C(C)(F)c2ccccc2)=O)CCN(C(=O)CCc2ccon2)CC1 N1(C(C2OCC(C)C2)=O)CCCC2(CC(NC(=O)CCC3CC(C)(C)CO3)C2)C1 N1(C(CCC#C)=O)CCCCC1CNC(=O)CCCC1CCOCC1 n1(CC)cc(C(=O)NCC(C)CN(C(=O)C(C)n2cccc2)C)c(C)n1 CCC1=C(C(=O)N2CC(C)(C(=O)NCc3c(F)cncc3F)C2)CCCO1 C(=O)(CC(C)(C)CC)N(CC(=O)NC(CCN(CC)CC)C)C CC(O)CC(=O)N(CC(C)NC(=O)NC(=O)CC(C)NC1CCCC1)C C(CCc1ccccc1)(C(=O)O)NC(N(CCC(=O)NCCCC#CC)C)=O N1(C(C2(CC#C)CCC2)=O)C2CCC1C(CNC(C1CC(OCC)C1)=O)C2 c1(OC)cc(C)nc(N(C2CNCC2(F)F)C(C)=O)n1.c12ccc(c(C)c1)NC2 N1(C(=O)Cc2ccc(O)cc2)CCN(C(c2cscn2)=O)C2CC12 C(CS(=O)(=O)c1ccc(Br)cc1)NC(N(C)Cc1cnsn1)=O C(=O)(CC1CCc2ccc(O)cc21)N(C1CCN(C(C(C)N(C)C)=O)C1)C C(CC1=CCC2CC1C2(C)C)NC(=NCCN1C(=O)CCC1)NCC1CC1 C1(CNC(=NCC=C)NCC2CCCOC2)Cc2ccccc2O1 N1(C(CCC2(C)CC2)=O)CCOCC2(C1)CN(Cc1ccccc1)CCO2 CC1(C)C(C(=O)NCC23CCC(NC(=O)CC4(O)CCCC4)(CO2)C3)CC1(F)F N1(C(C(CC)CN(C)C)=O)CC2(CCN(C(C3CCCN3C(N)=O)=O)CC2)C1 Cn1ncc(C(=O)NC2CC(NC(C3CN(c4nncs4)C3)=O)C2)c1N c1(CN(C2(C(N(C3(c4nn[nH]n4)CC3)C)=O)CCC2)C2CC2)cc(C#N)ccc1N C1(NC(C2SCCS2)=O)CN(C(C2CCCC(C3CC3)O2)=O)CCC12CCC2 C1(NC(CCC2C(C)(C)C2)=O)CN(c2ncc([N+](=O)[O-])cc2F)CCC12CCC2 c1(C(N2CC3(C2)CN(C(C2(Cl)CC2)=O)CC3CO)=O)cnc(O)c2ccccc12 CCCC(C(=O)N(C1CC(CCn2cc(-c3nccs3)nn2)C1)CC)S(N)(=O)=O C(=O)(CCC(C)(C)C)N1C(CNC(C2C(C)(C(=O)OCC)C2)=O)CC1 c1(C(N2C(CC)CN(C(C3(CC(=O)OC)CC3)=O)CC2)=O)cc(C)c(Cl)cc1F N1(C(c2csc(C)c2C)=O)CCC(CCNC(c2nocc2Cl)=O)CC1C C1(C(=O)NCCc2c(C)cccn2)CN(C(c2cc(C)n(C)c2C)=O)CC1(F)F c1(C(N(C2CCN(C(=O)COC3CCOC3)CC2)CC)=O)cc2cnn(C)c2s1 CC(C)C(C(=O)NC(C1CCCN(C(=O)Cc2ccc(O)cc2)C1)C)C(C)C Cc1c(C(N2CCCC2C(C)NC(C2(O)CC(C)(C)C2)=O)=O)nn2ccccc12 c1(C(N2CCCCC(CNC(C(CC=C)C)=O)C2)=O)cc2n(n1)CCCO2 c1(C(C)=O)ccc(C(=O)NC(CNC(C2CC(=O)N(C)C2)=O)CO)c(F)c1 C1(N(C(c2scnc2C)=O)CC)CCCN(C(C2(NC(=O)OC(C)(C)C)CC2)=O)C1 N1(C(CN(CCC#C)C)=O)CCCC(CN(C(=O)CC(C)F)C)C1 c1(SC)cnn(C)c1C(=O)NCC(C)NC(=O)C=Cc1cnc[nH]1 c1(C(N(CC(C)NC(C(C(CC)CC)C)=O)C)=O)csc(=NC2CCCCC2)[nH]1 C1(N(C(c2c(CC)ncs2)=O)C)CCCC2CN(C(C3CCCOCC3)=O)CC12 c1(C(=O)NC(c2cccc(Cl)n2)CC)cccc(Cc2cccnc2)c1 C1(N(C)C(C2CC2C(F)(F)F)=O)CCN(Cc2cccs2)CC1 C1(C(N2C3C(NC(c4c(C)occ4)=O)CC(C3)C2)=O)CN(S(=O)(=O)N(C)C)C1 N1(C(c2c(C)sc(Cl)n2)=O)CCC(C)N(C(C23CCCC2(C(N)=O)C3)=O)CC1 c1(CNC(Cc2c(C)non2)=O)cc(O)nc(CNC(C2C(C)CC2C)=O)n1 N1(C(c2c(CC)nn[nH]2)=O)CCN(C(=O)C(F)n2ccnc2)CC1C1CC1 N1(C(Cn2cnc(C#N)n2)=O)CC2(CCC(CNC(C3C4CCCOC34)=O)O2)C1 Cc1ccncc1CC(=O)NCCc1ocnc1CNC(=O)CO N1(C(c2[nH]cc(C(C)=O)c2)=O)CCOC(C(C)NC(=O)CSCc2ncc[nH]2)C1 C(=O)(C(F)(F)C(C)O)NCC(C)NC(c1ccn(-c2ccccc2)n1)=O CCCC(CC)C(c1nnnn1CCC1CC1)NCc1cc(C(=O)OC)co1 N1(C(c2c(F)ccc(C)c2F)=O)CC2CCC(NC(=O)COC(F)(F)F)CC2C1 c1(N2CCC(C3(NC(c4ccc(OC)cc4)=O)CC3)C2)ncc(C)cc1[N+](=O)[O-] Cc1cn2cc(C(=O)NC3COCC3NC(=O)CSc3ccccc3)sc2n1 C1(CC)CCN(C(=O)CC23CCC(CC2)C3)C1C(=O)NCC1CNC(=O)O1 CCCC(CC)C(=O)N1CC(NC(=O)C2=C(Cl)CC2)C(C)C1 CCCCCCC(CC)C(=O)N1CC2CCC2(CNC(c2cc(OC)cs2)=O)C1 C1(C(=O)NCc2nc(CC)on2)(CC)CCCN(C(C2CC(=O)NC2(C)C)=O)C1 c1(C(=O)NCC(C2CC2)NC(CN(CC(=O)NC(C)C)C)=O)ccns1 CC(CCN=c1[nH]c2ccc(F)cc2s1)NC(=O)C=C(Cl)Cl Cc1cc(C(F)(F)F)cc(NNC(=O)c2ccc(C(O)CF)cc2)n1 c1(C(=O)NCC2(CNC(CN(C3CC3)CC)=O)CC2)cccc2c1OCCCO2 C1(C(C)NC(C(c2ccccc2)OC)=O)CCN(C(=O)C=Cc2cc[nH]n2)C1 c1(CC(N2CC(F)(CNC(COC3(C)CCC3)=O)C2)=O)sc(=N)[nH]c1-c1cccs1 C(CCCN=C(NC1CCS(=O)(=O)C1)NC1CC2(CCC2)C1)N1CCCC(C)C1 C1(NC(c2cc3cccnc3s2)=O)C2COCC1CN(C(c1coc(O)n1)=O)C2 C1(OC)C2CC3CC1CC(C(=O)NC1CC1CNC(C1CC(F)(CO)C1)=O)(C3)C2 N1(C(=O)Nc2ccn(CC)n2)CCC(C(C)NC(=O)OC)CC1 c1(OC)ccc2c(c1)CCC(C(=O)NC1CCC(C(=O)Nc3cncnc3)C1)C2 N1(C(c2c(OC)noc2C)=O)CC(N(C)C(C2CC2(C)C)=O)C(C)(C)C1 c1(CC)nn(C)cc1C(=O)NCC1CN(C(=O)CC2CC2C2CC2)CC1O Cn1c(C(N2CCC(CNC(c3c(F)cc(N)cc3F)=O)C2)=O)cc2occc12 CCCCCCC(=O)NC1CC(CCNC(c2ccn(C3CC3(F)F)n2)=O)C1 C=CCCCCCCCCC(=O)NCCN(CCOC)C(C1OCCC1CC)=O C1(CNC(C2(C(=O)NC)CC2)=O)CCCCC1NC(=O)Cc1ccc(Cl)cn1 C1(NC(C(C)c2ccco2)=O)CN(C(C2CCN(C)CC2)=O)C2(CCCC2)C1 C(=O)(C#CC1CCOC1)N1C2CC(NC(c3ccc4nc[nH]c4n3)=O)C1CC2 C(=O)(C(CC(C)C)ONC(c1cncc(Cl)c1)=O)NCc1cn(CC#C)nc1 C1(C(N(CC(=O)NC(C(C)C)CN(C)C)C)=O)CCCC(C#N)C1 C1(CNC(C23OCC(COC)(C2)C3)=O)CCN(C(=O)COC(C)=O)C1(C)C C1(C(N2C(CCC(=O)N(CCCF)C)CCC2)=O)(CO)CC(C)(C)C1 N1(C(C2OCCN(C(C(CCC(C)C)O)=O)CC2)=O)CC=C(C(C)(C)C)CC1 C#CCCCCC(=O)NC(C1CCN(C(=O)C(C)(C)C)CC1)CO c1(C(N2CCCC(N(C(=O)C=C(C3CC3)C3CC3)C)C2)=O)ccc2cc[nH]c2n1 C1(NC(=O)C=Cc2cnc[nH]2)CCCC(NC(c2cnc(C(F)F)nc2)=O)CC1 c1(C(C)NC(CC2(C(=O)OC)CC2)=O)ccc(CNC(C2C3COCC23)=O)cc1 C(=O)(C(C)CC(N)=O)NC1CCN(C(CC2CCC(C(=O)OC)CC2)=O)C1C CCCC(C#N)C(=O)N1CCOCC(NC(=O)CCc2nc(C3CC3)no2)C1 C1(N(C(C(C)OC)=O)C)CCCC1(C)CNC(=O)CCc1cnc(C2CC2)o1 N1(C(C(CC)n2cccn2)=O)CC2(CCN(C(=O)COC3CC3)C2)C1 C#CC1(O)CC(C(N2CC(CC(F)C(=O)N(CC(C)O)CCO)C2)=O)C1 S(=O)(=O)(CC(F)(F)F)N1CC(C(N2C(C(=O)OC)CC2)=O)OCC1 CCC(C)CN=c1[nH]c(N2CCN(CC(F)F)C(C)C2)nc2cc[nH]c12 N1(C(C(C(C)C)C)=O)CCN(C(=O)CC2CCCC23CC3)C(c2ncc[nH]2)C1 C1(C(=O)NCC2OCCN(C(c3on(C)c(=O)c3)=O)C2)COc2ccccc2C1 Cc1cc(N2CC(F)CC2CNC(C2(C(C)C)CC2)=O)ncc1C#N C(=O)(CC(F)(F)C(F)(F)F)NCCC1CCN(C(c2c(N)ccc(OC)c2)=O)C1 C(=O)(C1CCCc2sc(=N)[nH]c21)N1C(CNC(C(C)(C)SC)=O)C(C)(C)CCC1 C(C)(C(=O)NCCN(C(=O)C(C)NC(=O)Cn1cnnn1)C1CC1)OC c1(C(C)C)ccc(OCF)cn1.c12cc([nH]n1)CNC(=O)C(O)C1CN(C1)C2=O c1(CN(C(=O)CC2(C)CCCCC2)C)ccc(-c2nn[nH]n2)cn1 c12cc(cc(Br)c1)CNC(=O)N2.C(CC(=O)OC)N(CCO)CC C1(CCC(c2cnc(CC(C)(C)C)s2)=O)C(C)CCCN1.C(C(=O)NC1CC1)OC N1(C(C(C(C)C)OCC)=O)CCC(NC(=O)C(F)CN(CC)CC)C(C)C1 c1(C2(CN3C(COC)C=CC3)CC2)cccc(CN)c1 c1(C(=O)NC(CSC)(C)C(=O)NCC(C)(C)CC(C)O)cc(C)nc(C)c1 c1(C(=O)NCCCn2cc(CNC(C)=O)nn2)ccc2c(c1)N(C)C(=O)C2 C1(NC(C(C)(C)n2cncn2)=O)CC2CC1CN(C(C1CC1F)=O)C2 Cc1cc(Cl)cc(C)c1C(=O)NCC1CC1NC(=O)Cn1ncc2ncccc12 c1(N2CCC(NC(CC3N(C)CCCC3)=O)C(O)C2)nccc(C#N)c1[N+](=O)[O-] C(=O)(CC(C)C(C)C)N(CCC)CCNC(=O)CCc1cc(Br)cs1 N1(C(CNC(c2c(C)[nH]cc2)=O)=O)CCN(C(C2C(C)C2C)=O)CC1 N1(C(C2CC(CNC(c3cnn(CCF)c3)=O)OC2)=O)CCCC(F)CC1 CC1(C)CN(C(=O)CC2CC=CC2)CC2(CN(CC3CCc4ncnn43)C2)O1 c1(C(N2CCCCC(NC(C(C)(C)c3nccs3)=O)C2)=O)ccc(F)c(Cl)c1F c1(C(N2CC(NC(c3cn(C)nc3)=O)C2)=O)cnc(C#N)s1 N1(C(C(C)Oc2c(OC)cccc2)=O)CCC12CN(C(c1cocc1C)=O)C2 C(=O)(C1=NOC2(CCC2)C1)NC(C(=O)N1CC(C(CC)CC)C1)CC(C)(C)C CCCC(C(=O)N1CCOCC(C(=O)NC2CN(C)CC2(F)F)C1)C(C)C C(c1ccc(O)cc1)=CC(=O)NCC1N(C(COCCC=C)=O)CCOC1 c1(C(N2C(C(=O)NCC3CC3)CC2)=O)cccnc1C(F)F C1(CNC(c2cc(COC)sc2)=O)CN(C(C2CCC3(CC3)C2)=O)CC1O C(=O)(CC(C)(O)c1ccccc1)NC(CC)CNC(c1ccsc1Cl)=O C1(C(=O)NCC(C)(CO)NC(C2C(Cl)(Cl)C23CC3)=O)(OCC)CCSCC1 c1(C(=O)N)cc[nH]c2nccc1-2.C1(C(=O)NC)C=CC(NC(c2occc2)=O)C1 CC(Cc1cnc[nH]1)C(=O)NC(C)(C)CNC(c1sccc1SC(F)F)=O c1(N(C)C)cnn2c1CN(C(c1ccc3c(c1)ncn3C)C(=O)NC1CC1)CC2 Cc1nc(NC(=O)C(C(C)C)NC(=O)Cn2cnnn2)ccc1C(F)(F)F CCC(C(=O)N(CC(C)(C)CNC(=O)CNc1ccc(C#N)cc1)C)C(F)(F)F N1(C(c2c(C)n(C(C)C)nc2)=O)CC(N(C(=O)C(C)C)C)C(C)(C)C1 Cn1cnc2nc(N3CCC(c4nccs4)C3)nc(NC3CCCCC3)c12 N1(C(c2c(CC)cccc2)=O)CC(C(N2CCOCCC2C)=O)C(F)(F)C1 N1(C(C2CC(=O)NC2)=O)CCN(C(c2ncccc2-c2ccccc2)=O)CC1 N1(C(c2cn(CCC)nc2)=O)CCC(C(=O)NC2CC3CC3C2)=C(F)C1 N1(C(C(CC)n2cncn2)=O)CC2CC2(CNC(=O)C=CC=Cc2ccco2)C1 C1(NC(c2n(CC)ncn2)=O)CC2CC1CN(C(=O)CCc1ccccc1F)C2 c1(C(N2C(CNC(C(c3ccnn3C)C)=O)COCC2)=O)cncc2nc[nH]c12 Cc1nc2c(C(N3CCCCC(CNC(C4CC(C)(F)C4)=O)C3)=O)cccc2o1 C1(C(=O)NCC(CO)NC(=O)Cc2ccccc2)CC2COCC(C1)C2 c1(C(=O)NCC(CO)NC(C2CC(=O)NC2)=O)ccc2[nH]nc(C(F)(F)F)c2c1 N1(CC)CCN(C(C(=O)NCC)C2CCC2)C(C)C1 c1(C(N2CCC(N(C(C3CCC(C)C3)=O)C)CC2)=O)cncc2ccc(F)cc12 C1(CNC(CC(C)C)=O)CCC(C)(C)CN1C(=O)CCC1CC(C)(C)CO1 Cc1cnc(C(N2CCC(C(N3CC(CO)C3)=O)C2C)=O)cn1 c1(C(=O)NC2CN(C(c3[nH]cc(C)c3)=O)C2)cnn(CC(C)C)c1C C12(C(N3CCC(SC)C3)=O)CCCC1CCN2C(c1cc(C)c[nH]1)=O C1(CC=C)(NC(=O)C(O)C=C)CCCN(C(=O)CCc2cncs2)C1 C(=O)(C1(C)CCCc2ccccc21)NC1C(CNC(c2c(CC)c[nH]c2)=O)C1 N1(C(c2cc(C)c(C)s2)=O)CCC(C)(C)C1CC(=O)NC(c1nc(=O)o[nH]1)C c1(C(N(CC(O)CNC(C2(C)CCCS2(=O)=O)=O)C)=O)c(F)ccc2[nH]ccc12 c1(C(=O)NCC2C(NC(CC(C)F)=O)CCC2)ccccc1C#N c1(C(C)(C)OC)nc(=NCCCC(C)NC(C2CCCCC2)=O)s[nH]1 c1(CC=C)ccccc1C(=O)NCC(C)CN(C)C(C1(C)CCN(C)C1)=O CC1CCN(C(=O)CN(C)C)CCN1C(C1CC1c1cccs1)=O C(CCCCC(=O)NCC1COC(CNC(c2cn(C)cn2)=O)C1)OC C(CC(C(=O)NCC1CN(C(C)=O)C1)NC(c1cc(C)[nH]n1)=O)OC C1(C(=O)O)CC2(CCCC2)CCN1CC1CCCS(=O)(=O)C1 CC(C)C(C)C(C)CC(=O)NCCN(C(=O)C=Cc1ccc(F)c(F)c1)C c1(NC(N2CCCC2C2(C)CC2)=O)ccc(C(N2CCOCC2)C)c(F)c1 N1(C(c2nnn(C)n2)=O)C2CCCC1CN(C(=O)CCN1CCCC1)C2 C(=O)(CS(=O)(=O)CC(C)C)NC(CCNC(C1(c2c(C)ccc(F)c2)CC1)=O)C c1(NC)ccccc1C(N1C(C(N2CCCCC2C2CCC2)=O)CC1C)=O c1(C(N2CC(NC(C(COC)C)=O)C(O)C2)=O)ccc2nc[nH]c2c1 C(=O)(C1=CN=C2N=CNN2C1)N1CCOCC(NC(c2coc(C(F)F)c2)=O)C1 C1(CNC(CC(CC)(F)F)=O)CC2CCC(C1)N2C(C1COC(C)(C)C1)=O c12ccc(s1)C(=O)C(=O)NC(C1CCC1)CNC2=O.C1(C(F)F)(CC)CC1 C(CC(F)(F)C(C)C)n1cc(C(c2nnnn2C)NC2C(CC)CCCC2)nn1 C1(C(N(C2CN(C(C(CC=C)NC(C)=O)=O)C2)C)=O)CCN(S(=O)(=O)NC)CC1 CC1CC(C(N2CCN(c3nnc(-c4ccccc4)o3)CC2C)=O)CC(C)C1 c1(C(=O)NC(C(=O)NCC(=C)CC)C2CCC2)cnncc1O C(=O)(C1CCCc2ccccc21)N1CCC(NC(=O)CN2CCS(=O)(=O)CC2)C1 N1(Cc2onc(C(C)OCC)n2)CCC(N(C)C(C2(O)CCCCC2)=O)CC1 N1(C(C(COC)C)=O)CC2CCN(C(=O)Cn3cnnc3)CC2C1 CCC(CC(=O)N1CC2CC2(NC(c2cnnc(O)c2)=O)C1)OC C1(CCOC)(C(=O)NCCCC2(NC(C3CSC3)=O)CC2)CCC1 C1(NC(C(F)=C(C)C)=O)CCN(C(c2cn(CCF)nn2)=O)C1 C1(NC(CCC#C)=O)CN(C(=O)Cc2cncc(Br)c2)CCC12CCC2 c1(N(C(=O)CNC(N)=O)C)ccc(Sc2cc(-c3ccccc3)ccn2)cc1 Cc1ccnc2sc(C(=O)NC3CN(C(c4ccncn4)=O)CC3(C)C)c(C)c12 C1(C2(O)CCOCC2)(CNC(N2CC3(C2)OCC2CC32)=O)CCC1 c1(C(N(CC(CNC(c2ccc(C=C)cc2)=O)O)C)=O)cc(F)cc2ccoc12 N1(C(c2cc(C)n(C(C)C)c2)=O)CC2CC(NC(C3CCCC(C)C3)=O)C(C2)C1 C(C(C(F)(F)F)NC(c1nc(-c2cccc(C(F)(F)C(F)F)c2)cs1)=O)N(C)C C1(C(N2CC(NC(c3n(C=C)ncc3)=O)C(C)C2)=O)Cc2ccc(OC)nc2N1 c1(C(C)=O)cc(=NCCCCNC(c2cnc3scc(C)n23)=O)[nH]cn1 C1(Cl)(C(N2CCC(OC3CN(C(C4CCCO4)=O)C3)CC2)=O)CC2CCC1O2 N1(C(CC(CC)C)=O)CC2(C1)CN(c1nc(C3CCCC3)nc(=N)[nH]1)C2 Cc1cccc(CCC(=O)NC2CCCN(C(c3ncccn3)=O)C2)c1Br C1(CC(N2CCC(N(C(C(CSC)O)=O)CC3CC3)C2)=O)OCCC1(C)C C1(NC(C2C(C=C)CC2)=O)CC(CNC(=O)C(CO)N(C)C)CC1O c1(C(=O)NC(CCNC(C=Cc2scc(C)n2)=O)C)ccc(F)c2ncccc12 Cc1ccccc1C1(C(=O)NCC(C)NC(=O)C(N2CCSCC2)C)CC1 C1(CC(=O)NCCOCCNC(c2ccc(O)nc2Cl)=O)CCCC2(CCC2)O1 C(=O)(CCC(=O)NC(C)C=CC(N1CCC(C(=O)NCC)C1)=O)NCCC N1(C(C(=O)NCCCSC)c2ccco2)CCCC1NC(=O)NC(C)(C)C C1(c2n(CCSC)nnn2)(NCc2c(C)cccc2Cl)CC(C)N(C)C1 c1(OC)c(C)cnc(Cn2cc(C3(O)CN(C(=O)Cc4ncc[nH]4)C3)nn2)c1C C(CC(C(=O)NC1(c2noc(C)n2)CC1)NC(=O)CC1CN(C(C)C)C1)OC CCC(C(=O)N1CCC(CNC(=O)CCCSC)(COC)C1)C(C)(C)CC N1(C(c2c(CC)cc[nH]2)=O)CC2CC2(CNC(=O)C(CCC)NC(N)=O)C1 c1(C(=O)NCCCNC(CCCCNC(C)=O)=O)nc(C)c(N)cc1C CC1(C)CC(NC(=O)CC2COC3(CCC3)CO2)CN(C(c2ccsc2Cl)=O)C1 N1(C(C2(C)CCN(C(C3CC(=C)C3)=O)C2)=O)CCC2(C=CCO2)C1 C(=O)(NN(C(C)=O)c1ccccc1)C1C(c2cccc(OC)c2Cl)C1 c1(C(N2CCC(C3N(C(C(CC#C)C)=O)CCCC3)CC2)=O)c(C)ncnc1C NC(=O)CCC(C(=O)NCCc1ccc2c(c1)CC2)n1cc(C2CC23CC3)nn1 c1(C(N2CC(CC=C)(NC(c3csc(C(F)F)c3)=O)C2)=O)cncc(OCC)c1 c1(C(N2CCN(C(Cc3c(C)cco3)=O)C(C)C2C)=O)oc2ccccc2c1C N1(C(C(C)SC)=O)CC2CCC2(CNC(c2sc(Cl)c(Cl)c2C)=O)C1 c1(C(C)OC(CCc2cc(C)on2)=O)c(Cl)cccc1Cl N1(CC)CCCCC1C(N1CC(CNC(=O)C(C2CCCOC2)OC)(OC)C1)=O C1(C(N2CCCC(C(N)=O)C2)=O)(CC)CCN(C(C2CCSCC2)=O)C1 O=C1NCCC2CCN(C(C3CN(C(C4CCCS4)=O)CC34CC4)=O)C12 c1(S)ccc(O)cc1.C1(C(=O)NC2CCC2N)CCN(C(C23CC(F)(C2)C3)=O)CC1 CCCCC(CC)CC(=O)N1CCN(C(=O)C(C)=C2CCCC2)CC1C1CCC1 c1(C(=O)NCCN(C(C(C)OCC#C)=O)C2CCCC2)cc(F)c(C#N)c(F)c1 C(=O)(C1CCCn2cncc21)N(CCN1CCN(C(C(C(C)O)(F)F)=O)CC1)C C1(NC(COCCCOC)=O)COCCN(C(=O)CC2CCCCC2)C1 c1(OC)ccncc1C(=O)NC(CCN(C)C)C(=O)N(C)Cc1cnnn1C C(=O)(CCC(=O)NC1CC(NC(=O)C(c2cnn(C)c2)C)C(O)C1)NC N1(C(c2nn(C)c(=O)cc2)=O)CCC2CN(C(=O)CCC3CCC(O)CC3)C2C1 CCC(CC)C(=O)NC1CCOC(C(=O)N(C2COCC2OCC=CC)C)C1 c1(C(N2CCC(OC)(CNC(=O)Cn3ccnn3)CC2)=O)ccc(N=[N+]=[N-])cc1 Cc1cnn(C(C)C)c1C(=O)NCCC(C)NC(C1CC(F)C(=O)N1)=O C1(C(=O)Nc2ccc(OC)cc2C)CC2(CCN1C(=O)Cn1cnnc1O)CC2 Cc1sc(O)nc1C(=O)NC1CCN(C(C2(n3ccnn3)CC2)=O)CC1 Cc1nc([N+](=O)[O-])cn1CC(N1CC(NC(=O)CCCCCF)CC1C)=O c1(CC(=O)NCC2(NC(c3ccc(O)nn3)=O)CCC2)ccc(Br)c(F)c1 C1(NC(C(C)(C)OCC)=O)CCOCC1C(=O)NCC(C)C1CCC1 c1(C(=O)NCCOC2CN(C(C#CC(OCC)OC)=O)C2)cc(F)ccc1CC c1(C(=O)NC(c2ccccc2F)CNC(=O)CCC2CC2)c[nH]c2ccccc12 Cc1cc(C)c(C(=O)NC(CNC(c2conc2C(C)(C)C)=O)C2CC2)cc1N C(=O)(C(CC(C)C)NC(=O)C(N1CCS(=N)(=O)CC1)C1COC(C)C1)OC CCC(CC(F)F)C(=O)N1CCN(C(=O)C(C2CCC2)C2CCC2)CC1CC c1(C(=O)NCC(CCC)NC(c2cc(C3CCC3)[nH]n2)=O)ccccc1C(C)C N1(C(CCCOCC=C)=O)CCCN(C(=O)C2=CCOCC2)CC1C(C)C c1(N(CC#CBr)C(c2cc(Cn3cc(Br)cn3)on2)=O)cccc(F)c1Br c1(NC(C2C3CC2N(C(=O)C=Cc2ccccc2)C3)=O)ncc([N+](=O)[O-])cc1I Cc1cccc2c1N(C1CCCCC1)C2=O.c1(OC)nc(Cl)ncc1Br c1(C(=O)NCC(CCCC)NC(=O)Cn2cnc(C)cc2=O)ccc(O)nc1Cl Cc1nccnc1C(=O)NCC1C2CC1N(C(=O)CCCCc1cnn[nH]1)C2 Cc1ccc(C(=O)NC(C)(C)CCNC(C2CCC(C3CC3)C2)=O)nc1O C1(C(N2CCC(C#CC)C2)=O)CC2CCCC2N1C(c1occ2c1CCC2)=O Cc1cc(C(=O)NCC(C2CC2)NC(c2cnc(C3CCCO3)s2)=O)c(C)cn1 N1(C(CCOCC)=O)CCC2CCC(NC(c3nnc(CC)s3)=O)C1C2 CCCC(C(=O)OC)C(=O)N1CC2CC2(C(=O)Nc2cccc(C)c2C)C1 CCCC(CC(=O)NCCSC)NC(=O)C(F)OC(F)(F)F C1(NC(c2ccc(CSC)cc2)=O)CC2CCC1N2C(c1ccc(F)cc1Cl)=O c1(C(C)C)nc2n(n1)CC(CC1CC1C)CC2.N1C(=NCCCF)NCC1 N1(C(C)C(=O)N(C)C)CC2CC1CC2C(N1CCN(C)CC1)=O O(NC(=O)C(C)(C)C(C)(C)C)CC(=O)NCC(C(C)C)(C)CO C#Cc1ccccc1NC(c1nnnn1C1CCCC1)c1cccs1 CC(C)C(C(=O)NCC(C)NC(=O)C(C)(C)c1ccncc1)c1ccc(Cl)cc1 c1(C(N2C3CC(CNC(=O)CC4(CO)CCC4)C2CC3)=O)cccc2cnnn12 CC1(C)COCCC1C(N1CC2CC(NC(C3(O)CCSCC3)=O)C2C1)=O C1(NC(C(n2ncc(C)c2)C)=O)CN(C(=O)CC2C(C)(C)C2(C)C)CC12CCC2 C1(CNC(CC(C)N(C)C)=O)CC2(CO1)CN(C(=O)CCn1cccnc1=O)C2 C(C(CC(C)C)C(=O)N1CCCC1C(C)NC(=O)CCc1ccc(F)cc1)OC c1(N2C(C3CCN(C(C4(C)CC4(F)F)=O)C3)CCC2)ncc(O)cn1 CCC(C)(CO)C(=O)NCC(=O)NCC(=O)NCC12CC(C)(CCO1)C2 C1(C(=O)OC(C)(C)C)Cn2cnnc2CN1C(=O)C(F)CC1CCNCC1 c1(C(N2CC(CC(C)NC(CC(=C)Br)=O)C2)=O)nccc2ncccc12 c1(CN(C2CCOCC2)C)cnc(C(C(=O)NC2CCCC2)N2CCC2CF)s1 C1(C)(CCC(=O)N(CC(C)SC)C)CN(C(c2nonc2N)=O)C1 c1(C(N2CCN(C(C(CC(C)C)N(C)C)=O)CC2)=O)[nH]nc2c(=O)n(C)cnc12 C12(C(N(C3CC(NC(c4c(CC)nc[nH]4)=O)C3)C)=O)CCCC1(C(=O)OC)C2 c1(NCC2(O)CN(C(C(c3ccc(C)s3)C)=O)C2)ncnc2c(Cl)cc(Cl)cc12 C(CCCCC(=O)NC(C1CCN(C(C2(C)CCSCC2)=O)C1)C)OCC CC1(C)CCC(CO)N(C(=O)C(C2(O)CCCCC2)NC(=O)CCC(F)(F)F)C1 Cc1ncccc1C(=O)NCC(C)NC(=O)CC1(n2nccn2)CC1 N1(C(c2ccc(SC)o2)=O)CC(NC(=O)C(Cl)=CCl)C(N=[N+]=[N-])C1 C1(C(N(C)CC2CCCCN2C(C2(C#N)CCC2)=O)=O)CC(=O)OC1(C)C c1(CN2CC3C(C(=O)NCc4ccc(SC)cc4)(C3)C2)ccc(Cl)cc1[N+](=O)[O-] C#CCCCC(C)C(=O)N1CCC(C(N2CCC23CC(C)(CO)C3)=O)C1CC N1(C(C2C(C)(CCC)C2)=O)CC2(C)CN(CCNC(=O)OC)CC2(C)C1 C1(SC)CN(C(c2ccc(C#N)cc2)C(=O)NC2CCC2)C2(CCC2)C1 c1(NC(c2csc(Br)c2)=O)ccnc(-c2cnn(Cc3ccncc3)c2)c1 c1(C(=O)NC(CNC(CCCC=C)=O)C(C)C(C)C)cc2nc(C)ccc2o1 CC(F)(F)CC(=O)N1CCCCC1c1ccc(CNC(=O)CSC(C)(C)C)cc1 C12(C(N(C3CC(NC(C4(C5CC5)CCOCC4)=O)C3)C)=O)CCC(=O)N1CCS2 N1(C(CC(CNC(C2(C)CCCOC2)=O)OC)=O)CCCC(C)(C)CC1 C1(NC2(C(=O)OCC(C3CCCC3)OCC)CCC2)CCCSC1 c1(C(N2CC(NC(C3C(F)(F)C34CCC4)=O)C(O)C2)=O)cc([N+](=O)[O-])cnc1O c1(OCCCC)ccc(CNC(=O)NCCCC2CC2(Cl)Cl)c(Cl)c1 c1(OC)ccc(C=CC(=O)NCC(C)(C2CCC2)NC(=O)C(F)OC)c(C)c1 C(=O)(C(C)(C)CCNC(c1ccnc(CO)c1)=O)N(CCC(=O)OC)CC O=C(C1CCCn2ccnc21)NCC1CC2(CC2)CN1C(C1CC=CC1)=O Cc1nc(C)c(C(=O)NCCN2CCCC(C(=O)NCC3CC3)C2)[nH]1 C1(NC(c2ccc(C(C)=O)[nH]2)=O)CC12CC(NC(c1cc(C)ns1)=O)C2 c1(C(N(C2CC(NC(=O)Cc3ccc(O)nc3)C2)C)=O)[nH]nc2c1COC2(C)C C(=O)(C1=CC2CCCCCCC12)NC1CC(F)(CNC(CCS(C)(=O)=O)=O)C1 Cc1ccc(N(C2CC(C)(C)C(=O)N2)C(=O)Cn2nc(C(C)(C)C)cc2N)cc1Cl c1(C(=O)NCC(CNC(C2(COC)CC2(F)F)=O)C)cn(C)nc1C N1(C(C(=O)NCC(C)=CC(=O)NCC2(O)CSC2)C)CCCCC1 C#CC1(C(=O)NC2CCCCCC2CO)CCN(C(C2CC=CCC2)=O)C1 C12(C(=O)NCC(C(C)C)NC(=O)CCc3ccc(C(C)C)cc3)CC(C1)C(C)O2 N1(C(c2c(CC)cco2)=O)CCC2(CCN(C(C3CCCC(O)C3)=O)CC2)C1 c1(CC(C)NC(=O)C(N2CCC(n3cc(C(N)=O)nn3)C2)=O)ccccc1Cl c1(C(C)OC)nc(C(=O)NCC(O)CNC(C2(F)CCCC2)=O)cs1 c1(NC(CN2C(CC)COCC2)=O)cc(N)c(C)cc1C N1(c2c(OC)cncn2)CCOCC(CNC(=O)C(c2ccc(F)cc2F)C)C1 C(=O)(C(C)(C)C(C)NC(c1cnc[nH]c1=N)=O)N(CCCC=C)CC N1(C(C(CC)CO)=O)CCC2(CCCN2C(c2cncc(-n3cccc3)c2)=O)C1 c1(NC(=O)NCC(C2CCCC(=O)N2)C)noc2ccc(F)cc12 c1(C(N2CC3CCN(C(C(CCC)O)=O)CC32)=O)cnc2ccccc2n1 N1(C(=O)Cn2nccn2)CC2CCN(Cc3ccc4cc[nH]c4n3)C2C1 c1(NC(C2CNCCN2Cc2c[nH]c3cccnc23)=O)cc(Br)cc2cn[nH]c12 CCC(C(=O)N1CC(O)(CNC(c2ccn(C)c2C2CCC2)=O)C1)C(C)C N1(C(C2C(C(=O)NCC#C)C2)=O)CC(NC(=O)CCn2nc(C)nc2C)C(F)C1 N1(C(C(n2c(C)ncc2)C)=O)CC(NC(C2(O)CCC2)=O)C(CO)C1 c1(NC(C2N(Cc3cnc(SC)nc3Cl)CC2)=O)cc(Br)cc([N+](=O)[O-])c1C N1(C(C2C(=C)C2)=O)CC2(COC(CNC(=O)C(CC)OCC)C2)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1C(CNC(C(=C(C)C2CC2)F)=O)C(C)CC1 C12(C(N3CC(N(C(C4CN(S(CC)(=O)=O)C4)=O)C)C(O)C3)=O)CCC(CC1)CC2 C(=O)(C1Cc2ccccc21)NC(C1(O)CCN(C(C2CCC3(CCC3)O2)=O)C1)C c1(CC(=O)NC(CN(C(C2(COC)CCCO2)=O)C)C)ccc(C(C)(C)C)cc1 c1(OCC=CC(=O)NC2CC2NC(=O)C=CC2CCCC2)ccccc1 C1(C)(CC)CCN1C(=O)C(C)NC(C1CS(=O)(=O)C1)=O CC(CN(C)C(c1cc(C2CC2)[nH]n1)=O)C(=O)N=c1ccn(C(C)(C)C)[nH]1 C1(COC)(NC(=O)C(C)CO)CCN(C(c2sc(C)cc2Cl)=O)C1 C(=O)(CC(C)(C)C(F)(F)F)NC(C)CNC(C1CC1c1cnn(CC(C)C)c1)=O C(C1CN(C(C2CC3CSCC(C2)C3)=O)Cc2ccccc21)NC(CC)=O N1(C(c2n[nH]c(C)c2O)=O)CC2CC(C(=O)NCC(c3ccco3)O)CC2C1 c1(C(N2C(C)(CNC(C(C)SCCCC)=O)CCC2)=O)cc2scnc2[nH]1 Cc1c(NCc2ccco2)ncnc1N(C)CCF c1(C(C)N(C)C(C2CC(NC(=O)C=Cc3cc[nH]n3)C2)=O)ncccc1Cl c1(OCC(=O)N(CCC(N2CCCC(C#C)CC2)=O)CC)cc(C)nc2ncnn12 C1(NC(COCP(C)(C)=O)=O)CCCC(NC(=O)CCc2ccc(N)cn2)C1 CC1COC2(C1)CN(C(c1cnn(-c3ccccc3)c1Cl)=O)C2 Cc1ncc(C(=O)NCC(n2cc(CCCN(C)C)nn2)C)n1C c1(CC)[nH]ccc1NC(N1CCC(CCNC(=O)OC(C)(C)C)C1)=O Cn1ncc(NC(=O)NC2CCn3nccc3C2)c1S(N)(=O)=O C1(NC(C)=O)CCN(C(c2conc2C(C)NC(c2c(C)n[nH]c2C)=O)=O)CC1 c1(C(=O)NC(C(C)NC(c2ccc(OC)o2)=O)C)ccc(-n2ccnn2)cc1 O=C(CC1OCCc2ccsc21)NCC1CNCCC12CCC2 c1(C(=O)NC(CC)CNC(=O)CCN2CCC(F)C2)cncnc1C C1(NC(c2cc(C)on2)=O)CN(C(=O)C(N2CCN(C)CC2)C)CCC1CO C1(NC(C(n2ccc(C3CC3)n2)C)=O)CC2(C1)CN(C(=O)Cc1cccs1)C2 c1(SC)ccc(CCC(=O)NC(C)CN(C(=O)CC(C)C)C)cc1 c1(C(C)NC(C2CC(NC(c3cnc(C)n3C)=O)C2)=O)cccc(C#N)c1 CCCCC(CC(=O)NCCOCC(F)(F)F)NC(C1(c2ccno2)CC1)=O c1(COC(C2OCC(C)(C)C2)=O)cccc2[nH]ncc12 c1(C(=O)NCC2(OC)CCN(C(COC)=O)C2)cnn2c(O)cc(C)nc12 C1(CC=C)(C(=O)N(CC(C)N(C)C(C)=O)C)CCCN1C(=O)C=C1CCCCC1 Cc1ccccc1C(=O)N(C)CCN(C(=O)CCC=CBr)C N1(C(c2nccc(CNC(CCN(C)CC)=O)c2)=O)CCCSCC1C CCC(CCC(=O)N1CC(NC(c2c(Cl)cnn2C)=O)C(O)C1)OC C1(OC)(Cn2nnnc2CNC(C)=O)CCN(C(=O)COCc2ccccc2)C1 C(CC(C(=O)NC1C2CC1N(C(c1cncc(Cl)c1)=O)C2)NC(N)=O)SC Cc1ccc(C(CNC(c2nccnc2C)=O)NC(C2(C)CCCS2)=O)cc1 CC1(C)COCC1C(=O)NCC1CCN1C(c1cnc(C(F)F)nc1)=O C#Cc1cnn(CC(=O)NCCCC(C)NC(=O)C(C)SCCCC)c1 C(=O)(CS(N)(=O)=O)N1CC(c2c(C(C3CC(C)(C)CO3)NC(C)=O)nco2)C1 Nc1nc(C(=O)NC2CC(NC(=O)CC3(CO)CC3)C23CCC3)ccc1O c1(C(=O)NC(CCNC(CCc2ccn(C)n2)=O)(C)C)ccc2c(c1)OCCN2 c1(C(=O)NC(CC=C)CNC(c2csnc2OC)=O)cc(Br)ccc1F N1(C(CN(C)CCNC(=O)C(C)(C)n2cnnn2)=O)CCCC1c1ccon1 C#CCC(CC(=O)NC1CCCCCC1F)NC(=O)CC1CC(OCC)C1 c1(C(N)CNC(C2(O)CCNC2)=O)cccc(OC(F)(F)F)c1 C1(F)(C(=O)NCC(C(C)C)CO)CCCN(C(c2cccnc2O)=O)C1 Cc1ccc(C(N2CCS(=O)C(C)C2)C(=O)NCc2ccccc2)c(F)c1 c1(OC)cc(C(N2CCC(O)(CCNC(C3CC3C)=O)CC2)=O)cc([N+](=O)[O-])c1 Cc1[nH]nc(CO)c1C(=O)NC1CC2(C1)CC2C(N1CC(N2CCC2)C1)=O C(=O)(C1=C2CCCN=C2NN1)NCC1N(C(c2cccc(C)n2)=O)CC1 C1(C(N(CCN(C(=O)Cc2ccsc2Cl)CC)CC)=O)CCc2cncn2C1 Cc1nn(CC(=O)NCC2CC2CNC(=O)CC=CC(C)(C)C)c(C)c1Br C1(CNC(C=Cc2n(C)ncc2)=O)CC(NC(=O)CCCC2CCC2)C12CCC2 CC1(C)CN(C(=O)C(O)C2CC2)CC1NC(=O)Cc1ccn(C(F)F)n1 c1(C(N=c2c(OC)c[nH][nH]2)=O)cnc2c(F)c(F)ccc2c1 c1(C(=O)NC2(CC)CCCN(C(c3ncc(Cl)n3C)=O)C2)ccc2[nH]ccc2c1 c1(C(=O)NC2C(C(=O)NCC(C3CCC3)OCC)CC2)ccc(C2CC2)cc1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCC1(NC(c2c(C)ncnc2)=O)CC1 N1(C(C(OCC)OCC)=O)CCC(C)(C)C1CC(N1CCC1C(C)C)=O c1(C(=O)NC(C)CN(C)C(C2CCCCC2C(F)(F)F)=O)cccc2cnsc12 N1(C(C(=O)NCC2(C(=O)OC)CC2)C)CCCCC1C(=O)OC.c1(CC(=O)N)ccon1 C1(C(CC)C)CCN(C(=O)COCCF)CC1.C1=CC(=O)NC1(C)C C1(C(=O)Nc2nc(C)c(I)s2)CN(C(c2cc3sccc3s2)=O)CC(F)(F)C1 N1(C(CC2CC(=O)OC2)=O)CCN(C(C2CCCC2F)=O)C2CC12 C(=O)(C(CNC(=O)C=Cc1ccncn1)CC1CC1)NC(C(C)C)C1CCC1 N1(C(c2cc(C)n(C)n2)=O)CCN(C(c2ccsc2C(F)(F)F)=O)CC1CCO c1(C(C)C)ccnc(N2CC3CC2C3C(=O)NCc2cc(C3CC3)n[nH]2)n1 c1(OC)cnc(Br)cc1C(=O)NCC(C)N(C(=O)Cn1ccnc1C)C C(C)(CCCCNC(C1(P(C)(C)=O)CC1)=O)NC(c1nc(C)oc1)=O C(=O)(C(F)C(F)(F)F)NCC=CCNC(CC1(CC)CCCCO1)=O CC1CNc2c(C(=O)NC(C)(C)CCCNC(C3CCCC3)=O)cccc2C1 c1(C(N2CCC(C(=O)NCc3n(C)ncc3)C2)=O)cc(F)c(C(F)(F)F)c(F)c1 Cc1cc(Br)cc2c1CN(N1CCN(c3ncc(-c4ccccc4)cn3)CC1)CC2 CCCCC(O)C(C)C(=O)NC(CCCC)CC(=O)NCc1cnns1 Cc1cn2ccc(C(N3CCCN(C(=O)CN4CCOCC4)C(C)C3)=O)cc2n1 c1(C(=O)NCC2(C)CCCN(C(CC(=O)OC)=O)C2)cc(Cl)c([N+](=O)[O-])[nH]1 N1(C(c2c(CNC(=O)C=CC3CCOCC3)noc2)=O)CC2CC=CC1C2 CCC(O)C(=O)NC(CNC(c1cnn(C)n1)=O)C(C)C C1(C(=O)NCC2C=CCC2)(SC)CN(C(=O)CC2CC2)C1 N1(C(CC(=C)Br)=O)CCCCC(NC(C2(C)CCCOC2)=O)C1 C1(C(=O)OCC)OCCNCC1N1CCCC(C)C1.N1(CCCN)CCOCC1 CCC(C)(C)CCCC(=O)NC(C)CNC(=O)COCCOCCO C(=O)(C1CCCc2c1ncn2C)NCC(CC)NC(c1ccc(C(F)F)nc1)=O Cc1ccc(C(=O)NC2CC(CNC(C3(C4CC4)CC=CC3)=O)C2(C)C)c(F)c1 C(=O)(C1=CC2CCCC12)NCC12CC(NC(CC(CC)(F)F)=O)(C1)C2 C=C1CCC(C(N2CCC2CNC(=O)CSCCC)=O)CC1 c1(C(=O)NCC(CC)NC(c2ccc(F)c(Cl)c2F)=O)cccc2cc[nH]c12 c1(C(=O)NCC(C)NC(C23C(CN(C(C)=O)C2)C3)=O)ccc(O)c(C(C)(C)C)c1 C(C(C)(C)C(=O)NCC1CCC(C)N1C)N(C(c1cc(OC)ns1)=O)C N1(C(c2ccc(C(C)C)nc2)=O)CCCC2(C1)CN(C(=O)C(C)(C)C(C)(F)F)C2 C1(C)(CC)CC(NC(c2cn(C)cc2C)=O)CN1C(c1sccc1C#N)=O c1(NCc2cc(F)c(C(=O)N=c3cccn[nH]3)c(F)c2)ncnc2[nH]cc(I)c12 N1(C(CN(CCOC)C)=O)CC2CC(NC(c3c(OC)noc3C)=O)C1C2 C1(CC)CN(C(c2cc(Cl)ncc2C)=O)CCN1C(c1cnc(OC)nc1)=O C1(NC(CCS(C)=O)=O)CC2CCC1(NC(c1cc(Br)no1)=O)C2 Cc1cc(=NCCc2cc(O)nc(O)n2)[nH]c(=NCc2c[nH]nc2C(C)(C)C)[nH]1 c1(C(N2CCC(CNC(c3ccc(CC)nc3)=O)C2)=O)cc(F)cc2cc[nH]c12 c1(OCC(=O)N(C2CCC(CNC(C3CC4CC34)=O)CC2)C)cccc(C#N)c1 N1(C(C(C)Oc2ccc(SC)cc2)=O)CCC(NC(C2CCC2)=O)CC(C)(C)C1 C1(NC(C(C(C)C)NC(C)=O)=O)CCC2(C1)CN(C(=O)Cn1cc(Cl)cn1)C2 C1(C(N2CCCC(C)C2CNC(C2CCC(=O)N2)=O)=O)CC2(CCOCC2)CO1 c1(CCC(=O)N(C2CCN(C(c3cc(C(C)C)no3)=O)C2)CC#C)ccccn1 c1(C(N(C2CCCN(C(C(c3cccc(O)c3)C)=O)C2)C)=O)cc(F)ccc1F c1(C(=O)NC2CN(C(Cc3nc(CC)sc3)=O)C3C2C3)ccc(Cl)c(O)c1 C#Cc1ccc(C(=O)N(C(C)CN(C)C(C2(c3ccccc3)CCC2)=O)C)cc1 O=C1CCC(C(=O)NCCCCC(=O)N2CCOCC2C(F)F)CN1 c1(C(C)=O)ccc(C(=O)NC(CNC(=O)CN2CCCC2C)C(C)(C)C)c(F)c1 C1(C(N(C2CCN(C(c3n(C)ccc3)=O)CC2)CC2CC2)=O)CCC2(CCC2)C1 c1(CNC(=O)C(=O)Nc2ccc(OC3CCOC3)cc2)ccc(Cl)cc1O c1(C(=O)NC(C#C)CC)ncoc1CNC(=O)Cc1ccn(C)n1 CC(CCCN=c1cc(C(N)=O)nc(Cl)[nH]1)NC(c1cnc2cc(C)ccn12)=O n1(-c2ccn(CC)n2)nc(C2CC2C)nc1-c1oc(CCOC)nc1C c1(C(N2CCN(C(CN(C(CC(C)OC)=O)C)=O)CC2)=O)cc(C)ccc1F N1(C(C2(CC=C)CCCC2)=O)C2CCC(C(=O)N(C)C)C1CC2.c12ncnn1C2 Cc1nc(C2(NC(C3(NC(N)=O)CC3)=O)CC2)n[nH]1.C1(=O)C(C2CC2)N1 C(C(C)(C)CNC(c1cnn(CC)c1)=O)N(C(c1csnn1)=O)CC c1(C(N2CC3(CC(NC(C4CC4C(F)F)=O)C3)C2)=O)ccnc2cc(Cl)ccc12 c12cc3nncn3c(n1)N2.N1(c2ccc(CC)cc2)CC(C)OC(C)C1 CCCCC(O)CC(=O)N1CCC(OCCNC(C2(c3cccs3)CC2)=O)C1 c1(Cn2c(C3C(C(C)(C)C)OCCC3)nc(-c3cncs3)n2)cc(Cl)cc(Cl)c1 CCC(CC)CCC(=O)NC(CO)C(C)NC(C1CCC(c2ccccc2)O1)=O N1(C(C=CC=CC=CC)=O)CCCC(C)(C)C1CNC(c1cc(N)c(Cl)cn1)=O Cc1c(Cl)ccc(C(N2CCN(C(=O)CC3CCOC3(C)C)CC2)=O)c1O C1(NC(C(C)NC(CC)(C)C)=O)CCN(C(c2ccccc2)=O)C1(C)C c1(C(=O)NC2CCC(CNC(C=C(CC)C)=O)C2)oc(Br)cc1C C1(NC(C2CN(C3CCC3)C2)=O)CCN(c2ncnc3[nH]ccc23)C12CCCC2 c1(CN(C(CCOC(C)C)=O)C)cnn2c1CN(C(=O)C(O)C1CC1)CC2 C1(C(=O)OCC2CC2(C)c2cccs2)CCc2nncn2C1 c1(OC)cccc(NC(=O)C(c2sccc2OC)N2CCC2C(C)C)c1 Cc1cccc2[nH]c(C(N3CCC(C(C)NC(c4cn(C)[nH]c4=N)=O)C3)=O)cc12 C1(NC(C2(COC)C=CCN2C(=O)CN2CCOCC2)=O)CCCN(C)CC1 c1(CCNC(N2CCSCC2c2cccc(Cl)c2)=O)ccc(F)cc1Br Cc1ccc(C(N2CCC(N(C(=O)C(C(C)C)c3cccnc3)C)C2)=O)c(N)n1 C1(NC(C2N(C(C)C)C(=O)CC2)=O)COC2(CCCN(C(=O)OC(C)(C)C)C2)C1 C(CN=C(NC1CC1)NC1CCCN(C(=O)OC(C)(C)C)C1C)OC N1(C(c2cc(COC)no2)=O)CC(F)(F)CC1CCNC(=O)CC12CCCC1C2 N1(C(c2c(=N)[nH]cnc2)=O)CCC2CC1CN(C(=O)CCNC(=O)CO)C2 Cc1nc(C(N2CCCC2C2(C(N3CCC(c4ccon4)C3)=O)CC2)=O)co1 c1(OC(C)C(=O)OC(C(=O)NC2(CNS(C)(=O)=O)CCC2)C)ccc(Cl)c(Cl)c1 Nc1cnc(C(=O)NC(CCC2CC2)C(=O)NC2(c3nn[nH]n3)CC2)cn1 C(=O)(C1=CS(=O)CCC1)N1CCC(C)C1CNC(c1cc(F)ccc1Cl)=O c1(C(N2CCCC(CNC(COCCOC)=O)C2)=O)ccc(C#N)cc1[N+](=O)[O-] C1(C)(NC(CCS(C)=O)=O)CCCN(C(=O)Cn2cccc(N)c2=O)C1 N1(C(C(C)OCC2CC2)=O)CC2CC(NC(=O)CC3(c4ccccc4)CC3)C2C1 CN1N=C(CC(=O)NC23CC2CN(C(c2cc4ccc(Cl)nc4s2)=O)C3)CC1=O c1(C(N2CC(NC(C(c3cn(C)nc3)O)=O)C2)=O)cc(O)nc(Br)c1 N1(C(C(=O)NCCC(=O)OCC)C2=CCSC2)CCc2cccc(O)c2C1 N1(C(CCc2ccc(C)o2)=O)CCC(C(=O)NCC(C)CCCO)(CF)C1 C1(CNC(C2(CC#C)CCOC2)=O)CC(C)CCN1C(c1ccsc1C#N)=O C(=O)(C1=C(CC)OCCS1)NCC1CN(C(C2CCC(CCC)CC2)=O)C1 Cc1n[nH]c(=NC2CC3CC(C2)N(C(=O)CCSc2nnnn2C)C3)o1 C(=O)(CCCNC(=O)C(C)C)N(C(C(=O)NC(CC)(C)C)C)CC1CC1 N1(C(C2(C)C(C)C2)=O)CCC2(CCCC2N2CCC23CCCCC3)CC1 C1(CNC(C(C)OCCOC)=O)CCCCN(C(=O)CCCn2cc(C)cn2)C1 CCN=c1cc(-c2nc(-c3occc3C)n(CCN(C)C)n2)cc[nH]1 CC1(C)CCN(C(=O)NC(CCO)c2cccs2)C1 c1(C(=O)NCC(=O)NCCC(C)(C)NC(C(CC)C)=O)cccc(Cl)c1 C(C(F)(C(=O)NCC1(CN(C)C)CCC1)C(C)C)NC(Cn1ncc(C#C)c1)=O c12cccc(n1)CN2.c1(C(=O)NC(c2n(CC)ncc2)C2CC2)cccc(CO)c1 c1(C2(CNc3cc(NC(C=C)C)ncn3)CC2)c(F)cccc1F n1(CC)cc(C(=O)NCC2CCCN2C(=O)CC2(C)CC2(F)Cl)c(C(C)C)n1 c1(CN(CC=C)C(C2CCC(C(=O)O)S2)=O)ccc(C(=O)OCC)cc1 N1(C(C(C=C)OC)=O)CCC(C)(C)C1C(=O)NCC1CC(C(C)C)C1 C(=O)(CCCS(C)(=O)=O)N1CCCC(O)(CNC(c2c(C)nco2)=O)C1 C(c1ccccc1)=CCC(=O)NCC1CC1C(=O)NCc1c[nH]ccc1=O C(=O)(CC(C(=O)N1CCC(O)CC1)S(=O)(=O)CC(C)(C)C)Nc1c(C)cccc1 C=CC(CCC)CC(=O)N1CCN(CC(C)NC(c2coc(C3CC3)n2)=O)CC1 N1(C(CSCC=C)=O)CCN(C(C2(O)CCOCC2)=O)CC1CO C1(NC(C2(CC#C)CC=CCC2)=O)CN(C(c2n[nH]c(CC)n2)=O)CC1(C)C C1(C(=O)NC(C2(O)CCN(C(=O)CCS(C)=O)C2)C)CC12CCCCCC2 Cc1ccc(CN2CCCC(C(=O)Nc3cccnc3I)CC2)cc1[N+](=O)[O-] C(=O)(CCCc1nccs1)N(C)CC1(NC(c2cnn(C3CCOC3)n2)=O)CC1 CN1CCCCC1CC(=O)NCC(C)(O)CNC(C1CCC(C(N)=O)CC1)=O C1(COC)(NC(=O)CCC(C)O)CCN(C(=O)Cc2cnnn2C)CC1 C(C(CC(C)C)C(=O)NC1CCC1NC(c1ccsn1)=O)OC C1(CCNC(c2c(C)nco2)=O)CN(C(=O)CCc2nc(O)n[nH]2)CC(C)O1 N1(C(COCC=C)=O)CCC(CNC(c2cccn(C)c2=O)=O)CC1C N1(C(CC(C)N2CCCC2=O)=O)CC2CC1C2NC(=O)C(c1ccccc1)O CC1(C)CCOC(CNC(C2N(C(=O)C=CC(=O)N(C)C)CCC2(C)C)=O)C1 O=S(=O)(c1ccc(Br)cc1NCCCC(F)(F)F)NC(Cc1ccccc1)CO C1(C)(C(=O)NC2(CC)CCOC2)C=CCN1C(c1cccnc1C)=O C1(C(=O)NCCC2(CNC(C3(C)CC=CCO3)=O)CC2)CCC2CCCCN12 c1(OC)nc(C)sc1C(=O)NC1(C)CC(NC(c2cccnc2N(C)C)=O)C1 c1(OC)ccc(C(N)=O)cc1C(=O)NCC1CN(C(=O)C(C)N2CCC2)CCO1 O=C1CC(c2cccs2)CC(=O)N1C.c1(SSC(CC2CC2)CO)ccccc1 CCCCCC(O)CC(=O)NC(C)CC(=O)NC(C)(CO)C(C)(C)O C(=O)(C1=NOC(C)(C)C1)NC1(C)CCN(C(CCSC)=O)C1 C1(S(N)(=O)=O)(C(N(CC(C)NC(c2cccnc2C(F)F)=O)C)=O)CCCC1 c1(NC(C2(C)CN(c3nnc(C)o3)C2)=O)nccnc1C(N1C(C)CCC1C)=O C1(CC)CCCN(C(c2ccc(O)c(F)c2)=O)C1C(=O)N(CC(F)Cl)C CCN=c1[nH]c(C)c(C(=O)NC(C)C(C)NC(=O)C(F)(F)c2nccs2)s1 C(=O)(C1c2ccccc2CN1C(=O)C(O)CC(F)(F)F)OC(C)(C)C c1(NCC(CCCC)NC(=O)C(C)(C)C(C)(F)F)cc(C)c([N+](=O)[O-])cc1Br N1(C(C2CCC(=C)CC2)=O)CC(NC(=O)CCn2cc(C)cn2)CC(O)C1 C1(C(=O)NCCN(C(=O)CC2(CC)CCC2)CC)Cc2cncn2C(=O)N1 C1(F)(C(N2CC(F)(CNC(CNC(C(C)(C)C)=O)=O)C2)=O)CCCOC1 C=CCC(CC=C)C(=O)N(CC(CC)NC(C1(CO)CCOC1)=O)CC c1(CN2CCC(CC(=O)Nc3cc(Cl)c(F)cc3Br)CC2)ccc(F)c(F)c1Cl c1(CC)oc(C(=O)OC)cc1S(=O)(=O)NC1(c2ccccc2OC)CCC1 c1(C(N2CC(O)(COC)C2)=O)cc(CNC2CCCC2)cc(Br)c1 c1(C(=O)NC2CC3CC(NC(c4cccnc4O)=O)CC23)ccc2occc2c1 C(=O)(C1=CS(=O)CCC1)NC1CC(NC(C(C)OCCN(C)C)=O)C1 n1(CC(=O)NCCCCN(C(C(C)CN(C)C)=O)C)ccc(=O)n(C)c1=O Cc1ccc(-c2nc(CS(=O)(=O)CC3OCCCO3)cs2)c(C)c1 c1(C(N2CC(CNC(=O)CC34CCCC3C4)C(O)C2)=O)cccn2nnnc12 CC(C)CC(C(=O)NCc1cnnn1C)ONC(=O)CCc1nc(O)n[nH]1 c1(NC(c2c(NC(=O)C=Cc3cnc[nH]3)c[nH]n2)=O)c(F)cc([N+](=O)[O-])cc1Br c1(C(N2CC3CC3(CNCc3ccc(F)c(O)c3F)C2)=O)ccc(F)c(F)c1F c1(C(N2CC(CCC)N(C(C3CCCS3(=O)=O)=O)CC2)=O)c[nH]c2cccnc12 Cc1nc(C(N2CC(C)CC2(C)C)=O)ccc1-c1ccc(N(CCC#N)C)cc1 CC1CCN(C(C2(O)CCCCC2)=O)CC1CC(N1CCC2(CSC2)C1)=O Cc1nc(C=CC(=O)N(C)CC2(O)CCN(C(=O)C(O)C(C)(C)C)C2)[nH]c1C C1(NC(C)=O)CC(c2ccccc2)(NC(C2CCC(CN(C)C)C2)=O)C1 c1(C(N2CC(NC(Cc3c(C)n[nH]c3)=O)C2)=O)ccc(S(=O)(=O)N(C)C)cc1 c1(CC(N2CC(C(C(=O)NCCN(C3CC3)CC)O)C2)=O)ccc(O)cc1 Cc1n[nH]c(C)c1CNC1CCCC1C(=O)NC(C)Cn1cnnc1 c1(C(C(=O)NC(CNC(C2(C(C)C)CCC2)=O)CO)C2CC2)cccc(Cl)c1 CC(CNC(c1cc(C#N)c[nH]1)=O)CC(=O)NC1(c2ncccn2)CC1 N1(CCC(=O)NC2CCN(C(CCC#CC)=O)C2C)Cc2ccccc2C1=O CC(N=c1[nH]c(=NCc2cc(Cl)ccn2)[nH]c2c1COC2)C1CCCO1 c1(OC(C)C)c(C(=O)NCC(n2cc(C(C)(C)F)nn2)C)cccc1F N1(C(CC2CC(C)(C)OC2)=O)CC(CO)C2(C1)CN(C(C1CS(=O)(=O)C1)=O)C2 CC1(CNC(C2CCCCC2n2cc(CO)nn2)=O)CCCNC1=O.C1C(=O)N1 Cc1cccnc1CC(=O)N(CC(C)NC(c1cnc(S)n1C1CC1)=O)C CC1OCCC1(F)C(=O)NCCOCCOCCNC(c1cnc(C(N)=O)s1)=O C1(NC(CCN(C(=O)CC#N)C2CC2)=O)CCC2(CC1)N=N2.CC(=O)OC c1(C(=O)NC2CN(C(c3c(CC)con3)=O)CC(O)C2)ccc2ccsc2c1 N1(C(c2c(CC)cco2)=O)CCC2(CC1)CC2C(=O)NC1(CC)CC=CCC1 n1(CCC)nc(C)c(C(=O)NCCC2CCN(C(=O)CC3CC=CCC3)C2)c1C CC(C)C(C)C(=O)N1CC(NC(c2ccc(CC(=O)N(C)CC)cc2)=O)C(C)C1 C1(C(=O)NCc2ccc(CCNC(C(CC)C#N)=O)cc2)CN2CCN1CC2 C1(C(C)NC(c2cnn(C3CCCC3)c2)=O)CN(C(C2CCC2)=O)CCO1 Cc1cccc2c(C(=O)N(CCCCCNC(C3(Cl)CC3)=O)C)cnn12 CCCCC(C(=O)NC12COC(C1)C(NC(C1CC(OC)C1)=O)C2)OC CC(C)CC(CNC(C1CCCC(C(F)(F)F)C1)=O)NC(=O)COC1CC=CC1 c1(C(N(C2CCN(C(=O)Cn3cc(C)cn3)C2)CC#C)=O)cc(C(F)F)ncn1 C1(C(N2C3CC(NC(C4C(C)CC(C)O4)=O)C(C3)C2)=O)CN2CCN1C(C)C2 CC1=NOC(C(=O)NC23CC(CNC(=O)CC4CCCCC4O)(C2)C3)C1C c1(C(=O)NC(C(=O)NCCCN(C)C2CC2)C2(C)CC2)c[nH]c(C#N)c1 C(N=c1[nH]c(C2CC2)nc(C)c1I)C1(OC)CC(CC)C1 C(=O)(C1=C(Cl)CCC1)NCC1(OC)CN(C(=O)CCOCC(F)(F)F)C1 N1(C(c2c(CC)cns2)=O)CC(C)C(C)(CNC(=O)CN2CCC(C)(C)C2)C1 C1(NC2CCC(NC(N(c3cccc(C)c3)CC)=O)C2)CC(=O)N(O)C1 C1(C2CN(C(c3ccc(-c4cnco4)cc3)=O)C2)(NC(C=CCC)=O)CC1 C1(CN(C(=O)CSC(F)F)CC)CCCCN1C(c1cnc(C(C)=O)s1)=O C1(NC(c2c(OCCOC)scc2)=O)CCCCC1c1scc(CNC(N)=O)n1 C1(O)(CNC(CN(C(CNC(CC)=O)=O)C(C)C)=O)CCC(C)(C)C1 C1(NC(CNC=O)=O)CC12CCC(NC(c1cn(C3CCOC3)nn1)=O)CC2 c1(C(=O)NCCN(C(c2cncc(F)c2)=O)C2CC2)cnc2nccn2c1 N1(c2cc(C)nc(N3CCC(C(F)F)C3)n2)CCC2(CCN(C)C2=O)C1 N1(C(C(CC(C)C)NC(C)=O)=O)CCCN(C(C2C=CCCC2)=O)CC1C c1(C(=O)NCCN(C(C)C(=O)NC2CCCCC2)CC)cccc2c1CCOC2 C1(NC(c2c[nH]nc2-c2ccc(Cl)cc2)=O)CN(C(C2(CCF)CC2)=O)CC1F C12(CSC)CC(C(=O)NCC=C3CCN(C(=O)Cc4ccnn4C)CC3)(CO1)C2 N1(C(c2c(C)n[nH]c2)=O)CC2OCC(NC(=O)CC3CCC3)C2C1 c1(OC)ccc2nnc(CNC(=O)CC3(C(F)(F)F)CCC3)n2n1 Cc1noc(C)c1S(=O)(=O)N1CCc2cc(-c3n[nH]c4c3CNC4)ccc21 C1(CNC(Cc2c(C)cc(N(C)C)cc2C)=O)CC12CCS(=O)(=O)CC2 c1(C(=O)NC(CCN(C(CC)=O)C)C)cc(OC)ccc1OC N1(C(c2c[nH]c(=NC)s2)=O)CCCC(CNC(C2CCN(C(N)=O)CC2)=O)CC1 N1(C(CCOCCOC)=O)CC(NC(=O)C(C)NC(=O)COC)C(O)C1 c1(C(=O)NC(C2(O)CCN(C(CC(=C)Br)=O)C2)C)ccc(F)c(F)c1F c1(C(=O)NC2C(CC)N(C(=O)CSc3cccs3)CC2)c2ccccc2nn1C N1(C(C(CC)F)=O)CCN(C(=O)CN2Cc3ccccc3C2)CCC1C c1(NC(C2N(c3cc(OC)nc(C)n3)CC(O)C2)=O)ccc(C)c2ncccc12 CC1CC(C(=O)NCC(O)C(C)O)CN(C(=O)CN2CC3CC3C2)C1 C12(CNC(=O)Cc3ccc(F)c(Cl)c3)CN(C(=O)C(C)OCO)C(CC)(C1)C2 c1(C(=O)NC(C)CNC(=O)CC2CC2C2CC2)ccc2oc(=N)[nH]c2c1 N1(C(COC(CC)(C)C)=O)CCN(C(=O)C(=Cc2c[nH]cn2)F)CC1CC1CC1 n1(CC)ncc(Cl)c1C(N1CCC(C(C)NC(c2cc(C)on2)=O)C1)=O C1(CCCCC)CCC(NC(c2csc(CC(C)C)n2)=O)CC1 C1(C(=O)NC2C(CC(=O)N(C)Cc3cn(C)nn3)CCC2)COC(=O)N1C c1(OC)ccc(CC(=O)NC2(C3CCCN3C(C3CC(C)(O)C3)=O)CC2)cc1Cl c1(C(=O)NC(C2N(C(C(C)OCCC=C)=O)CCC2)C)cc2c(C)cccc2[nH]1 C1(NC(CN2CC(C)C2)=O)CCCC2CN(C(C3CCc4nncn4C3)=O)CC12 Cc1cccc(C(c2nnnn2C(C)C)NC(C)Cc2c(C)noc2C)n1 c1(C(=O)NC2CCC(CCC(=O)N(CCOC(C)=O)C)C2)cccnc1O N1(C(Cn2cc(C(C)O)nn2)=O)CCN(C(c2cnn(C)c2N)=O)C(CCO)C1 Cc1cc(C(=O)NCc2ccc(C(=O)NC(C)C(C)O)cn2)[nH]c1C Cc1ccn2cc(C(N3CCOCC(CNC(=O)C(C)C(C)O)C3)=O)nc2c1 c1(N2CCCC(C)(CNC(c3c(CC)nc(C)[nH]3)=O)C2)nc(C)cc(C)c1C#N N1(Cc2ccc(C)s2)CC(C2CCCN(C(c3c(Cl)cccc3Cl)=O)C2)C1 N1(C(C2C(C)C2)=O)CC(NC(C2CC(O)(c3ccccc3)C2)=O)CC12CCC2 CC1(NC(c2cscc2C2CC2)=O)CCN(C(=O)COCC2CCC2)C1 c1(CC(=O)NC(C(=O)NCC=C)C2CC2)ccccc1O CC(C)S(=O)(=O)C(C)C(=O)NC1CC(CO)N(C(=O)COC2CCOCC2)C1 C1(NC(C2(CC=C)CC=CC2)=O)CCCCC1NC(=O)C=Cc1cccs1 N#Cc1ccccc1C1(C(=O)NC2CC2NC(=O)C2=COCCC2)CC1 C12(NC(C(Cc3ccco3)NC(c3ccc(CC)nc3)=O)=O)CCC(C1)OC2C C1(C(=O)N(c2cncnc2)Cc2cccc(OC(F)F)c2)COC2(CCNCC2)C1 N(C(=NCc1nc(Cl)cs1)NCc1ccccc1)CCNC(c1ccoc1)=O C=CC1OCCCC1C(=O)NC1CC1NC(=O)CCc1cccc(OC)c1OC CC1(NC(=O)C=Cc2ccncc2)CCN(C(C2CCCC2C(F)(F)F)=O)C1 c1(C(N2CC(C(C)NC(CSCCN(CC)CC)=O)C2)=O)ccccc1C C1(NC(C(c2cccnc2)NC(C2C(C)C2)=O)=O)CCCN(CCO)C1 C1(NC(COCCC=C)=O)COCCN(C(c2c(C)nn(CC)c2C)=O)C1 CCC(F)(F)CC(=O)N1CC(C)C(C)(C(=O)NCC2Cc3nccn3C2)C1 CC(C)CS(=O)(=O)CC(=O)N1CCCCC1CNC(=O)C=Cc1nccs1 c1(C(=O)NCC(CC)NC(=O)C(C)NC(=O)NC)ccnc2ccsc12 c1(C(C)C)cccc(C(=O)NCC2CCCC2NC(=O)C=Cc2cncn2C)c1 Cc1ccccc1C(F)(F)C(=O)NCCCN(C)C(c1ncoc1C1CC1)=O C1(C)(C(=O)NC2(CC(=O)N(CC(CC)(C)OC)C)CC2)CC2CC2C1 C1(C(=O)NC2(CCCNC(C(C)=C3CC3)=O)CC2)CC(C)=NO1 C1(C(N2CCC(C=C)C2)=O)CCc2nnc(Br)n2C1 C12CCCC1N(C)C2=O.N1(CC)CCC(NC(C2(n3nccn3)CC2)=O)C1 C(=O)(C(C)C(O)C(C)C)N(CCC(=O)NC(C)(C)CC1CCC1)CC=C N1(CCOC)CC(C(=O)NCC(C)CN(C)C(C2CCS(=O)(=O)C2)=O)CCC1=O C1(NC(CC2CCCC(C)C2)=O)CC2(CCCCN2C(=O)CP(C)(C)=O)C1 Cc1ccc(C=CCC(N2CCC(O)(CNC(c3ccc(Cl)o3)=O)CC2)=O)cc1 C1(CNC(=O)C(c2ccccc2F)F)C2CN(C(=O)C=CC3CCOC3)CC12 CC1C(NC(=O)Cc2cccs2)CCN1C(=O)CC1CCN(C)C1=O Cc1ccc(C)c(SCC(=O)NC2COCCC2NC(c2cc(C)nn2C)=O)c1 C1(C)(C(=O)NCCC2CCCC(C)C2)CCCN(C(=O)Cc2n[nH]c(=N)s2)C1 CC1CCC(n2cc(C(N3CCC(O)(C(N)=O)C3)C(=O)NC(C)(C)C)nn2)CC1 N1(C(C2CC(C)(CC)C2)=O)CC2(C1)CN(C(C13CCCC(O)(CC1)C3)=O)CCO2 C1(NC(C2(C#C)CCC2)=O)CCOCC1NC(C1CCCN1C(=O)OC(C)C)=O N1(C(C(C)OCCCC)=O)CCN(C(=O)COCC2CC2)C(C2CC2)C1 c1(C(N2C(C)(CC(=O)NC(CO)C3(O)CC3)CC2)=O)cccc(CC#N)c1 N1(C(C2C(CNC(CCOCC)=O)CCC2)=O)CCN(CC)C(C)C1 C1(CNC(C(C)OCC)=O)CC(C)(C)CN1C(c1csc(-c2cccnc2)n1)=O c1(C(N2CC=CCC2)C(=O)NC(C(=O)OC)C)cnn(C(F)F)c1 Cc1cnc2n1C(C(=O)NC1CN(C(C3CCOCC3)=O)CCC1(C)C)CCC2 CC1(CSc2cn(CC(=O)O)nn2)CCCO1.C12CCC1C(=O)N2 c1(C2N(C(c3ccsc3C(=O)OC)C(=O)NCCOCC)CC2)cccc(Cl)c1 C1(C2CN(C(=O)Cc3cc(F)ccc3O)C2)(NC(C2CCOC2)=O)CC1 C1(CNC(c2nnnn2C2COC2)(CC)C2CCC2)CC2C(C1)C2(F)F N1(C(=O)CCC2CC(F)(F)C2)CCCN(C(c2csc(C3CC3)n2)=O)C(CO)C1 C#CCCCCCCC(=O)NC(CC#C)CC(=O)NC(c1nn[nH]n1)CC c1(CC2CCN(C(=O)NCc3cccc(-n4cnnn4)c3)C2)ccccc1F c1(C(N2CC(F)CC(NC(C(CC)O)=O)C2)=O)noc2c1CC(F)(F)CC2 c1(COC(C(CCCOC)C)=O)csc2cc(Br)ccc12 Cc1c[nH]cc(-c2nc(-c3cccc(C(F)F)c3)nn2CC2CC2C)c1=O O=C(C#CC1CCC1)N1CCC(NC(C2(F)CCC2)=O)C(O)C1 CC(C(=O)N(C1(CNC(=O)OC2CCCC2)CC1)C)N(C(=O)CSC(C)(C)C)C CCS(=O)(=O)CC(=O)NC1CCC(C)N(C(c2cc(C(=O)OC)cs2)=O)C1 n1(CC)nc(C(=O)NC2CCC(CNC(=O)C(C(C)O)N(C)C)C2)cc1C1CC1 c1(OC)cc(=O)n(C)cc1C(=O)NCC1CC(O)(CNC(c2coc(C)n2)=O)C1 C(=O)(C(C)CN(C)C)NCC(C)C1(CC=C)N=N1 N1(C(c2ncc(C)cc2C)=O)CCC2(CC1)OCCC2NC(=O)C1=CCCCO1 CCCCC(CNC(=O)CC(F)(F)Cl)NC(c1csc(-c2ccccc2F)n1)=O C(=O)(C(C)CCCC)N1CCC(CCC2N(C(CC=C=C)=O)CCC2)CC1 C(CCCCNC(C1CC1c1ccsc1)=O)NC(CSC(C)(C)C)=O N1(C(c2nc(CC)[nH]n2)=O)CCN(C(=O)CCNC(C2CCCO2)=O)C(C)C1 C1(CC=C)(NC(=O)C(C)c2cccs2)CN(C(c2cn(CCOC)nn2)=O)C1 C1(C(=O)NC2C(C)CCN(C(C3(C(N)=O)CC3)=O)C2)CCc2nnc(O)cc2C1 CC1=NNC(=O)C1CC(=O)NCC(C)NC(c1[nH]cnc1Cc1ccccc1)=O C1(NC(c2[nH]c(=NC)sc2)=O)C2CC(O)C1N(C(C1CN3CCN1CC3)=O)C2 CC1CCC(NC(=O)CCn2ccnc2)CN1C(C1COC(C)(C)CO1)=O c1(C(=O)NCC2CC(C(=O)NC3CC(OC)C3)C2)ccc2[nH]ccc2c1 C1CC(O)C(=O)N1.c1(C(=O)OC(C)(C)C)nc(C2CCCCC2)cs1 Cc1nc(CO)ncc1C(N1CCCCC(NC(=O)CCC2CC2(C)C)C1)=O c1(CNC2CC3CN(C(C4CC(N(C)C)C4)=O)CC32)ccnc2ncnn12 CC(C)CC(CNC(=O)CC1CC(C)(C)CO1)NC(c1cccc(Cl)c1)=O Cc1nc(O)ccc1C(=O)NC1CC2(C1)CN(C(=O)CN(C)CCO)C2 c1(CO)cccc(-c2cn(C(C3CCCCC3)CN3CCCC3)nn2)c1 C1(NC(COCC=C)=O)CCCC2CN(C(=O)C=Cc3ccc(F)c(C)c3)CC12 n1(C(C)C(=O)N2CC(NC(C3CC3c3ncon3)=O)C2)cnc(C#N)n1.C1CC1 c1(OC)ccc(OC)c2sc(=NCCCCC3CCCCC3)[nH]c12 N1(CC(N2CCC(C(C)(C)NC(C3(F)CCOC3)=O)C2)=O)CCCCCC1=O Nc1nc(C(=O)NCC2CC2CNC(c2cnc(-c3cccs3)o2)=O)ccc1O C12(C(=O)NCC3N(C(c4ccc(Cl)o4)=O)CC(F)C3)CCCN1S(=O)(=O)CC2 C1(CN(C)C)CCN(C(c2ccc(CNC(=O)CSCCF)o2)=O)C1 C=CC(C)(CC)C(=O)N(CCCCCC(=O)N1CCC(OC)C1(C)C)C c1(COC(c2cn(CCC)nc2C)=O)ccncc1C#N C1(OC)CC(NC(c2ccc(F)cc2Cl)=O)CN(C(=O)Cc2ccc(O)nc2)C1 C1(C(=O)NC(CN(C(c2c(COC)cc[nH]2)=O)C)(C)C)CCC(F)(F)C1 N1(C(COC(CC)C)=O)CCC(NC(c2ccc(C)c(N)c2)=O)C2(CCC2)C1 c1(N2CCN(CCNC(CC(CC)OC)=O)CC2)cc(=O)n2oc(C)cc2n1 c1(NC(c2nc(-c3ccc(C)c(C)c3)sc2C)=O)cc([N+](=O)[O-])ccc1Br N1(C(COC)=O)CCC(CCNC(=O)CCc2ccc(Cl)c(Cl)c2)CC1C CC1(C)CCCC(C)(C)C1C(N1CCN(C(=O)C(F)F)C(C2CC2)C1)=O Cn1ncc2c1CCCC2N=c1[nH]c(=N)[nH]c(=NCC2COC(C)(C)CO2)[nH]1 CC#CCC(C(=O)NCc1cccc(CSC)c1)NC(=O)CCCNC(N)=O N=c1cc(C(=O)NC2(c3cccc(F)c3)CCN(C(=O)C(=O)N(C)C)C2)cc[nH]1 C(=O)(C(CC(C)C)OC)NCc1c(CNC(CC=CC=C)=O)cccc1 C1(NC(Cc2n(C)nnc2)=O)CCC2CN(C(=O)Cc3ccccc3O)CC2C1 Cc1nc([N+](=O)[O-])cn1CCC(=O)NC(C)CNC(c1n[nH]cc1C(C)(C)C)=O c1(NC(CC2C(NC(CCOC(C)=O)=O)CCC2)=O)cc(Cl)ccc1C Cc1nc(C(=O)NCC2(C)CCN(C(=O)CC3CCCO3)C2)c(C)s1 N1(C(=O)NC)CC2C(C(=O)NC3(NC(C4CCOC4)=O)CCC3)C2C1 C1(C(=O)NCc2ccc(CN(C)C(c3ccco3)=O)cc2)CC2OC1C1CC21 c1(C(=O)NC(C2CN(C(c3ncccn3)=O)C2)C)ccc([N+](=O)[O-])c(C#N)c1 C#CC1(C(=O)NC(C)CC(C)C)CN(C(=O)CN2C(=O)CNC2=O)C1 CC12CCC(C(=O)NC3COCCC3NC(c3ccncc3Cl)=O)(C1)OC2 C1(CNC(CCN(CCC(C)(C)C)C)=O)COCCN1C(=O)Cc1ccnn1C C=CCCCCCCCC(=O)NCC1CCCN(C(C2(COC)CC=CC2)=O)C1 c1(C(=O)NC(C)CN(C(=O)CCc2cscn2)C)nn[nH]c1C(F)(F)F Cc1nc(C(=O)NCC(C)N(C)C(c2ccn(C3CCCC3)n2)=O)c(C)n1C Cc1nc2c(NC3C(C)CN(C(=O)C4=CCCOCC4)CC3C)ncnc2s1 Cc1scc(C(=O)NC2CCC(CCNC(=O)C(F)(F)c3ccncc3)C2)c1C CC(C)CCCCC(=O)NC1CCN(C(=O)C(F)C2CCOC2)C12CCC2 C12(CNC(Cc3c(C)non3)=O)CCC1CCN2C(c1cnn(C(C)C)c1N)=O C(N=c1cc(CO)n(CCO)[nH]1)(c1cc(F)ccn1)c1n(C(CC)(C)C)nnn1 c1(-c2ccn(CCCNC(=O)NC(C)C)n2)ccc(F)cn1 N1(C(c2c(C)ncn2C)=O)CC(CO)C2(C1)CN(C(C1CCCCC(=O)N1)=O)C2 c1(C(=O)NCCC(CNC(CC(C)C(F)F)=O)O)sc2nccnc2c1N C1(NC(C(F)=CCC)=O)CC2(C1)CC(CNC(=O)C(c1ccccc1)N(C)C)C2 CCC(CCC(=O)NC(C)(CO)C(=O)N1CC(CC(F)(F)F)C1)OC O=C(CCCC(F)(F)CO)NCC1CC2CCCC2N1C(=O)Cn1cnnc1O N1(C(C(COCC)C)=O)CC2(CC)CC1(CNC(=O)C(c1ccccc1)C)C2 C(=O)(CC(C)CC(=O)NCC1CCC1C(=O)NCC1(CO)CCN(C)C1)OC CC1C(NC(=O)C(F)(F)Oc2ccccc2)CCCN1C(=O)CN1CCCC1C c1(C(N(CC(C)NC(=O)Cc2c[nH]c3ccccc23)C)=O)cc(S(N)(=O)=O)cs1 c1(C(=O)Nc2scc(C(C)(C)C)n2)cccc2occc12 C1(CC(=O)NCC(CNC(C(C)n2ccnc2)=O)O)CC(C)(C)C(=O)N1 C1(C)(C(=O)NCCCCC(=O)NC2(COCC)CC2)CCC(=O)NC1 C1(F)(C(N(C(CC(=O)N(CC(CCC)O)C)(C)C)C)=O)CCC(C)CC1 CCCCC(F)(F)C(=O)N1CCN(C(=O)Cc2cc(C3CC3)on2)C(C(C)C)C1 N1(C(C(C)(C)C)=O)CCC(C(F)(F)F)C(CNC(=O)CCc2ccc(Cl)s2)C1 c1(OC)ccc2occ(C(N3CCOC(Cc4ccccc4)C3)=O)c2c1 C1(NC(C2CC(SC)C2)=O)CCC2(CC1)CC(NC(=O)C(c1cccn1C)=O)C2 N1(C(C(=O)N(C(C)C)C)C)CCC2(CN(C(=O)CC3CCC4CC34)CC(C)O2)C1 c1(C(N2CC(C)N(C(c3ccn(C)n3)=O)CCC2)=O)cc(F)cc2c1C(=O)CC2 c1(C(N2CC(C(N(C(C)C)CC3CCCO3)=O)(CO)C2)=O)cncn(C)c1=O c1(C(=O)NC(C2CCCN(C(COCCOC)=O)C2)C)cccc(CO)c1C C(=O)(C(F)CC(C)(C)NC(=O)C=C1CCCCC1)N(CCCC)CCO c1(CC)cc(C)ccc1C(N1CCC(C)(NC(C2CC(=O)C2C)=O)CC1)=O c1(C(=O)NC(CNC(c2cnc(SC)s2)=O)C)cc(Cl)cc([N+](=O)[O-])c1 C1(OC)CC2CC1CN(C(c1ncoc1CNC(C13CCC(CC1F)C3)=O)=O)C2 C1(F)(CNC(C2C(C)C2C)=O)CCCN(C(=O)C=Cc2ccc(C(N)=O)o2)C1 C1(CNC(CCOCC(C)C)=O)CC(C(=O)N(C)CCSCCCO)=NO1 c1(CC(=O)NC2CC(C(N(C(C3CCC3)C)C)=O)C2)ccc(O)cc1 c1(C2CCN(C(=O)Oc3ccccc3)C2)cccc2ccccc12 C1(C(=O)NC(C2CCN(C(=O)CN3CCOCC3=O)C2)C)CN(S(N)(=O)=O)C1 C1(CNC(c2cncc(Cl)c2)=O)(CO)CCCN(C(=O)C(F)CC2CCOC2)C1 C1(CN(C)C(c2ccncc2Br)=O)CN(C(=O)CCc2ccc(=N)[nH]c2)CCO1 c1(CC(C(=O)N(C2CC2)CC2COC(C)(C)O2)N)cc(Br)cc(Br)c1 Cc1nc2n(n1)CCCC2NC(C1(S(C)(=O)=O)CC1)c1nnnn1C(C)C c1(OCC)ccc(CC(=O)NCC2CCCN2C(c2cccc(F)c2)=O)cc1 c1(CC(=O)N(CC(C2CCOC2)NCC)CC)cccc(OCCOC)c1.C(C#N)O N1(C(c2ccc(C)cc2N)=O)CCC2(CC1)COCC(CNC(C1CC1C)=O)O2 C1(C(N(CC(CC)NC(=O)CC2(CC)CCC2)CC)=O)CCCCCN1C c1(CNC(C(N2CC3CN(C(C)C)CC3C2)C)=O)cc2ccccc2n1C C1(C2CC2)(NC(c2ccncn2)=O)CCN(C(C2(C3CCCCO3)CC2)=O)C1 C1(CCC(=O)N(C2COCC2O)C)CCCCN1C(=O)CC1CCCC1 C(CC(C)C(=O)NC(C)(CNC(=O)Cc1ccccc1)C1CC1)=CC Cc1cc(-n2cc(CN(C(=O)C(c3cccc(Cl)c3C)O)C)nn2)ccc1F c1(C(N2CC(CCNC(c3[nH]ccc3C)=O)(OC)C2)=O)ccc(C)cc1 CC1(NC(C2CCNC(=O)C2)=O)CCC(NC(c2cc(F)cnc2O)=O)CC1 c1(C(=O)NCC2CN(C(C3(SCC)CC3)=O)C2)cc(F)cc(F)c1N N1(C(Cc2c(C(C)C)con2)=O)CCC(NC(=O)CCC(=O)N(C)C)C(O)C1 C1(N(C(=O)C(F)=C2CCC2)C)CCCCC1N(C(=O)CCCc1cnccn1)C C1(=O)C(C(C)C)O1.CCCC=CCCOC(C1(CN)CC1)=O c1(C(=O)NC2CN(C(CCCC=C)=O)CC2C=C)ccn2[nH]c(=N)nc2c1 c1(N2CC=CC(NC(C(CCCC)(C)F)=O)C2)nccc(C(=O)NC)c1[N+](=O)[O-] n1(Cc2c(CNC(=O)C(=O)N3CC(SCC)C3)cno2)nc(C)cc1C Cc1[nH]c(C#N)cc1C(N1CC(NC(=O)C(c2ccc(F)cc2F)(F)F)C1)=O Cc1nn(CC(C)C)c(C)c1CC(=O)NCCNC(C1CCCC(O)C1)=O C1(C(N2CCC(NC(=O)CCCc3ccccn3)C2)=O)CC(=O)N(C2CC2)C1 Cc1[nH]nc(C(=O)NC2CC(C)CN(C(=O)C(=O)NCC(F)(F)F)C2)c1[N+](=O)[O-] CC1CCCN(C(=O)CN2CC(=O)NC2=O)C1CCNC(c1nc(=N)cc[nH]1)=O c1(N2CC3N(C(C4CC(=O)NCC4)=O)C(CC3)C2)[nH]cnc2nc(Br)cc1-2 CC12CN(C(C34CCCC3C4Br)=O)CC1CN(C(=O)CCC1CC1)C2 N1(C(C2C(C(=C)C)OCC2)=O)Cc2ccc(CNC(=O)C(F)C3CCC3)cc2C1 c1(OC)cccc(I)c1C(=O)Nc1cc(-c2ccccc2C)nn1C C1(C(C)C)C(=O)N1.N1(CCNC(COCCSC)=O)CC2CC2C1.C(C)O C1(CNC(c2ncc[nH]c2=O)=O)CN(C(C2CCCC3(CC3)C2)=O)CC12CCC2 Cc1c(C(=O)NCC2CCC(C)CN2C(c2cc(F)c[nH]2)=O)cncc1N N1(C(C2CCCN(C)C2)=O)CCN2C3CCC(C3)C2C1.c12cn(nn1)CC(=O)S2 CC1CN(C(C2CCN(C)CC2)=O)CCN1C(c1ccn2c1CCC2)=O C1(C(=O)NCCC(O)CCO)(NC(c2cncc(Cl)c2)=O)CCOCC1 C1(NC(C(F)=C(C)C)=O)Cc2ccccc2C1NC(c1ccc(Cl)nc1O)=O N1(C(COCC=C)=O)CC(NC(=O)CC2CSC2)CC12CCCCC2 C1(C(=O)NC2CC2c2ccccc2)C2CCC(C2)N1C(c1cccnc1O)=O C1(CC=C)(NC(=O)C(C)(C2CCC2)NC(c2ocnc2C)=O)CCCC1 c1(OC)ccc(C(N2CCC(C)C(CNC(c3cnc(Cl)n3C)=O)C2)=O)cc1C C=CCC(CNC(C12CC(CO)(CN1C(c1cc[nH]c1)=O)C2)=O)CC(C)C C1(C(N(C2CCN(C(=O)CC3CSC3)CC2)CCC)=O)CN2CCN1CC2C c1(C(=O)OCC)cc(C)ccc1NC(=O)C(=O)N(C1CCS(=O)CC1)C c1(C(=O)NC(C(C)NC(=O)CC2CCCC2)CO)cc[n+]([O-])cc1 c1(C(N2CC=CC(C(=O)N(CC3CC3)CC3CC3)C2)=O)ccc(O)cc1F C(=O)(C(C(C)(C)C)NC(N)=O)NCC=CCNC(C(C1CC1)OC)=O.[nH]1cncn1 C1(C(N(CCC(=O)OC)C)=O)CC2(CC(NC(C3CC3(Cl)Cl)=O)C2)C1 c1(COC)ccc(C(c2nnnn2C2CC2)NCC(N)=O)cc1 Cc1n[nH]c2cc(-c3nc(C4CCC4)nn3Cc3ccccn3)ncc12 c1(CN(CC#C)C(=O)NCC2(C)CC(C(F)(F)F)C2)ccccn1 N1(C(CCC(=O)N(C)C)=O)CC(=O)NCCS1(=O)=O C1(CC(N2C(CN(C(=O)CC(C)(O)C3CC3)C)CCC2)=O)CCC(C)(C)CC1 CN1CCCCC(C(N2CCC(CCN(C)C)C2)=O)C1=O C=CC1(C(=O)NC2C3CCCOC23)CCN(C(c2cncc(C#N)c2)=O)CC1 c1(C(N2CC(C)(C)C(NC(C3(C)CCC(F)(F)C3)=O)C2)=O)c(N)cc(Cl)cc1F CC1CC(=O)CCC1C(N1CCC(NC(=O)C2=COCCO2)C(F)C1)=O c1(OC)ccc(OC(C)C(=O)NC2CCCCC2NC(c2nnsc2C)=O)cc1 c1(C(=O)NCC2C(CNC(CC#N)=O)C2)occc1F CC(C)CC(Cn1cc(C(O)CC(C)C)nn1)NC(C1(C(=O)O)CC(C)C1)=O N1(c2c(C(=O)OCC)cncc2)CCC(NC(c2ncc[nH]2)=O)C2(CCC2)C1 c1(C(=O)NC(CCNC(C(C#C)(C)C)=O)C)coc2c1CS(=O)(=O)C2 Cc1cc(C(=O)NCC(O)CNC(=O)CSc2ccncc2)c(C)nc1C Cc1cc(C)c(NC(=O)C(=O)NC2CCC2CNC(C2CCC(O)C2)=O)c(Cl)c1 C1(C(F)(F)F)(C(=O)NC(C)CCNC(=O)C(c2ccnn2C)C)CC=CCO1 C12(C(N3CC(O)(CNC(CS(C)(=O)=O)=O)C3)=O)CC=CC(C1)OC2 N1(C(C2CCN(OC)CC2)=O)CCC(C)C(NC(c2nc(C)no2)=O)C1C c1(C(=O)NCCN(C(c2cccc(F)c2Cl)=O)CC)c(N)cccc1F c1(OC)ncc(Cl)cc1C(N1CCC(NC(c2cc(C)c(Cl)s2)=O)C(CO)C1)=O N(C)(C1c2ccccc2CCC1N(C)C)C(=O)NCC(C)OCC C1(CNC(=O)CCC2CCOCC2)CCN(C(C2CCOC(=O)CC2)=O)C12CC2 c1(CNCC2CCC(CC)O2)ccc(N2CCCCC2)cc1 c1(OC)ncc(Cl)c(C)c1C(N1CCOCC(CNC(C2CCCN2C)=O)C1)=O C(=O)(N=c1cc2n([nH]1)CCCC2)C12N(C(C3(NC(N)=O)CC3)=O)CC(C1)C2 C1(C(=O)NCCc2nc[nH]n2)C=CCCN1C(=O)CC1CC(C2CC2)C1 C(=O)(C(C)(F)C(C)(C)F)N(CC(CNC(c1c(CC)n(C)nn1)=O)(C)C)C c1(C(=O)NC2(CC)CCCN(C(=O)C3=CCC3)C2)ccnc2c1CCO2 Nc1nccnc1C(=O)NCCC1(O)CN(C(=O)C(F)CC2CCCC2)C1 C1(CNC(C=CC=CCC)=O)CCN(C(c2snc(C)c2N)=O)C12CC2 C#Cc1ccc(C(N2CCC(O)(C(C)NC(=O)COCCN(C)C)C2)=O)nc1 C1(C(=O)NC2C(NC(=O)COCc3nccs3)C2)CN2CCCN1CC2 c1(OCC(=O)NCC(C)CN(C(=O)CC2CCC(=O)N2C)C)cc(F)ccc1F C(=O)(C#CC1CCOCC1)N(CCN(C(c1sccc1COC)=O)CC)CC C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(NC(=O)C=Cc2ccccc2Cl)CC(C)C1 N1(C(C2(C)CNC(=O)N2)=O)CC2(CCOCC2)CC1CNC(=O)CC1CCCO1 c1(CN2C(CC(N3CCC(CNC(C)=O)C3)=O)CCC2)cnccc1Cl c1(C(=O)NC(CNC(C2(CC=C)CC2)=O)C2CC2)ccc(F)c(COC(C)C)c1 Cc1cc(CC(=O)NCC2CN(C(=O)CCC3CC3(F)F)CCO2)cc(C)c1 C1(NC(CC(C(=O)O)NC)=O)CC2CCC(C1)N2C(c1c(OC)cccc1F)=O c1(C(=O)NC2(CCOC)CCN(C(=O)CCC3CC3(C)C)C2)ccc(Cl)cc1C Cc1oc(C)c(C(=O)NC2CCN(C(C3(C)CC4CC4C3)=O)C2)c1C c1(NCC2(OC)CC2)[nH]c(=NCCc2cnco2)nc2scnc12 CCC(CC)(CO)C(=O)NC1CCOC(CNC(=O)CC2(C)CCOCC2)C1 C1(C(c2ccccc2)NCC23CC(C#N)C(C2)C3)CC2(CCC(F)(F)CC2)CO1 c1(OC)cccc(C(=O)NC2CCC(CNC(C3CC3C(C)(F)F)=O)CC2)c1F c1(CC(=O)NCC2C(NC(Cn3c(C)cnc3)=O)CC2)n[nH]c2ccccc12 C1(CNC(CCC)=O)CCC(C)CN1C(c1ccc(SCC)nc1)=O N1(C(C(=O)NCCOCC)C2CC2(C)C)CC2CN(C)CC(C1)O2 N1(C(C2(C)C(CC)CCC2)=O)CC(CO)C2(C1)CN(C(=O)CSCC#N)C2 Cc1cc(CC(=O)NCC2CCCC(NC(c3ccncc3N)=O)C2)cc(C)c1 C1(NC(C(CC)n2cncn2)=O)CCC2CN(C(=O)Cc3csnn3)CCC2C1 n1(-c2ccc(OC)cc2)nc(C2CCC2)nc1C1=NOC2(CCC2)C1 C(=O)(C1=CCOC1)NCC1CC(NC(CN(CCOC)Cc2ccccc2)=O)C1 C1(N(C(=O)CC2CCCNC2=O)C)CN(C(c2cc(C3CC3)on2)=O)CC12CC2 c1(C(=O)NCCC(C)(C)NC(c2cc(O)cs2)=O)cc(Cl)ccn1 C(=O)(CCC(C)(C)C#N)N(CC(C)C(=O)N(C)CC1CCCC2CC12)C C1(NC(=O)CC2CCOC2)CC12CCN(C(=O)C1=CC3C=CC1C3)CC2 c1(C(=O)NCCCN(C(=O)C2=CCOCC2)C)ccc2ncccc2c1F C1(C(C)(C)C)CCC(C(=O)NCCCNC(=O)C(O)CC2CCCCC2)CC1 C(=O)(C(CN(C)C)C(C)C)NCC12N(C(c3cc(C)c(Cl)s3)=O)CC(C1)C2 C1(N(C)C)CN(C(C2CCCC(N)CC2)=O)CC12CC2 C1(n2c(C)cnc2)CCN(C(=O)C(n2ccc(C(F)(F)F)n2)C)CC1 C1(CC(=O)NCC2C3CN(C(=O)Cc4sccc4Cl)CC23)CCCOCC1 c1(N(CC(CN(C)OC(=O)C2CC2)O)C)ncc(C(F)(F)F)cc1Cl Cc1ccn2ncc(C(=O)N(C3CCC(NC(C4(CCF)CCC4)=O)C3)C)c2c1 C12CC(CCO1)NC2=O.c1(C(N(CCC(=O)OCC)C)=O)cc(CC)no1 C1(CCO)CCCN(N(Cc2cccs2)Cc2cccc([N+](=O)[O-])c2)C1 CCC(F)(F)C(=O)NC1CN(C(=O)Cc2cc(OC)no2)CC1O C(C(CC)(CC)C(=O)NCC(O)CC(F)(F)F)NC(c1oc(CC)c(C)c1)=O C(CN=c1[nH]c(=NCC2CCOC2)[nH]c2cccc(F)c12)C1CCC(C)(C)CO1 N1(C(c2ccc(C(C)=O)nn2)=O)CC2(CCN2C(c2cc(C(N)=O)cn2C)=O)C1 C1(CC#C)(C(N2CCN(CCNC(C3(C#N)CC3(C)C)=O)CC2)=O)CC=CCC1 c1(C(N(CC(N2CC(c3onc(C)n3)C2)=O)CC2CC2)=O)oc(C)cc1C C=CC(C)(O)C(=O)NC(C)CCNC(=O)CC1COCC1(C)C C1(CC(N2C(CCNC(c3c(CC)occ3)=O)CCC2)=O)CCC(C#N)C1 Cc1nc(C)c(CC(N2CCC(NC(C3CC(O)C3)=O)CC2)=O)c(O)n1 CCC(C)C(CO)NC(C1C=CCCN1C(=O)C(C)N(C)C(C)=O)=O C1(NC(=O)CC(F)(F)c2ccccc2)CCN(C(=O)C=C(Cl)Cl)CC1F C=CCCCCCCC(=O)NCC=C1CCN(C(c2ccc(Cl)nc2N)=O)CC1 c1(CCCCC(=O)N(C(CS(CC)(=O)=O)C)C)ccnc2ccccc12 C1(C(N)=O)CCCC(C(=O)NCC2(CNC(c3csnc3Cl)=O)CC2)C1 Cc1noc2cc(C(=O)N(CC(C)NC(=O)COc3ccc(F)cc3)C)ccc12 c1(C(N(C)CC2(O)CCN(C(Cn3c(C)ncc3)=O)C2)=O)cnc2n1CCCC2 C1(N(C(=O)CCN(C)CCO)CCC)CCN(C(C2(OC)CC(CF)C2)=O)CC1 Cc1ccc(-n2cc(CNC(C3(F)CCCCC3)C)c(C)n2)cc1 c1(C(N(CCNC(=O)C(C2CCCCC2)F)CC)=O)ccc2ccoc2c1 c1(CNC(C2N(C(C3(N(C)C)CCCC3)=O)CSC2)=O)ccncc1Cl CC(C)(CC(F)(F)F)C(=O)NCC1CC(F)CN1C(C1Cc2nccnc2C1)=O N1(C(C2C(CNC(C3C(C(C)C)CCO3)=O)CCC2)=O)CC2(COC(=O)N2C)C1 c1(COC(C(C2CCCOC2)OC)=O)ncccc1Cl C12(NC(C=C(CC)CC)=O)CCCCCC1N(C(c1cnc(F)c(Cl)c1)=O)CC2 C(=O)(CC(C)(C)C(F)F)NCC(C)(Cn1cccn1)NC(CC(C)C1CC1)=O N1(C(C(c2ccccc2F)C)=O)CCN(C(c2cc(Cl)ccn2)=O)CCC1C C1(F)(Nc2cn(-c3c(C)ccs3)nc2)CCCN(C(=O)CC2CCC(=O)N2C)C1 c1(C(N(CC(C)NC(C(C(CC)CC)C)=O)CC)=O)cccc2ncnc(O)c12 c1(CC)nn(C)c(NC(CNC(c2coc3ccc(C)cc23)=O)CC)c1[N+](=O)[O-] C(=O)(CCCCC(C)C)N1CC(C)(C(N(CC(CC)O)C)=O)C1 C1(OC)CCC2(C(=O)NC(C)C(C)(C)NC(c3cnc(O)c(C)c3)=O)CCC12 c1(C(N(CC(O)CN(C)C(C2(C)COCCO2)=O)C)=O)cnc(C2CC2)nc1O C1(CC)CN(C(C2COCCN2C)=O)CCN1C(c1csc(C(F)(F)F)c1)=O C1(C(N2C(CN(C(c3[nH]cc(CC)n3)=O)C)COCC2)=O)CCn2nncc2C1 c1(C(=O)NC2CC(CNC(C34CCCCC3C4)=O)C2)coc(=O)c2ccccc12 c1(C(=O)NC2(CC=C)CN(c3cc(Cl)c(O)nn3)C2)cc2ccccc2[nH]1 N1(C(c2c(C)nc[nH]2)=O)CCN(C(=O)C(C)C2(O)CCC2)CCC1C C(CCCC(=O)NCC(C)(Cn1cccn1)NC(=O)CC1CC(OC)C1)OC C1(NC(C2CCSCC2)=O)CC2CN(C(=O)CCCCCF)CC2C1 C(CC(CC)C(=O)NC1(CO)CCN(C(c2cnn3c2OCC3)=O)CC1)=CC C1(CC)CN(C(c2cnc(CO)nc2C)=O)CCN1C(=O)C=C(C)c1ccsc1 CC1(C)CCCC(C(=O)NCC(O)CC(=O)NCC2CCOCC2)C1 CCC(CC)CC(=O)NCC(C1CCCC1)NC(C1(COC)CCC(=O)N1)=O c1(C(N2CCN(C(CS(=O)(=O)NC)=O)CC2C(C)C)=O)cc2n(n1)C(C)CCC2 c1(C(=O)NC2CCC(NC(=O)C(c3ccccc3)O)C2)ccc2c(n1)CCOC2 Cc1ccc(C(=O)NCCCN(C(=O)CCCC#N)C2CC2)c(N)c1Cl c1(C(=O)NCc2ccc(CNC(C(C)O)=O)cc2F)cccc2c1OCCC2 c1(CN2C(C(=O)Nc3cc(C)cc(Cl)n3)CC(F)C2)cncc2ccccc12 S(=O)(=O)(c1ccc(C)c(C)c1)NCCC(=O)NC1C(CNC(C(C=C)(C)CC)=O)C1 c1(NC(C(C)C)=O)ccc(N2CCC(n3cc(C4CCN(C)C4)nn3)C2)cn1 c1(C(C(=O)NC2CC(NC(c3ccc(OC)o3)=O)C2)N(C)C)ccc(Br)cc1 C(c1cc[nH]c1)=CC(=O)NCC(CNC(=O)Cc1ccsc1)OC CC1CCN(C(c2ccnn2CCF)=O)CCN1C(=O)CNS(N)(=O)=O C(C(C)(C(=O)NCC(C)C(F)F)NC(=O)COc1cc(C)on1)SC c1(CC)ccc(C(C)=CC(=O)NC(C2CCCN2C(C2CC2F)=O)C)cc1 CC(C)C(C(=O)O)NCC(N1CCC2CC12NC(=O)OC(C)(C)C)=O C1(C(N(CC(C)(C)CNC(=O)C=CSC)CC)=O)CCc2ccccc2O1 C1(NC(CCCOCCC)=O)CC(C)CN(C(c2ccccc2OCCC)=O)C1 C(=O)(C(F)(F)CC(C)C)NC(CC=C)CNC(=O)Cc1c[nH]ccc1=O C1(C(N2C(C(=O)OC)CC2)=O)CCCCC1(C)NC(=O)Cc1cccnc1F CCC(CC)CCC(=O)NC1CN(C(=O)C(c2ccc(C)cc2)=O)CCC1C C1(NC(C(C)Cc2cnn(C)c2)=O)CC2(CCC(NC(=O)C=C(Cl)Cl)CC2)C1 N#Cc1ccc(CS(N2CCCN(C(c3c(F)ccnc3Cl)=O)CC2)(=O)=O)cc1 Cn1nnnc1C(C1CCOC1)NCCCCF S1(=O)(=O)CC(C2CC2)ON1C.c1(-c2nnc(C(=O)N(C)C)o2)ccccc1Cl c1(NC(C)=O)ccc(C(=O)NCC(C2C=CCN(C(C)(C)C)C2)=O)cc1F C1(CNC(Cc2nc(C)c(C)[nH]2)=O)CCN(C(C2C3C4CCC(C4)C23)=O)C12CC2 C1(NC(C2C(CC(C)(C)C)C2)=O)C2CC1CN(C(=O)OC(C)(C)C)C2 N1(C(C(N2CCOCC2)C)=O)C2CCC1C(CNC(=O)CCCC1CC1)C2 C1(O)(CNC(=O)CC(=O)NC2CC2)CCN(C(C2CC3(C2)CC(O)C3)=O)CC1 C(C(CNC(c1ccnc(C2CC2)n1)=O)S(C)(=O)=O)NC(C1C(CC)CCO1)=O Cc1nn(C)c(=O)c(C(N2C3CCC(C3)C2CNC(c2cc(F)c[nH]2)=O)=O)c1C C1(C(N(C)Cc2ccc(C)s2)=O)CC(F)(F)CN1C(=O)CCOC1CCCC1 c1(C(=O)NC(C)CNC(c2cc3sccc3cn2)=O)cc2n(n1)CCCC2O Cc1ccccc1C(=O)NC1(CF)CCN(C(=O)CCCn2cncn2)C1 N1(C(CC(=O)NC)=O)CCCOC(CNC(c2cnoc2-c2ccoc2)=O)C1 C12(C(=O)NCc3ccc(C)nc3)CCN(C(c3c[nH]cc3C)=O)CC1C2 N1(C(C(CCOC)C)=O)CCC2(C1)CN(C(c1ccnc(F)c1F)=O)CC(C)O2 N1(C(CCCOC(C)C)=O)CCCC(C2CCCN2C(C2CCCC(=O)N2)=O)C1 C1(NC(C2C(C)(CC)C2)=O)CC2CN(C(=O)Cc3ccc(Cl)nc3)CC12 N1(C(C(CC)C)=O)CCC(NC(c2cnc(C(C)(C)C)[nH]2)=O)C1(C)C C(=O)(C1=NNC(=O)CC1)NC(C1CCCN1C(=O)CCCCCC#N)C C1(CCC)C2CN(C(c3ccc(NC)cc3)=O)CC12.C12(CCOCC1)C(=O)N2 c1(C(=O)NCC(CCOC)NC(c2ncn(CC)n2)=O)cc(C(C)C)ccc1F c1(CC)cc(C(N2CCC2CNC(c2ncccc2CSC)=O)=O)sc1C Cc1csc(=NCC(=O)N2CC=CC2CNC(C2CCc3nccn3CC2)=O)[nH]1 CCC(C(=O)NC1CC(C)(NC(=O)Cc2csc(COC)n2)C1)C(C)O N1(C(c2n[nH]c(C)c2F)=O)CC2(CCN(C(=O)CCc3ccccc3Cl)C2)C1 Cc1ccc2c(=O)c(C(=O)NC3CCCC3NC(c3ccc(F)s3)=O)c[nH]c2c1 N1(CCCC(=O)NCCCC2CCN(C(CC=C=C)=O)CC2)C(=O)CN(C)C1=O c1(C(=O)OC(C)(C)C)cccc(NC(N2CC(C3C(C(=O)O)C3(F)F)C2)=O)c1F c1(C(N2CC3(N(C(c4cc(C)cc(C)c4)=O)CC3)C2)=O)cc(C)c2[nH]nnc2c1 c1(C(=O)NC(=O)CCC2(C(N3C(C4C(C)C4)CC3)=O)CCCC2)ccc(N)cn1 C1(C(C)C)CN(C(c2c[nH]ccc2=N)=O)CCN1C(C1OC2CCC1CC2)=O CCCC(C(=O)N1CC(N(CC)CC)C1)NC(=O)C(C)c1ccco1 C(=O)(CC(C)(C)C(=O)N1CC2(CCNC(C3CCS(=O)(=O)C3)=O)CCC1C2)OC c1(C(=O)NCC2CCC(NC(c3cc(C)[nH]n3)=O)C2)cc2c(s1)CCSC2 N1(C(COC(C)(C)C)=O)CCC(NC(c2cc(Cl)c(Cl)[nH]2)=O)C12CCCC2 C(=O)(CCP(C)(C)=O)N(CC(C)CNC(c1cc(-c2cccs2)on1)=O)C C1(C)(NC(CC2(N(C(CNC(CC)=O)=O)C)CC2)=O)CCC(C)C1 Cc1cc(C(=O)NC(C(=O)NC2CC3CC3C2)C2(C)CC2)cnc1C c1(N(C)Cc2cc(C)no2)ccc(S(=O)(=O)NC2CCC(C)(C)CC2)cc1F C1(N(C2(c3cc[nH]n3)CCC2)C(=O)CN2CC=CC2)CCN(CCC2CCC2)C1 Cc1ccc(CNC(=O)C=C2CCN(C(c3cc(Cl)cc(Cl)n3)=O)CC2)cc1C Cc1nocc1C(=O)NCC(C1CCOC1)NC(c1cnoc1C)=O c1(-c2onc(CN(CC(C)NC(c3c(CC)occ3)=O)C)n2)ccc(Cl)cc1 c1(C(=O)NC2C(NC(C(C)(C)SC)=O)CC2)cc2c(s1)CCCNC2=O c1(C(=O)NC(C)CCNC(=O)C(O)CCn2cncn2)c(Cl)cccc1Cl c1(N(CC(c2ccccc2)CC)C(=O)NC(C2CCOC2)C)ccccc1 c1(C(C)C)n[nH]c(=NCC2CCC(NC(c3cccc(NC(N)=O)c3)=O)C2)o1 C1(C(=O)NC2CN(C(C(C)SC(F)(F)F)=O)CC(F)C2)Cc2ccccc2C1 C(=O)(C(CC(F)F)NC(=O)C(C)=CC1CC1)N1CCN(CC(=O)NC)CC1 c1(C(=O)NCC2C(NC(c3ccn(CC)c3C)=O)CC2)cc2c(s1)CCCC2 Cc1ncc(NC(=O)C(C2CCCCC2)NC(c2cccnn2)=O)c(C)n1 c1(NCC2OCC(CNC(C(=Cc3cnc[nH]3)C)=O)C2)ncc(C#N)cc1Cl c1(CN(C)CC)cccc(C#N)c1.C1(=O)CCC(=O)N2CCOC(C2)N1 N1(C(C(=O)NCCC2CC2)=O)C2CCC1CC(n1cc(C3(O)COC3)nn1)C2 C1(CC(=O)NCc2c(NC(C3(c4ncc(C)o4)CC3)=O)[nH]cc2)NC(=O)NC1=O Cc1ncnc(O)c1C(=O)NC1CC(C)(CNC(C23CCCC2CCC3)=O)C1 C1(F)(C(=O)NCC2N(C)CCCC2)CCCN(C(=O)C(C2CCOCC2)O)C1 C1(NC(C2C3CCC2(c2cccnc2)C3)=O)CC2(CNC2)C1 N1(C(COC(C)=O)=O)CCOC2(CCC(NC(c3cnc(C(C)C)[nH]3)=O)CC2)C1 C1(CNC(C(OCC)OCC)=O)COCCN1C(=O)CCN1CCC1 CC(O)CCCCCC(=O)NC(C)(C)CCNC(c1ccc2nc(S)oc2c1)=O N1(C(c2scc(C)c2C)=O)CC2CCC1CC2NC(C1(c2ccccc2)CC1)=O C(=O)(C(CNC(C1CC(O)(CC)C1)=O)N(C)C)N(CCC(=O)OCC)C C1(C(=O)N(C)CC2(C)CCCC2)(SC)CN(C(c2cc(C)co2)=O)C1 C(C(CNC(=O)C(=Cc1cnn(C)c1)C)S(C)(=O)=O)NC(C(CCOC)OC)=O c1(CC)cc(C(N2CCN(C(=O)CC(C)COC)CC2C2CCC2)=O)cc(F)c1 c1(-c2cc(C(=O)NCC3CC3CNC(C3CC4(CC4)C3)=O)on2)ccccc1F C(=O)(C(Cc1cn[nH]c1)NC(=O)C(C)O)NC1(CC=C)CCC1 N1(C(c2ccc(C(C)C)s2)=O)CCC2(CC(NC(C3OC4CCC3CC4)=O)C2)C1 c1(C(=O)NCCCCC(C)NC(c2cscc2Cl)=O)cc(N)cc(N)c1 C1(CN(C(Cc2cn(CC)nc2)=O)C)CCCN(C(c2oc(C)nc2C)=O)C1 C(=O)(CC(O)C(C)C)NC1C(OC)CN(C(c2c(CO)n[nH]c2C)=O)C1 C(=O)(C1=C(C)CCC1)N1CC(CCNC(C2(c3c(OC)cccc3)CC2)=O)C1 c1(C(N(C2CN(C(C3C(C)CCC3)=O)C2)C)=O)cnc2c(F)c(F)ccc2c1 C1=C(CN=C(NCC2CCOC2)NC2CC(n3cncn3)C2)CCOC1 CC(CCC(=O)N(C1CCN(C(C2CN(CP(C)(C)=O)C2)=O)C1)C)S(C)(=O)=O c1(N2CCC=C(C(=O)Nc3cc(O)nc(O)n3)C2)ncnc2sc(Br)cc12 C1(C(N(C)CC2N(C(c3cnc(C)[nH]3)=O)CCC2)=O)CCC(NC(N)=O)CC1 c1(C(=O)NC2C(CNC(c3cc(C)on3)=O)CCCC2)n[nH]c2c1NCCC2 Cc1cc(Cl)ccc1C(=O)NC1CCN(C(=O)CC(C)NC(N)=O)C1C Cc1c(C(=O)NC2CCN(C(=O)C(C)Sc3ncccn3)C2)cccc1[N+](=O)[O-] C(=O)(CCCCCC)NC1CC(CNC(CSCCCC)=O)OCC1 N1(c2snc(CC)n2)CC2(CN(C(=O)C=CCN(C)C)CC2CO)C1 N1(C(CC(CC)C)=O)CCCCC2C1CCCN2C(c1cnc(O)n1CC)=O C(=O)(C(O)CCn1cncn1)NCC(C(=O)N1C(C(=O)OC)CC1)OC N1(C(=O)CC(C(F)F)n2ccnc2)CC2CCN(C(=O)CCN3CCCC3)C2C1 c1(OC)cc(CN2CCC(O)C2C(N2CC(F)C(F)C2)=O)ccc1Cl C1(CNC(C(C)=C2CC2)=O)CN(C(=O)Cn2ncccc2=O)CCO1 Cc1sc(C(=O)NC(C(C)NC(c2cc(O)ncn2)=O)C(C)C)cc1[N+](=O)[O-] c1(C(N(CC(C)C#N)CC)=O)ccc(CNC(C2CN(C)CCO2)=O)cc1 CCCCCCCCC(C)C(=O)N1CCCC(CN(C(=O)C2=CCSC2)C)C1 C(C(N=[N+]=[N-])C(=O)NC1CCOCC1NC(=O)C=CCOCCOC)OCC C(=O)(C#CC(=O)N(C)C)NC.c1(C2CN2)ccc(OC(=O)CC2CCOC2)cc1 C=C=CC(C)C(=O)N1CCN(C(c2ncoc2-c2ccc(C)cc2)=O)CC1 C(C)(CCCCN=c1nc2[nH][nH]cc-2c(O)n1)NC(c1cnc(C)o1)=O CN1CCc2nc(O)c(C(=O)NC34CCC(CN(C(=O)C5CC5)C3)C4)cc2C1 C1(CC)CC(C)N(C(c2csc(-c3cnn(C)c3)n2)=O)C1 CCC(C)(CNC(=O)Cc1cnn(C)c1)C(=O)NCC(C)(C)CN(C)C c1(NCC(c2ccccc2)(C)C)nc2ccccc2n1CC(=O)N(C)SC C1(CNC(CC2CCN(C)CC2)=O)CCCN(C(=O)CC2COCCO2)CC1 C1(NC(C2C(c3ccn(C)n3)C2)=O)CCCCCN(C(=O)Cn2nccn2)C1 c1(C(N(C2CCC(NC(C(C#C)(C)C)=O)CC2)C)=O)cc(C)c(N)c(C)c1 c1(C(=O)NC(C(C)NC(c2c[nH]c(C(N)=O)c2)=O)CO)cnn2ccncc12 C(CCCCC(=O)N(C)CC1COCCN1C(=O)CCc1cnoc1)=CC N1(C(c2cc(Br)cc(Cl)n2)=O)CC(CO)C2(CCC2)C1 Cc1ccc(F)c(CC(=O)NC2CC3CN(C(=O)CCc4nc(C)no4)CC23)c1 CC1CCCCN1CCC(N1CCN(C(=O)C=CC2CCCO2)CC1)=O N1(C(C2CCN(CC(C)(C)C(F)(F)F)CC2)=O)CCC12CCCSC2 C1(CC)CCN(C(=O)OC)C1C(=O)NCCOCCCSc1ccns1 Cc1cc(C(=O)NC(CCN(C(=O)Cc2ccn(C(C)C)n2)C)C(C)C)cnn1 c1(C(=O)NCC(C)N(C(C2CC23CCCC3)=O)CC)ccc(F)c2ccccc12 c1(C(C)C(=O)NCC(C)(C2CC2)NC(C2CN(C)C2)=O)ccc(F)cc1 c1(C(=O)NC2CCCN(C(C(C)=C3CCCC3)=O)C2)cc(C)nc(C)c1O C1(O)(CCNC(c2cc(COC)on2)=O)CCN(C(c2[nH]cnc2C)=O)C1 C1(NC(c2ccc(CC(C)C)nc2)=O)C2CCC1N(C(C1CCC(=O)N1C)=O)C2 c1(C(c2nnnn2C)NCc2c(CC)nn(C)c2)ccc([N+](=O)[O-])cc1F c1(C(=O)NCC(CC)NC(=O)C(=Cc2ccc(F)cc2)C)ccn2nccc2n1 N1(C(C(CC#C)C)=O)CCCN(C(=O)C(c2c(F)cccc2F)(C)C)CC1CO C(=O)(CC(CNC(=O)COC1CCC1)C1CCC1)NCC(CC)CO C1(C)(C(=O)NC(C)Cn2cnnc2)CN(C(=O)CC2COCC2O)C1 c1(C(=O)NC2CCC(C)N(C(=O)C(=O)C(C)(C)C)C2)c[nH]c2nccc-2c1 c1(CCC(=O)NC2C(C)CN(C(C3(O)CCOC3)=O)C2)nc2cccnc2[nH]1 CC(C(=O)NCC1(F)CC(NC(c2ccnc(S)c2)=O)C1)C(C)(F)F N1(C(C(C)OCC2CC2)=O)CCN(C(=O)CN(C)C(C2(C)CC2(F)F)=O)CC1 Cc1cccc2c1CC(C(N1CCCC1CNC(C1C3CCCCC13)=O)=O)O2 c1(C(=O)NCCN(CCC)C(C2CC2(C)CN(C)C)=O)ccc(F)c(COC)c1 c1(OC)cc(Cl)c(Cl)cc1CN1CCCC1CC(=O)Nc1cnc(OC(F)F)nc1 c1(C(=O)NC(C(=O)NC(C#C)CC(C)C)c2ccoc2)cc(O)ccc1F c1(C(=O)NC(CC)(CNC(=O)C(C)OCC(C)C)CC)cc(Cl)cc(Cl)c1N c1(C(=O)NC2C(NC(C(C(C)C)OC)=O)CCC2)nc2ccc(C)cn2c1N N1(C(C2C(OC)(OC)CC2)=O)CCN(C(=O)Cc2cc(C3CC3)no2)CC1CF Cc1cc(CC(N2CC(O)(c3cn(CC4C(C)C4(F)F)nn3)C2)=O)nc(O)c1 c1(C(=O)NCCC(CNC(C2(CSC)CCC2)=O)O)cc(F)c(F)cc1F C1(C(=O)NC(CCNC(C(C)C2CCOC2)=O)C)(C2CC2)CCCO1 C1(C(=O)NC(CC)CNC(C2(C)CC2C(F)(F)F)=O)CCCS(=O)(=O)C1 c1(C(N2CCC(CN(C(COC(CC)C)=O)C)C2)=O)ccc(Cl)cc1COC CC(C)CC(C)(C)C(=O)NC1CCCC1NC(=O)C(C)CCc1ccccc1F C1(N(C(C2C(=C)C2)=O)C)CCCN(C(c2ncoc2CC(=O)N)=O)C1.C(C)(C)(C)O Cc1ccc2cc(-c3cccc(N4CCN(Cc5ncn(C)n5)CC4)c3)[nH]c2c1 c1(CC(=O)NCCC2(OC)CN(C(C3(CCCC)CC3)=O)C2)cc(C)n(C)n1 C1(C(C)(C)C)CN(C(c2ccc(O)nc2Cl)=O)CCN1C(C1CCNC1=O)=O C12(C(NOC(C)(C)C)=O)CCC(CC1NC(C1CCCC3(CC3)C1)=O)C2 c1(NCC(C)CNC(C2CC=CC2)=O)ncnc2sc3c(c12)CCC(C)C3 c1(C(C)NC(C(CC)n2cc(CCOC)nn2)=O)ccc(C)c(Cl)c1 CCC(CC(=O)NC1CN(C(=O)CN(C)CC)CC12CCCC2)C(C)(C)C c1(C(=O)NCC2(OC)CN(C(C=CC)=O)C2)cn2ccc(F)c(C)c2n1 Cc1cc(NC(c2cnn(CCNC(=O)CC3CC=CC3)c2)=O)cc(C)c1F C(=O)(CCCCC(C)=O)N1CCC(NC(Cc2ccc(C#C)cc2)=O)(CC)CC1 Cc1cccnc1C(=O)NC(C)C(C(C)C)NC(c1ncccc1N)=O C12(C(=O)NC3C(C)CN(C(=O)COC4CCOC4)C3)CC3CC(C1)CC(C)(C3)C2 C(=O)(C1CCCc2c[nH]nc21)NC(CCNC(c1nc(C)sc1)=O)C(C)C N1(C(c2scc(C)c2Br)=O)CC2CCN(C(=O)C3=CCCC3)CC2C1 C1(NC(c2cccnc2CO)=O)CCCC(CO)C1.C12(CCCO1)C(=O)NC2 n1(CC(=O)OC)ccc2cc(Br)ccc12.C(C)(C(F)(F)F)OCCN1C(=O)C1 C1(CNC(C2C(CC)C2)=O)CC2(CC2)CN1C(c1ccc(C#N)[nH]1)=O c1(C(=O)NC2(CC(N3CC4C(C(C)(C)O)C4C3)=O)CC2)ccn2nccc2c1 CC#CCCCCNC(=O)C(=O)NCc1ccc(Cn2cc(C)cn2)cc1 CN1CCC(O)(CC(=O)N(CCN(C(=O)C(F)C(C)(C)O)C)C(C)C)CC1 Cc1cc(N)c(C(N2CC(C)(NC(C3CN(C(N)=O)C3)=O)C2)=O)nc1C c1(C(=O)NCC2=CCN(C(C(C(CC)O)(F)F)=O)CC2)ccc2ccn(C)c2c1 N#Cc1ccsc1C(N1CCC2CC12C(=O)NCCCC1CC1)=O c1(CC(=O)NCCC2(CNC(C(C)(C)OCC)=O)CC2)c(C)cccc1C C1(NC(COCC)=O)CN(C(c2cc(=O)c(OC)c[nH]2)=O)CC2(CCC2)C1 C1(C(=O)NCCC2CCCN2C)(CC)CCN(C(c2cnn(CCF)c2)=O)C1 Cc1nn(C)c2c1CC(NC(=O)NCCCC(C)(C)C1CC1)CN2 c1(C(=O)NC2CCCCC2CO)ccccc1-c1nnnn1C1CC1 CN(C)NC(=O)CCC(=O)NC1CCCCCC1NC(c1cnc(Cl)c(N)c1)=O C(CCN(C)C)(C(=O)NCCCCS(C)=O)NC(C(CC=C)OC)=O C=C(C)CCC(C)NC(C1C=CCN(C(=O)CCCN(C)C)C1)=O n1(CC(=O)NCC(C)(CC(C)C)NC(C(CCOC)C)=O)c(C)cc(C)nc1=O c1(CNC(C(C2CC2)SCC)=O)c(C(=O)NCC2CCOC2C(C)C)cnn1C CC1CCCC(OCC(=O)NC(CNC(c2cc(C(C)(C)C)on2)=O)C2CC2)C1 C1(NC(C(N)=O)=O)COC2(C1)CN(C(C1(C(F)(F)F)CC=CCO1)=O)C2 c1(CC(=O)NCC(C)CNC(=O)C(C)CF)cc2ccccc2o1 N1(c2cc(C)nc(N3CCOC(c4cc[nH]n4)C3)n2)CC2CCC(C1)N2C CC1CC(NC(C2CCCC23CC3)=O)CCN1C(c1cnn2ccsc12)=O C=CCCC(F)(F)C(=O)N1CC2CC(C(=O)NCCNC(N)=O)CC2C1 N1(C(C2(C(C)(C)O)CCC2)=O)CC2CC1C2NC(=O)CN1CCCCC1 C1(CNC(CN(c2cnccn2)C)=O)CN(C(=O)CC2CCC2)CCN1C c1(OC)c(C(=O)NC2CCC2NC(=O)C(N2CCCCCC2)C)c(C)nn1C c1(C(N2C(C(=O)NC(CC)C(=O)NC)CC=CC2)=O)cnc(O)cc1C c1(CN2C(C)(C(N(C(c3ccc(OC)cc3)C)C)=O)CC2)cc(Br)cc(Cl)c1F N1(Cc2c(SC)cccc2)CC2CN(C(=O)C(C)S)CC12 N1(C(C(C)S(C)(=O)=O)=O)CCC(NC(=O)C(F)(F)CC2CC2)C(CO)CC1 N1(C(c2cccc(NC)n2)=O)CC2CC(NC(=O)C(N3C(=O)CCC3=O)C)C1C2 c1(NC)scnc1C(=O)N(C(C)C(=O)NCC1CCC(=O)N1)C C12CCC(O)CN1OC2=O.c1(C(=O)NCCNC(N)=O)ccc(O)nn1 N1(C(=O)NC(c2nc(COCC)on2)C)CC2CCCS(=O)(=O)C2(C(F)(F)F)C1 N1(C(COCC=C)=O)CC(NC(=O)C=Cc2nonc2C)CC(O)C1 C(=O)(CCS(=O)(=O)c1ccccc1)NC(C)CCCNC(=O)C1=CCCS1 c1(C(=O)NC(C(C)C)(C)CNC(C2CCCOCC2)=O)ccc2c(c1)OCC2 N1(C(C2(C)CCC(C)C2)=O)CCC(C(=O)N(C)CC2(C#N)CC2)C(C)C1 c1(C(N2CCC(C)C(N(C(=O)Cc3ccco3)C)C2)=O)cc2cccnc2cn1 N1(C(Cc2c(C)noc2C)=O)CCOC2CN(C(C3CCCC(F)(F)C3)=O)CC12 c1(CSC)ccc(C(=O)NC2CC(CO)N(C(=O)C=CC3CCOC3)C2)cc1 C1(C)(C(N(CCCCCNC(c2cc(CC)sn2)=O)C)=O)CC(OC)CN1C c1(N2CC3CN(C(C4Cc5nccnc5C4)=O)CC3C2)ccc(Br)cc1[N+](=O)[O-] N1(C(C(CC2CCOCC2)NC(CC2CC(=C)C2)=O)=O)CC2(CO)CCC1CC2 N1(CC)CC(C(=O)NC2(C)CC(NC(=O)Cc3ccc(F)cn3)C2)CC1=O N1(C(C)C2CC2)CC(C(=O)NCCNC(=O)CC2CCCC2)CC1=O CN1CCC(ONC(=O)C(F)C2CCCN(C(c3cc(C#N)c[nH]3)=O)C2)CC1 c1(OCC)cnc(=NCC2CCC(NC(=O)CNc3ccc(C)cc3)CC2)[nH]c1 C1(CNC(CSCCC)=O)(CO)CCN(C(=O)CCCCc2ccccc2)CC1 c1(COCC(=O)NCC(C)CNC(=O)CNC(N)=O)cccnc1 C(CO)(CCCCNC(c1cc(C2CC2)cs1)=O)NC(c1c(SC)cn(C)n1)=O C1(NC(CC2CC(OCC)C2)=O)COCC1CNC(c1ccoc1C)=O N1(CC)CCC(C)C(CNC(C2(n3cc(CN(C)C)nn3)CCC2)=O)C1 c1(C(N(CCC(C)NC(=O)C(C)(C)C(F)(F)F)C)=O)cn(C)c(=O)nc1O C1(NC(=O)CC2CC(F)(F)C2)COCCN(C(=O)CCCCc2cnn[nH]2)C1 C1(CNC(C=CC=CC)=O)C(OC)C(OC)CN1C(c1csc(O)n1)=O C(C(N=c1[nH]c(N2CCOCC2)nc(=NCCCCC#N)[nH]1)C(C)C)OC Cc1cc(C(=O)N(C)CCOCCNC(=O)Cc2nccs2)[nH]c1C c1(CC)cncc(C(N2CCC(NC(C34CC(C)(CO3)C4)=O)CC2)=O)c1 CCCCC(O)CC(=O)NCC(C)C(F)C(=O)NCc1cnc(C)s1 N1(C(c2cnc(C(=O)OCC)s2)=O)CCC2CN(C(=O)C(F)(F)C(C)O)CCC12 c1(C(=O)NC2(C3CN(C(C(CC(C)(C)C)O)=O)C3)CC2)cc(O)c2ccoc2c1 N1(C(=O)CC2CCSC2)CCC2(CC2C(N2CCC(O)C2)=O)C1 CCC(CC)C(C(=O)N1CC(C)CCC1C(N1CC(S(C)(=N)=O)C1)=O)OC N1(C(CC2CC(=C)C2)=O)CC(NC(c2cnc(C3CC3)o2)=O)C2CC12 c1(COC(CSC)=O)ccc(C)c(C)c1.C12CN(C3CC13)C2=O.CC(=O)NCCOC N1(C(C2C(O)CCN2C(C2COCCO2)=O)=O)CCN2C(=O)CCC2C1 N1(C(C(C(C)C)NS(N)(=O)=O)=O)CCC(C)N(C(c2cn(C(C)C)nn2)=O)CC1 N1(C(C2N(C(C(CCCC)F)=O)CCC2)=O)CCOCC(C2CC2)C1 C#CC1(O)CC(C(=O)NCC2(C)CCN(C(c3ccnc(OCC)c3)=O)C2)C1 c1(C(N2CCC(CNC(CC3(O)CCCN(C)C3)=O)C2)=O)cnc2c(c1)CCC2 C(=O)(C(F)C(F)(F)F)NC1(CCCNC(C2N(C(CC)=O)CCCC2)=O)CC1 c1(C(C)NC2CC(N3CCN(C(C)C)CC3)C(=O)N2)ccc(F)cc1Cl c1(-n2cc(CCNC(C3CC(O)C(F)C3)=O)nn2)cccc(Cl)c1 c1(NC2CCC3CN(C(C(CC)C)=O)CC32)nc(C)cc(C)c1C#N C(=O)(CCCCC(=O)NCC1CN(C(c2n[nH]c3c2CC2CC32)=O)CCO1)NC C1(C(N(C(CC#C)C)C)=O)CCC2CCC1N2C(c1ccccc1O)=O C1(CNC(c2cc(C)c(C)[nH]2)=O)CCN(C(c2ccsn2)=O)C(C)C1 c1(C(N2CC(C(=O)NC3(CC(=O)OCC)CCCC3)C2)=O)cccc(CO)c1 C1(NC(c2c(C)cc(C)o2)=O)CC2(NC(=O)CCC3CC3(C)C)COC1C2 C1(NC(c2ccc(N)cn2)=O)CN2CCC1CC2 C=CCC(CC)C(=O)NCC(CNC(=O)C(O)Cc1ccc(OC)cc1)OC c1(C(=O)NC(C)C(C)(C)NC(=O)CC2CCCN2C)cc([N+](=O)[O-])nn1C c1(C(=O)NC2(COC)CCN(C(c3conc3C)=O)C2)cc2cccn2c(O)n1 CC(CC(F)F)C(=O)N1CC=CC1CNC(=O)Cn1cnc([N+](=O)[O-])n1 N1(C(=O)Cn2cnc(Br)c2)CCCN(C(C2CCCS2)=O)CC1 C1(C(N2CC(CC=C)(NC(=O)COC(C)CC)C2)=O)CCC2(C1)CC2(F)F c1(C(=O)NC2CC(F)(CNC(C(CC)OCC)=O)C2)c(N)sc2c1CCSC2 c1(C(=O)NCC2(C)CC(NC(C3(COC)CC=CC3)=O)C2)ccnc(F)c1OC c1(C(N(C)CC2(O)CN(C(CCC#C)=O)C2)=O)cnn(CCC)c1Cl N1(C(c2cncs2)=O)CCCC2(CCN(C(C3CCC3(F)F)=O)C2)C1 N#Cc1cn(CC(=O)NCC2CCCN2C(c2ccns2)=O)c(=O)nc1O CC(C)(C)C#CC(=O)N1CCCCC(CNC(=O)CCC2CCCC(=O)N2)C1 N1(C(C23CC(OC)C2C3)=O)CC=C(CCNC(c2ccnc3c2CCO3)=O)CC1 C#Cc1cc(C(=O)NCCOCCNC(c2cnc(CO)nc2C)=O)ccc1C C(C(C)(C)C(=O)NC1CC12CC(NC(=O)CCOC1CC1)C2)N(C)C Cc1cn2ccnc(C(=O)NCC(C)CNC(=O)C(N3CCCCCC3)C)c2n1 N1(C(CC=C)=O)CCCC(NC(c2n[nH]c(O)n2)=O)C1C C(=O)(CCCCN=[N+]=[N-])NC1CN(C(C(C(C)C)SC)=O)CC1n1ccnn1 CCC(C)CCCCC(=O)NCCC1(C(N2CCC(C)C2(C)C)=O)CC1 N1(C(C2C(C)C2C)=O)CC(CNC(C2(C3CCCO3)CCCC2)=O)C(O)C1 C(C)(N=c1nc(N2CCSC2)c2sccc2[nH]1)c1c(OCC)cccc1 N1(C(c2cn(C)c(=O)cc2)=O)CC2CN(C(C3CCC(C)(C)CO3)=O)CC2(C)C1 N1(C(c2nn(C)c(CO)c2)=O)CCN(C(c2cnns2)=O)C2(CCC2)C1 c1(C(=O)NC2(CC)CCN(C(=O)CNC=O)CC2)cc2cccnn2n1 N1(C(Cn2ccc(C)n2)=O)CC(C(=O)NOCC(C)(C)O)C(C)C1 C1(CCNC(C(CC)n2ccnc2)=O)CCN(C(c2csc(C#N)c2)=O)CC1 C1(=CCNC(=O)C=Cc2ccco2)CCN(C(C2OCCC2C(F)(F)F)=O)CC1 CCC(O)C(C)C(=O)N1CCCC(CN(C(=O)CC(C)(C)O)C)C1 N1(C(C2CC(F)CN2C(c2ccc(O)c(Br)c2)=O)=O)CCc2ccc(Cl)cc2C1 C#CCCC(O)CCNC(=O)CCCCN(C(=O)COC1CCOC1)C N(S(=O)(=O)N1CCCc2ccccc21)CC(C)(O)c1ccsc1 N1(C(CCC)=O)CC2(CC(NC(=O)CC3CSC3)C2)C1 c1(N2CCc3c(cn(C)n3)C2)nccc(=NC2COc3cc(F)cc(F)c32)[nH]1 c1(C(N2C(C)CC(CNC(C3(C4CC4)CCC3)=O)C2)=O)cn(C)c(=O)nc1O C(C)(CO)(C(=O)NC1CC1CCOC)NC(C(CC)NC(C)=O)=O Cc1cc(C(=O)NC2CN(C(=O)C(Cl)(Cl)Cl)CC2O)cc(O)c1 C1(C(=O)NCCCOCCN(C)C(C2(C)C=CCC2)=O)CCc2ccccc2O1 O=C(C1=CCOC1)NC1(CF)CCN(C(c2ccc(C(N)=O)nc2)=O)C1 C(C(=O)NCCOCCCN(C(=O)C(c1ccn(C)n1)C)C)(C(C)C)OC C1(C(N2CCC(NC(C3C(C)=CCS3)=O)C(O)C2)=O)COC2COCC2O1 N1(C(C2(CSC)CC2)=O)CC(NC(c2ccc(-n3cncn3)nc2)=O)C(C)(C)C1 C12(NC(Cn3c(C)c(Cl)cn3)=O)CCN(C(=O)C=C(Cl)Cl)CCC1C2 C(=O)(C(CC)C(F)(F)F)N1CC(OC2CCN(C(CCC(=C)Cl)=O)CC2)C1 CC1CN(C(C2(C#N)CC2)=O)CC1NC(=O)C(C1CCCCCC1)N(C)C c1(C(C(=O)NCCOCCNC(c2cnnc(O)c2)=O)(F)F)ccc(F)c(F)c1 C1(OC)CC2CCCC2C1.C12(c3cc(C)n(C(C)C)n3)CN(CO1)C2CC1CCC1 CC(C)CC(C)CC(=O)N1CCCC(C(N2CC(C)(CCO)C2)=O)C1 C(=O)(C(C)C(C)NC(C1CC(=O)C1)=O)NC(C(=O)OC)(C)C C1(C(N(CCC)C(C)C)=O)C2CC(O)C(C2)N1C(C1CC1(C)C(F)F)=O C1(CNC(CC(C=C)C)=O)CN(C(c2nn(C)nc2Br)=O)CCCO1 C1(CCOC)CN(C(=O)CCn2ccnc2)CCN1C(=O)CCF C(=O)(C(CC#CC)NC(=O)C=C(C)C1CC1)NCC(CC#C)(C)C c1(C(=O)NC(C(=O)NCC2CC2)C2CCCC2)cccnc1 c1(C2C(C(N3CC(NC(=O)C=Cc4cscn4)C3)=O)C2)c(F)cccc1F Cc1c(C(=O)NCC2CC2NC(c2cc(F)cc(Cl)c2N)=O)sc2ccccc12 c1(CCC)ncoc1C(=O)NC(C)CC(C)NC(=O)C(C)C c1(C(N2CC(O)(CN(C(=O)C3=COCCO3)C)C2)=O)ccc2c(c1)COC2 c1(C(=O)NC2(CCNC(C3CC(C)CC(C)C3)=O)CC2)cc(C#N)ccc1N c1(C(C)=O)cc(C(=O)NCCNC(=O)C(F)n2ccnc2)cnc1C c1(C(N(C(CNC(c2ccc(C)c(Cl)c2)=O)C)C)=O)cnc2c(c1)nnn2C c1(C(=O)NCCCN(C)C(C23CCC(CC2)O3)=O)c[nH]c2cc(F)c(F)cc12 N1(C(Cc2cc(C)[nH]n2)=O)CC2CC(NC(=O)C=Cc3cncnc3O)CC2C1 C1(CCC)CCCC1(c1nnnn1CCC1CC1)NCC=CCOC C1(CNC(Cc2ccc(C)s2)=O)CCC(NC(C23CC(C2)C(C)O3)=O)CC1 O=C(C(F)C1=CCCCC1)NCCC1=CCN(C(=O)CSCC(F)F)CC1 C1(CNC(c2cccc(O)c2)=O)CN(C(=O)CC2CC2(Cl)Cl)CCC1(F)F c1(CN2CC3N(C(c4c(C)cc(F)cc4C)=O)C(C3)C2)ccc2c(C)c[nH]c2c1 N1(C(c2c(C)cc(C)s2)=O)CC(C(=O)NCCC(C)N2CCCC2)C2(CC2)C1 Cc1ccc(C)c(NC(=O)CNC(=O)CNC(C2(C)CC(O)CN2C)=O)c1 C(c1c(F)ccc(Cl)c1F)=CC(=O)NCC(CNC(C1C(CC)C1)=O)F CC1Cn2nccc2CN1C(=O)CCCCN(C(=O)CCC1CCC(=O)C1)C c1(C(=O)NCC(C)N(C(c2c(C)cncc2)=O)C)cccn2nccc12 C1(NC(C(CSC)O)=O)CC2(C1)CN(C(c1ccc[nH]1)=O)C2 N1(C(CC2(C=C)CN(C(C3CC4(C3)CC(O)C4)=O)C2)=O)CC(S(N)(=O)=O)C1 N1(C(=O)CCC2CCCCO2)CCN(C(C2(CO)CCOCC2)=O)C2(CC2)C1 c1(C(=O)NCC2(C)N(C(CS(CC)=O)=O)CCC2)cc(C2CC2)n(C)c1C C1(NC(C=CC)=O)CC2CC(NC(C3CC34CC(OCC)C4)=O)C2C1 C1(NC(c2nc(COC)oc2)=O)C2CC3CN(C(=O)CS(=O)(=O)N(C)C)C1C3C2 Cc1ccc2nonc2c1C(N1CC(CNC(=O)COC2CCOC2)C1)=O c1(C(N(CCCCCC)CCNC(=O)C(C)OC)=O)cc(C)cc([N+](=O)[O-])c1 C1(CNC(c2nocc2Br)=O)COCCN(C(=O)Cc2cnoc2)C1 CC1CCN(C(=NCCF)NCC2COC3(CCC(C)CC3)O2)CC1 N1(C(C(CCC)OC)=O)C(C(=O)N(C2CCC(O)CC2)C)CC2CCCC12 C1(C(=O)NCCN(C(c2cc(C(C)(C)C)on2)=O)C(C)C)(OCC)CCCC1 c1(CCC)cc(C(=O)NCCNC(c2c[nH]nc2Br)=O)ccn1 c1(C(=O)NC(c2cn(-c3ccccc3Cl)nn2)C)ccc2c(c1)NC(=O)CCC2 c1(C(N)=O)cncc(NC(C2CN(C(c3cccc(C(F)F)c3)=O)CCO2)=O)n1 c1(N(CCCCN(C(C=CC)=O)C)C)cc2ncnc(O)c2cc1[N+](=O)[O-] c1(C(N2CC=CC2Cn2cc(CC(O)C3CC3)nn2)=O)ncc2c(n1)CNC2 c1(C(=O)NCC(CC)NC(=O)CC(O)CN(C)C)cc(SC)oc1C C1(C(=O)NCC(CCOC)NC(=O)CC2COC(C)(C)C2)CN(C)CC(C)O1 c1(C(=O)NC2(C3N(C(c4nc(N(C)C)oc4)=O)CCC3)CC2)ccc2c(c1)CC2 N1(C(CNC(C)=O)=O)CCCCC1C(=O)N(C)Cc1ccsc1 c1(SCC(=O)NC(C2CCOC2)CNC(=O)C2CC2)cc(C(C)=O)ccn1 N1(C(C2(CF)CCN(C(c3ccn(C4CC4)n3)=O)C2)=O)CCN(C2CC2)C(=O)C1 c1(NC(C2CC(NC(c3cc(F)ccc3O)=O)C2)=O)ccc2c(n1)CCC2 Fc1cc(CCCNC2CCCC2c2ccccc2Br)ccc1Br C12(CCNC(C3(OC)CC3)=O)CCC(C1)N(C(=O)CC=Cc1ccc(F)cc1)C2 c1(C(N2CC(CNC(C3CC=C(C)C3)=O)C(O)C2)=O)ccc2c(n1)CCO2 Cc1ccc(C2(C(=O)NC(C3CCN(C(=O)CC4COCCO4)C3)C)CC2)cc1 N1(C(C2C(C(=O)NCC#C)C2)=O)CC2CC(NC(C3CC3(F)F)=O)CC2C1 c1(OC)cc(Br)ccc1C(N1CCOC(CNC(c2csc(NC=O)n2)=O)C1)=O N1(C(C2CC(C)CN2C(c2cnc(Cl)n2C)=O)=O)CC(O)C(N=[N+]=[N-])C1 C1(COC)(CNC(c2csc(C3CCCO3)n2)=O)CN(C(=O)Cc2cncs2)C1 c1(CC)c2n[nH]c1C(=O)C(C)COC2=O.C(C)(C)(C1(O)CC1)NCC1(CO)CC1 C(C(C)(O)C(F)(F)F)N(C(=O)C(=O)NCC1(F)CCOC1)C C1(NCCC(C(F)F)N2CCOCC2)CCCC2(CC1)OCCO2 C1(OC)CC2(CCN(C(C3CC(NC(=O)CCOC)C34CCC4)=O)C2)C1 c1(SCCCC(=O)OC)ccc(NC(c2ncsc2C(F)(F)F)=O)cc1 C=C(Cl)CCC(=O)N1CC(OCC(=O)NCc2nc(C3CC3)n[nH]2)C1 c1(NC(C2C(NC(C3(C(F)F)CC(=C)C3)=O)COC2)=O)cc(C)ccc1COC N1(C(CNC(CS(=O)(=O)NCCCNC)=O)=O)CC(C)CC(C)C1 CS(=O)(=O)c1cc(F)c(Cl)cc1NC(=O)NC1COC2(CCCC2)C1 Cc1cc(Cl)ccc1C(=O)NCC1CC2CCC1N2C(=O)CC1CC1(Cl)Cl c1(CC(N2C(CN(C)CC3CCC3)CCC2)=O)ccc(F)cc1C(F)(F)F C1(CCCNC(CC(C)OC)=O)CCCCN1C(c1cccnc1C)=O N1(C(c2c(C)[nH]c(=N)s2)=O)CCCN(C(=O)C(N2CCOCC2=O)C)C(C)C1 C(C(=O)N1CCC(C)(NC(=O)CCc2cccs2)C1)(C(C)C)SC CC(C)(C(=O)O)C(CCO)N1CCC(C(=O)NCCc2n[nH]c(=N)s2)CC1 C1(C(=O)NC(C(=O)OC)C)CCN(C(C2CCC2(OC)OC)=O)C12CC2 c1(C(=O)NCC2(F)CC(NC(C3CCC(C)C3)=O)C2)ccc(S(N)(=O)=O)cc1F CCC(CC(=O)N1CCCC(O)(CNC(c2ccc(C(N)=O)o2)=O)CC1)C(F)F N1(CC(=O)N(c2ccc(Cl)cc2F)c2scc(C)n2)CCCCc2ccccc21 c1(C(=O)NCC23C(CN(C(c4c(C)nsc4N)=O)C2)C3)cc2oc(C)c(C)c2[nH]1 C1(NC(c2cc(CCC)on2)=O)CCC2CC1CN2C(c1cnccc1CC)=O C(=O)(C(C)CCC(C)(C)C)N(CCN(C(C)C)C(C12CC(CO)(C1)OC2C)=O)C c1(C(=O)NCC(CN(C(Cc2c(C)ocn2)=O)C)C)cc2c(nc1O)CCCC2 C1(NC(c2nn(C)c(C3CCCO3)c2)=O)COC2(C1)CN(C(c1cocn1)=O)C2 c1(C(=O)OC)cncc(CNC(=O)CCC(C)NC(=O)CCOC2CC2)c1 c1(C(=O)NCCCC(C)NC(C(CCCC)C)=O)ccc2c(=N)[nH]cnc2c1 c1(NC(N2CC(CC)C(CC(=O)OC)CC2)=O)nc2c(s1)COCC2 Cc1c(F)ccc(C(N2CC3COCC3(CNC(=O)OC(C)(C)C)C2)=O)c1C#N N1(C(c2nc(C)oc2)=O)CCCCC(C2CN(C(=O)CCCCF)C2)C1 N1(C(CCOC)=O)CCC(OC(C)(C)C)CC1.C1(=O)C(O)C2CN(C2)C(=O)N1.O CCCCC(O)CC(=O)N1CCN(C(c2cc(CC(C)C)nn2C)=O)C(CF)C1 c1(OC)cc(I)c(CNC(=O)C(C)Oc2ccccc2C(F)(F)F)cc1OC N1(C(CCC=C(C)C)C(=O)NC(c2ccccc2Br)C)Cc2ccccc2C1 N1(C(c2n(C)c(O)nc2)=O)CCC(NC(c2cccc(=O)n2C)=O)C(C(N)=O)C1 C1(NC(C2(CC(C)C)CCCC2)=O)CCN(C(=O)C2CC2)CCC1CO N1(CCC(=O)NC2CC(C)N(C(=O)CN(C)C(N)=O)C2)Cc2ccccc2C1=O C12(CNC(c3c(C)cc[nH]3)=O)CC(C1)C(NC(=O)Cc1cn3ccsc3n1)CO2 c1(CC(=O)NCCC(CNC(CCCC#C)=O)(C)C)ccc(S(=O)(=O)CC)cc1 C1(NC(CC2OCCN(C(CN(C)C(N)=O)=O)C2)=O)CCn2ncnc2C1 O(C=CC(=O)N1CCCC1CCCNC(c1n[nH]cc1-c1ccncc1)=O)CC c1(C(=O)NCC(CC)NC(=O)C(CC)CC(F)F)c(F)cc(Cl)cc1Cl N1(C(C(CC)c2ccccc2)=O)CCCC(CNC(c2cc(F)n[nH]2)=O)CC1 C1(CC(N2CC(COC)(CNC(C3(C(N)=O)CCC3)=O)C2)=O)CCC=CCC1 C(=O)(C1CCOc2ccccc21)NC(CNC(C1CN(CCOC)C(=O)C1)=O)C C1(COC(C(CC(C)C)N(C)C(=O)OC(C)(C)C)=O)CCCCC12CCC2 CC1CCc2nc(C(N3CCC(N(C)C(c4cc(F)c[nH]4)=O)CC3)=O)cn2C1 N1(C(CC(=O)NCC#C)=O)CC(C)CC1C(=O)NCC(C)(CC)CO c1(C(N2C(CN(C(C3(CC#C)CC3)=O)CC)CCC2)=O)cnn(CCC)c1CC C(CCCC(C)(C)NC(C1CCS1(=O)=O)=O)NC(C1CN(C)C1)=O c1(C(=O)NCCC(C)N(C)C(c2ccc3c(c2)NCC3)=O)cc(S(N)(=O)=O)c[nH]1 c1(C(N2C(C)CC(CNC(C3CCC3)=O)C2)=O)cc2oc(Br)cc2[nH]1 C1(C(=O)NC2CN(C(C=NOC)=O)CC(O)CC2)CCc2cn(C)nc2C1 C(=O)(C1=CC2(CN(C(=O)C3=CCCOCC3)C2)OC1)N1CCC(C)(CC)C1 N#CC1(C(=O)NCC2CN(C(=O)Cn3cc(C4CC4)cn3)C2)CC12CCC2 n1(CC(=O)NC2CN(C(C3(CCOCC)CCC3)=O)C2)ccc(C)cc1=O c1(OC)cc(Cl)ncc1CN1CC(C(=O)Nc2csc(C(F)(F)F)n2)C1 Cc1ccc(F)cc1N(C(=O)C(C)C(C)NC(C1CC(=C2CC2)C1)=O)C C1(O)(CCNC(C2(CC(C)C)CC2)=O)CCN(C(=O)CC2CCC(C)CO2)CC1 C=CC1(C(=O)NCC2CC(F)(CNC(=O)C(C)SCc3ccccc3)C2)CCC1 c1(C(=O)NCC2N(C(c3nc(C(C)OC)sc3)=O)CC2)c[nH]c(C)c(Cl)c1=O c1(C(c2cn(CC3CCCC3)nn2)NC(CC(=O)OC)=O)ccc(F)cc1 C#Cc1cccc(C(=O)NC2CC(CCNC(C3CCC(C)C3)=O)C2)c1F C1(C(=O)NCC(CC)NC(=O)CS(=O)(=O)CC)CCc2ncnc(C)c2C1 CC(C)(C)CC(O)C(=O)N1CCC(C(=O)NC2C=CC(C)(C)CC2)(CC)CC1 C1(C)(CNC(CCCOCC)=O)CCCN1C(=O)C(O)CSC N1(C(C)C)CC2(CN(C(C3(NC(=O)C(c4ccnn4C)C)CC3)=O)C2)C1 C1(CC)(NC(c2ns[nH]c2=O)=O)CCCN(C(=O)C(N2CCNC2=O)C)C1 N1(C(Cc2n(C)nnc2)=O)CCC=C(CNC(C2CC3C=CC2C3)=O)C1 C1(NC(c2ccc(C#C)cn2)=O)CN(C(=O)CCCOCC)CC1S(C)(=O)=O C1(CCNC(COc2ccn(C)n2)=O)CCN(C(=O)CC23CCCC2C3)CC1 N1(C(C2(NC(C)=O)CCC2)=O)CCN(CC(C)(C)NC(=O)CC(C)(C)F)CC1 N1(C(c2cc(CC)ncn2)=O)CCC(C)(C)C1C(N1CCOC(C)C1CO)=O N1(C(C(CC)N(C)C)=O)CCC(OCCNC(=O)CN(C)C(c2cccs2)=O)CC1 c1(C(C=CC)=O)cccc(C2CCN(C(C3CC(O)(c4ccccn4)C3)=O)CC2)c1 c1(CC)cc(OC)c(NC(C2CC(C)OC2C)=O)cc1C C(=O)(CC(C)(O)CCC)N(C(c1cn(-c2ccc(OCC)cc2)nn1)C)C c1(SC)cc(F)ccc1C(N1CCCC1CNC(C1(F)CCCOC1)=O)=O CCCCC(C)CCC(=O)N1CCC(C2CCCN2C(=O)C(C)=CC2CC2)CC1 C#CCCCCCCC(=O)N1CCC(C(C)NC(=O)C(C)OCCC=C)CC1 c1(C(N(CCNC(=O)C2=CCSC2)CC2CC2)=O)cccc(F)c1Br C1(CNC(CCN(C(C)=O)C)=O)C2CN(C(c3conc3C(C)(C)C)=O)CC12 N1(C(CC2CN(C(C(c3cnn(C)c3)C)=O)C(C)C2)=O)CCC(F)(F)CC1 C(CCSC)(C(=O)NC(C)C(CO)NC(C1(CSC)CC(F)(F)C1)=O)OC C1(C(=O)NC2C(NC(c3c(C)nc(CC)o3)=O)C2)CCC(=O)N(C(C)C)C1 C1(c2n(C3CC(C(C)C)C3)nnn2)(NC2(C3CC3)CC2)CCCN2CCCCC12 Cc1csc(CC(=O)NC2(C3CCCN3C(c3ccns3)=O)CC2)n1 C1(C(=O)NC2CCC(N(C(C=CC(=O)OCC)=O)C)CC2)CCn2ncnc2C1 c1(C(=O)NC(C2(O)CCN(C(c3cc(F)cc(F)c3)=O)C2)C)nn(C)c(Cl)c1Cl C(CC(C(=O)N1CC(CC(F)F)C1)NC(=O)CCn1ccnc1)OC c1(C(N(C2CCN(C(c3cc(SC)oc3C)=O)C2)C)=O)ccc2[nH]c(C)cc2c1 N1(C2C(NC(Cn3nnc(C)n3)=O)COC2)CCN(C(c2scnc2C)=O)CC1 N1(C(C2C=CC=CC=C2)=O)CC2CCC(C1)N2C(=O)CC1(O)CCCCCC1 C1(C(=O)NCC2N(C(C(OC)OC)=O)CCOC2)(C(=O)O)CC2(CCC2)C1 C(C)(C(C(=O)NCC(C)(C)C(C)(C)O)C(C)C)NC(CCCOCCC)=O N1(C(COC2(C)CCC2)=O)CCC2CC1CN(C(c1csc(O)n1)=O)C2 N1(C(COCCCCC)=O)CCC(C)N(C(c2nc(COC)oc2C)=O)CC1 C(=O)(C1CNC(=O)c2ccnn21)NC(C)C(C)(C)NC(=O)C=Cc1cccnc1 CN1C(=O)CCC1C(=O)NCC(C)(O)CNC(=O)CC1CCCCC1O CC1CC(CC(=O)NC2CC(N(C)C)C2)CN1C(=O)C(CC1CC1)N(C)C C1(CN(C(C2(CCCC)CCC2)=O)CC)CCCN1C(C1CC1c1nc[nH]n1)=O c1(Cn2c(-c3cccnc3O)nc(C(CCC)C)n2)c(Cl)cccc1Cl N1(C(c2c(CC)n(C)cc2)=O)CCN(C(c2cc(O)nc(N(C)C)n2)=O)C2CC12 N1(C(CC(CNC(c2cncc(OC)c2)=O)C)=O)C2C=CCC1CCC2 CCC(C)C(=O)NCC#CC(=O)N(CC)Cc1cccnc1 C#CCC(C)C(=O)NCC#CCNC(C1(c2ccn(C)n2)CC1)=O C(=O)(CCCS(N)(=O)=O)NC(CCN(C(C)=O)C)C(C)(C)C N1(C(C(C)Cc2ccco2)=O)CCCC2CN(C(=O)Cc3cc[nH]c(=N)c3)CC12 C1(C)(COCC)CCCN(C(C2CCOCC2)C(=O)NCCSC)C1 N1(C(CCC2CCN(C(C(C=C)CC)=O)C2)=O)CCCCC(CO)C1 N1(C(c2cccc(COC)c2)=O)CCN(C(=O)COCCCC(C)C)C2CC12 O=C(C1=CCS(=O)(=O)C1)N1CC2CC(C1)N(C(c1cc(C3CC3)no1)=O)C2 c1(-n2cc(OCC(=O)OCc3nnc(CCOC)o3)nn2)cc(F)cc(F)c1 c1(CNC(=O)NCC(C)SCc2ccccc2)ccn(CC(F)F)n1 c1(CC)cc(C(=O)NCC2(O)CCCN(C(=O)CN3CCCC3=O)C2)ccc1O C1(CN(C(=O)C(c2ccc(Br)nc2)(C)C)C)CCCN(C(C2(C)CC2)=O)C1 C1(C(C)C)(C(N2CCC2CF)=O)CCN(C(=O)C(C)OC(C)(C)C)C1 c1(C(N2CCC(OCCNC(CC(=O)OC(C)(C)C)=O)C2)=O)cc(Cl)c(Cl)s1 Cc1ncc(C(=O)NCCC(C)N(C(=O)Cc2ccnn2C)C)cc1N c1(C(=O)OCC(n2cc(C(=O)OC)nn2)C)cc(OC)cc(OC)c1Cl C(=O)(C(C)(F)C(=O)NCCCN(C(=O)C=CC=Cc1ccccc1)CCO)OC C1(NC(=O)C2=CCCO2)CC2CCC(C1)N2C(c1c[nH]cc(F)c1=O)=O CC1CN(C(=O)C2CC2)CCCN1C(C1CCCC(=O)CC1)=O N1(C(c2nc(CCC)oc2)=O)CCC2CCCC12C(N1CCC2(CC2)C1)=O C1(NC(c2cc(OC)n[nH]2)=O)CN(C(=O)CCOCCNC(C)=O)CC2(CC2)C1 C1(C(=O)NCCNC(C(C)(C)C)=O)CC(O)CCN1C(=O)C1=NOCC1 N1(C(C2CC(NC(C3(CC)CC3)=O)C2)=O)CCC(c2ccon2)C(O)C1 C12(CNC(CS(=O)(=O)N(CC)CC)=O)CCC(CC1)N(C(c1ocnc1C)=O)C2 C12(CC)CCC(C(=O)NCC3CCCN(C(=O)Cc4nc[nH]n4)C3)(CO1)C2 C#CC1CCCN(C(=O)C(CNC(C2CC3(CSC3)C2)=O)OC)CC1 N1(C(CC(CC)SC)=O)CCC2(CC1)CC2CNC(C12CC(C(F)F)(CO1)C2)=O Cc1ccc2cc(COC(C3(C)CNC(=O)N3)=O)c(Cl)nc2c1 N1(C(Cc2n(C)c(S)nn2)=O)CCC2CN(C(c3ccc4nc[nH]c4c3)=O)C2C1 c1(CC(=C)C)nc(C2CN(C(=O)COC)C2)n(-c2ccccc2C(C)C)n1 c1(CN(C(C(CCC)n2cc(-c3cnc(OC)s3)nn2)=O)CC)ccccc1Cl Cc1nccc(C(=O)N(CCC(C(C)C)NC(C2C3CCC(F)(F)C23)=O)C)c1C C(=O)(C#CC1CCOC1)N1C2(CNC(c3cncc(OC)c3C)=O)CCC1CC2 c1(CC)n[nH]c(=NCC2CC(NC(=O)C(C3CCOCC3)F)C2)s1 C(=O)(CCCC(=O)N(C)C)N1CC(C(C(=O)NCCS(CC)(=O)=O)O)C1 Cc1nn(C2CCC2)cc1NC(=O)C(=O)Nc1ccc(CCC(N)=O)cc1 C(C(O)CC(F)(F)F)NC(C(C1CCC1)NC(CC1C(CC)C1)=O)=O C(=O)(CC(C)(C)C(F)(F)F)NC(C(C)NC(CC)=O)(C)C C12(NC(C(c3c(C)noc3C)C)=O)CCCC1(F)CN(C(c1cc[nH]c1)=O)C2 C1(C(=O)NC(CC)CN(C(=O)CCc2cnc(C)s2)C)CN(C)CCO1 CN1CCOC(C(N2CCCC2CC(=O)NCc2cnsc2)=O)C1 Cc1ccc(CC(=O)NCC2CC(NC(=O)CCCOCC(C)C)C(O)C2)cc1 C(CN=c1[nH]c2cccc(Br)c2o1)C1N(C(C(C)NC(CC)=O)=O)CCCC1 c1(CCC(=O)NC(=O)CC2CCCN(CCNC3CCCC3)C2)ccc(Cl)cc1 C1(COC)CC2(CCN2C(C2CCCC(NC(=O)CC3CCC(C)(C)C3)C2)=O)C1 N1(C(C(CC)SC)=O)CCCCC(CNC(=O)Cc2ccc(C)cc2F)C1 C=CCCCC(C)(C)CNC(=O)CC(CC(C)C)NC(C1C=CCC1)=O C(=O)(C1=NOC2(CCOC2)C1)N(C)CCNC(C1(c2ncco2)CCC1)=O CCC(C(=O)N1CCCC1C1CCN(C(=O)Cn2ccc([N+](=O)[O-])n2)C1)C(C)C Cc1cc(N)c(C)nc1NC(C1CCN1C(=O)CSCCC(F)(F)F)=O C1(CNC(c2nc(OCC)oc2)=O)CC(NC(=O)C=Cc2cc[nH]n2)C12CCC2 Cc1cc(C(N2CCC(C)C(CNC(=O)COCC3(F)CC3)C2)=O)c(Cl)cc1N c1(CCC(=O)N(CCNC(c2c(C)cc(Br)o2)=O)C2CC2)c(C)nc(O)nc1C C=CC1(C(=O)NCCCNC(N)=O)CCN(C(=O)NC2CCO2)C1 c1(C(=O)NCC(CNC(c2ccc(O)c(F)c2)=O)CO)cc(Cl)c(F)cc1F c1(C(=O)NCC(=O)N(CC(C)NC(c2cscc2F)=O)CC)cc2c(s1)CCC2 N1(C(C(CC2CC2)OC)=O)CC(C)(CNC(c2c(F)cccc2Cl)=O)CC1(C)C c1(C(N2CCC(NC(C3CC(=C)C3)=O)C(OC)C2)=O)c(F)cc(C#N)cc1F C1(NC(c2cc(CC)n(C)n2)=O)CN(C(=O)Cc2cc[nH]c2)CC2(CC2)C1 C(=O)(C(C1=NOCC1)N(CCc1ccccc1)C1CC1)NCC N1(C(CCC2CC(C)C2)=O)C(CNC(c2cccnc2)=O)CC2CC12 N1(CCOCCNC)CCC(NC(=O)CC2(C)CCN2)CC1 c1(NC(C2CC(NCC3CCN(C)C3)C2)=O)nc2cc(F)ccc2s1 C(=O)(N(OC)C1CCC1)C1C(CNC(C2C(CCC)C2)=O)CCC1 N1(C(c2cc(OC)no2)=O)CCCC2(CCN(C(C3CCCCNC3=O)=O)C2)C1 c1(C(=O)NC2C(CNC(C(c3ccc(F)cc3)C)=O)C2)ccc(C#N)cc1O c1(C(=O)NCC2(NC(COCCC=C)=O)CCCC2)cc(F)cc(Cl)c1 CC(C)CCCCCC(=O)NC(C(=O)NC(C1CCC1)C)C(C)(C)C c1(C(=O)NCC2(CO)CCN(C(C(CC=C)(C)C)=O)CC2)cn2ccccc2n1 CC(C)CC(C(=O)NC1(CN(C(=O)CNC(=O)C2CC2)C)CC1)N(C)C CC(C)CC(C(=O)NCC(C)NC(c1c(F)ccc2n[nH]cc12)=O)C(C)C c1(OC)cccc(-n2c(-c3ccc(F)cc3)cnc2SC(=O)CC2CCCO2)c1 C1(NC(CC2CC(C)(C)OC2)=O)CCC12CCN(C(=O)C1=C(Cl)CCOC1)CC2 N1(C(C(C)(C)C(F)F)=O)CCC2(CC1)CC2CNC(c1ccsc1C(F)F)=O c1(C(=O)NC(c2cnn(C)c2)CNC(C2C(CC)C2)=O)ccc(C(C)(C)C)nc1 CC1(O)CCC(C(=O)NC(C(=O)NC2C=CCCC2)C2CCCC2)CC1 c1(CC)nc(O)c(C(=O)NC2CC2CNC(c2oc(C(F)F)cc2C)=O)cc1C Cn1nccc(C(N2CCOCC2CCNC(c2ccc(C(F)F)o2)=O)=O)c1=O N1(C(C=CSC)=O)CCC2(CC1)CN(c1ncc(C#N)cc1C)CCO2 Cc1nnc2n1CC(C(N1CCC(C)N(C(C34CC(C)(CO3)C4)=O)CC1)=O)CC2 N1(C(C(C)N(C)C)=O)CCC2(CC1)CC2NC(c1cc(C2CCC2)[nH]n1)=O N1(C(C=CC)=O)CCCC12CCCN(C(C1CCCN(C(C)C)C1)=O)C2 C(CC(=O)N1CC2(COC(C)C2)C1)(C(F)(F)F)NC(C1CC=C(C)CC1)=O N1(C(c2c(C(C)C)[nH]cc2)=O)CCOC2(C1)CN(C(=O)CSCCN(C)C)C2 C(CCCC)(CC(=O)N(C)CCc1cccnc1)NC(CCCCC)=O c1(C(=O)OC)ccc(O)c(CN2CC(C)CC2C(=O)NCc2cccc(F)c2)c1 CC1CCC(C2CCCC2)CN1C(=O)NCc1csc2ccccc12 c1(-n2c(C)cc(C)n2)c(C)cc(NC(c2cnc(O)n(C)c2=O)=O)cc1C c1(CN2CCC(C(=O)NCc3c(C)cccc3)CC2)cnc(C2CC2)nc1O c1(CC(=O)OCCNC(C2CC(OC)C2)C)coc2cc(C)c(C)cc12 C(N=c1[nH]ccnc1F)C1C(NC(c2ccccc2COCCO)=O)CCCC1 C(=O)(C1COc2ccc(F)cc21)NC1C(NC(Cc2cc(CC)no2)=O)CC1 Cc1ccc(C(=O)NCCCCC(C)NC(c2cc(Cl)ns2)=O)c([N+](=O)[O-])c1 C1(NC(C(N2CCOCC2)C)=O)CC(F)(F)CC1NC(=O)CCc1cnc[nH]1 C1(CNC(c2ccc(C)n2C)=O)CCN(C(c2csc([N+](=O)[O-])c2)=O)CC1C N1(C(CCc2ccc(C)cc2)=O)CCN(C(c2csc(S)n2)=O)C(C)C1C c1(-c2nc(NC(=O)NC3(CSCC(=O)OC)COC3)sc2)cc(C)ccc1C N1(C(COCCC(C)C)=O)CC(O)(C2CCN(C(=O)C=CCF)CC2)C1 C(C(C)(C)C(=O)NC1COCC1CNC(C1(C)CCNC1=O)=O)N(C)C CC1(C)CCC(C)(C(=O)NCCC2(O)CN(C(c3ccc(F)cc3Cl)=O)C2)CC1 C1(C(=O)NCc2cccc(CC)c2)COC2(CCN(C(=O)C(C)CN)CC2)C1 CC(=O)CC(C)(C)C(=O)NC(C)CNC(=O)C(C)CCc1cccc(F)c1 c1(C(=O)NCCn2cc(-c3ccc(=N)[nH]c3)nn2)cc2cc(Cl)c(Cl)cc2[nH]1 N1(C(COC(CC)C)=O)CC(NC(=O)CCc2cc(C)[nH]n2)C2(CC2)C1 O=C(C1CCCc2ccccc21)NC1CC1NC(c1cccc2c1OCCN2)=O C(=O)(C1=Cc2cc(C)ccc2OC1)N(CCC)C(=O)C1CC1.n1(C)ncnn1 C1(CC(=O)NC2CCC(NC(C3(C)ON=C(C)C3)=O)CC2)CCCCC12CC2 c1(C(N(C2CN(C(=O)Cc3cscn3)CC2(C)C)C)=O)cc2c(s1)CCC2=O Cc1ncc2ccccc2c1C(N1CC(C(=O)C2CC2)(C(=O)O)C1)=O c1(C(=O)OCC(CCCC)O)nn(CC)c(Br)c1Cl Cc1ccc2cc(C(=O)NC3CCN(C(C4CC4F)=O)C3C)ccc2n1 c1(OC)nn(C)cc1C(=O)NCc1cc(C)c(C(=O)NC(C2CCOC2)C)o1 C1(NC(c2c(C)ccnn2)=O)CN(C(C2CCN(C)CC2)=O)CC12CCC2 c1(C(=O)NC(CNC(c2c(C)ccc(F)c2N)=O)C)[nH]c2ccc(F)cc2c1Cl N(C1CCc2ccccc21)C(CC=CCNC(C1(C)N(C)CCC1)=O)=O CCC(CC)CC(=O)NC(CC(F)F)C(=O)NCCCCCOC C1(N(C(C(C)c2ccsn2)=O)C)CC2CC1N(C(c1ccc(Cl)c(O)c1)=O)C2 C1(NC(C2(COC)CC2)=O)CC2CC1N(C(=O)CSC1CCS(=O)(=O)C1)C2 C1(C(N2C3CC(CC(NC(CC4(C)CC4)=O)C3)C2)=O)C2C3CC4C1C1C2CC3C41 CC#CCC(C(=O)NCC1CN(C2CC2)C1)NC(=O)CN1CCC(C)C1 Cn1ncc2c(=O)n(CC(=O)NC3(CF)CCN(C(=O)CC4CC4)C3)cnc12 c1(C(C)C)ncoc1C(=O)NCC1CCN1C(c1cocc1C(N)=O)=O O=C(C1=C(Cl)CCOC1)NCC(C1CCC1)NC(c1cc(Br)ccn1)=O C1(CNC(c2ccc(OC)c(Cl)c2)=O)CC2CCC1N(C(C13COCC1C3)=O)C2 c1(OC)cc(C)c(C(=O)NCC(O)CNC(=O)CNC=O)cn1 c1(C(N(CC(CN(C(COCCCC#C)=O)C)O)C)=O)nnsc1NC C1(CNC(C(CCCOC)C)=O)CC2(CCC2)CN1C(=O)C(C)(F)F CC1(C)CCC(C(=O)NC2CCN(C(=O)CCc3ncc(F)cn3)C2)OC1 c1(C(=O)NCCC2(CNC(CC3C(C)CCC3)=O)CC2)cncnc1C(C)(C)C C1(NC(CCCc2cc(C)sc2C)=O)CCN(C(c2nc(=O)cc(N)[nH]2)=O)CC1O N1(C(CCOCCN(C)C)=O)CCC(CNC(c2c[nH]cc(Cl)c2=O)=O)C1(C)C C=CCCCCCCCC(=O)NC(CNC(=O)CSCCC)CCC c1(OC)cc(C(N2CC3CC3(C(=O)NCc3cc[nH]n3)C2)=O)nn1C c1(C(=O)NC2CN(C(C3(C(=O)NC)CC3)=O)CC(F)C2)cc(C)c(Cl)c(C)c1 C(=O)(C1=NOC(C)(C)C1)N(C)CC1C(NC(C(CCC)NC(N)=O)=O)CCC1 C1(C(=O)NC(COCCOC)C)CC2CCCC2N1C(=O)CC1NC(=O)NC1=O N1(C(C2C(C(N)=O)C2)=O)CCN(C(C23CC(c4ccccc4)C2C3)=O)CC1 N1(C(=O)NCC(c2cc(Cl)sc2Cl)n2ccnc2)CCC2CCCCCC2C1 C12(CNC(CS(=O)(=O)NC(C)(C)C)=O)CCCC1CCN2C(c1csnn1)=O CC(C)CC(C(=O)NC1(CO)CN(C(c2nnc(S)n2C)=O)C1)c1ccccc1 N1(C(C(CC)(C)CO)=O)CCC2(C=C(C(=O)NC(CO)C(O)CCC)C2)C1 CCCC(C(O)C(=O)NC1(C)CCCC(C)(C)C1)NC(=O)CNC(=O)CC Cc1cc(C(=O)NC2CC(O)CN(C(c3cccc(F)c3Cl)=O)C2)c(C)cn1 N1(C(C(=O)NCc2ccccc2)=O)CCC(CO)(Nc2cncc(Cl)n2)CC1 C1(O)(C(C)NC(=O)CCc2nc[nH]n2)CCN(C(c2ccc(N)cn2)=O)CC1 N1(C(C=CC(CC)C)=O)CCOCC1CCNC(c1ccc(C)n1C)=O n1(CC(=O)NCC(C)N(C(c2[nH]cc(C)c2)=O)C)ncc(O)nc1=O CC(Cc1ccccc1)C(=O)NC1(C)CC(NC(c2coc(C3CC3)n2)=O)C1 c1(C(N2CCC(CC)C2CNC(=O)CC23CCCC2C3)=O)ccc(N)c(Cl)n1 C(C)(C(C(=O)N(CC1=CCCOC1)C)C(C)C)NC(c1ncnc(C)c1C)=O CC(CCNC(C1CSCCN1C(c1cc(F)c[nH]1)=O)=O)CCO Cc1c(NC2CN(C(=O)CCCc3ccsc3)CCC2C(F)(F)F)ncnc1Cl N1(C(C(CO)NC(C(C)CC#N)=O)=O)CC2CSCC2(C)C1 c1(CC)nnc(C)cc1C(N1CC(NC(=O)CCC#N)CC(O)C1)=O Cc1oc(C)c(C(=O)NCC2(O)CN(C(c3cc(Cl)sc3Cl)=O)C2)c1C c1(OC)ccc([N+](=O)[O-])c(NCC(C)(C)NC(=O)Cc2cc(O)nc(O)n2)c1 N1(C(C=C(CC)C)=O)CCC(CCNC(=O)CCCn2cc(C)cn2)C1 C1(CNC(C(CC=C)C)=O)CCN(C(c2ccc(C(F)F)nc2)=O)C1(C)C N1(C(c2nc(COC)sc2)=O)C2CCC1CN(C(=O)C(C)(CO)OC)C2 O=S(=O)(c1cnc(NCC(O)Cn2cccn2)c(Cl)c1)N1CCSC1 N1(C(CNC=O)=O)CCC2CCN(C(C3CCC4(CCCC4)C3)=O)CC12 N1(C(C2OCCN(C(C(C)(C)CCCF)=O)C2)=O)Cc2cc(O)nnc2C1 c1(C(N2C3CN(C(CCN4C(=O)CCCC4)=O)C(C3)C2)=O)nnn2c1COCC2 C1(C(N(CCNC(c2ccc(SC)s2)=O)CC)=O)CC2C=CC1C2 C(CCCC(C)(C)C(=O)NNC(=O)C(C)NC(N)=O)NC(C1ON=C(CC)C1)=O C1(SC)CN(C(c2csc(-c3n[nH]c(C)n3)n2)=O)CC1NC(=O)CC(C)(C)C C(=O)(C1CCc2c[nH]nc21)N1CC(SC)C(NC(C23CCC(F)(CC2)C3)=O)C1 C1(C(=O)NC2CCN(C(CCC=C)=O)C2C(C)(C)C)CC12CCCCC2 C1(O)(N(C(=O)COCCCF)C)CCN(C(=O)COCC2CCOC2)C1 C1(CNC(C2ON=C(CC)C2)=O)CC(C)CN(C(c2cc[nH]c2C)=O)C1 c1(CN(C(=O)C(=O)N(C)CC2COC(C)(C)C2)C)cn(C)nc1-c1ccccc1 C1(C(N2CC(CNC(CC#N)=O)OCC2)=O)C2CCC(F)(F)C12 C#Cc1ccc(C(N2CCC(CC(=O)NCC(C)(CC)CO)C2(C)C)=O)cn1 C1(CC)CN(C(C2(C3(C)CC3)CC2)=O)CC1C(=O)NOCc1nc[nH]n1 C(CCC(O)C(=O)NCCC(C)CO)NC(CSC)=O C(=O)(C1Cc2ccccc21)N(CCCCN(C(=O)CCn1cccn1)C)C c12ccc(C(N3CCC(CCSC)C3)=O)cc1O2.C(=O)(C(F)C1CCC1)NCC C(c1ccncn1)=CC(=O)NCCN(C(CC1CC(OCC)C1)=O)C(C)C C1(n2cc(C3(C)CCCN3C(C3CCC4CC34)=O)nn2)Cc2ccc(Br)cc2C1 C1(C(=O)NC2(C(C)O)CC2)COC(CNC(=O)CCc2cnn(C)c2)C1 N1(C(C2CC(C(F)F)(OC)C2)=O)CCOCC(NC(=O)C=Cc2nccs2)C1 C(C(CNC(c1ccnn1CC(F)F)=O)CO)NC(C1(CS(N)(=O)=O)COC1)=O CC1(C(=O)NC2CCN(C(=O)CCNC(=O)CO)CC2)COc2ccccc21 CN1CCC(C(=O)NCCCC(C)(C)O)(NC(=O)CCC2CCCCC2)C1 C(=O)(CCC(C)C)N(CCNC(C=CCN(C)CC)=O)C1CC1 c1(OC)ccccc1C(=O)N(CC(O)CN(C(=O)CSC(C)C)C)C c1(C(N2C(C)(CNC(C3C(C(C)C)C3)=O)CCC2)=O)ccc(Br)c(F)c1F N1(C(C2N(C(C3CCCC(CF)C3)=O)CCN(C)C2)=O)CCC2CCCC2CC1 N1(C(C2CCC(C)CN2C(=O)CC(C)O)=O)CCC(O)C(C)(O)C1 c1(N2CCN(C(c3c(CC)noc3)=O)CC2CCO)nc2cccc(C)c2o1 c1(CC(N2CCOCC(NC(=O)CC(O)C3CC3)C2)=O)cc2ccccc2o1 C(=O)(CCCC(=O)N1CCCC(NC(c2ncoc2C2CCCO2)=O)CC1)NC N1(C(C2(OC)CCCCCC2)=O)CCC(C)N(C(=O)CCC(C)CN(C)C)CC1 C1(C(=O)NC(c2ncc(C)s2)C)(CNC(C2CC(=C3CCC3)C2)=O)CC(C)(C)C1 C(C(C)(O)C(=O)NCC(CNC(=O)CN(c1ccc(Cl)cc1)C)CO)OC CC1CC(NC(=O)CC2CC2C(F)(F)F)CN(C(=O)C(C)(C)COCC(F)F)C1 N1(C(c2cccc(OC)c2)=O)CCc2n[nH]cc2C1.N12CC(OC)CC1C2=O c1(C(=O)NCC2(NC(C3CC(C)OC3)=O)CCC2)cc(O)nn1C C1(C(=O)NCCCCCN(C(C2(CC)CCC2)=O)C)CCOC(=O)CC1 C(CCCCCC(=O)NC1CCN(C(=O)CCc2c[nH]c(=N)[nH]2)CC1(C)C)SC c1(C(N2C(CNC(C3C4CCC34)=O)CC2)=O)cnc(O)c(C(F)(F)F)c1 c1(C(=O)NCCN(C(C(C)NS(C)(=O)=O)=O)Cc2ccccc2)cnnc(O)c1 c1(CNCCC(=O)CCO)ccc(Br)c(Cl)c1 Cc1nc(N)cnc1C(=O)NC1CN(C(c2ccc(C(N)=O)cc2)=O)CC12CC2 C(=O)(CC1=CCCC1)N1C(CNC(C(C)OCC)=O)COCC1 C#CC1(C(N2CC3(CCC3O)C2)=O)CCN(C(=O)C(C)CCC)CC1 N1C(=NCc2ccccc2)N2CCCC(C2)C1=O.O=C1OCC(CSC2CC2)O1 C(=O)(C(C1CCCO1)NC(=O)C(C)C)N(CCCOCCOC)C.C1(=O)CO1 c1(Nc2ccc[nH]2)cc(Cl)ccc1C(N1C(C(=O)NCC(C)(C)C)CCC1)=O O(NC(=O)C(O)CNC(C1CCCCN1C)=O)CC(C(C)C)O N1(C(C2N(C(Cc3n(C)ncc3)=O)CC=C2)=O)CCC2(CC1)CC(O)C2 N1(C(c2c(CC)oc(C)c2)=O)CC2CCCC1C2CNC(c1cn(C)nc1O)=O N1(C(C(C)(CO)NC(=O)C(C2CC2)C2CC2)=O)CC2(CCOC2)C1 N1(C(CCc2cccc(OC)c2)=O)CCC2C(C1)CN2C(C1CC2C=CC1C2)=O N1(C(CC=C)=O)C2CCC1CC(F)(CNC(c1cccc3sccc13)=O)C2 Cc1ccnc(C(=O)NC2CC=C(C(=O)NC34CC(F)(C3)C4)C2)c1N N1(CCNC(C(C)NC(CC)=O)=O)CCC(NC(=O)C(CSC)OC)CC1 C(=O)(CCCCC(F)(F)F)NCCCc1cn(CCOC)nn1 C(=O)(C1=COc2ccccc2O1)N(C1CC(NC(C(CCOC)C)=O)C1)C C(=O)(C(O)CC(C)(C)C)N1C(C(N(OC)C)=O)C=CC1 C1(CNC(C2CCC(OC)C2)=O)(OC)CCN(C(=O)Cc2cnccc2C)CC1 N1(C(Cc2c(C(C)C)con2)=O)CCN(C(c2cc(N)nc(Cl)c2)=O)CC(O)C1 N1(C(CC(C)(C)SC)=O)CC23CCCC2(C1)CN(C(C1CCC12CCC2)=O)C3 c1(C(=O)NC2CC(NC(C3CCC(=O)C3)=O)CC2O)cccc(F)c1Br N1(C(c2cn(CCC)nc2)=O)CCC(C(N2CC(N(C)C)C(C)C2)=O)C1(C)C N1(C(c2c(OC)ccs2)=O)CCN(C(=O)C=Cc2cncn2C)C(C)CC1C c1(C2(C(=O)NC(C)CNC(c3cccnc3O)=O)CC2)ccc(Cl)cc1Cl Cc1ccc2sc(C(=O)NCCC3CN(C(C4(O)CC4(C)C)=O)CC3C)cc2c1 N1(C(C(C(C)C)(C)C)=O)CC(NC(c2cn(CC(N)=O)nn2)=O)C2CCCC2C1 c1(C(N2CC(C(=O)N(c3c(C#C)cccc3)CC)SCC2)=O)ccc(C)c(C)c1I C1(CNC(C2C(OC)CC2)=O)CC2CCC1N(C(c1ccc(F)c(C#N)c1)=O)C2 C1(C(=O)NC)(OC)CCN(C(=O)CN2CC3CCC2C3)C1 c1(C(N2C(C(=O)OC)(CC)CCC2)=O)cnn2cc(C)cnc12 C1(OC)CCN(Cc2cccc(I)c2)CC1C CC1C(NC(=O)COC2CCCC2)CCCN1C(=O)CNc1ccccn1 CC1=CCC(C(=O)NCC2(F)CC(CNC(c3cnoc3C3CC3)=O)C2)CC1 C12(CNC(c3c(CC)nccc3)=O)CCC1CCN2C(c1cnoc1C)=O c1(C(=O)NCC2CCN(C(c3cc(OCC)no3)=O)C2)ccc(Cl)c(C#N)c1 C1(C(C)C)CCC(C(N2CCC(CC(C)C)C2)=O)N1C(=O)CC1COCCO1 C1(C(=O)NC(CCCC)(C)C)CN(C(C2CCCN2C)=O)CC1(F)F CCCCC(O)C(=O)NCCC1CC(NC(C2(c3ccc(Cl)cc3F)CC2)=O)C1 Cc1oc(C#N)cc1C(N1CC(C(=O)NCC2(C#N)CCC2)CC1(C)C)=O Cn1cnc(Br)c1C(=O)Nc1ncc(Cc2ccccc2)s1 c1(C(N(CC(CNC(C(CCOC)C)=O)C)C)=O)ccc2c(c1)C(=O)CCCC2 N1(C(C2(C#C)CC2)=O)C2CCC1CN(C(C1(O)CCCN(C(C)=O)C1)=O)C2 C1(C(N2C(CC(C)C)CC2)=O)CCN(C(=O)c2cccn(C)c2=O)O1 C#CC1(OCC(=O)N(C)CC2(O)CN(C(=O)Cc3nnc(C)o3)C2)COC1 c1(COC(C23N(C(=O)OC(C)(C)C)CCC2CC3)=O)cc(C)c(C)c(Br)c1 c1(CC)nc(CC(=O)NCC(C)NC(=O)CC23CCCC2C3)cs1 S(=O)(=O)(c1ccc(CS(C)(=O)=O)cc1)Nc1n(-c2cc(C)nn2C)ccc1 C(CCCCN=[N+]=[N-])N(C(N(C)C)=O)CC1CC1 N1(C(CC(=C=C)C)=O)CCC(NC(c2cnn(C(C)(C)C)c2C)=O)C(F)C1 C1(O)(C(=O)NCCC(C)(C)NC(C(CN(CC)CC)F)=O)CN2CCC1CC2 C(=O)(CCCC(C)(C)CC)NCC(Cn1cc(C(=C)C)nn1)OC c1(C(=O)NCC(CO)NC(C(C)OC)=O)cccc(CC#N)c1 N1(C(C(C)OCC)=O)CC2CCN(C(=O)Cn3c(C)csc3=O)C(C2)C1 C(=O)(CC(O)CC(C)(C)C)N1CCCC(C(=O)NCC(C)CC2CCC2)(CC)C1 c1(C(=O)NC(CC)CNC(c2cccnc2C(F)F)=O)cc(C#N)cc(C)n1 c1(CC)scnc1C(=O)NCC(=C1CN(C(=O)CC(C)C2CCCCC2)C1)F c1(C(=O)NC23CC(CNC(c4ccc(OC)cc4)=O)(C2)C3)ncc(Br)cc1C C1(CCNC(CC2CC(OC)C2)=O)CCCCN1C(C1CC(C)(O)C1)=O n1(CCCC)nnnc1C(C)(CC1CCCCC1)NC(c1cccs1)(C)C1CC1 C1(F)(CNC(C(C(C)C)OCC(C)C)=O)CCN(C(C2CCCOCC2)=O)CC1 CC(C)C(O)C(C)(C)C(=O)NCC(C(=O)N1CC(OCC(F)F)C1)N(C)C N1(C(C2N(C)CCN(C(C3C4CCC(C4)C3C)=O)C2)=O)CC(=O)N(C)C(=O)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1CCCC(CNC(C(C)(C)C#N)=O)C1 c1(C(C)C)nccc(NC(C2CCN(CC3CN(C)CCO3)C2C)=O)n1 C1(NC(=O)C=CCN2CCOCC2)CC12CCN(C(C1OCCCO1)=O)CC2 C1(CC(=O)NC(c2ccccc2)C)CCCN(C(c2cc(Cl)n[nH]2)=O)CC1 Cc1oc(CNC(c2cn(C)nc2O)=O)nc1C(=O)NC1CCC(CN(C)C)C1 c1(NC(=O)NCCC2CCCC(C)C2)ccc2c(c1)C(O)CC2(C)C C1(NC(c2nccc(CC)c2)=O)CCC(C(F)(F)F)NC1=O C1(NC(c2c(C3CC(=O)NC3)cccc2)=O)COC2(C1)CN(C(=O)CO)C2 c1(C(=O)NC(C#C)(CC)CC)ccc(OC)c2ccccc12 C1(NCc2nc(CC)on2)CCN(C(=O)CC(c2ccccc2)C2CC2)CC1C C1(C(=O)NCC2(CCC)CCC2)CCCN(C(=O)Cc2cc(C)n(C)n2)C1 N1(CC(=O)N(CCCCN(C)C(c2cc(Cl)ns2)=O)C)CCCCS1(=O)=O C1(C(N2C(CNC(c3[nH]nnc3C3CC3)=O)CC(OC)C2)=O)Cc2nccn2C1 c1(OC)cc(CNC2CCN(C(C3CCCCC3)=O)CC2O)ccc1C(F)F C1(C(=O)NCCCCCNC(=O)CCCC2CCCC2)(CC)CCCC1O N1(C(C2(CC(C)C)CCC2)=O)CC2CC(NC(=O)C(C)NC(=O)C(C)(C)C)C1C2 CN1C(=O)CCCC1C(N1CCC(C)(C)C1CC(=O)Nc1cccc(CO)c1)=O C12(C(=O)NC3C(CNC(CN(S(C)(=O)=O)C)=O)C3)CCC(C(F)(F)F)(CC1)C2 C1(C(=O)NCC(c2ccc(C(C)C)cc2)NC(=O)CO)CC12CCCCC2 n1(CC)cnc2c(N3CCCN(C(=O)C(C)O)CC3)ncnc12 C12(CCC)CC(C(=O)NCCC3CC(NC(=O)C(C)CN4CCOCC4)C3)(C1)C2 C1(CCC)COCCN1C(=O)CC1CCCN1C(=O)CC(=O)OCC C(=O)(CCCCCCCCC(=O)N1CCCCC2(CCN(C(=O)C3CC3)C2)C1)OC C1(NC(CCN(C(C)=O)C)=O)CCC2(C1)CN(C(C1CNC(=O)O1)=O)C2 C(=O)(N=c1[nH]nc(OC2CCCCC2)s1)NCc1nccc(N(C)C)c1 C1(C)(C(N2CCC(NC(CC=CC=C)=O)C(O)C2)=O)COC2COCC2O1 Cc1cccn2c(C(N3CC(CNC(c4ccc(C)n4C)=O)C(O)C3)=O)cnc12 c1(C(=O)NC2C(CNC(C(=O)NC(C)C)=O)C2)ccc(-c2ccccc2)cc1F Cc1cc(C(=O)NCC23CC2CN(C(=O)CC2(O)CCCOC2)C3)nc(C)n1 N1(C(C2C(C)CCCC2)=O)CCC(NC(=O)Cc2cnnn2C)C2(CCC2)C1 C(C)(CCCCNC(c1nc(C2CC2)oc1C)=O)NC(COCC#C)=O c1(C(=O)NCC(=CC(=O)N(CC(=C)C)C)C)cnnn1CC C1(CCC)(Nc2ncnc(C)c2Br)CCN(C(C2(C)CC(C)=NO2)=O)CC1 N1(C(c2c(OCC)n[nH]c2)=O)CCC(CNC(C2CCCC(OC)C2)=O)CC1 N1(C(C2(C)COCCO2)=O)CCC(NC(c2ccc(Cl)s2)=O)C(CO)C1 C12(C(N3CC(=CC)C3)=O)CC(CO)(CN1C(=O)C(C)(O)C(C)C)C2 Cc1cccc2c1OCC2C(=O)N1C2CCC1C(NC(c1[nH]cnc1C)=O)C2 N1(C(CCN(C(C)=O)C)=O)CCCC2C(CCCN2C(=O)CNC=O)C1 c1(CCC(=O)NCC2C(NC(C(CC)C)=O)C2)cccc(F)c1 c1(CC)noc(C(N2CCC(CCNC(=O)Cc3cccnc3)C2)=O)c1C c1(CNCC23C(CC(=O)N2)CCC3)[nH]c2ccccc2c1Br c1(C(N2CCCN(C(C(C)=C(C)C)=O)CCC2)=O)ccc2n[nH]c(C)c2c1 C=CCCC(C(=O)NC1CC(C)(C(N)=O)C1)NC(=O)CC1CCCCO1 C#Cc1cc(C(N2CCC(C)(CCNC(=O)COC3CC3)C2)=O)cc(Br)c1 N1(C(c2c(C)nsc2)=O)CC2CCC(CNC(C3CC4CCC(C3)N4C)=O)(C2)C1 C1(OC)(CNC(c2ccoc2C)=O)CCN(C(C23CC(CCO2)C3)=O)C1 C1(NC(C(CCC)O)=O)CN(C(C2CCC(C(C)(C)C)O2)=O)CC2(CC2)C1 c1(OCCOC)cncc(C(=O)NC(C)(CNC(=O)Cn2cc(C)cn2)CO)c1 Cc1ccc(C2CCN2C(=O)C(CN=[N+]=[N-])c2ccccc2)cc1Cl C1(CC=C)(NC(c2ccc(C(O)CF)cc2)=O)CCN(C(=O)Cc2csc(C)n2)C1 C1(NC(C(C)N2CCCC2)=O)CC2CCC(C1)N2C(=O)CCC1CC(C)(C)CO1 C1(C(=O)NC2CCN(C(C(C)CSC(F)(F)F)=O)CC2)CCc2nn[nH]c2C1 C1(O)(CNC(=O)CCCF)CCCN(C(c2cc3n(n2)CCC3)=O)C1 C12(CC)CCC(C(N3CC4(CCN(C(=O)CCn5cnnn5)C4)C3)=O)(CC1)CO2 N1(C(c2c(CC)non2)=O)C(CC(=O)Nc2ccc(O)nc2)C2CCCC12 N1(C(c2cncc(NCC)c2)=O)CC(O)C(O)C1CNC(c1nnccc1C)=O c1(OC(C)C)ccc(C(=O)OCc2ccc(C#N)o2)cc1 C#Cc1c[nH]nc1C(=O)NCCN(C)C(c1cccnc1O)=O CCCCCC(=O)N(C)CC1(C(=O)NC2CCCC2c2nc(S)n[nH]2)CC1 c1(C(=O)NCC(C(=O)NC2C3COCC23)OC)cccc(C)c1O Cc1onc(-c2ccccc2F)c1C(=O)NC1CCCC1NC(C1(C)CC1)=O N1(C(c2c(C)occ2)=O)CCC(NC(=O)CC2CC3(CC3)C2)C1C CC1CCCc2cc(C(N3CCC4(C3)CC4(F)F)=O)nn21 Cc1cc(CCC(=O)NCC2CN(C(c3ccnn3CC3CC3)=O)C2)cc(F)c1 C(=O)(CCCN=[N+]=[N-])NC1(c2ccccc2)CN(C(c2ccc(CC)[nH]2)=O)C1 N1(C(Cc2ccc(OCC)cc2)=O)CC(CNC(=O)CC(C)(C)C)C(C)(C)C1 C1(CC(=O)N(C2CCCN(C(=O)Cc3ccoc3)CC2)CC)CCC(=O)NC1=O C1(COC(C)=O)CN(C(=O)C=C(C)CNC(=O)C(C)CC#N)C1(C)C C1(c2ccc(F)cc2)(NC(C=CC(CC)C)=O)CCN(C(=O)C=CS(C)=O)CC1 N1(C(C(CCC)N(C)C)=O)CCN(C)CC1CNC(=O)CC1CCCC1(F)F c1(C(=O)NCC2CCN(C(c3ncc(C)nc3)=O)C(C)C2)nccc2nn[nH]c12 c1(C(=O)NCCN(CCC)C(C2(NC(C)C)CC2)=O)cccc2nc(O)ccc12 C1(C(N2CCN(CCN(C(CC=C=C)=O)C)CC2)=O)CC2CCCCN2C1 N1(C(C(C=CC)O)=O)CCCN(CCCCNC(c2cccc(CC)c2)=O)CC1 CC1CCC(CC(N2CC(F)(CNC(c3cncs3)=O)C2)=O)C1 N1(C(Cc2cc(C(C)C)no2)=O)CCC(C(C)(C)C)(CNC(=O)C(C)(C)CF)C1 N1(CCCc2ccc(C)cc2C)CC2CC1CC2(C)O C1(NC(c2ccc(C)c(C)n2)=O)CN(C(=O)Cc2ccno2)C2(CCOC2)C1 c1(CC(C)NC(N2CC(N(C)C(=O)C3CC3)C2)=O)ccnc(O)c1 C1(CNC(=O)C(O)(C2CC2)C2CC2)CCC(NC(C2CC23CCOC3)=O)CC1 CCC(C)(CO)C(=O)NCC1(NC(c2cc(=O)c(Br)c[nH]2)=O)CCOC1 CC1CC(NC(c2ccsc2F)=O)CN1C(C1CCOC(C)C1)=O c1(C(=O)NC2(COC)CN(C(=O)Cn3ncccc3=O)C2)ccnc(N(C)C)c1 c1(C(N2CC(CNC(C3(CCOCC)CCC3)=O)C2)=O)ncc2[nH]ncc2n1 N1(C(C=CC(CC)=CC)=O)CCC(O)(CNC(=O)COC(C)(C)CC)C1 C1(NC(CCOCC)=O)CCN(C(c2sc(CC(F)(F)F)nc2C)=O)CC1C c1(C(N2CC(C)OCC2)=O)cn2c(n1)CCN(Cc1cc(Br)co1)CC2 c1(C(=O)NC2CC3CN(C(c4c(C)onc4)=O)C2C3)cccc2c1SCCC2 C(=O)(CC(C)(C)CC(F)F)N(CCCNC(CCCC=C)=O)CC c1(SC)cc(C(=O)NCC2C3CC2N(C(C2CC(F)(F)C2)=O)C3)c(C)o1 N1(C(c2c(COC)ncs2)=O)CCCC(CO)(NC(=O)C(O)Cc2cnc[nH]2)C1 c1(OC(C)C)cc(C(N2CC=CC2CNC(=O)CNC=O)=O)nc2ccccc12 C1(CC(=O)NCC2CN(C(C3CCCCO3)=O)CC2O)CCC=CCC1 N1(C(=O)OCC)CCC(C(C(F)F)NCCC(C)OC)CC1 N1(C(C2CC=C(C)CC2)=O)CC(NC(=O)Cc2cnsc2)C(C2CC2)C1 Nc1c(C(=O)NCC2(c3cn(C4CCC4)nn3)CC2)cnn1CCO CCCCCC(C)(C)C(=O)N1C(C(=O)NCC2CCCOC2)CC2CC12 N1(C(COC2(C#C)COC2)=O)CCCC(F)(C(=O)NCc2ccc(OC)nc2)C1 c1(-c2cnc(=NC)[nH]c2)cnc2[nH]cc(C(=O)NCc3cncc(C)c3)c2c1 C1(CN(C(C=CC(C)C)=O)C)CCC(CNC(c2cn(CCO)nn2)=O)CC1 N1(C(Cc2cc(CC)no2)=O)CCOC(C(N2CCC(F)(F)C2C2CC2)=O)CC1 C1(CC(=O)OC)C(=O)NCCN1C(c1c[nH]nc1C(C)(F)F)=O N1(C(c2on(C)c(=O)c2)=O)CCOC2CCN(C(=O)C=Cc3ccoc3)CC12 C1(CCCCC(=O)NCCCCCCN(C)C)SCC2NC(=O)NC12 CC(C)CCC(C)N(C(=O)CC1CCCN1C(c1nc[nH]n1)=O)C C12(CC(N3CC=CC(OC)C3)=O)CCC1CN(C(c1cc(C)ncc1C)=O)C2 C(C)(C(C(=O)NCCC1(O)CCOC1)NC(=O)COC(C)(C)C)OC c1(CNC(C2CCCCCC2)CO)cccc(F)c1Cl c1(C(=O)NCC2(C(N(CCN(CC=C)C)CC)=O)CC=CC2)cncc(O)c1 C1(CNC(C(CC)N(C)C)=O)CC2(CCN(C(C3CN(C)C(=O)N3)=O)CC2)CO1 N1(Cc2cc3ccc(F)nc3[nH]2)CCC(N=c2nc[nH]n3ccc(Br)c23)C1 c1(C(=O)NCCC2CCC(NC(C=Cc3cnc(C)s3)=O)C2)c[nH]c(=N)cc1C Cc1cc(C)c(C(C)NC(=O)C(=O)NC2CCCC2)c(C)c1 C1(O)(CNC(Cc2cc(C)sc2)=O)CCCN(C(C2(C#N)CCCCC2)=O)CC1 CN=c1ccc(C(=O)N(C2CCC(CNC(=O)CCNC(=O)NC)CC2)C)c[nH]1 c1(C(=O)NC(C(=O)N(CC(=O)OCC)CCC)C)ccn(C)c1 c1(C(C(=O)NCCS(C)(=O)=O)N(C(C)C2CC2)C)ccc(N(C)C)nc1 c1(OC)ccc2c(C(N3CCC(NC(C4CCCC(C)(C)C4)=O)C3)=O)cnn2c1 C1(C(=O)NCCc2ccnc(C)n2)CCCN1NC(=O)C(C)Cn1ccnc1 CC(F)(F)C(F)(F)CC(=O)N1CC=CC(NC(c2cc(Cl)sc2Cl)=O)C1 C(=O)(C#CC1CCCCO1)N1CC(OC)(CNC(=O)C(C)N2CC(C)C2)C1 c1(CC(=O)NC2CC(C(C)NC(=O)C=CC3CCCCC3)C2)cccc(Cl)c1F N1(C(C(C(C)OC)O)=O)CCn2ncc(CNC(c3cnoc3C)=O)c2C1 c1(C(=O)NC(C2N(C(CCSCC)=O)CCC2)(C)C)ccc(F)c2[nH]ccc12 CCC(CC)C(C)C(=O)N1CCC(NC(c2cc(N)c(C)c(N)c2)=O)C(C)C1 N1(C(C2N(C(C(CCC)NC(N)=O)=O)CC2)=O)CCCC2(CCOC2)C1 C1(C(=O)NCC2OCCC2C(=O)NCC2CCC(O)C2)CCCCC1O N1(C(c2cn(C)nc2)=O)CCCC(C2CCN(C(=O)C(C)(C)C(C)(F)F)CC2)C1 N1(C(C(=O)NCc2cnsc2)=O)CCc2c([nH]c3ccc(F)cc23)C1 C1(CNC(CCCOC(C)C)=O)CCN(C(C2CN(C(C)C)C2)=O)C1(C)C C1(N(C)C)CCCC(C(=O)NC2COCC2CNC(C2(CO)CCCCC2)=O)C1 C1(O)(CNC(CN(C(C)C)C)=O)CCCN(C(=O)C(C)Cc2ccccc2)CC1 c1(C(N(C(CNC(COC)=O)C)C)=O)cc(C)n(-c2ccc(C(=O)OC)cc2)n1 Cc1ccccc1-n1cc(C2(CC(=O)Sc3ccc(Cl)cc3)CCOCC2)nn1 c1(C(=O)OCC(=O)Nc2ccc(Cl)cc2)cc2c(nc1O)CCSC2 C1(C(=O)OCc2ccc(OC)c(C)n2)(CO)CC(F)(F)C1(F)F C(c1ccc(C(C)C)cc1)=CCC(N1CC(N(C(CCN(CCC)C)=O)C)C1)=O c1(OC)ccc(C(N2CCOC(CNC(=O)C(C)C(C)C)C2)=O)c2ccncc12 C(Cc1cc[nH]n1)(C(=O)N(C)Cc1cn[nH]c1)NC(C(C1CCC1)OCC)=O C1(C)(CNC(C2(C#C)CCC2)=O)CCCN(C(c2ccc(OC(F)F)cc2)=O)C1 C=CC1(CC(=O)NC2CCN(C(C)C)C2)CN(C(=O)CC2CC(OC)C2)C1 O=C1NC2(C(=O)NC3(c4ccc([N+](=O)[O-])cc4)CCC3)CCCC1C2 c1(C(COC)N(C)C(C2CC2Cc2cc(C)[nH]n2)=O)ccc(Cl)cc1 c1(C(=O)OC(c2ccccc2[N+](=O)[O-])C(=O)OC)cc2n(c1)CC(C)NC2=O CCC(C)C(C)(O)CNC(C1CCCC(NC(=O)C(O)CC(N)=O)C1)=O Cc1cc(N)c(C(N2CC3(CCN(C(C4(n5ccnn5)CC4)=O)C3)C2)=O)cc1F N1(C(C2N(C(C)=O)CCCC2)=O)CCOC(C)(CNC(c2c(C)ccn2C)=O)C1 c1(C(C)C)cc(C(N2CCC(N(C(=O)CSc3ccncc3)C)CC2)=O)n(C)n1 c1(SC)noc(C)c1CNC(C1(NC(=O)C(C)NC2CC2)CC1)=O C1(C(=O)NC2CCC(CN(C)C(C3(CCF)CC3)=O)CC2)CCOC(=O)CC1 C12(C(=O)NC(C)Cc3cccnc3)CCN(C(=O)C(F)C3CCCC3)CCC1C2 N1(C(c2c(Cl)cnc(C)n2)=O)CC(NC(c2cc(CCO)on2)=O)C(N=[N+]=[N-])C1 N1(C(COC)=O)CCOCC1CC(=O)NCCC1CC(=O)N(C)C1 C1(C(N2C(CNC(C3N=C(C)SC3)=O)CC(F)(F)C2)=O)CCc2ncncc2C1 N1(C(C(CC)CC)=O)CC2(NC(=O)C(CC(C)C)OC)CCC1C2 C12(NC(c3n(C=C)ncc3)=O)CCCN(C(=O)C(C)CC(C)C)CC1C2 c1(OC)cc(C(O)C(=O)N2CC(CC(=O)Oc3cn[nH]c3)C2)c(F)cc1O Cc1nc(O)[nH]c1C(=O)NCCC1CCCN1C(C1CCOC1C(C)C)=O c1(C(=O)NC2C(C)N(C(c3cc4ccccc4s3)=O)CC2)snc2ccccc12 CCCCCC(C)(C)C(=O)N1CC(CNC(=O)Cc2cc(C)no2)C2(CC2)C1 c1(NCC(CCC)CCO)cc([N+](=O)[O-])ccc1OCCCC(=O)OCC c1(NCC)cc(Cl)ccc1C(N1CC(NC(c2cccc(C)c2)=O)CC1CO)=O S(=O)(=O)(CC(=O)N1CC(OCCOC2(F)CC2)C1)N(C)C1CC1.C1(=O)CO1 C1(O)(CCNC(C2(CC#C)CCCO2)=O)CCN(C(C2CCC2=C)=O)CC1 C(c1cccc(Cl)c1)=CC(=O)NC1CN(C(C(CC#C)O)=O)CC1CC(C)(C)C N1(C(Cc2n(C)ccn2)=O)CC(NC(=O)Cc2ccco2)CCC(O)C1 c1(C(N2C(CC)CN(C(=O)C(F)=CC3CC3)CC2)=O)cc(OC)cc2c1CCC2 c1(OCC)ccc(Cl)c(C(N2CC(NC(=O)CCC(CC)OC)CC(C)C2)=O)n1 c1(CC)cc(NC(=O)NN2CCCC2(C(C)O)CO)sc1C(=O)OC C1(CNC(=O)CC2(CO)CC2)C2CN(C(=O)C=C(C3CC3)C3CC3)CC12 C=C1CC(C(=O)NCc2ccncc2)N(C(c2ccoc2C(F)(F)F)=O)C1 c1(-c2cn(CC3CC(NC(C4(OC)COC4)=O)C3)nn2)cnc(C)nc1 CCC(=O)CCC(=O)NCC(C)(C)C(N1CC(CO)C(C)(C)C1)=O c1(CC(NNC(CSCCOC)=O)=O)ccc2c(c1)OC(F)(F)O2 C1(C(=O)NC(CC)CSC)(CCOC)CCN(C(c2ncc(F)cc2C)=O)CC1 N1(C(c2cncc(OCC)c2C)=O)CCOC2(CCC(C#N)CC2)C1 CN=c1ncc(-c2ccc(NC(=O)C(C(C)C)NC(=O)OC(C)(C)C)nc2)c[nH]1 c1(COC)cc2c(c(=O)o1)C(c1ccc(OC)cc1)NC(=S)N2CCC(C)=O CC1CCCC=C1C(=O)NC(CN=[N+]=[N-])C(=O)NC1CCC(C(N)=O)C1 C(C(C)(C)CCN=c1nc2scnc2c(NC(CCO)C(F)F)[nH]1)OC CS(=O)(=NC(=O)Cn1nnc2c(C(F)(F)F)cccc12)c1cccc(Br)c1 N1(C(CNC(N)=O)=O)CC2CCN(C(c3cccc(C4CCC4)c3)=O)CC12 CCCC(CNC(=O)CC1CCOC1(C)C)C(=O)N(C1CCCC(=O)C1)CC c1(NC(c2c(C)nc(C3CC3)s2)=O)ncc(C#N)cc1C#N c1(CC(N2CCC(C(C)NC(=O)Cc3ccnc(Br)c3)C2)=O)cc(F)ccc1O C(=O)(C1CCCn2nccc21)NCCN(C)C(c1cnc(=N)[nH]c1)=O N1(C(C2(NC(N)=O)CC2)=O)CC2(C=C(C(=O)N3CCC(O)C(F)(F)C3)CO2)C1 C=CC1(C(=O)NC2CC(O)CN(C(=O)Cn3ncccc3=O)C2)CCCCC1 n1(CC)ccc(C(=O)NCC2(C)CCCN2C(c2cnc(C(N)=O)s2)=O)cc1=O C=CC1(C(N2CC(NC(c3cc(C)nnc3O)=O)C(C)C2)=O)CCCCC1 C1(F)(CNC(C(C)OCCOCC)=O)CCCN(C(c2csc(C#N)c2)=O)C1 C1(CNC(=O)CC2CCCC2)COCCN1C(c1cccnc1O)=O N1(C(C(CSC)(C)NC(=O)C(O)C2CCC2)=O)CC(=O)NC(=O)C1C N1(C(C(CN(C(C=CCOCCOC)=O)C)C)=O)CC(C)CC1CO C1(CNC(C(=O)NCC)=O)CCCCN(C(=O)C(C)(CC)CO)CC1 c1(NC(C2CCN(Cc3cnc(Cl)c(F)c3)CC2)=O)cc([N+](=O)[O-])ccc1Cl C(=O)(C(C)(C)S(C)(=O)=O)NC1C(NC(C(C(C)C)N2CCCCC2)=O)C1 CCC(CC(=O)NC(C(=O)NCc1nnn(C)n1)C(C)(C)O)CC(C)C N1(C(C(CC)N(C(=O)CCn2cccn2)C)=O)CCCC(C#N)C1 CN(CCc1cnc(O)nc1)N1CCN(C2CC3CCC(C2)N3C)CC1 c1(OC)cc(F)c(C(=O)O)cc1S(=O)(=O)NCc1cc(O)ccc1O c1(N2C(CNC(C3(C4CC4)CCCO3)=O)CCCC2)ncnc2[nH]cnc12 CCCC(CNC(c1ncnn1CC)=O)C(=O)N1CC(O)CC1COC C#Cc1cccc(CC(=O)NCC#CC(N2CCCC(C)C2CCO)=O)c1 C(=O)(C1=CCCN(C(c2cc(Cl)c(O)cc2F)=O)C1)N(CCC(=O)N(C)C)C Cc1nc(CC(C)C)c(C(=O)NC(c2ccccc2)CNC(C2CC2F)=O)s1 C1(C(N2CC(C=C)(CC(=O)N(C)Cc3ccns3)C2)=O)CCOC(C)(C)C1 N1(N(c2ccc3occc3c2)C(c2nc(C)sc2)=O)CCN2CC(O)CC2C1 C(CC(C)(C)CNC(=O)CC1CCCC(C)C1)NC(C(C1CCCC1)OC)=O c1(C(N2CCC(N(C(=O)CC3CNC(=O)C3)C)C2)=O)ccc(C#N)cc1F C1(C(N(CCCCN(C)C(C2CCCN2S(C)(=O)=O)=O)C)=O)COCCOC1 CC1CCC(C(=O)N(CC(=O)NC2CC2)C)N1C(C1CC2(CSC2)C1)=O N1(C(C(C2(OC)CCCCC2)(F)F)=O)CCC(NC(C2(N(C)C)CC2)=O)C(C)C1 c1(C(=O)NCCC2CC(NC(C34CCCCC3C4)=O)C2)ccnc2[nH]nnc12 CCC(Cc1ccccc1)C(=O)NC1CCC(NC(c2n[nH]c(C)c2F)=O)C1 C(CCC(C)NC(C1CCC(C)C1)=O)NC(C(C)OCC)=O C1(NC(C(COC)(C)O)=O)CCN(c2ccnc(C3CC3)n2)CC(C)(C)C1 CN1CCNCC1C(N1CC2C(CF)C2C1)=O C1(C(N(C)CC2CCCS2)=O)CC12CCN(C(c1ccc(O)cc1)=O)CC2 C(=O)(C(F)CC(C)(C)C)NC1CC(CC(=O)NC(CC)CCOC)C1(C)C Cc1ncc(F)c(=NCC2COC(C)C2)[nH]1 O(S(=O)(=O)CCc1cccc(F)c1)CC(=C)C C(CCN=C(NCC1CCC(NS(C)(=O)=O)CC1)NC1CCS(=O)(=O)C1)OCC N1(C(C(CC)CC(C)C)=O)CCC2(CC1)CN(C(c1ccc(Cl)cc1O)=O)C2 c1(C(C(=O)NC(C)CCN(C)C(C23COCC2C3)=O)(C)C)cccc(Br)c1 c1(C(=O)NC2C(NC(c3cc(C(C)(C)C)n[nH]3)=O)CCC2)ccncc1F C1(C(=O)NCCCCCCN(C(CCCC=C)=O)C)C2Cc3ccccc3C12 C12(C(N3CCC(C)(COC)C3)=O)C(NC(c3ccc([N+](=O)[O-])o3)=O)C3CC1C2C3 C1(C(=O)NC(C2CN(C(c3c[nH]c(Br)c3)=O)C2)C)CCCCC1C n1(CCOC)cc(C(=O)NC2CCCC2NC(c2coc(C(F)(F)F)c2)=O)nn1 C1(OC)(CNC(C2(Cl)CCCCC2)=O)CCN(C(c2cc(C)sc2C)=O)C1 N1(C(COc2cccc(C)c2F)=O)C(NC(=O)C(C)CN(C)C)CC2COCC12 C1(CNC(C2C(NC(c3cc(CCC)on3)=O)C2(C)C)=O)OCCCC1(C)C C(=O)(C1=CC2(CCOC2)C1)N1CC(CNC(CCCC(=O)OC)=O)C(C(F)F)C1 N1(C(C=CC)=O)CC2CC(C1)CN(C(=O)Cc1csc3ccc(Cl)cc13)C2 C1(NC(CCC(C)=O)=O)CCCCCCC1NC(=O)C(C)C1CCCO1 c1(C(=O)NC2CCC(NC(C(C)(F)F)=O)C2)ccc(C2(F)COC2)cc1 C#Cc1ccc(C(=O)NCC2CC2NC(c2cc(C3CCCC3)[nH]n2)=O)cc1Cl c1(C(=O)NC2C(NC(Cc3c(C)ccnc3)=O)CC2)nc(Br)cnc1N c1(C(=O)NCC(CC)NC(=O)C(C)(COC)OC)ccc(C(=O)C2CC2)cc1 CC(C)(CCNC(C1CC(CC2CC2)C1)=O)NC(=O)C(CO)c1ccccc1 n1(CC)cc(Cl)c(C(N2CCC(C)(NC(=O)Cc3cccc(OC)c3)C2)=O)n1 N1(C(C=CCCC)=O)CCCC(CC(=O)N(C2(C=C)CCC2)CCC)C1 C1(NC(c2cn(CC)nn2)=O)CCCC(C(N2CCC(OCCN(C)C)C2)=O)C1 C=CC(C)(O)CC(=O)NC(C)CC1CCN(C(=O)C(c2ccc(C)cc2)C)CC1 N1(C(CCCOCCOCC)=O)CCOCC1CN(C(=O)C=Cc1cscn1)C Nc1cc(C(N2CC(CNC(=O)CC3CC4(CC4)C3)C2)=O)cnc1Cl CC1(OCC(=O)NC2CC(CC(=O)NC3CNC(=O)C3)C2)CCCC1 N1(C(C(=O)NCc2ccc(-c3c(C)n[nH]c3C)cc2)=O)CCC(O)(C2CC2)C1 C1(CN(C2CCN(C)C2)C(C(=O)NCC)=O)CCN(C(C)=O)CC1 c1(C(=O)NC2C(NC(CC(C)F)=O)COC2)cnc2[nH]ccc2n1 c1(OC(CC)C(=O)NC23CC(CNC(=O)CC4CC4(Cl)Cl)(C2)C3)ccccc1C C1(CC)CN(C(=O)Cn2ncn(C)c2=O)CC1C(=O)N(C1CC2CCC1O2)C N1(C(C2CC23CCCC3)=O)CCC2(CCC2)C(CNC(C2(CCO)CC2)=O)C1 C1(C(=O)NC(C=C)(C)C)CCC(C)N(C(C2CN3CCC2CC3)=O)C1 c1(C(N2CC(F)(CNC(C3C4CCC3CC4)=O)C2)=O)cc2ccccc2cc1Cl Cc1cc(C(N2CC(NC(=O)C(C)N(CC(F)(F)F)C)C(O)C2)=O)nc(O)n1 N1(C(c2c(C)oc(Cl)n2)=O)CC2CCCC(CNC(C3CC=CC3)=O)C2C1 C1(NC(Cc2c(C)nn(C)c2C)=O)CCCC12CCN(C(=O)C1=C(Cl)CC1)C2 C1(NC(C=NOC)=O)CCC2(CC1)CC2NC(=O)CSCc1ccncc1 Cc1cc(P(C)(C)=O)oc1C(=O)NC1CCN(C(=O)C(O)C(C)C)CC12CCC2 C(=O)(C1=C(Cl)CCOC1)NC1CC(C)CN(C(=O)Cc2cnccn2)C1 N1(C(CCN(C)CC)=O)CC=CC(NC(=O)Cn2ccc(C3CC3)n2)C1 C(=O)(C(CC)C(F)(F)F)NCC1(CNC(CC=CCC)=O)CC12CCC2 C1(NC(c2c(C)n(C)nc2)=O)CC2CCC(C1)N2C(c1cc2cccn2cn1)=O c1(C(=O)NC2CCN(C(C(=O)NCC)=O)C2)ccc(F)c(SC)c1 N1(C(c2cnn(C(C)C)n2)=O)CCCC1(C)C(=O)NC1(CN(C)C)CC1 N1(C(C=CC(=O)N(C)C)=O)CCCC(CNC(=O)CC23COC(C2)C3)CC1 N1(C(C2C(C=C)C2)=O)CCCCC12CC(NC(c1ccc3ncsc3c1)=O)C2 C1(C(=O)NC2C(NC(c3c(CC)con3)=O)CCOC2)CCCCC1(C)C c1(NC(c2n(CC)nnn2)CCc2ccccn2)cc(Cl)c(C)cc1OC N1(C(c2cc(C)sn2)=O)CC2CN(C(=O)CC(O)C(C)C)CC(C1)O2 C(=O)(N1CCCc2nccn21)c1c(CNC(c2c(CC)n[nH]c2)=O)ocn1 N1(C(C(CC(C)C)C)=O)CCC2CCN(C(c3cc(C(F)F)ccc3Cl)=O)C2C1 N(C1CCCc2ccccc21)(C(C(=O)NC1C(CN(C)C)COC1)=O)C1CC1 Cc1cc2ccc(C(N3CC(F)CC3CN(C)C(C3CC34CC4)=O)=O)cc2o1 C(=O)(C(C1CCOC1)NC(=O)CNC(C1CC1C)=O)N(CC(=O)OC)C c1(C(N2CC(CC)N(C(C3CC(C(C)C)C3)=O)CC2)=O)cccc2cnsc12 C(C(CC(=O)N1C2CCC(C2)C1CNC(C1(O)COC1)=O)C(F)F)N(C)C c1(C(N(CC(CC)NC(=O)COCC2CCOC2)C)=O)cnc2[nH]ncc2c1 CC(C)C(C)(F)CNC(C1CC(NC(=O)CC(C)N(C)C)C(O)C1)=O C(C)(CC(=O)NCCC(c1cccs1)NC(=O)CCC(N)=O)(C1CCC1)N(C)C C1(CNC(=O)CN2CCSCC2)CN(C(=O)C(F)=C2CCC2)CCCO1 C(=O)(CC(C)C(F)F)NCCC1CC(NC(C(C)NC(c2ccccc2)=O)=O)C1 CC(C)C(CN=c1[nH]c(N2CC3CC3(CO)C2)nc2cc[nH]c12)N1CCCC1 c1(OC)ccc(C(C)CC(=O)NC(C)CNC(=O)Cn2nnc(C3CC3)n2)cc1 C1(NC(C#CC(C)(C)C)=O)CCCC2CN(C(C3(C)CCCC3)=O)CC12 c1(C(=O)NC(C(C)C)(C)CNC(=O)CC(C)(C)C)cnc(O)c2cnccc12 C1(NC(C2CCCCN2C(=O)Cc2ccccc2F)=O)C(O)C2CCOC12 c1(C(N(C(CC)CC)C)=O)nc(CNC(=O)C(F)C2CCOC2)oc1C C1(C(=O)NCCCC2(CNC(C(C)NC(C)(C)C)=O)CCCC2)CCC(F)CC1 C1(NC(C(C(C)O)C)=O)CCSC12CN(C(C1(O)CC(C)(C)C1)=O)C2 c1(C(=O)NCC(CNC(c2cn(CC)nc2C)=O)F)cc(F)cc2cccnc12 c1(C(N(CC(C)CNC(C2(C(C)(F)F)CCOCC2)=O)C)=O)c(O)cccc1F Cc1ccc(Cn2cc(CC3CCCN3C(=O)CC3COC(=O)C3)nn2)o1 C1(N(C(C(CCCC)O)=O)C)CCC2CN(C(c3cccc(Cl)c3F)=O)CC12 C(=O)(N1CCC(C(N2CCC2CF)=O)O1)C1(CCOC)CCC1 c1(C(N2CCOCC(NC(C34CC(C)C3C4)=O)C2)=O)nc2cc(O)ccc2[nH]1 c1(N2C(C3(NC(c4cc5c(o4)CCCC5)=O)CC3)CCC2)ncnc2scnc12 Cc1cc(C)c(NC(=O)NC(Cc2c[nH]c3ccccc23)CO)cc1Br C1(NC(c2snc3ccccc23)=O)CS(=O)(=O)CC1N=c1nc[nH]n2cccc12 C12(NC(CS(CC)(=O)=O)=O)CCCC1N(C(c1cnc(N(C)C)nc1)=O)CC2 C1(CCNC(c2cc(C)sn2)=O)CSCCN1C(=O)CCc1cnn[nH]1 n1(C(C(=O)NC(C)C)C)cc(CC2CCCN2C(=O)C(N2CCNC2=O)C)nn1 Cc1cccn2cc(C(N3CC=CC3CNC(=O)C=CC=C(Cl)Cl)=O)cc12 CCC(CC(=O)N(CC(=O)NC(c1ccccn1)C)C1CC1)C1CCC1 Cc1c[nH]c2ncnc(N3CC4CC(NS(=O)(=O)CC(C)C)CC4C3)c12 c1(C(=O)NCCCOC2CCN(C(CC(C)(C)OC)=O)CC2)ccc(O)c(N)n1 c1(-c2n(-c3n(C)ccn3)nc(C3CSC3)n2)cc(F)c(Cl)cc1F C1(CNC(CCN(C(C2CC(C)C2)=O)C)=O)CCC=CCC1 C1(F)(CN(C2CC(O)C2)C(C2N(C(=O)OC(C)(C)C)CCC2)=O)CCOCC1 c1(C(=O)NCCN(C(c2c[nH]c(=N)o2)=O)CC)c[nH]nc1-c1ccco1 CC1(C)CN(C(=O)CC2CCC(=O)C2)CC1NC(=O)CC1CC(F)C1 C12(CC(=O)N(CC(CC)NC(C3CCN(C)C3)=O)CC)CCC(CC1)CC2 C1(C(C)NC(C2(CCC)CC2)=O)CCCN(C(c2ccc(=O)oc2)=O)C1 N1(C(C2C(C)OCC2)=O)CC2CCC1C2NC(c1cccc(C(F)(F)F)c1)=O c1(OC)cnc(Cl)c(C(=O)NCC2CCCN(C(c3cc(Cl)ccc3Cl)=O)C2)c1 C1(C(N(CCCCC)CC=C(C)C)=O)CNC(C)C1 C(=O)(CC(O)CC(C)(C)C)N1CCC(CC=C)(NC(C2CCC(=O)O2)=O)C1 Cc1onc(C(F)(F)F)c1C(=O)NC1CCN(C(=O)CC(C2CC2)C2CC2)C1 C(CNC(=O)COC1CCCC1)(CC(F)(F)F)NC(C(COC)N(C)C)=O c1(C(N2CC(OC)(CNC(C3(C)COC(=O)C3)=O)C2)=O)cc(F)c2[nH]nnc2c1 n1(CC(=O)NC2(C3CN(C(C(C)CC4CC4)=O)C3)CC2)cc(C#N)c(O)nc1=O N1(C(=O)NC(c2ccc(-c3ccccc3)cn2)C)CCC2CCC(C2)C1 C1(C)(CC)CC(NC(c2cc(C(C)C)oc2C)=O)CN1C(c1cccc(O)n1)=O N1(C(c2ccc(C(CC)=O)s2)=O)CC(CNC(=O)C2CC2)C2(CCC2)C1 C1(F)(CNC(c2c(C)ncs2)=O)CCN(C(C2CNC(=O)N2C)=O)CC1 C12(C(N(CCOCC)C)=O)COC(C1)C(NC(c1ccc(F)cn1)=O)C2 C1(C(N2CCC(F)(C(=O)N(C)CC3CCCCC3)C2)=O)(OC)CCOCC1 c1(C(=O)NC2C(C(=O)NCCC(C)(O)C3CC3)COCC2)cccc2ccnn12 C1(CC(=O)N(C2CCN(C(c3cnoc3C3CC3)=O)C2)CCC)CCC(=O)NC1 C12(C(N3C(C=C)CCC3)=O)C(NC(c3cnns3)=O)C3CC1C2C3 C1(NC(c2c(C)onc2)=O)CN(C(C2CC3(CCO3)C2)=O)CC12CCOCC2 C=C=C(C)CC(=O)NCCCC1CN(C(c2conc2COC)=O)CCO1 C1(CC)CCCN(CC(N2CCC(NC(=O)Cc3nncn3C(C)C)CC2)=O)C1 N1(c2c(OC)cncn2)CC2(C)CN(C(c3cc(F)c(Cl)cc3F)=O)CC2(C)C1 CN=c1[nH]cc(C(=O)NCC2CC(F)CN2C(=O)CNC(c2cscn2)=O)o1 c1(NCC(OC)OC)ccc(S(=O)(=O)NCC(CC)N2CCCC2)c(Br)c1 C1(C(=O)OCC)(C(=O)NCC2CC2NC(=O)COC2CC2)CCCC1 c1(CC)cc2c(CNC3(CO)CC4C=CC3C4)cc(=O)oc2cc1O N1(C(c2ccn3nccc3n2)=O)C2CCCC1CN(C(C13CCCCC1C3)=O)C2 C1(C(N2CCC(CNC(CCS(C)(=O)=O)=O)C(O)C2)=O)CCc2nc[nH]c2C1 CCC(CNC(c1cc(CC2CC2)on1)=O)(CC)NC(=O)C(F)C1CCC1 C1(C(C)NC(c2cc[nH]n2)=O)CCN(C(=O)C2=CCC2)C1 c1(CC)cccc(C(N2CCC(F)C(NC(=O)CSC(C)C)C2)=O)c1O CC(C)(N=[N+]=[N-])C(=O)NC1CC(C(=O)NCCCCC(F)(F)F)C1 c1(C(=O)NC(C2(O)CCN(C(C(CO)OC)=O)C2)C)cc2ccccc2n1C C(=O)(N1CCC(C(N2CCOC(C)C2)=O)O1)C1CCC(CN)O1 C(=O)(CCC(=O)N(C)CCNC(C1(c2cncnc2)CCCC1)=O)NC NC(=O)C(N)CCC(=O)N(C1CC2(CNC2)C1)Cc1cccc(OCCO)c1 C1(CC)CCC(C(=O)N(CC(C)NC(c2cnn(CCOC)c2)=O)C)CC1 Cc1nnn(CC(=O)NCCCCCN(C(=O)C(c2ccncc2)C)C)n1 C1(C(=O)NC(CNC(C(C(C)C)NC=O)=O)(C)C)OCC2CCCC12 N1(C(C2(CNC(c3cncn(C)c3=O)=O)CCCC2)=O)CCC(C2CCOC2)C1 N1(C(C(C=C)(C)C)=O)CC2CCCC2(CNC(c2ccc(C)o2)=O)C1 C12(CNC(C(C(=O)OC)(C)F)=O)CCC(NC(C3CCN(C)C3)=O)(CC1)CO2 c1(N2C(CC)CCC2)cc(C(=O)NCc2csc(C)n2)ccc1C(=O)O N1(C(C(=O)N(C)C)=O)CC2CC(NC(c3cn(-c4ccccc4F)nn3)=O)C1C2 C1(C#N)(C(=O)NCCCCCCN(C)C(c2ccccc2)=O)CCCOC1 c1(OC)ccc2ncccc2c1NC(=O)C(c1cccc(C(F)(F)F)c1)(C)C CCCCCC(=O)N1CCCC(C(N(C)Cc2ccccn2)C)C1 c1(C(=O)NC2CC(C)(NC(=O)CN3CC4CC4C3)C2)cc(Br)ccn1 c1(OC(C)=O)cc(NC(c2ccc(F)c(F)c2F)=O)c2ccccc2c1 CCCCC(CC)C(=O)N1CCC(COC)(NC(c2cc(C(F)(F)F)ns2)=O)C1 C#CCCCCCC(=O)N1CCC(CNC(=O)C(O)Cc2cnc[nH]2)C1(C)C Cc1nnc(COCC(N2CC(C(C)NC(=O)C(N3CCNC3=O)C)C2)=O)s1 c1(OCCC(=O)NC2(C)CCN(C(C(COC)(C)O)=O)C2)cc(F)ccc1F N1(C(CCSC)=O)CC(C2CCN(C(c3cc(Cl)ccc3C(C)C)=O)CC2)C1 c1(CCC)[nH]ccc1C(=O)NCCCC(C)NC(=O)CC1CC12CC2 N1(C(C(C)NC=O)=O)CC2(CC(C(N3CCCCC(C)(F)C3)=O)CO2)C1 C=CC(CCC)CC(=O)NC1CN(C(=O)CCCc2ccccn2)CC1O O=C(C1Cc2ccc(Br)cc21)Nc1cn(C(c2nccc(Cl)c2Cl)C2CC2)nn1 c1(C(=O)NC(CC)(C)CNC(=O)Cn2c(C)c(C)sc2=O)ccc(C)c(C)c1N CC1C(C)N(C(c2cnc3n2CCCC3)=O)CCN1C(c1ccc(Cl)o1)=O c1(C(=O)NC2CC(CCNC(C(COC)(F)F)=O)C2)sc(Cl)c(Cl)c1OC C1(NC(C(=O)Nc2c(C)scc2)=O)CC(=O)N(C2CN(C(=O)NC(C)(C)C)C2)C1 C1(C(=O)NCC2CC(F)CN2C(C2CCCN2C)=O)(COC)CCC(=O)N1 c1(C(N(C(CN(C(C2=C(C)OCC2)=O)C)C)C)=O)cccc2c1OC(C)C2 N1(C(C2=CCC(NC(c3sccc3F)=O)C2)=O)CCc2nc(O)[nH]c2C1 C1(NC(C2(CCCC)CC2)=O)CN(C(=O)CC2(CSC)CC2)CC1OC Cc1cnc(CNC(C2(NC(=O)C(O)C3CCC3)CC2C)=O)o1 C(=O)(C(O)CCNC(=O)C=CCC(C)(C)NC(C1(C)CCCS1)=O)OC C1(NC(=O)CCc2cccc(C(F)(F)F)c2)CCCC2CCNCC12 C1(O)(CNC(c2c(CC)nn[nH]2)=O)CCCN(C(=O)C=CC2(C)COC2)CC1 c1(C(=O)NC2CCN(C(c3c(CC)n[nH]c3)=O)CC2)cccc(OC)c1N c1(NC(CN(CCC)CCNC(c2snnc2C)=O)=O)ccc(Br)cc1 C1(NC(CCc2n(C)ccn2)=O)CCCC(NC(=O)C=Cc2nnn(C)n2)C1 CC(C)C(CCN(C(=O)C(C)C1CCC1)C)NC(=O)C(C)(C)O N1(C(c2ncn(C(C)C)c2)=O)CCC2(C1)C(F)(F)C2(F)F N1(C(c2cc(C)sc2)=O)CCC(C)C1CNC(c1sccc1-n1cnnn1)=O C12(CC)CC(C1)NC2=O.C12CC1C2.C12CC1NC2=O.C(C)(C)(C)NC(=O)OC N1(C(C(C)C2CCCO2)=O)CC=C(C(=O)NCc2cccnn2)C1 N1(C(c2c(C)c[nH]n2)=O)CCC(C(C)CNC(c2cc(Br)n(C)c2)=O)CC1 C1(F)(C(N2CC(C)C(CNC(c3cc(F)cnc3Cl)=O)C2)=O)CC2(CCC2)C1 N1(C(C(C(C)C)n2ccnc2)=O)CC2CC1CN2C(c1ccc([N+](=O)[O-])o1)=O c1(NCCN(CC)CC)ccc(S(=O)(=O)N2CCCCC2CO)cc1F C(=O)(CC(O)CC(C)(C)C)NCC(CC=C)C(=O)Nc1cccn2ncnc12 c1(CNC(=NCC2C(C(=C)C)OCC2)NC(CC)C(F)F)ccc(S(C)(=O)=O)o1 c1(C(=O)NC(C)C(CO)NC(=O)C=Cc2cncs2)ccn2cnnc2c1 c1(C(=O)NC2(C3CCN(C(CCSC)=O)C3)CC2)nccc2c(C)cccc12 N1(C(C23N(C(C4C(CC)CCC4)=O)CCC2CCC3)=O)CCC(O)(C2CC2)CC1 C1(c2onc(C)n2)CN(C(C2CCN(C)CC2)=O)CC(C)O1 n1(CC2CN(C(C(C)N3CCCC3)=O)C2)cc(CC2COC2)nn1 c1(C(N)=O)nccnc1C(=O)NC1CCC1NC(C1CC(F)(CO)C1)=O C1(CCNC(=O)CC(F)(F)c2ccccc2)CN(C(C23CC2C3)=O)CCS1(=O)=O CCCC(C)(O)CC(=O)N1CCC(C=CC(=O)NC(C)CCCCO)CC1 c1(C2C(CN(CC(c3ccco3)O)C)C2)ccccc1Br N1(C(CSCC#C)=O)CCCCCC(NC(c2cc(C(=O)NC)ccc2C)=O)C1 C12(NC(C(c3cn(C)nc3)=O)=O)CC1CN(C(c1ccncc1C1CC1)=O)C2 C=C(C)CC(=O)N1CCC(n2cc(CNC(C3CCCN3C(C)=O)=O)nn2)C1 c1(NCC2(CN(C)C)CCCC2)ccc(S(=O)(=O)NCC2CC23CC3)c(Br)c1 C1(NC(C(CC)C)=O)CCN(C(=O)CCNC(=O)OCCCO)CC1(C)C c1(C(N(CCNC(c2cnc(Cc3ccccc3)s2)=O)CC)=O)cccc(O)n1 CC(F)(F)C(C)(C)CC(=O)Nc1ncc(C(C)(C)C)s1 c1(CNC(=O)CC2COCCN2C(C2CCCS2)=O)cc(Br)ccc1F C#Cc1c[nH]nc1C(=O)NC(C)(CNC(=O)Cc1csc(COC)n1)C1CCC1 N1(C(c2ccc(C(=O)OCC)cn2)=O)Cc2nnc(C)n2CC1C(=O)OC c1(C(=O)NC(CCN(C(c2c(OC)nn(C)c2)=O)C)C(C)C)cc[nH]c(=N)c1Cl CS(=O)CCC(=O)NCCC1CN(C(c2cc(C(F)F)[nH]n2)=O)CCO1 Cc1ccc(C=CC(=O)NCC(C)(C2CC2)NC(c2coc(CO)c2)=O)s1 C(CC(CNC(C1(F)CC1)=O)NC(=O)CC1CCC1)OC CC1=C(c2cc(C(=O)Nc3cccc4[nH]ccc34)c3cc[nH]c3c2)CCCC1 n1(CCCONC(C2C3CN(C(CCN)=O)CC32)=O)nc2n(c1=O)CCCC2 c1(OC)ccc(C(=O)NCCCC2(NC(c3ncc(Cl)cc3F)=O)CC2)c(F)c1 C#CCC(CC(=O)NCC1CCCCN1CC)NC(=O)CCc1ccncc1 C12(C(N(C)Cc3c(C)ccs3)=O)CC3CC(C1)CC(O)(C3)C2 C1(NC(=O)NCC2(CO)COCCN2)CC2(CCC2)C12CCC2 N1(CC(=O)NC(C)C(C)NC(=O)C2=C(Cl)CC2)CCCCS1(=O)=O C1(C(=O)NC2(CCCC(N3CC(C=C)C3)=O)CCC2)CCOC(CC)C1 c1(CC)ccc(C(C)(C)NC(=O)N(C2CC2)CC2CC3(CC3)C2)cc1 Cc1c(C(N2CCCOC(CNC(C3(F)CC=CCC3)=O)C2)=O)nc2sccn12 N1(C(c2c(C(C)(C)C)ocn2)=O)CCN(C(C2CCC2CF)=O)C(CCO)C1 N#Cc1ccc(CC(=O)NC(C(=O)NCC(=O)N2CCCO2)C2CCC2)cc1 c1(C(=O)NC2CC(CCNC(CSc3cn(C)nc3)=O)C2)cc2n(c1)CCOC2 N1(C(CNC(CCCCC)=O)=O)CCC(C2(NC(C3C=C3C)=O)CC2)C1 CC1(C)C(CO)CN1C(=O)C(F)C1CC(C(=O)Nc2ccc(O)cc2)C1 N1(C(C(=O)NC2CC3CN(C(=O)OCC)C2C3)=O)CCC2(CC1)COC(C)C2 C(=O)(CC(C)(C)C(=O)N1CCCN(C(C2CCC23CCC3)=O)C(CO)C1)OC N1(C(CCC=CC)=O)CCN(C(c2ccc(C(F)(F)F)cc2Cl)=O)CC1CC c1(C(=O)NC2CC(CNC(C3CCCCC3F)=O)C2)cccc2ccnn12 N1(C(c2c(C)onc2Cl)=O)CCC2C(CCCN2C(c2ccnnc2)=O)C1 c1(C(N2C(C(C)NC(c3c(C)ccnc3)=O)CCCC2)=O)cc2ccncc2[nH]1 c1(NC(CC=C)CC(F)F)cc(C)c(S(=O)(=O)N2CCN(C(C)CC)CC2)cn1 c1(-n2c(-c3c(F)ccc(CC)c3)nc(C3CSC3)n2)cc(O)nc2ncccc12 C1(NC(C=C(C)Cl)=O)CC2(C1)CN(C(=O)CC1CCC(C(F)(F)F)O1)C2 c1(C(=O)NCC(CN(C(CSCCN(C)C)=O)C)O)ccc(NS(C)(=O)=O)nc1 Cc1nc(F)ccc1CNC(C1CN(C(=O)CCC(=O)N(C)C)CC1(C)C)=O CCC(CC(=O)N1CCOC(C(=O)NC(C2CCCCO2)(C)C)CC1)CC(C)C C12(C(N3CC(C=C)C3)=O)CC(CO1)N(C(=O)C=Cc1cc(C)no1)C2 CC(C)(CCC#N)C(=O)NC1CC(NC(=O)CCSc2ccccc2)C12CCC2 c1(NC(C(C)C)=O)ccc(C(=O)OCC2CC23CC3(F)F)cc1 C1(NC(c2c(C)oc(C3CC3)n2)=O)CCC12CN(C(c1cn3ccnc3s1)=O)C2 C1(N(C(=O)CCN2CCOC2=O)C)CN(C(=O)CN2CCSCC2)CC1(C)C C(=O)(C(F)(F)C(F)F)N1CC(NC(c2ccn(CC)n2)=O)(COC)C1 N1(CC)N=C(C(=O)NCCC(C)NC(c2cc3c(nn2)CCCC3)=O)CCC1=O n1(CC(=O)NC2CCC2CNC(c2ccc(C3CC3)cn2)=O)cnccc1=O CP(C)(=O)C(O)C(=O)NCC1CCN1C(c1cncc(NS(C)(=O)=O)c1)=O c1(NC(CCSCC)C)nc(-c2ccsc2)oc1C C12(C(=O)NC3COCC3n3cc(CCCCO)nn3)CC3CC(C(=O)N1)C2C3 CCC(C(=O)N(CCCNC(c1ncc(F)c(OC)n1)=O)C(C)C)C(C)C C1(CN(C(=O)Cc2cccnc2)C)C2CN(C(=O)CCCC3CCCCC3)CC12 C(c1ccc(C(=O)OC(C)(C)C)cc1)=CC(=O)NC(C#CC)(C)C c1(N(C(=O)CC(c2ccccc2)N2CCOC2=O)C)ccc(I)cc1 c1(C(=O)NC2CC(N(C(C=C(COC)C)=O)C)C2)c(Cl)ccc2c[nH]nc12 Cc1nc2ccc(C(N3CCC(C)C3CNC(C3CCC(C)(C)O3)=O)=O)cc2o1 CC1=NC(C)(CNC(C2(CNC(C3CCCCN3C)=O)CCCO2)=O)CS1 CC1CN(C(C2CCCO2)=O)CCCN1C(c1noc2c1CCCC2)=O c1(CC)ncc(C(=O)N(C)CC=CC(=O)NCCC2CCC(C)C2)cn1 C(C(=O)N1CC2C(NC(=O)CN3CCCS3(=O)=O)C2C1)(C(C)C)OCC(C)C N1(C(=O)NC(c2ccc(OCC)cc2)COC)CCC2(CC1)COCC(=O)N2 C(=O)(C(CCC1CC1)NC(C1CC(C#N)(OC)C1)=O)NCC(C(=O)NC)OC CCC(CC(=O)NC(CNC(c1ccc(OC)s1)=O)CCOC)C1CC1 C(CCCCCN=c1nc(OC)c(F)c(C)[nH]1)NC(C(CCCOC)C)=O N1(C(C(CCC)(C)C)=O)CCC(C2CCN(C(c3c(F)cc(F)cc3Cl)=O)C2)C1 CC1C(C)N(C(c2cc(C#N)ccc2O)=O)CCN1C(c1ccoc1)=O Cc1nc2cc(CNCCC3CCCN3)ccc2s1 C=CCCC(C(=O)NC(C)CCOC)NC(c1cc(C)c[nH]1)=O N1(C(C=CCC(C)(C)NC(C2CC3CC(=O)C2O3)=O)=O)CCC2CCC(C1)S2 N1(C(c2cc(CC)no2)=O)CCC2CCN(C(=O)CCC(CC)CCC)CC12 C1(NC(c2n(CC#C)cnn2)=O)CN(C(C23CSCC2C3)=O)C2(CCCC2)C1 N1(C(C(CC2CCC2)NC(C2CC(O)C(F)C2)=O)=O)CC=C(CO)CC1 Cc1cnccc1C(=O)NCC1CC1NC(c1n[nH]cc1Cl)=O c1(C(=O)NCC(=O)NCC2OCCN(C(C3(C)CC3)=O)C2)ccc(Cl)c(Cl)c1 CC(CNC(=O)NC1C(NC(=O)OC(C)(C)C)C1)S(C)(=O)=O N1(C(CCN(C)CC)=O)CCN(C(C2C(C)C2C)=O)CC(C)(C)C1 Cc1ccc(C(=O)NC(C)C(C(C)C)NC(C2COC2)=O)cc1NS(C)(=O)=O O=C1CN(C(C2CC2C2CCCNC2)=O)c2cc(Br)ccc2N1 C1(NC(C2CCN(C)C2)=O)CN(C(c2ccoc2C(F)(F)F)=O)CCC1CO N1(C(C(C2CCC2)OCC)=O)CC2CC1C2CNC(=O)CN(C(=O)COC)C N1(C(CN(C)Cc2ccccc2)=O)CCC(NC(c2c[nH]c(Br)c2)=O)C(F)C1 c1(C(N2CCCC(O)(CCNC(=O)C3=CCCOC3)C2)=O)ccnc2[nH]nnc12 c1(C(=O)NC(C2CCN(C(CCC3(C)CC3)=O)C2)(C)C)cc2occc2n1C C1(NC(C2(C)CC(NC(c3cn(C)c(=O)n3C)=O)C2)=O)CCC=CCCC1 c1(SC)ccc(OC(C)C(N2CCC(C)(NC(=O)CNc3nccs3)C2)=O)cc1 c1(C(C)=O)nc(N2CCC(NC(c3ncoc3CC)=O)C(F)C2)c(C)c(Cl)n1 N1(C(CCOC)=O)CC(C)CC1C(=O)NCC12CC(CN1C)C2 C1(C(N(CCCCN(C(c2c(C)cnnc2O)=O)C)C)=O)CCN2CCCC2C1 c1(OC)cccc(NC(C2(C)CCN2C(=O)C(C)(C)OC)=O)c1Cl n1(CC(=O)NC(CCC)CNC(c2ccc(=O)oc2)=O)cc(C)ccc1=O Cc1n[nH]c(C)c1CNC(=O)CC1CCCN1C(=O)C1=NOCC1 C#CC1(C(=O)NC(C)C(C)CO)CN(C(=O)C=Cc2cnn(C)c2)C1 C12(C(=O)NCCc3cnco3)CCN(C(c3cnccn3)=O)CCC1C2 c1(OC)cccc(Cl)c1CN=C(NC1CCCC1)NC1CCCC(F)C1 CC(O)C(C(=O)N1CC(CNC(c2cc(C(F)F)no2)=O)C1)N(C)C c1(C(=O)NC2C(C)CCN(C(=O)CCC3CCC3)C2)cccc2cnnn12 O(NC(=O)CC(C(C)(C)C)NC(C1(O)CCOC1)=O)CC1(C)CCC1 n1(CC)nc(C)c(C(=O)NC2CN(C(=O)C(O)CC3CC3)CC2SC)c1C C1(NC(C2COCC(C)O2)=O)CN(C(=O)CCc2ccsc2)CC12CCCC2 N1(C(C2(C(CC)=O)CC2)=O)CCCC(CC(F)F)C1C(N1CCCC(O)CC1)=O C(c1ccc(Cl)cc1Cl)=CC(=O)N(C1CN(Cc2ccc(C#N)cn2)C1)C c1(NC(CN2CCCN(CC)CC2=O)=O)cccc2[nH]nc(O)c12 C1(CNC(C(C)=C(CC)C)=O)C2CCC1CN(C(C1CC13CCSCC3)=O)C2 c1(C(N2C(C)C(NC(c3cn(C)c(=O)cn3)=O)CCC2)=O)cc2sccc2n1C C(=O)(C(C)(C)CCCN)C(=O)C(F)OC(F)(F)F.CN1CC(CN)CC1=O C1(C)(C(=O)NCC2(F)CN(C(Cn3cc(C(C)=O)nn3)=O)C2)CCCCC1C CC(C)C(C(C)NC(=O)CN(C)C(c1cccs1)=O)NC(c1nn[nH]c1Cl)=O C1(NC(C2(CC=C)CCOCC2)=O)CCN(C(C2C3CC4C(C3)C24)=O)CC1(C)C C(=O)(C1=CCCC1(C)C)NCCC1(C)CCN(C(C(C)C(F)F)=O)C1 C(=O)(CC(CC)C(C)C)N(C1CCN(C(=O)Cc2cc(OC)ccc2F)C1)CC C(=O)(CCCC(F)(F)F)NC(C)CC(C)NC(=O)C(C)(C)CN1CCOCC1 Cc1nc(C)n(CC(=O)NCC2CC2CNC(C23CC(C)(C2)C3)=O)n1 S(=O)(=O)(c1ccc(Cl)c(F)c1)NC(COC)C(C)C N1(C(C2(NC(c3ccc(CC)o3)=O)CC2(C)C)=O)CCC2(CNC(=O)C2)C1 C1(O)(C(C)C)CCCN(C(=O)C(C2CC=CCC2)NC(=O)CCn2cncn2)C1 N1(C(C)=O)CCC(C)(C(=O)NCCCCNC(C2CCOC2C(F)(F)F)=O)CC1 C(=O)(C1=NOCC1)NC1CC(CC(=O)NC(C#C)CC)C1 c1(OC)cc(C(=O)N(CCCNC(C2CC(=O)N(C(C)C)C2)=O)C)ccc1C#N C(=O)(C#CC1(C)COC1)N1CC(OC)C(NC(=O)CCc2ccncn2)C1 C1(C)(C(=O)NC2C(NC(c3scc(C)c3)=O)CCC2)CC(C(F)(F)F)=NO1 N1(C(Cn2nnc(C)n2)=O)CCCC2CN(C(C3CCC(F)CC3)=O)CC12 Cc1cc(C)n(C(C)C(N2CCC(CC(N3CCOCC3C3CC3)=O)C2)=O)n1 c1(CC)nc(C)ncc1C(=O)N(C)CCN(C)C(c1csc(COC)c1)=O N1(C(c2ccc(C(C)(F)F)cc2)C(=O)NC(CC)C)Cc2cnc(CC)nc2C1 N#Cc1cc(CN2CCOCC2C(=O)Nc2ccc(F)c(Cl)c2)ccc1Br c1(C(=O)NC2C(OC)CN(C(=O)C(O)CC(C)C)C2)cccc2ccsc12 C1(OC)CC2(C1)CC(C(N1CCC(CNC(=O)CCSC(F)(F)F)CC1C)=O)C2 Cc1cnc(NCC2(O)CN(C(c3cc(C(C)C)oc3C(C)C)=O)C2)nc1O c1(N2CC3CC(NC(c4n(C)ncn4)=O)C3C2)ncc2c(n1)CCOC2 C1(CNC(C2CCC(=O)O2)=O)CC(F)CN1C(=O)CC1CCC(C(F)(F)F)O1 c1(-c2ccc(-c3ccc(C(N(CC(F)(F)F)C)=O)cc3)cc2)cccc(C#N)c1 N#CC1(C(=O)NCCC(O)CNC(=O)CCSc2ccc(F)cc2)CCCOC1 CC1CCN(C(=O)C(C)(C)C(N)=O)CC1NC(c1cc(F)c[nH]1)=O C12(C(=O)NCC3N(C)CCN(C(c4n[nH]cc4Cl)=O)C3)C3CCC(CC13)C2(F)F c1(C(=O)NC2C(C(N3CCC(C#CC)C3)=O)CCOC2)cccc2[nH]ncc12 C12(CC(=O)NCCn3cc(CNC(c4cc[nH]n4)=O)nn3)CCC(CC1)C2 c1(CNC(C(C)(C)OC)c2ccccc2)ccc(NC(C)=O)cc1 c1(C(N2C(C3(NC(C4CCCN(C)C4)=O)CC3)CCC2)=O)cccc2cn[nH]c12 c1(C(=O)NC2CCN(C(c3ncn(CC)c3)=O)C(C)C2)ccc2[nH]ccc2c1 c1(C(N2CC3C(CNC(C4OCCN(CC)C4)=O)C3C2)=O)cncc2ccsc12 N1(C(C2C3CC2N(Cc2n[nH]cc2Cl)C3)=O)CCC2(CC1)OCCc1ccsc12 C1(NC(CC2(C)CCN(C(C3(C(C)C)CCC3)=O)C2)=O)CC2C(C1)C2(F)F C(=O)(CCCN=[N+]=[N-])NC1CCC(C(=O)NCc2c(COC)noc2)CC1 c1(C(=O)NC2CN(C(C(=C)F)=O)C2)cnc2ccoc2c1 C(N=c1cc[nH]cc1C#N)C1(NC(C(C)CC(C)(C)C)=O)COC1 C=C(Cl)CCCN=c1cccc(S(=O)(=O)NCC(c2csc3ccccc23)O)[nH]1 C=CC1(C(=O)NCC2(C)CCOCC2)CCN(C(=O)C(C)COC)CC1 C1(NC(c2cnc(CC)[nH]2)=O)COC2(C1)CN(C(c1nc3ccccc3[nH]1)=O)C2 C#CC1CN(C(C2CC2(C)CC)=O)CCN1C(c1[nH]nnc1C(F)F)=O c1(C(N2C(C(C)NC(C(C)OC)=O)CCC2)=O)cc(Br)c(C)s1 C1(NC(C2CC2(F)F)=O)CN(C(=O)CNS(=O)(=O)C2CC2)CC1C(F)(F)F N1(C(CC(C)(C)C)=O)CC(NC(C2CCCCN2CC(F)F)=O)CC(F)(F)C1 CC(C)C(C#N)C(=O)NCc1cn(CC(=O)NCC2Cc3nccn3C2)nn1 CC1C(=O)NC(=O)CN1C(=O)CC(C(F)(F)F)NC(c1nnsc1N)=O CC(C)C(C)C(C)CC(=O)N1CC(CN(C)C(C2Cc3cc(F)ccc3O2)=O)C1 c1(NC(c2cccc(NC(C)=O)c2)=O)c[nH]c2c(C(F)(F)F)cccc12 c1(-n2c(C3(NC4(C=C)COC4)CCC(=O)N(C)C3)nnn2)sc2ccccc2c1C O=C(CN1C(=O)Cc2ccccc21)NC12CCCC1N(C(c1cncs1)=O)CC2 Cc1ccc(C(=O)NCC2CC(F)(CNC(=O)CC(C)C3CC3)C2)c(F)c1 CC1SCCCC1C(=O)NCCC1(O)CN(C(c2cn(CCCC#N)nn2)=O)C1 c1(C(=O)NC2(CN(C(=O)C(O)c3ccsc3)C)CC2)cn2ccccc2n1 C1(C(=O)NCCC2CN(C(C3(n4cccn4)CC3)=O)CCO2)(CC)CCNC1=O CCCCC(F)C(=O)NC(C)CN1CCN(C(=O)CC(CN(C)C)CC)CC1 c1(C(N(C(C)CNC(c2cnc3[nH]cnc3c2)=O)CC)=O)cnc2[nH]ccc2n1 C(=O)(CCP(C)(C)=O)N(CCN(C(C)C)C(C1CS(=O)(=O)C1)=O)C c1(C(=O)NC2CCC(NC(C3ON=C(C)C3)=O)C2)c[nH]c2cccc([N+](=O)[O-])c12 N1(C(c2c(C)cc(C)o2)=O)CCOCC(CNC(=O)CSc2ccccc2)C1 c1(OC)cccc(OC)c1C(N1CCC(C)(C(=O)NCC2(O)COC2)CC1)=O C1(CNC(C2C=CCC2)=O)CCCN(C(c2cccc(N3CCOC3=O)c2)=O)C1 c1(CC)cccc2c1N(CC(=O)NC1(CO)CCCCC1)CC2 n1(CC)c(C)cc(C(=O)NC2(C)CC(NC(c3cnc(CC4CC4)s3)=O)C2)c1C C1(NC(C(C)OCC(C)C)=O)CC2(C1)CC(CNC(c1ccc(N)c(Cl)c1)=O)C2 c1(OC)ncc(C(N2CCC2CNC(c2ccc(OC(C)C)cc2)=O)=O)cc1Cl N1(C(CC2C(C)(C)OCC2)=O)CCN(C(c2cnc(Cl)s2)=O)C(CC(F)(F)F)C1 N1(C(CCC(=O)NC)=O)CCCCC(CCC(N2CCC(C#N)C2)=O)C1 Cc1ccncc1C(C)(C)C(=O)NCC1CC1CNC(c1ccc(CO)s1)=O C(=O)(C1CCCc2ccnn21)NCC1(CNC(C=Cc2n(CC)ccn2)=O)CC1 C1(N(C)C(C2(CO)CCCO2)=O)CCCN(C(C23CC(C)(CO2)C3)=O)C1 C(CCCS(=O)(=O)NCC(c1ccc(OC)cc1)C(=O)OC)OC CCS(=O)(=O)CC(=O)N1CCC(c2n[nH]c(CNC(=O)CC(C)(C)O)n2)CC1 Cc1nn(C)c(C(F)(F)F)c1C(=O)NC1CCC(C)N(C(=O)CP(C)(C)=O)C1 O=S1CCC(NC(c2cscc2Br)c2nnnn2CC2CCCO2)CC1 N1(C(CCC(C)SC)=O)CCC2(CCC(NC(=O)C(CC)N(C)C)C2)C1 Cc1ccnc(F)c1NC(C1C2CCC(C2)N1C(C1(C(F)(F)F)CCC1)=O)=O C1(C(C(=O)O)F)CCCCCC1.n1(CCCN(C)CC)cc(CNS(N)(=O)=O)nn1 c1(C(N2C3CC(NC(CC(C)OC)=O)C3CC2)=O)cc2c(C(F)F)nn(C)c2s1 c1(OCC)ccc(O)c(C(=O)NCC2COC(CNC(=O)Cc3cscn3)C2)c1 c1(C(=O)NC2C(NC(C(CCOC)C)=O)CCOC2)ccc(C)c(OC)c1F N(C(=NCCN1CCCC1)N1CCC(CF)C1)CC(C)Oc1ccc(F)c(F)c1 C#CC1CCCN(C(C2CCC(C)N2Cc2ccc(-n3cncn3)cc2)=O)C1 CCC(CNC(c1ccccc1OC1CC1)=O)N=c1[nH]nc(CCOC)s1 CC(C)(C)C1=CCN(C(=O)CC(C(C)(C)C)NC(C2CCC3(CCC3)O2)=O)CC1 C1(C(=O)NC2(CNC(c3scc(C(C)=O)c3)=O)CC2)CC1C1CCC1 C1(CNC(=O)C=CC2CCCO2)CCCN(C(C2Cc3cscc3C2)=O)CC1 C(=O)(C(CC)C(=O)NCC1CCCC(NC(=O)CC23COC(CF)(C2)C3)C1)OC c1(C(N2CCCC(NC(C3C4CCCOC34)=O)C2)=O)cccc2nc(O)ccc12 CC1CCCCN(C(C23CC2CN(C(c2cc(Br)ccn2)=O)C3)=O)C1 C1(N(C(=O)NC(CNC(=O)OC)C)CCN(C)C)CCCC(C)C1 n1(C(C)C)cnc(C(=O)NCC(O)C(=O)N(C)CC2CC(O)C2)n1 c1(C(=O)NC2C(C)CCN(C(c3cnc[nH]3)=O)C2)cc2ccccc2c(=O)o1 C(=O)(C(C)CC(F)(F)F)N(CCCNC(c1ccc(CCC)cc1)=O)CC c1(C(N2C3C(NC(CCc4ccnc(C)n4)=O)C(C3)C2)=O)cc2nccnc2[nH]1 N1(CC)CCOC(C(=O)NCCNCC(C2(C(=O)OC)CC2C)=O)C1 C1(C(N(CCCOCC)C)=O)(CO)CCN(C(=O)CC2(CO)CCCC2)C1 C1(NC(=O)CC2CCCOC2)CCCN(c2ccnc(C3CCC3)n2)C1 N1(C(COCC(=O)NC)=O)CC(NC(c2cn(C)nc2C2CC2)=O)C2(CCC2)C1 C#Cc1cc(C(N2CCOC(C)(CNC(c3nccn3CC)=O)C2)=O)cc(F)c1 N1(C(C(CC#C)C2CC2)=O)CCC2(C=C(C(=O)N(C3CCCNC3=O)C)C2)C1 c1(NCCOCCN(C)C(C2CC3CC2C2CC32)=O)cnc(C#N)c(C#N)n1 C(CC(C(=O)NCc1cscc1C)NC(C1CC(C)(C)C1)=O)OCC C1(CNC(C2C(CCC)CCC2)=O)CN(C(C2(CSC)CC2)=O)CCC1(C)C c1(NCCOCC(=C)C)[nH]c(=NC2CCN(CC)CC2C)nc2ccc(OC)cc12 c1(NC(C2N(C(C3(COC)CC3)=O)CCC2)=O)ccc(C2=NCCN2)cc1 N1(C(CNC(=O)CNC(=O)CC2CCCC3CC23)=O)CC2C(C1)C2(F)F CC(C)(CC#N)C(=O)N1CCN(CCNC(C2CCCN2C2CCCC2)=O)CC1 O=S(=O)(C1CCCOC1)NCC1C2CCCC12 CCC(C(=O)NCC(CNC(c1cn(C)c2cnccc12)=O)OC)C(C)(F)F CCCC(C(=O)NCC1COC(CNC(=O)C=Cc2sccc2C)C1)N(C)C O=C(C(CCC1CCCO1)N1CCCCC1c1cc[nH]n1)NN1CCOCC1 C1(NC(C(C)(C)OCC)=O)CC(C2CCN(C(=O)Cc3ccn(C(F)F)n3)C2)C1 N1(C(CC(CC)C)=O)CCOC2CN(C(c3cccc(C4CC4)c3)=O)CC12 C1(CN(C(CC2(C(=O)OCC)CCCC2)=O)C)CN(C(=O)CCOC)CCO1 CC1OCCN(C(=O)CCn2ccnc2)C1C(=O)NCCC[Si](C)(C)C C1(NC(CCC(C)CN(C)C)=O)CN(C(=O)CCCCC#N)CC1C1CC1 c1(C(C(=O)NCc2cccs2)N(C)Cc2cncc(Br)c2)cccc(C#N)n1 C1(CNC(C(F)=C(C)C)=O)CN(C(=O)C(c2cccc(C)c2)C)CC(C)(C)C1 c1(CCCNC(C(c2ccccc2)N(CC)CC)=O)ccc(F)cc1OC N1(C(C(CCC)N(C)C)=O)CCN(C(c2ccc(CO)cc2)=O)C(COC)C1 Cc1cnc(NC(C2CC3CC3N2C(C2CNC(=O)O2)=O)=O)c(C)n1 C1(C)(C(=O)NCCN(C)C(c2ccc(-n3ccnc3)cc2)=O)CCCOC1 N1(C(C(C2(O)CCC2)NC(C(CC(=C)C)OC)=O)=O)CC2CCC(C1)C2O CC(C)(F)C(C)(F)C(=O)NC1CCCCC1NC(c1cccc(Br)c1F)=O N1(C(=O)Cn2nccn2)CCCC2(CCN(C(=O)C(C3CC3)C3CC3)C2)C1 N(C1CCCc2ccccc21)CCc1nccc(N2Cc3n(C)cnc3CC2)n1 C(=O)(C1=CCC(C)CC1)C(N(C12CC(n3cc(C4CCC(F)(F)CC4)nn3)C1C2)C(C)(C)C)=O c1(-n2c(CC(=O)NC(CCC)CC(=O)NCC)nnn2)ccc2c(c1)OCO2 C1(NC(c2occc2CN2CC2)=O)CN(C(=O)C(F)=CC2CC2)CC1O C1(N(C(CN2C(C)CC2)=O)CCO)CCN(C(=O)CC(C)F)CC1 C1(O)(CNC(C(C)SC(F)(F)F)=O)CC(CNC(=O)C=Cc2cscn2)C1 c1(C(=O)NCCOCCCNC(c2ccc(Cl)cc2)=O)ccc(O)c(CO)c1 Nc1cc(C(=O)NCCCNC(=O)CNC(=O)CC(F)(F)F)c(F)c(O)c1 C1(C2(O)CN(C(C3CCCCC3C(=O)O)=O)C2)(NC(C2C3CNC(=O)C32)=O)CC1 C1(NC(C(C)N(C)C)=O)CN(C(c2ccc(Cl)cc2)=O)CC12CCCC2 CC1(C(N2CCC(NC(C3CCCO3)=O)CC2)=O)CCCCCCC1 O=C(C1=CC2(CCOC2)C1)NCC1CC(F)(F)CN1c1ccc2nccnc2n1 N1(C(C2(OC)CCCC2)=O)CC2(C)CC1(C(N1CC3CCC3(CO)C1)=O)C2 C(C)(N=c1[nH]c(=NC)[nH]c(=NCC(C)C#N)[nH]1)c1ccc(C)o1 c1(C2C(C)OCC2)nc(-c2ccsc2)nn1C(C)C1CC1 C1(CC)(NC(C2C3COCC23)=O)CCCN(C(C2CC(=C3CC3)C2)=O)C1 C1(CC=C)(NC(C2(C)C=CCN2C(C2COC(C)C2)=O)=O)CCCCC1 C1(CNC(c2cnc(C)[nH]2)=O)CN(C)CCN1C(=O)CSc1ccccc1Cl C#CCCCC(=O)NCC(C(=O)NCCCc1c[nH]nc1C)N(C)C Cc1ccnc(C)c1C(=O)NCC1CN(C(c2ncc(Br)cc2N)=O)CC1C C1(C(=O)NC2(CC=C)CCN(C(c3cc(OC)cnn3)=O)C2)C(C)OC(C)C1C C1(C)(NC(c2cc(CC)sn2)=O)CCCN(C(c2cnn(C)c2)=O)C1 c1(C(N2CCC(CN(C)C(C3(F)CC3)=O)C2)=O)c(F)ccc(Cl)c1F C=CC(CCC)CC(=O)NCCCC1CCCN1C(=O)C(=O)N=S(C)(C)=O C(N=c1[nH]c(=NCCOC2CCCC2)[nH]c2c1SCC2)C1C=CCC1 c1(C(N2CCC3CN(C(CCC(C)OC)=O)CC32)=O)ccc2nc(C)[nH]c2c1 S(=O)(=O)(c1c[nH]ccc1=NC1CCC2(CCC2)C1)NCCC1(C)CC1(Cl)Cl CC1CCC(CNC(=O)Cn2ncccc2=O)N(C(c2csc(S)n2)=O)C1 C(C(O)(C(=O)N1CCCC(CNC(C2(C(F)(F)F)CC2)=O)C1)C(F)(F)F)N(C)C CC(C)CC(C)C(=O)NC1(C)CN(C(C2CC(=O)N(C3CN(C)C3)C2)=O)C1 c1(C(c2nnnn2CC2CC2)NCCNC(c2ccccc2)=O)sncc1Br C1(C(=O)NCC(=O)NCC)CCC(O)CN1C(c1cc(O)ccc1F)=O c1(C(=O)NCC2(C)CCC(NC(=O)C=CBr)C2)nccc2ccccc12 C1(C(=O)NCCN(C(=O)Cc2c(Cl)cnn2C)CCOC)CCCNS1(=O)=O CC1(C)CC2(CC2C(=O)NCC2C3CN(C(c4cc[nH]c4)=O)CC23)C1 c1(C(N2C(C3(NC(c4c(C)cno4)=O)CC3)CCC2)=O)sc2cncn2c1C N1(C(C(N2CC(C=C)C(CC(=O)O)CC2)=O)=O)CCC=C(c2ccncc2)C1 C1(NC(C2C(OCCC)CCCC2)=O)CC2(C1)CC(F)(F)C2 N1(C(CCC(C)OC)=O)CC2C=CC1C(C(=O)NCCCCN=[N+]=[N-])C2 n1(CC)nc(CNC(C2(NC(=O)CC(=O)OC)CCCC2C)=O)c(C)n1 C#Cc1ccnc(NC(=O)NCC2COC(C)(C)O2)c1 C1(C(=O)NCc2ccc(OC(F)F)cc2)CNCC12CCOCC2 C=Cc1ccc(C(=O)N(C)CCN(C)C(c2cccc(C(N)=O)c2C)=O)cc1 CC1C(NC(C2(CC#N)COC2)=O)CCN1C(c1ccc(OC(F)(F)F)cc1)=O C(CC(=O)NC(c1ccoc1)C)(C(C)C)NC(C(=O)NCC)=O N1(c2n(CCCOCC)c(-c3ccccn3)nn2)CCCC(C)(CCOC)C1 C(c1ccnn1C)=CC(=O)N(C(C)CNC(=O)CN1CCOC1=O)CC C1(C(N2CCCC2CN(C)C)=O)(CC)CCCN(C(c2cccc(C)n2)=O)C1 CN1CCN(CC(=O)NC2(CF)CCN(C(C3COCCO3)=O)C2)CC1 C1(C(C)C)CN(C(=O)COc2ccc(F)cn2)CCC1NC(c1nonc1N)=O C(C)(C)(CCC(=O)N(CCCCCC(=O)Nc1cnccc1CO)C)OC c1(OC)ccc(C(=O)NCC2(F)CN(C(c3cc(Cl)cn3C)=O)C2)c(Cl)c1OC N1(C(=O)CC(O)C2CCCC2)CCC2(CC1)CN(C(=O)C(F)(F)C1CCCC1)C2 c1(C(N(C2CCN(C(=O)C(C3CCCC3)OC)C2)CC#C)=O)nccnc1OC c1(C(=O)NCC(C)NC(=O)CC(C)n2cccn2)cccc(N2CCOC2=O)c1 c1(OC)ccc(COCC(=O)NC2CN(C(=O)CNc3nccs3)CC2F)cc1 C1(C(=O)NCc2cnn(-c3cccc(Br)c3)n2)CCCC2(CNC2)O1 N1(C(C(C)OC2CCCCCC2)=O)CCC(C)C(CNC(=O)CSC(=N)N)C1 C12(C(=O)N(CCO)CC3N(C(=O)Nc4ccccc4)CCCC3)CNCC1COC2 c1(C(=O)NCCN(C(c2ncc(C)o2)C)CC)cc(C)oc1C CC1CN(C(c2cn(CC(F)F)cn2)=O)CC2(CCN(C(=O)CCF)C2)O1 c1(C(N(CCN(C(Cc2cc(C)sc2C)=O)C)C)=O)cncc(F)c1Cl N1(C(c2coc(Cl)n2)=O)CCC2(CC1)CC(C(N1CC3OCCOC3C1)=O)CO2 Cc1ccc(C)c(CNC(C2CC(O)(CNC(c3ccccc3Cl)=O)C2)=O)c1 c1(C2(CC(=O)OC)CCC2)ccc(Sc2ccc(Cl)cc2)c(F)c1 N1(C(CC(=O)NCC)=O)CCCC(C2CCN(c3snc(Cl)c3C#N)CC2)C1 c1(C(N(C2CCCC2)CCCNC(C2(CC)CC2)=O)=O)cnc2c(c1)CCCO2 C1(C(=O)NC2(CN(C)C)CC2)CN(C(=O)C(F)C2CC2)CC12CC2 N1(C(C(CNC(C(CC)CN(C)C)=O)O)=O)CCC2(CCC(OC)C2)C1 C(=O)(C(F)(F)C1=CCOCC1)NC1C=CCN(C(c2cncc([N+](=O)[O-])c2)=O)C1 CCC(C)CC(=O)C(=O)NC12CC(C(N3CCSC(C)(C)C3)=O)(C1)C2 C1(NC(c2n(CC)nc(C)c2)=O)CS(=O)(=O)CC1NC(=O)Cc1cc[nH]c(=N)c1 N12CCN(C1=O)C(=O)C2.C(=O)(CCCn1ccnc1-c1ccccc1)NC Cn1c(C(N2CC(F)(CNC(C3CCNC(=O)C3)=O)C2)=O)cc2ccccc12 Cc1cc(C(=O)N(C)CC2(CNC(=O)Cc3ccsn3)CC2)n(C2CC2)n1 n1(CCNC(c2ccc(Cl)cc2)=O)c(O)nc2cc(Cl)ccc12.CC1CC(=O)N1 N1(C(C2C(CCC)C2)=O)CCC2C(C1)CN2C(=O)CCC(CC)CC C(=O)(C1Cc2ccc(Cl)cc21)NC(C1CN(C(c2c(C)ccc(OC)c2)=O)C1)C N1(C(CCC=C)=O)CCCCC1C(=O)NCC1CNC(=O)C1 Cc1csc(C(=O)N(C2CC(NC(c3ncn(C)n3)=O)C2)C)c1Br c1(CNC(C(=O)N(C(C)COC)CC=C)=O)ccc(N2CCN(C)CC2)nc1 C1(NC(C=CC(C)(C)NC(C=CCOC)=O)=O)CCCN(C)CC1 C(=O)(CCCS(C)(=O)=O)N1C(C)C(NC(C2CC(N(C)C)C2)=O)CCC1 c1(C(=O)NCC2N(C(CSc3nc(C)[nH]n3)=O)CC=C2)cc(F)ccc1Br CCC(C)C(C(=O)N1CCC(OC2CCCC2)CC1)c1ccccc1 C1(CC=C)(NC(C2CC(F)(F)C2)=O)CCCN(C(=O)CC2CCOC(C)(C)C2)C1 C1(CNC(C(C)=CC)=O)CC2(CCC2)CN1C(=O)C(CC=C)C(C)C N1(C(c2c(CSCC)cccc2)=O)CC2CN(Cc3[nH]c(C)cc3C)CC2C1 c1(OC)ncc(C(=O)Nc2cc(O)nc(-c3ccncc3)n2)cc1C(N)=O c1(CC)nn(C)c(Cl)c1C(=O)NC1CC(n2cc(-c3cccnc3F)nn2)C1 S(=O)(=O)(c1c[nH]c(C(=O)NC2CC(NC(C3CCC4C3C4(F)F)=O)C2)c1)N(C)C c1(C(=O)NC2CC(C)(NC(c3c(C)n[nH]c3C)=O)C2)cc2n(n1)CC(C)NC2 c1(C(=O)NCc2c(C)ccc(Br)c2)ccc(C)c(O)c1O c1(CCC(N2C(c3cn(C(C(=O)OCC)C)nn3)CC2)=O)ccc(Br)c(C)c1 Cc1ccc(C(N2CCC3CN(C(C4CC(=O)NC4(C)C)=O)C3C2)=O)c(F)c1F n1(CC(=O)NCCCN(C(CCCOCCC)=O)C(C)C)ccc(O)nc1=O c1(C(N2CCC(C(C)NC(C3CC(O)(CC#C)C3)=O)C2)=O)ncc[nH]c1=O N1(C(c2cnc(C)[nH]2)=O)CC2CC(NC(C3NC(=O)CC3C)=O)CC1C2 C1(NC(C2N(S(C)(=O)=O)CCC2)=O)CC(F)CN(C(C2C3CC4C(C3=O)C24)=O)C1 c1(CN2C(c3ncc(-c4n(C)ncc4)[nH]3)CCC2)cncnc1Br C1(C(N2CCC(NC(c3nc(CC)oc3)=O)C(CC)C2)=O)CCc2ccnn2C1 Cc1cnc(C(=O)NCc2cc(I)cc(F)c2F)c([N+](=O)[O-])c1 CC1CCN(C(=O)COc2ccsc2)C1CNC(=O)Cc1cccc(C2CC2)c1 N1(C(C2(C(C)(F)F)CCC2)=O)CC2(CNC(=O)CCn3ccnc3)CC1CO2 c1(C(CN(C(=O)C(=O)OC(Cc2c(C)nc(SC)s2)=O)C)=O)c(F)cccc1F C(C)(CCC(=O)NC1CCOC(CNC(c2cnc(C)n2C)=O)C1)SC [N-]=[N+]=NCCCCCCNC(=O)CCN(C(C1CCC(F)C1)=O)C1CC1 c1(OCCCCCC)c(CN=C(NCC2(CF)CCC2)NCC)cccc1C c1(CNC(=O)NC2CCN(C(=O)OCC)C2)cn(C)c2ccccc2c1=O CN1CCCC(C(=O)NC2(CCNC(c3cn(C)nc3O)=O)CCCC2)C1 c1(C(N2CC(O)(C(C)NC(CSCCOC)=O)C2)=O)cccc(F)c1C1CC1 CN1CC(=O)N(CC(=O)NCCC2CN(C(c3cc(F)cs3)=O)CCO2)C1=O c1(CC)onc(C(N2CCC(O)(CNC(c3cccn3CC3CC3)=O)C2)=O)c1C C12(CNC(c3c(C)nc[nH]3)=O)CCCC1CCN2C(C1CCc2nn[nH]c2C1)=O c1(OC)ccc2c(C)c(C(=O)NCC(C)NC(c3coc(C(F)F)n3)=O)[nH]c2c1 C(=O)(C1=C(c2ccc(F)cc2)CCC1)Nc1c(Cl)ccc(CC)c1 c1(OCC)oc(C)nc1C(=O)N(CCC(C)NC(c1cccnc1)=O)C N1(C(C(C)SCC)=O)CC2C(CNC(c3ccccc3C(N)=O)=O)C2C1 C1(C)(C(=O)NC(CC)CNC(c2cnn(C)c2Br)=O)CCCC1(F)F c1(-n2cc(C3C(NC(=O)C(C)CC#N)C3)nn2)cccc(Cn2c(C)ncc2)c1 C1(NC(C2C(C(N(C3CCN(C4CC4)C3)C)=O)CCC2)=O)CCOC1(C)C C(=O)(C1=CC2CCCCCC12)N1C(CCNC(=O)CCc2ncc[nH]2)CCCC1 c1(C(N(C(C)CCNC(C2CC3(CC3)C2)=O)C)=O)ccc2c(c1)CCCC(=O)N2 c1(C(CNC(C2(C)C(C(=O)OCC)CC2)=O)O)ccc(C(C)(C)C)cc1 C1(NC(c2c(C)nc(CC(C)C)o2)=O)CC2CC1N(C(C1(S(C)(=O)=O)CC1)=O)C2 N1(C(CC2(CC(=O)OC)CC2)=O)CC2CC(N(C(=O)CNS(=O)(=O)NC)C)C1C2 C1(N(C(=O)Cc2ncc(Cl)s2)CCNC(c2ncccn2)=O)CCCCCC1 C1(NC(C(CC)CC2CCCCC2)=O)CC2(CCN(C(=O)Cc3cnsc3)C2)C1 C1(CC=C)(C(=O)NCC(C)(CO)NC(=O)C2CC2)CCOCC1 c1(C(N2CC3(C(NC(CCCCC#C)=O)CC3)C2)=O)cccc2occ(Br)c12 C1(OCC)CC(N=c2[nH]c3c(c(=NCCS(C)(=O)=O)[nH]2)CSC3)C1 c1(C(=O)NC(CNC(c2[nH]cc(C(C)=O)c2)=O)(C)C)cnc(C(C)(C)C)nc1 C1(C(N2CC(CNC(c3cc(C4CC4)n(C(F)F)n3)=O)C2)=O)CCC2CCC(=O)N12 c1(C(=O)NCCN(C(=O)CC2CCCCN2C)CC)ccc2c(c1)CCC(C)N2 c1(C(C)=O)cc(CCC(N2CC(NC(=O)COC3CCCC3)C(O)C2)=O)oc1C CC1CCCN(C(=O)CC(O)C2CC2)C1CNC(c1cnn(CC(F)F)c1)=O CS(=O)(=O)CCC(=O)NC12CC1CN(C(c1cc3occc3s1)=O)C2 N1(C(c2c(C)n(C)c(C(C)(C)C)c2)=O)CC2=C(C1)CN(C(C1C3COCC13)=O)C2 c1(C(N2CCN(C(c3c(OC)cc(O)nc3)=O)C3C2C3)=O)ccc([N+](=O)[O-])nc1 CN1CCC2CN(C(c3ccc(C(=O)NCc4cnn(C5CC5)c4)s3)=O)CCC12 C1(C(=O)NC(CC)C(=O)NC)(C(C)C)CCN(C(c2nnccc2C)=O)C1 C1(C(N2CCC(CC#C)C2)=O)CCCCC1CNC(=O)CCCC=C C1(C(N(C2C(C)CC2)C)=O)CCC(NC(C2CCC2C(C)(C)C)=O)C1 c1(C(=O)NC2(C)CN(C(=O)C(F)(Cl)c3ccccc3)C2)ccc(C#N)c(F)c1 C1(NC(C(C)OCCOCC)=O)CC2C(NC(=O)C(C)(C)Cl)C2C1 Cc1cccc(C)c1C(O)C(=O)NC1COCCC1NC(c1cnc(Cl)[nH]1)=O C1(CC(=O)NCCCN(C(c2ccnc(F)c2OC)=O)CC)CC(C)(C)CCO1 CC1(C2(C(=O)NC3C=CC(CC(N4CC(O)(c5cc[nH]n5)C4)=O)C3)CC2)CC1 C1(C(=O)NC(CNC(C2(C=C)CCC2)=O)CC(C)C)CCc2nnnn2CC1 c1(CC)n[nH]c(CC)c1CC(=O)NC(CNC(C1COCCO1)=O)C(C)C O=C1CC2C(CCCN2C(C2(CF)CCN(C(c3ccc([N+](=O)[O-])o3)=O)C2)=O)N1 N1(C(CC2CC(C)C2)=O)CCCN(C(c2ccc3c(c2)CCC3)=O)C(C)C1 c1(C(=O)O)ccccc1-n1cc(C(N2CCOCC2CSC2CC2)=O)nn1 CC1CCN(C(c2cccnn2)=O)C1C(=O)N(C)OCC(F)(F)F.CCO C(=O)(CCCS(N)(=O)=O)NC1C(CNC(CC2ON=C(C)C2)=O)CC1 C1(NC(c2c(N)cc(Cl)cc2F)=O)CN(C(=O)C=C(Cl)Cl)C2(CCCC2)C1 CC(O)C(C)C(=O)NCC1(CNC(c2ncnn2C2CCOCC2)=O)CCC1 O=C1CCc2cc(C(N3CCn4c(-c5cccnc5)nnc4C3)=O)cnc2N1 C(=O)(C#CC1CCCO1)NC1(CC=C)CCN(C(C2(SC)CC2)=O)C1 N1(C(c2ccc(C(=O)NC)cc2)=O)CC2CN(C(C3CC(O)C3)=O)CC2C1 Cc1nc(C(N2CCC(C(=O)NC(C)CN(C)C(C)C)(C(C)C)C2)=O)cn1C c1(C(=O)NC(C(C(C)C)C)CNC(=O)C=CC2CC2)cc2ccccc2c(O)n1 C(=O)(C(C)C(=O)N1CCC(CCNC(c2oc(C(F)F)cc2C)=O)C1)OC c1(N(CC(=O)NCCOC2CN(C(C=CCCC)=O)C2)C)nnc(C)n1C c1(CC(=O)NCC(CCOC)NC(C2(CCC)CC(=O)C2)=O)ccc(OC)cn1 C12(CNC(C3(CC)CC3)=O)CCC(NC(C3CN(C)CCO3)=O)(CC1)CO2 c1(C(N2CCC(NC(=O)CC)CC2)C(=O)NCC(=C)C)cc(Br)nn1COC C1(C(=O)NCC2(O)CCN(C(C3CC(=C4CC4)C3)=O)CC2)CCCCC1C1CC1 C1(NC(CC2CC(=C)C2)=O)CN(C(c2c(C)cccc2Br)=O)CC12CCC2 C1(C(=O)NC2CC(=O)N(C)C2=O)CCN(C(=O)CC2(C)CCCCC2)C12CCC2 C12CCN(CCC1(F)F)C2.c1(-c2cn(C3C(SC)CCC3)nn2)sc(C)nc1C c1(C(=O)NC2CC(C(=O)NCC(C(=O)OC)C)C2)cnn2ccccc12 Cc1cccc(C)c1CNC(=O)CC(C(C)C)NC(C1(C)CC1(F)F)=O N1(C(C(C)SC(F)(F)F)=O)CCCC12CCN(C(=O)CC1CCC1)C2 c1(C(C(=O)NCCOCC)N(CCCCCCCC)C)ccc(Cl)c(Br)c1F N1(C(Cc2c(C)occ2)=O)CC2CCC(C1)N2C(=O)Cc1cccc(C(N)=O)c1 c1(OC)ccc(C(=O)NC2CCN(Cc3ccc(C)nc3)CC2F)c(C)c1C CS(=O)CCC(=O)NCC1CCN1C(c1cc(N2CCOCC2)ncn1)=O CC1(C(=O)Nc2nc(C(N3CCCN(CCO)CC3)=O)co2)CCC2CC2C1 CC(C)C(C)CC(=O)NC1CCN(C(C2CC=CC(O)C2)=O)CC1CO Cc1nn(CC(N2CC(C(C)NC(c3nc(Cl)oc3C)=O)C2)=O)c(C)c1Br c1(OC(C)C(N2CC(C)(C(=O)NCCN3CCN(C)CC3)C2)=O)ccc(F)cc1 Cn1cnc2cncc(C(=O)NCC34CC3CN(C(=O)CC3CCCOC3)C4)c12 c1(NC(C(c2ccc(SC)o2)N(CC(C)(C)OC(C)C)C)=O)ccc(F)cc1 C1(C(=O)NC(C2CCCCC2)C2CCCO2)CC12CCC2=O CCC(CC)CCC(=O)NCC1(NC(=O)C(n2cc(C)cn2)C)CC(OC)C1 c1(CC(C)C)ccc(C(C)NCC2(NC(=O)OC(C)(C)C)CC=CC2)cc1 C1(=CC(=O)NC(CNC(C(C)CC(F)F)=O)(C)CO)C(=O)Nc2ccccc21 CC1CCC(CCNC(C2(NC(=O)CN3CC(C)(C)C3)CCCC2)=O)C1 c1(C(C(=O)NC2C(C)CN(C(=O)Cc3cnc[nH]3)C2)=O)ccc(F)c(F)c1 N1(C(Cc2ccc(C)s2)=O)CCC2(CC1)CC(NC(=O)C(Cl)(Cl)Cl)CO2 N1(C(COC)=O)CCc2cc(C(=O)Nc3cc4[nH]c(C)cc(=O)n4n3)ccc2C1 C=CC(CC)CC(=O)N(CC(O)CN(C)C(c1cccc(OC)c1)=O)C C(=O)(CCCC(F)(F)F)NCC1CN(C(C2C(OC(C)(C)C)C2)=O)CC(F)C1 C#CC(CNC(C1(N(C(=O)C=C(C)C(C)C)C)CC1)=O)CC C(=O)(C1=CCS(=O)(=O)C1)N1CC(CCCCNC(CC(COC(C)=O)(C)C)=O)C1 CC1CC(CNC(c2cnoc2C2CC2)=O)CN1C(c1cccnc1F)=O C1(NC(C(C)=CC)=O)CCN(C)C12CCCN(C(C1(C(F)F)CC(F)(F)C1)=O)C2 CCCCCCCC(=O)NC(C)C(C)NC(=O)C(C)OCCC(C)C Cc1ccc(CO)cc1NC(=O)CC1CN(C(=O)C(C)C2CCC2)CCO1 Cc1cc(C(F)(F)F)ccc1NC(=O)C(=O)Nc1csc(F)c1 n1(C(CC)(C)C)nnnc1C(c1cccn1C)NCC1(CO)CCCO1 C(=O)(CCN(OC)C(=O)c1ccnn1C1CNC1)Nc1c(OC)cnnc1 C(=O)(C(N)C(=O)NCCCOc1ccncc1)OC c1(C(=O)NCc2c(C(NOCC(C)(C)C)=O)c[nH]n2)cc2n(n1)CCO2 c1(C(=O)NC2C(CNC(CC(C=C)C)=O)C2)cnn2c(N)cc(C)nc12 C1(CC)OCCC1C(N1CC(c2ccccc2)(NC(=O)Cc2c[nH]nc2C)C1)=O N1(CCCNC(C=CC=CC)=O)CCN(C(=O)COCc2ccncc2)CC1 N1(C(C2CCCN2CC(F)(F)F)=O)CCN(c2ccc(I)cn2)CC1 CC1c2cccn2CCN1C(C1CC=CC(n2cc(CCO)nn2)C1)=O N1(C(C2C(C)(C)CC2)=O)CC2(CCC(CNC(c3ccnc(C4CC4)c3)=O)O2)C1 C1(C(C)(C)NC(C2CC(N3CCCC3)C2)=O)CCN(C(=O)CCn2cccc2)C1 c1(C(=O)N(CCNC(C23CCC2CC3)=O)C2CC2)cc(Cl)c(Br)s1 N1(CC(=O)NC(CCN(C(C(C)SC(F)(F)F)=O)C)(C)C)CCN(C)CC1 N1(C(Cc2cc(C)[nH]n2)=O)CC(F)CC1CNC(=O)CCc1ccc(F)cc1 c1(C(=O)NC(CNC(c2c(OC)cc(C)s2)=O)(C)CO)n[nH]c2cc(C)ccc12 CC1C(C)S(=O)(=O)CCN1C(C1(N(C)C)COC1)=O.C(C)(C)(C)C(=O)O N1(C(C(C)=CCOC)=O)CC(NC(c2ccc(Cn3ccnc3)o2)=O)CC1CO C(CCN(C)C)(C(=O)NC1C2CCCOC12)NC(COCCC)=O C1(C(=O)NCC2(F)CCCN(C(=O)CN3CC4CC4C3)C2)CCCCC12CCC2 C1(NC(c2ccc[nH]2)=O)CC2COCC(C1)C2NC(c1cc2n(n1)CCCC2)=O N1(C(C(C=C)(C)O)=O)CC2CCN(C(C3(O)CCCCCC3)=O)CC2C1 CCC(CCOC)N=c1nc(N2CCN(C)CC(C)C2)c2c([nH]1)CSC2 N1(C(CCOC(C)=O)=O)CC(C)(CNC(C2CCCCC2O)=O)CC1(C)C N1(C(COCCCC#C)=O)CCN(C(=O)C(O)Cc2[nH]cnc2C)CC1CO CC(CCC(=O)N1CC(CNC(=O)Cc2cc[nH]n2)C(C)C1)S(C)(=O)=O c1(C(=O)NC2CC(F)(CNC(C3CCCC3)=O)C2)c[nH]c2ncccc12 C1(NC(=O)CC2CC(F)(F)C2)CCC2CCN(C(c3c[nH]nc3C3CC3)=O)C1C2 Cc1cc(C(=O)N(C)CC2CCC(NC(=O)C(C)OC(C)C)CC2)c(O)cc1F CC1CCC(NC(c2ccnc(OCCO)c2)=O)CN1C(c1c[nH]ccc1=N)=O c1(CC)ccc(S(=O)(=O)NC(c2cc3ccccc3n2C)C)c(C)c1 C1(CNCc2c(C)nn(-c3ccccc3F)c2)C2CCCCCC12 N1(C(C(CC)C#N)=O)CCC(CNC(c2ocnc2C(F)F)=O)C12CC2 c1(C(=O)NC2C(CC)N(C(=O)Cc3cncnc3)CC2)ncc(Br)cc1C CCC(C)C(O)C(C)C(=O)NCC1(C(=O)NCCCC(C)CO)CCCC1 c1(C(=O)NC2(C(=O)NCCC(CC)O)CC2)ccc(O)cc1 N1(C(C2(SC)CC2)=O)CC2CN(C(=O)C=CCF)CC(F)(F)C2C1 c1(C(=O)NCC=C(C(=O)NC(C2CCOC2)CC)C)cnn(C)c1C#N C1(COC)(CNC(c2cccc(C)n2)=O)CCCN1C(c1csc(O)n1)=O C(=O)(C(C(C)(C)O)NC(=O)C(C)O)N1CCC(CNC(COC)=O)C1 C1(C(N2CCC(OCCNC(c3cc(Cl)sc3Cl)=O)C2)=O)CN2CCC1CC2 Cn1nnc(CNC(C2(C)CCOC2)=O)c1C(=O)NCC1(O)CSC1 C(=O)(C1=CCCCO1)NCC(CC)NC(=O)Cc1ncc(-c2ccc(Cl)cc2)o1 C1(C2(O)CCOCC2)(C(=O)NCCN(C(c2cccc(CC)n2)=O)C)CC1 c1(CC)nnc(N2CC3C(NC(=O)CCC4CCCN4C)C3C2)nc1CC CCC(CC(C)C)C(=O)N1CCC(NC(c2ccc(Cl)c(O)c2)=O)C1 Cn1cnc2nc(N3CCC(C)(OC)CC3)nc(NCCC3CCC3)c12 c1(CNC(C2COC3(CCC3)C2)=O)ccc(C(F)(F)F)cc1Cl CCC(CC(C)C)C(=O)NCCC(C)(C)NC(=O)C(F)n1cccn1 Cc1ncc(C=CC(N2CCCC(CCNC(=O)COC3(C)CCC3)C2)=O)s1 CC(=O)C(C)CC(C)C(=O)N1CC(C)C1C(=O)NCCc1cncs1 Cc1cn2nc(C(=O)NCC3CCC(NC(=O)Cn4cncn4)C3)cc(C)c2n1 C1(NC(CC)CC(C)O)CCC2CCCCC2C1 N1(C(C(CC)O)=O)CC(C)(C)OC2(C1)CN(C(C1(C#N)CC1)=O)C2 N1(C(CCCOC(C)C)=O)CCN(C(C2CCOC2)=O)C2CCC12 Cc1ccc(C(N2CCCC(C(C)NC(C3(c4ncco4)CC3)=O)C2)=O)cc1C C1(NC(C2(C=C)CC2)=O)CCN(C(C2CCC(COC)C2)=O)CC1 N1(C(c2[nH]nc(OC)c2Cl)=O)CCCN(C(=O)CCC2C(=O)NN=C2C)C(C)C1 Cc1cc(NS(C)(=O)=O)ccc1C(N1CCCC1(C)CNC(=O)C(C)N(C)C)=O C1(C(=O)NC2(C)CCC(C)(C)C2)CCN(C(=O)CCC(F)(F)F)CC1(C)C C1(CC(=O)NC)CN(C(c2cnco2)=O)CCN1C(=O)Cc1cncnc1 C=CCC(CC=C)C(=O)NCCC1CN(C(=O)C=C(C)Cl)CC1C N1(C(c2nn(C)c(Cl)c2)=O)CC2CCC(NC(=O)CCOCC(F)F)(C2)C1 N1(CCNC(CC(C)C)=O)CCCN(C(=O)CSc2ccc(F)c(F)c2)CC1 C1(NC(CCN(C(CC)CC)C)=O)CC(CNC(=O)CC2CC=CC2)C1(C)C c1(N2CCC(COC)(NC(c3cnc(OC)cc3C)=O)C2)cc(C)nc(CO)n1 C1(CC(=O)NCCC(C)NC(CC2CCC(C)O2)=O)CC2CCC1CC2 C(C(C(C)(C)C)NC(c1ccc(NC(C)=O)cc1)=O)NC(C1CC(SC)C1)=O CCCCC(C)(F)C(=O)NCCC1=CCN(C(=O)Cn2cccc(O)c2=O)CC1 Cc1cnc(C(=O)NCCN(C(=O)CNC=O)C(C)C)c(F)c1 C1(C(=O)NCc2c(C)cc(C)s2)CN(C(=O)CCOCCN(C)C)CCC1(C)C C(C(=O)NOCC1CCOCC1)(c1ccoc1)NC(CC1(C)CC1)=O N1(C(c2cc(C)[nH]c2C)=O)CCC(CNC(=O)CC2(O)CCCCCC2)C(O)C1 c1(C(N2CC(CC(C)NC(C34CC(OC)C3C4)=O)C2)=O)ccc(=N)[nH]c1 C1(C2CCN(c3nc(OC)nc(OC)n3)C2)(NC(C2N(CC)CCCC2)=O)CC1 CCCCC(CNC(c1sc(C)cc1C)=O)NC(=O)C(F)n1ccnc1 c1(NCC(c2cn(C)nc2)O)ccc(S(=O)(=O)NC(C2CCC2)C2CC2)c(Cl)c1 N1(C(CCn2cc(-c3ccc(C)c(F)c3)nn2)=O)CC2CCCC2(CO)C1 CC1(C)CN(CCO)CCN1C(c1cnc(-c2ccc(C(F)(F)F)cc2)cn1)=O CC1(C(N2CCOCC2CNC(c2cnc(CC(C)(C)C)o2)=O)=O)CC(F)(F)C1 N1(C(c2ccc(OC)o2)=O)CC(NC(=O)CCc2conc2C)C(C2CC2)C1 c1(C(=O)NC2CN(C(C(CC)C)=O)C(C)C2)ccc(F)c2occc12 C1(C=O)(NC(=O)CCOCCCOC)CCC(C)(C)C1.C(=O)(CO)N(CCC)C(C)C C(=O)(C1CC(=O)c2ccccc21)N1C2(COC)CC(NC(C3CCOC3)=O)(C1)C2 Cc1cccc2c1OC(C(=O)NC1CCCC3OCCC13)C2 c1(N(CC(C(C)C)O)C)ncc(S(=O)(=O)N2CCC(CO)C(F)(F)C2)cc1Cl c1(C(N2CC(N(C)C(c3ccc(C(C)(C)C#N)cc3)=O)C2)=O)cc(O)ccc1O CC1CC(NC(=O)Cc2cnns2)CN(C(c2ccc(NCC(N)=O)cc2)=O)C1 C#Cc1cc(F)c(C(=O)NCC(CNC(C2C=CCCC2)=O)CO)cc1F Cc1cnccc1C(=O)NCC1CCN1C(=O)CCc1cncc(Br)c1 C12(CNCC(=O)NCCCC3CCCCO3)CC3CC(C1)CC(Cl)(C3)C2 C(CC1CCCC1)(C(F)(F)F)N(C=O)Cc1cc(-n2cccn2)ccn1 N1(CCN(C)C)CCC(C(=O)NCC(c2ccc(F)cc2)N(C)C)CC1 N1(c2c(S(=O)(=O)N3CCCC(OCC)C3)cccn2)CCN2C(CNS2(=O)=O)C1 C1(C(N(C(CC)C)Cc2ccccc2C)=O)CC2CCC(C1)S2(=O)=O c1(C(N(C)CC2CCCN(C(=O)CSCc3ncc[nH]3)C2)=O)cc(Cl)ncc1O C=CCCCC(C)(C)C(=O)NCC1CCN1C(c1cn(C)nc1-c1nccs1)=O C1(CC=C)(NC(c2ccn(C)c2)=O)CCN(C(=O)C=Cc2cnc[nH]2)C1 C(=O)(C(C)S(N)(=O)=O)N1C(C2CCCN(C(CC(C)(C)OC)=O)C2)CCCC1 C(=O)(CC(C)CC(C)C)N(CCC(C)NC(Cn1nc(C)oc1=O)=O)C C1(CC)CCN(C(c2cn(C3CC3)cn2)=O)C1C(=O)NCc1ccc(Cl)cn1 c1(C(=O)NC)c(NC2CC(CNC(=O)OC(C)(C)C)C2)csc1C n1(CCC)nc(C)cc1C(=O)NC1CCCCC1NC(=O)C=CBr c1(NCCN(C(CC)C)C)cc(N2CCCC(NC(=O)C(C)C)C2)ncn1 Cc1ccc2c(c1)CC(C(=O)NCCOC1CCN(C(=O)CCCCCO)C1)O2 c1(C(N2CC(CNC(c3ncc(Cl)cc3F)=O)OCC2)=O)cc2ncccn2n1 C1(NC(C(C)=C2CCC2)=O)CC(C)CN(C(c2ccc(CO)o2)=O)C1 n1(CC)nc(C)cc1C(=O)NCC1CC1C(=O)NC.C1(=O)CN1 C1(NC(C(C)NCC=C)=O)CC(Oc2ccccc2)C1(C)C O=C1CCOC(C(=O)NC(C(=O)NCC2(CO)CC=CC2)C2CC2)C1 c1(CC)cnc(C(=O)NCC(C)=CC(=O)NCCC(C)N(C)C)nc1 C(c1ccc2occc2c1)=CC(=O)NC1CC(C)(NC(c2cnc[nH]2)=O)C1 N1(C(C2N(C)CC(F)C2)=O)CCC2CN(C(=O)Cc3nc4c([nH]3)CCCC4)CC12 C1(CC)C(NC(=O)CC2COCC(C)O2)CCCN1C(C1CC(=O)NC(C)C1)=O Cc1nc(C(=O)NC2(C)CC(NC(c3ccc(Cl)cc3)=O)C2)n(C)n1 N1(C(=O)CC2CCC2)CC2CCN(C(C3C=CCCC3)=O)C(C2)C1 N1(C(C2CN(C(CC(COC)(C)C)=O)CC2(F)F)=O)CCOCC(C2CC2)C1 CC(CCC(=O)NCC1CCCCN1C(=O)C(C)(C)C1CCOCC1)N(C)C C(=O)(CC(O)(C(F)(F)F)c1ncc[nH]1)N(CCCCCC)CC C(=O)(C1=CC(O)C(NC(=O)C(C(C)(C)C)OC)C1)NCC(CC)(C)C N1(C(c2c(C)scn2)=O)CC2CC1C2C(N1CCC(c2ccccn2)C1)=O Cc1cccc2c1OC(C(=O)NC1C=CC(CNC(C34CCC(CC3)O4)=O)C1)C2 CC(C(=O)N1CCC(NC(=O)CN2CC3CC3C2)C1(C)C)C(F)(F)F CCCCC(C(=O)NCCN(C(=O)CCN(CC)CC)C1CC1)C(C)C N1(C(c2cc(COC)sc2)=O)CCC(NC(=O)CC2CCCN2C(C)=O)CC1 CC(CC(=O)NCC(CNC(c1cc(C2CCC2)on1)=O)CO)n1cccn1 C1(C)(NC(c2cnn(C)c2N)=O)CN2CCC1CC2.n12cc(cn1)C(=O)CC2 N1(C(COc2cccc(CC)c2)=O)CCN(C(C2Cc3cscc3C2)=O)C(C)C1 c1(C(N2CC=C(CNC(C(C(C)OC)O)=O)CC2)=O)cnc2ccoc2c1 Cc1nc(F)cc(=NCCc2cccc(C(F)(F)F)c2)[nH]1 S(=O)(=O)(c1cc(NC(c2cc(OCC#C)cc(Br)c2)=O)ccc1OC)NC C1(NC(C2C(NCc3cnc(OC)c(Br)c3)C2)=O)CCc2nc[nH]c2C1 C(=O)(C(CCCC=C)NC(c1ccc(F)cc1F)=O)NC(C#CC#C)(C)C c1(CC(=O)NC(C)CCN(C)C(C2CCC(=O)N2)=O)cnccc1C(F)(F)F C(=O)(CN=c1cc[nH]cc1)N1C2(C(=O)NC)CC(CO)(C1)C2 N1(C(c2cc(C)c(C)s2)=O)CCN(C(C2CN(C3CCC3)C2)=O)CC1C1CC1 c1(CCC)ccc(N)c(C(=O)NCCCNC(=O)CCN(C)CCC)c1 c1(OCC#C)cc(CN2CCCC(C(=O)OC)C2)ccc1Cl Cc1ccnc(C)c1C(=O)NCc1ccccc1CNC(=O)C(=O)NC1CC1 C(=O)(C(C)CCC(C)(C)C)NCC(CC)(C)NC(=O)C#CC1(C)COC1 c1(C(=O)NCC2N(C(c3c(C)cc(SC)o3)=O)CCC2C)cnc(C)c(C)c1 c1(CC)nc(C)oc1C(=O)NCC1(OCC)CN(C(=O)C(C)(C)Cl)C1 c1(C(=O)NC(c2ccccc2)C(C)NC(=O)CC2CN(C)C2)nscc1N C12(C(=O)NC3CCC(C(=O)OC)C3)CCC(CC1NC(=O)C(C)CSC)C2 C(CNC(=O)Cc1cnc(C2CC2)[nH]1)(CCNC(C1CNC(=O)O1)=O)OC N1(C(c2c(CC)nc(C)nc2)=O)CC(NC(c2ccc(N)cn2)=O)CC(C)(C)C1 c1(C(=O)NC(C2CCCC2)CNC(CCC=C(C)C)=O)cc2c(Cl)nccc2o1 c1(C(N2CCC(N3CCN(C(c4c(C)occ4)=O)CC3)C2)=O)cc(N)cc(O)n1 c1(CC(N2CC(C3(NC(CC#N)=O)CC3)C2)=O)c(Br)ccc(F)c1F N1(C(c2ccc(F)s2)=O)CC2CCC1C(NC(C1(c3ccccc3Cl)CC1)=O)C2 c1(SC)cc(C(N2CCCC(C)C2)=O)n(C)n1 c1(C(CO)NC(CNC(=O)CNC(=O)CC(F)(F)Cl)=O)ccc(F)cc1F c1(OC)ccc(C(=O)N(C2CN(C(c3n[nH]cc3Cl)=O)CC2F)C)n2nccc12 C(=O)(C(C(C)C1CCC1)NC(c1cc(C(=O)C(C)C)c[nH]1)=O)OC N1(C(c2cc(F)ccc2F)=O)C2CCC1CC(C(N1CC3CCC1C3)=O)C2 C1(C(N(CCOCC)C)=O)CCC(C)N1C(c1cnn(C(C)C)n1)=O CC1=C(C)CC(C(N2CCCC(NC(=O)CCNC(N)=O)C2C)=O)CC1 Cc1cc(NCc2csc(Br)c2)c(Br)cc1[N+](=O)[O-] C(CCC(C(=O)N1CC2CC1CO2)NC(=O)CC(C)n1ccnc1)OC Cc1cc(N2CCC(C3CCCC3)CC2)nc(=NCCC2CN(C)CCO2)[nH]1 Cc1cc(N)c(F)c(C(=O)NCC2CC2CNC(=O)CCCC(=O)N(C)C)c1F C(=O)(C#CC1CCCO1)N1CC(CCNC(c2c(CC)nn(C)c2)=O)C1 c1(NCC(C)(C2CC2)NC(c2cc(OC)nc(C)c2)=O)ncc2ncn(C)c2n1 c1(C(=O)NCC2N(C(C(C3CCOCC3)OC)=O)CCC2)cnc2nccn2c1 c1(C(=O)NC2C(NC(Cc3nnc(C)o3)=O)COC2)nc(Cl)sc1Br CC1CCN(C(=O)C(C)(C)F)CC1CNC(c1cc(Cc2ccccc2)c[nH]1)=O C(=O)(C(F)Cc1ccccc1)NCC1C(NC(=O)CCC2CCCC2)CC1 C=C(C)C(O)CC(=O)NC(C1CCN(C(c2sc(C)cc2Br)=O)C1)(C)C C(=O)(CC(C)(C)CC(F)F)N1CCC(CC(C)NC(C2CN(C)C2)=O)CC1 c1(C(=O)NC(CNC(C2C(CC)CCO2)=O)(C)C2CC2)occ2c1CCC2 c1(CN2CCC(C(=O)NCC(COC)O)(OC)CC2)nc2cc(Cl)c(F)cc2[nH]1 Cc1cc(CC(N2CC(Cn3cc(CC4CCOCC4)nn3)C2)=O)cc(C)c1 c1(CC)cccc(CC)c1CC(N1CCC(NC(c2cnc(C)s2)=O)CC1C)=O CCCCC(O)C(C)C(=O)N1CCN(C(c2cccc(CO)c2)=O)C2COCC12 CC(C)C(C)(O)CNC(=O)C(Cc1cn[nH]c1)NC(=O)Cc1cnns1 c1(C(C(=O)OC(CC(=O)OCC)C2CC2)F)cccc(F)c1 C1(NC(COCc2ccc(C)s2)=O)CCC(C)N(C(C2CCSC2)=O)C1 N1(C(c2ccc(C(C)C)nn2)=O)CCOC(C)(C)C1CO N(C(=NC)N1CC2CC(C1)N(C)C2)Cc1cc(COc2cccc(OC)c2)on1 C(=O)(C1=Cc2ccccc2C1)NCCC1(C(=O)NC(CC)(CC)CC)CC1 C12(CNC(CC(C=C)C)=O)CC(NC(C3OCCC3C)=O)(C1)C(C)(C)O2 N1(C(C(C(C)C)SCC)=O)CCC(C(F)(F)F)C(NC(=O)CNS(C)(=O)=O)C1 C(=O)(C(C)(C)C1=CCSCC1)NCC1CN(C(Cc2cccc(C)c2)=O)C(C)C1 C#CCCCC(=O)NCC1(C(=O)NCCC(=O)NCC)CCCO1 n1(CCNC(=O)CCc2ccccc2)cnc2cccnc12 N1(C(C=CC(CC)=CC)=O)CCC2(CCCC2CNC(=O)C(C)(C2CC2)OC)CC1 C(=O)(C(CNC(=O)Cc1ncccc1F)C(C)C)NC(CC)CSC CCCCCCC(C)C(=O)N1CC(COC)(NC(=O)C(C)(F)c2ccon2)C1 C1(CNC(=O)NC(c2ccc(I)cc2)(C)C)CCCC1(F)F N1(C(C(C)=C2CC2)=O)CCC2(NC(c3cnc(O)cc3C)=O)CCCCCC12 CN1CCN(C(=O)Cc2ccc(Cl)cc2Cl)C(CNC(C2CC23CC3)=O)C1 C(=O)(C(C)(C)C(F)(F)F)N1CCC(NC(c2[nH]cc(C(C)=O)c2C)=O)C(C)C1 C(CC[Si](C)(C)C)N(C1(C(F)(F)F)CCOCC1)C N1(C(CCC(=O)OCC)=O)CC(C)CN(C(c2cnn(C)c2)=O)CC1C N1(C(c2nc(C)c(C)s2)=O)CCC2(CC2)CC1C(=O)NC(c1ccccc1O)C C1(NC(c2ccc(-c3c(C)c[nH]n3)cc2)=O)CC2CC1N(C(C1CC=CC1)=O)C2 N1(C(c2cc(CC)c(C)s2)=O)CCCCC(NC(c2cc(C)ccn2)=O)C1 CC(CC(=O)NCC1(C(=O)NCc2cncc(F)c2)CCCC1)C(F)F C(C(C)(C)CC(=O)NCC1CCN(C(C2CC(=O)N2)=O)CC1C)OC C1(C(N2CCCCC(CNC(C3CC(OC)C3)=O)C2)=O)CC2(CCCCC2)C1 c1(C(N2CC(N(C(COCCCC)=O)C)C(O)C2)=O)noc2c(F)cccc12 c1(OC)cc(C(=O)NCCCNC(c2cnn(C)c2)=O)cc2cccnc12 CC1CCN(C(=O)C(=O)NC(CNC(c2ncc(C(F)F)s2)=O)CO)C1 C1(NC(C2(CCCC(=O)NCC3(C(C)C)CC3)CCC2)=O)CCC(O)CC1 C12(OC(C(CCC)NC(=O)OC(C)(C)C)=O)CC(CC(C)O1)C2 N1(C(C(c2ccccc2)NC(c2cc(C)nn2C)=O)=O)CC2CC(C)C2C1 N1(C(C(CC(C)C)O)=O)CCn2ncc(C(N3CCNCC34CCC4)=O)c2C1 CC1C(NC(=O)C2CC2)CCCN1C(c1ccc(F)s1)=O c1(C(=O)OC)ccc(C(=O)NC2(CNC(=O)C=C(C)C)CCC2)s1 N1(C(C2(C#C)CCCC2)=O)CCC(F)(CNC(=O)COc2ccc(Cl)nc2)CC1 c1(OCCOC)ccc(CC(=O)N(C2CCN(Cc3ccnn3C)C2)C)cc1 C1(CC)(CC)CC(O)CN1C(C1CC12CCN(C(c1ccoc1Cl)=O)C2)=O C(C(=O)NCC1CC1NC(C1CC1)=O)(C1CC1)SCC c1(C(N2CC(NC(c3c(C)ccnc3)=O)C(F)C2)=O)cccc2c1CCCC2 N1(CCc2noc(C)c2Br)C(=O)NC(C)C(C)C1=O N1(C(c2cc(N)cc(O)n2)=O)CCC2CN(C(=O)CCCNC(N)=O)CC12 c1(C(CCN(C(=O)C(O)CC2CCNCC2)C)O)ccccc1 c1(CNC(N2CC=CC2C(=O)Nc2ncccc2F)=O)ccncc1C(F)(F)F C1(C(=O)NC(CCOC)C(=O)O)CCCC2(CC2)C1 C1(C(=O)NC2(C(=O)NC3(CC=C)CCC3)CC(F)(F)C2)CC12CCCCC2 N1(C(c2c(C)nsc2)=O)CCC(F)(F)C(C(=O)Nc2c(C#N)cnn2C)C1 C(=O)(C1=CC2(CN(C(=O)Cc3cccnc3C)C2)OC1)Nc1ccc(C#C)nc1 N1(C(c2c(N)c(C)n(C)n2)=O)C2CCC1CN(C(c1c[nH]c3ncccc13)=O)C2 O=C1CN(C(C2CC(n3cc(C4CC4)nn3)C2)=O)CC(COCCO)N1 Cc1cc(C(N2CCCC2CCNC(C2CC2c2ccco2)=O)=O)nn1C(C)C c1(NCC(C)N(CC)CC)ncc(C)cc1S(=O)(=O)NCCc1ccns1 CC(C)CCCC(=O)NCC12COC(CNC(=O)C(C)(O)C(C)C)(C1)C2 c1(OC)cccc(F)c1C(=O)NCCCCNC(=O)C(C)C=Cc1ccccc1 C(=O)(C(C)CCCC(C)C)NCCCC(C)NC(CCCC(C)=O)=O Cc1cc(O)c(F)cc1NC(C1CC2CCCC2N1C(C1CC2(CC2)C1)=O)=O Cc1cc(C)c(-c2cn(CCCN(C(=O)CC3CCSC3)C)nn2)cn1 N(C(=NCC1COC2(CCCCC2)O1)N1CCC(F)(F)C2(CCC2)C1)C(CC)C C=CC1(C(N2CCC(C)(C#N)C2)=O)CCN(C(=O)C(O)CN2CCCC2)CC1 C#Cc1cc(C(=O)NC2COCCC2NC(=O)C(CC=C)C(C)C)cc(F)c1 N1(C(C(CC(N)=O)NC(=O)CN2CCCCC2)=O)CCc2nncn2CC1 C1(C(N(C)CC2N(C(CC(C)F)=O)CC(F)C2)=O)CC2(C1)CC(C)(C)C2 C1(CCNC(C(C2CCC2)OCC)=O)(C(=O)NC(C)CCO)CCCC1 C(CCCOC)(C(=O)N(CC(=O)OCC)C)NC(C(CC=C)C)=O CS(=O)(=O)CC(=O)N1CC(NC(C2COCCN2CC2CCC2)=O)C(O)C1 c1(OCC=C)ccc(CN2CCC2C2CCCC2)cc1OC C12(CC=CC1)C(=O)CCC1CC1C(=O)NC2.N1(OC)CC(N2CC(O)C2)C1 N1(C(C(C)c2ccco2)=O)C2CCCC1CN(C(C1CC(=O)OC1(C)C)=O)C2 N1(C(CCCC(CC)NC(CCCC#C)=O)=O)CCC(O)(C2CC2)CC1 C(=O)(CCCN=c1nccc[nH]1)NC1CCN(C(CCCCC=C)=O)C1(C)C c1(C(N2CCCCC(CNC(=O)COCCF)C2)=O)noc2c1COCC2 N(C(=NCC(C(C)C)C(C)C)NC1CCCC1)C1CC(OCC)C12CCC2 c1(N2CCc3c(cn(C)n3)C2)[nH]c(=NCC(Cl)=CCl)nc2sccc12 CN1CCN(C(=O)C2=CCCSC2)C(CNC(=O)CC2CS(=O)(=O)C2)C1 c1(N2CCC(OC)(CO)C2)nc(N(CCC#N)C)c2c(n1)CCOC2 Cc1ccc2c(=NCC3(Br)CC3(F)F)[nH]c(=NCc3ccnc(O)c3)[nH]c2c1 c1(NC(C2N(Cc3cnc(C)[nH]3)CC(F)(F)C2)=O)c(Cl)cc(Br)c(C)c1Cl N1(C(Cc2ccc(C(N)=O)nc2)=O)CCCC12CCN(C(=O)CCCC(N)=O)C2 CC(C)C(C(=O)NCCC(C)CCNC(=O)CC1CCN(C)C1)NC(N)=O c1(C(=O)NC2(CNC(C(C(=O)OC)OC)=O)CC2)cc2nccnc2[nH]1 N1(C(COCC#C)=O)CC(O)C(O)C1CNC(C1CCCN1C)=O N1(C(C(CCSC)O)=O)CC(NC(c2c(Cl)ccc(O)c2N)=O)CC2(CCC2)C1 N1(C(CC(C)(C)C)=O)CC(NC(c2ncc3[nH]ncc3n2)=O)C2CCCC2C1 C(c1cccnc1)=C(C(=O)NC1CCN(C(C(C)(F)c2ccccc2)=O)C1)F Cn1c(=O)n(C)c2cc(C(N3CCC(C4CCC(=O)N4)CC3)=O)c(Br)cc12 n1(C(C)C)ncc(C(=O)N(C2CCC(NC(=O)C(C3CC3)C3CC3)CC2)C)c1N c1(OC)cc(C(=O)NC2CC(C)(NC(C3NC(=O)CC3C)=O)C2)ccn1 C1(O)(CCNC(C=CSC)=O)CCN(C(=O)CS(=O)(=O)Nc2ccccc2)C1 C1(C(=O)NCc2ccc(F)nc2F)(NC(CC2CC(CC)C2)=O)CCC(C)(C)C1 N1(C(c2c(C)nns2)=O)CCC(O)(CC(=O)NCC(c2cccc(O)c2)O)CC1 C1(C(c2nnnn2C)N(c2cc(C)ns2)CCN2CCOCC2)C2CC=CCC12 c1(-c2cc(C(=O)NCC=CCNC(CC3C(C)C3)=O)on2)cccc(Cl)c1 C1(NC(=O)NCCN(CCCNCC(C)C)CC)CCCC1C c1(C(N2CC(CC)N(C(C)=O)CC2)=O)cc([N+](=O)[O-])c2c[nH]nc2c1 C1(C(=O)NC2(C)CN(C(C3CCCN3C(C)=O)=O)C2)(OC)CCCCCCC1.CN Fc1cnccc1COc1ccccc1.C12CCN(CC1)CC1CCC1CN2 C(=O)(C1=C(C#N)CCC1)NCc1cn(CCNC(CSC(C)(C)C)=O)nc1 N1(C(C(F)OC)=O)CC(NC(=O)CCc2cc(C)on2)C(C)C1 C(=O)(C1=C(C)OCC1)N(CC(CC)NC(c1ccc(-c2cccs2)[nH]1)=O)C c1(C(=O)NCC23CC(NC(c4nc(C)c(C)s4)=O)(C2)C3)cnc2n1CCCCC2 Cn1ccc2cc(C(=O)NN3CCOC4CN(C(C5CC5C#N)=O)CC43)ccc12 c1(C(=O)NC(C2(O)CN(C(C34CC(F)C3C4)=O)C2)C)cc(C2CC2)nn1C c1(CS(=O)(=O)Nc2c(C)ccc(CSC)c2)cccc([N+](=O)[O-])c1 S(=O)(=O)(c1cccnc1N(C)CCc1ccccc1Br)NC(C)CCOC(F)F C12(CC(N3CC(NC(C=CCN(CC)CC)=O)C(O)C3)=O)CCCN1CCC2 C(C)(C)(CC(=O)Nc1cnccn1)N(C(=O)C(N)=O)C Cn1cc(CCC(=O)NCC2CCN(C(C3CC(C(F)(F)F)C3)=O)C2)cn1 C1(NC(c2cc3ccncc3[nH]2)=O)CCC12CCN(C(=O)CSC1CC1)CC2 N1(C(c2cccc(SC)c2Cl)=O)CCC2CN(C(=O)C3=NOC(C)C3C)CC12 c1(C(N2CCCC(C)(CNC(c3ccnc(F)c3)=O)C2)=O)[nH]nc2ncccc12 C12(NC(=O)CN3CCC(OC4CCCC4)CC3)CC(C(F)(F)F)(CO1)C2 C12(C(=O)NCCOC3CN(C(c4c(CC)con4)=O)C3)CCCC(=O)N1CCC2 CCC(C)CC(=O)NCC(C1CCCN1C(=O)CCc1cccc(OC)n1)(C)C C1(CNC(CCC#C)=O)CN(C(c2ccc(Br)c(N)c2)=O)CCC1(C)C N1(C(C(C)c2cc[nH]n2)=O)CC2COCC2(C(=O)N(C(C)C)CC2CC2)C1 C(=O)(C(O)P(C)(C)=O)N1CCN(C2CCN(C(C=C(C)c3cccs3)=O)C2)CC1 C1(N(C(C(C)OC)=O)C)CC2CCC(C1)N2C(=O)CNC(C)=O Cc1nn2ncccc2c1C(=O)NC1CCCC1CNC(=O)Cc1ccsc1C CC(C)CCCCC(=O)N1CCCC1CC(=O)NC1(C)CC1(C)C c1(C(N2CCC3(NC(C(=O)NC4CC4)=O)C(C2)C3)=O)cn2cccnc2n1 c1(C(=O)NCC(CNC(CCc2c(C)ncs2)=O)CO)cnn2ccc(O)nc12 C1(C(=O)NC2(CCC=C)CN(C(=O)NC3CC3)C2)CC12CCCOC2 C(=O)(C1CCCc2nccn21)N1CCC2CN(C(c3ncn(CC)n3)=O)CC1C2 c1(C(=O)NCC(C)(C(C)C)NC(C(CC)F)=O)c(F)cncc1Cl C1(NC(c2ccn(CC)n2)=O)CCCCC1CNC(=O)CC(C)c1ccncc1 C1(NC(c2cnc(C3CC3)nc2O)=O)CN(C(C2CCCC2)=O)CCC1CO CCC(C#N)C(=O)NC(C)(C(=O)N(C)CCc1ccccn1)C1CCC1 C1(C(N(C2CCCN(C(c3cn(CC)cn3)=O)C2)CC)=O)CCS(=O)(=O)C1(C)C C1(NC(c2cc(F)cc(Cl)c2)=O)CC2CC1N(C(C1SCCS1)=O)C2 C1(NC(c2ccc(N(C)C)cc2)=O)CCN(C(c2cc(C(F)F)no2)=O)CC1O c1(C(=O)NCCCCOC)noc2cc(-c3sccc3C)ccc12 C(=O)(CCN=c1ccc(S(=O)(=O)NCC(CO)C2CCOC2)c[nH]1)NC CC12CC(C(=O)NCC3(F)COCCN(C(=O)CN4CC5CC5C4)C3)(C1)C(C)(C)O2 c1(C(=O)NC2(C)CC(NC(c3cscc3F)=O)C2)cnc2ccccc2n1 C1(C)(NCC(N2CC(O)(CN(C)C(c3cccc(C)c3)=O)C2)=O)CCCCC1C Cc1cc(=O)c(-c2nc(Cc3cnn(C)c3)nn2CC(F)(F)F)cn1C c1(C(=O)NCCC2N(C(C(C(=O)OC)C)=O)CCC2)sc(Cl)c(Cl)c1C c1(NC(C2(C)CCN(C(C(C)NC=O)=O)C2)=O)c(Cl)cc([N+](=O)[O-])cc1Br c1(C(CC)C)nc(CC2CC(F)(F)C2)n(-c2c(C)noc2C)n1 C1(NC(C(C(C)C)(C)O)=O)CC2CCC1CC2NC(=O)Cc1nn(C)cc1Cl c1(-c2c(C)n(C)nc2)cnc2[nH]c(C(=O)NCCN3CCCC3)cc2c1 CCC(C)C(CC(=O)N(C(CO)C(C)C)C)NC(C1CC1c1ccccc1)=O CC(C)(C)C(=O)NCCCC(=O)NCCNC(=O)C=CCN1CCOCC1 c1(C(=O)NCCC(C)(C)NC(=O)CCNC(=O)CO)cc(Cl)ccn1 c1(C(=O)NC2C(C(=O)NC3C(OC)COC3)C2(C)C)ccccc1O c1(C2(C(N(CCNC(CC(=O)OCCC(C)C)=O)C)=O)CC2)ccc(F)c(Cl)c1 C#CCC(C(N)=O)NC(=O)C(C(C)C)NC(c1ccc(C(N)=O)[nH]1)=O C(=O)(C(F)C(F)(F)F)N1CC(CNC(c2csnn2)=O)OCC1 C(CCOC)(C(N)=O)NC1CCN(C(c2nn(C)cc2CC)=O)C1.c1(C)ccccc1 C(C(C)(C)CNC(=O)C(C)(C)N1CCCC1)N(C(CCOCCOCC)=O)C C=C1CC2(C1)CC(C(=O)NCC(CNC(c1ccsc1C)=O)C(F)(F)F)C2 Cc1oc(C#N)cc1C(N1CC(NC(c2cnc(C(F)(F)F)s2)=O)C2(CC2)C1)=O C1(NC(C(C)n2cccn2)=O)CCN(C(C2(O)CC3CCC2C3)=O)CCC1CO C1(C(N)=O)(OC)CN(C(c2ncoc2CNC(=O)Cc2cncn2C)=O)C1 N1(C(CC2CCCC(C)C2)=O)CC2CCC1C(CNC(C1CC1C)=O)C2 c1(OC(CC)C(=O)NCCN(C(=O)CSSC)C)cccc(C)c1 C(C(=O)NC1CCCC1SC)(C(C)O)NC(C(C1CC1)OC)=O N1(C(C2CNCCC2c2ccccc2)=O)CCCCC1C1(C(=O)O)CCC1 C(=O)(C1=CC2C=CC(C1)C2)N1C(C(=O)NCC2C(CC)C2)CNC(=O)C1 C(=O)(CCCCCC(C)(C)C)NCC(C)N(C(=O)C1=CCCCC1C)C C1(C(=O)NC(C)CNC(c2cc(Cl)n(C)n2)=O)CCN(CCO)C(=O)C1 N1(c2nc(C)cc(C)n2)CCN(C(=O)C(=O)C2CC2)C(C#N)C1 Cc1nc2cc(C(=O)NC(C)(CNC(=O)C(C)(O)C3CC3)C(C)C)ccc2s1 C1(CNC(CCCC#C)=O)CN(C(=O)C(F)=C(C)C2CC2)CC1(F)F O(NC(=O)CC(CC)C(CC(=O)OC)C)CCCOC C(C(O)CC(F)(F)F)NC(C(C)NC(CCNC(C)=O)=O)=O c1(OC)ncc(Br)cc1CC(=O)NCC1CC1NC(=O)C(C)(C)CO c12cccc(Cl)c1CC(=O)N2C1CCC(F)(F)C1.N1(CC)CCCC1 N1(C(c2sc(CC)c(C)c2)=O)CC(C)CN(C(c2cccc(N)c2C)=O)CC1C CCC(CCCC(=O)NC1(CSC)CCCC1)NC(c1cn[nH]c1)=O c1(SC)cc(C(N2CCC2CNC(C2CCCC23CCC3)=O)=O)ccc1F.C1(C)CC1 C(=O)(C1CCCn2nccc21)NCC1CCCCN(C(C(F)=CCC)=O)C1 Cc1nc(C)c(CC(=O)NC(C)CCNC(c2c[nH]nc2-c2ccsc2)=O)s1 c1(OC)ccc(CC(N2CCCC2CNC(=O)C(C)(C)CSC)=O)cc1F C(CN=c1cc(CC)nc[nH]1)(C1CC1)NC(c1ccc(OCC#C)cc1)=O C1(CC(=O)N(CC(C)N(C(CCOCCOCC)=O)C)C)CCCS(=O)(=O)C1 N1(C(c2cc(C(=O)OC)cc(Br)c2)C(=O)NCCCF)Cc2c[nH]nc2C(C)C1 c1(C(=O)Nc2cnc(CC(C)C)nc2)n[nH]c2c1CCC(C)C2 N1(C(COC(CC)C)=O)CCC(NC(=O)CC2CN(C(=O)OC(C)(C)C)C2)C1 N1(C(c2c(SC)snn2)=O)CC(CNC(c2ccc(C(F)F)cc2)=O)CC1C N1(C(C(Br)=C(C)C)=O)CC2(C1)CN(C(C1CCC(=O)C(C)C1)=O)C2 N1(C(C(C2(C)CC2)NC(C=C(C)C2CC2)=O)=O)CCC2(CCCC2)CC1 CC(CCCCCO)NC(c1csc(CNC(=O)CC2(C)CCCCC2)c1)=O Cc1cc(CC(=O)NCC=CCNC(C2CCCC(C)C2)=O)ccc1O C1(NC(COC2CC(NC(C(C)SCC)=O)C2)=O)CCn2nnnc2C1 CCC(C(=O)NCC1CC(NC(=O)Cn2cc(N)cn2)C1)c1ccccc1 CC(C)(C)C(O)CCC(=O)NC1COCCN(C(c2cc(Cl)ncc2F)=O)C1 c1(CNC2CCC(C(=O)NCC3CCC(C(=O)O)CC3)C2)c(O)cc(O)cc1O N1(C(c2cccc(C#C)c2)=O)CCC2CCN(C(=O)CC3CC(C)(C)CO3)C2C1 C#CCC(C(=O)NC1(c2noc(C)n2)CC1)NC(C1CC1(F)Cl)=O CC(C)(CC(F)C(=O)NCC1CCc2nccn21)NC(C1COCC1(C)C)=O CC1CCc2[nH]nc(C(N3CCOC(CNC(C45CC(C4)C5)=O)C3)=O)c2C1 C1(C(=O)NCC2NC(=O)OC2)C(F)CCN1C(C1CN(C(N)=O)C1)=O Cc1ncc(C(=O)NCC(C2CC2)NC(c2c(Cl)cnn2C2CCCC2)=O)n1C c1(OC)ccc(C(N2CC(C)CC2C(=O)Nc2ccc(C(F)F)nc2)=O)cc1Br c1(NC(C2(C)CCCN2)=O)nc2ccc(Cl)cc2s1.N12CCCC1C2=O C(C)(C(C(=O)N1C(=O)NC(CC)(CC)C1=O)C(C)C)NC(CCC=C)=O c1(C(=O)OC)cc(F)cc(NS(=O)(=O)Cc2cc(F)ccc2Cl)c1C C(=O)(C(CCS(C)(=O)=O)NC(c1cccc(Br)c1)=O)NCC(COC)C N1(C(=O)Cc2ccno2)CCN(C2CCCN(C(C3(C(F)F)CC3)=O)C2)C(=O)C1 C1(C(C)C)CN(C(c2ocnc2C(F)F)=O)CCN1C(=O)C=Cc1ccn(C)c1 c1(OC)cc(C)c(NC(c2nnnn2C2CCOC2)c2cc[nH]n2)cc1F N1(C(C(N2CCSCC2)C)=O)CC2CN(C(c3ccccc3Cl)=O)CC2C1 C1(NC(CCCCC=CC)=O)CC2CCC1CN2C(=O)CCC(C)(C)N(C)C CN1C(=O)N2CCC(C(=O)NC3CN(C(=O)C=CBr)CC3O)C1C2 c1(C(=O)NCCCCCN(C(=O)Cc2cnoc2)C)ccc(Cl)c(F)c1 C1(O)(CNC(C(COCC)C)=O)CCCN(C(=O)Cc2cccc(F)c2)C1 C1(CCNC(C2CNC(=O)N2)=O)CCCCN1C(=O)CC(F)F CC(CN=c1[nH]c2ccc(S(=O)(=O)N3CCC(F)(CF)C3)cc2s1)OCCO N1(C(c2nc(CC)oc2C)=O)CCC(NC(=O)C=Cc2ccc(C)o2)C12CCC2 N1(C(c2sccc2CO)=O)CCC(CO)(CNC(C23COCC2C3)=O)C1 CC1=C(C(=O)NC(c2ccco2)CO)C(C)n2ncnc2N1C C(=O)(CCCNC(c1ccsc1)=O)NCC(C)NC(c1cnn(C)n1)=O c1(NC(CC2N(C(c3c(C)nc(C)s3)=O)CCC2)=O)cc(C)c(F)cn1 Cc1nc2c(o1)CCN(C(C(=O)NCc1ccccc1Br)c1csnn1)C2 c1(OC(C(=O)NC2CC(CC)(CO)C2)C)cccc(C(C)C)c1 CCC(C)(COC)C(=O)NC1CC(OC)CN(C(=O)CC2CCC(F)(F)CC2)C1 c1(C(N2CC3C(C(=O)Nc4n[nH]c(C)c4Br)C3C2)=O)ccc(Cl)cc1C#N c1(NCC(=O)NCC2OCCN(C(C3(OCC)CCC3)=O)C2)ccc(C#N)cc1 c1(C(N2C(C)CC(NC(c3ccc(F)cc3)=O)C2)=O)ccc(=O)n(C)n1 CCC1=NOC(CC(=O)N(CCC(=O)NCc2nn(C)cc2C)CC)C1 c1(C(=O)NC2CN(C(CCC)=O)CC2C)cnn2c1OCC(C)(C)C2 c1(OC)cccc(C(C)CC(=O)NCC(C)CNC(C2CN(C)C2)=O)c1 CCC(CC(=O)NCC(C)Cn1cccn1)NC(c1cn(CC)nc1C)=O N1(C(C)C)CCc2onc(C(N3CCCC3CNC(c3cccn3C)=O)=O)c2C1 C1(NC(C2CC(OC)C2)=O)CC(NC(=O)CCc2cccnc2Cl)CC1O Cc1sc(C(=O)Nc2nc(C(=O)Nc3cccc(O)n3)cs2)cc1Br c1(OC)ccc(C)cc1C(=O)NC1CN(Cc2cc(C)ccc2OC)CC1O Cc1cc(F)ccc1CC(N1CCC(CNC(C2CN(C)CCO2)=O)C1(C)C)=O c1(C(=O)NC2CN(C(c3c(CC)occ3C)=O)CC2C)ccc([N+](=O)[O-])c(C)c1 C1(C)(NC(CCCCSC)=O)CCCCC1C(N1CC2CC1CS2=O)=O c1(N(CC)CC)noc2cc(-c3cccc(OC)c3)ccc12.c1(CO)ccco1 C(N=c1nc(N2CCCC(C3CCC3)CC2)c2ccccc2[nH]1)C1C(CCC)C1 c1(CC)c(C(=O)NC23CC2CN(C(c2sncc2C)=O)C3)csc1C c1(CCC(=O)NCC2CN(C(C(C)c3cccs3)=O)C2)cccnc1 c1(C(=O)NCC(CNC(C(C)CSc2ccccc2)=O)O)cc(N)c(F)cn1 N1(C(C(C2CN(C(C3CC4CC4C3)=O)C2)O)=O)CCCCC1 N1(CCCN=O)C(CCCC)C(N=[N+]=[N-])CN(C)CC1 C=CCCCC(C(=O)NCc1c(C)nn(C)c1C)NC(c1ccsn1)=O C1(C(=O)OC(C)(C)C)OCC2COCCC12.C1(C(=O)OC)CN(C=O)CCN1C(C)=O C(=O)(C1COc2c(C)cccc21)NC1CC(NC(C(CCCC)O)=O)C1 C(CC(C(=O)NCCC(=O)NC1CC1)NC(C1(C#N)CC1)=O)N(C)C C1(C(N(CC(C)NC(c2c(C)cn(C)n2)=O)C)=O)C(C)OC(C)C1C c1(C(N2CC(CN(C(CC(C)SC)=O)C)OCC2)=O)cccc2c1OCCN2C Cn1nc2c(c1C(=O)NCC1C=CCN1C(c1cc(F)ccc1O)=O)CCC2 CCCCC(=O)NCCC1CCC(NC(=O)CCCN(C)C(C)C)C1 N1(C(CN(CC(=O)N(C)Cc2ccc(C)o2)C2CC2)=O)C(C)CCCC1C c1(OC)sc(C(=O)NC(C)(C)CNC(c2cnc(S)nc2)=O)cc1Br C1(C)(NC(c2cc(C)c(C)s2)=O)CCCN(C(C2CCC2C#N)=O)C1 O=C1NC(c2ccccc2)C2=C1C(c1cc3ncccc3s1)NC(=O)N2C1CC1 c1(C(=O)NC2CCC(CNC(C3CC(F)C3)=O)CC2)cc(F)c(F)c(F)c1F CC(C)C(F)(F)CCN=c1[nH]c(=NC(C)C2CCCC2O)c2cccc(F)c2[nH]1 Cc1cc(NC(CN(C)C)C(C)C)ncc1S(=O)(=O)N1CC(C)C(C)C1 C(C)(CNC(=O)C=CC1C(C)C1(Cl)Cl)(CC(C)C)NC(C)=O C12(CC)CC(CC(c3cnn(C4CCC4)c3)C)C(C1)C2.N C1(C(N)=O)CN(C(=O)C(=O)Nc2cc(C3CC3)sn2)CCC1CO C(=O)(CCC[N+](=O)[O-])NCC(C(C)(C)C)NC(C(C(C)C)NC(=O)OC)=O C(=O)(CCCC(C)O)NCCCOCCNC(c1ccc(CC)s1)=O N1(C(C(C=C)O)=O)CC(CNC(c2ccccc2CN(C)C)=O)OC2COCC12 c1(-c2c(-c3ccn(C(C)C)n3)ccnc2)ccc(F)cc1Cl C1(CNC(C2CCC(C)C2)=O)CN(c2cc(Cl)ncn2)CCC12CCOCC2 N1(C(C2OCCC(N(C)C)C2)=O)CCCC(O)(CNC(c2ccccc2Cl)=O)C1 c1(C(N(C2CCN(C(C3C(C)=C3)=O)C2)CCO)=O)cc(C)c2[nH]cnc2c1 c1(C(N(CCC#C)C)=O)cc(CNC(C2(O)CCOC2)=O)no1 N1(CCN)CC2C3C=CC(CC3)C2C1.c1(CC)n[nH]c2c1CCCC2 CC(C)(C(=O)NC1CC(C)(NC(=O)CCCNC(c2cccs2)=O)C1)C1CCC1 c1(NC)ccc(C(N2CCC(NC(C3(Br)CC3)=O)CC2C)=O)cc1F N1(C(C(CC=C)N(C)C)=O)CCC(C)(CNC(c2cn(C)nc2C)=O)CC1 c1(C(=O)NC(CSC)C)ccc(C2OCC2(C)C)cc1 C1(O)(C(C)NC(c2ccn(C(C)C)n2)=O)CCN(c2ncncc2I)CC1 C1(C(=O)NC2CCCC(CNC(=O)CCOCC3CC3)C2)(CC)CCCCO1 C1(CC(=O)NCC=CCNC(CCCNC(=O)OC)=O)CCCCC12CC2 Cc1cccc(Br)c1CC(=O)N(CCCNC(C1CC2CCCC2C1)=O)C c1(CNC(=O)NCCC2CC(=O)NC2)cccc(F)c1 N1(C(c2c(CC)con2)=O)CC(CC(=O)N(CC(C)C(C)C)C)CC1(C)C C(=O)(C(C(=O)NCC1(O)CCN(C(C2(CO)CCCC2)=O)C1)OC)OCC c1(C(=O)NC(CC=C)CNC(C2CC2c2cccnc2)=O)cnn(C2CC2)c1C c1(C2CCC(NC(=O)NC3COC(=O)C3)CC2)nnc2n1CCCC2 C1(CC=C)(NC(=O)Cc2n[nH]cc2Br)CCN(C(=O)CS(=O)(=O)N(C)C)C1 C1(C(NNC(Cc2n(C)nc(C3CC3)c2)=O)=O)C2CCCC(=O)C12 c1(O)ccccc1CN(CCO)CC.C(C)(CCNC(=N)N)S N1(C(c2ccc(Cl)c(F)c2)=O)CCCN(C(=O)C(F)n2cccn2)C(CO)C1 N1(C(=O)NC(c2ccc(Cl)cc2)COC)CCN(c2n[nH]c(C3CC3)n2)CC1 C(C1CC1)(C1CC1)=CC(=O)NC(C(=O)NCCN(CCOC)C)C1CCC1 C1(NC(C23CC(CO)(C2)C3)=O)CCCC(NC(C2(COCC)CCOCC2)=O)C1 c1(C(=O)NC(C)CCn2cncn2)c[nH]c(C#N)c1.n12cc(nn1)CNC21CC1 N1(C(C)C(N)=O)CCS(=O)(=O)C(CCNC(c2cnc(F)c(Cl)c2)=O)C1 Cc1cc(O)ncc1C(=O)NCC(C)N(C(=O)CC1CCCCN1C)C CCCCCCC(CC)C(=O)N1CC2CC(NC(c3cccc(CC)c3)=O)C1C2 C1(O)(CC(=O)NCC2C=CCC2)CN(C(C2(CCc3ccccc3)CC2)=O)C1 c1(C(N(CCCNC(C2(C(N)=O)CC2)=O)CC)=O)ccc(C(C)C)cn1 N1(C(C(=O)NCC(C)N(C(C2C(C(=O)OC)COC2)=O)C)C)C(=O)CCC1=O C(=O)(C(O)CCC(C)C)NCCCCCN(C(C1(C)CC=C(C)CC1)=O)C c1(SC)ccnc(NC(N2CCCC2CCCF)=O)c1 c1(CO)nc(Br)ccc1NCc1csc(-c2cnc(CC3CC3)nc2)n1 C1(C(N2CC(COC)C2(C)C)=O)CCC2CCC1N2C(c1cc(F)cnc1O)=O N1(C(CCC2C(C)(C)C2)=O)CCC(C(=O)NCC2(C)CC2(C)C)C1(C)C c1(OCCCC)ccc(C(N2CCC2CNC(C2C(C#N)C2(C)C)=O)=O)cc1 c1(NC(=O)OC)ccc(C(=O)NCC2(C)CCN(C(c3ncccn3)=O)C2)cc1 C1(CC(=O)NCCCO)CN(C(=O)C=C(C2CC2)C2CC2)CC12CC2 c1(C(N2CC3C(CNC(CCCCC)=O)C3C2)=O)c(C)c(O)nc2ccccc12 CC1CCCCC1CCNCc1ccccc1Br C1(N(C(=O)CC2CSC2)CCC)CCN(C(=O)CC2CCCOC2)CC1 Cc1cc(CC(=O)NC(C2CN(C(=O)CC3C=NN(C)C3=O)C2)C)cc(F)c1 N1(C(C(C)CC2CCC2)=O)CCOC(CCNC(C2(C(N)=O)CC2)=O)C1 c1(C(=O)NC2CCCC(CNC(C3CCCC3)=O)C2)cccc2occc12 C1(C(=O)OC)CCC(C(N2CCCC2C(C)(C)NC(=O)C=CCO)=O)CC1 c1(C(=O)NCC(CC=C)NC(C2(C)CC2C)=O)cccc([N+](=O)[O-])c1Cl c1(OC)cccc(C(=O)NCC(C)NC(=O)Cc2cn(C)nn2)c1C c1(C(N2CCCC(C)C2CNC(=O)C2=CSCS2)=O)[nH]nc2ncccc12 C(=O)(CC(C(C)NC(=O)C(CN(C)C)CC)N(C)C)N1CCC(COC)C1 CC(C(=O)NCC12CC(NC(c3cocn3)=O)(CO1)C2)C1=CCCC1 C1(NC(C(CCC)OC)=O)CN(C(c2ccc(C)cc2OC)=O)CC2CC12 C(=O)(C(CC(C)(C)C)NC(=O)CC1(N(C)C)CC1)N1CCCC(COC)C1 c1(C(=O)NCCNC(c2onc(CC)c2C)=O)occ2c1CCOC2 c1(C(N(CCNC(C23CC(C2)C(C)O3)=O)CC)=O)cnc2ccc(C)cc2c1 N1(Cc2nc(CCCC)[nH]c2Cl)C2CCC1CC(NC(C1CCCN1CC)=O)C2 c1(C(=O)NCC(CNC(c2ccc(C#N)cn2)=O)F)c[nH]c2cccc(Cl)c12 N1(C(c2ccc(C)o2)=O)CCOC(C(C)NC(C23CC(CF)(CO2)C3)=O)C1 c1(C(N2CCC(CCNC(c3cc(C#N)sc3)=O)C2)=O)csc2ncnc(O)c12 C1(NC(C2(OCC)CCOC2)=O)CCC(CCC(=O)N(C)CC2(CO)CCC2)C1 CCC(O)C(C)C(=O)N(CCCCNC(C1COC(C)(C)CO1)=O)C N1(CCCCCNC(c2c(CC)nc[nH]2)=O)CCN(C(=O)C(C)=C2CC2)CC1 CC(C)CC(CNC(=O)COc1ccsn1)C(=O)NCC1CC=CCC1C Cn1nc(C(=O)NCC2CCN(C(c3scnc3C(F)F)=O)C2)cc1C(N)=O N(C(=NCc1ncccc1OC)NC(C)C)CC(COC)F C1(C)(CC(=O)NC2CCC(NC(Cc3cnc(C)s3)=O)C2)CCCCC1 C1(NCC(CNC)O)(ON)CC(C)(C(C)C)C1 C1(NC(C2(NC(C3CCN(C)C3=O)=O)CSC2)=O)CCN2CCCCC12 CC(F)(F)CCCC(=O)NC(C)(CNC(c1ccccc1[N+](=O)[O-])=O)C1CCC1 N1(C(CCc2cccc(C)c2)=O)CCN(C(C2COCC2(C)C)=O)CC1CO c1(CC(=O)NCC2(F)CC(CNC(C3N(N=O)CCC3)=O)C2)nc([N+](=O)[O-])n[nH]1 C1(CN(C(CCOCCN(C(C(C=CC)O)=O)C)=O)C)CCCC2CC12 C1(NC(CC(CCC)(C)C)=O)CC2CCC1CN(C(C1C3CCOCC13)=O)C2 C1(C(=O)NC2C(NC(c3c(Cl)ccc(F)c3F)=O)C2)COCC2(CCC2)O1 CC1(C)C(NC(C2C(C#N)C2(C)C)=O)CC1C(=O)NC(CF)C(F)(F)F c12ccc(cc1)C(C(C)C)NC2c1nnnn1C.C1(F)(C)CCOC1.CC C1(C(NOCC(=C)Cl)=O)CCN(C(C2CC23CCC3)=O)C1(C)C c1(CC)cc(C(=O)N(CC(Cc2ccccc2)NC(=O)C(N)=O)C)ccc1C c1(C(N2C3(CNC(CNC(CC)=O)=O)CCC2CC3)=O)c(C)ccc(C)c1O Cc1ccc2sc(N(CC(C)CNC(=O)C3=NOC(C(C)(C)C)C3)C)nc2c1C c1(C(N(CC(C)(C)NC(C=Cc2cnc(C)s2)=O)C)=O)cc2cc(Cl)ccc2o1 Cc1ccn(CC(N2CCC(CN(C)C(c3cn(C4CC4)cn3)=O)C2)=O)n1 C(=O)(CCCCCCCO)N1CCN(C(c2c(C)csc2)=O)C2C1C2 c1(C(=O)NC2C(CNC(C)=O)C2)nccc2c(S(N)(=O)=O)cccc12 c1(N2CC(CNC(c3ccc(O)nc3)=O)OCCC2)nc(Cl)nc2c1CCOC2 CC(C)C(C)C(C)CC(=O)NCCCC1(NC(C2SCCS2)=O)CC1 C1(C)(C(C)C)CN(C(C2CNC(=O)CN2C(C2CC(OC3CC3)C2)=O)=O)CCO1 N1(C(=O)OC(C)(C)C)CC(C(=O)NCCn2cc(F)ccc2=O)CCC12COC2 Cc1ncc(C(=O)N(C)CCNC(=O)Cn2[nH]cnc2=N)cc1C(F)(F)F C1(NC(C2C(OC)C2)=O)CCC(O)CN(C(c2cccn3ccnc23)=O)C1 C1(O)(COC)CCOCC1NC(=O)C(C)(C)n1ccc(C(F)(F)F)n1 Cc1cc(C(=O)Nc2cc(NC(c3cn(C)c(C(F)F)n3)=O)no2)ccc1Br Cc1ccccc1C(C)C(=O)N1CC(Cn2cc(CN(C)C)nn2)C1 C1(C2CC2)(OC)CN(C(=O)C(C)NC(C2CC3CCCC3C2)=O)C1 c1(C(N2CC3(C2)CN(C(C2CCCO2)=O)CC3CO)=O)cc2ccccc2cn1 Cc1cc(CC(=O)NCCN(C)C(C2COCCC2C)=O)cc(C)c1 C(C(=O)NC1(CNC(=O)C(O)C(F)F)CCC1)(C(C)C)SCC N1(CCC(=O)NCC(C)(C)NC(=O)CCN2CCCC2)CCSC(C)(C)C1 c1(C(=O)NC2CCC2CNC(C2(CO)COC2)=O)ncsc1-c1ccccc1 C1(O)(CC(=O)NCc2c(C(=O)NCc3n(CC)ccn3)cco2)CCOCC1 C12(NC(C3(O)CCC3)=O)CCC(CC1)N(C(=O)COC(F)(F)F)C2 C1(CNC(C2CC(C)OC(C)C2)=O)C2CCCC1N(C(=O)C1=CCCS1)C2 c1(NC(=O)NCCS(CC)(=O)=O)ccc2c(c1)c(C)nn2C C1(C(=O)NCCOCCNC(c2ccc(CO)cc2)=O)CCCC(C(F)(F)F)C1 N1(C(CSc2n(C)ccn2)=O)CCN(CC(=O)Nc2ccc(CC3CC3)o2)CC1 c1(C(N(CC(C)NC(C2C(C)(CC)C2)=O)C)=O)cnc2sccc2c1 C1(CNC(C(N2C(CC)CCC2)=O)=O)C2CN(C(=O)CP(C)(C)=O)CC12 C1(C(N(CC(C)C(=O)N2CC(N3CCOC3=O)C2)C)=O)Cc2nccn2C1 c1(C(N2CCC(c3nc(C)no3)C2)C(=O)NCCCC)nnc(C2CC2)s1 CC(C)CC(C)CC(=O)N1C(CNC(c2cc3ccsc3s2)=O)CC2CC12 C=CC(C)(O)CC(=O)N1CCC(CCCNC(C2Cc3nncn3C2)=O)CC1 N1(C(c2c(C)n[nH]c2C)=O)CCC2CN(C(=O)C(C)(C)CNC(N)=O)CCC2C1 C1(NC(C2CC3CCC2O3)=O)CCCCN(C(=O)CC2CSCCS2)C1 C1(C(=O)NCCC(C)OC)(COCC)CN(C(=O)CN2CCCCC2)C1 c1(C(=O)OCC)cccc(NC2CCN2C(=O)CCN2CCN(C)CC2)n1 c1(C(=O)NCC2(CNC(C3(C)N(C)CCC3)=O)CCC2)cc2ncccc2o1 C12(CNC(c3c(C)nn(C(C)C)c3)=O)CCC1CCN2C(c1ccc(N)cn1)=O C1(C(=O)NCCCC2OCCN(C(c3n(CC)ncn3)=O)C2)(OC)CCCOC1 N1(C(Cc2cn(SCC)nn2)=O)CC(NC(=O)CCC2NC(=O)NC2=O)C(C)C1 c1(C(=O)NC2C(CNC(=O)C=CC(F)(F)F)CCC2)cncc(Cl)c1Cl CC1CCN(CCc2cn(CC3CCCN3C(C3(C)COCCO3)=O)nn2)CC1 C(=O)(CCCC(=O)N1CC(CC(F)C(N2CCCC(C(C)C)CC2)=O)C1)OC C(=O)(C(C)(C)CS(C)(=O)=O)NC1CCN(C(C=CSC)=O)C(C2CC2)C1 c1(SC)ncc(C(=O)N(CCCN(C)C(C2CCCN(C(N)=O)C2)=O)C)n1C c12cc(cnc1F)OCC1CN(CCO1)C2=O.C(C)(C)(C)OC(N(CC)CC)=O C=CC(C(=O)NC(c1ccccc1)C(=O)NCCC1COCC1O)OC C1(C(=O)NCCOCCOCCNC(CCC#C)=O)COc2cc(O)ccc2C1 Cc1nc(C)c(C(=O)N(C2CCN(C(=O)COC3CC3)C2)C)nc1C c1(NCCCOC=C)ccc(S(=O)(=O)NCc2ccc(F)c(C3CC3)c2)cc1F C1(CNC(CCN(C(COC2(C)CCCC2)=O)CC2CC2)=O)CC(O)CCO1 n1(NCC(=O)NCC(N2CCCC(C)C2)C)nc(C2CC2)n(C)c1=O C1(C2CCCN(C(c3cn(-c4ccccc4)cn3)=O)C2)(NC(=O)CC(F)F)CC1 C#CCC(O)C(=O)NC12CC(C1)N(C(c1cc(Br)c(OC)s1)=O)C2 c1(C(C2CC2)NC(=O)NC(c2cccs2)C)cccc(O)c1 N1(C(C(C(C)(C)C)NC(c2cc[n+]([O-])cc2)=O)=O)CCC(O)C(F)(F)C1 c1(N2CCC(CNC(CCS(=O)(=O)NC)=O)C2)ccc2cnccc2c1[N+](=O)[O-] c1(C(=O)NCCC(C(C)C)NC(=O)Cc2nccs2)ccc(N=[N+]=[N-])cc1 C1(NC(c2c(C(C)(C)C)noc2)=O)CC2CC1N(C(C13CC1COC3(C)C)=O)C2 CP(C)(=O)CCC(=O)NCCC1CCCN1C(C1CCCOCC1)=O C1(NC(C(OCC)OCC)C)CC2CCCN(C1)S2(=O)=O CC1(NC(=O)Cc2cncnc2)CCCCC1C(N1CCSCC1)=O O=C1CC(C2CC2)(CNc2ccc(CN3CC(c4ccccc4)C(O)C3)cc2)C1 c1(C(C(=O)NC2CC(C#N)C2)NC(CCSCCC)=O)ccccc1 C1(C(N2C(C(C)C)CN(C(=O)C(C)(C)F)CC2)=O)CCC2(CCCC2)C1 C12CCN(C1)C(=O)c1ccsc1NC2.C1(c2ccccc2)(C(=O)OC)CCOC1 C12(C(=O)NN3C(CNC(c4cccc(OC)c4)=O)CC(C)C3)CCC(C1)OC2C C1CCCCOC(C)C(=O)N1C.C(C=CC(=O)OC)(CC)=CC=CC N1(C(c2cc(NC(CCC)=O)ncc2)=O)CC(NCC)CC1(COC)CC c1(C(=O)NC(CNC(CN(C)C(N)=O)=O)(C)C2CCC2)cccn2ccnc12 C1(CCNC(C(C2CC2Cc2ccco2)N(C(C)C(F)F)C)=O)CCCCC1 c1(C(N(CCCOCCN(C(c2ccc(C)o2)=O)C)C)=O)cc(C)c(C)cn1 N(C1CCNC(=O)c2[nH]ccc21)C(=O)Nc1cccc(F)c1[N+](=O)[O-] C=CCC(C(=O)N(CC(=O)NC(C(O)CO)C1CC1)CCOC)OC C1(CNC(C(CC)CC)=O)CN(C(c2coc(O)n2)=O)CC(C)(C)O1 Cc1nc2ccccc2cc1C=CC(=O)N(C)CCNC(C1CC1F)=O c1(C(N(C)C)=O)ccc(Cn2nc(-c3ccncc3)nc2CC(C)C(C)C)cc1 C1(CC)CCCC(N=c2cccc(S(=O)(=O)N3CCC(CSC)CC3)[nH]2)C1 c1(C(N(C2CC(C(=O)NC3CNC(=O)C3)C2)C)=O)ccc(=O)n(C)n1 CC1(C)CC(C)(C(N2CCC(C3CCCN3C(=O)CCc3cnoc3)C2)=O)C1 CCCC(C)C(=O)N1CC(O)CC1C(=O)Nc1cncc(N(C)C)c1 c1(CCNC(N2CCN(CC(=O)O)C(=O)C2)=O)ccc2c(c1)CCO2 c1(C(=O)NC(CCC)CO)cc2ccc(-c3ccoc3)cc2n1C c1(C(=O)NCCCN(C(CCN(CCCCC)C)=O)C(C)C)oc(C)nc1C N1(C(=O)CCc2ccon2)CCCC(CCNC(C2(CF)CCOCC2)=O)CC1 c1(CNC(C23CCCN(C(=O)CN4CCSCC4)C2C3)=O)ccc2c(c1)CCC2 C1(C(=O)NC(C2CCC2)C)(NC(c2cn(CC=C)nn2)=O)CCN(C)C1 c1(C(=O)NC(CN(C(c2sc(OC)nc2C)=O)CC)C)ccc(C)c(Cl)c1 CCC(C(=O)N(CC(=O)NCCOCC(C)(C)CN(C)C)CC)N(C)C C1(NC(C(C)OCCC=C)=O)CN(c2nncs2)CC12CCOCC2 CC1CN(C(C2CCC(=O)NC2)=O)CCN1C(=O)CCc1cccc(N(C)C)c1 CCCCC(CNC(c1ccon1)=O)NC(=O)C(F)(F)CC1CCCO1 N1(C(c2c(C)nc(CCC)o2)=O)CCCC(NC(=O)CCCC(C)C)C1C C1(C(N(CCCCNC(CCC=CC)=O)C)=O)CCCCN1C(C)C C1(N(C(C2CCN(C(C(C)CC3CCCC3)=O)C2)=O)C)CC2CCC1O2 N1(C(C2CCC3CC23)=O)CCN(C(c2noc3c2CCCC3)=O)C2(CC2)C1 N1(C(=O)CO)CCC(C(=O)NC2CCC2Nc2ccnn2C2CCOCC2)CC1 N1(C(C(c2ccc(F)cc2)OC)=O)CCC(O)C(NC(=O)C2=CCOCC2)C1 C1(O)(C(N2CCC(OCCNC(c3cccc(O)c3O)=O)C2)=O)CC2CCC1C2 C1(O)(CNC(C2(CCCC)CC2)=O)CCN(C(=O)Cc2c(C)cnn2C)C1 C(=O)(C(C)(C)CNC(=O)C(Cn1ccnn1)NC(=O)C=Cc1nccs1)OC C1(NC(c2ccc(C)o2)=O)(CO)CCN(C(=O)CCc2scnc2C)CC1 N1(C(c2c(C)snn2)=O)CCCN(C(=O)C(O)Cc2cnn(C)c2)CC1CO CCC(C)C(CC(=O)N1CCC(N2CC(O)C2)C1)NC(=O)C(N1CCOC1=O)C Cc1nc([N+](=O)[O-])cn1CC(=O)NCCCN(CCO)C(C1CCCOC1)=O n1(CC)cnc2c(N(CC(C)NC(=O)C(C)(C3CC3)NC(C)=O)C)ncnc12 c1(C(N(C(C)CNC(C2CCC=CCCC2)=O)C)=O)cc2c(nc1N)CCC2 C1(C(N2CC(c3ccccc3)(NC(CSCC)=O)C2)=O)CCCCC1(F)F c1(C(=O)NCC(c2ccc(OC)cc2)NC(=O)C2CC2)cnc2c(n1)CCCC2 c1(OC)cc(CNC2CN(C(c3cn(C)nc3C(F)(F)F)=O)CC2C)ccc1F C(=O)(C1=CC(C)(CC)C1)NCc1cn(CC(NOC(C(=O)OCC)(C)C)=O)nn1 N1(CC(N2CCOCCC2C)=O)CCC2(CC1)CC2NCCCCCC c1(CC)cc(C(=O)NCC(C)(C)CCNC(=O)CCSCC(C)C)n(C)n1 C#CCC(C)(C)C(=O)NCC1CN(C(c2cnc(C)s2)=O)CC1O c1(C(c2nnnn2C2CCOCC2)NC(COCC)(C)C)scnc1Br N1(C(C(=O)NCCCNC(=O)OC(C)(C)C)[Si](C)(C)C)CCC2(CC=CCO2)C1 n1(CC)ccc(C(=O)NC2CC2CNC(=O)CC2CC(C)(C)CO2)c1C c1(-c2cn(CCCCCC=C)nn2)cnc(OC)c(OC)c1 C1(NC(c2cc(C)no2)=O)CN(C(=O)C=Cc2cncn2C)CCC1C(F)(F)F c1(C(N2C(CNC(=O)Cn3ccnn3)CCC2)=O)cccc2c1OCCN2 CC1CCCCC1(CNC(=O)C=CC(N)=O)NC(=O)Cc1ccc(F)nc1 C(CCC)(C(O)C(=O)N1CC(C2CCCC2)C1)NC(c1c(CCC)n[nH]c1)=O C(=O)(CS(=O)(=O)CC)N1CC2C(CNC(C=CSC)=O)C2C1.c12cn(nn1)CC2 C1(NC(C(C2CC2)OC)=O)CC2(C1)CC(NC(C1CC(F)(F)C1(C)C)=O)C2 CC1(NC(c2c[nH]nc2CCNC(=O)CSC2CC2)=O)CCCC1O c1(CNCCOCCC)ccc(-c2cc(F)ccc2OC)cc1C Cc1cn(C)cc1C(=O)NC(C1CC1C(=O)NC(c1nc[nH]n1)CO)C C1(CC)CCCN1C(=O)C(Cc1cn[nH]c1)NC(=O)CC1COCCO1 N1(C(c2cc(C)cc(F)c2)=O)CCC2(CC1)CC(NC(=O)CC(C)(C)C)C2 c1(CC)cnc(Cl)[nH]c1=NC1CN(C(C2OC(C)CC2C)=O)CC1C C12(CNC(CCCN(C)C)=O)CCCC1N(C(=O)COC1CCCCCC1)CC2 c1(CC(C)(C)OC(=O)NC2CC(C)N(C3CC3)C2)c[nH]c2cc(F)ccc12 c1(C(=O)NC(CCOC)CNC(c2[nH]nnc2C2CC2)=O)cncc(C#N)c1 N1(C(C(c2cccc(C(=O)OC)c2)OCCOC)=O)CCC(C(N)=O)(N(C)C)CC1 CC(C)CC(C(=O)NC1CCCN(C(=O)Cc2ccc(F)cc2F)C1C)C(C)C C(N=c1[nH]c(C#N)c(Cl)s1)C1C(C)CN(C(=O)C=Cc2ccc(F)nc2)CC1 N1(CCNC(=O)C(=O)NC2CC(F)(F)C23CCC3)CCc2ccccc2C1 Cc1nc2c(cnn2C(C)C)c(C)c1CCC(N1Cc2cccc(N)c2C1)=O N1(C(CC(C)C)=O)CCC(NC(=O)C(CO)NC(N)=O)CC1 c1(C(N2C(C)(C(=O)NC)CC2)=O)cc(CC)c(C)[nH]1 c1(C(N2C(CNC(c3c(CC)ocn3)=O)CC(O)C2)=O)nc(Br)n2ccccc12 c1(SCC)cc(C(=O)NC2CC(C)(NC(=O)CN(C3CCCC3O)C)C2)ccn1 N1(C(c2nc(C)sc2C)=O)CC2CC(NC(c3ccc(C)s3)=O)C(C2)C1 c1(C(=O)NC2C(NC(C(C)SCC)=O)CCC2)[nH]c(C)nc1C C(CCC(=O)NC(c1cn(CC2CNC(=O)C2)nn1)(C)C)SC C1(C(N2CCC(N(C(=O)C=Cc3cn(C)cn3)C)C2)=O)CC(F)(F)CCC1(C)C CCCCCC(O)C(=O)NC1COCC1CNC(=O)C=CCOC N12CCSC(C1)C2=O.c1(C(=O)N(CCCO)CCCO)ccccn1 C1(NC(C2CC(SC)C2)=O)C2CCCN(C(=O)CN3CC4CC4C3)C2C1(C)C c1(C(=O)NCC2C(C(=O)NC(C#C)(C)C3CCC3)C2)cc(Cl)ns1 Cc1ccc(C=CC(=O)NCC2CCC(NC(C3CCC(C)C3)=O)CC2)cc1C C1(C(=O)NCc2cn(CCC)nc2)CCN(C(=O)CCC(F)(F)F)CC1O C(CC(C)C)(C(=O)NCC1CN(C(C2CC(O)(C(F)(F)F)C2)=O)C(C)(C)C1)OC Cc1ccc(CC(N2CCCC2C(C)NC(c2cnsn2)=O)=O)cc1 C(CCC(=O)NC1CCCC1CNC(c1ccn(C2CC2(F)F)n1)=O)SC N1(C(CN(C2CCC2)C)=O)CC2OCCN(C(C3CCCC(C#N)C3)=O)C2C1 c1(CCCC)nc(-c2cccc(Cl)c2)nn1C1CCc2ccccc21 N1(C(C2CC2(F)F)=O)CCCC(CCNC(C23CC(F)C2C3)=O)CC1 C(=O)(C(O)C(F)(F)F)N.C1(NC(C(=O)NC2CCCC2)=O)(CO)CCOC1 c1(C(N(C2CCN(C(C(C(CC)O)(F)F)=O)C2)CC)=O)cncc2nc(O)[nH]c12 N1(C(c2cc(OC)no2)=O)CC(C)(C)CC1CNC(=O)COCc1cc(C)on1 N1(C(c2c(C)nc(C)[nH]2)=O)CCCCC(NC(C2(C(F)(F)F)CC(F)(F)C2)=O)C1 C(CCC(C)C)(C(=O)NC1(CC(C2CC2CC(C)(C)C)C)CCCC1)NC(C)=O c1(NC2CCC(C(=O)OC)NC2)cccc(S(=O)(=O)C2CCCC2)c1 C=C(C)C(CC(=O)NC(C)CCN(C)C(C1(CC)CC1)=O)OCC C=CCC(C(=O)NCC(CC)NC(c1cnsc1)=O)c1ccccc1 c1(CC(=O)NCCCn2cc(C3CCC3C(F)(F)F)nn2)ccc(Cl)nc1F N1(C(c2cc(OC)c(Cl)cc2)=O)CC2CCN(Cc3ccc(I)cc3C)C2C1 c1(C(=O)NC2CCCN(C(C3CCSCC3)=O)C2)onc2c1CCCC2 c1(OC)ccc(NC(=O)C(CCO)NS(C)(=O)=O)c(OC)c1 c1(CC)ccc(O)c(NC(=O)C(C2(O)CCC2)NC(=O)C(C)C2(O)CCC2)c1 N1(C(CC2C(C)(C)C2(C)C)=O)CCN(C(c2ccsn2)=O)CC1C1CC1 C1(C(C)=O)CC(CC(=O)NCCNC(=O)C(C)(C)Sc2ccc(C)cc2)C1(C)C N1(C(C2=CCN(C)C2)=O)CCC2CCC(NC(=O)C(C)(C)F)C1C2 N1(C(C2N(C(N)=O)CCC2)=O)CCc2sc(CNC(=O)CNC=O)nc2C1 c1(C(=O)OCCCOCCOCC)csc(C(=O)OC)n1 c1(CCSCCNC(c2cc(OC)no2)=O)ncc(C(F)(F)F)cc1Cl C1(C(=O)NCc2c(C)nco2)CN(C(=O)CCC(N)=O)CC1O C(=O)(CC(C)(O)COC)NCCC1CN(C(COC(CC)(C)C)=O)C1 c1(CNC(CN(C(c2ccnnc2)=O)CC)=O)conc1C N1(C(CCN(C(C)C)C(c2ccsc2Cl)=O)=O)CCOCC(C)(F)C1 Cc1c(C(=O)NCC(CO)NC(=O)C(O)Cn2cncn2)cnn1C(C)C N1(C(Cn2ccc(C(=O)OC)n2)=O)CCCC(N(C)C(C2CCCCO2)=O)C1 c1(CC(=O)NCC(C2(O)CCN(C(CC=C=C)=O)C2)C)ccc2c(c1)CCOC2 O(NC(=O)CC(C)(C)NC(C)=O)CC(=C)Cl CCS(=O)(=O)CC(=O)N1CCC(CNC(C2CCCC2OC)=O)(OC)CC1 CC1CN(C(=O)C(C)(C)NC(c2ncn3c2CCC3)=O)CC(C)O1 c1(-c2cn(C)nn2)nc(-c2ccoc2)nn1Cc1cccc(Br)c1 N1(C(c2n(CCC)ncc2)=O)CCN(C(CNC(=O)CCC#N)C(F)(F)F)CC1 CC1(C)CC(CC(=O)NCC2CC(CNC(=O)C=C3CC3)CO2)C1 N1(C(C2(C(=O)OC)CC2)=O)CCC(C#N)(NC(C)=O)C1.c12ccc(o1)CNC2 c1(-c2cn(CCN(C(C3(C)CCNC3=O)=O)CC)nn2)ccc2cnn(C)c2c1 CCCCC(O)C(=O)N1CCC2C(NC(C3(c4ccno4)CCC3)=O)C2C1 N1(C(C(C=C)(C)C)=O)CCC2CCC(C1)N2C(=O)C(C)=CCO C1(C(=O)NCC(C)(C)CC2CC2)CC12CCCC2.C1(=O)C(=O)NCCOCCN1 N1(C(C2C(CCOC)C2)=O)CCCCC12CC(NC(=O)CC1C=CCC1)C2 N1(C(c2c(C)oc(CO)c2)=O)CCCN(C(c2cnn(C3CC3)c2)=O)C(CO)C1 C12(C(=O)NC(C3CCN(C(C4CC4(C)Br)=O)CC3)C)CCC(F)(CC1)CC2 N1(C(c2cn(-c3c(C)nccc3)nn2)=O)CCCS(=O)(=O)CC1c1cnn(C)c1 S(=O)(=O)(c1cccc2cnccc12)NCC1CCC(NCC2(C)CCC2)CC1 C(CCSC)(C(=O)NCCCC1CCOC1=O)NC(C1N(CC)CC1)=O C(=O)(CCCCCN(C(c1cnc(C(C)C)nc1)C(=O)NC)C)OCC C1(NC(Cc2cc(C)on2)=O)CCC(CNC(=O)CCc2c(C)noc2C)CC1 c1(C(N2C3C(CNC(C(C)CO)=O)CC(CC3)C2)=O)ccc2c(c1)COC2=O C12(NC(c3cnc(OCC)s3)=O)CC1CN(C(=O)CC1C=NN(C)C1=O)C2 c1(C(N2CC(OCC#C)C2)=O)cnccc1OC1CCCCC1n1cc(Br)cn1 C1(CN(C(=O)CCN(C(=O)C(c2ccccc2)F)C2CC2)C)CC2CCC1O2 C(=O)(CCC(C)(C)C#N)NCC(C(=O)N(CC)Cc1cnn(C)c1)(C)CC C1(NC(C(CC=CC)C)=O)COC2CN(C(c3ccccc3N)=O)CC12 CC(C)(CC(=O)N(C1CCCC1O)C1CC1)n1cc(C2COCCC2O)nn1 c1(N2CCC(NC(CCCCOCC)=O)CC2)nc(C)nc2c1cnn2C N1(C(c2cccc(C(=O)NC)c2)C(=O)NCC(C)C)CCCCCC1C N1(C(c2ccc(C(=O)OC)[nH]2)=O)CCCC(NC(=O)CNC(C)=O)C1 Cc1nc(CC(=O)NCC(=C2CN(C(C3CCC(C)S3)=O)C2)F)n[nH]1 c1(C(=O)NC2(CCCNC(Cc3c(C)ocn3)=O)CC2)cccc(F)c1F C(=O)(C(CO)C(C)(C)CCCCN)NC(c1cn(C)nc1)C1(CO)CCC1 C(CC(C(=O)NCC1(C2CCC2)CC1)NC(C1CCC1C#N)=O)SC c1(C2CCN(C(C3CCN(C(c4c(C)ncs4)=O)C3C)=O)C2)ccc(O)cc1F Cc1nnc2n1CCCN(C1CCN(C(c3ccccc3)C)C1=O)C2 c1(C(=O)NCC(CC=C)NC(C2CC(=O)NC(=O)N2)=O)cc(Cl)ncc1OC C1(NC(Cc2c(CC)con2)=O)CC=C(C(=O)N(c2csnc2C)CC)C1 Cc1nc(S)sc1CC(N1CC(CNC(c2ccccc2C(C)O)=O)C1)=O CCC(C)CC(=O)NCCN1CCC(NC(=O)COc2ccccc2F)CC1 C1(C(N2CCOC3(CC3)C2)=O)C2CC(F)C(C2)N1C(c1ccccc1)=O N1(C(c2cccc(Br)c2O)=O)CCC2(CC1)CC2C(N1CCSCC1)=O N1(c2scc(C(=O)O)n2)CCC(C(=O)NC2CC(=O)N(c3cn[nH]c3)C2)CC1 CCC(C)(Cl)CNC(C1COCC1NC(C12CCC(C1)C2)=O)=O CN1C(=O)CCC1CC(=O)NCC1CCCN1C(c1ccc(OC(F)F)cn1)=O c1(C(N(C2CC=C(C)CC2)CC(CNC(C)=O)O)=O)c(C)cccc1Br c1(C(=O)NCC(CC)(C)NC(=O)CSc2nc(C)cc(C)n2)c(C)nn(C)c1Cl C(CCCCC(=O)N1CCC(CCN(C(=O)CC2OCCC2C)C)CC1)OC C1(C(=O)NCC2C(CNC(C(C)CC3CCCC3)=O)C2)C2CC3C(C2)C13 Cc1cc(N2CCC(c3cc(O)n[nH]3)CC2)nc(=NCCC2CCCO2)[nH]1 c1(C(C(c2nnnn2C(C)C)NCCC(C)SC)(C)C)ccccc1Br CC(C)C(C(=O)N1CCOC(C(=O)NOCC2CCOC2)CC1)C(C)C N1(C(CC(CCC)(C)O)=O)CCCC2CN(C(C3CN(C)CCO3)=O)CCC12 c1(OC)cc(C)c2cc(NC(C3CCCN(C(=O)C4CC4)CC3)=O)ccc2n1 n1(CCCC)nccc1C(=O)N(CCCNC(C1CC1[N+](=O)[O-])=O)CCC n1(CCNC(C2CCC(O)C2)=O)ccc(C(=O)NCC2CC2CO)c1 Cc1ccc(C(=O)N(CC(=O)NCc2cnc(C)c(C)c2)C2CCC2)cc1O c1(C(=O)NC2CC3CC(NC(C(C(C)C)OC)=O)CC32)ccc2c(c1)OCCN2 C1(NC(c2c(C)snc2)=O)CN(C(C2(C(=O)OC(C)(C)C)CCCC2)=O)CC1C N1(C(CC(CC)C2CC2)=O)CCCN(C(=O)CNS(=O)(=O)NC)CC1CO CC1(C)COCC1C(=O)NC1CC1CNC(=O)C(c1ccccc1Cl)(F)F Cn1c(CCNCCC(=O)Nc2ccncc2)nnc1S C(=O)(NNC(=O)CN1CCC(N(C)C)C1)N(C1CN(C(C2C(C)OCC2)=O)C1)C C1(CC(=O)N(C)CCNC(C2CCCC2c2ccccc2)=O)COCCOC1 N1(C(CCC(=O)NC)=O)CC23CCCC2(C1)CN(C(c1nc(=N)cc[nH]1)=O)C3 Cn1nc(-c2ccc(Cl)s2)cc1NC(=O)NCCCCC1CC1(C)C(F)F C(=O)(C#CC(C)(C)CNC(=O)C(C)(O)C1CC1)NCC(COC)C(C)C N1(CC)CCC12CCN(C(=O)NCC1(C(F)(F)F)CC(C)(C)C1)CC2 C1(NC(c2cc(C)oc2)=O)CCC(NC(=O)COCCc2cccs2)CC1 C(=O)(C1=CCCSC1)NCC1(C(N(CC(C2CC2)OC)C)=O)CC12CCC2 N1(CC(=O)NC2CCCC(NC(c3[nH]cc(C)c3)=O)C2)CC(=O)N(C)C1=O CC1CCCN2C1C2=O.c1(OCCCC(=O)N(C(C)(C)C)CC#N)ccccc1Cl c1(N2CC(CNC(COCC)=O)N(C)CC2)cc(C)c([N+](=O)[O-])cc1C(=O)OC C1(CO)CC(CO)CN(CCc2cn(CCC3CCCCC3)nn2)C1 C1(NC(c2c(C)scn2)=O)CC(CNC(C2(C)CCC(=O)N2)=O)C(O)C1 c1(CNC(c2c(N)non2)=O)ccc2c(c1)CCC2NC(=O)C#CC1CCCO1 C1(N(C(=O)CSC(C)C)CCC)CCN(C(c2cncnc2C)=O)CC1 N1(C(c2cn(C(C)(C)C)nn2)=O)CCCC(n2ccnn2)CC1 Cc1nnc2n1CC(C(=O)N(C)CC1(NC(c3csc(Cl)c3)=O)CC1)N(C)C2 c1(C(N2CC(CC(=O)Nc3c(CCC)onc3C)C2)=O)cnc2ccccc2n1 C1(C(N(CCCC#C)C)=O)C(C2CC2)CCN1C(c1ccncc1)=O Cc1nc(C(N2CCC2CNC(C2CCC3CC23)=O)=O)c(C)s1 C1(NC(C(CC)O)=O)CC2CCC1CC2NC(C1CCC(C(=O)N(C)C)CC1)=O CC(=O)C(C)CC(C)C(=O)N1CCC(NC(c2cccc(C)c2C)=O)C1C(C)C n1(CC(=O)N(CCN(C(C)=O)C(C)C)C)cnc2c(N)ncnc12 CC(C)(CC(=O)N1CCCC(NC(C2CC(n3cccn3)C2)=O)C1)C(F)(F)F CC(C)CC(C)C(=O)N1CCC(C)(CNC(C2(c3cccnc3Cl)CC2)=O)C1 N1(C(CN(CCC)C)=O)CC(OC)C(OC)C1C(=O)NC1CCC(N(C)C)C1 N1(C(C(CCN(C)C)O)=O)CCC2CCN(C(=O)Cc3cncnc3O)C2C1 C(CCC(=O)NC(C)CNC(C1(CCc2ccccc2)CC1)=O)OC C1(NC(c2n(C=C)ncc2)=O)CC2(CCCCN2C(=O)CC2CCN(C)C2=O)C1 c1(C(N2CC(C3OCCN(C(CC(C)(C)OC)=O)C3)C2)=O)cnc2[nH]c(=N)sc2c1 Cc1cc(N)cnc1C(=O)NCCCCC(C)NC(=O)Cn1ccc(O)nc1=O c1(C(C)C)ccc(C(C2CCN(C(=O)CCN3CCOCC3)CC2)O)cc1 N1(C(C(C)(O)C2CCCCC2)=O)CCN(CCNC(=O)C=Cc2ncco2)CC1 c1(OCCC(=O)NC(CNC(C2(CCC=C)CC2)=O)CC)cccc(Cl)c1 C(=O)(C(C)CC(C)C)NC(CCC)C(=O)NCCC1NC(=O)NC1=O C=CC(C)CC(=O)N(CCCCNC(=O)C(C)(C)NC(=O)Oc1ccccc1)C C1(CC(=O)OC)CN(C(C2CCCOC2)C2CC2)C(C)(C)CO1 C1(CC(=O)NCCC(=C)C)CN(C(=O)CNC(C)=O)CCC1C CCCC(C)C(C(=O)Nc1ccccc1Cl)N1CCCC(N2C(=O)CCC2=O)C1 c1(N2CCC(O)(C(C)NC(=O)Cn3cccn3)C2)nc2ccc(N)cc2s1 C1(C2CCCOC2)(NC(c2c(CNC(C3CC(CC)OCC3)=O)occ2)=O)CC1 C1(C(=O)Nc2ccc(C(=O)OC(C)(C)C)cn2)CN(S(C)(=O)=O)CCC1CO CCCC(C(=O)NC)NC(=O)CC1CCC(NC(=O)C(C)=C2CC2)CC1 C1(C(=O)NC(C2CCOC2)C#C)C=CCN(C(=O)C(C)(Cl)Cl)C1 C1(F)(CNC(C2CC(=O)NCC2)=O)CCCN(C(C2(c3cnc[nH]3)CC2)=O)C1 c1(C(N2CCCC(NC(C(=O)N(C)C)=O)C2)=O)cc2n(n1)CC1(CC1)C2 CC(C)C(C(=O)NC1CCN(C(c2ccnn2CCF)=O)CC1F)C(C)C N1(C(c2c(OC)csc2)=O)CC(NC(=O)CC=Cc2ccccc2)CC(C)C1 c1(C(=O)NCC2CCC(NC(C3(n4cncn4)CC3)=O)C2)ccc(Cl)cc1Cl C(=O)(C(CC(F)(F)F)c1ccc(Cl)cc1)N(C)CCNC(c1cccc(C#N)c1)=O n1(CC(N2C(C(C)NC(=O)CNC=O)CCC2)=O)ncn(C)c1=O C1(NC(C23CC(COC)(OC2)C3)=O)CN(C(=O)CN2CCC(C)CC2)CC1(C)C c1(C(N(CCCN(C(CC(C)C(F)F)=O)C)C)=O)cnc2cc[nH]c2c1 c1(CCC(N2CCCC(NC(C(CC)NC(C)=O)=O)C2)=O)ccc(OC)cc1F N1(C(C(CC)CN(C)C)=O)CCC2(CC2)CC1C(=O)Nc1cnn2c1CCCC2 c1(C(=O)NCCC2CCN(C(C(CCCOC)C)=O)C2)cc2cnccc2[nH]1 N1(C(CCC2CC(c3ccc(OC)cc3)C2)=O)CC(C)(C)OCC1(C)C C(CCC(=O)NC1(CNC(c2cnn(-c3cccnc3)c2)=O)CCOC1)N(C)C C1(CNC(c2cccc(CC)n2)=O)CCN(C(=O)C(O)CC(C)C)CC1C c1(C(N2CC(CNC(C(C)SCC)=O)C(C)C2)=O)c(O)nnc2c1CCC2 c1(C(=O)NC2CN(C(c3c(Br)cn(CC)n3)=O)CC2C)sc(C)c(C)c1C c1(NC(N(CC(=O)N(C)C)C(c2cccnc2)C)=S)ccc(F)c(Cl)c1F C(=O)(CC(C)(C)CC(C)=O)N1C(CN(C(C=CCC)=O)C)COCC1 C(=O)(C#CC1CCOCC1)NC1CC(NC(c2c(C)ccc(CC)c2)=O)C(O)C1 N1(C(C2(c3cccc(OC)c3)CCCC2)=O)CC(OCC(F)F)CC(O)C1 Cn1cnnc1C(=O)NC1(C)CN(C(=O)COCC2CCCO2)C1 CCC(C)(C(=O)NCC1(OC(C)(C)C)CN(C(N)=O)C1)N(C)C.C1(=O)CCC(C)N1 S(=O)(=O)(c1ccsc1C(=O)OC)NCCCC(CCC)N C12(C(=O)NC(CC3C(C)C3)=O)CCC(CC1)N(C(=O)COCP(C)(C)=O)C2 c1(C(N2CCC(C(CNC(COC)=O)(C)O)CC2)=O)c(C)cccc1[N+](=O)[O-] N1(CC)CCC2CN(Cc3cc(C(=O)OC)ccc3N)CC12 N1(C(c2c(OC)csc2)=O)CC(CNC(=O)CN2CCCC2C)C(C)(C)C1 C1(CC)CC(C(=O)NOCc2cn(CC(C)O)nn2)CCN1C(c1ccnnc1)=O CC1(C)CC(NC(=O)CSCC(F)(F)F)CN1C(c1cncc(-n2cccc2)c1)=O c1(C2(C(=O)NC3C(CNC(C(C)C#N)=O)CC3)CC2)ccc(Cl)cc1 C1(CNC(c2cnc(C)[nH]2)=O)CC2CCCC2N1C(c1cn(C2CC2)cn1)=O C1(C(N(CCN(CC)CC)C)=O)CCC(C)N(C(c2csc(Cl)c2)=O)C1 Nc1cc2c(cc1C(=O)NC1CCCCC1NC(=O)CN1CC3CC3C1)CCC2 c1(CNC(N(C)CCc2nccs2)=O)cnc(N(C)C)c(Br)c1 N1(C(c2c(CC)nn(C)c2)=O)CCC2(NC(c3cnc(S)n3C)=O)CCCCC12 C1(NC(c2c(C)oc(CO)c2)=O)CCN(C(=O)CNS(C)(=O)=O)CC1F C1(O)(CN(C(c2c(C)onc2)=O)C)CCN(C(C2CC(O)C2)=O)CC1 N1(C(C(C(C)C)F)=O)Cc2ccccc2C(NC(=O)Cc2ccnn2C(C)C)C1 c1(CC(=O)NCC(CNC(=O)CCc2nncs2)OC)ccc(F)c(Cl)c1F C(CS(=O)(=O)NCC(=O)N(C)CC1(O)CN(NC(C2CC2COC)=O)C1)OCC N1(C(C23N(C(C(COC)(F)F)=O)CC(C)(C2)C3)=O)CCCC(N=[N+]=[N-])C1 C1(OCC=C)CCN(C(=O)C(=O)NCC(C)CC2CCCC2)C1 C(=O)(NNC(=O)CC(C)(C)n1cc(CNC2CCOCC2)nn1)OC(CC)C c1(-n2ncc(C)c2)cccc(C(=O)NCC2CC(NC(C3CCC(C)S3)=O)C2)c1 N1(c2ncc(CN3C(C)CCCC3C)cn2)C(=O)c2ccccc2C1=O N1(C(=O)CN2CC=CC2)CCC2C(CCCN2C(=O)CC2CC2)C1 c1(C(N(CCN(CCCc2cccs2)C)C)=O)cc(CCO)on1 c1(C(=O)NCC(CC(C)C)NC(c2c[nH]cc2Br)=O)ccnc2ccsc12 CC(C)CC(=O)C(=O)NCC1(C(N2CCCCC2C2CC2)=O)CC2(CC2)C1 C1(NC(c2ccc(C#N)o2)=O)CCCC(NC(=O)CCc2ccncn2)CC1 Cc1ccc(C=CC(N2CCC(O)(CCNC(C3(C)C=CCCC3)=O)C2)=O)cc1 N1(C(C2CC(C3CC3)C2)=O)CCC2CCCC12C(=O)NCCC1CC1 c1(C(=O)NC(C)CCNC(=O)CC2COCCO2)ccccc1C(C)(C)C c1(C(N2C(CNC(CCC(=C)Cl)=O)CCCC2)=O)cc(Cl)ccc1CC CC1C2CCC(C2)C1C(=O)NC1(C(=O)NCc2cc[nH]n2)CCN(C)C1 N1(CC#C)CCN(C(=O)C(CC2CCC2)NC(=O)CCN(C)CC)CC1=O C(=O)(CCCC(CC)CC)N1CCN(C(C=C(CC)C)=O)CC(CO)C1 C1(C(=O)NC(CCCC)COC)CN(C)CCN1C(c1cc([N+](=O)[O-])n[nH]1)=O C=CCC(CNC(C1(C(N)=O)CC1)=O)NC(=O)Cn1cc(Cl)cn1 C1(NC(=O)NCCc2cccc(CC)c2)(CO)CCC12CCC2 C1(NC(C2(C)COC2)=O)CS(=O)(=O)CC1C(=O)NCc1cc(C2(C)CC2)n[nH]1 N1(C(c2c(COC)cco2)=O)CC2CC1C2C(=O)Nc1ccc(C(N)=O)cc1 Cc1cc(=NC(C)c2c(Cl)ccc(F)c2Cl)[nH]c(NCC2C(F)(F)C23CCC3)n1 c1(SC)cc(C(N2CC3CC(NC(=O)CC4C=CCC4)C2C3)=O)ccc1N N1(C(c2cc(C)on2)=O)C2CCC1C(C)C(NC(c1ccoc1Br)=O)C2 c1(C(=O)NC(C(=O)N(CC=C)C(C)C)C)cnoc1 N(S(=O)(=O)N1CC(CO)C(C2CC2)CC1(C)C)(CCCC)CC C(C)(c1ccco1)=CC(=O)NCC(COC)NC(=O)C=CC1CC1 CC1=C(C(=O)NC(C)CN(C(=O)C(C)C)C)Cn2nnnc2N1C C#CC12CC(CN1C(=O)CC(C)CNC(=O)C=CC1CCCC1)C2 c1(OC)cc(S(=O)(=O)NC(=O)C(N)C2CC2)c(Cl)cc1Cl c1(C(=O)NC2C(C)(CNC(C3(OCC)CCC3)=O)CCC2)cc2n(n1)CC(F)C2 C(C)(C(=O)NCC=CC(=O)NCc1ncc[nH]1)NC(C)=O CC1CCN(C(=O)CC2NC(=O)NC2=O)CCN1C(C1CC(C)(F)C1)=O C1(C(N2CC(O)(C(C)NC(C3C(OC)CCC3)=O)C2)=O)CCC(C(N)=O)CC1 C#Cc1ccc(C(N2CCCCC2C(=O)NC2C=CCCC2)=O)cn1 C1(CNC(C(C)OCC=C)=O)CN(C(=O)C=CSc2nc[nH]n2)CC12CCC2 c1(C(N2C(CNC(c3ccc(SC)o3)=O)C(C)CC2)=O)nc(O)nc(O)c1N C(CCCC(C)(C)C)N(C(=O)NC(C)C)C C1(CNC(CC2C(=O)NC(=N)S2)=O)CC2(CCN(C(=O)CC3CSC3)CC2)CO1 c1(C(=O)NCC2(CCNC(C3CCC(C)C3)=O)CC2)cc2c(F)cccc2[nH]1 NC1CCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CC12CCC2 C(CCCC(CO)NC(C1CCC(F)(F)C1)=O)NC(C1(OC)CCC1)=O c1(C(N2CC(C)C(CNC(c3cc(CF)on3)=O)C2)=O)cc(O)nc(Cl)c1 c1(SCC(N2CCC(Sc3ccc(CN4CCCC4)cc3)C2)=O)ccc(Cl)cc1 c1(C(N2CCC3(NC(C4CC5(C4)CC(F)C5)=O)C(C2)C3)=O)cccc2cncn12 CC(C)C(CCNC(c1cc(CO)[nH]n1)=O)NC(C1(Cl)CC1(C)C)=O CC1=C(C(=O)NCc2cncc(C(N3CC(CN(C)C)C3)=O)c2)CCO1 CCCCCC(C)CC(=O)N1C2CCC1C(CNC(=O)CC1(CO)CCCC1)C2 C(c1ccc(Cl)s1)=CC(=O)NCCCN(C(C1N(C(=O)NC)CCC1)=O)C(C)C C1(C(N(CCC(C)NC(c2c(Cl)cnn2C)=O)C)=O)CCC(=O)N1C CON1CCC(C(=O)NCCC2CN(C(c3cc4n(n3)CCC4)=O)C2)CC1 C1(C(N(c2cc(C(F)(F)F)ccn2)CCC)=O)CCc2ccccc2N1C(=O)OC C#Cc1ccc(CC(=O)N(C(CNC(C2CNC(=O)C2)=O)CC)C)c(F)c1 c1(N(C2CCN(C(C3CCN(C)C(=O)C3)=O)CC2)C)ncc(Cl)cc1[N+](=O)[O-] N1(C(=O)OC)CCCN(C(=O)CC2CC3(COC3)C2)CC1 c1(NC(CC(C)C)CCNC(=O)NC(C)(C)C)cc(C(=O)O)ccc1[N+](=O)[O-] C1(N(C)C(c2c[nH]ccc2=O)=O)CN(C(=O)C(O)C(F)F)CC12CC2 S(=O)(=O)(c1ccc(C#N)cc1)N1C(C(=O)NCc2c(C)nn(C)c2Cl)CCC1 N1(C(=O)CCc2ccc[nH]2)CCOC(c2cn(-c3cccc(Cl)n3)nn2)C1 c1(C(=O)NCC(CC=C)NC(C2C=CC=CC=C2)=O)cc(C)c(N)cc1F C12(NC(CCCC(C)O)=O)CCCN(C(c3cc(O)ccc3N)=O)CC1C2 C1(C(N2C(CC)CC(C)C2)=O)CCOCCN1C(=O)C(C)NC(N)=O c1(OC)cc(C)c(C(=O)N(C(C)CCNC(=O)CCc2cccc(C)c2)C)cn1 c1(C(=O)NCC2CC3CC3N2C(c2sccc2F)=O)cc2cc(Cl)ccc2o1 c1(C(=O)OC(C(=O)NC)C)cc(C#N)[nH]c1C C1(CCC=C)(C(=O)NC(C)C(C)SC)CN(C(=O)C(C)OCC=C)C1 c1(NC(c2nnnn2C(C)C(=O)OC)CCSC)nc2c(Cl)c(Cl)ccc2s1 C1(CCNC(=O)CC2CC(F)(F)C2)CCCN(c2nc(C3CCCCC3)ns2)C1 N1(c2n(CC)nnn2)CCC2(CCCCN(C(C3CCC4CCCCN34)=O)C2)C1 C1(C(=O)NC(CCCNC(CSC)=O)C)CCCN1S(=N)(=O)N(C)C C(c1ccc(Cl)cc1)=CC(N1CC(NC(C2(CCC=C)CC2)=O)C(OC)C1)=O C1(CC)CCCN(c2nnc(C3CC3)cc2C(F)(F)F)C1C(=O)OC C1(CNC(c2n(C)nnn2)(COCc2ccc(F)cc2)CF)CC2OC1C1CC21 C1(COC)(NC(c2ccc(C(C)C)nc2)=O)CCN(C(C2CSCC(=O)N2)=O)C1 C1CC(=O)N1C(C)C.C(CC(C)C)SCC(=O)NC1C(CC(=O)OCC)C1 N1(C(CC(C)NC(C2CCCC2)=O)=O)CCN(C(=O)Cn2cncn2)C2(CCC2)C1 C(=O)(C(O)C(F)(F)F)NC1(CNC(C2CCN(C(C)=O)C2)=O)CCCC1 N1(C(C)(C)C)CCN(C(=O)C(N2CCC(C(C)(C)C)(CN)C2)=O)CC1 C(=O)(C1CCc2c[nH]nc21)NCC(CNC(c1n[nH]c(C)c1Br)=O)F C(CCCNC(=O)CC(C)C1CC1)(c1ccccc1)NC(C=CCCC)=O C1(OC)COCC1NC(=O)C(c1ccnn1C)C.C1(=O)C(C)(C)N1C1CC1 N1(C(C(C)(C)N(C)C)=O)CCC(O)(C2(NC(c3cc([N+](=O)[O-])c[nH]3)=O)CC2)CC1 C1(NC(C=NOC)=O)CN(C(C2CC(=O)N(C(C)C)C2)=O)CC1n1ccnn1 N1(C(C(C=C)C)=O)CCC2(CCCN2C(c2csnc2C)=O)C1 c1(CNC(CNC(C(C)NC(CC)(C)C)=O)=O)ncnn1C C(=O)(CC1=NNC(=O)C1)NCC1(NC(c2ccc(CC)c(N)c2)=O)CCOC1 CC(C)CC(C(=O)N1CC(C)C1C(N1CCC1C1CCC1)=O)N(C)C CCC(C)C(C)(O)CNC(=O)C(F)C1CC(NC(c2cncc(C)c2)=O)C1 c1(C(=O)OC(C(C)SC)C)cc([N+](=O)[O-])ccc1N(C)C C1(NC(C(C(C)C)C)=O)C(C)(C)CN(C(c2ccc(C(C)(C)C)s2)=O)CC1(C)C CC1CC(C(=O)Nc2c(F)cccc2Cl)CC(C)C1 C1(C2CC2)(C(N2CC(CNC(COC(CC)C)=O)C(O)C2)=O)CC=CC1 C1(CN(C(C(C)C2CCCC2)=O)C)CCC(NC(C2(C)CC=CCC2)=O)CC1 c1(OC)cccc2cc(C(=O)NCc3ccnn3C(C)C)oc12 c1(OC)ccnc(F)c1C(N1CC(CO)(NC(=O)CC2CCCN(C)C2)C1)=O CCCC(C)CC(=O)N1CC=CC(NC(c2c[nH]nc2C(C)(C)C)=O)C1 Cc1cc(C)nc(-c2cn(CC3CCN3C(=O)CO)nn2)n1 C1(C(=O)NCC(C)NC(=O)C(C)NC(=O)OC(C)(C)C)C2CCCCCC12 c1(C(=O)NC2C(CNC(C(C(C)(C)C)O)=O)CC2)ccc2nc(O)[nH]c2c1 C12(CNC(c3cc(COC)on3)=O)CCC1CN(C(=O)C(F)(F)c1nccs1)C2 C(=O)(C(C)(F)C(C)(C)F)N1CCCC(N(C(c2ccc(CC)c(Cl)c2)=O)C)CC1 CCC(C)C(C)C(=O)NCC1CC(NC(=O)C=CC)C1.c12ccccc1C(=O)N2 n1(CC#C)cc(CNC(=O)C(CNC(=O)CCC2CCOC2)N(C)C)cn1 CC1CC(CNC(C2CC2c2cccs2)=O)CN(C(C2(C)CCSCC2)=O)C1 O=C1CC(C(=O)NC2CN(C(c3cccnn3)=O)CC2n2ccnn2)CCN1 CCCC(Cc1ccccc1)NC(=O)CN(CCc1nccs1)C(C)C CCCCC(C)(c1nnnn1CC(F)F)NC(CC(N)=O)c1ccccc1 CN1CCC(C)(C(N2CCC(C)(CCNC(=O)CC3CCC3)C2)=O)C1 C1(CNC(c2ccc(C(N)=O)nc2)=O)CC(F)(F)CN1C(=O)C(F)OC(F)(F)F CCCCC(=O)N1CCCC1C(C)NC(=O)C(C)SCC C1(CNC(C(C2CCCC2)NC(c2cn(CC)nn2)=O)=O)OCCC1(C)C c1(C(=O)NCCC(C)NC(CC2ON=C(CC)C2)=O)c[nH]c2c(Cl)cccc12 C1(NC(C=CCN(C)C)=O)CC(CNC(=O)C=CI)C1 C1(c2cn(C3CCC(N(C(CC(C)(C)C4CC4)=O)C)CC3)nn2)CCC(C)CC1 C1(CNC(=O)C=Cc2cc[nH]n2)CC2CCC1N(C(=O)CSC1CC1)C2 c1(C(N2CCC(CC(=O)Nc3ccc(C)cc3Br)CC2)=O)c[nH]nc1S(N)(=O)=O N1(C(C2C(CC)CCO2)=O)CCN(C(c2ccc(C)o2)=O)CC1COC N1(C(C(CCCC)O)=O)CC2CC(C)N(C(=O)C(CC(C)C)C(N)=O)C2C1 c1(C(=O)NCC(C)CNC(=O)C=Cc2ccc[nH]2)cc2ccnc(Cl)c2s1 C1(CNC(=O)CC(F)(F)F)CC2CCC1N2C(C1(F)CCOCC1)=O c1(C(N2CC(NC(c3c(CC)n(C)nn3)=O)C(C)CC2)=O)cnc2[nH]cnc2c1 c1(C(N2C(CCCNC(C(F)OC)=O)CCC2)=O)nc(SC)n2ccccc12 C(=O)(CC1CCC(C)(C)c2ccccc21)NCCN(C(=O)CC(C)(O)COC)CC C1(NC(CC(C)C2CC2)=O)CN(C(=O)CCCC2CC2)CCC12CCC2 CCC(C)(F)C(=O)NCCN(C(=O)C(C)SC(C)C)C c1(C(=O)NCCC)ccc(N=S(C)(C)=O)s1.C12CSCN1C(=O)COC2=O c1(C(=O)NCCC2CCC(NC(c3c(C)onc3)=O)C2)ccc(F)cc1Br Cc1[nH]nc(NC(=O)CN(CCO)CCn2ccnn2)c1C C1(C(N2CCC(CN(C(C(CCC)N(C)C)=O)C3CC3)CC2)=O)CC2COCC2C1 c1(CCNC(CC(CCSC)O)=O)c(C)[nH]c2ccc(Br)cc12 N1(C(C2C(CCC)CN(C(=O)CC3OCCO3)C2)=O)CCOCC(C)C1 C1(C(N2CC(NC(c3oc(CC)c(C)c3)=O)C(C)C2)=O)CC2OC(C)(C)OC2C1 CCCC(CC)CCC(=O)N1CCCC(CC)C1C(N1CCCC1C)=O n1(CC)cnc2nc(N3CC(C)C(C)C3)nc(NCC(C)(C)SC)c12 c1(C(=O)Nc2c(NC(C)=O)cccc2)c(C)nc2c(OC(F)(F)F)cccn12 N1(C(C2C(NC(=O)C(c3ccccc3)O)CC=CC2)=O)CCC(CO)(CO)CC1 C1(C(=O)NCC2CN(C(=O)CCOCC(F)(F)C(F)F)C2)CCC(C2CC2)CC1 C1(CNC(c2c(CC)cco2)=O)CCC(C)N(C(=O)Cc2csc(C(C)C)n2)C1 N1(C(c2ccc(OCC#C)cc2)=O)CCC(NC(=O)CCC2CCOC2)C(O)C1 c1(C(=O)NC2C(C)CN(C(C3CC3(C)C)=O)CC2)cn(C)c(=O)nc1O CN1CCC(C(=O)NCC2(CF)CC2)(NC(=O)CCC2(C#N)CCC2)C1 N1(C(c2nc(C)sc2)=O)CCCC2CC(NC(=O)CC3OCCC3(C)C)CCC12 c1(N(CC(C)C)C(=O)NC(C#C)C2CC2)cccc(N(C)C)c1 c1(C(N2CCCC(N(C(c3c(C)ncn3C)=O)CC)C2)=O)cc(F)c(O)c(F)c1 C12(CNC(c3n[nH]c(C)c3Cl)=O)CCC(CC1)N(C(c1cc[nH]n1)=O)C2 C(=O)(CCC(C)CC)NCc1c(C(=O)NC(CCCC)CO)n[nH]c1 C(=O)(C(O)C(F)(F)F)N(CC(CC)NC(=O)C(C)(C)c1ccccc1)CC CCC(C(=O)NC(C)(C)CC(=O)NC(CF)C(F)(F)F)C(F)(F)F C1(NC(CSCCC)=O)CC2C1CCN2C(=O)C=CCN(C)Cc1ccccc1 CCCCC(O)CC(=O)NCC1CC2CCC(C1)N2C(=O)C=CC(C)(C)C CC1=C(C(=O)NCC=C2CCN(C(C3CCC4(CCC4)C3)=O)CC2)CCCC1 N1(C(c2cnn(CCCC)c2CC)=O)CCC2(CCCN2C(=O)C=CC2CC2)C1 Cc1ccc(C(=O)NC2CCCC(CN=c3[nH]nco3)C2)nc1 C1(CCOC)(NC(=O)C(c2cnn(C)c2)C)CCN(c2nc(Cl)c(C(C)=O)s2)C1 S(=O)(=O)(CC(=O)NCC1CCN(C(c2cnco2)=O)C1)N(CC)CC c1(C(=O)NC(CCCC)CNC(c2cnn(C)c2)=O)ncccc1S(=O)(=O)CC C1(C(=O)OC)(CC)CCCCN1C(C1C(C)(C)C1(C)C)=O C1(CN(C)C(C2(C)CCCO2)=O)CCCN1C(C1(CC2CC2)CCCC1)=O C(C(C)(C)C(=O)NCc1ccc(C#N)s1)N(C(C(SC)SC)=O)C CC(CC(C)NC(=O)C(CO)NC(N)=O)NC(=O)CC1CCC(=O)N1 N1(C(C(C)Sc2cccnn2)=O)CCC(C)C1c1cn(C2CC2)nn1 C1(c2n(CC)nnn2)(Nc2ccc(N(C)C)cc2)CCCCCC1C C1(CC=C)(NC(C2CC2C)=O)CCN(C(c2cnc(OC)c(Br)c2)=O)C1 N1(C(C(C)=C(C)C)=O)CCCN(CCNC(C2CCC(O)C2)=O)CC1 N1(C(=O)Cn2ncnn2)CCN(C(C2CC2(Cl)Cl)=O)C2CCC12 Cc1ccc(SCC(=O)NC2(COC)CN(C(C3CC3C(N)=O)=O)C2)cc1 N1(C(CCSC)=O)CCC(N(CCO)C(C2CC2C(C)(C)C)=O)C1 C1(C(N(C2CCCNC2=O)C)=O)C2CC3C(C2NC(=O)CCc2cnn(C)c2)C13 C1(C(=O)NCC(=C)CCNC(C2CC(CC(C)(C)C)C2)=O)CCN(C)C(=O)C1 C1(C(=O)NCC(C2CCCCC2)NC(c2nocc2Cl)=O)COCCOC1 C1(=O)CCCCN1.C(=O)(CCC=CC)NCCOCCC=C N1(C(C2N(C(CC(C)C)=O)CCCC2)=O)CC=C(CNC(=O)C(C)C2CC2)CC1 CC(C)(C)CCCCC(=O)NCC1CC(C(=O)NCc2ccnc(O)c2)C1 C(=O)(CC(C)(C)CNC(=O)C(C)(C)C(N)=O)N1CCC(C(=O)NC)C1C N1(C(c2c(C)ccnc2O)=O)CC2CCN(C(=O)CC3CC34CC4)CCC2C1 CCC(C)(C)C(O)C(=O)N1CCCCC(NC(C2CCOCC2(C)C)=O)C1 C12C(C)CCN1C(=O)C(C1CC(C(=O)OC)C1)C(C)NC(=O)C2.N(C)C.OC CCC(CC)C(CNC(C1(C(=O)N(C)C)CCCOC1)=O)N1CCOCC1 N1(C(c2c(CC)n(C)nn2)=O)CC(CNC(=O)CN2CCCNC2=O)CC(C)C1 CCCC(C)CC(=O)NCC1CC(C(F)(F)F)CN1C(C1CC(F)(F)C1)=O CCC1=C(C(=O)NC2CCC2NC(C2CC(C3CCOCC3)=NO2)=O)CCCO1 C1(C(=O)OCC(=O)N(C)Cc2cccc(SCC(F)(F)F)c2)CC(=O)NC(=O)N1 c1(CCC)ccc(C(=O)NC(C)CN(C(=O)C2=CC(C)(CC)C2)C)cc1[N+](=O)[O-] Cc1c(C(N2CC(CC(C)NC(C3(O)CC3)=O)C2)=O)sc2ncnc(N)c12 c1(C(=O)OC)cccc(-c2cccnc2)c1.C12(CCCO1)C(=O)OC2 C(=O)(C(C)(C)C(O)CC)NC1(CC=C)CN(C(=O)CC=C(Cl)Cl)C1 Cc1c(F)cc(C(=O)NCC2CCN(C(c3ccc(C#N)cc3)=O)C2)cc1F N1(C(CNC(CCC)=O)=O)CC2CC(C(N3CC(C)(C#N)C3)=O)C(C2)C1 c1(C(=O)NC2CCCCCN(C(=O)CC34CCCC3C4)C2)cnc2ccoc2c1 C(=O)(CC(F)(F)C(F)(F)F)N(C1CCN(C(C2CC2(F)F)=O)C1)CC n1(CC)nc(CCC(N2CC3COC(C2)C3O)C(=O)NC2CC2)c2ccccc12 C1(C)(C(=O)NCC2(O)CN(C(CN(C)C(=O)OC(C)(C)C)=O)C2)CCCC1C N1(CC)CC2(CN(C(C3CCOCCN3C(=O)C=CCOCCOC)=O)C2)C1 CCCCC(O)CC(=O)NC1(CO)CN(C(=O)C=CC2(C)CCOCC2)C1 CC(C)CC(F)C(=O)NC1CCCCCC1NC(=O)CC(=O)N(C)C C1(CNC(C2(C(C)=O)CC2)=O)CCCN1C(C1(C)CC1(F)Cl)=O C(=O)(C(C)(C)CC(F)F)N1CC(C(=O)NCC(F)CO)CC(C)C1 c1(C(c2nnnn2-c2ccccc2)NC(c2ccccc2F)C)cc(C)ccn1 C(=O)(C(O)C(C(C)C)OC)NCC1(NC(C(CC)SC)=O)CCOCC1 C1(COC)(CNC(=O)CC(C)C(C)C)CCN(C(c2ccc(C(C)C)s2)=O)CC1 N1(C(C(C=C)O)=O)CCC(NC(c2ccc(N3CCOCC3)nc2)=O)C(F)C1 Cc1nccn2ncc(C(=O)NC(C)(C)Cc3cc(F)cc(F)c3)c12 CC1=C(c2ccco2)CN(CC2CCCC2C(F)(F)F)CC1 N1(C(C=CC(CC)C)=O)CCCC1(C)CNC(=O)C=Cc1cscn1 C#CCCCCCC(=O)NCC1CCN(C(c2cnn(CCO)c2)=O)C1 c1(C(=O)NCC2(NC(c3cnn(C)c3N)=O)CCOCC2)cnn2c1CCC2 N#Cc1cccc(S(=O)(=O)N2CCC(C(=O)NC(=O)N=c3[nH][nH]cc3C#N)CC2)c1 C1(CS(=O)(=O)N)CC2(CCC2)C1.C1CCCC(F)C1 CCC(CC(=O)NC1CCN(C(c2nscc2Br)=O)C1C(C)C)OC N1(C(C2(C)CCSCC2)=O)CC2CCN(C(=O)CCCN3CCOC3=O)C2C1 C1(O)(COC)CCN(C(=O)C(C2CC2)NC(c2cc(F)c[nH]2)=O)C1 CC1C(NC(=O)C(C)S(C)(=O)=O)CCCN1C(c1ccnc(C2CC2)n1)=O N1(C(c2cc(C)no2)=O)CCCOC(CNC(c2ncccc2C(F)F)=O)C1 CC(N=c1[nH]c2c(c(=NCCN(CC(F)(F)F)C)[nH]1)CCCC2)C1CCOC1 CCC(CC)(C(=O)NCC=CCC(N1CC(C)(O)C1)=O)C(C)C c1(NC(C)=O)cccc(C(=O)N(C2CCN(C(=O)CC(F)(F)F)CC2)CCO)c1 C(=O)(CCCCCC(C)C)NCC12CN(C(c3n[nH]c(C)c3Cl)=O)C(C1)CCO2 c1(C(C)C(=O)NCC2CN(C(C34CC(C3)C4)=O)C(C)(C)C2)ccc2c(c1)OCO2 c1(OC)cc(C(=O)NC2CN(C(=O)CC(C)C)CC(C)(C)C2)cc([N+](=O)[O-])c1Cl c1(C(=O)NC(CC=C)CNC(c2c[nH]c(=N)o2)=O)cc(Cl)c(F)cc1F c1(C(N2C3CC(NC(c4cc(SC)c(N)cc4)=O)(C3)C2)=O)cn2ncccc2n1 c1(C(N(CCC2CCN(C(C(CN(C)C)O)=O)CC2)C)=O)cc(O)c(F)cc1N N1(C(C2(Cl)C(C)(C)C2)=O)CCCCC(CNC(=O)CCn2cc[nH]c(=O)c2=O)C1 CCCC(CCC)C(=O)N1CCC2CC12C(=O)NC1CCC(C)(O)CC1 c1(OC(C)(C)C(N2CC(C)(C)C2c2nccn2C)=O)ccnc(Cl)c1 CC1CCN(C(C2CN(C(c3cccc4[nH]ccc34)=O)CC23CC3)=O)CC1(F)F C1(NC(C(CC)C)=O)CCCC12CCN(C(c1cc(O)ccc1Br)=O)CC2 C1(NC(C(C)CC2CCCC2)=O)CC2CCC(C1C)N2C(c1ncccc1F)=O Cc1c(C(=O)NC(C(=O)N2CCCCC2CF)C(C)(C)C)cccc1O c1(N2CCCC(C)(C(=O)NCc3c(C)cccn3)C2)ncnc2[nH]cc(C#N)c12 C1(CC)CCC(NCc2cn(C(C)C)nc2C(C)(C)C)CC1 CC1(C)C(C(N2CCC(NC(=O)CNC(c3ccncc3)=O)C2)=O)CCS1(=O)=O CC12CCN(CC1)CC2C(=O)NCC(O)CNC(=O)CSCC(N)=O C12CC(C(F)(F)F)CN1C2=O.c1(C(=O)NCC(=O)NC2CC2)nc[nH]n1 C1(SC)COCC(C)O1.C12(CN(C(=O)CNC(C)=O)C1)C(=O)N2 Cc1cc(C(=O)NC2CC3CCC2CN(C(C2CCCS2)=O)C3)c2[nH]cnc2c1 N1(C(C)C)CCC(N(C(=O)CNC(=O)CCc2cccs2)C)C1 C1(CNC(=O)C(F)CC2CCOC2)CN(C(C2CCCSC2)=O)CCCO1 C(=O)(C(n1nnnc1C)=Cc1ccc(F)cc1)N(CC)CC1CCCO1 N1(C(C2(CC=C)CCCC2)=O)CCOC(CNC(c2cc(C(F)F)ncn2)=O)C1 C1(C(C)C)(C(=O)NCC(C)(O)CNC(C2CN(C3CCC3)C2)=O)CCNC1=O C1(F)(c2cn(C(C)C(=O)N3CC3)nn2)CCN(C(c2cccc(C(=O)O)c2)=O)C1 C1(C(=O)NCCN(C(c2c(C)noc2C2CC2)=O)CC)CCN(C)C(=O)C1 N1(C(C2C(C)C2)=O)CCC(F)(CNC(c2cccc(CC(F)(F)F)c2)=O)CC1 C1(C(=O)NCC2N(C(C3N(C)CC(O)C3)=O)CCOC2)CN2CCC1CC2 CC1(C)COCC(CC(=O)NCC2(C)CCN(C(=O)C3=CCCO3)C2)O1 c1(C(N2C(C(COCC)(C)C)CCC2)=O)c(NC(=O)C2CC2)sc(C)c1C c1(C(N(C(C)CN(C)C(C23CSC(C2)C3)=O)C)=O)ccnc(CN(C)C)c1 C1(CNC(C(C2CCCCC2)OC)=O)CC2CCC1N2C(c1cc(Cl)on1)=O Cc1ccc(C(=O)NC2CCC(C)N(C(=O)COCc3ccccc3)C2)nc1C c1(C(N(CC(C)NC(C2CCC(O)C2)=O)C)=O)cn2cccnc2n1 CC1(C)COC(CC(=O)NC2CCCC(CNC(c3sccc3F)=O)C2)C1 C1(NC(C=C2CCC(C)C2)=O)CC(Nc2ncc3ccnc-3[nH]2)C12CCOCC2 c1(N(C)Cc2cccnc2)ccc(SC2CCC2)nc1.C12CCN(C1)C(=O)NC2 C1(N(C)C(c2cc(C(N)=O)[nH]n2)=O)CN(C(c2ccnc(Cl)c2)=O)CC12CC2 N1(C(c2c(C)ocn2)=O)CCN(C(C2(CC(F)F)CCC2)=O)CC12CCC2 N1(C(C(C)NC(C)(C)C)=O)CCC(NC(c2ccccc2CO)=O)C(C)(C)C1 N1(c2nc(C)nc(C(C)C)c2)CCN(C(=O)C2=CC(C)(C)C2)CC(C)(F)C1 C1(NC(CC(C)(F)F)=O)CCN(C(c2c[nH]cc2C(F)(F)F)=O)CC1(C)C c1(OCC)c(C)cc(-c2cnc(C(=O)NCC(C)(C)F)nc2)cc1C c1(OC)ncc(C=CC(N2CCC(CNC(=O)C=C(C)C3CC3)C2(C)C)=O)cn1 C1(C(=O)NC(CC=C)CNC(=O)CCc2cc(C)[nH]n2)CC12CCCCC2 C1(CCCCNC(C(C)C2CC2)=O)CCCN(C(=O)CCN2CCCC2)C1 C1(C(=O)NC(C2CCCC2)CNC(c2ccncc2)=O)CCCC2CCCN12 c1(C(N2C3CC(NC(=O)CC4(N5CCCC5)CC4)(C3)C2)=O)occ2c1CCCC2 c1(COC(CCn2cc(C(CCC)OC)nn2)=O)n[nH]c(-c2cccs2)c1C CCCCC(C)CCC(C)(c1nnnn1CCC)NCCCc1ccco1 c1(C(=O)NCCC2CCN(C(c3ccn(COC)n3)=O)C2)ccc2nn[nH]c2c1 C(C1=CCN(C(=O)COC2CCN(C)CC2)CC1)NC(CC(C=C)C)=O N1(c2n(CCOC(C)C)nnn2)CC2CCN(c3ccc(Cl)cc3)C2C1 C1(CC(C(=O)OCC)F)(NC(c2ccc(C)c(Cl)c2)=O)CCCCCC1 N1(C(CNC(CCC)=O)=O)CC2CC1(CNC(c1cccc(CC(C)C)c1)=O)C2 C1(C)(C(N(CCC(C)NC(=O)C(C)(C)CF)C)=O)CNC(=O)C1 c1(C(N(C)CC2C3CN(C(C4(C)CCNC(=O)C4)=O)CC23)=O)cc2n(n1)CCCN2 N1(C(C(C(C(C)C)OC)O)=O)CCC2CCCC(C1)N2C(=O)COC1CCOC1 c1(C(N(C2CC3CC2CN3)C)=O)ccc(Oc2ccc(Cl)cc2)cc1 C1(O)(C(N2CCC(O)(CNC(C3CCC(C)CC3)=O)CC2)=O)CCC(C)(C)CC1 N1(C(c2nccc(C)n2)=O)CC(CNC(c2n[nH]cc2C(C)C)=O)OC(C)(C)C1 c1(NC(CC2(C)CCN2C(=O)CCCC(F)(F)F)=O)ccc2c[nH]nc2c1 C1(C(N(CC(CC)NC(C2(C)CCOCC2)=O)C)=O)CC2(C1)CC(O)C2 CCCCC(CC)C(=O)N1CC2CCC(CNC(C3SCCS3)=O)C2C1 c1(C(N2CC(C(C)NC(=O)C(C)(Cl)Cl)C2)=O)cccc2c1CCC(=O)N2 Cc1ccc(C(=O)NC2CCC2)cc1C1CNC1.N12CCOCC1CCOC2=O c1(C(N2CC(C)(NC(C(COC)O)=O)C2)=O)c(C)cc(C)nc1S CC(C)(C(c1nnnn1C1CCC1)Nc1cn(CC2CC2)cn1)C1CCCCC1 CCCCCCCC(=O)N1CCC(CF)(NC(=O)Cc2cncn2C2CC2)C1 N1(C(Cc2c(C(=O)OC)n(C)nc2)=O)CCN(C(c2cnnn2C)=O)C(CO)C1 c1(C(=O)NCC2(O)CC(CNC(C3CCC(C)(C)C3)=O)C2)cnn2c1CCC2 N1(C(C2CC(=O)C2)=O)CCC2(CCC2)C(NC(=O)Cc2cnccn2)C1 C1(C(N2C(CNC(=O)C(F)CC3CC3)CCCCC2)=O)C2CCC3C(C2)CC13 N1(C(C2C(COC)(CC)C2)=O)CCC(C(=O)OC(=O)CC(C)(C)OC)CC1 c1(NC(=O)NC(C(F)(F)F)c2ccccc2)cccc([N+](=O)[O-])c1 c1(C(N2C(C(N3CC(n4cccn4)C3)=O)CC2)=O)ccnnc1O C=CC1(C(=O)NCCC2CC2C2CC2)CCN(C(=O)C(=O)CC(C)C)C1 C#CC1(C(N2CC3C(COC)C3C2)=O)CCN(C(C2CC(C3CC3)=NO2)=O)C1 C(=O)(CC(C(F)(F)F)n1ccnc1)N(CCN(C(CC(C)(C)SC)=O)C(C)C)C c1(C(=O)Nc2cccc(NC(CS(C)(=O)=O)=O)c2)cccc2nccnc12 C(CCCCC(=O)NC1CCN(C(=O)Cc2[nH]cnc2C)CC1CO)OCC N(C1CCCc2cc(CNC(C3(C)CCC3)=O)ccc21)C(CC(C)(C)OC)=O C=CCC(CNC(=O)CC(C)NC(C)=O)NC(=O)C=CSC C1(NC(=O)C(F)(F)C(O)C2CC2)CCN(C(=O)C(F)C2CCC2)CCC1CO N1(C(c2cc(C)sc2)=O)CCN(C(=O)CCN2CCC(F)C2)CC12CC2 c1(OCC)ccc(CNC2CCCCCC2c2ccccc2)c(Cl)c1O N1(C(CC(C)C2CCCC2)=O)CCC=C(CNC(C2CC(=O)NC2(C)C)=O)C1 CCC(C(=O)OC)C(=O)NC1CCN(C(C2C=CC=CC=C2)=O)CC1CC c1(C(=O)NCC(C2CC2)NC(C(C(C)C)O)=O)nn(C)c2ccccc12 N1(C(C=CC=CCCCCC)=O)CCCC(C(=O)NCC(C)C(C)O)C1CC C1(C(=O)OC)CC2CCC1N(C(c1c(Br)ncn1C)C(=O)NCC1CCOC1)C2 N#Cc1cncnc1C(=O)NCC1CC(CNC(=O)C=C2CCCC2)CO1 C1(C2CC2)(CNC(C2OCC(C)C2)=O)CCN(C(c2cc(Cl)cc(F)c2N)=O)C1 C#CCC(C)(C)C(=O)N(CC(O)CN(C)C(c1cnc[nH]1)=O)C O=C(CC(F)(F)C(F)F)N1CCCC(N(c2ncc(I)cn2)CCO)C1 c1(C(N(C2CCN(C(=O)CC3CCC(C)C3)CC2)CCOC)=O)cc(C)cnn1 c1(C(N2CCC(CNC(COC)=O)CC2)=O)cc(Cl)c(F)cc1O Cc1cc2[nH]c(C(=O)NC3CC(C)N(C(=O)C(C#N)=CC4CC4)C3)cc2s1 Cc1cn2ccnc(C(=O)NCC(O)CCNC(=O)C3=COCCC3)c2n1 C1(NC(c2cccc(F)c2)=O)CC2CC1CN(C(c1coc3ccccc13)=O)C2 CC1CN(C(C2(F)CC=CCC2)=O)CC1c1cn(CCNS(C)(=O)=O)nn1 C(C)(c1ccccc1C)=CC(=O)NCC1N(C(C2CC(CC)C2)=O)C2CCC1C2 CC(CNC(c1ccsc1)=O)(CO)NC(=O)CCCNC(N)=O Cc1c(C(=O)NC(C)CNC(c2cnn(C)c2C)=O)cccc1O C12(CCC1)CC(=O)N(CCOC)CC(=O)N2.C1(SC)CN(C2CCC2)C1 C1(CC(=O)NC2C3CN(C(C(CC)NC(N)=O)=O)C2C3)CC(C)(C)CCO1 Cc1ncoc1C(=O)NCc1cn(CC(=O)NCCC(=O)N2CCCC2)nn1 N1(C(CCCOC)=O)CCCC(NC(c2oc(SC)cc2C)=O)C1C C1(C(=O)NCC(CNC(c2cnc(OC)c(F)c2)=O)O)CC2CCCCCC12 c1(CCC)ccc(C(=O)NC23CCC2CN(C(=O)C(C2CC2)OCC)C3)cc1N Nc1cc(C(N2CCCC(C(N3CC(OCc4cccs4)C3)=O)C2)=O)cc(O)c1 N1(Cc2c(OC)ccc(C)c2)CCC2(CCN(C(=O)CN3CCCS3(=O)=O)C2)C1 N1(C(N2CC=CC(NC(=O)COC3CCCC3)C2)=O)CCC2CC1CO2 C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC1(C)CCCN(C(C(C(=C)Cl)(C)C)=O)C1 N1(C(C(C)OC(C)(C)C)=O)CC=C(C(=O)NCC2(C)CCCC(=O)N2)CC1 Cc1cccc(-c2cccc(C3(NC(c4ncncc4I)=O)CC3)c2)c1 c1(NC(=O)NC(c2ccccc2F)c2cc(C)no2)cc(F)cc(Cl)c1 C(=O)(C1=CCCCC1P(C)(C)=O)NC1CN(C(C2CN(C)C2)=O)CC1(C)C c1(CC(=O)NC2CC(C)(NC(=O)C3=CCC3)C2)ccc(Br)cc1[N+](=O)[O-] C1(O)(C(N(CCCN(C(c2nn(CC)c(=O)cc2)=O)C)C)=O)CCCC(C)(C)C1 C1(Nc2nccc(C)n2)CCN(C(c2c(C)cccc2C)=O)CC1O c1(C(N2CC(COC)N(C(=O)Cc3nnc(C)s3)CC2)=O)c(Cl)ccc(F)c1C C1(NC(c2c(Cl)cc(C)s2)=O)CC2CCC(C1C)N2C(c1nc(C)n(C)n1)=O n1(CC(=O)NCCCC(C)NC(c2nn(C)cc2Cl)=O)ccccc1=O O=C(CC(C(F)F)c1cccc(F)c1)N1CCC(N2CC(O)C2)C1 C1(C(=O)NCC2CCC=CCC2)CC=CCN1C(c1ncccc1O)=O N1(C(c2nn(CC)nc2C)=O)CCCC12CCCN(C(=O)CC1CC(C)C1)C2 C1(C2CC2)(NC(C23N(C(C4CCCC(C#N)C4)=O)CC(C2)C3)=O)CCCCC1 C1(NCC)CCC(N=c2nc(NCCC3CCC3)c3c([nH]2)CCS3)CC1 N1(C(C2C(OCC)CC2)=O)CCC2(CCC2NC(c2nc(=O)n(C)[nH]2)=O)CC1 c1(OC)ccccc1C(N1CCCCC1CCNC(c1ccoc1Br)=O)=O c1(OCC(C)(C)C)ccc(CC(=O)NCCC(C)(C)NC(C2CC(O)C2)=O)cc1 c1(C(N2C(CCNC(c3c(C)ccs3)=O)CSCC2)=O)ccc(F)c(C(F)F)c1 CCC(C)(C)C(O)C(=O)N1CC2(CC2)CC1CNC(=O)Cc1cccc(Cl)c1F C(=O)(C(F)CC(C)(C)NC(C1CCSCC1)=O)NCc1nc(O)cc(C)n1 c1(C(=O)NCC2CC(NC(C(CCC)N(C)C)=O)C(O)C2)nc2cnccc2s1 CCCCC(C)(F)C(=O)NCCCOCCCNC(=O)CC1CC1(Cl)Cl c1(C(=O)NCCCN(C(C(C)=C2CC2)=O)C2CC2)ccc2nc(CO)[nH]c2c1 C(CCN=c1nc2ncn(C)c2c(COC2CCOC2)[nH]1)NC(c1nccs1)C CCCC(F)C(=O)NC(Cn1ccnn1)C(N1CCCC(CN(C)C)C1)=O Cc1cc(Br)cc(C(=O)NCC2(NC(c3cncn3C)=O)CC2)c1C c1(CCC(=O)NCC23CC(CNC(CC=C=C)=O)(OC2)C3)nc2ccccc2s1 c1(C(=O)NCC2CN(C(C3(Br)CC3)=O)C2)ccccc1Cn1cccn1 C1(CNC(C(C)(C)CC2CCOCC2)=O)CC2CN(C(=O)C3=CSCS3)CC12 C1(CNC(C=CC(CC)=CC)=O)CC(C)N(C(c2cc(CC)c[nH]2)=O)C1 N1(C(c2cc(F)cc(Br)c2)C(=O)NCCOCC)C2CCC1CN(C)C(=O)C2 C(=O)(C1c2c[nH]nc2CN1CC1ON=C(C)C1)NCC1CC(C)(C)CCO1 O=C(N=c1cc(C2CCC2)o[nH]1)NCC1CCCN1CC1CC1 CC(C(=O)NCCN(C(c1ccsc1)=O)C1CC1)C(C)n1cccn1 N1(C(c2cc(C)sc2)=O)CCC2(CCN(C(c3cc(C#N)cn3C)=O)C2)C1 c1(C(N(CCCN(C)C(C2(n3cccn3)CC2)=O)C)=O)cccc2oc(O)nc12 c1(SC)nc(NC2CC3CN(C(=O)COC4(C)CCCC4)CC23)cc(C(F)F)n1 Cc1nc(C(=O)NCC2CCC(NC(=O)C(CO)N(C)C)CC2)c2ccnc-2[nH]1 N1(C(c2ccc(C)o2)=O)CC2(CCCC2)C1C(N1CC(c2ncc[nH]2)C1)=O C1(NC(CCCC#C)=O)CCN(C(=O)C=C(C)c2ccsc2)CC1O C12(CC(=O)NC(COCCCNC(C3(C)CC(=C)C3)=O)(C)C)CCC(CC1)C2 c1(C(=O)NCC(C2CCC2)NC(C(=O)NCC)=O)cc(C(F)(F)F)ccc1Br c1(OCC(N2CCC(CNC(C3(OC(C)=O)CC3)=O)C2)=O)ccc(F)c(Cl)c1 N1(C(c2nnn(CC)c2C)=O)CCN(C(=O)C=CCOCCOC)CC1C Cc1c(CNC(=O)C(C)CNC(=O)CC(C)CN(C)C)cnn1C Cc1cc(F)c(C(N2CC(C(N3CCOC(CN(C)C)C3)=O)C2)=O)c(Br)c1 Cc1c(Br)c(C)n(NC(=O)Cc2ncc(-c3cccc(Cl)c3F)o2)c(=O)c1C#N c1(C(=O)NC(CC=C)C(=O)N(C)CCC2CCOCC2)c[nH]c2ccncc12 C1(C)(NC(C(C(=O)OC)C)=O)CCC(NC(c2ccc(C)o2)=O)CC1 c1(C(=O)NCC2C(CNC(C3(CC#C)CCC3)=O)C2)cnn(C(C)(C)C)c1C C(=O)(CCS(N)(=O)=O)N(CCCNC(CCCN(CCC)CCC)=O)C C1(C(N(C2CN(C(C=CCCC(C)C)=O)C2)C)=O)COCCC1C N1(CCC(=O)N(C(C)(C)C)Cc2ccccc2)CC2CCC1CN2C(N)=O N1(C(c2nn(CC)c(O)c2)=O)CCN(C(=O)Cc2ccoc2C)C2CCC12 C1(C(=O)NC(C(=O)NCCC)CC)CC2(C1)CC21CCC1 n1(CCC)c(SCC(=O)N(C)CCC2CCNCC2)nc2ccccc12 c1(C(N2CCC(NC(c3cc([N+](=O)[O-])cs3)=O)C2)=O)cnc(Cl)c(F)c1 c1(NC(=O)C(N2CC(F)CC2C(c2ccccc2)O)=O)cn2cc(F)ccc2n1 N1(C(C2C(COC)CC2)=O)C(C(=O)NC2CC2c2cncs2)CC1C N1(C(=O)CN2CCCC2CO)CCCN(CC2CCCC2)CC1 C1(NC(Cc2c(C)nc[nH]2)=O)CCCC12CN(C(=O)COC1CCC1)C2 S(=O)(=O)(c1cccs1)Oc1ccc(C(=O)NC(c2ccccc2)(C)C)cc1 c1(OC)cc(Br)cnc1OC(N1CCCC(n2ccc(C)n2)C1)=O.C(C(F)F)O c1(C(=O)NCc2ccc(C(F)(F)F)o2)cc2n(c1)CCN(CC)C2 c1(C(=O)NCC2CCC(NC(=O)CCc3cc[nH]n3)C2)cccc2c1C(=O)NC2 C1(O)(C(C)CNC(c2cocn2)=O)CCN(C(=O)CCOc2ccccc2O)C1 C1(NC(c2cccc[n+]2[O-])=O)C2CCC1N(C(=O)C(F)CC1CCCCC1)C2 N1(C(=O)Cc2ncsc2Cl)CC2(CCN(C(c3c(F)cccc3F)=O)CC2)C1 Cc1cc(O)nc(SCC(n2cc(COc3cccc(C#N)c3)nn2)C)c1C#N C1(C(=O)NC2C(CNC(c3c(CC)n(C)nc3)=O)CCCC2)CC2CCC(C1)O2 c1(N2CC3C(NC(C(CC)(C)C)=O)C3C2)nc(C)c(C#N)cc1Cl c1(C(CNC(c2ccc(N(CCC)CC)cc2)=O)O)c(C)nn(C)c1Cl N#Cc1cc(F)c(NC(C2CC23CCN(C(C2(Br)CCC2)=O)C3)=O)cc1Cl N1(C(Cc2c(C)occ2)=O)CCN(C(C2CCCN2N=O)=O)C2COCC12 c1(CC)cn2c(C(N3CC=CC(NC(=O)C(COC)N(C)C)C3)=O)cccc2n1 N1(C(Cc2n(C)ncc2)=O)CC2OCC(NC(C3CC34CC(F)(F)C4)=O)C2C1 c1(OC)cnc(F)c(C(=O)NCC(C)(C)NC(=O)CC2CC3(CC3)CO2)c1 N1(C(=O)NCc2cc(C)oc2C)CC2C3CCC(CC3)C2C1 c1(SC(C)C)ccc(C(=O)NCCOCCNC(=O)CSS(C)(=O)=O)cc1 N1(C(=O)OC(C)(C)C)CCC(CC(O)C(=O)NCc2ccoc2C2CC2)CC1 C12(CNC(CCN(C(c3ccncc3O)=O)CC)=O)CC(CN1C)C2 c1(C(N2CC(NC(C3CC(OC)C3)=O)C(CO)CC2)=O)cc(C)c(C)nc1C C1(C(=O)OCC)COC2CN(C(c3cc(=NS(C)(=O)=O)cc[nH]3)=O)CC2O1 C1(CC(=O)N(CC(=O)NCCS(=O)(=O)NC)C2CC2)CCOC1(C)C CCCCC(CNC(C1(C)CC=CC1)=O)NC(C1CC(=O)N1)=O c1(C(=O)NC(CCOC)CNC(c2cc(F)c[nH]2)=O)cnc(OCC2CC2)cn1 C1(C(=O)NCc2nccc(C(=O)NC(C#CC#C)(C)C)c2)CCCCC(=O)C1 C(=O)(C#CC1CCCCO1)N1CCN(C(CNC(c2ccns2)=O)=O)CC1 C1(C(N(C(C2CCCCC2)CO)C)=O)CC(F)(F)CN1C(c1cncn1C)=O CCC(CCOC)C(=O)NCC1CC(OC)CN1C(c1nonc1N)=O N1(C(C2N(CC)CC2)=O)CCOC(CCNC(c2ccn(CCF)n2)=O)C1 N1(C(C2(F)CN(C(C3CC(CC#C)C3)=O)C2)=O)CCCC(C#C)CC1 c1(C(=O)NC2C(CC(=O)N(CCN(CC)CC)C)CCCC2)cc(C)nc(C)c1 CC1(F)CN(C(=O)C(N)=O)CCN(C(=O)C(F)(F)Cc2ccc(F)cc2)C1 c1(-n2cc(CNC(CC(C)C)CCO)nn2)cc(F)c(O)c(F)c1 c1(C(=O)NCC2N(C(CCC=CC(C)C)=O)CC(F)C2)ccncc1N=[N+]=[N-] Cc1cc2[nH]c(C(=O)N(C3CC4CCC(C3)N4C(=O)C=CC(N)=O)C)cc2s1 C12(C(=O)NCC3CC(F)(CNC(=O)C=C4CCOCC4)C3)CCCCC1C2(F)F S(=O)(=O)(CCC(=O)NC1CC(C)CN(C(=O)CCC=CC(C)C)C1)NC C1(C(=O)NC2(CNC(=O)CCc3ccccc3Cl)CC2)Cc2cc(Cl)ccc2O1 c1(CC)cc(CC(=O)N(C2CCCN(C(c3cc(C4CC4)on3)=O)C2)C)n(C)n1 N1(C(c2cc(C(N)=O)[nH]n2)=O)CC(NC(=O)CC2CCOC2)C2(CC2)C1 c1(CNC(c2ncn(CC)c2)=O)cnn(C)c1C(=O)NC(c1ccccc1)(C)C CC1CCC(C(=O)NCc2cccc(NC(=O)Cc3cncn3C)c2)C(=O)N1 CN1CC(NC(C2CN(C(=O)CCc3ccc(N(C)C)cn3)CCN2)=O)CC1=O c1(C(N2C(C(=O)Nc3ncc(C(C)=O)s3)CCC2)=O)ccc(CF)cc1 CC(CC(=O)NCc1ccncn1)C(C)(C)NC(c1cccc(CO)n1)=O c1(C(=O)Nc2ccc(C(=O)NCCC(CSC)OC)cn2)ccc2c(n1)CCC2 C(CCCCC(=O)NCC12CC(CO1)N(C(c1cc3sccc3s1)=O)C2)OC c1(CNC(C2(C)CCN(C(c3ccc(NC)cc3)=O)C2)=O)cccc(C)c1F c1(SCC(N2CCN(CCNC(C3C(=C)C3)=O)CC2)=O)cccc2ccccc12 C(=O)(CC1=Cc2ccccc2C1)N1CCN(C(C2N(C)CCC2)=O)C(C2CC2)C1 N1(C(C(C(C)C)O)=O)CC2CC(NC(=O)C(C)(C)n3ccc(C4CC4)n3)C2C1 S(=O)(=O)(c1cc2sc(=NC3COCC3C)[nH]c2cc1Cl)NC(CCCC)(C)C Cc1nccn1CCN(C)C(C1CC(C)N1C(=O)Cn1cc(CO)nn1)=O c1(C(=O)NC2(CNC(c3cc(C(=O)OC)on3)=O)CCC2)cccc(Cl)c1Cl c1(-c2cn(CC3CC(c4cccc(F)c4)(O)C3)nn2)cc(Cl)ccc1F C=CCCCC(C(=O)NCC1CC2CCC2C1)NC(=O)C(C)N=[N+]=[N-] c1(NC(C2CC(=C)CN2C(c2nc(C3CC3)cs2)=O)=O)ccc(Br)c(Br)c1 CC(C)(C)C(C#N)C(=O)NC(C(N1CC(O)(C2CC2)C1)=O)C1(O)CCC1 C(c1cccnc1)=C(C(=O)NC(C(C)CCNC(C(C)NC(N)=O)=O)CO)F c1(NCC)cncc(C(N2CC(CCNC(=O)CNC(=O)CCC(C)C)C2)=O)c1 C1(NC(c2c(OC)scc2)=O)C(C)CN(C(c2cc(Br)ccn2)=O)CC1C Cc1cc(C(=O)NCC2CCCCC2NC(C2CC23CCCCC3)=O)nc(C)n1 n1(CC(=O)NCCC(Cn2cc(CC)nn2)F)c(SC(F)(F)F)nc2ccccc12 C12(C(=O)NCC(C)N=[N+]=[N-])CC(C)(CN1C(=O)C(C)CC1CC1)C2 N1(C(C2N(C(C3C(CC)C3)=O)CCC2O)=O)CCn2cc(C)nc2C1 c1(C(=O)NC2CCC(NC(CC3(C)CCCO3)=O)C2)cccc(O)c1Cl c1(-c2nc(-c3ccc(NC(c4ccc(O)c(F)c4)=O)s3)on2)ccc(Cl)cc1Cl O=C(C1CCc2scnc21)NC1CC(NC(C2(CCF)CCC2)=O)C12CCC2 Cc1cc(Cl)c(C(=O)NC2(CF)CCN(C(C3(C)CCCC3C)=O)C2)cn1 C(=O)(C1=C(C(C)OC)N(CCSC)C(=O)NC1c1nc(C2CC2)no1)OCC Cc1ccc(CC2CCCC2NC(=O)NOCC(O)C(C)C)cc1 c1(-c2ccc(C)cc2)csc2ncn(CC(N3CCN(C)CC3)=O)c(=O)c12 S(=O)(=O)(CCN=C(NC1CCOCC1)NC12CC(C)(C1)C2)N1CC(C)OC(C)C1 c1(C(N(C(CNC(C(COC)O)=O)C)C)=O)cc(S(=O)(=O)N(C)C)oc1C C1(CCC(=O)NC2(CN(C)C)CCCC2)CCCCN1C(C1CC(=C2CC2)C1)=O N1(C(C(C)O)=O)CCCC(CCCNC(c2ccc(C3CC3)cn2)=O)C1 c1(C(=O)NCC(C)NC(C2CCN2C)=O)ccc(Cl)c(Cl)c1.C(C(C)C)O.CS C=CC(C)(C)CC(=O)NC1(CCO)CN(C(C2CCN(OC)CC2)=O)C1 N1(c2nc(C)nc3c2CCC3)CCc2cc(-c3cccc(O)c3C)ccc2C1 c1(CNC(C2C(C)CCC2)=O)ncccc1NC(=O)NCC1CNC(=O)O1 C1(NC(C=CC)=O)C2CCN(C(c3ccc4cnoc4c3)=O)CCC12 c1(C(N2CC(OCCNC(c3cc(C)[nH]n3)=O)C2)=O)cc2c(C)cccn2n1 c1(C(N(CC(C)CNC(=O)C(C)C2CCCC2)C)=O)cnc2ccnn2c1O N1(C(CCCCC=C)=O)CC2CCN(C(=O)C(C)C(F)F)C2C1 N1(C(C=C(C)C2CC2)=O)CCC2(CC1)CC(C(=O)NCCOC(C)C)C2 C1(O)(CNC(c2ncccc2C2CC2)=O)CC2CCC(C1)N2C(c1ccsc1)=O c1(C(N2CC3CC(NC(C(CCC)(C)C)=O)C3C2)=O)c[nH]c2ccccc12 C=CC(C)(O)CC(=O)N1CC2CC2(CNC(c2nnn(C3CC3)c2C(F)F)=O)C1 C1(NC(C2CC(C)=C(C)CC2)=O)CN(C(c2coc(Br)c2)=O)CC2(CC2)C1 CC1(C)Cc2ccc(-c3nc(CSc4ncc5cc(Cl)ccn45)no3)cc2O1 Cc1cc(OC(C)C(N2CCCC(N(C)C(c3ccncc3)=O)C2)=O)cc(C)c1 c1(C(=O)NCC(CC)NC(c2occc2Cl)=O)ccc(N(C)C)c(F)c1 C(=O)(CC(COCC1(C(=O)NC(C)C)CC1)OCC)N(CC#C)CC=C C#CC(CNC(C)=O)N(C)N(C)CCCc1nccs1 N1(C(CC(C)OC)=O)CC(CNC(c2ccc(CN(C)C)cc2)=O)CC1C CCC(C)C(=O)NCC(=O)NC1(C(=O)NC(C)C(C)(C)O)CCCC1 C(=O)(C(CCC(C)C)SCC)Nc1ncc(-c2cn(CCOCC)nn2)cc1C c1(C(N2CC(C(C)NC(CCC(=O)NC)=O)C2)=O)ccc(OC)c(Cl)n1 CC1(C)CC(CNC(C2C3CN(C(C4CC5OC4C4CC54)=O)CC23)=O)CCO1 c1(OC)ccc(-c2nn(C(C)C(=O)OC3(CC(N)=O)CC3)c(=O)o2)cc1 c1(N(CCC(C)C)C)nc(N2CCCC(C3CC3)CC2)nc2ccsc12 c1(C(N2C(CNC(C3(C(C)C)COC3)=O)CC3(CC3)C2)=O)cc[nH]c2nccc1-2 c1(OC(C)C)cnccc1C(=O)NC1(CF)CCN(C(c2cnn(C)n2)=O)C1 CN1CCCC1CC(=O)NC1(C(=O)N(CCO)C2CC2)CC1 O=C(C1CCc2nccn21)NCC1CC12CCN(C(C1(C3CC3)CC1)=O)CC2 C1(C(=O)NC2CN(C(CCCOC)=O)C(C)CC2)Cc2cncn2C(=O)N1 C1(C(N2CCN(C(CC(C)CF)=O)CC2C)=O)CCc2nnc(O)n2C1 C(=O)(CS(=O)(=O)CCO)N1C(C)CC(NC(=O)CN2CCN(C3CC3)C2=O)CC1 CC1COC(C(=O)NC23CC(NC(c4cc(-c5cccs5)on4)=O)(C2)C3)C1 Cc1c(C(N2CC(C)N(C(=O)CCc3nncn3C)CC2C)=O)sc2cncn12 CC1CN(C(C2CCCCCC2C)=O)CCN1c1ccncc1 c1(C(=O)NC(COC)CNC(C2(C)CC2F)=O)ccc([N+](=O)[O-])c(Cl)c1 C1(NC(C2(C)N(C(CC(=O)NCC)=O)CC=C2)=O)CN(C)C(=O)C12CC2 C#CCC(CC(F)F)C(=O)N1CCC(C(=O)NCC2CC3CCC3C2)C1C(C)C C1(NC(CCC2CC(NC(C(C)C3CC3)=O)C2)=O)CC(F)(F)C1(C)C C(=O)(C(=O)N=c1cc(-c2ccc(F)cc2)o[nH]1)c1ccc(OC)c(-n2cncn2)c1 C(C1CN(C(=O)C(C)OCC2CC2)CC1C(N1CCSC(C)C1)=O)=CC n1(CC)ncc([N+](=O)[O-])c1C(=O)NCC(O)CNC(=O)CC1(CSC)CC1 N1(C(C=CC(=O)OCC)=O)CCC(C(=O)NCc2cnn(C)c2C)(COC)C1 N1(C(c2cc(C(=O)OC)sc2C)=O)CCC2CN(C(=O)Cc3cnccn3)C2C1 N1(C(C(C)Cn2ccnc2)=O)CCn2nc(C(=O)N(CCCCl)CCCCC)cc2C1 C1(C2CC2)(NC(CCCC)=O)CCN(C(c2ccc(F)cc2C(F)(F)F)=O)C1 N1(C(C2C(OC)C2)=O)CC=C(CC(=O)NCCn2nc(C)nc2C)CC1 c1(OC)cc(F)c(CN2CCC2(C)C(=O)NCc2cccc(C#N)c2)c(F)c1 c1(C(=O)NCCCCCNC(COCCC=C)=O)cncc(C)c1Cl N1(C(C(CCC)NC(C2CC=CC2)=O)=O)CC2CC(CO)C(C2)C1 CCCCCC(C)(C)CNC(=O)C(C1CCN(C(C2CCC(CO)CC2)=O)C1)C C#CCC(C)(C(=O)N(C)CCOC)NC(c1ccon1)=O C1(NC(C2(C#C)CC2)=O)C(CN=c2[nH]ncs2)CCC12CCC2 c1(C(N2C(CNC(C(CC)COC)=O)CC2)=O)c2ccc(Br)cc2nn1C c1(C(N2C(C)CN(C(C3CC34CC4)=O)CC2)=O)cccc([N+](=O)[O-])c1Br c1(CN2CC(N3C(=O)CC(C(C(=O)O)NC(C(N)=O)=O)C3)C2)cc(F)cc(Br)c1 N#Cc1cc(Br)ccc1NC(C1CCCN(C(C2CC(O)C2)=O)C1)=O C1(O)(CN(C(c2c(CC)non2)=O)C)CCN(C(=O)CCC2CC(C)C2)C1 c1(NC(=O)NC(C(=O)OCCC)CC2CCC2)ccc(OC(C)(C)C)c(Br)c1N Cc1cccc(C(=O)NC(C(=O)NC2C=CCCC2)C(C)C)c1O CCC(CC(=O)NC1CCN(C(=O)Cc2ccns2)C1C(C)C)SC c1(CN(C)CC2CCCCC2O)c(O)ccc(Br)c1Cl C12(C(=O)NC3CC4CN(C(C(CCC)(C)O)=O)CC43)CC(C)(C1)OC21CCC1 C(C(CO)N=c1[nH]c(Cl)nc(CC)c1Cl)Nc1cc(SCC)ncc1 Cc1ccnc2ccc(C(=O)NC3CCC3NC(=O)CCCS(C)(=O)=O)cc12 c1(C(N2CC=CC(NC(C3N(N=O)CCC3)=O)C2)=O)csc2c(O)ccnc12 CC(CNC(=O)C(CN(C)C)NC(=O)CCc1nc(O)n[nH]1)N=[N+]=[N-] Cc1nn(CC(=O)NCC(C2CCCCC2)NC(=O)CC(F)F)c(=O)n1C C1(CC)CN(C(=O)C(C)N(C(=O)CCc2cn(C)cn2)C)CC(=O)N1 N1(c2ncc(C(=O)OCC)nc2)CC2CC(NC(c3cnn(C)n3)=O)CC1C2 C1(NC(CCC(=O)NCC)=O)C2CCC1N(C(=O)Cn1nnc(C3CC3)n1)C2 Cc1cnc(C(=O)NCCCN(CCO)C(c2cnc(C(C)C)o2)=O)cn1 C(=O)(C(C(C)C)N(C)CCNC(=O)NCc1ccc(C2CC2C)o1)OC c1(C(N2CC(NC(c3n(C(C)C)ccc3)=O)C2)=O)cc2[nH]ccc2s1 N1(C(C2(F)CC(C(=O)OCC)C2)=O)CCOC(CNC(=O)CC2(C)CCCC2)C1 N1(CC(=O)NC2(CNC(CCC(C)OC)=O)CC2)CCCNS1(=O)=O C1(NC(c2csc(C(F)F)c2)=O)CCC2CCN(C(c3ccc(F)cn3)=O)C1C2 C1(CC(NOCC(C)(C)O)=O)CN(C(C2C=CCCC2)=O)C(C)(C)C1 N1(C(C2C(=C)C2)=O)CC(CNC(C2(CCN3CCOCC3)CC2)=O)C(C)(C)C1 CC(C)C(F)C(=O)NCCCN(C(=O)CCC1CC(C)(C)CO1)CCO N1(C(C)C)CCN(c2cc(CNC(C3CCOC(CN)C3)=O)ccn2)CC1 c1(NC(C2CC3CC3N2Cc2cnc(Cl)cn2)=O)nccc(Cl)c1Cl c1(C(=O)NC(CC(C)NC(C=C(COC)C)=O)C)ccc(C)n1C c1(C(C(=O)N(CCCCCCNC(c2c[nH]c(=N)o2)=O)C)O)ccc(F)c(Cl)c1 C1(NC(C(C2CN(C(c3ccc(C)nc3)=O)C2)O)=O)C2CCC(C2)C1CO c1(CC(=O)NC(C(C)C)CCNC(=O)C(C)(O)C2CCC2)cn2ccccc2n1 C1(CN(c2cn(C)nc2OCC(F)F)C)CCC(NC(N2CCOCC2)=O)CC1 N1(C(C2C(C3C(C)C3)C2)=O)CCC(N=c2[nH]nc(C(F)F)s2)(CO)CC1 N1(C(C2CCCC(C(=O)OC)C2)=O)CCC2(NC(c3ccn(C)c3)=O)CCCC12 Cc1cc(C(=O)NCC2CC2NC(C2(C(C)(C)C)CCCC2)=O)ncc1CO C(CCC(C)C(=O)NCC(C1CCCN1C(=O)Cc1cncn1C)(C)C)OC C1(OC)CCCC(C(=O)NCC2(F)CC(NC(c3ncccc3Br)=O)C2)C1 C(C(=O)N1CCC(C)(CCO)C1)(C(C)O)NC(c1c(C)csn1)=O C1(CNC(C2CCN(C)C2)=O)C2CCC(C2)N1C(C1(S(C)(=O)=O)CC1)=O C1(C)(C(=O)NCC(C)CN(C)C(c2conc2C2(C)COC2)=O)CCCCO1 Cc1nn(C)cc1C(=O)NCCC1CCCN1C(=O)C=CSc1ccccc1 C1(NC(CN(CCC)C)=O)CC(CNC(c2ccc(CC(N)=O)cc2)=O)C1(C)C N1(C(C2N(CC)CC2)=O)CC(CNC(c2cc(=O)c(OC)c[nH]2)=O)OC(C)(C)C1 Cn1nc(NC(=O)NCC2CCN(C(=O)CCc3cnc[nH]3)C2)cc1OC(F)F Cc1ccc(CCC(=O)N(C)CC2(CNC(=O)CCc3cnccn3)CC2)cc1 C(CCSC)(C(=O)Nc1cn(C2CN(C(C3C=CC(CO)C3)=O)C2)nn1)OC N1(C(c2n(C)ncn2)=O)CCN(C(C2CCS(=O)(=O)CC2)=O)CC(C)(F)C1 C(=O)(C(C(C)(C)C)c1cc(F)cc(F)c1)NCC(CC)NC(=O)C(F)CC N1(C(c2c(OC)ccs2)=O)CCC(NC(c2ccnn2C)=O)C1C(C)(C)C C(C(=O)OCC(=O)Nc1nnc(C(C)C)s1)(C(C)C)SC O=C1OCC2CN(C(=O)C(N3CC4CC5CC4C3C5O)=O)CCN12 C1(NC(=O)Cc2ccon2)CC=C(C(=O)NC2Cc3cscc3C2)C1 c1(C(N(CCN(C(C2C(CC)N(C)CC2)=O)C(C)C)C)=O)ccc(N)cc1Cl C1(C(=O)Nc2cccc(C(=O)OCC)c2)CC12CCN(c1ncncc1OC)C2 C(=O)(C1=NNC(=O)C1)NC1CC(CNC(CCCn2c(C)cc(C)n2)=O)C1(C)C c1(C(C(=O)NC)N(C)Cc2csc(C(C)C)n2)csc(C(C)C)n1 C(N=c1nc2c(cnn2C)c(NCC(C)OC(C)(C)C)[nH]1)c1ccc(C)s1 C1(C(=O)NCCOCC(=O)NC)CNC(=O)CN1C(=O)C(C)Cn1cccn1 C1(CNC(c2c(CCC)nns2)=O)CC(OC)CN1C(=O)C(C)OCCN(C)C c1(C(N2CCC(CNC(CC3C(CC)C3)=O)C2(C)C)=O)nccc2occc12 C(=O)(CCCCCCSC)NCC1(CNC(C2(CCC)CC(=O)C2)=O)CCC1 Cn1cc(C(F)(F)F)nc1C(=O)NCCCNC(C1CCCN1C1CC1)=O C1(C(C)C)C(NC(=O)CN2CCOCC2)CCN1C(=O)CCn1cccn1 Cn1cc2c(C(N3CC(NC(C45CCC(C4)S(=O)(=O)CC5)=O)C3)=O)cccc2n1 C1(C(=O)OC)C(C)CCCN1C(c1ncc(F)cc1F)C(=O)NCCCC1CC1 S(=O)(=O)(c1ccc(S(=O)(=O)Nc2ccc(C(F)F)cn2)cc1)NC(C(C)CO)C CC(C)CC(O)C(=O)NC1CCCN(C(c2ccc(C(C)(F)F)cn2)=O)C1 CC(C)CC1CC(=O)NCC2(CCOC2)C(=O)N1.C1(CO)CC1 c1(C(=O)NC(c2cnn(C)c2)C(=O)NC2(CC)CC2)cn(C2CC2)cn1 N1(C(C2CC(=C)C2)=O)C2CCC1(CNC(c1cnc3n1CCS3)=O)CC2 c1(CCC(=O)NC(C(C)NC(C2CNC(=O)C2)=O)(C)C)cccc(F)c1F n1(CC)c(C)nn(CC(N2CCOC(CCNC(=O)C=CS(C)=O)C2)=O)c1=O N1(C(C2(C#C)CC2)=O)CC2CCC1CN2C(=O)COc1cc2c(s1)CCC2 n1(CCC(=O)NCC2CCCCN2C(=O)Cc2ccsn2)cccnc1=O CCCS(=O)(=O)C(C)C(=O)NCCN(C)C(c1c(N)sc2c1CCC2)=O S(=O)(=O)(c1ccc(NCC2CCC3(CC3)CO2)c(C#N)c1)NCCC(C)OC CCC(CC(C)C)C(=O)N1CCCC(C)(C)C1C(N1CCc2nn[nH]c2C1)=O C(=O)(C(C)CC(F)(F)F)N1C(C(N(C2CC(C)C2)C)=O)C(O)CC1 C12(NC(CCCC=C)=O)CCC1CN(C(c1ccc(OCCOC)cc1)=O)C2 C12(CCNC(C3(OC)CC3)=O)CCC1CN(C(c1c(C)ccn1C)=O)C2 c1(CN2CCC(C(N3CCC(C(=O)OC)C3)=O)C2)ccncc1O C1(c2cn(C(=O)OCC)nn2)N(C(=O)CN2C(C)CCC2C)CCCC1(C)C.CC=O C=C(C)CN=C(NCC1CCSC1)NCC1(OCC)CCOCC1 CC(C)C(O)C(F)(F)C(=O)NCCN1CCCN(C(=O)Cn2nccn2)CC1 Cc1nc(C(=O)NC(C)CN(C)C(C2(C)CC2)=O)c(-c2ccc(F)cc2)s1 C1(C)(C(=O)NCC(CNC(CCOCC(C)C)=O)(C)O)CCCNC1=O c1(SC)ncc(C(=O)N(C(C)CN(C)C(C2C=CC=CC=C2)=O)C)n1C C1(C(N(CC(C(=O)NC)C)C)=O)COCCN(C(c2ccccc2NC)=O)C1 N1(C(C(C)(C)CNC(c2cnccn2)=O)=O)CCC2(CCCOC2)C1 N1(CCN(C(C(C)NC(C2CCC2)=O)=O)C)CCN(C(=O)CC(C)(F)F)CC1 C1(COC)(NC(=O)Cc2nccs2)CN(C(=O)C(c2ccc(C)s2)C)C1 c1(C(N2CCC(CCNC(CSCC=C)=O)C2)=O)ncccc1-c1ccccc1 N1(C(CCCC2C(C)C2)=O)CC(C)(C)OCC1CNC(c1c[nH]cc(Cl)c1=O)=O c1(C(N2CCC3(NC(CCNC(=O)NC)=O)C(C2)C3)=O)c(F)ccc(Cl)c1N C(=O)(CC(C)C(F)(F)F)NCC(N(C(=O)CSc1ccnn1C)C)C1CC1 CC(C#N)C(=O)N(C)CC=CC(=O)NC1CC1CC(C)(C)C C1(CNC2C(F)C3N(C(=O)OC(C)(C)C)C(CC3)C2)CCc2nc(CO)cn2C1 N1(C(C2C(=C)C2)=O)CCN(C(C2(c3ccc(Br)s3)CCC2)=O)CC1 N1(C(c2n[nH]c(C)c2Cl)=O)CC(C(=O)NCC(=O)NC(C)C)CC(C)(C)C1 Cc1nc(C(C)C)oc1C(=O)NCC(C)N(C(=O)CCc1cccnc1F)C c1(NC(C2(CNC(c3cnn4ccccc34)=O)CC2)=O)nc2cc(F)ccc2s1 C(C(C(=O)N1CC=CC1CF)NC(C1CCOC1C(C)C)=O)OCC C(=O)(CCCC(F)F)NC1CCC(C)(CNC(c2ccc(C(N)=O)o2)=O)C1 c1(C(=O)NC2CN(C(=O)CCn3ccnn3)CC2F)ccc2cccc(F)c2n1 N1(C(CCSCCCC)=O)CCC(F)(CNC(C2CC2c2ccccn2)=O)C1 c1(CCCCNC(C(c2cnn(C)c2)OC)=O)nnc(C)n1C C(CC)(CC)(CCNC(=O)C(C)(O)C1CCC1)NC(C(CCC)NC(C)=O)=O Cc1ccc(F)c(NC(c2ccccc2OCC(N2CCCCC2CO)=O)=O)c1 c1(OC)cc(C(N2CCC(NC(=O)Cc3nnc(O)s3)C2)=O)ccc1OC(C)C C(C)(C(C(C)C)NC(c1cc(Cl)ns1)=O)NC(CCC=CC(C)C)=O C(=O)(C1=CC2CCCCCC12)N1CCCC(c2cn(C(C(C)O)C)nn2)C1 C=C(Cl)CC(C(=O)NCCc1ccn(CC)n1)NC(C1CCC2CC12)=O C(=O)(C1=CCCC1C)NCCC(C(C)C)NC(C1(C2CC2)CC1)=O C(=O)(CCC(C)(C)C)NC1CCC(NC(c2n(COC)ncc2)=O)CC1 CC1(C)CC(NC(c2cc(C3CCC3)n[nH]2)=O)CN1C(C1CC1F)=O N1(C(C2C(CC)C2)=O)CCC(CN(C(=O)COCC(F)(F)F)C)C1 C#Cc1cncc(C(=O)NCC(CNC(c2cnn(C)c2CC)=O)S(C)(=O)=O)c1 C(=O)(C#CC1CCOC1)NC1CC(C)(NC(=O)C(c2ccccn2)N2CCOCC2)C1 N1(C(C2C(C)(C(F)F)C2)=O)CC(NC(=O)COc2ccsc2)CC12CCOCC2 C(=O)(CCC(=O)c1ccc(Cl)cc1)NCCN(C(C1(CC#C)CCC1)=O)C CC1CCC(CNC(=O)CNc2nccs2)N(C(c2cc(C3CC3)ns2)=O)C1 C1(C(=O)OC)CCN(C(=NCCc2ccccc2)NC2CC2)CC1 C(=O)(C(CCCC(OC)OC)N1CCN(S(=O)(=O)CC)CC1)NCCCCCC N1(C(C2C(OC(C)=O)C2)=O)CC(C(=O)NCCC2(C)CCCO2)C(C)C1 c1(-c2nc(NC(C(=O)N(C3CCC(C)CC3)CC)C)sc2)ccc(F)c(F)c1 C1(NC(CCSCC(N)=O)=O)CC2(C1)CC(CNC(C1CCCCC1F)=O)C2 N1(CC(=O)NC(CNC(C2(CCC=C)CCCC2)=O)C(C)C)CCCOC1=O C(N=c1[nH]c2c(c(=NC3COC(C4CC4)C3)[nH]1)COC2)c1ncn(C)n1 C1(C(=O)NCC2(C(F)(F)F)CCC2)CC(F)CN1Cc1cccnc1Br c1(NC(N(C2CCCC2NC(=O)CO)C)=O)cccc(Br)c1.C1(C)CC1 c1(CNC(C(N2C(C)CC(c3ccccc3)CC2)=O)=O)ccc2c(c1)CCO2 c1(CNC(C(F)OC)=O)cccc2c1CN(C(c1cc(C(C)=O)[nH]n1)=O)C2 c1(C(=O)NC(C(C)NC(C(=O)NCCNC(C)=O)=O)(C)C)c(N)cc(Cl)nc1Cl Cc1nc(C(=O)NCCCN(CCCNC(=O)CC2CCOC2C)C)cc(O)n1 C1(NC(C(CCC)=CCC)=O)CN(C(c2cc(C)c(F)cc2O)=O)CCC1(C)C CC1=NOC(CC(=O)N(C2CCCC2)CCNC(=O)CCC2CCCO2)C1 c1(OCC=C)c(OC)cc(CNCC2CCCCC2c2ccccc2)cc1Cl C(=O)(N=c1[nH]n(-c2ccccc2)cc1C)c1ccn(C(c2ccccc2)OC)n1 C1(NC(C(C)OCCCC)=O)C2CC3C(C2)C13C(=O)NCc1ccc(C)cc1F CC1CC(=O)NCC1NC(=O)Nc1cccc(CCC(=O)NCc2ccns2)c1 N1(C(CC2(CC)CCOCC2)=O)CCCC(CCNC(c2csc(Cl)c2)=O)CC1 O(NC(=O)C(CSCC)NC(c1cccnn1)=O)CC C(CCC(=O)NCC(C)CNC(=O)C(c1cnn(CC)c1)=O)OCCC CC(C)(O)C(C)(CO)NC(=O)C#CCNC(=O)C(F)C(F)(F)F Cc1csc2c(N3CCC(CCNC(C4CC4(C)C)=O)C3)ncnc12 N1(C(c2n(CC)ccn2)=O)CCN(C(C2CCCC2(C)C)=O)C(C(C)C)C1 CCC(CC(=O)NC(C)CN(C)C(C1CN(S(N)(=O)=O)C1)=O)C(F)F c1(C(=O)NCC2CN(C(C3(CC)CCOC3)=O)C2)csc2cc(OC)ccc12 c1(CNC(C(=O)Nc2n(CC(C)C)ccn2)=O)cn(C(F)F)c2ccccc12 N1(C(c2cc(C)c(C)s2)=O)C2CCC1CC(CNC(C1(CF)CCC1)=O)C2 C(=O)(CC(C)(C(F)F)N(C)C)N1CC(CCCCNC(c2c(C)oc(CO)c2)=O)C1 CN1CCCCCC1C(=O)NCC1(CNC(C2(C)CCOC2)=O)CCC1 c1(COC)noc(CNC(=O)C(C2CC2)NC(c2sncc2C)=O)n1 n1(CC(=O)NC(CCCNC(C(C)OCCC(C)C)=O)C)cnccc1=O c1(C(N2CC3C(NC(C=C(CC)C)=O)(CCC3)C2)=O)ccc2ncccc2n1 c1(C(N2CCC(N(C(c3c(C)con3)=O)C)C(C)C2)=O)ccc2cc[nH]c2c1F CN=c1nc(N2CCC(CCCO)C2)[nH]c(=NCc2ccnc(O)c2)[nH]1 c1(C(=O)NC2(C)CCN(C(C3(C4CCCO4)CCC3)=O)C2)ccc(F)c(CO)c1 c1(CSCC)cccc(C(=O)NC2C3CCN(C(C4CCC(CC)CC4)=O)C23)c1 c1(C(=O)NC2CN(C(CSCC=C)=O)C(C)(C)C2)cnc2n1CC(C)CC2 C(=O)(C1CCc2cc(F)ccc21)NC1C2CCN(C(CCS(C)(=O)=O)=O)C21 C12(C(=O)NCC3(F)CCN(C(Cc4c(C)n(C)cn4)=O)C3)CC1COC2(C)C C(=O)(CCCC(=O)N(C)CCNC(C1CC12CC2(F)F)=O)OC C(CN=c1ccnc(NC2CCC2)[nH]1)NC(C1CCCCN1CC(F)F)=O N1(C(CC(C)CNC(=O)CCc2cccn2C)=O)CCNC(=O)CC1 CN1CC(NC(C2CC=CCN2C(c2nocc2Cl)=O)=O)C(C)(C)C1 c1(CC)ccc(C(=O)NC(C)CCNC(c2cc(C(C)CC)no2)=O)cn1 c1(C(N(CCCNC(C2(OCC)CCC2)=O)C)=O)nc(C(F)(F)F)sc1C N1(C(=O)Cc2cn[nH]c2)CCN(C(c2c(O)cc(F)cc2F)=O)CC2(CC2)C1 C12(C(=O)NC(c3cn(C)nc3)(C)C)CCCC1N(C(=O)CCCN(C)C)CCC2 Cc1nc(C(=O)NC2(C)CC(NC(C3(C)CCOC3C)=O)C2)c(C)n1C N1(C(c2cc(CC)ncn2)=O)CCC(NC(C2CC(C)(F)C2)=O)C(F)C1 c1(CC(=O)NC2CC(NC(C=CC(c3cn(C)nc3)=O)=O)C2)c(F)cccc1Br C(=O)(C(C)(F)C(=O)NC1CCCC1CC(=O)NCC(C)C(C)(F)F)OC C(=O)(CCCC(C)CC)N(CCCCNC(c1nc(COCC)sc1)=O)C CC1CC(=O)NC(C(=O)NC2C=CC(CC(=O)NC34CCC(CC3)C4)C2)C1 C1(C(=O)NCC(N2CCCCC2)C)CC2CCC(C1)O2.C1(C)C(=O)N1 c1(N2CC(CC)N(Cc3nocc3C(=O)OC)CC2)ncnc2c1CCCC2 c1(CC(=O)N(CCNC(C2CSC2)=O)CC)cc(=O)n(C2CCS(=O)(=O)C2)[nH]1 Cc1ccc(=N)[nH]c1C(=O)N(C1CCCCC1N(C)C(c1cc(=O)n(C)o1)=O)C c1(C(N(CC(C)NC(C2(C(F)F)CC(F)(F)C2)=O)C)=O)cc(S(N)(=O)=O)c[nH]1 C(Cc1ccccc1)(CCNC(c1ccc(C(F)(F)F)o1)=O)NC(COCC)=O c1(C(=O)NC2CC3CN(C(C(C(CC)O)C)=O)CC32)cc(C)c2c(c1)CCCN2 C(C)(CNC(=O)C=C1CCOCC1)(C(C)C)NC(C(C)SCC)=O c1(C(=O)NCC(CNC(CC2(CCC#C)OCCO2)=O)C)cnc(Cl)cn1 c1(C(=O)NC2C3CCN(C(C(C)OCCOC)=O)C32)coc2cccc(O)c12 C1(C(=O)NCC2(C(C)NC(c3cncnc3)=O)CC2)CCC2(CC2)C1 CCC(F)C(=O)NCCN(C(=O)C(C)(C)N1CCCCC1)CC c1(C(C(=O)NC2C(CNC(C3C4(CC(OCC)C4)C3)=O)C2)O)cc(F)cc(F)c1 c1(C(N(C2CN(C(CC(CC)(F)F)=O)CC2(C)C)C)=O)cc(C)cc(C)c1O N1(C(CC(n2c(CC)ncc2)C)=O)CCC(NC(=O)C(=O)NC)C(CO)C1 Cc1cc(C(=O)NC(CNC(C2(O)CC(CF)C2)=O)CO)ccn1 C(=O)(C(C)(CSC)NC(C1COCC(C)O1)=O)N(CC(CCC)O)C c1(N2CCC(C(F)(F)F)(OC)C2)cc(C)nc(NC(=O)CCOC(C)C)n1 c1(OC)ccc(-n2cc(C3CCCN3C(=O)CN3CCCOC3=O)nn2)cc1 c1(CN2CCCN(CC(=O)NC(C(=O)OC)C)CC2)c[nH]c2ccccc12 Cc1nc(C)c(C(N2CC(N(C(C3(C4CCCO4)CCC3)=O)C)C2)=O)s1 C1(C)(CC)CN(C(C2(CCNC(=O)C(CC3CC3)OC)CCCC2)=O)CCO1 c1(C(N2CC(O)CC(NC(C(C)(C)C#N)=O)C2)=O)cc(Br)c([N+](=O)[O-])[nH]1 c1(OC)c(C(=O)NC(C)CC(C)NC(=O)C(=O)NCCC(N)=O)occc1=O CC1(NC(=O)CCNC2CCN(c3ccccc3)CC2)CCC(=O)N1 c1(C(=O)NC(C(C)NC(c2c(CC)nn(C)c2)=O)C)c(C)cccc1Cl c1(CN(CCOC)C)ccc(Cl)cc1Oc1ccccc1.C12(CC1)C(=O)N2 N1(C(C2(C#C)CCCC2)=O)CC(C#N)(S(C)(=O)=O)C1 c1(OC)ncc(Br)cc1CNC(Cc1cccs1)CC(=O)NCCCO C1(CC(=O)N(CC#C)CC=C)CN(C(c2cccc(F)c2)=O)CCC1C c1(C(=O)NCCCCNC(CCC(CC)OC)=O)coc2c1CCCC2 N1(C(CN(CC)CC)=O)CCC(C(C)NC(c2csc(C(=O)OC)n2)=O)C1 c1(C(N2C(C)C(NC(=O)CCC3CC3)CC2)=O)cncn(C)c1=O C123CCC(CN(C1)C2=O)C3.c1(CNC(C2CC2C(F)F)=O)ccc(F)cc1 C1(NC(C2(CCC)CC2)=O)CC2CCC(C1)N2C(C1CCSC1)=O Cc1cc(Br)ccc1-c1cn(C2CCCC2C(C(N2CCOCC2)=O)C)nn1 C1(C(=O)NCCCCNS(C)(=O)=O)COCC2(CNC2)O1 CN1C(=O)C(F)CC1C(N1CCC(NC(c2ccc(-c3ccncc3)o2)=O)C1)=O C=C=CC(C)C(=O)NC1(CN(C(=O)C(C)SC(C)C)C)CC1 Cc1cncc(CCC(=O)NC2CN(C(c3c(C)noc3C)=O)CC2C)c1 C1(NC(C2(S(N)(=O)=O)CC2)=O)CN(C(=O)COCC2CCCO2)CC2(CC2)C1 CC1CN(C(=O)CCC(C)(C)F)C(C)CN1C(=O)Cc1ncc(F)cc1F n1(CC(=O)NC(C2CCOC2)CNC(=O)CCc2cnoc2)cccc(O)c1=O C1(CC=C)CCCCN1c1nnc(-c2ccccc2Cl)n1CC c1(C(=O)NC2CCC(CNC(C3CSC3)=O)C2)cccc2c(O)nncc12 C1(C)(CNC(c2c(CC)scc2)=O)CCN(C(=O)C(C)(C)CF)C1 C12(NC(CC3N(C)CCC3)=O)CCOC(CNC(c3cncc(C#N)c3)=O)(C1)C2 Cc1ccc(F)c(C(=O)NCC2CC(O)CN2C(c2cc3n(n2)CCO3)=O)n1 N1(C(CCCCC#C)=O)C2CCC1CC(NC(c1cc(C(F)F)ncn1)=O)C2 CC(C)C(O)C(C)C(=O)NCC(C(=O)N1CC2CCC2(CO)C1)C(C)C C1(NC(COc2ccn(C)n2)=O)CCN(C(C2CCNC2=O)=O)CC1(C)C c1(C(N2C(C)(CNC(C3ON=C(C(C)C)C3)=O)CCC2)=O)ccccc1[N+](=O)[O-] N1(C(C(C)N(CCC)C(c2cc(CN(C)C)n[nH]2)=O)=O)CCC(F)(F)CC1 n1(CC)c(C)ccc(C(N2CCOC(CC(N3C(C)CCCC3C)=O)C2)=O)c1=O Cc1c(C(=O)N(C)CCN(C(=O)C(C)Sc2ccccn2)C)ccc(F)c1F c1(CNC(=O)NCCCn2ncc(C(=O)OCC)c2)c(C)nn(C)c1OC N1(C(C(CC=C)CC(C)C)=O)CCCCC2(CCN(C(=O)C(=O)C(F)(F)F)C2)C1 C=CCC(CNC(=O)C(F)=CC1CC1)NC(c1ncoc1CCCC)=O c1(C(=O)NCC2OCC(CNC(c3n(CC)nnc3)=O)C2)cc(Cl)ncc1O C1(CC)CN(C(=O)CC2CC(=O)NC2=O)CCN1C(=O)Cn1cc(C(F)F)cn1 N1(C(CCCc2onc(CCC)n2)=O)CCC=C(CNC(=O)COC(F)F)C1 c1(OC)ccc(S(=O)(=O)N2CC=CC2C(=O)Nc2ccc(Cl)c(C#N)c2Cl)cc1 c1(CN(Cc2onc(C)n2)Cc2cccc(F)c2)n[nH]c(C)c1Cl C1(CCCC)CCC(C(=O)NC2CCC(NC(C3(O)CCC3)=O)CC2)CC1 c1(CC)ccc(C(=O)NC2CN(C(=O)C(C)N(C)C)CCC2CO)cc1Br CC1CC(C(=O)NCC2(CCO)CC2)N1C(=O)CSCCN(C)C c1(C(N(CCNC(CC(C)C(C)(C)C)=O)C2CC2)=O)cnc2c(cnn2C)c1N c1(C(=O)NC2(C)CCCN(C(CCC(C)C#N)=O)C2)n[nH]c2c1CCSC2 C=CC(C)(O)CC(=O)N1CCC(O)(CCNC(c2sccc2OC)=O)C1 c1(CC)ocnc1C(=O)NC1CC1CNC(=O)C(F)=CCCF C1(CNC(=O)Nc2c(OC)csc2)COCCN1C(=O)C(C)c1cccs1 C(=O)(C(C(C(C)CC)OC)N1CCCCCCC1C)NCC C(C)(CCC(=O)NCC(C)(C1CCC1)NC(=O)C=CC(C)(C)SCC)OCC C1(NC(C2(OCC)CCOC2)=O)C=CCCC1C(=O)NCCCC(N)=O C(=O)(C1=CC2(CCOC2)C1)NC(CNC(CCC1CC(OC)C1)=O)C(C)C C1(C(N(CC(c2ccccc2)O)C)=O)CC12CCN(Cc1cccc(O)c1Br)C2 C1(CNC(C(C)(C)C)=O)C(C2CC2)CCN1C(=O)Cn1cnc(C(N)=O)n1 c1(OC)ccc2onc(NC3CCCN(S(=O)(=O)C(C)(C)C)C3)c2c1 C1(NC(c2c(CC)n(C)nc2)=O)CN(C(c2cc(F)c[nH]2)=O)CC1C1CC1 Fc1cc(Br)ccc1C1CCN(CN2CC=C(Br)CC2)C1 CC1CC(C)(C(N2CCC(CNC(=O)CC3CCSCC3)C2)=O)CC(C)O1 C(=O)(C1CCCc2nnn(C)c21)NCCC1(NC(C(CC=C)CC(C)C)=O)CC1 c1(SC(C)CNC(=O)N(CCC(c2ccccc2)O)CCO)ccc(Cl)cc1 C(=O)(C(CC(N)=O)NC(C1CCCSC1C)=O)NCC(C(C)O)O c1(-c2nc(-c3cccc(C)c3)nn2CC2CCSC2)scc2c1CCCC2 CCC(CC(=O)NCC1(C)CCCN(C(=O)COCCCOC)C1)C(F)F N1(C(CC(CCC)CC)=O)CC2(C)CN(C(=O)C(C3CCC(=O)N3)C)CC2(C)C1 C12(NC(C(CN(C(=O)OC(C)(C)C)CC)F)=O)CC1CN(C(c1ccnn1C)=O)C2 c1(-c2cc(C(=O)NCc3cccnc3Br)c(Cl)nc2)cnc2c(F)cccc2c1 [N-]=[N+]=NC1CCC(C(=O)NCC(O)CNC(C2(C3CCC3)CC2)=O)C1 c1(C(=O)NCCC(CNC(C2(C)CCCO2)=O)O)c(Br)ccc2n[nH]cc12 C(=O)(CC1NC(=O)c2ccccc21)NC1(CC=C)CN(C(C2CC2=C)=O)C1 S(=O)(=O)(c1cccc(Cl)c1F)NC1CN(C(c2ccnc(OC)c2F)=O)CC1O C1(NCc2cccc(OC)c2)CCC2CC(F)(F)CC2C1 C1(CS(CN(C)C(N)=O)(=O)=O)CCC2(CC(NC(N3CCc4ccccc43)=O)C2)O1 N1(C(C(=O)NCC2CCC(NC(C(CC)=CC)=O)C2)C2CC2)CCN(C)CC1 C1(C(N2CCCC(F)(CNC(c3ccoc3Cl)=O)C2)=O)CCc2ccnn2C1 c1(SCC(=O)NC2CCCC2n2cc(Br)cn2)ccc(C(=O)OC)cc1[N+](=O)[O-] CC(C)C(C(=O)N1CC(NC(C2CN(C(N)=O)C2)=O)C(O)C1)c1cccc(Cl)c1 C1(CC)CCCN(C(c2cc(C(=O)OCC)on2)C(=O)NCCCSCC)CC1 C(C)(C)(CC(=O)NCCc1cnn[nH]1)NC(COCCC=C)=O CC(=O)C(C)CC(C)C(=O)N1CC(O)CCC1C(=O)NCc1noc(C)n1 CCCCC(C)CCC(=O)NCC1CCC(C(=O)NOCC(F)F)C1 C1(NC(CCC=C)=O)CC2CCC(C1)N2C(=O)COc1ccc(Cl)nc1 c1(C(N2CCCC(CN(C(C(COC)C)=O)C)C2)=O)csc2cnccc12 C(=O)(CC(C)(C)C)NC1CC(NC(C(C)NS(C)(=O)=O)=O)C1.C1(=O)CCN1 c1(C(=O)NCC2CCN(c3sc(C(=O)OC)c(Cl)n3)C2)noc2cc(Cl)ccc12 CC(C)(C(=O)NCCCCC(N)=O)C1=CCN(C(c2ccc(C3CC3)o2)=O)C1 C(=O)(C1=NOC(C)(C)C1)NCCCOCCC(=O)NC(CCOC)C(C)C N1(CC(=O)NCC2C(NC(CN3CC(C)(OC)C3)=O)COC2)CCNC(=O)C1 C=Cc1ccc(C(N2CC(NC(=O)CCCn3cncn3)C(C=C)C2)=O)cc1 C1(CN(C(=O)C(c2cccnc2)O)C)CCCN1C(c1c[nH][nH]c1=N)=O N1(C(c2nc(CC)sc2N)=O)CC2CC(C1)CN(C(C1C3CS(=O)(=O)CC13)=O)C2 c1(C(N(C(C(=O)N(C)Cc2snc(C)n2)C)C)=O)cn(CC)nc1C C1(CNC(C(N2CCNC2=O)C)=O)CCCCC1C(=O)NCC#CC#CCO N1(C(C2C(C(N)=O)C2)=O)CC2CC(C1)N2C(=O)CC1(N(C)C)CC1 C1(C(=O)NCC2(OCC)CCCC2)CCC=CC1NC(c1cn(C)cn1)=O C(=O)(CC(C(C)(C)C)NC(=O)Cc1cncs1)NC(C1CCOC1)C C(C(CC(C)C)OC)NC(c1nccn1C)=O.C1(C(=O)NC)(C)CC1 c1(C(=O)NC2CCC3CCN(C(C(CC)CC)=O)C32)ccc2c(c1)C(=O)C(=O)N2 c1(-c2c(C)occ2)nc(CC(O)CF)n(C(C)C2CC2)n1 c1(C(N(C(C)CCNC(c2ccc(C3CC3)cc2)=O)C)=O)ccc(S(C)=O)cc1 N1(C(C=CCN(C)CC)=O)CCN(C(=O)Cc2ccsc2)C(c2ccccc2)C1 c1(OC)cc(C)c(CN2CCC(O)(C(=O)Nc3ccc(O)cc3C)C2)cn1 N1(C(c2n(C(C)C)ccn2)=O)CC2(CC(C(N3CC(C)C(F)(F)C3)=O)CO2)C1 c1(CC(=O)NCCNC(C(CC)(C)F)=O)cc(F)cc2c1OCOC2 C1(C(C)(C)C)CC(C(=O)NCC2CCCCC2NC(=O)COC2CCCC2)=NO1 c1(C(N(CC(=O)OC(C)(C)C)C)=O)ccc(C2CC2)o1.C1(=O)C(C2CC2)CN1 C(=O)(C(C)(C)CO)N(CCCCN(C)C(C1C(F)(F)C12CC2)=O)C c1(C(=O)NC(C2CC=CCC2C(F)(F)F)CC(=O)OC)nccc(SC)n1 c1(NC(=O)CN2CC(CO)C(O)C2)ccc(Cl)c([N+](=O)[O-])c1 C1(NC(C2CCCC2)=O)CCN(C(C2CCCCO2)=O)CCC1CO c1(C(N(C)CC2CCCN(C(CC3(NC(C)=O)CC3)=O)C2)=O)ccc(C#N)n1C c1(OCCN2C(COC)C(C)CC2)ccc([N+](=O)[O-])cc1.n12cc(nn1)C2 CCCC(CNC(c1cccc(CNC(=O)C(C)CC(C)C)n1)=O)CCO c1(CCCC)ccc(C=CC(=O)NC2CC2CN2C=N2)o1.C(C)(c1ccsc1)=CC C(=O)(C(N=[N+]=[N-])C(C)C)N(CCC(=O)Nc1cc(C)c(F)nc1)CCO CCC(C(=O)NC1CCCC1CCNC(c1ccoc1)=O)NC1CCC1 c1(CCC(N2CC(COC)C3(C2)CC3)=O)ccnc2ccccc12 N1(C(C(C(COC)C)C)=O)CCC2(CCOC2)C(CNC(C2(COC)CC2)=O)C1 C12(NC(C(C)CO)C)CCC(C)(CC1)OC2 c1(C(N2CCC(F)(C(=O)NC3CCCC(O)C3)C2)=O)ccc(O)cn1 c1(CNC(C(N2C(C)CCC2C)C)=O)nnc2n1CCC2 C1(C(=O)NC(C(C)(C)OC)C)CCC2CCC1N2C(=O)C(C(C)C)C1CCC1 C1(C(C)NC(C2C(COC)C2)=O)CCN(C(=O)CC(=O)Nc2nccs2)CC1 c1(OC)ccc(C(F)(F)C(=O)NC(C)CC(C)NC(=O)CCCCC2CC2)nc1 C1(C(=O)OC)COCC1COC(=O)C(F)C1CC(C(C)(C)C)C1 c1(OCC)nn(C)cc1CNC(=O)NC(COC(C)C)CO N1(C(COc2cn(C)nc2)=O)CCCCC1C(=O)NC(C1CCCO1)(C)C N1(CCC=CCCC)CCC(N(C(=O)CC(C)n2ccc(C)n2)C2CC2)CC1 N1(C(=O)CCC2CCC2)CCC2(CCCC2C(N2CCCOCC2)=O)C1 N1(C(c2cnn(C)c2C#N)=O)CC(C)(C(N2CC(CO)C(O)C2)=O)CC1(C)C n1(C(CC)C)nnnc1C1(NC(CC2CC2)C2CC2)CC(OC(C)C)C1 Cc1ccc(C(=O)NCC2CN(C(=O)C(C)C3CCCO3)CCC2C)c(F)c1F c1(C2(CN(C3CCCN(C(c4cc(C)on4)=O)C3)CCO)CC2)cc(F)ccc1Cl C1(CC(=O)NC(C(=O)NCC2(COC)CC2)Cn2ccnn2)CC=CCN1C Cc1cc2c[nH]nc2c(C(=O)N(C)Cc2ccc(Oc3cccnc3)cc2)c1N n1(CC(N2CCCCC(N(C)C(=O)OC(C)(C)C)C2)=O)cc(F)ccc1=O N1(C(C2=CCN(C(CC(CC)SC)=O)C2)=O)CCCC2(CCC2)C1 c1(C(N(CC)CC2CCCN2CC(O)COC(C)C)=O)cc2ccccc2[nH]1 c1(CCn2cc(CNC(c3c(C)cc[nH]3)=O)nn2)ccc(Br)nc1 c1(-c2c(OC)cccc2C)cc2c(s1)CCN(C(c1ccno1)=O)C2 C1(NC(c2ccn(COC)n2)=O)CC2CCC(C1)N2C(=O)C(F)(F)C(C)O N1(C(C2CCN(C(=O)OC)CC2)=O)CCC2CN(C(=O)C(C)CC(C)(C)C)CC12 C12(C(N3CC(C(C)NC(C4CC4C)=O)OCC3)=O)CC(CO)(C1)OC21CCC1 c1(C(=O)NCC2CC(NC(CNC(c3c(C)occ3)=O)=O)C2)c(Cl)ccc(O)c1N Cc1ccc(NC(=O)NC2CCN(C(=O)NN(c3ccccc3)C)CC2)cc1C C1(C(=O)Nc2cccnc2CO)CC(F)(F)CN1C(=O)CC1(O)CCC1 c1(C(=O)OC)cncc(C(=O)NC2(CNc3ncncc3Br)CCCC2)c1 c1(OCC)nccc(C)c1C(=O)NCCc1ccc(OC)cc1F c1(OC)ccc2cccc(NC(=O)C(n3nc(C)cc3C)C)c2n1 Cc1cc(N(C)Cc2ccc(Cl)cc2)ncc1S(=O)(=O)NC1CCN2CCCCC12 Cc1ccnn1CC(=O)NCCn1cnc(C(=O)NCC=CCl)c1 Cc1oc(CO)cc1C(N1CCC(CO)(NC(C2CC2c2ccncc2F)=O)C1)=O N1(C(Cc2cc(C)cc(C)c2)=O)CCN(C(=O)C2=CCCCC2)CCC1C N1(C(c2cnc(C)nc2O)=O)CCC2CCC(NC(=O)CC3C=CCCC3)C1C2 C(=O)(CCC(=O)NC1(C2CCCN2C(=O)CC(C)C2CC2)CC1)SC N1(C(C2N(C(c3n(OC)cnc3C)=O)C(C)C2)=O)CCC2(CNC(=O)N2)C1 CC1CN(C(c2cccc(=O)n2C)=O)CC(CCNC(c2sccc2CO)=O)O1 N1(C(C2(CNC(C3CN4CCC3C4)=O)CC2)=O)CCC2OCCCC2C1 c1(N2C(C)CN(C(=O)Cc3cccs3)CC2)c(O)nc(=O)n(CCN(C)C)c1N C1(=CCNC(CC(C)n2cccn2)=O)CCN(C(C2CCCNC2=O)=O)CC1 c1(C(N2CCOCC2Cc2cn(CC(F)(F)F)nn2)=O)ccc2scnc2c1 n1(CC=C)cc(C(=O)N(C(C)CNC(=O)C(O)CN2CCOCC2)CC)cn1 c1(CN(C(N2CCCC(CS(C)(=O)=O)C2)=O)C2CC2)ccc(C#N)cc1 CCC(C)(COC)C(=O)NCCCCC(=O)Nc1cc(C)ccc1CO Cc1cc(CNC(=O)CCOCCCNC(c2ncccc2N)=O)sc1C C1(C)(N(C(=O)CN2CCN(c3nncs3)CC2)C)CCCOC1 C1(NC(C(C)OC2CCCC2)=O)CN(C(=O)C=C2CCN(C)C2)CCC12CCC2 C1(C)(C(=O)NC2CCCN(CCC)C2)CCCN(C(=O)C=Cc2ccc[nH]2)C1 c1(NC(CCC)(C)c2nnnn2-c2c(C)cccc2C)cc(F)c(Br)cc1C n1(CC)ncc(C(=O)NC(C)CCNC(c2ccc(C#N)[nH]2)=O)c1C(F)(F)F C(=O)(C(C)(C)CCC)N(C)CC1N(C(Cn2c(CCC)ncc2)=O)CCC1 c1(OC)c(Cl)cc(C(=O)NCCOCCN(C)C(C2CN(C)CC2C)=O)nc1Cl c1(CC)ncc(C(=O)N(CC(O)CNC(c2nocc2C(C)C)=O)C)s1 N1(C(COC(C)C)=O)CCC2(CC1)CN(C(c1csc(=N)[nH]1)=O)c1ccccc12 C1(C(=O)NCCCCN(C(C(C=C=C)C)=O)C)(OC)CCC(C)(C)C1 C=CC1CN(C(=O)CCC2(C)CCC(=O)N2)CC1NC(=O)C=CC(C)(C)SC N1(C(c2ccnc(C)c2N)=O)CC2CC(C(=O)NCCN=[N+]=[N-])C(C2)C1 c1(C(N2CC(N(C(c3c(COC)noc3)=O)C)C(F)C2)=O)c([N+](=O)[O-])cnn1C S(=O)(=O)(c1cccnc1NCC1(CC2CCC2)CC1)N1CCN(CC(C)O)CC1 CC(C)CC(O)C(C)C(=O)N1CC(C(=O)NCC(C)(O)C(F)F)C(C(C)C)C1 C1(NC(=O)Cc2cn[nH]c2)CCC(NC(c2ncoc2C(F)F)=O)C1 c1(C(N2CC3(OCCN(S(C)(=O)=O)C3)C2)=O)c2n(c(=O)n1C)CCCC2 c1(C(=O)NC2CN(C(c3n(C)ncc3)=O)CC2O)ncc(Cl)cc1O C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)NC1CCC(NC(CCP(C)(C)=O)=O)C1 c1(CN(C)C(C2CC(c3ccc(Cl)s3)C2)=O)sccc1Cl CC(C)C(C(=O)NC1C=CCCCC1)NC(=O)CCN(C)CCO C1(C)(C(=O)NCC2(CC)CN(C(CCOCCCOCC)=O)C2)CCN(C)CC1 C1(C)(NC(COCCSC)=O)CCN(C(C2CCC(=O)C2)=O)CC1 c1(CC=CC=C)nc(C2CCOC2)nn1C(C)C c1(CC)cc(C(=O)NCc2cccc(NC(=O)C(C3CC3)C3CC3)c2)cc(N)c1 C(=O)(C(C(C)O)NC(C)=O)N1C(CNC(c2c(CC)nc[nH]2)=O)C=CC1 N1(CC)C(=O)CCC1CC(=O)NCC(C)(C)CNC(C1CCN(C2CC2)CC1)=O c1(C(N2CC(C(=O)NCC3CCCC(OC)C3)C(C)C2)=O)ncc(C)cc1C C(CN=C(NCCF)NCc1occc1C)c1ccc(SC)cc1 C#CC1(NC(C2CCC3(CC3)N2C(C2C3CCC(F)C23)=O)=O)CCCCCC1 O=C(C1=NOC(CNC(C2(O)CCCOC2)=O)C1)NC1CCCC1O CC1(C)Cc2cc(C(=O)NCC3C4CN(C(C5CCC(=O)O5)=O)CC34)ccc2O1 c1(CNC(C)=O)cc(C(=O)N(C(=O)CO)Cc2ccccc2)ccc1C c1(C(N2C3CN(c4ncc(CC)cn4)CC2C3)=O)cc2ncccc2o1 C=C(C)C(C)(C)C(=O)NCC1CC(F)(CNC(c2cc(Cl)sc2NC(C)=O)=O)C1 C1(O)(C(C)NC(=O)CCOc2ccc(Cl)cc2)CCN(C(=O)C(=O)N(C)C)CC1 C1(NC(C2N(C(CN3CC(C)(OC)C3)=O)CCCC2)=O)CN(C)CC1(F)F N1(C(C(=O)NCCC#N)c2cn[nH]c2)CCC2(CCC2)C1 Cc1cc(=NC(=O)C2C(NC(=O)C(CO)C(C)(C)C)C2(C)C)[nH]n1C(C)C C(=O)(C1=C(C)CC1)NCCn1cc(C(N2CC(C(=O)OC)(OC)C2)=O)nn1 C1(C(=O)NC2CC(CN=[N+]=[N-])C2)CC2CCCCC2C1 N1(C(CN(C)C)=O)C2CCC1CC(N(C)C(C1C(C)(C)C1(C)C)=O)C2 Cc1cn2c(n1)CC(C(=O)NCC1CN(C(=O)C(C)OC3CCCC3)CC1O)C2 C(=O)(C1=CC2CCC(C1)C2)NCC(C(=O)NCC(CC)CO)N(C)C O=C(C1=COCC1)NCCC1CCN(C(c2oc(Br)nc2C(F)F)=O)C1 N1(C(C(CC2CCCC2)OC)=O)CCNc2cc(Cl)ccc2C1 c1(CNC(N2CCC2CC2CC(=C(F)F)C2)=O)ccnc(OC(F)F)c1 C1(CNC(c2nn(CC)c(C)c2)=O)CC2CCCC2N1C(=O)C#CC1CCCO1 C1(C(N2C(CSC)CCC2)=O)CN(C(C2CC3(CSC3)C2)=O)CC1(F)F S(=O)(=O)(c1ccccn1)NC1CCN(C(CN(CC(=O)O)C2CC2)=O)CC1(F)F c1(C(N(C)CC2CN(C(CN(C)C(N)=O)=O)CC2O)=O)cccc2[nH]ncc12 c1(C(=O)NCC(C)(C2CCC2)NC(C(COC)N(C)C)=O)cc2cccnc2s1 CC1(OCC(=O)NC2(C)CN(C(=O)C(F)C3CCOC3)C2)CC(O)(CO)C1 N1(C(c2c(CC)scn2)=O)CC(CNC(c2cn(C(C)(C)C)nn2)=O)CC1C C1(N(C(=O)CCOCCCOC)CCC)CCN(C(=O)C(C)SC(F)(F)F)C1 c1(OCC)c(Cl)cc(C)nc1C(N1CCC(NC(=O)C(n2nccc2C)C)C1)=O CCC(CC)C(=O)N1CCC(CNC(C2CC2C(=O)OC(C)(C)C)=O)C1 N1(C(c2cnc(N)c(Br)c2)=O)CCCN(C(C2CCSC2)=O)CCC1 C1(C(=O)NCCCNC(C(C(=O)NC)(C)C)=O)CC12CCc1ccccc12 C1(N(C(CC(=C)C)=O)C2CCCC2)CCCN(C(=O)CCC2C(=O)ON=C2C)C1C CCC(C(=O)NC1CCCC1C(N)=O)N(C(=O)CC1CCCSC1)C C1(CC(C(=O)NC2CC(F)(F)C2)N(C)C)COC(C)(C)C1 c1(C(=O)NC(CC2CN(C(COC(CC)C)=O)C2)C)cnc2n1CCS2 c1(C(C)NC(=O)NC2C(CC(=O)OC)CCC2)ccc(OC)cc1 C12(C(=O)NC3CC(CNC(C4(c5ccc(F)cc5)CC4)=O)C3)CCC(CC1O)C2 CC(CC(=O)NCCCN1CC=CC1)NC(c1ccn(CCF)n1)=O c12ccc(cc1)-c1cn(nn1)CCO2.C(C)(C(=O)NC(C)(C)C)NC(CC)=O N1(C(C2C(C)=CCS2)=O)CCCCC2(CCN(C(c3cc(Cl)ccn3)=O)C2)C1 C(C(O)CC(=O)NCCOC1CCN(C(=O)CC(C)(C)C)C1)N(C)C C(=O)(C1=CC2(CCOCC2)C1)N1CC(N(C)C(=O)C2CC2)C(F)C1 c1(C(N2C3CCC(NC(c4ccc(C)cn4)=O)(C3)C2)=O)cnc([N+](=O)[O-])n1C C=CC1OCCC1C(=O)N(C(C)(CNC(=O)Cc1cccnc1O)C1CCC1)CC c1(C(=O)NC(C(C(C)C)NC(c2sccc2C#N)=O)C)nc[nH]c2ncnc1-2 C1(CC)C(C(N2CC(F)(CO)C2)=O)CCCN1C(=O)Cc1ccnc(O)c1 c1(C(=O)NC2CC(NC(=O)CC3C=CS(=O)(=O)C3)C2)cc(Cl)cc([N+](=O)[O-])c1O N1(C(C(CCC)OC)=O)CC(NC(c2cn(CC)nn2)=O)C(S(C)(=O)=O)C1 CC(C)C(O)CC(=O)N1CCC(CNC(=O)C(=O)NCCC(N)=O)C1 N1(C(C(COC)(C)C)=O)CC2(CC(CC(N3CCCNC(=O)C3)=O)C2)C1 CC1CCC(NC(C2CCCC2C2CC2)=O)CN1C(=O)Cn1cccn1 c1(C(=O)Nc2ncc(-c3c(C)cc(Cl)nc3)cc2O)cc(C)c2c(cnn2C)c1 N#Cc1ccc(CNC(c2conc2CNC(c2ccncc2)=O)=O)nc1 c1(C(=O)NC2C3CCN(C(CCNC(=O)CO)=O)C32)cc2cccc(F)c2o1 c1(C(N2CCCC(C(N(CCO)CC)=O)C2)=O)ccc(Br)c2ncccc12 Cc1nc(CC(=O)NCC(C)(CO)NC(=O)CC2CCCC2)c(C)s1 Cc1cc(C(=O)N(CC(C)NC(C2(C)CCCO2)=O)C)c(O)c(C)n1 C1(OC)CCCC(CC(=O)NCCCCC2(CNC(=O)CC3CCCC3)CC2)C1 N1(c2cc(OC)nc(OC)n2)CCC(NC(=O)CC2CCCCN2C)C12CCC2 N1(C(C2CCN(C)C2)=O)CC2OCCN(C(=O)CC3(C(F)F)CC3)C2C1 CCC(C)(C)CCCC(=O)N1CC(O)(C(F)C(=O)N(C2CCC3CC23)C)C1 CC(C)CC(CNC(C12CCCC1C2)=O)NC(c1ccnn1C1CCCCC1)=O S(=O)(=O)(C1CC1c1ccccc1Br)NCC1(C(=O)OCC)CCC1 N1(C(CCCCC)=O)CCC2CCC(C1)N2C(C1CCS(=O)(=O)N1C)=O c1(OC)ncnc(C(=O)NC2(CCCNC(=O)CC3CCCOC3)CC2)c1F C#CC1CN(C(C2CCC(C)(C)CC2)=O)CCN1C(C1CC(n2ccnc2)C1)=O C1(NC(C2CC(C)(CC)C2)=O)CCN(C(C2CCCC(C)C2)=O)CC1 C1(OC)(CNC(=O)C(CC)SC)CCN(C(=O)C(F)(F)c2nccn2C)C1 c1(C(=O)NC)cccc(C(=O)N(C)CC2CCCN2C(c2cnn(C)c2)=O)c1 N1(C(c2cc(C#N)oc2)=O)CC2=C(C1)CN(C(c1ncnc(O)c1Br)=O)C2 c1(C(C(=O)NC(CC)CNC(=O)Cn2cnnn2)=O)cc(F)ccc1C C1(C(C)C)C(C(N2CC(O)C(O)C2)=O)CCN1C(c1ccccc1F)=O c1(N2CC3(C)CN(C(CSCCC)=O)CC3(C)C2)ncnc2c(Cl)cc(Cl)cc12 N1(C(CCNC(COC)=O)=O)CC2CCN(C(C3OC(C)CC3C)=O)CCC2C1 C12(C(N3CCC(C)(NC(CCNC(=O)OC)=O)C3)=O)CCC(C(F)(F)F)(CC1)C2 C1(C(N(C2CCN(C(=O)CCCn3cncn3)C2)C)=O)CCc2cnn(C)c2C1 c1(C(N2C(CNC(c3nc(Cl)cs3)=O)CC(OC)C2)=O)cc(C)cc2c[nH]nc12 N1(C(C(CNC(C2(OC(C)=O)CC2)=O)C)=O)CC2(COC(C)C2)C1 CC1CN(C(=O)CSC2CC2c2ccccc2)CC1(C)C(=O)O N1(C(C2C(C3(C)COC3)C2)=O)CCC(C(=O)N2CC3CC2CS3)=C(F)C1 N1(C(C(C)SCC)=O)CC2(C1)CN(C(=O)CC1=CCCCC1)CCO2 c1(OCc2nc(-c3ncn(CC(=O)OC)n3)on2)ccc(Cl)cc1Cl C1(C(=O)NC2CC(C)(CNC(COCC#C)=O)C2)CCc2nnc(C)n2C1 c1(C(N2CCC(C(=O)NCc3cnccn3)O2)=O)cccc([N+](=O)[O-])c1 CCC(C)CCCCC(=O)N(C)CCN(C(C)C(=O)NC1CCCCC1C)C N1(C(CC2N(C)CCCC2)=O)CCC2(CC1)CN(C(=O)Cn1cccc1)CCO2 C1(NC(c2c(CCC)n[nH]c2)=O)CCC(C)N(Cc2cc(-c3cccs3)on2)C1 c1(C(=O)NC2CC(CCNC(CC3CC(C)C3)=O)C2)cc2ccccc2cc1O N1(C(CCCC#N)=O)CC(C2CCCN(C(C3CCC(C(N)=O)O3)=O)C2)C1 N1(C(Cn2c(C)ccn2)=O)CCC(N(C(C2CCCCO2)=O)CC2CC2)CC1 CCCC(C)C(C)(c1nnnn1CCCSC)NCc1cc(CC)nn1C N1(C(c2ccc(OC)s2)=O)CC2CCC(CNC(c3ccnnc3)=O)(C2)C1 N1(C(c2n(C)nnc2)=O)CC2CCCC(CNC(=O)C=Cc3ccncn3)C2C1 N1(C(c2c(N)cc(F)c(Cl)c2)=O)CC2CC(C1)CN(C(c1ccnc(S)c1)=O)C2 C(=O)(C(C(C)C)OC)NC(COCC)C(=O)NCC(C)(C)CCOC C(=O)(C(CC(F)F)c1ccccc1)NCC(CN(C(c1nccc(C)n1)=O)C)O CC(C)(C)C#CC(=O)NC1CC(C(=O)NCCN=S(C)(C)=O)C12CCC2 C1(NC(CNC(c2c(C)occ2)=O)=O)CCCC(NC(c2nc(O)sc2C)=O)C1 C=CCC(CC(C)C)C(=O)NCC1C2CC1N(C(=O)CCC1CC(F)(F)C1)C2 Cc1nn(C)c(C)c1C(N1CC2(CC2C(=O)NCCN2CCNC2=O)C1)=O C=CCCCC(C(=O)NC1COCC1SC)NC(C1CC12CCCC2)=O S(=O)(=O)(c1ccc(F)c(F)c1)N(C1CCC(CC)CC1)C1CC2CC1CN2 c1(Cc2nc(C(CCC)C)nn2-c2ccnc(F)c2)c(C)nc(CC)nc1C C1(C(=O)NCCCC2CCC2)CCCN(C(=O)C(F)n2ccnc2)CC1 C(=O)(C(C)C(C)S(C)(=O)=O)NCC1CCN(C(c2cncc(NC)c2)=O)CC1 C1(C)(CNC(CCCC)=O)CCCC1NC(=O)COc1ccsn1 N1(C(Cc2cc(C)on2)=O)CCOC(CNC(c2[nH]ccc2C)=O)C1 C1(C(=O)NC(c2ccccc2O)C)CCCCCN1C(=O)CC1CCC1 C1(C(N2C(CN(C(CCCN(C(C)C)C)=O)C)CCC2)=O)CCCCC12CC2 c1(C(O)CNC(=S)Nc2ccccc2F)ccccc1[N+](=O)[O-] c1(C(N(CC(C)Nc2ncc(C)c(C)n2)C)=O)c(C)cccc1[N+](=O)[O-] N12CCCC1(C)C2=O.c1(CCC(=O)NC2CC(OC)C2)nc(C)c(C)o1 c1(SCC(N2CC(n3cc(-c4cnn(C5CC5(F)F)c4)nn3)C2)=O)ccc(Br)o1 CCCC(CCC)CC(=O)NC1C(C)CN(C(c2cc(Br)n[nH]2)=O)CC1C C1(CN(C(C)=O)C)CN(C(=O)C(Cc2cccc(C)c2)N(C)C)CC12CC2 c1(OCC(=O)N(CCCN2CCOC2=O)CC)c(F)cccc1F Cc1ccc([N+](=O)[O-])c(N(CCCNC(=O)Cn2cnc([N+](=O)[O-])c2)C)c1 c1(CC(=O)NCC(CCNC(C(C)(C)SC)=O)O)cnccc1C c1(C(=O)NC(CNC(CCCSC)=O)C(C)C(C)C)cc2nc[nH]c2cc1N C=CC(C)(C)CN(C(=O)C(C)OC1CCCC1)Cc1nnn(C)n1 c1(CC(=O)N(CC(C)NC(CCC=CCC=C)=O)C)ccc(C#N)cc1F C(=O)(C(C)C1=CCCC1)NCC(=C)CCNC(=O)C1=CCCCC1 c1(C(N(CCNC(=O)CC2(C)CCCO2)CC)=O)n[nH]c2c1CN(C)CC2 N1(C(c2ncn(CC)c2)=O)CCN(C(c2ccco2)=O)C(C(C)C)C1 CCCCC(O)C(=O)Nc1ccc(CNc2c[nH]nc2C2CNC(=O)CO2)cc1 c1(CC(=O)OCCC(F)(F)C(F)F)c[nH]c2cnccc12 c1(C(N2C(CNC(Cc3scc(CC)n3)=O)CC2)=O)ncccc1C c1(C(=O)NCC(C)N(C(=O)C(C(C)C)NC(C)=O)CC)cc(Cl)ncc1F N1(C(C(C)OCC=C)=O)CCCC(CCNC(C2CC(=C(F)F)C2)=O)C1 CCC(C(=O)NCC(C1CCN(C(c2cc(C(C)C)oc2C)=O)CC1)C)C(C)C C(C)(C)(CCCC(=O)NCC1CCCCO1)NC(COCC(=C)C)=O c1(NC(C(C(C)NC(C=CCC)=O)C)=O)ccc2nc[nH]c2c1 C1(N(CCN(C)C(C2CCC3(CCC3)O2)=O)C)CC2CCCCC2NC1=O C12(C(N(CCNC(C(CCCC)O)=O)CC)=O)CCCCC1CCCC2 C1(NC(C2N(C(COCCSC)=O)CC=CC2)=O)CC=C(C(C)C)CC1 N1(CCN2C(=O)NCC2)CCCCC1CCO N1(C(CCOC(C)C)=O)CCC(N(C)C(C2CCC2C(c2ccccc2)=O)=O)C1 N1(C(CCN(CCCCC)CC)=O)CCCC(CNC(=O)C(F)CC2CC2)C1 Cc1cn2cc(C(N3CCC(C(C)NC(=O)C4=CCCC4C)CC3)=O)nc2s1 O=C(C1=CC2C=CC(C1)C2)NC1(CNC(c2cncc(O)c2)=O)CCOC1 c1(CCC(=O)NC(CN(C(c2n(CC)ccc2)=O)C)C)c(F)cccc1Cl c1(CN2CCC(NC(C3(N=[N+]=[N-])CC3)=O)C2)nnc2n1CCCCC2 Cc1nc(C2CCCCC2)sc1C(=O)NC1C2CN(C(c3cc(C)ns3)=O)CC12 N1(C(C2(COCC)CC2)=O)CC2(CCCCN(C(=O)CCSCC)C2)C1 N1(C(C(C)CC2CC2)=O)CC(NC(c2ccc(-c3nccs3)cc2)=O)C(CO)C1 C1(CC)(NC(=O)CCN(C)CCO)CCN(C(C2(COC)CC2)=O)CC1 C(C)(C)(CCN=c1cc(C(C)(C)C)nc(Cl)[nH]1)NC(C(C)Cc1ccccc1)=O N1(C(CCCC#CC)=O)CC2ON=C(CNC(=O)CCn3ccc(C)n3)C2C1 N1(C(c2c(CC)nccn2)=O)CCCN(CCNC(C2(C(N)=O)CC2)=O)CC1 c1(C(C)=O)ncc(NC(=O)NCC2(N3CCOCC3)CCCC2)s1.C1(C(=O)N)CC1F c1(CN(C(=O)C(=O)NCCCc2cccnc2)CCN(C)C)ccc(F)cc1 C1(CCNC(c2ccc(C)cc2)=O)CC(N=c2[nH]c(C(=O)O)nc(C)c2C)C1 C1(Nc2ccc(O)cn2)CC2CCC(C1)N2.N1(C(CO)=O)CC(N(C(C)(C)C)C)C1 C1(C(C)NC(CN(C)CC)=O)CN(C(=O)C(C)C(C)c2ccc(F)cc2)CCO1 CC1(C)C2CCC(C(=O)NCCC3(O)CN(C(C4(F)C(C)(C)C4(C)C)=O)C3)C1C2 C1(CC)CC(C)CN(C(C2(C(C)C)CCCN2C(c2ccn(COC)n2)=O)=O)C1 Cc1ccc(S(N)(=O)=O)cc1C(=O)NC1CCC1CNC(=O)C(C)(C)n1cnnn1 Cn1nc2c(c1NC(C1(C)CCN1Cc1nccc3ccccc13)=O)CCCC2 C#Cc1cccc(C(=O)NCC2CC(F)(CNC(C3(F)CCOC3C)=O)C2)c1C C#CCC(C)(CNC(=O)CSCCNC(C1CCSCC1)=O)CO Cc1ccc2c(C(=O)NNC(C3(C)CCCS3(=O)=O)=O)[nH]nc2n1 Cc1cc(C(=O)N(CCCNC(C2CCC2C(C)(C)C)=O)CCO)cs1 CC1(C)CC(C(=O)NCCSCCCO)CN1C(=O)C1=CCCOC1 CCC(C)C(C(=O)N(C1CCN(CCCOC)C1)C)NC(N)=O C(=O)(CC(C)CC(=O)NCc1ccc(C(N(C)Cc2ccccc2)=O)cc1)OC C1(O)(CCNC(=O)CC2(O)CCC2)CCCN(C(=O)CCc2cscn2)C1 N1(C=O)CCCC(N(C)C(C2CCCN2CCOc2ccccc2C)=O)C1.CN N1(C(c2ccc3scnc3c2)=O)CCC2(CCN(Cc3ccc([N+](=O)[O-])o3)C2)C1 CC1(C)CCCN(C(=O)C(=O)NC2CCCC(C(N)=O)C2)C1 c1(CC(N2CCCC(CN(C)C(c3csc(=N)[nH]3)=O)C2)=O)ccc(F)c(F)c1 c1(C(=O)NC(C)C(=O)N(C)CCC2CCC2)cncn1C c1(NC(C2CCCN(Cc3ccc(OC)nc3Cl)CC2)=O)cc(=O)n(C)c(O)n1 N1(C(C=CCCC)=O)CC2CCN(C(C3CCC4CC3CO4)=O)CCC2C1 C1(C(N2CCC(C(C)NC(=O)C(F)CC(C)C)CC2)=O)(OC)CCCCCCC1 C12(C(=O)NC3C(C)(C)CN(c4nc(Cl)c(C#N)s4)C3)CC3CC(C1)CC(O)(C3)C2 C1(CNC(C(C(=O)OC)C)=O)CN(C(c2cc(CC(C)C)on2)=O)C(C)(C)C1 N1(C(C2(CCCC)CCC2)=O)CCOC2(CCN(C(C3CCCCS3)=O)C2)C1 n1(C(C(N2CC(F)CC(NC(CCC=C(C)C)=O)C2)=O)C)nc([N+](=O)[O-])cc1C C1(CC)CN(C(=O)C(C)CSc2ccc(F)cc2)CCN1C(=O)C1=C(C)OCC1 c1(CCC)cc(C(=O)NC2CC(CCNC(c3ccnc(S)c3)=O)C2)n(C)n1 C(C(CC(C)C)C(=O)NC(C)CC1CC1)NC(CCOCCC)=O N1(C(c2n(C)c(S)nn2)=O)CC(CNC(=O)CC2COC(C)(C)C2)OC(C)(C)C1 N1(C(Cc2scc(C)c2)=O)CCCC(F)(C(=O)NCCCN2CCOC2=O)C1 C1(F)(CNC(COCCC)=O)CCN(C(c2cnc(O)o2)=O)C1 CCCC(C)(CC)C(=O)NC1CCCCCC1C(N1CC(O)(C2CC2)C1)=O Cc1ccc(COCC(=O)NC2CC2NC(=O)C(c2nc(C)cs2)C)cc1 C(=O)(CCCCC(N)=O)NC1(CCNC(C2C(C)=CCS2)=O)CCC1 c1(C(N2CC(N(C(c3cc(C)ncc3)=O)C)C(C)(C)C2)=O)cn(C)c(=O)cc1C CC1(C)CN(C(c2nocc2Cl)=O)CC1NC(=O)CC1CC1(Cl)Cl C=CCC(C(=O)N1CC(NC(c2cn3ccnc3cn2)=O)C(SC)C1)C(C)(C)C CCCC(C)(C)C(=O)NC1CCC1NC(C1CN(CP(C)C)C1)=O CC1(CCNC(c2cc[nH]c2C2CCCC2)=O)CCN(C(=O)COC(F)F)C1 N1(C(C2CC(=C)C2)=O)CCSC(C(=O)NC(c2ccc(F)cc2)CO)C1 N1(C(C2C(c3c(C)n[nH]c3)C2)=O)CC(S(=O)(=O)N2CCNCC2)C1 C#CC1C(C(=O)NCCOCCS(C)(=O)=O)C1(C)C c1(NC2CC3CN(C(COC(CC)C)=O)CC32)ccc(Br)c(C)c1[N+](=O)[O-] C1(CNC(CC)=O)CC2(CCN(C(c3ccc(-n4cnnc4)cc3)=O)C2)CO1 c1(C(=O)NC(CNC(c2ccc(NC)cc2)=O)C(C)(C)C)ccc2c[nH]nc2c1 N1(C(c2cnc(C)s2)=O)CC(NC(=O)C(C)(C)CN2CCN(C)CC2)CC(F)C1 C(=O)(CCCCC(=O)NCCC(C)CCNC(=O)CC1C=CCC1)NC c1(C(=O)NCCC(C)N(C(C#CC(C)C)=O)C)cc2cccnc2nc1N Cc1c[nH]c(=NCCCC(C)NC(=O)CCC2CC2)nc1S(C)(=O)=O N1(C(c2ccc(C)s2)=O)CCOC2(CCC(NC(=O)C(C)N(C)C)CC2)C1 C1(O)(CNC(c2ccsc2)=O)CC(NC(c2cn(CC3CCOC3)nn2)=O)C1 N1(C(C=CCOCCOC)=O)CCC(C(=O)NCC(C)(O)CCO)(OC)C1 S(=O)(=O)(c1ccc(Cl)cc1)NC1(NC(=O)Cc2cc(Cl)nc(Cl)c2)CCC1 C1(CN(C(=O)C(O)CC2CCOCC2)C)CCN(C(=O)CC2CS(=O)(=O)C2)CC1 CC(C)(CCNC(=O)CC1CSCCS1)NC(=O)CC1CCSC1 c1(C(=O)NCC(CSC)OC)cncc(CNC(c2ccc(O)cc2)=O)c1 C1(C(N2CCOC(CO)C2)=O)C2C3CC4C1C2C34C(=O)NC(C)C(C)(C)C N1(C(C2C(C)(C)CO2)=O)CCN(C(=O)CNC(N2CCCC2)=O)CC(O)C1 S(=O)(=O)(c1cc(C(F)(F)F)cc([N+](=O)[O-])c1)Nc1c(C(=O)OCC)c(F)ccc1 C1(F)(C(N(CCCCCNC(c2cncc(C(F)F)c2)=O)C)=O)C2CCCCC12 c1(C(=O)NCC2(F)CN(C(C3CC4CCC3O4)=O)C2)cccc2ccncc12 C1(CC)C(NC(=O)Cc2cc(F)ccc2C)CCCN1C(c1coc(Cl)n1)=O c1(NC(C)=O)cnccc1C(N1CCOC(CC(N2CC(C)(C(N)=O)C2)=O)C1)=O c1(N2CCC(C)SCC2)nc2ccccc2c(=NCC2(C)CC2(F)F)[nH]1 N1(C(c2ccc(CCC)cc2)=O)C2CCC1CC(NC(C1CSCC(=O)N1)=O)C2 C1(C(N2CC(C(N)=O)(CNC(C3CSCCS3)=O)C2)=O)CSCC(=O)N1 C1(C(=O)NC2CCc3nc(C)sc3C2)(CN)CC2(C1)CC(F)(F)C2 C#Cc1ccnc(C(=O)NC2(CC(=O)NC3(CC)CCNC3=O)CCC2)c1 CC1CN(C(c2ccc(F)s2)=O)CC1CC(N1CCSC(C)C1)=O c1(OC)ccc(C(=O)NCc2cnc(Cl)nc2OC)cc1S(N)(=O)=O c1(NCc2c(Br)ccc(OCC)c2)ccc(S(=O)(=O)NCC(C)(C)OC)cc1Br C=C(C)CC(C(=O)NCc1cnc(C)n1CC)NC(C1CCOC1C(C)C)=O CC(CS(C)(=O)=O)C(=O)N1CC2CC1CC2CNC(c1cnc(S)n1C)=O C(C(=O)NCCN(C(=O)C(F)(F)c1cncs1)C1CCCCC1)(C(C)C)SC c1(N(C(c2c(C)nc(-c3cnn4c3CCC4)cc2)=O)CCO)nccc2ccccc12 C1(C(N2CCC(OC)(CNC(c3cnc(Cl)s3)=O)C2)=O)Cc2cccc(F)c2O1 C1(NC(CCCN(C(C)C)C)=O)(CF)CCN(C(=O)CC2CCC(=O)N2)C1 Cc1c(C(=O)NCC(C)CNC(=O)CCc2ncccn2)sc(Cl)c1Cl CC1(C)OCc2c1n[nH]c2C(=O)NC1CCCN(c2nnc(C3CC3)s2)C1 C(C)(CCCCNC(c1c(C)coc1C)=O)NC(CCOCCOC)=O C1(CNC(C23CCCN2CCC3)=O)C2CCC2CN1C(=O)C=CC1CCCCC1 c1(CC)[nH]nc(Cl)c1C(N1CCCC(CNC(C2(SC)CC2)=O)C1)=O C(C(=O)NC(C)CCN(C)C)(C(C)OC)NC(CCCOCCC)=O c1(OC)cc(C(=O)N(C(C)CNC(=O)CCc2cnoc2)C)cc(F)n1 c1(CNC(C2CC(C(=O)OC)C2)=O)nc(C(=O)NCC2CCNC2=O)co1 C(=O)(C1=NN(C2CC2)C(=O)CC1)N1CCN(C(C2C(C(N)=O)C2)=O)CC(O)C1 c1(C(=O)NC2CCC(CNC(c3c(C)[nH]cc3)=O)C2)ccc(-c2cnco2)cc1 C(CC(CNC(C1C=C(C)CS1)=O)NC(=O)CCc1cccnc1)OC Cc1c(CN2CCN(C3CCc4nccn4C3)CC2)sc2cncn12 C(=O)(CCC(=O)N1CCC(O)CC1)N(C)CC1CCCN1C(C1(F)CCC1)=O C#CCC(C)C(=O)NC(C1CCCC1)CNC(=O)Cc1csc(C2CCCC2)n1 C1(CN(C)Cc2ccccc2)CCN(C(=O)COCCSc2ccccc2)C1 N1(C(C2(CC=C)CCOC2)=O)CCC(CNC(c2c(C)coc2C2CC2)=O)CC1 c1(C(=O)NCC2(F)CCC(NC(CSC)=O)C2)ccc2ncc(Br)n2c1 c1(C(=O)NC(C(C)NC(CC=C=C)=O)CO)cn(C)nc1C1CCCC1 C1(NC(C2C(C)CCS2)=O)CCN(C(=O)C=Cc2ccsc2Br)CC1 c1(CCC(=O)NC(C)(CNC(C2(C)CNC(=O)C2)=O)CO)cnc2n1CCOC2 c1(OCCCC)ccc(CC(=O)NC2CC(C(=O)NC(=O)CC(C)CF)C2)cc1 c1(C(N2CCCC(N(C(COCC)=O)CCOC)C2)=O)cc(S(N)(=O)=O)cn1C C=CC(C)(C)C(=O)N1CCC1CNC(=O)C(Cc1ccc(F)cc1)N(C)C Cc1ccc(C(C)(C)C(=O)N2CC(CNC(c3nc(=N)cc[nH]3)=O)C2)cc1Br N1(CCc2ccc(C(=O)OC)cc2OC)CC(C)CS(=O)(=O)CC1 N1(C(c2n(CC)ccc2)=O)CC2CCCC2(NC(=O)CS(=O)(=O)NC(C)(C)C)C1 c1(C(=O)NCC2N(C(CC(C=C)C)=O)CCOC2)cnc2ccc(OC)nn12 C1(C(=O)NC2CCC(C(=O)NCc3cccc(F)n3)C2)CCC(F)(F)C1 Cc1cc(O)c(C(=O)NC(C2CCN(C(c3nc(O)[nH]c(=O)n3)=O)CC2)C)nn1 c1(COC(c2cccc(I)c2O)=O)cc(F)cc(Cl)c1 c1(C(=O)NC2CCC(NC(C34C=CC(CC3)C4)=O)C2)c(F)ccc2ccncc12 c1(CC)cc(C(=O)NCC2(C)CC(NC(C3(C4CCC4)CCC3)=O)C2)cc(O)n1 C(CN=c1nc(N(C)C)cc(C)[nH]1)N(C(c1nc(OCC)oc1)=O)C c1(CNC(C(C2CCN(C(CC3(OC)CCC3)=O)C2)C)=O)ccc(F)cc1F C1(NC(c2onc(C)n2)C)CN(C(c2cnn(C3CCC3)c2C)=O)CC1C c1(C(=O)NCCC(C)(C)NC(C2C(C)(C)C2(F)F)=O)cncc2cnccc12 CC1CCCCC1(CNC(c1ccc(CO)nc1)=O)NC(=O)CCC1CC1(C)C O=C(C1CCc2ccccc21)N1CC2C(C1)N2C(c1cccc(O)c1Cl)=O c1(CC)ccc(C(N2CC(NC(=O)C=Cc3ccco3)C(CO)C2)=O)cc1CC Cc1cc(CC(N2CCC(NC(=O)COCP(C)(C)=O)C(F)C2)=O)cc(C)c1 C(=O)(CC(C(F)(F)F)n1cccn1)NCC1CC(OC)CN1C(=O)CO C1(C(N(C(C(=O)OC)C)C2CC2)=O)CC(O)CN1C(c1oc(C)cc1C)=O C(CC(C)C)(C(=O)NCCC1(O)CN(C(C2CN(C(N)=O)C2)=O)CC1)OC c1(C(=O)NCC(CNC(CNS(C)(=O)=O)=O)F)ccc(C2CC(=O)C2)cc1 N1(C(c2n(CC)ncn2)=O)CC(NC(c2occ(C)c2C)=O)CC12CCCCC2 CC1CCC(F)(F)CN1C(=O)C(C(C)(C)C)NC(=O)C=Cc1cc[nH]c1 C(=O)(C1=COCCO1)NC(C)CCCCNC(c1cc(C(N)=O)cn1C)=O c1(OC)cccc(C(N2CC(CO)(NC(C3CCCN3N=O)=O)C2)=O)c1OC c1(C(N(c2nnc(-c3ccccc3)s2)C(C)C)=O)cc(Cl)c(Cl)s1 C1(C(=O)NCCNC(CN(CCC(C)(C)C)C)=O)CC2(CCC2)CO1 C1(C(N(C)CCN2CCCC2)=O)CCN(C(C2C3CCCCC23)=O)C12CCC2 C1(C)(NC(C(C(C)(C)C)NC(c2ccn(C)n2)=O)=O)CCCCC1(C)C c1(CC(=O)NCCNC(CCCCC#N)=O)ccc2c(c1)CCC2 C1(NC(CCCC)=O)CCN(C(=O)C(c2cc(C)cc(F)c2)C)C(C)C1 c1(CC(N2CCC(F)(CNC(C(CCC)CC)=O)C2)=O)coc2ccc(C)cc12 c1(C(=O)NCc2n(CC)cnc2)cc2ncc(-c3ccc(C)cc3F)cc2[nH]1 N1(C(CNC(=O)NC)=O)CC(NC(=O)CC2(CO)CCC2)CC12CCOC2 CC(C)C(F)(CNC(C1CN(C)C1)=O)C(=O)NC1CCN2CCC1C2 c1(C(=O)NCC2CN(C(c3c(OC)scc3)=O)C(C)CC2)cc(F)c(C)cc1O c1(C(=O)NC2C(NC(Cn3c(C)ncc3)=O)COCC2)cc(O)nc(O)n1 C1(C(=O)NC(c2cnn(C)c2)C)(CO)CCCN(C(=O)CCc2nncs2)C1 c1(C(=O)NC(c2cccc(OC)c2)CNC(=O)C=C2CC2)cc(C)nnc1O c1(OC)ccc(NC(=O)C(N2C(C)CN(C)CC2C)=O)c(NC(=O)C2CC2)c1OC Cc1cc(C)c(C(=O)NCC2(CC(=O)NC(c3ncnn3C)C)CC2)cn1 c1(CC(=O)NCC(CC)(CC)NC(C2(C)CC3(CCC3)C2)=O)cc(F)cc(F)c1 C1(CC(=O)NCC2(CNC(=O)CC3CCCC34CC4)CC2)CCCC2(CCC2)O1 CC1CC2(C(=O)NCC3CCCN3C(c3cocc3C(N)=O)=O)CC12 C1(CNC(c2c(CC)n(C)nc2)=O)CN(C(=O)C(CO)OC)CC1(C)C CC(O)(CNC(=O)Cn1cnnn1)CNC(=O)CC1(CO)CCCC1 CC1CN(C(=O)CC2COCCN2Cc2ccc(Cl)cc2F)CC(C)O1 CCC(CC)(CN=c1[nH]c2c(c(=NC3CCS(=O)(=O)C3)[nH]1)SCC2)c1cccs1 c1(C(N2CC3C(NC(=O)COCC4CCC4)C(C3)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 N1(C(c2cn(CC)nc2)=O)CC(F)CC1CNC(=O)CC1CCCC(C)C1 C1(C(N(C)Cc2cc[nH]c2C2CCC2)=O)CC12CC(NC(=O)OC(C)(C)C)C2 CC1CC2(CCN(C(=O)Nc3cccc(C(=O)Nc4cncc(C#N)c4)c3)C2)CO1 Cc1cc(C(N2CCN(C(c3ncsc3C)=O)CC2CCO)=O)c2occc2c1 C1(CN(C(c2cnc(C)[nH]2)=O)C)CCCCN1C(=O)CSCCN(C)C CP(C)(=O)c1ccnc(C(=O)NC2CC3(C2)CC3NC(=O)CNc2nccs2)c1 C1(C(=O)NC2(C(COC)O)CC2)(CNC(c2cnn(C(C)C)c2)=O)CCCO1 c1(C(N(C)C)=O)ccc(C(N2CC(CCO)(NC(c3cccnc3)=O)C2)=O)cc1 C#CCCCCC(=O)N1CC=C(CNC(C2CCN(C(C)=O)C2)=O)CC1 c1(C(=O)NC(C)CC(C)NC(c2cnccc2Cl)=O)nc2cccnc2s1 C(=O)(C1c2ccccc2CN1Cc1ccc(C)nc1Cl)Nc1c(OC)cccn1 CCCC(C)(CCC)C(=O)NC1CC2CC(NC(c3cnns3)=O)C1C2 N1(C(Cc2cccc(C)n2)=O)CC2CCC(NC(=O)C(c3ccccc3)C)C2C1 c1(C(=O)NCC2C(C)CCN(C(c3cnccc3Cl)=O)C2)ccc2scnc2c1 c1(C(=O)NC2C(NC(CCC#C)=O)CCCC2)cnn2ccc(Cl)c(F)c12 c1(C(N2CC(NC(c3c(OC)n[nH]c3)=O)C2)=O)c(C)nc(O)nc1C C(=O)(C(F)CC(C)(C)NC(c1ccccn1)=O)Nc1ccc(COC)cc1 C1(CNC(c2c(Cl)cc(C)s2)=O)CC2CCC(C1)N2C(=O)CC1C(C)(C)C1(C)C c1(SCNC(C(c2ccc(I)s2)N(C(C2CSC2)C)C)=O)ccccc1 C1(C(=O)NCC(C)OCC#C)CN(C(c2cc(CC)n(C)n2)=O)CC1(C)C C1(NC(CCC2C(C)=NOC2=O)=O)CN(C(c2cn(C(F)F)cn2)=O)CC12CC2 c1(CC)nc(Cl)cc(=NCCCCN(C(=O)CS(=O)(=O)N(C)C)C)[nH]1 CCCC(C(=O)N1CC(C)(C(N2CCC(O)CC(C)C2)=O)C1)C(C)C C(=O)(C1=CCCC1)NCC1(C(N2CC(CCO)(CC)C2)=O)CCCO1 c1(CN(C)CC2CC(OC(C)(C)C)C2)ccc(-c2ccco2)cc1F N1(C(=O)NCc2c(C)cncc2)CCC(C2=NOCC2)C1 C#CCCCCC(=O)NC1CC2CC1N(C(c1ncc(F)cc1C)=O)C2 c1(OCC)oc(C)nc1C(N1CCCC1CNC(C1C=CCCC1)=O)=O C1(NC(C2C(=C)C2)=O)CCC(NC(c2oc(CCC)nc2C)=O)CC1 CC1(CNC(c2ccc3c(c2)CCO3)=O)COCCN(C(C2CC3(CC3)C2)=O)C1 C1(NC(c2cnc(SC)s2)=O)CCN(C(c2cn(CCF)nn2)=O)C1(C)C c1(-c2ccc(N)cc2)cccc(F)c1O.CC1(C(=O)Nc2cscn2)CCCN1C c1(C(N2CCC(NC(=O)COc3ccc(Cl)cc3Cl)C2)=O)ccnc2cc[nH]c12 Cc1oc(CNC(=O)C=CC2CCCN2C)nc1C(=O)NCCc1ccco1 C(=O)(C1CCc2cccnc21)N(CC(C)CNC(c1cccc(=O)n1C)=O)C c1(C2C(CNC(C=CC(CC)C)=O)C2)cccc(NC(C2CC(C#N)C2)=O)c1 C1(c2nnnn2C)(NC(C2(C)CC3(CCC3)C2)c2scc(C)n2)CCC(=O)NC1 CC12CCN(C(c3coc(CC4CC4)n3)=O)C1CN(C(c1cnc(S)nc1)=O)C2 N1(C(CC2CCC(C)(C)CC2)=O)CC2(CCCN(C(=O)CN3CCSCC3)C2)C1 c1(C(N2CC(CNC(c3cc(Cl)c[nH]3)=O)CC(C)C2)=O)cc([N+](=O)[O-])ccn1 CC(F)(F)CCCC(=O)NC1(CF)CCN(C(C2CCCOC2)=O)C1 C=CCC(C(=O)NCC1CC2CC2N1C(C1CN(C(C)C)C1)=O)c1ccccc1 CC1CN(C(c2c(Br)cnn2C)=O)CCC1CNC(=O)CCn1cccn1 CCC(CC(=O)NCC(C1CC1)N(C(=O)C(C)SC(F)(F)F)C)C1CCC1 n1(CC)cc(C(=O)C(=O)NC2(CN(C(=O)C(C)N(C)C)C)CC2)cn1 c1(C(N2CCN(C(CC(CC)C)=O)C(CF)C2)=O)cc(C)cc([N+](=O)[O-])c1N CC1CC(CO)N(N(C)Cc2cccc(C(C)(C)C)n2)CCO1 C(C(C(C)C(C)C)NC(=O)CCCCCF)NC(c1ccc(N(CC)CC)nc1)=O Cc1ccc(Br)c(C(=O)NC2CC(CN=c3nn[nH]n3C)(c3ccccc3)C2)c1 c1(CNC(c2n(C(CC)(C)C)nnn2)c2ncc(SC)s2)ccncc1C C1(C(N(CC(C)(C)NC(c2ccc(C)s2)=O)C)=O)CC2(CC2)CO1 Cc1ccncc1CC(=O)NCCC1CCCN(C(c2cnc(C(C)O)s2)=O)C1 C1(O)(C(=O)NCCCNC(=O)COC2CC2)CCc2cc(Br)ccc2C1 C(CCCCCN(C(=O)C(C)(C)CO)C)NC(C1C(C)C1)=O N1(C(C(C)OCC#C)=O)CC(NC(c2ccc(Cl)cc2CC)=O)C(N=[N+]=[N-])C1 CC(C)(C#N)CCC(=O)N1CC(F)(F)CC1CCNC(=O)C=Cc1ncc[nH]1 c1(COC)ccc(CNC(C2CC2NC(=O)C(C)OC2CCCC2)=O)cc1 c1(N2CCC(O)C(F)C2)ncnc2cc(C(F)(F)F)ccc12 c1(OC)ncc(F)c(=NC(=O)C2CC2NCc2cc([N+](=O)[O-])ccc2N(C)C)[nH]1 c1(C(=O)NC2CN(C(CC3CCC(C)CC3)=O)CC2O)cnc2[nH]ccc2n1 C1(NC(c2cc(CC)nn2-c2ccccc2)=O)CN(C(=O)C(N)=O)C2(CCC2)C1 C=Cn1nncc1C(=O)NCC(CC(=O)NCCC1C=CCC1)C1CCC1 C=CCC(CC=C)C(=O)NCC1CCCN1C(=O)C(C)Cc1ccnn1C c1(N2CCCC(COC)C2)nc2c(c(=NC(C)Cn3cncn3)[nH]1)COC2 c1(CCNC(C(C2CCCO2)NC(c2ccco2)=O)=O)ccccc1F c1(NC(C2CCCC(NC(c3cncc(C)c3)=O)C2)=O)cccc2ccoc12 c1(C(N2CC(O)(CN(C)C(C3CCC3)=O)C2)=O)c(C2CC2)cnn1C C(=O)(C1CCCc2nccn21)N1CCN(C(c2ccn(C)c(=O)c2)=O)CC1CF C(=O)(C(COC)NC(=O)CCn1ccc(C)n1)NCC(C#C)OC C1(C2CCCO2)(C(N2CC(C)(NC(c3cn[nH]c3)=O)C2)=O)CCCO1 N1(C(c2cc(C)no2)=O)CCCCC(N(C)C(C2CC2c2cccs2)=O)C1 c1(CC)cccc(C(=O)NC(c2ccccc2)CNC(=O)CC2CC2(C)C)n1 c1(C(=O)NCCC2CCN(C(c3cc(C(F)F)[nH]n3)=O)C2)cc(Cl)cnc1O N1(C(C2(CC#C)CCN(C(C3CCC(CC)O3)=O)C2)=O)CC2CCCC(O)C2C1 C1(C(N(CCCCCCNC(C2(CO)CCCCC2)=O)C)=O)CCCCN1N=O C1(C(N2C(CNC(C3(C=C)CCCCC3)=O)CC(O)C2)=O)CCc2n[nH]cc2C1 c1(OC)ccc(S(=O)(=O)N(C(C(=O)O)C(C)C)C)cc1-c1cc(Cl)c(O)cc1C N1(C(C2CCC(NC(C(C(=O)OCC)OC)=O)C2)=O)CCn2cnnc2C1C C=C(C)C(C)(C)C(=O)NCC1CCC(NC(=O)Cc2cccc(OCC)c2)CC1 Cn1ncc([N+](=O)[O-])c1N1CCN(C(c2cnn(CC3CC3)c2)=O)CC1.C1CN1 C1(NC(C2(CCOCC)CCCC2)=O)CCCCC1CNC(=O)CCF c1(C(=O)NC2(CCNC(CC3(OC)CCCC3)=O)CCCC2)csc(C)c1N CC(C)C(C#N)C(=O)NC1CCC(CCNC(=O)COC2CCCCC2)C1 CC(C)C(O)CC(=O)NC1CN(C(=O)CCCC2CCCCC2)CCC1CO C1(C(N(CC(CCC=C)O)C)=O)C(C2CC2)CCN1C(C1CCN(CC)C1)=O C1(NC(COC(CSC)(C)C(=O)Nc2ccc(Cl)c(O)c2)=O)CC2(C1)CC(O)C2 CCCC(CCC)CC(=O)NCCCC(CO)NC(=O)C(C(C)C)SCC CC1CCN1C(=O)NCCCNC(=O)CNS(N)(=O)=O C(=O)(C1=C(C)OCC1)NC1CCCC(NC(C2CCC(CC)O2)=O)C1 CCCCCC(C)CC(=O)NC1CC(NC(c2cc(Cl)nnc2O)=O)C1 C1(CNC(c2cnc(O)s2)=O)(NC(C2CC(CCO)C2)=O)CCOCC1 C1(F)(C(N2CCC(NC(c3c(C)oc(C(F)(F)F)n3)=O)C2)=O)CCC(F)(F)CC1 CCCCC(CC)C(=O)N1CCC(C)(C(N2CCOC(C)(C)C2)=O)CC1 c1(C(=O)NC2(CF)CCN(C(c3c(C)ncn3C)=O)C2)cc2cccn2c(O)n1 CC1CCCc2ncc(C(N3CCN(C(=O)C(F)=C4CCC4)C(C)C3)=O)n21 CCCC(C)(C)C(=O)NCC(F)CNC(=O)Cn1nnc(C(C)(C)C)n1 c1(NC)cnncc1C(N1CCOC(C(C)NC(=O)CN2CCOCC2)C1)=O c1(C(=O)NCCOCCCNC(C(CCC)CC)=O)cc(=O)n2ccsc2n1 O=C1CCCC(C(=O)NC2CCOC(C(N3CCC4(CC4)C3)=O)C2)C1 C1(C(=O)NCC(C)Cn2cccn2)CC2(CC2)CN1C(=O)CN1CC2CC2C1 CCC#CCCNC(C1(NC(=O)CNc2ncccn2)CC(CO)C1)=O n1(C2CCN(Cc3cc(C)cc(C(F)(F)F)c3)C2)c(C)nc2ccccc12 c1(C(=O)NCC2CC(NC(CC(C=C)CC)=O)C2)cccc2c1ccn2C(C)C c1(CNC(N(CCCF)C)=O)ccc(Br)c(Br)n1 c1(OCCOC)ccc(CNC(=O)NC2CC(CCC(N)=O)C2)cn1 C#Cc1cccc(NC(=O)CCC)c1.C1(CC=C)(C2CC2)CN(C(=O)C(F)C2CCOC2)C1 C1(CC)CN(C(=O)C(C)(C#N)CC)CCN1C(=O)COc1ccc(C)cc1C CC1CCSCCN1C(=O)CCN(C)C(C1CCC(F)CC1)=O N1(CC2C(c3cn(C)nn3)OCC2)C2CCCC1CC(=O)NC2 c1(C(N2CCC(OC3CC3)C2)C(=O)NCC(F)F)cccc(-c2ccccc2)c1 C1(C)(CNC(C2(CC(C)C)CCCC2)=O)CCN(C(=O)C2=CCOC2)C1 c1(C(=O)NCC2C(NC(COCC(C)C)=O)COC2)cc2c(F)c(F)ccc2[nH]1 C1(C)(CC(N2CC(CC(C)NC(c3cc(CO)[nH]n3)=O)C2)=O)CC1(F)Cl S(=O)(=O)(c1cnc(Cl)nc1)N1CC2C(C(=O)NCc3cccc(Cl)c3F)(C2)C1 CN1C(=O)c2ccccc2C1CC(=O)NC1CCC(NC(C2CCOC2)=O)CC1 c1(Cc2cnc(NC(C3CC(C)OCC3)=O)s2)ccc2nc[nH]c2c1 c1(CNC(C2CC(C(C)=O)C2(C)C)=O)ccc(-c2cncnc2)c(C)c1 N1(C(Cc2c(C)occ2)=O)CCN(C(c2cc[n+]([O-])cc2)=O)C2CCCCC12 C(=O)(C1=NOC(C)C1)NCC1CCCN(C(c2c(C)cccn2)=O)C1 N1(C(c2cc(SC)oc2)=O)CCC(NC(=O)COC(c2ccccc2)C2CC2)CC1 N1(C(C=CCN(CC)CC)=O)CC(NC(C2(c3cccnc3)CCC2)=O)C(C)C1 c1(C(N(C(C)C(=O)NC2(CF)CC2)CCC)=O)cc(C)c(O)nn1 c1(CC)nc(C)[nH]c1C(=O)NCC1CC1NC(C1CCC(C(=O)OC)CC1)=O C12(CNC(C3CCN(CCO)C(=O)C3)=O)CCCC1CN(C(c1cnsn1)=O)C2 N1(C(CC=C=C)=O)CCC(C)(CC(=O)NC(C)Cc2nncn2C)C1 C1(=CCCN(CC)Cc2cccc(CCCC)c2)COCCN(CCc2c(C(C=O)OC)c(F)ccc2)C1 Cc1ccccc1C(F)(F)C(N1CCC(CNC(C2CC23CC3(F)F)=O)CC1)=O N1(C(c2c(OC)n[nH]c2)=O)CC(CNC(=O)Cc2cncnc2)C(F)(F)C1 N1(C(CCC)=O)CCCOC(CNC(=O)CSc2nccn2C)C1 N1(C(CCNC(C)=O)=O)CCC(C)(CNC(C2CC2c2ccc(F)cc2)=O)CC1 C1(C(=O)NCC2N(C(C3CCC(CN(C)C)O3)=O)CC2)CCC(C)C(C)C1 C=C(C)CN=C(NCC(c1c(C)noc1C)C)N1CCOCC2(C1)CC2(F)F c1(CNC(CCOC(C)=O)=O)cc(C(=O)NCCCc2nncn2C)no1 C(=O)(C1Cc2ccccc21)NC1(CC(=O)NCc2ccnc(Cl)c2)CCC1 C1(C(=O)NCCCCCCN(C(c2cc(COC)on2)=O)C)CCS(=O)(=O)CC1 c1(CC(N2CC(CNC(Cc3cc(C)no3)=O)OCC2)=O)ccc2occc2c1 C(CCNC(C1(CC(C)=O)CC1)=O)(C(=O)N1CCCC1CCC(C)C)OC C(=O)(C1COc2ccccc21)NC1CCN(C(Cc2c(OC)ccc(Cl)c2)=O)C1 C1(CNC(C=C(C)CNC(=O)COCC2CC2)=O)CC2(CCC2O)C1 C(C)(C(O)C(=O)N1CC(O)(CCNC(c2ccnc(C3CC3)c2)=O)C1)SC N1(C2CCN(C(C=CC=CC)=O)CC2)CCN(C(c2scc(C)c2C)=O)CC1=O c1(C(N2CCC(CNC(C3CCCC(C)C3)=O)C2)=O)cn2cccnc2n1 c1(NC(C2CCCCN2Cc2ncsc2Br)=O)nccc(-c2ccccc2F)n1 N1(C(C2(C(=O)OCC)CC2)=O)CCCC(CCCCNC(c2cc(=O)cc[nH]2)=O)C1 Cc1ccccc1C=CC(=O)NCC1CCCC1NC(C1(C)CCCS1(=O)=O)=O N1(C(CSC)=O)CC(C(=O)NOCC(F)(F)F)C(C)C1 c1(C(N2CC3C(CNC(CC4ON=C(CC)C4)=O)(C3)C2)=O)c(C)cc(C)c(C)c1 C1(C(=O)NC(c2nc(-c3cccc(C(F)(F)F)c3)no2)C)CCCOC1(C)C C1(NC(CCCCC(C)C)=O)CCC2(CCCN(C(=O)Cc3ccsc3)C2)C1 C1(NC(C(CSC)C)=O)CC2(CCCCN2C(C2(O)CCCC(C)CC2)=O)C1 CC1OCCCC1C(=O)NC1CC(N(C(=O)CCc2nncs2)C)C1 C1(CC)C(NC(=O)Cc2nnc(C)o2)CCN1C(=O)C=CCOC1CCOCC1 C1(C)(CNC(C(COC)O)=O)CCCN1C(c1nc(OC)c(C)s1)=O CCC(C)(CNC(=O)CCC1CCOCC1)NC(=O)COC1CCC1 N1(C(Cn2cnc(C#N)n2)=O)CCOCCC1C(=O)NCC1CCC(F)(F)C1 c1(C(N2CC(NC(c3c(Cl)nc4ccccn34)=O)C2)=O)cc2cccnc2cn1 N1(C(CSCC)=O)CC(NC(=O)Cc2cnccn2)CC(F)C1 C1(OCCNC(C2C(C(N(CC(C)C)CC(C)C)=O)C2)=O)CCOCC1 C1(C(N2CCC(C(=O)NCCOCC(=O)OC)(C(C)C)C2)=O)CC2(C1)CC2(F)F c1(C(=O)NCC2CC(COC)CN2C(=O)C2=NNC(=O)C2)cc(C)nc(C)c1 C(c1cccc(CO)c1)=CC(=O)NCC1N(C(C2C(C=C)C2)=O)CC1 N1(C(CCC2CC(OC)C2)=O)CCN(C(=O)CCn2cnnn2)CC1c1ncc[nH]1 c1(C(=O)NC23CC(CNC(=O)C=C4CCC4)(OCC2)C3)ccc2nnn(O)c2c1 C#CC1CC2(CC(C(=O)NCC3CCCN3C(=O)C(O)Cc3ccccc3)C2)C1 N1(C(=O)COc2cc(-c3ccccc3)ncn2)CCC(CF)(OCC(F)F)C1 N1(C(c2cnc(O)[nH]2)=O)CCC(O)(C(=O)Nc2cnnc(Cl)c2)C1 Nc1ccc2c(c1)CCC(C(=O)NC(c1c(F)cccc1F)CC1CCCC1)C2 C1(C(N2CCN(CCOC)CC2)=O)CCCN1NC(=O)C1CCOC1C(C)C c1(CC(=O)NC2(C)CN(C(=O)COC3(C)CCC3)C2)c[nH]ccc1=O Cn1ncc(C#N)c1C(N1CCC(C)(CC(=O)NC(C(N)=O)C2CC2)C1)=O c1(C(=O)NC2CC(C(=O)NC(C#C)C)C2)c(F)ccc(F)c1OC C(C(C)(C)C(=O)N1CCC(CNC(c2cncc(Br)c2)=O)C1)OCC C1(NC(C(C2CCS(=O)(=O)CC2)(C)C)=O)CCCCN(C(=O)CCC2CCCO2)C1 c1(N(CCNC(C2CC(=C3CC3)C2)=O)CC)ncccc1S(C)(=O)=O c1(OC(C(=O)NC2C3CN(C(COCCOCC)=O)CC32)C)cc(Cl)cc(Cl)c1 N1(C(CC2CC(=O)NC2=O)=O)CCOC2(CCC(NC(C3CC3(Cl)Cl)=O)CC2)C1 CCCCC(C)CCC(=O)N1CCC=CC1C(N1CCCC1CC1CC1)=O C1(N(c2cc(C)nn2-c2ccncc2)C(C2(Br)CC2)=O)CCNCC12CC2 C(C)(C(=O)N(C)CC1(CNC(=O)CSC)CCC1)SCC C(=O)(CC(O)CC(C)(C)C)NC1CN(C(C)C)C(CO)C1 c1(N(C)C)cc(C(c2cccc(F)c2)NCC2(c3cccc(Cl)c3)CC2)ncn1 Cn1nc(C(N2CC3CC3(NC(=O)Cn3nccn3)C2)=O)cc1C(N)=O CC(C)S(=O)(=O)CC(=O)NCC12CC(CN1C(=O)CCC=Cc1ccccc1)C2 N1(C(C23CN(C(C4C=C(C)CS4)=O)CC2(CO)C3)=O)CC2CCOC(=O)C2C1 c1(OC)cccc(Cl)c1CC(=O)N(CC(C)NC(=O)CC1CCCO1)CC CC1CCN(C(=O)C(c2ccc(I)cc2)F)C(CN)C1 C1(NC(C(CCC)CC)=O)CC12CCC(NC(c1cc(C(F)F)nn1C)=O)CC2 CC(C)C(O)C(C)(C)C(=O)NCC1CCCC(CNC(=O)CC(F)(F)Cl)C1 C1(NC(C2=C(C)OCC2)=O)CCC2CC1CN2C(c1ccnc(CN(C)C)c1)=O C12CCN(CC1O)C2.Cc1cncc(C(=O)NCC2(Cc3ccccc3)CC2)n1 c1(N(C(C)(C)CNC(c2nc3cccnc3s2)=O)CCO)cccc(P(C)(C)=O)c1 C=C1CC(C(=O)N(c2ccsc2)C)(CNC(=O)C(O)CN2CCCC2)C1 C(=O)(C(C)(C)n1ccc(NC(=O)OC(C)(C)C)n1)N(CCCN(C)C)C1CC1 N1(C(c2cc(C)ncc2C)=O)CCCC12CCC(NC(c1c[nH]nc1F)=O)CC2 c1(CNC(=NCC)NCC2CC(C)OC(C)C2)c(C)cccc1[N+](=O)[O-] c1(-c2cn(CCNC(C3C4CCCCC34)=O)nn2)cncc(F)c1 Cc1nc2c([nH]1)CN(C(C1CN(C(=O)C3=CCCOCC3)CC1(C)C)=O)CC2 CCC(O)C(C)C(=O)N(C(CNC(c1ccc(OC)nc1OC)=O)C1CC1)C c1(CCC)ccc(C(C)NCc2nc(C(=O)OC)n[nH]2)s1 C1(CC=C)(C(=O)NCCN2CCOCC2)CCCN1C(=O)CCN1CCOCC1 C1(CNC(=O)NCC2C(C)C2(F)F)CCC2COCCC2O1 N1(C(c2nc(COC)[nH]n2)=O)CC(CNC(=O)C(F)CC2CCCC2)CC1C N1(C(c2ncc(C)nc2)=O)CCC2CCCC(C1)N2C(c1cnc(N(C)C)s1)=O N1(C(c2c(C)sc(Br)n2)=O)CCN(C(=O)C(=Cc2c[nH]cn2)F)CC1C CN1CCN(C(C2CN3CCC2CC3)=O)C(CNC(c2cnc(N)cn2)=O)C1 c1(-c2nc(-c3cn(OCCOC)nc3)n(CCF)n2)ccc2nc[nH]c2c1 C12(CC(=O)N(CCC)CCNC(=O)C(c3ccnn3C)O)CCC(CC1)C2 C1(C(=O)NC(C(=O)NCC=CCCOC)(C)C2CCC2)CC(O)CN1C N1(C(C2C3CCN(C(C(C)(C)O)=O)CC32)=O)CC2(C)COCC2(C)C1 CC(CS(C)(=O)=O)C(=O)N1CCOCC(CNC(c2cnns2)=O)C1 N1(C(CCCC(C)=O)=O)CC2(CNC(c3[nH]cnc3C)=O)CCC1CC2 C1(C(=O)NC(CC)CNC(c2cscc2C(=O)OC)=O)CCOC(C)(C)C1 C(=O)(C(C)C(C)S(C)(=O)=O)NC(C1CN(C(=O)CCN2CCCCC2)C1)C c1(CCCC(=O)OCC)cc(=NC(C)c2ccn(-c3ccccc3)n2)[nH]c(C)n1 C(=O)(C1Cc2ccccc21)NCC1OCCCN(C(CCC=C)=O)C1 CC1OCCC1(C)C(=O)NCC1CCC(C(=O)NCC2(O)CCOC2)CC1 c1(C(=O)NCC(CN(C(c2cc(C)sn2)=O)C)C)ccc(C)c(F)c1F C(C)(N=c1[nH]c2c(c(=NCC(C)C(F)F)[nH]1)COCC2)c1ncc(C)cn1 Cc1cc(Cl)cc2[nH]c(C(N3CCC(N(C(=O)CC4CCOC4)C)C3)=O)cc12 C1(O)(COCC)CCCN(C(=O)NC2CC2)CC1.c12ccnc(c1)N2.C(C)(C)(C)O c1(C(=O)NCC(CCNC(=O)CC2CCCCC2)O)cccc2c[nH]nc12 CC(C)(CC(=O)NCCCCCNC(c1csc(C(F)(F)C(F)(F)F)c1)=O)C(F)F N1(C(C(CC)OC)=O)CC(F)CC1CNC(=O)Cc1cc(C)[nH]n1 c1(CC(N2CCC(F)(C(N(CCC#N)C3CC3)=O)C2)=O)cc(F)ccc1Br C1(C#N)(OC)CC(C(=O)NC(Cn2cncn2)C(=O)NC2(CO)CC(O)C2)C1 c1(C(=O)NCC(C2CC2)NC(c2cc(C)c(Cl)s2)=O)cc2ccncc2cc1F c1(C(=O)NCC2(CN(C(C(CCC)O)=O)C)CC2)ccc2cccnc2c1 c1(C(=O)NC2CN(C(CC=C=C)=O)C(C)CC2)ccc2ccccc2c1 C(=O)(CCCCCCCS(C)(=O)=O)NCCOC(CNC(CCC=C=C)=O)(C)C C1(C(C(C)C)NC(=O)C(C)(C)C)CCCN(C(C2(Cl)CC2)=O)C1 Cc1cc(CCCC(=O)N2CC(CC(C)NC(=O)C(C)N(C)C)C2)on1 S(=O)(=O)(c1ccc(C(=O)OCCOC)cc1)NCC(CNCC#C)O CCC(O)CC(=O)NCC(C)(C1CC1)NC(=O)CC1CN(C(C)=O)C1 N1(C(C2C3(CN(C(c4cc[nH]c4)=O)C3)C2)=O)CC=C(c2ccccc2)CC1 c1(CCC(=O)NCC2(NC(C3CC3(F)Cl)=O)CCCCC2)ccc(F)cc1 C1(CNC(C(COC)(F)F)=O)CCC2(CCCC2)C1 Cc1ccc(CNC(=O)CN(C(=O)CCc2cc(C)[nH]n2)CC(C)C)cn1 CS(=O)(=O)C(C(=O)NC1CN(C(=O)CCc2ncc(F)cn2)CC12CC2)C1CC1 CN1CC(C(=O)NNC(c2ccc(C#N)cc2)=O)OCCC1=O CC1CC(C(=O)NC2CCCC2NC(=O)Cc2ccc(O)cc2C(F)(F)F)=NO1 c1(C(N2C(C(=O)NCC3CCS(=O)(=O)C3)CC(=C)C2)=O)cc(F)c(Cl)c(F)c1 CC1C(C)N(C(c2cc(C3CC3)cs2)=O)CCN1C(=O)Cc1sc(S)nc1C N1(c2n(CC(=C)C)c(Cc3ccccn3)nn2)CCCCC(C)(F)C1 N1(C(c2c(CNC(C=CC(=O)N(C)C)=O)occ2)=O)CC2OCCOC2C1 c1(C(=O)OC)ccc(CC(=O)NC2C(CNC(=O)CC3CC3)C2(C)C)cc1 C(C(C)(C1CC1C(=O)O)NC(=O)NCC1(C(F)(F)F)CCC1)OC C1(CC)(NC(=O)C(C)C2CCCC2)CCN(C(=O)C(F)C(F)(F)F)CC1 c1(OC)ccc(Br)c(C(N2CCCC(C)(CO)C2)C(=O)NC2CC2)c1 N1(CC)CCN(CCN(C(=O)CSCC(=O)NC(=O)Cc2ccccc2)C)CC1 N1(C(C)C)CCC(C(=O)NCCC2CCCN(C(c3c[nH]c(Br)c3)=O)C2)CC1 c1(C(=O)NCC(C)CNC(c2ccc[nH]2)=O)cc2cc(Br)cc(F)c2o1 N1(C(CSCC)=O)CC(NC(c2cc(-c3ccc(C)cc3)n[nH]2)=O)C(SC)C1 c1(-c2cnc(OCC)nc2)ncc(C(=O)OC)cc1NC(C)=O C1(C(=O)NCC2(F)CN(C(C(F)=C(C)C)=O)C2)CCCC2(CCCCC2)C1 c1(C(=O)NC(CNC(c2[nH]cc(C)c2)=O)C(C)C)ccc2c(c1O)OC(C)(C)C2 C1(NC(N2CCC(O)(c3n(Cc4n(C)nnc4)cnn3)C2)=O)CCCCC1(C)C c1(C2N(C(C3=CCCCO3)O)CCC2)nc2cc(F)c(F)cc2[nH]1 Cc1nn(-c2ccc(Cl)cc2)c(C)c1C(=O)NC1CC2C=CC1C2 c1(-n2c(C)ncc2)cc(C(=O)NCC2C3CN(C(=O)C4=CCC4)CC23)ccn1 C=CCC(CNC(=O)COC)C(=O)NC12CCC(CC1)C2 C(=O)(C(C)CC(C)(F)F)NCCN(C(c1nc(C)c(C)s1)=O)CC1CC1 Brc1scnc1OC1CCN(CC2CC2)C1 C=CCC(CC(F)F)C(=O)N(C(C)CCNC(C1CCC2(CCC2)C1)=O)C N1(C(c2cncc(OCC)c2)=O)CCCC(O)(CNC(C2CC2C2CC2)=O)CC1 CC1CCCC(C(=O)NC(C)CNC(=O)CCn2cnnn2)O1 C1(O)(C(C)NC(C=C(C)c2ccsc2)=O)CCN(C(=O)CC2(C)CC2(F)F)CC1 C1(NC(CS(CC)(=O)=O)=O)CCN(C(c2ncc(F)cc2C)=O)CC12CCC2 C(=O)(CCCC(C)(C)C#N)NC(CC(=O)Nc1c(C)noc1C)C(F)F N1(C(c2c(CC)cncc2)=O)CCCC12CCN(C(C1OCC1(C)C)=O)C2 C1(C(=O)NCC2(F)CN(C)C2)CCN(C(C2(F)CC=CCC2)=O)CC1(C)C C12(C(N(CC(C)C(=O)NCCC(=O)NC3CC3)C)=O)CCCN(CC1)C2 N1(C(c2ccc(C(C)(C)C)o2)=O)C2CCC1CC(CNC(c1ccon1)=O)C2 C#Cc1ccc(C(=O)NCCCC(CCC)NC(=O)C(C)CC(OC)OC)nc1 N1(c2scc(C)n2)CCC(C(=O)N(CC(C)(C)NC(C2C3CCCC23)=O)C)CC1 c1(C(=O)NCC2CCN(C(C(C(CC)C)C)=O)C2)c[nH]c2ncccc12 C1(NC(C(=O)N(C)CC#N)=O)CCC2CC2CC1 C1(NC(c2cnc(O)[nH]2)=O)CC2CC1CN2C(C1CC=CCC1)=O C(CN=c1nc(N2CCN(C)C(CO)C2)c2c([nH]1)CCCC2)OC N1(C(c2cc(C(C)C)no2)=O)CCC(NC(c2cnn(C3CCC3)c2)=O)C12CC2 c1(C(N2CC(CNC(c3cnccn3)=O)OCC2)=O)n[nH]c2ccccc12 C=CCCCN=C(NCc1ccnn1C1CCCC1)NC1CCOC(C)C1 Cc1c[nH]c2ncc(C(N3CC(CNC(=O)CNC(N)=O)CC(C)(C)C3)=O)cc12 Cc1cccc(C(N2CCN(C(=O)CC34CCCC3C4)CC2)=O)c1Cl C(CC1CCC1)(C(=O)N1CC(c2cn(C(C)CO)nn2)(C(=O)OC)C1)OC.N(C)C C1(C(=O)Nc2ccc(COC)cn2)CC(C)c2nc(C)cn2C1 CC1C(C)N(C(c2ccnn2CC#N)=O)CCN1C(=O)CCc1cccnc1Cl C1(C)(NC(CC(C)(C)SC)=O)CCCN(C(=O)CCc2cc(C)n(C)n2)C1 O(P(C)(=O)CCCC)C(N1CCCC1C(C)C(=O)OC)=O C12(CNC(c3cn(CC=C)nc3)=O)CC1CN(C(=O)CC(CC)C1CCC1)C2 C(=O)(C1=CCCCC1C)N1CC(OC)C(NC(=O)C(=O)N=S(C)(C)=O)C1 c1(C(N2CC(C(F)(F)F)C(C)C2)C(=O)NCC=C)cnc2c(c1)COC2 N1(Cc2cccc(OC)n2)CC2CN(C(C3CCN(C)C3)=O)CC12 c1(NC(C2N(Cc3ccc(C#C)cc3)CC(F)C2)=O)cc(C#N)ccc1Br CCCCCCC(C)CC(=O)N1CC(NC(C23CC(C#N)(C2)C3)=O)C1 CCC(C(=O)NCC=CCNC(=O)C(C)Cc1cnc[nH]1)c1ccccc1 Cc1nc[nH]c1CNC(C1CCOC1CNC(c1ccsc1)=O)=O CCC(F)(F)CC(=O)NC1CC(C)(NC(c2ccc(Cn3ccnn3)cc2)=O)C1 c1(C(=O)NCC(CC)(C)NC(C2CCOC2)=O)cc2cc(Cl)ccn2n1 C1(O)(CCNC(C2(NC(C(=O)NCC3CC3)=O)CSC2)=O)CCCOC1 C(=O)(C1=CS(=O)(=O)CCC1)NC(C)(CNC(c1ccc(SC(F)(F)F)o1)=O)C1CC1 N1(C(c2ccc3ncnn3c2)=O)CCC2(CCCN2C(C2CC2Br)=O)CC1 Cc1cc(C)c(C(N2CC(CNC(C3CCCN3N=O)=O)CC(C)C2)=O)c(O)n1 C1(NC(C(C)S(N)(=O)=O)=O)CCCC12CN(C(c1cnc(O)s1)=O)C2 N1(C(c2cc(CC)[nH]n2)=O)CC2CCOCC2(NC(=O)C2=CCCCC2)C1 c1(CCOC)ncc(C(C(=O)NC(C)C(C)OC)N(C)CCC(=O)OC)s1 C(=O)(C(C)(CC)CCC)NC(CCCC)CNC(=O)CC1CCCC(C)(C)O1 C(=O)(C=C(Cl)Cl)N(CC(CNC(C1C(=C)CC1)=O)O)C n1(-c2c(C)cccc2)[nH]nnc1=NC(=O)NCc1cc(C(C)C)on1 Cc1ncc(Cl)c(C(=O)NC2C3CN(C(=O)C(O)CC(=O)OC(C)(C)C)CC23)n1 c1(CC)cccc(C(=O)NC2COCCC2NC(=O)C=C2CCOCC2)c1F c1(C(=O)NC2CC(C)(NC(COC(CC)C)=O)C2)cc2ccccc2cc1C N1(C(C=C(CC)CC)=O)CCC(O)(C2(NC(=O)CCCSC)CC2)CC1 CN1CC(N=c2nc3sccc3c(NC3C4CCOC4C3(C)C)[nH]2)CC1=O Cc1ccncc1CC(=O)NC1CN(C(c2cccnc2)=O)CC1C N1(C(COc2ccc(C(C)C)nc2)=O)CCC(C)C2CNC(=O)C12 c1(C(=O)NC)cccc(C(=O)NCC2CC(NC(=O)Cc3csnn3)C2(C)C)c1 C(=O)(C(C)(CO)NC(=O)Cc1cccnc1O)N(C1CC2CC2C1)C C(=O)(CCCCC(C)(C)C)N1CCOCC(CNC(C2ON=C(C)C2)=O)C1 C#CCCCC(C)C(=O)NC1CC(CC(=O)NCc2nocc2CC)C1(C)C N1(C(C(C)=C(CC)C)=O)CC2(CCC2)CC1CNC(c1nccc(OC)c1F)=O c1(NC(C)=O)ccc(C=CC(N2CCC(C)C(NC(=O)CP(C)(C)=O)C2)=O)cc1 C(CC(C)(O)C(=O)NCc1cc(C(=O)NCCC(C)(O)C2CC2)no1)N(C)C c1(C(CNC(=O)C(F)(F)CO)NC(C(C)SCCCC)=O)ccc(F)cc1F C1(N(C(CCCC)=O)C)CN(C(c2cc(C)n(-c3ccc(Cl)cc3)n2)=O)CC1O CCC(CC)CC(=O)N(CCCNC(=O)C(C)(C)Nc1ccccn1)CCO N1(C(c2nc(C)sc2)=O)CCN(C2CCC(NC(=O)CC3(C)CCC3)CC2)CC1 N1(C(c2c(CC)ncs2)=O)CCC(C)(C(N2CCC(C)C2C(=O)OC)=O)C1 N1(C(c2cc(CNC(C3C(C)CCOC3)=O)ncc2)=O)CCCC2(C1)N=N2 CC1=NN(c2ccc(Br)cc2)C(=O)C1CC(=O)NCC(CO)C(C)C CCC(CC(=O)NCC1CCC2(CN(C(=O)Cc3cc(C4CC4)no3)C2)O1)C(C)C C1(NC(CN(C)C2CC2)=O)CCOCC1NC(=O)Cn1ncccc1=O c1(C(N(C2CN(C(=O)CC3(C)CC3(F)Cl)C2)C)=O)ccnc(-c2ccco2)c1 S(=O)(=O)(c1cccnc1NCc1cn(CC)nn1)N(CCCC=C)CCOC N1(C(Cn2nnc(C)n2)=O)CC2(CO)CC1(C(=O)NC(C)CC(C)(C)C)C2 N1(CC#Cc2ncn(C)n2)CCc2ncncc2C1 C(CCC)(CCCNC(C1(n2nccn2)CC1)=O)CC.N1(CC(=O)N)CC(=O)NC1=O C1(CC)(CO)CCCN(C(=O)CC2CCCN(C(=O)CC(C)(C)O)C2)C1 C(=O)(C1=CC(C)(C)C1)N1CC(CC(C(=O)NCCc2n(CC)cnn2)F)C1 c1(C(=O)NCC(C(C)(C)C)NC(C2CC(=C(F)F)C2)=O)cc([N+](=O)[O-])ccn1 C1(CCNC(=O)C2=CCC2)CC2CCC(C1)N2C(=O)CCc1ccncc1 C=CCCCCC(=O)N1CCCC(C)(NC(C2CN(C(C)=O)CCO2)=O)C1 C1(NC(CC(C)OC)=O)CCCC2CN(C(c3ccc[nH]3)=O)CC12 N1(C(Cc2nc(C)[nH]n2)=O)CCC(NC(=O)CCCOc2ccccc2)C(O)C1 c1(C(=O)NC2CC(CNC(C=Cc3c(C)nccc3)=O)C2)ccn2nnnc2c1 c1(C(=O)NC(C)CNC(=O)C(C)NS(C)(=O)=O)ccc2nnn(C)c2n1 C1(SC(C)C(=O)NC(C)(C)CN(C(=O)Cc2ccccc2)C)CCCCO1 c1(-c2n(-c3cccc(O)c3)nc(C3CSC3)n2)nccc2c1[nH]c1ccccc21 C1(CC(N2CCC(N(C(=O)COc3ccon3)CC#C)C2)=O)CCCCC1C c1(SCC(=O)NC(C(F)(F)F)C2CCCNC2)ccc(O)cc1 CC(F)CC(=O)N1CCC(CCC(=O)NCC2(C3CC3)CC2)C1 C(=O)(C1=CCCCO1)N1C(CNC(=O)CC2CCSCC2)CC(COC)C1 N1(C(=O)OC(C)(C)C)CCC2(OC(c3nccc4occc34)=O)CCCC12 c1(CNC(CCSCC)=O)ccnc(N2CCN(C(C3CCOC3=O)=O)CC2)c1 N1(C(C2N(C(C(CC)COC)=O)CC=CC2)=O)CCc2nnnn2CC1 c1(C(=O)NC2C3N(C(Cc4cc(C)no4)=O)C(CC3)C2)nc2ccccc2s1 C(=O)(C(CCC1CC1)NC(=O)CC(C1CC1)C1CC1)N(CC(COC)C)C C(CCNC(c1nc[nH]c1C(C)(C)C)=O)(C(C)C)NC(C(n1ncc(C)c1)C)=O CCC(O)C(C)C(=O)N1CCC(NC(c2cn(-c3ccccc3Cl)nn2)=O)CC1 N1(C(C(CC)NC2CCN(Cc3cccnc3)C2)=O)CCCC(CC)C1 N1(C(c2cc[nH]n2)=O)CC(NC(=O)C(C2(O)CCOCC2)(F)F)CC12CCCC2 c1(CC(N2CCN(CC#N)CC2)=O)c(F)cccc1Br c1(C(=O)NC(CCN(C(C2(CC=C)CCOC2)=O)C)C)nnc(S)n1C C1(CCNC(CC2(OC)CC2)=O)CSCCN1C(=O)CC(C)CF CC1CN(C(=O)C#CC2CC2)CCN1C(=O)COCc1ccc(C#N)cc1 C(CC(C)(C)C)(C(=O)N1CC(O)CC1C(=O)N(C)CC1CCC(=O)N1)OC c1(N(C(C)=O)C)cccc(OC(C)C(=O)NCCCc2nncs2)c1 Clc1cccc(CNC2CCCS2)c1-n1ccnc1 Cn1ncc(C(=O)NC2CCOC(C(=O)NCCCC3CCC3)C2)c1Cl c1(C(=O)NC2CC(C)(NC(C(CC)=CCCC)=O)C2)cncc(C)n1 c1(C(=O)NC(C2CCOC2)CNC(C2(SC)CC2)=O)ccc(OCCF)cn1 CCCC(C)(C)CNC1CCOCC1OCc1ccccc1 C=C(Cl)CC(C(=O)NC1CCOCC1C)NC(=O)C(C1CCC1)OCC n1(CC)nnnc1C(c1cc(F)c[nH]1)NCc1occc1C CC(C)C(C(C)NC(C1(F)CC1)=O)NC(c1cc(-c2cccs2)on1)=O N1(CC(=O)N(CCCCN(C)C(C2CC2(C)Br)=O)C)CCC(O)CC1 N1(OC(CS(=O)(=O)NCC(c2ccccc2)N(C)C)=O)CCCOC(C(C)Cl)C1 N1(C(c2cc(N)c(F)cc2)=O)CCCN(C(c2ccc3c(c2)CC3)=O)CC1CO c1(NC(C2(NC(C(C3CCCC3)OC)=O)CSC2)=O)csc(C(N)=O)c1 N1(C(COCCC)=O)CC2C(CN(C)C(c3oc(Br)cc3C)=O)C2C1 N1(C(=O)NC(COC(C)C)C)CC2CCCC2(C(=O)OC(C)(C)C)C1 C(C(C)(CC)C(N)=O)NC(CN(C(=O)C(O)CCCC)CC#C)=O c1(CNC(C(COC)(C)C)c2ccccc2)cnc(C)c(Cl)c1 c1(C(=O)NCCC(CNC(c2cc(OCC)n[nH]2)=O)O)ccc2ncc(C)n2c1 C(CCCCCNC(=O)C(C)(C)C)n1cc(CC(=O)NCCCCCC)nn1 N1(C(Cn2ncc(C)c2)=O)CC=C(C(C)(C)C(=O)N2CCC2CC(C)(C)C)C1 N1(C(C23CCC(C(=O)OC)(CC2)C3)=O)CC(CN)C(S(C)(=O)=O)C1 CC(CNC(C1CCCC(NC(=O)C2=CCSC2)C1)=O)CC(F)(F)F CC(C)(C(=O)N1CC(CCCCNC(=O)C=Cc2cncs2)C1)c1cc[nH]n1 C(=O)(C1=NNC(C(F)(F)F)C1)NC1C=CC(CNC(c2c(C)ccnn2)=O)C1 C12(CCN(C)C1)C(=O)NC2.c1(C(C)=O)cc(C(=O)NC(C)(C)C(=O)N(C)C)no1 Cc1nc(CO)sc1C(=O)NCCOCCN(C(C)C(=O)NCC(C)C)C C(=O)(C1Cc2ccccc21)NC(c1ccc(OC)cc1)CNC(C=CCC)=O c1(CC(=O)N(C(C)CNC(c2c[nH]c(=N)s2)=O)C)cnn2ccccc12 N1(C(CCC)=O)CCC(CO)(CNC(c2cc(C)cc(Br)c2)=O)CC1 c1(N2CC(C(=O)NCC(c3cc(C)oc3C)C)C2)ccc(Cl)cc1C#N C(=O)(C(O)C(F)(F)F)NC1C(OCC(N2CCC(C)CC2)=O)CCCC1 C#CCCCC(=O)NC(C(C)NC(c1ccc(CSCC)cc1)=O)C(C)C Cc1[nH]nc(C(=O)N(C2CCN(C(=O)CC3CCCCN3C(C)=O)C2)CCO)c1F c1(C(C(=O)N(CC2N(C(CCC#C)=O)CCC2)CC)C)ccc(CC)cc1 c1(C(CC)O)nnc(N2CCC(O)(c3ccc(C)cc3)C2)n1CC(C)C N1(C(C(C)C)=O)CCC2(CC1)CC(NC(c1ccc(S(C)(=O)=O)cc1)=O)CO2 c1(NC(=O)NC2(c3cc(C)no3)CCCC2)cnc(O)c(C(F)(F)F)c1 C(c1ccncn1)=CC(=O)NC1(CC(=O)NCC2(C(C(C)C)O)CC2)CCC1 CCC(C)(O)CNC(=O)CC1CCN(C(=O)CC2CN(C(C)=O)C2)C1 c1(CC)cc(=NC(=O)CC(CC)NC(C2CNC(=O)O2)=O)[nH]n1C CC(C(=O)NC1CCCC(NC(C2CCC=CCC2)=O)C1)C(C)O Cc1cn(C)nc1C(C(=O)NC1CCOC1)N(CCC#N)Cc1ccccc1 CC1CC2(CCN(C(=O)Cc3ccc(F)cc3Cl)CC2)CN1C(=O)C=CC1CC1 Cc1cc(C(=O)NC2CC(CNC(=O)CC3CN(C)C3)CC2O)cc(C)c1F c1(C(=O)NC(CC=C)CNC(=O)CC(=O)NCC)cc(S(=O)(=O)NC)cn1C C1(N(C(=O)Cc2ccsc2)C)CCCC(NC(c2nnn(C)c2C(F)F)=O)C1 N1(CC)CCCC2C1CCCN2C(C(=O)NCc1ccccc1Br)C(CC)OC c1(CC(=O)NCC2CCCN(C(C3(C)CC(C#N)C3)=O)C2)ccc2ncsc2c1 c1(C(=O)NC2CCCCN(C(C(C)C(C)(C)C)=O)C2)ccc2c(c1)NC(=O)C2 c1(C(=O)NCc2ccc(C)cn2)coc2c1CN(C(=O)C1=CCCC1C)C2 CCC(CC)(C(=O)NCC1CCC(N(C)C(c2nnsc2N)=O)CC1)OC c1(C(N2CC3CCC2CN3C(C2(C(F)(F)F)CC2)=O)=O)cc(O)cc([N+](=O)[O-])c1 C=C1CCC(C(=O)NCC=CCNC(c2ccncc2N(C)C)=O)CC1 C(=O)(CC(C)P(C)(C)=O)NC1CC(CCNC(c2[nH]cc(C(=O)OC)c2)=O)C1 Cc1cc(F)ncc1CNC(=O)NC(C)COCc1ccccc1 CCCCC(C)N(C(=O)C(=O)N1CC(OCCOC)C1)C N1(C(C2=CCC(NC(C(CC)=CCCC)=O)C2)=O)CCc2c(cnn2C)C1 n1(CC)cc(C(=O)NC(CNC(=O)COC2CCC2)C(C)C)c(C(C)C)n1 c1(C(=O)NC(c2cccnc2)C(=O)NCC2CC(C(C)C)C2)cnc(Cl)s1 c1(C=O)ccc(S(N)(=O)=O)o1.CC1(C)CCC(C(=O)NCC2C3CNCC23)C1 C(c1cccc(F)c1F)=CC(=O)NCC12C(CN(C(C=CC)=O)C1)C2 N1(C(C2CCCN(C(COCCCN(C)C)=O)C2)=O)CC2(C1)OC(=O)NC2C CC1=NN(C)C(=O)C1CC(=O)N(C1CN(C(=O)C(=O)Nc2ccccc2)C1)C N1(C(CC2ON=C(CC)C2)=O)CC2CCOC2(CNC(=O)C2=C(C)CCCC2)C1 CCCC(CNC(=O)C(N)=O)C(=O)N1CCC(COC(C)=O)C1 C(=O)(CS(=O)(=O)CCOC)N1C2CN(c3cc(CC)ncn3)CC1C2 c1(C2(CNCC3CCC(C(=O)OC)CC3)CC2)ccc(Cl)c(F)c1 C1(CC(=O)N(CCN(C(C(C(CC)O)C)=O)C)C)C2CC3CC(C2)CC1C3 C1(CNC(C(C=C)CC)=O)CN(C(=O)C(C)OC2CCCC2)CC12CC2 c1(C(=O)NC2CCC(N(C(c3occ(C)c3)=O)C)C2)ccn2ccnc2c1 C(C)(CCCCNC(c1ccc(Cl)cn1)=O)NC(CCN(C(CCC)C)C)=O C1(N(C(c2c(C(C)C)nco2)=O)C)CCCN(C(=O)C(c2ccccc2)F)CC1 CC1(C)C2CCC(C(=O)NCC3CCCC3NC(c3cnc(C4CC4)[nH]3)=O)C1C2 C1(C(CC)CC)CC(NC(=O)NC2(C(=O)OC)CS(=O)(=O)C2)CCO1 c1(OC)nc(N(C2CNCC2(F)F)Cc2ccc([N+](=O)[O-])s2)ncc1C Cc1cc(C(=O)N(CCCN(C(=O)COCC(F)F)C)C)nc(O)c1 c1(C(C)NC2(c3nnnn3C)CC(CC)C2)ncccc1C c1(OC)ccc(CNC(=O)C(C2CC2)NC(c2ccc(F)s2)=O)cc1 C(=O)(CC(C)(C)CC(F)(F)F)NCC1CCN(C(C(c2ccc(F)cc2)C)=O)C1 C1(NC(CC2CCC(NC(C(CC3CCC3)OC)=O)CC2)=O)CCC2(CCC2)C1 c1(C(N(C)CC2N(C(C(C)CC3CCC3)=O)CC(F)C2)=O)ccc2ncsc2c1 C1(CNC(c2c(C)nns2)=O)N(C(=O)COc2cccnc2Cl)CCCC1(C)C N1(C(c2sccc2Br)C(=O)NCC(=C)C)CC(C)(C)c2cc(Cl)ccc21 CCCC(CC(=O)N1CCOCC1CC(N)=O)NC(=O)CC(C)CC C1(CNC(c2cc(OC)no2)=O)CN(C(=O)C2=CCC2)CCC1C(F)(F)F CCCCCCC(C)C(=O)N(CCNC(c1c(F)cc(O)cc1F)=O)C(C)C N1(C(C2C(COC)C2)=O)CCC(NC(c2ccnc(F)c2OC)=O)C2(CCC2)C1 c1(C(N2CC(NC(C(C)N3CCC3)=O)C(F)CC2)=O)ccc(O)c2ncccc12 c1(C(=O)NC2(C)CCN(C(C3CC(n4cnnc4)C3)=O)C2)cc2c[nH]cnc-2n1 C1(C(N(CC)CC2CCCCN2C(=O)C=C(C)C)=O)CCCCCN1C N1(C(=O)CC2CC2)CC2(Cc3ccccc3)CC1(C(=O)O)C2 C(=O)(C1Cc2ccc(Cl)cc21)NCCS(C(C)(C)C)(=O)=O C1(C(N2CC(c3c(CNC(c4ccns4)=O)nco3)C2)=O)CCc2cnnn2C1 c1(C(N2CC(NC(c3ccnn(C)c3=O)=O)C3C2C3)=O)ccc2c(c1)OCCO2 N1(CC)OCC(NC(C2CC(CCNC(=O)CC3CN(C(C)=O)C3)C2)=O)C1=O C1(NC(CC=CCC)=O)CCCC12CCN(C(=O)C(C)(O)CC(C)C)CC2 Cc1cccc(OCC(=O)NC(C)(C)CN(C(=O)CC2CCC(C)(C)O2)C)c1C N1(C(C2CCCN(S(CC=C)(=O)=O)CC2)=O)CCC2(CC1)OCCc1ccsc12 N1(C(C(C)(C)CC2CC2)=O)CCOC(C)(CNC(C23CC=CC(C2)OC3)=O)C1 C1(C)(CNC(C(C2CC2)OC)=O)CN(C(=O)Cc2ncoc2C)CCO1 c1(CC)c[nH]c2ncnc(N3CC4(CN(C(c5ccc(C6CC6)cc5)=O)C4)C3)c12 CC(C(=O)N1CC2C(NC(C3CC(n4cnnc4)C3)=O)C2C1)C1=CCCC1 c1(C(=O)NCC(C2CCCN2C(C2CNC(=O)O2)=O)(C)C)cnn(CCO)c1N c1(CC(=O)N(C2CCN(C(C3CCN(S(C)(=O)=O)C3)=O)C2)CC)ncn(C)c1C N1(C(c2c(C(F)F)ccc(C)c2)=O)CC2(CCC(CNC(=O)C(C)O)O2)C1 N1(C(C(C)=CC2CC2)=O)CC2(NC(c3ccc(C)nc3O)=O)CCC1C2 Cn1cc(C(N2CCC(O)(c3ccccc3)C2)=O)c(OCc2ccccc2)n1 C1(NC(CC(C)CN(C)C)=O)CN(C(=O)C(C)n2ccnn2)CCC1O c1(C(N2CCC(C)(NC(CC(CCC)(C)O)=O)C2)=O)cc2ccccc2[nH]c1=N c1(C(=O)NCC23CC(NC(c4c(CC)cco4)=O)(C2)C(C)O3)cn2ccccc2n1 N1(C(c2cnc(CCC)s2)=O)CCC(CCNC(c2cnnn2C(C)C)=O)CC1 c1(OC(C)C)ccc(C(=O)N(C2CCCCC2NC(c2c[nH]c(=N)o2)=O)C)cn1 c1(C(N(C2C(C)CCN(C(C3CC(=C)C3)=O)C2)C)=O)ccc(Cl)c(Cl)c1O C(=O)(C(C)(C)NC(=O)NC1CC(C(=O)NCCc2ccccc2)C1)NCC CC(C)CC(C(=O)NCC1CC(NC(c2ccc(C(C)C)o2)=O)C1)C(C)C C1(C(=O)NCC2C=CCN2C(c2cnc(C(C)(C)C)o2)=O)(OC)CCSC1 c1(N(C)C)ccccc1C(=O)NCC1CCCC1NC(=O)CC1(C2CC2)CC1 C1(C(=O)NCC(C)C(=O)OC)(OC)CCN(C(=O)C=CCN(C)C)C1 N1(C(Cc2cccc(C)c2)=O)CC(NC(C2(F)CCS(=O)(=O)C2)=O)C(C)(C)C1 C1(=O)C(N(C)C)CCC2C(C(C(=O)OC)N1)C2.C1(SC)CC1C CCCCCCCCCCC(=O)NCC(C)CNC(c1ncoc1C(C)(C)C)=O c1(-c2cn(C(C)C(=O)NC3CCCN(O)C3=O)nn2)cc2ccccc2s1 Cc1cc(C(=O)NC2CC3CC(NC(=O)C4=NNC(=O)CC4)C3C2)c(F)cc1Cl c1(C(=O)OCCc2cc(C)on2)ccc(Cc2ccc(Br)cc2)cc1 C(=O)(C(=O)N=S(C)(C)=O)N1CC(CC)C(NC(C2CC(CC)(CC)C2)=O)CC1 C12(CNC(CC(C)(C)OC)=O)CCCC1N(C(=O)C=C(C)C1CC1)CCC2 Cc1ccc(NC(=O)N(C)C)c(SCCN(C(C23CCC(CC2O)C3)=O)C(N)=O)c1 C1(NC(C2(CSC)CN(C(=O)CN3CCOCC3=O)C2)=O)(CO)CC2CCCC12 C1(CC2CCC(NC(N(C(c3ccncc3)C)CC)=O)CC2)CC2C(C1)C2(F)F Cc1cccc(CNC(C2CC(C)CN(C(=O)CCNC(=O)CO)C2)=O)c1F N1(C(C2CCCC(C)O2)=O)CC(C2(NC(=O)Cc3ccc(F)cc3)CC2)C1 C1(c2nnnn2CC)(Nc2cccc(NC(CCC)=O)c2)CCN2CCCCC12 c1(NC(N2CC3C(CC(=O)NC(CCO)C(F)(F)F)C3C2)=O)cc(Cl)ncc1F c1(C(=O)NC(CC)(C)CNC(=O)C=Cc2cccnc2)cncc2cnccc12 N1(C(Cc2cccc(C#N)n2)=O)CC=C(c2cccc(Cl)c2)CC1 Cc1ccc(CCCC(N2CC(NC(c3ccn(C)c3)=O)CC2C)=O)cc1 c1(C(N2C(CNC(c3c(C)coc3)=O)CC3CC32)=O)cc2c(Br)cccc2[nH]1 c1(CN(C(c2c(CC)c[nH]n2)C(=O)NCc2cccs2)C)nc2ccccc2o1 S(=O)(=O)(c1cnc(N(C(C)=O)C2CC2)s1)N1CCC(F)(CC)CC1 N#Cc1ccccc1-c1cccc(C(C2N(CC3CC3)CCCC2)=O)c1 C1(C(C(=O)NCCN(C(C(CCC)=CCC)=O)CCC)O)CCS(=O)(=O)CC1 C1(NC(C(N2CCCCC2)C)=O)CCCCN(C(c2cnc(C(N)=O)s2)=O)CC1 c1(C(N2C(CN(C)Cc3nnc(C)s3)CCCC2)=O)cn2nccc2nc1C c1(OC)ccc2c(c1)CC(C)N2C(c1cncc(Br)c1)=O c1(COC)ocnc1C(=O)NCC1(NC(C23CC(CO2)C3)=O)CCC1 C1(C(=O)NC(c2nn[nH]n2)CC)CSCN1C(=O)C=CC(C)C C(=O)(C1CCCc2c(O)cccc21)N1CC(CNC(CC=CC=C)=O)C2(C1)CC2 C#Cc1ccc(NC(C2(CNC(=O)CCC)CC3(CC3)C2)=O)cn1 C(C)(C(=O)NCC1(CC(=O)N(CC(O)CC)C2CC2)CC1)OCCOCC N1(C(CCc2cnc(C)s2)=O)Cc2cccc(F)c2C1 Cc1sc2ccccc2c1S(=O)(=O)NCC(C)S(C)(=O)=O c1(C(C(=O)NC(CNC(c2ccn(CCC)n2)=O)C)(C)C)ccc(Cl)c(Cl)c1 N1(C(C2N(C(c3c(C)n(C)nn3)=O)CC3CC32)=O)CCCC(C)(O)C1 C1(CNC(c2cc(C)oc2)=O)COCCN1C(c1ccc(C(C)F)cc1)=O N1(CCNC(c2c(O)nc(=O)n3c2CCC3)=O)CCS(=O)(=O)C2(CCCCC2)C1 N#Cc1ccc(O)c(C(N2CCC(NC(c3ccsc3C(F)F)=O)C(O)C2)=O)c1 N1(C(C2(OCC)CCC2)=O)CCN(C(c2c(F)cc(O)cc2F)=O)CC(CO)C1 C(C(C(=O)NC1CC(NC(N)=O)C1)NC(=O)C(C)c1cccs1)OC N1(C(C(COC)C)=O)CCN(C(c2cn(-c3ccccc3OC)nn2)=O)C(C)C1 c1(C(=O)NCC#CCNC(c2cocn2)=O)ccc(Cl)cc1C(F)(F)F C1(CC(N2CCC(C(N(CC#C)CCOC)=O)C2)=O)CCC(=O)N1C N1(C(C2N(N=O)CCC2)=O)CCN(C(=O)CCF)CC2(CC2)C1 C1(NC(c2cnc(CC)s2)=O)CCCC(NC(c2cccn2C2CC2)=O)C1 CC(CNC(=O)C(O)CC1CCCCC1)(CO)NC(=O)CCc1csc(=N)[nH]1 C(=O)(C(C)(C)CCC#N)NCCN(C(C1CC(CC(=O)OC)C1)=O)C(C)C CP(C)(=O)C(O)C(=O)N1CC2(CNC(c3cnnc(O)c3)=O)CC2(C(F)(F)F)C1 C1(C(N(CCCNC(c2c(CC)non2)=O)C)=O)CC2(C1)CC(C)C2 CCC(C)C(CC(=O)NCC(O)C(C)(C)O)NC(c1cc(C)sn1)=O CC(C)(C(=O)NCC(CO)NC(=O)C=C1CCC1)c1cccnc1 c1(C(=O)NCC(CNC(c2c(C)csc2)=O)(C)O)cc(S(N)(=O)=O)cn1C c1(NC(C(=O)N(C(C)CS(C)=O)C)=O)ccc(Br)nc1Cl N1(C(c2c(C)c(O)ccc2)=O)CCC(C)N(C(c2cc(Cl)cnn2)=O)CC1 C1(NC(C2(CC#C)CC=CCC2)=O)CCN(C(=O)CCCCOC)CC1C1CC1 N1(C(CNC(c2c(C)cccc2)=O)=O)CCC2(C1)CN(C(c1cccs1)=O)CCO2 C(=O)(C1Cc2ccccc21)NC1(CO)CCCN(C(c2c(C(C)C)c[nH]n2)=O)C1 n1(-c2cn(C)nc2)ncc(Br)c1C(=O)Nc1ccc(C2CC2)cc1 C(=O)(CC(=O)NC(CO)C(=O)N1CCC1(C)CCO)N(C)C C(=O)(C1=CCOCC1)N1CCC(C(=O)NC(COC)C)(OC)C1 C1(F)(C(N(CC(CCC)O)C)=O)CCN(C(=O)COC2CCC2)C1 C1(C(C(=O)N(C2(COC)CC2)C)NC(=O)Cn2cccn2)CC=CCC1 C1(NC(C2CC(CC)OCC2)=O)CCN(C(=O)C(C2CC(F)(F)C2)O)C12CC2 C(=O)(C(O)CCCc1ccccc1)NC(CNC(c1ncc(C)nc1)=O)CO c1(C(N2C(CC(=O)N(C)Cc3ccccc3)CCC2)=O)c(Cl)cccc1Cl C1(C(=O)NCCCCC#C)CCN(C2CCN(C(c3cc[nH]c3)=O)CC2)CC1 c1(C(=O)NC(C2(CNC(CCOC)=O)CC2)C)c[nH]c2nc(Cl)ccc12 c1(C(C(=O)NCCC2(CNC(CNC(=O)NC)=O)CC2)O)ccc(F)c(Cl)c1 C#CCC(CC(=O)NC12CCN(CC1)C2)NC(=O)C(CO)OC c1(C(N(CC(C)NC(=O)CSCC(F)F)C)=O)cnc(C2CC2)[nH]1 N1(C(c2c(C)cnnc2)=O)CCC(C)N(C(=O)CCOc2ccccc2Cl)CC1 c1(OC)cc(C(O)C(=O)NC2CCCN(C(=O)C(F)=C3CCC3)C2)c(F)cc1O C(C(C)(C)CC(C)C)NC(C(CCC1CCC1)N(C1CC1C(C)C)C(C)=O)=O O=C(CC(C(F)(F)F)NC(=O)CSC1CC1)NCC12CC(CO)(CO1)C2 NS(=O)(=O)c1ccc(C(=O)NC2C=CCN(C(C3CC34CCC4)=O)C2)nc1 C1(NC(c2c(C)nc(CC3CC3)s2)=O)CCN(c2cncc(Cl)n2)CC12CCC2 CCCCC(O)C(C)C(=O)NCCC1CCN(C(c2cc(F)ccc2CC)=O)C1 C12(C(=O)NCC(C3CC3)NC(CCSCC(N)=O)=O)CC(F)C1C2 N1(C(c2ccc(S(C)(=O)=O)s2)C(=O)NC2COC2)CCOC2(CCSC2)CC1 c1(C(=O)OC)cccc2nc(COC(=O)C(C3CCCCC3)N(C)C)cn12 N1(C(CC(=C)Br)=O)CCC(CCCNC(c2ccnc(OC)c2)=O)CC1 C(=O)(C1c2c[nH]nc2CN1C(=O)CC(O)C(C)C)N(CCSC)C C(=O)(C(C)C(O)C(C)C)NC1(CO)CCN(C(Cc2c(C)cccc2)=O)C1 C1(NC(C)=O)CCN(C(=O)C(=O)Nc2cc(C)n(C(C)C)n2)C(c2ccco2)C1 N1(C(C(COC)(C)O)=O)CCC(C)(CCNC(=O)CNC(=O)CN(C)C)CC1 Cc1c(C(=O)NCc2ccc(C(F)(F)C(F)(F)F)s2)cnn1C(C)(C)C N1(C(c2c(C)nsc2)=O)CCC2(CCN(C(C34CC(CO3)C4)=O)CC2)C1 C1(NC(CCN(C)CC)=O)CN(C(c2cc(C)c(O)nn2)=O)CC1S(C)(=O)=O c1(NCC(=O)NCC(C)CNC(=O)CCC2CCCC2)ccccn1 c1(OC)cc(C)cc(F)c1CNC12CC(C(=O)NCc3cccc(Br)c3)(C1)C2 c1(C(N2CCCC(N(C(=O)C=C3CCCCC3)C)C2)=O)cccc(P(C)(C)=O)n1 c1(C(=O)NC(C(C(C)C)NC(C2(O)CC(F)(F)C2)=O)C)cn(C)c(=O)n(C)c1=O N1(C(c2cn(-c3ccccc3)nc2C)C(=O)NC(CC)C)CCC(C)OC(C)C1 N1(C(c2ccc(CN(CC(F)(F)F)C)o2)=O)CC2C(CNC(C3(F)CC3)=O)C2C1 c1(C(=O)NC(CNC(C2(CF)CC2)=O)CO)cc([N+](=O)[O-])c(Cl)cc1Cl c1(C(=O)NC(CCOC)CNC(=O)C(C)c2cccs2)ccc(S(N)(=O)=O)s1 C1(C(=O)NCC(CCNC(C2(NC(N)=O)CC2)=O)O)OCC2COCCC12 C(=O)(C(C(C)(C)C)C1CCC1)N1C(C(C)NC(c2cccnc2)=O)CCCC1 c1(C(N(CCN(C(CC2C(C)CCC2)=O)C)C)=O)ncccc1S(C)(=O)=O N1(C(c2c(OCc3c(C)cncc3)cccc2)=O)CCN2CCOCC2C1 c1(CC)cc(C)ccc1C(=O)NCC1CC(O)CN1C(c1cnc(CC)s1)=O N1(C(CCC(C)OCC)=O)CC2CC1CCN2C(c1ccc(F)cc1Cl)=O C1(F)(CNC(c2c(C)scc2)=O)CCN(C(=O)CC(C)C2CCCO2)CC1 C(CN=C(NCC1CCC1)NCC(c1ccccc1)(C)O)c1ncc(C)cn1 c1(NC(c2nnnn2-c2c(CC)cccc2C)(CC)C)cnc2n1CCCC2 c1(-c2cn(C3(NC(C(CC)=CC)=O)CCC3)nn2)ccccc1C(=O)O CCCN=C(NCC1CCOC1C(C)C)NCCSCc1ccccc1F N1(C(C(C(C)(C)C)NC(C(C(CC)C)N(C)C)=O)=O)CCC2(CC=CCO2)C1 C1(NC(N2CCC(c3scc(C)n3)C2)=O)CC2CN(C(=O)OC(C)(C)C)CC2C1 C1(NC(CCC2CCCN(C(CCC#C)=O)C2)=O)CCN(C)CC1(C)C Cn1cnc2sc(C(N3CC(NC(c4cc(C#N)c[nH]4)=O)C(C4CC4)C3)=O)cc12 c1(OC)cccc(CNC2CCC(CCN)C2)c1C C(=O)(C1=C(CC)N(c2ccc(Cl)cc2)C(=S)NC1c1cc(COC)[nH]n1)OCC CC(C(=O)NCCC(C)N(C(=O)Cn1ccc(C(F)F)n1)C)S(C)(=O)=O c1(CC(=O)N(C)CC2N(C(c3cc(C)oc3)=O)CCOC2)ccc(S(C)=O)cc1 c1(C(=O)NCC2C(NC(C3(COC)CCC3)=O)C2)ncc2ccccc2c1O c1(CC(=O)NCC(C)NC(c2csc(C(F)(F)F)n2)=O)cccc(F)c1Cl c1(C(N(CCCCCNC(=O)C(C)C2CCOC2)CC)=O)cccc2c1OCC2 C1(NC(c2c(C)coc2C)=O)CN(C(=O)Cn2[nH]cnc2=N)Cc2nccn2C1 O=C(C1=COCCC1)NCC1CCCCN(C(=O)CSCc2cccnc2)C1 c1(CNC(CN2CC(C)(C)C(NCc3ccccc3)C2)=O)cc2ccccc2[nH]1 C(C1=NOC2COCC12)N1CC(N2CCN(C(CCCCCN(C)C)=O)CC2)C1 c1(NC(C2CCN(C(c3cnc(C)[nH]3)=O)CC2)=O)cc(F)cc(C)c1Br c1(N2CCN(CC=C)CC2=O)ccc(C(N2CCCCCC2)=O)cc1F c1(C(NOCCC#C)=O)n[nH]c2c1CN(C(=O)CC(CC)C(F)F)C2 C(=O)(C1=CC2CCC(C1)C2)N1CC2(OCC(C(N(C(C)C(=O)OC)CC)=O)C2)C1 C(=O)(CC(CC(=O)O)C(F)(F)C(F)(F)F)NCC(N1CCCCC1)C C1(C(=O)NC(C)C(N2CCC(OC(C)C)CC2)=O)(CC)CC(C)(C)C1 C=CCC(CC=C)C(=O)NC1(C(=O)NCCCC(=O)NO)CC1C O=C(C1=C(Cl)CCOC1)NC1CCC1NC(c1ccc2nc[nH]c2n1)=O C1(NC(C2(CCCC)CCC2)=O)COC2CN(C(=O)C=C3CCOCC3)CC12 C=CCCC(C(=O)NCC)N(C1CCCCCC1)CC1CCOC1C C1(CNC(c2n(CC)c(O)nc2)=O)CCN(C(c2cc(=N)[nH]n2C)=O)CC1C c1(C(=O)NCC2N(C(C(C)CF)=O)CCN(C)C2)cc2cc(Cl)ccn2n1 c1(C(=O)NC(C(=O)N(CCC#C)CC)CC2CC2)ccccc1CC c1(OC)ccc(NC(=O)CCN(C(=O)CC2CCCC(C)O2)C)cc1F CCC(C(=O)NC(C)C(CO)NC(C1(C2CC2)CC1)=O)OC.C1(C(=O)N)CCCC1 C(=O)(C1=NOC2(CCC2)C1)N(C1CCN(C(C(CC(C)C)N(C)C)=O)C1)CCO c1(CN2CC(CS(=O)(=O)NC)NCC2)cc(Cl)cc(Br)c1 c1(CC)cc(C)[nH]c(=NCCCCCCN(C(=O)C2=CCOCC2)C)n1 c1(C(=O)NC2C3CN(C(C(CC=C)(C)C)=O)C2C3)cnc2c(C)nsc2c1 S(=O)(=O)(c1ccc(NCC2COCC2(C)C)c(Cl)c1)NCC1(S(CC)=O)CC1 N1(C(C(COC)(C)C)=O)CC(C)CN(C(c2cnc3ccncc3c2)=O)C(C)C1 C1(C(=O)NCC2(SC)CC2)(NC(CCC)=O)CCC(C)(C)C1 CCC(C(=O)N(CCCCO)CC)NC(N)=O N1(C(c2c(CC)nc(C)nc2)=O)CCCC2(C1)CN(C(=O)CSC(C)C)CCO2 CCC(C)C(O)CC(=O)N1CC2COCC2(C(N2CCOCC(C)(O)C2)=O)C1 c1(C(N2CC(OC)(CO)C2)=O)coc2c1CN(C(=O)CC(=O)NC1CCCC1)C2 C#CC1(CNC(=O)CCN(C(c2cncc(C)c2)=O)C2CC2)CCCC1 C1(C)(C(N(CC(C)(C)CNC(C2CC(CC(C)(C)C)C2)=O)C)=O)CCSCC1 Cc1cc(C)c(C(N2CCCCC(NC(C34COC(CCO3)C4)=O)C2)=O)cc1C C1(NC(CCC2C(C)(C)C2)=O)COCCC1C(=O)NCC1CN(C(=O)O)C1 n1(CC(=O)NC(CNC(C2CCC(NC(=O)OC)CC2)=O)C)cc(C)ccc1=O Cc1nc(C(=O)NCC2CCN(C(C3CCCN3CC(F)(F)F)=O)C2)cc(O)n1 N1(C(C(C)(CO)NC(C2CCCC2F)=O)=O)CCN2C(=O)NCC2C1 CC1CCCC1C(=O)NCCCOCCNC(=O)C(C)n1ccnc1 C1(NC(C(C(C)C)O)=O)CCCCN(C(=O)CN2CC(C)(C)C2)C1 c12cccc(c1)N2.N1(C(C2(C)C(C)C2)=O)CCC(C)(c2cn(C3CCC3)nn2)C1 c12cn3ccc(cc3n1)OC2=O.c12cncc(c1C)C(=O)N1CCN2CC1.CO.OC c1(N2C3C(NC(CC(C)C4CC4)=O)(CCC3)CC2)ncnc2c1cnn2C C1(C(=O)OCC)CCCCN1C(C1CC(O)CN1C(C1CC1C)=O)=O CC(C(=O)N1CCN(C(c2cc(-c3cn(C)nn3)on2)=O)CC1)S(C)(=O)=O N1(C(c2ccc(CC)cc2O)=O)CCC2CN(C(=O)C(CC)CC(C)C)CC2C1 CCC(O)C(=O)N(C)CCN(C(=O)CC1CCCOC1)C N1(C(CN(S(CC)(=O)=O)C)=O)CCOCC1CCNC(=O)C=C1CCN(C)C1 c1(C(N2CC3C(NC(C4CCCN(C)C4)=O)(C3)C2)=O)cc(Cl)ccc1Cl N1(C(COCC)=O)CCCC(C)(C)C1CNC(=O)CC1(C)CCOC1 C1(C(N2CC(C(C)NC(c3cnn(C4CCCC4)c3)=O)C2)=O)CC2CC1C1CC21 c1(OC)ccc(CCC(=O)N(C)CC2CCCN2c2nccnc2F)cc1 C1(NC(=O)NC(C2CCOCC2)CC)CCCN1Cc1ccncc1 C(=O)(C(C)C(O)C(C)CC)N(CC(=O)NC1CC(O)C1OCC)CC#C C(=O)(C1=C(Cl)CC1)NCC(CO)NC(C(C)(C1CC1)OC)=O C(CC(O)C(F)F)NC(c1ccn(CCNC(=O)CC2CCCC2)c1)=O O=C(CCCCCCn1cc(-c2ccsc2)nn1)NCC1CCC12CC2 c1(C(N2C(C(=O)NCC(=O)NC3CCCCC3)CSC2)=O)cc2scc(Cl)c2[nH]1 c1(OC)c(Cl)cc(C(N2CC(N(C(=O)Cc3c[nH]nc3O)CCO)C2)=O)cc1Cl c1(C(=O)NC2C(NC(=O)C=Cc3cc[nH]c3)CC2)n[nH]c2c1CSCC2 C1(C(=O)NC(CCNC(=O)C=CC(=O)NC2CC2)C(C)C)(OC)CCCCCC1 C1(COC)CC(CNC(c2cc(C(C)C)nn2C)=O)N(C(c2ncoc2C)=O)C1 c1(C(=O)NC2CC2)ccnc(N(C)Cc2nc(NC(C=NOC)=O)sc2)c1 c1(OC)cncc(NC(C2COCCN2C(=O)C(n2ccc(C)n2)C)=O)c1 N1(C(c2cn(CC)nc2)=O)CCC(CC2CN(C(C3CCC(O)CC3)=O)C2)CC1 S(=O)(=O)(CC(=O)N1CCC(C)(NC(=O)CC(C)C2CCCCC2)C1)NCC c1(N2CC(NC(=O)CN3CCCCC3)C3(C2)CC3)ncnc2c1CCCC2 C(CC(=O)N1CC(NC(c2c(C)cnn2C)=O)C(F)C1)(C(F)(F)F)OC CCCCCCc1ccc(C(N2CC(O)(C(C)NC(=O)C(C)=CC)C2)=O)s1 CCCCCCC(C)(C)C(=O)NC(C)CCCNC(=O)C(C)NC(C1CC1)=O N1(C(c2ncn(CC)c2)=O)CCCOC(CNC(=O)C(C)C2CCC2)C1 c1(C(C)C)cc(F)c(C(=O)NCC2(NC(C3CCC3C)=O)CCCCC2)cc1F c1(C(N2CCC3(C2)CN(C(C2CCCO2)=O)C3)=O)cc(F)cc(Br)c1Cl C1(C(N2CC(SCC)C2)=O)CC(C)(C)CCN1C(c1cc(C)co1)=O CCC(C(=O)OC)C(=O)NC(CC)CCC(=O)NCCC1(OC)CCC1 n1(C(C)C)cc(CC(=O)N(CCCNC(=O)C(C)c2cccs2)C2CC2)nn1 c1(C(N2C(C)CCN(C(c3c(C)nn(C)n3)=O)CC2)=O)cnc2n1CCC(C)C2 C(C(C)N=c1cc(NCCCC(C)CO)nc(C)[nH]1)c1ccc(C)cc1C C=CC1CN(C(c2occc2COC)=O)CC1NC(=O)CC1CCSC1 Cc1nc(NC(C23COC(CNc4ccc(F)cc4F)(C2)C3)=O)c(C)c(Cl)n1 c1(NC(N(CC)CC2(CO)CCN2C(C)C)=S)ccc(NC)cc1 C1(CN(C(=O)CC2(CO)CC2)CC)CN(C(=O)Cn2ccc(C)n2)CCO1 N1(c2nc(N3CCC(C)(COC)C3)nc(C)c2)CCC2(CC1)COC(C)(C)C2 C1(NC(c2c(CC)nc[nH]2)=O)CCCCN(C(C2CC2(C)C(C)C)=O)C1 c1(CC)nc(C)[nH]c1C(=O)NCC1(F)CCN(C(=O)C(=Cc2ccccc2)C)C1 N1(C(c2ccn(CCO)c(=O)c2)=O)CCC2(COC(CSc3ccccc3)C2)C1 CN1C2CCC1CC(CC(=O)NCC1CN(C(=O)CC3CC4(CCC4)CO3)C1)C2 CS(=O)(=NC(=O)c1ccc(Cl)o1)c1cnn2c1CN(C(=O)CC=C(Cl)Cl)CC2 Cc1cc(S(C)(=O)=O)cc(C(N2CC3CCN(C(=O)C=CC(C)C)C3C2)=O)c1C C(CC(F)(F)F)N(C(=O)C(C1CCOC1)NC(c1c[nH][nH]c1=N)=O)C C(=O)(C(CC(C)C)C(N)=O)NC(CCNC(COc1cc(C)on1)=O)C(C)(C)C C1(CNC(C2CCC2)=O)CN(C(C2CCCCC2C2CC2)=O)CCC1(F)F N1(C(c2[nH]cc(C(C)=O)c2)=O)CCC(NC(=O)C(C(C)C)C2CCC2)C(C)C1 N1(C(C(C)(C)C2CCOCC2)=O)CCC2CN(C(=O)Cc3cccnc3)C2C1 N1(C(C2N(C(C(c3n(C)cnc3)O)=O)CC2)=O)CCC(C)(C)C1 C(=O)(C1=CC2C=CC(C1)C2)NCC1(O)CN(C(c2n(C)ncc2C(F)(F)F)=O)C1 c1(OCC(=O)NC(C(C)NC(c2cc[n+]([O-])cc2)=O)CO)ccc(C#N)cc1Cl N1(C(CSCCC)=O)CCC2OCCN(C(c3ccc(S(C)(=O)=O)cc3)=O)C2C1 N1(CC(c2c(OC)cccc2)O)CCC(F)(C#N)C1 C12(NC(C=CCOCCOC)=O)COC(CNC(=O)CC3CCNC3=O)(C1)C2 C1(C(=O)OC)CCN(N2CC(O)CC2C(=O)OC)CC1C C=CC1CN(C(=O)NCCC(C)(C)COCC)CCO1 C#Cc1cnn(C)c1C(=O)NC(C)C(=O)N(C)CCn1cnnc1 C1(NC(CCCCC)=O)CCN(C(c2cccc(-c3nc[nH]n3)c2)=O)C(C)C1 C(=O)(CCC(=O)OC)N1CC(c2cn(CC)nn2)(NCc2cn(C3CC3)cn2)C1 C(=O)(CCC1=CCCCC1)N1CCC(=CCNC(c2csc(CO)n2)=O)CC1 N12CC(CC1C)CNC(=O)Cn1cc(nn1)C2=O.c1(CC)ccc(OC)cc1 Cc1cc(C)c(C(=O)NCC2CCC2NC(=O)CC2CCN(C)C2=O)c(O)n1 c1(C(=O)NCCOCCn2cc(CSCC)nn2)noc2c1CC(C)CC2 c1(C(N2C(C3(NC(C4CCCC4CF)=O)CC3)CCC2)=O)cc2ncccn2n1 c1(OC)c(C(N2CC(CC(F)F)C2)C(=O)OC)cccc1C C1(CC=C)(NC(=O)CC)CCN(C(=O)C(C)(C)OC(C)C)C1 c1(NC(N2CCC(N3C(C)CC(O)C3)CC2)=O)cnn2c1C(=O)N(C)CC2 c1(C(=O)NCCCC(=O)NCC(C2CC=CCC2)=O)nc2ccccc2s1 C1(NC(c2c(CC)nn(C)c2)=O)CCN(C(=O)CCCC(C)(F)F)CCC1CO C(c1cccc(CO)c1)=CC(=O)NC1CN(C(C2(C(C)(F)F)CCC2)=O)CC1O C1(C(=O)NCC2(NC(c3cc(SC)oc3)=O)CC2)Cc2ccc(F)cc2C(=O)O1 N1(c2ccnc(NCC3(C)CCOCC3)n2)CCC2(CNC(=O)O2)C1 S(=O)(=O)(c1ccc(Br)cc1)NC1C2CN(C(=O)C3=COCC3)C(CC2)C1 CC(C(=O)NC1C2CC1N(C(=O)C#CC(C)(C)O)C2)C(F)(F)F C1(CCC)CN(C(c2cccc(C)c2)=O)CCN1C(=O)CN(C1CCC1)C(=O)CC c1(CNC(C2CC3(CC3)CN2C(=O)CC2(O)CCOCC2)=O)nc(Cl)ccc1F c1(NC(c2c(CC)scc2)=O)cc(-c2ccc(COC)nc2)c2cn[nH]c2c1 N1(C(c2c(C)nc[nH]2)=O)CCCC(C2CCN(C(c3cnn(C)n3)=O)CC2)CC1 c1(C2N(C(c3c(C)cns3)C(=O)NCCC3(C)CC3)CCC2)cccc(Br)c1C C1(CNC(c2n(CC)ncc2)=O)CCC(NC(c2ccc(C)cc2)=O)CC1 N1(C(CC2(NC(C)=O)CC2)=O)CC2CCCN(C(C3CCCOC3)=O)C2C1 C1(C(N(CCCO)CC#C)=O)CCCN(C(c2cccc(CO)c2)=O)CC1 c1(C(N(CC(=O)NCc2c(CC)nn(C)c2)C)=O)cnn2c1CCC2 Cc1cc(C(N2C3CCC2C(NC(C2CC4C=CC2C4)=O)C3)=O)ncc1C(F)F c1(C(=O)OC)cnc(NC2CCN(C(=O)CC34CCCC3C4)C2)c(C)c1 c1(OCC(=O)NC2CC(NC(c3nccs3)=O)C2)ccc2c(c1)CCC2 c1(C(N(C2CCN(C(C3CC4C=CC3C4)=O)CC2)CCOC)=O)ccnc(Cl)c1O Cc1nn2ncccc2c1C(=O)NCC1C2CN(C(C3CC(F)C(=O)N3)=O)CC12 c1(C(=O)OCC)cccnc1N(CCCCCNC(C1CCC(F)C1)=O)C N1(C(c2c(C)cnnc2)=O)CCC(C(=O)Nc2ncccc2F)C(O)C1 CC1(C)CC(COC(c2cnc3n2CCCC3)=O)NC(=O)N1 Cc1cc(C(=O)NCC2CN(C(=O)C(C)C3CCCC3)CC2C)c(F)cc1N N1(C(C2CCCCCS2(=O)=O)=O)CC2CC(C1)N(C(=O)Cc1ncncc1Cl)C2 C=CCC(C)C(=O)NC1(CNC(c2ccc(NC)cn2)=O)CC(OC)C1 S(=O)(=O)(c1cc(C)cc(Br)c1)NC1C(C(=O)Nc2cc(SC)ncc2)C1 C=CC1(NC(=O)CC2(C)CCN2C(=O)Cc2sccc2C)CCOCC1 n1(C(C)C)cnnc1CSCC(=O)N(CCCCNC(=O)CC1CCC(C)O1)C N1(C(CC(C)c2ccccc2)C(=O)NC2CCC2)CCC(C2CCOC2)C1 C1(CNC(=O)COC(F)F)CC2(C1)CN(C(=O)CN1CCSCC1)C2 N1(C(C(C)OCC)=O)CC2CC2(C(=O)N(CC(O)CO)C(C)C)C1 C1(C(N(C(CC)CSC)C)=O)CCN(C(=O)C2=COCCC2)CC1(C)C c1(C(=O)NCC2C(C(N(C(CC(C)C)C)C)=O)CCO2)cnccc1C#N C(=O)(C(O)CCC(C)C)NC1C(CNC(CCCCOCC)=O)CC1 N1(C(C2C(C=C)CC2)=O)CCS(=O)(=O)C(CCNC(=O)CC(C)(C)C)C1 C1(NC(c2cnn(CCF)c2)=O)CC2(C1)CN(C(=O)C(C1CCC1)C1CCC1)C2 c1(NC(C2N(C(Cn3c(C)ncc3)=O)CCOC2)=O)c(Cl)cc(F)cc1Cl C=C1CC2(C1)C(=O)NCCCOCC(=O)N2.C1(C(N)=O)COCC1NC(=O)OC C(C1CCCCCC1)=CC(=O)N(C)CC1N(C(C2CC(CC)(CC)C2)=O)CCC1 Cc1cc(C(=O)NC2CCC(C)(CNC(=O)C3=CSCS3)C2)cc(C)c1Cl N1(C(c2cncc(C#C)c2)=O)CC2CC(NC(=O)COc3ccsn3)CC2C1 Cc1ncc(Br)c(C(=O)NCCCNC(=O)C(n2cc(Cl)cn2)C)n1 C1(C(N2CC(NC(C)=O)C2)=O)C2CCC(C2)C1NC(=O)C(C)N(C)C(C)=O CN1CC(NC(=O)C(c2ccccc2)NC(c2ncc(F)cc2F)=O)CCC1=O N1(C(=O)NCCC2CC(C)(C)OCC2)c2ccccc2NC(=O)C12CCCC2 C1(C(=O)NCCOC(C)(C)CNC(C2CC(O)CN2C)=O)(OC)CCCOC1 c1(OC(C)C)ccccc1C(=O)OCc1cn(CCSc2ccno2)nn1 c1(C(=O)NC2CC(F)(CNC(c3cc(CCC)[nH]n3)=O)C2)cccc(C)c1CC N1(c2nc(C)cc(OC)n2)Cc2ccccc2CC1C(=O)Nc1cc(F)ccn1 CN1C(=O)CCCc2occ(C(=O)NCC34CCC(CF)(C3)OC4)c21 C1(C(N(C(C(=O)NC(CCC(C)C)C)C2CC2)C)=O)CCCCC(=O)N1 c1(C(=O)NC(CCN(C(c2cncc(C)n2)=O)C)C)cc(Cl)nnc1O N1(C(CC=CC=C)=O)CC(NC(c2ccnc(C)n2)=O)C(c2ccccc2)C1 C1(NC(C2CC3CCC2O3)=O)CCCN(C(C2(CO)CC2)=O)CC1 N1(C(c2cncc(F)n2)=O)CCC(N=c2nc[nH]c3[nH]c(Cl)cc23)C1 c1(CCC(N2CCC(NC(CC(C)(C)F)=O)C2)=O)cccc2cnccc12 c1(C(=O)NC2C(C)CN(C(c3cc(C(N)=O)[nH]n3)=O)C2)cccc2c1OCO2 C1(C)(C(N2CC(C(C)NC(c3cc(OC)n[nH]3)=O)C2)=O)COC(C)CO1 C1(CNC(C2(OC)CCC2)=O)CCN(C(=O)CCc2c(C)nn(C)c2C)C12CC2 C1(COC)(CNC(C2CCOC2C)=O)CCCN1c1ccc(C(F)(F)F)nn1 C1(C)(NC(c2ccc(NC(C)=O)s2)=O)CCN(C(=O)CC2SC(=N)NC2=O)C1 C12(CNC(C(CC3CC3)OC)=O)CCCC1CN(C(c1ccc([N+](=O)[O-])[nH]1)=O)C2 C1(C(=O)N(CCC(C)C)Cc2cccc(C)n2)(OC)CCN(Cc2cccs2)CC1 Cc1nonc1CC(=O)NCCCCCNC(=O)CCc1nncn1C N1(C(C(F)=CC)=O)CCC2(CC1)C(OC)CC2NC(=O)C1=CCC(C)(C)CC1 N1(C(CCC=CC)=O)CC2CCCCN2CC1CNC(c1cc(C2CC2)on1)=O c1(C2N(C(=O)NCC3C(C(C)C)OCC3)CCC2)nc2cc(Cl)ccc2o1 C1(CN(C(c2c[nH]c(=O)cn2)=O)CC)CCN(C(=O)CC2CCC(=O)N2C)CC1 C(=O)(C(CC(C)C)OC(C)=O)NCCC1(C(=O)NC(c2ccnn2C)CC)CC1 C(=O)(C(F)CC(C)(C)NC(=O)CC(C)(C)C)NC(C(CCC)C)C c1(CC)cc2c(NC(CNC(=O)C(C)CC(C)(C)C)CC)nc(C)nc2s1 O(NC(=O)C(C)(C)C(C)NC(=O)C(C)S(N)(=O)=O)CCCC CC1(C(=O)NC23CC2CN(C(c2nnn(C(C)(C)C)n2)=O)C3)CC2(CCC2)C1 C(=O)(CCCCCC#N)N1CCN(C(c2c(CC)nc(C)o2)=O)CC1C(C)(C)C C#Cc1ccc(C(=O)NCC(O)CN(C)C(C2CC(CC(C)(C)C)C2)=O)cc1Cl C1(C(N(C2CCSC2)CC)=O)CC2CCC(C1)N2C(=O)CN(C1CCOCC1)C C(=O)(C(C(C)(C)C)OC)N1CCCC(N(C(Cc2nc(CC)sc2)=O)CC)C1 N1(C(c2cc(F)cnc2O)=O)CC2CN(C(=O)C(F)C3CCOC3)CC2C1 CCCC(C(=O)NC(C)CC1CN(c2ncc(Br)cc2C#N)C1)S(N)(=O)=O Cc1nc(N2CCCCC2CNC(c2cnoc2CC(C)C)=O)c(F)c(C)n1 c1(NCC(=C)Cl)ccc(S(=O)(=O)N2CCN(CCC#N)CC2)c(Cl)c1 C1(C(N2CC3(CN(C(=O)CCC(F)F)C3)OCC2)=O)CC12CCc1ccccc12 C1(CC(C)NC(C2C(C)C(=O)C2)=O)CCN(C(C23CCC(C2)C3)=O)CC1 N1(C(C(C(CCc2nc(C)sc2)=O)CCCC)=O)CC(O)CC1COC CC(C)(CC(=O)NCC(C)(C)C#CC(=O)N(CC(F)F)C1CC1)C(F)F C1(NC(c2cc(-c3ccc(C)cc3)no2)=O)CC(C)CN(C(C2(O)CCC2)=O)C1 CCCCCCCCC(C)CC(=O)NCC1OCCC1C C1(CNC(Cn2c(C)ccc2C)=O)CCC(C)N(C(=O)CCC2CCC(=O)C2)C1 C1(C(=O)NCc2cn(CC(=O)O)nn2)CC(=O)N(O)C1 c1(C(N2C(C(N3CC(N4CCOC4=O)C3)=O)C=CC2)=O)ncc2ccccn12 C1(NC(c2ccn(C3CC3)n2)=O)CN(C(c2cn3c(n2)CCC3)=O)C2(CCC2)C1 N1(C(CC(C)NC(c2sccc2CO)=O)=O)CCC2(C1)CN(C)C2 Cc1ccc(=O)n(CC(N2CCC(C)C(NC(C3CC(C4CC4)=NO3)=O)C2)=O)n1 C(c1cc[nH]c1)=CC(N1C(CNC(c2cnn(C3CCOC3)n2)=O)CC1)=O Cc1onc(Cl)c1C(N1CCC(CNC(=O)C(c2ccccc2)O)CC1)=O c1(C(=O)NC(CNC(c2n(C=C)nnc2)=O)C2CC2)cccc(Cl)c1Cl N1(C(C2CCC(=O)N2)=O)CC(NC(=O)CN(CCO)CCO)CC2(CCC2)C1 N1(C(C2C(C=C)CC2)=O)CCCC(C)(CNC(c2ocnc2C2CC2)=O)C1 Cc1ccc(CCN(Cc2ccc(C3OCCO3)cc2)Cc2cccs2)nc1 C(N=c1[nH]c(C(N2CCC(N3CCCC3)C2)=O)cs1)c1c(C)cco1 C1(C(=O)NC(CN(C(C(CC)n2cccn2)=O)C)(C)C)C2CCCOC12 C(CC(C)(C)CC(=O)N1CC2CCC(CNc3cc(O)nc(O)n3)(C2)C1)OC C(=O)(CC(O)C(C)CC)NCCCOCCC(=O)NC(CC=C)CC(=O)OC Cc1cc(O)c(C(N2CCOCC2CNCc2c(F)ccc(Cl)c2Br)=O)cc1Br Nc1cccc(Cl)c1C(N1CC(N2CCCC2)C(F)C1)=O c1(OC)nccc2c(NC(=O)NC3(CO)CCSC3)c[nH]c12 n1(C(C)C)cnc2c(NC(C)CN(C)C)nc(N3CC(=O)NC(C)C3)nc12 N1(C(C2CCCN(CC)C2)=O)CCC(NC(=O)CSCCC(C)C)C(F)C1 C12(NC(c3c(C)oc(C(C)C)n3)=O)CCCC1CN(C(=O)C(C)N(C)C)C2 c1(CC)ncccc1C(=O)NC1CCC1C(N1CCC(CN2CCCC2)C1)=O c1(C(N2CCC(O)(CC(=O)OC)C2)C(=O)NCCC)ccc2c(c1)CCC2 N1(C(CNC=O)=O)C2CCC1CN(C(c1ccc(-c3nnc(O)o3)cc1)=O)CC2 c1(C(N2CC3(CCN(C(c4ccns4)=O)C3)C2)=O)nc2n(c1Cl)CCCC2 C1(C(=O)NCC(C=C)C)CC2CC1CC2O C1(C(N(CC(C)N(C(Cc2c(C)n[nH]c2)=O)C)C)=O)CCc2cc(F)ccc2O1 C1(NC(CC2N(C(CCC#C)=O)CCC2)=O)CCN(C2CC2)C1=O Cc1cc(Br)ccc1C(=O)NC1CC(CNC(=O)CN(C)C(C)C)C12CCC2 C(=O)(C(C)CC(C)(C)C)NCc1c(C(N2CCC(C(=O)NC)C2C)=O)n(C)nc1 N1(C(C(CC)OC(C)=O)=O)CCCCC(CNC(=O)C(C)(C)COCC(F)F)C1 C1(C)(C(=O)NCCc2ccc(C)nc2)CC(O)CN1C(c1nc(C)c(C)s1)=O Cc1nc(NCCC2(CO)CCCC2)cc(N2CCCC(N(C)CCO)C2)n1 C(CC(C(C)C)NC(C1CC1c1ccc(F)cc1)=O)N(C(C1C(C)=CCS1)=O)C C1(C(=O)NC(C2CCCC2)C)CCCN(CC=Cc2ccccc2)C1 C1(NC(Cc2cn(CC)nc2)=O)CN(C(C2CCCC2O)=O)C2CCCC12 C1(C(N(C(C)CC(C)C)CCOC)=O)CC(NC(=O)CSC)C(O)C1 C1(C(N2C(CNC(CC(C)(C)SC)=O)CC(F)C2)=O)COc2ccc(Cl)cc2C1 C1(NC(c2c(C)csc2)=O)CC2(CCN(C(c3nc(C)c(C)[nH]c3=O)=O)CC2)C1 C1(CNC(C(C(C)C)OC)=O)CN(c2nccc(CO)n2)CCCO1.C1C(=O)N1 C=C(C)CCC(C)NC(C1(C)CCN(C(=O)CSC)C1)=O c1(C(N(CC(CN(C(=O)CC2CCC(=O)N2)C)O)C)=O)cnn(C)c1Br C1(NC(c2csc(C)c2N)=O)CCN(C(c2cc(O)nn2C)=O)CC1(C)C c1(C(N2C3C(NC(c4n(CC)ncn4)=O)CC(C3)C2)=O)nc2cc(F)ccc2s1 c1(C(=O)NCC(CNC(C(C)c2ccsc2)=O)F)scnc1C1CC1 c1(C(=O)NC(CCOC)CNC(=O)C(CC(C)C)N(C)C)cnc2c(c1)COC2 N1(C(c2cc(CC)on2)=O)CC(NC(=O)C=Cc2ccncn2)C2CC12 Cc1cn(C(C)C)cc1C(N1CCCC1CNC(C1(OC(C)C)CCOC1)=O)=O c1(OC)ccc(C(N2CC3CC3(NC(c3cnn[nH]3)=O)C2)=O)c(Cl)n1 c1(C(=O)NC2C(CNC(CC(C)C(F)F)=O)C2)cc(=O)c2ccccc2n1C c1(CN2CC(F)CC(C(=O)N(CCO)CCO)C2)ccc(F)c2ccoc12 N1(C(C(C2CCC2)OCC)=O)CC2OCCN(C(c3ccc(N)cc3Cl)=O)C2C1 n1(CC(=O)NCC(C)(C)NC(C(C)C2CCCC2)=O)cc2ccccc2n1 c1(C(=O)NCCCN(C(C2CC(F)C2)=O)CC)ccnc(OC(C)C)c1 C1(CNC(c2cc(COC)no2)=O)CN(C(=O)C2=CCC2)CC1C C1(C(N2CC3CCOC3C2)=O)(CC)CCCN(C(=O)C=CC(F)F)C1 N1(C(C2CC(CC)C2)=O)CCN(C(c2cc(Br)sc2C)=O)CC1C N1(C(c2cc(C)no2)=O)CCC(C(C)(C)CNC(C2(CO)CCCO2)=O)CC1 C1(N(C(CSCCC)=O)C)CC2CCC(C1)N2C(C1(C)CCC(C)=C(C)C1)=O CCCC(C(=O)N(CC(=O)Nc1cnc(C)nc1)CC)NC(N)=O c1(CC(C(=O)NCC)OC(=O)CNC(c2ccon2)=O)cccc(C(=O)O)c1 N1(C(C(c2ccoc2)NC(=O)CC2(O)CCCCC2)=O)CCC2(CCCCO2)C1 N1(CCc2scc(CC)n2)C(=O)NC2(CCS(=O)(=O)CC2)C1=O c1(C(=O)NC(c2nocc2C(=O)NCc2nncn2C(C)C)C)cc(=O)cc[nH]1 c1(C(=O)NC2CCCCN(C(C(C)C3CCOC3)=O)C2)nc2cccnc2s1 CC1(F)COCCN(c2cc(NCCC3CC3)nc(C(=O)O)n2)C1 C1(C(N(c2cnn(C)c2)CC)=O)CCN(C(=O)CCc2cnc(C)o2)CC1 c1(OC)c(O)cc(C(N2CCC(C(N3CCOC(C(C)C)C3)=O)C2)=O)cc1O c1(C(C(=O)NCCSC)N(C)CC)cnccn1.c1ncc(C(N)=O)s1 c1(OC)ccc(F)c(C(=O)NCC2C(C)CCN2C(c2cc(C)ccn2)=O)c1 S(=O)(=O)(c1cccs1)NCC(N1CCC(O)(Cn2cc(-c3cccs3)nn2)C1)=O N1(C(c2c(OC)nn(C)c2)=O)CCN(C(c2ccns2)=O)CC1c1cnn(C)c1 N1(C(C2C(C(C)=O)C2(C)C)=O)CC(C(N2CCC(C#N)CC2)=O)C(C)(C)C1 C#CC1(C)CCCN(C(=O)CC2CCCN(C(=O)CCC(C)(C)OC)C2)C1 Cc1ccc(-c2nc(C3CCC3)nn2C)c(C(F)(F)F)c1 CCC(C)C(O)CNC(=O)CCCNC(C1(CC(C)C)CCC1)=O c1(C(N(CC)CC2CCCN2C(=O)C(CC2CC2)OC)=O)nccnc1OC C1(COC(CN(C(C)=O)C(c2csnc2Br)=O)=O)CCCC(CF)C1 C1(C)(C(=O)NC2CN(C(c3c(CC)occ3C)=O)CC2F)CC(C2CC2)=NO1 Cc1ccc(S(=O)(=O)N(c2nccc(C3CC3)n2)C2CNCC2F)cc1C Cc1nccc(Br)c1NC(C1CC(O)CCN1c1nccc(C(F)F)n1)=O N1(C(CC(=C)C)=O)CC2CCC(C1)N2C(c1cnn(C(C)(C)C)c1Br)=O C(C)(CC(C)N=c1nc(C2CC2)[nH]s1)NC(C(C)=C1CCC1)=O N1(C(C(CC)CC)=O)CC2CCCCC2(CNc2ncnc(C)c2F)C1 N1(C(C(C)Oc2ccccn2)=O)CCC(C)CC1CNC(c1c(Cl)nn(C)c1Cl)=O CCCCC(O)C(C)C(=O)NCC(C)NC(=O)C(C(C)C)N(CC)CC N1(C(c2n(OC)cnc2C)=O)CCC(C2CC(NC(c3cnc(O)n3C)=O)C2)C1 C1(CC(=O)NC(C2(O)CN(C(C3CCN3C(C)(C)C)=O)C2)C)CCCCC1 N1(c2n(CCOC)c(-c3cc[nH]n3)nn2)CCC2C(C1)C2(F)F c1(CC)cccc(CNC(=O)C(Cc2cnc[nH]2)NC(c2cc(Cl)cs2)=O)c1 c1(C(N(C2CCN(C(=O)COCC3CC3)C2)CC)=O)cc2ccccc2s1 n1(CC)c(C)cc(C(N2CCOCC(NC(=O)C#CC3CC3)C2)=O)c1C C1(CNC(CN2C(C)CC2)=O)CC12CCN(C(=O)COc1ccsn1)CC2 c1(C(=O)NCC(CC(C)C)NC(=O)C(F)C(F)(F)F)cc2c(cc1Cl)CCCC2 CC(C)CC(C(=O)NC1CCCC1NC(c1ccc(Cl)[nH]1)=O)C(C)C c1(C(=O)NCC(CC=C)NC(=O)CC2CC3CC3C2)c(C)ccc(C)c1N C12(NC(CC=C(C)C)=O)CCCC1N(C(c1cc(C(N)=O)ccc1O)=O)CCC2 CC(CC(=O)N1CC(C(=O)NCc2nc(CO)n[nH]2)CC(C)C1)C(F)F N1(C(C=CC)=O)CCN(C(=O)CCC(=O)N(C)C(c2ccccc2)C)C2CC12 C1(CNC(CCC2C(C)C2)=O)C(C2CC2)CCN1C(c1cc[nH]c2nccc1-2)=O N1(C(c2nn(CC)c(C(F)(F)F)c2)=O)CC(CNC(c2cnsn2)=O)CCC1C c1(C(N2CC(NC(C3(CO)CC3(F)F)=O)C(F)C2)=O)c[nH]c2cccc(Cl)c12 Cc1nc(OC(C)C)ccc1C(=O)O.C1(=O)CC2(CC2)N1 C(C(=O)NCC1CCOC1)(C1=CCCCC1)N1C(c2onc(C)n2)CCCC1 Cc1cnc(NC(C2CCCCN2C(=O)Cc2ccc(Cl)s2)=O)c(Cl)c1 C(CCN=C(NCC1(C)CC1)NC(C)C)(C1CCCC1)OCC C(=O)(C(Cc1cc[nH]n1)NC(=O)CSCCC#N)N(CC(C)C#N)C c12cnc(cc1C)NC(=O)C2N(CCCCC)C.c1(C(=O)OC)ccccc1 c1(C(=O)NCCC(CC)(C)NC(c2ncnc(C)c2C)=O)ccc2nc[nH]c2n1 c1(C(=O)NC2CCN(CC)C2)cc(-c2nn[nH]n2)cc(O)c1 C1(C(=O)NCC=CCNC(C(C)NC(c2ccoc2)=O)=O)CC2CCC2C1 C=C1Cn2c(C(=O)NCC3CC(NC(c4cc(C)[nH]n4)=O)CC3O)nnc2S1 c1(C(N(CCC(=O)N(CCC#C)C)C)=O)cncc(Cl)c1 Cc1ccc(C)c(-c2cc(NC(=O)NC3CCC(O)CNC3)no2)c1 N1(C(C2N(C(C(CCCC)F)=O)CSC2)=O)CCCC2C(O)CC12 NC(=O)CCC(=O)NCC1CCCC1NC(=O)CN1CCCCCC1 C1(c2cn(C)nc2)CCCCN1C(c1c(I)cnn1C)C(=O)NC1CC1 c1(NC(c2ncc(-c3c(C)ccs3)s2)=O)cc(C(N)=O)n(C)n1 N1(C(C2(OC)CC(C)C2)=O)CC2C=CC1C(C(N1CCC3C(C(N)=O)C3C1)=O)C2 c1(C(=O)NCC2CCC(NC(C=CCN)=O)C2)noc2c1CCCC2.CC(C)(C)OC c1(C(N2CCC(N(C(=O)C3=C(Cl)CCC3)CC)C2)=O)ncc([N+](=O)[O-])cc1C C(=O)(CCC(C)(C)C)N1CC(O)(C(C)NC(C2CCC(F)(F)C2)=O)C1 N1(C(CC2(C)N(C(C3(CC(=O)OC)CC3)=O)CC2)=O)CCC(F)(F)CC1C c1(C(N2C(C)(CNC(=O)C(F)C3CCC3)CCC2)=O)cc2ccccc2nc1F C1(CC(=O)N(C)CC2(CNC(=O)Cc3ccc(Cl)s3)CC2)CC(O)C12CCC2 Cc1ccncc1CC(=O)N(C(C)CO)CCC1CC1 Cc1cc(Cl)cc(C)c1OCC(=O)NC1CN(C(C2CC(C)(O)C2)=O)C1 N1(Cc2cc(C)cc(O)c2)CCC(F)(F)C(C(=O)NCc2ccnc(C)c2)C1 c1(C(=O)NCC(CCOC)NC(c2cccnc2OC(C)C)=O)ccc(C)nn1 CC(C)C(C(=O)N1CCN(C(c2cc[nH]n2)=O)CC1c1ccnn1C)C(C)C Cc1c(C(=O)NC2C3CC(NC(C4C5CCCOC45)=O)CC23)cncc1F c1(C(=O)NC(C2(CNC(C3CC4(C3)CC4F)=O)CC2)C)cn(C)c(=O)n1C C1(C(C)N)CN(C(c2coc(C3CCOCC3)n2)=O)CCO1 N1(C(C=CCN(C)CC)=O)CC2CCC1C1CN(C(=O)C#CC(C)(C)C)CC21 c1(CC)c(C(N2CC(C)(NC(=O)CNC(c3ccoc3)=O)C2)=O)ccn1C c1(C(CC)(C)C)cn(CC(C2CN(C(=O)NC3(Cl)CC3(C)C)C2)F)nn1 Cc1cccn2ncc(C(=O)NC(C)(C)CCNC(c3cnc(C)n3C)=O)c12 c1(C(=O)NCCC(C)NC(c2cnn[nH]2)=O)cccc(-c2cc[nH]n2)c1 c1(C(=O)NC2CCCC2SCCCO)cnc(C2CC2)nc1 N1(C(c2nc(C)[nH]n2)=O)CCOC(C(C2CC2)NC(=O)COCc2cccnc2)C1 C(=O)(C1=Cc2ccccc2C1)NC(CC(=C)C)C(=O)NCc1noc(C(C)C)n1 c1(C(N2C3C(NC(CCN4CCC(C)CC4)=O)C(C3)C2)=O)ccc(C#N)c(F)c1 N1(C(C(C)NC(CC)(C)C)=O)CC(C(=O)NCCNC(=O)NC)CCC1C c1(NC(N2CCCC(CN(C)CO)C2)=O)cc(CC2NC(=O)NC2=O)ccc1Cl C(=O)(CCCCC(=O)N1CCN(C(c2cnc(C(F)F)cn2)=O)C2CC12)OC Cc1scnc1C(=O)N(CC(O)CN(C(=O)CC1CC1C(F)(F)F)C)C Cc1noc(C(=O)N(CCCNC(C2CC2F)=O)Cc2ccccc2)c1C C(=O)(CC(C(F)F)C(C)(C)C)N1CCCC(O)(CN(C(=O)CNC=O)C)C1 c1(C(=O)NC(C)(C)CNC(C2(CC3CC3)CCCO2)=O)cc(Cl)cnc1O CC1CC(N=c2nc(O)c3cnn(C)c3[nH]2)CN1C(=O)CCC(F)(F)CN=[N+]=[N-] c1(C(N(CC(CNC(C=C(COC)C)=O)C)C)=O)cc(C(=O)C(F)(F)F)c[nH]1 C1(O)(CN(C(=O)C(C)(C)N2CCCCC2)C)CCCN(C(C2CC2(C)C)=O)C1 CCC(C)CCCCC(=O)NCCC(C)NC(C1(C)CC(OC)CN1C)=O C=C(F)C1(CC(N2CC(O)(CNC(=O)COC(C)CC)C2)=O)CCOCC1 C(=O)(CCCCC(=O)NC(C)CNC(c1cncc(Cl)c1Cl)=O)NC c1(CN2CCC3(C(C(N4C(C#N)CC(F)C4)=O)C3)C2)ccc2nonc2c1 C1(CNC(CC(C)N(C)C)=O)CN(C(=O)CC2CCCCCCC2)CC(C)(C)O1 c1(C(=O)NCCC(=C)CNC(=O)C=CC2CCCCC2)[nH]nc(C)c1Cl c1(CC(=O)NCCNC(C2C(COC)CC2)=O)cc(OC)ccc1OC N1(C(C(C)NS(CC)(=O)=O)=O)CC2CC2(CNC(c2ccc(N(C)C)cc2)=O)C1 c1(C(CC)O)nc(-c2ccnn2C(F)F)n(-c2cccc(Br)c2)n1 c1(Cn2cc(CC(CC)(C)O)nn2)cccc(CNC(=O)C(F)(F)F)c1 N1(C(CC=CC=C)=O)CCC(C2CCC2)(CNC(=O)C(C)O)CC1 C1(NC(C(C)(C)CC2CC2)=O)CCN(C(C2CC3(CCC3)C2)=O)CC(O)C1 c1(C(N2CCOCC(NC(C3CC3[N+](=O)[O-])=O)C2)=O)cc(F)cc2ccccc12 C1(N(C)C(c2cc[nH]n2)=O)C2CN(C(C3(C)CC3Br)=O)CC12 c1(SCCCCCC)ccc(NC(=O)C(N2CC(O)(c3cscc3Br)C2)=O)cc1 C(=O)(C(F)C(CC)CC)NCC1CCN(C(CCCOCC)=O)CC1O CC1(C)CCC1CC(=O)NC1(C(=O)NCCNC(=O)CC2CCCOC2)CCC1 c1(CNC(C2CN(C(c3ncn(C)c3C(F)(F)F)=O)C2)=O)ccc(F)nc1F Cc1cccc(OCCCNCCCOC(=O)C(C)Oc2cccc(F)c2)c1 c1(CC)ccc(OCC(N2CC(NC(c3cc(C)nn3CC)=O)C(C)C2)=O)cc1 N12CC(CC(C)C1)C2=O.c1(CC)n[nH]cc1C(=O)NC1(C(O)CO)CC1 C(=O)(CC(C)(F)F)NCC(C)(C)CNC(=O)C(C1CCCO1)C1CC1 N1(C(CC(CC)N(C(=O)C(O)CSC)C)=O)CC2(CNC(=O)N2C)C1 C1(C(=O)NCCn2c(CSC)ncc2)CN(C(C2(O)CCOC2(C)C)=O)CC1(C)C CCC(C)(CNC(C1CCOC(C)(C)C1)=O)C(=O)NCc1ncccn1 CP(C)(=O)C1CCCC=C1C(=O)NC1CC(=O)N(CC2CCCCC2)C1 C(Cc1ccc(C)cc1)(CC(=O)O)NC(CCCOCCC)=O c1(COC)nc(C)ncc1C(N1C2CCC(C2)C1CNC(=O)C(C)SC(C)C)=O N1(C(c2c(C)cc(OC)nc2)=O)CCC2CN(C(C3CC(=O)N(C)C3)=O)CC2C1 c1(C(N(CC(C)NC(=O)CS(=O)(=O)NC(C)(C)C)C)=O)cccc(O)c1[N+](=O)[O-] N1(C(Cc2c(C)noc2C)=O)CC(NC(=O)C2=CC(O)CCC2)C(N=[N+]=[N-])C1 C1(CNC(COCc2cccc(OC)c2)=O)CCN(C(=O)C(C)N(C)C)C1(C)C N1(C2CCN(C(c3cnc(CC)s3)=O)C2)CCC(N=c2[nH]nc(COC)s2)CC1 N1(C(C(CC)OCC)=O)CCCC(CC)(NC(c2ccccc2F)=O)C1 C12(COC)CC(CNC(C3CCN(C)C3=O)=O)(CN1C(c1nccnc1N)=O)C2 C1(CNC(c2n[nH]c3c2COC3)=O)CN(C(c2ccccc2)=O)CCCO1 C1(CNC(c2n(CC)cnn2)=O)C2CCCC1N(C(C1CC=CC1)=O)C2 CC1(CNC(=O)C(Cn2cncn2)NC(=O)COC2CC=CC2)CCCC(=O)N1 c1(C(=O)NCC2C=CC(NC(c3cnc(CC)s3)=O)C2)nc(C)c(C)nc1C C(=O)(CCN1C(=O)CCc2ccccc21)NCC(CO)NC(C1=NOC(C)C1)=O c1(C(=O)NC2CCN(C(CC(CC)SC)=O)CC2)cc2ccc(F)cc2s1 c1(NC(Cc2cc(CC)no2)=O)ccc2c(C)cc(C)nc2n1 c1(C(=O)NC(CC)(CNC(=O)CC2CCCC(OC)C2)CC)ccc(N)c(O)c1 Cc1noc(C2CC2NC(=O)CNC(=O)CNC(=O)C(N)=O)n1 c1(C(=O)NCC2(OC)CN(C(c3cnsc3C)=O)C2)cnc(O)c(F)c1 C1(C(=O)OCC)CCN(C(C23CCCCC2C3)=O)CC1C1CC1 c1(C(=O)NC2(C)CCN(C(c3cc(Br)no3)=O)C2)cccc(C#N)c1 c1(C(=O)NCC2(CCNC(=O)COc3cn[nH]c3)CC2)ccnc(F)c1F N1(C(C(c2ccccc2)OCC)=O)C2CCCC1CC(NC(C1CC1CC)=O)C2 N1(C(C2CC(OC)C2)=O)CCC2(C1)CN(C(C1CC=C(C)CC1)=O)CCO2 C(CC)(CS(=O)(=O)c1ccccc1)NC(=NCC)NCC(C1CC1)C1CC1 C1(C(=O)NC2CC(NC(c3n(C)c(C#N)cc3)=O)C2)CC2CC(O)C(C1)C2 C1(NC(c2nc(CC)oc2)=O)CC2CCC(C1)N2C(C1CC1c1cccs1)=O Cc1ccc(Br)c(C(=O)N(C2CC(NC(c3sccc3C3CC3)=O)C2)C)c1 C1(CNC(CCC=CCC=C)=O)CCC2CN(C(c3ccon3)=O)CC12 C1(CNC(CSCC#C)=O)Cc2ccccc2CN1C(=O)C(C)(C=C)CC C(CCC[Si](C)(C)C)N(CC#CC(OC)OC)C(c1ccc(Cl)s1)=O c1(C(=O)NC(C(CO)NC(CN(C2CC2)CC)=O)C)cccc2ccccc12 c1(C(C)(C)C)nc(=N)[nH]c(=NCCC2CCN2C(=O)Cc2nc(=N)[nH][nH]2)[nH]1 c1(CCC(=O)NCCN(C(C(C)(C)C2CC2)=O)C2CC2)cccc(Br)c1F N(C(=NCCCn1ccnn1)N1CCC(c2cc(OC)ccn2)C1)CC(=C)C N1(C(CN(C(C(C=C)OC)=O)C)=O)CCS(=O)CC1 c1(C(=O)NCCc2c(C)cccn2)nc2n(c1Cl)CCN(C(=O)CCBr)C2 Cc1ccc(C(N2CC3(CC3)CC2CNC(C2CCCS2)=O)=O)cc1C c1(OC)ccc2c(c1)CC(C(=O)NC1CC1NC(c1csc3cncn13)=O)O2 C1(C(N(CCCC(=O)NC(C#C)C(C)OC)C)=O)CC(=O)NC1(C)C C1(C(=O)NCCCNC(c2n(C)c(=O)ccc2)=O)CCN2CCOCC12 c1(NC(c2ccc(CCC(=O)NC(c3cccs3)CC)[nH]2)=O)cc(F)ncc1C N1(C(C2CCC(CC(=O)OC)CC2)C(=O)NCCOC)CCn2ccnc2C1C C1(N(C(C(CC)COC)=O)C)CN(C(c2nc(C)oc2OC)=O)CCC1O C(=O)(C1CCc2nccn21)N(C1CCCN(C(c2c(N)cn(C)n2)=O)C1)CCF N1(C(=O)NC(C2CCCCC2C(F)(F)F)CSC)CCN(c2cnccn2)CC1 N1(C(c2cn(CC)nc2)=O)CCC(C)C(NC(c2cc(NC)ccc2O)=O)C1C C1(NC(=O)CCc2nn[nH]n2)CCCC(c2ccccc2)C1 c1(C(C(=O)NCCCCCC)N(C)Cc2cnn(CCOC)c2)cc(C)nn1C O(N1CCC(CC(=O)NC2CCCN(C(C3(NC(N)=O)CC3)=O)C2C)CC1)CC N1(C(C2N(C)CC(C)(C)C2)=O)C2CCC1CN(C(C1CC(C)(C)CN1C)=O)C2 c1(C(=O)NC(CC)(C)CNC(=O)C(C)C(F)F)cc2sc(Br)cc2[nH]1 C1(NC(CC(C)c2cccnc2)=O)CN(C(=O)CC(Cl)Cl)CC12CCC2 C1(C(N2C(CNC(c3occc3Br)=O)CCCC2)=O)CC2(CCC2)CO1 CC(C)CCCCC(=O)N1CCCCCC1CNC(c1ccc(C(F)(F)F)s1)=O C1(CC(=O)NCc2c(C)csc2)CCC(NC(=O)CN2CCCCCC2)CC1 C1(C(C2(C3CCCCO3)CC2)=O)(CNC(c2ccc(SC)s2)=O)CCOCC1.OC CCC(O)C(F)(F)C(=O)NCC12CCC(CC1)N2C(=O)CSc1ccccc1C c1(C(=O)NCC(C(C)C)NC(c2cnc(CC)[nH]2)=O)cccc(F)c1SC C(CCC(C)(C)C(=O)N1CC2(CC(CO)CO2)C1)NC(C(C)S(N)(=O)=O)=O c1(C(=O)NC(C2OCCN(C(C3C(=C)CC3)=O)C2)C)ccnc2c1ncn2C Cc1cc(C(=O)NCC2CN(C)CCN2C(=O)C#CC(C)C)ccc1Cl C12(CNC(C(Cc3ccoc3)NC(CC(C(C)C)C)=O)=O)CC3CC(CC1C3)C2 CN1C(=O)OCC1C(N1CCN(CCNC(c2ncncc2Cl)=O)CC1)=O c1(C(=O)NC(CN(C(C23CCC(OC)C2CC3)=O)C)(C)C)ccc2c(c1)CCN2 c1(C(N2CC(CC)N(C(=O)C(CO)OC)CC2)=O)cc2c(C)cccc2o1 C1(CNC(C(n2ccc(Br)n2)C)=O)CN(C(C2CC(C)(C)C2)=O)C(C)(C)C1 CC1=C(C(=O)N2CC3(CCCC3)C2C(N2CCCC(F)(CO)C2)=O)COCC1 C1(CNC(c2n(CC)nnc2)=O)CCN(C(c2nc(Cl)cs2)=O)C1(C)C CC(C)CC(CNC(c1cnsc1)=O)NC(C1(c2cccc(Cl)c2)CC1)=O C1(CNC(C(C(C)C)O)=O)CN(C(c2cc(CCCO)on2)=O)CCC1(C)C c1(C(N(CCC(C)NC(=O)CC2CCC=CCC2)C)=O)ccc(=N)[nH]c1 C(c1ccc(C)cc1)=CCC(=O)NC(CC)(C)CCNC(C1OCCC1(C)C)=O CC1(C)CCCN(C(C2CC23CCSCC3)=O)C1CNC(c1ccc(O)cn1)=O c1(C(=O)NCC#CCNC(C2C(C(=O)OC)C2)=O)n[nH]c2nccc(Cl)c12 c1(NCC)cccnc1C(=O)NC(C)CC(C)NCC(C)(C)CNC C(=O)(N=c1ccn(CCS(C)(=O)=O)[nH]1)N1CCC(CC#C)C1 c1(C(C)(C)C)cc2c(N3CC(C)CC3C(N3CCC(Br)CC3)=O)ncnc2s1 c1(OCC)ccc(NC(C2CCC(C)N2Cc2cc(O)ccc2Cl)=O)nc1C N1(C(C=C(CC)C)=O)CCN(C(=O)CC2(C)CCCO2)C(C)C1 c1(NC(c2n(CCC)ncc2)=O)ccc(CNS(C)(=O)=O)cc1.C12(O)CN(C1)C2 N1(C(COCC#C)=O)CCC(NC(c2ccc(OC(C)C)nc2)=O)C(C)C1 C(C)(C(CO)NC(C1CNC(=O)N1)=O)NC(C(C)n1cccn1)=O N1(C(c2ncc(C(F)F)s2)=O)CC2C(CN(CCO)C3CC3)C2C1 c1(C(C)C)nc(NCCN(C)C)cc(=NCc2noc3c2CCCC3)[nH]1 CCCCCCCCNC(=O)CC(CN(C)C)NC(=O)CC1CC(N(C)C)C1 C(CCCC(CO)NC(C1CCCN(CC(F)F)C1)=O)NC(CCCN(C)C)=O c1(CC)cnccc1-c1nc(CCSC)nn1CCN1CCN(C)CC1 C1(CNC(c2n(CC)c(O)nc2)=O)CN(C(=O)C(C)n2ccnc2)CC1(C)C N1(C(=O)OCC=C)CCC(Oc2cccc(C(N)=O)c2)CC1 C1(CNC(c2ccc(C(C)C)cc2)c2n(CCOC)nnn2)CCCC(C)O1 Cc1nc(CC(=O)NCC2CCN(C(=O)C(C)CC3CCCC3)CC2)[nH]c1C c1(C(=O)NCCN(C(C2C(C)(CC)C2)=O)CC2CC2)cc(C(F)F)ncn1 C1(NC(c2cnco2)=O)CCCCN(C(=O)CCc2ccc(F)c(F)c2)C1 C1(N(C(C(C=C=C)C)=O)C)CCCN(C(=O)C(F)=CC2CC2)CC1 C1(NC(c2cc(O)ncn2)=O)CCS(=O)(=O)C12CN(C(C1CCCCC1)=O)C2 Cc1sncc1C(=O)NC1CCCC1CC(=O)N(C)CCC1CCCO1 CC1CN(C(=O)CCc2nc(Br)cs2)C2(COC2)CO1 c1(C(=O)OCC23CC(C)(OCC2)C3)c(F)ccc2c1OCC2 CCC(C)(C)C(C)CC(=O)N1CC(F)CC1CN(C(=O)COCCOC)C N1(C(C2(C(=O)OCC)CC2)=O)CCC(NC(C2CC3CCN2CC3)=O)C(C)C1 Cc1ccc(C(=O)NCC(C(C)(C)C)NC(=O)CN2CC3CC3C2)cc1N C1(C(N2CCC(CCC)(CO)C2)=O)CC2CCC(C1)N2C(=O)C(=O)NOC c1(NCCS(CC)(=O)=O)ccc(S(=O)(=O)NCCOC)cc1[N+](=O)[O-] C(=O)(C(CC)CCc1ccccc1)N(CCOCCCNC(C1C(=C)C1)=O)C c1(OC)cn(C)c(C(=O)NCCCC(C)NC(=O)C2=NOC(C)C2)cc1=O C(=O)(CCC(C)N(C)C)N(C(C)C(=O)NC)CC.C1(=O)C(C(C)C)N1 N1(C(COC(CC)CC)=O)CC(O)(CNC(c2ncsc2C)=O)C1 c1(C(=O)NCCCCCN(C(=O)CCc2cccs2)C)ccc2oc(O)nc2c1 N1(C(c2cc(C(=O)OC)sc2)=O)CCC2(CC1)OCCC2NC(=O)CN(C)C1CC1 c1(C(N2C(C)CCC(NC(c3c(CC)ocn3)=O)C2)=O)cc(F)c(F)c(Cl)c1F N1(C(C2N(C(COCC#C)=O)CC2)=O)CC2CCCC(C1)N2C N1(C(C2CCC(=O)NC2)=O)CCC2CCCC12C(=O)NC1CCCOC12CCC2 C(c1nc2ccccc2o1)=CC(N1CC(OCCNC(C=CCCC)=O)C1)=O N1(C(C(C)=C2CCCC2)=O)CCCC(C(=O)NC(C)CCN(C)C)(OC)C1 c1(C2(NC(=O)NCC(C(C)C)Cc3ccccc3)CCCC2)ccc(F)cc1F C1(NC(=O)CCN2CCCC2)CC2CC(NC(=O)C(F)(F)c3cnccn3)C1C2 N1(C(c2c(CC)cco2)=O)C2CCCC1CN(C(=O)C(F)Cc1ccccc1)C2 n1(C(C)C)cc(C(=O)NC2CCC(NC(C3(CCO)CC3)=O)C2)ccc1=O C(=O)(C(CC1CCC1)NC(C1(NC(=O)CC(C)C2CC2)CCCC1)=O)OC c1(C(=O)NCCC2CN(C(C(COC)OC)=O)CC2C)cc(C#N)ccc1F N1(C(C(CSC)OC)=O)CCCC(N(C)C(c2ccn(C(C)(C)C)n2)=O)C1 N1(C(c2cccc(OCC)c2)C(=O)NC2CCC2)CC(CO)OC(C)(C)C1 C(=O)(CCCCCCCBr)N1CCC(N(C)C(=O)NCCc2ccccc2Br)C1 C#CC1(C(N2CCC(C(C)CNC(=O)C(CN(C)C)N(C)C)CC2)=O)CCCC1 C#CC1CN(C(=O)CCCNC(=O)C=Cc2cnccn2)CCO1 C1(NC(C(C=C)(C)C)=O)CN(C(C2CC3CCC3C2)=O)CC1N=[N+]=[N-] C1(C(N2CCCC(OC)C2)=O)CC12CCN(CC(=O)NC1CCCC1)CC2 C1(NC(C(C)OCCC(C)C)=O)CN(C(=O)C=Cc2ccccc2)CC2(CC2)C1 c1(OC)c(Cl)cc(-c2cn(C3(CNC(=O)CCCSC)CCCC3)nn2)cc1Cl c1(NC(C2CC(CNc3ccsn3)C2)=O)ncnc2c1ncn2CCO CCC(CC(=O)N1CC2CC(NC(=O)CN3CC(C)C3)C1C2)C(C)C c1(NC(C2CCCN(C(=O)Cn3cc(Br)cn3)C2)=O)c(Br)cc(Br)cc1[N+](=O)[O-] N1(C(C(C)=CC2CC2)=O)CCC(C(F)(F)F)C(NC(c2ncnn2C(C)C)=O)C1 c1(C(N2CC(C)C(C)(C(=O)NC(C)CS(C)(=O)=O)C2)=O)cc2cccnc2[nH]1 Cn1oc(C(=O)NCC(CO)NC(c2ccc(CSCC(F)(F)F)o2)=O)cc1=O c1(CCC(=O)NC(CC(C)NC(c2c(C)nn[nH]2)=O)C)c(F)cccc1Cl N1(C(C(CC(F)F)NC(c2cncnc2)=O)=O)CC23CCC2(COC3)C1 c1(C(N(C2CCN(C(=O)C(F)CC3CCCC3)C2)C)=O)cnc2nccnc2c1 CC(C)C(C(=O)NC1CCC(NC(=O)CC(C)(F)F)C1)c1ccccc1 c1(CC)cc(S(N)(=O)=O)cnc1SC1COCCOC1 C1(CC)(NC(c2cccc(N)c2)=O)CCCN(C(c2cnccc2N(C)C)=O)C1 C1(C(C(N2CC(=C)C2)=O)C)CCN(C(c2ccncc2)=O)CC1 C1(C(=O)NC2CCCC2(C)C)CCCC(CNC(=O)OC(C)(C)C)CC1 CCC(C)CC(=O)N(C)CCOCCCNC(=O)Cn1cc(C(F)(F)F)nn1 C=CC(CC)CC(=O)NC1CN(C(=O)C(C)(C)SC)CC1C(F)F c1(C(=O)NCC2CCCN(C(C=CSC)=O)C2)cc(OC(F)F)cc(Cl)c1 C(CCCCC(=O)NCCc1ccc(F)nc1)NC(C1(CC)CC(C)(C)C1)=O C1(C)(NC(C2(NC(c3n(COC)ncc3)=O)CC2C)=O)CCCC1C N1(C(C(C)(F)F)=O)CCC(CO)(CNC(=O)CCC2CCCCC2)CC1 c1(C(=O)NCC(CCOC)NC(C2CC(=O)N2)=O)ccc(C2CCC(=O)N2)cc1 CC1(C)C(NC(c2ccn(CCNC(=O)CC3CCSC3)c2)=O)CC1(F)F c1(C(C(=O)NCC2CC3CCC23)=O)c[nH]c2cc(F)ccc12 C=CCC(CC=C)C(=O)NCCC1CCN(C(c2cc(Br)co2)=O)C(C)C1 Cc1ccc(=O)n(CC(=O)N(CC(C)NC(c2scc(C)c2Br)=O)C)c1 N1(C(CCCCOC)=O)CC2ON=C(CNC(c3cn4c(n3)CCC4)=O)C2C1 C1(CCC)COCCN1C(=O)CC1(OC)CN(C(C2CCCN2CC)=O)C1 c1(C(N2C(C3(O)CN(C(C(CCC)OC)=O)C3)CCC2)=O)cnc(N)c(Cl)c1 C(CC(C)C)(C(=O)N1CCCC1C(=O)N(CC(F)(F)F)C1CCC1)NC(C)=O C1(C(=O)NC(CN(C(CCn2c(C)ccn2)=O)C)(C)C)C2CC3C(C2=O)C13 c1(C(N(CCNC(C2(CC#C)CCCCC2)=O)C(C)C)=O)ccc([N+](=O)[O-])s1 C1(C(=O)NCC2(OC)CN(C(c3n(CC)ncc3)=O)C2)OCCC1(C)C CCCCC(C)CCC(=O)NC1CCOC1C(N1CC(C2CCCCC2)C1)=O N1(C(CC=CC)=O)CCN(C(=O)CN2CC=CC2)C2CC12 C(C(CNC(C1CN(C2CCC2)C1)=O)S(C)(=O)=O)NC(CC(C)O)=O C1(C(=O)NC23C(CN(C(c4cc(C(C)=O)sc4)=O)C2)CC3)CCC2(CCC2)CC1 c1(C(N2CCC(N(C(C)=O)C)C2)=O)cn2c(n1)CCN(CC(=O)O)CC2 CS(=O)(=O)CC(F)(F)CC(=O)N(CCNC(c1ccc(O)cc1F)=O)CC1CC1 CCC(CC(=O)NCC1CC(C)(O)C1)N(C)C(C1CCN1C(C)(C)C)=O C1(C(N2CC(O)(CCNC(C3(CC)CCNC3=O)=O)C2)=O)CS(=O)(=O)CC(=O)N1 CSC1=C(C(=O)N2CCCC2(C)CNC(c2ncccc2C)=O)CCCC1 N1(C(Cc2cccc(SCC)c2)=O)CC(NC(c2cocn2)=O)CC12CCOC2 N1(C(C(=O)N(CCOC)CCNC(c2n[nH]cc2Br)=O)C)CCCC(O)C1 C(=O)(CC1COc2cc(O)ccc21)NCC(C)NC(c1c(C)cc(OC)nc1)=O CCN=c1ccc(C(N2CC(OC)C(NC(c3ncoc3C3CC3)=O)C2)=O)c[nH]1 c1(C(C)(F)F)ccc(CN)nc1.N1(C(=O)CSC2CCCCO2)CCC(O)(C)C1 Cc1cc(C(=O)NCC2CN(C(c3ccn(C(C)C)n3)=O)C3CC23)cc(N)c1Cl C(C(=O)N(C(C)CC(=O)NCCCN(C)C)C)(C(C)C)SC C12(NC(c3ccc(OCC(F)F)cc3)=O)CCCC1CN(C(=O)C1=C(Cl)CC1)C2 c1(CC)c(C(=O)NC2CCC(NC(=O)C=CSC)CC2)nnn1-c1ccccc1 N1(C(C(C)c2cncs2)=O)CC2(CC(NC(=O)CCC(C)(C)C)CO2)C1 C1(C(F)(F)F)(C(N(C)CC2CCCN2C(=O)C(F)OC(F)(F)F)=O)CCCCC1 C1(CNC(CCC(C)(F)F)=O)CC2(CO1)CN(C(C1CC3(C1)CC(C)(C)C3)=O)C2 C(C(C)(C)CC(C)O)NC(c1n(CC(=C)C)nnn1)C1(CF)CC1 c1(OCC(N2CC3(CN(C(C4CCOCC4)=O)C3)C2)=O)cc(Br)ccc1F c1(C(=O)NCC2CCCN2C(c2ccc3nonc3c2)=O)cnc2snnc2c1 C1(NC(NCC=C(C)C)=NCCc2ccccc2C#N)CCn2c(C)cnc2C1 C1(C(=O)NCc2n[nH]cc2C(N2CC=CC(O)C2)=O)C2CCC(F)(F)C12 c1(NC(=O)C(F)F)cccc2c(C3=COCCC3)cccc12 C(=O)(C(F)(F)C(F)(F)C(F)F)NCC(C)CNC(c1nnn(C)n1)=O c1(NC2CN(C(c3ccc(C)c(F)c3)=O)C(C)C2)ncnc2cc(C3CC3)nn12 C1(NC(c2n(CC)c(O)nc2)=O)(CC)CCCN(C(=O)CN2C(=O)CNC2=O)C1 N1(C(C(C2CCCO2)NC(Cc2cc(C)n(C)n2)=O)=O)CCC(O)CC(C)(C)C1 c1(OC)ncc(C(=O)NC(C(=O)NCCCn2cncn2)c2ccco2)s1 n1(CCOC)cc(C(C(=O)OC(C2CS(=O)C2)=O)OC)nn1 c1(NC(C2CN(Cc3cccs3)CCC2O)=O)cc(Br)cnc1[N+](=O)[O-] N1(C(c2c(OC)c(Cl)ccc2)=O)CC2CCN(C(=O)C(C)(C3(C)CC3)OC)CC12 N1(C(C2N(C(=O)CC3COCCO3)CSC2)=O)CCC2(CCC(O)C2)C1 C1(OCC#C)CCCN(C(=O)C(C)CNC(=O)Cc2ccc(C)nc2)C1 CC1CN(C(c2cnn(-c3ccccc3)c2Br)=O)CCN1C(=O)C(C)(C)O c1cnc2cc(CNC(c3nnnn3Cc3cccs3)c3nc[nH]n3)oc2c1 c1(C(=O)NC)ccc(C)c(NC(C)CCN(C)C(=O)OC(C)(C)C)c1 C1(NC(Cc2nc(-n3c(C)ccc3C)sc2)=O)CCN(C(=O)CC(C)F)C1(C)C N1(c2nc(OC)cc(OC)n2)CCCC1C1OCCO1 N1(C(CC2C(C)(C)CCN2C(C2CC(=O)CS2)=O)=O)CCc2ccccc2C1 CC(C)(C)C(C(=O)NC1CN(C(c2cc(F)cnc2O)=O)CC1O)C1CCCC1 C1(C(N(C(CN(C(C(=O)Nc2ccc(C)cc2)=O)C)C)C)=O)CC(C)(C)CCO1 CN1CC(C(N2CC(NC(=O)CCC(=O)N(C)C)C2)=O)C(C)(C)C1.c1(O)ccsn1 C1(NC(c2c(C)cccc2O)=O)CN(C(=O)CC2=CCOCC2)CC1C1CC1 N1(C(C2N(C(=O)CCc3ccccc3F)C3C(C2)C3)=O)CCC2(CCOC2)C1 C(=O)(CC(C)(C)CC(=O)N1CCC(NC(C2CCCN2C)=O)C1)OC C1(CNC(c2[nH]cc(C)c2)=O)CCN(C(=O)C(C)c2ccsn2)C(C)C1 CCCC(CCC)CC(=O)N1CCC(CO)(NC(=O)CC2CCC(=O)NC2=O)C1 C(=O)(CC(C(F)F)NC(=O)C(C1CCC1)OC)N(CC(COC)C)C N1(CC(=O)NCC)CCCCC1NC(C)CCCOCC c1(-c2cnc(C(=O)NCCc3ccc(C)cc3)nc2)ccc(F)c2cccnc12 C1(C(N(C(C)C(C)(C)O)C)=O)(NC(c2cn(C)cn2)=O)CC(F)(F)C1 N1(C(COC)=O)CC2(CCCCN2C(c2ccc3c(C)[nH]nc3c2)=O)C1 c1(COCC(=O)NCCC2CC(NC(c3cnc(Cl)[nH]3)=O)C2)ccncc1 C12=NNC(=NC(=O)N1)S2.N1(CC)CCCC1.C1CO1 N1(C(C(COCC)NC(=O)C(C)NC(C)=O)=O)CC(S(N)(=O)=O)C1 C1(C(=O)OCC)(C(=O)NCCCNC(C2CC(C)=NO2)=O)C=CCC1 c1(OCC(C)C)ccc(S(C)(=O)=O)cc1NC(=O)N(c1cnc[nH]1)C C1(C(=O)NCc2ccc(C)s2)CC2CCC1N2C(c1ncsc1Br)=O C1(C2(O)CCOCC2)(CNC(N(C)Cc2c(C)occ2)=NCc2ccccc2)CC1 N1(C(C2(C)CCC(=O)C2)=O)CCCCC(CNC(c2n[nH]c3c2CCC3)=O)C1 c1(OC)ncc(C(N2CCCC(N(CCF)C(C3CC3C)=O)C2)=O)cn1 CC(CC1CC1)C(=O)N1C(C(=O)NC2CC(C(F)(F)F)C2)CC1C c1(C(=O)OCC)c(C)sc(C(N2CCCC(CSC)C2)C(=O)NCC(F)F)c1Cl CCCC(CC)C(=O)NC(CO)CCCNC(C1CCCS1)=O c1(C(N(CCCNC(C2(C)CC2C(F)(F)F)=O)CC)=O)[nH]nnc1C(=O)OC n1(CC(=O)NC(CC)CN(C(=O)C(COC)OC)CC)cccc(C)c1=O N1(C(CCc2n(C)ncc2)=O)CCC2CN(C(=O)CN3CCCC3=O)CCC2C1 CC(C)(CC(=O)NCC(F)CNC(c1cccc(-c2cc[nH]n2)c1)=O)C1CC1 c1(C(N(CCNC(Cc2cc(CC)no2)=O)C(C)C)=O)ccc2cc[nH]c2c1F C(N1CCC2(CCCCO2)C1)c1n(CC)c(C)nn1.n1(CCC)c(C)nc(C)c1C CC1CCN(C(c2cc(C3CCC3)nn2C)=O)CC1CNC(C1(Cl)CCC1)=O S(=O)(=O)(CC(=O)NC(C)CC1CN(C(=O)C(C)Cc2ccc(C)cc2)C1)NC C1(NC(c2cncc(OC)c2)=O)CCCC(NC(c2ccnc(O)c2)=O)CC1 CC1(NC(=O)C=CCC(C)(C)NC(c2cnsn2)=O)CC(O)(CO)C1 Cc1cn2cc(C(N3CC4CCN(C(=O)CC5CCN(C)CC5)C4C3)=O)sc2n1 N(C(=NCCc1csc(C(C)C)n1)NC(CC)C=O)CC(=C)C C(C1(C)CCOCC1)=CC(=O)NC(C1CN(C(c2ccc(C(F)(F)F)o2)=O)C1)C C(N=c1cccc(S(=O)(=O)NCC2CC3CC3C2)[nH]1)C1(C(C(C)C)O)CC1 CC(C)(C)C(CNC(C1C2CCC1(c1ccccn1)C2)=O)NC(c1nncs1)=O c1(C(C(=O)N(CCNC(=O)CCn2cncn2)C2CC2)O)ccccc1Br c1(NC(C2C(CNC(C(n3ccc(C)n3)C)=O)C2)=O)ccccc1N=[N+]=[N-] CC#CCCCC(=O)NC(C)C(C)(C)C(=O)NC(c1ncn(C)n1)C c1(C(=O)NC2C3N(C(C(C)(C)N(C)C)=O)CC(CC3)C2)c[nH]c(=O)c2ccnn12 c1(C(=O)NCC(CC=C)NC(=O)CN2CC(C)(OC)C2)c(C)ccnc1O C1(NC(=O)C(F)OC(F)(F)F)CCCCC1OC(CNC(C(C)(C)OCC)=O)=O CN1CCC(C)(C(N2CC(NC(=O)Cc3ccon3)C(n3ccnn3)C2)=O)C1 N1(C(C(C(=O)OCC)C(C)C)=O)CCCC2(NC(=O)C3=C(Cl)CC3)CCCC12 c1(CNCC(C(=O)NC)(C)C)ccc2oc(Cl)cc2c1 C=CCC(CC)C(=O)NC(C)CNC(=O)CC1NC(=O)NC1=O C1(NC(c2cnc(OC)nc2)=O)CC2CC(C1)N(C(c1snnc1C1CC1)=O)C2 C1(CCN(C(c2nc(COC)sc2)=O)C)CCN(C(C2(SC)CCC2)=O)CC1 c1(C(N(C2(CC(N3C(C(C)O)COCC3)=O)CC2)C)=O)ccc(=O)n(C)c1 N1(C(c2c(=NCC=C)[nH]ccn2)=O)CCC2(CCCCN(C(=O)C=CC)C2)C1 c1(C(N2CCC(F)(C(N(CC(O)CF)CC)=O)C2)=O)c[nH]c(C#N)c1C C1(CC)(NC(=O)CCOCCN(C)C)CCN(C(c2cc(Br)c(C)o2)=O)C1 N1(C(C2N(CC)CC2)=O)CC2CCC1CN2C(=O)Cn1cnnc1O CC1CC(C)(C(=O)NC2CC(CNC(=O)CCc3cccc(F)c3)C2)CC(C)O1 CCCCC(=O)N(C)CC1CCN(C(c2cscc2Cl)=O)C1 N1(CC(N2CC(C(=O)NCCC3CCC(C)O3)(SC)C2)=O)CCC(O)CC1 C(=O)(C1CCOc2ccc(Cl)cc21)NC1(C)CCN(C(=O)COC(F)F)CC1 c1(C(N2CC(OC)(CNC(C3CCCOC3)=O)C2)=O)cc(O)cc(N)c1C N1(C(COCC#C)=O)CCN(C(c2cccnc2)=O)CC(C)(F)C1 Cc1cc(C(=O)N(C)CC2CN(C(=O)C(c3ccnn3C)C)CCO2)ccc1Cl Cc1ncnc(C)c1C(N1CCC(CN(C)C(C2(C)CC=CCO2)=O)C1)=O Cc1cc(C(=O)NCCN(C(=O)C(C)CC2CC2)C2CC2)ccc1-n1cnnn1 N1(C(=O)NCCC#C)CCC2(CCCCN(C(=O)COCC(=C)C)C2)C1 S(=O)(=O)(c1ccccc1F)NC(C)C(N1CCC(N)C(C)(C)C1)=O c1(C(=O)OC)cc2cc(SCCCOc3cccc(F)c3)sc2[nH]1 c1(C(=O)NC2CN(C(C=CCCC)=O)CC2O)cnc(C2CCCC2)[nH]c1=N C1(CC=C)(NC(c2cc(CO)[nH]n2)=O)CCN(C(c2nncs2)=O)C1 N1(C(C)C)CCCC(NC(=O)CC(C)(C)N(C)C(C2CC2C(C)(F)F)=O)C1 C(CC1CC1)(CC(=O)N1CC(O)CCO1)NC(C1CCCC(OC)C1)=O c1(C(=O)NCCCN(C(C2CN(C(N)=O)C2)=O)CCO)cnn(CO)c1C(F)(F)F c1(C(=O)NC2CC(OCC(=O)NC(CC)CC)C2)snnc1CC c1(C(=O)NCCC2CCC(NC(=O)CCc3ccco3)C2)occ2c1CCCC2 c1(NC)cc(C(=O)NCc2ccccc2CNC(=O)CNC(N)=O)ccc1F c1(C(N2C(CO)CC(NC(C(CC)(C)O)=O)C2)=O)cc(C#N)cc2ccccc12 N1(C(c2c(NC)cnnc2)=O)CCC=C(C(=O)N2CC(CO)C2)C1 C1(CC)C(NC(C2(OC)CCSC2)=O)CCCN1C(c1nccnc1C)=O C(C(=O)NCC1(C2CCCN2C(=O)CCOC2CC2)CC1)(C(C)(C)C)N(C)C N1(C(C(CCC)NC(c2cncc(OC)c2)=O)=O)CCOC2(CC2)C1 N1(C(CSCC(C)C)=O)CCC2(CC1)CN(C(c1cncs1)=O)C2C(C)C C1(NC(C(C)NC(C)=O)=O)CCC(C)(CNC(c2cc(C)sc2C)=O)CC1 CC1(C)CC(CNC(c2ccc[nH]2)=O)CN(C(=O)C(c2ccc(F)c(F)c2)=O)C1 C1(C(N(CCCCC(=O)NCCN2CCC(O)C2)C)=O)CC2(C1)CC2(F)F C1(C(=O)NCC23CC(NC(=O)CCC(C)OC)(C2)C3)(CC)CCCCC1 n1(CC(N2CCC(CN(C(C3C(C(C)C)C3)=O)C)CC2)=O)nnc2c1CCCC2 C1(O)(CC(=O)NCC(C)(C2CCC2)NC(=O)CSc2n[nH]c(O)n2)CCCOC1 N1(C(CC(CCCC)O)=O)CCCC2(CCCN2C(=O)CC(Cl)Cl)C1 n1(CC(C)C)cc(NC(=O)C(N2CCC(NC(C3CCNCC3)=O)C2)=O)cn1 N1(C(C2(CCC)CC2)=O)CC(NC(c2cnc(C)c(C#N)c2)=O)C(C2CC2)C1 N1(C(CNC(CC)=O)=O)CC2CCCC2(NC(c2cc3cccnn3c2)=O)C1 C(C(C)(C)C1=CCCCC1)NC(C(=O)NCCOc1c(C)cccc1C)=O CC1CCOC(C(N2CCOC(CCNC(=O)C(F)(F)c3ccccn3)C2)=O)C1 CC1CCC(NC(=O)Cc2ccccc2Cl)CN1C(=O)COC1CC=CC1 C1(O)(CC(=O)N(C(C)CCNC(c2ccsc2C(F)F)=O)C)CCN(C)CC1 c1(CCC(=O)NC(C=C)C)ccccc1-n1cc(CCCNC)nn1 C=C(Cl)CC(C(=O)N(CC#CC)C)NC(C1C=CC=CC=C1)=O C(=O)(CN=S(C)(C)=O)NCCCCC1(NC(C(C)C(=O)N2CCOCC2)=O)CC1 c1(CC)cnc(C(=O)NC2CCN(C(=O)CCc3nncs3)C2)nc1 Cc1ccc2c(n1)CN(C(C1C3CC(O)C(C3)N1C(c1nc(C)c(C)s1)=O)=O)C2 c1(C(C(=O)NCCN(C(C(C)OCCC(C)C)=O)C(C)C)(F)F)ccc(Cl)nc1 [N-]=[N+]=NCCNC(=O)C(C1CCCC1)NC(=O)CCc1cnoc1 C1(n2c(C(c3ccoc3)NC(C(=O)NCC)CC)nnn2)CCCCCC1 c1(C(N2CC(F)CC(NC(c3coc(C4CC4)n3)=O)C2)=O)cn2ccnc2cn1 C12(C3CC3)CCN(C1)C(=O)C(=O)N2.c1(OC)c(OC)cccc1C(N)=O N1(C(C(C)SC)=O)CCN(C(C2(c3cccc(F)c3F)CCCC2)=O)CC1CO C12(C(N(C)CC3(O)CN(C(c4ccc(N)c(N)n4)=O)C3)=O)C3C4C1C1C2C3C41C N1(c2nnc(C(c3ccc(C)c(C)c3)O)n2C)CCCCC(S(C)(=O)=O)C1 c1(NC(CC2(NC(CC3CCN(C)CC3)=O)CCC2)=O)ccc(C#N)nc1 C(C(C)(C)CC(=O)NC1CCN(CCNC(=O)C(CSC)OC)CC1)OC c1(C(=O)NCC2N(C(c3n(C=C)ncc3)=O)CC2)c(Cl)cc(Cl)nc1N C(=O)(CC(C)C1CC1)N(CC(C)N(C)C(c1[nH]ccc1-c1ccccc1)=O)C Fc1ccc(Br)c(C(c2nnnn2C2CCOCC2)NC(CF)C2CCC2)c1 C(=O)(C1CCCc2c[nH]nc21)NCCCCCN(C)C(C1(C)CNC(=O)C1)=O N1(C(C(CC)(C)C(N)=O)=O)CC2OCCN(C(=O)Cc3ccoc3C)C2C1 Cc1nc(CN2CCC(NC(=O)Cc3cccnc3)C2)ccc1Br C(=O)(CC(C)CC(F)(F)F)N1CCC(CNC(CCc2nc(C)c(C)o2)=O)C1 N1(c2nnc(C3C(OCC)C3)n2CC)CC(C)c2ccc(OC(F)F)cc21 C(=O)(C1CCc2nccn21)N1CC(C)N(C(C2CCC(=O)NC2)=O)C(C)C1 N1(C(c2n(CC)ccn2)=O)CCCC(C(=O)NCCC(=O)NO)C1C C12(NC(c3cc(CC)no3)=O)CCC(CNC(c3cc([N+](=O)[O-])c[nH]3)=O)(C1)OC2 C1(CNC(C(CO)N(C)C)=O)CCN(C(=O)CCCC2CCC2)CC1CO c1(CC(=O)OC(c2ccccc2OC)CC)cccc(Br)c1 c1(C(N2CCC(NC(C(CC)=CCCC)=O)C(C)C2)=O)cn(C)c2ccccc12 O=C(CC1=NNC(=O)C1)NCCC12CCC1CN(C(=O)Cn1nnc(=O)[nH]1)C2 C(=O)(C1=NOC(C)(C)C1)NC(c1cn(C)nn1)C(N1CC(F)(C(=O)OC)C1)=O C(=O)(C1=CC2(CCOC2)C1)NC(CNC(c1c(OC)cc(=O)n(C)c1)=O)C1CC1 C1(C(=O)NC2CC(=C)C2)COCCC1NC(c1cscc1OC)=O N1(C(C2C(=C)CC2)=O)CC2CN(C(c3cc(C)ccc3Br)=O)CC2C1 C1(C(F)F)(NC(c2cn(-c3cccc(OCC)c3)nn2)=O)CCN(C)CC1 c1(C(=O)NCC#CCNC(c2n(CC)nnc2)=O)coc2c1N(C)C(=O)CCC2 c1(OC)nc(C(=O)NC(C)(CNC(c2ccn(CCF)n2)=O)CO)cc(O)n1 c1(OCCC)ccc(CNC2CC2C(=O)NC(c2cccc(O)c2)C)cc1 c1(C(c2noc(C)n2)N(C(CNC(CC(=O)OC)=O)=O)C2CC2)ccc(Cl)cc1 C=CCC(CNC(=O)CC1CC2CC2C1)C(=O)N(C)CCOC(C)=O C1(CCC)CN(C(=O)C(C)Cn2ccnc2)CC1C=O.c1ccnnc1 C12(CNC(CCOCCC)=O)CCC(C1)N(C(c1cc(=O)n(C)cn1)=O)C2 S(=O)(=O)(c1ccc(N2CC(C)CC(O)C2)nc1)N1CCCC(CC=C(C)C)C1 c1(C(=O)NC(CC)COC(=O)C=CCNCOC)ccc(OCC(F)(F)F)cn1 c1(C(N(CCN(C(=O)CC2CCC(O)C2)C)C)=O)ccc(NS(C)(=O)=O)cc1O C1(CC)CCCN(C(c2n[nH]c(=N)[nH]2)=O)C1C(=O)N(C)CCOC1CC1 CONC(=O)C(=O)NCCNC(C1(OC)CCOCC1)=O C1(C(=O)NCCOCC)(CC)CCCN(C(C2CCOC2C)=O)C1 C12(CNC(c3c(C(C)C)con3)=O)CCC(CN(C(c3ncncc3N)=O)C1)C2 C#CCC(CC#C)C(=O)N1CC2CC1CN2C(=O)CC1(CC)CCC1 C1(CCC(=O)N(C)Cc2cccnc2)CCCCN(C(C2(O)CCSCC2)=O)C1 C1(C(N2C(CCNC(COC)=O)CSCC2)=O)CN2CCCN1CC2 c1(C(CCOC)NC(C2CCOCC2)CC)ccc(OC)cc1C C#Cc1cncc(C(=O)NC2CCN(C(=O)Cc3cc(C(F)(F)F)n[nH]3)C2)c1 C(=O)(C1CCCn2ccnc21)NCC(C)(CO)NC(=O)Cc1ccsc1 Cc1cnc(C(=O)NC(C)CN(C)C(c2ccc(OCF)cc2)=O)c(F)c1 C1(C(N(C(C=C)C2CC2)C)=O)CCN(C(=O)C#CC2(C)COC2)C1(C)C CC(C)CC(C)(C)C(=O)NC1CC(NC(=O)CCC(C)N(C)C)C(O)C1 C(C(=O)N1CCC(F)(C(=O)NC2(CF)CCCC2)C1)(C(C)C)SCC C1(C(N(CCOCCNC(c2c(OC)cccn2)=O)C)=O)CCn2cnnc2C1 C1(N(C(=O)C(=O)N(C)C)CC#C)CCN(C(=O)CN(C)C(=O)OC)CC1 C1(CNC(C(C=CC)O)=O)CCCN(C(=O)CNC(=O)Cc2ccc(O)cc2)C1 C1(CC(=O)NCCOC2CCN(C(C3CC3C(F)F)=O)C2)CCCCCC1 C1(C(=O)Nc2c(C)cc(C#N)cc2)CC12CCc1cc(Br)ccc12 O=C1COc2c(C(=O)NC3CCN(Cc4ccccc4I)CC3)cccc2N1 C1(C(=O)NC(CC=C)CO)COCCN(C(=O)CCC2CCC(=O)C2)C1 N1(C(c2c(C)c(F)ccc2)=O)CCCN(C(=O)C(C)P(C)(C)=O)CC1C(C)C C1(C(=O)NC2CC(C)(C)C2)(CC)CCN(C(c2cnn(C3CC3)c2)=O)C1 N1(C(c2c(CCC)n[nH]c2)=O)CCC(NC(=O)C(O)Cc2cn(C)cn2)C1(C)C C1(CNC(C2CCOC2C(F)(F)F)=O)CCN(C(C2C3COCC23)=O)CC1 c1(C(C)C)cc(C(=O)NC(C)(CNC(C2CC(N(C)C)C2)=O)CO)n[nH]1 C(C(=O)NCC1(NC(C2CC3(CSC3)C2)=O)CC1)(C(C)C)OCC C(CC(C)C)(C(=O)NCC(CO)NC(c1cnc(C)nc1C(C)C)=O)OC N1(c2n[nH]c(=N)s2)CCc2nc(C(=O)Nc3ccc(F)c(O)c3)cn2CC1 c1(NC(C(CCC)C)C)ccc2[nH]ccc2n1 Nc1ccc(CCC(N2CC3CC(NC(C4CNC(=O)C4)=O)C2C3)=O)cc1F N1(C(C2CCOC3(CCC3)C2)=O)CC2(CCN(C(=O)C(F)n3cccn3)CC2)C1 CC1CCC(N(C)C(c2ccc(CNC(=O)CCc3cnn[nH]3)s2)=O)C1 c1(NC(CN(C(C2CC(O)(CC#C)C2)=O)C)C)cccc(F)c1[N+](=O)[O-] c1(CC(N2CCC(C(C(=O)N(CCCOC)CCO)F)C2)=O)ccc(C#N)cc1 c1(CC)ccc(C(=O)NC2CN(C(C3CC(=O)N(C)C3)=O)C(C)(C)C2)c(N)c1 N1(CC(c2ccc(F)cc2)C)C(=O)CN(CC2CCCC(C3CC3)O2)C1=O N1(C(C(CO)OC)=O)CC2(CCCC2)C1C(=O)NCC1CCOC1C N1(C(Cc2nnc(C)o2)=O)CC2CCC(CNC(C3(F)CCC(C)CC3)=O)(C2)C1 c1(CC(N2CC(C)(C(=O)NC(CC)CN(C)C)C2)=O)cn(C)nc1C CCCC(C)(CCC)C(=O)NC(C)CNC(=O)Cc1ccc(Br)c(Cl)c1 c1(C(N(C2CN(C(=O)C#CC(C)(C)C)C2)C)=O)cc(Br)c2occc2c1 N1(C(CC2(OC)CCCC2)=O)CC2(CCCCN2C(C2CCCC(=O)N2)=O)C1 C(=O)(CC(C)(CN(C)C)C(F)(F)F)NC(CNC(COCC)=O)C1CCC1 S(=O)(=O)(c1ccc2[nH]c(=NC3CCC(C4CC4)C3)sc2c1)NC(C(CC)CC)C CC1CC(C(=O)NCC2(C)NC(=O)NC2=O)CCN1C(c1ccn(C)c1)=O c1(C(N2CCCC2CC(F)(F)F)C(=O)NC(CC)(C)C)ccn(C2CC2)c1 N1(C(c2cc(CNC(CN3C(C)CCC3)=O)[nH]n2)=O)CCN2CCC1C2 C1(C(=O)NCCC(CCC)O)CC2(CCC2)CN1C(c1cccn2cncc12)=O c1(SC)cnc(NCc2ncccc2-c2cncc(CN3CCOCC3)c2)nc1 CCCC(O)C(=O)N1CCC(CO)(NC(=O)CCC2CCCCC2)C1 N1(C(CCS(N2CCS(=NC)(=O)CC2)(=O)=O)=O)c2ccccc2Sc2ccccc21 C1(N(C(CSC)=O)CCO)CCCN(C(=O)C(C)=C2CC2)C1 c1(C(N2CCC(CCNC(CNS(NC)(=O)=O)=O)C2)=O)ncnc(O)c1Cl c1(C(N(CCCNC(C2(C)CC3CC3C2)=O)C(C)C)=O)c2c(nn1C)CCCC2 c1(NC)nc(C)ccc1C(=O)NCC(C)CNC(C1(OC(C)=O)CC1)=O C1(C(=O)NC2(CNC(c3c(C)nc(CCCC)s3)=O)CC2)CN=C2N=CNN2C1 N1(C(C(c2ccc(F)c(Cl)c2)N)=O)CCC2OCC(=O)NC2C1 c1(OC)cccc2ccc(NC(C3CC(NCc4ccc(F)nc4)C3)=O)nc12 C1(N(C)C(C2CCCCN2C)=O)CCC2CN(C(c3cccc(F)c3O)=O)CC12 C1(NC(=O)COCCF)CCC12CCN(C(=O)Cc1ccc3c(c1)COC3)CC2 N1(C(CC(C)N(C)C)=O)CCCC2CN(C(=O)CC3CC4(CC4)CO3)CC12 c1(C(=O)NC(CC)CN(C(=O)C(N2CCOCC2)C)CC)cc(C)n(C)c1 N1(C(c2ccc(OC)o2)=O)CCN(CCCNC(=O)CCC=CC(C)C)CC1 C(=O)(C1=CCC(C)CC1)NC(CC(=O)NC1CC=C(C)CC1)C(F)F N1(CCC(C)SC)CCC(NC(c2cc3n(n2)CCC3)=O)C(C)C1 C1(C(=O)OC)CC2CCC(C1)N2C(c1cc(CO)co1)=O.C12CC(C1)NC(=O)C2 N1(C(c2c(C)nc(C(C)C)o2)=O)CC(C)N(C(=O)CSCC(F)(F)F)CC1C C1(C)(C(C(N2C(C(C)N(c3ccccc3)C(=O)CC3CC3)CCC2)=O)F)CCOCC1 C1(NC(c2cnc(OCC)nc2)=O)CCN(Cc2ccc(OC)c(Cl)c2)CC1C N1(C(C2C(=C)C2)=O)CC(OC)CC1CNC(c1ccc(C(C)(F)F)cn1)=O CN1CCc2[nH]nc(C(=O)NC3CC(NC(c4c(N)cc(Cl)cc4Cl)=O)C3)c2C1 N1(C(C(COCC)C)=O)CCOC(C(=O)NCCN(CC(C)C)CC)C1 Cc1cc(C(=O)NC(CNC(=O)CC2CCC3CC23)C2CC2)cc(N)c1O c1(OC)c(C(=O)NC)csc1C.C1(CC(C)C2CCC2)CCN(C(=O)CO)CC1 C(=O)(C(C)(C)C(C)(F)F)NCC1CC(C)CN(C(=O)Cc2csc3nccn23)C1 c1(C(=O)OC)ccc2cnnc(N(C3CC3)Cc3ccc(F)c(F)c3)c2c1 c1(C(=O)NCC2COCCN2C(c2ncccc2Cl)=O)cncc([N+](=O)[O-])c1 CC1(C(=O)NCc2ccc(CO)s2)CCCN1C(C1CCCC1)=O C1(C(=O)NCCC(=O)NCC(=C)F)(CC)CNC(=O)C1 c1(CC)cc(C(=O)NCC(N2CCN(C(=O)C(C)(C)C)CC2)C)cc(Cl)c1 C(=O)(C1COc2ccccc21)N(CC(C)NC(C1(C)CCNC(=O)C1)=O)C c1(C(N2CC(NC(c3ccc(C(C)=O)[nH]3)=O)C(O)C2)=O)ccc(S(C)(=O)=O)[nH]1 C(C1OCCc2sccc21)NC(CNC(=O)CN1CCCC(C(F)(F)F)C1=O)=O N1(C(c2nc(CC)oc2)=O)CC2CCC1C(NC(=O)CCC1CCC(C)O1)C2 N1(C(COC2(C)CCC2)=O)CCCC1CNC(C12CC(c3ccccc3)C1C2)=O C1(CC(=O)NC(CC)CNC(=O)CCC2CCOCC2)CC(C)(C)C(=O)N1 N1(C(CN2CCC(C)CC2)=O)CCC2(CC1)CC2NC(=O)CN1CCC(C)(C)C1 N1(C(C2CC23CCOC3)C(=O)NCC(C)C)CCC(C2CC2)C1 N1(C(CC(n2ccc(C)n2)C)=O)CCN(C(=O)C=Cc2cccc(Cl)c2)CC1C O(N1CCC(NC(=O)CC(C(F)F)N(C(=O)C=CCN2CCCC2)CC)CC1)CC c1(NCCOc2ccc(C)cc2)nc(NC2CC3CC(O)C2C3)c2c(ncn2C)n1 C1(NC(C2CCN(C(c3ccncc3)=O)C2)=O)CCC2C(CC1)C2(F)F c1(C(=O)OC)cc(C)cnc1N1CC(C)(NC(c2c(Cl)cnn2C)=O)C1 c1(C(N2CC(NC(C(CC)(C)O)=O)C(O)C2)=O)occ2c1CCC2 CC#CCC(C(=O)NC(c1ncccn1)CC)NC(=O)C(CC)=CC CC(CCC(=O)N1CCCC1c1ncc[nH]1)NC(C1CC(=C2CC2)C1)=O C=C(C)CC(C(=O)N(CCCCCCNC(c1ccccc1CC#N)=O)C)OC Cc1c(C(N2CC(OCCNC(c3cc4occc4s3)=O)C2)=O)sc2cncn12 N1(C(C(CC)n2cncn2)=O)CCC(C)C1N(C(=O)C(F)=C(C)C)C1CCCC1 C(c1ccc2c(c1)COCC2)=CC(N1Cc2ccc(Cl)nc2C1)=O C12(NC(CN(C)C)=O)CCCCC1N(C(c1cnc3c(cnn3C)c1)=O)CC2 c1(C(=O)NCC2C3CN(CC(=O)NCC=C)CC32)cc(C)nc(O)n1 CCC1=C(C(=O)N2CCCC2(C)CNC(C2CC3(CCCC3)CO2)=O)CCCO1 N1(C(CCSCCC)=O)CC2CCOC2(CNC(=O)C(C)(C)CCSC)C1 c1(C(=O)NCC(C(=O)NCC(C)N(CC)CC)N(C)C)cnn2c1OCC2 c1(CC)[nH]c(=N)sc1C(N1CC(NC(=O)C=CC(c2ccccc2)=O)CC1C)=O c1(CCNC(C2C(CNC(CCC)=O)CCC2)=O)cccnc1F CC1CC(C(=O)Nc2ncccc2O)N(C(c2cnn(C3CCCC3)c2)=O)C1 Cc1ncc(C(=O)NCCOCCN(C(=O)CCc2cnoc2)C)n1C(F)F C12(NC(C3OCCN(C)C3)=O)CCCC1N(C(c1scc3c1CCCC3)=O)CC2 c1(C(=O)NCC2CCN2C(C2CN(CC(F)(F)F)C2)=O)cccc(C2CCC2)c1 C#CC1C(C(N2CCC(OCCNC(=O)Cc3ccn(CC)n3)CC2)=O)C1(C)C C1(n2ncc(C)c2)CCN(C(=NCCCCc2cn[nH]c2)NCC(C)(C)C)C1 CC1CCC(NC(c2csnn2)=O)CN1C(=O)Cc1cnc(C2CC2)[nH]1 C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC(C)C(CNC(=O)COCC(F)F)C1 S(=O)(=O)(c1ccc2c(c1)CNC(=O)O2)NCc1ccc2nnc(C)n2c1 N1(C(C(CC)n2cccn2)=O)CCOCC1COC.c1(C2C(=O)O2)ccccc1 C1(N(C(=O)CCc2ccn(C)n2)C)CN(C(=O)CCC2CCOCC2)CC1F C1(CNC(c2cc(SC)oc2)=O)CC2CCC1N2C(=O)C(C)C1CCCO1 c1(C(N(C)CC2CCCN(C(C(C(CC)C)O)=O)C2)=O)cc2n(n1)C(C)CCC2 N1(C(c2c(C)nc[nH]2)=O)CCCCC1C(=O)Nc1ncc(C#N)s1 c1(C(=O)NC23CC(NC(C4CCC(OC)C4)=O)(C2)C3)c(C)nn2cc[nH]c(=O)c12 n1(CC)cnc2nc(=NCC(C)C(F)(F)F)[nH]c(NCCS(=O)C(C)(C)C)c12 C=CC1CN(C(=O)COCC(F)(F)F)CC1NC(=O)CCCCC1CC1 c1(C(N)=O)ccccc1OCC(=O)NCC=CCNC(C1CC2CC2C1)=O c1(C(=O)NC(C2CCCN(C(c3cnc(Cl)c(Cl)c3)=O)C2)C)cccc(Br)c1F CC1(C)CCCN(C(c2cocn2)=O)C1CNC(c1cc(O)cc(Br)c1)=O C1(C(N(CCNC(c2ccc(OCCOC)nc2)=O)C)=O)CCCNS1(=O)=O C1(N(C(CC=C=C)=O)CC)CCCN(C(c2cc(C)sc2C)=O)C1 c1(-c2nc(NC(c3cnc(OC)s3)=O)sc2)ccc(COCCO)cc1 N1(c2snc(CC)n2)CCC2(CC1)C(NC(=O)C=Cc1nc(C)cs1)CS2(=O)=O N1(C(CCNC(=O)NC)=O)CC(n2cccn2)(C(=O)NCCCNC(C)=O)C1 c1(OC(C)C(=O)Nc2ccccc2)cc2ccccc2cc1C(=O)OCCO Cc1ccc(S(=O)(=O)N2CCC(CC(N3CCCC(C)(O)C3)=O)C2)cc1C(=O)O N1(C(=O)C(O)C2CC2)CCC(c2cn(CCCCO)nn2)C1 c1(CC)nnc(N2CCN(C(C3CCOCC3)C)CC2)n1CC(=O)OC(C)(C)C c1(-c2n(CC=C)c(N3CCCC4OCCC34)nn2)cnc2cc(Cl)ccc2c1 c1(COC)ccoc1C(=O)NC1(C(=O)NC(c2cnc[nH]2)C)CC1(C)C C1(NC(CC(=O)N(C)C)=O)CCC(N(C)C(c2nc(C3CC3)n[nH]2)=O)CC1 C1(NC(c2cc(SC)c(CNC(C)=O)cc2)=O)CCCCC1S(C)(=O)=O N1(C(c2cc(C(C)=O)sc2)=O)CCN(C(=O)CCCc2ccsc2)CC(CO)C1 c1(C(C)(C)C)ccc(CNC(C2CCC(=O)O2)=O)cc1 N1(C(C(F)=C(C)C)=O)CCC(N(C)C(c2ccnn2CCF)=O)CC1 C1(NC(C(C)SC)=O)CCCCC1CNC(C1(CCF)CCOCC1)=O C1(C(N2CC(C(=O)O)(NC(=O)C=C[N+](=O)[O-])C2)=O)CCC2C(CC1)C2(F)F CC(C)C(CNC(=O)NCCCS(=O)(=O)N1CCCC1)CO C(CC(=O)N1CCC2CC12)(C(C)OC)NC(COCCSC)=O N1(C(C(CC)SC)=O)CCCC(N(C(=O)C=CCCC(C)C)C)CC1 C1(CCNC(C2(C)CNC(=O)C2)=O)CCN(C(c2csnc2Cl)=O)CCC1(F)F C1(CCC=C)(C(=O)NC(CO)C(N)=O)CN(C(c2cnn(CC)c2)=O)C1 C1(NC(C2(CC)CC(=C)C2)c2nnnn2Cc2cccs2)CCCN(C)C1=O C1(CN2C(C(=O)NCC3(C(=O)NC4CC4)CC(=C)C3)CCC2)(CC)CCCCC1 C(C)(CCC(=O)N1CC(C)(C(=O)N(C)Cc2ccc(F)cc2)C1)OCC N1(C(C(C)C2(O)CCC2)=O)CC(C(=O)NC2CN(C)CC2C)CC1(C)C N1(C(C2(OCC)CCC2)=O)CC2CN(C(C3C=CCC3)=O)CC(C1)O2 C1(C(N2CCC(F)(CNC(c3c(CC)nccc3)=O)C2)=O)CC2(CCO1)CC2 Cc1cc(Cl)c(C(=O)NCCC(C)(C)NC(=O)CC2(C)CC2)c(Br)c1 c1(C(=O)OC)ccc(C(=O)N(C(C)CNC(C2(C)CC2(F)F)=O)C)n1C C1(OC)CN(C)C(C)(C(N2CC(CC(C)NC(=O)Cc3cccc(Cl)c3)C2)=O)C1 N1(C(C=CSC)=O)CCC(C)(NC(=O)COCC2CC2)C1 c1(C(=O)NC2CCN(C(c3c(COC)scc3)=O)C2C)cnn2c1CCCC2 C(=O)(CS(=O)(=O)C(C)C)NC1C(O)CCN(C(c2c(C)ccc(O)c2)=O)C1 N1(C(C(C)SCC)=O)CCN(C(=O)C(COC)COC)CC2(CC2)C1 C(C(C)(C)CCl)(c1nnnn1C1CCC1)NCC(CCSC)OC C1(NC(c2c(C)[nH]cc2)=O)CN(C(=O)C(C2(O)CCCCCC2)(F)F)CC12CC2 N1(C(Cc2cccc(C)c2)=O)CCC2(CC2C(N2CC3COCC3C2)=O)C1 N1(C(C2(c3nn[nH]n3)CN(C)C2)=O)CCc2c(Cl)ccc(Br)c2C1 C1(n2cc(CC(C=C)O)nn2)CC2CCC1(NC(=O)COCC(F)(F)F)C2 CCC(CN=c1[nH]nc(Cl)c(C)c1[N+](=O)[O-])Oc1ccccc1C(F)(F)F C(c1cncn1C)=CC(=O)N(C1CCC(NC(=O)Cc2cnnn2C)C1)C C1(OC)CCC(C)(C(=O)NCCOCCCN(C(=O)C(F)(F)CO)C)CC1 N1(c2ccc(CNC(C)CCOCc3ccccc3)cc2)CCS(=O)(=O)CC1 c1(SC)ccc(-c2cncc(C(N3CCCC(Br)C3)=O)n2)cc1 c1(C(=O)NCC2CN(C(CSC)=O)C2)ccncc1NCc1ccc(C)cc1 c1(CC(=O)NCCN(CCC)C(C2CCC(C)S2)=O)cnccc1Cl C1(C(C)C)C(NC(C2(C(=O)N(C)C)CC2)=O)CCN1C(=O)CC1CC(=O)NC1=O C(C1=CCCN(C)C1)NC(C1C(C)CCN1C(C1OC2CCC1C2)=O)=O N1(C(C(C)C(F)(F)F)=O)CCCCC12CN(C(c1ccn(C3CC3(F)F)n1)=O)C2 c1(C(N2CCC(NC(C3COCCO3)=O)C2C2CC2)=O)cc2cnccc2[nH]1 C(=O)(CCCCC(N)=O)NC1(CN(C(=O)Cc2cccnc2O)C)CC1 Cc1ccc(C(C)(C)CC(=O)N(C)CCOCCNC(=O)C(C#N)C2CC2)cc1 C=C(C)C(CC(=O)NC1CCC(F)(CNC(c2cc(O)n(CC)n2)=O)C1)OCC C1(C2(CC)CCC2)CCCN1C(=O)C(n1nccc1C)C.C12CCN1C(=O)C2 N1(C(c2cnc(C)[nH]c2=N)=O)CC2(CCCC(CNC(c3cc(Cl)on3)=O)O2)C1 CC1(C)CC(=O)NCC1C(=O)NCC1CN(C(C2CCC(=O)N2)=O)CCC1(F)F N1(C(=O)CCn2ccccc2=O)CC(C2CN(C(C3SCCS3)=O)C2)C1 c1(C(N(C(CNC(=O)COCP(C)(C)=O)C2CC2)C)=O)c(F)cc(F)cc1Cl C(C(CC)CC(F)F)C(=O)NC(c1cccc(C(F)(F)F)c1)CCC C(=O)(C1COc2ccccc21)N(C(CNC(C1CC1c1ccn(C)c1)=O)C1CC1)C c1(NC(C2(CN(C3CCCN(C(=O)NC)C3)CCO)CC2)=O)cnc2sccn12 c1(C(=O)NCC(COC)C)oc(CNC(C2CNC(=O)C2)=O)cc1C Cc1oc(C)c(S(N)(=O)=O)c1NC(N1CCC(F)(c2ccccc2OC(F)F)C1)=O c1(CC)ccoc1C(=O)NCC(C)CNC(=O)C(=O)Cc1cccs1 C1(NC(C2CCCO2)=O)CCC2CN(Cc3ccc(Cl)c(F)c3)CC2C1 c1(CC(N2CCC(c3cn(CC(=O)OC)nn3)C2)=O)cccc2c1OC(C)(C)C2 c1(NC(=O)CCn2cc(CCC3(CCO)OCCO3)nn2)cscc1Br C12(COC)CCC(CC1)N(C(=O)C=Cc1ccccc1N)C2 c1(CNC(C2C(C(=O)NC3(CC)CCOCC3)C2)=O)ncc(Br)cc1C c1(C(N2C(CNC(c3cc(OC)ncc3)=O)CC2)=O)cc2c(o1)CCCNC2=O CCC(O)C(C)C(=O)NC1CCN(C(c2cc(C(F)F)ccn2)=O)C(C)C1 c1(SCC(=O)NC2CCC(C(=O)NCCNC(C)=O)C2)ccc(O)cc1 Cc1ncc(Cl)cc1C(=O)NCCC1CN(C(=O)C=C2CCN(C)C2)C1 C1(C(N(C2CCN(C(=O)C(O)P(C)(C)=O)CC2)CC)=O)CCC(=O)N(C(C)C)C1 c1(OC(CC)C)nccc(=NC2CC(NC3CCN(CC4CC4)C(C)C3)C2)[nH]1 C(=O)(C(C)(C)C(=O)NC(C1CCN(C(=O)Cc2cncc(C)c2)C1)C)NC N1(C(C(C)OCCOC)=O)CC(Nc2ccnc(C#N)n2)CC2(CCC2)C1 C1(C(N(CC(=O)NC)CC)=O)CC(CNC(=O)C(C)c2cc[nH]n2)C1 C1(CC#C)(C(N2CC=CC(NC(=O)C(F)(F)c3cnn(C)c3)C2)=O)CCCCC1 Cc1cc(C(=O)NCC(CO)NC(c2nccn2C)=O)c2cccc(O)c2n1 c1(CC(N2CCC(N(C(=O)CC3CC(OC)C3)CC)CC2)=O)c(F)cncc1Cl CC1CN(C(c2ccn(CCF)n2)C(=O)NCC(F)F)CC(C)(C)O1 CCC(O)C(C)(C)C(=O)NCC(c1ccc(F)cc1F)NC(c1ccc(C)s1)=O C1(C(=O)NCC2N(C(C(C)=C3CCC3)=O)CCCC2)CC(=O)c2ccccc2O1 Cc1cccc(NC(=O)CC2CC(C)N(C(=O)CNC(C3CC3C)=O)C2)c1 N1(C(C(C(C)C)NC(C)=O)=O)CC(C(=O)Nc2nc(Br)ccc2Cl)CC(F)C1 C1(OCC=C)CCN(C(=O)CC2(C)CCN2C(=O)C(C2CCOCC2)=O)C1 c1(C(N(CC(C)N(C(=O)C(=O)NCC(F)F)C)C)=O)cc2c(cc1N)CCC2 N1(C(c2ccc(F)c(F)c2F)C(=O)NCC(C)C)CCCC2(CCN(C)C2=O)C1 C(=O)(CCCCCCN=[N+]=[N-])N1CCC(NC(CCSCCCC)=O)C12CCC2 N1(C(C(CC#C)(C)C)=O)CC2CC(NC(=O)CN3CCCC3C)C(C2)C1 C1(C)(C(=O)NCCOCCN(C)C)C=CCN1C(c1ccnc(CO)c1)=O C(CC(=O)NC1CC(NC(=O)C(c2ccc(N(C)C)cc2)C)C1)(C(C)C)OCC N1(C(C2(CC)CC2)=O)CCCCC12CC(NC(=O)CN1CC(=O)N(C)C1=O)C2 C(=O)(CCC(C)(C)C#N)NCCC1C(C)CCCN1C(=O)Cn1ccnn1 c1(C(N(C)CC2C3CN(C(C4CCC(C)CC4)=O)CC32)=O)csc2nccn12 c1(NCC(C(C)(C)C)SC)cc(Br)ccc1S(=O)(=O)NCCNC(=O)C(C)(C)C N1(C(C(CNC(C(CCCCC)O)=O)(C)C)=O)Cc2nncn2C(C)C1 Cc1cnc(C(=O)NCC2CCCCC2NC(c2[nH]cnc2C)=O)nc1 c1(OC)cc(C(=O)Nc2cccnc2Oc2ccccc2C#N)ccc1C C1(NC(CCCC)=O)CCN(C(=O)CN(C)C(=O)OC)CC1CC c1(CCNC(C(C2CCCC2)NC(C2CC=CCC2)=O)=O)ccncn1 C1(CNC(c2c(C)cn(C)c2)=O)CCN(C(=O)Cc2cc(Cl)ccc2O)C1(C)C C1(C#C)(C(N(CC#C)CCOC)=O)CCN(C(=O)C(C(C)C)C(C)C)CC1 N1(C(c2c[nH]nc2CC(F)(F)F)=O)CCN(C(=O)Cc2nccs2)C(CCO)C1 C12(C(c3nnnn3CC)NCc3cn(CCC=C)nn3)CCCC1C2(F)F C1(CNC(C2C3CC4C(C3)C24)=O)COCCN(C(=O)COC2CCCC2)C1 C1(C(N(C)Cc2ncnn2C)=O)CN(C(C2CCCO2)=O)CCC1(C)C c1(C(N2C(C(=O)NCC3(CC)CCCO3)CC2)=O)cc(N)cc(F)c1 N1(C(CC2(C)CCC2)=O)Cc2n[nH]cc2C1C(=O)N1Cc2ccncc2C1 N1(C(C(C)(C)OC)=O)CC(NC(c2csc(=NC)[nH]2)=O)C(n2ccnn2)C1 C1(C(=O)NC2(C)CC(NC(C3CC(OC)C(OC)C3)=O)C2)CCS(=O)(=O)N1C C12(C(=O)NCCC3CCN(C(=O)COCC4CCCO4)CC3)CCCC1C2(F)F CC1(CNC(=O)C(CC2CC2)NC(=O)CC(C2CC2)C2CC2)CC2CC2C1 N1(Cc2c(OC)nccc2)CCC2C1CCCN2C(=O)C(C)NC(C)=O C1(C(=O)Nc2cc(C)c(NC(C3CC(F)(CO)C3)=O)cc2)CSc2ccccc2O1 c1(C(N(CCC)CCNC(c2coc(O)n2)=O)=O)nc(OC)ccc1OC.C1CC1 C1(C(N2CC(CN(C(CN(C(C)=O)C)=O)C)OCC2)=O)CC2(CCO1)CC2 c1(C(=O)NCCN(C(CCCCOC)=O)C)cn(C(C)C)c(=O)nc1O c1(C(N(C(CSCC)C)C)=O)[nH]c2ccccc2c(=O)c1Br Cc1ccccc1CSc1ccc(N2CCC2)cc1.C12CCN(C1)C2=O C1(C(N2CCCCC(CNC(C3C(=O)NCC3)=O)C2)=O)CC2(CCCC2)CO1 C1(c2nc(C(C)OCC)nn2CCOCCC(F)(F)F)CC(c2ccccc2)=NO1 C1(C(=O)NC(C)Cc2ncn(C)n2)(CC)CCN(C(=O)CC(C)O)C1 Cc1cc(C(=O)NC2CCOCC2C(N2CCC(CCO)CC2)=O)cnc1C CCC(C)(C)CC(=O)N1CC(O)(C(C)NC(c2csc(C(C)OC)n2)=O)C1 C1(C(=O)Nc2cncc(C)c2C)CC12CCc1cc(Br)ccc12 c1(C(C(=O)NCC(C)NC(C2(C)CS(=O)(=O)C2)=O)C)ccc(C(C)(C)C)cc1 C(CC(=O)N1CCC(C)(NC(=O)CC2(CS(C)(=O)=O)CC2)C1)(C(F)(F)F)OC c1(CC)ccccc1CC(=O)NC(C)C(c1ccccc1)NC(c1c[nH]nc1C)=O C1(CNC(c2cc(O)cc(O)n2)=O)CN(C(=O)C(F)(F)CO)CC2(CCC2)O1 C1(C(N2CCCC(N(C(C(=O)NCCOC)=O)CCO)C2)=O)CCC2(CC1)CC2 c1(CC(=O)NCC2C(NC(C(C)Cc3cnc[nH]3)=O)CC2)ccc(Cl)cc1 CCCC(O)C(CO)NC(=O)C(C)NC(C1CCC(C)(C)OC1)=O N1(C(c2ccn(CCC)n2)=O)CC(CNC(C2CCCS2)=O)CC12CCOCC2 c1(OC)ncc(C)c(C(=O)NC(C)C(c2ccccc2)NC(=O)CC#N)c1Cl C1(C(N2CCN(C(CC(C)(C)OC)=O)CC2CO)=O)CC(C(C)(C)C)=NO1 Cc1cccc(C(F)(F)C(=O)N(C)CC2CCN(C(C3CCCC34CC4)=O)C2)c1 C1(NC(c2cc(OC)no2)=O)CC(NC(=O)C=CSCc2ccco2)C12CCC2 N1(C(C(C)(C)O)=O)CCC2(CCCN(C(=O)C3Cc4c(Cl)cccc43)C2)C1 c1(C(N2C(C3CCN(C(CCCC)=O)CC3)CCC2)=O)ncnc(O)c1F c1(CC)oc(C)cc1C(N1CC(NC(C2CC2c2ccsc2)=O)C(CO)C1)=O c1(C(N2C(CCNC(C3C(=C)CC3)=O)CSCC2)=O)nc(O)nc(O)c1N C(=O)(C(C)C(C)(F)F)NCC(CN(C(Cc1c(C)nc(C)s1)=O)C)(C)C CC1CCN(C(C2(c3ccc(Cl)cc3)CCCC2)=O)CC1NC(C1(O)COC1)=O C1(C(=O)NCCSCCCO)C=CCCN1C(c1ccc[nH]1)=O C1(C(N(C)Cc2ccn(CC)n2)=O)CCOCCN1C(=O)CCn1ccnc1C c1(OC)ccc2c(c1)OCCC2N(C)C(=O)NCc1ccc(C)cc1OC(F)F C(=O)(C#CC1(C)CCCO1)N1CC(CNC(c2ccc(OC)nc2C)=O)C1 c1(C(=O)OC)n[nH]cc1-c1cn(CCCC(=O)NC2(C)CC2C)nn1 CCC(CC(=O)N(CCCNC(C1CC(COC(C)=O)C1)=O)C)C(C)C CC1CCN(c2nnc(CCc3ccc(Br)cc3)n2C)CCC1(F)F c1(C(=O)NC(C(=O)NCCc2cn(CC)nc2)C2CCCO2)ccc(O)cc1 C(=O)(C1CCCc2nn[nH]c21)NC(C(C)C)(C)CNC(=O)Cc1nn(C)cc1Cl CCCCC(C(=O)NCC1CCC=CCC1)ON=C(C)C c1(N2C(CCNC(CCc3nnc(C)n3C)=O)CCCC2)ccc([N+](=O)[O-])cn1 C(=O)(CC(C)OC)NCC(CC)N(C)C(c1nc(C)co1)=O C12(CNC(C(C)N(C)C)=O)CCC(CN(C(c3ccccc3O)=O)C1)C2 C(=O)(C(C(C(C)C)OC)N1CC(C#N)C2(CC2)C1)NCCCNCC CC(C)C(O)C(C)C(=O)N1CCC(C)(CNC(c2ccc(S(N)(=O)=O)s2)=O)CC1 c1(C(N2CCC(Cc3onc(C(C)C)n3)C(F)(F)C2)=O)ccc2n[nH]cc2c1 C1(CNC(C=Cc2cnc(C)s2)=O)CCCCC1N=c1cc(C(C)C)nc(Cl)[nH]1 CP(C)(=O)c1cnc(C(N2CCCC(CNC(c3ccc[nH]3)=O)C2)=O)nc1 C1(CC(=O)N(CCNC(c2sc(N(C)C)nc2C)=O)CC)OCCOC1(C)C C1(CC(N2C(C(N(CCn3ncc(C)c3)C)=O)CCC2)=O)CCCC(=O)N1 c1(C(N2CC(NC(c3c(COC)nn[nH]3)=O)C(O)CC2)=O)ccc(C)c(F)c1F N1(C(C(c2cccc(C)c2)C)=O)CCN(C(c2cccc(=S)n2O)=O)CCC1C C123CCC(CC1)(CC2)C(=O)N3.c1(C(N2CC3CCC2C3)=O)cc(F)ccc1Cl N1(C(c2c(C)n(C(C)C)nc2)=O)CC2CC(NC(=O)COC3CCCC3)C(C2)C1 c1(C(C(=O)OC)NC(C2CC2c2cnn(C)c2)=O)cc(F)c(Br)cc1OC c1(NC(C2CC2NCc2c[nH]c3cccc(Br)c23)=O)c(Cl)cc(Cl)cc1[N+](=O)[O-] c1(N2CCC(C(C)NC(c3ccc(CC)cc3)=O)C2)nc2cccc(C)c2o1 C1(NC(=O)COc2ccsn2)CCOC12CCN(C(=O)C1=CCCOC1)CC2 Cc1cnc2nc(C(=O)NC(CNC(c3n[nH]c(C(C)(C)C)n3)=O)CO)nn2c1 c1(NC(C(C(C)C)C)CNC(=O)C(n2cc(Cl)cn2)C)ccnc2ncnn12 C=CCCCC(=O)NCC(C)(C1CC1)NC(=O)C(C)Oc1ccc(OCC)cc1 c1(C(=O)O)cc2ccccc2cc1S(=O)(=O)N1CCSCC1c1nccs1 C(C(C)(C(C)C)NC(=O)C(n1cc(Cl)cn1)C)NC(C1(CCC)CCC1)=O c1(C(=O)NCCC(C)NC(=O)Cn2cnc(=N)[nH]2)ccc(C(F)F)c(F)c1 C1(NC(C2CCC(=O)N2)=O)CN(C(c2nccc(Cl)c2F)=O)CCC12CCC2 c1(C(=O)NCC(CNC(c2c(COC)noc2)=O)C)cn2ccsc2n1 C(=O)(C(CNC(=O)CC1(CC)CCC1)CCC)NC(CC#C)CC CN1CCC(NC(c2conc2CNC(=O)CC(=O)N(C)C)=O)C1 C=CC1(NC(C23CCC(NC(C4CCN(C)C4C)=O)(CC2)C3)=O)CCOCC1 c1(CCC)ccc(C(N2CCC(C(C)NC(C3CCO3)=O)CC2)=O)cc1 C(CCC1CCC1)(C(=O)N1CCC2CCC12)NC(C(C)OC)=O Cc1cc(Cl)c(C(N2CCOCC2CCNC(c2n[nH]cc2Cl)=O)=O)cc1C C1(NC(c2cnc(C(C)C)s2)=O)CCN(C(=O)CCC(C)CN(C)C)CC1CO c1(O)ccc(F)cc1.C1(N(CC(=O)O)CC)CCN(C(C)=O)CC1.C1(=O)CO1 c1(C(=O)NCCC2CC(NC(CN(C)C)=O)C2)ccc2nccn2n1 C1(CNC(C=CC(=O)N(C)C)=O)CCCCN(C(c2cc[nH]n2)=O)C1 CC1(C)CN(C(=O)CC(F)(F)C(F)F)CCN(C(c2cn[nH]c2)=O)C1 c1(CNC(CCNC(C(C)(C)c2ccno2)=O)=O)ccc(O)c(F)c1 Cc1nc(C=CC(=O)NC2CCN(C(=O)Cn3nccn3)C23CC3)[nH]c1C C(=O)(C1=NOC(C)C1)Nc1cn(-c2ccc(CCCCOC(C)=O)cc2)nn1 C1(C(=O)NC(C)(C)CC(=O)NCCc2cscn2)CCCC(C#N)C1 C1(NC(C2(CC=C)CCC2)=O)C=CCN(CC(=O)Nc2cncc(Cl)n2)C1 S(=O)(=O)(c1ccc(N2CC=C(Br)CC2)nc1)N1CC(C)CC(OC)C1 c1(CC(=O)NCC2C(NC(=O)CCN3CCOCC3)CC2O)csc(Cl)n1 N1(C(C(CC)OC)=O)CC(NC(c2cnn(CCN(C)C)c2C)=O)CC2(CC2)C1 C(=O)(C(F)(F)CCCC)N1CCC(N(CC#C)C(C2CCCCCN2C)=O)C1 Cc1cc(C(N2CCC(NC(C3CCS3(=O)=O)=O)C2C)=O)ncn1 c1(C(C)NC(CCCc2nnc(C)n2C)=O)ccc2ncsc2c1 N1(C(C(CCC)NC(C2(CC)CCOC2)=O)=O)CCc2cncnc2C1 [N-]=[N+]=NC1CN(C(=O)CC2CCN(C(c3cnc(S)nc3)=O)CC2)CC1O C(CN=c1[nH]c(N2CCC(OCC(C)C)C2)nc2c1CSC2)(CC(C)C)OC c1(C(N2CC(C)(NC(CN(S(CC)(=O)=O)C)=O)C2)=O)cn2c(n1)COCC2 C1(C(=O)NCCCN(C(=O)CCCNC(=O)OC)CC)CCNC(=O)C1 CCCC(C)CC(=O)NCC1CCCC1NC(C1CC(OC)CN1C(C)=O)=O c1(NC(C)=O)ccncc1NC(=O)CC1CCN(Cc2cnc(Cl)cn2)C1 C1(SCC(=O)NC2CC(NC(c3nc(COC)oc3)=O)C2)CCS(=O)(=O)C1 Cn1cc(C(N2CC3C(NC(=O)C=Cc4cnc[nH]4)C3C2)=O)c(Br)n1 c1(OCC=C)cccnc1C(=O)NC(CNC(=O)C(Cl)=CCl)C(C)C N1(C(c2cc(C(=O)OC)[nH]c2)=O)CC(=O)Nc2cnccc21 N1(C(C(=O)N(CCNC(C=CCN(C)CC)=O)CC)C)CCNC1=O c1(C(C(=O)NCC(C(C)C)NC(C2CC(C#N)C2)=O)O)ccc(F)c(F)c1 C1(NC(C2CCCN2CC(F)(F)F)=O)(CO)CCCN(C(C2C3CCCC23)=O)C1 C(=O)(C(F)(F)CO)NCc1scc(C(=O)NC(C)(C)COC)c1 c1(CC(N2CC=CC(NC(C(CC)COC)=O)C2)=O)cc(Cl)ccc1O C1(N(C(=O)CC(C)F)CCC)CCN(C(c2csnc2C)=O)CC1 CCC(C(=O)N1CC(Cn2cc(CCC3CCCO3)nn2)C1)c1cccnc1 c1(C(=O)NCC2CCN(C(C(CC=C)(F)F)=O)CC2C)cc2cccnc2[nH]1 C1(C(N2CC(O)(NS(C)(=O)=O)C2)=O)CN(C(=O)CCCn2cccc2)CCS1 C1(CNC(COCCN(C)C)=O)CCCN1C(=O)CCn1cncn1 N1(C(C2C(C)=C2)=O)CCCC2(CCN(C(c3cc(F)c(O)c(Cl)c3)=O)CC2)C1 c1(N2CCCC(NC(C3CC(C#C)(O)C3)=O)C2)ncnc2cc(C(C)C)nn12 CC1CC(NC(c2csc(C(C)(C)C)n2)=O)CN(C(c2ccc(Br)o2)=O)C1 N#Cc1c(C(=O)NCC2(NC(C3CSCC(=O)N3)=O)CCCCC2)cccc1F c1(COC)nc(C)c(C(=O)NCc2ncccc2CNC(=O)C(C)CC2CC2)s1 Cc1cnc(N(C)Cc2cnsc2)c(S(=O)(=O)NC2(CO)CC2)c1 c1(C(=O)NC(CC)C(=O)NCCN=[N+]=[N-])cc2ccccn2c1 C(=O)(CC(C)(C)c1cn(Cc2cnn(C(C)C)c2)nn1)NCCn1ncc(C)c1 c1(C(N2CCC3(NC(c4c(CC)cc[nH]4)=O)C(C2)C3)=O)cn2cc[nH]c(=O)c2n1 Cc1cnc2[nH]cc(CN3CCNCC3C(=O)NC(c3ccno3)C)c2c1 c1(C(=O)NC(CN(C(c2c(OCC)ccs2)=O)C)C)ccc(Cl)c(F)c1 CCCC(C)(CCC)C(=O)NC1CC(O)C1CC(=O)NC(c1cc[nH]n1)C CC(CC(=O)NCC1C=CC(NC(C2CC=CC2)=O)C1)c1cccnc1 c1(C(=O)NC2CN(C(c3cccc(CC#N)c3)=O)CC2O)nccc(Cl)c1F C1(NC(CCN(CCC)C)=O)CN(C(c2nn(C)cc2SC)=O)CCC1C c1(SC)ccccc1C(N1CCC(CN(C(=O)Cc2c(C)noc2Cl)C)C1)=O c1(C(N2CCC(CCC=C)(C(=O)NCCC(=O)NC)C2)=O)nccc2[nH]ccc12 CC1NC(=O)C=C1N1C(=O)N(C)C(CSCCS)C1 C1(C(N(C)CC2CCCN(C(c3ccc(SC)s3)=O)C2)=O)CCn2cncc2C1 C1(C(=O)NCCCCCNC(c2c(C)nc[nH]2)=O)COCC2(CCC2)O1 c1(CNc2c(C(N3CCC(C)CC3)=O)n[nH]c2)ccc2oc3ccccc3c2c1 N1(C(CC(C=C)C)=O)CC(C2CCCN(C(c3cc4c(C)n[nH]c4cn3)=O)C2)C1 c1(NC(C2CCN(C(C3CCCN(C)C3)=O)C2)=O)ccc(CO)c(F)c1 C#CCC(C)(C(=O)NCC1C=CCOC1)N1CC(C)CN(C(C(=O)OC)C)C1 C1(CNC(CCC#C)=O)CC(C(F)(F)F)CCN1C(c1cncc(C2CC2)c1)=O N1(C(CNC(=O)CCCCO)=O)CCC2(C1)CN(C(=O)Cc1ccccc1)C2 C1(NC(CS(C(C)C)(=O)=O)=O)C2CC3CN(C(c4ccc(F)c(O)c4)=O)C1C3C2 CCC(CC(C)C)C(=O)NCC1CC(O)CN1C(=O)Cc1cnc(C)s1 N1(C(=O)CC(C2CC2)C2CC2)CCC2(C1)CN(C(c1cnc3c[nH]nc3c1)=O)C2 C1(CNC(c2c(CC)nco2)=O)CCCCC1NC(=O)Cc1nc(C)cs1 C1(C(N2CC(NC(c3cc(Cl)nnc3O)=O)CC(C)C2)=O)CNC(=O)C(C)(C)C1 C12(NC(C(CC)N(CC)CC)=O)CCCC1N(C(=O)C(c1ccc(F)cc1)=O)CC2 c1(CC)cc(C(=O)N(C(C)CNC(c2sccc2F)=O)CC)nn1CCO N1(C(C2CCC(COC)C2)=O)CC2C(CNC(=O)Cc3cccn3C)C2C1 Cc1c(C(=O)NC(C)CNC(c2cnc(C(C)C)s2)=O)sc2cccc(F)c12 CC1(C)CN(C(C2CN3CCN2CC3)=O)CC1NC(c1cccc(CO)n1)=O c1(C(=O)Nc2n(CCCC)ncc2)ccc(-c2cncc(-c3cccs3)c2)cc1 C1(O)(C(C)NC(C2C(C(C)O)C2)=O)CCN(C(C2CCN(C)C(=O)C2)=O)CC1 CCCCCC(C(=O)Nc1cccc(NC(=O)C(C)SC)c1)C(C)C CC(C)C(C(C)NC(=O)CCCc1csc(=N)[nH]1)NC(c1nc(Cl)cs1)=O c1(C(N2CCC(C)(CCNC(C3CCCOC3)=O)C2)=O)cc2ncccc2s1 C1(OC)CC(CNC(=O)CCn2cc(Br)cn2)N(C(=O)CC2(C#N)CCC2)C1 C1(NC(c2c(OC)nccn2)=O)CCN(C(=O)CCC(C)(F)F)CC1OC C1(C(=O)N(CC)CC2CCCN2C(=O)C2=C(Cl)CC2)CCN(C2CCSC2)CC1 C1(C(=O)NC(c2nncn2C)C)CN(C(C2(C)SCCCS2)=O)CC1F C(=O)(C1=CC(O)C(NC(=O)C(C)NC=O)C1)N1CCOCC(=C)C1 c1(C(=O)NCC(C)NC(c2ccn(C(CC)CC)n2)=O)csc2nccn12 C1(CC)CN(C(=O)CCc2cc(F)ccc2F)CCN1Cc1ccc(C)cn1 Cc1noc(N)c1C(N1CC2CC1C2CNC(=O)CSc1ccc(F)cc1)=O C12(CC)CN(C(=O)COc3ccc(Br)cn3)C(CNC(=O)CCF)(C1)C2 C(C(C)C(=O)N1CC(CNC(=O)C=CCN2CCOCC2)(OCC)C1)OC C(CN=c1[nH]c(NC(CCC(=C)Cl)=O)nc(=N)[nH]1)NC(C12COC(CF)(C1)C2)=O N1(C(CC(C=C)(C)O)=O)CC(C)(CNC(=O)C(C(C)C)C(C)C)CC1(C)C CC(C)(CNC(=O)Cc1ccc(F)cn1)CCNC(=O)COCC1CCOC1 C(CC(C(=O)NCc1ccncn1)NC(c1ccn(C)c1C)=O)OC c1(C(=O)NCC2CCCN2C(=O)CC(O)C2CCCC2)cc(C2CC2)nnc1O n1(CC(=O)N(CCCNC(=O)COC)CC)cc(C2CCC2)nn1 c1(C(=O)OCC(=O)Nc2c(OC)ccc(NC(C)=O)c2)c(N)cc(F)cc1Br C1(C2CCN(C(=O)CCC3CCOC3)C2)(NC(c2nc(C)c(C)s2)=O)CC1 C1(NC(C2CC(N(C)CC)C2)=O)CCN(C(c2cccc(SC)c2)=O)CC1CO C1(C(=O)NC(C)(C)CC=CC(=O)NCC(O)CC2CCCC2)Cc2nccn2C1 C12(CCNC(c3nc(C)sc3)=O)CCC1CN(C(=O)COc1ccc(F)cc1)C2 Cc1cc(C)c(C(=O)N(CCC(C)NC(=O)CC2CCC(=O)N2)C)[nH]1 CC1CCOCCN1C(c1c[nH]nc1CNC(=O)CCC(C)(C)F)=O N1(CC(C(=O)OCC=C)NCc2ccco2)CCc2ccccc21 N1(C(C2CC(CCNC(C(C)NC(=O)NC)=O)C2)=O)CCN2C(=O)NCC2C1 c1(C(=O)NC23CC(CNC(C4CC(=O)NC4)=O)(C2)C3)cnn2ncccc12 c1(C(N(C2CCCN(C(CCC#C)=O)C2)CCO)=O)cc(Br)ccc1N N1(C(C2CC(N(C)C)C2)=O)CC2CCC1C2NC(=O)CN(C)S(=O)(=O)N(C)C CC(CCC(C)(C)C)C(=O)N1CCC2(C1)CN(C(C1CC(O)CN1C)=O)C2 c1(C(=O)OC(c2ncc(Br)cn2)C)ccccc1-c1nc[nH]n1 C1(NC(c2c(CNC(CCCSC)=O)cnn2C)=O)CC2C(C1)C2(F)F Cc1ccc(S(=O)(=O)N2CCN(C(=O)N(C(C)CC(F)F)C)CC2)cc1 CC1CC(NC(c2ncnc(O)c2Cl)=O)CCN1C(=O)CCCc1nncn1C C#Cc1cnc(N2CCC(CNC(C3CCC=CCCC3)=O)C2(C)C)nc1 C(C(=O)NCCCN(C(=O)Cc1cc(C(F)(F)F)n(C)n1)C1CC1)(C(C)C)SC Cc1nccnc1C(=O)NC(C)C(C)NC(c1cncnc1C(C)(C)C)=O N1(C(c2ccc(O)cn2)=O)CC2CN(Cc3ccc(O)c(O)c3)C2C1 N1(C(Cc2noc(C)c2C#N)=O)CCN(C(=O)C(C)C(F)F)C2(CCC2)C1 c1(OCC(=O)NC2(C3N(C(C(CC)O)=O)CCC3)CC2)cccc(OC(C)C)c1 c1(C(=O)NC2(CF)CCN(C(CC3OCC(C)(C)C3)=O)C2)coc2c1CCCC2 c1(OC)ncnc(CNCc2ccccc2-c2ccco2)c1OC C1(C(N2C(C(C)O)CC2)=O)N(C(=O)CC2CCC(=O)C2C)CCC1(C)C c1(N2CC3C(CNC(=O)C(C4CC4)C4CC4)C3C2)nc(Cl)nc2c1S(=O)(=O)CC2 O=C(CCCc1cnn[nH]1)NCC1CCC(NC(=O)Cc2n[nH]cc2Br)C1 Cc1cc(C(=O)NC2(C(=O)NCCC3CCCO3)CC2(C)C)nc(O)c1 c1(CC(C)OC(C2CCC(F)CO2)=O)ccc2c(c1)CCC(C)(C)O2 C#Cc1ccc(C(N2CCC(C)(CNC(=O)C(C)=C(C)C)C2)=O)cc1F C1(NC(C(C(C)C)OCC)=O)(CC)CCCN(C(=O)C(C)OCC(C)C)C1 N1(C(CCC2CC(OC)C2)=O)CCN(C(=O)C=Cc2cncn2C)C(CF)C1 C(N=c1[nH]nc(-c2ccon2)s1)C1(CCN(C(C2CCCC23CCC3)=O)CC)CC1 c1(OC)cccc(Cc2nc(-c3ncccn3)n(C3CCC(C)C3)n2)c1OC Cc1cc2[nH]c(=NC(C)CCNC(=O)CC3C=CCC3)c3ccccc3n2n1 c1(C(N2CC(CNC(C3=C(C)OCC3)=O)OCC2)=O)cccc2c(Br)ccnc12 c1(CNC(=O)NCC2CSCCN2Cc2ccccc2)ccc2c(c1)COC2 C(=O)(C1COc2ccccc21)NCC1(NC(CC2C(C)C2(F)F)=O)CCC1 N1(C(c2cc(C(N)=O)oc2)=O)CC2(CCN(C(c3cccc4nonc34)=O)C2)C1 C1(NC(c2n(COC)ncc2)=O)CC(C)CN(C(=O)CC2CC(SC)C2)C1 c1(CC(=O)NCCNC(CC(c2ccc(Br)cc2)C)=O)cc(O)nnc1O Cc1c(C(N2CCC(NC(=O)C(C3(O)CCCC3)F)C2)=O)cc(C2CC2)n1C C1(NC(c2cnsc2)=O)CC(F)CN(C(c2sccc2-n2ccnn2)=O)C1 N1(C(C(C)NC(C)=O)=O)CCCC(c2cn(-c3ncc(C)s3)nn2)C1 c1(C(=O)NCC2CC(NC(CC(CC)SC)=O)C2)cc2cccnc2o1 c1(CC(=O)OCC(n2cc(-c3cscn3)nn2)=O)c[nH]c2ccc(Cl)cc12.C(CO)S C(=O)(C1=CCCN(C(c2cc[nH]c2C2CC2)=O)C1)N1C(CN=[N+]=[N-])CC1 C(C)(CC)(CCNC(C1CC(CC)C1)=O)NC(c1c(CC)con1)=O CC(O)C(C(=O)NCC12CC(CCO1)C2)NC(c1cnc(S)nc1)=O N1(C(c2ccc(CC)o2)=O)CCC(NC(c2c[nH]nc2OC)=O)C(CO)C1 c1(CCC)cc(C(=O)NCC(C)N(C(=O)C=Cc2cccs2)CC)no1 CON(CCC(=O)NC(C)CCO)C(=O)C12CCC(C)(C1)OC2 N1(C(C2(OC)CCCC2)=O)CCCC(C2CCCN(C(c3cc[nH]c3)=O)C2)C1 C1(CC(N2CC(NC(CSc3n(C)ccn3)=O)C(O)C2)=O)CCCC(C)(C)C1 C1(N(C(C=NOC)=O)C)CCN(C(=O)C=Cc2ccsc2C(F)(F)F)CC1C c1(CC)cc2c(CC(=O)N(C3CCS(=O)(=O)C3)CC3CCCO3)csc2s1 C=CCC(CC)C(=O)N1CC(O)(C(C)NC(c2nc(-c3ccco3)sc2C)=O)C1 c1(CC(N2CCC(OC)(CNC(C3(Cl)CC3(C)C)=O)C2)=O)cc2ccccc2o1 CCC(O)C(C)C(=O)N(CCCN(C(=O)CC1CCN(CC(F)(F)F)C1)C)C C1(F)(CNC(C2CCC(C)(C)C2)=O)CCCN(C(C2(C)CC2(C)C)=O)CC1 O(C1CC2(CCC2)Oc2ccccc21)C(c1cc(OC)cc(CON)c1)=O C1(NC(CCCc2ccc(OC)cc2)=O)C2CC1CN(C(c1nn[nH]c1Cl)=O)C2 c1(C(=O)NC(C#C)CC2CCCC2)oc(CNC(C2CCC2C#N)=O)cc1C c1(C(N2C(C(C)NC(C(CC)F)=O)CCC2)=O)cnc2nc(C)[nH]n2c1=O O=C(CC(F)(F)c1ccccc1Br)NCCCN1CCCC1=O C1(NC(C(c2cccc(O)c2)C)=O)CCCN(C(=O)CC2CCNC2=O)CC1 c1(C(CNC(=O)OC(C)(C)C)N(C)C(=O)NCc2ccccn2)ccccc1F c1(NC(C(CC)N(C)C(C2CC=CCC2)=O)=O)ccc(C)nc1 N1(C(c2c(F)ccc(OC)c2)=O)CC2(C1)SCCC2NC(=O)CCC1CCCO1 c1(C(=O)NCCN(CC(C)O)C(c2cnn(C)n2)=O)c[nH]c2cc(C#N)ccc12 N1(C(COc2ccc(OCC)cc2)=O)CCN(C(=O)CCCC2CCC2)CC1C C(=O)(C1CCc2cccnc21)NC(C1N(C(CC(C)(C)OC)=O)CCC1)(C)C C1(C)(NC(C(C2CCC2)NC(c2n(C)ccn2)=O)=O)CN2CCC1CC2 N1(C(Cc2cc(CC)no2)=O)CC2(CCCC2NC(c2coc(Cl)n2)=O)C1 N1(CC(=O)NCC2C(NC(c3cn(C)nn3)=O)CCC2)CCOCC1=O C12(NC(c3occ(C)c3C)=O)CCC1CN(C(C1(F)CCS(=O)(=O)C1)=O)C2 N1(C(c2nc(OCC)oc2)=O)CCC(CNC(=O)C=C(CC)CC)(COC)CC1 CC1(NC(C2CC2[N+](=O)[O-])=O)CCN(C(=O)CSCc2cccnc2)CC1 N1(C(Cc2cnc(C)[nH]2)=O)CC2C(NC(=O)C(C)N(C)C)CS(=O)(=O)C2C1 c1(C(C)=O)c[nH]c(C(=O)NCC2CCCC2NC(=O)COc2cnn(C)c2)c1 C(CCCCC(=O)N(CC(C)CNC(c1cnc(O)n1C)=O)C)OCC c1(N2C(=O)CC(NCC(c3cn(CC)nc3)O)C2)ccc(Br)cc1C C(=O)(CCCCC(C)=O)NC1CC=C(C(=O)NC(CCCC)C)C1 N1(C(C2(C)CC2(Cl)Cl)=O)CCc2[nH]nc(CNC(C3CC4C=CC3C4)=O)c2C1 N1(C(CC2(OC)CCC2)=O)CC(N(C(=O)C(C)OCCC(C)C)C)C(C)(C)C1 Cc1nc(N)cnc1C(=O)NCCC1CN(C(C2CCCS2)=O)CCO1 C(N=c1nc(N2CCOC(C)CC2)c2sccc2[nH]1)C1N(C(C)=O)CCC1 C(=O)(C1=CS(=O)(=O)CCC1)NC1CCCC(NC(c2c(C)ncnc2)=O)CC1 N1(C(c2n(C)ncc2)=O)CCC(CF)(NC(C2CC23CC(O)C3)=O)C1 C#CC1(C(=O)NCC(c2cccc(C)c2)NC(C2(C)CC(C#N)C2)=O)CCCC1 N1(C(C2(C)C(C)CN(C(=O)CCCC3CC3)C2)=O)CCCC2(CCCC2)C1 N1(C(C2N(C(CN(C3CCC3)C)=O)CC=C2)=O)CC2CCCCC2C1 C(=O)(C(C)(C)CC(C)C)N(C)CC1N(C(c2cc(C)n(C3CC3)n2)=O)CCOC1 c1(CC(N2CCCC(NC(C3C(CCC)C3)=O)CC2)=O)ccc2c(c1)CCC2 CCC(C)CC(=O)NCC1(CNC(c2csc(C(C)(C)C)c2)=O)CCC1 c1(C(C)C)nnnn1CC(N1CCC1CNC(=O)Nc1nsnc1O)=O Cc1cccn(CC(N2CCC(NC(C3(n4cccn4)CC3)=O)C2C)=O)c1=O Cc1cc(C(=O)NCC2(CO)CCN(C(=O)CCN3CCOC3=O)C2)ccn1 O=C(NNc1ccc2ccccc2n1)NCC1Cc2ccccc2CO1 C1(CC)CCCC1(C)NC(=O)CCCC1CCCCO1 c1(C(N(CCCNC(=O)CCOCCCOC)CC)=O)csc(C)c1 N1(CCCc2occn2)CCc2c(ncn2C2CCCNC2)C1 N1(C(CCCc2cc(C)no2)=O)CCCN(C(C2CCO2)=O)CC1C c1(CNC(C(C)NC(C2C(C(=O)NCC=C)C2)C)=O)nncn1C c1(CN2CC(CC(=O)NCC3(C)CCC3)OCC2)cccc(Cl)c1O C(=O)(C(C)CC(F)F)N(CC(C(N1CCC(CC)(CO)C1)=O)(C)C)C C1(C(=O)NCC(C)CNC(=O)C=C2SCC(=O)N2C)CCc2cc(F)ccc2O1 C=Cc1cccc(CN2CCSC(C(=O)Nc3cc(O)nc(O)n3)C2)c1 c1(NCCC2CCC(NC(C3(C)CC3Br)=O)C2)ccc([N+](=O)[O-])c2cccnc12 C1(NC(C(C)NC(C2(CC=C)CC2)=O)=O)CCCN(C2CC2)C1 c1(C(=O)NC2CN(C(c3c(C)nc(N(C)C)s3)=O)C(C)(C)C2)cncc([N+](=O)[O-])c1 C1(C(=O)N(CCCCCNC(=O)COCCCF)C)(CC)CCCCC1 CCC(CC(=O)NC(C)CCCCNC(=O)CCN(c1ccncc1)C)OC C1(C)(CNC(COCC(=C)C)=O)CN(C(=O)CCSc2nccn2C)CCO1 C1(CNC(=O)C=Cc2cnc[nH]2)CC12CCN(C(c1nnc(O)nc1O)=O)CC2 C(=O)(CC(F)(F)C(F)F)N1CCCC(CCNC(=O)C(O)C(F)(F)F)C1 N1(C(C(C(C)(C)C)(C)C)=O)CCC2(CC1)CC(NC(=O)C#CC1CCCOC1)C2 N1(CC(=O)NC2CC(NC(C3N(C)C(=O)NC3)=O)C2)CC(C(F)(F)F)CCC1=O c1(CC)cncc(C(=O)NC2CCCC(N(C(=O)Cc3cnc[nH]3)C)C2)c1 C(CC(O)C(=O)NC(c1cncs1)C)NC(Cc1cnc(C)s1)=O c1(-c2cn(CCCN(C)C)nc2)nc(CC(F)(F)F)nn1CC1CCCCO1 CC(C)C1=NOC(C)(C(=O)NCC2COCCN(C(=O)C(F)=C3CCC3)C2)C1 N1(C(C(CN(CC)CC)F)=O)CC(C)(C)CC1CNC(c1ccc(Cl)cc1)=O CCC1=NOC(CC(N2CC=CC(C(=O)N(C(C)C)CC)C2)=O)C1 C(=O)(CCP(C)(C)=O)NCC(CCOC)NC(c1cc(C(C)C)ccc1C)=O c1(CC(=O)N(CC(C)(C)CNC(=O)C2=CCOC2)CC)cn2ccsc2n1 N1(C(=O)C=CC(F)(F)F)CCN(C(=O)C(C2CCOCC2)O)C(C2CCC2)C1 c1(Nc2cccc(NC(C)=O)c2C)cc(S(C)(=O)=O)c(Cl)cc1Cl C1(C)(NC(CN(C(c2c(C)scc2)=O)CC2CC2)=O)CCCC(C)(C)C1 c1(CC)ccccc1CC(=O)NCC1CCCCN1C(C1CC(=O)C1C)=O CN=S(C)(=O)c1cccc(C(N2CC(CCNC(=O)CCCNC(N)=O)C2)=O)c1 N1(C(CC(C)O)=O)CCCC(O)(CNC(c2cn(C3CCCCC3)nn2)=O)CC1 n1(CC)ncc2cc(C(N3CC(CNC(C4C(F)(F)C45CCC5)=O)C3)=O)cnc12 c1(C(=O)OC)ccc(NC(=O)C(F)(F)CC2CCCO2)c2ncccc12 C(=O)(C(CC)(CC)CC)NC1C(C(=O)NC(CC)C2CCC2)CC=CC1 N1(C(COC)=O)CC(O)CC1Cn1cc(COC(C)C)nn1 C12(C(=O)NC(C(=O)NC(C)CC3CC3)C3(C)CC3)COCC1C2 Cc1cc(C(=O)NCC23CCC2CCN3C(C2CN(S(N)(=O)=O)C2)=O)c(C)cn1 O=C(N=S1(=O)CCCC1)c1ccc2c(c1)CCO2 c1(C(=O)NCC(CNC(C(C)NC(c2ccoc2)=O)=O)F)cn(C)nn1 c1(CC)cnccc1C(=O)NCCC(=O)NC1CCSC1 CCC(C)(CCO)NC(C1CN(C(c2cc[nH]n2)=O)CC1OC)=O N1(C(C2C(C)OCC2)=O)CCCCC(CNC(c2cc(CO)ccc2Cl)=O)C1 N1(C(CCSCCC)=O)CC2CC(NC(=O)COCCCC(C)C)C(C2)C1 Cn1[nH]cc(C(=O)Nc2cccc(OC(=O)NCC3CCCO3)c2)c1=O N1(C(C(C)=O)C)CCC(O)CC1.c1(OC)nc[nH]n1 c1(CN=C(NCC2CCCC(C)(C)C2)NC2CCCCC2)ccc(C#N)c(Cl)c1 C1(NC(c2c(C(C)C)c[nH]n2)=O)CN(C(c2cc(C3CC3C)on2)=O)C(C)(C)C1 C(C)(C)(C(=O)NCCC1CC1(F)F)OCC(=O)N(C1CC(C(N)=O)C1)C c1(CN2C(CNC(C3(C)CCOCC3)=O)CCC2)ccc(F)c(I)c1 Cc1ccc(Br)nc1N(C1CCNCC1)C(=O)Cn1cc(C2CC2)nn1 CCC(=O)CCC(=O)NCC(C)(C)OCC(=O)NCc1ccccc1OC Cc1ccoc1CC(=O)Nc1nc(C2CCOC2)cs1 NC(=O)CC(O)C(=O)NC1CCCN(C(c2ccc(O)cc2Cl)=O)C1 CCS(=O)CC(=O)N1CCN(CC2CCCN(C(=O)Cn3ccnn3)C2)CC1 C(=O)(C(O)CC(F)(F)F)N1CCN(C(CCC=CCC=C)=O)C(C(F)F)C1 c1(C(=O)NC2(CNC(=O)CC3C=CCC3)CC2)cc(Br)c2n[nH]cc2c1 c1(C(=O)NCC2CC(C)N(C(=O)CCC(N)=O)C2)cnc2c(ccn2C)c1 N1(C(C2CCN(C(c3ccccc3)=O)C2)C(=O)NC)CCCC1C#N C1(C(N(C)OCc2ccccc2)=O)CC(O)CN1C(=O)CCCC1CC1 C=CCCCC(C(=O)NCC(C)C(=O)OCC)NC(c1ccsc1OC)=O C1(NC(C2CC3(CCCCC3)C2)=O)CC2CC(C1)N(C(=O)CCCCNC=O)C2 c1(C(=O)OC)ccc(N(C2CCCC2c2ccccc2)CCO)c(C#N)n1 C=CCCCCCC(=O)NCC=C1CCN(C(C2CC2(C(C)C)CC)=O)CC1 Cc1nn(C)cc1CC(=O)N(C1CCC(NC(C2C3COCC23)=O)CC1)C Cc1csc(CCC(=O)NCC2(C(C)(C)O)CN(C(c3cncnc3)=O)C2)n1 c1(C(C(=O)NCCN(C(C2COCCO2)=O)CC)C)ccc(C)cc1 C1(C(N2C(C)CC2CO)=O)CCOCCN1C(c1nc(Cl)cs1)=O c1(C(N(CC(CC)NC(C(CC)SC)=O)C)=O)c(C)nn(C)c1F c1(C(=O)NCCOC(C(CC)OC)=O)cc([N+](=O)[O-])ccc1OC(C)(C)C c1(CC(N2CC(NC(C3C(C=C)CC3)=O)C2)=O)c(C)cccc1Cl Cc1ccncc1C(N1CC2CC1(C(N1CCC(F)CC1)=O)C2)=O C=C(C)C(C)(O)C(=O)N1CCCC(CNC(c2sc(-c3ncc[nH]3)nc2C)=O)C1 c1(C(=O)NCC2(O)CC(NC(=O)CC3CCC3)C2)cccc2c1CCO2 CCCC(CC)CCC(=O)N1CCC1CCC(=O)NOCC12CCC(CC1)CC2 C(=O)(CCCC(F)F)N(C1CCCN(C(C2(CCOC)CCCC2)=O)C1)C C1(CCNC(c2cc(N(C)C)ncc2)=O)CN(C(c2csc(Cl)c2)=O)CCCO1 c1(CC)cc(C(=O)N(C2CN(C(c3c(C)ccn3C)=O)CC2O)C)c(C)o1 C(c1ccc(C)c(C)c1)=CC(N1CCN(C(CSC)=O)C(c2ccccn2)C1)=O C12(CNC(c3nc(C#C)sc3)=O)CC(CO1)N(C(=O)C(C)CC(C)C)C2 c1(C(N2CC(F)CC(NC(C3(C)C(C)C3)=O)C2)=O)cc(F)c(F)cc1O N1(C(C=C(COC)C)=O)CCC2(NC(c3cc(SC)oc3C)=O)CCCCCC12 c1(C(N(CCC(C(C)C)NC(c2c(C)[nH]cc2)=O)C)=O)cc2occ(Br)c2[nH]1 C1(CNC(=O)N(CC(C2CCCO2)O)CCO)CCS(=O)(=O)CC1 c1(C(N2CC3C(CNC(c4cnc(=N)[nH]c4)=O)C3C2)=O)cnc(O)c([N+](=O)[O-])c1 c1(C(N2C(C(C)NC(C(C(C)C)OC)=O)CCC2)=O)cccc([N+](=O)[O-])c1C Cc1csc(C(O)CC(=O)NCC(C)N(C(=O)C=Cc2ccsc2)C)c1 N1(C(COCC)=O)CCC2(CCC(NC(=O)CCNC(=O)C=CCl)CC2)CC1 CC1(C)C(CNC(=O)CC2=CCCC2)CCN1C(c1ccc(N)c(Cl)c1)=O Cc1ccn(CC(C)C(=O)NCC(C(C)C)NC(c2cocc2C)=O)n1 N1(C(C(C)N(C)C)=O)CCN(CCCCCNC(C2(CF)CC2)=O)CC1 Cn1ncc(Cl)c1C(=O)NC1CC12CC(NC(=O)CCc1ccncn1)C2 C1(NC(C(C)OCCOCC)=O)CC2CCC1N2C(=O)CCC1CC1(Cl)Cl c1(N(CC(=O)NC(C)C)C)nc2cccc(F)c2c(=NCC2(Cl)CC2(F)F)[nH]1 c1(CC(N2CC(O)(CN(C(c3[nH]c(=NC)sc3)=O)C)C2)=O)cccc2c1CCC2 CCCC(C)(CC)C(=O)N(CCCNC(=O)C(C(C)C)n1cnnc1)CC C(c1ccc(F)cc1)=CC(N1C(C2CCN(C(=O)CC(O)C3CC3)C2)CCC1)=O c1(C(=O)NC(CCCCNC(c2ccc(C)nc2)=O)C)cccc2oncc12 C(=O)(CC(O)C(C)C)N1C(CNC(CC(n2c(C)cc(C)n2)C)=O)C=CC1 N1(C(CNC(C)=O)=O)CCC(NC(=O)C(c2ccc(F)cc2)F)C(O)C1 C1(CNC(c2nnc(C)s2)=O)CC(C)N(C(c2nccc(C(F)(F)F)n2)=O)C1 c1(C(N(C(=O)C=CC2CCC2)CCNC(CC#N)=O)C2CC2)ccccc1 CCCCC(O)C(C)C(=O)NCCCC(CO)NC(=O)CC1(CSC)CC1 Cc1ccc(C(=O)NCCC2C(C)CCCN2C(=O)CN2CCSCC2)c(N)n1 CCC(CC(=O)N(CCCCCCNC(C1(C)CC1(F)F)=O)C)C1CCC1 N1(C(C(N2CC(C)C2)C)=O)C(CNC(=O)Cc2ccnn2C)CC2CCCC12 C(=O)(C(C(C)(C)C)N(C)C)NC(c1ccccc1)CNC(C1CC(N(C)C)C1)=O C1(C(=O)NC2(CNC(CNC(=O)NC)=O)CCC2)NC(=O)C2CC12 C1(CC(=O)NCCC2CCCC2)CCCN1C(c1cnn(C(C)C)n1)=O C1(NC(c2ccoc2Cl)=O)CCCCC12CCN(C(c1ccc(F)s1)=O)C2 C(=O)(C(CC(N)=O)NC(c1ccnc(C)n1)=O)N1CCCC(CCC#C)C1 c1(OC)cc(C(=O)NC(c2c[nH]ccc2=O)C)ncc1Br Cc1ccc(C2CC2)c(C(N2CCOC(CNC(=O)CCC(=O)N(C)C)C2)=O)c1 CCCCCCC(CC)(CC)C(=O)N1CC(NC(C2CS(=O)(=O)CC(=O)N2)=O)C1 C(=O)(C(CC(C)(C)C)OC)N1C(CCC)CN(C(=O)CN(C)C)CC1 C(=O)(CS(=O)C(F)(F)F)NCCCNC(c1cc(C)cc(F)c1)=O CC(C)C(C#N)C(=O)NCC1CCN1C(c1ccnn1CCF)=O C1(NC(C2CC23CC3)=O)CN(C(=O)C(F)=CC2CC2)CC12CCCC2 C1(CC)(NC(=O)C(C)CCO)CCN(C(c2ccc(F)c(SC)c2)=O)CC1 c1(C(N2CC(NC(c3cc(C)nn3C)=O)CC2(C)C)=O)ccc2nccn2n1 CC(C)C(C(=O)N(C(C)CNC(C1(C)CCSCC1)=O)C)c1cccnc1 C1(C)(NC(C2N(CC#C)CCC2)=O)CCN(C(=O)Cc2nc(C3CC3)cs2)C1 C(=O)(C1CCCc2c(O)cccc21)N1C2C(NC(CSC)=O)CC(CC2)C1 C(=O)(C1=C(CF)N(C2CCOCC2)C(=S)NC1c1ccc(Cl)c(O)c1)OC c1(C(=O)NCC(CNC(=O)CC2CC(n3cnnc3)C2)CO)cc(F)cc(Cl)c1 c1(C(=O)NCC2C(NC(c3c(C)cnnc3)=O)C2)c[nH]c(=O)c2ccncc12 C1(NC(c2c(COC)nn(C)c2)=O)CC2CC(C1)CN(C(=O)CC1CCC1)C2 C(=O)(C(C)CC(F)F)N1CCC(N2CCC(NC(c3cnc(C)[nH]3)=O)CC2)C1 Cc1cccc(OCC(N2CCC(CCNC(=O)CC34CCCC3C4)C2)=O)c1C c1(COC)nc2n(n1)CC(SC1CCC(=O)N(C)C1)CC2 N1(C(C(C(C)O)C)=O)CC2CC(C)N(C(c3cn(CCO)nn3)=O)C2C1 c1(C(N2CCN(C(c3ccc(C)o3)=O)CC2CC#N)=O)ccc(F)c(C)c1Cl N1(C(C(C)C2CC2)=O)CCC2CCC(C1)N2C(=O)CCSC1CCCC1 N1(C(c2cn(CC=C)nn2)=O)CCC(C)(C)CC1C(=O)NC1COC(C)(C)C1 c1(N2CC=CC(OC)C2)nc2c(c(=NCc3ccc(Cl)cc3Br)[nH]1)CC(C)CC2 CCC(C)CC(=O)N1CCCC1CN(C1CCN(C2CCC2)C1=O)C CC1(C)CC(NC(c2cc(C(N)=O)co2)=O)CCN(C(=O)C(O)C2CCC2)C1 c1(C(=O)NC(CCCC)CNC(c2snnc2C)=O)ccc(OC(F)F)cc1F N1(C(C2CCC(CNC(=O)CCc3nccs3)C2)=O)CCC(CC(N)=O)CC1 c1(CNC(=O)NC2CCCC2CO)c(Cl)cc(Cl)cc1Cl Cc1ccc(CC(=O)N(CCNC(c2ncc(N)cc2C)=O)C2CC2)c(C)c1 C1(NC(c2ccc(N)cn2)=O)CCN(C(=O)C=C2CCC2)CCC1(F)F c1(OC)ccc(Cl)c(C(=O)NC2CCC(F)(CNC(C3CCCCO3)=O)C2)n1 C1(CN(C)C(c2cccc(CCO)c2)=O)CCCCN1C(=O)CC1CC=CCC1 N1(C(CCC2N(C)CCC2)=O)CCCC(C)(CNC(c2ccccn2)=O)C1 N1(C(C2CCCC(=O)C2)=O)CCCCCC1CNC(=O)CC1CC=CC1 S(=O)(=O)(c1ccc(N2CC3CC3(CO)C2)c2cnccc12)NC(C=C)(C)C N1(CC)CC(C)N(C(=O)CC2(C=C)CN(C(=O)Cc3ccccc3C)C2)CC1C c1(N(C(c2cc(C(F)(F)F)ccc2Br)C(=O)NCC)C)cnn2c1OCC(O)C2 CCCCCCC(C)C(=O)NCC(C(C)(C)C)NC(c1c(Cl)n[nH]c1C)=O CC1(C)CCC(CS(N2CCCC2c2ccc[nH]2)(=O)=O)OC1 C=C(Cl)CCC(=O)NCC1C=CCN1C(c1cccc(C(C)(F)F)c1)=O C1(C(N2CCN(CCC)CC2)=O)CCN(C(=O)CCc2cncs2)CC1C C(=O)(CCCCC(N)=O)NC1(CCNC(c2c(C)cccc2F)=O)CC1 C(CN=S(C)(C)=O)NC(C(CO)NC(C(CC)n1ccnc1)=O)=O C1(C(=O)N(C2CC3CNC2C3)CCc2ccccc2O)CC2(C1)OCCO2 c1(C(=O)NC(CCNC(c2nc(CC)oc2C)=O)C)ccnc(S(N)(=O)=O)c1 N1(C(C2C(NC(Cc3nc(=N)[nH][nH]3)=O)COC2)=O)CC(O)C(O)C1 CC(C1Cc2ccccc21)NC(c1cnc(C(=O)O)c(Cl)c1)=O Cc1nn(CC(N2CCOCC2CNC(C2(CF)CCOCC2)=O)=O)cc1Cl C12(COC)CCC(C(N3CC(CNC(=O)C(C)(C)OC)C(C)C3)=O)(CO1)C2 N1(C(C2(N)CCCC2)C(=O)OC)CCc2[nH]c3ccc(F)cc3c2C1.OC C(C1CCCN1C)=CC(=O)NC1(CC(N2CCC(OCCNC(C)=O)C2)=O)CC1 c1(C(=O)NCCC(C)NC(=O)CCCCC(F)F)cn(C)c(=O)c2c1CCCC2 C(=O)(CCC(C)(C)[N+](=O)[O-])N(C(C(=O)N(C(C=C)C1CC1)C)C)C N1(C(C=CC=CCC)=O)CC=CC(NC(c2ccc(-c3nnc(S)o3)cc2)=O)C1 Cc1cc(C(=O)NCCCC(C)NC(c2ccnn2C2CCCC2)=O)cc(N)c1 N12CCOC(CC1)C2=O.c1(NC)cnccc1C(N1CC=CC(OC)C1)=O N1(C(C2(OC)CCC2)=O)CCC(CO)(CNC(=O)CC2CCCCC23CC3)CC1 c1(SCC)ccc(NC2CCC(COC(c3ccccc3)=O)C2)cn1 C1(NC(c2c(C)nns2)=O)CC2(C1)CC1(CC(NC(=O)CN3CCCCC3)C1)C2 CCC(C(=O)NCCSc1cc(C(C)(C)C)no1)NC(c1ccco1)=O N1(C(C2CCC(C)C2)=O)CCC(C2CN(C(c3ccsc3Cl)=O)C2)CC1 c1(C(N2CCC(F)(C(N3CC(C#N)OCC3)=O)C2)=O)ccc2scnc2c1 S(=O)(=O)(c1cncc(Br)c1)N1CC(C(=O)Nc2cc(F)c(Cl)cn2)C(F)(F)CC1 c1(N(C)Cc2cscn2)ccc(S(=O)(=O)N2CC3COCC3C2)cc1F CC1CN(C(=O)CCOCCNC(C2CC2F)=O)CC1O.C1CCO1 c1(C(=O)NC2C(C)CN(C(=O)C=Cc3ncc[nH]3)C2)cc(O)nc(O)c1 Cc1cc(C(=O)NCC(C2(O)CCN(C(c3cnnc(O)c3)=O)C2)C)c(C)s1 C(=O)(CC(C)CC(F)(F)F)NCC1(NC(Cn2c(C)c(Cl)cn2)=O)CCCC1 C(=O)(C1=NOC(C)C1)N(CC(C)O)CCNC(c1cccc(OCCC2CC2)c1)=O c1(C(=O)NC2CC(NC(c3ccccc3CN)=O)C2)ccc(F)cc1O c1(C(C)C)nn(C)cc1C(N1CC(NC(=O)Cc2cnc[nH]2)C(O)C1)=O C1(c2ccc(OC)cc2)(C(N2CC(n3cnc([N+](=O)[O-])n3)C2)=O)CCN(C)CC1 c1(-c2nnn(C(COCCOC)(C)C(=O)O)n2)ccccc1-c1ncn(CCl)n1 C(=O)(CCC(=O)NCC#CCNC(C1CCCN1C1CC1)=O)NCCC CCCC(O)CC(=O)NCC1CC(F)(CNC(=O)CC2CCCO2)C1 c1(CC(=O)N(CC(C)CNC(=O)CCc2ccccc2F)C)ccc(C#N)cc1 n1(CC(CCC)OC)c(-c2ccc(Cl)cc2)csc1=Nc1ccc(OC)cc1 c1(COCCOC)nc(-c2c[nH]nc2C)n(C2CCC2)n1 CCCCCC(F)C(=O)NCC1CN(C(=O)C(C)(C)C(O)CC)CCC12CCC2 N1(C(c2cc(C)[nH]n2)C(=O)NCC=C)CCCSCC1C c1(OC)cc(C(=O)NC(C)CCCNC(=O)CCc2cn(C)nn2)c(C)cc1O CC1CCOC(C(=O)NOCC(=O)N(C2CC2)CC2(C)CCN(C)C2)C1 C1(CCNC(c2ccc(OC)o2)=O)CN(C(C2(CC(F)F)CC2)=O)CC1C C1(CNC(CCc2nc(C)sc2)=O)CCN(C(C2CCCC2)=O)C(C)C1 N1(C(c2cscn2)=O)CCC2C(CCN2C(c2c(F)ccc(F)c2F)=O)C1 C(CCO)(CC(C)(C)C)Nc1cn(-c2c(F)ccc(C)c2)nn1.N12CCC1C2 CCCCS(=O)(=O)CC(=O)NCC=CCNC(c1cn(CCCC#N)nn1)=O N(C(=NCCc1cccs1)N1CCCC(C(F)(F)F)C1)C1CC(O)C1 C1(NC(CCS(C)=O)=O)CCC2(CCN(C(c3ccc(Cl)c(N)c3Cl)=O)CC2)C1 C(CSC)(CN=c1[nH]c2c(c(=NCCOC3CCS(=O)(=O)CC3)[nH]1)SCC2)OC c1(CC(C)C)ccc(CO)cn1.c12ccc(cn1)C(=O)NCC(C)n1cc-2nn1 N1(C(c2c(CC)cco2)=O)CCC(NC(C2(CC3CC3)CCC2)=O)C(CO)C1 C=CC(C)(C)CC(=O)NCc1ccccc1CN(C)C(c1cccnc1S)=O C1(CC)C(=O)NCCN1C(=O)C(C)(C)C(C)NC(c1nnsc1C)=O c1(OC)cc(C)cc(C(=O)NCC(C2CC2)NC(c2ccnnc2)=O)c1O c1(C(=O)NC2CCN(C(c3nc(C)n(C)c3)=O)CC2O)n[nH]c2ccc(Cl)cc12 C(CCC(CCC)NC(=O)Cc1cnsc1)NC(C(C=C)(C)C)=O CCCCC(C)(F)C(=O)N1CCC(O)(C(C)NC(c2ncc(C(F)F)s2)=O)CC1 c1(C(N2CC(C(CC)NC(=O)C(C)N(CC(F)(F)F)C)C2)=O)cnc(C)[nH]1 C1(NC(c2cnsn2)=O)CC2CCC(C1)N2S(=O)(=O)c1ccc(Br)s1 N1(C(C(C)N(C(=O)CCCC2CC2C)CCO)=O)CC2(C)CC1CCO2 CCCCCCC(C)C(=O)NCC1C(C)CCN1C(C1CCC1)=O c1(C(=O)NCC2CC2NC(C2(n3cncn3)CC2)=O)cnc2nccnc2c1 Cn1c2c(ccc1=O)C(NC(C1CCCC(C)(C)CC1)=O)CCC2 C1(NC(C2(C)CNC(=O)C2)=O)CC(F)(F)CC1NC(=O)Cn1nccn1 O=C1Cc2ccc(C(N3CC=CC3CNC(=O)C(F)CC3CCC3)=O)cc2N1 c1(OCC(=O)NC2CCC(NC(C(C)(C)CO)=O)C2)cc(Br)ccc1F N1(C(C(COC)C)=O)CC(OC)C(CNC(=O)C(c2cccc(OC)c2)(F)F)C1 CC12CCCCC1CN2C(=O)C(C1CCC1)NC(=O)C(F)CC1CCOC1 N1(C(C(CCCC)O)=O)CCC(C(=O)NCc2cc(F)cc(F)c2)=C(F)C1 c1(C(=O)NC(CNC(CN(CCCCCC)C)=O)C)ccc(Br)c(C)n1 N1(C(C2CN(C)C(=O)N2)=O)CC(=O)NCC1C(=O)Nc1cnn(C)c1 Cc1cc(C(=O)NC2CCC(NC(=O)C(C)NC(C3CCCCC3)=O)C2)sn1 S(=O)(=O)(c1cc(C)cnc1N1CCC(C)CC(C)C1)NCCC(CCC)O CC1(C)CN(C(C2(C)CC=CCO2)=O)CC(CNC(=O)CCc2ccsc2)O1 C(=O)(C1=CC(C)CC1)N(CCCNC(C1C(OC)(OC)CC1)=O)C c1(NC(C)=O)ccc(Cl)c(C(N2CC(O)(CCNC(=O)CC(C)C(F)F)C2)=O)c1 c1(C(=O)NC2(CNC(c3cnc(CCCC)s3)=O)CC2)cnn(CCC#N)c1C C12(CNC(c3cnccn3)=O)CCCCC1N(C(c1ncc(F)cc1F)=O)CC2 Cc1cc(C(c2nnnn2CC2CC2)O)cc(C)n1.C1CCOCC1NCC1CC1 N1(C(c2nc(C)n(C)n2)=O)CCC2(CCCCC2NC(C2CC3CCC2C3)=O)C1 C1(COC)(CNC(C2(C)CCOC2)=O)CCCN1C(c1cccnc1S)=O C(=O)(CC(O)C(C)C)NCC(C)NC(=O)Cc1ccc(-n2cnnn2)cc1 C1(NC(C2CCN(C)C2)=O)(CF)CCN(C(=O)C=Cc2ncc[nH]2)C1 N1(c2nnn(C)n2)CCC(C)(C)C(CNC(C2CCCS(=O)(=O)C2)=O)C1 c1(C(N(CCCCNC(=O)CC2NC(=O)NC2=O)C)=O)ccn(CCO)c(=O)c1 c1(CC(N2CCC(CNC(c3c(C)c(O)ccc3)=O)C2)=O)cccc2nc[nH]c12 Cc1cccc(C(N2CCC(O)(CNC(=O)CCC3CCN(C)CC3)C2)=O)c1O N1(C(C2N(C(C)=O)CCC2)=O)CCC2CN(C(c3c(C)nn(C)c3Cl)=O)CC12 c1(C(=O)NC(C)C(CO)NC(=O)Cn2nnc(=N)[nH]2)ccnc(C(N)=O)c1 N1(c2c3ncn(CC(CC)CCO)c3ncn2)CCc2c(F)ccc(Br)c2C1 c1(OC)ccc(-c2cc(C(N3CCC(N(C(C)CC(N)=O)C)C3)=O)no2)cc1 C1(C)(C(C)C)CN(C(C2(F)CN(C(=O)CC3CCOC3(C)C)C2)=O)CCO1 c1(C(=O)NCC2N(C(CCc3ccc(C)s3)=O)CC=C2)ccc[n+]([O-])c1 c1(-c2ccc(CCC)s2)cccc2c(CN3CCC(CC(C)C)CC3)[nH]nc12 c1(C(N2CCCCC(CNC(C3CC(O)C3)=O)C2)=O)ccc2ccc(Cl)cc2n1 c1(NC(c2cnn3c2CCC3)=O)ccc2occc2c1 c1(C(N2CCC(O)(C(C)CNC(=O)CN(C)C)C2)=O)cccc(F)c1N n1(CC(=O)NC2CC(NC(C3C(C(=O)OC)C3(C)C)=O)C2)nc(C)ccc1=O c1(CC)ccc(OC)c(CN2CC(C)CC2C(N2CCCC(O)C2C)=O)c1 c1(C(=O)NC2(CNC(COCCCC#C)=O)CC2)cc(Br)cs1 N1(C(CCC=C)=O)CCC(C)N(C(C2CCOC(CC)C2)=O)CC1 C1(C(=O)NCCOCCCNC(=O)OC(C)(C)C)CCCN1c1ccncn1 N1(C(C(CC)(C)C)=O)CCC(CNC(c2cccc(C)c2)=O)C(F)(F)CC1 CC1CC(CC(=O)NC2(C(N)=O)CC2)CN1C(c1cn(C2CC2)cn1)=O C(=O)(C(C)(C)CS(N)(=O)=O)N(CC(C)N(C(C=Cc1ncc(C)[nH]1)=O)C)C C1(NC(=O)Cc2ccsc2)COC2(C1)CN(C(c1cc(Cl)ns1)=O)C2 C1(CC(=O)Nc2cccc(O)c2Br)Oc2ccccc2NC1=O C1(C(=O)NCc2ncn(C(C)C)n2)C2CC2CN1C(c1cc(Cl)no1)=O Cc1c(C(=O)NCCC(O)CNC(c2c[nH]nc2C2CCC2)=O)cnn1C(C)C C(CN=c1cc(C)c(S(=O)(=O)NCC2CN(C)CCN(C)C2)c[nH]1)OCCOC C12(CNC(CSCC)=O)CCC(CC1)N2C(C1CCC(F)(F)CC1)=O C1(C(C)C)CN(C(c2cc(O)n(C)n2)=O)CC1C(=O)NCC1(C)CCCCO1 c1(NC(C2CN(C(C(=O)NC(C)C)=O)CC2C)=O)cccc(C2CC2)c1Cl c1(C(=O)NCCS(CC)(=O)=O)ccc(I)cc1F CC(C)CC(CC(=O)N(CC(C)C)C)NC(=O)CC1CCCCCC1 Cc1nn(CC(=O)NC2CCC(NC(=O)CN3C(=O)CCC3=O)C2)c(C)c1Br N1(C(c2nc(CC)sc2)=O)CC(NC(=O)C(C)NC(C2CCC2)=O)C2CC12 N1(C(c2cc(C)sn2)=O)CC=CCC1C(=O)NCC1CC(F)(F)CO1 C12(C(=O)NC(CN(C(c3c(C)n(C)nc3)=O)C)C)CCCN1CCC2 C(=O)(C(C)CCC(C)(C)C)NCC1OCCN(C(c2c(C)cc[nH]c2=N)=O)C1 C1(C(=O)NC(C=C)CO)CCOCCN1C(c1nocc1C)=O C(=O)(C1=CC2CC(C1)CC2O)NCCNC(c1c(CC)cccn1)=O N1(C(CCCNC(C(C)(C)C)=O)=O)CCOC2(C1)CN(C(=O)CC1(C)CC1F)C2 C1(CNC(C(C)OC2CCCCC2)=O)C2CC1N(C(C1CCCC(CF)C1)=O)C2 C1(CC)CCC(C)N(CCNc2cc(C(=O)OC)nc(C)n2)C1 CC1(CNC(=O)CCN(C(=O)CC2OCCCO2)C2CC2)COCCO1 CCC(C)(C)C(=O)C(=O)N1CCC(C2(NC(=O)C=Cc3cncc(F)c3)CC2)C1 CN1CCN(C(c2ccccc2Cl)=O)C(CNC(=O)CCCC(N)=O)C1 C(=O)(C1Cc2c(Cl)cccc21)N1CCC(C)(CNC(c2c(CC)cccc2)=O)C1 N1(C(C(CC)n2ccc(C3CC3)n2)=O)CCC(NC(=O)Cc2n[nH]c(C)n2)CC1C c1(CC)cc(C(=O)N(C(C)C(=O)NCC2C=CCOC2)CC)no1 C1(C(=O)NCC(CC)N(C(=O)CC(C)(C)SC)C)CC12CC2(F)F c1(C(N2C(C(C)NC(COCCCCC)=O)CCC2)=O)oc(C(F)F)cc1C N1(C(c2cccnc2S)=O)CC2CCN(C(C34C=CC(CC3)C4)=O)CC12 C1(C(=O)NCCC2CC(NC(c3cc(C(C)=O)on3)=O)C2)CC(=O)N(C)C1 N1(C(C(=O)N(CCCC)Cc2cc(-c3cccs3)on2)=O)CCC(C)CC1 CC1(CNC(C2(C#N)CCCO2)=O)CCN(C(=O)CCCn2ccnc2)C1 N1(C(C(C)C)=O)CCCC(n2cc(CNC(C3(C(F)(F)F)CCO3)=O)nn2)C1 N1(C(CN(C(=O)OC)C)=O)CC2=C(C1)CN(C(=O)CC1CCC(F)(F)CC1)C2 c1(OC)cc(-c2ccc(NC(C3CCC3)=O)cc2)c(OC)nn1 c1(C(N2CCOCC(NC(CCc3ccn(C)c3)=O)C2)=O)cc(S(C)(=O)=O)co1 n1(C(COC)C)cc(C(=O)N(C2CC(NC(c3ccc(C)cn3)=O)C2)C)c(C)n1 C1(F)(CNC(c2cncc(OC)n2)=O)CCN(CC2CNC(=O)CO2)CC1 Cc1cc(CC(=O)NC(C2CCCN2C(=O)CCCOCC2CC2)(C)C)ccn1 N1(CC(=O)NC2CN(C(=O)CSc3cccs3)C2)CCCCS1(=O)=O C1(NC(c2c(CC)ncs2)=O)CN(C(C2CCC(C)(C)O2)=O)CC1(C)C c1(CC(=O)NC2CCC(F)(CNC(C3CCCC3CF)=O)C2)ccc(F)c(F)c1 C12(CNC(C=CC)=O)CN(C(c3ccc4cc3-4)=O)CC1CCO2.O(C)CC c1(C(N2CC(N(C(C=C(C)C(C)C)=O)C)C(F)C2)=O)c[nH]c2c(Cl)cccc12 c1ccc(OCC)cc1C1CC1.C(=O)(CC(=O)C)NN(C)CC1CC1C(=O)OC Cn1nc(C2CC2)cc1NC(C1(C)CCN(C(c2ccc[n+]([O-])c2)=O)C1)=O CC1CC(NC(C2CC(N(C)C)C2)=O)CN1C(=O)Cc1cccc(O)c1 CC(N=[N+]=[N-])C(=O)N1C(C(=O)NC2CCC(O)CC2)CCC1C(C)C C(CC(C(C)(C)C)NC(c1c[nH]nc1-c1ccnn1C)=O)N(C(COCC)=O)C CP(C)(=O)C1CCCCC1C(=O)N(CCOC)Cc1ccccc1 c1(CCC(=O)NCC2(O)CC(NC(C(C)CO)=O)C2)cccc(C(F)(F)F)c1 c1(C(=O)NCC(C2CCCC2)NC(C2C(C=C)C2)=O)ccnc(CN(C)CC)c1 C=CCC(C)(CC)C(=O)N1CC2CC(NC(C3(SC)CCC3)=O)C(C2)C1 c1(C(=O)NC2C(NC(c3cccnn3)=O)C2)ccnc2c1CCC2 c1(C(=O)NC2CCCC2C(=O)N(C2CC2)CC2CCCCC2)cc(O)cc(F)c1 c1(C(=O)NC2C3CCN(C(C4(C5CC5)CCCO4)=O)CC23)cc2ncccn2n1 C1(COC)CCCCC1C(=O)NCc1cccnc1SC1CCC1.C12(CC1)CS2 Cn1nnc2c1CC(C(N1C3CCC1C(CNC(=O)CC1(C#N)CC1)C3)=O)CC2 c1(NC(=O)N(C2CC2)Cc2cccs2)ncnc2c1ncn2CCO C1(N(C(C2CC(CC)C2)=O)C)CCN(C(c2sc(C)nc2Br)=O)CC1 C1(O)(C(C(=O)NCCCCOC)NC(C2C(OCC)CC2)=O)CCCCC1 n1(CCC)ccc(C(=O)NCC2CCC(NC(=O)COCC(C)C)C2)n1 O=C(CCC1CCc2ccccc21)NCC12CC1CN(C(c1cocn1)=O)C2 N1(C(C2CCC(SCC)CC2)=O)CCC2(CC(NC(=O)CC3=CCCCC3)C2)C1 n1(CCC=C(C)C)cc(C2CCCN2C(=O)C(CC)N(c2ccccc2)C)nn1 N1(C(C2(C#C)CCCCC2)=O)CCC(CNC(=O)C=CC(=O)N(C)C)C(F)(F)C1 c1(OC)ncnc(OC)c1CN1CC2(CC(C(=O)Nc3cncnc3)C2)C1 C1(C(N2C(C)COCC2C)=O)C2C3CC4C1C2C34C(=O)NC1CCC(O)CC1 c1(OC)cccc(NC(=O)C=CC(=O)NC(CNC(=O)C(O)C(C)C)CO)c1 C(c1ccc(C(C)(C)C)cc1)=CC(=O)NCC(C)N(C)C(C1CCN(C)CC1)=O CC(=O)C(C)CC(C)C(=O)N1CCC1C(=O)NCC(C)(O)C1CCC1 C1(C(=O)NC2CN(S(C)(=O)=O)C2)(CC)CCCN1C(C1OCCC1(C)C)=O c1(OC)nc(N(C)C)ccc1NC(=O)Cc1ccc(Cl)c(F)c1 C(CC(C(=O)N1CCC1CC(=O)NCC1CN2CCC1C2)OC)OC C(=O)(CC(=O)NC(Cn1cncn1)C(=O)NCc1nn[nH]n1)OCC CCC(C)CCC(=O)N1CCCC(O)(CCNC(=O)Cc2cnn(C)c2)C1 c1(CNCC2(NC(c3c(CC)n[nH]c3)=O)COC2)c(OC)cc(OC)cc1Br CN1CC(C)(C)CC1C(N1CCC(Cn2cc(CCN3CCCCC3)nn2)C1)=O C=CCC(C)(C)C(=O)NCC=CC(=O)NC(C1CCCCO1)C c1(C(=O)NCC(CCOC)NC(C2CCNC2=O)=O)cc(C(F)F)ccc1Cl c1(C(C)=O)cc(C(=O)NC(C)CC(C)NC(C2(C)CC(C)(C)C2)=O)cnc1C CN1CCCC(NC(C2CCN(C(=O)CC3CC=CCC3)C2(C)C)=O)C1=O N1(C(C2C(CC)C2)=O)CCOC(C2CN(C(=O)Cc3cc(C)[nH]n3)C2)C1 c1(CNC(C(C)n2cccn2)=O)ccccc1CNC(=O)CC1CCC(=O)N1 N1(C(c2c(CC)ncs2)=O)CC2CC1C2NC(=O)CN(C)C(=O)C1CC1 c1(NC(c2cccnc2)C)ncccc1S(=O)(=O)NC1CC(C#N)C1 Cc1cc(C(=O)NC2CCC(NC(=O)Cc3csc(S)n3)C2)c(C)n1C(C)C c1(C(=O)Nc2cccnc2Cl)cnn2ccc(-c3cc(F)c(F)c(F)c3F)cc12 C(CCCC(=O)NCC(CCOC)NC(=O)CCC(C)N(C)C)OCC CN1CCC2(CCN(C(=O)CC3CC(C)(C)CN3C(=O)CCC3CCCC3)C2)C1 C1(CC(=O)NCC(CC)(C)NC(C2CCN(C)C2C)=O)CC(=O)NC(=O)C1 C(CS(=O)C(C)(C)C)NC(c1n(CC=C)nnn1)COC1CCC1 c1(C(=O)NC2CC2CNC(C2CC2(Cl)Cl)=O)ccn2c(O)nnc2c1 C1(NC(C(CC2CCOCC2)NC(=O)COCCF)=O)CCCC(F)C1 N1(C(CCCOCCC)=O)CC2CC2(CNC(=O)CC2CCNC(=O)C2)C1 c1(C(=O)NC2C(NC(c3cnc(CCC)s3)=O)CCC2)ccc2c(c1)CCCO2 c1(C(=O)NCCCC(C)NC(C(c2nc(C)sc2)=O)=O)cc2ccc(O)nc2s1 Cc1nc(Br)oc1C(=O)NC(C)CNC(=O)CCN(C)CCO C1(CCNC(=O)C(C2CCC2)C2CCC2)CC(N=c2cnc(F)c[nH]2)C1 c1(C(N2CC(CNC(C(CN(C)C)(F)F)=O)C(O)C2)=O)cc(Cl)ccc1O C(=O)(CCS(N)(=O)=O)NCCCCCCN(C)C(C1CC1(F)Cl)=O N1(C(c2coc(-c3ccsc3)c2)C(=O)NCC2CC2)CCCC2CCC(O)CC12 Cc1c(-n2cc(CC3(F)CCCN(C(=O)OC(C)(C)C)C3)nn2)cccc1Br CCC(C)CCCCC(=O)NCC(C1CC1)N(C)C(c1cc(Cl)c([N+](=O)[O-])[nH]1)=O N1(C(=O)CCCn2cc(CCc3nn[nH]n3)nn2)CCCNC(=O)C12CCC2 N1(C(C(CC)c2ccccc2)=O)C2CCC1C(NC(c1ccccc1C)=O)C2 C1(NC(CCN(c2ccccn2)C)=O)CN(C(C2CCC2)=O)C2(CCOCC2)C1 Cc1cnc(C(=O)NC2CCCC(CN(C(=O)CCCn3cccc3)C)C2)cn1 C1(CC(=O)N(CCNC(c2cc(COC)sc2)=O)C(C)C)CCCC1(F)F N1(S(C(C)C)(=O)=O)CCC2CCC(C1)N2C(=O)Cc1ccc2c(c1)CCC2 C1(NC(c2n[nH]c(C3CC3)n2)=O)(CO)CN(C(c2scnc2C(F)(F)F)=O)C1 N1(C(C(CCC2CCC2)NC(C(COCC)C)=O)=O)CCC(F)(F)C(F)C1 C1(CNC(C(CC=C)OC)=O)CC2(C1)CN(C(=O)CCCCCC)C2 CCC(CCC(=O)N1CC(CCn2cc(CC3(O)CCSC3)nn2)C1)OC N1(C(c2[nH]c(=N)sc2)=O)CCCN(C(c2cccc3cncn23)=O)CCC1 Cc1c(C(C)NC(=O)C(CNC(=O)Cc2cccnc2O)CC2CC2)cnn1C CN1CCC(O)(CNC(=O)COCCNC(C2CCOC2)=O)CC1 C12(NC(C3C(C)OC(C)C3C)=O)CCCC1CN(C(c1c(F)cccc1Cl)=O)C2 c1(C(=O)NCC(CNC(C=CC=CCCCCC)=O)O)cc(F)cc2cnccc12 C1(CC(N2CC(F)(CNC(CN3CCN(CC)CC3)=O)C2)=O)CC(O)C12CCC2 c1(C(C(=O)NC)N(C)CC2C3CNCC23)ccc(C#N)cc1Br CCC(CNC(=O)CC1CC2(CCC2)C1)(CC)C(=O)N1CCC(F)C1 C(=O)(CC(C)(C)C(=O)N1CCCC(C(C)(O)CNC(c2cnnn2C)=O)C1)OC N1(C(CN(C)C)=O)CC2C(CC(=O)N(C(=O)CCc3ccccn3)CC(C)C)C2C1 c1(C(N2CCC(C(C)(C)NC(C(C)OC)=O)C2)=O)cc2c(s1)CN(C)CC2 c1(NC(C(N2CCCCC(C)C2)C=C)=O)c(C)cccc1C C1(C(N(CC(=O)NCC#CCOC)CC2CC2)=O)C2(CC2)C12CC2 N1(C(C2(c3cc(C)no3)CC2)=O)CCN(C(C2CCC(C)C2)=O)CC1CCO N(C(=N)N1CC(O)CC(C)(C)C1)c1nn(C)c(=O)n(C)c1=O C=CCCCCCCC(=O)NCC1CCCN1C(=O)CNS(N)(=O)=O C(=O)(C1=CN(C(=O)OC(C)(C)C)CCC1)N1CC2C(NC(CSCC)=O)C(C2)C1 N1(CCS(CC)(=O)=O)CCN(c2nnc(CCC#N)n2CC(C)C)CC1 c1(C(=O)NCC2(O)CCN(C(CCCC(C)=O)=O)C2)ccc(S(C)=O)cc1 N1(C(C2C(C)CC=CC2)=O)C2CCCC1CN(C(C13CCC(C)(CC1)OC3)=O)C2 C1(C(N(CC(C)NC(c2c(C)con2)=O)C)=O)Cc2cc(F)cc(F)c2O1 C(C)(CCC(=O)NCCN1CCC(NC(=O)C=C2CCN(C)C2)CC1)OCC C(=O)(C(F)CC(C)C)N1C(CC)C(NC(=O)COC(C)(C)C)CC1 c1(OC(C)(C)C)ccc(Cl)c2c1CCCC2NCC1CCC(F)(F)CC1 N(C1CCCc2ccoc21)C(c1n(CCOC)nnn1)c1cnn(CC(C)C)c1 CC1(C)CC(C(=O)NC2CCCC(NC(=O)C=Cc3ccco3)C2)CC(C)(C)C1 N1(C(CC2CC(C(=O)OC)C2)=O)CCCC1CNC(c1scnc1C)=O CC1CN(C(=O)CCSCC(N)=O)CC1NC(C1CCC(=O)C1)=O N1(C(C(CC)COC)=O)CCN(C(=O)Cc2sccc2Br)C(C)C1 CC(C)C(CCN(C(=O)C(C)(C)C1CCOC1)C)NC(=O)Cc1nc(=N)[nH][nH]1 C12(NC(C3(C)C(C)CCC3)=O)CCC(NC(c3cnn(CCO)c3N)=O)(CC1)C2 C1(NC(C(C)CN(C)C)=O)CCC12CN(C(=O)CSc1cccc(F)c1)C2 Cc1cc(C(C)C)ccc1C(=O)NC1CCC12CN(C(=O)Cc1csc(=N)[nH]1)C2 C(C(=O)NNC(=O)c1ccccc1Cl)NCc1cc(SCC)ncc1 N(C(=NCc1ccccn1)NCc1nnc(-c2ccc(C)cc2)o1)C(CC)CC C(=O)(CCCCCC(C)O)NC1CN(C(c2ccc(C)nc2O)=O)CC1O S(=O)(=O)(c1ccc(NCC(O)CS(C)(=O)=O)c(Cl)c1)NC(c1c(C)nccn1)C C1(C(=O)NCC(C2CCC2)NC(C2(CC#C)CCCC2)=O)CCOC1C=C C(C)(C(=O)N(Cc1ccc(C)o1)OC)NC(COC)OC c1(C(=O)NC(C(=O)NC(C=C)C)CC2CCC2)cnc(O)n1CC C(CCCCC(=O)NCCc1cncc(C)n1)NC(C1(CC=C)CCCC1)=O c1(C(N(C2CN(C(=O)CC3(C(F)F)CC3)CC2(C)C)C)=O)ccc2[nH]ccc2n1 c1(C(=O)NC2CCN(C(C3C(OCC)CCC3)=O)CC2)cc(Cl)cc(F)c1F c1(OC)cc(F)ccc1-n1nc(C2CCOC2)nc1C1CC1c1ccnn1C C1(C)(CC)CCN(C(=O)C(Cc2cn[nH]c2)NC(=O)CN(C)CCOC)C1 CCC(CC(F)(F)F)C(=O)N1CCN(C(c2cnc(C#N)s2)=O)CC1COC c1(C(=O)NCCN(C(C2(C(=O)OCC)CCC2)=O)C2CC2)ccnn1C(C)C N1(Cc2cc(C)no2)CCC(NC(=O)Cc2ccccc2F)CC(C)(C)C1 O=C(CC1=CCCC1)NC1CCCC(NC(=O)C(F)CC2CC2)C1 CC(C)CC(C)(C)C(=O)NC(C)Cc1ccc(CNC(=O)C2CC2)cc1 C(=O)(CCCCC(F)F)NC1CCCN(C(C2(CC(C)C)CCNC2=O)=O)CC1 c1(C(N2C(CN(C(C(C)OCC#C)=O)CC)CCC2)=O)ccc(O)cc1C Cc1c(C(N2CC=CC(NC(=O)CC3CC4(CC4)C3)C2)=O)cnn1CC(C)C C=CCC(C)(C)CC(=O)NC1CC2CCC1(NC(=O)C(O)CC1CCOCC1)C2 CC1CCN(C(=O)CC2C=NN(C)C2=O)C(C(=O)NCC23CCCC2CCO3)C1 N1(C(C2N(C(=O)OC)CCC2)=O)CC2CC(C1)N(C(=O)CCN(C)CCO)C2 c1(C(N2CC(F)(CNC(=O)CN3CCS(=O)CC3)C2)=O)ccc2cccnc2c1 C(N=c1[nH]c(=NCCCC(C)C)[nH]c2c1CCC2)c1cccc(OC)c1 C1(C(=O)NC2C(NC(C(C)(C)OC(C)C)=O)CCC2)CCC(C)CC1 N12CCC3CN(CC13)C(=O)COCC2=O.c1(Oc2ccc(C)s2)ccc(Cl)cn1 c1(N2CC3(C(C(=O)Nc4c(C)c(Cl)c(Cl)cc4)C3)C2)[nH]cnc2nc(Br)cc1-2 N1(C(c2ccnn2C)C(=O)NCCOCC)CCc2c(C(=O)OC)cccc21 C(C(O)CF)N(C(=O)CNC(=O)COC(F)F)CC CC(=Cn1ccnn1)C(=O)N1CC(C)(CNC(=O)COCC(C)C)CC1(C)C CC(C)C(O)C(F)(F)C(=O)NC1CCN(C(c2cc3n(c2)CCSC3)=O)C1C c12cc(cc(O)c1)C(=O)OC2.C(=O)(C(O)C(F)(F)F)C1CC(CC(=O)OC)NC1 c1(C(=O)NCC(CN(C(c2c(C)cc(F)s2)=O)C)O)ccc(C)c(C)c1F C1(C2CC2)(C(=O)NCC2(C)C(C)CN(C(c3cc(CF)on3)=O)C2)CCOCC1 c1(OC)cc(C(N2CCC(NC(C34CC3C4)=O)C(F)C2)=O)ccc1O C1(NC(C=CC(CC)=CC)=O)CCN(C(C2CC(=O)N(C(C)(C)C)C2)=O)CC1O c1(C(N2C(CCOC)CN(C(C3CCCO3)=O)CC2)=O)ccc2n[nH]cc2c1F c1(CNC(CCNC(N)=O)=O)c(F)c(Br)c(F)c(Br)c1F C(C(O)C(=O)NC(C)(C)CCNC(C1CCN1S(C)(=O)=O)=O)SC N1(C(Cc2ccc(OC)cc2)=O)CCN(C(C2CC3(C2)CC(C)C3)=O)C2CC12 Cc1ccc(C(=O)NC2CCCC2NC(c2ccc(C(C)C)cn2)=O)cn1 c1(CC(N2CCC(NC(C(C)SC(C)C)=O)C2C)=O)cc(F)c(F)cc1F C1(OC)CC(OC)C12CCN(C(=NCC1CCC1)NCc1cc(C)no1)CC2 Cc1ccnc2nc(C(=O)NC(C)CCNC(c3ccn4ccccc34)=O)nn12 N1(C(=O)CCCC2CCOCC2)CCC2(C1)CN(C(C1CC(=C(F)F)C1)=O)C2 CCCCC(CCCC)NC(=O)CCCCCNC(C1(CO)CC1)=O C1(C(=O)NC2C3(CN(C(CC(CC)(C)C)=O)C3)CC2)CC2CCCC(C1)C2(F)F c1(C(=O)NCC2N(C(C(C)Cc3ccco3)=O)CCCC2)cc2cc[nH]c2cc1Cl C(c1ccccc1)(C(F)(F)F)=CC(=O)NC1COC2CN(C(=O)C(Cl)=CCl)CC12 N1(C(c2nc(C)sc2)=O)CCCCC(N(C)C(C2CC(N3CC(O)C3)C2)=O)C1 CCCCN=c1[nH]c(=NC(CC)C2CCCO2)c2[nH]ccc2[nH]1 Cc1ccnc(C(C)NC(=O)Nc2cccc(C(C)C)c2)n1 C1(COC)(NC(=O)CC2CCCNC2=O)CCN(C(C2(NC(C)=O)CCC2)=O)C1 c1(C(C)C)nnc(C(=O)NCCCC2CCCN2C(C2CC(=O)N2)=O)s1.C1CC1 N1(C(CCC(=O)NC2(c3cccc(OC)c3OC)CC2)=O)CC(C)OC(C)C1C C1(n2cnc(C)c2C(=O)O)CCN(C2CCc3c(F)cc(F)cc32)CC1 C1(C(N2CC(CNC(=O)CCc3cnoc3)C2)=O)(CO)CCCCO1 c1(OCCCCCC)ccc(CNC(=O)CC2(Cc3ccccc3)CCC2)cn1 S(=O)(=O)(c1[nH]c(=NCC2(C(F)(F)F)CCC2)ccc1Br)NCC1(N(C)C)CCC1 CCC(C)C(O)C(C)C(=O)NC1COCCC1C(=O)NCCCOCC(C)C C(=O)(C(=O)C(C)(C)C)NCC1(CNC(C(CC)F)=O)CCCCC1 C1(NC(=O)OCC)CCN(C(C2CCN(C(C3CC(C)(CC)C3)=O)C2)=O)C1 C(=O)(C1=CCCN(Cc2c[nH]nc2-c2ccccc2)C1)NCc1nc(C)sc1 C[S+](C)CCC(O)C(=O)NC1C2CC1N(C(c1cc(F)c(N)cc1F)=O)C2 c1(OC(C(=O)N(CC(C)(C)NC(Cc2nc(C)[nH]n2)=O)C)F)ccc(Cl)c(F)c1 CCCCCCCC(=O)NC1CCCC(C(N2CCCC(O)CC2)=O)CC1 C12(C(N3CC=CC(NC(C(C)NC(=O)NC)=O)C3)=O)CCC(=O)N1CCS2 C1(C(=O)NCCCOC)(CNC(c2ccc(-c3ccco3)nc2)=O)CC(C)(C)C1 N1(C(CCC2(C)CC2)=O)CCC2(CCCN(C(=O)Cc3ccc(Cl)nc3)C2)C1 CC(C)(C(=O)NCCOC1CCN(C(=O)CCc2ccncc2)C1)n1cnnn1 c1(C(=O)NC(C)CN(C(=O)C(F)(F)c2cscn2)C)cccc2c1OC(C)C2 CC1CN(C(C2(O)CCC2)=O)CC1NC(c1ccccc1CC(C)(C)C)=O c1(C(N(C2CCN(C(CC3(C)OCCO3)=O)C2)CC2CC2)=O)cc(F)cc(F)c1 N1(C(CCCC(=O)NC)=O)CCC(CNC(=O)CCCOC)C(F)(F)CC1 N1(C(C=C(C)C2CC2)=O)Cc2n[nH]cc2C1C(=O)N(C)CC1CCCN1C C1(CC(=O)N(CC)CC2CCCN2C(=O)Cn2nccc2C)CCNC(=O)C1 c1(CN(C(C(=O)NCC)CCc2cccc(F)c2)C)ccc(F)cc1 C1(NC(Cc2c(OC)ccc(F)c2)=O)CCC2(CC1)CC2NCC1CC1 CCC(CC(C)C)C(=O)NCc1ccc(C(=O)NCCOCC(N)=O)o1 c1(SC)nc(Cl)cc(=NC2(CNC(=O)CNC(C3CCC3)=O)CCCC2)[nH]1 n1(CC(=O)Nc2cc(Br)nn2C2CCCCO2)c(C2CC2)nc2ccccc12 C1(CNC(Cn2c(C)ccc2C)=O)CCN(C(=O)CCS(C)(=O)=O)C(C)(C)C1 c1(C2CCCN(C(C(C#N)C3CC3)=O)C2)ncc2n1CCCC2 Cc1ncc(C(=O)NCC2CCCC(NC(c3cc(F)cc(Cl)c3)=O)C2)cc1N N1(C(c2cnc(C(C)C)s2)=O)CCC(C)(NC(=O)C(C)OC2COC2)C1 C1(NC(C(CN(C)C)O)=O)CN(C(C2(NC(N)=O)CC2)=O)CC2(CCOCC2)C1 C(=O)(CCCC(=O)NC(C(=O)NCCOCC(F)(F)F)C(C)O)OC N1(C(c2nc(C)n(C(F)F)c2)=O)CCC(C)C(NC(=O)CSc2nncn2C)C1 c1(C(=O)Nc2c(C)cnc(O)c2)ccc2c(C)nn(C3=CCC(O)CC3)c2c1 CCCCC(CNC(=O)CC1C(=O)NN=C1C)NC(=O)C(C)=CC(C)(C)C N1(C(c2ncc(I)s2)C(=O)NCCCSCC)CCC(C)C(F)(F)CC1 N1(C(CC2(OC)COC2)=O)CCOCC1CCNC(c1cnc(C)[nH]1)=O CC(C(=O)N(C1CCCC1)CCNC(=O)CCCc1ccccc1)C(F)F C1(NC(COCCC=C)=O)COC2(CCN(C(=O)Cn3ncc(C#N)c3N)C2)C1 c1(C(=O)NC2CC(NC(C(C)OCc3ccoc3)=O)C2)ccc2n[nH]cc2c1 c1(CCOC(C2CC(C(F)(F)F)(OC)C2)=O)ccc(O)cc1F c1(NC(CC(C)N(C(c2c(C)ccnn2)=O)C)=O)ccc(Cl)nc1C C1(C(N2CCC(O)(CNC(C(C=C)(C)CC)=O)CC2)=O)CCS(=O)(=O)C12CCC2 C12(NC(CC)=O)CCCC1CN(C(c1n[nH]cc1Cl)=O)C2 C=CCCCCCCCC(=O)NC1(CNC(=O)C(C)CC(N)=O)CCCC1 CC1=C(C(=O)NC(C)(CNC(=O)CC2CCOC2(C)C)CO)C(C)(C)CCC1 c1(C(CNC(C=CC(CC)C)=O)N(C(=O)CCCSC)C)ccccc1 c1(OC)ccc(C(C)C)cc1C(N1CCCC(n2cc(C3CCC3)nn2)CC1)=O C1(CCC(=O)NCCCNC(C)=O)CCN(C(=O)CCc2ccc(F)cc2)CC1 N1(C(CC(C(C)C)C)=O)CCOC2(CCN(C(=O)CCN3CCOCC3)CC2)C1 c1(C(N2CCC(C)(CCNC(c3cc(Cl)no3)=O)C2)=O)cc(C2CC2)nnc1O C1(F)(CNC(=O)Cc2cnn(-c3ccccc3)n2)CCN(C(c2cncs2)=O)C1 C(=O)(C1=NN(CCO)C(=O)CC1)NC12C(CN(C(c3c(C)noc3)=O)C1)CCC2 c1(C(=O)NCCc2ncc(C)cn2)n[nH]c2c1CN(C(C1(O)CC(CF)C1)=O)C2 Cc1c(N)ccc(C(=O)NCC2(CNC(=O)Cn3nnnc3C)CCC2)c1F C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(CCNC(C(CC)(CO)OC)=O)OC CC(C)(CO)C(=O)NC1CC(NC(C2CCCN2C(=O)Cc2cccs2)=O)C1 C(C)(C(O)C(F)F)NC(C(C1CN(C(CC)=O)C1)O)=O CON(CC1CC1)C(=O)CC1CN(C(=O)Cc2ccc(O)nc2)CCC1C C=CCCC(C)C(c1nnnn1C1(C)CC1)NCCCn1ccnn1 C(=O)(C(O)CC(F)(F)F)NCC(C)(C1CCC1)NC(c1c(C)cccn1)=O c1(C(N2CC(O)(CN(C(C(C)n3ccnc3)=O)C)C2)=O)ccnc2[nH]ncc12 c1(CC(N2CC(C(C)NC(C3C=CCC3)=O)C2)=O)ccc(S(C)(=O)=O)cc1 CCCCC(CC)C(=O)NCC1C2CCC(C2)N1C(=O)COC1CCOC1 n1(CC#C)nccc1C1CCCCN1C(N1CCC(O)(CC(C)C)C1)=O N1(C(c2cccc(C)c2C)=O)CCC(NC(C23CC(F)C2C3)=O)C(C)(C)C1 CN1CCC(C)(CNC(C2(NC(=O)Cn3cnnc3)CCOCC2)=O)C1 CCCCS(=O)(=O)Nc1cnc(-c2ccccc2C(=O)N(C)C(C)C)cn1 CCCC(CC(C)C)C(=O)NC1(CNC(=O)CS(=O)(=O)CCO)CCC1 N1(C(CC=CC=C)=O)CCCC(C(C)NC(=O)CN(C2CCCCC2)C)C1 C(CCC)(C(=O)NC1CN(C(=O)CCN2CCN(C)CC2)C2CC12)=CCC Cn1cnc2c1CCCC2C(=O)N1CC=CC(NC(C2CCCC(F)(F)C2)=O)C1 C(N=c1nc(N2CCCC(CO)C2)c2c([nH]1)CCC2)c1scc(C)c1 C1(CC(N2CCC(C)(COC)C2)=O)CCCN(C(=O)C(O)CC(N)=O)CC1 c1(C(=O)NC(COC)CNC(=O)C(C2CC2)OC)cccc(F)c1F c1(OC)ccc(C)c(C(=O)N(CCCCNC(=O)CC23CCC(CC2)C3)C)c1 C1(NC(C2CC(C)(C)C2)=O)CC(Nc2cc(O)ncn2)C12CCC2 c1(C(C)C)ccc(S(=O)(=O)NC2(C)CCOC2)cc1 C1(CC(=O)N(CC(CC)NC(c2ccc(C(C)C)cc2)=O)CC)CCC12CCC2 C1(NC(C(COC)O)=O)CC2CCC(C1)N2C(c1ccccc1SC(F)(F)F)=O N1(C(C(=O)Nc2ncn(C(C)(C)C)c2)=O)CCCC(c2cc(F)cc(F)c2)CC1 c1(C(=O)Nc2nc(-c3ccnnc3)cs2)c(F)cccc1Br c1(C(N(C2CCN(C(C(C)OC3CCCC3)=O)C2)C)=O)cccc(CO)c1 c1(NCCNC(COC(c2c(C(C)C)ocn2)=O)=O)ccc(Cc2scnc2C)cc1 Cn1c(=O)c2cc(C(=O)NCCOCCNC(C3CC3CF)=O)sc2n(C)c1=O N1(C(C(F)=C(C)C)=O)CCC2C(C1)NC(=O)CN2C(=O)Cc1csc(C2CC2)n1 c1(C(=O)NC2CCN(C(c3cc(Cl)c(Cl)s3)=O)C2)c(F)cc(F)cc1Cl C(=O)(CC(C)(C)NC(c1cccc(Cn2ccnc2C)c1)=O)NC N1(C(Cc2ccc(C)s2)=O)CCC2C(CCN2C(c2cnn(C)c2C(F)F)=O)C1 Cc1nc2c(o1)CCCC2CC(=O)NCC1(NC(=O)CCC2CCCO2)CCC1 C(=O)(C1=CCCSC1)N(C)CC1CCCN(C(c2ccn(C(F)F)n2)=O)C1 c1(C(=O)NCC2(F)CC(NC(C3CC3c3ccsc3)=O)C2)cc(F)cc(Cl)c1O C1(C(=O)NC(C)CCNC(=O)CC2CSCCS2)CCCC2CCCN12 N1(C(C(F)OC)=O)CCC(CNC(=O)C(F)(F)C2CC2)C(C)C1 Cn1ccc2ccc(C(=O)NC3CCCCN(C(C4C=CCC4)=O)C3)cc12 N1(C(c2cc(OC)ns2)=O)CCC2(CC1)CC(NC(C1C3CC4C(C3=O)C14)=O)C2 C1(CNC(C(C=CC)O)=O)CN(c2ncc3ccccc3n2)CCC12CCC2 c1(NCC=CCCOC)ncc(S(=O)(=O)NCCS(=O)CC(F)(F)F)cc1Cl C12(CCNC(C3CC(F)(F)C3)=O)CCC1CN(C(C1(CO)CC1)=O)C2 c1(CC(=O)N(CC)CC2CCCN2C(C2(CCOC)CC2)=O)c(C)noc1Cl Cc1ncccc1C(=O)N(CCNC(=O)CCC1CCCCO1)C1CC1 CC(C)CC(C(=O)NCC1CN(C(c2nnc3ccccn23)=O)C1)C(N)=O c1(C(=O)NC2(CN(C)C(C3C4CS(=O)(=O)CC34)=O)CC2)csc(S(N)(=O)=O)c1 C1(CC(=O)NCC2(COC)CN(C(C(CC)OC)=O)C2)CCCC(C)(C)O1 N1(C(C2CC(C(C)C)C2)=O)CCC(C(=O)NCC2(C)CCOC2)=C(F)C1 CC1CCCN1CC(=O)NC12CC(C(N3CCC(CO)C3)=O)(C1)C2 N1(C(c2ccc(CN(C)C)[nH]2)=O)CCN(C(=O)COCC2CCCO2)C(CF)C1 C12(NC(C(C)C3CCOC3)=O)COC(CNC(C3CC(O)CN3C(N)=O)=O)(C1)C2 C1(C(=O)NC(CCNC(c2c(C)[nH]nc2Cl)=O)(C)C)CC2(CCC2)CO1 C12(NC(C3CN(C)C(=O)N3)=O)CCC(CC1)N(C(c1cc3ncccc3s1)=O)C2 c1(C(=O)NCC(CNC(c2n(CC#C)ccc2)=O)OC)ccc(OC)cc1O C1(C)(CNC(C(CC)OC)=O)CCN(C(c2cn(C(C)C)cn2)=O)CC1 C1(C(=O)N(C2CC(C)(C)C2)C)(CC)CCCN1C(C1C=CCS1)=O Cc1nc(S(=O)(=O)N2CCC3CN(C)CCC23)sc1Br C1(CC)CCC(C)CN1C(=O)CC1CCCN1C(c1cnsc1)=O CN1CCC(C(=O)NCC2CC(NC(=O)CN3CSCCSC3)C2)CC1=O N1(C(C(CCC)N(C)C)=O)CCC(C2(NC(c3cnc(Cl)c(Cl)c3)=O)CC2)CC1 C1(NC(CSC(C)C)=O)CCN(C(c2cccnc2SC(F)F)=O)CC1C(C)C N1(C(c2c(CC)noc2C)=O)CCC(C2CN(Cc3cc(Br)ccc3I)C2)CC1 Cc1[nH]c(C)c(C(=O)NCC(C)(C)NC(=O)C(O)C(C)C)c1C N1(C(C2C(C(=O)OC)C2(F)F)=O)CC(C)(C)CC1CNC(=O)CSC(F)F c1(SCNC(C2C3(CC3)N2C)=O)ccc(Br)cc1.C1(CCCOC)C=CCC1 C(=O)(CC1=NN(c2cccc(Cl)c2)C(=O)C1)NC1C(CNC(C(C=C)O)=O)C1 C(CCC(C)(C)C(=O)NC(CCO)C(F)F)NC(C(C)Cn1ccnc1)=O c1(C(=O)NC2CN(C(C(C)(C)CC3CC3)=O)CC2F)ccc(C2CC2)cc1F CCCCS(=O)(=O)NC(C)C(=O)NCC(CC(C)C)NC(C1(CO)CC1)=O c1(N(CCC)CCNC(c2cncc(F)c2)=O)ccc([N+](=O)[O-])c(SC)c1 c1(C(CN2CCN(CCOC)CC2)=O)c(C)nc2ncnn2c1C.N12CCCC1C2=O C1(NC(C(C=C)C)=O)CN(C(=O)C(C)(C)COCC)CC1CO CCCCCCC(CC)(CC)C(=O)N1CC2CCC2(NC(c2nnsc2C)=O)C1 C12(CC)CCC(C(=O)NC3CCC(CNC(=O)CC4OCCC4C)C3)(CC1)CO2 CCCCCC(C)CC(=O)N1CCC(COC)(NC(c2scnc2C2CC2)=O)C1 Cc1cc(C#N)cc(C)c1C(c1nnnn1C1(C)CC1)NCCCCS(C)=O c1(CN(C(c2cccc(F)c2I)C(=O)NC)CCC)ccc(F)cc1F C1(CC=C)(NC(=O)Cn2cnc(Br)c2)CCCN(C(=O)C(COC)OC)C1 c1(C(C(=O)NCCC2CC2)N(C)CC)cn2c(F)cccc2n1 c1(C(C)C)ccc(F)c(C(=O)NCC2CC(F)CN2C(=O)Cn2cccn2)c1 c1(C(N2CC3C(CNC(CN(CC)CC)=O)(C3)C2)=O)ccc(C)cc1OC c1(CCCNC(CCC)(C)c2nnnn2-c2ccccc2)ccccc1C N(C(=NCC1CC1)NCc1ccco1)CC1N(CC)CCC1 CCC(C(=O)NCC(CNC(=O)CC1CCN(C)CC1)OC)C(C)(F)F c1(SC)nccc(N2CCCC2C(=O)NC(CC(C)C)c2ccccc2)n1 c1(C(=O)NCC(CC=C)NC(c2ccc(OC)c(F)c2)=O)cc(C)c(CO)cn1 CCC(C(=O)OC)C(=O)N1CCCC(CCC(=O)NCc2nn(C)c(=O)n2C)C1 c1(OC)cc(CO)ccc1NC(=O)CC1CCCN1Cc1ccc[nH]1 Cc1nc(S)sc1CC(=O)NC1COCCC1NC(=O)C=CBr O=C(O)CN1C(=O)COc2ccccc21.C1(CO)C(=O)N1CCc1ccccc1 N1(C(C2(CC)CC(C)(C)C2)=O)CCN(C(c2cn(C)nc2CN)=O)C(C(C)C)C1 N1(C2C(NC(CCN(CC)CC)=O)COC2)CCN(C(c2nn[nH]c2Cl)=O)CC1 c1(OCC)ccc(-c2cc(C(=O)OCC3CCC(C)(CC)O3)n(C)c2)cc1F c1(NCC2CCCC(NC(C(C)(C)C(F)F)=O)C2)ncnc2[nH]cnc12 C1(NC(CCCOCC=C)=O)CCC(=O)NC1c1ccnn1C c1(C(N(C2CCCCC2N(C)C(C2CCN(C)CC2)=O)C)=O)cc(Cl)nc(=N)[nH]1 C1(C(=O)NC(CCC)CNC(c2cncnc2)=O)CCn2cncc2C1 C12(C(=O)NCCCN(C(C3ON=C(CC)C3)=O)CCO)CCCC1OCC2 CCC(C(=O)NC(C(=O)NC1(C)CCSCC1)C(C)OC)C(C)(C)CC C12(C(=O)NCc3scc(C)n3)CC(CN(C(c3cc(C#N)oc3C)=O)C1)C2 N1(C(CNC(CC)=O)=O)CCC2CCN(C(=O)COc3ccc(F)cn3)C2C1 Cc1cccc(C(=O)NC(Cc2ccco2)C(=O)NC(CCO)C2CC2)c1N Cn1cc(F)c(C2CCN(C(=O)CC(c3cccc(C(F)(F)F)c3)N)CC2)n1 N1(C(CC(C)SC)=O)CCC(C2CCN(C(=O)CC(C)CC(C)C)CC2)C1 Cc1cc(=NC(=O)C2COCCC2NC(=O)C(C)C(F)F)[nH]n1C C1(C(C(=O)NCCOCC)N(CCC(F)(F)F)CC#N)C2COCC12 c1(C(=O)NC(C(C)NC(C2CCC(F)(F)C2)=O)(C)C)cc(Cl)c2c(c1)OCO2 C12(CNC(C(C)CN(C)C(c3cnn(C)n3)=O)=O)CCCC(CO1)C2 c1(C(C)NC(=O)CCC2CCC(NC(=O)C(C)(C)n3cncn3)C2)cccnc1F C(=O)(CC(C)(C)CC(=O)NC1CN(C(=O)C=Cc2cccc(F)c2)C1)OC Cc1cc(-c2noc(-c3cc(Br)cs3)n2)c(C)o1 C(=O)(CC1=CCN(C(=O)CS(=O)(=O)CCOC)CC1)NC1(CC)CCOCC1 C1(NC(c2c(CC)scc2)=O)CCCN(C(C2(C)CCCC2)=O)C1 c1(C(=O)NC2(C3CCCN3C(C3CC34CCC4)=O)CC2)cc(C2CC2)ccc1Cl C1(CN(C)C(c2cc(=O)n(C)o2)=O)CCCC(NC(=O)C=Cc2ccoc2)C1 c1(CC)occ(C)c1C(N1CCC(CO)(NC(=O)CCc2nc[nH]n2)C1)=O N1(C2C(C(C)(C)C)OCCC2)C(=O)NC(c2ccc(N3CCCC3)cc2)C1=O c1(C(N2CC(N3C(=O)CC(NC(=O)Cc4ccon4)C3)C2)=O)csc(=NC2CC2)[nH]1 CCC(CC)C(CNC(c1cc(C2CC2)[nH]c1C1CC1)=O)CO N1(C(=O)CCC2CCOCC2)CC=C(C(=O)N2CCC(O)CC2C2CC2)CC1 C(=O)(CC1=CCCCC1)N1CCCC(NC(CCC2CCC(C)O2)=O)(CO)C1 c1(C(N2CCC(N(C(=O)C=C3CCOCC3)C)C2)=O)c(Br)ccc(F)c1N N1(C(c2c(CC)noc2)=O)CCC(C)(C)C(C(=O)NC(c2c(C)n[nH]c2C)C)C1 CCC(CC)N=C(NCC1(N(C)C)CCCCC1)NC1CCn2c(C)cnc2C1 Cc1cn2cc(C(=O)NC3CCN(C(=O)CCn4cccn4)CC3(C)C)sc2n1 C1(CNC(C2CC(C)(C)O2)=O)CCCCN1C(=O)CSCc1ccccc1 N1(C(COC2CCN(C(Cc3c(C)scc3)=O)C2)=O)CCC2CN(C)CC2C1 C(CCC(=O)N1CC(CCCCNC(=O)Cc2ccsc2)C1)SC c1(CC)nc(C(=O)NCC(C2CC2)N(C)C(C2C(C(F)F)C2(C)C)=O)co1 c1(C(=O)NC23CC2CN(C(c2cnn(C4CC4(F)F)c2)=O)C3)cc(Cl)ccc1O C12(CCOC)CCN(CC1)CC(=O)N2.C(=O)(C(C)C1CCC1)NC(C)C N1(C(CC(C=C)C)=O)CC2CCC(NC(=O)C=C3CCC(C)CC3)(C2)C1 C(=O)(CC(F)(F)C(F)F)NC(CC)CN(C(C1(C(=O)OC)CC1C)=O)CC N1(C(CC2(COC)CCCC2)=O)CC(NC(c2cnc(C)nc2C)=O)CCC1C N1(C(C(NOC)=O)=O)CC2CC(C(N3CC(OCC(C)C)C3)=O)C(C2)C1 c1(C(C(=O)NCCOCCN(C(COC(CC)C)=O)C)C)ccncc1C C1(C(C)NC(=O)CCF)CN(C(c2cccn2C2CCCC2)=O)CCO1 C(C(COC)CC(=O)NCC(C)(C)CNC(C12CC1CCC2(F)F)=O)OC C(CC(C)C(=O)N1CC(O)CC1C(=O)NCc1snnc1CC)=CCC CC(C)(C)CC(O)CNC(C1CC(CCNC(=O)C=CCF)C1)=O C12(CNC(c3cnn(C4CCOC4)n3)=O)CC1CN(C(C1CSC1)=O)C2 N1(c2cc(C#CC)cc(Br)c2)CCn2ncc(S(C)(=N)=O)c2C1 c1(C(N2C(C)C(NC(=O)CNC(c3ccco3)=O)CC2)=O)cccc(F)c1F c1(C(=O)NC(CNC(c2ccccc2OC2CCC2)=O)CO)cc2cscc2s1 C1(CC)CC(OC)CN1C(=O)C(N1CCN(c2ccccc2OC)CC1)C CCCC(C(=O)NCCN(C(=O)C(C(C)C)n1cccc1)C)c1ccc(Cl)cc1 c1(CC)cc(NC2CC3CC2CC3C(=O)O)cc(CC)c1 c1(SCCC(=O)NC2C=CC(NC(=O)C3CC3)C2)ncnc2[nH]cnc12 C(=O)(C(CNC(C1(OC)CCOC1)=O)CC(C)C)N(CC(C)OC)C C1(NC(CN2CCN(C)CC2)=O)CC2CC(NC(=O)Cc3nn(C)cc3Cl)CC12 n12cnc(c1)NC(=O)C1(CC1)C(=O)NCC2.C12(CSC)CCCC1C2 N1(c2ncc(CCC)cn2)CCC(NC(c2snnc2C)=O)C(F)C1 N1(C(C=CSC)=O)CCCC2(C1)C(NC(=O)CCc1cnc(C)o1)CCN2C C(=O)(C(C)(C)C(C)(C)O)N1CC2C(C(N3CCC(C(=O)OCC)CC3)=O)C2C1 C1(CN(C)C(C2CCCC2CNC(C2(n3cccn3)CC2)=O)=O)CCCC2CC12 c1(NC(CN(c2ccco2)C(N(CC(C)C)C)=O)=O)ccc(Br)cc1 CC1CC=C(C(=O)N2CC=CC2CNCCn2cc(F)ccc2=O)CC1 C1(C(=O)NCCN(C)CCNC(=O)CCc2ccco2)CCCO1 C1(CNC(C2(C)CC(F)(F)C2)=O)COCC2(CCN(C(=O)C=CBr)CC2)O1 N1(C(C(C(C)O)NC(C(C(CC)C)N(C)C)=O)=O)CCOCC(C)(C)C1 c1(C(N(CC(C)O)CCNC(c2cnns2)=O)=O)ccc2nccn2c1 N1(C(C(=O)N(CCNC(CN(CCC#C)C)=O)CCC)=O)C(C)CCCC1C CCCC(C)CC(=O)N1CCCC1CN(C(c1ccc(CSC)o1)=O)CC Cc1cc(C(N2CCOCC2CNC(C23CC(C)(CO2)C3)=O)=O)nc(C)n1 c1(NC(c2ccc(N(CC)CC)nc2)=O)cc(C)c(C)cc1C(=O)OC c1(C(N(C(CN(C(Cc2c(C)con2)=O)C)C)C)=O)ncnc2sccc12 C1(C)(C(=O)NCCN(CC(c2ccccc2)C)C)CCCN1C(N)=O CC1CN(C(c2ccc(Cl)[nH]2)=O)CCC1NC(c1c(Cl)nn(C)c1Cl)=O c1(C(=O)NCC(C)N(C(=O)CCS(C)=O)CC)cc(C)cc(Cl)c1 N1(C(c2c(C)nns2)=O)CCC2(CC2)CC1C(N1CCCC(C(C)(C)O)C1)=O CCCC1C(=O)NNC(=O)C23CN(C1=O)C(CC2)CC3.C(CC)(C1CC1)C(=O)OC C1(CNC(c2[nH]nnc2C2CC2)=O)CC2CCC1N2C(c1ccc([N+](=O)[O-])s1)=O N1(C(C2CCOCC2)C(=O)NCC(C2(C)CC2)=O)CCN(c2nc[nH]n2)CC1 CC1Cc2ccc(CNC(N3CCCC(N4CCCCC4)C3)=O)cc2C1C N1(C(CCCCSC)=O)CC(F)(F)CC1(C)CNC(C1CC12CCSCC2)=O C1(NC(=O)Cc2cccs2)CC2CN(C(=O)COCCF)CC2C1 c1(C(=O)NCCNC(C2CN(CC)C(=O)N2)=O)cc(N)c2ncccc2c1 C12(NC(c3cc(O)cc(=O)o3)=O)CCCC1CN(C(C1CC3(CC3)CO1)=O)C2 c1(C2(NC(C3C=CCN(C(CCC#C)=O)C3)=O)COC2)cccc(Cl)c1Cl N#Cc1cc(C(=O)NC2CCN(C(c3ccc(F)c(O)c3)=O)CC2F)ccc1F c1(C(N2CC3C(NC(C(CC)N(C)C)=O)(CC3)C2)=O)ccc(F)c2[nH]ccc12 N1(C(COCCOC)=O)CCC2(CCCN(C(=O)Cc3ccc(C)cc3)C2)C1 C(=O)(CC1=CCN(C(=O)C=CC2CCOC2)CC1)NC(C(CCC)C)CO N1(C(c2nccc(CC)c2)=O)CC(CNC(=O)C(C)(C)CCSC)CC(C)C1 c1(C(=O)NCC2C(C)CN(C(=O)CSCC(N)=O)C2)noc2cc(Cl)ccc12 c1(OC)cc(C(=O)NCC=C2CCN(C(C3CCC(=O)N3C)=O)CC2)cc(C)n1 Cc1cc(C(=O)NC2(CC=CC(N3CCCC(C(N)=O)C3)=O)CCC2)nn1C C1(NC(c2nc[nH]c2C(F)(F)F)=O)COCCN(C(C2CCCNS2(=O)=O)=O)C1 CCC(F)(CNC(=O)CC(COC)NC(=O)CCC1CCC1)CC C#CC1(CC)COCCN1C(C1CN(C(=O)OC(C)(C)C)C1)=O C#Cc1ccc(C)c(NC(=O)NC2CCC(C(=O)OCC)CC2)c1 C1(CNC(c2nn(C)c(O)c2)=O)CC2CCC1N2C(c1cc2[nH]ccc2s1)=O C1(C#N)(NC(c2c(C)cccn2)=O)CCN(C(c2ccnnc2)=O)C1 C1(O)(C(C)NC(C2CC(n3cnnc3)C2)=O)CN(C(=O)C(C2CCOCC2)O)C1 CC(C)C(C)(C(N)=O)NC(C1CCCCC1NC(=O)C(F)C1CCCC1)=O CC1CN(C(C2CC3(C2)CC(O)C3)=O)CCC1CNC(c1cc(CO)[nH]n1)=O C(=O)(CC(C)CC(C)C)N1CCC(C(NOCCCC(=O)OC)=O)C(O)C1 c1(OC)cc(=NC(=O)C(C2(O)CCCCC2)NC(=O)Cc2cnc(C)s2)[nH]n1C CCS(=O)(=O)CCN(C(=O)C(n1cc(-c2cc(C(=O)OCC)ns2)nn1)C)C N1(C(C(c2cc3ccccc3s2)C)=O)CCOc2ccccc2C1C(F)F C1(CC)CCC(C(=O)NC2CCCC2CNC(c2sccc2C(C)(C)C)=O)CC1 CC(c1cccc(Cl)c1)=CC(N1CCC(N(C(=O)CN2CCCC2)C)C(C)C1)=O Cc1ccc2c(c1)CN(C(C1(c3ccc(Cl)c(F)c3)CC1)=O)C2 C(C(CC1CC1)CO)CNC(C=CC(=O)NC(c1ncoc1C1CCC1)=O)=O C(C(O)C(F)(F)F)N(C(C)CNC(c1csnn1)=O)C c1(CNC(CCCOCC)=O)ccc(CCNC(=O)C(C)(C)C2CCC2)cc1 N1(C(COCCC)=O)CCN(C(=O)C(C)CSCc2ccccc2)CC1C c1(N2CC(c3c(OC)cccc3)OCC2)nc(C)c2c(n1)CCCC2 Cc1ccc(C(=O)NC2C3CCC2N(C(=O)CCN2CCC(C)CC2)C3)c(O)c1 C1(NC(c2cc(N(C)C)ccn2)=O)C2CN(C(=O)CC3CC(OC(F)F)C3)CC12 C=CC1CC(NC(=O)C(C2(O)CN(C(=O)C=Cc3ccco3)C2)F)CCO1 C12(C(=O)NCC(CC)N(C)C)CC(C)(CN1C(=O)C(C)SC)C2 C(=O)(C(C)CCC(C)(C)C)N1C(CN(C(C2CC2(F)F)=O)CC)CCC1 N1(C(C2(COC)CCCO2)=O)C2CCC(C2)C1CNC(C1C(C)(C)C1(C)C)=O C(=O)(CCCC(=O)NC1CCN(C(C2CC=CCC2C)=O)C12CC2)NCC Cc1oc(C#N)cc1C(=O)NCc1ccc(C(=O)NCc2cncc(F)c2)cc1 C=CC1(C(=O)NC(C2CC(NC(c3cc(CC(C)C)[nH]n3)=O)C2)C)CCCC1 C1(CNC(C=C(C)C)=O)CCCC1NC(c1ccc(-c2cc[nH]n2)s1)=O C1(NC(c2cc3ncccc3[nH]2)=O)CC12CCC(NC(C1CC1F)=O)CC2 c1(OC)ccc(OC)c(OC)c1CN1CCC(C2(C)NC(=O)NC2=O)CC1 C1(C(N(CC(C)NC(=O)C(c2cccc(Cl)c2)C)C)=O)C2CCC1CC2 CCC(C(=O)NCC(CCOC)NC(=O)Cc1c(C)nc(O)nc1O)C(F)(F)F N1(C(C2C(C)CCO2)=O)CCN(C(c2cnn[nH]2)=O)C(CC(F)F)C1 CC(C)(C)C(CCc1cccc(F)c1)NCCCc1ccc(C(=O)O)cc1 C(=O)(C(O)C(F)(F)F)NCCC1(NC(CCOCC(C)C)=O)CCCC1 C1(CNC(c2cnccn2)=O)CC12CCN(C(c1n[nH]c3c1CSCC3)=O)CC2 C(=O)(CS(=O)(=O)CCO)NCC1CN(C(Cc2ccc(C)c(C)c2)=O)CC1O c1(-n2cnc(C(=O)NCCCNC(C3CC(CF)C3)=O)n2)cccc(Cl)n1 N1(C(=O)C=Cc2ccco2)CCN(C2CCCN(C(c3cnns3)=O)C2)C(=O)C1 N1(C(C2C(C=C)OCC2)=O)CCC=C(C(=O)N2CC(F)(C(=O)OC)C2)C1 Cc1ccc(NC(C2CC(NC(=O)Cc3ccccc3O)C2)=O)cc1 N1(C(c2cn(C)nc2)=O)CCN(C(=O)Cn2ccnn2)CC(C)(F)C1 N1(C(CN(C)CCO)=O)CCCC2C1CCCCN2C(=O)Cn1cnc(=N)[nH]1 C=C1Cn2c(C(=O)NC3CC(NC(C4(OC)CCSC4)=O)C3)nnc2S1 C1(C(C)=O)CC2N(C1)C2=O.c1(CC(=O)NC2CC(C)(F)C2)sc(C2CC2)nc1C C1(C(=O)NC(C2CCN(C(c3cc4ccsc4s3)=O)C2)(C)C)CCCCN1N=O C1(NC(C2CC(=O)N2)=O)CN(C(c2cc3occc3s2)=O)C2(CCOCC2)C1 C12CCCC(CC1)C(=O)N2.C1(NC(C(=O)NCC)=O)CC(F)(F)C1 Cc1cc(Cl)cc(Cl)c1OCC(=O)NCC1CC1NC(=O)CSC(C)C CC(C)C(F)(CNC(C1(CO)CCCO1)=O)C(=O)N1CCCCC(CO)C1 C1(CC)(NC(=O)CCOc2cc(F)cc(F)c2)CCCN(C(=O)C(C)N(C)C)C1 S(=O)(=O)(c1ccc(F)cc1)N(CC(N1CCC(NC(C)=O)C1)=O)C C1(C(N(CCC#N)C2CC2)=O)CCCC12CCN(C(C1CCC3(CC1)CC3)=O)C2 c1(CC)cc(C(N2CCCCC2CNC(C2CC2COC)=O)=O)ccc1O Cc1ncc(C(N2CC(C(=O)NCc3ccc(Cl)cc3)C(C(C)C)C2)=O)c(C)n1 CC1(C#CC(=O)N2CCC3CC23C(=O)NC2CC3CC4C(C3)C24)COC1 c1(OC)ccccc1C(N)C(=O)OC(=O)N(CCC#N)C N1(C(CN(S(CCCC)(=O)=O)C)=O)CCN(C(=O)CCOCCOC)C2CC12 c1(CC)ccc(F)cc1NC(=O)C(C(C)C)NC(=O)Cc1sccc1C C(=O)(C(C(C)C)C(C)C)N1CCC(NC(c2ncc(C)c(Br)c2)=O)CC1C CN1CCn2ncc(C(=O)NC3CN(C(=O)C=Cc4cccs4)CC3O)c21 CC1(C(N2CCC2CNC(c2cccc(N)c2O)=O)=O)CCCS1(=O)=O C(=O)(C1=CCOCC1)NCCC1OCCN(C(C(C)(O)Cc2ccccc2)=O)C1 c1(C(=O)NCC(C)N(C(Cc2c(C)ncs2)=O)C)cc(OC(F)F)cc(F)c1 N1(C(Cn2cnc(C#N)n2)=O)CCCC2CN(C(C3CCCC3(F)F)=O)CC12 C1(NC(CSCCNC(CCC2CCC(=O)C2)=O)=O)CC2C(O)C(O)CC12 N1(C(c2cc(C)c(F)cn2)=O)C2CCC1CC(NC(=O)CC1(N(C)C)CCC1)C2 C(CCC(=O)NC(C1CN(C(C2(N3CCOCC3)CCC2)=O)C1)C)OC(C)=O n1(CC)nc(C)c(C(=O)NCC2(CN(C(=O)C=CI)C)CC2)c1Cl N12CC3CC(C1C3)C2=O.O=C1NC(C2(c3ccnn3C3CCC3)CC2)CO1 N1(CC(Cn2cc(CCC(=O)NC)nn2)O)CCN(C(=O)C(C)(C)C)CC1 C1(C(=O)NCCOCCCN(C(=O)CC2CC(n3cnnc3)C2)C)CC1[N+](=O)[O-] C(=O)(CC1=Cc2ccccc2C1)NCC1N(C)CCN(C(C2(C=C)CCC2)=O)C1 N1(C(c2cnc(OC)nc2)=O)CCC(C2CC2)C1C(=O)N(C1CN(C2CC2)C1)C CCC(C(=O)N1CCC(CC2CCN(C(C3(O)COC3)=O)CC2)CC1)C(C)C C1(C(N(C2CCN(c3nncs3)CC2)C)=O)CCC2(CC1)N=N2 C1(CNC(C2N(C(=O)NC)CCC2)=O)CCCCN1C(c1sc(F)cc1Cl)=O O=S(=O)(c1ccc(Br)cc1NCC1COCO1)NCc1cc(F)c(Cl)cc1F C(=O)(C(C)S(C)(=O)=O)N1CCC(O)(CNC(COCC(=O)NC)=O)C1 C12(C(N3CC(F)(CNC(COCCOCC)=O)C3)=O)CCC(CC1)CO2 N1(C(Cc2c(C)scc2)=O)CCc2sc(CNC(C3(F)CC4(CCC4)C3)=O)nc2C1 C1(CCC)C(=O)NCCN1C(=O)N(CCCN(c1ccc(C)cc1)C)CC C1(NC(c2cc(C3CCCCC3)on2)=O)CCC2(CC1)CC2NC(=O)C1CC1 C(=O)(C(CC)C(=O)OC)N1C(C(=O)NCc2c(C)nc(CC)o2)CC2CC21 N1(C(C=C(CC)CC)=O)CCC(CNC(=O)C(c2cnn(C)c2)O)CC1C N1(C(C2C(C)C2C)=O)CC2CCN(C(=O)CCc3nc4ccccc4s3)C(C2)C1 C(C)(CNC(c1ccnn1C)=O)(CC(C)C)NC(C(C)OCCC(C)C)=O c1(CC)cc([N+](=O)[O-])ccc1C(=O)NC1CN(C(c2ccncc2N)=O)CC1C C1(CNC(C2CC(=C)C2)=O)CN(C(=O)CCc2ccc(C(F)(F)F)cc2)CCO1 C1(C(N2CC(NC(c3cn(C)c(=O)cn3)=O)C3C(C2)C3)=O)CCn2cnnc2C1 C=CCC(CC)C(=O)NC1CCC(NC(=O)CSc2nncn2C)CC1 C1(C(N2C(C#C)CCC2)=O)COCCN(C(C2CN(C3CCC3)C2)=O)C1 C=C=CC(C)C(=O)NCC(O)CCNC(c1ccc(CO)s1)=O C12(CNC(c3c(C)cco3)=O)CCC1CN(C(=O)CCC1CC1(Cl)Cl)C2 c1(C(=O)NCC(CNC(C(CCCCC)O)=O)F)[nH]nc2c1CCCC2(C)C N1(C(C2CN(C)C(=O)N2)=O)CCN(C(c2scnc2Cl)=O)C2COCC12 c1(OCC)nc(C)ccc1C(N1CCC(O)(CNC(=O)CC(C)SC)C1)=O CN1CCCC(C(C)(C)C(=O)NC2CC(N(C(=O)CSc3cnn(C)c3)C)C2)C1 C(=O)(C=C1SCC(=O)N1C)N1CC2(CNC(C(CC)N(C)C)=O)C(C1)CCO2 Cc1nc2cc(-c3ccc(CN4CCCCC4c4nn[nH]n4)c(C)c3)ccc2s1 c1(C(=O)NC2(CNC(c3ccc(F)s3)=O)CC2)c[nH]c2ncccc12 CCCCC(C)(F)C(=O)NCC1(CNC(=O)CSCCOC)CCC1 N1(C(c2cnc(C3CCC3)o2)=O)CC2CCN(C(=O)C=CC(F)(F)F)C2C1 CCC(O)C(C)C(=O)NCC1CCN(C(=O)C=C(Cl)Cl)C1(C)C N1(C(c2c(CC)n[nH]c2)=O)CCC(F)(CNC(C2(CC3CC3)CCC2)=O)CC1 c1(C(=O)OCc2cc(F)ncc2F)ccc(NN2C(=O)CCC2=O)cc1 Cc1csc(NC(C)C(N2CCC(CCNC(c3cscc3C)=O)C2)=O)n1 C1(OC)CN(C(c2cc(C)on2)=O)CC1NC(c1cc(F)cs1)=O C1(C(=O)NCc2n(C)c(O)nn2)CCN(C(C2C(C#N)C2(C)C)=O)C1(C)C C(C(N=[N+]=[N-])C(=O)NCCCC(=O)NCc1cc(F)ccc1O)OCC N1(C(C=C(CC)C)=O)CCC2C1CCCN2C(c1cnccn1)=O C1(CNC(c2ccc(SC)o2)=O)CN(C(c2cscc2F)=O)CCC1(C)C c1(C(=O)NC2CN(C(c3c(Cl)ccnc3Cl)=O)CC2O)cc2cccnn2c1 c1(SC)cc(C(N2CCCC2CNC(C2CC2c2cccc(C)c2)=O)=O)n(C)n1 N1(C(CC2CN(C)C2)=O)CCC(NC(=O)CCc2ccsc2)C(CO)C1 C1(CCNC(=O)Cc2cc[nH]n2)CN(C(c2nc(Cl)c(Cl)s2)=O)CCO1 c1(C(N2CC(CNC(C(C)(C)C)=O)C(C)(C)C2)=O)n[nH]c2ccc(Br)cc12 N1(C(C(C)(C)n2cccn2)=O)CC2(CO)CC1CO2.C12CCC(CC1)CNC2=O Cc1ccc(C)c(C(=O)NC(C2CCCN2C(=O)C(N2CCCCCC2)C)C)n1 C1(C(=O)NCC2N(C)CCC2)CN(C(c2c(F)cncc2Br)=O)CCC1(F)F C1(CNC(C2CCC(OC)C2)=O)(NC(c2nccc(Cl)c2C)=O)CCCCCC1 N1(C(c2c(C)csn2)=O)CCCC(CNC(C2(CO)CCCC2)=O)CC1 C1(C)(C(=O)NCCCOCC=C)CN(C(=O)CC2CC2C2CC2)CC1C c1(OC)cc(C(N2CCN(C(c3cn(C)cn3)=O)C3CC23)=O)ccc1I Cc1ccc(F)cc1CC(=O)NC1CN(C(=O)COC2CCC2)CCC1F N1(C(CCSC)=O)Cc2ccccc2C(NC(C2(F)CCOC2)=O)C1 N1(C(CCCC)=O)CCCC(C(=O)NC2CCC(N(C)C)C2)C1.C1CNC(=O)N1 c1(COC)nc(NCC(C)(C)CC2CC2)cc(N2CCC(OCC(C)C)CC2)n1 c1(C(N2CC3C(CNC(C4(COC)COC4)=O)C3C2)=O)cncc(C(F)F)c1 N1(C(CN2CC(CC)C2)=O)CC2CC2(NC(=O)CCOCc2ccccc2)C1 c1(C(C)C)n[nH]c(=NC2CC3CC(C2)N(C(=O)CC2COC(=O)C2)C3)o1 CN1C(=O)OCC12CN(C(=O)CN(C(C1CC13CCOC3)=O)C1CC1)C2 N1(C(CC(C)C2CC2)=O)CCC(NC(c2nn(C(F)F)cc2Cl)=O)CC(C)(C)C1 Cc1cncc(C(=O)NC(C)CCCNC(c2cc[nH]c2C2CCCC2)=O)n1 C1(NC(Cn2ccc(C)n2)=O)CC2CCC(C1)N2C(=O)CCc1nc(C)no1 c1(CC(=O)NCC(C)NC(=O)Cc2csc(C3CCCC3)n2)ccc(N)c(F)c1 Cc1ccc(C(C)CC(=O)OCc2cccnc2C)cc1 N1(C(=O)CN2CCSCC2)CCC2CC1CN(C(C13CC(F)(C1)C3)=O)C2 C1(OC)(CNC(=O)Cc2csc(=N)[nH]2)CCN(C(c2nocc2C(C)(C)C)=O)C1 C(=O)(CC(C)(C)C(F)F)N1CCN(C(C2C(=C)C2)=O)CC1c1ccncc1 c1(OC(C)C)cnc(C(=O)NCCC2CCC(NC(C3CC(C)(F)C3)=O)C2)cn1 N1(C(CN(CCC)C)=O)CC2CC(C)N(C(c3cc(C)n(C)c3)=O)C2C1 C1(C(N2CC(C)C(N(C)C)C2)=O)CC2(CCN(C(C3C4CC5C(C4=O)C35)=O)C2)C1 C1(C(=O)NCc2ccnc(OC)n2)CN(C(=O)CC2(O)CCCOC2)CCN1C c1(C(C(=O)NC(CC)C)N(C)Cc2ccc(F)cn2)ccc(C)cn1 N1(C(COC(C)C)=O)CC(F)(F)CC1CCNC(c1cc2c(s1)CCC2)=O CC1(C)CCC(C(=O)NC(C)(CNC(=O)COc2ccon2)C2CC2)C1 C(=O)(CC(CNC(C1(C)COC1)=O)OC)NCc1onc(CC)n1 c1(C(N(CCCNC(c2c[nH]nc2OC)=O)CC)=O)cc(C)cc(Cl)c1 Cc1cc(C)c(C(=O)NC(C(=O)N(C2CC2(C)C)C)c2cccs2)cn1 C1(C(=O)NCCC(=C)C)CC(NC(=O)CCc2cnn[nH]2)CCO1 Cc1c(C(C)NC(C2CCC2c2ccccc2)=O)c(C#N)c2n1CCC2 C1(C(=O)NCC(CC=C)NC(C2CCCC2OC)=O)(COC)CC(F)(F)C1 c1(N2CC3CC(NC(CCC=C(C)C)=O)C3C2)ncnc2sc(C(C)C)cc12 CC1(CSc2ccccc2)CCCOC1.C12CN(CCO1)CCc1nnc2o1 n1(CC(=O)NCC2CC(OC)CN2C(c2ccccc2F)=O)ccc([N+](=O)[O-])n1 C(=O)(CCCc1cnn[nH]1)NC(c1nocc1C(N1CC(O)(C(F)(F)F)C1)=O)C C1(C(C)NC(C2CN(C)C2)=O)CCN(C(C2CCCN2C(=O)C2CC2)=O)C1 c1(C(=O)NC2(c3scc(C)n3)CCC2)cc(I)ncn1 c1(C(N(C2CCN(C(c3cnn(C)n3)=O)CC2)CCC)=O)ccccc1CC#N Cc1cccc(F)c1C(=O)NCCC(C)N(C)C(c1cnn(C)c1Cl)=O N1(C(C(C)NC(C)=O)=O)CCOC(CCNC(c2ccsc2Br)=O)C1 Cc1nc(NCCOc2ccc(I)cc2)ccc1-c1cccc(O)c1 c1(-c2c(C)c(C#N)ccc2)ccc2c(c1)CCN(C(c1ccc(Br)cn1)=O)C2 c1(C(N2CC3CCC3(C(=O)NC3CCSCC3)C2)=O)cnc2c(Cl)cccn12 CC#CCCCC(=O)N1CCC(C(=O)N(C2CCN(C(C)=O)C2)C)O1 C(=O)(C(O)C(C)(C)CC)NCC(=C)CCNC(C1(C)CCCOC1)=O CC(CC(=O)NC12CC(CNC(C3(F)CCOC3)=O)(C1)C2)C(F)F C1(N(C)C(C2CSCCS2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C C(=O)(CC(C(C)OC)NC(=O)C(N1CCCCC1)c1csnn1)NCC=C c1(N2CCCC(NC(C3CCC(C)(C)O3)=O)CC2)nc2cc(F)ccc2o1 CCC(C)CC(=O)C(=O)N(CCC(=O)N1CC2(CC(OC)C2)C1)OC CC(C)C(CC1CCCCC1)C(=O)N1CC2CC1C2NC(=O)Cn1ncnn1 C1(C(=O)NC(CNC(c2cc(-c3ccc(C)s3)[nH]n2)=O)(C)C)CC2C(C1)C2(C)C c1(Cn2cc(C3N(C(c4sc(SC)c(Br)c4)=O)CCC3)nn2)cc(Cl)ccc1Cl C=C1CCC(C(=O)NC2CC(NC(c3cc(C)[nH]n3)=O)C2)CC1 Cc1cc(N2CCCC(CNC(c3scc(C)c3Cl)=O)C2)nc(C)n1 c1(CC(=O)NCCC2N(C(CN(C)S(N)(=O)=O)=O)CCCC2)ccc(F)c(F)c1 N1(C(CCC=C)=O)CC2ON=C(CNC(=O)CSCc3ccccc3C)C2C1 C1(C(C)NC(=O)Cn2cnnc2)CCCN(C(=O)CN2CCC(C)(O)C2)C1 N1(C(C(CC)CC2CCCC2)=O)CCN(C(=O)C(C)(C)CF)CC1CCOC C1(C(CNC(CCC=CCC=C)=O)C)CCN(C(C2CCC(CC)CC2)=O)CC1 N1(C(COC)=O)CCN(C2CCCN(C(=O)Cc3ccco3)C2)C(=O)C1 c1(C(=O)NC(CCOC)CNC(=O)CC(C)CF)cc(F)c(F)cc1O C(=O)(C(C(C)(C)C)NC(=O)Cc1ccon1)NC(c1cnc[nH]1)C c1(CCNC(C(C)C)Cc2ccc(F)cc2)cnc2c(C(=O)O)cnn2c1 CC(C)(CCC(=O)NCC1(C(N)=O)CC1)NC(C1CC2(CC2)CO1)=O C1(C(N2C(C)CC(NC(CC=C)=O)C2)=O)CC2CC1C1CC21 Cc1ccc2oc(N3CCC(NC(C4CC4(F)F)=O)CC3C)nc2c1 Cc1cc(F)ncc1C(=O)NCC(C)N(C(=O)C(C(C)C)N1CCCC1=O)C C1(CN(C(CCNC(=O)OCC)=O)C)CC(C(=O)N(C)C2CC2)CO1 C1(OC)COCCC1C(=O)NCC1(C(N)=O)CN(C(=O)Cc2cnn(C)c2C)C1 C1(CNC(C2(CC(C)C)CCC2)=O)CCC(NC(=O)Cc2c(Cl)cnn2C)CC1 N1(C(C2(C#N)CC=CC2)=O)CC2(CCC2)CC1CNC(=O)CCc1cnccn1 N1(C(C(CCC)CC)=O)CCN(C(C2(CC(F)F)CCC2)=O)CC(O)C1 C1(NC(C(CC=C)CC(C)C)=O)CC(N=c2[nH]c(C3CC3)nc(Cl)c2C)C1(C)C N1(C(=O)CCn2ccnn2)CCOC2(CCN(c3ncnc(O)c3Br)CC2)C1 C1(C(N2CCC(N(C(c3ccc(COC)o3)=O)CC)C2)=O)CC(=O)CCO1 C(=O)(C1=NOC2(CCOC2)C1)NC(CCNC(c1cnc(C)o1)=O)C C1(C(N2CCC(F)(F)C2)=O)CC2(C1)CN(Cc1ccc(Cl)cn1)C2 c1(C(=O)NCC2CN(C(C(C)n3cccn3)=O)C(C)(C)C2)ncn2c1COCC2 C1(C(N(C)CC2(NC(c3cc(CC)ncn3)=O)CC2)=O)CC(C)(C)OC1(C)C C1(CN(C)C(=NCCCF)NCC2CCOC2)CC2COCC(C1)C2(F)F n1(-c2ccn(CC)n2)nc(COC)nc1C1CC(n2cccn2)(OC)C1 CC1(C)CC(C)(C(=O)NCC2CC(C(=O)NCCCCC3CC3)C2)C1 N1(C(CCOC(CC(C)C)C)=O)CCC(O)(CNC(c2cnnn2C(C)C)=O)C1 C1(C2(O)CN(C(=O)C(O)C3CCC3)C2)(CNC(=O)C=Cc2cncc(O)c2)CC1 c1(CSC)nc2ccccc2n1CC(=O)NCC1COCCC1(F)F C1(CN(C(CCN(C(CSCCCC)=O)CCC)=O)C)CCCCC1O c1(C(c2nnnn2C2CCOCC2)NC(CCSC)C)cc(C2CC2)nn1CC c1(-c2c(C)c(N3CCC4(CCC4)C(O)C3)ncn2)ccc2c(c1)OCCO2 C12(NC(C(C3CCC3)OC)=O)CCCC1N(C(C1(F)CCC(=O)CC1)=O)CC2 CCCCCC(O)CC(=O)NC1(CNC(C2CCCCN2CCC)=O)CC1 C1(C(=O)NCC(CN(C(c2cnnc(C)c2)=O)CC)(C)C)CCC12CCC2 CCCCCCC(C)(CCC)C(=O)NC1CCN(c2ccccc2OC)C1=O CC1CCC(NC(C2CC3(CSC3)C2)=O)CN1Cc1ccc(C(F)F)cn1 C1(NC(C(COC)C)=O)CCN(C(=O)CNC(=O)OC(C)(C)C)CC12CCC2 N1(C(=O)NC(c2cccc(OC(C)C)c2)CC)CCOCC1C1CCOCC1 CCCC(C)CCCC(=O)N(CCC)CCNC(=O)CCn1cccn1 C1(NC(C2(CCC)CCC2)=O)CCN(C(=O)CNC(=O)CC)CCC1CO c1(C(N(C2CCN(C(C3CCOCC3)=O)C2)CC)=O)ccc(C)nn1 C1(CN(C(C(CC)N(CC)CC)=O)C)CCC(CNC(c2occc2C)=O)CC1 N1(C(C2C(OC)C2)=O)CC2CCC1CN2C(=O)Cn1ccc(C(F)F)n1 C1(NC(C=NOC)=O)CCN(C(c2cc(C)nc(C)c2)=O)CC(C)(C)C1 C(=O)(CC(CC)C(C)C)N(CCC(C)NC(C1(COC)CCCC1)=O)C N1(C(C2CN(C(C(C(=O)OCC)OC)=O)CC2F)=O)CC2CCC1CC2 N1(CC(=O)NC2(C(N(CCCO)CC)=O)CC2C)CCNC(=O)C1 c1(N(CCC(O)C(C)(C)C)C)nccc(=NC2CSC2)[nH]1 c1(SCC)cnc(O)c(C(=O)NC2CCCCC2NC(c2snnc2CC)=O)c1 c1(C(=O)NCCN(C(=O)C=C(C)C(C)(C)C)CC)ccc(C(C)=O)c(F)c1 NC(=O)C#CC(=O)N1CCC(C(c2ccc(F)cc2)O)CC1 C1(C)(C(N(CCC(F)(F)F)C)=O)CCCN(C(C2(C(C)(C)O)CC2)=O)C1 c1(C2C(NCC(CNC(=O)OC(C)(C)C)(C)C)C2)ccc(F)cc1Cl c1(C(=O)NCC2COCC2NC(c2cnc[nH]2)=O)cncc(CO)c1 CCC(C)CC(=O)NC1CC(CNC(c2ccnc(N(C)C)c2)=O)CC1O N1(C(C(CC#C)C2CC2)=O)CC(C(=O)N(C)CC2(O)CCCCC2)CCC1(C)C c1(C(N(CC(=O)N(C)CC2CCC(C)CC2)C)=O)cc2n(n1)CCC2 N1(C(CSCC#C)=O)CCC(C(=O)NC2CCN(c3nc(COC)ns3)C2)CC1 Cc1ccc2[nH]cc(CC(C)NC(=O)CC3CCCCNCC3)c2c1 CC1(C)Cc2cc(CNC(=O)CN3OC(C)(C)CC3=O)ccc2O1 N1(C(C2(CF)CCN(C(C(CCC)OCC)=O)C2)=O)CCOC(C(C)C)CC1 C#CCCC(C(=O)NCC1(O)CC2CCC1O2)NC(=O)Cn1ccc(C)c1 C1(CC(=O)N(C(CNC(c2ccc(C)nc2)=O)C)C)CCCCC1(F)F Cc1cc(C(=O)NCc2csc(CNC(=O)C(C)(C)F)n2)ncc1C#N C1(CNC(=O)Cc2cncnc2)CCN(C(C2CCC(F)(F)CO2)=O)CC1(F)F c1(C(=O)NC(C)CO)ncn2cc(-c3cccc(CCO)c3)sc12 Cc1cc2c(C(=O)NC(C)CC(C)NC(c3c(C)ccn3C)=O)ccc(C)c2[nH]1 C1(C(N2CCC(N(C(C(C)OCOC)=O)CCO)C2)=O)CC(S(C)(=O)=O)C1 N1(CC(=O)NC2C(CNC(CCCC)=O)C2)CCN(C(C)=O)CC1 N1(C(CNC(C)=O)=O)CCC2CCCN(C(c3ccccc3O)=O)C2C1 c1(C(N2CCC3CN(Cc4ccc(F)nc4)CC23)=O)cc(F)c(F)cc1F c1(C(=O)NC2C3OCC(NC(C(C4CC4)OC)=O)(C3)C2)ccc2c(c1)OCCO2 C1(C2CCCNC2)(NC(c2c(C(C)(C)C)con2)=O)CC1 C(CC(C(C)(C)C)NC(=O)Cc1cnco1)N(C(c1c(C)snc1)=O)C c1(C(=O)NCC(CNC(=O)CCSC(F)(F)F)F)ccc(Cl)c(F)c1O N1(C(c2ccn(C)n2)=O)CCCN(C(c2coc(Sc3ncccn3)n2)=O)CC1 C1(NC(C(C)Cn2cccn2)=O)CC12CC(NC(=O)C(c1ccc(F)cc1)=O)C2 c1(C(C)OC(c2nscc2Br)=O)ccc(-n2ccnn2)cc1 C1(C(N(CC)Cc2ccccn2)=O)CN(C(=O)CCC2CCC2)CCS1 C(=O)(CC1=CCCCC1)NC(c1ccc(C)cc1)CNC(C(C)N(C(C)=O)C)=O Cc1ccnc(-c2noc(C(C)Sc3sc(Cl)nc3Cl)n2)c1 n1(CC)nc(C)c(C(=O)NCC2(NC(C3C4CCCC34)=O)CC2)c1Cl C12(C(=O)OCC(C(C)C)OCc3ccccc3)CCC(C(F)F)(CO1)C2 N1(C(Cc2c(C)ccs2)=O)CCN(C(=O)C(C(C)C)c2cccc(Cl)c2)C(C)C1 S(=O)(=O)(c1ccccc1N1CCC(NC(c2ccccc2CC)=O)C1)NCC CCCCCC(C)CC(=O)N1CCCC1(C)C(N1CC(C)(O)C1)=O C1(NC(C(C)CSC2CC2)=O)C2CC1N(C(=O)CC1(c3ccccc3)CC1)C2 N1(C(C(C(C)(C)C)SC)=O)CCN(C(=O)CCC(C)(C)C)CC12CC2 C1(NC(CC(C)F)=O)CC12CCN(C(C1(C)CCOC1)=O)CC2 c1(C(=O)NC(C2CCN(C(C3CNC(=O)N3)=O)CC2)C)ccnc2c1ncn2C C#CCC(C)(C(=O)NC(c1nnc(O)n1C)C)NC(=O)C(O)C(C)(C)C O(NC(=O)C(Cc1cn(-c2cccc(C)n2)nn1)C(C)C)C(c1ccccc1)C C1(C(=O)NCC(CNC(c2cc(CCC)n(C)n2)=O)OC)CS(=O)(=O)CC(=O)N1 C(=O)(C(Cc1cc[nH]n1)NC(c1cnsn1)=O)NCC(C)F N#CC1(C(=O)NC2CCCC2n2cc(C3CCCCCC3)nn2)CC2CC2C1 N1(C(C2CCC(C)CC2)=O)CCN(C(C2CCCCCN2C)=O)CC1C c1(CCCN(C2CCOC2)C(=O)NCc2cn[nH]c2)cccnc1F c1(C(N2C(C(=O)Nc3cc(C)cc(Br)c3)CC2)=O)cc(F)c(Cl)c(C#N)c1Cl c1(C(=O)NC(CCN(C(C2CN(C)C(=O)CC2)=O)C)(C)C)nc[nH]c2nccc1-2 N1(C(c2cc3ncccc3[nH]2)=O)CCC2CCC(NC(C34CCC(C3)C4)=O)C1C2 Cc1ccc(F)c(C(=O)OC2CCCCC2OCC(C)C)c1 N1(C(C2CCCCC2)C(=O)NCC(F)F)CCCCCC1c1ccccc1 CCCC(CC(C)C)C(=O)N1CC(C)(C)CC1CNC(=O)C=C(C)C(C)C C1(C(N(C)CCNC(C2CC(Cc3ccccn3)C2)=O)=O)CC2C=CCC(C1)C2 N1(C(CCCCNC(COCC(=O)OC)=O)=O)CCCC(C)(C#N)C1 c1(NC(N(c2ccc(Br)cc2)CCOC)=O)cccc2c(F)ccnc12 CCS(=O)(=O)CC(=O)NCC(C)(C)OCCNC(=O)CCc1cccnc1C c1(C(=O)NC2(C)CN(C(C(C)=CC)=O)C2)[nH]c2c(c1C)C(=O)CCC2 C(=O)(C#CC(C)(C)CNC(C1CC=C(C)CC1)=O)NCCSCC#C c1(CC(=O)NC2CC(NC(C=CCCC(C)C)=O)C2)ccc(S(=O)C2CC2)cc1 c1(SCCC(N)=O)ccc(C(=O)NC2CC(NC(C3CCC34CCC4)=O)C2)cc1 C12(CCNC(c3c(C)nsc3)=O)CCC1CN(C(=O)C(C)(O)CCN(C)C)C2 O=S(=O)(c1[nH]c(=NC2CC(CF)C2)ccc1Br)NC1CCOCC1O Cc1c(C(=O)NC(CNC(=O)C(C)C(C)(C)C)C2CC2)cnc2ccccc12 N1(C(c2c(CC)ocn2)=O)CCn2nc(C(=O)NCC3CCCCC3C)cc2C1 C1(C(=O)NCCN(CCOC)C(C2COCCOC2)=O)CC12CCOC2 CC1(C)CC1(Br)C(=O)NCC(c1ccccc1)NC(C1(C(F)(F)F)CC1)=O c1(N(CCN(CC(F)(F)F)C)C)nnc(C2CCOC2)n1CC1OCCC1(C)C N1(C(C=CCN(C)CC)=O)CCCC(O)(CNC(C2CC2(Cl)Cl)=O)CC1 N1(C(c2ccc(C)cc2C2CC2)=O)CCC2CN(C(=O)C(C)(C)OC(F)F)CC12 C1(S(N)(=O)=O)(C(=O)NC(C2CN(C(=O)CC(C3CC3)C3CC3)CCO2)C)CCC1 n1(CC(N2CC(C(C)NC(C(CCSC)O)=O)C2)=O)ccc([N+](=O)[O-])n1 c1(SCCC)ccc(C(=O)NC2CC2CNC(=O)COC(C)C)cc1 C1(OC)CN(C(C2CC2(C)C)=O)CC1C(=O)NCC(C)C1CCC1 C(=O)(CC(C)C(C)(C)CC)N1CCN(C(C(CC)=CC)=O)CC(CO)C1 N1(c2nccc(N3CCC(CC(=O)N(C)CC)C3)n2)CCCN(CC(C)O)CC1 C(=O)(CC(C)C(=O)NC1CCC(NC(=O)C=C(C)C(C)C)CC1)OCC N1(C(c2cccc(CSC)c2)=O)CC(NC(=O)CCC2CCC2)CC(O)C1 c1(C(N2CC(C)N(C(c3ccc(Cl)c(C#N)c3)=O)CC2)=O)ccc(F)c(Br)c1F C(=O)(CS(=O)(=O)c1ccccc1Cl)NC(CNC(C(COC)C)=O)(C)CO c1(OC)cc(Cl)ccc1NC(=O)NCC(c1ccnn1C)(F)F CCC(C)(C(=O)N1CC2CC1C2NC(=O)CC1(CN(C)C)CCOCC1)C(N)=O c1(CCNC(c2ncn(CCNC(CCOCC(C)C)=O)c2)=O)ccccc1O N1(C(c2csc(Cl)n2)C(=O)NCCSC)CCOCC1c1c(C)n[nH]c1C CCCCCC(C)C(=O)N1CCC2C1CCN2C(=O)CN1CCOC1=O Cc1cnn(C(C)C)c1C(=O)NC1CCCCC1NC(c1cscn1)=O CC1CCC=C1C(=O)N1CCC(N(C(=O)C=Cc2ccoc2)CCO)C1 c1(OC)ccc(CN2CC(C(=O)NCC(C)(C)O)CC(F)C2)c(F)c1F C1(CNC(Cc2cc(C)c(F)cc2)=O)C2CCC1CN(C(=O)CCCN(C)C)C2 C1(CC(=O)NCc2ccc(CNC(C3CCCS3)=O)cc2)CC2(CCC2)CCO1 CCCC(O)C(CO)NC(=O)CN1CCN(C(=O)CC2CCCOCC2)CC1 C(=O)(CCCC(N)=O)N1CCC(COC2CCN(C(C(CCSC)O)=O)C2)CC1 C12(C(=O)O)CN(C1)C(=O)CCOCCOCC2.n1(CC(=O)OC)cnnn1 c1(C(=O)NC23CCN(C(c4cc(OCC)n[nH]4)=O)CC2C3)ccc(F)c(C#N)c1 n1(CC=C)cc(C(N2CC(F)CC2(C)CNC(=O)C(N)=O)=O)c2ccccc12 Cc1[nH]c2c(F)cccc2c1CCNC(N1CCC(Cc2cnccn2)CC1)=O N1(CC(=O)NC23CC(C2)N(C(=O)C(F)C2CCOC2)C3)CCCCCC1 Cc1ccc(I)c(C)c1NC(C1CCCC1NC(=O)CCN1C(=O)C=CC1=O)=O N1(C(C(n2nnnc2C(C)(C)C)C)=O)CCC(N(C)C(C2(O)CCC2)=O)CC1 CCCC(O)C(CO)NC(=O)CC1CN(C(c2cnco2)=O)CCO1 CCCCC(C)(CO)NC(C1CC2CC2N1C(C1C2CCC(F)C12)=O)=O c1(C(C)OC)nc(C(=O)NCC(=C2CN(C(=O)CCc3cnc(O)[nH]3)C2)F)cs1 c1(OCC)nc(C)cc(C)c1C(c1nnnn1CC)NCc1ccc(Cl)cc1Cl N1(C(C(CCC)C)=O)CC(NC(c2oc(CC3CC3)nc2C)=O)CC(F)(F)C1 CCC(C(=O)N1CCN(C(c2ccc(C)o2)=O)C(CC(F)(F)F)C1)C(C)C C#CCCC(O)CCNC(C1C2CC2CN1C(c1cncc(OC)c1)=O)=O c1(C(=O)OCC)nc(C)ccc1NC(=O)NCC1(COC)CC2CC2C1 C(C)(C)(CC(=O)N1CCC(NC(=O)CSc2nc[nH]n2)C1C(C)(C)C)SC c1(C(=O)NC2C(CNC(c3n(CCCC)ncc3)=O)C2)cc2ccc(Cl)cn2c1 N1(C(=O)Cc2cn[nH]c2)CC2CCN(C(c3ccc(C4CCOC4)cc3)=O)C2C1 c1(C(=O)NC(C2CN(C(c3nncn3C)C)C2)C)cc2sccc2s1 C1(NC(c2cc(C)nn2C)=O)C2CC3CN(C(=O)CCOCC(C)C)C1C3C2 CC(C)CC(O)C(=O)NC1(CNC(c2ccc(Oc3cccnc3)nc2)=O)CC1 n1(CC)nc(C(N2CCC(CC(N)=O)(NC(C3CC3(Cl)Cl)=O)CC2)=O)ccc1=O Cn1cc(C(=O)NCC(C)(O)CNC(=O)CC2(C(F)F)CC2)c(C2CC2)n1 C1(CNC(C2(CSC)CC2)=O)(NC(c2ncc(OC)cn2)=O)CCCCC1 C1(OC)CC2(C1)CC(NC(=O)NC1CCN(C(=O)OC(C)(C)C)C1)C2 C1(C(N2CC(C(C)OC)C2)=O)(CC)CCOCC1.C12CC(C1)C(=O)NCC2 N1(C(COC2(C)CCC2)=O)CC2CCC2(NC(=O)CN2CCC(=O)NC2=O)C1 N1(C2C(C)CCN(C(c3ccc(Cl)s3)=O)CC2)CC2C(=O)NC(=O)C2C1 C1(CN=[N+]=[N-])CCCN1C(=O)CCn1cc(Cl)cn1 Cc1ncnc(C)c1CNCc1cccc(NC2CCCCC23CC3)c1 C(N=c1cc(C)[nH]cc1-c1nn[nH]n1)C1N(CC=C(C)C)CCCC1 C#CC1(C(=O)NCC2CC(C)N(C(=O)COCc3cc(C)on3)C2)CCCC1 C#Cc1cccc(-c2ccccc2C2(C(c3ccc(C4CC4)c(F)c3)=O)CC2)c1 C(c1ccc(F)c(F)c1)=CC(=O)NC1CCN(C(CCCC=C)=O)C(C)C1 n1(CCCC)ncc(C(N2CCCC(NC(=O)C(C)OCC(C)C)C2)=O)c1C C1(CNC(CN(C(C)=O)C)=O)C(C)CCN(C(=O)CCOCCN(C)C)C1C C1(C(N(C)CC2(O)CCCC2)=O)COCCC1NC(=O)CCC1(C#N)CCC1 C1(C)(CNC(C2(COC)CCOC2)=O)CCCNS1(=O)=O C(=O)(C(CC(C)C)NC(N)=O)NCC12CC(NC(CC3(OC)CCC3)=O)(C1)C2 CC(O)C(C)(C)CN=c1[nH]c(N2CCC(C)(CC#N)C2)nc2cc[nH]c12 C1(C(=O)NC2CCCC2NC(=O)CSC(F)F)(COC)CC=CCC1 c1(C(=O)NC2(CCCNC(COCC)=O)CC2)cc(S(N)(=O)=O)cn1C N1(C(C(C)SC)=O)CC(CNC(c2cc(Br)no2)=O)C(O)C1 Cc1cnc(C(=O)NCCCCC2CCN(C(=O)CCCC3CC3)CC2)c(C)c1 c1(C(=O)NCCCC(C)NC(C2CCN(C)C2)=O)ccc(C#N)c(Cl)c1 CC(C)C(CCN(C(=O)Cn1cncn1)C)N=c1cc[nH]cc1C#N C=C(C)CC(C(=O)N(C)Cc1nccn1CC)NC(c1oc(CC)nc1C)=O c1(CNC(C)=O)ccc(C(=O)NC(C2(O)CCN(C(=O)C=CCF)C2)C)cc1 c1(C(=O)NC2CCCN(C(C3N(C(C)C)CCC3)=O)C2)cc(Cl)ncc1F c1(OC)cc(C(=O)NC(C)C(C)NC(c2cncs2)=O)ncc1Br C1(O)(C(=O)NCC(C)CN(C)C(c2ccc(CF)cc2)=O)CCSCC1 c1(CC(=O)N(C(C)CCNC(=O)C=CC2CCC2)C)ccc(F)cc1C(F)(F)F C1(CC#C)(C(=O)NCCc2c(C)n[nH]c2C)CCN(C(=O)COC2CCOC2)C1 N1(C(C=COCC)=O)CCCC(CCNC(c2ncccc2N(C)C)=O)C1 c1(-c2cc(C(=O)NC)c(Cl)nc2)ccc(S(=O)(=O)NCc2ncccn2)cc1 CC1CCN(C(=O)C=CC2CCCC2)CCN1C(C1CCCS(=O)(=O)N1)=O N1(C(C(C)(C)c2cnsc2)=O)CC2CCC(CNC(=O)CCF)(C2)C1 C1(C(N2CCC(NC(c3c(CC)nc(C)o3)=O)C2)=O)CC2(C1)CC1(CC1)C2 Cc1cccn2cc(C(N3CCC(N(C(=O)CCC(C)C)CCO)C3)=O)nc12 C1(CNC(C(CC)C(C)C)=O)CN(C(c2nnn(C(C)C)c2C)=O)CC(C)(C)C1 C(CCCC(C)NC(c1cc(C(C)(F)F)n[nH]1)=O)NC(c1cc(CCC)[nH]n1)=O c1(C(=O)NC2CC(CNC(C(=O)NCCOC)=O)C2)ccccc1NC(N)=O C1(O)(CC(=O)NCc2cn(CCN(C(=O)C(C)(Cl)Cl)C)nn2)CCCCC1 N12CCCC(C1)C(C)C(=O)NC(=S)NC(SC)C2=O.N1(CC)CCOCC1 c1(C(=O)NC2CCCC(NC(C(C)SC)=O)C2)cc(C)nc2c1c(C)nn2C CC(C)(F)CCC(=O)N(CCCNC(=O)CCNC(C1CCC(=O)N1)=O)C1CC1 C(=O)(C(C)C(C)NC(c1cccnc1O)=O)NC(c1nc(CC)on1)C C1(CC)C(C(=O)OC2CC2)CCCN1C(=O)C(=O)NC(C)C.C12COCC1C2=O C1(NC(CNS(N(C)C)(=O)=O)=O)CCN(C(C2(C(N)=O)CC2)=O)CCC1CO c1(C(N2C(CCNC(C3CC(CCC)C3)=O)CCCC2)=O)cc(C)cnc1N N1(C(c2cncc(C)c2)=O)CCC2(CC1)CC(NC(=O)C=C(Cl)Cl)CCO2 CCC(C)(C)CC(=O)N1CCCCC1C(=O)Nc1cc(CO)cc(F)c1 N1(C(c2n(CC)ccn2)=O)CCN(C(=O)C(C)(c2ccccc2)OC)CC1C c1(OC)noc(C)c1C(=O)NCC1CCCCC1C(=O)N(C)CCOC Cc1cc(C(=O)NC2(C(=O)NC3(C(C)O)CC3)CCCC2C)nc(C)c1 C1(C(=O)NCC(=O)NCC(C)C)OCCC1NC(=O)CC1CCCCC1 c1(CC)c(C(=O)Nc2cccc(NC(c3ccoc3Br)=O)c2)ccn1C c1(CC(N2CCN(C(C(N)=O)=O)C(CC(F)F)C2)=O)ccc(F)cc1[N+](=O)[O-] N1(C(=O)OCc2cc(F)n[nH]2)CCCCC1CNC(=O)C(F)(F)F c1(C(N2CC(N(C(Cc3cn(C(C)C)nc3)=O)C)C2)=O)cnc2c(cnn2C)c1 C1(NC(c2ccc(C(C)C)o2)=O)CCN(C(=O)CC(=O)NC2CC2)C(C)C1 C1(C(=O)NC2CN(C(C3CC(=O)NC3)=O)CC23CC3)COc2cc(Cl)ccc2C1 N1(C(C(CCC2CC2)OCC)=O)CCC(CO)C(O)C1.C1(C)CCC(=O)N1 c1(OC)ncccc1S(=O)(=O)NC(c1ccccc1N(C)C)=O C1(O)(C(=O)NCCC2(O)CN(C(c3c(C)c[nH]n3)=O)C2)CCc2ccccc2C1 CCC(C)(C(=O)NC1(CCCNC(c2ccnc(C(F)(F)F)c2)=O)CC1)C(N)=O c1(OC)ccc(CN2CCOCC2CC(N2CCC(C)C2)=O)cc1I c1(C(N2CCCC(NC(C(CC)CO)=O)CC2)=O)cncc2c(O)nccc12 c1(C(N2C(C)CCC2)=O)ccc2c(c1)CN(C(c1ccc3ncnn3c1)=O)C2 CC1Oc2ccccc2OC1C(N1CCN(C(c2ccco2)=O)CC1)=O C1(CNC(c2ccc(C)cc2F)=O)CN(c2ccnc(NCC)n2)CC(C)(C)O1 C1(COC)CC(CNC(c2c(Cl)cnn2C)=O)N(C(=O)C=C(C)C(F)F)C1 C(C(C(C)(C)C)NC(c1ncccn1)=O)NC(C(C)Cc1ccncc1)=O CCC(C)(C(=O)NCCN1CCCN(C(=O)CC2CCC(=O)N2)CC1)C(F)F C1(NC(=O)C2=COCCO2)CCC2CN(C(=O)CO)CC2C1 C1(C(=O)NCc2c(CC)cncc2)CCC(O)CN1C(=O)CC1(C)CCOC1 CC1OCCC1(C)NC(C1CN(C(=O)CNC2CCSC2=O)C1)=O.C1C(=O)N1 c1(N2CCN(C(C)C)CC2C)ncnc2c1ncn2CC1(O)CCCC1(C)C N1(C(C2C=CC(NC(c3cccc4[nH]ccc34)=O)C2)=O)CCc2ncccc2C1 C12(C(=O)O)CCCC(C(=O)NCc3cc(-c4ccccc4)on3)(COC1)C2 c1(C(=O)NCc2ccc(CNC(C3C(COC)C3)=O)cc2)cccc2ncnn12 C(=O)(CC(C(F)(F)F)c1ccon1)N1C(CNC(C(N)=O)=O)COCC1 C(CC(F)F)(C(=O)NC1CC1F)NC(C(C)=NOCC#N)=O c1(COCC(N2CC3C(NC(=O)C4=CCCCO4)(C3)C2)=O)nc2ccccc2s1 c1(NC(C2CC(F)CN2Cc2cccnc2F)=O)ccc(Cl)cc1O C1(NC(c2ccc(OC)c(C)c2)=O)CCCCN(C(c2cnco2)=O)CC1 C(C)(C(=O)NC1CN(C(c2scnc2C2CCCC2)=O)C1)(C1CC1)OC N1(C(CCN(C)CC)=O)CCN(C(=O)C(c2ccc(Cl)cc2)=O)C2CC12 c1(NC(C2CCOCC2)C(C)OC)cc2c(N(C)C)ncnc2n1C c1(-c2cnc(C3N(C(=O)Cc4cncnc4)CCC3)[nH]2)ccccc1I C1(CC)CC(O)CN1C(=O)CCCCNC(C1(COC)COC1)=O c12cc(OC)ccc1NC(=O)COC2=O.C(=O)(C(C)(C)SC)NC c1(OC)cc(CN2CC3C(C2)N3C(=O)C(c2ccc(Cl)cc2)=O)cc(C(F)(F)F)c1 C(CCC(C)(C)C(=O)NCC(C)CC(=O)NCC1CC2(C1)CC21CC1)OC c1(C(=O)NCC2(OC)CN(C(C3CC=CCC3)=O)C2)cc2cnccc2o1 C1(C(N2C(=O)CC(N(C3CC4C3CCN4C(=O)C3CC3)C)C2)=O)CC2(C1)CC(F)C2 C1(C(N2CCCCC(CNc3nccc(CO)n3)C2)=O)CCc2c[nH]nc2C1 C(N=c1[nH]c(=NCc2ccc(O)nc2)c2cc(OC)ccc2[nH]1)C1C(SCC)C1 CC(C(=O)N(CCO)C1CC1)NC(=O)CCOCCN(C)C C12(C(=O)NCC#CCNC(C(C=C)c3ccccc3)=O)CC1Cc1c[nH]nc12 C(=O)(C(CC(C)CC(C)(C)C)N1CCCS(=N)(=O)CC1)NCCCSC c1(C(=O)NC(C)CNC(=O)C(F)=CC2CC2)cc(N)cnc1Cl C1(NC(CC(C)(C)C)=O)C(C)CN(C(c2cccc(C3CCC3)c2)=O)CC1C C=CC(C)(C)CC(=O)N1CC(CNC(c2cc(CC)cnc2O)=O)C(C(F)F)C1 Cn1cc(C(N2CC3CC3(CNC(=O)COc3ccccc3F)C2)=O)ncc1=O c1(C(=O)NC2C(CNC(CCOC(CC(C)C)C)=O)CC2)c(O)cccc1Cl C12(C(N3CCCC(OCC)C3)=O)CCCC1CCN2C(c1cnnc(O)c1)=O C1(O)(CNC(C(n2nnnc2C(C)(C)C)C)=O)CN(C(c2n[nH]cc2C2CC2)=O)C1 c1(N(CCCCC=C)C)cccc(S(N)(=O)=O)c1S(C)(=O)=O C1(C(=O)NCC2CC(NC(=O)COCC3CCCO3)C2)CCC(F)(F)C1 C1(NC(c2c(COC)cco2)=O)CN(C(C23CC4CC2C3C4O)=O)CC1(C)C Cc1nn(C)c(Br)c1C(=O)NC1CC(CNC(=O)C(O)CF)C1 C1(NC(CN2CCN(C(c3n(C)nnc3)=O)CC2)=O)CCC2(CC1)N=N2 CC1CCCC1CC(N1CC(=C(F)CNC(c2scnc2C2CC2)=O)C1)=O C1(CNC(Cc2c(OC)ccnc2)=O)CN(C(C2C(C)C2C)=O)CCN1C c1(CC)ccc(C(=O)NCC=CC(=O)NC(C)CC(C)(C)C)cc1 C12(C(=O)NC3CC(CNC(CSCCN(C)C)=O)C3)CCCCC1OCC2 N1(C(CN(C(=O)Cn2nnnc2C)CCOC)=O)CCC12CCC(O)CC2 c1(C(N2C(CNC(=O)C(C)CO)CC(OC)C2)=O)occ2c1CCC2 N1(CC(=O)N(CCC(=O)NCC(=O)NCC#C)C(C)C)CCC(C)CC1 N1(C(C(CC=CC)CC)=O)CC2(CCCC2)C1C(=O)NCc1cccc(O)n1 C1(C(=O)NCCc2cc(C)ncc2)N(C(=O)C(C2CCOCC2)=O)CC12CCCC2 C1(C(=O)Nc2cnc(O)c(C(F)(F)F)c2)CCC2(CN(Cc3ccsc3)C2)O1 CC1(C)Cc2ccccc2C1NC(=O)NCCc1ccc(C2CCCCC2)cc1 CCC(C)(O)C(=O)N1CC(CO)(NC(c2csc(C)c2OC)=O)C1 C(=O)(C(C(C)C)c1cccs1)NCCCN(C(C(CC)N1CCCC1=O)=O)C c12cc(Oc3ccccc3F)ccc1C(=O)N2.C1(C(=O)O)C=CC(C(=O)O)C1 Cc1cc(C(N2CCC(N(C(=O)C(C(C)C)NS(C)(=O)=O)C)C2)=O)nn1C C1(C(=O)NCC2(C(C)(C)O)CN(C(C(=O)NCCOC)=O)C2)CC=C(C)CC1 CCC(CC(=O)NC(C)(CC)CO)N(C)C(c1ccncc1OC)=O c1(C(=O)NC2C(NC(COc3ccc(OC)cc3)=O)C2)ccc2c(c1)COCO2 CC1CC(C)(C(N2CCOC(CN(C)C(C3(CCO)CC3)=O)C2)=O)CC(C)O1 CN1CCC(=CC(=O)N(C2CCC(NC(c3cc(F)n[nH]3)=O)CC2)C)CC1 C1(N(C(=O)C(C)SC(C)C)CC)CCN(C(c2cc(C(C)(F)F)on2)=O)CC1 N1(C(CCNCCOCCOC)=O)CCC(NC(C2(C3CC3)CCC2)=O)C1 C(C(C)(O)CC(=O)N(CC(C)CNC(=O)Cc1cccnc1)C)OC N1(C(c2cncc(OC)c2C)C(=O)NCCC)CC(C)(C)C12CCOCC2 N1(C(C(=O)NCC)=O)CC(NC(=O)C(F)C2CC2)C(C)C1 c1(C(N2CCC(NC(CC3C(C)CCCC3)=O)C2)=O)c[nH]c2cccnc12 C1(CNC(c2ncn(CC)n2)=O)CCC2(CCC2)CN1C(C1CCCC(C)C1)=O C(CCCCCNC(=O)C(C)(O)C1CCOC1)N(C(=O)CN1CC(C)(C)C1)C C(=O)(CCS(=O)(=O)C(F)(F)F)N(CC(CC)NC(C1CCSC1)=O)CC C(CCC)(C(=O)N1CCCCC1CNC(c1nocc1CC)=O)=CCC N1(C(CC2(C)CC2(Cl)Cl)=O)CCC(C2CC2NC(c2cc3n(c2)CCC3)=O)CC1 N1(C(C(C2CC2)OCC)=O)CCN(C(c2occc2C2CC2)=O)CC1CC(F)F C1(C(=O)NCC(C)(C2CCC2)NC(COCCC=C)=O)CCCOC1C CCC(C)(CNC(=O)C(CCOC)NC(=O)CC1C(=O)NN=C1C)CC c1(C(N(CCCNC(=O)CC2(N(C)C)CCC2)C)=O)cc2cccnc2[nH]1 c1(C(N2CCC(C)(CNC(=O)CC3CCCC3)C2)=O)ccc(O)c(Cl)n1 C1(NC(c2c(C)csc2)=O)CC2CN(C(C34CCC(C)(CO3)C4)=O)CC12 c1(C(=O)NC2CCC(NC(C3(COC)CCOC3)=O)C2)ccc(C#N)nc1O c1(C(=O)NC2(CNC(CC(C)F)=O)CCOC2)cc(Br)cn2ccnc12 c1(OC)cncc(C(N2CC(C)(NC(=O)CCCN3C(=O)CCC3=O)C2)=O)n1 CC(CC(=O)N(CCCCNC(=O)C(C)(Cl)Cl)C)c1ccccc1 C(N=c1[nH]cnc2cc(Br)ccc12)C1CN(C(c2c(CC)noc2)=O)CC1C c1(CC(=O)NC(CN(C(C(CC)OCC)=O)CC)C)c[nH]c2cc(Cl)ccc12 N1(C(C(CCC)O)=O)CC2CN(C(c3c(C4CCCC4)noc3C)=O)CC2C1 Cc1ccncc1CC(N1CC(CCNC(=O)C(C)(O)C2CCC2)C1)=O C12(C(=O)Nc3cc(CC)nn3C)CCCC1CCN2C(c1nsnc1NC)=O c1(C(=O)NCC2(C)N(S(CC(C)C)(=O)=O)CC2)cc2cc(Cl)ccc2[nH]1 c1(C(=O)NC2CN(C(C3ON=C(C(C)C)C3)=O)CC2C)ccc2c(c1)C(C)CN2 c1(NC(=O)NCCC(CCC)OC)c(C)n(C)n(-c2ccccc2)c1=O C(=O)(C1=Cc2ccccc2C1)NCCC1CC(NC(C2(C(C)C)CCCO2)=O)C1 c1(C(N(CC(C)(C)CNC(C2(C)CC2(F)F)=O)CC)=O)cccc(CF)c1 C#Cc1ccc(C(=O)NCCC2CC(NC(=O)CC(C)C(F)F)C2)cc1C c1(C(c2cccs2)C(=O)N(CCCC(F)(F)F)CC)cccc(Cl)c1 N1(Cc2n(CC)ncc2)CCC(C(=O)NC2CSC2)CC1 c1(CCCC(N2C(CN(C)C(C3(C)CCC(=O)N3)=O)CCC2)=O)cccc(Cl)c1 C1(NC(CC2(CC)CCC2)=O)C2CC3C1C3C2C(=O)Nc1cnc(C2CC2)nc1 N1(Cc2ncn(C)c2)CCc2[nH]nc(C(=O)Nc3c(Cl)cnn3C)c2C1 C=CCC(CNC(=O)CN1CCOCC1)C(=O)N(C)Cc1ccccc1C C1(C(=O)NC(CC(C)NC(=O)C(c2ccc(F)cc2)(C)C)C)CC1C1CCCC1 Cc1ccc2nonc2c1C(=O)NCC1=CCN(C(C2CC2(C)C(C)C)=O)CC1 C(C)(C)(CCN=c1cc(C(F)F)nc[nH]1)NC(c1n(C)ncc1Cl)=O c1(CCC(=O)NCCCCC2CN(C(C3(C(N)=O)CC3)=O)C2)cccc(F)c1F CCCCCCCCC(=O)N1CCCC2C1CCN2Cc1ccncc1F c1(CC(C)NC(c2c(CC)c(C)ccc2)=O)c[nH]c2c(C)cccc12 C1(O)(CC(=O)N(C2CCN(C(C3(OC(=O)CO)CC3)=O)C2)C)CCOCC1 CCCC(CC)CCC(=O)N1CCN(C(=O)C=CCN(C)CC)CC1CCO c1(C(N(C2CCCN(C(CCCOC(C)C)=O)C2)C)=O)cc2scnc2[nH]1 C#Cc1cccc(C(N2CC3CCC(CNC(C4CCCOC4)=O)C3C2)=O)c1C N1(C(c2cc(C(=O)OC)n(C)c2)=O)CCCC(O)(CCNC(=O)CCC(F)F)C1 c1(C(=O)OC(C)(C)C)cc(C(F)(F)F)ccc1Br.c12nc(co1)NC(=O)CO2 C1(C)(C(N(CCCNC(C(C2(OC)CCCC2)(F)F)=O)C2CC2)=O)CCCC1O c1(NCC(N2CCOCC2)(C)C)nc(-c2nn[nH]n2)cc(=N)[nH]1 C1(C(=O)NCCC(C(C)C)NC(c2cn(CCO)nn2)=O)CNC(=O)CC1C N1(CC(=O)N(C2CCN(C(=O)CCCOc3ccccc3)C2)C)CCOCC1=O C1(=CC(=O)NCCCCN(C(=O)C2=C(Cl)CCOC2)C)CC2CCC(C1)N2C C(=O)(C(C)(F)CC1CCC1)NCCN(C(Cc1ccn(C(C)C)n1)=O)C CC(C)(C(=O)NCC(CO)NC(=O)C(F)(F)c1ccncc1)C1CCCCO1 c1(C(=O)NCC(C2CCN(C)C2)OC)cccc([N+](=O)[O-])c1C C(C(O)C(=O)NC1(CNC(C2CCC(=O)C2)=O)CCC1)SC C1(C(=O)NC(C=C)C)CC2(CC2)CN1C(c1ccc(OC)nn1)=O CC(C)CCCCC(=O)N(C(C)CN(C(=O)CNC(=O)Nc1ccccc1)C)C c1(C(=O)OC)nc(=NCC(CO)c2ccc(Cl)cc2)cc[nH]1 C1(C(=O)OC)(OC)CN(C(c2ccc(I)cc2C)=O)CC1OC C(C)(C(C(=O)N1CCC(C)(N(C)C)CC1)C(C)C)NC(CCCOC)=O N1(C(C2CCCCO2)=O)CCN(C(c2cc(Cl)cnc2O)=O)C(CC2CC2)C1 C=CC(O)(C(=O)NC(CNC(c1ccc(C2CCC2)cc1)=O)CC)C(F)(F)F C1(C(=O)NC2CCN(CC(C)O)C2)CCS(=O)(=O)N1 Cc1cc(CC(N2CCC(NC(C3CCC=CO3)=O)CC2C)=O)cc(C)c1 c1(C(CC)C(=O)NCC(C)N(C(=O)C(=O)NCC)CC)cccc(C(F)(F)F)c1 c1(OC)cccc(C(=O)NCC#CCNC(=O)CC2(C(F)F)CC2)c1 Cc1cn(C)cc1C(=O)NCC1CC(CNC(c2nn(C)cc2Cl)=O)C1 c1(CC(=O)NC(CN(C(CCSCCCC)=O)C)(C)C)csc2c(F)cccc12 c1(C(N2CCC(CCNC(CN(C)C3CC3)=O)CC2)=O)ccc2c(c1)C(=O)NC2 CCCC(C)(CCC)C(=O)N1CCCC(CNC(C2(OC)CC(C)C2)=O)CC1 CC(C)CCCC(C)C(=O)NCC1CC(C(=O)NC2(C)CCSCC2)C1 N1(S(C(C)C)(=O)=O)CCCC2(CCCN(Cc3c(F)ccc(Br)c3F)C2)C1 c1(C(N2CCCCC(CNC(C3(CCC)CCC3)=O)C2)=O)c(C)ccc(Cl)c1N c1(OC)ccc(O)c(NC(=O)CC2C(NC(c3cnc(S)nc3)=O)CC2O)c1 n1(CC(=O)NCCN(C(C23CCC(CC2)C3)=O)CC)nc(C2CC2)n(C)c1=O C1(NC(C=CCOC)=O)COC2(CCN(C(=O)Cn3nc(C)c(Cl)c3C)C2)C1 CC1(NC(=O)CC2(c3ccccc3)CC2)CCN(C(C2CC23CC3(F)F)=O)CC1 c1(OC)ccccc1C(C)CC(=O)NC1CC(CCNC(=O)C=CC(=O)N(C)C)C1 C12(CNC(=O)CCc3cncs3)COCCN1C(=O)CN(C(c1cnc[nH]1)=O)C2 C1(CC(N2CCC(N(C(=O)CC3CCCCO3)CC)C2)=O)CC(=O)NC1=O c1(C(N2CCC(NC(CN(c3ccccc3)C)=O)C2)=O)ccc(Cl)nc1O Cc1noc(C)c1C(=O)NC1(CNC(C2CCN(C3CC3)C2=O)=O)CCC1 C1(C(=O)NC(c2nncn2C)C)CCN(C(=O)COCC2CC2)O1 Cc1ccc(C)c(C(=O)OCc2ccnc(Br)c2)c1O c1(CCC(=O)N(CCNCC)CC)cc(Cl)no1.C1(COCC=O)CCCCO1 C1(CC=C)(C(=O)NC(c2nccn2C)C)CN(C(c2csc(=N)[nH]2)=O)C1 CC#CCCC(=O)NC(C)(C(=O)NC(C)C(C)CC)C1CCC1 C1(OCCNC(C)=O)CCN(C(=O)NCC2(CO)CCCOC2)CC1 Cc1nc(C(N2CC(C(C)(C)O)(CNC(=O)C(=O)NCCC(N)=O)C2)=O)sc1C CC1(C(=O)NC2CCN(C(=O)Cn3cnc(C(N)=O)n3)CC2F)CCCNC1=O C1(C)(CNC(c2c(CN(C)C)ccs2)=O)CCN(C(c2nn(C)cc2Cl)=O)C1 N1(C(CC2(OC)CN(C(=O)Cn3cnc(C#N)n3)C2)=O)CC(CO)CC(C)(C)C1 c1(SC)nccc(C)c1-c1noc(C2CCCN2C(=O)C(C)(CO)SC)n1 CCCCC(C)CCC(=O)N1CCCC2(NC(c3cccn3C)=O)CCCC12 C1(N(C(C(C(C)(C)C)OC)=O)C)CC2CCC(C1)N2C(=O)C(C)(C)CF C(=O)(CC(C)C(F)(F)F)NCC1(C)CCN(C(C2CC(OC)(OC)C2)=O)C1 CCCCC(C)C(=O)NC1(CNC(C2(F)CCOCC2)=O)CCCCCC1 c1(C(=O)NC2C(NC(C3C(C)(C)C3)=O)CC2)cc2c(cc1N)CCCC2 C(C1CCN(C(=O)C#CC2CC2)CC1)=CC(=O)NCC1(CO)C(C=C)C1 CC1(C)CCCC(C)(NC(C2C=CCN(C(=O)CN3CCCC3=O)C2)=O)C1 c1(C(=O)NCC2C(C)CCN(C(=O)C(=O)NCC3CC3)C2)cc([N+](=O)[O-])cn1C c1(C(=O)NCc2c(C(=O)Nc3c(C)cc(Cl)cc3)c[nH]n2)cnc2ccccn12 N1(C(CSCC#C)=O)CCCC2(CCC(NC(c3cc(C)cc(O)n3)=O)C2)C1 Cc1cc(C(=O)NC2CC2NC(=O)CC2CN(C(C)C)C2)cc(C)c1 c1(C(N(C2CCN(C(CC(=O)OCC)=O)C2)CC)=O)cc(C(C)C)nn1C C(=O)(C(C(C)(C)C)N(C)C)NC(CNC(c1c(C)coc1)=O)(C)C(C)C C1(CC(N2C(CNC(=O)CCn3cccn3)CC2)=O)CC=CCC1 c1(C(C(=O)N(C)CCN(C(=O)C(C)c2ncco2)C(C)C)SC)ccccc1 C12(CC)CCC(C(=O)NC(C)CNC(C3(N4CCOCC4)CCC3)=O)(CC1)CO2 C1(C(N(C)CC2CCCS2)=O)C=CCCN1C(C1CCCC(=O)N1)=O C12(CNC(c3c(=N)[nH][nH]c3)=O)CCC(CC1)N(C(=O)CSc1ccccn1)C2 C1(COC)NC(=O)N(C2CCCCc3c(Cl)ccc(F)c32)C1=O Cn1nnc2cc(C(=O)NCC3CCCN3C(=O)CC3CC(C)(C)OC3=O)sc12 N1(C(C2C3C(NC(C(CC=C)CC)=O)C4C(C3)C42)=O)CCC(O)CC(C)(C)C1 N1(C(C(CCCC)O)=O)CCCC12CCCN(C(C1(C#N)CCSCC1)=O)C2 N1(CC)CCN(Cc2nc(C3CC3)no2)CC1.c1(NC(C)=O)nc(CC=O)cs1 c1(C(N(C(CC)C(N2CC(OC)C(O)C2)=O)C)=O)ccccc1F C(CC(C)(C)C)N(C(c1ccccc1)C)CCc1cnn(C)c1 C1(N)CC2CCCC(C1)N2.c1(C(S(=O)(=O)CCCl)=O)ccc(-n2cnnn2)cc1 CC1(C)CCCC(NC(C2CC(O)CN2C(c2scnc2Cl)=O)=O)C1 c1(C(NNC(C2C(C)c3c[nH]nc3CC2)=O)=O)ccc(N=Nc2ccccc2)[nH]1 C(CCCC(=O)N(C)Cc1ccccc1)N(C(=O)CNC=O)C c1(Cn2cc(C(=O)NC(CC)CO)nn2)cccc(NC(C)=O)c1 C1(C(=O)NCCc2n(C)cnn2)CC2CC1CN(C(c1cncnc1)=O)C2 N1(C(c2ncc(F)cn2)=O)CCC(C2(c3ccccc3)CC2)C1 C=CC(C)(C)C(=O)NCC(O)C(=O)NC1CC(O)C1OC C1(C(C(=O)NC(CCNC(C(c2ccc(C)s2)C)=O)(C)C)O)CCCCCC1 N1(C(C(C)c2cccs2)=O)CCC(C(=O)N(C)CC2CCCS2)C1 C1(C(=O)NCCC2CCOC2)C2CN(C(=O)CN3CCC(F)CC3)CC12 N1(CCN(C)C(C2CCNC2=O)=O)CCN(C(=O)CSc2ccccc2Cl)CC1 C(=O)(CCCS(C)(=O)=O)N1CC(CNC(C(C=C)c2ccccc2)=O)(OC)C1 c1(NC(C(F)=CCC)=O)ccc(C(N2CCC(OCCN(C)C)C2)=O)cc1 C1(NC(=O)COCc2ccccn2)CC2(C1)CN(C(=O)Cc1cnccn1)C2 N1(C(c2n(C)cc(C#N)c2)=O)CCC(C2CC2)C1CNC(=O)COCCN(C)C C(=O)(C1=NOC2COCC12)NCCN(C(=O)C(c1cccc(Br)n1)(F)F)C c1(C(=O)OC)sc2ncnc(N(CCCN(C)C(C3(O)CCCC3)=O)C)c2c1C c1(N(C(=O)C(C)=CCNC(=O)C(C)n2ccnc2)CC)ccccc1 N1(C(c2cccc(C(=O)OC)c2)C(=O)NCC=C)CCCC1P(C)(C)=O C1(C(N(CC(C)NC(c2cc(C)[nH]n2)=O)CC)=O)CC(=O)N(C(C)C)C1 CCC(CC(=O)NCC(C)C(C)O)NC(=O)CC1(COC)CC1 c1(OC)ccc(C(=O)C(N2CCC(O)(CNC(c3cc(C)on3)=O)C2)=O)cc1 CCCCCC(C)(C)C(=O)NCC(C)CN(C)C(c1cnn(C)c1C(F)F)=O C1(NC(C2N(N=O)CCCC2)=O)COC2(C1)CN(C(=O)C(F)(F)C(O)C1CC1)C2 N1(C(C2CCN2C2CCCC2)=O)CCN(C(=O)C2=CCCC2)C(CO)C1 C12(CNC(c3c(C)ncs3)=O)CC(NC(=O)C(F)C(F)(F)F)C(CO1)C2 c1(C(=O)NCC2CCCN2C(c2sccc2C(F)F)=O)cnn2c(=O)cc[nH]c12 CC(C)CC(C(=O)NCC1CCN1C(c1ncoc1C1CCCO1)=O)C(C)C c1(CCC)cc(C(=O)NCCc2cc(C(=O)N(C)Cc3ccccc3)no2)no1 CC1(n2nnnc2CC(O)C(C)(C)C)CN(S(=O)(=O)Cc2ccncc2)CCO1 c1(CC)ncccc1C(=O)NCc1cc(C)c(C(=O)NCCC2CCCO2)o1 Cc1c(C(=O)NCC(C)NC(C2(C)CCCO2)=O)cccc1S(N)(=O)=O C1(CNC(c2cc(C)ns2)=O)CC2(CCN(C(C3C(C)(C)C3(C)C)=O)C2)CO1 c1(NC(C(c2cccnc2)NC(c2cccnn2)=O)=O)cccc([N+](=O)[O-])c1 C12(C(=O)NC3CC(F)(CNC(CCCOCCOC)=O)C3)CCC(=O)N1CCS2 C1(NC(COC(CC)C)=O)CCC(C)N(C(c2ccc(=O)n(CCF)n2)=O)C1 CCCCC(CC)CCC(=O)N1CC(NC(=O)C(N)=O)CC(C)C1 CC(C)S(=O)(=O)C(C)C(=O)NC1CC(C)(NC(=O)C=CC2CCCN2C)C1 C(=O)(NN1CCCC1C(N1CC(O)C(O)C1CO)=O)C1CCC(C)(C)O1 C#CCC(O)C(=O)NC1C(C(=O)NCCOc2ccccc2)C1(C)C C1(C2CN(C(C3CC3(F)F)=O)C2)(NC(CC(C)c2ccccc2)=O)CC1 N1(C(C(F)=CC)=O)CC2CCC2(NC(c2ccc(OC3CCOCC3)cc2)=O)C1 c1(OC)ccc(C(=O)NC(C)(C)Cc2ccc(Br)cc2F)c(F)n1 Cc1cnc(C)c(C(=O)NCC2CCNC2)c1C C(=O)(CC1OCc2ncccc21)N1CCC(CCNC(c2cc(CC)[nH]n2)=O)C1 C(CCCC(CO)NC(C1(CCF)CC1)=O)NC(c1cc(C)ncc1)=O c1(NC(C(CC(=C)Cl)NC(=O)CCn2ccnn2)=O)ccc2nncn2c1 N1(C(C(N2CCOCC2)C)=O)CC2CCN(C(C3CNC(=O)N3)=O)CC12 C12(NC(N(CC(N3CCOCC3)C)CCOC)=O)CC1COC2(C)C c1(C(=O)NCC2(O)CC(C(=O)NCC(C=C)(C)C)C2)ccc2cncn2c1 c1(CC(=O)NCCN(CCOC)C(C2CCN(C)CC2)=O)cccc2nsnc12 c1(CN2CCC3(C(C(N4CCC(NC(C)=O)CC4)=O)C3)C2)cccc2c1OCO2 C1(CC)(CO)CCN(C(C2CCCN(c3cncc(N)n3)CC2)=O)CC1 C1(C(=O)NC2(C(COC)O)CC2)CSCCN1C(=O)CN1CCOCC1=O C(=O)(C(C(C)(C)O)NC(c1cc(C(C)=O)on1)=O)NC(C#C)C(C)(C)C CC1(C)CCC(C(N2CC3(C(=O)NCc4nncn4C4CC4)CC2CO3)=O)CC1 N1(C(Cc2scc(C)n2)=O)CCCC(NC(c2cc(C3(O)COC3)on2)=O)C1C C(=O)(CC(CNC(C1CC(CF)C1)=O)C1CCC1)N1C(COC)CCC1 c1(C(=O)NC2(C3N(C(CCCC#C)=O)CCC3)CC2)cc2scc(Cl)c2[nH]1 N1(C(C(COC)O)=O)CC2CC(NC(c3conc3C3CCCC3)=O)CC1C2 CC(Cc1ccccn1)C(=O)N1CCCC1CCNC(c1ccn(C)n1)=O C(=O)(C(CC(C)C)CC(C)C)NCCN(C(=O)C(C)(C)CCOC)CC N1(C(c2cc(C)sc2)=O)CCC(F)(CNC(C2CCC(CN(C)C)C2)=O)CC1 C1(C(=O)NCC(=C2CN(C(C3(C)CCC(=O)N3)=O)C2)F)CCc2nncn2CC1 c1(CC(N2C(c3cn(C(C(=O)O)C4CC4)nn3)COCC2)=O)nc2ccccc2s1 N1(C(C(CC)N(C)C)=O)CCC(C(C)NC(=O)C=Cc2ccn(C)c2)CC1 C(=O)(C(C)CCCC(C)C)NCc1cc(C(=O)NCC(C2CCC2)OCC)n[nH]1 Cn1nc2c(c1C(=O)NCC13CC1CN(C(c1cc(C(F)F)no1)=O)C3)CCC2 C1(OC)CC2CC(NC(=O)C(C)(C)C(C)NC(c3cc(Cl)cs3)=O)CC12 S(=O)(=O)(CCCNC(=O)CCC1CCCCN1C(=O)OC(C)(C)C)N(C)C C(=O)(CN=c1ccc(Cl)n[nH]1)N1CC=CC(NC(C2CC(F)C(=O)N2)=O)C1 N1(C(CNS(NC)(=O)=O)=O)CCN2C(=O)C(NC(=O)Cc3ccco3)CC2C1 N1(Cc2nc(OC)sc2)C(=O)NC(C2CCCO2)C1=O N1(C(C(COCC)n2cc(C3(C#N)CCOC3)nn2)=O)CCc2nn(C)cc2C1 CS(=O)(=O)c1ncc(C(=O)NC2(CO)CCCN(C(=O)CCOCC3CC3)C2)s1 C=CCC(C)(C)C(=O)N(C1CC(NC(=O)CC(C)C(=O)c2ccccc2)C1)C c1(CC(=O)N(CC(C)NC(c2csnc2Cl)=O)C)ccc(C(N)=O)nc1 C1(C(=O)NC(CCC)CCC)CC12CCN(C(C1(C)CC(=O)C1)=O)C2 N1(C(CC(CC)C2CC2)=O)CC(C2CCCCC2)CC1C C1(c2n(C(C)C)cnn2)CCN(N(C)CC2CC2c2ccccc2)C1 C1(CNC(CNC(CCC)=O)=O)CC2CCC1N2C(c1cccc(OC)c1N)=O C=CC1CCN1C(c1cc(CNC(c2nscc2C)=O)no1)=O Cc1cc(C)c(CNC(C2CC(F)CN2C(=O)C(F)C(C)(C)O)=O)cn1 c1(NC2CN(C(C(C=C)(C)O)=O)CC(C)(C)C2)ccc([N+](=O)[O-])c(C)n1 Cc1cc(=NCCSCC2CCCC2)[nH]cc1S(=O)(=O)N1CCn2ncnc2C1 CCCC(C)(O)CC(=O)N(CCCCCC(=O)NC(CN(C)C)C(C)C)C c1(NC(CCC(C)(C)NC(C2CC2(F)F)=O)=O)cccc(N=[N+]=[N-])c1 C1(OC)(CNC(=O)C(C)(C)n2cccn2)CCN(C(=O)C(C)NS(C)(=O)=O)C1 C(=O)(C(C(C)C)n1ccnc1)N1CC(CC(C)NC(CN(CCC#C)C)=O)C1 c1(C(=O)NCC2CC(F)(CNC(CC3ON=C(C)C3)=O)C2)ccc(C(N)=O)cc1 C=CC1(C(=O)NCCc2nccs2)CCN(C(=O)C(CO)OC)C1 N1(C(=O)NC2(C)CCCO2)CC(F)CC1CNC1CCC1CO c1(CNC(c2cnn(CC3CCC3)c2)C)cccc(Br)c1 c1(NC(CSc2n(-c3ccc(C)cc3)c(C)nn2)=O)nc2c(s1)CCC2 C1(CNC(C2C(CC(C)C)C2)=O)(CNC(c2cn(C)nn2)=O)CC(F)(F)C1 Fc1cc(F)cc2c1CCN(c1nc(NC3CCSCC3)c3ncsc3n1)C2 c1(C(N2CC3CC(NC(CCNC(=O)OCC)=O)C3C2)=O)cn2ncccc2n1 C1(C(N(C2CCOC2)C)=O)CCN(C(=O)COCC2CCCO2)C1 N1(C(CCNS(CC)(=O)=O)=O)CCN(C(=O)CN2CCOC2=O)CC1CCO C1(NC(CCNS(C)(=O)=O)=O)CCC2(CC1)CC(NC(C1CC1C1CCCO1)=O)C2 Cc1nc(C)c(C(=O)NCCN(C)C(c2ccc(C(C)(C)C)cc2)=O)c(C)n1 c1(C(N2CCC(O)(CNC(C(COC)(F)F)=O)CC2)=O)noc(C)c1[N+](=O)[O-] C1(NC(C=CC(C)NC(c2c(C)[nH]cc2)=O)=O)C=CCCC1CO N1(C(C(CCC)O)=O)CCn2ncc(S(C)(=O)=NC(=O)C=C(C)C(C)(C)C)c2C1 c1(C(=O)Nc2ccc(OCC)nc2)nn2c(c1-c1ccc(NC)nc1)CCCC2 N(C1CCc2cc(CNC(c3n[nH]cc3C3CCC3)=O)ccc21)C(C=CCC)=O c1(C(=O)NC(CCCC)CNC(c2[nH]nnc2C)=O)cc(C)c(C)c(C)c1 N1(c2nnc(C)o2)CC2CCCC(NC(c3cc(C4CC4)ncn3)=O)C2C1 C1(C)(CC(=O)N(C)CC2CCN(C(CN(CCC)C)=O)C2)CCOCC1 c1(CSC)nc(C)ncc1C(N1CC(C2(NC(C3CC3(C)C(F)F)=O)CC2)C1)=O c1(CC(=O)NCC(C(=O)N2CC(CO)(CO)C2)OC)c(C)n[nH]c1C C(=O)(C(F)CCC(C)C)N1CCC2C(NC(CCOCCC)=O)C2C1 N1(C(C2(CC=C)CN(NC(=O)CC3CCCC3)C2)=O)CC2CC2(C(=O)OC)C1 C(=O)(C(CNC(=O)C(O)c1ccsc1)C(C)(C)C)NC1(C#C)CCCCC1 c1(CC(=O)NCC(CO)NC(=O)CCCCn2ccnn2)cc(O)nnc1O C1(C(=O)NCC2(F)CC(CNC(C(=O)N(C)C)=O)C2)CCCN(S(N)(=O)=O)C1 Cc1cc(O)ccc1C(N1CCCC(C(=O)NCCc2ccc(F)cc2)C1)=O C(=O)(C1=NOCC1)NC1(CCCCNC(c2c(CC)occ2)=O)CC1 N1(C(C(C)(C)OC(C)=O)=O)CCc2c(CNC(=O)NC(=O)C(C)(C)C)cccc2C1 C=CCC(Cc1ccccc1)C(=O)NC1CC2CC1N(C(C13CSC(C1)C3)=O)C2 C1(NC(Cc2cnc(C)[nH]2)=O)CCC12CN(C(=O)C(C)CN(C)C)C2 CC(CS(C)(=O)=O)C(=O)NCC1CC1CNC(C1(C(F)F)CCCO1)=O c1(C(=O)NCC(C2CC2)NC(COCCCC#C)=O)ccc(OCCF)cc1 c1(NC(CC2(N(C)C)COC2)=O)cc2c(cc1C(=O)O)OCO2 Cc1nn(C)c(C(=O)NCC2(O)CN(C(C3(C#N)CCCC3)=O)C2)c1[N+](=O)[O-] C#CC(CC(C)(C)C)NC(C1(NC(=O)COC(CC)CC)CC(O)C1)=O N1(C(CCOCCC)=O)CC2CC(C1)CN(C(c1ccncc1Br)=O)C2 c1(CC(=O)NCCN(C(C2CCC3CC23)=O)CC2CC2)ncn2c1CCCC2 C1(CCNC(c2c(SC)ccs2)=O)CCN(C(C2CC(F)(F)C2)=O)C(C)C1 N1(C(C(C)Oc2ccccn2)=O)CC(NC(c2cncc(Cl)c2)=O)CC(C)(C)C1 c1(CNC(C2C(C(=O)OCC)C2)=O)ccc(C(=O)Nc2ncn(C(C)C)n2)cc1 N1(C(C2CN(C(C)C)C2)=O)CCC(F)CC1C(=O)N(C)CC1CC1 CCC(CC(F)(F)F)C(=O)N(CCCCNC(c1ccc(CN(C)C)o1)=O)C C#Cc1cccc(C(N2CC(C(=O)NCC(C)COCC)C(CCC)C2)=O)c1 c1(OC)ncc(F)cc1C(=O)NC1CCCC(CN(C(=O)C=C2CCC2)C)C1 C1(C(=O)NCc2cc(C)cc(O)c2)CN(C(=O)CS(C)(=O)=O)CCC1(F)F n1(CC(=O)NCC2(NC(C3C(C)(Br)C3)=O)CCCCC2)ncc2cccnc12 C1(NC(C(CC)CC2CCCCC2)=O)CC2CCC(C1)N2c1nnccc1C#N N1(C(C=C(C)Cl)=O)CC2CCC(NC(=O)Cc3cnc(C)nc3O)CC2C1 C1(NC(c2c(CC)nns2)=O)C2CN(C(C3(N(C)C)CCCCC3)=O)CC12 C1(CC)CCCCC1OCC(=O)NCCN(C(=O)CCc1cnc(C)o1)C(C)C C(=O)(CCC(=O)N(C)C)N(C(C1CCCN(C(c2cn(C3CC3)cn2)=O)C1)C)CC N1(C(COC(CC)C)=O)CC2CC1CC2NC(=O)CCCC1CCCC(=O)N1 CC(=O)CCCC(C)C(=O)N1CCC(CC(=O)NCC2(CO)CC=CC2)C1 N1(c2cc(OC)ncn2)CCCOC(CNC(c2cnc(SC)s2)=O)C1 C(C)(CCC(=O)NCC1(C)CC1(F)F)NC(CSCC=C)=O N1(C(=O)C(O)C2CCCC2)CC2CCN(C(=O)C(F)C3CC3)CCC2C1 C(CC(=O)N=c1ccn(C)[nH]1)N(CC(C)C)C(C1CCC(C#N)CC1)=O c1(C(=O)NC2CCN(C(C=Cc3c(C)ccs3)=O)CC2)ccc2nccn2c1 c1(N2C(C(=O)Nc3ccc(OC)nc3)CCC2)ncc(Br)c(N2CCOCC2)n1 N1(C(CC2CC(NC(=O)C(C3CCOCC3)=O)C2)=O)CC(CO)C(C2CC2)C1 Cc1nc(-c2ccccn2)sc1C(N1CC(NC(c2coc(N(C)C)n2)=O)C1)=O C(=O)(C1=CCCCC1C)NC1C(OC)CN(C(=O)C(C(C)O)N(C)C)C1 N1(C(C2CCC(O)CN2C(=O)C2=CCCCO2)=O)CCCc2occc2C1 Cn1cncc(C(N2CC3(CNC(c4cccn(O)c4=O)=O)CC2CO3)=O)c1=O c1(CN=C(NC2CCC(C(F)(F)F)CC2)NC2CCCCC2)ccc(Br)c(F)c1 Cc1nc(C(=O)NCC2(F)CCC(NC(C3(F)CC=CC3)=O)C2)c2ccccn12 C(=O)(CCCCC(F)F)N1CCC(CN(C(C2COC(=O)N2C)=O)CC)CC1 c1(CC(=O)NCCCN2CCC(NC(c3ccn(C4CC4)n3)=O)C2)ccc(F)cc1 n1(-c2cc(C)cc(C)c2)nc(C2Cc3ccccc32)nc1CCCC1CC1(F)F C(C)(C(O)C(=O)NCCc1ccc(CNC(C2(SC)CCOCC2)=O)cc1)SC N1(C(Cc2nc(C)oc2)=O)CCCC(C(C)C(=O)N(CC(F)F)C2CCC2)C1 N1(C(c2c(Cl)ccc(OC)c2)=O)CCC2(CCN(C(c3ccc(C)[nH]3)=O)C2)C1 c1(CNC2CCN(C(C3(C(F)(F)F)CCCC3)=O)C2)cc(O)nc(O)n1 C#CCC(C)(C(=O)N1CCC(C)(COC)C1)NC(c1cccc(C)c1O)=O c1(CCC(N2C(CNC(C(C)=C(CC)C)=O)C=CC2)=O)cccnc1Br c1(C(=O)NC2CCC(NC(c3cscn3)=O)C2)ccc(O)nc1 CC(C)(C)C(C(=O)N1CCCC(O)C1)NC(C1CCCC(=O)N1)=O c1(OC)n[nH]cc1C(=O)NCC(O)CNC(=O)CN1CC2CC2C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CN(C(=O)C(O)C1CCC1)C)(CO)CO N1(C(c2cc(C)ns2)=O)CCOC(C)(CNC(=O)C(C)(C)C2CCCCO2)C1 O=NN1CCCC1C(=O)NC12CC(NC(C3(F)CCOC3)=O)(C1)C2 N1(C(c2cn(CC)nc2C)=O)CCC(NC(=O)CCC2(C)CC2)C(F)C1 CCCCC(C)C(=O)NC(C)CCN(C)C(c1cc(O)ccc1C(F)(F)F)=O C(=O)(CCC(=O)NC)NCC1C(NC(CC2(OCC=C)CC2)=O)C1 C12(C(=O)NC(C)CCCCNC(C3CCOC3C)=O)C3CC(CC13)C2(F)F c1(C(=O)NC2C(NC(C#CC3(CC)CC3)=O)CCC2)ccc(C)c(S(C)(=O)=O)c1 c1(OC)c(F)cc(NC(=O)Cc2csc(Nc3ccccc3)n2)c(Br)c1F.C(C)=O C(=O)(CCC(C(C)C)NC(C1CC(O)CCO1)=O)Nc1cccc(CC)c1C C1(NC(C(C)(C)CF)=O)CCC2CN(C(=O)CSc3ccccc3)CC2C1 C#CCCCCCC(=O)NC1CC2CC(C1)N(c1nccnc1F)C2.c1ccccc1 c1(C(=O)NCC(C)N(C)C(c2cnsn2)=O)cnc(O)c2cnccc12 C1(OC)CN(S(=O)(=O)c2ccc(C(F)F)o2)CC(F)(F)C1 C1(Cl)(NC(CNC(CC(C)C)=O)=O)CC12CCOCC2 C1(C(=O)NCC2CN(CCC)C2)CCN(C(=O)CCC(=O)NC)C(CC)C1 N1(c2nccc(C(F)(F)F)n2)CC2(CCCC2)C1 N1(C(CN(C)C(N)=O)=O)CC(NC(C2(C#N)CCCO2)=O)CC12CCOCC2 CC1CN(C(C2CC2C(F)(F)F)=O)CCCN1C(=O)Cc1ccsc1 c1(CC(=O)N(C2CC2)CC2(OCC)CCC2)nccn1C.C1(=O)CCN1 C#Cc1ccc(C(=O)NC2CCCC(N(C)C(c3coc(C)n3)=O)C2)cc1F Cc1nc2ccc(C(N3CCC4CN(C(=O)C(C)CC5CC5)CC34)=O)cc2[nH]1 N1(C(c2c(CC)n(C)nc2)=O)CCN(c2ccnc(C#N)n2)CC(C)(F)C1 C12(NC(=O)C=CC3CCOCC3)CCOCC1CN(C(C1(Cl)CC1)=O)C2 c1(C(=O)NCC2CN(C(CCC(=O)NCCC)=O)C2)ccc2ccnc(O)c2n1 C(C)(C)(CC(=O)NCCC1(O)CCN(C(=O)C(F)Cc2ccccc2)C1)SC N1(C(c2c(C)cc(N)cn2)=O)CCCC2(C1)CN(C(=O)Cn1ncc(Cl)c1C)C2 C=C(CNC(C1CC1(F)Cl)=O)CCNC(c1ccnn1CC(F)F)=O CC1=NN(c2ccc(C(=O)NCC(O)CN(C(=O)C3=CCCS3)C)cc2)CC1 c1(N(C(c2scc(C(NOCCCC#C)=O)c2)=O)CC)cncc(C#N)c1 c1(C(C)NC(c2nnnn2C(C)(C)CC)(C2CC(=C)C2)C)cnccn1 CC(C)C(C)(O)C(=O)NC(CNC(c1ncsc1C(F)(F)F)=O)C1CCC1 CC1(C)CCOC(C(N2CC=CC(C(=O)NC3CC(C)(C)OC3=O)C2)=O)C1 C1(NC(c2cccc(CC)c2)=O)CCN(C(c2ccnn2C(C)(C)C)=O)CC1F C1(CS(C)(=O)=O)CCC(C(=O)NCC2CN(C(=O)C(O)Cc3cn(C)cn3)C2)O1 CC1CC=C(C(=O)NCCC2CCCCN2c2ncnc3c2CCC3)CC1 C1(CCCCNC(c2ccc(C(F)F)o2)=O)CCCN(C(=O)COCC(F)F)C1 C12(C(N3CCCC(CC4CCN(c5scc(OC)c5)C4)C3)=O)CC1CCC2(F)F C(=O)(C(C)C(O)C(C)C)NCCCOCCCNC(CC(CCC)C)=O Nc1ncc([N+](=O)[O-])cc1C(=O)NC1CCC(NC(C2CCCN2N=O)=O)CC1 C1(NC(CC2C(C)(C)C2)=O)CC2(CCCCN2C(c2cccc3c[nH]nc23)=O)C1 c1(CN2CCCC(C)(C(=O)NCc3ccc(Br)cc3)C2)ccc(S(N)(=O)=O)cc1 N1(C(C)=O)CC(O)CC1C(=O)N(C1CCCN(C(C2CCCO2)=O)C1)CC1CC1 C1(CNC(c2cnc(C(C)OCC)s2)=O)CC2(CC2)CN1C(c1cnsc1C)=O c1(C(=O)NC(C)CC(C)NC(C23CCC(CC2)CO3)=O)cc(Cl)c(F)cc1O c1(C(=O)Nc2c(C(C)C)nsc2)ccnc(CNC(C2CCC(=O)C2)=O)c1 C1(CNC(C(N)=O)=O)CC2(CCOCC2)CN1C(=O)CC1CCCOC1 c1(NC(CNC(c2c(C(C)C)ncs2)=O)(C)Cn2cccn2)ccc(C#N)nn1 C(=O)(CN=c1ccc(C#N)c[nH]1)N1CCC(CN(C)C(C2(C3CC3)CC2)=O)C1 Cc1ncnc(C)c1C(=O)NCC(CO)NC(=O)CSc1nnnn1C1CC1 c1(C(=O)NCCN(CCC)C(C2(CS(C)(=O)=O)COC2)=O)cc(Cl)cnn1 n1(C(C)(C)C)nnnc1C(C)(CSCCF)NCCC1CCOC1 C1(C(N2C(CNC(C3CCCC4CC34)=O)CCC2)=O)COc2ccc(O)cc2O1 C(=O)(C(C)CC(F)(F)F)NCc1c(C(=O)NC(CC)C2CC2)con1 N1(C(c2c(CNC(C3C(C)(C)C3(F)F)=O)ccs2)=O)C2CCCC1CC2 CC1C(NC(=O)C(C)(C)C2CCC2)CCN1c1nncs1 c1(C(N(CC(CC)NC(=O)C(C)S(N)(=O)=O)C)=O)cc2ncccc2[nH]1 c1(C(=O)NOCC2C=NNC2=O)ccc2c(c1)OCO2 Cc1cncc(C)c1C(=O)NC1CC(C)(NC(C2CCC(F)C2)=O)C1 CCCCCCN(CCNC(=O)CN1CSCC1=O)C(C1CCCSC1)=O N12CCN(CC1)C(C1CC1)c1cn(nn1)CCC2=O.C(CCCC1CC1C)OC C1(NC(CN(CCOC)C(C2CCCSC2)=O)=O)CCCC(O)CC1 C1(CC(=O)NCC(C)(C2CC2)NC(C(CCCC)C)=O)CC2(CCCC2)CO1 C1(C(N(CCN(C(=O)CN2CCC2C)C(C)C)C)=O)COc2ccc(Cl)cc2O1 C1(C(=O)NC(C(C)SC)C)CCN(C(=O)CC2C=CCC2)CC1O C(=O)(CCCCC(C(=O)NC(C)(C)C)NC1(C)CCCC1C)OC N1(C(C(C)c2cccs2)=O)CCCC(F)(C(=O)NCCN2CCCC(O)C2)C1 N1(C(C(C)SC(F)(F)F)=O)CC2(CC(NC(=O)C(C)(O)C3CC3)CO2)C1 c1(CNC(C2(C(C)(F)F)CCC2)=O)ccccc1CNC(C1(C)CC1(C)C)=O CC1CN=NC(=O)C2(CCN(Cc3cccc(-c4nnsc4Cl)c3)CC2)N1 O(NC(=O)COCCNC(c1ccoc1C1CC1)=O)C(CC)C CC(=O)CCCC(C)C(=O)NC(C)C(C)NC(C12CCC(CC1)CO2)=O C(C(C)(O)CC(=O)N1CC(C2CN(C(c3cccc(F)c3Br)=O)CCO2)C1)OC Cc1ccccc1NC(=O)C(C(C1CC1)C1CC1)N1CCC(N2CCCC2)C1 C(=O)(C#CC(C)(C)O)N(C)CC1COCCN1C(c1ccc(F)cn1)=O O=S(=O)(c1cnc(NCCCc2nncs2)c(Cl)c1)NCC1CCC1(F)F c1(C(N2CCC(CCNC(c3n(CC)ncc3)=O)C2)C)ccc(Br)cc1 Cc1ccc(C(N2CCCC(CNC(=O)C(c3ccc(F)cc3)=O)C2)=O)cc1 c1(OC)ccc2c(c1)CCCC2.C1(=O)CCC(=O)NC(OC)C2C(COC)C2O1 N1(C(c2n(C)cnc2)=O)CC=C(CC(=O)N2CC(c3nncs3)C2)CC1 C1(NC(C(CC)O)=O)(CNC(=O)Cc2ccc(C(C)=O)cc2)CCOCC1 N1(C(COc2cccc(C)c2)=O)CCC(CNC(C2(C)CC(F)C2)=O)C12CCC2 C(=O)(C(C)(C)Cc1cnn[nH]1)N(CCCNC(C(c1scc(C)n1)(F)F)=O)C C(=O)(C(CC)CC=CC)N1C(C(=O)NCCC#C)C(C)C1 C1(OC)C(C)(C)CN(c2nc(C)ns2)C1(C)C C(C(O)C(=O)NOCCc1ccccc1)NC(c1cccc(F)c1)=O Cc1ncc(CC(=O)NC(CNC(C2(c3cncnc3)CCCC2)=O)C2CC2)s1 C1(NC(C2CSCCS2)=O)CC1C1CCN(C(=O)CCC2CCC2)CC1 c1(CC(=O)N(CCN(C(c2cnc(OC)s2)=O)CC)CC)nc(C)c(C)s1 CC1CCC(C(=O)N(C)CC2CCCS2)N(C(=O)COCCCN(C)C)C1 N1(CC(=O)NCC(C)(CO)NC(CC)=O)C(=O)CC(C)(C)C1=O c1(OC)cc(F)c(C(N2CC(C)(NC(=O)CC3C=CCC3)C2)=O)c(Cl)c1 c1(C(c2nnnn2C2CCC2)NC(C)C(C)(C)F)ccccc1C(C)(C)C C#CC1CN(C(C2(C(C)C)CCN(C(=O)CCc3nncs3)C2)=O)CCO1 N1(C(C(C)OCCCC)=O)CCC2C(CCN2C(c2ccnc3[nH]nnc23)=O)C1 c1(OC)csc(C(N2CCN(C(=O)Cc3ccccc3Cl)CC2)=O)c1OC C1(C(C(=O)NCC2N(C(C(CCC)N(C)C)=O)CCC2)OCC)CCCCCC1 n1(CCC(N2CC(CNC(C3(C#C)CC3)=O)OCCC2)=O)cc(S(N)(=O)=O)cn1 N1(C(C(CC)(C)F)=O)CC(NC(c2cc3c(s2)CCC3)=O)C2CCCC2C1 c1(C(N2CCC(CCC(=O)NC(C3C(C(=O)OC)C3)C)C2)=O)sc(O)nc1C c1(C(C(=O)N(CCCNC(C(C(=O)OC)(C)F)=O)CC)O)cccc2c1OCC2 C1(CNC(CC=C(C)C)=O)CC2CCC(C1)N2C(c1ncc([N+](=O)[O-])n1C)=O Cc1nc(CC(=O)NC2CCCC(NC(C3(O)CCSC3)=O)C2)c(C)s1 c1(C(=O)NC(CCNC(CC(CC)OC)=O)C(C)C)cccc2oc(C)cc12 C1(C(=O)NCC2(CC)CCC(=O)N2)CN(C(c2ccsc2C)=O)CC1C1CC1 C1(C(=O)NCC2(NC(=O)CC3(n4cncn4)CC3)CCOC2)CC2CCC(C1)O2 c1(CC)nnc(N2CCC(C(F)F)CC2)n1CCCSc1csc(C)c1 C1(NC(c2c(C)cc(C)[nH]2)=O)CN(C(=O)C=Cc2cnc(C)s2)C2(CCOC2)C1 N1(C(c2cc(C)sn2)=O)CC2CS(=O)(=O)CC2(NC(=O)C2=CC(C)(C)C2)C1 c1(CC(N2CCCC(N(C(C(OC)OC)=O)C)CC2)=O)cn2cccc(C)c2n1 C1(C(N(CC(C)NC(C2(CO)CCC2)=O)C)=O)CCCC(N(C)C)C1 C1(OC)CCCC(C(N2CC(C(C)NC(=O)CCC3CCCC3)C2)=O)C1 c12cc(ccc1F)NC2=O.CC(C)(C(=O)NCC(=O)NOCCC(F)F)C1CC1 N1(C(CC2C(C)C2)=O)CC(C2CCCN(C(C3CCC(=O)N3C)=O)C2)C1 C1(CC(=O)NCCCCCN(C(C2(F)C(C)C2)=O)C)COc2ccccc2O1 c1(C(=O)NC2CC(N(C)C(C34CCC3C4)=O)C2)cccc(-c2ccc[nH]2)c1 CCC(C)C(=O)C(=O)N1CC2CC1C2NC(c1ccccc1)=O C1(C(=O)NC(C#C)(C)C2CC2)CN(C(C2CN(C(=O)NC)C2)=O)CCN1C N1(C(C(=O)NCC)=O)CCC2CN(C(=O)CC34CCC(CC3)OC4)CCC2C1 CCC1c2ccsc2CCN1C(c1c(OC)ccc(Br)c1C)=O C(=O)(CC(C)P(C)(C)=O)N(C(C)CCNC(c1c[nH]nc1C1CC1)=O)C Cc1ncc(Cl)cc1C(=O)NC1CCCCC1NC(c1conc1C1CCC1)=O c1(CC(=O)OCC(c2ccc(F)cc2)C)ccc(C(F)(F)F)cc1 N1(C(c2c(C)cn(C)n2)C(=O)NCCC2(C)CC2)CCC(C)CC(C)C1 c1(C(=O)NC2C3CN(C(C(C)C(C)(F)F)=O)CC32)cnc2nccn2c1 c1(C(=O)NCC2CCN2C(c2scnc2C(F)F)=O)ccc2c(c1)NCC2 C(=O)(C1=CCCN(C(=O)Cc2ccn(C)c2)C1)N1CC(C)C(N(C)C)C1 CCC(C(=O)N1CCC(CNC(c2ccc[n+]([O-])c2)=O)CC1)C(C)O C1(=CC(=O)NCCNc2nn(C)cc2Br)CCN(SCC)CC1 Cc1cc([N+](=O)[O-])cc(C(=O)NCC(O)CN(C)C(C2CC(CF)C2)=O)c1Cl c1(CC(=O)Nc2nc(C)c(-c3ccc(N)c(Cl)c3)cc2)cccc([N+](=O)[O-])c1 Cc1nc(N(C)C)sc1C(N1CCC(CCNC(c2ccc(F)o2)=O)C1)=O c1(C(NC(=NC)NC(C)COCCOC)C#C)ccccc1Br C1(CC(=O)NCc2nc(C(=O)NCc3nc(N(C)C)n[nH]3)co2)CCC(=O)NC1 C1(C(=O)NCC(C2CCN(C(CC(C)(F)F)=O)CC2)(C)C)CC2C=CC1CCC2 C1(NC2(CC=C)CCCCCC2)CCc2c(cnn2CC)C1 c1(C(N2CCC(O)(CN(C(=O)C3=CCCOC3)C)C2)=O)cc(O)cc(F)c1 c1(-c2nnc(N3CCC(CCOC)C3)n2C)cc2sccc2s1 C1(CCC)(NC(=O)C(CC(C)C)OC)CCCN(C(=O)CN2CC3CC3C2)C1 C1(C(=O)NC(C(C)NC(CCNC(C=C(CCC)C)=O)=O)C)CCCCN1CC c1(CC(=O)N(C)CCOCCCNC(=O)C(N)=O)nnc(-c2ccccc2)o1 N1(C(C(COC)NC(=O)OC(C)(C)C)=O)CC(NC(C2CCCN2C)=O)C(O)C1 N1(C(CCCNC(=O)NCC#C)=O)CC2CC1CCN2C(=O)CC(C)(C)OC N1(C(c2c(C)noc2C)=O)CCOCC(NC(=O)C=Cc2ccn(C)c2)C1 c1(OC)ncc(C(=O)NCCOCC(C)(C)NC(=O)CC2(C)CCOCC2)cc1C C(=O)(CS(=O)C(F)(F)F)NCC1(F)CCN(C(c2c(CC)cncc2)=O)C1 C12(CNC(c3c(COC)noc3)=O)CC(NC(C3CC3(C)C)=O)(CCO1)C2 C(C1CCCCC1)=CC(=O)NCC(CNC(C(N)=O)=O)O C1(NC(C(C)N)=O)CCC(CCC2CC2)C1.CCC(=O)C1(C(=O)NNC=O)CC1 CCCCS(=O)(=O)CC(=O)N1CC(NC(c2cc(F)ccc2Cl)=O)C(C)C1 N1(C(C(CC)N(C)C)=O)CCCN(C(c2ccc(OC)c(OC)c2C)=O)CC1C C1(CNC(CCC(N)=O)=O)(NC(c2cnn3c2OCC3)=O)CC2CCC1C2 c1(-n2cc(C3(C)CC3)nn2)ccc(F)c(C(F)(F)F)c1.C12CCCN1CC(=O)N2 C1(C(=O)NCC(n2ccnn2)C)CCN(C(=O)CSC2CC2)C12CCC2 c1(NC(=O)CCN(C(C2CC2(F)Cl)=O)C2CC2)cccc(CCO)c1 c1(C(N2C(CC)CN(C(c3cnn(C)c3)=O)CC2)=O)cnc2ncnn2c1O c1(C(=O)NCc2c(C(=O)NCCC3(C)CC3(F)F)nco2)cccc(O)n1 C(=O)(CS(=O)(=O)C1CCCC1)NCC(C)(C)CNC(C1CC12CCCOC2)=O CCC1=C(C(=O)N2CCCN(C(C3CCCN(C(C)=O)C3)=O)CC2)CCCO1 C1(NC(C2(CC)CC2)=O)CCOC(CNC(C2CC3(CCC3)C2)=O)C1 CCC(CC(=O)NCC1CC(F)(CNC(c2cc(C#N)c(C)cn2)=O)C1)C(C)C C1(C(=O)NC23C(CN(C(c4cc(C)sc4C)=O)C2)C3)Cc2nncn2C1 C1(CC(=O)NC(C2CN(C(C3(C)C(C(=O)OC)C3)=O)C2)C)CCCN(C(C)C)C1 N1(C(c2cc(CC)no2)=O)CC(NC(=O)CN(CC)CC)CC2(CCC2)C1 NS(=O)(=O)c1sc(Cl)cc1C(N1CC2CCN(C(=O)CNC=O)CC2C1)=O N1(C(CC2C(C)C2)=O)C2CCC1CC(N(C)C(C13COCC(C1)C3)=O)C2 C(=O)(C(C(=O)N1CC(CCC(=O)NOC2CCCCC2)C1)OC)OC c1(C(=O)NCC(CNC(=O)CCn2cccn2)F)ccc(Br)cc1F CN(C)C(=S)NCC1(CN2CCCC2)CC1 c1(NC(C2N(C(Cc3nc(C)on3)=O)CCC2O)=O)c(Br)c(C(C)C)nn1C Cc1c(C(=O)NC2CCCCN(C(C3(C(F)(F)F)CCC3)=O)C2)nn(C)c1N C12(CNC(C(C(C)C)O)=O)CCC1CN(C(=O)CCC(C)(C)F)C2 c1(CC)nn(C)c(CC(=O)NCC2(F)CC(NC(=O)Cn3cccc3)C2)c1Cl CC(CC(=O)NCCC1(C)CCCC1)C(C)(C)NC(c1coc(CO)c1)=O c1(C(N2CCC(O)(CNC(c3[nH]c(=NC)sc3)=O)C2)=O)cc(OC)cnc1F N1(C(C(C)C(F)F)=O)CCOCC(NC(=O)C(F)(F)CN(C)C)C1 CC(C)C(CN=c1ccc2nnc(-c3cccc(C(F)(F)F)c3)n2[nH]1)N(C)C C1(C(N2CCN(C(C(CCC)OCC)=O)CC(O)C2)=O)CCc2nnc(O)n2C1 C=C=C(C)CC(=O)N(C1CCN(C(=O)C(C)C2CC2)CC1)CCOC c1(CCC(N2C(C(N3CCCC4(CCO4)C3)=O)CC2)=O)ccc2c(c1)CCO2 N1(CC)CCC2CN(S(=O)(=O)N3CC(NC(=O)Nc4ccc(NC)cc4)C3)CC12 n1(CC#C)c(C)cc(C(=O)NC2(CC=C)CCN(C(=O)CC(CC)OC)C2)c1C c1(COC)ccc(NC(C2CCCN(Cc3cc([N+](=O)[O-])cs3)CC2)=O)c(C)c1 C1(CC(=O)NCCCCN(C(C)C)C)CN(C(C2COC(=O)N2)=O)CCO1 c1(CC)cc(C(=O)NCC=CC(=O)NC)ccn1.N12CCCC1C2 C(=O)(C(F)C(C)(F)F)NC1CC(C(N(c2ccc(O)cc2)CC)=O)C1(C)C O=C(CCC(=O)c1cccc(Cl)c1)NC1CC(NC(=O)Cn2cnccc2=O)C1 C1(NC(C2N(C)CCCC2)=O)COC2CN(C(c3scnc3Cl)=O)CC12 c1(C(=O)NCC(C2CCN(C(C(C=C)O)=O)CC2)C)cc2ncccn2n1 C1(NC(C2CCCC2)=O)C2CC3CN(C(C45CCCC(C4)OC5)=O)C1C3C2 c1(OC)cc(OC)c(OC)cc1CNC(=O)NCC1(CO)CC=CCC1 Cc1ccc(C(=O)NCC(C)CNC(=O)C(C)N(C)C)c2cccnc12 N1(C(C2N(C)CCC2)=O)CC2(C1)CN(C(C1(CO)CCCO1)=O)CC2CO CCC(C)(F)C(=O)NC1CC(O)(CNC(c2ncn(-c3ccccc3)n2)=O)C1 CC(C)(CC(F)C(=O)NCC1CSCCO1)NC(=O)CC1CCCCC1 C1(NC(CCCC#C)=O)CN(C(c2ccnn2COC)=O)CC12CC2 c1(C(C(=O)NCCOCC)N(c2cc(F)ccc2F)CC)ccc(F)c(Cl)c1F CCS(=O)(=O)c1ccc(Cl)cc1NC1CCCOC1c1ccc(Cl)cc1 c1(C(=O)NC(C(C)(C)C)CNC(=O)CC2(C3CC3)CC2)cccc2ccnn12 c1(C(=O)NCC(C2CCC2)NC(C2N(C)CC2)=O)cn2c(n1)CCCC2 C1(O)(C(=O)NCC(CNC(C(C)c2ccco2)=O)F)CC(C)(C)C1 c1(CC(=O)NC2C(F)CCN(C(C3(OC)CCC3)=O)C2)ccc2c(c1)COCC2 C1(CC(=O)NCCOCCCNC(C=CC(CC)=CC)=O)CC2C=CC1C2 C1(C2(O)CCC2)(C(=O)NCCC(C)(C)NC(=O)CCc2ccnc(Cl)c2)CC1 CC1(C)CC(N)CC(C(=O)NCc2csc(-c3ccco3)n2)O1 C1(C(=O)NC2CC(C)N(C(c3cccc(N)c3N)=O)C2)CCc2c[nH]nc2C1 C1(CC(=O)NCCN(CC(C)O)C(C2C=C(C)CS2)=O)CC(CC)=NO1 c1(C(=O)NC(CC)CN(C(=O)CCOCCOC)CC)cc[nH]c(=N)n1 N1(C(=O)CO)CC2CCN(C(c3cnc(N4CCS(=O)(=O)CC4)nc3)=O)C2C1 C(=O)(C(C#N)C(C)C)NC(C(=O)NC(c1c(C)nc(C)[nH]1)C)C(C)C c1(C(=O)NCC2N(C(C(CCC)C)=O)C3C(C2)C3)cnc2sccc2c1 C1(CC(=O)NC2(CC)CCN(C(c3c(C)ncn3OC)=O)C2)CCCNC(=O)C1 C1(C(=O)NC2C=CCN(C(C3(CC(C)C)COC3)=O)C2)CC1C1CCCCC1 c1(C(=O)NC(C(C)NC(=O)COC2(C)CCCC2)C)ccc(N)cn1 C1(C(N(CCNC(CSCC)=O)Cc2ccccc2)=O)COc2ccccc2O1 c1(OC)ccc(Cl)c(C(=O)NC2CN(C(=O)C3=C(C)CCC3)C3(CCC3)C2)c1F CCC(C)(CNC(C1CC(OC)(OC)C1)=O)C(=O)N=c1ccn(C)[nH]1 C1(NC(C2(NC(C3N(C(C)=O)CSC3)=O)CCCC2)=O)CC(=O)N(C(C)C)C1 N1(c2nnc(C(=O)OC)s2)CC2C(NC(=O)CCCCc3ccccc3)C2C1 C(=O)(CC(C)CC(C)C)N1CCCC(O)(CN(C(c2cnc(C)o2)=O)C)C1 C(=O)(C(O)CC(C)(C)C)NC(CNC(C(c1c(OCC)cccc1)(F)F)=O)CC C(C(C)(F)CNC(=O)CNC(c1ccccc1)=O)NC(CN(CC)CC)=O N1(C(c2ccc(=NCC)[nH]c2)=O)CC(C)CN(C(=O)C(C)COC)C(C)C1 C1(CC)CN(C(=O)CCNC(=O)CCC(C)(C)F)CC(=O)N1 C1(C(=O)NC2CCN(C(=O)CCCN3CCCC3)C2)CCCC2(C1)CC2(F)F n1(C(C)C)ccc(C(C)NC(c2csc(C(F)F)n2)=O)n1 C1(C(=O)NCC2(NC(C(C)OC)=O)CCC2)CN(S(N)(=O)=O)C1 C1(C(=O)N(C2CCN(C(c3coc(C)c3)=O)CC2)C)(OC)CCS(=O)(=O)C1 c1(C(=O)NC(CCOCC)C)c[nH]nc1CCNC(C1CCCO1)=O c1(CN(C(=O)CCC2CCC(=O)N2)C)cc2nc(Cl)ccc2s1 c1(CC(=O)NC(C2CCN(C(C(CSC)C)=O)C2)(C)C)ccccc1CO Cc1cc(C#N)cnc1C(=O)NC(Cc1ccco1)C(N1C2CSCC1C2)=O c1(OC)ccc(CC(N2CCCC(CN(C(=O)Cc3cnccn3)C)C2)=O)nc1 c1(C(=O)NC2(CNC(c3c(C)n[nH]c3C)=O)CCOC2)ccc(S(C)(=O)=O)s1 C12(CNC(c3cc(CNC(CC)=O)c(N)cc3)=O)CCC(CO)(CC1)CO2 N#Cc1ccncc1C(N1CCC(C(=O)NCCN2C(=O)CSC2=S)C1)=O C(C(O)C(=O)N1CC(C(N)=O)(CNC(=O)C(C)(C)C2CCCCC2)C1)OC N1(C(C(CC2(N(C(=O)CC3CC=CCC3)C)CCC2)F)=O)CC(CO)CC1CO c1(C(N2C(C(=O)OCC)CC(C)(C)C2)=O)nc2ccccn2n1 C(=O)(C(C)(C)C(F)(F)F)NCC1CCN(C(c2c(CC)n(CC)nc2)=O)CC1C O(N(C(=O)c1coc(C)n1)C(C)C)Cc1cnn(C)c1C.CCOC c1(C(N2CCC(CNC(Cc3cc(C)cc(F)c3)=O)C2)=O)cnn2ncccc12 c1(OC)cccc(C(=O)NCCC2(NC(C3CC(O)C(F)C3)=O)CCC2)c1F N(C1CCCOc2cc(F)cc(F)c21)c1ccc(S(=O)(=O)N2C(C)CC2)c(Cl)c1 N1(C(C(CC(C)C)NC2C3CC2(c2ccco2)CO3)=O)CCCC(C2CC2)CC1 c1(OC)cccc(C(F)(F)C(=O)NCCCCNC(=O)CC2(C)CC2F)n1 c1(C(=O)NCC2C(NC(c3nn(C)c(=O)cc3)=O)CC2)cncc2cccnc12 Cc1nc(C)c(CNC(C2CCC(CNC(c3cccnc3C)=O)CC2)=O)[nH]1 CC1CCC(F)(F)CN1C(=O)C#CC(C)(C)CNC(c1ccn(C(F)F)n1)=O c1(OC)cc(C(=O)NCC2CCCCC2NC(=O)C(C(C)C)SC)cnc1OC n1(CC)c(N2CCCC2C23CCC(CC2)C3)nnc1-c1cc(Br)co1 N1(C(c2c(C)ncs2)=O)CC(NC(=O)Cc2cc(C)n(C)n2)C(F)C1 c1(NCC(C)C2CCC2)ccc(S(=O)(=O)NCC#CCCO)c(Cl)c1 C1(NC(=O)Cc2ccc(O)nc2)(CF)CCN(C(=O)Cc2ccccc2)C1 c1(C(N2CCCC(F)(CNC(c3cnn[nH]3)=O)C2)=O)cc(F)c(Cl)cc1Cl C1(CN(C)C(c2ncsc2Br)=O)CCN(C(=O)C(=O)NCC(F)F)CC1 N1(C(C(CC)N(C)C)=O)CC2CCN(C(c3cccc(CCO)c3)=O)CC2C1 CCC(O)CC(=O)N=c1ccn(CC(=O)NCc2ccoc2)c(O)n1 C1(CC(N2CCC(NC(CC(=O)OC)=O)C2)=O)CCCC(C)(C)O1 N1(C(C2CC(C#C)(O)C2)=O)CCC2(C(=O)NCCc3cn(CC)nn3)CCCC12 C(=O)(CP(=O)(C(C)C)C(C)C)NCCN(C(=O)Cc1ccc(F)cc1C)CCC C(CC(C)C)(C(=O)NC1CN(C(c2ccn(C(C)C)n2)=O)CC1C)OC c1(C(=O)NCC2N(C(CC(C(C)C)OCC)=O)CCC2)cccc(C#N)c1Br C1(C(N2CCC(C)(COC)C2)=O)CN(C(=O)CN2CCCCC2C)CCN1C C=CCC(C)(C)C(=O)N1CC(F)(F)CC1C(=O)NCc1c(Cl)cncc1Cl C1(NC(CN(CCC#C)C)=O)CN(C(c2ccc([N+](=O)[O-])n2C)=O)CC1C1CC1 C1(C(N2C3CN(C(c4c(C)cccc4)=O)CC2CC3)=O)CC2(CCOCC2)CO1 c1(NCCC)nccc(C)c1C(=O)C(=O)NC(CNSS(C)(=O)=O)CC c1(C(N2CCN(C(C3CCCS3)=O)CC2C(F)(F)F)=O)cc2ccc(Cl)cc2s1 C(CC(C)C(F)(F)F)NC(=O)NC1C(C=C)COC1 c1(CC)nn(C)cc1C(N1CCC(C(=O)NC(C)C2CC2)(CF)C1)=O c1(OC)ccc(C=CC(N2CCC(NC(=O)CC3CCC4CC34)CC2)=O)cc1Cl c1(-c2c(C)ncs2)ccc(F)c(CN(CC(N)=O)C(C)(C)C)c1 S(=O)(=O)(C1CC2(CC2)C1)NC(c1ccccc1)CSC N1(C(c2c(CSC)cccc2)=O)CC(C2CN(C(c3c[nH]nc3C(F)F)=O)C2)C1 c1(C(N2CC(O)(C(C)NC(=O)CC(C3(C)CC3)C3CC3)C2)=O)cncc(CO)c1 C1(CNC(C(c2cnccn2)C)=O)CCCC2CN(C(C3(C4CC4)CC3)=O)CC12 CC1CN(C(C2CCOC2)=O)CC(C)N(C(c2ncnn2C2CCOCC2)=O)C1 Cc1cc(N)c(C(N2CCC(CNC(C3(n4cnnn4)CC3)=O)C2)=O)c(F)c1 CC(C)C(F)(CNC(=O)C(C)SC1CC1)C(=O)NOC1CC2CCC1C2 c1(C(N2CCC(CCNC(C(=O)NCC)=O)C2)=O)cnc2onc(C)c2c1 c1(C(C(=O)N2C(CNC(c3c(C)nc[nH]3)=O)CC2)(C)C)c(C)noc1C C(=O)(CC(C(F)F)NC(=O)C(F)=CC1CC1)N1CCC(OC)C1 CCC(C(C)(F)F)NC(=O)CN(C(=O)C=C(C)C1CC1)C Cc1ccc2c(c1)CC(C(N1CCC1CNC(c1cnc3nccn3c1)=O)=O)S2 n1(CC(=O)NC(C(C)NC(CCCC(C)C)=O)C(C)C)c(O)nc2ccccc12 c1(N2C3CC(=O)NCC2CC3)cc2c(O)nc(O)nc2cn1 c1(C(=O)NCC2CN(C(CC(C)(C)O)=O)C3C2C3)sccc1S(N)(=O)=O c1(OC)cnc(F)cc1C(N1CC(NC(=O)CCn2cc(C)cn2)CC(C)C1)=O c1(CC)cc(Cl)ccc1C(=O)NC(CNC(c1cnc(C(C)(C)C)[nH]1)=O)C1CC1 c1(N(CC(=O)NCC2CN(C(=O)CCC(C)(F)F)CC2F)C)ccccc1[N+](=O)[O-] C1(C(=O)NCC(CCC=C)O)CCN(C(C2CS(=O)(=O)C2)=O)C12CC2 n1(-c2noc(C3CC(O)(CCNC(=O)CS)C3)n2)nccc1O.c1(COC)nnnn1C N1(C(C2C(C(F)(F)F)CC(=O)N2)=O)CCC12CN(C(=O)C=CC1CCOCC1)C2 Cc1cn2c(=O)c(C(N3CCSCC3C(=O)NCc3ccncn3)=O)cnc2s1 c1(CC(=O)NC2C(NC(CC(C)n3cccc3)=O)CC2)cnn2c1CCCC2 Cc1cc(COC(=O)CN(C)C(C2CN(c3nnnn3C)C2)=O)cc(Br)c1 N1(C(C(C)n2cccn2)=O)CC2(CCCN(C(C3(CF)CCC3)=O)C2)C1 C1(NC(C=CC)=O)CCSC12CN(Cc1cncc(-c3ccc(C)cc3)c1)C2 Cc1cc(C)c(C(=O)NCC2CCCCN2C(c2cnco2)=O)c(O)c1 N1(C(C)COCCO)C(=O)NC(Cc2ccccc2)C1=O C1(CC(=O)N(C(CNC(Cc2cc(C)sc2C)=O)C)C)Cc2cc(F)ccc2O1 C1(N(C(c2ccsc2)=O)CC)CCCN(C(=O)C(C2CCOCC2)F)C1 N1(C(COCc2n(C)ncc2)=O)CCCC(C)(NC(c2ccc(F)o2)=O)C1 C(=O)(C1CCCn2c(Br)cnc21)NC1C(CNC(C2(C(N)=O)CC2)=O)C1 C(=O)(CCCCC(F)(F)F)NC1CN(C(CS(CC)=O)=O)CC(C)(C)C1 CCCCC(CNC(c1oc(CC)cc1C)=O)NC(C1CC(C)CN1C(C)=O)=O C(=O)(C1=CS(=O)CCC1)N1CCC(CN(C)C(c2nccc3ccsc23)=O)C1 C1(C(N(C2CCS(=O)(=O)C2)CC#C)=O)CC2(CCOC2)C1 C1(C2CC2)(NCc2ccc(C3C(C)C3)o2)CCC1 C=CCCCC(C(=O)NCC1(CO)CC(C)(C)C1)NC(c1coc(C)c1)=O c1(NC(=O)NC2CCC2Nc2ccccc2)cnc(Cl)c(Cl)c1 C1(NC(Cn2nc(C)c(Cl)c2C)=O)Cc2ccccc2N(C(C2CC2F)=O)C1 N1(C(Cc2onc(C)n2)=O)CCOCC(NC(C2CCN2C)=O)C1 CCCC(CCCNC(c1n[nH]c(CC)c1C)=O)NC(=O)C=CC1CCCN1C c1(OC)nc(=N)nc(N2CCC(O)(C(N3CCC(N4CCC(O)CC4)C3)=O)C2)[nH]1 N1(c2snc(SC)n2)CCCC(NC(c2ccc(-n3cccn3)c(C)c2)=O)C1C CC(C)CC(C)C(=O)NCC=CC(=O)NC(C)C(=O)NCCF Cc1ccc(C(CNC(C2(C)CCCS2)=O)NC(C2OCCCO2)=O)cc1 N1(C(C(C)n2cccn2)=O)CCOCC(F)(CNC(c2ccoc2Cl)=O)C1 C1(NC(C2C(C)(C)CO2)=O)CCCC2CN(C(=O)C(C)(O)C3CCC3)CC12 c1(C(N(CC(CC)NC(c2nn(C)nc2Br)=O)C)=O)cccc(C)n1 CS(=O)(=O)CC(=O)N1CCOC(CNC(=O)Cc2c[nH]ccc2=O)C1 N1(C(c2cc(CC)no2)=O)CC2CC1CCN2C(=O)C(C1CCOCC1)O Cc1cccc(CNC(=O)NCc2cc(C)n(-c3cccc(C(F)(F)F)c3)n2)c1 C1(C(=O)NCc2c(C)c[nH]n2)N(C(=O)COCc2scnc2C)CCCC1(C)C N1(CCC)C2(CCC(CCO)C1=O)C(=O)N2.C(CCS)N(C(C)C)C=O Cc1c(C(N2CCCC2CNC(=O)CC2CCCCC2(C)C)=O)cccc1N N1(C(C(CC)n2ccnc2)=O)CC2(CCCC2)C1C(N1CCC=C(F)C1)=O c1(C(=O)NCC2(OCC)CCSCC2)ccc2[nH]nc(C3CCCO3)c2c1 N1(C(=O)OC(C)(C)C)CCC(C)(OC(=O)NCc2nc(C(=O)O)n[nH]2)C1 C1(NC(C(CC=CC)C)=O)CN(C(=O)CS(=O)(=O)NC)C2(CCCCC2)C1 c1(C(=O)NCCC(C)N(C(c2nc(CCC)oc2)=O)C)ncc2c(F)cccn12 C1(C(=O)NC(CNC(=O)CC(=O)NC2CC2)C2CC2)CCC(F)CC1 C1(C)(NC(C(CCOC)NC(=O)CN2CCNC(=O)C2)=O)CCC(=O)NC1=O C(=O)(CC1CCc2cc(Br)ccc21)NCC(CNC(CSCCCC)=O)O Cc1ccc(S(=O)(=O)N2CC(NC(c3cc4cccnc4[nH]3)=O)C(C)C2)c(C)c1 CCC(CC)C(=O)N1CC=CC(NC(c2coc(O)n2)=O)C1 S(=O)(=O)(c1cnc(C(=O)OC)s1)N1CCN(c2ccc(OCC)cc2)CC1 C(C(C)C(=O)NCC(F)CNC(c1cn(C)cn1)=O)OC c1(C(=O)NCC2(C)C(C)CN(C(C3(F)C(C)C3)=O)C2)cccc2[nH]ccc12 N1(C(C=CS(C)=O)=O)CCCC2(C1)CN(C(c1[nH]nnc1-c1ccccc1)=O)C2 C1(C(=O)NCC(C=C)(C)C)(CNC(C2CC(F)(CF)C2)=O)CC12CCC2 N1(C(C(C)NC(CC)=O)=O)CCN(C(c2c(Cl)cnn2CC)=O)C(C(F)F)C1 C(CCC(C)C(=O)N1CCN(C)CC1CNC(c1cnccn1)=O)OC N1(C(CSCC=C)=O)CCC(=O)NC2CN(C(=O)CCc3cc(C)no3)CCC12 C1(C(N(C(C)C(=O)NCC2(C#N)CCC2)C2CC2)=O)CCCC1(C)C c1(OC)ccc(C2(C(=O)NC(COC(C)(C)C)CO)CCOCC2)cc1 N1(C(C2(NC(N)=O)CC2)=O)CC2CCC1CN2C(=O)CN1CC2C=CC1C2 Cc1cc(C#N)ccc1C(=O)NCC#CC(=O)NCc1ncn(C2CC2)n1 C1(CNC(COCCCC)=O)CN(C(=O)C(c2ccc(Cl)nc2)(F)F)CC1(C)C C(=O)(C(C(C)(C)C)OC)N1CCC(OCC(=O)NCC(C(=O)NC)C)C1 CCCC(C)(O)CNC(C1(C)C=CCN1C(c1cc(COC)on1)=O)=O N1(C(c2cnn(C)n2)=O)CCC(C(=O)NCCC2CCC(C)(C)O2)=C(F)C1 C1(C(N2C(COC)CN(C(=O)CN(C)C(N)=O)CC2)=O)CCc2c(nnn2C)C1 C12(CNC(CC(C=C)CC)=O)CCCC(CN(C(c3n[nH]c(C)c3C)=O)C1)C2 N1(C(CCOCCC)=O)CCC(O)(CCNC(c2cccnc2CC)=O)CC1 C(c1ccccc1)=CC(=O)NCCN(C(=O)CC1(C)CC1)CCOC Cc1ncc(C#N)cc1NC(c1cc(CNC(C2(C)CC2C)=O)no1)=O c1(C(=O)NCc2ccc(C(N(C)CCc3nnc(O)o3)=O)s2)ccccc1C#N Cc1nc2ncccc2cc1CC(N1CC(O)CC1CNC(C1CC=CC1)=O)=O C(=O)(C#CC1CCCCO1)NC1C(C)N(C(=O)CCc2ncccn2)CC1 C1(CC(=O)c2ccccc2)C(=O)O1.c1(NC(=O)OC)ccc(OCC(=O)O)nc1 CCCCCCC(CC)C(=O)NC(C)C(C)NC(c1conc1C1CCC1)=O C=C1CCN(C(=O)CC2OCCC2(C)C)C(C(=O)NCc2cncn2C2CC2)C1 c1(-c2scc(C(N(C3CCCN(C(C4CC4(F)F)=O)C3)C)=O)n2)ccc(F)cc1 N1(C(CN(C(CCN(CCC)C)=O)C2CC2)=O)CCC(CO)C(F)(F)C1 C1(CNC(C(C=C=C)C)=O)CCCC2(CN(C(c3snnc3CC)=O)C2)O1 N1(C(c2n(CC)ccc2)=O)CCC(CNC(c2cnc(C)n2C)=O)CC1 CC(O)C(F)(F)C(=O)N1CCC(C(N2CC(C#N)C2)=O)C(C)C1 C(c1cnc(C)nc1O)=CC(=O)NCC(CC(C)C)NC(CC1(C=C)CCC1)=O N1(C(C2CC(SC)C2)=O)CC(CNC(=O)CN2CCC(C)C2)CC1(C)C N(C1COc2cc(Br)ccc21)C(c1ccc(C)c(C(C)(C)C)c1)=O C(C(CNC(=O)Cc1cncc(NCC)c1)S(C)(=O)=O)NC(CC1C(CC)C1)=O CC(C)CC(C(=O)NC1CCC(NC(=O)CC(O)c2ccccc2)CC1)N(C)C S(=O)(=O)(c1cnccc1NC1CC(C)c2ccccc21)N(CC=C)CCC N#Cc1cc(S(=O)(=O)NCc2ccc(C3CC3)cc2)ccc1NCC1COCO1 N1(C(CC(=O)OCC)=O)CCCC2(CCCN2C(=O)C(C)COC)C1 C(c1ccc(Cl)nc1)=CC(=O)NCC1(OC)CN(C(=O)C(=O)C(C)(C)C)C1 C1(C(=O)NCC2CC(C(=O)O)C2)CN(C(C2CC3C=CC2C3)=O)CC12CC2 CC1CC(CO)CN(C(C2CCN(C(=O)COCc3nc[nH]n3)C2)=O)C1 c1(-c2ccc(C(C)=O)cc2)nc2c(s1)CC(C(=O)N(C1CCOC1)CCO)CC2 N1(C(c2cc(C)sc2C)=O)C(C(=O)NCCN2CCC3CC23)C2CC(O)C1C2 N1(C(=O)OC(C)(C)C)CCn2nc(C(N3CC(CO)CC4OCCC34)=O)cc2C1 c1(C(N(CCC(C)NC(C(C=C)O)=O)C)=O)cccc(F)c1 N1(C(c2c(C)nc(O)cc2)=O)CCC2(CCOC2)C(CNC(=O)C(C)(C)F)C1 N1(C(C(=O)N(C(C)COC)CCOC)=O)CCOC2(CCOC2C)C1 Cn1cc2c(CN3CCc4nc(-c5ccc(F)cc5)sc4C3)cccc2n1 C(CCOCCO)(C(=O)N1CCC(F)(CF)C1)NC(c1c(CC)cno1)=O C1(CC=C)(C(=O)NC(C)Cc2nc[nH]n2)CCCN1C(c1nc[nH]n1)=O C(C1=NOC2CN(C(=O)Cc3ccccc3O)CC12)NC(c1cc(CC)no1)=O Cc1ccc(NC(=O)CN(C2CN(C(c3ccncc3Cl)=O)CC2F)C)cc1C n12c3c(cc(cc3)c1=O)CC2.C1(C(N(CC(C)NC(C)=O)C)=O)COCCN1C c1(NCC2CCC(CC)CC2)cccc2c1NCCC2C C=CC1(C(=O)NCCc2cc[nH]n2)CCN(C(c2ccoc2CC)=O)CC1 c1(OC)ccc(C(N2CCC(OC)CC2)C(=O)OCC(=O)N(C)C)c(C)c1 C1(C(=O)NC(CNC(C(C(C)C)OCC)=O)C)Cc2cc(OC)ccc2O1 C(=O)(CCC(F)(F)C(F)F)NC(C)CCNC(=O)CCC1CC1(F)F C(=O)(C(C)(C)CC(C)(C)C)N(CCOCCNC(CC(C)n1cccn1)=O)C N1(C(CCc2n(C)cnn2)=O)CC(CNC(=O)C2=CCC2)C(F)(F)C1 c1(C(=O)NC2(CNC(=O)CC3CC(O)C34CCC4)CC2)cnc2ncccc2c1 c1(OCCOC)ccccc1C(N1CCC(CNC(c2nccnc2N)=O)C1)=O CC(C)(C#N)C(=O)N1CC(N2CCN(C(c3cnc(C4CC4)nc3)=O)CC2)C1 C1(C(N2CCCC(C(=O)NC3CCCCC3(F)F)C2)=O)CCCC2(CC2)C1 C1(OC)CC(CNC(=O)Cc2ccon2)N(C(c2cc(Br)c(C)o2)=O)C1 C=CCC(CC=C)C(=O)NCCC(C(=O)N(C1CCCC1(F)F)C)OC C1(F)(CNC(C(=O)NCCOC)=O)CCCN(C(c2ccccc2C(F)F)=O)C1 N1(C(C2(C#C)CC2)=O)CCC2(CC1)CC2NC(c1cc(C)n(CC(F)(F)F)n1)=O N1(Cc2ccc(O)c(C)c2O)Cc2ccc(NC(c3cc(O)n(C)n3)=O)cc2C1 Cc1cc(C(=O)NC2CC(CC(N3CCNC(=O)CC3)=O)C2)cc2c[nH]nc12 N1(C(CC)=O)CCSCC1CCNC(=O)CC(F)(F)Br C12(C(=O)NC)CCC(COC(C)=O)(CC1)CO2.C12CCN1C2=O c1(C(=O)NCC(CNC(c2cc(C)c(N)cn2)=O)CO)cccc2c1ncn2C N1(C2(C(=O)OCC)CC2C)CCC(C)(C(=O)N(CC)C(c2cn(C)nn2)CC)CC1 C(=O)(CCCCC(=O)N1CC(C2CN(C(=O)C(C)(O)C3CCC3)CCO2)C1)NC CC(C)(C)C(C)(O)C(=O)N1CC(NC(=O)CCNC(=O)C=CCl)CC(F)C1 CCCC(C)(C)CC(=O)NC1(C)CCCN(C(=O)C(C)CC2CCC2)C1 c1(CNC2CCN(C(=O)OC(C)(C)C)CC2C(=O)O)cc2cnccc2[nH]1 N(C(=NCc1cc(Cl)cs1)NCc1ccco1)Cc1cn(CC(F)F)nc1 C(=O)(C1CCCc2n[nH]cc21)NC1CN(C(c2cc(C)c(F)nc2)=O)CC1C Cc1coc(C(C)C)c1C(=O)NCC(C(C)(C)C)NC(=O)CC(C)C1CCCC1 CC1(C)CN(C(C2CC3CC2CO3)=O)CC1NC(=O)Cc1ccnc(O)c1 C(=O)(C1=NOC(C)C1C)N1CCC(N(C(=O)Cc2cn(C3CC3)cn2)CC)C1 C1(C(=O)NCCCCC2CN(C(c3n(C)ccn3)=O)C2)(N(C)C)CCCCC1 Cc1cncc(C)c1C(=O)NC1CCOCC1C(=O)NCc1cnn(C(C)C)c1 C1(F)(CNC(COCC)=O)CCN(C(=O)CN(C)CC)CC1 C1(CC=C)(C(=O)NCCN2CCOCC2=O)CCCN1C(=O)Cc1cnc(C)s1 CC(O)C(CO)NC(=O)CCC1CCN(C(=O)C(N)=O)C1 C=CC(C)(CCOC)C(=O)NCCC1(C(=O)N(C2COC(C)(C)C2)C)CCC1 C1(C(N(C)Cc2cccnc2)=O)CCC2(CN(Cc3ccc(CO)o3)C2)O1 C1(C)(NC(CCCOC(C)C)=O)CCC(NC(=O)CC2(O)CCCCC2)CC1 c1(CC(N2C3CN(C(C4(O)CCC(C)CC4)=O)CC2C3)=O)c[nH]c2cnccc12 C1(C)(OCC(=O)NC2(CCOC)CCC2)CN(C(C2CCCOC2)=O)C1 C1(CNC(c2cc(COC)on2)=O)CC2(CO1)CN(C(=O)CC1(C)CCCC1)C2 Cc1nnc2ccc(NC(=O)C(=O)NCC(C3CCCOC3)(C)O)cn12 C(C)(N=c1[nH]c(=NC(C)c2ccco2)[nH]c2c1COC2)c1ncc(C)o1 C(=O)(CCCC(C)(C)NC(=O)C(n1ccc(C)n1)C)NC(CC)C(=O)N(C)C C(C(N=c1nc[nH]s1)C(C)C(C)C)NC(CCn1c(C)nc(C)n1)=O C12(OC)CCC(C(N3CCN(C(C4(CF)CC4(F)F)=O)CC3)=O)(CC1)C(=O)C2 c1(C(=O)NCc2c(-c3n(C)ncc3)nccc2)ccc(Br)c(C(F)(F)F)c1F c1(C(=O)NC(C2CCN(C(=O)CC#N)C2)C)ccc(Cl)nc1OC(F)F c1(CNC(C(C)COc2ccccc2)=O)nnc2n1CCN(C(=O)CNC=O)C2 Cc1ccc(C(=O)NCC2CN(Cc3cccc(C)c3Cl)CCO2)c(C(C)C)n1 S(=O)(=O)(CC(CC(C)(C)C)OC)N1C(C(=O)OC)C=CC(OC)C1 CC12CC(C(=O)NC3CC4CN(C(=O)CN5CCC(=O)NC5=O)CC34)(CCO1)C2 c1(OC)cc2nn[nH]c2cc1C(=O)NC(C)CNC(c1n[nH]c2c1CCCC2)=O C1(NC(C(C)O)=O)CC2CC(NC(=O)Cc3cc(C4CC4)no3)CC2C1 C1(C(C(=O)N(C)Cc2cn(-c3ccccc3)nn2)F)CCCNCC1 C(CCC(C)C)(C(=O)N(CC(C1CCC1)OC)C)NC(c1ccnc(OC)n1)=O CC(C(=O)N1OC2C=CC1CC2)C1CCN(C(=O)C2=NOC3COCC23)C1 CC1Oc2cc(Br)ccc2C1Nc1cc(NC2CC3(CC3)C2)ncn1 N1(C(c2ccc(C(C)C)cc2)=O)CCCC(O)(CCNC(=O)Cn2cnnn2)C1 C1(OC)(CNC(c2cnccn2)=O)CCN(C(=O)CN2CCC(O)CC2)CC1 c1(C(=O)NC2CCC(F)(CNC(c3ccc(C)o3)=O)C2)c([N+](=O)[O-])cnn1C c1(CCC(=O)NC2(C)CC(NC(C(CC#C)(C)C)=O)C2)c(C)nc(SC)nc1O c1(NC(C2C(C(=O)OC)(C(C)C)C2)=O)c(C#N)cnn1-c1ccccc1Cl C(=O)(CCC(C)C)NCC(=O)NCCCC(C)NC(C1(CC)COC1)=O C1(C(=O)NCC(CC)N(C(=O)CC2COC(=O)C2)C)CCn2nnnc2C1 S(=O)(=O)(C1CCN(C(=O)Nc2cccc(C(C)C)c2C)CC1)NC N1(C(C(C)=C2CCC2)=O)CCOCC1CCNC(=O)C(C)n1ccnn1 C(=O)(C1=COCCO1)NCCC1CCCN(C(CCC=CCC=C)=O)C1 CCC(CC)(CC)C(=O)NCCCC(O)C(=O)NCC(=O)NC1CCC1 Cc1c(-c2nc(C3CCCCC3)nn2C2CCSC2)cnn1-c1cccc(F)c1 C1(NC(CC(COC)(C)C)=O)CN(C(=O)CCc2cc(C)n(C)n2)CCC1(C)C C1(C(C)=O)CCN(C(c2nc(-c3cnccn3)no2)=O)CC1 c1(C(N(C2CC3CNC2C3)C(C)C(C)(C)C)=O)ccc2cncn2c1 C(=O)(N=S(C)(=O)C1CNC2(CCOCC2)C1)C1(OC)CCC1 N1(C(c2cn(C)nn2)=O)C2CCC1CC(CN1CCCC1)C2.C12(CC1)C(=O)NC2 C1(CNC(C2CC(CC)(CC)C2)=O)C(C2CC2)CCN1C(c1nc(Cl)cs1)=O c1(NC(C2CCC(NC(c3c(C)ocn3)=O)C2)=O)ccc(C#N)c2ccccc12 C1(C(=O)NC(C2CCN(C(c3cnccn3)=O)C2)C)CCc2ccnn2C1 C12(CNC(c3ccc(CC)s3)=O)COCCN1C(=O)CN(C(=O)CCS(C)=O)C2 Cc1cc(C)c(C#N)c(NCc2ccc(C(C)CC(=O)O)cc2)n1 C1(CCCNC(C(C=C)O)=O)CCN(C(C2CCN(c3nccn3C)C2)=O)CC1 N1(CCCCCOC)CCC(NC(=O)CC2(C)CC2(Cl)Cl)C(O)C1 CC(C)C(C(=O)N(CC(C)NC(C1(CCO)CC1)=O)C)Oc1ccc(Cl)cc1 c1(N2CCC(NC(C3C(C)CCC3)=O)C(C)(C)C2)ncnc2c1ccn2C N1(C(Cc2ccc(C(N)=O)cc2)=O)CC(NC(C2(F)CCC2)=O)CC12CCC2 c1(C(N(C)CCOCCNC(c2cc(Br)no2)=O)=O)cc2n(c1)CCC2 C1(NC(c2c(CC)scn2)=O)CN(c2cc(C3CC3)nc(Cl)n2)CC(C)(C)C1 C1(C(=O)NCC2C(NC(CC3(OCC)CC3)=O)COC2)CC(=O)NC(C)C1 CC1CC(C(=O)N2CCCC(C(C)(C)C(=O)NC(c3ccncc3)C)C2)=NO1 c1(SCC(=O)NC2CC(C)(NC(c3ncn(CC)c3)=O)C2)ccsc1[N+](=O)[O-] c1(C(=O)Nc2c(C(=O)NC3CC4(CCC4O)C3)cn(C)n2)ccc(C#N)cc1 C1(C2(O)CCN(C)CC2)(C(N2CCC(C)C(NC(C3CC4(CC4)C3)=O)C2)=O)CC1 N1(C(C(=O)NCc2ccnc(Nc3ccccc3)n2)=O)CCC(CO)C(O)C1 CC(COCC(F)(F)F)N=c1[nH]c(N2CCOCC2)nc(=NCCN(C)C)[nH]1 c1(C(=O)NCC2(CNC(C(CC)C(C)O)=O)CC2)ccc2nccnc2c1 C=CCC(F)(F)CNC(C1(CCNC(=O)C(C)=C2CCC2)CCC1)=O CC(F)(F)C(F)C(=O)NC1CCC(CNC(c2ccccc2CC#N)=O)C1 N1(C(C(COC)C)=O)CC2CC(NC(=O)C=CSCc3ccco3)C1C2 C1(CNC(c2cnsn2)=O)CCCC12CCN(C(C1CCC1(F)F)=O)CC2 C(=O)(C(C)(C)C(N)C1CC1)NC1C(c2ccc(OC)cc2)CCCC1 CCC(C)CN=c1[nH]c(N2CC3CC=CCC3C2)nc2c1CC(C)CC2 N1(C(C(C)CNS(=O)(=O)c2ccccc2)=O)CC2CCCC(C1)C2O C(=O)(C(O)CC(N)=O)NC1CCCC(NC(CCC2(C)CC2)=O)C1 N1(C(C(CC)COC)=O)CCN(C(C2(C)CC2(F)F)=O)CC12CCC2 n1(CCC(C)C)cc(C(=O)NC(C)CN(C(=O)CC(C)N(C)C)C)nn1 CC(c1cccnc1)=CC(=O)NCC1CC(C)N(C(=O)C=CC2CC2)C1 C1(N(C(c2c(COC)ccs2)=O)CCF)CCCN(C(=O)CCC=CC(C)C)C1 C1(CC)C(=O)N(C)CCN1C(=O)C(CCC1CCC1)NC(=O)C1=C(C)OCC1 N1(C(C2CC(CC)(CC)C2)=O)CCSCC1C(=O)N(C)CC1(F)CCC1 C1(C(=O)NCC(CN(C(C2CCOC2C)=O)CC)(C)C)CC(=C(F)F)C1 C1(C(=O)OC)CC2(CC(C(=O)OC(C)C(N3CCCCC3)=O)CCO2)C1 C(C(C(=O)NC1CCCC1N(C(=O)CCCCOCC)C)C(C)(C)C)OCC=C CC(C)CC(C(=O)NCc1csc(CNC(=O)CCOCC(F)(F)F)n1)C(N)=O c1(C(N)=O)ccc(C(N2CC3(CC3C(N3CCC3c3ccccc3)=O)C2)=O)cc1 c1(CC(=O)NCC(C)(CO)NC(c2ccon2)=O)coc2cc3c(cc12)CCC3 c1(CNC(CCSCCC)=O)ocnc1C(=O)N(C)CCF N1(C(C(C2CC2)SC)=O)CC(C(=O)NC(C2CCCC2)CO)OC(C)C1 C1(NC(c2ccc(=N)[nH]n2)=O)CCCCCN(C(c2ccnc(O)c2)=O)C1 Brc1ccc(-n2nccc2CN2CCCCC2n2nccn2)cc1 C1(NC(CC(=C)C)=O)CC2CCC1N(C(c1ccc(C(F)(F)F)cn1)=O)C2 N1(C(C2C(=C)C2)=O)CCCC2(NC(c3cc(C)cc(F)c3)=O)CC2C1 c1(OCC=C)cc(OC)ccc1C(N1CC(NC(=O)CC)CC1C)=O c1(COCC)nc(C(=O)NCC2CC2NC(c2ccoc2Br)=O)cs1 C(N=c1[nH]cnc2ccc([N+](=O)[O-])cc12)c1ccc(CNC(COC)=O)cc1 C1(C(CNC(c2cc(CC)[nH]n2)=O)C)CCN(C(c2n[nH]cc2C2CC2)=O)CC1 CCCCCCCC(=O)N1CCC(C)(C)C1C(N1CC(=O)N(C)C(C)C1)=O CC(C(=O)N1CCC1C1CCC1)SC(F)(F)F N1(C(c2ccccc2C)=O)C(CNC(C2(n3cccn3)CC2)=O)CC2CC12.CO C(CNC(C1(C(N)=O)CC1)=O)(C(C)C(C)C)NC(Cc1c(C)noc1C)=O c1(C(=O)NC2CCCC(CNC(C(C=C)(F)F)=O)C2)cc(C)c(Cl)c([N+](=O)[O-])c1 CC(C)(C)CCC(F)C(=O)NCCCOCCNC(C1CCNC1=O)=O CC1CN(C(=O)CN(c2cnccn2)C)CCCN1C(=O)C1=CCCOC1 c1(C(N2CCC(C)C2CNC(=O)CC2(O)CCCOC2)=O)cc2cnccc2o1 c1(CC(N2C(C(C)NC(c3cn(CC)nc3)=O)CCC2)=O)c(C)cc(C)cc1C N1(c2nc(C(=O)OC)c(C)s2)CCC(C)(NC(=O)C(C)C(C)O)CC1 c1(C(C)NC(=O)C(C)(C)NC(=O)C(CO)NC(N)=O)nnc(O)n1C C1(NC(=O)C(F)(F)c2cncs2)CN(C(C2(CC3CC3)CCC2)=O)CC1F N(C1CCCn2ccnc21)C(C1OCCC(NC(CSC)=O)C1)=O C1(C(N2CCCC(N(C(=O)CCOCC3CC3)CC)C2)=O)CC2(C1)CS(=O)(=O)C2 CCC(C)C(C(=O)NCCC(C)F)N(C)C(C1CN(C(C)C)C1)=O CC1(NC(C2CC2Br)=O)CN(C(=O)C(C)(C)c2cnc[nH]2)C1 [N-]=[N+]=NC1CCC(NC(=O)CC2(c3ccccc3)CS(=O)(=O)C2)C1 CCCCN=C(NCc1nncn1C)N1CCC(C(F)(F)F)(C(=O)NC)C1 c1(C(=O)NCC2C(C)CCCN2C(=O)C=C2CCC2)ccc(P(C)(C)=O)cn1 c1(OC)ccnc(C(N2CC(CNC(=O)CC3CCCN(C)C3)C2)=O)c1O C1(NC(CNC(C)=O)=O)CN(C(=O)CCc2ccc(Cl)s2)CCC1C C#Cc1cccc(OCC(=O)NCC(C)(O)CNC(C2CCN(OC)CC2)=O)c1 c1(C(C)=O)cccc(C(N2CC(O)(CN(C(=O)C(F)(F)CO)C)C2)=O)n1 c1(C(C)NC(c2csc(Br)n2)c2nnnn2-c2ccccc2Cl)ccccc1O c1(C(N(C(=O)CN2CCOCC2)Cc2ccco2)=O)ccc2c(c1)CCO2 C(=O)(N=S(C)(=O)C1CC(C(=O)OC)C1)c1cc(OC)cc(C(=O)OC)c1 c1(C(N2CCC(C3CC3)(NC(CCC#C)=O)C2)=O)ccc(F)c2c1OCC2 N1(C(c2c(C)con2)=O)CCCCC(NC(C2CCC(C)O2)=O)CC1 N1(C(Cn2cnc(=N)[nH]2)=O)CCN(C(c2cncc(F)c2Cl)=O)C2CC12 CC(CC(=O)NC1(C(=O)NCCCC(N)=O)CCN(C)C1)C(C)(C)C C1(O)(CNC(CCN(C(C(C)C2CCCC2)=O)C)=O)CCCC1(C)C C1(C(N2CCN(C(CCCC#N)=O)C(CF)C2)=O)CC(c2ccccn2)=NO1 N1(C(C2CC(=O)NCC2)=O)CCC(C(=O)NC(c2ccc(Cl)cc2)CO)C(O)C1 Cc1cc2[nH]c(C(=O)N(CCC(C)NC(C3(C)CC4CC4C3)=O)C)cc2o1 C(=O)(CCC(=O)NCC(C)N(C(=O)C(C1CCCC1)SC)C1CC1)N(CC)CC c1(C(=O)NCC(CNC(c2ccn3nccc3n2)=O)F)ccc2ccncc2n1 Cc1cc(NC(c2conc2CNC(c2cnc(C)s2)=O)=O)cc(Cl)c1 N1(C(C(C)OCCN(C)C)=O)CCN(C(CCc2c[nH]c(=N)s2)=O)CCC1C S(=O)(=O)(c1cccs1)N(CC(=O)NC(CC)CN(C)C(C1(C)CCCN1C)=O)C N1(C(=O)CCNc2ccccc2)CCOC2(CCCN(C(C3CCCO3)=O)C2)C1 CC1(CNC(C2C=CCCN2C(C2CC2Cl)=O)=O)CCC(=O)N1 Cc1ccccc1OCC(=O)NCC1C2CC2CN1C(c1csc(Br)c1)=O c1(CC)ncc(C(=O)NC2CC(C(N3CC(C)(O)C3)=O)C2)s1 C#CCCCCCCN=c1ccc(N(C)CC=C)n[nH]1 Cc1cc(C)c2[nH]c(=NC3CCCCC3NC(C3(O)CCCC3)=O)sc2c1 C1(CNC(CCCCC)=O)CC2(CCN(C(C3COC3)=O)CC2)CO1 CN1CC(C(=O)NC2CN(C(C3C4CCCCCC34)=O)C2)OCCC1=O c1(N2C(CNC(c3cnc(F)c(F)c3)=O)CC(C)(C)C2)ncnc(Cl)c1[N+](=O)[O-] c1(C(=O)NC2(CCCCNC(c3c(C)cco3)=O)CC2)cc(N)cc(F)c1 c1(C(N2C(C(=O)Nc3cc(C)cc(O)c3)CC3CC32)=O)cccc2ncccc12 N1(C(C(C)c2ccsn2)=O)CCC2(CC(NC(c3cnc4cc[nH]c4c3)=O)C2)C1 n1(CC)cc(S(=O)(=O)N2CCC(NC(=O)CCN(C)C(C)=O)C(F)C2)cn1 C1(C)(C(N(CCC(=O)NC(C2CCC2)C)CC2CC2)=O)CCCO1 c1(NC(C)=O)ccc(NC(c2ccc(-c3c[nH]nc3C)cc2)=O)cc1Cl N1(C(C2CCC(=C)CC2)=O)CCCC(O)(CCNC(c2cnn(C)c2CC)=O)C1 C1(NC(Cn2cnc(=N)[nH]2)=O)CCOCC1NC(c1cnc(C2CC2)nc1)=O CC(C)(C)C(Br)C(=O)N1CC2CC1(C(=O)O)C2 C1(CC(=O)NCCN(C(C)C)C(C2CCOC2)=O)C=CS(=O)(=O)C1 C1(CNC(C(CC)C2CCC(=O)N2)=O)COc2ccc(F)cc2C1 c1(C(=O)OC)ccnc(C(=O)NC2(C)CC(NC(=O)Cc3cn(C)nc3C)C2)c1 C1(NC(C=CC(=O)OCC)=O)CC2C1CCN2C(=O)CCC(CC)OC C1(C(=O)NC2C(C)CN(C(=O)C=CCn3cncn3)C2)CCC(=O)N(C2CC2)C1 c1(OC)cc(C=CC(=O)NC(C(C)NC(=O)C(=O)NC(C)C)C(C)C)ccc1F C(CC)(CC(=O)NOC)NCC(CC)CC c1(NC(N2CC(N(OC)C)C2)=O)cccc(S(=O)(=O)C(F)F)c1 C#CCCC(O)C(=O)N1CCCC(CCNC(=O)Cc2csc(COC)n2)CC1 C(=O)(CC(CNC(=O)C(N)Cc1ccccc1[N+](=O)[O-])C(F)(F)F)OC C12(NC(CC=C)=O)CCCC1N(C(c1sc(CC(C)C)nc1C)=O)CC2 c1(C(=O)NC2CC(N(C(C3CC(C)(C(=O)OC)C3)=O)C)C2)[nH]nc([N+](=O)[O-])c1Cl S(=O)(=O)(c1c(C(=O)OC)cccc1Cl)NCCCC(COC)(C)C c1(C(=O)NC(C)CC2CN(C(=O)Cn3nnc(=N)[nH]3)C2)ccnc2c1cnn2C c1(OC)cc(Br)ccc1CSC.C12CCCN(CC1)c1cc(ncn1)C(=O)N2C Cc1cc(Cl)cc(C(N2CC3(CCC(CNC(=O)CCS(C)=O)O3)C2)=O)c1N c1(C(OC(=O)NCC=C)SCC(N2CCCCC2CCC)=O)ccc(C)cc1C c1(OC)ccc(C(c2ccc(NC(c3nccn3C)=O)cc2)=O)cc1Br c1(N(C)CC2N(C(N)=O)CCC2)cncc(C#N)n1.CC(C=O)N C12(NC(c3c(OC)cccc3)=O)CCCC1(F)CN(C(=O)C(C)N(C)C)C2 N1(C(c2cc(C)c(C)o2)=O)CCCC(C)C1CNc1nccnc1F n1(CC)nc(C2CC2)cc1C(N1CC2CC2(CNC(=O)CCS(C)=O)C1)=O N1(C(C(C)OCC=C)=O)CCCC(C)(C)C1CNC(c1ccc(=O)oc1)=O C(=O)(CC1NC(=O)c2ccccc21)NCCCCNC(=O)CC1CCS(=O)(=O)C1 C#CCCCC(C)C(=O)NCC(CO)NC(=O)CCOc1cccc(OC)c1 c1(C(=O)NC2C(SC)CN(C(=O)C(C)C3(O)CCC3)C2)ccn2ccccc12 n1(CC(C(C(=O)OC)C2CC2)=O)cnc2ccccc12.C12CC(C)CN1NC2=O Cc1cccc(C(C)(C)C(=O)N2CCC(CNC(C3CCCN3C(C)C)=O)C2)c1 C1(NC(Cc2cc(C)no2)=O)CN(Cc2ccc(C(C)C)cc2)CC1F S(=O)(=O)(c1ccccc1)C(N1CC(C2CCNCC2)OC(C)C1)C(C)C C1(C)(CNC(C2N(CC)CC2)=O)CCN(C(C2CCC(N(C)C)CC2)=O)CC1 C(=O)(CC(C)(C)CCOC)NC1CC(C(=O)NC(C#C)CC2CCCC2)OCC1 c1(C(C(=O)NCCC#N)N(C)CC2(C#N)CC2)ccc(F)c(Cl)c1F C(=O)(N=c1[nH][nH]c2c1CN(c1ncc(F)cn1)C2)C1(C(C)C)CCC1 c1(OCC#C)ccc(Br)c(CNCc2cnc(CC)s2)c1 C1(C(=O)N(C2CC(=O)N(C)C2)C)(OC)CCN(C(=O)Cc2ccsc2)CC1 c1(CCC(C)C)cc(C(=O)NC(C)CNC(c2cnc(C(C)O)s2)=O)no1 C1(C2CCN(Cc3ccccc3[N+](=O)[O-])CC2)(NC(C(CC)OCC)=O)CC1 N1(C(CCC2C(C)C2)=O)CC2(CCN2C(c2ccc(C3CC3)cn2)=O)C1 C=CCCC(C)C(C(=O)NCc1ccco1)N1CC(N(C)C)C(C(=O)OC)C1 c1(C(N(CC(C)NC(C2CC2CC(C)(C)C)=O)CC)=O)[nH]c2c(C)cccc2c1C C(=O)(C1=C(C)OCC1)NCC1C=CC(NC(C2C(OC)CCCC2)=O)C1 C#Cc1cc(C(=O)NCC2CN(C(C3CSC3)=O)CCO2)ccc1Cl O=C(C1=C2CCCN=C2NN1)N1CCC(N2CCN(C3CC3)CC2)C1 c1(SC)ccnc(O)c1-c1nccn1C1CN(Cc2ccon2)C1 C1(N(c2ccc(O)c(F)c2F)C(Cc2ccc(C)o2)=O)COC2(CCNCC2)C1 c1(N2CC3(CCC(C(=O)Nc4cc(Cl)nc(Cl)c4)O3)C2)ncc2ccccc2n1 C(=O)(C(=O)N=c1cc(C(C)(C)C)o[nH]1)N1C(C)CS(=O)CC1 c1(CC(N2CCC(CC(=O)N(CC)Cc3cccc(F)c3)C2)=O)cccc(Cl)c1 C1(C(CNC(c2c(C)occ2)=O)C)CCN(C(=O)C(C)(C)c2cccs2)CC1 c1(OC)ccc(CCC(=O)NC2C3CN(C(c4c[nH]c(Br)c4)=O)CC23)c(OC)c1 N1(CC)CC(NC(=O)CC2CCN(Cc3cc(C)n(C)n3)C2)CC1=O CC1(CCNC(=O)CCCNC=O)CCN(C(=O)CCC(N)=O)C1 Cn1nnc2cc(C(=O)OC(C)(C)C)ccc12.C12C(C)CCN1C2=O c1(C(N2CCCC(N(C(C3C(CC(C)C)C3)=O)C)CC2)=O)ccccc1[N+](=O)[O-] N1(C(CCCCN(C(=O)CSC(F)(F)F)C)=O)CCCC2CCCC12 N1(C(C(C)CO)=O)CCN(C(C2(C(N)=O)CC2)=O)CC(C)(F)C1 n1(C(C)C)cncc1C(=O)NCC1(O)CN(C(=O)Cn2nccn2)C1 c1(SC)nc(NC(=O)Nc2ccc(C)c(Br)c2)ncc1Br c1(CC)c(C(N2CCCC(C3CCCN3C(=O)Cc3ccco3)C2)=O)csc1C N1(C(C2C(CNC(Cc3ccc(C)nc3)=O)CC2)=O)CCCC(O)CC1 Cc1ccc(CC(=O)N(C2CN(C(=O)C(O)C(F)F)C2)C)cc1C c1(C(=O)NCC2(CNC(CCCOCCC)=O)CC2)ccc(F)c(F)c1 c1(CNC(C2CCN(C(=O)CCCCC3CCSS3)C2)=O)ncc[nH]c1=O Cc1cc(C(=O)NC2CN(C(c3cc(F)ccc3O)=O)CC2C)cc(Br)c1 C12(C(N3CCC(C#N)(F)C3)=O)CC(CCO1)N(C(c1ccc(O)cn1)=O)C2 c1(N2CC(C(C)NC(CC(COC)C)=O)C2)nc(C#N)c(Cl)s1 C1(CNC(CC(C)(C)C)=O)N(C(C2CCCN(S(C)(=O)=O)C2)=O)CCC1(C)C C1(C(=O)NOCc2cnn(C)c2)(NC(CCOC)=O)CC(=O)C1 N1(C(C(CSC)(C)NC(=O)CC2CCC=CCC2)=O)CCC12CCC(C)CC2 C1(CNC(c2c(C)cnn2C)=O)C2CCCC1N(C(C1CCC(C)O1)=O)C2 c1(C(N2CC3C(CNC(C4CCCS(=O)(=O)C4)=O)C3C2)=O)cn2cnnc2cn1 C1(n2cc(CC(CC)(C)O)nn2)CON(C(=O)C2CC(=O)N(C(C)(C)C)C2)C1 CC12CN(C(C3CCCCS3)=O)C(C(=O)NCCOCCO)(C1)C2 N1(C(C(C(=O)OC)C)=O)CCC2(CC1)CN(C(C1CCC1(OC)OC)=O)C2 c1(C(=O)NCC2C(NC(c3csc([N+](=O)[O-])c3)=O)CC2)ccc2snnc2c1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CCC(NC(=O)CSC(C)C)C(CC)C1 C(=O)(CC(C)(C)C(F)F)NCC1CC(COC)CN1C(=O)C1=CC2C=CC1C2 Cc1cc(C(N2CCC(F)(CNC(C3CN(C)C3)=O)C2)=O)c(N)s1 c1(OC)cc(C(=O)NCC(C)(C(C)C)NC(=O)C(F)=C(C)C)cc(OC)c1C c1(NC(N)=O)cccc(C(=O)NC2(CCNC(=O)C(C3(O)CCCC3)F)CC2)c1 c1(OC)cc(C(=O)Nc2ncc(-c3ccc(C(F)F)c(F)c3)s2)c(F)cn1 c1(CC(=O)NC2CN(C(CNC(CC(C)C)=O)=O)C2)ccc(Br)cc1F C1(NC(CCCC)=O)Cc2ccccc2C1NC(=O)CCCn1ccnn1 C(C)(CCC(=O)N1CC(CCO)(NC(=O)CCC(C)SC)C1)OCC C1(C(=O)NN2CC(OCCN(C(COC(C)=O)=O)C3CCC3)C2)CCCN1C=O c1(C(C(N2CC(CNC(=O)Cc3csnn3)OCC2)=O)O)cc(F)c(F)c(F)c1 N1(C(CCN(C(C2CC(C(=O)OC)C2)=O)CCO)=O)CCN(C)C(C(C)C)C1 N1(CCC)C(=O)CCC1C(N1CC2C(N(C(=O)CCCc3ccsc3)C)C2C1)=O c1(C(C(N2CC(C(C)NC(CCCNC(COC)=O)=O)C2)=O)C)ccc(C)cc1 c1(C(=O)NCC(C)NC(c2c(C)nccc2Cl)=O)cccc2c1CCO2 CCCCCC(O)C(C)C(=O)NCC(CNC(c1cc(C)sc1N)=O)CO C(=O)(C1=COCCO1)NC(CCCNC(CC1C(C(=O)OC)CCC1)=O)(C)C C1(NC(C2(N(C)C)CC2)=O)C2CC1N(C(=O)CCCn1ccnn1)C2 C1(C(=O)NC(CC#C)CC#C)CCN(C(=O)C(CC=C)CC=C)O1 N1(C(COC(CC)C)=O)CCN(C(c2sc(C)nc2C)=O)CC(O)C1 c1(C(=O)NC2C(C)C(C)N(C(=O)CC(C)N(C)C)CC2)cc2ccccc2n1C C(=O)(CC(C(F)F)NC(=O)C(F)OC)NC1(CCOC)CCN(C(C)=O)C1 C(=O)(C(C)(C)C(C)(F)F)NC1C=CC(CNC(Cc2cc(C)[nH]n2)=O)C1 c1(C(=O)OC)[nH]c(=NC(C2=CCCCC2)C2CCOCC2)[nH]c2ncnc1-2 CCC#CCN=c1[nH]c(=NC(C)c2nc(C(C)C)n[nH]2)[nH]c2c1CCCC2 N1(C(c2cc(C)no2)=O)CCC2(CO)CN(C(c3ccn4ccsc34)=O)CC2C1 C12(C(N3CCC(C(C)NC(C4CCCSS4)=O)CC3)=O)CC3CC(C(=O)N1)C2C3 C1(C(N2CC(C)=C(C)C2)=O)CC2C=CC1N(C(c1cccc(F)c1C)=O)C2 C1(C(N2CCC(OCCNC(=O)C=C(Cl)Cl)C2)=O)CC2(C1)CC(F)C2 [N-]=[N+]=NC1CCN(C(C2(F)CCCN(C(C3CC4(CCO3)CC4)=O)C2)=O)C1 N1(C(C(c2ccc(C)cc2)(C)C)=O)CCN(C(C2CCC(C)O2)=O)CC(O)C1 N1(C(C(C)CCO)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)Cc1ccco1 C(C(=O)NCCC1(C(N2CCC2(C)C(=O)OC)=O)CCC1)(C(C)C)OCC C(CC(=O)NC1CCC1O)N(CC#C)C(C1CC(SC)C1)=O c1(C(N(C2CCN(C(=O)CNc3ncccn3)C2)CC)=O)c[nH]c(C(N)=O)c1 c1(C(N2C(C)CCC2C(=O)NCC2CN(C)CCO2)=O)cc2c(cc1Br)OCO2 C=C1CC2CCC(C1)N2C(=O)C(CCNC(=O)C(C)(C)C(C)O)OC c1(C(c2nnnn2CCNC(C)=O)NC(CCC(=C)C)C)cc(C)cc(C)c1 N1(C(C=C2CCN(C)CC2)=O)CC(C)(C)OCC1CNC(C1CC1Br)=O CC(C)C(CC(=O)NCC1(NC(C2CN(C(C)C)CCO2)=O)CC1)c1ccon1 c1(COC(C)=O)ncc(-c2ccco2)n1CCC(F)(F)F c1(-n2ncc(C(=O)NCC(C(C)(C)C)NC(C3C(C)(C)C3)=O)n2)cccc(Cl)c1 Cc1cc(C(=O)NC2CC2C(=O)Nc2cccc(Cl)c2Cl)nc2nccn12 c1(C(=O)NCC(O)CNC(C2CCCCS2)=O)cc2nccnc2cc1F c1(CCC(=O)NC2CC(N(C)C(c3ccc(Cl)o3)=O)C2)cnc2n1CCCC2 c1(C(=O)NCCCC(=O)NC2(C(N)=O)CCCC2)cnncc1O c1(C(=O)NCC2(CNC(C3(O)CCC(CC)C3)=O)CC2)nccc(C)c1N CCC(CN(C)C)N=c1nc(N(CC(C)OC(C)(C)C)C)c2c(ncn2CC)[nH]1 N1(C(CC(=O)NCC)=O)C2CCC1C(C)C(NC(C1CCCS(=O)(=O)C1)=O)C2 CC1CN(C(=O)CCC2CCC(=O)NC2)CC1NC(=O)C(=Cc1c[nH]cn1)F C1(CC(N2CC(O)(COC)C2)=O)CC(NC(=O)CCc2cccs2)C1(C)C c1(S(CC(F)CN2CCOC3(CCCCC3)C2)=O)nc2ccc([N+](=O)[O-])cc2s1 CC(C)CC(C(=O)N(CCO)CCO)N(C(=O)CCc1ccn(C)n1)C C1(C(N2CCN(C(C3(CC)COC3)=O)CC23CC3)=O)CC2CC(O)CC(C1)C2 N1(c2nc(C(C)C)nc(N(C)C)c2)CCC2(C=CC2)CC1 N1(C(C2CC(Cl)(Cl)C2)=O)CCCC2CN(C(C3(O)CCCC3)=O)CCCC12 CCCCCN(C(=O)C(C)OC1CCOC1)C(C)C.c1(NC(C)=O)cnn(C)c1 N1(C(C2CC(SC)C2)=O)CC2C(CNC(c3ccc(CS(N)(=O)=O)cc3)=O)C2C1 Cc1ccnc(C(=O)NCCC(O)CNC(=O)Cn2ccccc2=O)n1 C#Cc1cccc(C(N2CCN(C3CN(C(=O)C(C)c4ccsc4)C3)CC2)=O)c1 N1(C(CC2(OC)CN(C(=O)Cc3cccc(Br)c3)C2)=O)CCCC2CCCCC12 Cc1cc(C)cc(C=CC(N2CC3CCC2CN3c2ncnc3[nH]cnc23)=O)c1 C=CCCCCCC(=O)N1CC(N(C(=O)C(C)CCCC)C)C(C)(C)C1 c1(C(=O)NC(C)C(=O)N2CC(n3ccnc3)C2)sccc1CC1CCC1 CCN=c1ccc(C(=O)NCC2CC(F)CN2C(C2(CCF)CC2)=O)c[nH]1 C(CCCCC)N(CC(=O)N(C(C)CNC(=O)CCc1conc1C)OCC)C C(C(C)(O)CNC(=O)CNC(=O)C(F)(F)F)NC(COCCOCC#C)=O C1(C(=O)NCCCC(=C)C)(C(C)C)CCN(C(C2CCOCC2)=O)C1 c1(OC)cccc(C(c2nnnn2CCCF)NC2C=CCCC2CO)c1 C(=O)(CCC(C)CN(C)C)C1(OC(C)C)CCC1.CC1CNC(=O)NCC(=O)NC1 N1(C(C=C2CCC(C)CC2)=O)CC(C(N2CCCC2(CO)CO)=O)C(F)(F)C1 c1(C(=O)NC(Cn2cc(-c3c(C)cncn3)nn2)C)cccc([N+](=O)[O-])c1 c1(C(=O)NC2C(NC(c3cccc(OC(F)F)n3)=O)C2)cccc(F)c1 C1(NC(C(CC)CC)=O)CCN(C(=O)C=Cc2c(C)noc2C)CC1C C1(NC(C2CC(O)(CNC(c3oc(C)c(CO)c3)=O)C2)=O)CC2(CCC2)C1O C1(CCNC(C=C(C)C(F)F)=O)CN(C(c2ccncc2C)=O)CCO1 c1(CC)nc2c(C(=O)NCC3CCC3NC(=O)CC(O)C3CC3)ccnc2[nH]1 O=C1OCc2cc(COC(C3CC4CC3C3CCCC43)=O)ccc21 c1(OC)ccc(C(N2CC(NC(=O)C(O)Cc3ccccn3)C(O)C2)=O)cc1N CC(CC(=O)NNC(=O)c1cc(Br)c[nH]1)NC(=O)OCc1ccccc1 N1(C(C(C2CCOC2)CCNC(=O)C(CN(C)C)N(C)C)=O)CCC(OC)C1.CO N1(C(c2cncc(C)c2)=O)CCC(CNC(C2CCCC(CF)C2)=O)C(O)C1 C1(C(=O)NC2C(CNC(C(CO)NC(=O)OCC)=O)C2)(CC)CCCCO1 c1(CC(=O)NCCN(C(C2CC(C)CC(C)C2)=O)CC)nc([N+](=O)[O-])n[nH]1 C1(C(=O)NC(C(=O)NCC2(COC)CCC2)c2ccco2)CCCN1C=O N1(C(c2cnc(C)[nH]2)=O)CCC(N(C(=O)CC(C)c2ccco2)C)C2(CC2)C1 c1(CC(C)C(N2CCOC(CNC(c3nc(C4CC4)cs3)=O)C2)=O)cccc(F)c1 c1(C(=O)NC2C(NC(C(CC#C)C)=O)CCOC2)ccc(Br)c(O)n1 N1(C(C2(CF)CN(C(C3C(C)CCC3)=O)C2)=O)CC(CO)C1(C)C C(=O)(CCCCC(F)F)N1CC(O)(CNC(C23CCC(OC)C2CC3)=O)C1 N1(C(Cc2c(C)nc[nH]2)=O)CC2CN(C(c3cccc[n+]3[O-])=O)CCC2(CO)C1 N1(C(CCC(C)OC)=O)CCN(C(C2CC2C)=O)CC(C)(F)C1 C1(C(=O)NCCC(CC)(C)C)CC2(CC(NC(C3COCCO3)=O)C2)C1 c1(C(N2CCC(NC(C(F)=CCC)=O)C2)=O)oc(SC)cc1C c1(C(N2CCC(N(C)C(c3ccc(O)c(F)c3)=O)C2)=O)cn2ccc(Cl)cc2n1 N1(C(CCCSC)=O)CC(NC(C2CC(=O)NC2(C)C)=O)CC(C)(C)C1 CCCC(C)(O)CC(=O)NCc1cc(C2CCN(C(c3ccoc3)=O)CC2)no1 N1(C(C(CCSC)O)=O)CC2CCN(C(=O)CCc3ncc(F)cn3)CC(C2)C1 CC1(C)CC2CN(C1)C2=O.C1(NC(=O)COC(F)F)CCCCC1n1cccc1 c1(NC)ccccc1C(N1CCCCC1CCC(=O)N1CCC1CF)=O C(C(C)CC(=O)NCC1CC(CNC(=O)CCN2CCCCC2)C1)OC c1(C(=O)NC(CNC(C(CC)(C)CC)=O)C)c(C)oc2ncn(C)c(=O)c12 c1(C(N2CCC(C)C(NC(C3CCCC3)=O)C2)=O)n[nH]c2c1CCOC2 c1(OC)cc(Cl)c(Cl)cc1C(N1CCC1(C)C(=O)NCCOC(F)(F)F)=O C1(OC)CN(C(c2cc(C(N)=O)c[nH]2)=O)CC1NC(=O)CNC=O C1(NCC2(C)N(C(=O)OC(C)(C)C)CCC2)COCC(C)(C)C1 c1(C(N2C(Cn3cc(-c4cc(=N)[nH]cc4)nn3)CCC2)=O)ccc(Cl)c(F)c1 C(=O)(C(C)CC(C)(C)C)NC(CNC(CC(CC)CC)=O)C(C)C c1(CN(CCCC)C(=O)NC(c2ccncc2)c2ccccn2)ccc(C)cc1 c1(C(C(N2CCCC(NC)C2)=O)(F)F)cccc(F)c1F C12(CN(C)C(=O)OC(C)(C)C)CCOC1CN(C(=O)CCc1ccccc1)C2 CC1(CO)CCN(C(C2CCC(NC(c3c(O)cccc3O)=O)CC2)=O)CC1O c1(C(=O)Nc2scc(-c3ccc(OC)c(F)c3)c2)cccc2oc(=N)[nH]c12 c1(CC)ccc(C(C)C(=O)NC2CC(NC(=O)CCn3cccn3)C2)cc1 c1(CC(=O)NCC(CNC(Cn2c(C)ccn2)=O)(C)C)cccc(C(F)F)c1 N1(C(C2(C(=O)NC)CC2)=O)C(C(=O)N(C2C3CCCC23)C)CC1C N1(C(c2cnns2)=O)CCCC2(CCN(c3nc(Cl)nc4c3SCC4)C2)C1 Cc1cc(NC(=O)CSS)cc(C)c1.C1(C(=O)OCC)CCC(=O)N(c2cnn(C)c2)C1 CCC(C)(C)C(C)NC(=O)COCCNC(C1CN(C(C)=O)C1)=O C1(NC(C2CC(=C)C2)=O)CCOCC1NC(=O)C(C)n1cccn1 C1(C)(C(N(C)CC2N(C(C=CC)=O)CC(F)C2)=O)CCCCNC1=O C1(CNC(c2c(C)ocn2)=O)CCCCN1C(=O)Cn1cccc1 N1(C(C(C)(C)SC)=O)CC2CCCC(CNC(=O)C(C)(C)CNC(C)=O)C2C1 C1(CC#N)CN(C(c2c(O)cccc2Br)=O)CCN1C(c1ccc(Br)cc1F)=O c1(NC(C2C(CC)C2)=O)ccc(NC(=O)CC23CCC(C)(C2)OC3)cc1C C(C)(C)(CCCNC(c1c(Cl)cnn1C)=O)NC(C1C(OCC)C1)=O c1(NC(C(=O)NCC(CC)NC(c2cc(CO)ccn2)=O)=O)ccc(C)c(F)c1 CCCC(CCCNC(=O)CNS(=O)(=O)N(C)C)N=c1cc(C)nc(C(C)C)[nH]1 C1(NC(C2CCC(OC)CC2)=O)CN(C(C2CCN(C)C2)=O)CCC1C(F)(F)F CCCC(C)(O)C(=O)NCC1CCCN(C(c2occc2Br)=O)C1 c1(Cn2cc(CC3N(C(C(C)CF)=O)CCOC3)nn2)ccc(Cl)c(F)c1 c1(OC)ccc(CNC(c2ccc(Sc3ncccn3)o2)C)c([N+](=O)[O-])c1 c1(C(=O)OC)ccc(I)cc1NC(C1CC(O)CN1Cc1ccc(C)nc1)=O N1(C(c2c(CC)ocn2)=O)CC2CCC2(CNC(=O)Cc2nccn2C)C1 n1(C(C)C)ccc(=NCc2nnnn2C(C)(C)C)[nH]1 c1(N2CC(CC(C)C)C(O)CC2)nc(N2CCC(CF)CC2)c2ncccc2n1 N1(C(C(C)OCCOCC)=O)CC2CC1CN(C(c1cncc(COC)c1)=O)C2 C1(CC(=O)NCC(CO)NC(c2n(CCC)ncc2)=O)CC(C)(C)OC1=O C=CC(C)(C)CC(=O)NCCC(C)NC(=O)C(c1ccc(Cl)cc1)(C)O C1(NC(CC2C(C)CN(C(C3CCCCC3O)=O)C2)=O)C2CCCC1CC2 C(C1CCOC1)=CC(=O)NC1CCN(C(=O)CCCC2CCC2)C1 c1(OCC)cc(C(C)NC(=O)Nc2ccc(Br)cc2-c2ccccc2)cc(F)c1 c1(C(=O)NCC=C2CCN(C(CC(C)CN(C)C)=O)CC2)cc(F)ccc1F Cc1oc([N+](=O)[O-])cc1C(=O)NC1CCN(C(=O)CC2CCOC2(C)C)C1C N1(S(CCOCC)(=O)=O)CCC(N2CC3CCCCC3C2)C(C)CC1.N(C1CC1)CC CC1CN(C(c2ccc(Br)c(N)c2)=O)CCN1C(=O)CC1(O)CCC1 S(=O)(=O)(c1ccc(NCCC2CCSCC2)c(Br)c1)N1CC(C)S(=O)C(C)C1 C1(N(C(CC(C)c2ccccc2)=O)CCO)CCCN(C(=O)CC(C)(C)O)C1 C(=O)(CCCC(=O)NC)N(C1CCCN(C(c2cc(C)nc(CO)n2)=O)C1)CC Cc1[nH]c(=N)sc1C(=O)NC(CCN(C)C(c1nc(Cl)sc1Cl)=O)C(C)C c1(OC)cnc(C(N2CCOCC2CCNC(=O)COC2CCOC2)=O)cn1 CC(C)CC(O)C(C)C(=O)N1CC(O)CC1CC(N1CCC12CCCC2)=O c1(C(N2C(CN(C(=O)C(C)C)CC)CCC2)=O)cnn(C2CCCC2)c1C C12(C(N3C(CCC)C=CC3)=O)CCC(N)C1CC2 N1(CCC)CCCC(C(=O)NC2CC(CCNC(c3csc(=N)[nH]3)=O)C2)C1 c1(C(=O)NC(C2(CNC(C(C=C)O)=O)CC2)C)ccc2oc(C)nc2c1 C12(CNC(CC3CN(C(C)=O)C3)=O)CCN(CC1)CC2 CCC(CC(F)F)C(=O)NCC(C1CCCC1)NC(c1ncn(C)c1C)=O n1(CC)nc(C)c(C(=O)NCC2CCN(C(=O)CCCC(=O)OC(C)(C)C)C2)c1Cl c1(C(=O)NCC2N(C(C(C(C)C)SCC)=O)CCC2)cc(O)ccc1N N1(C(C(CC=CC)NC(=O)CCOCC(F)F)=O)CCC2CCN(C)CC12 C1(C)(CC)C=C(C(=O)N2CCCC2CNN(C)C(c2ccc(C(C)=O)nn2)=O)C1 c1(C(=O)NC2C3(CC(NC(C(C4CCC4)OC)=O)C3)C2)cc(C#N)c(F)cc1F S(=O)(=O)(c1ccc(F)c(C(=O)OC)c1F)NC(CS(CC)(=O)=O)CO C1(C)(OC)CN(CC(=O)NC(C2CCN(C(C3(O)CCC3)=O)C2)(C)C)C1 n1(CC(=O)NC2C(C(C)(C)C)CCC2)ccc([N+](=O)[O-])n1 C(=O)(N=c1cc(C)n(C2CC2)[nH]1)C1(NC(CCCC(C=C)C)=O)CCCC1(C)C N1(C(C(C)OCC)=O)CCN(C(c2c[nH]c(=N)c(C)c2)=O)CC1C1CCCC1 [N-]=[N+]=NC1CCCN(C(=O)CCN(CCCO)C(C2C=CCS2)=O)CC1 N1(C(C2(C(F)(F)F)CC2)=O)CC(O)CC1Cn1cc(-c2ccc(Cl)cc2)nn1 c1(NC(=O)OC2CCN(c3n(C)nnn3)C2)ccc(S(C)=O)cc1 C=CCC(C(=O)NC(CN(C)C(c1nccnc1CC)=O)CC)C(C)C Cc1sc(C)c2sc(C(N3CCC(CN(C)C(C4CCNC(=O)C4)=O)C3)=O)cc12 C(=O)(C(C)CCCOC)N1CCC(C2N(C(CCC(=O)NC)=O)CCC2)C1 Cc1nc2c(o1)CCN(C(=O)C(C(C)O)NC(=O)C(C)CO)C2 c1(C(N2CCC(N(C(=O)Cn3cnccc3=O)CC)C2)=O)ccc(C)c(F)c1N C(=O)(C(O)CC(C)C)NC1C2CC(NC(CS(CC)=O)=O)CC21 c1(C2C(C(=O)NC3C(SC)CN(C(=O)C(O)C(C)C)C3)C2)ccc(F)c(Cl)c1 C1(C(=O)NC2(CC=C)CN(C(=O)CCCN3CCCC3)C2)CCOC2(CCC2)C1 CC1(C)CCCN(C(=O)CC2CC(F)(F)C2)C1CNC(C1CN2CCC1CC2)=O c1(COC)nc(NCCC2CCC(OC(F)F)CC2)cc(=NCCOC(C)=O)[nH]1 c1(CC(CC(=O)NC2CC2O)NC(=O)CCc2cn[nH]c2)ccc([N+](=O)[O-])cc1 C1(NC(C(=O)N(CCO)Cc2cnc(CC)s2)=O)CNCCC1C CC(C1=CCN(C)CC1)NC(C1CCCN1C(=O)CCc1ccco1)=O C(C(C(C)C(C)C)NC(c1ccc(C(C)=O)c(O)c1)=O)NC(C1(CC)CC1)=O c1(C(N(CCCNC(=O)CCC2CC2(Cl)Cl)C)=O)sc([N+](=O)[O-])cc1Cl c1(C(=O)NC(CC)CN(C(=O)CCc2nc[nH]n2)C)ccc(Br)c(C)c1 c1(NC(C(C(=O)OC(C)(C)C)(C)F)=O)nccc2[nH]ccc12 c1(C(N2C3CN(C(c4c(OC)ccnc4F)=O)CC32)=O)cnn2cccc(C)c12 c1(C2(NCc3ccn(C)c3)CC2C)ccc(F)cc1 c1(C(N2CC(NC(CC(CC)OC)=O)C2)=O)cc2cccc(Cl)c2cn1 c1(C(N2CCC(NC(C3N(CCCC)CCCC3)=O)C2)=O)ccn2cncc2c1 c1(C(N2CCC(N(C(C3CCC(C)CC3)=O)C)C2)=O)cnc2c(Cl)cccn12 c1(OC)ccc(Cl)cc1C(=O)CN(C)Cc1ccc(C(C#N)C#N)cc1 N1(C(CNC(C(CC)C)=O)=O)CC2CCN(C(=O)C=C3CCN(C)CC3)CC2C1 CC1C(C(=O)NCC(F)F)CCCN1C(=O)C(C)c1cc[nH]n1 C(CCCC(C)NC(c1cncnc1C1CC1)=O)NC(CSCCC)=O N1(C(c2ccc(NC)c(F)c2)=O)CC2=C(C1)CN(C(=O)C1=CCCC1C)C2 C(C)(N=c1[nH]c(=NCCCS(C)=O)c2c(F)cccc2[nH]1)c1nccc(COC)n1 O=CN1CCCC1C(=O)NCCC1CC(NC(=O)C2CC2)C1.C12CN(C1)C2=O c1(CC(=O)NC(CNC(c2ccc(C)c(C)n2)=O)C)cn2c(C)csc2n1 C(=O)(C1=CCCC(C)(C)C1)NC(C)CCCCNC(=O)CSc1ccncc1F N1(C(C(CC)O)=O)CCC(CNC(c2oc(SC)cc2C)=O)(OC)CC1 c1(C(=O)NCC2C(NC(C(c3ccc(F)cc3)C)=O)CC2)csc(=NC2CC2)[nH]1 c1(C(=O)NCC(C)N(C(c2cnnc(O)c2)=O)CC)cnc(O)cc1C C(CNC(=O)COCC(C)(C)C)(C(=O)NC(c1ccc(C)s1)C)OC C(=O)(C(C)CC(C)(C)C)N1CCC2C(C(=O)NCc3c(CC)cccc3)C2C1 C1(O)(CC)CCC(C(=O)NC(C)CNC(=O)CN2CCCCC2)CC1 C#CCCCC(C)C(=O)NC1(CNC(C2(c3cc[nH]n3)CCC2)=O)CCCCC1 CCCC(C(=O)Nc1cccc(N(C(c2cc(Br)no2)C(=O)NC)C)c1)OC Cc1cncc(F)c1C(=O)NC1CC(CNC(=O)C=Cc2cccc(F)c2)C1 N1(C(C)=O)CCCC1(C)C(=O)NCC1(C)CCN(C(C2(O)CC(F)(F)C2)=O)C1 C(=O)(C(CCC)=CCC)N(CC1N(C(C(F)=CCC)=O)CCC1)CC N1(C(C2(NC(=O)COc3cnn(C)c3)C(C)CCC2)=O)CC(C)C12CCOCC2 CC1CCC(NC(=O)CC(C)(C)C#N)CN1C(C1CCCS(=O)(=O)C1)=O C#Cc1cc(NC(C23CC(NCc4ccc(Cl)c(O)c4)(C2)C3)=O)ccc1C Cc1ncc([N+](=O)[O-])cc1C(=O)NC(CNC(c1nccc(Cl)c1O)=O)C1CC1 Nc1cccc(C(=O)NC2CN(C(=O)CCCC3CC3)CC2n2cccn2)c1F N1(C(CN(CC(C)(C)C)C)=O)CC(NC(c2cccnc2O)=O)C(F)C1 C(=O)(C1=CCCSC1)NCCCOCCNC(CCN(C)C(=O)OC(C)(C)C)=O Cc1cccc(F)c1NCC(=O)N=S(C)(C)=O C(=O)(C(C)(C)CC(=O)NCCC1CCCCN1C(=O)CCCCN(C)C)OC N1(C(C(C)OC)=O)CCc2c(c(CNC(C3CCOCC34CCC4)=O)nn2C)C1 N1(C(c2c(C)nc(Br)s2)C(=O)NC2CCOC2)CC(C)OC(C)(C(F)F)C1 c1(C(C(C)C)N(C(C2CC2c2cn[nH]c2)=O)C(C)C)ccccc1 Cc1[nH]nc2cc(C(=O)NC3CCN(C(C4CC5CCCCC45)=O)C3)ccc12 C1(C(=O)NCC(C2CC2)NC(c2[nH]cc(C#N)c2)=O)SC2C=CC1CC2 N1(CCC)CCCC(C(=O)NC2CCCC(NC(=O)Cn3nnnc3C)C2)C1 c1(CCCNC(=O)C(=O)NCC2CC23CC3(F)F)ccc(F)cc1 Cc1ccc(C(N2CC3(CC3)CC2CC(=O)N(C2CC2(C)C)C2CC2)=O)nc1C N1(C(CCCC(C)=O)=O)CCCN(C(=O)Cn2cnc([N+](=O)[O-])c2)CC1C(C)C C1(C(=O)NC(CCCNC(c2c(C)nc(CC3CC3)o2)=O)C)CCCCNC1=O C1(NCc2ncc(C3CCC3)cn2)COC2(CCNC2)C1 c1(C(N2CCC(NC(C(C)(C)C(N)=O)=O)C(O)C2)=O)n[nH]c2ccccc12 N1(C(C2C(C)(CC)C2)=O)CCCC(C2CC2NC(=O)CC2CC2C)C1 C1(CNC(c2c(CC)non2)=O)CC2(CCN(C(=O)CCC(F)F)C2)CO1 CCC(C)(C)CS(=O)(=O)N(C(c1ccc(Br)c(F)c1)C(=O)O)C1CC1 N1(C(COCCOCC#C)=O)CCN(C(=O)CC2C=CCC2)C2COCC12 CC(C)(C(=O)NCC=CCNC(C1(c2cc[nH]n2)CCC1)=O)n1ccnn1 Cc1ncnc(N2CCC(C)(CNC(=O)CCCN3C(=O)CCC3=O)CC2)c1Br Cn1ncc(CCC(=O)NC2CN(C(C3CC3(C)C(F)(F)F)=O)C2)n1 c1(C(=O)NC(C)CNC(c2cc[nH]n2)=O)cccc2ncnc(O)c12 C1(CCC=C)(C(=O)N(CC(=O)OC)CC)CCN(C(=O)CC=CCC)C1 Cc1cc(Cl)c(C(=O)NC2CC(C)(NC(=O)C(C)Cc3cccc(F)c3)C2)cn1 c1(NC(C2N(Cc3ccc(OC)cc3)CC(O)C2)=O)ccnc(F)c1Br C1(NC(=O)CCC2CCOC2)CC(N=c2[nH]nco2)C12CCC2 CN1CCCC1C=CC(=O)NC(c1ccccc1)CNC(C1(C#N)CC=CC1)=O C(C(=O)N1CC(O)CCO1)N(CCC)C(c1cnc(C)[nH]c1=N)=O CC(C)(C)C1=NOC(C(N2CCC(CNC(c3ccc(Cl)c(Cl)c3N)=O)C2)=O)C1 S(=O)(=O)(c1cn(C)c2cc(Br)ccc12)NC(c1ccc(C)c(C)c1)C N1(C(c2cc(C)oc2)=O)CC(NCCNC(=O)CCCN2CCCC2)CC1C Cc1cnn(C)c1CNC(=O)C(Cc1cc[nH]n1)NC(=O)C=C(C1CC1)C1CC1 C12=CC=C(C=C1)C2.C(CCO)(C1CC1)NC(=O)NCC1CC1.c1(S)ccco1 C1(CC)CC(C(N2CCCC2(CNC(=O)C=CC(=O)NC)COC)=O)CC(=O)N1 N1(C(c2c(C)nns2)=O)CC2CCCC2(C(=O)NCC(C)(C)N2CCCC2)C1 N1(C(C(C)Cc2ccncc2)=O)CCN(C(C2CC2C(F)(F)F)=O)CC1 CCC(CC)(CO)C(=O)NCC(C)(C)CN(C(=O)CC1CN2CCC1CC2)C CCC(CC)CCCC(=O)NC1CN(C(=O)CCc2cccs2)CC1CO N1(C(C2CC=CCC2)C(=O)NC2CC2)CCC(O)c2ccccc2C1 c1(C(N2C(C)(CNC(C(CC)(C#N)CC)=O)CCC2)=O)oc(P(C)(C)=O)cc1C N1(C(C2ON=C(CC)C2)=O)CC=C(C(C)(C)C(=O)NC(CC)C(N)=O)C1 c1(CNC(C2(N(C(C(CO)OC)=O)C3CC3)CCC2)=O)ccc(O)nn1 C(=O)(C1=CSCCO1)NCCN(C(=O)C1=NOC(C2(O)COC2)C1)CC Cc1ccc(CC(=O)NCC2(CC(=O)NCc3ncsn3)CC2)cn1 C1(CNC(C=CC(=O)N(C)C)=O)(NC(=O)CC2NC(=O)NC2=O)CCOCC1 C=CC(C)(C)CC(=O)NC1C2CC1N(C(=O)Cc1c(F)cncc1Cl)C2C Cc1ncc(C(=O)N(CC(C)C(=O)N(C)C(C2CCOCC2)C)C)s1 C(=O)(C1CCN(C)c2ccccc21)N(CC(CC)NC(c1cccc(O)n1)=O)C Cc1ccn2cc(C(=O)NC3CC4(C3)CN(C(=O)CC(C)C(F)F)C4)nc2c1 c1(C(N2C3CN(C(c4cccc(C#C)c4)=O)CC2C3)=O)c[nH]c2ccncc12 N1(C(c2cc(C)nc(O)n2)=O)CCN2C(=O)C(NC(=O)CC3CCCC3)CC2C1 C1(CNC(C=C(COC)C)=O)COC(CNC(c2nccn2C)=O)C1 c1(N2CCC(NC(C(C)S(C)(=O)=O)=O)C(C)C2)cc(C#N)ccc1[N+](=O)[O-] C=CC(C)CC(=O)N1CC(NC(=O)Cc2csc(Br)n2)C(CC)C1 C1(N(C(CN(C(COC)=O)C)=O)C)CN(C(=O)C(C2CCCC2)OCO)CC1O C#Cc1cc(C(=O)NCCC2(O)CCCN(C(c3cc(F)c[nH]3)=O)C2)ccc1C c1(C(N2C(C(N3CCC(C(=O)NC)CC3)=O)C(O)CC2)=O)ccc(Cl)c(Cl)c1Cl C1(C(=O)NC2C(C)CN(C(=O)C=C3CCC3)CC2)C2CCCCCCC12 C(=O)(C(O)CC1CCCCC1)NCC1C(CNC(CNC(=O)NC)=O)C1 n1(CCOC)nccc1C(=O)NCCN(C(C)C(=O)NC(C)(C)C)C(C)C O=C(CCCC#Cc1ccccc1)NCCNC(=O)CCCC(F)(F)CO Cc1noc(C(=O)O)c1CN1CCCC2CC12 N1(C(C(C(CC)C)OC)C(=O)NCCSC)CC2CCC(C1)C2(F)F C1(C(=O)NCC2(C)CCN(C(=O)C(O)CC3CCCC3)C2)CCC2(CCC2)CO1 c1(C(C(=O)NCc2nnn(CC(F)(F)F)n2)(F)F)ncccc1Br c1(CC)cccc(NC(N2CC3CC2CN3Cc2noc(C)n2)=O)c1C c1(OC(C)C)cccnc1C(=O)NC1CC(N(C)C(C2(C)COC2)=O)C1 c1(C(=O)NCCN(C(C(CC#C)C)=O)C2CCCC2)c(C)cc(OC)cc1F N1(C(=O)CSC(F)(F)F)CCC(N(C(=O)CCc2ccnn2C)CC)CC1 C1(N(C(CN(C(=O)C(C)C(C)O)CC)=O)C)CN(C(=O)OC(C)(C)C)CCO1 Cc1csc2cc(C(N3C4CCC3CC(CNC(=O)C(C)(C)C3CC3)C4)=O)[nH]c12 N1(C(CCC)=O)CCC2(CCC(CNC(C3CC3CC(C)(C)C)=O)O2)CC1 c1(OC(C(N2C3CC(NC(c4ccc(CC)[nH]4)=O)(C3)C2)=O)C)ccc(Cl)c(C)c1 Cc1cc(NC(=O)C(N2CCC2CNC(c2ccc3c(c2)CC3)=O)=O)ccc1Cl N1(CC2(CNC(=O)OC(C)(C)C)CN(CC(F)(F)F)C2)CCC(O)CC1 C1(S(N)(=O)=O)(C(N(CC(C)NC(c2cnc(C(C)OC)s2)=O)C)=O)CCCC1 C1(C(N2CC(=C(CNC(C(CO)N(C)C)=O)F)C2)=O)COc2ccccc2O1 N1(C(c2ccc(C)c(C)c2)C(=O)NCc2cccc(Br)c2)CC(C)C(O)C(C)C1 c1(CC(=O)NCC(C)N(C)C(C2CCOC2C2CC2)=O)cnc2ccccc2c1 C1(OC)CCN(C(=O)CNC(c2c[nH]nc2-c2cccnc2)=O)C1 Cc1c(Br)ccc(C(N2CC3(CC(NC(c4cn[nH]c4)=O)C3)C2)=O)c1C CC1C(NC(=O)CC2CCCC(=O)C2)CCN1C(c1cncc(C(N)=O)c1)=O Cc1ccc(C(CNC(c2c(C)ccn2C)=O)NC(=O)CS(C)(=O)=O)cc1 C1(NC(C(CC)C)=O)CC2CC(C1)N(C(=O)CCCN1CCCCC1)C2 CC1CCC(C(=O)NCC(C)(CO)NC(=O)Cc2cc(C3CC3)on2)CC1 c1(C(=O)NC(CC)CNC(c2cc(C3(C)COC3)no2)=O)cc(Cl)cn1C Cc1cnc(C(=O)NCCC2CCN(C(=O)CCCC3CCCCC3)C2)nc1 N1(C(C(C(=O)OCC)C2CC2)=O)CCCCC(NC(c2ncc(OC)cn2)=O)C1 C(C(CC(C)C)C(=O)NCCC1COCCO1)NC(c1nc(C)n(C)c1)=O c1(NC2C3(CN(C(CCN(C)CC)=O)C3)CCC2)cc(C(C)=O)c([N+](=O)[O-])cn1 N1(C(=O)CN2CCCCC2)CC2CCCN(C(C3CN4CCCN3CC4)=O)C2C1 C1(NC(c2cc(C)sn2)=O)CCC2CCN(C(C3CCC4CC3C4(C)C)=O)C1C2 N1(C(C2=C(C)OCC2)=O)CC2(CCCC2NC(c2cc(N)c(F)cn2)=O)C1 c1(OCC)cc(C(=O)NCC2(NC(C3CC4CC4C3)=O)CCOC2)oc(=O)c1 CC(C(C)(C)C(=O)N1CC2CC1CC2CF)NC(C1CCCN(C)C1)=O Cc1nc2c(s1)CC(C(=O)NC1CC(CNC(c3csc4cncn34)=O)C1)CC2 n1(CC(=O)NCC2N(C(C=Cc3c(C)ccs3)=O)CCC2)cc([N+](=O)[O-])c(C)n1 c1(CC)ccc(NC(C2C=CCCN2C(=O)CC2CCOC2(C)C)=O)cn1 C1(N)(C(=O)NCC2(CC)CCCCC2)CCC2CCCC12 c1(NC2C(OC)CCCC2)ccc(Br)c(C)n1 N1(C(C(OCC)OCC)=O)CCC(C)(C)C1CNC(C1C=C(C)CS1)=O C(=O)(C(C)C(=O)NCCCOCCNC(=O)CNC(=O)C(F)(F)F)OC Cc1cc(Br)c(N)cc1C(=O)NC1CN(C(=O)Cc2c(C)cccc2C)C1 CC(C)C(CC1CCCCC1)C(=O)NCC1CCCN(C(=O)CCCN(C)C)C1 C1(NC(CSc2nc(C)[nH]n2)=O)CN(C(=O)C(C)C)CC1CC(C)(C)C N(C)(C(=NCCC1(O)CCOCC1)NCC1CCC12CC2)CC1CCOCC1 N1(C(C(CCOC)(C)C)=O)CCCN(C(=O)CCC2(C)CCC(=O)N2)C(CO)C1 C1(C(C)NC(=O)CN(C)C(N)=O)CCN(C(C2CC=CC2)=O)C1 CC(C)(C)CC(O)C(=O)N1CC(O)(C2(CNC(C3(C(F)F)CCCC3)=O)CC2)C1 Cc1cncc2cc(C(N3CCC(C(CO)NC(=O)CCC(N)=O)CC3)=O)sc12 c1(C(N2C(C)(CNC(=O)C(O)C3CC3)CCC2)=O)nc(Br)n2ccccc12 C(=O)(C1CCCc2n[nH]cc21)N(C)CC1CCCN1C(c1cc(=N)[nH]n1C)=O c1(C(=O)NC(C(C)NC(c2c(Cl)cc(C)s2)=O)CO)ccn2c1CCCC2 N1(C(C(CC)(C)CO)=O)CCCC(C2(NC(C3CCCCC3)=O)CC2)C1 C#CCCCCNC(=O)COCCNC(c1ccc(C)o1)=O CCCCCCC(F)C(=O)N1CC2CC1CN2C(=O)C(=C1CCCCC1)F C1(NC(=O)C(c2cccc(C3CC3)c2)O)CCCN(C(=O)Cc2cc[nH]n2)C1 c1(C(=O)NC(C2CC(NC(c3c(C)oc(C)c3C)=O)C2)C)cnc2[nH]cnc2c1 c1(C(N2CC(C)C(CNC(c3ccoc3)=O)C2)=O)sccc1S(=O)(=O)C(F)F N1(C(C2C=CCN(C(c3c(C)cnnc3)=O)C2)=O)CC(F)(F)CCC1C c1(CC(N2CC(C)(NC(C(n3cc(Cl)cn3)C)=O)C2)=O)ccc(CN(C)C)cc1 c1(OC)ncc(F)cc1C(=O)NC1CC(NC(c2cc(F)ccc2O)=O)CC1O C1(NC(c2c(OC)n(C)nc2)=O)CN(C(=O)C(C)(C)C2CC2)CC1(C)C Cc1nnc2ccc(C(N3CCC(CF)(NC(=O)Cn4ncnn4)C3)=O)cn12 c1(C(N2CC(NC(CC3CC(SC)C3)=O)(CO)C2)=O)csc2nccn12 N1(C(COCC#C)=O)CCC(C(O)C(F)F)CC1 c1(OC)ncnc(N(C2CCCN(C(=O)C3=CCSC3)C2)C)c1OC C=C(C)CC(C(=O)NCCOC)NC(=O)CN1C(=O)CCCC1=O N1(C(C2OCCC(C)C2)=O)CC(C2CCN(C(=O)Cc3cccc(O)c3)CC2)C1 C1(NC(C(C)NC(CC)=O)=O)CCCC(NC(=O)CNC(=O)CC(C)C)C1 c1(C(=O)NC(c2cnc(C)s2)C)c(CNC(=O)CNC(=O)C(C)(C)C)cnn1C c1(OC)cccn2ncc(C(N3C4CCC3CN(C(C3CCCO3)=O)C4)=O)c12 c1(C(=O)NCC2(O)CN(C(CC=CC)=O)C2)ccc(-c2nn[nH]n2)cc1 c1(C(=O)NCCC(C)N(C(CCCOCCC)=O)C)ccc(C(C)C)c(C)c1 N1(c2ccc(S(=O)(=O)NCC#CC)cn2)Cc2ccccc2OC2(CCOC2)C1 O=S(=O)(c1cc(F)c(F)c(F)c1)NCC1CN(Cc2cnccc2Cl)CCO1 C1(NC(CCc2onc(CN)n2)=O)COc2ccc(F)cc2C1 C1(C(C)C)CCC(C(=O)NC(C)Cc2cccnc2)N1C(c1cnc[nH]c1=N)=O c1(CC)cccc(N2CCC(NC3(C(=O)OC)CC3C(F)(F)F)CC2)c1 CC(CC(=O)N1CCCN(C(c2ccc(F)c(C3(C)CC3)c2)=O)CC1)C(F)(F)F c1(C(=O)NCCCC2(NC(C(CC)O)=O)CC2)cc(C)cc2c1OCC2 c1(C(=O)NCCCC(C)NC(C(CC(C)C)OC)=O)cc2c(cc1F)NCCC2 n1(CCC)ccc(C(=O)NC(C(=O)N2CC(OC(C)=O)C2)c2cccs2)n1 C1(CNC(C(=O)NC(C)C)=O)CN(C(=O)C(=O)CCc2ccccc2)CCCO1 c1(C(=O)NC2CC(F)(CNC(C3(C)CC3F)=O)C2)cc(N)c(F)cn1 C(CC(=O)N1CC2CC2(CNC(=O)CC(C)=C(C)C)C1)(C1=CCCC1)OCC N1(C(C2C(CC)C2)=O)CC(NC(=O)Cc2ccc(O)nc2)C(N=[N+]=[N-])C1 Cc1cc(C(=O)N(C2CCN(C(=O)C=CCOCC(F)(F)F)C2)CC)ccc1Cl C1(NC(CCNC(C)=O)=O)C2CC3CN(C(=O)Cc4c[nH]nc4C)C1C3C2 Cc1sc(C)c(C(N2CCC(C)(NC(=O)C=Cc3cccnc3)CC2)=O)c1C c1(C(=O)NC2CCN(C(C(CC)C(=O)OC)=O)C2)cc2cc(F)cc(F)c2[nH]1 CN1CCC(C(=O)NC2CC23CC(NC(=O)CC(O)CC2CC2)C3)CC1 CCC(C)CCC(O)CC(=O)N1CC(F)(CNC(=O)CC2CCC=CCC2)C1 N1(C(c2cnn[nH]2)=O)CCOC2(CCC(N=c3ncc4ccccc4[nH]3)CC2)C1 c1(CCC(=O)NCC2CC(NC(CCC)=O)C(O)C2)nc2ccccc2[nH]1 C(=O)(CCCCCNC(=O)C(C)(C)O)NCCN1CCN(C)CC1 c1(N2CC(C)=C(C)CC2)[nH]c(=NCCN2C(=O)CCC2=O)nc2sccc12 Cc1cc(C(C)(C)C(=O)N2CC(NC(c3cnc(C4(C)OCCO4)s3)=O)C2)cs1 C1(n2cc(-c3cnc(OC)s3)nn2)CN(C(C2CC2(C)C(F)F)=O)CC1O Cc1ncc(OCC(N2CC(NC(=O)C(N3CCC(C)C3)=O)C(F)C2)=O)c(C)n1 c1(C(=O)NC2CC(CNC(=O)Cc3cncnc3)C2)cccc2sncc12 N1(C(c2c(C)cn(C(C)C)c2)=O)CC(NC(c2cnco2)=O)CC(C)C1 c1(C(=O)OC)ccc(C)nc1N1CCOC(CNC(C2(C)CCCOC2)=O)C1 CC1CN(C(=O)C(=O)Nc2ncc(-c3ccccc3)s2)CC(C)(C)O1 C=CCC(CC(=O)NC(C)(CC)C(F)(F)F)NC(c1csc(=N)[nH]1)=O C1(C(=O)NCCN(C(C2(C=C)CC2)=O)CC)CC2(C1)C(C(=O)OC)C2(F)F N1(C(c2cn(CC(=O)OC)nn2)=O)CCC(N(C(=O)C(COC)N(C)C)C)CC1 c1(NCC2C(NC(c3nc(OC)cc(OC)n3)=O)CCC2)ncc(C)cc1[N+](=O)[O-] c1(C(=O)NCC2CC(NC(C(CC)n3ccnc3)=O)C2)ccc(Cl)c(C)c1N C1(CC(C2CCN(C(=O)Nc3nc(C)on3)CC2)=O)CCC2C(CC1)C2(F)F C1(COC)(NC(=O)C(F)(F)c2cnccn2)CN(C(=O)CC2CCCCO2)C1 CCCCC1C(=O)N2CC(C3(CC3)OCCSCC(=O)N1)C2.N1(C(N)=O)CCCC1 C1(C(N2CCCN(C(c3c(C)cccn3)=O)C(C)C2)=O)CCCN(S(N)(=O)=O)C1 c1(CCc2scc(C)n2)nc(Cn2cccn2)nn1-c1ccnc(Br)c1 N1(C(C2(C#C)CN(C(=O)C(C)OCCN(C)C)C2)=O)CCCC(O)(CO)C1 N1(C(C2C(CNC(C3(COC)COC3)=O)C2(C)C)=O)Cc2cccnc2C1 Cc1ccccc1OCCC(=O)N(C)CC1CCCN1C(C1CCSC1)=O c1(C(=O)OC)c(NC2CCCCC2C)ccc(F)c1Cl c1(CC(=O)NC(CNC(c2c(C)[nH]nc2Cl)=O)C(C)(C)C)cc(Cl)cc(Cl)c1 c1(OCC)ccccc1C1CCN(Cc2nccn2C)CC1 c1(OCCN(CCCc2ccn(C)n2)CC)c(C)cccc1C C1(C)(CC)C=C(C(=O)N(C2(CC(=O)NCCC#CC(C)(C)C)CC2)C)C1 N1(CCc2cccc(C)c2)CC2CCC(NC(=O)COC3CCCC3)CC2C1 C1(NC(C(=O)NC(C2CCCOC2)C)=O)CCC2(C1)CC2(F)F C=CC(C)(O)CCCC(C)C(=O)NCC1(NC(C2(CN(C)C)CC2)=O)CCCC1 Cc1ccc2c(c1)C(N(C(c1ccn3ccc(O)nc13)=O)C1CC1)CCCO2 N1(C(c2c(C)ccc(O)c2)=O)CCC2CN(C(c3ccc(Br)cc3Br)=O)CC12 c1(C(=O)NC23CC(CNC(C(C(CC)CC)C)=O)(C2)C3)cc2c(nn1)CCOC2 c1(C(C(=O)OC)N(C)C(=O)N(C)C(C)C)ccc(OC)c(Cl)c1 N1(C(CCCCC#C)=O)CCC2(CCN(C(=O)C=CC=C(Cl)Cl)C2)C1 C1(NC(C2(C)CCOC2)=O)CCOCC1NC(c1ccnn1CC(F)(F)F)=O O=S(=O)(c1ccc(Cl)cc1Cl)N1CC2CC(CN(Cc3cccs3)C2)C1 C1(CC(N2CC(CC(C)NC(c3ncoc3Br)=O)C2)=O)CCCCC1 C1(NC(C(CC=C)CC)=O)CN(C(C2(NC(N)=O)CC2)=O)C2(CCOCC2)C1 C1(NC(c2ccc(C(C)=O)cc2)=O)(CO)CCCN(C(c2sncc2C)=O)C1 C=CCC(C)(CC)C(=O)NCC1C(C(=O)NCc2ccc(C)c(O)c2)C1(C)C C1(CNC(c2c(NC)c(F)ccc2)=O)CN(C(=O)C(C)(O)C2CC2)CCC1(C)C c1(C(=O)NCC(CCO)OC)ccc(F)c2occc12 c1(CC(=O)N(C2CCN(C(C(C)(C)SC)=O)C2)C)oc2ccccc2c1C C1(CNC(c2nc(C)oc2)=O)CC2(CCN(C(=O)CCC=CBr)C2)CO1 N1(C(CCC(C)(C)C)=O)CC2CC(C(N3CC(O)CC3(C)CO)=O)C(C2)C1 N1(C(C23CC(C)(C2)C3)=O)CCCC(N(C(=O)CSc2ccccc2O)CCF)C1 c1(C(=O)NC(C2CCN(C(c3cnn(C)n3)=O)C2)C)c(F)ccc(Cl)c1N C(=O)(CC(C)(C)CC)N(CCCC(=O)NCCCCOCC)C C(=O)(C1=CCCN(C(=O)CC2CCC(C#N)C2)C1)NCCN(C)CC C1(N(C(C(=O)NC(CN(C)C)CCO)=O)C)COC(C)(C)C1 c1(COC)nc(C(=O)NCC(C(C)C)NC(c2conc2C2CCC2)=O)co1 n1(CC(c2ccccc2Cl)O)cnc2c(N3CCC=CCC3)ncnc12 C1(C(N2CCC(OC3CN(C(c4cn[nH]c4)=O)C3)CC2)=O)CC2CCC1O2 Cc1nc(CO)ncc1C(N1CC=CC1CNC(=O)CC(C)n1cccn1)=O N1(C(C)=O)CC(O)CC1C(=O)N(C)CCNC(=O)C=Cc1ccn(C)c1 N1(C(CCN(C(C(c2ccn(C)n2)C)=O)C2CC2)=O)CCC(C2CCCC2)C1 N1(C(CC2CC(=O)OC2)=O)CC2(CNC(C3CCS(=O)(=O)C3)=O)CCC1CC2 C#CCCCC(C)(N)C(=O)NC(CN1CCC1)CC CCCC(C(F)(F)F)NC(C1(CCNC(=O)CN2CC(C)(C)C2)CC1)=O CS(=O)(=NC(=O)C1CC(c2ccccc2)O1)c1ccccc1Cl C1(C(=O)NCc2cn(CC(C)NC(C3(F)C(C)C3)=O)nn2)CC(=O)N(C2CC2)C1 N1(c2onc(C3N(C)CCC3)n2)CCN(C(=O)NCCC2CC3(CCC3)C2)CC1 c1(C(N2C(C)(CNC(C34CCN(CC3)C4)=O)CCC2)=O)ccc(O)nc1Cl c1(-c2cc(OCC)cc(F)c2)cc(C(=O)NCCCS(N)(=O)=O)c2[nH]ccc2c1 c1(NC(C)=O)ccc(C(=O)NC2CN(C(=O)COCCO)CCC2C)cc1F c1(OC)ccc(C(=O)N(C)CC2CCCN2C(c2nn(C)cc2N)=O)cc1O Cc1cc([N+](=O)[O-])cc(C(=O)N(c2nccc(-c3c(F)cccc3F)n2)C)c1Cl Cc1ccc2c(c1)c(CNC(=O)C1=CCCN(CC(=O)NC3CC34CC4)C1)cn2C N1(C(c2ccc(C)nn2)=O)CC2(CC2)CC1C(=O)NCC1CCSCC1 C1(NC(c2cn(C3CCC3)nn2)=O)CC(=O)N(C2CN(Cc3scnc3Cl)C2)C1 c1(CNC(C(=O)OC(CC)C)C(C)C)cc(Cl)cc(I)c1 c1(C(=O)NC(C)(C)CNC(=O)Cc2cccc(Br)c2)ccc(N)c(Cl)n1 c1(NC)cnccc1C(=O)NC1(CNC(c2ncsc2C2CC2)=O)CC1 n1(CC)cc(CC(=O)N(CCC(C)NC(=O)C(c2ccnn2C)C)C)cn1 N1(C(CC2C(C)C(=O)CC2)=O)CCC2CCC(NC(=O)C=CC3CCOC3)C1C2 C=CCCC(C(=O)NCc1nn[nH]n1)NC(=O)CC1CC(=O)NC1=O Cc1cc(NC(=O)COc2ccsn2)ccc1NC(C1CCC(=O)N(C)C1)=O c1(N2CC3C(CN(C)C)(C3)C2)nc(Cl)c2c(ccn2C)n1.C12CCN(CC1)C2=O N1(C(CC=C)=O)CCCC1(C)CCC(=O)NCCCC1CCCCO1 Cc1ccc(Cl)cc1OCC(=O)NCC(C)(C)NC(=O)CC1CCNC1=O CN1CCC(C(=O)Nc2ccc(O)cc2)(NC(=O)CC2CC3CCC2C3)C1 c1(C(=O)NCC2C(CNC(C3C(C)C3)=O)C2)cnn(C2CCC2)n1 C(c1ccc(F)c(F)c1)=CC(=O)NC(C1(O)CN(C(c2cnn[nH]2)=O)C1)C c1(C(C)C)ccccc1NC(C1CCCC1NCc1ncccc1Cl)=O CC(CC(C)(C)C)C(=O)NCC1(C(C)(C)O)CN(C(=O)CCCNC(=O)C2CC2)C1 Cc1ccc(SCCC(=O)NC2(C)CC(NC(=O)CCCN(C)C)C2)cc1C c1(CCCC(=O)NC2(CC=C)CN(C(=O)C(C)OCC)C2)ccc(F)cc1 N1(C(c2c(CC)n(C)nc2)=O)CC(NC(=O)CC(=O)OC)CC12CCCCC2 Cc1c(C(=O)N(CCCNC(=O)CCCC(C)(C)C)CCO)ccc2c1CCC2 C1(C(=O)NCCOCCNC(=O)CC2CCC3CC23)CC(=O)N(O)C1 N1(C(N(c2c(C)cccc2)C)=O)CCCN(C2COC2)CC1 c1(OCC)ccc(F)c(C(=O)NCC(O)CNC(C2(C)CCCC2)=O)c1N c1(C(C)SCC(=O)NCC23CC(CN2C(=O)C=CCO)C3)nc2ccccc2[nH]1 C#CCC(CC(F)F)NC(=O)C=CC(C)(C)SC.C1(=O)CCN1 C(C)(C(=O)N(CCCC(=O)NC)C)(N(C(CC1C(CC)C1)=O)C)C1CC1 CCC(CC)(CCC(=O)NC1(CNC(c2c[nH]c(=NC)s2)=O)CC1)[N+](=O)[O-] Cc1nn(C)cc1CC(N1CCN(C2CCCN(C(=O)C(C)C(C)C)C2)CC1)=O c1(NCC)ncc(C(=O)NCC(C)N(C(C2(F)CCC2)=O)CC)cc1Cl c1(CC(=O)OCC2CC(C)CC(C)C2)cccc2cn[nH]c12 c1(NC(=O)OCCOCCC)ccc(-c2cc(CO)ccc2C)c(F)c1 CC1CN2CC1N=C1C3=C(CBr)NC2=C1CCC(C)C3.C1(C)CCOCC1 N=c1c(C(N2CCCCC2CCNC(C2(F)CCCC2)=O)=O)c[nH]cc1Br C12(CNC(=O)CSc3ccccc3)CC(CO1)N(C(C1(Br)CC1)=O)C2 N1(C(c2nnn(C)n2)=O)CC2(C)CN(C(c3ccc(=N)[nH]c3)=O)CC2(C)C1 c1(NC(=O)NCC=C(CCC=C(C)C)C)c(C)[nH]c2ccc(F)cc12 C(CC(C(=O)N(CC(=O)OC)C)OC)NC(C(C)OCC=C)=O CC1CN(C(c2ccc(C(F)F)nc2)=O)CCCN1C(=O)CCCN=[N+]=[N-] N1(C(C2(OC)CCN(C(c3c(OC)cncc3)=O)C2)=O)CC(C)(C)OCC1C N1(C(c2cccc(OC)n2)=O)CCC2CCCN(C(=O)CCCS(N)(=O)=O)C2C1 c1(C(C(=O)NCC(c2cccc(Cl)c2)NC(CC=C(C)C)=O)O)cccc(F)c1 c1(N(C(=O)C(N2CCC(CC3CC3)C2)=O)C)cnc(Cl)c(Cl)c1 C1(NC(C2CCN2C(=O)C(F)C2CCCC2)=O)CN(C2CC2)C1 c1(-c2cn(C3CN(C(C(C)Cc4ccccc4)=O)C3)nn2)ccc(Br)cc1O C(=O)(C1=CCC(F)(F)CC1)NC1C(CC)N(C(c2cc(C)cc(O)n2)=O)CC1 c1(C2CCN(C(C3CCCN(C(CC)C)C3)=O)C2)cc(CN(C)C)cc(OC)c1 Cc1nn(C)c(Cl)c1CC(=O)NC1CCC(NC(c2[nH]ncc2C#N)=O)CC1 N1(C(c2cc(C)nnc2O)=O)CC2CCC1CN2C(C1CC(=O)N(C)C(=O)N1)=O c1(C(=O)NCCOC2CCN(C(C(CC)CC)=O)CC2)ccc(S(C)(=O)=O)cc1 C1(OC)CCC2(C(=O)N(CC(=O)NCCS(C)(=N)=O)C)CC12 Cn1ccc(C=CC(=O)NC2COCC2n2cc(CC3CCCOC3)nn2)c1 Cc1ccc(Cl)c(OCC(=O)NC2(CO)CN(C(c3cccc(F)c3C)=O)C2)c1 c1(OC)cc(C)c(C(=O)NC2CN(C(C3CCCC(C)(C)O3)=O)C2)cc1Br C12(NC(CCOCCOC)=O)CCOCC1CN(C(=O)C(C)SC(C)C)C2 Cc1c[nH]cc(C(=O)NC2COCC2NC(c2ccc(Cl)c(F)c2)=O)c1=O c1(N(CCOC)C)ccnc(NC(C2CCN(C(=O)C(O)CC3CCCC3)C2)=O)c1 c1(C(=O)NC(CCCNC(c2c(CC)n[nH]c2)=O)(C)C)cnc2n1CCOC2 c1(C(=O)OC(c2c(Cl)cccc2Cl)C)cc2c(s1)CCCCC2 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C(=O)NCC1C2CCCCC12)C1(C)CC1 N1(C(C(CC)(F)F)=O)CCN(C(=O)CC2CCCNC(=O)C2)C2CCCC12 c1(NC(C)C)ccc(Cl)c(NC(CC2CCN(CCc3nccs3)CC2)=O)c1 C1(C(=O)NCCC(C)(C)F)CCCCN1C(=O)COCCN(C)C C1(NC(c2cc(OC)ns2)=O)CC2CCCC(C1)N2C(C1(F)CCN(C)CC1)=O C1(C(=O)NC2CCN(C(C(C(C)(C)C)NC(C)=O)=O)C2)CCn2nccc2C1 c1(C(=O)NCC=CCNC(C2(C)CCC(C)C2)=O)csc(=NC2CCCCC2)[nH]1 c1(NC(C2CC(NCc3cccc(NS(C)(=O)=O)c3)C2)=O)ccc(C#N)cc1I C(CC(C)C(C)(C)C)ONC(C1C(C)CCN1C(c1ccccc1)=O)=O C(CN(C)C)(C(C)C)NC(CN1C(NC(C=CCN(CC)CC)=O)CC1)=O N1(C(C=C(CC)C)=O)CC2C(CNC(=O)COCc3cccnc3)C2C1 C1(C(=O)NCC2(CNC(c3c(CC)[nH]cc3)=O)CC2(F)F)CC2CCC(C1)N2C Cc1cncc(C(N2CC(F)(CNC(C3CCN(C)C3C)=O)C2)=O)c1 CC1(C)CCC(CC(N2CCC2C(=O)NCCN=S(C)(C)=O)=O)O1 C1(NC(C(CCOC)NC(c2ccc(C)cn2)=O)=O)CC2CC3C(C2)C13 Cc1noc(C(=O)NC(Cc2ccccc2)C(=O)NC(=O)NC2CCC2)c1C CC1(C)CCCCC1C(=O)N(CCC(=O)NCC1CC(C(N)=O)=NO1)CC1CC1 C12(C(N3C(CCNC(C4C(COC)C4)=O)CCC3)=O)CC(C)(C1)OC21CCC1 C(=O)(C1=CCCOCC1)NCCOCCCN(C)C(c1[nH]cc2c1CCCC2)=O C1(CCC)CCCC1CNC(=O)NCCCN(C(=O)CNC(=O)CC)C CCCC(C(=O)N1CCC1CCOC)NC(=O)C(C1CC1)OCC n1(CC(=O)NC2CCC(F)(CNC(c3cc(C)nn3C)=O)C2)cc(F)ccc1=O C(C(CNC(C12CCCC1(C(N)=O)C2)=O)C(F)(F)F)NC(Cn1c(C)ccn1)=O c1(C(=O)NC2CCN(C(Cn3ncn(C)c3=O)=O)CC2)cnn2cccc2c1 c1(CC)ccc(C(=O)NC(CO)CCCNC(=O)C2CC2)cn1 c1(NCCC(C)(C)NC(C(C(CC)(C)C)O)=O)ncc(C)c(S(C)(=O)=O)n1 c1(CC)cnsc1C(=O)NC1(C)CC(NC(C2CC2(C)C(F)F)=O)C1 C1(OC)CN(C(=O)C=CCN(C(=O)Cc2cnn(C)c2)C)C2(CCC2)C1 C1(C(=O)NC(CNC(C2(C)CCCCO2)=O)C(C)C)(COC)CCCCO1 c1(C(N(C2CCN(C(=O)C=Cc3ccoc3)C2)C)=O)cc(OCC(F)F)ccn1 c1(N(C(=O)CNCC2(c3ccccc3)CC2(C)C)C)cnn(-c2ccccc2)c1 c1(C(N(C(C)CNC(C2(C3(O)CCC3)CC2)=O)CC)=O)cccn2nnnc12 Cc1cc(CCC(N2CC(C)(NC(=O)CC3(C)CCOC3)C2)=O)on1 c1(C(N2CC(N(S(CC)(=O)=O)C)C2)=O)cnoc1-c1ccc(Cl)s1 c12ccc(cc1)COC2=O.C1(C(F)(F)F)(NC(=O)OC)CN(C(C(C)CO)=O)C1 N1(C(C2C(C)(C(F)F)C2)=O)CCN(C(c2csc3nnsc23)=O)CC1C(F)F c1(OC(C)C)ccc(C(=O)NCC(C)(O)CNC(C2CCC(CO)O2)=O)cc1 C1(C(N(C)CCn2cccn2)=O)C(C2CC2)CCN1C(=O)C=Cc1ccc[nH]1 c1(C(=O)OC)c(C(c2nnnn2C)NCC(C)COC(F)(F)F)ccn1C N1(C(C=C(C)C)=O)CC2(C=C(C(=O)N3CCC(O)C34CCCC4)CO2)C1 CCCCC(O)C(=O)N(CCCCNC(c1oc(C(F)(F)F)nc1C)=O)C c1(C(=O)NC2CCCN(C(C3OCCN(C)C3=O)=O)C2)cnn2c(=O)cc[nH]c12 CCC(C(=O)N1CC(C(F)(F)F)CC1CNC(c1ccn(C)n1)=O)C(C)C CC1(NC(c2ncncc2Cl)=O)CCC(NC(c2ccc(CO)cc2F)=O)CC1 C1(NC(C=C(C)C(C)C)=O)CC(N=c2ccnc(C(C)C)[nH]2)C12CCC2 C1(NC(C(CC)CC)=O)CN(C(c2cc(C(C)(C)C)n[nH]2)=O)CC(F)(F)C1 c1(SCC(=O)NC(CCCCNC(C(C)OC)=O)C)ccc(F)cc1F C1(C)(C(=O)NC(C2(O)CN(C(C3N(CC)CCOC3)=O)C2)C)CCN(C)C1=O N1(C(COC(CCC)C)=O)CC(F)CC1CN(C(=O)CS(=O)(=O)N(CC)CC)C C1(CNC(C(C=C=C)C)=O)CN(C(c2sccc2Cl)=O)CCC1(F)F c1(OC)cc(NC(=O)C(N2CCC(O)(CC#N)C2)=O)ccc1C CC12CC(NC(c3csc(Cl)c3)=O)(C1)C1(CN(C(C3(O)CCSC3)=O)C1)O2 c1(C(N2CCC(O)CC2)C(=O)NCCCSC)nc(C2CC2)n(C)n1 C(C(O)CCNC(=O)Cc1ccn(CC(F)(F)F)n1)NC(C1(OC)CC1)=O c1(C(=O)NC2C3CN(C(c4c(CC)ccs4)=O)CC32)cccc2c1C(=O)CCN2 c1(C(C(=O)NC(C)CCNC(=O)Cc2nc[nH]n2)N(C)C)ccccc1F C(C(O)CC(=O)N(C)CC1CCN(CC)C1)NC(C1(OCC)CCCC1)=O c1(C(=O)OCC)sc(NC(=O)C(=O)N(C)Cc2cccs2)nc1-c1ccccc1 c1(OC)ncc(F)cc1C(=O)NC1C2CN(C(=O)C(c3ccccc3C)C)CC12 Cc1ncccc1CC(N1CCC(CC(=O)NC(C)(C)CCO)C1)=O N1(C(c2c(C)ccnn2)=O)CC(O)CCC1C(=O)NC1CCOCC1F C12(C)CC(Sc3ccc(F)cc3F)CN1C2.C(=O)(C(F)=C(C)C)OC c1(NC(C2CC(O)CN2C(=O)C=CCBr)=O)ccc(N2CCOCC2)c(Cl)c1 c1(CC(=O)NC2C(C)N(C(C3CCC(F)C3)=O)CCC2)cn2c(n1)CCCC2 N1(C(CC(=O)OC)=O)CC(CNC(=O)C=Cc2ccc(C)o2)CCC1C c1(CCC)cc(C(N2CCCC(C)(NC(C3CCN(C)C3=O)=O)C2)=O)cc(O)n1 c1(C(=O)NC2CC(NC(c3sccc3C(F)F)=O)C2)ncccc1Br C1(C(c2nnnn2C2COC2)(CC(C2CC2)(N)SC)CC)CCC2(CC1)CC2 c1(C(=O)NC2(CC=C)CCNC2)ccc(C(F)(F)F)c(O)c1 C1(COC)(NC(=O)C=Cc2cnn(C)c2C)CCCN(C(=O)COC(F)(F)F)C1 c1(C(=O)NCCC(=O)NCCN(C(=O)CS(=O)CC)CCC)ccc(C)c(C)c1 c1(OC)cncc(C(=O)NCCC2CN(C(C3(F)CC3C)=O)C2)n1 N1(C(CC(C)c2ccccc2)=O)CCCC(CC(=O)NC(C)C(F)(F)F)C1 C1(CNC(=O)COC(CNC(=O)C(=O)NCC(F)(F)F)CO)CCCCO1 c1(N2CC(CNC(COC(CC)(C)C)=O)OCC2)c(C#N)nnc2ccccc12 C(=O)(C1=CSCCO1)N(C1CCN(C(=O)CC2CCC(C)(C)CO2)C1)C Cc1cc(C(=O)NC(C)(C)C(C)NC(=O)CCC2CC(C)C2)nn1C(C)C c1(C(C(=O)NC(C(=O)NCCN(CCOC)C(=O)C2CC2)C)C)cccc(Cl)c1 N1(C(C=CCCC)=O)CCOC(C)C1C(N1CCC(OC2CCC2)C1)=O C1(C(N(C(C)C)CC)=O)CCc2cnn(CNCC(C)(C)OC(=O)NCC)c2C1 n1(CC(=O)N(C(CNC(C2CC2C(F)F)=O)C2CC2)C)cccc([N+](=O)[O-])c1=O N1(C(c2ncc(C)cn2)=O)CCC2(CCCC2NC(C2CCSCC2)=O)C1 Cc1cc(Br)ccc1C(=O)NCCC1(NC(C2CC23CCCC3)=O)CC1 C1(C(=O)NCC2CCC(C)CN2C(c2cc(Cl)sc2Cl)=O)CCn2nnnc2C1 N1(C(COC(CC)(C)C)=O)CCCC(NC(c2ccccc2SCCO)=O)C1C O=C(CC=C(Cl)Cl)N(C1(C(=O)NOCCCCC2CC2)CCC1)C1CC1 N1(C(c2n(CC)ccn2)=O)CCC(CCNC(c2nccc(C)c2N)=O)CC1C C1(CO)CC2(CC(Nc3ncc(Br)s3)C2)C1 Cc1cc2c(C(=O)NC3CCCC3NC(=O)CC3(C)CC(F)(F)C3)cccc2o1 C1(c2cn(Cc3c(C)c[nH]n3)nn2)CCCN(C(C2CCCN2C)=O)C1 c1(C(N2C(C(=O)NCC3(C#N)CC3)C3CCC2C3)=O)cc(Br)cc2[nH]ccc12 c1(OC)nn(CC(=O)NC(=O)Cc2ccc(C)s2)cc1I N1(C(CCN(CCCCC)C)=O)CCOC(CNC(=O)CC2CC2(Cl)Cl)C1 c1(OC)cc(CCNC(C2C3CN(CC(N)=O)CC23)=O)ccn1 N1(C(C2C(C3C(C)C3)C2)=O)CC(C2CCCN(C(c3ncccc3F)=O)C2)C1 C(=O)(CC(C)(C)CN(C)C)N1CC(CC(C)NC(C(CC)C)=O)C1 C1(NC(c2nc(CC)sc2)=O)CN(C(c2cccc(COC(C)C)c2)=O)CC1C C1(NC(C(C(C)C)NC(C)=O)=O)CCN(C(C2CCCCC2O)=O)CC1(C)C c1(C(C)NC2CCOCC2N2CCOCC2)nc2ccccc2s1 N1(C(C2C(OC)C2)=O)CC(CO)C2(CCN(C(=O)C=CSc3nc[nH]n3)CC2)C1 N1(C(c2cnc(OC)s2)=O)C2CCC1CN(C(=O)CC1CCOC1)CC2 CC1(CNC(c2c(F)cccc2Cl)=O)CCCN(C(C2(S(N)(=O)=O)CC2)=O)C1 C1(N(C(c2nc(=N)[nH][nH]2)=O)CC)CCCN(C(=O)Cc2cnn(CC)c2)C1 c1(C(=O)OC)ncc[nH]c1=NCC1CN(C(c2nc(Cl)ccc2F)=O)CCO1 N1(C(C(=O)Nc2ccc(C#C)cc2)=O)c2ccncc2CC1C c1(C(=O)NC(C2CCN(C(c3c(C)ncn3C)=O)C2)C)cc(N)nc(Cl)c1 CCCCC(C)(CO)NC(=O)C=C(C)CNC(=O)Cn1ncccc1=O C(=O)(C(C)C(C)NC(C1(CNC(C23CCC(OC)C2C3)=O)CC=CC1)=O)OC c1(OC)cc(CNC(C(=O)c2ccccc2)C(C)CC)c(OC)cc1Cl C(C(C)(O)CC(=O)NCC1CCCN(C(c2ccc(N(C)C)c(F)c2)=O)C1)OC c1(C(=O)NC2CCC(N(C(CC(CC)C)=O)C)CC2)cn2cccc(F)c2n1 C(CCCC(C)C)(c1n(C(CC)(C)C)nnn1)NC(C1CN(c2ccccn2)C1)=O C#CCC(CC(F)F)C(=O)N1CC(C)CN(C(=O)C(CO)C(F)(F)F)C(C)C1 C1(CC=C)(NC(c2ccc(=O)n(C)n2)=O)CCCN(C(=O)Cn2cnc(=N)[nH]2)C1 C12(CNC(C(CC)(C)C)=O)CC(NC(=O)CSCC(C)C)(C1)C(C)O2 C1(CC)C(C(=O)NC(CC(=O)N(C2CC(C)(C)C2)C)C2CC2)CCN1C N1(C(CC(C)OC)=O)CCCCC(NC(c2cc(F)ccc2Cl)=O)C1 C1(C(=O)NCC(CO)N(C)C)CCC2(CC2)N1C(c1ncc[nH]1)=O c1(C(N2CC(O)(CNC(C3(C)CC=CCC3)=O)C2)=O)ccc2c(c1)NCCC2 c1(NC(C)=O)ccc(C(=O)NCCN(C(C2CCN(C)S2(=O)=O)=O)CC)c(Cl)c1 c1(C(=O)NC2C(n3cc(CC(C)O)nn3)CCC2)ccc2nncn2c1 C(=O)(CC1COC1)NC(C)C.C1(OC)CN(C(=O)C=CC(=O)NCO)CC1OC C1(OC)CC2CC(C(=O)N(CCN(C)C(c3ccccc3Cl)=O)C(C)C)CC12 c1(OC)c(F)cc(F)c(N2CCN(C(c3cc(Br)c[nH]3)=O)CC2)c1[N+](=O)[O-] Cc1ccccc1SCC(=O)NC1CCCC1CNC(=O)CNC=O C1(CC)CCC(C)CN1C(C1(COC)C=CCN1C(=O)C(C#N)CC1CC1)=O C1(NC(COCCCC#C)=O)CCN(C(c2sc(C(C)C)nc2C)=O)CC1(C)C Cc1cn(C(C)(C)C(=O)NCCCNC(=O)CCOC(C)CC(C)C)cn1 N1(C(c2[nH]cc(C)c2C)=O)CCN(C(c2ccc(N(C)C)cc2)=O)C2CC12 CC(C)(CCCNC(c1c(F)cccc1F)=O)C(=O)NC1CCC2CCCC1O2 N1(C(c2ccsc2Cl)=O)CCN(C(C2C3CCCCCCC23)=O)CC(O)C1 N1(C(c2cc(OCC)ncc2)=O)CC2CCCC2(NC(=O)Cc2cnn(C)n2)C1 C1(C)(C(N(CC(=O)N(C)Cc2cc(C)no2)C)=O)CCC(=O)NC1 c1(C(=O)NCC2N(C(C3C(C(=C)C)OCC3)=O)CC2)cc(Br)c2n[nH]cc2c1 OC1(C2CC2)CCCN(N2CCOC(c3ccc(F)c(Cl)c3)C2)C1 c1(C(C(=O)NCC2N(C(CCN(CCCCC)CC)=O)CC2)=O)cc(F)cc(Cl)c1 CCC(C)(Br)C(=O)N1CCOC(CC(C)C)C1 CCCC(C)(CCC)C(=O)N1C2CCC1CN(C(c1occc1Cl)=O)CC2 n1(CC(=O)NCCC2(O)CN(C(CC3CN(C)C3)=O)C2)ncn(C)c1=O c1(C(=O)NCC=C(C(=O)NC(CCOC)CO)C)cnnc(C)c1 c1(CCc2c(C)cccc2)ncnc2c1nnn2CC1CC1 N1(C(c2cncc(C)n2)=O)CCCC2C1CCCN2C(=O)Cc1cnc(C)o1 N1(C(c2n(CCC)ccc2)=O)CCC=CC1C(N1CCCCCC1)=O C12CCCCN1C(=O)CCCNC2.C1(C(C)NC(=O)NC(C)(C)C)CC(F)(F)C1 N1(C(C(CC)=CC)=O)CCC2(CC1)COC(CNC(=O)C(C(C)C)SCC)C2 Cc1cc(C)n2ncc(C(N3CCC4CN(C(=O)C(F)(F)C(C)O)CC34)=O)c2n1 C1(NC(C(C)=C(C)C)=O)CCN(C(=O)CCc2nnc(O)nc2O)CC1F c1(C(=O)NCC(CNC(C2(C(CC)=O)CC2)=O)C)cn2ncccc2n1 c1(NC(c2[nH]c3c(Br)cccc3c2C(O)C(F)F)=O)cc(Cl)cc2ccccc12 c1(C(N(CCC(C)NC(C2(O)CCOC2)=O)C)=O)cncc(C(F)(F)F)c1 c1(OC)cc(N)c(C(=O)NC2(CCNC(c3cncnc3C)=O)CC2)cc1OC N1(C(c2ccc(Cl)cc2Cl)C(=O)NCCC)CC(C(=O)OC)C(C2CC2)C1 N1(C(c2c(C)nc(C)s2)=O)CCC(CNC(=O)CSC(F)(F)F)C(C)C1 c1(OC)ccc(Br)cc1CSC1CCN(C(=O)CSC2CCCC2)C1 C1(OCCNC(C(N2CCOCC2)c2cc(C(=O)OC)sc2)=O)CCN(C)CC1 c1(OC)cc(C(N2CC(C(=O)Nc3cc(F)c(Cl)nc3Cl)C2)=O)cc2n[nH]cc12 C1(CCC#C)CCCN1C(=O)C(CC1CCCC1)NC(c1cc(CCC)[nH]n1)=O Cc1noc2ncc(S(=O)(=O)C(=O)NCC3CCC(NC(=O)OC(C)(C)C)C3)cc12 Cc1cc(=NC(=O)Nc2ccc(-c3csc(=N)[nH]3)cc2)cc[nH]1 C=CCCC(C(=O)NCCNC(C)=O)NC(=O)C(C1CCC1)OCC Nc1ncc(Cl)cc1S(=O)(=O)Nc1ccc(N2CCS(=O)(=O)CC2)cc1 N#CC1CN(Cc2ncc(Cl)nc2Cl)CCN1C(=O)Cc1ccccc1 Cc1cnc(C(=O)NCC2(C)CCCN2C(=O)CN2CCC(C)(C)C2)c(F)c1 C1(CCC=C)(C(N2CCCC2CNC(C)=O)=O)CN(C(=O)C(C)N2CCC2)C1 c1(C(N2CC3CC4C(NC(C=C(C)Cl)=O)C2C3C4)=O)ccc2c(c1)NCCC2=O C(=O)(CCC(=O)c1cccc(F)c1)N(C(CNC(CC1(OCC)CC1)=O)C)C c1(C(N(C2CN(C(=O)Cc3cc[nH]n3)C2)C)=O)cc(F)c(O)c(Br)c1 Cc1ccc2nc(SCC(=O)NCC3CN(C(c4nn[nH]c4Cl)=O)C3)[nH]c2c1 c1(C(N2C(C(N(CCCCC(C)C)C)=O)CC2C)=O)cccc2[nH]ccc12 C1(COC)(NC(=O)C(C)N(C)C)CCCN(C(c2ccc(SC)cc2)=O)C1 C1(NC(C(CCC)NC(=O)Cc2cccnc2F)=O)CCCCCC1CO N1(C(c2cc(C)oc2C)=O)CCN(C(C2CC3C(C2)C3(C)C)=O)CC1C(C)(C)C C1(C(=O)NCC(CC)NC(=O)CCC(=O)N2CCC(O)CC2)C2CCC(F)(F)C12 C12(C(N(C3CCN(C(=O)CC4CCCC4O)CC3)C)=O)CCN(CC1)C2 C1(NC(COc2c(C)cccc2)=O)CCN(C(=O)CCC2CCCO2)CC1C N1(C(C)=O)CS(=O)(=O)CC1C(=O)NC1CC(NC(c2cc(C3CC3)ncn2)=O)C1 N1(C(C(C)(C)NC(C)=O)=O)CCCCCC(NC(c2cnncc2C)=O)C1 C(=O)(CCCCC(F)F)N1C(CNC(C2N(S(C)(=O)=O)CCC2)=O)CCCC1 c1(C(=O)NCC(C)(C2CCC2)NC(CCSC)=O)ccc([N+](=O)[O-])c(C)c1 C1(C(N2CCC(CNC(c3occc3F)=O)C2)=O)CCc2ncsc2C1 CC(C)C(F)C(=O)NC1CCCCC1CNC(c1ncoc1C(C)(C)C)=O c1(C(=O)NC2CC(F)(C(=O)NC3C(C(=O)OC)CCC3)C2)c(C(F)(F)F)cnn1C CCC(CNC(c1coc(C(C)(C)C)n1)=O)(CC)NC(=O)COC1CC=CC1 C(=O)(C(CC(F)F)NC(c1c[nH]cc1C)=O)N(CC#C)CC1CCCO1 Cc1cc(C(=O)NCC(C2CCOC2)NC(=O)CCF)cc(C)c1OC(F)F C1(CNC(C(C2CN(C(c3n(CC)ccn3)=O)C2)OC)=O)OCCC1(C)C O=C(C(F)(F)c1nccs1)NCC(F)C1CCC1 N1(C(c2cncc(C(C)(F)F)c2)C(=O)NC(CC)C)CCCC12CCC2 Cc1nn(C)c2sc(C(=O)NCCC34CN(C(C5CC5C)=O)CC(F)(C3)C4)cc12 N1(C(CCN(C(C(C)OC2CCCC2)=O)C)=O)CC(N(C)C)C(C)(C)C1 N1(C(CC(COC)C)=O)CCN(C(=O)C=Cc2cccnc2)C(CC(C)(C)C)C1 Cc1cc(NC2(CC(=O)O)CCC(C)C2)c(F)cc1[N+](=O)[O-] N1(C(CC=C)=O)CCC2CN(C(=O)Cc3ccc(F)cc3Br)CCC2C1 N1(C(c2ccc(OC)cc2N)=O)CC(C)(C)CCC1CNC(=O)C(O)CN(C)C c1(CS(=O)(=O)N(CC(CN(CC)CC)N)C)cc(C)sc1C C1(C(N(C(CC)CNC(c2cc(C)ccc2N)=O)C)=O)C2Cc3ccccc3C12 n1(CCCSCC)nnnc1C(C)(C1COC1)NCC(CC1CCOCC1)OC C1(O)(CC(=O)NCC(CC)(CC)Nc2cncc(C#N)n2)CCN(C)CC1 C1(C(=O)NCC2C(NC(C3CSCC(=O)N3)=O)CC2)CCc2nc[nH]c2C1 c1(NC(=O)NC(C)(CN2CCOCC2)C2CCC2)ccc2c(c1)OCO2 C(=O)(CC(O)Cc1ccccc1)N(C1CN(C(=O)C=Cc2ccc(C3CC3)s2)C1)C N1(c2nnc(CC)s2)CC(C(=O)NCCSCC(C)=O)CC1=O c1(CCC)cnnc(C(=O)NCC(CNC(=O)Cc2c(C)noc2Cl)CO)c1 c1(C(=O)NCC(CC=C)NC(=O)C(C2CCCCCC2)C)cc[nH]c(=NC)c1 c1(C(F)(F)F)cc2n(n1)CC(OCc1ccc(-c3cccnc3)cn1)CO2 C1(CNC(=O)C2=NOCC2)CN(C(C2CC(OC(F)(F)F)C2)=O)CCCO1 C1(C(N2CC(COC)(NC(=O)C(C)CC3CC3)C2)=O)CCCCC(F)(F)C1 C(C(C)(C)C(=O)NC1CCC(N(C(=O)CCc2nnc(C)n2C)C)C1)OCC C1(NC(c2nc(C)n(C)n2)=O)CCC(C)(NC(=O)CC2CCCO2)CC1 N1(C(C(C)(C)n2cnnn2)=O)CCC2(CCC2(C)C)C1 C#CC1CN(C(=O)C(CCN(C)C)NC(=O)C(C)OCC(C)C)CC1O C#CCCCCCC(=O)NCC(F)CNC(=O)C(n1ccc(C(F)(F)F)n1)C C(=O)(C(C)CCC(C)(C)C)N1C(C(=O)NCC(CCC)C)CCCC1 c1(C(=O)NCCC2(C)CCN(C(C3C=CCC3)=O)C2)cc2cnc(Cl)cc2s1 CN1CCCC1C=CC(=O)NC1CC(NC(C2CCCCC2c2nc[nH]n2)=O)C1 N1(C(C2(CCC)CC2)=O)CCOC2(CCN(C(C3CCCC4CCCN34)=O)C2)C1 C12(NC(C=C3CCC(C)C3)=O)CC1CN(C(c1cc(-n3cccn3)ccn1)=O)C2 N1(C(C(C2CCN(C(=O)CC3OCCC3(C)C)C2)C)=O)CCCC(CN(C)C)C1 O=C(C1=CC2CCCCC12)NCCCCCNC(c1ncc(F)cn1)=O c1(C(N(CC(C)(C)CNC(=O)CC23CCCC2C3)C)=O)cc2ncccc2[nH]1 C(C)(C(C(C)C)NC(c1cnn(C(C)(C)C)c1Cl)=O)NC(COCCCC#C)=O c1(C(N2CCC=C(CNC(c3cc(Cl)ncc3O)=O)C2)=O)cccc2nccn12 C1(C)(C(N2CCN(C(CCCSC)=O)CC2)=O)CCC(C(C)(C)C)CC1 N1(C(c2c(NC)cccc2)=O)C(C(=O)NCC2CC(CF)C2)CC2CCCC12 C1(C(N2C(CCC)COCC2)=O)CCCN(C(C2CC3(C2)CC(C)C3)=O)CC1 c1(C(N(CC(C)C)CC(C)C)=O)cn(CCNC(=O)C(n2cccn2)C)nn1 C1(C(=O)NCC2(CNC(c3ccc(C4COC4)cc3)=O)CC2)COC2COCC12 C1(C(=O)NCC2(CO)CCCN(C(CC(C=C)C)=O)C2)CCn2c(C)nnc2C1 N1(C(c2ccc(C(F)(F)F)c(F)c2)=O)CC2CN(C(C3CC4CC4C3)=O)CC2C1 c1(CC(=O)NCC2CN(C(C3(C(N)=O)CCC3)=O)C2)csc(Cl)c1 c1(OC)nc(C(=O)NCC(C)(C2CC2)NC(=O)CC(=O)N(C)C)co1 n1(CCN(C(=O)C(O)CC2CCOCC2)CC)cc(CC2CCCOC2)nn1 c1(CNC(C)=O)ccc(C(F)(F)F)cc1Cl.C12CCN(CC1)CC(=O)N2 CC1=C(C(=O)N(CC(C)(C)C(=O)NCC(c2ccncc2)C)C)CCC1 c1(-n2c(C(C)NCC(CC3CCCCC3)SC)nnn2)ccc(F)cc1.SC C(O)(CN=C(NCc1ccco1)NCC1(C2CC2)CCCO1)c1n(C)ncc1 N1(C(=O)OC(C)(C)C)CCC(OC(CC(F)C2CC2)=O)C1 N1(CCOC)CC(C(=O)NC2(COC)CN(C(C3CCC(=O)NC3)=O)C2)CC1=O N1(C(C(C)C)=O)CC(NC(=O)CCc2nc(-c3ncccn3)no2)CC(C)C1 C1(C(=O)NC(c2nccs2)CC)C=CCN(C(=O)C(CO)N(C)C)C1 C#CCCC(=O)N1CC(CN(C)C(C2(OCC)CCOC2)=O)C1 c1(C(=O)NC(C)CC2CN(C(C3CCOC3)=O)C2)cccc2c1CCCCC2 C1(CC(=O)NC(COC(C)C)C)CCN(C(C2CCOC2C)=O)C1(C)C c1(C(N2C(CNC(=O)CCCC3CCCO3)CC(F)C2)=O)cnc2n1CCC2 CCCCCC(C)CC(=O)N(C1CCCN(C(c2cnn(C)n2)=O)C1)CCF c1(C(=O)O)ccc(-n2cc(C3CC(NC(=O)CC4CCCO4)C3)nn2)cc1 c1(CNC(C2(CC)CNC(=O)C2)=O)ccc(F)cc1Cl C1(C(=O)NC2CCOC(CO)C2)(NC(CC(=O)NCC(F)(F)F)=O)CC(F)(F)C1 c1(CN2CC(CC(N3CC(F)(F)C(F)(F)C3)=O)OCC2)c(Cl)cc(F)cc1Cl C1(NC(C2C(CC)CCC2)=O)CN(C(=O)CN2C(=O)CNC2=O)CC2CCCC12 [N-]=[N+]=NC1CN(C(=O)CC2CCN2C(=O)CSCC(F)F)CC1O n1(CC(=O)NC2(CF)CCN(c3snc(SC)n3)C2)c(=O)oc2ccccc12 Cn1cnc(CC(O)C(=O)NC(CNC(=O)CCn2cccn2)CO)c1 CC(c1ccsc1)=CC(N1CCOC(CCCNC(c2cc(C)cs2)=O)C1)=O N1(c2ccnc(C(=O)OC)n2)CCC(C2CCCN(C(c3cnoc3C)=O)C2)C1 N1(Cc2ccc(C(=O)OC)[nH]2)CCCC(C(N2CCC(NC(=O)CC)C2)=O)C1 N1(C(C2CC(C)(O)C2)=O)CCCCCCC1C(=O)Nc1cccc(O)c1 C1(F)(C(=O)NCC2CCC(=O)N2)CCCN(C(c2cccc(F)c2O)=O)C1 C1(C2CC2)(C(=O)NC2CC(CCNC(c3cnccn3)=O)C2)CCOCC1 C(=O)(CCC(O)C(C)(C)C)NC(C)CC1CN(C(=O)Cc2nncn2C)C1 Cc1cc(C)c(CC(N2CCC(CCNC(C3CCSC3)=O)CC2)=O)c(O)n1 N1(C(C2CC=CCO2)=O)CC2CCC(C1)N2C(=O)C=Cc1ccc(O)cc1 c1(C(=O)NC2C(C)CCN(C(C3(C(N)=O)CCC3)=O)C2)cccc2ccnn12 C1(C(=O)NCC2N(C(CC(C)c3ccccc3)=O)CC2)COC(=O)N1C Cc1cc(I)ccc1C(N1CCN(C(c2cnccc2Br)=O)C2CC12)=O c1(Nc2c(CC(=O)NCCCCCC)cccc2)cc(Cl)cnc1OC CCCCC(CC)C(=O)NCC(C(=O)Nc1ccc(C#N)cc1CC)C(C)(C)C c1(OC)ccc2c(c1)nc(OC)n2C.c1(N2C3(CCCC3)C2=O)ccc(F)cc1 c1(NCC2(CNC(=O)CC(O)C3CCCC3)CC2)cc2nn[nH]c2cc1[N+](=O)[O-] C1(C(=O)NC(CNC(c2cnc(S)[nH]2)=O)C2CC2)CCS(=O)(=O)C12CCC2 c1(OC)ccc2c(c1)C(C(=O)NCCC1CC(NC(C3(OC)CC3)=O)C1)CC2 C(=O)(CC1CS(=O)(=O)c2ccccc21)NCCNC(CC(C)OC)=O c1(C(=O)NC(C2(O)CN(C(CCC(=O)NCC)=O)C2)C)cc2nc(Cl)ccc2o1 n1(CCC)cc(C(=O)NCC(C)CN(C(=O)CSCC2CCCO2)C)cn1 c1(C(=O)NC2CCCN(C(CCCN(C(C)=O)C)=O)C2)nccc2c[nH]nc12 c1(NC(C2(C(N3CCC(C)C(C(F)(F)F)C3)=O)CC2)=O)ccnc2ncnn12 N1(C(C(=O)NCc2ccccc2)CC2CCCCC2)C(=O)c2ccccc2C1=O N1(C(C(F)=CCC)=O)CCC(F)(C(=O)NC23CC2CN(C)C3)CC1 CCCCC(C(=O)NCC1(F)CCOC1)NC(c1scnc1Cl)=O C1(NC(CN(C(C)C)C)=O)C2CC(CN(C(=O)CC3CCNC(=O)C3)C2)C1CO N1(C(C)=O)CCN(N(C)Cc2ccnn2-c2cccc(C#N)c2)CC1 C(CCNC(N)=O)(C(F)F)NC(CCNC(=O)OC(C)(C)C)F C(=O)(CC(C(C)(C)C)NC(C1CN(C)CCO1)=O)NCC(=C)C C1(C(N2CC(OC)(CNC(c3conc3C)=O)C2)=O)CC2(CCC2)CO1 C1(CNC(C2(CC=C)CC2)=O)CCCCN(C(=O)COCCF)C1 c1(CC(=O)NC2C(NC3(C(=O)OCC)CCCC3)CCC2)ccc(OCC)nc1 c1(C(N2CCCN(C(c3cnc(Cl)s3)=O)CC2)=O)nccc2c1NCCC2 c1(C(=O)OC)ccccc1C(=O)NC(C)CCNC(c1ccc(CCF)cc1)=O c1(C(N2CCCC(C)C2CCNC(=O)CCNC(N)=O)=O)ccn2ncnc2c1 Cc1cc(O)ncc1C(=O)NC12CCN(C(c3cc(N)cnc3C)=O)CC1C2 N1(C(C(COC)C)=O)CCN(C(=O)C(C2CCCCC2)C)CC1CC1CC1 Cc1cc(Br)ccc1C(=O)NCC1CC1CNC(C1CCCNC1)=O C1(C(=O)NCC2(C(C)C)CC2)CCCN(C(c2nocc2Cl)=O)CC1 N1(C(Cc2c(C)ccs2)=O)CCCCC(NC(=O)C(C)NS(C)(=O)=O)CC1 C(=O)(C(COC)CC(C)C)NCC(CCNC(C1(COC)CCC1)=O)O N1(C(c2cc(C(F)F)on2)C(=O)NC(CC)C)CCC2(CCCN(C)C2)C1 CC1CCCC(C(=O)NC2(CN(C(=O)CCOCC3CCC3)C)CC2)O1 C12(NC(c3c(C)snc3)=O)CCC(C(=O)NCCOCC3CCCC3)(CC1)C2.CON C1(C(=O)NCCn2cc(C(N(CC(C(=O)NC)C)C)=O)nc2)CC12CCOCC2 C1(CC(=O)NCC(CNC(CN2CCC(C)C2)=O)(C)C)SC2=NCCN2C1=O C(=O)(C(CC1CCOC1)NC(=O)OC(C)(C)C)N(CCCC)C(C)Cc1ccccc1 CC(CCC(=O)NCC1(O)CN(C(=O)CC2CC3CC3C2)C1)N(C)C c1(C(=O)NCCC(C)NC(c2c(F)cccc2Br)=O)ccc(=O)n(C)c1 CCCC(CCCO)C(=O)N1CC(NC(=O)C(C)=C2CC2)C(C)C1 c1(C2(C(N3CC(NC(CC4C(C)C4)=O)C3)=O)CC2)ccc2ccncc2c1 N1(C(C(C(C)(C)C)O)=O)CCC2(CC1)CC(NC(=O)Cc1cc[nH]n1)CCO2 CC1(NC(C2CCCCN(C(c3cc(C4CC4)on3)=O)C2)=O)CCCCCC1 c1(NC(C2CCCC(NC(CCNC(C)=O)=O)C2)=O)cccc(F)c1Br CCC(C)(C)C(O)C(=O)N(CC(C)NC(c1ccc(C)c(OC)c1)=O)C CC1(C)CCC(C(N2CCCCC(NC(C3(C(F)(F)F)CCCC3)=O)C2)=O)OC1 c1(NCCCC)nc(N(C)CC2(CO)CC2)nc2ncn(C)c12 CC1(C)C(=O)NCC1NC(=O)C(C1(O)CCC1)NC(C1CCCCC(=O)C1)=O C(=O)(C1CCCc2nc[nH]c21)NCC1(C)CCCN(C(=O)CCOCC(F)F)C1 c1(C(C(=O)NCCNC(=O)C(C)SCC)N(CC)CC)ccccc1 CCC1=NOC(C(N2CCC(C)C2CNC(c2ccc(C)cc2)=O)=O)C1 C1(NC(COC2CCN(C(c3n(C(C)C)ccc3)=O)C2)=O)(CO)CC2CCCC12 C1(C(=O)NCC2CC(C(=O)OC)C2)CC2CN(C(=O)C(C)CC(F)(F)F)CC2C1 c1(NC(C)=O)ccc(C)c(C(=O)NC2CN(C(=O)C(F)CC3CCC3)CC2O)c1 CON1CCC(C(=O)NC(CCN(C(=O)CC2=CCCC2)C)C(C)C)CC1 CC1CCN(C(C2CC(=O)C23CCC3)=O)CC1CC(=O)NC1CC2C=CC1C2 C1(C(N2CCC(NC(C(C)C(F)(F)F)=O)CC2)=O)CCc2cc(F)ccc2O1 N1(C(C(C)SCCCC)=O)CCN(C(=O)C=CSCc2ccco2)CC1C1CC1 Cc1nc(C(=O)NCC2CC2CNC(c2cccn2C(C)C)=O)ccc1Br CC1=C(C(=O)NC23CC2CN(C(=O)C(c2ccccc2)C2CC2)C3)CCS1(=O)=O N1(C(C(C#C)(C)C)=O)CCC2(CCCN(C(=O)CN(c3ncccn3)C)C2)CC1 C1(CCC)(NC(=O)C(C)COC)CCCN(C(=O)CCCc2cccs2)C1 c1(OC)cc(C(=O)NC2CN(C(=O)CN3CCC3C)CC2(F)F)cc(F)c1 CC(C)CC(C)C(=O)NCCCCC1CCN(C(=O)CCCC#N)CC1 c1(OC)cnccc1C(N1CCSCC1C(=O)NC(C)C(C)(C)O)=O CC1=CCC(C(=O)NCCC2(CNC(=O)Cc3ccc(C)s3)CC2)CC1 C1(CN(C)C(c2cc(C(C)(C)C)ccn2)=O)COCCN1C(=O)C=CC=C(Cl)Cl Nc1ccc(F)c(C(=O)NC2CCC2NC(=O)C=CC2CCCO2)c1 C1(C(=O)NCC2CCN(C(CCCCOC)=O)CC2C)CCc2ccccc2C1 N1(C(COCC(C)C)=O)CCC(NC(c2cc(Cl)cc(Cl)n2)=O)C(O)C1 C1(C(=O)NCC(=O)N(C)CCC2(CO)CC2)CCCN1C.C(C(N)=O)S n1(SCCOCC#C)nnc2c1CCCC2 CC1C(=O)NCCCN1C(=O)NCCN1CCN(c2ccccc2)CC1 c1(C2CC(=O)N2C2CC2)ccncc1Cl.C(=O)(C(O)COC1CCOCC1)OC c1(CC(N2CCCC(c3cn(CCN(CC)CC)nn3)C2)=O)ncnc(C)c1C c1(C(=O)NCCN(CCOC)C(c2coc(C3CC3)n2)=O)nnc(C)o1 N1(C(CC(CC)C)=O)CC(CNC(=O)C(C)(C)c2ncco2)CC12CCC2 NC(Cc1c[nH]nc1O)C(=O)NNC(=O)c1cn(C2CCOCC2)cn1 C1(CNC(C)=O)CCCN(C(C)C(=O)NCC(c2ccc(Cl)cc2)C)C1 CC(CC(C)NC(c1snnc1C1CC1)=O)NC(=O)C(O)CC1CC1 Cc1scnc1C(=O)NC1(C(=O)NCCN(C)CCOCF)CCC1 C1(CNC(CC)=O)CN(C)CCN1C(c1cc(OC)cc(Br)c1)=O N#Cc1cnccc1CNC12CC(C(=O)Nc3c(Br)ccnc3Br)(C1)C2 N1(C(C(CC)NC(N)=O)=O)CCOC(C2CN(NC(=O)C(CCOC)OC)C2)C1 Cc1cc(Cl)cc(C(=O)N(C(C)CN(C)C(C2CC3CCC3C2)=O)C)c1C C(N(C)N1CCC2(C(C(F)(F)F)C2)C1)c1c(C(C)=O)cccc1 c1(COC)ccccc1C(N1CC2CC2(CNC(c2cnnc(O)c2)=O)C1)=O C12(OC)CCCC(CC(NC(c3ccncc3-c3ccccc3C(C)C)=O)C1)C2 c1(COC)ccccc1C(=O)NCC1(COC)CCN(C(=O)C(C)(C)C2CC2)C1 c1(CNC(C2(C)CCC2)=O)ccccc1-n1cc(C2COC(C)(C)C2)nn1 C1(NC(C(c2ccc(C)cc2)(F)F)=O)CC2(CCN(C(C3(C(N)=O)CC3)=O)C2)C1 c1(CC(N2CC(NC(C3CC(C)(O)C3)=O)CC(C)C2)=O)ccc(F)cc1[N+](=O)[O-] C1(C(=O)NCCc2cnc(C)[nH]2)COCCN(C(C2Cc3nccn3C2)=O)C1 Cn1cc(C(=O)NC2CCC(CC(=O)NC(C)(C)C)CC2)c(C(F)F)n1 C(=O)(C1=NN(C)C(=O)CC1)N1CC(C(=O)NC(c2ncc[nH]2)C)N(C)CC1 CCC(C)(CNC(=O)C(C)(CSC)NC(=O)COC1CCC1)C(C)O N1(C(C#C)C)CCCN(C(=O)NCC2(CCN(C)C)CCCC2)CC1 c1(C(=O)NCC(C(C)C)NC(c2cc(C)nnc2)=O)cc(C)c2nc(C)cn2c1 C1(CCC(N2CC(F)(CNC(c3cncn3C3CC3)=O)C2)=O)CCC(O)CC1 N1(C(CSC)=O)CCC2(COCC(CNC(c3cncc([N+](=O)[O-])c3)=O)O2)C1 c1(C(N2CCC(C)C(C)(C)C2)=O)ccc2nc(S)[nH]c2c1 c1(OC)cnc(F)cc1C(N1CCN(C)CC1CNC(=O)CC12CCCC1C2)=O C(CNC(=O)C(c1ccccc1Cl)O)(CC(F)(F)F)NC(=O)Cc1ccsc1 CCC(C)(C(=O)NCCCN(C(=O)C(C)(C)CF)C(C)C)C(N)=O C=CC1(CC(=O)NC2(CCC)CC2)CN(C(c2cnn(CC)c2)=O)C1 Cc1ccc(C(=O)N(C2CCN(C(C3CC34CCC4)=O)CC2)C)c(C(C)C)n1 C(CC)(CC(=O)N(C)Cc1nncn1C)N(C(c1ccc(CC)s1)=O)C N1(C(C(C)N(C(=O)CC(O)C2CCCC2)C)=O)CC(CO)CC1CO c1(NCCN(CCOC)C)[nH]c(=NCc2scnc2C)nc2c1ncn2C(C)C C1(CNC(=O)C(O)COC(C)(C)C)CN(C(=O)C(F)C2CCC2)CC12CC2 N1(C(c2nccc(CNC(c3csnn3)=O)c2)=O)CC2CCC1C(O)C2 C1(CNC(c2c(CNC(=O)CC3CC=CCC3)cco2)=O)CC1C1CCC1 N1(C(C(CC)NC(C)=O)=O)CCC(N(C(c2ccccc2F)=O)CC2CC2)CC1 c1(CNC(C(N2C(C(N)=O)CC(O)C2)=O)=O)cc(F)ccc1F Cc1c(Br)ccc2c1CCC2NCc1ccc(F)c(C(F)(F)F)c1Cl N1(C(CCC(C)OC)=O)CC(C2CCCCN(C(C3(C)CCCC3C)=O)C2)C1 N1(C(C(C)n2ccnn2)=O)CCN(C(=O)CC2(CO)CC2)C2CCCCC2C1 c1(C(=O)NC2CN(C(Cc3ccc(C)nc3)=O)CC2C)cnc2c[nH]nc2c1 c1(CC)ncnc(CC)c1C(=O)NCCC1(NC(=O)CC2COC(C)(C)C2)CC1 C1(C(C)C)(CO)CCCN(C(=O)CCc2ccc(Br)c(F)c2)C1 C(CN=c1ccc(C#N)c(C)[nH]1)C1CCC(NC(C=CCC)=O)C1 C1(NC(C(Cc2ccsc2)NC=O)=O)CC2(CCN(C(C3(F)CC3)=O)CC2)C1 C#CC(C)(C)C(=O)NC1CCC(C)(CNC(=O)C=CBr)C1 c1(NC(C2(CNC(c3cccc(C(F)(F)F)c3)=O)CC2)=O)nc(F)ccc1Br NS(=O)(=O)c1ccc(C(=O)NC2CC2CNC(C2CC2C(F)(F)F)=O)c(F)c1 c1(C(=O)NC2CC(CNC(COCCC#C)=O)C2)c(O)cc(Cl)cc1Cl Cc1nc2c(C(=O)NC3C4CC3N(C(c3cc(C)sn3)=O)C4)ccnc2[nH]1 Cc1ccc(SCC(N2CCCCC2CNC(=O)CC2CCC23CCC3)=O)cc1 N1(C(C2OCCC(C)C2)=O)CC(NC(=O)C(C)n2cccn2)CC2(CCC2)C1 c1(CCC(=O)NCC(CC)NC(=O)C(C)C(F)F)c(C)noc1C Cc1ccc(OCC(=O)NCC(C)CN(C(=O)Cc2nc(C)sc2Cl)C)cc1 CCCCCC(C)(C)C(=O)NC1CC2CC(C1)N(C(=O)CCSCC(N)=O)C2 C12(C(N3CCCC(CN(C)C)C3)=O)CCCC1CCN2C(C1CCOC1)=O CC(CNC(C1(C)C=CCC1)=O)CC(=O)Nc1csc(Cl)c1 Cc1coc(C)c1C=CC(N1CC2CC(NC(C3CCC34CCC4)=O)C1C2)=O N1(C(C=C(C)C(C)(C)C)=O)CCC(CO)C(NC(c2cc(O)nc(O)c2)=O)C1 c1(C(=O)NC2(C(C)C)CCC2)cccnc1CNC(=O)C(F)CC1CCOC1 C(CCCCCOC)NC(c1cnc(C(=O)OC)s1)c1nnnn1C1(C)CC1 Cc1nc2ncc(C(=O)N(C3CN(C(=O)CCC=CC(C)C)C3)C)c(=O)n2[nH]1 N1(C(c2ccc(OC)cc2Br)=O)CCCC2C1CCN2C(c1ccnc(O)c1)=O C(CCCCC(=O)N1CCCC(F)(C(=O)Nc2ccccc2)C1)NC(N)=O Cn1c(C(=O)NCC(=O)NCC(N2CC(C#N)C2)=O)cccc1=O C(CCCCC(=O)N1CCC(F)(F)CC1)NC(c1c(CCC)[nH]cc1)=O C=C(Cl)CC(C(=O)NCC(C)C1CCC1)NC(=O)C(F)OC(F)(F)F Cc1c(NC(C)C)cccc1C(N1CCOC(CNC(c2cncs2)=O)C1)=O c1(CN=c2cc(C)nc(N3CCn4nccc4C3)[nH]2)cc(O)n2nc(C)cc2n1 Cc1cc(O)ccc1NC(=O)CC1CCC(NC(C2(F)CCC2)=O)CC1 N1(C(CCCn2c(C)ncc2)=O)CCC(N=c2[nH]c3ncc(Cl)cc3o2)C(C)C1 C1(C(=O)OCC)CN(C(C2CC3C=CC2O3)C(=O)NCCOCC)CCO1 N1(C(C(CC#C)(C)C)=O)CCC2(CC1)CN(C(c1cc(S(N)(=O)=O)co1)=O)C2 c1(C(=O)NC2C(C)CN(C(c3cccnc3C3CC3)=O)C2)cnn2ccncc12 CS(=O)(=O)c1ccc(OCCC(=O)NCC2CC2CF)cc1 N1(C(c2cc(C)c(Br)s2)=O)CCC(F)(CNC(C2CCOC2)=O)CC1 C1(C=O)C(n2cc(C(=O)NCCOCCO)nn2)C1(C)C.C1(CC2CC2)CN(C)C1 Cc1ccc(CNC(=O)CC2CN(C(c3cn(CCO)nn3)=O)CCO2)nc1 Cc1csc(=O)n1CCC(=O)NC(C1CCCN1C(=O)C(C)C(C)C)(C)C N1(C(C2CCC3CCCCN23)=O)CCCC2(CCN(C(C3CCOC3)=O)CC2)C1 N1(Cc2ccc(CNC(C)=O)cc2)CCC2OC(=O)OC2C1 C(CC(CC)C(=O)NC(C)CC(=O)N1CCC1C1CCCCC1)=CC N1(C(CCCCN(C(C(CCCC)N(C)C)=O)C)=O)CCn2nc(C)cc2C1 N1(C(C2CCC(CCCCC)O2)=O)CCC(C)(C)C(C(=O)NC2CC(C)(O)C2)C1 N#Cc1ccnc(N2CCCC(C(=O)NCCSc3cccs3)C2)c1 N1(C(C(CSC)O)=O)CCc2nc(CNC(C3CC4CCC(C3)S4)=O)sc2C1 c1(C(=O)Nc2ccc(C(=O)NC(CO)C(F)(F)F)cn2)ccc2sccc2c1O C(=O)(CCCCN=[N+]=[N-])NCc1occ(C(=O)NCC2N(C)CCN(C)C2)n1 N1(C(C2C(C(=O)OC)C=C2)=O)CCCC1C(=O)NCCOC1CCCCC1 C1(NC(C(C)(F)F)=O)CN(C(=O)Cc2cccc3nsnc23)CC2(CC2)C1 c1(OC)cc(OC)c2cc1O2.c1(C(C(=O)CN(C)CC2CC2)O)ccccc1C c1(OC)cc(C)cc(C(N2CC(Cn3cc(CNC(C)=O)nn3)C2)=O)c1C S(=O)(=O)(c1ccc(Cl)c(Cl)c1)NC(c1cc(Cl)cc(Br)c1)CC(=O)O O(C1CCc2c(Cl)ccnc21)C(C1CC1(Cl)C(=O)O)=O C12(NC(c3cnc(CNC(C4CC=CCC4)=O)nc3)=O)CCN(CC1)CC2 C(CCCCCn1cc(CC2(O)CCC2)nn1)NC(=O)CCCC1CC1 C(=O)(C(C)(C)NC(C1(N(C(=O)CC2CSCCO2)C2CC2)CCC1)=O)N(C)C N1(C(c2ncc(N)nc2)=O)CC(NC(=O)CC2(O)CCC2)CC12CCC2 Cc1cc(=NCCP(C)(C)=O)[nH]c(N2CC3CC(C)(C)C3C2)n1 c1(NC(=O)NC(c2ccc(N(C)C)cc2)C)ccc(F)cc1NS(C)(=O)=O CCCC(O)C(=O)N1CCOCC1CC(=O)OC.c12ccoc1C(=O)NOC2 c1(C(=O)NC(C)C(CO)NC(c2ccc(Cl)nc2O)=O)cnc2c(c1)CCCO2 Cc1ccc2c(C(=O)NC3CN(C(C4(C)CCCO4)=O)CC(F)(F)C3)csc2c1 N#Cc1ccc(-c2cn(C3CC(NC(=O)CCCCCF)C3)nn2)cn1 Cc1ccc(C(=O)NCC(CO)NC(=O)Cc2ccccc2CC(N)=O)c(O)n1 N1(CC)CC(NC(C2(CNC(=O)C=CC3CC3)CC2)=O)CCC1=O C(=O)(C(F)(F)C(F)(F)F)N1CC(CNC(c2c(C)ccc(NC)c2)=O)OCC1 C(CC(C(=O)NC1CC(O)C1OC)NC(c1cccc(O)n1)=O)OCC Cc1cccc2c1CN(C(=O)CC(CNC(=O)C=Cc1ccc[nH]1)C1CCC1)C2 C1(NC(C(c2cccs2)NC(CCNC(COC)=O)=O)=O)CCOC2(CCC2)C1 c1(OC)cc(C(=O)NCCC2(CN(C(C3CN(C(=O)NC)C3)=O)C)CC2)c(C)o1 c1(C(N2C(CNC(CC(=C)C)=O)C(C)CCC2)=O)nc2c(s1)CN(C)CC2 N1(C(c2ccc(CC)o2)=O)CC2(C1)CN(C(C1CCN(C(=O)OC)C1)=O)C2 c1(C(N(C(C)CN(C(=O)CSC(F)(F)F)C)C)=O)cc(F)cc2nn[nH]c12 C1(C(=O)NCCCOCC2CC2)COC2(C1)CN(C(c1nc(Cl)cs1)=O)C2 CC1(CCC(=O)NCc2ccncn2)CN(C(c2ccsn2)=O)C1 C1(CNC(c2nn(CC)c(C)c2)=O)CC2(CC(NC(C3CC3Cl)=O)C2)C1 Cc1cccc2nc(C(=O)N(CCC(C)NC(c3cc([N+](=O)[O-])c[nH]3)=O)C)cn12 c1(C(=O)NC23CC(NC(=O)CC4COCCO4)(C2)C3)cn2ncccc2n1 c1(C(=O)NC2CC3C(NC(Cn4ncc(CC)c4)=O)C3C2)cc(C)c(O)nn1 c1(C(C)(C)C)cc(C(N2CC3CNC(C3)C2)=O)cc(C(C)(C)C)c1O Cc1c(C(=O)NC(C)CCCCNC(=O)CSCC#N)nnn1C1CCOC1 C1(C(N(C2CCN(C(=O)CNC(C)=O)C2)CC)=O)Cc2nnsc2S1 C(C)(C)(CC(=O)NC1CC(N2CCCC2)C1)N(C(C(=O)NC)=O)C Cc1cncc(C(=O)NC2CCC(N(C)C(c3cc(Br)co3)=O)CC2)n1 N1(C(c2c(OC)n(C)nc2)=O)CCC2CC(C1)CN(C(=O)CC1CCCC1)C2 c1(C(N2CCCC(NC(=O)Cc3cnccc3Cl)C2)=O)cnc2scnc2c1 C1(C(=O)NCC#CCNC(c2c(N(C)C)cccn2)=O)CC2CCCCCC12 CC1(CNC(=NCCc2ccccn2)NC2CCCOC2)CCC(F)(F)CC1 N1(C(c2c(C)sc(C)c2C#N)=O)CCCC12CCN(C(=O)Cc1cscn1)CC2 C(CN=c1[nH]cnc(C)c1Br)N(C(C1(CC)CCNC1=O)=O)C C1(C(=O)NCCC(=O)NC(C)COC(F)(F)F)CCCCCCC1 N1(C(C(CC(C)C)(C)C)=O)CC2CS(=O)(=O)CC2(NC(=O)C(=O)N(C)C)C1 C=CCC(Cc1ccccc1)C(=O)N1CCCCC1CN(C)C(C1(CF)CC1)=O Cc1nccc(C(=O)N(C(C)C(=O)NC2CCN(C(C)C)C2)C)n1 N(C(=NCCF)NCC(=C)C)C1C(C=C)OCC1 C(=O)(C(C)CC(F)(F)F)NC1C2(CC(NC(c3c(C#C)c[nH]n3)=O)C2)C1 O=C1NC(C2CC=CCC2)C(=O)N1CC1(n2cccc2)CCCC1 C1(CCNC(CCC=C)=O)CN(C(=O)Cc2ccc(OC)cc2)CC(C)O1 N1(C(c2c(C)cns2)=O)CCC(C2CCN(C(=O)CC3CCC(=O)N3)CC2)CC1 C12CC3CN(CC3C1)c1nc(cn1C(C)C)CNC2=O.Cc1ccn(C2CC2)n1 C12(NC(c3ccnc(OC(F)F)c3)=O)CCC(NCc3sc(Br)nc3Br)(CC1)C2 C(=O)(C(C)(F)CC1CN(C(=O)OC(C)(C)C)C1)Nc1c(OC)scc1 c1(C(N2CCC(NC(C3(CC)CC3)=O)CC2C)=O)cc2ccc(Br)cn2n1 N1(C(c2ccc(OC)o2)=O)CC(F)(F)CC1(C)CNC(C1(C(F)F)CCC1)=O c1(C(=O)NC2CC(N(C(=O)Cn3cnnn3)C)C2)cccc2nc(C(F)F)[nH]c12 C1(CC=C)(NC(C2CCCN2C)=O)CCN(C(c2cncc(N(C)C)c2)=O)C1 C1(CC)(Nc2cc(C3CC3)nc(Cl)n2)CCN(C(=O)CC2C=CCC2)CC1 Cc1ccc2c(O)c(C(=O)NCC3CC4CCCCN4C3)cnc2n1 C1(C(=O)NCC(C)(C)OCCNC(=O)C2=CCCOC2)C(C)(C)CCCC1(C)C C12(NC(C(CC3CCC3)NC(c3ccnnc3O)=O)=O)CCC(O)(CC1)CC2 Cc1ccc(C(N2CCCCC2CNC(c2nc(Br)c(C)s2)=O)=O)c(O)c1 N1(C(COCC#C)=O)CCOC2(CCN(C(=O)CNC(=O)OC)CC2)C1 C1(NC(C2N(CCC)CCC2)=O)CC2(C1)CC2NC(=O)Cc1nnc(C)s1 C1(c2onc(-c3c(OC)nsc3)n2)CC2CC1CC2OC c1(C(N(C2CCN(C(=O)CN3CCS(=O)CC3)C2)CC)=O)ccc2n[nH]cc2c1 C#Cc1ccc(C(=O)N(C2CCCN(C(c3cc(C)c[nH]3)=O)C2)C)cc1 Cc1noc(C)c1C(=O)NC(CO)C(C)NC(=O)CC(O)CN(C)C N1(C(CC2CCCC(OC)C2)=O)C2CCC1CN(C(C1CC3(CC3)C1)=O)C2 C1(NC(CCOC)=O)CC2CCCC(C1)N2C(=O)C=CC1CCCO1 C1(O)(CC(=O)OC(=O)C(c2ccncc2)NCC)CCN(C(=O)C(C)(F)F)C1 c1(OC)ccc(Cl)c(C(=O)NCC(c2cccc(C)c2)NC(=O)C2=CCC2)n1 CCC(C)CC(=O)C(=O)N1CCC(NC(=O)CN(C2CC2)CC)C1 C1(C(C)NC(C(CN(CC)CC)F)=O)CN(C(=O)CCSC)CCO1 CC1CCN(c2nnc(-c3ccccc3)o2)CC12CCC2 N1(C(C)=O)CCCCC1C(=O)NCCC(C(C)C)NC(c1n[nH]cc1C1CC1)=O C12(NC(=O)CCc3nc(O)n[nH]3)CC=CCN1CCC2.c12cn(nn1)CCOC2 Cc1cc(C)cc(C=CC(N2CCN(Cc3ccccc3F)CC2C)=O)c1 CC1CCC(OC(C2CC(=O)C23CCC3)=O)CN1C(=O)NC1CCCCCC1 N1(C(C(c2ccc(C)cc2)=O)=O)CCCC(C)(CNC(C2CNC(=O)O2)=O)C1 C(=O)(C(C(C)C)C1CCC1)N1C(C(N2C(CSC)CCC2)=O)(C(C)C)CCC1 c1(C(=O)NC2CN(C(c3cc(Br)c[nH]3)=O)CC2F)cc(Br)ccc1I C1(C(=O)NC23CC(NC(C(C)c4ccsn4)=O)(C2)C3)CC2(CCCCC2)S1(=O)=O n1(CC(=O)NC(C2CCO2)C)ccc(C2CC2)n1 CCCC(CC)CC(=O)N(C1CC2CCC(C1)N2C(C1CCC(C)(C)CO1)=O)C c1(C(N2CCC(NC(CSCC=C)=O)C2)=O)ccc(OC(F)(F)Cl)cc1 C1(C)(CC)CCC(C(=O)NCc2cc(C(N3CC(c4nn[nH]n4)C3)=O)co2)O1 c1(C(=O)NCC2C(C)(C)N(C(=O)CCC3CCC3)CC2)cccc2oncc12 c1(C(=O)NC2CN(C(=O)CCCCCF)CC(O)C2)c(O)cnc2ccccc12 c1(OC)cc(C(=O)NC(C)C(C)NC(c2cc(Cl)c(F)cc2N)=O)cc(F)c1F c1(C(N(C(C)CN(C(=O)CC2CSC2)C)C)=O)ccc2c(c1)CN(C)C(=O)N2 CC1OC2(CNC(=O)CCC#N)CC1(NC(C1CCC(=O)N1C)=O)C2 C1(CCC=C)CCCN(C(=O)C(CNC(=O)CC(CC)OC)N(C)C)C1 N1(C(C(=O)N(C)C)=O)CCC(CCNC(C2CCC(O)CN2C)=O)C(F)(F)C1 c1(C(=O)NCC2C(NC(c3cc4c[nH]nc4s3)=O)CCC2)cccc2sccc12 C12(C(=O)NC3C(CNC(c4c(OC)c(Cl)sc4)=O)CCCC3)CCC(C)(C1)OC2 C1(C(=O)NC(C)C#N)Cc2ccccc2CN1C(c1ncc(Br)s1)=O Cc1ncc(Br)c(C(=O)NCC2CCN(C(=O)CCP(C)(C)=O)C2)n1 c1(C(N(C2CCN(C(=O)COC3CC=CC3)C2)C)=O)cnn(C2CCOCC2)c1 N1(C(c2cc(C)c(F)cc2)=O)CCC(F)(F)C(C(=O)NC2(CC#N)CCCC2)C1 C(=O)(C1=CC2CCCCC12)NC(C1CCCC1)CNC(c1c(C)nc(CC)o1)=O S(=O)(=O)(c1ccc(C(=O)NC(C)(C)CCNC(=O)CSc2nncs2)cn1)NC c1(C(=O)NC2C(CNC(Cc3nc(COC)sc3)=O)CC2)ccn2nnnc2c1 CN1c2ccccc2CC1C(=O)NCC12CC(CN1C(C1CCN1C(C)(C)C)=O)C2 c1(C(N(C2CCN(C(C3CCCC(=O)N3C)=O)C2)CC)=O)ccc(F)c(C)c1 c1(C(N2C(C3(NC(c4cc(OC)no4)=O)CC3)CCC2)=O)ccc2c(c1)NCC2 Cc1ccnn1CC(=O)NC(Cc1cn[nH]c1)C(=O)NCC(=O)NCCO C(CCC(=O)N(C1(CNC(C)=O)CCSC1)C)=CCC=C N1(C(C2C(CC)CCO2)=O)C2CCCC1CN(C(c1csc3cncn13)=O)C2 C(=O)(C1=CC(O)CCC1)NC(C1CCCC1)CNC(C(C)=CC1CC1)=O CC(C)(F)CCC(=O)N1CC(C(=O)NC(c2nc[nH]n2)C2CC2)C2(CC2)C1 N1(C(C2(C)CCN(C(C)=O)C2)=O)CCC2(CCC(NC(c3ccccc3)=O)C2)C1 CCCC(C)N=c1[nH]c(=NCCCN2CCCC(C(N)=O)C2)[nH]c2cccnc12 C1(CN(CC2C(C(=O)OCC)CCCC2)CC)CCC2(CCC2)C1 N1(C(CC(C(C)C)O)=O)CC2CCC1CN2C(c1cc(C(F)(F)F)cc(O)n1)=O N1(C(C(C)(C)NC(C)=O)=O)CCCCC1CNC(=O)C(c1ccc(F)cc1)C c1(C(=O)NCC2(NC(c3nc(OC)oc3)=O)CCCC2)cc(F)cc(Cl)c1O C1(CNC(c2cc(C(C)C)sn2)=O)CN(C(=O)C#CC(C)(C)C)CCCO1 c1(OCC(=O)N(C)C)ccc(C(N2CCCC(Nc3ccccc3)C2)=O)cc1 c1(CC(=O)NCCC(C)NC(C(COCC)C)=O)cccc(C)c1Br C1(NC(CCSC)=O)C=CCN(C(=O)CCN2C(=O)CCC2=O)C1 n1(CC)nc(C(N2CCC(C3CCCN3C(=O)Cc3csnn3)C2)=O)cc1O N1(CC(N2C(C)(CNC(c3csc(Cl)c3Cl)=O)CCC2)=O)CCS(=O)(=O)CC1 c1(CCCC)ccc(S(=O)(=O)NCC23CC2CN(C(=O)C=C(C)C)C3)cc1 CCC(O)C(C)C(=O)NC1(CNC(=O)C(c2ccc(F)cc2F)=O)CCC1 C1(CNC(c2cc(Cl)c(F)c(Cl)c2)=O)CN(C(c2cccnc2)=O)C2(CCC2)C1 C12(CNC(c3c(SC)cccc3)=O)CCC1CCN2C(c1[nH]cc(C)c1C)=O Cc1ccc(CCCNC(=O)C(C2CC2)NC(=O)C(=O)N(C)C)cc1C C12(C(=O)NC3CN(C(c4nc(C)oc4C)=O)CC3O)CC(CC(C)O1)C2 c1(C(N(CC(C)N(C(C(COC)OC)=O)C)C)=O)cnc(-n2cccn2)c(C)c1 C(=O)(C(C)(F)C(=O)N1CC(CNC(c2cc(C)sc2C)=O)(COC)C1)OCC c1(C(N2CC(CCn3cc(C(CC)(C)O)nn3)C2)=O)nnn2c1COCC2 C(=O)(CCCCC(=O)NC)NCCC(C)NC(c1c(SCC)cccc1)=O N1(C(C2(CC)CCCCC2)=O)CCC(C(=O)NCC(CO)C(C)C)CC1(C)C C1(C2CCCN(C(c3ccc(F)cc3N)=O)C2)(NC(C(CCCC)(C)F)=O)CC1 C1(NC(CN(C)C)=O)CCC2CCN(C(c3cc(F)cc(Br)c3)=O)C1C2 N1(C(C(C2CCCC2)OC)=O)CCCN(C(c2cccc3c2NCC3)=O)C(C)C1 C(c1cnccn1)=CC(=O)NC(CC(C)NC(C1CC(=C(F)F)C1)=O)C Cc1cc(C(=O)NCC(C)CNC(=O)C(C)NC(C2CCC2)=O)c2occc2c1 c1(NC)ccc(C(N2CC(NC(=O)C=Cc3cccs3)C3CC23)=O)nc1 CCCC(C)CC(=O)NC1COCCC1NC(c1cccc(OC)c1C)=O c1(C(N2CCC(C(=O)Nc3ccc(CC)nc3)(C(C)C)C2)=O)cccc(C)c1O Cc1ccc(-c2cnn(CCCO)c2)c2nc(C(N3CCC3CO)=O)cn12 N1(C(C2(C(=O)OC)COC2)=O)CC2CC(C1)N(c1ncnc(=N)[nH]1)C2 C(=O)(C1=CCCCO1)N1CC(C(C(=O)NC(C=C)C(F)(F)F)OC)C1 c1(CC)ncc(Cl)c(C(=O)NC2CCN(C(c3cc(=N)[nH]c(=N)[nH]3)=O)CC2C)n1 N1(C(C=COCC)=O)CCCC2(C1)CN(C(c1cc(C)ccc1C)=O)CCO2 C1(NC(CC)CCc2ccccc2)CN(C)CCN(C)C1 C(C)(C)(C(C)CC(=O)NC1(C)CCCCC1)NC(COC)=O Cc1c(C(=O)NCC2COCC2NC(=O)C=Cc2cnc[nH]2)oc2ccccc12 C1(NC(c2cc(Cn3ncc(C)c3)on2)=O)CCOCC1NC(C1C(C)C1C)=O C12(C(=O)NCCCCN(C(c3ccc(CCC)s3)=O)C)CC1COC2(C)C C1(c2n(CC=C)c(N(C)CC3CCCS3)nn2)COc2ccccc2C1 N1(C(CCCN(C(C)=O)C)=O)CC2CCC1CN2C(C12CCCC1(C(N)=O)C2)=O C=CCN=C(NC1CC1(COCC)COCCC)N1CCC2CS(=O)(=O)CC12 C(CCC(=O)NCC1(CN(C)C(C2(O)CCOC2)=O)CC1)OC(C)C C1(C(C)C)CCC(C(=O)N(C)CCN2CCCC2)C(=O)N1 Cn1cc(C(=O)NC2C3CC2N(C(=O)CC2CCCCC2)C3)cc1Br c1(C(C(=O)N(CC(C)NC(C2CC(C(F)(F)F)C2)=O)CC)O)cccnc1 N1(C(C=CC(C)NC(c2ccc(CC)nc2)=O)=O)CC(N(C)OC)C1 C(=O)(CCS(=O)(=O)CC(C)C)NCC1(C)CCN(C(C(C)OCC=C)=O)C1 C=C(C)c1ccccc1NC(C1(NC(c2cccc(CO)n2)=O)CC(O)C1)=O N1(C(c2c(CC)n(C)cc2)=O)CC(N=[N+]=[N-])CC1C(N1CC(O)C(C)(C)C1)=O C12(C(CNC(c3c(C)nsc3)=O)NC(=O)Cc3ccnn3C)CCC(CC1)C2 c1(C(N2C(C)CN(C(C3(C)COC3)=O)CCC2)=O)cnc2cn(C)nc2c1 C(=O)(C(CCC(N)=O)NC(C)=O)NC(C(=O)N(CC)Cc1ccccc1)C Cn1cnc2nc(N3CCC(c4ncccn4)CC3)[nH]c(=NC3C=CCC3)c12 CCCCCC(CC)C(=O)NCC1(C2CC2)CCN(C(C2CCCOC2C)=O)C1 C(CCCCCCO)CC(=O)OCC(=O)NC(c1ccccc1F)CC Cc1c(C(c2nnnn2CCCF)Nc2ccnn2C)cccc1C(F)(F)F C(=O)(C(C)(C)CO)NCc1c(C(N(C)CC2CC2(F)F)=O)occ1 c1(C(=O)NCC2(NCc3ccnc(F)c3)COC2)cccc(I)c1 c1(CC(=O)NC(C2CC=CCC2)C(=O)NC2(CC)CC2)cnc(O)cc1C CC1CCC(C(=O)NCC23CC2CN(C(C2CCN(CC4CC4)CC2)=O)C3)CC1 N1(C(c2nc(C)on2)C)CCc2ccccc2C1CNC(=O)CCn1ccnc1 c1(NCc2ccc(C(C)C)cc2)nc2ccccc2c(=NC(C)c2cnsc2)[nH]1 c1(N2CCN(C(Cn3c(C)cc(C)n3)=O)C3(C2)CC3)ncnc2ccc(F)cc12 c1(OC)c(Cl)cc(C(=O)N(CCNC(c2nc(Cl)cs2)=O)C2CC2)cc1Cl CCC1=C(C(=O)NC2(C3CCN(C(=O)C(C)COC)C3)CC2)CCCO1 C1(S(N)(=O)=O)(C(N2CC(C)C(CNC(=O)C3=NNC(C(F)(F)F)C3)C2)=O)CCC1 c1(C(N2C(C)CC(NC(C3=C(C)CCC3)=O)C2)=O)cn2nc(C)sc2n1 c1(CC)ccc(-c2nc(CCc3nc(C)no3)n(C(C)C(C)(C)C)n2)cc1 Cc1csc(CCCC(=O)NC(CNC(=O)Cc2cnccn2)C2CCC2)n1 N1(C(C(N2CCC(C)CC2)=O)=O)CCC=C(CNC(C2CC(O)C2)=O)C1 c1(C(N2CC(OC)(CNC(=O)Cc3ccnn3C)C2)=O)ccc(C(C)F)cc1 N1(CC)CCCCC1C(N1CC(N(C)C(C2CC(=O)CO2)=O)C1)=O c1(OC)ccccc1C(c1nnnn1C(C)C)NC1CCOC1c1cccnc1 c1(OC)cccc2c1CCC2(CO)NC(=O)N(C)Cc1ccnc(N(C)C)c1 N1(C(CN(CCOC)C)=O)CC(NC(=O)C=Cc2ccc(OC)cn2)C(C)(C)C1 C(=O)(CC1OCc2cc(Cl)ccc21)N(CCN(C(C1(CC=C)CCOC1)=O)C)C n1(C(C(=O)NC(c2nncn2C)CC)C)nnnc1C(C)C c1(OC)ccc2c(c1)OCC2CC(=O)NCCCNC(c1cc(C)ccc1N)=O C(C(C(=O)NC1CC1)N(CC(=O)NC(c1ccccc1)C)C)(C1CCC1)OCC N1(C(c2ncc(CC)cn2)=O)CC2CC1CN(C(C1CCN(C)C1=O)=O)C2 c1(NC(CSC)C)[nH]c(=NC2CC3C(C2)C3(F)F)nc2c1cnn2C c1(C(N2CCN(C(c3cc(CC)on3)=O)C(C)C2C)=O)nc2ncc(C)cn2n1 C(=O)(CCC(C)C(C(=O)NCCCSC)N1CCCOCC1C)OC N1(C(CN(CC)CC)=O)C2CCC1C(CNC(=O)Cc1cnc(C)[nH]1)C2 Cc1nn(CC(=O)NCC2CN(C(=O)CCCn3cncn3)CC2C)c(=O)o1 c1(C(=O)NCC(C2CC2)NC(c2c(CCC)[nH]cc2)=O)c(C2CC2)noc1C c1(C(=O)NC2(C)CC(NC(c3ccccc3-c3cc[nH]n3)=O)C2)ccc[n+]([O-])c1 c1(C(=O)NCCOC(CNC(CC(CC)SC)=O)(C)C)ccn2c(O)nnc2c1 c1(C2CC2)c(F)ccc2nc[nH]c12.C1(C(=O)NC2CNC2=O)CC2CC2C1 c1(OC)ccc(C(NC(=S)N(c2cc(C)ccn2)CCc2cc[nH]n2)C)cc1 C1(c2n(C)c(C3CCC4(CCC4)OC3)nn2)CC12CCCCCC2 Cc1cc2cccnc2nc1C(=O)N(C)CCN(C(=O)CN1CCC1C)C(C)C CCC(C)C(=O)NCC(=O)NCC1(C)CC(NC(=O)C=C2CCCC2)C1 C1(NC(C2C(C)C2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)C2(CCCCC2)C1 C1(NC(Cc2ccc(CCC)cc2)=O)CCN(C(=O)Cc2csnn2)CC1(C)C Cc1c(CNC2(c3nnnn3-c3ccc(F)cc3)CC(C#N)C2)cnn1C C1(C(=O)NCC2(F)CN(C)C2)CCCCCCN1C(C1CCC1(F)F)=O C12(NC(c3c(C)cccc3)=O)CCC(CNC(=O)Cc3ccsn3)(CC1)OC2 C#CCC(CC#C)C(=O)N1CCOCC(NC(=O)C(F)(F)CN2CCCC2)C1 C1(NC(c2ccc(OC)c(Cl)n2)=O)CN(C(=O)CP(C)(C)=O)CCC12CCC2 N1(C(c2c(F)ccc(C)n2)=O)CCC2(CCC(NC(=O)C(C)C3CCCO3)C2)C1 c1(C(N(CC(O)CNC(=O)C(c2ccccc2F)O)C)=O)cc(S(C)(=O)=O)co1 c1(C(CCC(=O)N(CCCN(C(C2C(OCC)C2)=O)C)C)=O)ccc(F)c(F)c1 n1(CCOC)nccc1C(=O)NCC1CCN(C(c2cnoc2C(C)C)=O)C1 N(C1CCc2cccnc21)C(C(N(C(c1ccc(C)cc1)=O)C)C1CC1)=O c1(OC)ccc(Br)c(F)c1CNC(=O)NC1CC(C(C)(C)C)C1 C1(C#N)(OC)CC(C(=O)N(C)CCN(C(=O)CC2CCCCO2)C)C1 Cc1ccc(I)cc1CNC1CCN(C(=O)CC(C)O)CC1 c1(C(N2C(C(=O)Nc3cncc(C)c3)C(C)CC2)=O)cc(C)ccc1C C1(C(=O)NCCC2(C)CCCO2)CC2CCCC2N1C(C1CCCN1C(N)=O)=O C1(NC(CC(CC)SC)=O)COC2(C1)CN(C(=O)C(C)(C)n1cncn1)C2 C(=O)(C(O)CCC(C)C)NC1CC(NC(C(CCC)OC)=O)C(O)C1 CC(O)(CC(=O)NC1CN(C(C2CCC3(CC2)CC3)=O)CC12CCC2)C(F)(F)F N(C1CCCn2ncnc21)C(C(=O)NCCCC1CCOCC1)=O CCCC(C(=O)N(C)CC1CCCN1C(=O)Cc1sc(C2CCC2)nc1C)OC N(C(=NCCN1CCOCC1)NCC(F)(F)Cl)C1CC(C)OC1 c1(C(=O)NCC(C(C)C)NC(c2cnc3c(c2)COC3)=O)nnn2c1CSCC2 N1(C(C(CC)Nc2ncccc2C)=O)CCN(C(c2ccco2)=O)CC1 c1(C(=O)NC(CC)CNC(c2cnc(O)o2)=O)sc([N+](=O)[O-])cc1Cl C=C(Cl)CC(C(=O)N(C1CC2CC2C1)C)NC(=O)C1=CCCCO1 C(=O)(C1=Cc2ccccc2C1)NCc1cnn(C)c1C(=O)NC1CSC1 C1(CNC(C(CSC)C)=O)CCCN(C(C2(OC(C)=O)CC2)=O)C1 Cc1cc(C(=O)NC(C(=O)N(C)Cc2ccco2)C2CCCO2)cc(O)n1 c1(C(=O)NC2C(NC(c3cccc(OC)c3N)=O)C2)cccn2nnnc12 N1(C(C2C(C)C2)=O)CCCC(N(C(=O)COc2cn[nH]c2)C)C1 C1(NCc2cnn(CCC)c2C)CCc2onc(C(=O)N=c3cco[nH]3)c2C1 C1(C(N(C2CCS(=O)(=O)C2)CC#C)=O)CCN(CC(N2CCCCC2C)=O)CC1 c1(C2(C(N(C)Cc3cn(Cc4ncoc4C4CC4)nn3)=O)CCC2)ccc(Br)cc1 C(=O)(C(F)(F)CC1CCCO1)NCC(C)(CO)NC(c1cnc(C#N)s1)=O c1(C(=O)NC(CNC(c2ncc(N(C)C)nc2)=O)(C)C2CC2)cnc(Cl)cc1Cl c1(C(N2CC3C(C2)N3C(c2ccc(F)c(O)c2)=O)=O)ccc(O)nc1Cl c1(C(=O)NCC2CC(F)(F)CN2C(C23CC2C3)=O)c[nH]c2cccnc12 C(=O)(C1CCOc2ccccc21)N1CC=C(CNC(c2c(C)scc2)=O)CC1 c1(C(N(C(C(=O)NC(CC#C)CO)C2CC2)C)=O)cc([N+](=O)[O-])c[nH]1 C1(C(N(CCC(C)NC(=O)CCC(C)(F)F)C)=O)CC(C)(C)OC1(C)C C(=O)(CCC(C)CN(C)C)NCC(C)CC(=O)NC(C)C(=O)NCCF c1(NC(C2C(C(N3CCCCC(C)C3)=O)C2)=O)ccc2scnc2c1Br N1(C(C(CC)C)=O)CC2(CNC(c3conc3C)=O)CCC1CC2 c1(C(=O)NCC2(NC(CC3(C)CC3)=O)CCOC2)cnc2n1CCCC2 Cn1cccc1CC(=O)NCC(C)(C1CC1)NC(=O)C(O)CN1CCCC1 c1(CN2CCCC(C)(C(N3CCCOCC3)=O)C2)ccc2ccsc2c1 C1(NC(C(CCCC)F)=O)CN(C(=O)CCc2c[nH]c(=N)[nH]2)C2CCCC12 CC1CN(C(=O)C=Cc2ccn(C)c2)CCCN1C(C1CCC12CCC2)=O C1(O)(CNC(C(C)Cc2ccccc2)=O)CCCN(C(=O)C(C)N2CCCC2)C1 c1(N2CCN(C3C(OC)CCC3)CC2)ncnc2ccsc12 c1(C(C)NC(=O)CC2(NC(c3cc(Cl)c[nH]3)=O)CCCC2)ccc(F)cc1 N1(C(c2cccc(F)c2)C(=O)NCCCCCC)CCC(CC(F)F)(CO)CC1 c1(OCC(=O)NC2C(C(C)C)N(C(C3CC(C)(C)O3)=O)CC2)ccc(F)cc1Cl N(C1CCc2cc(F)cc(Br)c21)C(N1CC(CC)N(C(=O)C2CC2)CC1)=O C(=O)(CC(C(C)C)OCC)NCC1(F)CCN(C(C=CCC)=O)C1 c1(CC)ccc(CS(N2CCC(n3cccn3)C2)(=O)=O)cc1 Nc1cc(F)cnc1C(=O)NCCCC(=O)NCCCC(C1CC1)C1CC1 Cn1c(C2CC2C(C)(F)F)nc2ccc(Cl)cc12 N1(C(C(C=C)CC)=O)CCN2CCN(C(=O)CC3CCCC(C)O3)CC2C1 c1(CC(N2C(C)CC(NC(C3(C4CCCO4)CC3)=O)CC2)=O)nc2ncccn2n1 CCCC(CC(=O)N(CC(N)=O)CC(C)C)NC(c1cnn(CC)c1)=O c1(OC)cccc(Cl)c1CC(N1CCC(O)(CNC(C2CC=CCO2)=O)C1)=O N1(C(C2(CCCC)CC2)=O)CC(CC(c2csc(C)n2)N)OC(C)C1 c1(NC(C)=O)cccc(C(N2CC(O)(CNC(=O)CSc3nc[nH]n3)C2)=O)c1C C1(C)(C(=O)NCCC(C)NC(c2ccc(OC)o2)=O)CCC(=O)NC1 N1(C(C2(NC(C3CCC4(CC4)C3)=O)C(C)(C)C2)=O)CC2CC2C2CC12 c1(C(N2CCC(N(C)C(c3cnc(O)[nH]3)=O)C2)=O)cccc(OC(F)F)c1 C1(C(=O)NCCN(C(c2conc2-c2ccc(Cl)cc2)=O)CC)CCCN1N=O c1(NC(C2C3CC2N(C(C2C4C=CSC24)=O)C3)=O)cccc2c1OCC2 c1(C(N(CC(C)N(C)C(c2cccc(C(C)(C)C)c2)=O)C)=O)ccc(N)c(Cl)c1 N1(C(CSC(C)(C)C)=O)CCN(C(=O)CC2CC3CCC2C3)C(C2CCCC2)C1 c1(OC)ccc2ccccc2c1CN1CCC(CN(S(=O)(=O)CC#N)C)C1 C1(C(=O)OC)CC(n2cc(-c3ccc(I)cc3)nn2)CN1C(=O)CC1CSC1 N1(C(C)C(=O)NCC2CCCCC2)CCCCC12CCC2 C1(NC(C2(COC)CN(C(C3CCC3)=O)C2)=O)CC2(C1)CC(O)C2 C12(NC(CCCOCC)=O)CCCCCC1N(C(c1cnc(O)c(F)c1)=O)CC2 c1(C(N2CC(NC(c3cc(C)n(CCO)n3)=O)C(F)C2)=O)cccn2cnnc12 CCCCC(CC)CC(=O)NC1CCCC2CN(C(C3(C)CC(C#N)C3)=O)CC12 Cc1nn(C)c(N)c1C(N1CCC(C)C(CC(=O)NCC23CCC(CC2)C3)C1)=O N(C1CCc2ccccc21)Cc1ccccc1-c1ccnc2c1CCC2 c1(OC)cc(-c2cnc(NC(c3cnc(NC(C)=O)o3)=O)c(O)c2)ccc1OC C(=O)(C#CC1(C)CCCO1)NC1CCC(C)(C)CC1CNC(=O)Cc1cccs1 Cc1nc(C)c(CC(=O)NCC(C)CNC(=O)C=C2CCC(C)C2)c(O)n1 N1(C(=O)CC2CC3(CC3)CO2)CC2CCC1CN2C(=O)CNC(c1ccsc1)=O C1(C(=O)NC(C)C(C)(C)NC(=O)CCSC(F)(F)F)CN2CCN1CC2 N#Cc1cn[nH]c1C(=O)NCC1CN(C(C2CCCC3CC23)=O)C1 c1(-c2cn(CCCC(=O)NC3CCN(C4CCCC4)C3)nn2)cc(O)nc(O)n1 CCC(C(=O)NCC1CCN1C(=O)CCNC(c1cc(F)ccc1F)=O)C(C)O CC(C)CC(C(=O)N1CCC(CCO)(CCO)C1)N(C)C C1(NC(c2n(C(C)C)ncc2-c2ccccc2)=O)CCc2ccccc2OC1 C(=O)(CCCCCN(C(=O)COCCOC1CC1)CC)NC1(CC=C)CC1 C1(N(CCC#N)CCC)CCN(C(=O)C(C)Oc2ccccc2C)CC1 N1(C(c2nc(C)oc2C)=O)CCCC(C)(C)C1CNC(C1(C)CC1(F)F)=O c1(C(N2C3CCN(C(=O)NC(C(=O)OC)C)C3CC2)=O)c(O)ccc2nc[nH]c12 c1(NC(C(C)OC(=O)COc2nn(C)cc2Br)=O)ccc(F)cc1Br c1(C(C)(C)C)cccc(OCC=O)c1.N1CCCCC1CNCc1ccsc1 C1(N(C)C)CN(C(=O)C(C)(C2CC2)N(C(=O)Cc2cccnc2O)C)CC1O c1(C(=O)OC(C(C)C)C(=O)N2CCC(O)CC2)nnc2c(C(F)(F)F)cccn12 c1(C(=O)NC2CC(CO)N(C(c3ccc(Cl)s3)=O)C2)ccc2oc(=O)oc2c1 CCCC(CNC(=O)C(n1nccc1C)C)C(=O)N(C1CCC1)C1CC1 Cc1n[nH]c(C)c1C(C)NC(=O)CC1CCCC1NC(C1C=CC=CC=C1)=O C(=O)(C(O)C(CCC)NC(c1ccnc(O)c1)=O)NCCCCC#CC N1(C(C2(C)CCCN2C(c2sc(Br)cc2Br)=O)=O)CCOC(C#N)C1 c1(CC(=O)NCc2cc(C)c(Br)c(C)c2)cc(F)c(Cl)cc1[N+](=O)[O-] CC#CCC(C(=O)N1CCCC(O)C1)NC(=O)CN(C)CC C(=O)(C1=C2CCCN=C2NN1)NC1(C(C2CCN(C(C(C)(C)CF)=O)C2)(C)C)CC1 C1(N(C(C(C(C)C)NC(c2cc(C)n(C)c2)=O)=O)C)CC(C)CC(C)C1 C1(C(N(C2CN(C(c3cc(C)sc3)=O)C2)C)=O)CC(=O)N(c2cccc(Cl)c2)C1 n1(CCOC)ncc(C(=O)NC(C2CCN(C(C3CCCCO3)=O)C2)C)c1C C1(O)(CCNC(C2C(C)CCCC2)=O)CCN(C(=O)CC2CCN(C)C2=O)CC1 CC(C(=O)N(C(C)CNC(=O)CCc1ccc([N+](=O)[O-])cc1)C)C(C)S(C)(=O)=O CC(CF)C(=O)NCC(CO)NC(=O)CNC(C1CCC1)=O C=Cc1cncc(C(N2CCCCC2CCN(C)C(c2c(C)ncn2O)=O)=O)c1 CC1CCCN(C(C2COC(C)(C)C2)=O)C1CNC(c1c[nH][nH]c1=N)=O C1(NC(CCC(C)C)=O)CCN(CC(=O)N(C)C)CC1O C1(NC(C=CCNC(C(C)(C)Cl)=O)=O)CCC12CCCC2 c1(C(=O)NCC2CCCCN2Cc2cc(Cl)nc(Cl)c2)cc2cc(F)ccc2s1 C(CC(CC)C(=O)NCC(C)NC(=O)C=Cc1ncccc1C)=CC C1(C(=O)NC2(CC=C)CN(C(=O)CC3CCCCCC3)C2)CCS(=O)(=O)N1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CC(C)CN(C(=O)C(C)(CC)OC)CC1C S(=O)(=O)(c1cnccc1N1CCN(C(C2CC2C)=O)CC1)NCC(C(C)C)(C)C C1(CC)OC2(CCN(CC(N3CC4(CC(C(F)F)=NO4)C3)=O)CC2)NC1=O Cc1ccc(C(=O)N(CCC(=O)N(CCCC(C)(F)F)C)C)c(O)c1 N1(C(CC)=O)CCCCC1C1CCN(C(c2c(Br)cnn2C(C)C)=O)CC1 C12(C(N3C(C(C)(C)CN)CCCC3)=O)CCC(CC1)CO2 c1(N2CC3CC(NC(C4=C(C)CCCC4)=O)CC3C2)nc(Cl)nc2c1CCOC2 N1(C(COCCOCC)=O)CC(NC(=O)C(O)COC)CC1(C)C C1(C(N2CC(F)(CC)C2)=O)CC(NC(=O)CN2CCCNC2=O)CCO1 N1(C(C(CC)O)=O)CC(CNC(C2(c3ccno3)CCOCC2)=O)C(O)C1 N1(C(c2c(CNC(COCC)=O)c[nH]n2)=O)CCOCC1CC c1(SC)ccc(C(=O)NC2(C)CCN(C(=O)Cn3cncc3C)C2)cc1 N1(C(C(C=C)OC)=O)CCCC(C2CN(C(c3cnnn3C=C)=O)C2)C1 N1(C(C(CC)N(c2cccnc2Cl)CC)=O)CCC(C)C1CNC(OC)OCC.COC c1(C(=O)NCC(C)C(=O)NC2CCn3cnnc3C2)ccc2cc[nH]c2n1 Cc1cc(CNC(C2CCCC(NCc3cnc(F)c(C)c3)C2)=O)cc(C)c1 C1(NC(c2ccn(C(C)C)n2)=O)CC12CCN(C(c1cc(F)ccc1Cl)=O)C2 Cc1ccc2c(C(=O)NC3CCC(CNC(=O)C=C4CCSCC4)C3)c[nH]c2c1 c1(OCC)ccc(C(N2CCCC(CO)(CNC(C3(OC)CC3)=O)C2)=O)cn1 C(CCCCC(=O)NCC1CC=CCC1C(=O)N(C(C)COC)CC)OCC C1(C(=O)NCCCCN(C(=O)CCNC(=O)C=CCl)CC)CCC1C(C)(C)C c1(NC(C)CNC(C2(O)CCSCC2)=O)ncnc2c1COC2 C1(CNC(C(COC)O)=O)CN(C(=O)CCc2ccc(C)o2)CC(C)(C)C1 C(=O)(C1CCC(=O)c2ccccc21)N1C(CNC(c2[nH]cc(C)c2)=O)CCC1 C1(NC(c2n(CC)ccn2)=O)CN(C(=O)C=Cc2cc(C)no2)CC1C N1(C(C2(c3cccc(OC)c3)CC2)=O)CC2CC1CN2C(C1CCCN1N=O)=O CC1CC(CNC(C2CC2C)=O)CCN1C(c1ccoc1)=O c1(OC)n[nH]c(C(N2CC(CNC(C3(CCF)CC3)=O)(OC)C2)=O)c1Cl CN(NC(N)=O)S(=O)(=O)c1cc(CN(C)C)c(Cl)s1 C1(C)(NC(C2C(NC(C3C(OC)CC3)=O)CCO2)=O)CCCC1(F)F N1(C(c2nc(C(C)OC)sc2)=O)CC(CNC(C2C(C)(C)C2(C)C)=O)C2(CC2)C1 N1(C(C2(CSC)CC2)=O)CCN(C2CCCN(C(=O)C(C)O)C2)C(=O)C1 C1(CNC(c2cn(CCO)c(=O)nc2O)=O)CC2(CO1)CN(C(=O)C=C(Cl)Cl)C2 C1(CCC)CN(C(c2c(C)csc2C)=O)CC1C(=O)N(C)Cc1ccccn1 C1(CNC(CCC(=C)Br)=O)CC(C)(C)CCC1NC(=O)C=CC1CCC1 C1(CC(N2CC(N(C(=O)CSc3nnnn3C3CC3)C)C2)=O)CC2C=CC1C2 C(=O)(C1=NNC(=O)C1)NCC(CC(=O)N(CC(C)C)C1CC1)C1CCC1 C(c1cnccc1C)=CC(N1C(CN(C2OCCN(C(C)=O)C2)C)CCC1)=O C(CN=c1nc(CC2CCCC2)[nH]s1)(N(C)C(c1cc(Cl)nnc1O)=O)C1CC1 C12(NC(C(C)OC)=O)CC(CNC(=O)CC(C)C(F)F)(C1)OC21CCC1 N1(C(CCC(=O)OC)=O)CCCC(NC(c2nccnc2C(F)(F)F)=O)C(F)C1 N1(c2ncc(C)c(O)n2)CCC2(NC(=O)CCN3CCCS3(=O)=O)CCCC12 N1(C(C(CC=CCC)C)=O)CC2(CCC2)CC1C(=O)N(C)CCOC(C)=O N1(C(C(C)OCCCC)=O)CCCC(N(C(=O)Cc2ccns2)CC2CC2)C1 c1(OC)c(N2CCC(N(C(=O)C(C)OCCC(C)C)C)CC2)ncnc1C N1(C(CCN(C)CCO)=O)CCCCC(C2CN(C(=O)C(C)(O)C3CCC3)C2)C1 C1(CNC(c2ccc(NC)cn2)=O)CC(C(=O)NCc2nnc(O)o2)=NO1 CON(CCC(=O)O)C(=O)N1CCCC(COc2ccccc2)C1 c1(C(N2CC=CC(C(=O)NC3CC(=C)C3)C2)=O)ccc(F)c(O)c1 C1(C(=O)Nc2cnc(OCC)nc2)CCN(C(c2ccnc(Cl)c2C)=O)CC1O C1(c2ccc(CC)cc2)CN(C(=O)CO)CCN1C(C1CCOC1(C)C)=O c1(C(N(CCCNC(CSCCCC)=O)CCO)=O)cn(CCOC)nn1 N1(C(C(C)OCC=C)=O)CC(C2CCN(C(c3scc4c3OCCO4)=O)CC2)C1 N(C(=NCC1CCS(=O)(=O)N1)NCc1cnccc1Cl)C(C=C)C S(=O)(=O)(c1c[nH]c(C(=O)NC2CCN(C(=O)C(C3CC3)SC)C2)c1)NCC C1(NC(c2nc(CC)oc2)=O)CS(=O)(=O)CC1NC(c1cccc(C2CC2)n1)=O CN1CCN(C(=O)C(c2ccco2)NC(=O)Cn2cnnc2)CC1C1CC1 C(C(O)C(=O)NCC1CCCC1NC(=O)CCc1cnoc1)N(C)C c1(OC)cc([N+](=O)[O-])ccc1C(=O)N(CCCNC(=O)Cc1ccncc1Cl)C C1(C)(NC(CNS(C(C)CCN)(=O)=O)=O)C2CC3CC(C2)CC1C3 N1(C(C2(C)ON=C(C)C2)=O)CC2CCCC1C2CNC(=O)C(=O)NC1CC1 c1(CC)cc(C(=O)NCC2CCCCN2C)ccc1C c1(C(N2C(CN(C(=O)C(O)C(F)(F)F)C)CCCC2)=O)cc(F)ccc1Cl CCCCCCCC(=O)NCC1CCCN(C(=O)CCNC(C2CCC2)=O)CC1 C(C(=O)n1c2ccccc2c(=O)n1C)c1c(C)cc(N)cc1 C(=O)(C(C)(C)C(F)(F)F)NC(C1CCN(C(=O)Cc2cncnc2)CC1)(C)C Cc1noc2nc(C(N3CCCC(NC(=O)CC4(C)CC4(Cl)Cl)C3)=O)ccc12 c1(CC)sc(CNC(C2CCC(NC(=O)Nc3ccncc3)C2)=O)nc1C N1(C(=O)COc2ccccc2F)CC2CC1CN2C(C1CC2(CC2)CO1)=O CC1(C)CN(C(c2ccoc2CNC(=O)C(C2CCOCC2)O)=O)CC1CO CCCCC(CNC(c1c(C)noc1C)=O)NC(C1CCN(CC(F)F)CC1)=O C1(NC(CCNC(C(C)(C)C)=O)=O)CC2CCC(C1)N2C(C1CCCOCC1)=O CC(C(=O)N1CCOC(CN(C)C(c2cc(O)nc(O)c2)=O)C1)C(F)(F)C(F)F N1(C(CCN2CC(=O)NCC2)=O)CCCC2C1CCCN2C(c1coc(Cl)c1)=O c1(C(N(C2CCN(CC(=O)N(CC=C)CC=C)C2)CC)=O)ccnc(F)c1OC C1(F)(CNC(=O)NC(C=C)(C)C)CC(O)C1 C(=O)(CCP(C)(C)=O)NC1(C(=O)NC(C2CCCCC2)C)C(C)CCC1 N1(C(C(C)(CO)OC)=O)CCC(CCNC(=O)C#CC2CCC2)C(F)(F)C1 CC(C)(C)C(C)(C)C(=O)N1CCCC(N(C(=O)C2=COCC2)CCO)C1 Cc1cc(C(C)(C)NC2(C3(NC(=O)OC(C)(C)C)CC3)CCCC2)nc(N(C)C)n1 n1(CC)ccc(C(=O)NC(C)C(=O)NCCC(N)=O)n1 c1(C(=O)NCC2(C)CC(NC(C34CC(F)C3C4)=O)C2)cc2cnccc2o1 C1(C(N2CCC(C(C)NC(=O)COCP(C)(C)=O)C2)=O)(CC)CCC(O)CC1 c1(C(N2CCC(NC(CC(=O)OC)=O)C2)=O)c(C)cnn1Cc1ccccc1 c1(NC(C2CCC23CC3)=O)cccc(Cl)c1N1CCCCC1 c1(C(c2n(CC)nnn2)NCC2SCCS2)cccnc1Cl c1(C(N(C(C)CN(C(=O)CCCc2nc(C3CC3)no2)C)C)=O)ncc[nH]c1=O C1(C(=O)NCC(C)(F)CNC(=O)CC2CCC2)CCn2nnnc2C1 CCCC(C(=O)NC1(CO)CN(C(=O)C(C)c2cc[nH]n2)C1)OCC C1(C(=O)NCC(CNC(c2c(NC)scn2)=O)O)CCCN1C=O c1(C(C)C)cc(C(=O)NC(C)CNC(=O)COCCN(C)C)on1 c1(C(=O)NCC2(C(=O)NOCC(F)(F)F)CC(=C)C2)cc(CO)c(C)o1 C1(C(=O)OC)(NS(=O)(=O)c2cccs2)COC(C)(C)C1 N1(C(c2n(C)ccc2)=O)CCCC2CN(C(C3(c4cccs4)CC3)=O)CCCC12 CC(C)C(F)(F)CC(=O)N1CC(NC(c2c(O)cccc2Cl)=O)C(C)C1 C#CC1CCC(C(=O)NC2CCN(C(c3c[nH]nc3OC)=O)C2C)CC1 c1(OCC=C)ccccc1C(N1CCCC(NC(=O)C(C)CO)C1)=O C1(N(C)C)CN(C(=O)CC2CC3(CC3)CO2)CC1CNC(=O)CC1CC1 C(C)(CO)(C(=O)NCc1ccc(Cl)nc1)NC(C(C)O)=O CCC(C)C(C)C(=O)N(CCCCNC(c1cc2n(c1)CCC2)=O)C C1(C(=O)NCC2N(C(c3cc(SC)oc3C)=O)CCCC2)C2(CCC2)C12CCC2 C1(NC(C(CC(C)C)C)=O)CCS(=O)(=O)C12CN(C(=O)Cc1c[nH]ccc1=O)C2 CC(C)C(CNC(c1ccnnc1O)=O)C(=O)NC(C(F)F)C(C)(C)C c1(CNC2CC(C(=O)Nc3c(C(=O)OC)ccnc3Cl)C2)cc(Cl)c(Cl)cc1F CC(C)CCCC(=O)N(CC(O)CNC(C1CC2C(C1)C2(C)C)=O)C C=CCC(CC(F)F)C(=O)NC1CN(C(=O)C(C)NC(=O)NC)C2(CCOC2)C1 c1(C(=O)NC2CC(C)(NC(c3ccc(SC)o3)=O)C2)cc(C2(Cl)CC2)n(C)n1 C1(C(F)(F)F)(Nc2c(N)cncc2Br)CCCN(C(=O)OC(C)(C)C)C1 C1(NC(c2c(C)n(C(C)C)cc2)=O)CC2CN(C(=O)C(=O)CCC(C)C)CC2C1 C1(C)(CC)CCN(C(C2CN(C(=O)C(CCN(C)C)N(C)C)CC2C)=O)C1 N1(C(C(COCC)C)=O)CCC2(CC1)CC(NC(=O)CC(C)CC(C)(C)C)C2 CC(C)C(C(=O)N1CCC(=CCNC(=O)CC2CCCCC2O)CC1)NC(N)=O C#CC1(C(N2CC3C(NC(=O)CSc4nc[nH]n4)C3C2)=O)CCCC1 Cc1cc2[nH]c(C(N3CC(O)(CNC(C4CC5CCCC(C4)C5)=O)C3)=O)cc2o1 C1(NC(CCCC=C)=O)CN(C(c2c[nH]nc2-c2cnn(C)c2)=O)CC12CC2 c1(CN2CCN(C(C(c3ccc(C)cc3)=O)=O)CC2C)cc(F)c(C)c(Br)c1 C1(Oc2ccc(F)nc2)CS(=O)(=O)CC1N1CCCC1.CC1C(=O)NCCN(CCO)C1 C=CCCCCCCC(=O)NC1C=CCCC1C(N1C(CO)CC1C)=O O(N(Cc1ccccc1)C(=O)c1c[nH]nc1-c1ccc(Br)s1)CC c1(C(=O)NCC(C(=O)NC2C(O)CCC(C)C2)(C)C)cc2cc[nH]c2cn1 C1(C(=O)NC(C2(O)CN(C(CCOC(C)C)=O)C2)C)CCC(F)(F)CC1 N1(C(C=Cc2cn(C)nn2)=O)CCCC(C)(CNC(c2ccc(CO)nc2)=O)C1 c1(C(N2C(CNC(c3scc(C)c3)=O)COCC2)=O)cnc2cc(C)[nH]c2c1 C(CC(C)C(=O)N1CCC(NC(c2c[nH]nc2C2CCCCC2)=O)CC1)OC CC(C)CC(C)C(=O)NCC1CC(F)(F)CN1C(C1CCCSC1)=O C1(NC(c2cc(CC)no2)=O)C=CCC(C(=O)NC2CC2O)C1 C12(CNC(C=C(CC)C)=O)CCCC(CN1C(=O)CCC=CBr)C2 c1(C(CC)C(=O)N(C)CCNC(=O)CC2(C)CC2(Cl)Cl)ccc(OC)cc1 C(C(C(C)C(C)C)NC(C1(C(=O)NC2CC2)CCC1)=O)NC(CC)=O Cc1[nH]nc(C(N2CCC(C)N(C(=O)Cc3ncn(C)c3C)CC2)=O)c1[N+](=O)[O-] N1(C(C(C=C)C)=O)CCC(CNC(=O)CSCC(F)(F)F)C(F)(F)CC1 Cc1ccc(C(N2CC(F)(CNC(c3ccn4ncnc4c3)=O)C2)=O)c(=O)n1C C1(C(=O)NC(C#C)C)CCCN1C(=O)C=CC1CCCC1 C1(CNC(Cc2ccc(C)s2)=O)C2CN(C(=O)Cc3ccccc3)CC12 c1(CNC(C(=O)NCC2C(C)OCC2)=O)ccc2c(c1)OCCC2 c1(NC(C2(CCC)CC2)=O)cc(Cl)c(C(F)F)cc1F N1(C(C2CC(=O)C2)=O)CC2Oc3cccc(NC(=O)CSC(F)(F)F)c3C2C1 C(=O)(C1=COCCC1)N1CC(CCCCNCC2CCC(NS(C)(=O)=O)CC2)C1 C1(CCNC(C(CC)O)=O)CCN(C(=O)Cn2cc(C3CC3)cn2)CCC1(F)F N1(C(c2cnc(CC(C)C)s2)=O)CN(C)C(=O)C1C C1(NC(c2nnnn2C)CCSc2ncn(C)c2Cl)CCCC(C)(C)C1 c1(OC(C)C)ccc(C(C(C)O)NC2CCC(c3nn[nH]n3)C2)cc1 Cc1ccc(OCC(=O)N(C)CC2(NC(C3CCC(=O)CC3C)=O)CC2)cc1C c1(C(C)NC(Cc2ccccc2)CCO)cc(Br)cnc1Br c1(CC)cc(C(=O)NC2CCN(C(c3cn[nH]c3)=O)CC2C)c(C)nn1 N1(C(C2CC(C)N(C)C2)=O)CCCCC(C(=O)N(C)CCOC2CC2)C1 C1(C(=O)NC(COCC)C(=O)NCC2CCCC23CCC3)CC(=O)N(OC)C1 C=CC1(C(N2CC(O)(C(F)(F)F)C2)=O)CCN(C(=O)CC#N)C1 CCC(CC)C(C)C(=O)N1CC(C(N2CCC(C)OC(C)C2)=O)CCC1(C)C c1(C(=O)NC(C(C)C)CNC(=O)CC(C)(C)c2cccs2)cc(F)cc(N)c1F c1(C(=O)NCC(CC=C)NC(C2(C)CCN(C)CC2)=O)cc(S(C)(=O)=O)cs1 C1(C(=O)NC(C)CN2CCOCC2)C=CCCN1C(c1ns[nH]c1=O)=O N1(C(C2(C)CC(F)C2)=O)CCC2(CC(NC(c3c[nH]nc3C3CCCO3)=O)C2)C1 C=C=C(C)CC(=O)NC(C1(O)CCN(C(=O)CN2CSCCSC2)C1)C C(=O)(C(O)C(F)(F)F)N1CCC(C(C)(C)NC(C2CC2C2CC2)=O)C1 c1(-n2cc(CN3C(COCC)CCC3)nn2)cnc(C(F)(F)F)cc1C Cc1c(Cl)c(C(N2CCN(C(C3CC(=O)N(C4CC4)C3)=O)C(C)C2)=O)nn1C c1(C(CN(C)C(=O)Nc2cnn(C3CCNC3=O)c2)O)cccc(C#N)c1 CC(CC(=O)NC1(CC(N)=O)CCN(C(=O)CC(F)F)CC1)CC(C)(C)C C1(NC(c2cnc(CC)[nH]2)=O)CCCN(C(=O)C(C)CSC)CCC1 c1(C(c2n(CCC)nnn2)NCC(C)C2CCC2)c[nH]ccc1=O C1(NC(c2ccc(OCCCC)cc2)=O)CCC2CN(C(C)C(=O)NC)CC2C1 Brc1ccc2nnc(CNCC34CCCNC3COC4)n2c1 CCCC(C)CC(=O)NCC(C)(C1CC1)NC(=O)CN(C)Cc1nnc(C)n1C c1(C(=O)NCCF)ccc2ccc(C3=CCOC3)cc2n1 C1(F)(C(=O)NCC2CC3CN(C(C(C)=C(C)C)=O)CC32)CS(=O)(=O)CC12CCC2 CC(=O)CCN=C(NCC(C)C)NC1CCC(C(N)=O)C1 C(CC(C)C)(C(=O)NC)NOC(CC1(c2ncco2)CCC1)OCC C1(CNC(c2c(F)cccc2F)=O)CN(C(c2ccccn2)=O)CC12CCC2 CC1(C)COC(C(N2CC3C(C(=O)Nc4cncc(Cl)c4)C3C2)=O)C1 c1(CC(=O)NCCC2CCCN(CC(=O)NC(=O)NC)C2)cccc(Cl)c1Cl C1(NC(C=CCC)=O)CN(C(c2cccc(C)n2)=O)CC1C1CC1 C1(CNC(C2(CC=C)CCOC2)=O)CC2(CO1)CN(C(C1(CO)CCCC1)=O)C2 N1(C(C(Cc2c(C)n[nH]c2C)C)=O)C2CCC1CC(NC(=O)CC1CSC1)C2 C(=O)(CCCCN=[N+]=[N-])N(C(C)(C)CC(=O)NCC(c1ccco1)O)C c1(C(N2CCC(c3nc(C)on3)C2)=O)cc2ccccn2n1 N1(CCOC)CCC(c2nnnn2C(C)C)(NCC2CCCSCC2)C1 C=C(CNC(=O)NC(c1ccccc1F)CF)C(F)(F)F C12(NC(CC(CC)O)=O)CCC(CN(C(C3CC3c3ccccn3)=O)C1)C2 C1(CC)C(C(N2CCC(O)CC2)=O)CCN1C(C1CCSCC1)=O N1(C(C(CC)CC)=O)CCN(C(=O)C(F)n2cccn2)CC1c1ccccc1Cl N1(C(COc2cc(C#C)cc(Br)c2)=O)CCOC2(C1)CN(C(C1CC1C)=O)C2 N(C1c2ccccc2CC1NC(=O)C(C)(F)C(F)(F)F)C(C(C(C)C)(C)C)=O C(CCC(C(=O)N1CCCC(O)CC1)NC(=O)CC(C)(F)F)OC N1(C(COCP(C)(C)=O)=O)CC(CNC(=O)CC2CC(=O)C2)CC12CCC2 C1(NC(c2nc(C)n(C)n2)=O)CCCCC12CCCN(C(=O)CC(C)F)C2 CC(CN(C)C)CC(=O)N(C)CCC1CCN(C(=O)C(F)(F)C2CCCC2)CC1 CCCCCC(C)CC(=O)N(CCC)CCNC(=O)CCn1cccn1 CC(=NOCC#N)C(=O)NC(C(=O)N1CCC(OC)CC1)C(C)C c1(C(=O)NC(c2ccns2)C)ccc(CNC(c2cnsc2)=O)nc1 c1(N2CCC(c3ccccc3)(NC(CC)=O)C2)cc(C)nc2ccnn12 CC1(CNC(=O)CCNC2COC2)CCN(C(=O)CCc2cnoc2)CC1 C(CCN(C(=O)C=Cc1ccoc1)C)(C(C)C)NC(C(COCC)C)=O c1(C(=O)Nc2cc(C(=O)OC)ncc2Br)cnc2onc(C)c2c1 c1(C(N2CC3C(CNC(c4c(C)noc4)=O)C3C2)=O)c2n(c(=O)n1C)CCCC2 N1(C(C(=O)N(C(C)C)C)C)CCCCC(NC(c2ccc(=O)n(C(C)C)c2)=O)C1 C1(NC(c2cc(COC)sc2)=O)CC2CCC1CN(C(C1CNC(=O)C1)=O)C2 N1(CC(CC)CC)CCC(C(C)NC(=O)CCCc2ccccn2)CC1 C=CCC(CNC(C1CCCCC1)=O)C(=O)N(C(C)C(C)(C)C)C C(S(C)(=O)=O)C1(CC(=O)NN(CCCNC(CSCCC#N)=O)C2CC2)CC1 N1(C(c2cccc(OC)c2)=O)CC2(CCCC2NC(=O)C(C)CC2CCC2)C1 N1(C(C=COCC)=O)CC2(NC(C3CC4(CCCCO4)C3)=O)CCCC2(F)C1 c1(C(N2C(C)(COC)CC2)=O)cc2c(Br)cc(F)cc2[nH]1 C(CC(C(=O)NCC(C)(C)C(N)=O)NC(=O)C(CCC1CC1)OC)OC C1(CNC(C(C(=O)OCC)F)=O)CC2CCC(C1)N2C(=O)C(C1CCOCC1)O C1(C(N(C)CC2CCN(C(c3c(C)noc3N)=O)C2)=O)OCC2CCCC12 n1(CC)cc(Cl)c(C(=O)NC(C2CN(C(c3c(Cl)cnn3C)=O)C2)C)n1 C(=O)(C(C)N=[N+]=[N-])N(CC(=O)NCC=C=C)CCOC c1(C(N(CCNC(c2ccc(CN(C)C)o2)=O)CC)=O)cc(C)cc(Br)c1 Cc1ccc(C(N)CC(=O)NC2(CO)CCOC2)cc1 CCC(C)(C)C(C(=O)N1CCN(C(=O)C(=Cc2ccncc2)C)CC1)OC c1(C(=O)NC(C)CCCNC(=O)C(=Cc2cccnc2)F)cccn(C)c1=O c1(CC)nnsc1C(N1CCC1CNC(=O)CC1CCNC1=O)=O c1(C(C)C)ccc(N)c(C(N2CCC(NC(C3(F)CC4(CCC4)C3)=O)C2)=O)c1 CCC(C)C(C)NS(=O)(=O)CCC1CN(C(=O)OC(C)(C)C)C1 N1(C(=O)OC)CCC(N)CC1.C(=O)(C(C(C)C)NC(=O)C1CC1)C(=O)C(C)N c1(OC)ncc(C(=O)NC23CCC(NC(c4cnns4)=O)(CC2)C3)cc1C c1(C(N2CC(CC)C(C(=O)NC3(COC)CC3)C2)=O)nc(C)ccc1C C=CC1(C(=O)NCC2(C)CCN(C(c3coc(CO)c3)=O)C2)CCCC1 CC(C)C(C(C)NC(C1(F)CCCCC1)=O)NC(c1coc(CO)c1)=O c1(C(N2C3C(NC(c4cncc(C)c4)=O)C(C3)C2)=O)cc(Cl)ccc1Br CCCCC(O)C(C)C(=O)N1CC(CC(=O)NC2CC=C(C(C)C)CC2)CC1C C(=O)(CCCCC(N)=O)N1CCC=C(CNC(c2c(C)ccnn2)=O)C1 C1(CNC(c2ccc(CC)cn2)=O)COCCN(C(C)C(=O)Nc2nncs2)C1 CC1=CCCN(C(=NCCC(C)(C)C)NCCN(CC(F)(F)F)C)C1 N1(C=O)CCCCCC1CNC(C1CC(Cl)(Cl)C1)=O.C1(N(C)C)(O)COC1 N1(C(CCCCCC#N)=O)CCC2CCN(C(c3ccnc4[nH]nnc34)=O)C2C1 N1(C(c2c(C)nc(C)s2)=O)CCCC2(CCC2NC(c2csc(O)n2)=O)C1 Cc1ccncc1CC(N1CCC(O)(CNC(c2coc(C(C)(C)C)n2)=O)C1)=O C(CC(=O)NC1CN(C(C)C)C1)(C(F)(F)F)NC(CCC)=O CCC(C(=O)N1CC(O)(CNC(C2CC2C)=O)C1)NC(N)=O C1(NC(C(C)NC(CC)=O)=O)C2CC3CN(C(=O)C(C)OC4CCCCC4)C1C3C2 C1(OC)CN(C(c2ccc(C(F)F)o2)=O)CCC1NC(=O)CC(C)c1ccco1 C1(NC(Cc2ccc(C)s2)=O)(CO)CCCN(C(=O)CSc2ccccc2O)C1 O=C1CCN(Cc2ccoc2)C(=O)N1CC1CCC2(CO1)CC(OCC(F)F)C2 CC(O)CCCCCC(=O)NC(C)CNC(=O)CCC1(C)CC1 C1(C(N(CC(C)(C)CNC(=O)CCn2cc(C)cn2)CC)=O)CCC2CC2CC1 CC1CCN(C(=O)C(F)(F)CC2CC2)CCN1C(=O)C(C)OCC1CC1 Cc1[nH]c2ccc(Br)cc2c1C(=O)CN1CCCCC(C)C1 Cc1cc(F)ccc1C(O)C(=O)NCC(C)(C)NC(=O)C=CC1CC1 n1(CC(=O)N(C2CCCN(C(=O)C=CI)CC2)C)ccc([N+](=O)[O-])n1 C1(C(=O)NCc2ccc(CC)o2)CC(O)CN1C(c1ccn(C)n1)=O CC(=O)CC(C)(C)C(=O)NCc1cnn(C)c1C(N1CCC(N2CCCC2)C1)=O CC(C(=O)NOC(C)(C)CO)C1CCN(C(=O)CCc2ccncc2)CC1 N1(C(COC2CC(NC(C(C(C)C)F)=O)C2)=O)CCn2ccnc21 CC1CCNCCC1N(C(=O)Cc1ccn(C)n1)Cc1cocn1 C(=O)(C(C(C)(C)C)n1ccnn1)NCCC(C)N(C(C=CC(C)(C)SC)=O)C Cc1cn(C)nc1C(=O)N(CC(=O)NC1CC(C(N)=O)C1)C1CCC1 c1(C(=O)NC(CN(C(=O)CSCC2CCCO2)C)(C)C)cccc2c1C(C#N)C2 C1(CNC(c2c(C)nc(C)o2)=O)CN(C(C23C(=O)C4CC2C3C4)=O)CC12CCC2 CC(C)C(CCN(C)C(C1CCC(F)C1)=O)NC(=O)CSC1CC1 N1(C(CC)C(N)=O)CC2CCC(NC(c3cc4n(n3)CCCC4)=O)CC2C1 CC1=C(C(=O)N2CC3CC2CN(C(c2ccc4cccnn24)=O)C3)CCCO1 CCCC(C)(CCC)C(=O)NC1C=CCC(C(=O)NOCCCC2CC2)C1 c1(C(=O)NCC2CN(C(COC)=O)CC23CC3)ccc2cc(F)ccc2n1 N1(C(C2(C)CNC(=O)C2)=O)Cc2nccn2CC(NC(c2ccnc(S)c2)=O)C1 C1(C(C)NC(N)=O)CCCN1C(=O)C(C1CCCCC1)C CC1(C)CCC(C)(C(N2CC3CCC3(NC(c3csc(C(F)F)n3)=O)C2)=O)CC1 N1(C(C=CC=CC)=O)CCOC(C)(CNC(=O)C(C)Oc2ccc(Cl)cc2C)C1 Cc1cc(C(=O)NCC(C)N(C(=O)CC2CCNC(=O)C2)C)c(Br)c(C)c1 c1(N(C)C)cc(C(=O)NC2CC2C(=O)NC2CC(O)C2)nc2ccccc12 C1(NC(c2csc(Br)n2)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CCC1CO Cc1ccc(C(=O)NC2CCC(C(=O)NCC(N)=O)C2)o1 c12cccc(c1F)NC(=O)C(=O)N2.C1(C(C)C)CC(C(=O)N(C)C)CCO1 C(c1cc2ccccc2o1)=COCC1(c2cn(CCCC(=O)NCC)nn2)CC1 c1(C(=O)NCC2CCCN(c3cc(SC)nc(C)n3)C2)cc2nc(C)ccc2o1 c1(CNC(C2N(C(C3N(C)CCOC3)=O)CCC2)=O)ccc(F)cc1F c1(CC)cccc(F)c1C(=O)NC1CCN(C(=O)C(=O)C(C)(C)C)C1 Cn1nccc1C(F)=CC(N1CCC(NC(=O)Cc2ccccc2)C1)=O C1(OCC)CC2CN(C(=O)C(C3CCN(C(=O)Cc4nccn4C)C3)C)CC12 c1(C(=O)NCCCC(C)NC(c2cccc(C(F)(F)F)n2)=O)csc2cncn12 c1(C(N2CC(NC(C3(O)CC3)=O)C3CCCC3C2)=O)cc2ccc(Cl)cc2o1 c1(C(=O)NCCC2N(C(C(CC)CC)=O)CCC2)cccc2cncn12 O=C1CC(C(=O)NC2CC3CC(NC(C4CC5(CSC5)C4)=O)CC23)CC(=O)N1 N1(C(c2c(CC)ncs2)=O)CCCCC(CNC(=O)Cc2conc2C)C1 C1(C(=O)NC(C)C(C)(C)NC(c2cc(C3CCC3)[nH]n2)=O)CC2COCC2C1 C=C(CNC(=O)C(O)C1CCCC1)CCNC(c1csc(C(C)C)n1)=O N1(C(c2cc(CC)c(F)cc2)=O)CCC2CCC(C1)N2C(=O)Cc1ccoc1 CC1(C)CC(NC(C2C3CCCCC23)=O)CN1C(c1csc(C#N)c1)=O c1(N2CC(NC(CCC(=O)N(C)C)=O)CC(C)(C)C2)nccc(S(C)(=O)=O)n1 Cc1c(C(=O)OCc2cn(Cc3nnn(C)n3)nn2)cc(F)cc1Br c1(C(N2CC3CC2CN(C(C2(CC)COC2)=O)C3)=O)cc([N+](=O)[O-])ccc1OCC N1(C(C23CC(OC)C2C3)=O)CCN(C(c2cnc(N)c(N)c2)=O)CC1CO N1(C(CC(COC)(C)O)=O)CC2CCC1C1CN(C(c3nc(C)no3)=O)CC21 C1(CNC(C2CCC(C)(C)C2)=O)COCCN(C(c2ccccc2O)=O)C1 n1(CC(=O)NCC2CCN2C(C2(C3CCC3)CC2)=O)sc(=O)c2ccccc12 N1(C(c2c(Cl)cn(C)n2)=O)CCC2CN(C(=O)CCc3cc(Cl)no3)CCC12 c1(C(N(C2CC2)CC2CCN(C(C=CCN(C)CC)=O)C2)=O)cccc(F)c1C C1(CC)CN(C(=O)Cc2c(F)cccc2F)CCC1NC(=O)Cc1[nH]cnc1C CC1CC(NC(c2cc(C3CC3)nc(O)c2)=O)CN(C(=O)CC2CCC(=O)O2)C1 N1(C(C(N2CCOCC2)C)=O)CCC(NC(=O)CCc2cc(Cl)no2)CC1C C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)NCC1C(NC(=O)CC2CCOCC2)CC1 C(=O)(C(C)(C)N=[N+]=[N-])NC(c1ccccc1)C(=O)NCC1CCC(C)CC1 C(=O)(C(O)Cc1ccccc1)NCCCN(CC(CC)Oc1ccccc1)C C1(C)(CC(N2CC(O)(CN(C(=O)CCC3CCCO3)C)C2)=O)CC(F)(F)C1 N1(C(CC2CC(SC)C2)=O)CC(C)CN(C(=O)Cc2c(C)cccc2F)CC1C N1(S(C2C(C)C2)(=O)=O)CCCCC(N2CCCC2)C1 n1(CCC(=O)NC(CCC)CCCNC(=O)CC2CC2)cc(C#N)c(O)nc1=O C12(CNC(CN(C)C)=O)CCCC1N(C(c1cc([N+](=O)[O-])ccc1O)=O)CCC2 N1(C(CNC(C)=O)=O)CCC(C2CC2)C1CNC(c1ccc([N+](=O)[O-])[nH]1)=O C(=O)(CCCCC#N)N1CCC(C(C)(C)NC(=O)CC2CC3(CCC3)C2)C1 S(=O)(=O)(c1ccc2nc(N(CC(C)CC)C)sc2c1)NC1(CC=C)CC1 C1(C)(CN(C)C(C2CC(=C3CC3)C2)=O)CCCC1NC(c1cc(C(F)F)cs1)=O c1(C(=O)NCC(CC)(C)NC(=O)CN2CSCC2=O)cnn2ncccc12 C(N=c1nc(O)c2ccc(Cl)cc2[nH]1)C1CCC(NC(c2n(C)cc(Cl)c2)=O)C1 NS(=O)(=O)c1cc(C(=O)NC2CN(C(=O)C=CC3CCOC3)CC2C2CC2)co1 N1(C(CCN(C(C2CC2Cl)=O)CC)=O)CCc2cncnc21 C(=O)(C(C)(O)C(C)c1ccccc1)N(CCOCCNC(c1c(C)scc1)=O)C N1(C(c2cc(CC)nn2C)=O)CCC(C2CC2)(CNC(C2CCCOC2C)=O)C1 c1(CC(C)Sc2nccc(COC)n2)c(Cl)cccc1Cl N1(C(C2CC(=O)N2)=O)CCC2C(C1)OCCN2C(c1cnc2ccc(Br)cn12)=O C(=O)(C1CCCc2ncnn21)N1CC(C)N(C(C2(C)C=CCC2)=O)CC1 c1(C(N2C3CN(C(C(C)C#N)=O)C(C3)CC2)=O)ccc2c(c1)CCNC2=O c1(C(C)C)ncc2c(n1)CCN(N1CCC(Cc3cccc(F)c3)C1)C2 c1(CC)c(C(=O)NC2CCN(C(c3ccccc3SC)=O)C2(C)C)cccc1F C1(F)(CNC(C(N2CC(C)C2)C)=O)CCN(C(=O)CCc2cccs2)C1 C1(CC(=O)N(C)CC2CCN(C(c3cnnc(Cl)c3)=O)CC2)CCCC2(CC2)C1 c1(SC)ccc(C=CC(=O)NCC2(F)CN(C(C3CC4CCC(C3)O4)=O)C2)cc1 S(=O)(=O)(c1ccc(CC(N2CC(NC(=O)CC3CCC3(C)C)C(O)C2)=O)s1)NC C(CC(C)(CC)NC(C12CCC(C1)C2)=O)NC(C(C)OCC#C)=O c1(C(N2CC=CC(NC(C3(CO)CC3)=O)C2)=O)cc2c(=O)cc[nH]c2s1 n1(CC)cc(C(=O)NCC2CC(NC(=O)OC(C)(C)C)C(OC)C2)c(C)n1 C(C1CCCCC1)=CC(=O)NC(c1ccnn1C)C(=O)NCC(CC)O c1(OC)ccc(Br)c(CNCC2(C(N3CCC(C#N)CC3)=O)CC2)c1O C(=O)(CC(O)CN(C)C)NCC(N(C(CC(=C)C)=O)C)C1CC1 c1(C(N2C(C(C)NC(C3(F)CCCC3)=O)CCCC2)=O)cnc2c(c1)COC2 C(C(C)(CC)C(N)=O)NC(C(CCOCCO)NC(COCCC=C)=O)=O C1(C(=O)NCCCOC=C)CCC(C(C)C)N1C(=O)C(C)COC c1(CC)oc2ccccc2c1C(=O)NC1CC1CNC(c1snc(O)c1Cl)=O S(=O)(=O)(c1ccc(Cl)s1)NC(C(CC)NCCNCCc1cnc(CC)s1)=O c1(C(N(CC(C)CNC(c2cc(Br)c[nH]2)=O)C)=O)cc(Cl)ncc1Cl CC1CCN(C(C2CCC3(CC3)N2C(=O)C(O)CN(C)C)=O)CC1(C)C C(=O)(C(C(C)(C)C)OC)N(CC(C)NC(c1cnc(C(=O)OC)s1)=O)C C(CC(=O)NCC(CC)CO)=CCC.C1CC(=O)N1 N1(C(CC2(C)N(C(CCC#CC)=O)CC2)=O)CCc2ccc(O)cc21 C1(NC(CCc2cnn(C)n2)=O)CN(C(C2COC3COCC23)=O)CC(C)(C)C1 c1(-n2c(C3CCN3)nnn2)ccccc1Cl.C(C1CC1)=CC.CCS c1(C(=O)NCC2C3CN(C(C(CC)N(C)C)=O)C(C3)C2)c(C)cc(C)nc1C CCC(CC)CCC(=O)N1CC(C(=O)NCCSC2(CCOC)CC2)(SC)C1 c1(C(=O)NCC2(NC(Cc3c(C)nn(C)c3)=O)CC2)ccc2ccn(C)c2c1 CCC(C)C(C)CNC(=O)C(c1ccoc1)NC(c1ncccc1Cl)=O C1(C(=O)NCCCC(=O)Nc2cnn(C)c2)(CC)CCCCO1 CC1(C)CC(CNC(C2CCCO2)=O)CN(C(c2cc(C(C)(C)C)on2)=O)C1 C1(CNC(CCNC(C)=O)=O)CN(C(c2ccnc(C(N)=O)c2)=O)CCC1(C)C C1(N(C)C)(C(=O)NC2CCCC2NC(=O)COCc2nc[nH]n2)CCCSC1 C(C)(C)(C(=O)N1CCC(OCCNC(C2CC2c2cnn(C)c2)=O)C1)N(C)C c1(C(N2C(CNC(C(C)C#N)=O)C3CCC2C3)=O)ccc2ncccc2c1Cl c1(-n2ncc(C)c2)cccc(NC(C)CC2CN(C(=O)OC(C)(C)C)C2)c1 C1(CC(=O)NCCOC2CN(C(CSC)=O)C2)CC1C1CC1 C1(CNC(C2CN(C)C(=O)C2)=O)CC12CCN(C(c1scnc1C(F)F)=O)CC2 C(CCCCC(=O)NC)NC(Cc1c(CC)ccs1)=O N1(C(C2C(OC)C2)=O)C2CCCC1CN(C(=O)Cn1cc(C)c(O)nc1=O)CC2 C#CCCCC(C)C(=O)NCC(CC(C)C)NC(=O)Cc1nocc1C c1(C(=O)NC2(C)CCCN(C(CC3(C)CCOCC3)=O)C2)cnc2c(c1)COC2 c1(C(=O)NCC=CCNC(Cc2c(C)cc(C)s2)=O)ccc2ccccc2n1 N1(C(c2cnccc2Br)=O)CCC2(CCCN2C(=O)CC2COCCO2)C1 Cc1cnc(NC2CCN(C(C)C)C2)c(S(=O)(=O)NC2CN(S(=O)(=O)N(C)C)C2)c1 c1(C(N(CC(=O)N2CC(NC(=O)OC)C2)CCC)=O)ccc(C(C)=O)[nH]1 Cc1cc(C(=O)NC2CC(CNC(c3ccc(C#N)n3C)=O)C2(C)C)ccc1F CC(C)(O)C#CC(=O)NC1CCC(CCC(=O)NCC2CSCCO2)C1 CC1CC=CCC1C(N1CCCCC1C1CCN(C(c2cc(Cl)cn2C)=O)C1)=O c1(CC)cc(C(=O)NC(C2(CNC(=O)CCC3CCOCC3)CC2)C)c(C)o1 C12CC3(CN3C1=O)C2.c1(C(=O)OC(C)(C)C)ccncc1NC(C(=O)OC)C CCCS(=O)(=O)C(C)C(=O)N1CC(NC(c2ccsc2COC)=O)C2(CCC2)C1 c1(C(N2C(C(C)(C)C(=O)NCC(C)(O)C3CC3)CCC2)=O)c[nH]c2ncccc12 C1(C(=O)NCC2C(NC(C3CN(C)C(=O)N3)=O)CCC2)OCCCC1(C)C N1(C(C2C(C)C2)=O)CC2(CCN2C(=O)Cc2cccc(OC(F)(F)F)c2)C1 CN(C)NC(=O)CCC(=O)NC1CC(NC(C2CCCC(C(N)=O)C2)=O)C1 c1(C(=O)NC(CCCC)CC)cccc(S(=O)(=O)N(C(C)C)Cc2ccco2)c1 c1(C(=O)NC(CNC(C(C)NC(C)=O)=O)C(C)(C)C)ncc(C2CC2)cc1C N1(C(C(CCCC)=O)=O)C2CCC1CC(NC(c1ncc[nH]c1=O)=O)C2 Cc1cc(C(=O)NCCN(C(=O)C(C)CC2CCC2)CC(C)O)c(C)n1C C(C(C)(C)CC(=O)NOCC1CCOC1)NC(c1nc(C)oc1C)=O c1(SCC(=O)NCC(C)CN(C)C(C2C3CCC2CC3)=O)ccccc1F c1(C(=O)NC2CC(CNC(CCNC(C)=O)=O)C2)cccc(C)c1O N1(C(C(CC)O)=O)CCCC(O)(CN(C)C(c2cn(C)nc2C(C)(F)F)=O)C1 CN1CCCCC(C(=O)NCC(C)(C)CNC(=O)CCCc2cccnc2)C1=O C(=O)(C#CC1(C)COC1)NCC1N(C(CCc2c(C)cccn2)=O)CCCC1C CC1CCCn2c(C(=O)NC3CCN(C(c4c(N)ccc(F)c4F)=O)C3)cnc21 N1(CC(=O)NC2CC3CCC(C2)N3C(C2C3CC4C(C3)C24)=O)Cc2ccccc2C1 C=CCC(C(=O)NCC1CC(=C2CC2)C1)NC(=O)CN1CC2CCC1C2 C12(NC(c3c(N)cn(C)n3)=O)CCCCC1CN(C(C1CC1C1CCCC1)=O)C2 C1(C(N2C(C(N(C)C)=O)CC2)=O)CC2(CCN1C(C1CC3CCC1CC3)=O)CC2 N1(C(C23CC(OC(C)=O)(C2)C3)=O)CCC(C(=O)NC2CCN(C)C2=O)CC1 CC(C)(C)C(O)CN1CCN(C(C2CCNCC2)=O)CC1 N1(C(C2N(C(c3sc(C)c(Br)c3)=O)CC2)=O)CCCCC(F)(F)C1 c1(CS(N2CCC(C)(OCC)C2)(=O)=O)ccc(Cl)cc1F C(=O)(C#CC1CCCCO1)NCc1ccc(CC(C)NC(c2ccoc2)=O)cc1 c1(C(N2C(CNC(c3n(C(C)C)cnc3)=O)COCC2)=O)cc2n(n1)CCCO2 C#CC1(C(=O)NC(CCO)C(C)(C)C)CCN(C(=O)CCc2cccnc2)C1 C1(CNC(CC2(OC)CCCCC2)=O)CC2CCC1N(C(C1(CO)CCC1)=O)C2 CN1CC(NC(C2CCOC(=O)C2)=O)C(C(F)(F)F)C1 Cc1ccc2[nH]cc(CC(=O)NC3CCCN(C(c4csc(Cl)n4)=O)CC3)c2c1 C(=O)(C1=CC2CCCCC12)N(CC(O)CNC(=O)Cc1ccccc1Cl)C C1(NC(CCC2(C)CC2)=O)CCN(C(=O)CC(=O)OC(C)(C)C)C12CC2 C1(C(N2C(CNC(CC(C)Cc3ccc(Cl)cc3)=O)CC2)=O)CC2CCC1CC2 C1(C(N2C(CCNC(C(C(C)O)C)=O)CCC2)=O)CC2C=CCC(C1)C2 N1(C(c2cc(C)c(Cl)cc2)=O)CCC2CN(C(=O)C(C)(C)F)CC12 CC1(CNC(=O)C(N)=O)CC(F)(F)C1.C1(=O)CCCN1C(=O)CO Cc1cc(=NCC(O)C2CC(C)(C)C2)[nH]cc1S(=O)(=O)NC(c1cccnc1)C CC1(C)CCC(CCN2CC(CNC(C3CCCCC3n3cccn3)=O)C2)C1 Cc1sc(=O)n(C(=O)N(C2CN(c3ncnc(C(C)(C)C)n3)C2)C)c1C c1(C(C)C)ccccc1OCC(N1CCC(C)C1CNC(c1ccsc1)=O)=O n1(CC)cc(C(=O)NC2CC(CC(=O)NCC(C)(F)C(C)C)C2)c(C)n1 C1(CNC(COCC#C)=O)(NC(C2CCCC2O)=O)CC2CCC1CC2 c1(C(=O)OC)nccc(C(N2CCN(CC(=O)OC)C(=O)C2)=O)c1OC1CCC1 c1(C(=O)NC(C)CC2CN(C(C3CCCC34CC4)=O)C2)cccc2c1OCCO2 CCC(C)(C#N)C(=O)NOCC(=O)NCC(C)F C(C)(C(C(=O)NC1CN(C(=O)OC(C)(C)C)CC1CSC1CC1)n1cccn1)OC C(=O)(C(C)(F)C(=O)NCC(O)C(=O)NCCN1CCOC1=O)OC C1(C(=O)NCCc2c(C(=O)NCC(C)F)c[nH]n2)CCCN1C=O N1(CC)CCCCC1C(=O)NCC1(F)CN(C(=O)C2=CCCC2)C1 c1(CC)cnc(C(N2C3CN(C(c4cccnc4OC)=O)CC23)=O)nc1 C(CO)(C(C)N=c1[nH]c(=NCC2(C(C)C)CCCC2)[nH]c2ccsc12)SC S(=O)(=O)(c1cc(C)cnc1)N1CCCC(C=C)C1.C(CCCCCSC#N)NCCC C(N=c1cc(Cl)nc(C2CC2)[nH]1)C1C(NC(c2cc3n(n2)CCCO3)=O)CCC1 Cc1cccnc1CCC(=O)NCCSCC(N1CC(O)C(O)C1)=O c1(CC(=O)NC2CC(F)(CNC(C(Cn3ccc(C)n3)C)=O)C2)cccc(F)c1 O(NC(=O)C(COC)Oc1cn(C2CCOCC2)nn1)C(CCC(=O)OC)C C12(C(=O)OC)CCC(C(=O)NCC(C)CNC(=O)C=Cc3scnc3C)(C1)C2 C(CC(O)CC(=O)NCC1CCN1C(=O)CCc1nccs1)SC c1(CN(C(C2C(C(C)NC(C=C)=O)C2)=O)CC)cccc(O)c1 C(=O)(CCCCN(C)C)NC1CC(CNC(CN(C)C)=O)C1 C=CC1(C(=O)NCCN(C(=O)C(CCC)NC(N)=O)C)CCOCC1 c1(C(=O)NCC2C(CNC(c3cccc(CO)c3)=O)C2)nccc2[nH]ccc12 CC1CC(CN(C2CCN(C(c3ccnc(OCCO)c3)=O)CC2)C)CCO1 Cn1nccc1NC(C1CCCN1c1nnc(C2CCCC2)s1)=O N1(C(c2cc3ccc(Br)cc3o2)=O)CCCC(S(=O)(=O)N2CCOCC2)C1 C1(OC(C)C(=O)NC2CCC2NC(c2nc(Cl)cs2)=O)CCCCCC1 N1(C(C(C(C)(C)C)NC(C)=O)=O)CC2CCCCC2(CNC(C)=O)C1 C1(CNC(CC=CC)=O)CCN(C(=O)CCCCOc2ccccc2)C12CC2 Cc1cc(NC(C2CCC(O)CC2)=O)ccc1NC(C1CC1(C)C)=O C1(C(N(C2CCN(C(c3n(CC#C)ccc3)=O)C2)CC)=O)CC2(C1)CC2F c1(CNC(C2N(C(c3n[nH]c(C)c3C)=O)CCCC2)=O)ccc2c(c1)CCO2 C(=O)(CCCN(C)N=O)NC(CN(C(c1ccc(=O)n(C2CC2)c1)=O)CC)C C1(C(=O)NCCC(=C)CNC(C2CCCC2(C)C)=O)CC2CCCC(C1)C2 C1(NC(CCOC)=O)C2CC3CN(C(=O)C(c4ccccc4F)C)C1C3C2 c1(C(=O)NC(C(=O)N(C2C(C)CC2)C)CC2CCOCC2)cncc(CO)c1 Cc1coc(C(=O)NC2(CF)CCN(C(c3c[nH]nc3C3CC3)=O)C2)c1C C1(NC(c2c(Cl)cc(C)s2)=O)CCN(C(=O)CCc2ccc[nH]2)C(C)C1 C1(C(=O)O)CN(C(c2ccc(F)c(Br)c2)=O)CC12CN(C(=O)CCCCCl)C2 C1(C(N(C2CC3CC2N(C(C2CC=CC2)=O)C3)C)=O)Cc2nncn2C1 Cc1nc(SC(F)(F)F)sc1CC(=O)NCCNC(=O)CNC=O c1(C2(C(=O)NC(CC=C)CNC(c3cnc(C(C)C)o3)=O)CC2)ccc(Cl)cc1 C12(CNC(=O)C=Cc3cnc[nH]3)CC1CN(C(=O)CC1CSCCS1)C2 C1(C(=O)NCC(CC)C)CC2CCC(C1)N2C(=O)CCCC#N c1(CNc2c(C(=O)OCC)[nH]c3ccccc32)c(C)cc(C)c(C(C)=O)c1C c1(C(N2CCC(CNC(C(C)SCCCC)=O)CC2C)=O)cc2ncccc2s1 c1(OC)ccc(CN2CCCCC2C(C)N)cc1Cl c1(CCCNC(C(Cc2ccccc2)NC(N)=O)=O)ccc2c(c1)OCO2 C1(NC(C2CCN(C(=O)C3CC3)CC2)=O)Nc2cc(C(F)(F)F)ccc2S(=O)(=O)N1 C12(CNC(c3cc(SC)oc3)=O)CC1CN(C(c1ccnnc1)=O)C2 C1(C(C)NC(=O)CC(C)C)CCN(C(C2CCCN2C(=O)C(C)(C)F)=O)CC1 C1(C(N2C(C(C(=O)N(CCOCC)C)(C)C)CCC2)=O)CCS(=O)CC1 Cc1nc(C2CC2)[nH]c1C(=O)NC(CNC(=O)Cc1cccnc1Cl)C1CCC1 N1(C(C(CN(C)C)(F)F)=O)CCOCC(C)(CNC(C2(C)CCN(C)C2)=O)C1 c1(NC(C(C)N(C(=O)C=CC(F)F)CC)=O)ccc(OC)cc1O n1(CC(=O)N(C2CCN(C(=O)CCCn3ccnc3C)C2)CCC)nnc(=O)[nH]1 N1(C(CC(C)NC(=O)OC(C)(C)C)=O)CCCC(C)(C)C1NCC1CCCC1 c1(N(C(=O)C(N)CCOCC(F)(F)F)C)ccc(C#N)cn1 c1(OC)cc(F)c2c(C(=O)N(CC(C)NC(=O)Cc3ccsc3C)C)n[nH]c2c1 C(=O)(CCC1=NNC(=O)CC1)NC(CNC(CSc1n(C)cnn1)=O)CO C(CCSC)(C(=O)NCC(c1cccc(Cl)c1)NC(c1cc(F)n[nH]1)=O)OC n1(CC)ncc(C(=O)NCCC2CCCCN2C(=O)C(C)c2ccco2)c1Cl c1(OC)ncc(C(=O)NCC2CCCN(C(c3ccc(CO)cc3)=O)C2)cc1F c1(NCc2cnc(SC)s2)[nH]c(=NCC(C)N2CCC(C)CC2)nc2sccc12 c1(C(=O)NCC(CNC(CCCC#CC)=O)F)cc(C)c(C)cc1Cl N1(C(=O)CCCc2cc[nH]n2)CC2(CCN2C(c2ncccc2Cl)=O)C1 C1(C(C)C)CC(O)CN1C(=O)CC1CCC(NC(C2COCC2(C)C)=O)CC1 N1(C(CN(C)C(N)=O)=O)CCC(CCCCNC(C2(C)CC2Br)=O)CC1 C(C1C(=O)Nc2c(F)cccc21)NC(c1ccc(OC)cc1)CC(C)C C1(N(C(CN(C2CCCCCC2)C)=O)C)CN(C(=O)C(O)C2CCC2)CC1(C)C c1(C(N2CCC(CNC(CCSCC(N)=O)=O)C2)=O)c(Cl)n[nH]c1C1CC1 C(=O)(C1CCCn2nccc21)N1CC(N2CCN(C(c3cn(C)nc3)=O)CC2)C1 N1(C(C(=O)NCCCSC)=O)CCOCCC1c1ccccc1 C1(C(N2C(CC)C(O)CC2)=O)N(C(C2CC(C)(O)C2)=O)CCCC1(C)C C1(C(=O)NCCCNC(C(C)OCCCCCC)=O)CC(=O)N(C(C)C2CC2)C1 C1(CNC(C(COC)(C)C)=O)CN(C(c2nnsc2SC)=O)CC12CC2 C(Cn1cccn1)(C(=O)NCC#CC1CC1)NC(c1csc(F)c1)=O C(=O)(C1=C(c2ccccc2)CCCC1)NC1C(C)CN(C(=O)C(C)C#N)C1 CCC(CC(=O)NCC#CCNC(C1(C)CC1(F)F)=O)C(F)F N1(C(CCCN(C(C)C)C)=O)CC(CNC(c2cc(=O)cc[nH]2)=O)C(C)C1 Cc1ccc(C2CCCN2C(=O)N(C2CC(CO)C(O)C2O)C2CCC2)cc1C CCC(C)C(O)C(=O)NC1CC(O)(CNC(C2(CC(F)F)CCC2)=O)C1 C1(NC(c2cccc(-c3ccoc3)c2)=O)CCC12CN(C(C1COCCO1)=O)C2 c1(OC)ccc(C(O)C(=O)NCC(C)NC(=O)C(=O)N(C)C)cc1 c1(C(=O)NCC(C)CNC(c2nonc2N)=O)cc(C(F)(F)F)ncc1[N+](=O)[O-] N1(C(C(OCC)OCC)=O)CC=CC1(C)C(=O)NCCC(C)(C)CC N1(CC(=O)NCC=CCC(=O)N(C2(C#C)CC2)C)C(=O)CNC1=O C1(NC(CC=C)=O)CC2CN(C(=O)C(c3cc(F)cc(F)c3)O)CC12 c1(C(N2C(CNC(C3N(C(C)C)CCC3)=O)CC2)=O)ccc2cc(O)ccc2n1 N1(C(COCCCCOCC#C)=O)CCC(C(O)CNC(=O)C=C)CC1 C1(C(N2CCCC(C(=O)NC(C)C)C2)C(=O)NC(CC)C)CC2CC1C1CC21 C1(C(=O)OC)N(C(c2cccc(OC(F)F)c2)=O)CC12CCC(F)(F)CC2 CC1CN(C(=O)CCCN=[N+]=[N-])CC(C)C1NC(=O)C1=CCCS1 C1(CC(C)NC(CCC=CC)=O)CCN(C(c2ccccc2SCC#N)=O)CC1 c1(OCC(N2CCC(C)(CNC(C(C(C)C)O)=O)C2)=O)ccc(Cl)c(C(F)(F)F)c1 CC(=O)CCCC(C)C(=O)NC1CC(CNC(C23CCC(CC2F)C3)=O)C1 Cc1cc(O)nc(C)c1C(=O)NCCCOCCNC(=O)C(C)(C)C Cc1cccc(CC(N2CCC(CNC(C3CN(C)C(=O)N3)=O)C2)=O)c1C C1(NC(=O)CC(Cl)Cl)C2CCC(C2)C1C(=O)NCc1cc(F)cc(F)c1 c1(N2CCC3(C(C(=O)OC)C3)C2)cc(NC(=O)NC2CC2)c2c(c1)COC2=O N1(C(CC=C)=O)CCCC2CN(C(=O)Cc3ccc4c(c3)CCCO4)CCC12 N1(c2nccc(SC)n2)CCC2C(CCCN2C(=O)CCCCN(C)C)C1 C(C(CC(=O)NCC(C)(Cn1cccn1)NC(c1cnc(Cl)s1)=O)C(F)F)OC C1(C2N(C(c3cc(CC)[nH]n3)=O)CCC2)CCN(C(C2C=CCS2)=O)CC1 C1(C(C)NC(C=CC(=O)OCC)=O)CN(C(c2cc(Cl)cnn2)=O)CCO1 C=CCC(CC=NOCC(=O)NCCNC(=O)N(C)C)C(=O)OCC CCC(CC(=O)NCCOC1CCN(C(c2nn(C)cc2C(C)=O)=O)CC1)OC CCC(C)(CCNC(c1ccsc1Cl)=O)NC(C1CC=CC(O)C1)=O C1(N(C)C(c2ccc(-c3ccco3)s2)=O)CCC(NC(C2COC2)=O)C1 c1(CC)cccc(C(N2CC=CC2(C)C(=O)NCCCN2CCCC2C)=O)c1 C1(NC(c2ccc(C(C)C)o2)=O)CN(C(c2cccc(O)c2Cl)=O)C(C)(C)C1 c1(C(=O)NC(C)CC2CCC(F)(F)CC2)cnc2c(c1)CCC2 N12CC3CCCC(C1)C3C2=O.n1(CC)cc(CNCC(=O)NC2CC2)cn1 CCCC(C)(CCC)C(=O)N1CC(CNC(c2cnn(CC)c2)=O)C(C(F)(F)F)C1 C1(C)(CNC(c2ccc(C)nc2C)=O)CN(C(=O)CC2CCC2(C)C)C(C)(C)C1 c1(C(=O)NC(C2(O)CCN(C(=O)CC3CC(=O)C3)C2)C)cc2n(c1)CCC2 C(=O)(C(CNC(c1ccc(C(N)=O)[nH]1)=O)C(C)(C)C)Nc1c(CC)csc1 Cc1cc(CNC(C2CCCSC2)=O)oc1C(N1CC(N2CCCC2)C1)=O C1(CC)CCCCC1C(=O)NCCC1CCCN(C(C2CCCC2OC)=O)C1 c1(CNC(c2ncn(CCNC(C3C(CCC)C3)=O)c2)=O)cc(C)c(C)o1 C1(C)(NC(c2cnc(CC)o2)=O)CCCCC1C(=O)NC(C)Cc1cnn(C)c1 C1(C(N(C)CC2CCSC2)=O)CCCCCCN1C(=O)Cc1ccsc1 C(=O)(C1(C)COc2ccccc21)NCC1CC(NC(CCC(C)OC)=O)C1 N1(C(c2c(CNC(CC3(NC(C)=O)CC3)=O)occ2)=O)CC2(CCNC2=O)C1 N1(C(CCC=C(C)C)C(=O)Nc2c(C)cccc2C)Cc2ccccc2CC1C N1(C(C2(CC)CC2)=O)CC2(COC(CNC(C3OCC3(C)C)=O)C2)C1 C1(C(N(C)C)=O)CCC(C(=O)O)N(C(=O)OC(C)(C)C)C1.c12noc(n1)NC2 C12COCC1N(CC)N2.c1(SCC2CCCN2C(=O)OC(C)(C)C)cnn(C)c1 C1(NC(CCC#C)=O)CN(C(c2nc3cnccc3s2)=O)C2(CCOCC2)C1 Cc1cccc2c(CC(=O)N(C)CCN(C)C(C3CC(F)(F)C3(F)F)=O)c[nH]c12 c1(CNC)c[nH]c2c(Cl)cccc12.c1(CCN2C(=O)C3(CC3)C2=O)cncn1C C1(OC)CC2CC(C(N3CCCC3CCNC(=O)C(C(C)C)C3CCC3)=O)CC12 C1(C(C)(C)C)(CNC(C2C(CC)C2)=O)CCN(C(c2cncc(Br)c2)=O)C1 CC1CCCC=C1C(=O)N1CC(CNC(C2CC(=O)CCO2)=O)C2(CC2)C1 c1(C(N2CC(CNC(C(COC)(C)OC)=O)OCC2)=O)cc2sc(C)cc2[nH]1 N1(C(C(C)N(C)C)=O)CCN(C(=O)C(C)(C)N2CCOCC2)CCC1C C1(F)(CNC(c2cccnc2-n2ccnn2)=O)CCCN(C(c2cnsc2)=O)C1 O=C1NC(Cc2ccccc2-n2ccnc2)C(=O)N1C1CC2CCC1C2 C(=O)(CC(F)(F)Cl)NCC(CC)NC(c1csc(NC(C)=O)n1)=O c1(N2CCC(N(C(=O)C=CC3CCCO3)C)C2)nc2c(F)cccc2o1 N1(C(CC(C)N(C)C)=O)CCC(NC(=O)C(c2cncnc2)C)C(O)C1 c1(C(=O)NC2(CNC(=O)C(O)C(F)F)CCCCC2)cc2cccnn2c1 S(=O)(=O)(c1ccccc1F)NCC(=O)NCC1CCN1C(C1CC12CC2)=O CCCC(C(F)(F)F)NC(=O)CC1CCC(NC(=O)CCCCOC)CC1 N1(C(CNC(CC(C)C)=O)=O)CCOCC(C(=O)NCC(C)(O)C(C)C)C1 C(=O)(C(F)(F)CN(C)C)NC(CC(C)NC(C1(C2CCC2)CC1)=O)C N1(C(C2CC(C)OCC2)=O)CCN(C(C2(Cl)CC2)=O)CC2(CC2)C1 CC1OC(=O)NC1C(=O)NCCCCCCN(C(=O)CNS(N)(=O)=O)C N1(C(c2c(CCC)n[nH]c2)=O)CCOC2(CCCN(C(=O)C(F)=C3CCC3)C2)C1 c1(C(=O)OC)ccc(N(C(=O)C(C)(F)F)C(C)=O)c(C)n1 C#CCCCCCCC(=O)N1CCCC1(C)C(N1CCOC(C(C)C)C1)=O C1(C(=O)NCc2c(C(N3C(CN(C)C)CCC3)=O)cco2)CC(C)(C)CCO1 C(C(CNC(=O)C(C)Sc1ccccn1)S(C)(=O)=O)NC(c1c(CC)nn[nH]1)=O c1(CC)ccc(Cl)c(C(N2CCOCC(NC(C3CCS(=O)(=O)N3)=O)C2)=O)c1 C1(CC2C(C(=O)OC)(C(=O)O)C2)CCCN(c2cc(C(N)=O)ccn2)C1 N1(C(c2c(C)nns2)=O)CCC(C(=O)NCCN2CCC(CO)C2)(C(C)C)C1 c1(CC(=O)N(C2CCC(NC(c3cccnc3)=O)C2)C)ccn(CC(F)(F)F)n1 C1(C(N(c2cccnc2-c2ccncc2)C)=O)COCCN(C(=O)C(F)(F)CO)C1 c1(SCc2c(C(=O)NCC(c3ccc(Cl)cc3)O)c[nH]n2)ccc(F)c(F)c1 C1(C(=O)NC(C(=O)NCC(CCC)OCC)CCC2CC2)CC(=O)NC(=O)C1 C(=O)(C(C)P(C)(C)=O)NCCCN(C(CCc1ccc(C)o1)=O)C1CC1 CON(CCC(=O)N1CCn2c(C)nnc2C1)C(=O)C1CC(C)CC(=O)N1 c1(OCCCC(N2CC(CC=C)(NC(=O)C(F)=CCC)C2)=O)ccccc1Cl c1(C(N2C(C(C)NC(C3CC3C3CCC3)=O)CCC2)=O)ccc2cnccc2n1 N1(C(C)=O)CC2OCC(C(=O)Nc3ccc(Br)cc3C(C)=O)C2C1.C1C(=O)N1 CCC(CC(C)C)C(=O)N(CCC(C)(C)NC(c1cccc(C(C)C)n1)=O)C C1(CN2C(CNC(c3cnccn3)=O)CCCC2)CCCC2(CCC2)O1 n1(CC)cnc2c(NCC3CCOC3(C)C)[nH]c(=NC3CC(C(F)F)C3)nc12 c1(C(N2CCC(N(C(c3c(C)cnnc3)=O)C)C2)=O)cc(N)nc(Br)c1 c1(C(=O)Nc2cccc(C(N3CCN(C)CC3)=O)c2)cccc(C#CCO)c1 N(C(=NCCC(=O)N(C)C)NCCc1c(F)cccc1F)CC1C(C)C1 C(=O)(C1=CS(=O)CCC1)NCC12C(CN(C(CNC(CNC(C)=O)=O)=O)C1)CC2 c1(C(N2CCC(NC(CCCC(C)=O)=O)C2C(C)C)=O)ccc(N=S(C)(C)=O)s1 N1(C(CC2(CSC)CC2)=O)CCC(NC(c2cocn2)=O)CC1C1CC1 C(=O)(C(CC(=C)C)NC(C1CC1C(F)F)=O)NC(C1CCOC1)C#C CC1(C)CC(NC(=O)CC(C)(C)C2CC2)CN1C(C1CC(C#N)C1)=O CCC(F)C(=O)N1CCC(CNC(=O)CCN(CC)CC)C1 N1(C(C(C(CC)C)O)=O)CCC2(CCC2)C(NC(c2cc3c[nH]cnc-3n2)=O)C1 C1(SCC(N2CCC2c2cn(C3CC3)nn2)=O)CC12CCOc1ccc(Cl)cc12 C1(C(N2C(CNC(c3c(OC)nccc3)=O)CC3CC32)=O)CCCC12OCCO2 c1(C(c2nc(C3CCN(CC)CC3)nn2C(C)C)CC)ccc2c(c1)CC(C)O2 C1(CCNC(C2CCC(F)(F)C2)=O)CN(C(=O)COC(F)(F)C(F)(F)F)CCO1 N1(C(C2=C(C)CCC2)=O)CCC2CCN(C(=O)C3=CCS(=O)(=O)C3)CC12 C#CCCCCCCC(=O)N(C1CCCN(C(=O)C(c2cccc(C)c2)C)C1)C c1(C(N2CC3C(NC(C(C)N(C(C)=O)C)=O)(C3)C2)=O)cc(C#N)c(F)cc1F c1(OC)ncccc1C(=O)NC(CNC(=O)C(C)Oc1ccc(F)cc1)C(C)C CCC(C)C(=O)C(=O)N1CCC(O)(C(=O)NCCN2CCC(O)C2)CC1 C1(CNC(=O)C2CC2)COCCN(C(c2cnoc2C2CCC2)=O)C1 C1(C(=O)NCC(C)C(C)(C)C)(NC(C(COC)O)=O)CCc2cc(Br)ccc2C1 N1(C(C(C)CC2CCCC2)=O)CCC2CCCC(C1)N2C(C1(N(C)C)CC1)=O Cc1nn(C2CC2)cc1C(=O)NC1(C)CCN(C(c2coc(Cl)n2)=O)C1 C1(NC(Cc2cc(C)sc2C)=O)CCN(C(=O)C=Cc2cncs2)C(C)C1 C(C)(CN=c1[nH]c(=NCc2cc(O)n[nH]2)c2sccc2[nH]1)c1c(C)noc1C c1(C(=O)OC2CC2NC(=O)CC2CC2C(C)=O)cnoc1-c1cccs1 C1(C(C)NC(CCSC)=O)CCCCN1C(=O)CNC(=O)C1CC1 c1(CC(N2CCC(CNC(CNC(N)=O)=O)C(O)C2)=O)cn2ccccc2n1 N1(C(C(OC)OC)=O)CC(CNC(=O)C2=COCC2)C(c2ccccc2)C1 c1(C(N(CCCCNC(CC(C)CN(C)C)=O)C)=O)cc2ccc(Cl)cc2[nH]1 CC1CN(C(=O)CC2CCN(C(=O)C(C3CCOCC3)=O)CC2)CC(=O)N1C CCC(CC(=O)N1CCC(C(C)NC(C2CC(=O)OC2(C)C)=O)CC1)C(C)C c1(CC)ncc(C(=O)N(CCC(=O)NCCCC(=C)C)C2CC2)cn1 n1(CCC(=O)NC2CC(NC(C3CC4CCCC4C3)=O)C2)ccc2ccccc12 N1(C(C)C)C(=O)COCC1C(=O)NC1COCC1NC(=O)CC(C)(C)C#N c1(C(N2CCC3CCN(C(=O)CC4CCC4)C3C2)=O)cncc2cc(Cl)ccc12 C(C(=O)NCC1(CCCNC(c2cnoc2CC)=O)CCCC1)(C(C)C)SCC N1(C(C2(OC)CCCCCC2)=O)CCCCC12CC(NC(C1CC(C#N)C1)=O)C2 c1(C(N2C(CCNC(C3C(=C)C3)=O)CC(F)(F)C2)=O)cc2cc(Cl)ncc2[nH]1 C(=O)(C(C)CC(F)F)N1CC(CCC(=O)NC2(C(=O)OC)CCCC2)OCC1 N1(CC(=O)NC(C2N(C(CN(S(C)(=O)=O)C)=O)CCC2)(C)C)CCS(=O)CC1 N1(C(CC(C(C(C)C)C)C)=O)CCC2CC(CNC(=O)CCC3CC3)CCC2C1 N1(C(CC2(CN)CCC2)=O)CCN2CCCC2C12CCC2 C#CCCC(O)C(=O)NCc1nc(CNC(C23C=CC(CC2)C3)=O)cc(O)n1 N1(C(C2C(CC)OCC2)=O)CCN(C(c2cc(C)cs2)=O)C(CC(F)(F)F)C1 C1(C(N2CC(C3CC3)(C(=O)NCCCCCCC3CC3)C2)=O)CCC(C2CC2)C1 Cc1cc(=O)c(NC(C2CCC2NC(c2cnc(S)nc2)=O)=O)c(C)[nH]1 c1(CN=c2cncc(OC)[nH]2)cccc(N=S2(=O)CCCC2)c1 N1(C(=O)OC(C)(C)C)CCC1C=CC(=O)NC1CC(CCC(=O)O)C1 CC1CCN(CC(N2CCCC(CCNC(C3CCC4CC4C3)=O)C2)=O)CC1 CC1CCOCC1C(=O)NCCCN1CCN(C(=O)CCc2cnc(O)[nH]2)CC1 c1(C(=O)NCC(CC(C)C)NC(=O)Cn2cnnn2)cccc2cc(O)ncc12 C1(NC(COCC)=O)CN(Cc2ccc(C)cc2Br)CC1(F)F c1(OCCC)ccc(CCCC(=O)NC2CC2NC(=O)CCSC2CC2)cc1.OC C1(C(=O)NC2CN(C(Cc3nn(C)c(Cl)c3)=O)CC2F)CC12CCC1(CC1)CC2 c1(CC)ccc(C(N2CCC(CO)(NC(C3CC4OC3C3CC43)=O)C2)=O)c(Cl)c1 C(CC(C)C)(C(=O)NCC1(O)CC(C(=O)NCC2CC(C(C)C)C2)C1)OC C12(C(=O)NCC(C)N(C(C3ON=C(C)C3)=O)C)CCCC1CCC2 c1(C(=O)NC2CCN(C(Cn3c(C)cc(C)n3)=O)C2C)cc(S(N)(=O)=O)c(C)o1 N#Cc1cc(CNC2CC2C(=O)Nc2ccc(F)c(Cl)c2)cc(F)c1 c1(C(=O)NCC2OCCN(C(C(CC)F)=O)C2)cc(OC)cc(OC)n1 N1(C(c2nn(C)c(C(N)=O)c2)=O)CCC2(CO)CN(C(=O)C=CCF)CC2C1 CCC(C(=O)N(C1CN(C(=O)COc2ccc(OC)cc2)C1)C)C(C)(F)F c1(C(C(=O)NCCN(C(=O)Cc2cc(C3CC3)no2)CCC)C)ccccc1F c1(CNC(C(C2CCN(C(C)=O)CC2)C)=O)cccc2nccnc12 c1(C(N(C2CCN(C(=O)CC3OCCO3)C2)CC)=O)c(F)cccc1F c1(CC)cc(OC)ccc1C(N1CCC(CNC(=O)C(C)(C)C#N)C1)=O n1(CCNC2(C(N3CCC3CF)=O)CC2)cc(C2CCC2)nn1 N1(C(C(COC)O)=O)CC2(Cn3cc(Cn4cccc4C(=O)O)nn3)CC1CCO2 C(CCN(C(=O)CC1CCCCCC1)C)(C(C)(C)C)NC(c1c(C)cncc1)=O C(CCC(O)C(=O)N1CCOC(C#N)C1)NC(c1nc(C)oc1C)=O C1(NC(C(C)(C)NC(=O)CC2CC(=O)C2)=O)CCC(=O)NC1(C)C C1(NC(CCC(=C)Cl)=O)CN(C(=O)C(n2nccc2C)C)CC(C)(C)C1 C12(NC(C(CC)C(C)O)=O)CC(CO)(C1)OC21CN(C(C2CC3C=CC2C3)=O)C1 N1(C(CC2C(NC(c3cccnc3S)=O)CC2O)=O)CCCC12CC2 C1(C(=O)NCCCN(CCCNC(C2CCCC(C)C2)=O)C)CCS(=O)(=O)CC1 C(CN=c1[nH]c2cc(Cl)c(S(=O)(=O)N3CCOC(CO)C3)cc2s1)OC N1(C(C(CCC)C(C)C)=O)CCOC2(CCN(CCCS(C)(=O)=O)CC2)C1 Cc1cccnc1C(N1CCCCC1C(C)(C)CNC(c1ncn(C)c1C)=O)=O C1(NC(c2cncc(NC)c2)=O)CN(C(=O)CC2CCCC(=O)N2)CC12CCC2 c1(CCC(=O)N(C)CC2N(C(C(C=C=C)C)=O)CCCC2)nc2ccccc2s1 c1(C(=O)NC2CC3CN(C(C(CC(C)C)C)=O)C(C2)C3)noc2c(F)cccc12 C1(NC(CC=CC)=O)CC2CC(C1)N(C(=O)COc1ccc(C(=O)NC)cc1)C2 c1(C(C(=O)N(CC(C)N(C(=O)C2=CCSC2)C)C)=O)ccc(F)c(F)c1F CC1CCN(C(c2csc(Cl)c2)=O)C(C(=O)N(C)CCN2CCCCC2)C1 C1(C(C)C(=O)NCCn2cncn2)CCN(C(=O)C(C)(C)CC2CC2)CC1 c1(C(=O)NCCOCCN(C(C2CCC(C)O2)=O)C)cccc(CN(C)C)c1 CC(CC(C)(C)C)C(=O)NC1CN(C(c2cnc3ccccn23)=O)CC1C(F)F c1(N2C3CC(F)C(C3)C2)ncnc2n[nH]cc12 CCC(CNC(=O)C(C1CCN(C(=O)CC2CC=CCC2)C1)C)(CC)C N1(C(C(C)=C2CC2)=O)CCC2CN(C(=O)CSc3ccc(Cl)c(Cl)c3)CC2C1 CCCCCCCCOCC(=O)NC(CNC(C1CCCC1)=O)C1CCC1 C(CCO)(C(F)F)NC(C(COCC)n1cc(C2(C(=O)O)CCCC2)nn1)=O Cc1occc(=O)c1OCC(=O)NC(C1CN(C(C2CCCO2)=O)C1)C C1(N(C(CCC=C)=O)C)CN(C(c2nn(C)cc2C(C)=O)=O)CCC1O c1(C(=O)NCC2(O)CCN(C(C34CCC3CC4)=O)C2)c[nH]c2cnccc12 c1(C(N(C(CCNC(C(C)NC(COC)=O)=O)C)C)=O)cc2cc(F)ccc2o1 c1(SC)ccc(C(N2CCCC(CCNC(C3(CO)COC3)=O)C2)=O)cc1 Cc1nnccc1C(N1CCCC1(C)CNC(c1snc(C)c1N)=O)=O C(CC(C)C(=O)N(CC(C)C(=O)NCC)Cc1ncnn1C1CC1)=CCC c1(C(=O)NCC(C(=O)N(C)CC2(CO)CCC2)OCC)ccc(Cl)c(O)c1 C12C3CC4C(C3NC1=O)C24.C(=O)(C(C)(CC)OC)NC1CN(CCC)C1 c1(C(=O)NCC(CN(C(=O)CC2CCC(F)(F)C2)C)O)cc2n(n1)CCO2 C1(C(=O)NCC(C)(F)CNC(c2cc[nH]c(=N)c2)=O)(OC)CCC(C)(C)C1 C1(CCC)CC(NCCc2cccc(F)c2)CCO1 C(=O)(CCCCCCCC1CC1)NC(CCCNC(C1=C(C)OCC1)=O)C c1(C(N2C3CCC(NC(c4ccc(C=C)cc4)=O)(C3)C2)=O)cc2cc(Cl)sc2[nH]1 C1(NC(c2n(CCOC)ncc2)=O)CN(C(c2cc(O)cs2)=O)CCC12CCC2 c1(SC)ncc(C(=O)NC2CN(C(c3nnn(C)n3)=O)C2)n1-c1ccc(F)cc1 c1(OC)cc(C(C)NC(=O)CN2CC(=O)NC2=O)ccc1OCc1noc(C)n1 c1(OC)cccc(CC(C)(C)NC(=O)NC2CSC(C)(C)C2)c1 c1(CN(C(CCC)C)Cc2ccccc2)ccc2c(c1)CCCN2C C1(C(=O)NC2CCN(C(c3c(C)cc(C)[nH]3)=O)CC2C)CCc2nccn2C1 N1(C(C(c2cccnc2)OC)=O)CCOC(CC2CN(C(=O)OC(C)(C)C)C2)C1 c1(OC)cc(C(O)C(=O)N2CC(NC(=O)CC(C)F)C2)c(F)cc1O c1(NC)nc(C(N2CCC(NC(=O)C3CC3)C2(C)C)=O)ccc1[N+](=O)[O-] C(CC(=O)O)(CC(C)C)N(C(CC)CO)CCc1ccccn1 C(CC(CC)(CC)NC(=O)C(C)Cn1ccnc1)NC(C(CC)(C)O)=O N1(Cc2cn(CCC(C(C)C)NC(=O)CCC(F)(F)F)nn2)CCc2ccccc21 c1(C(C)NC(c2csc(C(=O)N(C3CC(O)C3)C)n2)=O)nc2c(s1)CCCC2 c1(CN2CCCC(C(N(C(C)C)C)=O)C2)cccc2ccncc12 c1(CC(N2CC(F)(CNC(CC3C(CC)C3)=O)C2)=O)c[nH]c2c(F)cccc12 C1(C2N(C(C3(CC)CC3(F)F)=O)CCC2)CCCN(C(=O)OC(C)(C)C)C1 CC(CC(N)=O)C(=O)NCCCN(C(=O)Cc1nc[nH]n1)C1CC1 C(=O)(C1CCCn2cnnc21)Nc1nc(C)nc(N2CCC3(CC2)COC3)c1 C1(NC(c2c(C)sc(Br)c2)=O)CC(C)CN(C(c2nonc2N)=O)C1 C#CCCCC(=O)NC1CCOC(CNC(=O)CC2COC(C)(C)C2)C1 c1(C(=O)NCC2CN(C(C3(C)CCC3)=O)CC23CC3)cccc2ccnn12 C1(CC=C)(NC(C2CCS2(=O)=O)=O)CCN(C(=O)Cc2n[nH]c(=N)s2)C1 C1(C(=O)OC)C(NC(=O)Nc2onc3c2CCCC3)C2CCCCCC12 c1(CC(N2CC(NC(C(C=C=C)C)=O)(CO)C2)=O)cc(F)c(C)cc1F N1(C(C(C(C)C)N(CC)CC)=O)CC2CCCC(C1)N2C(=O)C(C(C)C)N(C)C C1(CC(N2CC(C(N)=O)(OC)C2)=O)CCN(C(=O)Cc2cc[nH]c2)C1(C)C C(=O)(C(C(C)C)c1ccc(C)cc1)NCCN(C(CNC(=O)OC)=O)C Cc1cccc(C(N2CCN(C(C3CC3(F)F)=O)C(C3CC3)C2)=O)c1C(F)(F)F c1(OC)ccc(Cl)c(C(N2CCCC2CNC(=O)CCSc2nccn2C)=O)n1 C1(NC(C(c2ccn(C)n2)C)=O)CCCCCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C1 C1(CCCC)CCCN1C(=O)C(C)CN(C)C(C1CCCCS1)=O n1(C(CC)C)ccc(=NC(=O)CCN(C(=O)C(CCN(C)C)N(C)C)C)[nH]1 c1(C(N(CC(C2CCCCC2)OC)C)=O)ccc2c(n1)CCC(C)(C)C2 c1(CC(C(=O)NCC(C)NC(C2(CC)CC(C)(C)C2)=O)C#N)ccc(C#N)cc1 C12(NC(c3n(C)ccn3)=O)CC(C1)N(C(=O)C(C)(C)c1ccno1)C2 C(=O)(C(CC(C)C)ONC(=O)C=C(C)C(F)F)N(C(C(=O)OC)C)C1CC1 c1(CC)cc(F)c(C(N2CC3C(CNC(=O)C(C)C(O)CC)C3C2)=O)cc1F C1(CNC(C2N(C)C(=O)OC2)=O)CCCCN(C(=O)C(F)(F)c2ccccc2)C1 CC1CCN(C(c2cc(CO)[nH]n2)=O)CC1NC(=O)Cc1sc(O)nc1O N1(C(c2nc(C)sc2)=O)CC2(CNC(=O)Cc3csc(C4CC4)n3)CC1CO2 N1(C(CCCCSC)=O)CCC(CNC(c2cnc(C(C)C)s2)=O)C(C)C1 c1(C(=O)NC2C=CC(CNC(C(C)NC(=O)NC)=O)C2)cc2cc[nH]c(=O)c2s1 C(=O)(C(O)C(C)(C)C)N1CC(O)(C(CNC(C(C)C(F)F)=O)(C)C)C1 c1(C(CC)C(=O)N(CCCNC(=O)Cn2nccn2)C)c(C)noc1C c1(C(=O)NC2CC(C(N(C)CC3(O)CCC3)=O)C2)cnn2ccccc12 Cn1cc2ccc(C(=O)NC3(CCNC(=O)C(F)C4CCC4)CCC3)cc2n1 Cc1cccc(O)c1C(=O)NC(C)CCCCNC(C1CC(=O)N(C)C1)=O c1(C(N2CCC(NC(c3c(C)n[nH]c3)=O)C2CO)=O)cc2n(n1)CCCCC2=O N1(C(c2cn(CC=C)nc2)=O)CCC(C)(C)C1C(=O)NC(CO)C1(C)CC1 CC1(C)COCC(NC(=O)NCCOCCCSC[Si](C)(C)C)O1 C1(N(C(C(CC)F)=O)CC)CCN(C(C2(CC)CCOCC2)=O)CC1 CC(C(=O)N(C1CN(C(=O)C(CC(F)(F)F)c2ccccc2)C1)C)C1=CCCC1 C1(NC(CC2(NC(Cc3c(C)cnn3C)=O)CCCCC2)=O)CC1C1CCCC1 c1(OC(CNC2(C(c3n(CC)nnn3)OC)CC2)C2CC2)ccc(Cl)c(OC)c1 C(=O)(CCCC(C)(C)C(=O)OC)NC(CC=C)CNC(c1ccc(C(C)F)cc1)=O S(=O)(=O)(c1cnc(C(=O)O)s1)N1CCC(Oc2c(C(N)=O)cccc2)C1 N1(CC)CCC(OC2CN(C(C34CCC(CC3)CO4)=O)C2)CC1NC(=O)CCOC N1(C(C=CC(=O)N(C)C)=O)CCC(C(=O)NC2(C(N)=O)CCC2)C1 CCCCCCC(=O)NC1CN(C(=O)CCCN(C)C(=O)C2CC2)CC1OC N1(C(C2(CCC)CC2)=O)CC2(C1)CN(C(C1CC(CC(=O)OC)C1)=O)CC2CO c1(NC(CNC(c2c(C)cc(SC)o2)=O)(C)C)cnc(C#N)cn1 c1(OC)ncc(C(=O)NC(C)CCNC(=O)CC2CN3CCN2CC3)nc1C c1(C(=O)NC2(C)CCN(C(C(CCCC)=O)=O)C2)cnn2cc(OC)ccc12 N1(C(C2CC(C)N(C)C2)=O)CC2(CCN(C(c3ccn4nccc4n3)=O)C2)C1 N1(CC)CCCCC1C(N1CC(OC)C(C(=O)NC(C)(C)CO)C1)=O S(=O)(=O)(c1cc(C)sc1C)Nc1cc(C(=O)OC)cc(F)c1 C#CCCCC(C(=O)NCSc1ccccc1)N1CC=C(CO)CC1 Cc1cc2[nH]c(C(=O)NC(CNC(c3coc(CO)c3)=O)C(C)(C)C)cc2o1 C1(C(=O)NC2CC(O)(CNC(CN(CCOC)C)=O)C2)Cc2ccc(F)cc2C1 c1(C(N(CCNC(c2c(C)ncc(Br)c2)=O)C)=O)cc(F)cc(Cl)c1N CC1(C)CCN(C(=O)C(c2cccnc2)C2CCCC2)c2ccccc21 C(=O)C(C)C(F)(F)F.c1(C(=O)OC)sc(CNc2cccc(CO)c2)nc1C C1(N(CC(=O)NC(CN(C(c2sccc2Cl)=O)CC)C)C)CCCC1O CC(C)CC(F)C(=O)NCC(C(C)C)NC(c1[nH]nnc1C1CC1)=O C(CCCC(=O)N1CCC(C2CCCN2C(c2coc(C(F)F)n2)=O)CC1)SC N1(C(C2CCCN(C(C3CCCCC3)=O)C2)=O)CCC2C(CCN2C2CC2)C1 C(C(C)(C(=O)N(CC1CC1)CC1CC1)NC(c1ccc(=N)[nH]c1)=O)SC c1(C(=O)NCC2CN(C(=O)C(F)=CCCF)CCCO2)ccc2occc2c1 N1(C(C23C(CN(C(=O)CCc4cncnc4)C2)C3)=O)CCOC(CO)C1 C1(CNC(C(C)CF)=O)CC2(CC2)CN1C(=O)CC1(O)CCCCC1 C(=O)(CCC(F)(F)C(F)F)N1CCN(C(C(C)C2CC2)=O)CC(O)C1 CC1CCN(C(=O)C=C(Cl)Cl)C(C)C1NC(c1cc(C(C)(C)C)on1)=O c1(OCC(=O)NCC(CC)NC(=O)CSc2cncn2C)ccncc1 C1(CC)(NC(c2cnc(COC)s2)=O)CN(C(C2SCC=C2C)=O)C1 C(=O)(C(F)C1=CCCCC1)NC(C)(C)C.CC1CCCN2C1C2=O.C(=O)OC N1(C(CSCCC#N)=O)CC(NC(C2(C(F)(F)F)CC2)=O)CCC(O)C1 C1(C(=O)NCC(=O)N(CC(C)(C)C)C)CC(=O)C1C(F)(F)F CC(C)CC(F)(F)C(=O)N1CCC2(CC1)CC2CNC(=O)C#CC1CC1 CC1CC(CNC(=O)CNCP(C)(C)=O)CCC1(C)C Cc1cc2[nH]c(C(=O)NCC3CCCCN3C(C3CC(Cl)(Cl)C3)=O)cc2o1 S(=O)(=O)(c1ccc(C)cc1Cl)N(S(CC(=O)OCC)(=O)=O)C1CC1 N1(c2cc(NC3COCC3C)nc(C(C)C)n2)CCc2nc(=N)[nH]cc2C1 c1(NCC2(CNC(C(CC)(C)OC)=O)CC23CCC3)ncnc2sc(C)nc12 c1(C(=O)NC2(CN(C(c3c(C)nccc3)=O)C)CC2)cc2c(F)ccc(F)c2[nH]1 c1(C(=O)NCC(C)CNC(=O)CNC(c2cccs2)=O)ncncc1C#N c1(C(=O)NC2CCC(F)(CNC(CCC(C)OC)=O)C2)[nH]c(C)c([N+](=O)[O-])c1C c1(C(=O)NC2CC(NC(C(C)(C)F)=O)C23CCC3)cncc(S(C)(=O)=O)c1 Cc1ccccc1C(c1cccs1)C(C1(C)CCN(C(N2CCCCC2)=O)C1)=O CC1CN(C(C2CN(C(c3cnccn3)=O)CC2(C)C)=O)C(C)C1C c1(C(=O)NCC2N(C(CNC(CC)=O)=O)CCCC2)c(C)ccc2ncccc12 CC(c1cccc(Cl)c1)=CC(=O)NCCNC(C1CNC(=O)CC1C(F)(F)F)=O c1(C(N(CCNC(C2CCC(C)S2)=O)C)=O)cnc2c(N)cccc2c1 c1(SC)nc(C)c(Br)c(=NCCCNC(=O)CN(c2ncccn2)C)[nH]1 CC1CN(C(=O)CCc2cccc(F)c2)CCCN1C(C1COC2(C)CC1C2)=O Cc1cnc2cccc(C(=O)NC3CC(C)CN(C(c4nc(=N)cc[nH]4)=O)C3)n12 C(CNC(=O)Cn1c(C)c(C)sc1=O)(C(C)C(C)C)NC(COCCCCC)=O C(=O)(C(C)CC(F)(F)F)N(CCCNC(C(C=C)(F)F)=O)CC1CCCC1 c1(C(N2CCCCCC2CNC(C2(O)CCSCC2)=O)=O)cn2cnnc2cn1 C1(CNC(C=CC(C)(C)C)=O)CN(C(=O)COC2CCOC2)CC(C)(C)C1 N1(C(C(C(CC)CC)C)=O)CCC2(CCN(C(c3ccccc3C(C)C)=O)C2)C1 n1(CC(=O)NCCC2(O)CCN(C(CC3C(C)C3)=O)CC2)cc2ncccc2n1 Cc1ccc(C(=O)NCC(N2CCCC2NC(c2ncccc2C)=O)=O)c([N+](=O)[O-])c1 c1(C(N2C(C)CC(NC(c3c(CC)nco3)=O)C2)=O)cc(N)ccc1O Cc1c(C(N2CCOCC(C(=O)NC(c3ccccc3)CO)C2)=O)cccc1Br c1(NC(C)CN2CCCC2)[nH]c(=NCCSC(F)(F)F)nc2scnc12 c1(C(=O)NCCNC(C2CCC2c2ccc(Br)cc2)=O)cccc(C(F)F)c1F c1(OC)cc(N)c(Cl)cc1C(=O)NCC1CCN(C(C2CNC(=O)N2)=O)C1(C)C c1(C(N(CCC)CCNC(C2(C)CCCN(C)C2)=O)=O)ccc2nn[nH]c2c1 N1(C(C2C(CC)C2)=O)CCC(CN(C)C(c2snnc2C(C)C)=O)C1 c1(C(=O)NCCC2CCN(c3snc(SC)n3)C2)ccc2oc(O)nc2c1 N1(C(CCC#N)=O)CC(NC(c2ccc(C(F)(F)F)o2)=O)CC2(CC2)C1 C12CCCN(C1)C2=O.N1(CCN(C)C(c2ccnn2C2CCC2)=O)CC2CC2C1 c1(NC2CC2)ccc(COCC(=O)NC2CC(NC(C3(C4CC4)CC3)=O)C2)cc1 CC1(CC(=O)NC2CCCC2NC(c2ccc(CC3CC3)s2)=O)CC1(Cl)Cl N(C(=NCCCOC)NCC1SCCS1)CC1(SCC)CC1 c1(C(N2CC(C(N)=O)(CNC(c3cc(SC)c(C)o3)=O)C2)=O)c(C)nn(C)c1N Cc1sc2ccccc2c1C(=O)NC1CN(C(=O)CC2CCOC2(C)C)CC1C c1(CC)ccc(C)cc1C(=O)NCC(O)CCNC(c1cc(N)cc(F)c1)=O N1(C(c2c(NC(C)=O)c[nH]c2C)=O)CC2CCN(C(=O)CC(O)C(C)C)C2C1 Cc1ncc([N+](=O)[O-])cc1C(=O)NC1CC2CC1CN(C(=O)C(O)C1CC1)C2 c1(OCC(=O)NC2CCCN(C(CCC)=O)C2)ccc([N+](=O)[O-])cc1 C1(C(=O)NCCOC(C)=O)(NC(=O)Cc2ccon2)CCN(C)C1 c1(NC(=O)OC(C)(C)C)ccc(F)cc1NC(N1CCC1C1CCOC1)=O c1(OCC)nc(C(=O)NN2CC(C(=O)NC3CC(CC4CC4)C3)C2)sc1C C(=O)(C1=CC2C=CC(C1)C2)NC1CCC(C)(NC(=O)C=CC2CCOCC2)CC1 CCCC(C(=O)NCC(C)(F)CNC(=O)C(n1ccc(C)n1)C)N(C)C n1(CC(N2CC(CC(=O)NC(C)CCSC)(OC)C2)=O)cccnc1=O C1(C(=O)NCC2CN(C(C3(CO)CCC3)=O)C2)CC(=O)N(O)C1 C1(C(=O)NC(CCCNC(C2(CC)CC2)=O)C)CCCN(C(C)C)C1 C1(NC(C2(N(C)C)CCC2)=O)CCCCN(C(=O)C(c2ccc(N)cc2)(C)C)C1 N1(C(CCCNC(=O)OC)=O)CCOC2CN(C(=O)CC(O)CC(C)(C)C)CC12 N1(CC)CCN(C(C2CCC3CCC2N3C(C2CCC(=O)O2)=O)=O)CC1(C)C Brc1c(SCCC2CCCO2)n[nH]c1-c1ccccc1 c1(C(N2CCCC2Cn2cc(COC3COC3)nn2)=O)cc(Br)n2ccccc12 N1(C(C(CC#C)(C)NC(=O)C(O)C(F)(F)F)=O)CCC2CCCCC2C1 C=CCC(CC(=O)N1CCCN(CC)CC1)NC(C1(C)CCCCC1C)=O c1(OC)ccc(S(=O)(=O)Nc2cccc(Cl)c2)cc1NC1CCOCC1(C)C CC1(C)CCCc2ccccc2C1NC(CC1CCOC1)CO CC1CCC(CNC(=O)COCC2CC2)N(C(C23CCOC(C)(C2)C3)=O)C1 C(=O)(C(CC(C)C)NC(C)=O)N(CC(CC)NC(C12CC(CO1)C2)=O)C C(CC(C)(C)C)(C(=O)NC(C)C1CC1)NC(C1C(C(C)C)CCO1)=O C1(F)(CNC(CCOCCCOC)=O)CCN(C(=O)CC(C)SC)CC1 C1(NC(C2CCC(CC)O2)=O)CCN(C(C2(CN(C)C)CC2)=O)CC1C c1(NC(N2CCC(NC(=O)CCCC3CC3)C2)=O)cccc(Cl)c1F C(=O)(CCC1CC(NC(N2C(CN(C)C)CC2)=O)C1)OC(C)(C)C c1(C(=O)NC2(C)CC(NC(=O)C(=O)NCC(F)(F)F)C2)ccc([N+](=O)[O-])cn1 c1(CC)nn(C)cc1CNC(=O)NCC(C)(C)C(C)O C(N=c1[nH]c(=NCc2ccc3c[nH]nc3c2)[nH]c2ccsc12)C1C(C)CCCC1 N12CCC(O)(CC1)C2=O.c1(CN(C)C)ccc(-c2ncc(C(=O)NCCSC)s2)cc1 C1(NC(=O)CCc2cncs2)CN(C(c2conc2C2CCCC2)=O)CCC1F C(=O)(CCC(=O)NCC1CC(CNC(=O)C(C)(C)CO)C1)N(CCC)CCC c1(OCC)cccc(C(=O)NC(C)C(N2CC(O)(CO)C2)=O)c1 c1(OC)c(C)nc[nH]c1=NCC1CCCN(C(=O)C(c2c(C)nn(C)c2C)C)C1 c1(C(N2C(C(C(=O)OC)C)CCC2)C(=O)NCCC2CC2)ccc(C#N)cc1Br N1(C(c2cc(Br)c(CC)c(Br)c2)=O)CC(=O)NCC2CCCC12 c1(C(N2CC(F)CC(NC(=O)CN3CCCCC3)C2)=O)cc(O)cc([N+](=O)[O-])c1 C(=O)(C(C)(C)CC(=O)NC(C)(CNC(C12CC(CO1)C2)=O)CO)OCC c1(C(N2C3(CNC(=O)C=Cc4ncc[nH]4)CCC2CC3)=O)cc(O)c(O)c(O)c1 CC1C(C)N(C(=O)COc2cccc(C#N)c2)CCN1C(=O)Cc1cnccn1 N1(C(c2c(C)cccc2)=O)CCC(C2CC2NC(c2cc(C#N)c[nH]2)=O)CC1 c1(CC(C)C)ccc(C#N)c(NC2CN(C(=O)CC3CC(O)C3(C)C)C2)n1 C=CCC(C(=O)N1CCC(CO)(CNC(=O)C=CCCC=C(C)C)C1)C(C)C CC(C)C(C)C(CNC(=O)CP(C)(C)=O)NC(=O)CCSC1CCCC1 c1(OC)cc(SC)ccc1C(=O)NC(C1COCCN1C(=O)CC1CC=CC1)C C1(NCc2ccc(C(=O)Nc3c(C)cc(OC)cc3)o2)CC(O)C(O)CC1CN O=C(CCC(F)(F)Cn1cc(CCCO)nn1)NCCc1cc(Br)no1 c1(CC(=O)N(CCCCN(C)C(C2CCCC(O)C2)=O)C)ccc(F)cc1F C1(C(=O)NCC(C)(C)SC)CC(NC(c2c[nH]c(C)c2)=O)C1(C)C c1(C(=O)NC2C(CNC(Cc3ccc(C)nc3)=O)CC2)c(C)cccc1O C1(NC(c2cc(CCC)c(C)s2)=O)COCCN(C(c2ocnc2C(F)F)=O)C1 N1(C(C2C(=C)C2)=O)CC(C(=O)NCCCn2cnnn2)C(F)(F)C1 c1(C(=O)NC2CC(C)(NC(C3CCS3(=O)=O)=O)C2)ccc(F)c(OC(F)(F)F)c1 c1(C(=O)NC2CC(CNC(c3c(CC)ocn3)=O)CC2O)cc(SC)ccc1C C(=O)(C#CC1(C)COC1)NC1CCCN(C(C=CC(CC)=CC)=O)C1 C(=O)(CC(C)(C)c1ccccc1)NCC(C1CCC1)NC(c1c(C)con1)=O N1(C(C(CC)C(C)C)=O)CCN(C(=O)C(c2cccc(OC)c2)C)CC2(CC2)C1 C12(C(N(C(C(=O)OC)C)C3CC3)=O)CC(CN(C(=O)CCC3CCCC3)C1)C2 c1(NC(C2(F)CN(Cc3cccc(C#C)c3)C2)=O)cc(Cl)c(Cl)cc1Br C(=O)(C1=C(C)OCCS1)NCCCCN(C(C(C(C)(C)C)NC(C)=O)=O)C C(=O)(C(CO)C(F)(F)F)NC(CN(C)C(C1CCC2(CC2)C1)=O)(C)C C1(CC(=O)NCC(C(C)C)NC(c2ccsc2-n2cnnn2)=O)CCC(C)CO1 N1(C(COCCCN=[N+]=[N-])=O)CC(C(=O)NC2CC3CCCC3C2)C(F)(F)C1 c1(C(N2CC=CC(NC(COCCOC)=O)C2)=O)ccc2nc(C)nc(O)c2c1 c1(CC(N2C(CN(C(CCCOC)=O)C)CCC2)=O)ccc2nonc2c1 c1(SC)cc(C)c(C(=O)NCC2(F)CCN(C(c3c[nH]nc3C3CC3)=O)C2)o1 N1(C(c2c(CC)nns2)=O)CC(=O)CC1C(=O)NCC(C)(O)CCOC c1(C(N2CC3CCC2CN3Cc2cc3cc[nH]c3cn2)=O)cc(Cl)c(Cl)nc1Cl CCCC(C)(CC)C(=O)NC1CC(F)(CNC(c2cnccc2C)=O)C1 c1(CCC)c(C(N2CCC(C)(CNC(C3(C4CC4)CCCO3)=O)C2)=O)nnn1C N1(C(COCCC=C)=O)CC(NC(C2(CC3CC3)CCCO2)=O)CC(F)C1 C(C(C(C)(C)C)NC(=O)C(c1ccc(Cl)cc1)N(C)C)NC(c1c(C)ocn1)=O CC(C)C(CNC(=O)CNS(C)(=O)=O)NC(c1ncc(C(F)F)s1)=O c1(OC)cc(=O)n(C)cc1C(=O)NCC1=CCN(C(C2CC2(C)C(F)F)=O)CC1 C(CC(=O)NC1CCS(=O)CC1)(C(F)F)NC(c1cn(C2CC2)nn1)=O C12(NC(c3cc(C)ncc3)=O)CCCN(c3cc(C(C)C)nc(C(C)C)n3)CC1C2 C(=O)(CC(C)CC(=O)N1CC2(CC2)CC1C(=O)NCC(C)(C)n1ccnc1)OC c1(NC(CCc2c(N=[N+]=[N-])cccc2)=O)ccc(O)c2ncccc12 c1(C(N(C(C)CN(C(=O)CC2(C)CC2)C)C)=O)ccn(C(=O)OC(C)(C)C)n1 CC(CC(=O)N1CCCC(N(C(=O)CNC(c2cccs2)=O)C)C1)CC(F)(F)F C1(O)(C(=O)NCC2CC(NC(CN(C)CC)=O)C2)CCCC(C)CC1 C(CC(C)(C)C)(C(=O)N1CCC(CCNC(=O)CNC(=O)CC(C)(C)C)C1)OC c1(C(CNC(c2occ(C)c2C)=O)NC(=O)C(Cl)=CCl)ccc2ccccc2c1 c1(C(C)(F)F)ccc(C(=O)NC2CC(NC(c3ccc(C(N)=O)[nH]3)=O)C(O)C2)nc1 c1(C(=O)NCC2C(CNC(c3cc(C)nnc3)=O)C2)cccc2c1ccn2C c1(C(=O)NC2CN(C(c3c(Cl)cn(CC)n3)=O)C(C)C2)ccn2nncc2c1 C1(C(N2CC(CCCC)N(C(C34CC(C3)C4)=O)CC2)=O)CC2CSCC(C1)C2 C1(CN)CC2(CCCC2)CN1CCC(=O)Nc1cc(F)c(F)cc1F CCC(CNC(=O)C(Cc1cn[nH]c1)NC(=O)C(c1cnn(C)c1)=O)(CC)CO c1(C(=O)NC(CC=C)CNC(=O)C(CC)CO)cc(OCC(F)(F)F)cc(O)c1 N1(C(C2C(C)CN(C(=O)C(C(C)(C)C)C3CC3)CC2)=O)CCc2cccnc2C1 C(C(C)C(C)C(=O)N1CCCC1CNC(=O)C=Cc1cncc(O)c1)OC N1(C(c2ccc(CC)cc2F)=O)CCC(NC(=O)CC2CCOC2)C2(CCC2)C1 C(=O)(CC(C)(C)CC(=O)NCC(Cc1ccccc1)NC(=O)C(CC)CC)OC C1(C(=O)NC2C3(CCN(C(CS(CC)(=O)=O)=O)CC3)C2)COc2ccccc2O1 CC(=NOCC#N)C(=O)NC(CO)C(=O)N(CCCc1ccco1)C c1(C(=O)NC2CCC(C(=O)NCCS(C)(=O)=O)C2)ccc2nc(Br)sc2c1 N1(C(CN(CCC)C)=O)CCC(C(=O)NCCCn2nccn2)C1(C)C C1(C(=O)NCCC2OCCN(C(CNC(=O)CO)=O)C2)CCCC2(CCC2)O1 c1(C(N2CC(NC(c3n(C(C)C)cnc3)=O)C(F)C2)=O)sc(Cl)c(Cl)c1N C(C(C)(CC(=O)NCCN(C(C1CC(N(C)C)C1)=O)C1CC1)C(F)(F)F)N(C)C Cn1nc(C(F)(F)F)cc1NC(C1CCCC(C(F)(F)F)C1)=O C1(CC(=O)OCC)CC12CCN(C(=O)Cc1ccco1)CC2 c1(C(N2CCN(C(CC3C(C)(C)CCO3)=O)CC2)=O)nc2ccc(Br)cn2c1F C(CS(=O)(=O)c1ccccc1F)NC(C1C2(CC(OC(C)(C)C)C2)C1)=O C(=O)(C1=NOC(C)(C)C1)NC1C(CNC(Cc2cccc(OC(C)C)c2)=O)C1 C(=O)(CC(C)(C)C(F)(F)F)NC(C)(C)CCNC(=O)C(O)CC1CCOCC1 C=CC(C)(C)C(=O)NC1(C(=O)NCc2csc(C)n2)CC1 CC1(NC(c2cc(F)cs2)=O)CC(NC(c2cncn2C2CC2)=O)C1 C(=O)(CC(F)(F)CC(=O)OC)NC1CC2(CN(C(CCCC)=O)C2)C1 c1(CN2C(C(=O)NC3(C(=O)OC)CCOCC3)COCC2)ccc(O)cc1Cl C1(C2CC2)(NC(C2=CC(C)(CC)C2)=O)CCN(C(=O)C(C)(C)C(C)(C)C)C1 CCCC(CC)C(=O)NCC1CCCN(C(c2ccc(C3CC3)nc2C)=O)C1 c1(OC)c(C(N2CC=CC2CNC(C2CC2(F)F)=O)=O)csc1Cl c1(-c2onc(-c3c(C)cc(F)s3)n2)cc2occc2s1 c1(NC(C(Cc2cc[nH]n2)NC(=O)CCOC2CCC2)=O)ccccc1F C(C(C)(C)CNC(=O)CCCc1cccnc1)N(C)C(c1nocc1Br)=O C(=O)(C1=CCC(NC(c2ncnc(O)c2F)=O)C1)NC1CCC(CCCC)C1 c1(C(C)C)ncc(C(=O)NCC2CCC(NC(C3CC(C(F)(F)F)C3)=O)C2)[nH]1 N1(C(c2nc(OC)c(F)cn2)=O)CC2COCCC2(NC(=O)Cc2ccsn2)C1 C(CN=c1[nH]c(N2CCN(C3CC3)C(C)C2)nc2c1CCCCCC2)SCC=C C1(NC(=O)C=Cc2ccc(Cl)s2)CC2CC(NC(C3CC34CC4)=O)CC12 c1(C(=O)NCC(=C)F)ccc(CNC(=O)CC2C=CCC2)nc1 CC12CN(C(=O)C=CC3CC3)CC1CN(C(c1n[nH]cc1Cl)=O)C2 Cc1ccc2n[nH]cc2c1C(N1CCCC(C2(NC(C3CC3(C)C)=O)CC2)C1)=O C1(N(C(c2cnc(C(C)=O)s2)=O)C)CN(C(c2cc(C)sc2C)=O)CC1(C)C N1(C(C(=O)NCC(CC)OCC)=O)CC2(C(=O)OC)CCC1C2 c1(C(N2CCC(C3C(NC(=O)C(O)CF)C3)CC2)=O)ccc2cc(Cl)ccc2c1 C1(NC(c2cc(C3CC3)cs2)=O)CN(C(c2ncoc2Br)=O)CC1O C12(C)CCN(C1)C(C1C(CC)C1)C(=O)NC2.C(C)(C)(C)OC(=O)NC1CC1 C(CC(C(=O)NC1CC=CCC1)NC(=O)Cc1cccnc1C)SC c1(SCC(=O)NC2CCC(NC(=O)Cc3csnn3)CC2)ccccc1[N+](=O)[O-] N1(C(c2c(C)sc(Cl)n2)=O)CCN(C(=O)Cc2cnnn2C)CC(O)C1 C1(C(N2CCC(OCC=C)C2)=O)CCN(C(=O)C(C(C)C)SCC)C(C)(C)C1 n1(CC)ncc(CNC(C2CCC2NC(c2cc(C)n(C)n2)=O)=O)c1C N1(C(c2ccns2)=O)CCC2CCN(C(C3CC3CF)=O)C2C1 N1(C(C2(OC)CCSC2)=O)CCC2CCC(C1)N2C(C1COC1)=O Cc1cc(C(=O)NCC2CN(C)CCN2C(C2COCCO2)=O)cc(F)c1 C1(NC(c2cncc(C#C)c2)=O)CCCC12CCN(C(=O)CSC(F)(F)F)C2 c1(C(N2CC(C(C)NC(c3conc3C3CCC3)=O)C2)=O)cnc(N)c(CO)c1 C1(CNC(=O)Cn2ncc(Br)n2)CC2(C1)CN(C(C1C3CCCC13)=O)C2 c1(CNC(c2ccns2)=O)cn(C2CCCC2)nn1 CCC(C#N)C(=O)NC1CC(NC(=O)CCN2C(=O)CCC2=O)C1 N1(C(C2(CC#C)CCOC2)=O)CC(NC(C2(NC(N)=O)CC2)=O)C(C)C1 C1(CC)(NC(=O)CCc2nnc(C(F)F)o2)CCN(C(=O)CNC(C)=O)CC1 C1(CNC(C2CCN(C)C2=O)=O)CCCC2CN(C(=O)Cc3cc[nH]c3)CC12 Cn1cc(S(N)(=O)=O)cc1C(=O)NC1CC(NC(=O)C#CC(C)(C)C)C12CCC2 C1(Cc2nc(N(C)NC)c(C)cn2)CCN(C(=O)OC(C)(C)C)C(C)(C)C1 N1(C(C(c2c(C)cc(F)cc2)(F)F)=O)CC2(CCN(C(c3cnc(O)s3)=O)C2)C1 S(=O)(=O)(c1cc(Cl)c(OC(C)C)cc1Cl)N1CC2C(CC(=O)OCC)C2C1 CC1(C)COC(CC(N2CC(NC(C3(F)CCCCC3)=O)CC2CO)=O)CO1 C(CCC1CCC1)(C(=O)N(CCCO)CCO)NC(c1n(CC)nnc1)=O C1(C(=O)NCC2N(C(C(C)C(F)F)=O)CCC2)CN2CC3CC2(CO1)C3 C1(NC(C2C(c3ccn(C)n3)C2)=O)CCC12CN(C(=O)CC(C)(F)F)C2 C1(C(N2CC(CCCNC(C)=O)OCC2)=O)CCCN(S(N)(=O)=O)C1 c1(C(=O)NCC=C2CCN(C(C3CC(C)OC3=O)=O)CC2)cc(S(C)(=O)=O)co1 N1(C(=O)NCc2cc(C(C)(C)C)sc2)CCC(S(=O)(=O)CC)C1 c1(SC)ncc(C(N2CC(NC(=O)CN3CCSCC3)CC2C)=O)c(O)n1 c1(C(CC)C(=O)NCc2nnn(C(C)(C)C)n2)ccc(OC)c(OC)c1 Cc1c(C(=O)NCC2(O)CCN(C(C3CC(=O)NC(=O)N3)=O)C2)nn(C)c1N c1(C(=O)NCC(CC=C)NC(C2(CC#C)CCOC2)=O)nnn(C)c1CC N1(C(c2cn(CCC)nn2)=O)CC(O)CC1C(=O)NC(C)CCSCC C(=O)(C(C)(C)CC#N)NC(C)CNC(=O)CN(C)C CC1(C)OCCc2cc(C(=O)NCC3CN(C(c4ccccc4O)=O)C3)ccc21 C1(C(=O)NCC(C)(C)NC(C2CNC(=O)N2)=O)CCCC2(CCOCC2)O1 N1(C(c2ccc(F)cc2)CCOC)CC2CC1CN2C(=O)C(N1CCSCC1)C C1(C(N2CCCC(F)(CNC(C(=O)NCC(F)F)=O)C2)=O)CCc2c[nH]nc2C1 N1(C(c2nn(C)c(O)c2)=O)CCCC2(CCC(NC(=O)CCN3CCC3)C2)C1 c1(C(N2CCC(c3ccccc3)C2)=O)cc(N2CCC(O)C2)ccc1[N+](=O)[O-] C1(CC(=O)NC(CNC(c2nc(C)oc2)=O)CO)Sc2ccccc2NC1=O c1(CCC)cc(C(=O)NC(C2CCCN2C(=O)CSC(F)F)C)n[nH]1 C(C(CC(C)C)C(=O)NC1(C(=O)NCc2nc[nH]n2)CCCC1C)OC c1(C(N2C(C(C)(C)NC(CSCC#C)=O)CCC2)=O)cn(C)c(=O)cc1OC Cc1nc(C)c(C(=O)N(CCCCN(C)C(C2(N(C)C)CCCSC2)=O)C)[nH]1 CS(=O)(=NCC(=O)NCC(C(F)F)n1ccnc1)c1ccc(Cl)cc1.CC(=O)O N1(C(CCSC)=O)CCCC(N2CCN(C(C3CC=CCC3)=O)CC2)C1 c1(C(=O)NC2CC(F)(CNC(CC=C)=O)C2)cc(N)cnc1Br C1(C#CC(=O)NC2CN(C(=O)C(c3ccccc3F)C)CC2(C)C)(CC)COC1 c1(C(=O)NCC2CCN(C(C3(C)CSC3)=O)C2)nc(S(N)(=O)=O)c2ccccn12 N1(C(C2(CC(=O)OC)CC2)=O)C2CCC1CN(C(=O)CC1CC(CC)=NO1)C2 N1(Cc2c(Cl)ccc(Br)c2)CCC2(CC1)CSC2 N1(C(c2c(OC)ccs2)=O)CCC(NC(c2ccc(C)nc2OC)=O)CC1C c1(NC(C2C=CCN2C(c2cc(Cl)ncc2F)=O)=O)ccnc2c1CCO2 C=CCC(C(=O)N1CCOCC1CC(=O)N(C(C)CCO)C)OC C12(CNC(CC3(C=C)CC3)=O)CCC(CNC(c3nn(C)cc3Cl)=O)(CC1)CO2 c1(C(C)C)cc(C(=O)NCC2(NC(C3CCCC3O)=O)CCOC2)no1 C12(C(N3CC4(N(C)CC4)C3)=O)CCCC1CCN2C(=O)CC1CC(=O)C1 N1(C(c2cc(CC)c(O)cc2)=O)CCN(C(=O)C2=CCCSC2)C2CCCCC12 C1(C(=O)NCC(CC)NC(c2[nH]c(C)c(C(C)=O)c2C)=O)CCCS(=O)(=O)N1 N1(C(CC(C)=C(C)C)=O)CC(NC(=O)C=Cc2ccncn2)CC1C CC(C)CC(CNC(=O)CSCc1ccccn1)NC(=O)CCn1ccnn1 N1(C(C2CCCC(N(C)C)C2)=O)CC(C2CCN(C(C3(F)CC3)=O)CC2)C1 Cc1cn2cc(C(N3CCN(C(C4CCS4(=O)=O)=O)CC3CC3CC3)=O)nc2s1 c1(CCN(C)C)cn(CC2CC(F)(F)C2)nn1 c1(CCC(=O)N(C2CN(C(CCC)=O)CC2(C)C)C)c(C)nc2nc[nH]n2c1=O c1(C(=O)NCC2(NC(C(C3CC3)OCC)=O)CCOC2)cc(C)cc(C)c1O C(=O)(C(O)CC(N)=O)NCC(CNC(c1c(C)con1)=O)O C(C(C(C)C(C)C)NC(c1ccc[nH]1)=O)NC(c1nn(CC)c(C(F)(F)F)c1)=O C(=O)(C(C(C)(C)C)Sc1ccco1)NCC1C(C(=O)NCC(C)(C)C)COCC1 N1(C(CC)=O)CCC(CNC(=O)CCCC2CCCC(=O)N2)C12CC2 C1(NC(C(C)NC(C)=O)=O)CC2CCC1CC2NC(=O)C(C)C(C)(C)C C1(NC(C(C)(C)OCC)=O)CC(C)N(C(=O)CCCSc2ccc(C)cc2)C1 c1(OCCC)cc(C)c(Br)cc1CNC(=O)C(N1CC(F)(F)CC1C)=O c1(C(=O)OCC)cc2ccc(Br)cc2o1.c12cccc(C)c1NC2=O c1(C(N(CCC(N)=O)CC)=O)ccc(CNC(=O)COC2(C)CCCC2)o1 C=CCCC(C)(C)C(=O)NCCC1CCCN(C(=O)CNC(=O)CNC(C)=O)C1 CCC(C)CC(C)N(C)C(C1C=CCN1C(=O)CC1CCCCN1C)=O n1(CC)[nH]c(=NC(=O)c2cnccc2Cl)cc1C1CC1 c1(C(N2CCC(C)C2CNC(=O)C=Cc2cscn2)=O)cnc(O)c([N+](=O)[O-])c1 CC(C)(C)CC(F)C(=O)NC(C)(C)CCCC(=O)NC1(C)CC(C)(C)OC1=O N1(Cc2c(OC)cc(Cl)cc2)CC2CN(C(C3CC4C=CC3C4)=O)CC2C1 C(=O)(C1=CSCS1)N1CC(NC(C2N(C)CCC2)=O)(CO)C1 CN1CCC(C2CCN(C(c3cc(Cl)cc(Cl)c3F)C(=O)NC3CCOC3)C2)C1 C(=O)(CCC(=O)NN(C)C)N(CCCNC(C1CCN(C)C1=O)=O)C(C)C C(CC1CCc2ccccc21)n1c(CCC#C)nnc1N(CCOC)C(C)C C#CCC(C)(C(=O)NC(c1ccc(O)cc1)C)NC(=O)C=Cc1cncn1C N1(C(c2oc(C)c(CO)c2)=O)CC2N(C(=O)COCCCF)CCC2(C)C1 Cc1ccc(Br)c(CNc2cn(C)c(C(=O)Nc3cccc(C(C)(C)C)c3)n2)c1 C(=O)(C(O)CCCNC(=O)CC1CC2(CCC2)C1)NCCC#CCC c1(C(=O)NC2(C)CCN(C(C3C(=C)C3)=O)C2)ccnc2cc(Cl)ccc12 O=C(C(C1=CCCCCCC1)N1CC2CCCC1C2CO)NCCCF CCCCCCCC(=O)NCC1(F)CC(NC(c2ccc(Cl)c(C)c2N)=O)C1 CC(C)C(C(=O)NCC1(CN(C(=O)CCC2CCCCN2C)C)CC1)NC=O C=CC(C)(C)CC(=O)N1CC(CCCCNC(=O)CCC2CC2C)C1 Cc1nc(C2CC2)[nH]c1C(=O)NCC1CC(NC(c2c(Cl)cnn2C)=O)C1 c1(C(=O)NC(CSCC)C(=O)NC2CCN(C)C2)cccc(C)n1 Cc1ccc2[nH]nc(C(N3CCC3CNc3cc(C)ccc3[N+](=O)[O-])=O)c2c1 C(C)(C)(CC(=O)NCC1(F)CC(NC(=O)C=Cc2cnc[nH]2)C1)OC C1(C(=O)NCC2CC(Cn3cc(C(C(C)C)(F)F)nn3)C2)CCCC(F)(F)CC1 n1(CC(=O)NC2CN(C(CCN(CC)CC)=O)C3C2C3)ccc(=O)c([N+](=O)[O-])c1 CC(C)CC(CNC(c1ccc(CO)o1)=O)C(=O)NC(C1CCCC1O)C O=C1CC(C(=O)NCC2CCCN2C(=O)CC(F)(F)Cl)CCN1 C(=O)(CC(C)CN(C)C)NCCC1(NC(c2scc(C)c2)=O)CCC1 c1(C(=O)NC2(CNC(C34C(C(N)=O)(CCC3)C4)=O)CC2)cc(O)cc(Cl)c1Cl C1(C(N2CCC(C)(C)C(NC(=O)C(=O)NC3CC3)C2)=O)Cc2cccc(F)c2O1 Cc1cc(C(N2CCCCC(NC(=O)C=CC3(C)CCOCC3)C2)=O)ncc1F N1(C(c2c(C)nn[nH]2)=O)CCCC(C)(C)C1C(=O)N(C)CCOCCCO C1(NC(c2c[nH]c(Br)c2)=O)CCCN(C(c2coc(O)n2)=O)CC1 c1(C(=O)NCCN(CCC)C(C2(OC)CCSC2)=O)ccc2c(c1)C(=O)NC2 c1(OC)cc(CC(N2CC3(NC(=O)C(C)OC)CCC2C3)=O)ccc1[N+](=O)[O-] N1(C(C(CC=CC)C)=O)C2CCC1CN(C(C13CC(C(=O)OC)(CO1)C3)=O)C2 C1(C(N2CCN(C(CC(CC)C)=O)C(C)C2)=O)Cc2cccc(OC)c2O1 C1(N(C(C2CCOC2=O)=O)CC)CCCN(C(C2CCC2C)=O)CC1 C1(CCC(=O)OC)(CNC(=O)CNC(=O)CCOC2CC2)CCCC1 N1(C(CCC#C)=O)CCCC(O)(CCNC(=O)C=CI)C1 c1(COC)nocc1NC(=O)C(Cc1cn[nH]c1)NC(=O)C=CC(C)(C)C S(=O)(=O)(C1CCOc2ccccc21)NC(C1(c2cc(C)no2)CC1)=O c1(CC(N2CC(CC(C)NC(=O)CCc3ccsc3)C2)=O)cc[nH]c(=N)c1 C1(NC(c2c(SC)snn2)=O)CCCC12CCN(C(=O)COCCF)C2 N1(C(C(C)CO)=O)CCSCC1CCNC(=O)C(C)Oc1ccccc1 N1(C(C(C)SC(C)C)=O)CC2CC(C(=O)NC3(CCO)CCCCC3)CC2C1 C1(CNC(c2c(C)sc(Cl)n2)=O)CC2(C1)CN(C(C1CCCC1)=O)C2 Cc1ccccc1NCCc1nc(-c2cc[nH]n2)nn1-c1cccc(C(=O)O)c1 C1(C(=O)OC2CN(C(C(C)=O)=O)C(=O)C2)CCC(C)(C)CN1 C1(CNC(C=CC(C)(C)SC)=O)CC2CCC1N(C(c1nccc(Cl)c1F)=O)C2 CC1CC(O)CCN(C(C2CC(C)(NC(C3(CC4CC4)CC3)=O)C2)=O)C1 c1(CC(=O)N(CC(CNC(C(C(C)C)F)=O)O)C)csc2ccc(Cl)cc12 C12(C(N(CCC(=O)NC)C)=O)CC(CN(C(C3(F)CC3)=O)C1)C2 c1(OC)ccc2c(c1C(=O)NC(C1CN(C(=O)C3=COCC3)C1)C)CCC2 Cc1nn(C)c(C)c1C1CC(NC(C2CC2c2ccon2)=O)C1 CC(C)(C)CCCNC(c1sccc1CNC(=O)CCCC1CCC1)=O N1(C(c2c(C)nc(O)[nH]2)=O)CCC2(CC(NC(c3coc(Cl)n3)=O)CO2)C1 C1(C(N2CCCC(Cn3cc(CCCOC)nn3)C2)=O)CCc2nnnn2CC1 c1(CC(=O)NC(C)(C)CCCNC(C2(O)CCSCC2)=O)ncc(F)cc1F N1(C(C2(COC)COC2)=O)CCC(CCNC(=O)Cn2ncn(C)c2=O)CC1 Cc1nc(O)nc(O)c1CC(=O)NC1CCC12CN(C(C1CC3CCC3C1)=O)C2 C1(C(=O)NCC2(F)CN(C(C(C)(C)OC(C)C)=O)C2)CCC12CCCO2 C1(c2cn(C)nc2)CN(C(c2cnn(C3CCCCO3)n2)=O)CCO1 C1(C(N2CCCC(CC)(NC(=O)C(Cl)=CCl)C2)=O)CC2C=CC1CCC2 c1(C(C)NCC2CNC(=O)C2)c[nH]nc1S(=O)(=O)N1CC2COCC2(C(=O)OC)C1 N1(C(C(C)(C)n2cccn2)=O)C2CCC1CC(NC(C1Cc3nncn3C1)=O)C2 C(C)(C(=O)NCCC1(C(=O)NCC2CCCO2)CCC1)=C(C)C C(C(=O)N=c1ccn(CCO)[nH]1)CC(C1N(C(C=CC(C)(C)C)=O)CCC1)(C)C CS(=O)c1cccc(C(=O)NC2CN(C(c3ccc(Cl)cn3)=O)CC3CC23)c1 c1(CC)nn(C)cc1C(=O)NCc1cn(C2CN(C(=O)C(C)C(C)O)C2)nn1 c1(C(C)NC(=O)OCC)ccc(NC(CSC)C(F)(F)F)c([N+](=O)[O-])c1 c1(C(N2CC3(CCN(C(Cc4c(C)non4)=O)C3)C2)=O)cc2c(cn1)OCCC2 N1(C(C(C2N(C(c3cncc(C)n3)=O)CCC2)(C)C)=O)CC2(CCOC2)C1 c1(C(N2CC(OC)C(NC(=O)C(C)NC(C)=O)C2)=O)ccc(S(C)(=O)=O)c(C)c1 N#CC1(C(=O)NC2CC2CNC(c2cnn(C3CCCCC3)c2)=O)CCSCC1 Cc1nc(C(=O)NC2CC2NC(C2CCC(=O)N2C)=O)c(C)n1C C(=O)(C(O)C(F)(F)F)N(CC(C)N(C)C(c1cccc(CO)c1)=O)C Cc1nc(=N)[nH]cc1C(=O)NC1CC1NC(c1cnc(C(C)(C)C)nc1)=O Cc1cccc(Cc2ccc(CN(C(=O)C(=O)N(C)CCN3CCC3)C)cc2)c1 CC1CN(C(C2CCC(NC(c3cc(O)ccc3Cl)=O)C2)=O)CC(C)O1 Cn1cncc(C(=O)NCCCCCCNC(c2cccc(OC(F)F)c2)=O)c1=O C1(CC(=O)NCCN(C(=O)CC2SC(=N)NC2=O)C)COC(C)(C)C1 c1(OC)c(C(=O)NC(C2CCCN2C(C2CC2c2ccsc2)=O)C)c(C)nn1C C(=O)(CCS(=O)(=O)N(C)C)N1CC(CC(C)NC(c2ccnc(CO)c2)=O)C1 C(=O)(C1=NN(C(C)C)C(=O)CC1)N1CCC(F)(CNC(c2cccc(C)n2)=O)C1 c1(C(=O)NC2CC(C)(C(N3CC(NC(=O)NC)C3)=O)C2)cnc2n1CCC2 C1(C(=O)NC2C(C)N(C(=O)CN3CCOCC3)CC2)Cc2ccccc2C(=O)O1 C1(C(N(CCC(=O)NC)C)=O)C2CCC(C2)N1C(C1(O)CCOC1(C)C)=O Cc1ccc(-c2nc(C3CC3(C)C)nn2C2CSC2)c2c1CCCN2 CN1CCc2cc(C(=O)NCC(F)CNC(C3OCCOC34CCC4)=O)ccc21 c1(OC)cc(C(=O)NCCCN2CCCCCC2)cc([N+](=O)[O-])c1 N1(C(C(CC)COC)=O)CCN(C(=O)CCc2c(C)noc2C)CCC1C CC1CCC(CNC(=O)Cc2cc[nH]n2)CN1C(=O)CNS(C)(=O)=O C1(C(N2CC(N(C(=O)CC3CCC(=O)N3)C)C2)=O)CC12CC(O)C2 c1(OC)ccc(C(N2CCCC2CNC(=O)CCc2ncc[nH]2)=O)c(C)n1 c1(C(C)C)ccc(C(=O)NCC=CCNC(=O)C(C)Oc2ccccc2Cl)nc1 CC1C(NC(C2CCC(F)(F)C2)=O)CCN1C(=O)CCC(=O)c1cccc(F)c1 N1(C(=O)NCCn2cnc(C(=O)OC)n2)CCC(C(=O)OC(C)(C)C)CC1C CC(C)C(CNC(C1CCCS1)=O)C(=O)NCCN1CC=CCC1 C1(C)(C(=O)NCCCNC(CNS(CCOC(C)C)(=O)=O)=O)CCC(C)C1 N1(C(c2ccc(C)o2)=O)CC(NC(C23CC(F)(C2)C3)=O)C(C2CC2)C1 N1(C(C=Cc2cn(C)nn2)=O)CCC2(CC1)CC2NC(C1(Br)CC1(F)F)=O N1(C(c2c(=N)[nH]cnc2)=O)CCN(C(C2CCC(=O)NC2)=O)C2CCC12 N1(C(C(CC)C2CCOCC2)=O)CCC(CO)(NC(C2CCCSC2)=O)CC1 c1(C(N2CCC(C3(C)NC(=O)NC3=O)CC2)=O)n[nH]c2cc(N)ccc12 C1(OC)CCCN(C(c2ccnc(Br)c2)C(=O)Nc2ccc(F)cc2)CC1 c1(C(N2CC(CC=C)(NC(c3scnc3Cl)=O)C2)=O)c(Cl)cnn1C(C)C C(=O)(N=c1cc(-c2ccc(Cl)cc2)o[nH]1)NCC1CCN(S(C)(=O)=O)C1 C(CCCCCC(=O)N1CCN(C2(C)CC2)CC1)NC(C(CC=CC)C)=O Cc1ccc(CC(=O)NCC2CCN2C(C2CCOC2C(C)C)=O)cc1C CC(C(C)(C)C(=O)N(C1CC2CC2C1)C)NC(=O)C(O)C(F)(F)F C(N=c1[nH]c(Cl)c(C#N)s1)C1CC2N(C(CN3CCN(C)CC3)=O)C(CC2)C1 C(C1=NOC2CN(C(=O)C=C(C)Cl)CC12)NC(c1cc(CC)no1)=O Cc1ccc(C#N)c(NCC2(C)CCC(NC(=O)CSc3ccccn3)O2)n1 c1(C(=O)NC2CCC(N(C)C(C3CC4CCC3O4)=O)CC2)cccc2cnnn12 N1(C(C(C)NC(Cc2nc(C)oc2)=O)=O)CC2(CO)CCC1CC2 CCC(C)(C(=O)NC1C2CC1N(C(c1nnc(O)cc1O)=O)C2)C(N)=O C1(CNC(=O)NC(CCC)c2ccco2)CCC2(C1)CC2(F)F Cc1c[nH]c(C(=O)NCC(CC(C)C)NC(C2(C)CCCC2)=O)c1C C1(CC#N)CN(C(=O)C(=O)NCC2CCOC(c3ccccc3)C2)CCC1(F)F C(=O)(CCCCC(C)C)NCCC(CNC(c1c(OC)ncnc1OC)=O)(C)C c1(C(=O)NC(C2CCN(C(c3cc(O)no3)=O)C2)C)ccc(N)c(N)c1 c1(-c2cc(OC)cc(C#N)c2)n[nH]c2ncc(C(=O)NCCN(C)C)cc12 N(C(=NCCCCl)NC1CC1)CC1(C)CCCCC1O.c1ccccc1 C1(C(=O)NC2CC(Cl)(Cl)C2)CC(O)CN1C(c1cnns1)=O C=CCCCCCC(=O)N(CC(C)O)CCNC(c1cnc(NC(C)=O)o1)=O C1(CC(=O)NC2CCC(NC(c3cc(C)ncn3)=O)C2)OCCOC1(C)C c1(C(C(=O)NCC(c2c(CC)cccc2)N)O)ccc(Cl)cc1Br Cc1cnc(C(c2cccs2)NC(=O)CC2CCCCN2)s1 C(=O)(C(CCC1CC1)NC(=O)CSCCC)N1CCC(CCC=C)C1 C(C(CC(F)(F)F)NC(=O)C(C)COC)NC(c1cnc(OCC)s1)=O Cc1cc(C(=O)NC(c2cccnc2)C(=O)Nc2cccc(O)c2)nn1C C1(NC(c2nc(CCCC)sc2)=O)CS(=O)(=O)CC1NC(=O)C1CC1 N1(C(C(c2ccco2)NC(CCc2n(C)cnn2)=O)=O)CCOC2(CCC2)C1 c1(C(N2CCC(CCNC(C(COC)(C)OC)=O)CC2)=O)cc(F)cc(Cl)c1N c1(C2(C(=O)NC(C(=O)OCC)C(=O)OCC)CC2)c(C)[nH]c2ccnn2c1=O c1(CC)ccc(C(=O)NC2CCCCCN2C)c(C)c1 c1(C(N2CCCC(N(C(C(=O)NCC)=O)C)C2)=O)c(SC)nc(O)nc1C C1(C(=O)NC(CC)CNC(C2(C)CC(C)=NO2)=O)CC2CCCCCCC12 c1(COCCNC(C(=O)Oc2ccc(F)cn2)=O)ccc(OC2CCC2)cc1 N1(C(Cc2c(C)ccc(C)c2)=O)CC2CCC1C(C(=O)NCCC(C)O)C2 Cn1cc(Cl)cc1C(=O)NCC(=C1CN(C(c2cnnc(C3CC3)c2)=O)C1)F C1(C(=O)NCC(N2CCCCC2)C)CCN(C(=O)Cc2ccn(C)n2)C(C)C1 C12(CC(N3C(C)CC(NC(CCCC(C)=O)=O)C3)=O)CCC(CC1)C2(C)C N1(C(c2c(OC)ccnc2F)=O)CC2CN(C(=O)C3=CC(C)(CC)C3)CC2C1 C1(O)(C(N2CCC(COC)(NC(=O)Cc3cscn3)C2)=O)CCCC(C)(C)CC1 C(=O)(C(O)Cc1cnc[nH]1)NCC(CC)N(C(=O)CC(C)n1ccnc1)C Cc1ccc(OCC(=O)NCC(CO)NC(=O)C(C)(C)O)c(C)c1 CCC(CC(=O)N(CCCCNC(c1ccc(OC)cc1OC)=O)C)C(C)C C12(C(N3CCC(C)C3)=O)COCC1CN(C(c1ccc(O)c(I)c1)=O)C2 O=C(CC1=CCN(C(=O)C(F)C(F)(F)F)CC1)N1CCC(n2cncn2)C1 CC(F)C(C)N=c1[nH]c2c(c(=NCC3(c4cccc(C#N)c4)CCC3)[nH]1)COC2 CC(C)(CNC(=O)Cc1nncs1)CC1CN(C(=O)CSc2ccccn2)C1 N1(C(=O)Cn2cnccc2=O)CCN(C(C2CC(CF)C2)=O)C2CCCCC2C1 c1(C(=O)NC(CNC(C2(CCOC)CCC2)=O)(C)C2CC2)ccc(C)o1 N1(C(Cc2cc(CC)no2)=O)CC(CC(N2CC=CC2COC)=O)C2(CC2)C1 C1(CNC(c2snc(O)c2Cl)=O)C2CN(C(C3(CO)CC3)=O)CC12 C=CC(C)(CCOC)C(=O)N1CCC(O)(CCNC(C2CC2COC)=O)CC1 N1(C(C(CC)(C)O)=O)CCOC2(CCN(C(=O)C(C)(C)S(C)(=O)=O)CC2)C1 N1(C(C=NOC)=O)CCC=C(C(=O)N(CC(=O)NC(C)(C)C)C)C1 N1(C(Cc2nc(C)sc2)=O)CCC(NC(c2cnc(C)s2)=O)CC1C N1(C(CC(C=C)C)=O)CCC(CC)(NC(=O)CC(F)(F)c2ccccc2)CC1 c1(C(=O)NC(CNC(C(C(C)(C)C)NC(C)=O)=O)(C)CO)cc2c(o1)CCCC2 Cc1nnc(C(C)NC(c2conc2C(C)NC(c2ccoc2Cl)=O)=O)s1 CN1CCCC1C1CCCN1C(c1cc2c(Br)cccn2n1)=O S(=O)(=O)(c1ccc(N2CC3CCC2C3)c(Cl)c1)NCC1(C)CC(F)(F)C1 C(=O)(C(CCC(N)=O)n1cc(-c2cccc(Cl)c2F)nn1)NCC1(S(C)=O)CC1 CCCC(C(O)C(=O)NCC(F)F)NC(=O)Cc1cccnc1 N1(C(C=C(C)C)=O)CCC2(CCOCC2C(N2CCCC2CN(C)C)=O)CC1 C1(NC(CCC2(C)CN(C(C3CC3[N+](=O)[O-])=O)C2)=O)CCC=CCCC1 C1(C(=O)NCC(C)OC(C)(C)C)CCCCN1N=O.c12ncc(cc1Cl)[nH]2 CCC(CC)C(C)C(=O)N(CCNC(C1CC1C1CCOCC1)=O)C1CC1 CC(C)CC(CNC(=O)CC1CCC(C#N)C1)C(=O)NC1CNC(=O)C1 Cc1ncnc(C)c1C(=O)NC(C)CCNC(c1ncccc1CN(C)C)=O C1(C(N2CC(O)(C(C(=O)NC(C)(C)C)F)C2)=O)CC12CCCC2 Cc1cc(F)c2cc(C(N3CC(C)C(NC(=O)CN(C)C)C(C)C3)=O)[nH]c2c1 n1(CCNC(C2CC(OC)C2)=O)ccc(C(=O)NCC2CC(CO)CO2)c1 N1(C(C23CCC(NC(CN=[N+]=[N-])=O)(CC2)C3)=O)CCCC2CCCC12 Cn1ccc2ccc(C(N3CCC(NC(C4CC(C#N)C4)=O)C3)=O)cc12 N1(C(C(C)C2CCC2)=O)CCC(NC(=O)C(O)c2ccsc2)C1 C#CC1(O)CCN(C(=O)CC2(NC(C3CC(CCC)C3)=O)CCC2)CC1 C1(C(C)NC(CC=C)=O)CN(C(C2COCCN2C)=O)CCO1 C1(F)(CNC(CC(C=C)(C)C)=O)CCCN(C(C2CC=CCC2)=O)CC1 N1(C(CCOCC)=O)CCCC(C(C)C(=O)N2CC(CC(F)F)C2)C1 c1(OC)cc(Br)cc2c1C(NC(C1CC(S(C)(=N)=O)C1)=O)CC2 N1(C(C(C=C)O)=O)CCC(NC(C2CC(N(C)C)C2)=O)CC1 N#Cc1cc(-c2ccc(NC(c3ccc4c(c3)CCO4)=O)s2)cc(F)c1 N1(C(CC=C(C)C)=O)CCC2CC2(NC(=O)CN(C2CCCCCC2)C)CC1 C1(C(=O)OCC)CCN(C(=O)CCN(C(=O)CCOC2COC2)CCO)C1C C1(C(=O)OC)C=CCCN1C(=O)C(=O)N(C)Cc1cscc1Br c1(OC(C(=O)N(CC(C)NC(C2SCCS2)=O)C)(C)C)ccc(Cl)cc1 C1(C(=O)NC2CCC(NC(c3coc(O)n3)=O)CC2)CC2CCCCCCC12 c1(OCC)cc(C(=O)NCCCN(C)C(c2cnn(CC3CCOC3)c2)=O)[nH]n1 N1(C(C(c2cccc(C)c2)F)=O)CC2(CCN(C(=O)CC3CCCO3)C2)C1 Cn1nc2c(c1C(c1nnnn1-c1ccccc1)NCCn1ccnc1)CCC2 C1(CCOC)CN(C(c2ccc(OC)s2)=O)CCN1C(C1CS(=O)(=O)C1)=O C(CN=c1ncc(F)c[nH]1)NC(C1CC(=O)N(CCO)CC1)=O N1(C(C=C(C)CN2CCOCC2)=O)CCC(N(C)C(C2CCCC(=O)N2)=O)CC1 C1(C#N)(C(N(CC)CC2CCN(C(C3(C)CCCO3)=O)CC2)=O)CCCOC1 C(=O)(C1=NOC2(CCCN(C(c3cc4cccnn4n3)=O)C2)C1)NCC(C)O N1(c2cc(C)[nH]n2)CCN(C(C(=O)NC2CCOC2)C2CC2)CC1 C1(CN=C(NC2C(C)CN(C)CC2)NC2CCCC2)CCCCC(F)(F)C1 CCC(C)C(O)CC(=O)N1CC=C(C(=O)N2C(CO)CC2CO)CC1 C1(NC(CCC)=O)CCN(C(=O)CC(C)(C)C#N)CC1CO c1(CN2C(=O)CN(CC(CCCC)CC)C2=O)ccc2c(c1)C(=O)NCCC2 C(c1ccccc1)=CCSCC1C(=O)OCC1 C#Cc1cccc(C(N2CCN(C(C3CC(C)=NO3)=O)CC2C2CC2)=O)c1F c1(SCC)cccc(C(=O)NCC2CCCC(NC(c3sccc3OC)=O)C2)c1 C1(NC(C(CCSC)O)=O)(CO)CCN(C(c2cccc(Cl)c2Cl)=O)CC1 c1(C(=O)OCC)cnccc1C1C(C(F)(F)F)(C(=O)NCCC(=O)OC)C1 C1(C(=O)NCC2CCCN(C(=O)Cn3cnnn3)CC2)C2CCN(CC2)S1(=O)=O CCCC(CCC)CC(=O)N1CC(n2cc(COC3COC3)nn2)C(C)C1 C#CCCCC(C)C(=O)N1CC(CNC(C2CCS(=O)(=O)CC2)=O)OC(C)(C)C1 c1(NC)cc(Cl)ccc1C(N1CCC(C(C)NC(C2CC2OC)=O)CC1)=O N1(C(C(CC)COC)=O)CCC2(CCCN(C(c3nnc(C(C)(C)C)s3)=O)C2)C1 C1(NC(CC)=O)CCCN(c2nnc(CCCSC)n2CC2CC2)C1 c1(C(=O)NC2CC(CNC(CN3C(C)CCC3C)=O)C2)ccc2n[nH]cc2c1 c1(CC(=O)NCC(C)NC(COc2ccc(C)cc2F)=O)c(C)cc(C)cc1C CC(C)C(O)C(C)C(=O)NC(C(N1CCCC(F)(F)C1)=O)c1ccco1 CC(C)C(F)(CNC(c1cc(C#N)ccc1N)=O)C(=O)NC1(C)CCNC1=O c1(C(=O)NCCCC(C)NC(=O)C(C)(C)Cc2cnn[nH]2)cc(Cl)ccc1Cl c1(C(N(C2CCC(C)(C)C2)CC)=O)cc2nc(-c3ccco3)cc(C(F)(F)F)n2n1 CC1(C)CN(C(=O)CCC#N)CCN(C(C2CCC3(CCC3)O2)=O)C1 C1(C(=O)NCC2C(NC(=O)CC3CCCCC3)CCC2)CCCC2CCCN12 C1(NC(c2nccc(OC)c2)=O)CCN(C(=O)Cc2ccnc(F)c2F)C(C)C1 c1(CC(=O)NC(CNC(CCOCC)=O)C2CC2)cc2ccccc2c(=O)o1 C1(NC(C2(C(C)C)COC2)=O)CN(C(=O)CC2CC2)CC1C#N c1(C(=O)NC2CC(C)N(C(C3COCCOC3)=O)CC2)cncc2ccccc12 C1(C(=O)NC2CC(NC(c3ccn4ncccc34)=O)C2)CCOC2(CCCC2)C1 C1(NC(C=CC)=O)CN(C(=O)Cn2cc(C3CC3)cn2)CC(C)(C)C1 O=C1CC(CNC(=O)CC2CC2CNC(=O)COCC2CCC2)CCN1 c1(CC)ccc(Cl)c(NC(=O)C(N2CCCC(O)(c3nn[nH]n3)C2)=O)c1 N1(C(Cn2ncc(C(=O)OC)c2)=O)CCC(N(C)C(C2CC2C(N)=O)=O)CC1 c1(C(=O)NCCCCCCNC(C2C3C4CCC(C4)C23)=O)cc2c(o1)CCCC2 C1(C(N2CCC(CN=c3[nH]nc(CC)s3)C(C)C2)=O)C(O)C(=O)N(C)C1C N1(CC(=O)Nc2n(CCC)ncc2)CCCC(NCc2ccc(OC)cn2)C1 C(CF)(C(F)(F)F)NC(C1C=CCN1C(C1CC1(F)Cl)=O)=O C=C=CCCC(=O)NCc1cc(C(=O)NCCC(O)C2CCCC2)co1 C1(NC(CC2C(C)(C)OCCO2)=O)CCC2(CC1)CC(NC(C1CCSC1)=O)C2 C1(C(N2CCN(C(C#C)C)CC2)=O)CCCC(NC(c2csc(O)n2)=O)CC1 C(=O)(C1CSc2ccccc21)N1CC(O)(CCNC(C(C(C)(C)O)(F)F)=O)C1 N1(C(COC)=O)C(Cn2cc(-c3nccs3)nn2)CC2CCCC12 N1(C(c2cc(C)sc2C)=O)CCC(C)(C)C(CNC(=O)CC2CC=CCC2)C1 C1(NC(C2C(C(N)=O)C2)=O)CC12CC(NC(c1ccncc1)=O)C2 CC(CC#N)C(=O)NC(C(=O)NCCOC1(C)CCC1)C1CCCC1 N1(C(CC2(CC)CCC2)=O)CC(O)CC1(C)C(N1CCC(CC(N)=O)CC1)=O C1(CCCCC)CCC(C(=O)NC2CC(C)(NC(C3CCS3(=O)=O)=O)C2)O1 c1(CN2CC(CCC)OCC2)c2n(c(C)cc1=O)CCC2 C(N=c1[nH]c(=NC2C=CC(C)(C)CC2)c2[nH]ccc2[nH]1)C1(OC)CC1 CC(C)CC(C(=O)N(CCCCN(C(=O)CCc1cccnc1F)C)C)C(N)=O N1(S(c2ccc(C(=O)O)o2)(=O)=O)CCCCCCCCCCCC1 c1(NCC2(OCC)CCCCC2)nccc(=NCCc2cncc(F)c2)[nH]1 c1(NC(C2CCN(c3ncc4[nH]ccc4n3)CC2O)=O)cc(Br)ccc1[N+](=O)[O-] C1(NC(c2cc(C)no2)=O)CC2(CCC(CNC(C3(C)C=CCC3)=O)OC2)C1 C(CCN=c1[nH]c(=NCC(CC)(CC)C(N)=O)[nH]c2cc(C(F)(F)F)ccc12)SC N1(C(CCCOCC)=O)CCCC(NC(CN(C)CC2(C)CCCCO2)=O)C1 CC(CCNC(=O)CCc1ncc[nH]1)NC(C1CC1CF)=O c1(-c2ccc(NC(c3cc(Br)ccc3F)=O)cn2)ccc(F)c(O)c1F C(C1CCC(C)CC1)=C(C)C(N1CCC(CN(C)C(c2cccc(Br)c2)=O)C1)=O C1(C)(NC(C=CCC(C)(C)NC(CC(COC)(C)O)=O)=O)CCC2(CC1)CC2 C1(C(=O)NCC(C(C)C)C(C)C)CC2C=CC1N(C(=O)C1=NOCC1)C2 C#CCCCC(=O)NCC1(O)CCN(C(c2ccc(SCC)cc2)=O)C1 c1(CC)ccc(C(=O)N(C)CC2(NC(=O)C(CCSC)NC(N)=O)CC2)c(F)c1 CC(CCl)(CCl)CS(=O)(=O)Oc1c(Br)cccc1Br C(CC(=O)OC)N(C(=O)C(C)NC(C1CCSC1)=O)CC=C N1(C(c2ccn(C3CC3)n2)C(=O)NCCC(=O)OCC)CCOC(C)C1C c1(C(=O)NCC(C)(CC)NC(C(CC)C)=O)c(C)nc2sc(C)nn12 c1(OCC)cccc(C(=O)NCC(F)CNC(=O)CCOC(C)C)c1 c1(OC)cc(NCC2CCCN(C(=O)COCC3CCCC3)C2)nc(OC)n1 C(=O)(C1=NOC(C)C1)NCc1c(C(=O)Nc2c(CC)noc2)cccn1 N=c1nc(N2CC(C(N)=O)C(C(N)=O)C2)[nH]c(=NCCS(=O)CCNC)[nH]1 c1(CC)cc(C2CC2)nc(N2CCCC(C)(NC(=O)C#CC3CC3)C2)n1 N1(C(C2CC2C2CC2)=O)CC2CCN(Cc3ccc(Br)cc3O)C2C1 C1(NC(c2ccc(N(C)C)nc2)=O)(CO)CCCN(C(=O)CC2CC3CC3C2)C1 c1(C(N2CCN(CC(CNC(C3(SC)CC3)=O)C)CC2)=O)ccc2oncc2c1 C(=O)(CCCC(=O)NC1COCC1NC(=O)CN1CC(=O)NC1=O)OCC n1(CC)nc(CNC(=O)C(C2CCC(F)(F)C2)O)c(Br)n1 C1(C(=O)NCCCn2cc(C(CSCC)C)nn2)CCc2ccccc2OC1 C(CCCCC(=O)NC1CN(C(=O)CC2CN(C(C)=O)C2)CC1OC)OC CC(C)CCCCCC(=O)NCC1CCCCN1C(C1CC1F)=O c1(CCC)[nH]ccc1C(N1CC(NC(C2(COC)CC(=O)C2)=O)C1)=O C1(CC(=O)NC(C(O)CO)C2CC2)(OC)CN(C(c2sccc2F)=O)C1 c1(OC)ccc(C(=O)NC(C)CNC(C2(c3ccno3)CC2)=O)c(N)c1 C1(CNC(CCCC)=O)CN(C(=O)CC(CC)SC)CCC12CCOCC2 Cc1ccc(F)c(C(=O)NCC2C(C)CCCN2C(=O)CC2COCCO2)c1 c1(C(C)(C)C)nnc(C=CC(=O)NC2CC(Cl)C2)o1 c1(OCCCc2cn(C)nc2)ccc(Cl)c([N+](=O)[O-])c1.C1C(C2CC2)NC(=O)N1 N1(C(C2C(C)C(=O)C2)=O)CCOC(CNC(=O)CC2CC3CC3C2)C1 N1(C(C2(CCC=C)CC2)=O)CCCC(F)(C(=O)N(CC(C2CCCC2)O)C)C1 Cc1c(C(=O)NCCNC(=O)Cc2cn(C)nn2)oc2c1ccc1ccccc21 C(C1=CCCCCC1)(c1nnnn1C1CCCC1)NCCCC(=C)Br C(=O)(C(CC(C)C)C(C)C)N1CC(CC)N(C(c2sccc2OC)=O)CC1 CC1(C)CC(NC(=O)CC(C)(C)NC(c2ccc(CO)s2)=O)C(=O)O1 Cc1ccnc(O)c1C(=O)NC1CCC(NC(C2CC3(CCC3)C2)=O)C1 O=C1OCCc2ccc(C(N3CCC(CCNC(C4(Cl)CC4)=O)C3)=O)cc21 c1(C(=O)Nc2nnc(SC(C)C)s2)coc2c1C(O)CCC2 N(C(=NCCF)NCc1cn(-c2ccccc2OC)nn1)CC(C)(C)OC.C1(C)CC1 N(C(=NCCS(=O)(=O)C1CCOCC1)NC1CCC1)C1CCC(=O)NC1 C(c1cn(C)nn1)=CC(=O)NC(C(=O)NCCCN(CC)CC)CC1CC1 N1(C(CC(C)N(C(c2ccc(=NC)[nH]c2)=O)C)=O)CCC(C)C2(CCC2)C1 C=CC(C)(CCOC)C(=O)N1CC(N(C)C(c2csc(O)n2)=O)C1 c1(C(N2CCN(C(C3(C#C)CC3)=O)CC(CO)C2)=O)ncnc2c1c(Br)cn2C c1(C(N(C)Cc2ccc(Br)c(Cl)c2)=O)cc(F)cc(Br)c1Br C1(NC(=O)Cn2cnnc2)CCN(c2nnc(C(F)F)o2)CC12CCC2 N1(C(C(C=C)O)=O)CCn2ncc(CNC(C3CC3c3ccn(C)n3)=O)c2C1 CC1(C)CCC(C(=O)N(CC(N2CC3(CCC3O)C2)=O)C2CCC2)CO1 C#CC1CCN(C(C2CCCCC2CNC(C2CC(n3cnnc3)C2)=O)=O)CC1 C12(CNC(c3n(CC)ccn3)=O)CC(CNC(=O)CC3(CSC)CC3)(CO1)C2 c1(C(N2CC(C(N)=O)(CNC(=O)CC3CCC4CC34)C2)=O)n[nH]c2ccccc12 C1(CNC(C2C(SCC)C2)=O)OCC1(C)C C1(C(N(CC(=O)N(CC(F)Cl)C)CCC)=O)COCCN1CC N1(C(c2cccc(OC)c2Cl)=O)CCC2(CCCC2NC(=O)CNC(N)=O)C1 CC(O)CCCCCC(=O)N1CCC(CC(N)=O)(NC(=O)CNC=O)CC1 C1(NC(=O)C(F)CC2CC2)CC(F)CN(C(c2ccsn2)=O)C1 c1(C(=O)NCC(CNC(C2(COC)CC2(F)F)=O)O)cccnc1S CCCC(C)(O)CC(=O)NCC1(F)CC(NC(c2cc(Br)cn2CC)=O)C1 N1(C(CCNC(COC)=O)=O)CCC(O)(CNC(=O)CC2CC(NC(C)=O)C2)C1 Cc1n[nH]c2cc(C(=O)NC(CNC(=O)C3=CCCS3)C(C)C(C)C)ncc12 C1(NC(c2cc(F)n[nH]2)=O)COC2(CCN(C(c3cccc4nsnc34)=O)C2)C1 C1(C(N2C(CNC(C3CN(C)C(=O)N3)=O)CCC2)=O)CC2COCC(C1)C2=O CC1CCN(C(C2(N(C)C(C3CC(=O)CCO3)=O)CC2)=O)CC1O N1(C(CCc2scc(C)n2)=O)CCC(C2CCN(C(C3CCCSC3)=O)CC2)C1 c1(NC(C(CNC(C)=O)(C)C)=O)c(C)cc([N+](=O)[O-])cc1Br C=CC(CCC)CC(=O)N1CCC2CC12C(=O)NCC1CCN(CCC)C1 Cc1nnc2n1CCC2(C)C(=O)NCCNC(=O)C(C)(C)CC1CCCCC1 CN1CCCC(C(=O)NC2CN(C(C3(C#N)CCCO3)=O)CC2F)C1 c1(CC)nc(CCNC(=O)C(C2(C)CC2)NC(c2cocn2)=O)n[nH]1 C1(CCNC(c2scc(C)c2C)=O)CCCN(C(C2CC3(CCC3O)C2)=O)CC1 C1(C(=O)NCC2(O)CCN(C)CC2)(CC)CCN(C(=O)CCC2CCOC2)CC1 c1(CCC(=O)NCC2C(NC(c3c(CC)noc3)=O)CCC2)ccccc1SC Cc1cnnc(O)c1C(=O)N(C)CCOCCNC(=O)CC1CCCN(C)C1 Nc1cccc(CC(N2CCCC2CNC(=O)CC(C2CCC2)C2CCC2)=O)c1 Cc1cc(=O)n(C)cc1C(=O)N(CC(N1CCCC2(C1)N=N2)=O)C Cc1cc(CCC(N2CC(C)(NC(c3cc(C(F)F)ncn3)=O)C2)=O)c(C)s1 C1(NC(C2CN3CCC2C3)=O)CCCCC1C(N1CC(CCO)C1)=O C1(NC(c2ccc(OC)s2)=O)CCC2(C1)CN(C(c1ccc(F)c(F)c1C)=O)C2 C1(NC(c2c(OC)nccc2)=O)CCCN(C(=O)COc2ccccc2)C1C.C(C)(=O)O C1(CNC(CC(CC)SC)=O)CC(C)(C)CN1C(c1cnn2ccsc12)=O c1(CNC(C(C(C)C)(C)C)=O)ccc2c(c1)CN(C(=O)C(O)C(F)F)C2 C(C(C(C)C(C)C)NC(c1ccoc1C1CC1)=O)NC(C1(CCCC)CCC1)=O c1(NC)ccc(F)cc1C(=O)NCCC(C)(C)NC(=O)CC(C)n1ccnc1 C1(C(N(C)CC2CCC(CNC(CCCOC)=O)CC2)=O)OC2CCC1CC2 C#CC1(C(=O)NC(c2cccc(C)n2)C)CCN(C(c2ccn(C3CC3)n2)=O)C1 c1(CC)ccc(C(=O)NC2CCN(C(=O)CCn3cncn3)CC2CO)cc1Cl C1(C(N2CCCC(N(C(=O)CSC3CC3)CC)C2)=O)CCc2[nH]nc(O)c2C1 c1(C(=O)NCC2(NC(C3(CC)COC3)=O)CCC2)ccc(Br)cn1 C1(C)(CNC(C(N2CCCCCC2)C)=O)CN(C(=O)C(F)C(F)(F)F)C(C)(C)C1 C(=O)(C1=CC2(CCOC2)C1)NCC(C)NC(c1cccc2cccn12)=O c1(C(=O)NCC(CC)NC(=O)C(C)Oc2ccc(C(C)=O)cc2)cnccc1C c1(C(N(CC(CNC(CCc2cc(C)on2)=O)(C)C)C)=O)cnn(C)c1C N1(c2cc(COC)ncn2)CCC(NC(=O)C(F)F)C(C)C1 C(=O)(C(O)C1=CCCCC1)N(C(CNC(C(CC)(C)CC)=O)C1CC1)C C(=O)(C1=NOC(C(C)(C)C)C1)NCC1(CNC(C2ON=C(CC)C2)=O)CC1 c1(C(N(CCNC(C2CCCC(C)CC2)=O)CC)=O)cc(Cl)c(O)c(Cl)c1 CCCCCCN(C(=O)Cc1cc(C)no1)CCNC(=O)Cn1cc[n+](C)c1 c1(C(=O)NC(C(C)NC(C2(CC#C)CCOCC2)=O)(C)C)ccc2[nH]ccc2c1 c1(C(=O)OC)cc(C)nc(N2CCCC2CNC(c2[nH]c(C)nc2C)=O)n1 C(C(C)(O)C(F)F)NC(C(C)NC(COCCC)=O)=O C(=O)(CCCCCS(N)(=O)=O)N1CC2C(CNC(C(CCC#C)O)=O)C2C1 C1(C)(CC(=O)N(CCC(C)(C)C)C)CCN(C(C2CS(=O)C2)=O)C1 C1(NC(C=CCCC)=O)C2CC3CN(C(c4nccn5nccc45)=O)C1C3C2 N1(C(C(CC)NC(C)=O)=O)CCCC(C(=O)NCc2ccc(Br)s2)CC1 C1(C(C)(C)NC(c2cc(Cl)c[nH]2)=O)CCN(C(=O)Cc2cccnc2O)CC1 C(C(CC(=O)NC(CNC(c1ccc(Cl)c(F)c1O)=O)C1CC1)C(F)F)N(C)C c1(C(N(C)CC2CCN(C(=O)CCc3cn[nH]c3)C2)=O)cncc(F)c1Cl c1(CCCC)ccc(NC(c2nc(C(=O)OC(COCC)=O)cs2)=O)cc1.OC N1(C(C(C=C=C)C)=O)CCC(C)(C(=O)NC2CCCN(C)C2)CC1 N1(C(C=C(C)C(C)C)=O)CCCC(C(=O)NC2(CN(C)C)CCCC2)CC1 c1(NC(=O)CCC2CCCC(=O)N2)ccc(OC(F)F)c(O)c1 C1(CN(CCc2cnccn2)CC)CCN(C(c2ccc(C(N)=O)o2)=O)CC1 C#CCCCC(C)C(=O)N1CC2C=CCOC2C1 Cc1ccn2ncc(C(=O)N(C(C)CCNC(c3cc(O)ccc3N)=O)C)c2n1 C1(C(N2CC3CC3C2)=O)C2CC(O)C(C2)N1C(c1cc2cnccc2[nH]1)=O c1(C(N2C(C)CC(NC(C(C)SC(F)(F)F)=O)C2)=O)ccnc(Cl)c1N N1(C(c2cc(C)oc2C)=O)CCCC(C)(CNC(=O)CCc2cccc(F)c2)C1 C1(NC(c2cc(C)sc2)=O)CN(C(c2ocnc2C(F)(F)F)=O)CC1C1CC1 Cc1ccccc1C(=O)NC1CC(F)(CNC(C2(C)CCOC2)=O)C1 c1(C(N2CCN(C(Cn3ncc(C)c3)=O)CC(C)C2)=O)ccc2cccnc2n1 c1(C(=O)NCC(CN(C(C(CCC)(C)CC)=O)C)O)cc2cc(F)cc(F)c2[nH]1 C1(C(=O)NC(CC(C)NC(c2cccc(OC)c2N)=O)C)CS(=O)(=O)CC(=O)N1 c1(C(N2CC(C(C)NC(CCOCCOCC)=O)C2)=O)cccc(OC)c1Cl N1(C(c2csc(Cl)c2)=O)CCN(C2CCCN(C(c3ccns3)=O)C2)C(=O)C1 C1(NC(C2C(C)(CC)C2)=O)CN(C(c2ccn(CCF)n2)=O)CC1CO C=CC1CN(C(=O)C(CC)C(C)C)CC1NC(c1ccc(OC)s1)=O CCCC(C(F)(F)F)NC(=O)C1=CCC(NC(C2(COC)CC=CC2)=O)C1 C1(NC(CCNC(C)=O)=O)CC(CNC(C)(C)C)N(C(=O)COC2(C)CCC2)C1 C(=O)(CCC(=O)NCCC(C)NC(C1CCCSC1)=O)NCCCOC N1(C(CS(N)(=O)=O)=O)CC2(C1)OC1(CO)CC2(NC(=O)CN2CCOCC2)C1 c1(C(N2CC(C(C)NC(c3c(C)coc3C3CC3)=O)C2)=O)c(F)ccc(O)c1F c1(C(=O)NC(CCOC)CNC(c2cccc(F)c2Cl)=O)ccc2snnc2c1 N1(Cc2cnn(CC)c2C)CCCC(F)(F)C1C(=O)OC(=O)NC.C(C)(C)(C)O O(NC(=O)C#CC1CCC1)CC(=O)NCc1ccc2cc[nH]c2c1 C1(NC(c2c(C)scn2)=O)CCN(C(c2[nH]ccc2-c2ccccc2)=O)C(C)C1 C1(C(N(C)CCNC(c2ccc(-c3ccccc3)s2)=O)=O)CCCC2(CCC2)O1 C(N=c1[nH]c(C)cc(=NCC(C)N2CCc3ccccc3C2)[nH]1)c1n(CC)ccn1 CC(CC(C)N=c1[nH]c(=NCC23CCC(CC2)O3)[nH]c2cc[nH]c12)C(F)F c1(C(=O)NCC2(NC(c3csnn3)=O)CCCCC2)ccc2sncc2c1 Cc1cc(C=CC(=O)NCC2CN(C(C3CCOC3C)=O)CC23CC3)ccc1F N1(C(=O)CCF)CCC(NC(C2(C3CC3)CC2)=O)C1 C1(C(N(CCNC(c2cc(C3CC3)[nH]n2)=O)CC)=O)CCN(C2CC2)CC1 CC1(C)C(CNC(c2ccc(CO)o2)=O)CCN1C(C1CCCCC1O)=O Cc1nnc(N2CCC3(NC(c4ccc(Cl)o4)=O)CCCCCC23)c(C#N)c1C C(=O)(CC(C)(C)C)NCCC(CNC(=O)C(C)n1ccnn1)OC N1(C(CC2(C(=C)F)CCC2)=O)CCN(C(=O)C(C)C(O)CC(C)C)C2(CCC2)C1 CC(C)C(C(=O)NC1C2CC1N(C(C1CCCN1C1CC1)=O)C2)N(C)C N1(C(C(C)C#N)=O)CC2(CC(NC(=O)COCCc3cccc(F)c3)CO2)C1 N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CCCC(CNC(=O)C=CC(C)CC)C1 Cc1c(C(=O)N(CCCOCCN(C)C(C2C3CCCC23)=O)C)cnn1C c1(CC)ccc(C(=O)NCC(F)F)o1.C1(=O)C(=O)NCCN1 C1(C(=O)NC(C2(O)CN(C(COCCOCC#C)=O)C2)C)CC12CCCCCC2 C1(C(N2C(CC(=O)NCCC(CC)CO)CCC2)=O)CC12CCCCC2 CCCCC(C)(C)NC(C1CSCCN1C(=O)C=C(CC)CC)=O N1(c2nnc(CC)s2)CCC(C(C)NC(c2ccc(F)o2)=O)CC1 C(N=c1[nH]cnc2c1CCC2)C1(O)CN(Cc2c(OC)cc(Cl)cc2)C1 c1(C(=O)NC2C(NC(C(CCC)OC)=O)CCOC2)nn2c(c1Br)CCC2 C1(CC(=O)NCC2CCCCN2CCCC2CCOC2)CCC=CCC1 C(=O)(N1OC2CCC1C2)C1(CNC(c2ccco2)=O)CCCO1 c1(OC)cccc(CCC(=O)NCC=CCNC(c2ccc(COC)cn2)=O)n1 N(C1CN(C(C23CCCN(CCC2)C3)=O)CCc2ccccc21)C(C(F)OC)=O N1(C(C=CCN(C)CC)=O)CC2(C1)CN(C(=O)CC(c1csc(COC)n1)=O)C2 C1(C2CCCO2)(C(N(C(CNC(C2(CC)COC2)=O)C2CC2)C)=O)CCOCC1 c1(OC)ncc(C(c2nnnn2CCCC2CC2)NC2COCCOC2)cc1F Cc1ccc(-c2nn[nH]n2)cc1NC(C1CCC2CCC12)=O c1(CC)nn(C)cc1C(=O)NCC(O)CNC(=O)COc1ccc(C(C)=O)cc1 c1(C(N2CC(NC(C(C)C(C)(C)C)=O)(CO)C2)=O)cc(F)c(F)cc1NC(N)=O C1(NC(CCOCCOC)=O)COC2(CCN(C(c3ccc(O)nn3)=O)CC2)C1 c1(C(N(C2CCN(C(c3cc(Br)c[nH]3)=O)C2)C)=O)ccc2nc(O)n(C)c2c1 c1(N(CCCC=C)C)cc(Br)ccc1S(=O)(=O)NCCC(C)(C)F C1(NC(C2CCCC(C)C2)=O)CC2CN(C(c3cc4nc[nH]c4cn3)=O)CC2C1 Cc1cc(C(=O)N(CCCNC(=O)C(N2CCC(O)CC2)C)C)c(Cl)cc1F Cc1cc(Br)cc(C)c1CC(=O)NCCCCNC(=O)CC(C)C(F)F C(C(CO)(CO)NC(C1CC1C1CCCO1)=O)N(C(C(F)=C(C)C)=O)C N1(C(c2c(C)nc(CCC)s2)=O)CCN(C(=O)C(F)=C2CCC2)C(CO)C1 C(=O)(CC(C)C(=O)N1CCCC1CNC(=O)COc1ccccc1Br)OC C(CCCCCOc1ccccc1)NC(c1cnc(C)o1)COC N1(C(C(CC(C)C)(C)C)=O)CCC2CCC(NC(=O)Cc3c(Cl)cnn3C)C1C2 N(C(=NCCc1cncs1)NCC1CC1)CC(=O)OC(C)(C)C C(=O)(C(CC(C)C)OC)NCC1(CNC(c2c(OC)oc(C)n2)=O)CC(F)(F)C1 c1(OCC)ncc(C(=O)NC(C)CCCNC(c2c[nH]nc2C)=O)cc1Cl C1(N(C(CCSC)=O)C)CCCC2CN(C(C3Cc4ccccc4C3)=O)CC12 Nc1cc(Cl)cc(F)c1C(=O)NCCC(O)CNC(c1cnccn1)=O C1(CNC(=O)CCCCCO)CCC2CN(C(C3(C(F)(F)F)CC3)=O)CCC2C1 Cc1ccncc1C(N1CCOC(C(=O)NCc2ccc(Br)nc2)C1)=O C(CC(F)CN=[N+]=[N-])NC(C(Cc1cn[nH]c1)NC(c1ccc(C(C)C)o1)=O)=O c1(OC)cnc(Br)cc1C(=O)NCC1CCCCN1C(c1cc(C)ncn1)=O C(=O)(CN=c1[nH]c(=NCC2CC2)c2ccc(OC)cc2[nH]1)NCC=C c1(N2CCC(C)C(NC(c3c(CC)nns3)=O)C2C)cc2nnc(C)n2cn1 C1(C(=O)NCCOC2CN(C(c3ccc(COC)o3)=O)C2)CC(=O)C12CCCC2 C1(C(=O)NC2(C)CN(C(c3ccc(C4CC4)nc3O)=O)C2)CC1C1CCCC1 c1(C(=O)NCC2(C(N)=O)CN(C(CC3(COC)CC3)=O)C2)cccc(F)c1N C(=O)(C(C)(F)C(=O)NCC1CCCN1C(C1(c2cccnc2)CC1)=O)OCC C12(NC(=O)CNC3CC3)CCC(CNC(=O)CN3CC=CC3)(CC1)OC2 c1(C(N2CC(c3ccsc3)C(C)C2)C(=O)NC)ccc2c(c1)nc(C)n2C CC1C(C(=O)NC2CC=CCC2C(=O)Nc2cccc3occc23)=NOC1C c1(NCC(=O)NCC(CC)NC(=O)C(F)(F)F)nc(Cl)nc2c1SCC2 c1(OC)cc(NC(C2CCN(C(c3cn[nH]c3)=O)CC2O)=O)c(Br)cc1C C1(NC(C2(NC(=O)CCC3CCC(=O)C3)C(C)(C)C2)=O)CCC2(CCC2)CC1 N1(C(C2(CC#C)CCC2)=O)CCCC(N(C)C(c2cnn(C)n2)=O)C1 C#CCC(C)(C(=O)N1CCC(OCCF)C1)NC(C1CC(=C2CCC2)C1)=O C1(C(N(CCC(=O)NC)C)=O)COCCN1C(c1ncccn1)=O C1(NC(C(CC)C)=O)CS(=O)(=O)N(C)C12CCN(c1nnc(C3CC3)o1)CC2 C12(NC(CCN(S(C)(=O)=O)C)=O)CC1CN(C(c1nnn(C)c1C(F)F)=O)C2 C1(NC(=O)OC(C)(C)C)CC(NC2CCC(C)(C)CC2)CCC1(F)F C1(C(=O)NC2CC(CCC(=O)NCCC3(O)CCCC3)C2)CCC(C2CC2)CC1 N1(C(C2(CCC)CC2)=O)CCC(NC(=O)CSC2CCCCO2)C(O)C1 N1(C(C(c2ccc(Cl)cc2)C)=O)CC2CC1(CNC(=O)CCc1cccs1)C2 C(CC(C)NC(=O)Cn1cc(-c2ccc(Cl)cc2C)nn1)(C(=O)O)SC C1(NC(c2c(OC)cc3c(c2)OCC3)=O)C2CC3CN(C(=O)OC(C)(C)C)C1C3C2 C=C=CC(C)C(=O)N1CCC(N2CCC(NC(C34CC(F)(C3)C4)=O)C2)CC1 C1(O)(CNC(C2CCSC2)=O)CCN(C(C2(Cc3cccc(Cl)c3)CC2)=O)CC1 C(CCN=C(NCC12CCC(CC1)OC2)N1CCC(c2cccc(C)c2)C1)OC CC1CN(C(=O)CCc2nccs2)C(C)CN1C(=O)Cc1nc([N+](=O)[O-])n[nH]1 c1(CC(N2CCC(O)(CNC(CN(C)C3CC3)=O)C2)=O)nc([N+](=O)[O-])n[nH]1 C1(NC(C=C(C)C(F)F)=O)(CNC(c2ccc(N(C)C)nn2)=O)CC2CCC1C2 c1(C(=O)NCC(C)(C2CC2)NC(=O)Cn2nnc(C3CC3)n2)c(N)cc(Cl)cc1Cl Cc1cccc(C(=O)NC2COCC2C(N2CCC(F)(C#N)C2)=O)c1O Cc1cc(F)ccc1C1CC1C(=O)NC(C)CC(C)NC(=O)CCCC(C)O C1(CCC)CN(C(=O)CN2CCN(C(c3cc(C)sc3C)=O)CC2)CCO1 C(=O)(NNC(=O)Cc1cccs1)C1(C)CCCC1O c1(OC)ccc(-c2nc3c(s2)CCN(C(c2ccc(O)cn2)=O)C3)c2cn[nH]c12 C(=O)(C(O)CC(F)(F)F)Nc1ccc(C(=O)NCC2(CO)CC3C=CC2C3)cn1 CC1OC2(C(=O)NCC3C(O)C(O)CN3C(=O)CC3CCCC3)CCC1CC2 N1(C(c2cncc(F)c2)=O)CCN(C(C2CC2c2ccsc2)=O)C2CCC12 c1(C(=O)NC2CCC(CCNC(CC=C=C)=O)C2)ccc(Cl)c(OC)c1N C1(N(C(C2(NC(c3cnn(C)c3N)=O)CCN(C)C2)=O)C)CCCC(C)(C)C1 Cc1c(C(=O)NC2(C)CN(C(c3snc(O)c3Cl)=O)C2)cnc2ncnn12 c1(C(N2CC(CNC(C3CC(OC(F)(F)F)C3)=O)C2)=O)[nH]cc2c1CCC2 C1(NC(c2n(C(C)C)ncc2)=O)CC12CCN(C(C1CCCCC1(C)C)=O)CC2 N1(C(CC2CC(=O)OC2)=O)CC=C(CNC(=O)CSc2cn[nH]c2)CC1 N1(C(=O)C=Cc2cnccn2)CCC2CCN(C(=O)CC3CCCSC3)C2C1 C(=O)(CC(C)(C)CCC)NC(c1ccccc1F)CNC(C(C=C)C)=O Cc1cc(C(=O)NCC2CC(NC(=O)CCC(C)N(C)C)C2)ncc1S(N)(=O)=O C(=O)(C(C)C(C)CC)NC1CCC(NC(C(Br)=CC)=O)CC1 CCC1=NOC(CNC(=O)NC(c2ccncc2)CCSC)C1 CCS(=O)(=O)CC(=O)NC(C1(O)CCN(C(=O)COC(C)(C)C)CC1)C c1(C(N2CCC(NC(C3C(CC)OCC3)=O)C2)=O)ccc(Cl)c(Cl)c1O C(=O)(C#CC1CCCO1)NCCC1OCCN(C(c2c(C)[nH]c(=N)s2)=O)C1 N1(C(c2cc(C(=O)OC)sc2C)=O)CCC(NC(=O)CNC(N)=O)C(O)C1 c1(C(=O)NCC2OCCC(N(C)C(C3COC(=O)N3C)=O)C2)ncnc2c1CCC2 c1(CNC(C2(C(CC)(F)F)CC2)=O)ccc(C(N2CC(F)CC2CO)=O)nc1 C(C)(C)(C(C)CC(=O)NC(c1cncs1)C)NC(c1c(C)nccn1)=O CC1CN(C(=O)CCCS(C)(=O)=O)CC(C)C1NC(=O)CC1COCC1(C)C C(=O)(C1=COCC1)NC(CC(C)NC(C(CC)F)=O)C C(=O)(N1Cc2ccccc2CO1)C1CC(C)(NC(C(C(C)C)CN(C)C)=O)C1 c1(C(=O)NCCNC(C2N(C(CC)=O)CCCC2)=O)ccc(N)c2ncccc12 C1(CNC(C(C)OC)=O)CC2(CO1)CN(C(=O)CSCCN(C)C)C2 N1(C(CSCC(N)=O)=O)CC2ON=C(CNC(c3cc([N+](=O)[O-])n[nH]3)=O)C2C1 C=C(Cl)CC(C(=O)N1CC(=O)NC(C)C1)NC(=O)C(C(C)C)C1CC1 C1(N(c2n(-c3ccc(C)cc3)nnn2)C(C2(Br)CC2)=O)CCC2(CCNC2)CC1 c1(OCC)ncc(C(=O)NCC(CO)NC(C2(C(F)F)CCCO2)=O)cc1Cl N1(C(=O)CCC2CCOC2)CC=C(C(=O)N2CCC(F)(F)C2)CC1 C(=O)(CC(F)(F)C(F)F)NCCC1(CNC(C2(C(=O)OCC)CCCC2)=O)CC1 c1(C(=O)NC(C(NOCC(C(C)C)O)=O)(C)C2CCC2)ccc2occc2c1 C(C1=CCN(C(=O)CC(C)CF)CC1)NC(c1cn(CC(CC)O)nn1)=O c1(OC)ccc(Cl)cc1C(N1CC2C(C(=O)NC(C3CCOCC3)C)C2C1)=O CCC(C)C(C(=O)N(C1CCNCC1)CCN(C)C)OC N1(C(C(C2CC2)OCC)=O)CC(CC(=O)N(C(C)CO)CC2CCC2)CC1C N1(C(CCCCCC#N)=O)CCC(CNC(C2CCC23CCC3)=O)C(F)(F)CC1 c1(C(=O)NCC(CN(C)C(c2ccc3c(c2)NCC3)=O)O)ccnc2ncnn12 c1(C(=O)NCCCNC(c2c(C)nn(C3CC3)c2Cl)=O)cnc2ncccn12 C(=O)(C1=CCCCO1)NC1CCC(N(C)C(C2CCCCN2C)=O)CC1 C1(NC(CC2CN(C(CC(C)C3CC3)=O)C(C)(C)C2)=O)CN(C)C(=O)C12CC2 C(=O)(C(C)(CO)NC(=O)C(C)n1cncn1)NCC(CC)N(C)C N1(C(C2CCN(C(c3cc[nH]c3)=O)C2)=O)CCOCC2(CC2)C1 C1(C(=O)NC(c2cccnc2N)C)CCC2(CCCC2)C1 C=CC(C)(CCOC)C(=O)N1CCOC(C)(CNC(=O)CCc2cnc[nH]2)C1 C(c1cc(C)nn1Cc1cccc(I)c1)=CC c1(NC(C)=O)ccc(C(N2CCC(NC(=O)CC3CCCN3C(C)=O)C2)=O)s1 C(F)(C(=O)NCC(C)(C1CCC1)NC(C12CCC1C2)=O)=C(C)C C1(NC(c2nccc(C)n2)=O)CC(F)CN(C(c2c(C3CCC3)cnn2C)=O)C1 Cc1cc(C)c(NC(=O)CN(C)CCc2nnc(N(C)C)s2)c(Br)n1 N1(C(c2ccccc2-c2ccc(F)cc2)=O)CC2COCC2(CC2CCC2)C1 N1(C(CC)=O)CCC2(CCC(NC(c3sccc3S(C)(=O)=O)=O)C2)CC1 N1(C(c2ccc(C(C)=O)cc2F)=O)CCC2(CO)CCCC12 c1(C(c2ccc(Cl)s2)N(C(=O)C(C)OCC(C)(F)F)CC)cccc2nonc12 C1(C(=O)NCC(=O)N(CCCCC(=O)OC)C)CC2CC1CC2O C1(NC(C(COC)(C)C)=O)(CNC(=O)CCn2nc(C)nc2C)CCCCCC1 c1(C(N2CCN(C(CSC)=O)CC2CC(F)(F)F)=O)nc2nc(C)ccn2n1 C(C#Cc1cccc(F)c1F)OC(=O)Cc1csc(C2CCOCC2)n1 CCCCN=C(NCC(C)CC(F)(F)F)NCCS(=O)(=O)N(C)C c1(C(N2CC(O)(C(C)NC(C(N3CC(C)C3)C)=O)C2)=O)cccc(F)c1F c1(C(=O)NCc2scc(C(N(C3CC(C#N)C3)CC#C)=O)c2)ccc(CF)cc1 C12(NC(C3C(C=C)C3)=O)CCOC(CNC(=O)CCC(C)(C)C)(C1)C2 N1(C(=O)NCC(C)(C)OC)CCC(F)(F)C(C(N)=O)C1 C1(C(=O)NCCCCCNC(C2(CC)CCOCC2)=O)CCCCC(C)(C)C1 c1(C(C)(CN2CCC(F)C2)NC(=O)NC(CC=C)C)ccc(Cl)c(F)c1F N1(C(C(C)OCC)=O)CCCC12CCN(C(=O)Cc1ccc3nonc3c1)C2 c1(CC)cc(OC)cc(C(N2CC(n3cc(-c4cccs4)nn3)C2)=O)c1 c1(C(N2CCOCC2(C)C2CC2)C(=O)NC)ccc2cc(C)ccc2n1 c1(OCC(C)C)cccc(C(c2nnnn2C)NC(c2ccc(Cl)nc2)C2CC2)c1 Cc1cc(C)c(C(=O)NCC2CC3(CC(NC(=O)Cc4cc[nH]c4)C3)C2)c(O)n1 c1(C(C)(C)C)n[nH]c(=NC2CN(C(c3cnc4[nH]c(O)nc4c3)=O)CC2(C)C)s1 C#CCCCCC(=O)NCC1CC2(CC2)CN1C(c1n[nH]c(=N)[nH]1)=O c1(C(C(N2CCN(C(c3cccc(CSC)c3)=O)CC2)=O)C)cccc(C#N)c1 c1(C(=O)NC(CCNC(C2N(C)CC(F)C2)=O)(C)C)cc2n(n1)CCC2 C=C(CNC(C1CN(C(c2n[nH]c(C)c2O)=O)CC1OC)=O)C1CCOCC1 c1(C(NNC(=O)Nc2nc3cnccc3[nH]2)=O)cc2cn[nH]c2cn1 Cc1ccc2ccncc2c1C(=O)NCCC(C)N(C)C(c1cccc(N)n1)=O N1(C(=O)OC(C)(C)C)CC2C(N)C2C1.c1(OCN)cccnc1OCCO C1(CCNC(c2nc(CCC)oc2)=O)CCN(CCC2CCCC(C)C2)CC1 c1(-c2nc(Cc3c(C(=O)OC)cncc3)nn2C)nnc(C)c2ccccc12 c1(OCC)nc(C)ccc1C(=O)NC1CCC(C)(NC(C2C=CCC2)=O)CC1 c1(C(=O)NCCN(C(c2ccc(CC3CC3)s2)=O)CC)cnc2[nH]c(C)nc2c1 Cn1cccc1C(=O)C(=O)NCC1CCCN1C(=O)CCCc1nc(C(F)F)no1 N1(C(c2c(C)cns2)=O)CCCCC12CC(NC(=O)CCc1cnn[nH]1)C2 C(=O)(C(CC(F)F)NC(c1c[nH][nH]c1=N)=O)NCCCCS(C)=O c1(CNC(=O)CC2CCCN2C(C2C(C(=O)OC)C2)=O)cc(OC)ccc1OC C1(C(N(C)Cc2cnn(C)n2)=O)CCN(C(=O)OC(C)(C)C)C1(C)C N1(C(c2n(CCN(C)C)ncc2)=O)CC2CC1C2CNC(c1nc(Cl)cs1)=O.C1CC1 CC1CCN(CC(N2CCC(C(F)C(N3CCCC3C(O)CO)=O)C2)=O)C1 C1(C(N2CC(c3onc(C)n3)C2)=O)CNC(=O)CN1C(c1ccncc1N)=O [N-]=[N+]=NC1CN(C(C2(F)CCCN(C(c3cccc4cncn34)=O)C2)=O)CC1O c1(OCC#C)ccc(N)cc1.N12CCSCC1C2=O.C(=O)(CCNC(C)=O)NCC C1(NC(=O)Cc2csc(C(F)(F)F)n2)CC2(CCN(C(=O)C(F)CC3CC3)CC2)C1 C1(CC)C(NC(c2ccncn2)=O)CCCN1C(C1CC(C)=NO1)=O C(C1CSc2ccccc21)NC(c1ccnn1C1CCNCC1)=O C(CCN(C(=O)CC1COC(=O)C1)C)(C(C)C)NC(CSCC=C)=O c1(N2CCC(CCNC(C(CCCC)O)=O)C2)ncnc2c1nnn2CC1CC1 c1(C(=O)NC2(CO)CCN(C(c3nn(C)c(Cl)c3Cl)=O)C2)nccc2occc12 c1(N2CCC(F)(C(=O)OC)C2)nc(O)c2cc(Cl)ccc2n1 CC1(C)COC(CC(N2CCC(CNC(=O)CCC3CC3)C2)=O)CO1 CC(C)N=C(NCC(c1cc(F)cc(F)c1)(F)F)NC1C=CCCC1 C(CCN=C(NCCc1ccc(C2CC2)cc1)NCC1(Br)CC1)SC C1(C(=O)NCCC(=O)NC(C)(C)C)CC(O)CN1C(=O)CC1(C)OCCO1 C1(NC(C(CC)OCC)=O)CC12CC(NC(=O)CCOc1ccccc1)C2 n1(CC(N2CC(COC)N(C(=O)CCC(N)=O)CC2)=O)c(=O)oc2ccccc12 C1(C(N2CC(CCCCNC(c3[nH]cc(C(N)=O)c3)=O)C2)=O)CCCCC1(F)F C1(C(N(CCN(C=O)CC)CC)=O)CC2(CCC2)CCO1.c1(OCC)ccc(CO)s1 C=C(Cl)C(C)(C)C(=O)N(CCCN(C(=O)CC1CC(O)C1(C)C)C)C C(=O)(C(C)(F)C(=O)NCCC(=O)NC1CNC(=O)C12CC2)OC c1(C(=O)NCC2(C)N(C(C(C)OC)=O)CCC2)cc(C)nc2c1cnn2C c1(NC(Cn2cc(CN)nn2)=O)cc2ncc(-c3ccc4[nH]ccc4c3)cc2[nH]1 N1(C(C2CCC(C)O2)=O)CCN(C(c2ccc(C(F)(F)F)nc2)=O)C(C)C1 CC(c1ccsc1)=CC(=O)NCC(C)CN(C(=O)C(CO)N(C)C)C c1(CNCc2ccc(CCCCC)cc2)cc(C)cc(Cl)c1 C(=O)(C1CCCn2ncnc21)NCC1C(C)CCN(C(CC(C)OC)=O)C1 C(=O)(CCCC(C)(C)C#N)N1CCCC(N(C(=O)CSc2nnnn2C)C)CC1 C1(C)(C(N2CCCC(N(C(CN(C)CC)=O)CCO)C2)=O)CC(C2CC2)=NO1 c1(CC)cc(C(=O)N(CC(C)NC(=O)C(CCSC)OC)CC)ccc1OC c1(C(=O)NC(C(C(C)C)O)C)ncnc2c1CCCC2 c1(C(N2CCCC(COC)C2)=O)ccc2ccoc2c1.c1(C)cn(C(C)C(=O)O)nn1 C(=O)(C#CC1CCOC1)N1CCC(F)(C(=O)NC2CC(C(C)C)OC2)C1 N1(C(C2C(NC(C)=O)C3CCC2C3)=O)CC=C(C(C)(C)C)CC1 C1(C2CCCO2)(C(N(CCN(C(=O)Cc2cnn(C)c2)C(C)C)C)=O)CCCC1 Cc1ccc2cccnc2c1C(=O)NC(C)CNC(=O)C(F)Cc1ccccc1 c1(CC)cc(C(=O)NCC=CCNC(c2ccc(C(C)F)cc2)=O)cc(Cl)c1 c1(C(=O)NC2(CC=C)CN(C(c3cncc(O)c3)=O)C2)n[nH]c(C)c1Cl C1(C(=O)NCCN(CCC)C(c2nnsc2SC)=O)CC2C(C1)C2(F)F n1(CC#C)c(C)cc(C(=O)NC2CCC(NC(=O)CC(O)C(C)C)CC2)c1C c1(C(=O)NCC(c2ccccc2)C2CCCC2)ccc2ccccc2c1[N+](=O)[O-] n1(CC(=O)NCC#CCNC(=O)C(F)C(F)(F)F)ncc2ncccc12 C(=O)(C1=CCCC1C)NCCC(C)N(C)C(c1coc(CC2CC2)n1)=O c1(C(=O)NC2C(CNC(C3CCN(C(CCC)=O)CC3)=O)C2)cc(C#N)n(C)n1 c1(SCC)cc(C(=O)NC2CC2CNC(C2C(C=C(C)C)C2(C)C)=O)ccn1 c1(C(=O)NC2CN(C(CC(=O)OC)=O)CC2C)c(F)cc(OC)c(F)c1F n1(CC(N2CCN(C(=O)CNc3ncccn3)C(CF)C2)=O)cc([N+](=O)[O-])cn1 N=c1nnn(CC(=O)NCCCOCCOCCNC(=O)Cc2ccon2)[nH]1 CC(C)(Cc1ccccc1)CC(=O)NCC1COC(CNC(=O)Cc2cn[nH]c2)C1 N1(C(C(CC)n2cncn2)=O)CCCC(NC(c2c[nH]cc2Br)=O)C1 CC1=CCC(C(C)CC(=O)NCCNC(c2cnc(CCC(F)(F)F)s2)=O)CC1 C1(CC(=O)NCC(C(C)C)(C)NC(c2cncc(F)c2)=O)CCCCC(=O)N1 c1(C(C(=O)NCC)N(C)CCc2cccnc2)nc2cc(Br)ccc2s1 C1(NC(CC2(CSC)CC2)=O)CCCCC1S(C)(=O)=O CC(C)C(C(=O)NC(C)CC1CCN(C(=O)C2=NOCC2)CC1)N(S(C)(=O)=O)C1CC1 C1(NC(=O)CCN(CCCO)C(C2CC(=C3CC3)C2)=O)CN2CCC1C2 CC(CN=c1c(C#N)c[nH]c2c(F)ccc(Cl)c12)N(C)CC1CCC1 c1(OC)cc(C(=O)N(CC(O)CN(C(=O)CO)C)C)cc(Br)c1 C1(C(=O)NC2(C)CCN(C(C(C)(CO)OC)=O)C2)CC2(C1)CC(O)C2 c1(N(C)Cc2cccc(OC)c2)nc(N2CCC(F)C2)nc2cccc(F)c12 Cc1ccc(O)c(NC(c2ncccc2NC(c2cc(Br)cnc2O)=O)=O)c1 N1(C(C)=O)CCC(C(=O)Nc2cccc(NC(C3(N(C)C)CCC3)=O)c2)CC1 C1(CC(=O)NC(C)(C)CCNC(CCOCCOCC)=O)CC2(CCCC2)CO1 C1(OC)(OC)CC(C)(C(=O)NC(C2(CNC(c3ccc(O)nc3)=O)CC2)C)C1 CCC(CC(F)F)C(=O)NCC1CSCCN1C(=O)CCCC(=O)OC(C)(C)C C(=O)(C1c2c[nH]nc2CN1C(=O)CCc1cnn(C)c1)NCC1CC(SC)C1 N1(C(CCNC(CSCCC(C)C)=O)=O)CCC2CC2C1 c1(C(=O)NC2CC3CCC2N3C(C23CCC(CC2)C3)=O)cc(Cl)c(F)cc1F C(Cc1ccccc1Br)(C(=O)N(O)CC1CCCCC1)N(CC)CC C12(C(N3CCC(C(CNC(Cc4ncc(C)o4)=O)C)CC3)=O)CCC(CC1)CC2 C1(F)(CNC(c2cc(C)on2)=O)COCCN(C(c2ncn3c2CCCC3)=O)C1 Cc1cnc(C(=O)NC2CC(F)(CNC(=O)CC3CC4C=CC3C4)C2)cc1C N1(C(C2(C(=O)OC)CC2)=O)CC2(CC2C(=O)Nc2ccc(C(C)O)cc2)C1 c1(C(=O)NCC(C2CC2)NC(=O)C=CBr)cc2ccc(Br)cc2o1 c1(OCC=C)ccc(CC(=O)NC2COCC2NC(=O)C(F)OC(F)(F)F)cc1 c1(OC(C)=O)cccc(C(N2CCCC2)=O)c1C.N12CSCC1C2=O CCC(CC)CC(F)C(=O)NCC1CC12CCN(C(=O)C1=CC(C)C1)CC2 c1(OC)c(F)cc(C(N2CCN(Cc3cc(O)ncc3Br)CC2)=O)cc1F Cc1coc(C(=O)N(CC(O)CN(C)C(c2cc(C(C)(C)C)nn2C)=O)C)c1C c1(C(=O)NCCN(C(C2CCCC2Cc2ccccc2)=O)CC)cn(C)cc1C C1(NC(C(c2c(C)cncc2)C)=O)CC1C1CCN(C(c2cocn2)=O)CC1 c1(C(=O)NCC2(NC(C3C(=C)C3)=O)CCOC2)cnn(CCC(C)C)c1C c1(COC)nc(NCc2ccnc(N(C)C)c2)cc(=NCC2COCC2(C)C)[nH]1 Cc1cc(OCC(N2CCC2CNC(C2CCCCN2C)=O)=O)cc(C)c1 Cn1[nH]c(=NC(=O)C2CC2NC(=O)Cc2cc(F)c(F)cc2Br)cc1C(N)=O N1(C(c2c(C)sc(O)n2)=O)CCCC(C)(CNC(c2cnn(C(C)C)c2C)=O)C1 Cc1cccnc1C(F)(F)C(=O)NCC1CN(C(C2CCN2C)=O)C1 Cc1cc(C(=O)NCCNC(C2CC2c2ccccc2C)=O)n(C)n1 CC(=O)CC(C)(C)C(=O)N1CCC(CO)(CNC(=O)CC2CC3C=CC2C3)C1 C(c1cccc(C2CCN(C(C3CN(C)CCO3)=O)CC2)c1)=C(C)C Cn1ncc(Br)c1CN1CCCC(CNC(C2CCC(C(F)F)CC2)=O)C1 C(N=c1[nH]c(=NCCOCc2ccccc2)[nH]c2c1CCCC2)c1n(C)cnn1 CC1CN(C(c2ccc(CO)cc2)=O)CC(C)N(C(=O)CO)C1 c1(NC(C)=O)cc(F)c(F)cc1C(=O)NC1CCN(C(c2cncnc2C)=O)C1 C1(NC(c2cc(C)no2)=O)CC(NC(c2ccc(C(F)F)nc2)=O)C12CCC2 C1(NC(c2c(C)onc2)=O)CN(C(C2CCCCN(C)C2=O)=O)CC2(CC2)C1 N1(C(=O)COc2ccon2)CCC2CCCN(C(=O)CCC(F)(F)F)C2C1 N1(C(C(C)NC(=O)NCC)=O)CC2(NC(C3(C4CCCCO4)CCC3)=O)CC1C2 c1(OC)ccc(CC(=O)NC2CC3(C2)CC3NC(c2sc(F)cc2Cl)=O)cc1 C1(C(=O)Nc2c(I)ccc(C#N)c2)CCCC12CCN(S(=O)(=O)CC1CCC1)C2 C(C(O)CNC(C1CCOC1)=O)N(C)C(C1CC(CC(C)(C)C)C1)=O C1(CCC)(NC(=O)C2=CSCCO2)CCN(C(=O)CCNc2ccccn2)CC1 c1(OCC#C)cc(CNCC2CCCN2S(C)(=O)=O)cc(Br)c1 c1(C(N2CC(C(C)NC(=O)CC#N)OCC2)=O)ccc2cccc(F)c2n1 N1(C(CCC#N)=O)CCC2(NC(=O)CCc3c(F)cccc3F)CCCCCC12 N1(C(c2c(N)c(Br)ccc2)=O)CCC2(C1)CN(C(C1CCCC1O)=O)C2 N1(C(c2cc(C)ncc2)=O)CCCC(C)(C)C1CNC(=O)CC(C)C1CCCC1 C1(CN(C(c2c(CC)occ2)=O)C)CCCCN1C(=O)CCCF C1(CNC(C(C)=C2CCC2)=O)(NC(=O)CCC2OCCO2)CC2CCC1C2 C1(CNC(C2CCN(C)C2)=O)(CNC(c2cn(C)nc2O)=O)CCOCC1 C(C(=O)N1CCC(C2CCCN2C(=O)Cc2nncs2)C1)(C(C)C)SC CC1=C(C(=O)N2CC3CC(NC(c4c(C)cc(=O)oc4C)=O)C2C3)SCCO1 C12N(CC1(C)C)C2=O.n1(CCNC(CCC)=O)cc(C(=O)NN2CCCC2)nn1 N1(C(CC=C)=O)CCC(C2CCN(C(c3cc(CC)ccc3OC)=O)CC2)CC1 c1(C2(C)C(C(=O)NC3(CC(=O)OC)CCNCC3)C2)ccc(F)c(F)c1 n1(CCN(C)C)nccc1C(N1CCC1CNC(c1sccc1C(F)F)=O)=O C1(C(=O)OC)CC12CCN(C(=O)Nc1cccc(NC(C)(C)C)c1)C2 c1(C(N2C(CNC(c3ccc(C)[nH]3)=O)CCCC2)=O)cnc2c(Cl)cccn12 c1(NC(N(OC)Cc2ccccc2)=O)cccc(Br)c1OC(F)F N1(C(c2nn(C)c(C(F)(F)F)c2Br)=O)CC(N)CC2(CCC2)C1 C1(C(=O)NCCC2OCCN(C(c3nc(CC)oc3)=O)C2)CC2(CCC2)CO1 N(C(=NCCc1cccc(C)n1)Nc1ccc(OCC)c(OCC)c1)C(C=C)C C(=O)(CC(CC)C(C)C)NCCOCCCNC(C1N(C(C)=O)CSC1)=O C1(NC(CN(C)CC)=O)(CO)CCN(C(C2CCC(=O)NC2)=O)C1 N1(C(CSC)=O)CCOCC1C(=O)Nc1ccc(-c2ccccc2)nc1 c1(CN2C(C(=O)Nc3c(OC)ccnc3)CC3(CC3)C2)cc(C)cc(Br)c1O CCN=c1[nH]cc(C(N2CCCC(CNC(=O)C(C)=CC(C)(C)C)C2)=O)s1 N1(C(C2C3(CCN(C(COC(C)C)=O)CC3)C2)=O)CC2CCC(C1)C(=O)N2 C1(C(=O)NCCCN(C(c2c(C)nc[nH]2)=O)C)C2Cc3c(Br)cccc3C12 c1(C(N2CCC(NC(C(c3c(C)cncc3)C)=O)C2C)=O)cc(Br)cnc1O Cc1cc(CN(CCCCl)C)cc(NC(N2CCS(=O)(=O)CC2)=O)c1 N1(C(C)(C)C)CC(C(=O)NC2CC(CNC(c3cnn(C)c3F)=O)C2)CC1=O c1(OC)cc(CC(=O)NCC(C)CN(C)C(C2OCC2(C)C)=O)cc(Br)c1 C1(NC(c2cn(C)nc2)=O)CC2CC1CN(C(c1cc(Cl)ccc1Cl)=O)C2 Cc1cc(C)c(OCCNC(c2ccc(NS(=O)(=O)CC#N)cn2)=O)c(C)c1 C(CCN=c1[nH]c(Cl)ncc1[N+](=O)[O-])N(C(CCCC1C(C)C1)=O)CC1CCCC1 C1(c2nnnn2Cc2ccccc2)(NC(CCCC)C)CC2(CCC2)C1 C#Cc1ccc(CC(=O)NC2(CCNC(c3coc(N(C)C)n3)=O)CCC2)cc1 c1(OC(C)C)cccc(CN(C)CCNC(C(=O)CCN2CCCC2)=O)c1.OC c1(COC)cccc(C(=O)NCC2CCCC2NC(C2CCCN2C(C)=O)=O)c1 N1(C(C(C)C2CCC2)=O)CC2CC(NC(C3COCCN3C)=O)CC1C2 C1(C(N2CCN(C(c3cc[nH]n3)=O)C(CC(F)(F)F)C2)=O)CN2CCC1CC2 c1(OC)ccc(F)cc1-c1cc(C(=O)NC2CCC(F)(F)C2)ccn1 N1(C(c2c(C)onc2O)=O)CCN(C(=O)C(C)Oc2ccccc2Cl)C2(CC2)C1 CC(C)CC(C)C(=O)NCC1(C(C)(C)O)CN(C(c2ncn(C(C)(C)C)n2)=O)C1 CS(C)(=O)=NCC(=O)NC1CC(C)(NC(c2cnc(-c3cnccn3)s2)=O)C1 CCS(=O)(=O)NCC(=O)NCCCN(C(=O)CC1CCCC1)C(C)C n1(CC(=O)NC2CCN(C(C(=C(C)C3CC3)F)=O)CC2C)cnc2ccccc12 c1(C(=O)NCC(C(C)C)NC(c2ccc(CC3CC3)s2)=O)ccc(S(C)(=O)=O)o1 Cc1c(C(=O)NCC(O)CNC(c2cn(C)c(=O)n2C)=O)[nH]c2cc(F)ccc12 CCCC(C)CC(=O)N1CC(F)(CNC(=O)CC(C(F)F)n2cccn2)C1 N1(C(C(n2c(C)ncc2)C)=O)CCC(C)(CNC(=O)C(c2cccnc2)C)CC1 C1(NC(c2n[nH]cc2Br)=O)CCCCC12CCCN(C(c1cnnc(Cl)c1)=O)C2 N1(C(c2n[nH]c(CC)c2F)=O)CC(NC(=O)Cc2ccccc2Br)C(C#N)C1 C(C)(C)(CCCC(=O)NCC1CCC1C)NC(C(CC=CCC)C)=O c1(-c2n(CC)nc(CC(C)CC)n2)cnn2cc[nH]c12 C1(NC(c2cccc(N3CCC(=O)NC3=O)c2)=O)CCCCCCC1C(=O)O C(CNC(c1c(C)n[nH]c1C)=O)(CC(=O)NCCSC)OC Cc1n[nH]c(=NC2C3CC2CN(C(=O)CC2OB(O)c4ccccc42)C3)o1 N1(C(c2cc(COC)no2)C(=O)NCCC2CC2)CCSCC1c1ccccc1 c1(C(=O)OC)sc2cccc(F)c2c1CNC1CN(C(=O)C2=CCCSC2)C1 N1(C(CC2CCCC(=O)N2)=O)CCC(NC(C23CCC(C2)C3)=O)C(O)C1 N1(C(CCCSC)C(=O)NC2CCOC2)CCOC2(CCC2)C1 c1(NC(C(Cc2cccc(OCC)c2)N)=O)cc(OC)c(OC)cc1[N+](=O)[O-] C1(CNC(C2NCCC23CCOC3)=O)CC(c2ccc(F)cc2)=NO1 Cc1cc(C(=O)NCC(CC(C)C)NC(C2CC(C)N(C)C2)=O)ncc1C(N)=O c1(CC(N2CCN(C(C3CCC3)=O)CC(O)C2)=O)coc2c(Cl)c(Cl)ccc12 C(=O)(C1Cc2ccc(F)cc21)NC1C(Nc2nc(COC)c(C)s2)CS(=O)(=O)C1 N1(CC)CCC(NC(=O)CC2CCC(NC(C3CC3C(F)F)=O)C2)C1=O c1(OC)ccc(CO)cc1OC.C1(C)(CSC2CC(C(=O)OC)CN2)CC2(CC2)C1 CC1(c2cn(Cc3csc(Br)n3)nn2)CCN(C(C2(S(N)(=O)=O)CCC2)=O)CC1 C1(COC)(NCC(c2ccccc2I)C)CCOCC1 C=CC(C)(C)C(=O)NCCC1CN(C(C2CCCCN2CC(F)F)=O)CCO1 Cn1cc(C(F)=CC(=O)NCC23CC2CN(C(=O)CN2CCCOC2=O)C3)cn1 C=C1CCC(CNC(=O)C(CCC)NC(c2ncccc2O)=O)CC1 C1(Nc2nccc(OCCOC)n2)CCCCN(C(=O)CN2CCN(C)CC2)C1 N1(C(C(C)OCCN(C)C)=O)CCC(F)(CNC(c2csc(Cl)c2)=O)CC1 c1(OC)cc(C(=O)NC(C2CCN(C(=O)CC3CCC(C)CC3)C2)C)ncn1 C1(C(=O)NCCN(C(=O)CCc2nnc(C(C)C)o2)CCOC)CCS1(=O)=O CCCCCCn1cc(CN(C)CCNC(c2c[nH]nc2-c2ccccn2)=O)nn1 N1(C(C(F)=CCC)=O)CC2(CNC(=O)C(CCSC)N(C)C)CC1CCO2 CC1C(=O)CC2CCC1N2C(c1ccc2c(c1)CCN2)=O C1(C(=O)NC(C(C)SC)C)CCN(C(=O)Cn2cnnn2)CCO1 c1(CNC(C2C(C(N(CCC#N)C)=O)C2)=O)c(Cl)ccnc1Cl N1(C(Cn2ncc(CC)c2)=O)C2CCC1C(CNC(C1CC1(C)C)=O)C2 C(=O)(C(O)CC(C)C)NC1(CCOC)CCN(C(C2(CC#C)CC=CCC2)=O)C1 C(=O)(C(CP(C)(C)=O)C(F)(F)F)NC.N1(C(=O)OC(C)(C)C)CC2(CCOC2)C(F)(F)C1 c1(C(N(C(C)C)CCNC(c2cnc(Cl)s2)=O)=O)ccc2c(c1)C(=O)NC2=O C1(NC(=O)CCc2nccs2)CC2CCC1N(C(=O)CC1CCCC1)C2 c1(OC)ccc(C(=O)NCC2CCN2C(c2ccc(C3(O)COC3)cc2)=O)cc1 c1(C(N2CCC(CNC(CCC=C(C)C)=O)C2)=O)cc(Cl)cc(Cl)c1Br c1(C(=O)NCC2(COC)CN(C(CC(=C=C)C)=O)C2)ccc(F)cc1F C1(C(N(CCN(C(C)=O)C)C)=O)CN(C(C2(F)CC=CCC2)=O)CC(C)O1 N1(C(C)=O)CCOCC1C(=O)NC1CCC(CNC(=O)CCCn2ccnn2)C1 c1(OC)ccccc1C(N1CCC(C(=O)NC(C(F)(F)F)C2CC2)(C(C)C)C1)=O c1(C(C)(C)C(=O)NC2CC2CNC(=O)CC2(CO)CC2)cc(Cl)cc(Cl)c1 CC1(C)C2CC1CN(C(C1CSCCN1C(=O)CC(F)(F)F)=O)C2 C1(OC)CN(C(C2CCCO2)=O)CC1C(N1CCCC1CC1CCC1)=O N1(C(Cc2cn(CC)nn2)=O)CCC2CC12C(=O)NCC(C)C(C)(F)F c1(C(N2CCC(NC(c3cc(C)[nH]n3)=O)CC2)=O)ccc(OC(F)(F)F)cc1Br CC1(C)OCCN(C(=O)NCCCc2coc(S(N)(=O)=O)c2)C1CO C=CCC(C)(CC)C(=O)N(C)CC1CCN(C(C23CCC(C2)C3)=O)C1 C123CC(C1)(OC21CNC1)CNC3=O.C(=O)(N=c1[nH]nc(-c2ccsc2)s1)OC C1(C(=O)NCCC2CCN(C(C(CC(=C)C)C)=O)C2)CC2OC(=O)OC2C1 N1(C(c2nnn(C)n2)C(=O)NC2CC(F)(F)C2)CCN(Cc2nc[nH]n2)CC1 c1(C(C(=O)NCc2cc(N3CC(C)OCC3)ncc2)=O)ccc(F)cc1F c1(OC)cc(CCC(=O)NCCC(C)N(C(=O)C=C(C)C(C)C)C)ccc1F c1(CN2C(C(N3CC4CCCC4C3)=O)CCC2)ccc2nccnc2c1 Cc1cc(=NCC2(CC(C)C)CC2)[nH]c(=NCC(C)(C)CC(F)(F)F)[nH]1 C=C(Cl)CC(C(=O)NC(CCCC)C(=O)NC)NC(C1CCCC1C(C)C)=O C1(NC(CSCCC)=O)CCCC12CN(C(C1C3C4CCC(C4)C13)=O)C2 C12CN(C(C)(C)C1)C(=O)n1cc(cn1)CNC(=O)C2.C12CC3(CC(C3)N1)C2.CC c1(C(=O)NC2C=CCN(C(=O)C(O)C3CCCC3)C2)cncc2nc[nH]c12 c1(C(=O)NCC2(O)CN(Cc3cccc(OCCC)c3)C2)nccc2[nH]ccc12 C=CC1(CC(=O)N(C)CCOC(F)F)CN(C(C2CCC(CO)CC2)=O)C1 C1(C(N(CC(C)NC(C(CCSC)O)=O)C)=O)CCC2C(C1)C2(F)F c1(C(N2CCC(C3CC3)(NC(CC)=O)C2)=O)cc2c(Br)cccc2o1 N1(C(=O)NC2CCC(CNC(=O)C3CC3)C2)CCC(Oc2ncccn2)CC1 C1(C)(OC)CC(NC(C2(C)CC(O)CN2C(c2cc(=O)cc[nH]2)=O)=O)C1(C)C c1(C(C)C)nc(NCC(C)CCO)cc(N2CCC(CC(F)F)C2)n1 C(=O)(C1OCCn2ccnc21)NC1C(CC)N(C(c2ccc(F)cn2)=O)CC1 N1(C(C(CC)(C)C#N)=O)CCN(C(=O)CC2OCCCC2(C)C)C2(CCC2)C1 Cc1n[nH]c(C)c1CC(=O)NCC1CCCCN1C(C1(c2ccn(C)n2)CC1)=O c1(OCC)ccc(C(N2CCCC2CN)=O)cc1F C(=O)(C(C)CNC(=O)C(O)CNC(c1cnc(S)[nH]1)=O)OC(C)C C1(NC(Cc2c(C)ocn2)=O)CCN(C(=O)CC23COCC(C2)C3)CC1 CC1CCN(C(C2C(C)(C)C2(C)C)=O)C(CNC(=O)Cc2ccsc2Cl)C1 N1(C(C2C(NC(C)=O)C2)=O)CCC2(CCN(C(C3C4CC(=O)CC34)=O)C2)C1 C(=O)(CCCCCC#N)N1CC(CC(=O)NCC(C)C(C)(C)C)OCC1 N1(C(C(C)(C)OC)=O)CCOCC(F)(CNC(=O)Cn2cnc(C(F)(F)F)c2)C1 C1(COC)CN(C(C2CC(=O)N(C)C2)=O)CCN1C(c1ccc(C(N)=O)cc1)=O C1(C(C(=O)NC)N(CC(=O)OC)CC)(C(F)(F)F)CCOCC1.C1CCN1 c1(OC)coc(C(=O)N(C2CCC(NC(=O)CCN(C)C(C)=O)C2)C)cc1=O CCC(C)(CCNC(=O)Cc1cc(C)nn1C)NC(=O)Cc1cncc(F)c1 C=CCCCCCCCC(=O)N(CCN(C(=O)CCc1cncnc1)CC)CC N1(C(C2CC23CC3)=O)CC2CCN(C(C3C4CCC5C(C4)CC35)=O)C2C1 N#CC1(NC(C2CCN(C(c3c(I)ccnc3F)=O)CC2O)=O)CCOCC1 C(CC1=CCOCC1)NC(CCN(C(=O)C(CC(C)C)OC)CC#C)=O c1(-c2onc(-c3cnc(NC)c(C)n3)n2)cc(Cl)c2ncccc2c1F N#Cc1cccc(CCC(=O)NC(CNC(=O)Cc2cnn(C(F)F)c2)C2CC2)c1 C1(CNC(CCN(CCC)C)=O)CC(F)CN1C(C1CCC(C)(CC)O1)=O N1(C(C2(CCNC(C3(CC(C)=O)CC3)=O)CC2)=O)CCSCC(C)C1 C1(NC(=O)Cc2cnoc2)CC2CCC1CN(C(c1onc3c1CCCC3)=O)C2 Cc1c(NC(C2CC(C)CN2C(=O)C(=O)N(C)C)=O)cccc1CO C1(C(N(C2CC3N(C(CC=CC)=O)C(CC3)C2)C)=O)CC2(CCCCC2)S1(=O)=O C1(CC)(NC(C2CC(F)C(=O)N2)=O)CCN(C(=O)C(O)Cc2cnc[nH]2)CC1 N1(c2ccc(OC)c(OC)c2)C(=S)NC(c2cn[nH]c2)C2=C1CCCNC2=O C1(C#N)(C(N2CC(N(C(CCC)=O)C)C(F)C2)=O)CCSCC1 C1(C(=O)NC2CCOCC2NC(C2(CC3CC3)CCC2)=O)C2(CCC2)C12CCC2 Cc1cc(C(N)C(=O)Nc2cccc(N3CCCC3)c2)cc(C)c1 N1(C(C(CC)C(=O)OC)=O)CCN(C(=O)CC2CC(=O)NC2=O)CC(C)C1 C(=O)(C(C)(C)CC(F)(F)F)NCC(C)(C)NC(=O)CC1CC2(CCC2)C1 CC1CC(C)(C(N2CC(ON3CCN(C(=O)C4CC4)CC3)C(O)C2)=O)CCO1 N1(C2CN(C(c3cc(C(C)=O)sc3)=O)C2)CC(NC(c2nsnc2O)=O)CC1=O N1(C(=O)CCOC2CCOC2)CCC2(CC1)CN(C(C1CCC1(F)F)=O)C2 N1(C(c2c(C)cns2)=O)CC2CC1CC2NC(=O)C=Cc1csc(C(F)(F)F)c1 C1(NC(=O)CN2CC3CC3C2)CCN(C(c2ccc(C3CC3)cn2)=O)CC1F C(CCC(C)C)(C(=O)NCC1C=CCOC1)NC(C(C(=O)OC)OC)=O CC1COC(CO)CN1C(C1CC(C)(NC(=O)CC(=O)N(C)C)C1)=O C1(C(N2C(CNC(c3ccc(OC)nc3C)=O)CCC2)=O)CCCC2(CCC2)C1 C(=O)(C(O)C1CCc2ccccc21)N1CCCCC(CNC)C1 Cc1cc(=NC(C)CN(C)C(C)C)[nH]c(=NCC2CCCCC2O)[nH]1 C(=O)(C1CCc2nccn21)NCC1N(C(c2cc(Br)cc(C)c2F)=O)CC1 C12(NC(=O)COCC3CCCC3)CCCN(C(c3cccc(Cl)c3)=O)CC1C2 CCC(C(=O)NCCOCCN(C)C(c1sncc1C)=O)C1CCC(=O)N1 C#Cc1ccc(OC)c(C(=O)NCC(CC)(CC)NC(=O)CC2CCC(=O)N2)c1 N1(C(CNC(CC)=O)=O)C2CCC1C(NC(=O)CC1(C)CCC1)C2 c1(CNC(=O)NC(c2ncc(Br)cn2)C2CC2)ccc(F)cc1O Cn1cnc2nc(=NC(C)(C)CCN3CCCC3)[nH]c(NCc3cccnc3)c12 c1(C(=O)OC(C)(C)C)ccc(N2CCOC(CCC(F)(F)F)C2)nc1 C(=O)(CCCCCF)NCCn1cc(CNC(=O)CNC2CC3C=CC2C3)nn1 CC1CSCCN(CC(=O)N(C)C(c2n[nH]cn2)c2cccs2)C1 N1(C(C(C)N(C(C)=O)C)=O)CCC(N=[N+]=[N-])(C(N2CC(c3ccon3)C2)=O)C1 N#Cc1c[nH]cnc1=NCC1CCC2(CCC2)C1NC(c1cncnc1)=O C(=O)(C(O)C(F)(F)F)Nc1cccc(CNC(CC2C(CC)C2(F)F)=O)c1 N(C1CCCc2sc(Cl)cc21)C(Cc1c(C)oc(-c2ccco2)n1)=O N1(C(c2ccc(C)cc2O)=O)CCC(C)N(C(=O)CC2CC(O)C23CCC3)CC1 n1(C(C)C)cc(CC(=O)N(C)CC2CN(C(C3CCCN3C3CC3)=O)C2)cn1 C1(NC(C2(NC(CC=CC=C)=O)CC(F)C2)=O)CCCC2(C1)N=N2 c1(-n2c(C(c3c(C)scn3)NC(C)CCF)nnn2)ccc(Cl)cc1F C(CCC(C)CC(=O)N1C2CCC1C(NC(=O)CCC(N)=O)C2)=C(C)C C1(C(C)C)CCC(C(N2CCOCC2CN(C)C(C2CC2(C)C(F)F)=O)=O)CC1 c1(NC(C2CC(NC(CCCOC)=O)C2)=O)cc(C)ccc1Cl N(C(=NCc1ccccc1)NC1CC1c1ccc(F)cc1)c1snc(CC)n1 C(C)(C(C)(C)C(=O)N(C)CC1(C)CCCC1)NC(COCCSC)=O C(=O)(CCCCCC(C)O)N1C(CCC)CN(C(c2conc2COC)=O)CC1 c1(NC(C2CCCC2(C)C)CC)ncc(C)cc1S(=O)(=O)N1CCSC(C)C1 C(CN=C(NCc1ccc(F)cc1OC)N1CCC(OC)C(C)C1)OC N1(C(CSCC#C)=O)CCCC(C2CC2NC(=O)C(F)OC)C1 C12CCCN(C1)C(=O)C1CCCC21.c1(S)ccc(C(F)(F)F)cn1.CO C1(C(=O)NCCNC(=O)OCC)CCCCN(C(=O)C(C(=O)OC)OC)C1 N1(C(CCCC=C)=O)C2COCC1CC(NC(=O)CC1CCCO1)C2 Cc1ccc(C(C)(C)CC(=O)NC2CC(C)(NC(c3n[nH]cc3C)=O)C2)cc1 Cc1cccc(C=CC(N2CC3CC2C3NC(=O)C(C)Oc2ccccc2)=O)c1 N1(C(C2C(NC(c3cnc(C)s3)=O)COC2)=O)C(C)CCC1(C)C c1(C(=O)NC(CC2CN(C(C(CC=C)N(C)C)=O)C2)C)cnc2c(n1)CCCC2 O=C(CS(=O)(=O)CCO)N1CCN(C(C2CCCSC2)=O)C(CC(F)F)C1 C1(C)(C(N(CCC(N2CC(OCC#C)C2)=O)CC)=O)CCCN1C c1(OC(C(=O)NC(CC)(C)CNC(C2(C(C)(F)F)CC2)=O)C)ccc(Cl)cc1 C1(NC(c2cc(C3(C)CCC3)[nH]n2)=O)CN(C(C23COCC2C3)=O)CC1C(F)F N1(C(c2ccoc2Cl)=O)CC(C2CCCN(C(C3CCC4CCC3O4)=O)C2)C1 C(=O)(CCCCCF)NCCOCCC(=O)NCC1C(C)(C)COC1 C12(OC)CC(C(=O)NC3(CCNC(=O)Cc4sccc4C)CCC3)(C1)C2 c1(C(N2C(CNC(C(=O)OCC)=O)COCC2)=O)cc(F)c(F)cc1I C1(CN(C(C2(COC)CN(C(=O)CC3COC(=O)C3)C2)=O)C)CCCC1(C)C c1(N2CCC(C(=O)Nc3cncc(OC)c3)C2)ncc2c(ccn2C)n1 c1(C(=O)NC(C#C)CO)nnn2c1CSCC2 c1(C(=O)NC2(CO)CCN(C(Cc3c(C)ccs3)=O)C2)ccc2nn[nH]c2c1 c1(C(N(C2CCCC(NC(c3c(C)ocn3)=O)C2)C)=O)ccc2nnn(O)c2c1 N1(C(C(CC=CC)CC)=O)CC2(CCN(C(C3CCS3(=O)=O)=O)CC2)C1 N1(C(C(CCCN(C)C)OC)=O)CCC2CN(C(c3ccnc(OC)c3)=O)CC12 C1(N(C(Cc2c(C)ccs2)=O)C)CN(C(=O)C(C)C(F)(F)F)CC12CC2 c1(CNC(NC2C(C)C2)=NCCc2ccc(F)cc2)ccc2c(c1)CCC2=O CCCCC(C)CCC(=O)N1CC2CC(C1)CN(C(c1ccc(SC)cc1)=O)C2 C(=O)(C(F)C(F)(F)C(F)(F)F)N(C)CC1CCN(C(CN(C(=O)OC)C)=O)C1 c1(NC(C2(O)CCN(C(c3cnc(CC)o3)=O)CC2)=O)cc(F)c(O)cc1C C1(CC)CN(C(c2cc(C3CC3)n(C)n2)=O)CCN1C(=O)CSC1CC1 N1(C(C(C)C2CCC2)=O)CCCCC2(C1)CN(C(C1(CO)CCCC1)=O)C2 Cc1cc(C(=O)N(C2CN(C(=O)Cc3sccc3Br)CC2O)C)oc1C c1(C(=O)NC(c2cccc(F)c2)CC)cc(Cl)sc1Cl C(=O)(C(F)(F)C(F)(F)F)N1CCCN(c2cc(C(C)C)nc(Cl)n2)CC1 Cc1cc(C(=O)N(CCCCNC(=O)CC(C)C)C)c2c(C)n[nH]c2n1 c1(OC)cc(NC(=O)CCOCCCNC(=O)CSC)ccc1C N1(CC(=O)NCC2C=CC(NC(C3(O)CCSCC3)=O)C2)CCC(=O)NC1=O N#Cc1csc(C(=O)NCC2(NC(=O)CC3CCCS3(=O)=O)CCOCC2)c1 N1(C(c2nc(CCCOCC)co2)=O)Cc2n[nH]cc2C1C(=O)NC(=O)CNC Cc1sc(C)c(C(=O)NCC(CO)NC(=O)C2=CCSC2)c1C#N N1(C(C23N(CC(OC)C2)CCC3)=O)C2CCC1CN(c1cncc(Cl)n1)CC2 n1(CC)cc(C(N2CCCC2CN(C(=O)C(F)(F)c2csc(C)c2)C)=O)cn1 CCC(C)(CC)C(=O)N(CC(C)NC(c1cc(C)ccc1Cl)=O)C C1(NC(c2n(C)nnc2)=O)CCN(C(=O)CSc2cccc[n+]2[O-])CC(O)C1 N1(C(=O)OC(C)(C)C)CCC(n2cc(NC(=O)NC3(CCC)CC3)cn2)C1 O=C(C1COc2ccc([N+](=O)[O-])cc21)N1CC2(CC(NC(C3(Cl)CC3)=O)C2)C1 Cc1ccc(C)n1CC(N1CC2CC1(CNC(=O)CC1CC1)C2)=O C(CCCC(F)(F)F)NC(C(C(C)NC(=O)C(C)(F)c1ccon1)C)=O CCC(C)(CNC(C1CC1c1ccco1)=O)NC(=O)CCc1cnccn1 CC1(CNC(C2C=CC=CC=C2)=O)CCCN(C(C2(CO)CCCO2)=O)C1 c1(NCCSC)nc(N2CC(C)CC2C(=O)Nc2ccc(O)cc2Br)ncc1Br N1(C(CC(C)(C)C)=O)CC2CC(NC(c3cnn(CCO)c3C(C)C)=O)CC1C2 C(=O)(C1Cc2ccc(F)cc21)N1CCC(NC(C(c2ccc(C)s2)C)=O)C1(C)C CCCCCCC(C)(CCC)C(=O)NCC(C)NC(c1c(C)cc(C)oc1=O)=O O=C(C#CC1CCC1)NCC1CC(NC(=O)CCn2cccn2)C1 c1(C(=O)NC2CC(CNC(c3ccc(=N)[nH]c3Cl)=O)C2)nnn2c1COCC2 c1(CC)cc(N2CCOC(C)(CNC(c3ccc(=O)n(C)n3)=O)C2)nc(C)n1 Cc1ccc2[nH]cc(CC(=O)NCCCCCCNC(C3(C#N)CC3C)=O)c2c1 N1(C(CSSC)=O)CCC2(COC(CNC(=O)Cc3cn[nH]c3)C2)C1 C1(N(C(C(C)CS(C)(=O)=O)=O)c2cnc3ccccc3c2)COC2(CCNCC2)C1 CC(C)CC(C(N)=O)NC(=O)Cc1cnc(C(F)(F)F)s1 C1(C(N(C)C)C2CC2)CCCC(NC(N2CC3CC2C3C(F)(F)F)=O)C1 CC(C)C(CC(=O)NC1COCCOC1)NC(c1cc(C2CC2)on1)=O c1(C(=O)NC2CN(C(c3c(C)nc(Br)cc3)=O)C2)ccc(S(C)(=O)=O)c(Br)c1 C(CC)(C(=O)N1CC(CNC(=O)Cc2csc(S)n2)(COC)C1)OCC c1(C(=O)NCC(C)(C2CCC2)NC(C(CCC)O)=O)ccc2c(c1)N(C)CC2 C(c1ccc(C)cc1)=CC(=O)NCC1(CN(C(CC(CC)OC)=O)C)CCC1 C#Cc1cccc(N(C)C(C2C(NC(=O)C(CC)C(=O)OCC)C2(C)C)=O)c1 N1(C(CC(C)F)=O)CC2(C(F)(F)F)CC1(CNC(=O)CS(N)(=O)=O)C2 C1(NC(C2CCS(=O)(=O)CC2)=O)CCCCCC1NC(C12CCN(CC1)CC2)=O Cc1nccc(CCC(=O)N(C(C)CCNC(=O)COC2CCCCC2)C)n1 N1(C(c2c(C)nc[nH]2)=O)CCN(C(=O)C=Cc2ccc(Cl)cc2)CC1C C1(CNC(c2cc3sccc3s2)=O)C2CCC(C2)N1C(=O)CC1CC=CCC1 c1(C(N2C(C)CC(CNC(CN(C(C(C)C)=O)C)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 N1(C(CC(COC)NC(C2CCCCC2O)=O)=O)CCCNC(=O)C1 C1(C(C)NC(CSCC=C)=O)CCN(C(c2ccc(N(C)C(C)=O)cc2)=O)CC1 C1(C(=O)NCCn2ncc(CC)c2)CCCN(CC2CNC(=O)C2)C1CC N1(C(c2c(OCC)cccc2)=O)CC2CCC1CN2C(=O)CC1CCCS1(=O)=O C1(CONC(C2(COC)C=CCC2)=O)CC2(CCCC2)CO1 C1(CN(C(=O)Cc2ccc(Br)cn2)C)CCCCN1C(c1ccco1)=O CCCC(C)(C)C(=O)N1CC(CNC(c2cc(C(F)(F)F)ccc2N)=O)C(C)C1 C1(CC)CN(C(C2CCC2(F)F)=O)CCN1C(=O)CCCOC c1(CC(=O)NC2CC(F)(CNC(c3cc(CC)ncc3)=O)C2)c[nH]c(=N)nc1O c1(C(=O)NCC(CNC(C2(COC)CCCC2)=O)CO)cccc(Cl)c1 N1(C(CC=C(C)C)=O)CCCC2(CNC(c3cnc(C4CC4)s3)=O)CCCC12 Cc1c(C)c(C)c(C(N2CCCCCC(NC(C3CCCO3)=O)C2)=O)c(C)c1C Cc1cnc(C(N2CC=CC(NC(C3C=CCS3)=O)C2)=O)c(C)c1 C(C(C)(C)C(=O)NCC1CN(C(=O)C=C(C)c2ccco2)CC1O)SC N1(C(C(C)Cc2ccco2)=O)CCC2(CC(C(=O)N3C4CCC3COC4)=NO2)C1 CCC(C(=O)N1CCOC(C)(CNC(=O)COC2CCOCC2)C1)C(C)C N1(C(C2C(Cl)(C(=O)OCC)C2)=O)CCC(C)(NC(c2cc(C(N)=O)[nH]n2)=O)CC1 C1(C(N(CCN)Cc2n(C)ncc2)=O)C2CC1N(C(c1nc(Br)cs1)=O)C2 c1(C(N2CCC(OCC=C)C2)C(=O)NCC(=C)C)ccc(Cl)cc1 C1(CC(=O)NCCCNC(=O)CSCCc2ccccc2)(CO)CCCCC1 c1(C(C(=O)OCC(C)CN(C)C)Sc2ccccc2)cnn(C)c1 N1(C(CN(C)Cc2ccco2)=O)CC2CN(C(C3CC=CCC3)=O)CC12 c1(OC)cccc(C(C)O)c1OCC(C)C.n12ncc(c1C)NC(=O)CC2 C1(C(=O)OC)CS(=O)(=O)CCN1C(c1ccc2c(c1)CCC2)C(=O)NC(C)C C=CC(C)(CCOC)C(=O)N1CCC(C2CCCN2C(c2cnco2)=O)C1 N1(C(C(C)(C)C#N)=O)CCCC2(NC(C3CCC=CO3)=O)CC2C1 C1(C(N2CC(O)(C(CNC(CCOCC)=O)(C)C)C2)=O)CCN(CC(F)F)CC1 C1(COC)(NC(=O)C(C)C2CCCC2)CCN(C(c2cnccc2Br)=O)C1 N1(C(c2c(CC)c[nH]c2)=O)CC(NC(c2ccsc2SC)=O)C2(CCC2)C1 C(CCC(C)C(=O)N(CCCN(C(=O)C(c1ccc(F)cc1)CO)C)C)OC CCC(C)C(C(=O)N1CCC(C(=O)NCCCOC(F)(F)F)C1(C)C)N(C)C c1(CCC(=O)NCCCOCCNC(=O)C=CC=C(Cl)Cl)cc(Cl)no1 c1(OC)cc(C(N2CCCCC(NC(=O)CSc3ccccc3)C2)=O)cnc1Cl N1(C(C(C2CC2)OCC)C(=O)NC(c2ccccc2)C)CCC2(CC1)OCCO2 CCC(CC(C)C)C(=O)NCCSCC(=O)NCC(O)C(F)F c1(C(=O)NCC2N(C(COC(CC)C)=O)CCCC2)cc2cc(N)ccc2[nH]1 C(CC(C)C)(C(=O)NC(C)CCCO)ONC(CCNC(C)=O)=O C#CCC(C)(CC)C(=O)N1CCN(C(C2CCN(c3ccccn3)CC2)=O)CC1 C(C)(C)(CC(=O)NCC1(O)CN(C(C2(C)CCCCC2)=O)C1)SC c1(C(N2CCC(C(C)C(N3CC4CC4C3)=O)CC2)=O)cncc(OC)n1 c1(CC)nn(C)c(CC(=O)NC(C)CN(C)C(c2cc(Cl)c[nH]2)=O)c1Cl c1(C(=O)NCC2N(C(C3C(C=C)C3)=O)CCC2)c(C)cc(Cl)cc1C C(=O)(C1CNc2ccccc21)N1CCCC(CNC(=O)Cc2ccc(O)nn2)C1 C(=O)(C(COCc1ccccc1)NC(c1cc(-c2cccs2)[nH]n1)=O)OCC C(c1c(F)ccc(Cl)c1F)=CC(=O)NC1C(C)(C)CN(C(C2CCC2(C)C)=O)C1 c1(-c2nc(C)[nH]n2)cccc(C(=O)NCC(O)CNC(=O)C(C)OC(C)(C)C)c1 S(=O)(=O)(c1cc(C=CC(=O)NC(C)COC)cs1)NCC C=CC1CN(C(=O)CC2CC3(CC3)CO2)CC1NC(c1cccc(Cl)c1OC)=O C1(NC(CC(CC)O)=O)CCC2CN(c3ncnc(C)c3OC)CCC2C1 Cn1cnc2nc(=NCCC3CCOC(C)(C)C3)[nH]c(NCc3n[nH]c(=N)s3)c12 C1(OC)CCC(C(N2CCC3(C2)C(=O)N3)=O)CC1.O(C(=N)O)CCO CCCCCCCCCC(=O)NC(CNC(C1CC(C)(C)CN1C)=O)CC C(CC(C(=O)NCCn1cc(CS(C)(=O)=O)nn1)c1ccccc1)=C(C)C c1(C(=O)NCC(CNC(c2c(SCC)nccn2)=O)C)cc(C)c(Cl)c(C)c1 C1(CCCC)CN(C(c2cnoc2C)=O)CCN1C(=O)COCC(C)(C)C C1(C(=O)NCCC2CCCN2C(C2CCOCC2)=O)CC2CCC1O2 N1(C(C(=O)N(C)C)=O)CCC(C(F)(F)F)C(CNC(=O)C(O)c2cnc[nH]2)C1 N1(C(c2c(C)nccn2)=O)CCC2CC2(C(=O)Nc2ccc(CCO)cc2)CC1 c1(CC)nc[nH]c(=NCC2(CNC(C3(O)CC(C)(C)C3)=O)CC23CCC3)c1F Cc1ccc2c(n1)CN(C(=O)C(C)C(C)NC(C1CCC1C)=O)C2 C1(CNC(=O)Cn2ncnn2)COCCN(C(C2(C(F)F)CC2(F)F)=O)C1 c1(C(=O)NC2(C(=O)NCCN3CC(C)(O)C3)C(C)CCC2)cc2n(n1)CCC2 N1(C(c2cc(C)c(Br)cn2)=O)CC2(COC(CNC(c3ccncn3)=O)C2)C1 c1(CC)cc(O)ccc1NC(=O)CC(O)CNC(=O)C(C1CC1)OC C1(NC(C(CC#C)C)=O)CC2CCC1CC2NC(c1ccc2c[nH]nc2c1)=O C12(C(=O)NCC3CCC(NC(C(C(C)SC)O)=O)CC3)CC3CC(CC(C3)C1)C2 c1(C(N2CCC(C(=O)NC(CCC(C)C)C)(C(C)C)C2)=O)cccn2cncc12 c1(OC)nc(C)ccc1C(=O)NC1CC(CNC(C2C(C)CC2C)=O)C1 C(=O)(CC(C)(C)CC(=O)NCCC(C)(C)NC(=O)C(F)OC)OCC C(C(CC)(CC)C(=O)N1CCC(OC(C)C)C1)NC(C(C=C)CC)=O C(CC(C(=O)NC(C)CN1CCCCC1)NC(=O)C=C1CCC(C)CC1)OC c1(C2(C(=O)NCC3C4CN(C(C5C(C(C)C)C5)=O)CC43)CC2)cccc(Cl)c1F C1(NC(c2cc3n(n2)CCC3)=O)CCSC12CN(C(C1(C3CCCO3)CC1)=O)C2 c1(C(=O)NCC=CCNC(C2CCC2F)=O)ccnc2ccc(Cl)cc12 N1(C(=O)COCC(F)F)CCC(CF)(NC(C2CC(=C3CC3)C2)=O)C1 c1(CC)cc(=NCC(C2CC2)NC(c2[nH]cnc2C)=O)[nH]c(C2CCCCC2)n1 C1(C(N2CCC(O)(CNC(c3cccc(CC)n3)=O)C2)=O)CCCCC(C)(C)C1 C(CN(C)C)(C(=O)N=c1ccn(CCO)[nH]1)NC(CC(CC=C)(C)C)=O N1(CC(N2CC(C(=O)NC(CC=C)CO)(SCOC)C2)=O)C(=O)CNC1=O CC1CC=CCC1C(=O)NCC(CO)NC(c1cc(CO)[nH]n1)=O C(CCC(C)(C)NC(c1csc(C(=O)OC)c1)=O)NC(c1cc(CC)[nH]n1)=O N1(C(CC2(NC(C3(C#N)CC3)=O)CC2)=O)CCc2c(O)noc2C1 C1(C(=O)NC(C2CN(C(C3(CC#C)CC3)=O)C2)C)CC(C)(C)C1 C=CC(C(=O)N(CCCOCCNC(C1CCS1(=O)=O)=O)C)OC N1(C(c2cnc(CN3CCCC3)s2)=O)CCCC(c2cn(CCCCF)nn2)C1 O=C1CC(C2CC2)(C(=O)NC2CCN(C(=O)C=Cc3cncs3)CC2CO)C1 N1(C(C2CN(C(C)=O)C2)=O)CC(NC(C2CC(F)C(=O)N2)=O)CC1C c1(CC(=O)N(CCNC(C(C)OCCN(C)C)=O)C)cn2cc(F)ccc2n1 c1(C2C(C)CC2)nc(-c2ccncc2)nn1Cc1cccnc1 c1(C(=O)NC2C(NC(CCNC(=O)C=CCl)=O)COCC2)ccnc(Cl)c1O C1(O)(CNC(=O)C(O)Cn2cncn2)CCN(C(C2CC(F)(F)C2)=O)C1 C=C=CC(C)C(=O)N1CCC(OCCNC(C2(C(F)(F)F)CC=CCO2)=O)CC1 C(=O)(CC(C)(C)C(=O)N1CCCC(NC(C2CC=CCO2)=O)C1)OCC C1(CC)CC(C(=O)NC2CCC(C)CC2)CCN1C(=O)C#CC(C)C N1(C(C(C)OC2CCCC2)=O)CC2(CCNC(=O)C=CC(C)(C)C)CCC1C2 Cc1cc(C(N2CCN(C(C3CC3F)=O)C(CF)C2)=O)c(C)n1-c1cnn(C)c1 C1(C(=O)O)CCN(C(C2CC2C(F)(F)F)=O)CC1C(c1ccccc1)C1CC1 Cc1scc(C(=O)NCC2(C)CC(NC(=O)CC3SC(=N)NC3=O)C2)c1C Cc1nc(CNC(c2ccon2)=O)oc1C(=O)N(C)CC1CCOC1 c1(CC)nc(NC(=O)C(=O)Nc2ccc(OC)cn2)sc1C c1(C(CC(=O)OCC)NC(=O)N(CCCC(=O)NC)C)ccc(Cl)cc1 C1(NC(C(C)=CC)=O)COC2C(NC(C3(C)CCC34CCC4)=O)COC12 c1(CN(c2ccc(N)cc2F)C(c2cc(C)c(Br)s2)=O)c[nH]c2ncccc12 N1(C(c2c(C)ccnc2Cl)=O)C2CCCC1CC(NC(C1CCCC3CC13)=O)C2 C1(CCC)CC(C(=O)N(CC(=O)NC2CC2CCOC)CC)C1 C=CC(C)(CCOC)C(=O)N(C)CC1CCCN1C(=O)C(n1nc(C)cc1C)C CC(C)C(C(=O)NCC(N1CCCC1C(N)=O)=O)NC(=O)C1CC1 C(=O)(CCCC(C)(C)C)NCCC(CCNC(CC1ON=C(CC)C1)=O)C c1(C(=O)NC2C(NC(CCCOCCC)=O)C2)ccc(NC(C)=O)cc1 N1(C(CC2C=NN(C)C2=O)=O)C(C(N2CC(C3CC3)(CO)C2)=O)CC2CCCC12 C1(CC(=O)NCC=CC)COCCN1C(c1cnn[nH]1)=O c1(C(=O)NCc2nc(O)n[nH]2)ccc(S(=O)(=O)NCc2ccco2)cc1 C1(OC(C)=O)CCN(S(=O)(=O)NCC2CCCC3(CCOC3)O2)C1 CCC(C)C(CC(=O)NCC1(CC2CCC2)CC1)NC(=O)CCC(C)N(C)C N1(C(CC(CCC)O)=O)CC2CC1CCN2C(=O)CNc1ccc(C(N)=O)cc1 N1(C(c2c(CC)nco2)=O)C(C(=O)N(C)Cc2cn(C)nc2C)CC2CCCC12 N1(C(c2ccc(CCC)c(N)c2)=O)CC(C)N(C(=O)CSC)CC1C C(=O)(CCC(=O)N(C)C)N(CC(C)N(C(=O)C(c1ccsc1Br)(F)F)C)C C=C(CNC(c1ccc(CN)cc1C(F)(F)F)=O)c1cccc(F)c1 c1(C(C(=O)NCCCOCCNC(CSc2n(C)cnn2)=O)F)ccc(F)cc1 C1(NC(c2c(C)cc[nH]2)=O)CCC2CN(C(=O)CC3(C)OCCO3)CC12 c1(C(=O)NCC2N(C(C(F)OC)=O)CCCCC2)[nH]nc2c1CCC2(C)C C(=O)(C(=O)CC(C)C)NCC(C)(C(C)C)NC(c1[nH]cc(CC)c1)=O CC1=CCSC1C(=O)NCC(c1ccccc1)CNC(=O)COc1ccsn1 CC1=C(C(=O)N2CC(NC(c3scnc3Cl)=O)CC2C)C(=O)OC1(C)C C12CCCN(C1C)C(=O)C(C(C)CC)ONC2=O.C=C1CC(COC)C1 C1(CNC(c2ncccc2C2CC2)=O)CC2CCC(C1)N2C(c1cc(F)n[nH]1)=O C(=O)(C#CC1CCOC1)N(C(C)CNC(=O)Cc1sccc1Cl)C C1(NC(C)=O)CCN(C(C2CSCN2N2C(C)CCC2C)=O)C1(C)C C1(C(N(CCCNC(C2CCCO2)=O)C)=O)CCS1(=O)=O c1(C(=O)NC(CNC(C2CC(C)CC(C)C2)=O)C(C)(C)C)cc2c[nH]cnc-2n1 N1(C(C2CCN(C(c3c(CC)cns3)=O)C2C(C)C)=O)CCC12CCSCC2 c1(C(CNC(CN(C2CCCC2)C)=O)(C)C)ccn(C)n1 CN1C(=O)N(C)C2(CCN(C(C3CCCN3CC(F)(F)F)=O)C2)C1=O c1(CC(=O)NCC(C2CC2)NC(C2CCC(=O)NC2)=O)c[nH]c2cc(F)ccc12 N(C1c2ccccc2CC1NC(C1(C)CC=CC1)=O)C(c1cc(C)nc(O)c1)=O c1(C(C(=O)NCC(F)F)N(C(C)(C)C)CC=C)cc2cc(Cl)ccc2s1 C(=O)(C1CCCc2c(N3CCc4cc(F)ccc4C3)ccnc21)OC N1(CC)CCN(C(c2ncc(C)s2)C(=O)NC(C)C(=O)OC)CC1C CC1CN(CC(=O)Nc2cccc(F)c2)CCC1NC(c1cc(C2CC2)no1)=O CC1(C)CC(C(N2CC(F)(CO)C2)=O)CN(C(=O)COC2CCCCC2)C1 C1(C(=O)NC(CC)CN(C(=O)C=CCOC)C)CN2CCCN1CC2 N1(C(c2cnn(CCC)c2C)=O)CCN(C(c2ccoc2CC(N)=O)=O)C2CC12 c1(C(N2CC(CCNC(C(CCC)O)=O)C(C)C2)=O)cc(C)c(C)nn1 N1(C(C(C)NC(C)(C)C)=O)CC2CCN(C(=O)CNS(=O)(=O)N(C)C)C2C1 c1(C(=O)NCCN(C(=O)C(N)=O)CCCN(C)C)ccc2c3c(cccc13)CC2 CC(CCNC(=O)CC1CCOC1)N(C(=O)CCc1cn[nH]c1)C Cn1ncc(C(=O)NCC2C=CCN2C(c2cnc(=N)[nH]c2)=O)cc1=O c1(C(=O)NCC(C(C)(C)C)NC(CC(C=C)C)=O)c(C)nc2sccn12 CC(C)(C(=O)NCCOCCCNC(=O)C(O)c1ccsc1)C1CCC1 c1(OC)c(Cl)cc(C(=O)NCC2CCC(CO)CC2)c2ncccc12 c1(CC)cnccc1C(N1CCC(C(=O)NCC(O)CC(C)C)CC1)=O c1(C(N(C2CCN(CC3CN(C)C(=O)CC3)CC2)C)=O)c(Cl)ccc(F)c1F c1(CC(=O)NCC2CC(NC(C(C=C)O)=O)C2)cccnc1Br C1(NC(C2CN(C)C2)=O)CCOC12CCN(C(=O)C1CNc3ccccc31)CC2 c1(CC)cn2c(n1)CC(C(N1CCCC(F)(CNC(=O)CCCCF)C1)=O)CC2 C1(NCc2c(C)cnn2C(C)C)COCC(C)(C)C1 c1(CC(=O)NCC(C)CNC(=O)CC2CCCCCC2)ccc([N+](=O)[O-])c(N)c1 c1(N2C(CC)CN(C(C3C4COCC34)=O)CC2)nc(C)nc2c1CCC2 C(CN=C(NC1CCC1)N1CCC(F)(F)CC1)N1CCN(CC(C)C)CC1 CCCCC(CNC(=O)CC1COCCN1C(=O)CCc1cn(C)cn1)CCC Cn1cnc2ccc(C(N3CCC(C(O)CNC(C4CCCO4)=O)CC3)=O)cc12 Cc1cccc(C(=O)NCCCCCC(=O)NC2(C)CCCC2C)c1C Cc1c(C(=O)NCCC2=CCN(C(=O)CCOC3CC3)CC2)[nH]c2c1CCCC2 N1(C(CC(=C)C)=O)CCC(NC(=O)C(C)(C)C2CC2)CC1C Cc1c(C(=O)NC(C(N)=O)C(C)(C)C)[nH]c2ccccc12 c1(OC)ccncc1C(=O)NCCCN(C(=O)CCc1nc(C)cs1)C c1(C(=O)NC(C=CC(=O)NC(c2cc[nH]n2)C)(C)C)ccn2ccccc12 C(=O)(C#CC1CCCC1)NC1CC(OC)CN(C(=O)C=Cc2nc(C)co2)C1 Cc1cc(C(=O)NC2(CNC(=O)COc3cnn(C)c3)CCC2)c2nccn2c1 C1(NC(c2c(CC)onc2)=O)CCCC12CCN(c1ncn(C)c(=O)c1Br)CC2 CCC(C)(CCC(C)C)C(=O)N1CCC(CNC(c2ccc(O)c(F)c2)=O)C1 N1(C(C(C(=O)OCC)C2CC2)=O)CC2CCC(C1)N2C(=O)CS(=O)CC c1(C(=O)NCC(=C2CN(C(CSSC)=O)C2)F)ccc(=O)n(O)c1 CS(=O)CCC(=O)NCC1(O)CC(CNC(=O)CCNC(=O)OC)C1 N1(CC)CCC(c2nnnn2CC(F)F)(NCCCc2ccccc2F)C(C)C1 C1(Cn2cc(N(c3ccco3)C)c(-c3ccccc3)n2)CCCCC1(C)C C1(CNC(c2cnc(CC)s2)=O)CC(NC(=O)CC2CCC2C)C1(C)C C(N=c1[nH]n(C)c(C)c1[N+](=O)[O-])C1C(NC(c2scc(C)c2)=O)C2(CC1)CCC2 Cc1nnc(CC(=O)NCCOC2CN(C(C3CC(n4cccn4)C3)=O)C2)s1 C1(C(=O)NCC2C=CC(NC(CCc3c(C)nn(C)c3)=O)C2)CCC(C)(C)CO1 C1(C)(NC(c2c(CC)ccs2)=O)CCN(CC2CCCOC2)C1 C(C(C(C)C(C)C)NC(c1coc(C(F)F)n1)=O)NC(CC(=C)Br)=O c1(C(N2C(C)CC(NC(c3cc(F)n(C)n3)=O)C2)=O)cc(O)c2ccccc2c1 C(=O)(C1CCCc2ccccc21)N1C(CNC(CSCC)=O)CC(OC)C1 c1(C(N2C(C)C(NC(=O)CCC3CC(C)(C)CO3)CC2)=O)ccc2c(c1)CC2 N1(C(C(C)(C)C)=O)CCOC(NC(=O)NCC2(c3ccc(Cl)cc3)CC2)C1 S(=O)(=O)(c1cnn2ccc(N(C)CCOC)nc12)NCC1CC(=C)C1 C1(CC)CN(C(=O)C(C)c2cccs2)CCN1C(c1cc(F)cn1C)=O C(=O)(C(C)CC(=O)c1ccccc1)NC(CNC(C(n1cc(C)nc1)(C)C)=O)C c1(CC(=O)NCC(CO)NC(C2OCCC(C)C2)=O)c(F)cc(F)cc1F c1(NC(C2N(C(C3C(C)C3)=O)CCCC2)=O)cncc(C#N)n1 C1(CC(=O)NC(c2ncc[nH]2)C)CCCC(NC(c2ccncn2)=O)C1 CC(C)C(F)(F)CC(=O)N(CCCNC(C1C(C)C1C)=O)Cc1ccccc1 C(CS(=O)(=O)CC(=O)NCCOCCN(C(=O)C(=O)N=S(C)(C)=O)C)OC Cc1cc(C(N2CCCN(C(C3OC4CCC3C4)=O)CC2)=O)ccc1Br Cn1cc([N+](=O)[O-])cc1C(N1CCC(NC(=O)CSCc2ccccc2)CC1)=O C(=O)(CCCC(=O)c1ccc(Br)cc1)NC(C(=O)OC)Cc1cncn1C C(=O)(C1=CCN(C(=O)CSC2CC2)CC1)NCCc1cc(C)n(C)n1 C1(O)(CNC(c2cc(C(N)=O)ncc2)=O)CCN(C(C2CCS(=O)(=O)C2)=O)CC1 c1(CC)cc(C)nc(N2CC3CN(Cc4ccc(N5CCCCC5)s4)CC23)n1 N1(C(CCCCC#C)=O)CC(CO)C2(C1)CN(C(=O)C(CCC)N(C)C)C2 C1(C(=O)NCc2c(C)ncs2)CCC(C(C)C)N1C(=O)C=CC(=O)N(C)C N1(C(C2(NC(C)=O)CC2(C)C)=O)CCCC(CC(=O)NCC(=O)NC(C)C)C1 CC1(C(=O)N2CCN(C(c3cc(O)no3)=O)C(CO)C2)OC(=O)c2ccccc21 c1(CNC(=O)NCc2ccn(-c3ccc(Cl)cc3)n2)cnc2c(F)cccc2c1 c1(OC)cc2ccc(NC(=O)C(C)C3CCC3)cc2cc1OC C1(NC(C(C=C)O)=O)CC2(CCN(C(=O)C(C)(C)CC#N)CC2)C1 N12CCC(N(C)N3CCN(CC3)CCN(C)CC1)C2.S(C)(=O)(=O)CC C1(C(=O)OC)CCN(C(=O)CC2CC2CNC(C23C=CC(CC2)C3)=O)O1 c1(C(=O)NC2C(NC(C3NC(=O)OC3)=O)CCCC2)cc(F)cc(F)c1 c1(N2CC(OCC(=O)NCC)C(O)C2)ccc(Cl)cc1[N+](=O)[O-] CCCCC(=O)C(=O)NCC(C)(C)CC1CN(C(=O)CC2CCCCC2(C)C)C1 Cc1sc(C(=O)N(C2CCN(C(C3CCN(C)C3=O)=O)C2)C)cc1[N+](=O)[O-] C1(C(N(CCC#C)C)=O)CC2CCC1N2C(C1(CC=C)CCOC1)=O N1(C(c2c(CCC)[nH]cc2)=O)CC(C)(C)CC1C(=O)N(C)CC1(C)CCC1 c1(CNC(C(n2cc(COc3cnn(C)c3)nn2)C)=O)nncn1C Cc1nc2ccnn2cc1C(=O)NC1(CF)CCN(c2snc(C)c2C#N)C1 c1(C(=O)NCC(CCNC(CSCCOC)=O)O)ccnc(F)c1 c1(C(=O)NC2CC(F)(CNC(CCC3C(C)C3)=O)C2)c2c(c[nH]c1=N)CCC2 Cc1cc(C(=O)NCCOCCNC(=O)C(C2CCC(=O)N2)C)nc(O)n1 N1(C(CC2(CC)CCC2)=O)CCCC(O)(CN(C)C(C2CCC2C)=O)C1 N1(C(C(C)OCCC(C)C)=O)CCOC(C(=O)NC2CCOCC2F)C1 c1(C(=O)OC)ncc(OCc2nc(F)ccc2Cl)cc1F Cc1oc(C(C)C)cc1C(N1CC(NC(=O)CCN2CCCC2=O)C(CO)C1)=O c1(CC(=O)NC(C)CC2CCN(C(c3cn(C)cn3)=O)CC2)c(Cl)cccc1Cl N1(C(CC(C=C)CC)=O)CCC(NC(c2cc(OC)cc(Cl)c2F)=O)C(C)(C)C1 C1(NC(C(c2ccc(Cl)s2)C)=O)CC2(C1)CC2N=c1ccc(C(F)(F)F)n[nH]1 c1(C(N(CCN2CCN(C(C(CC#C)(C)C)=O)CC2)C)=O)[nH]nc2cnccc12 c1(CCC)n[nH]c(=NC2CCN(C(c3cc(C)cnc3Cl)=O)C2)s1 C(CC(O)C(=O)N(C1CCN(Cc2ccnc(OC3CCCC3)c2)C1)C)SCC Cc1[nH]c2ccccc2c1C(=O)C(=O)NC1(CNC(c2cncnc2)=O)CCC1 C(CS(=O)(=O)CC(=O)N(C1CCC(=O)NC1)C)OC N1(C(C(C)(CC2CCC2)OC)=O)CC2(CC(NC(=O)Cc3cnn(C)c3)CO2)C1 CC1C(NC2(CO)CCC2)CCN1C(=O)C=C1CCC1.C(=O)(CCN(C)C)N Cc1ccc(C(=O)NCCC2CSCCN2C(=O)C#CC(=O)N(C)C)cc1F N1(C(CC(C=C)C)=O)CCOC2CCN(C(=O)Cc3cccc(Cl)c3F)CC12 N1(C(c2cnc(CC)o2)=O)CCCC(F)(C(N2CCC(O)C(O)C2)=O)C1 C1(c2nc(CNC(C(F)OC)=O)[nH]n2)CCN(C(C2(CC3CCC3)CC2)=O)CC1 N1(C(C(CCNC(=O)CC2(O)CCC2)OC)=O)CCC2(CCOC2=O)C1 C(CC(=O)NCCn1cnc(C)c1C)(C(F)F)NC(C1(COC)COC1)=O C1(C(=O)OCCCC)CC(NC(=O)CNC(=O)CCCN(C)C(C)=O)CCO1 N1(C(CC(C)F)=O)CCC2(CCC2NC(c2ccc(C3CC3)c(Cl)c2)=O)CC1 C1(C(=O)NCC2C(C)CCN2C(C2CCCSC2)=O)CCCCN(C)C1=O CC(CCCNC(=O)CN1CCC1C)NC(C1(c2ccccc2)CCC1)=O Nc1c(C(=O)NCC2CCN(C(=O)CC3=CCCCC3)C2)cc(Cl)cc1F C(=O)(C1=C(C)CCCC1)NCC(C)N(C(c1nc(COC)[nH]n1)=O)C c1(OC)cc2ccc1CN1CC3N(C(C3)C1)C(=O)c1c-2cccn1.C(C)(C)OC C1(C(=O)NC(CCNC(CN(C(=O)OC)C)=O)C)Cc2n[nH]cc2C(=O)N1 c1(OC)ccc(OCC(=O)NCC2CCC(NC(C3CC(O)C3)=O)CC2)cc1 C1(C)(C(=O)OCC)CCN(C(c2sc(Cl)cc2Cl)C(=O)NCCSC)C1 c1(-c2c(C(=O)NCC(CNC(CC3(C)CC3)=O)F)c[nH]n2)ccc(Cl)cc1 c1(CCC)nc(C)c(C(=O)NCC2(C)CCCN2C(=O)C(O)C(F)F)o1 c1(N2CCC(S(C)(=O)=O)CC2)nc2c(c(=NCc3csc(Cl)c3)[nH]1)CCCCC2 N1(C(C2N(C(COCCOC)=O)CCC=C2)=O)CCCN(C)C(=O)C1 c1(NC(CC2CN(C(c3c(CC)n(C)nn3)=O)C(C)C2)=O)cc(C)c(F)cc1O c1(NC(C2CCCN(C(C(CC=C)OC)=O)C2CC)=O)cnc2c(c1)CCC2 CC(C)C(C(C)NC(=O)CNC(=O)CN(C)C)NC(c1c[nH]c(=N)o1)=O c1(C(=O)NCCN(C(=O)C(O)Cc2cnn(C)c2)CCOC)cc(CO)ccn1 C(=O)(CCCCC(N)=O)N1CC(CNC(=O)CCCN2CCCC2)CC(C)C1 c12cn(nn1)C1CCC(C1)C(=O)NC2C1CC1.C1(OOC(=N)O)CC(CF)C1 c1(C(N2CCC3CN(C(C4C(=C)C4)=O)C3C2)=O)ccc2c(c1)OCCO2 C(=O)(C(C)(C)C(C)(F)F)N1CCC(N(C(C2CN(C)C2)=O)C)C1 c1(COC)c(C(N2CC(NC(=O)CC(C)(C)C)C3CC3C2)=O)sc2ccccc12 C12(NC(c3ncc(OC)cn3)=O)CCC(CN(C(=O)CC(O)C(C)C)C1)C2 c1(CC(=O)NCC(CNC(C2(C)CCOC2)=O)(C)O)cnn2ccccc12 N1(C(c2cccc(C)c2)=O)CCN(C(c2nc(C)ccc2Br)=O)C2CC12 C(CC(C)C)(C(=O)NOCC1(COC)CCC1)OCC N1(C(c2c[nH]c(=N)s2)=O)CC(NC(c2ccccc2Cl)=O)CC(F)(F)C1 c1(C(N(C2CCCCN(C(C(C)OC)=O)C2)C)=O)oc2ccccc2c1C N1(C(C(C)c2ccco2)=O)CCC(C)(C)CC1C(=O)N1CC(O)CO1 C(=O)(CCCCC1CC1)NC(C1CCCCN1C(c1ccn(C)n1)=O)C Cc1nn(C)cc1C(C)C(N1CCCC1CNC(=O)Cc1cn(C)cn1)=O N1(C(C(CC#C)(C)NC(=O)CCCCC)=O)CC2CC(CO)C(C2)C1 CC1CN2CCN1CC2C(=O)NC1CN(C(c2cc(Br)c(C#N)s2)=O)C1 Cn1cc(Br)cc1CNS(=O)(=O)Cc1cscc1Br N1(C(c2ncc(C)nc2)=O)CCC2(C=C(C(=O)N3CC4CC5CC4C3C5O)C2)C1 N1(C(C(CN(C)C)NC(c2ncc(OC)nc2)=O)=O)CCCC(F)(CO)C1 C1(C)(CNC(C(C)C#N)=O)CCCN(C(c2ccc(Cn3cc(F)cn3)o2)=O)C1 N1(C(C(COC)C)=O)CCCCC1C1(CNC(=O)C(C(C)O)NC(C)=O)CC1 Cc1n[nH]c(C)c1C(=O)NC(C)C(C(C)C)NC(C1CCN(C(C)C)CC1)=O c1(C(C)C)ccc(C(=O)NCC(F)CNC(C2COC(=O)O2)=O)s1 N1(C(c2cc(C)n(C)c2)=O)CCCC2(NC(=O)CC(O)CC(C)(C)C)CCCC12 C1(OC)CCC2(CC1)CN(S(=O)(=O)Cc1ccc(Br)cc1)C2 c1(OC)c(F)cc(CNC2CC2C(=O)NCC2CCCOC2)cc1F c1(C(=O)NC(CNC(c2c(SC)cccc2F)=O)CO)cc(C)cc([N+](=O)[O-])c1 c1(C(=O)OC)cc(Br)c(NC(N2CCC(O)CC23CC3)=O)nc1C C(=O)(C1CCCc2ncccc21)NC1CCC(N(C(C2C(C(C)O)C2)=O)C)CC1 C(C(COC)CC(=O)NC1CN(C(c2ccon2)=O)CC1OC)OC c1(OC)ccnc(NCC(N2CCC(NC(=O)C(O)c3ccsc3)C2)=O)n1 c1(C(=O)NC(C)C(C)NC(c2c(Cl)cnn2C)=O)ccc(O)c([N+](=O)[O-])c1 C1(CN2C(=O)CCC2)CCCCN1C(c1cnn(CCF)c1)=O.C12CCN(C1)C2 Cc1[nH]nc2cc(C(=O)NC3(CCNC(C4SCCC4C)=O)CCC3)ccc12 c1(C(=O)NC(C2C(C(N3CC(CC(C#C)C)C3)=O)C2)C)csnc1Cl c1(N2CCC(C(C)NC(C(CC(C)C)C)=O)CC2)cc(C#N)c(F)cc1[N+](=O)[O-] CCCC(CCC)C(=O)N1CCC(C(=O)N(CC(N)=O)CC(C)C)CC1 C(=O)(C(C)(C)CC(F)(F)F)NC1C(CNC(c2cc(C)nc(O)n2)=O)CCC1 N1(CC(N2C3CN(C(c4ncn(C)c4)=O)C(C3)C2)=O)C(=O)CC(C)(C)C1=O N1(C(c2cc(C)c(Cl)cc2)=O)CCC(C2CCCN(C(=O)C(=O)N(C)C)C2)C1 C(=O)(C(C)CC(C)(C)C)N1CCC(C(=O)NCCCC(=O)N(C)C)(OC)C1 N1(CCCNC(C(C)NC(CC)=O)=O)CCN(C(=O)Cc2ncn(C)c2C)CC1 C1(C(=O)NC2C(OCC=CC)CCC2)(NC(=O)CC(C)CN(C)C)CC(C)(C)C1 C(=O)(C1=COCCO1)Nc1cccc(CC)c1.C12(OC)CCN(C1)C2=O c1(C(=O)NC2(CO)CN(C(C3C(C=C)OCC3)=O)C2)nccc2ncccc12 C(C(CC1CC1)C(=O)NCCc1cncs1)NC(C(=O)NCC(F)F)=O C1(NC(CN2CCC(C)(O)C2)=O)(CO)CCCN(C(c2cc(C(N)=O)[nH]n2)=O)C1 N1(C(CN(C)C(N)=O)=O)CCCC(CNC(=O)C(=Cc2c[nH]cn2)F)CC1 C12(NC(C3C(CNC(Cc4cc(COC)on4)=O)CCC3)=O)CCN(CC1)CC2 C(CC(C)(C)NC(C1CC2CC2C1)=O)N(C(=O)CCCO)C.C(C)(C)(C)OC C1(NC(c2c(N)nccc2)=O)CN(C(=O)C(F)C2CCC2)C2(CCCCC2)C1 c1(C(N(CC(C)O)CCNC(C2CCCO2)=O)=O)cc(Br)cc(F)c1F C(=O)(C1=COCCC1)NC1(C)CC(NC(C2C3CNC(=O)C23)=O)C1 c1(C(N2CC(CC(=O)Nc3c(CC)cccc3)OCC2)=O)cc(OC)cc(Br)c1 N1(C(C(C)N2CC(O)C2)=O)CCC(OCCNC(=O)OC(C)(C)C)C1.N(C)C CC(C)CC(C(=O)NC1C2CCC1N(C(=O)CCOCCN(C)C)C2)C(C)C c1(CC)ccccc1C(=O)NC(C)C(C)NC(C1(CSC)CC(F)(F)C1)=O c1(C(=O)OC)nc(=NC2CC(F)(CNC(=O)CC3CC3(Cl)Cl)C2)c(F)c(Cl)[nH]1 c1(C(C(N2CC3C(CNC(C4(C(=O)NC)CC4)=O)C3C2)=O)O)ccc(Cl)c(Cl)c1 CC1CCC(Cl)=C(C(=O)NCC2(O)CCCN(C(c3cc(Cl)n(C)n3)=O)C2)C1 c1(C(C)C)c(C(N2CC(F)(CNC(=O)C=C3CCN(C)C3)C2)=O)cnn1C N1(C(CCCC=C)=O)C(CNC(C2CC(C(C)C)C2)=O)CC2CCCCC12 c1(C(N2CCC3(NC(c4cnc(O)o4)=O)C(C2)C3)=O)cc(F)c(F)c(F)c1F c1(C(=O)NCC(C)(Cn2cccn2)NC(=O)C2CC2)cc2ccncc2[nH]1 C1(NC(CCc2ncc(C)[nH]2)=O)C2CCC1N(C(C1CC(C)C1)=O)C2 Cc1oc(CNC(C2CCCC(C)C2)=O)nc1C(=O)NC1CSC1 C1(CC)CN(C(=O)CC2CC(OC)C2)CCC1NC(c1cnc(S)nc1)=O C(=O)(C1CCCc2scnc21)NC(CNC(c1coc(C(F)F)n1)=O)CO c1c(CC2CCCN2CCC2CCCO2)nnn1CC1CCCO1 Cc1cccc(C(N2CC=C(CNC(=O)C(F)C3CCOC3)CC2)=O)c1C C1(N(C)C(c2cccc(OC(F)(F)F)c2)=O)CS(=O)(=O)CC1O C1(CC)(NC(=O)Cc2ccnn2C)CN(C(=O)CC2CC3(CC3)C2)C1 N1(C(c2cccc(CC=C)c2)=O)CCC(C)C(NC(C2(C(C)(F)F)CC2)=O)C1 CCC(C)(CC)C(=O)N1CCC(F)(CNC(=O)Cc2ccc(C(N)=O)cc2)CC1 C(=O)(C1CCCc2cncn21)N1CC2C(CNC(c3c(N)cn(C)n3)=O)C2C1 C12(CCN(C(c3nc(O)sc3C)=O)CC1)C(=O)N2.c1(COC)c(F)cncc1F N1(C(C(CCC)CC)=O)CC2(CC(C(N3CC(C(C)(C)O)C3)=O)CO2)C1 c1(OC)cccc(NC(C2CCC2C(=O)O)=O)c1Br C(CCC(C)C)(C(=O)NCCC1CN(C(=O)Cc2ncc(C)o2)C1)NC(C)=O c1(C(=O)NCC2CCN(C(CCCC(CC)C)=O)CC2)cc2cccn2c(O)n1 CC1CCC=C1C(=O)N1CCN(C)CC1CNC(c1ccn(C)c1)=O C=CC(C)(CCOC)C(=O)NCC1COCC1NC(c1cc(C)no1)=O c1(C(N2CCC(C(=O)NC(C(C)C)C)CC2)=O)ccnc2ncnn12 CC1(C)OCCOC1C(N1CCCC(Cn2cc(CC(O)C3CC3)nn2)C1)=O Cc1c(NC(=O)CC(C)(C)CNC(c2cc(C)n(C)n2)=O)cccc1Cl CC(C)CCC(=O)NCC1CCCC1NC(=O)CCC1CCC(=O)N1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C1(O)CN(C(C2(C)CCC2)=O)C1)C C(CCCCC(=O)N1CCC(C(=O)N(C(COC)CC)C)(OC)C1)=CC N1(C(C(CC)NC(N)=O)=O)CCC(F)(F)C(CNC(c2ccc(C)nn2)=O)C1 CC1(C(=O)NCC2(CO)CCN(C(=O)CC3CC(=O)C3)C2)CCNC(=O)C1 C1(NC(C2C(=C)C2)=O)CC12CCN(C(=O)CC1C=CCCC1)C2 Cc1ccc(F)c(N)c1C(N1CC=C(CCNC(=O)C(C)SC(C)C)CC1)=O C1(C(=O)NC2(CNC(C3=NNC(=O)C3)=O)CCOC2)CCc2nc(O)[nH]c2C1 c1(C(=O)NCC(CCNC(CCCc2ccc(C)s2)=O)O)cnc(O)n1C CCC(F)(F)CC(=O)NCC1CC(OC)CN1C(c1nc(C)ccc1F)=O C1(O)(C(C)Nc2ccnc(C(F)(F)F)c2)CCN(C(=O)Cc2ccccc2)C1 N1(C(CC(C)F)=O)CCCC2CN(C(=O)C(=Cc3ccccc3)F)CCC12 N1(C(=O)CC2CN3CCN2CC3)CCC2CCC(C1)N2C(C1CCCCCS1)=O N1(CC(=O)NCCN(C(c2c(CC)cco2)=O)CC2CC2)CCC(C)(O)C1 C1(CNC(C=CCCC)=O)CCN(C(c2ccc(Cl)c(C(F)F)c2)=O)C12CCC2 C(=O)(C(C)S(N)(=O)=O)NC1C2CN(C(C(C3CCC(=O)N3)C)=O)C1C2 C(c1ccccc1F)=CCC(=O)NC(CNC(c1[nH]cc2c1CCC2)=O)C1CC1 C(C)(CNC(C12CC(C)(C1)C2)=O)(CC(C)C)NC(C(CC)SC)=O c1(C(N2CC(NC(=O)CCC3CC3)CC23CCC3)=O)cnc2cccnc2c1 c1(C(=O)NC2C(C(=O)NC(C#C)C3CCC3)CCCCC2)cc(C)cc(C#N)c1 Cc1cc2c(cc1C(=O)NC(C)C(C)NC(c1cc(C(C)C)nn1C)=O)OCO2 N1(C(C(CNC(C2(C)CC2)=O)O)=O)CCCOC(C)(C)C1 CC12CC1CCN2C(=O)CC1C=CC(NC(C2CCCC2)=O)C1 C(=O)(C1Cc2ccccc21)N1CCCC(CCC)(NC(=O)C(F)CCC)C1 C1(NC(c2c(OC)nn(C)c2)=O)CC2CC1N(C(=O)Cn1ccc(C)cc1=O)C2 N1(C(c2c(C)cc(C3CC3)cc2)=O)CC2(CCCCN2C(=O)C2=CC(C)(C)C2)C1 N1(C(C(C2CC2)SC)=O)CCN(C(c2ccn(C)n2)=O)CC1CC(C)(C)C CN1CCOC(C(N2CC3CC2C3CNC(=O)CC2COC(C)(C)C2)=O)C1 c1(C(N2CCC(NC(C3C(C(N)=O)C3)=O)C2C2CC2)=O)cc(C2CC2)cc(F)c1 CC1(C)CCCN(C(c2cnn(CCO)c2)=O)C1CNC(C1CC2(C1)CC2F)=O CC(C)CCC(F)C(=O)NCC1CC1CC(N1CCC1C(C)(C)O)=O C=CC1(CC(=O)NC2CCCC(NC(C3CCC=CCCC3)=O)C2)CCCCC1 N1(C(CC2(NC(=O)C(F)CC3CCOC3)CC2)=O)CCCC(F)C1 c1(C(=O)NC2CCCC(N(C(CNS(CC)(=O)=O)=O)C)C2)c(C)cc(=O)oc1C C1(C(=O)N(C2CCOC(C)C2)C)(CC)CCN(C(c2c[nH]nc2OC)=O)C1 CCCCC(C(=O)N1CCC(N(C(C2CCCC(CF)C2)=O)CC)C1)C(C)C N1(C(c2nccc(C(N)=O)c2)=O)CCC2(CC1)CC2NC(=O)CCCC1CC1 c1(C(N2CC(O)(CNC(C(C)OCCC=C)=O)C2)=O)cnn2c(C)cc(C)nc12 N1(C(C(CC)(F)F)=O)CCC(CO)C(CN(C(=O)Cn2cccc(C)c2=O)C)C1 C1(NC(C(C)C)=O)CN(C(C2CCc3cncn3C2)=O)C2CCCCC12 C1(Nc2nc(C)nc(N3CCOC4(CC4)C3)c2)CCOC2(CCSC2)C1 Cc1cccn2nc(C(N3CCCCC3CNC(C3CCS(=O)CC3)=O)=O)cc12 C(N=c1[nH]c(Cl)nc2c1SCC2)C1(CNC(C2=CC(C)(CC)C2)=O)CCC1 c1(SCC=C)ccccc1C(N1CC2C(CNC(=O)CC3OCCCO3)C2C1)=O C(=O)(C1=CS(=O)CCC1)NCC1CCC(NC(c2cnc(OC)c(Cl)c2)=O)CC1 c1(C(N(C2CC(NC(C3(F)CC3C)=O)C2)C)=O)cccc(C(F)(F)F)c1 N1(C(=O)Cc2ccc(CO)cc2)CCN(C(c2nc(C3CC3)cs2)=O)C2CC12 c1(C(=O)NCC(C2CCCCC2)NC(C(=Cc2cscn2)C)=O)nc(C)n(C)n1 C1(NC(c2nc3ncccn3n2)=O)CN(c2ncc(Br)c(O)n2)CC2(CCC2)C1 C1(NC(C(C)=CC2CC2)=O)CC(O)CN(C(=O)CCOC2CC2)C1 Cc1nc(CC(=O)NCCC(C)N(C)C(c2ccn(CC(C)C)n2)=O)c(C)s1 CC(C)(C#N)CCCC(=O)NC(CO)C(=O)NCC1(C)CC(F)(F)C1 C1(CNC(C2C(C)CC=CC2)=O)CN(C(=O)CCSC(F)(F)F)CC2(CCC2)O1 C1(CC(=O)OC)CC(NCCC2CCSCC2)CCO1 c1(C(N2C(C)CC(CCNC(c3cc(Cl)c[nH]3)=O)CC2)=O)n[nH]c2c1CCSC2 CC1Cc2cccc(C#N)c2N1C(c1cc(C(F)(F)F)ncc1Br)=O c1(C(=O)NCC(CCOC)NC(=O)CNC(=O)OC)nccc2occc12 C1(N(CCOC)C(c2nccn2C(C)C)=O)CCNCCC1C.CC(F)(F)F CC1(C)COC(CC(=O)NC(CC2CCC2)C(=O)NCC2(C)CCC(=O)N2)C1 N1(CCCN=C(NC2C(OCC)C2)NCC)CCN(S(=O)(=O)N(C)C)CC1 C(CCC)(C(=O)NCCN(C)C(c1cccc(C2CC2(F)F)c1)=O)=CCC CCCC(C(=O)NCC(O)CNC)OCc1cn(CC(=O)O)nn1 CCCCCC(F)C(=O)N(CCCNC(=O)CCC=Cc1ccccc1)CCC CCC(O)C(=O)NCC1CC(F)(CNC(=O)CCc2cn[nH]c2)C1 c1(N2CCC(CCCN(C)C)CC2)nccc(=NC2CC3CCCCN3C2)[nH]1 C(=O)(C1=CCCN(C(=O)C(O)C(C)(C)C)C1)NC(C1(O)CCC1)C C1(C(C(=O)NC(CN(C(COC(CC)CC)=O)C)CC)O)CC(F)(F)C1 C1(C(=O)NCC(C)(C)O)CN(C(C2CCNC(=O)C2)=O)C2(CCC2)C1 C1(NC(C(CC#C)NC(c2cccc(C)c2O)=O)=O)CCc2nn[nH]c2C1 c1(C(=O)NC2CN(C(=O)Cn3cncn3)CCC2O)cnc2ccccc2n1 N1(S(C2C(C)OCC2)(=O)=O)CCC(N)c2cc(Cl)ccc21 C1(C(NOCC#C)=O)C(O)CCN1C(=O)C(C)C=C Cc1ccc2[nH]c(C(=O)NC(C)CN(C)C(c3ccccc3C3CC3)=O)cc2c1 N1(C(Cc2c(C)con2)=O)CCN(C(=O)C(C)(C)C(=O)OC(C)(C)C)CC1CF C1(C(=O)NCC2CCC2NC(=O)C(F)(F)c2nccs2)CCCS1(=O)=O N1(C(C(c2ccc(OC)cc2)C)=O)CCC2(C1)CN(C(c1oc(C)cc1C)=O)C2 C1(C(=O)NCCOCCOCCNC(CC(C)C)=O)CN(C)CC1C(F)(F)F CC(C)C(F)C(=O)NC1CC(C(=O)N(C)OCC(F)(F)F)CC1O n1(C(C)C)ccc(C(N2CC(n3cc(CNC(=O)CC4CCOC4)nn3)C2)=O)c1 C1(NC(CCN(CC)CC)=O)C=CCN(C(=O)C(=Cc2cccs2)C)C1 N1(C(C2CN(C)C2)=O)CCN(CCCNC(C2(C3CCCO3)CCCC2)=O)CC1 C12(C(=O)NC(c3ccc(C)cn3)C)COC(C1)C(NC(C1(C)CCC1)=O)C2 c1(NCC)ncccc1C(=O)NCC=CCNC(c1cncc(C2CC2)c1)=O N1(C(C=C=C(C)C)=O)C2CC1CN(C(c1coc(C(N)=O)c1)=O)C2 N1(C(C=COCC)=O)CCC2CCN(C(c3c(O)ccc(Cl)c3F)=O)CC12 N1(CC(=O)NC2C3CN(C(CC(CC)O)=O)CC32)C(=O)N(C)C2(CCCCC2)C1=O c1(OCC)cccc(CCC(=O)NC2CCN(c3nc(C(=O)O)co3)C2)c1 CCC(C)(C)CCCC(=O)N1CC(C(=O)NCC(C)(O)C(=O)OC)OC(C)C1 c1(C(=O)NC2CN(C(Cc3c(O)ccc(C)c3)=O)C2)c(C)[nH]c2ccccc12 C(N=c1[nH]cnc2c1CCC2)C1NCCCC1.c1(C=O)ccc2[nH]nc(I)c2c1 C12(C(=O)NC(C(C)(C)OC)c3cn(C(C)(C)C(=O)O)nn3)CC(C)(CCO1)C2 C1(C(=O)NC(c2nc(C)[nH]n2)C)CCCCN1C(c1csnn1)=O C(=O)(CCC(C)(F)F)NCCCCN(C)C(C1CC1C(C)(C)C)=O C(=O)(C(C)(CF)c1ccccc1)N1CC(N(C(=O)Cn2ccc(C3CC3)n2)C)C1 C12(CNC(CN(C)Cc3cccc(Cl)c3)=O)CC1CN(C(C1CC=CC1)=O)C2 C1(CN(C(=O)CC2CCCOCC2)C)COCCN1C(=O)CCc1ccn(C)n1 C12(NC(C3CCC(C)C3)=O)CC(C1)N(C(c1ccn(C)n1)=O)C2 c1(C(=O)NC2CCOCC2C(N2CC(F)C(F)C2)=O)ccc([N+](=O)[O-])[nH]1 CC(C(=O)N1CCC(O)C1C(=O)N(C(CCO)C(F)F)C)C(F)F C(=O)(C1=CC2CCCC12)NCc1ccc(CN(C(C(CSC)(C)C)=O)C)cc1 c1(C(c2nnnn2C(C)C)NCC)nccc(N(C)CC2CCC2)n1 N1(C(CCN(CC)CC)=O)CCC(F)(CNC(=O)CC(C)SC)CC1 C1(CNC(c2cc(C3CC3)ccn2)=O)CN(C(=O)CCCn2ccnc2)C2CC12 c1(C(C)(C)NCC(O)Cc2ccccc2Br)ccccc1F N1(C(C2C(CC)CCCC2)=O)CCC2(C1)CN(C(c1c(OC)cccc1C)=O)C2 N1(C(c2c(CNC(c3cnc(O)o3)=O)cc[nH]2)=O)CCOC2(CC2)C1 c1(CNC(C=C(COC)C)=O)csc(C(=O)NCCC2CC2C)c1 CC1CCCCC1n1nc(-c2ccc(N)cc2)nc1-c1cc(Cl)no1 C1(NC(C(CC=CC)C)=O)CCSC12CN(C(c1ccc(CCO)cc1)=O)C2 c1(C(C(=O)NCCCSC)N(C)C(c2ncc(C)[nH]2)C)nn(C)cc1C CC#CCN=c1nc(N(CC(COC)OC)C)c2c(ncn2CC)[nH]1 c1(C(N2C(C)C(NC(c3ncn4c3CCC4)=O)CC2)=O)ccnc2c1ncn2C CCCC(C(=O)NC1CCC(CC(N2CCC(CN(C)C)C2)=O)CC1)NC(N)=O CC(O)C(C(=O)N1CC(CCNC(=O)OC(C)(C)C)C1)NC(=O)C1=COCC1 N1(C(CCCC)=O)CCC2(COC(CNC(c3cccc(CS(C)=O)c3)=O)C2)C1 CC(C)C(C)(CNC(=O)CC1CCC(=O)N1)NC(=O)CC1CSCCO1 C#Cc1ccc(Cl)c(C(=O)NCCC2(CNC(C3CC3(C)CC)=O)CC2)c1 C1(OCCCNC(C(C)=O)=O)CCN(C(=O)CC2OCCC2C)CC1 C1(C(N2CC3(CC(F)C3)C2)=O)CN(C(c2csnc2Cl)=O)C2(CCC2)C1 NC(=O)CCCCC(=O)NC1CC(O)C1CC(=O)NC1(CC2CC2)CC1 c1(C(N2CCC(NC(c3c(C)cco3)=O)CC2C)=O)cnc(C)c(C#N)c1 CC(O)C(C(=O)NCC1CC(CO)CN1C(=O)CN(c1cccnn1)C)N(C)C C=CC(C)C(C)C(=O)N(CCCOCCNC(c1c[nH]ccc1=O)=O)C C(=O)(CC1=CCN(C)CC1)N1CCC(C2(NC(c3ccc(C)c(F)c3)=O)CC2)C1 C1(C(C)(O)CNC(=O)N(c2cnn(-c3nccs3)c2)C2CC2)CN2CCC1CC2 CC(C)CCCC(=O)NCC1(C)CCN(C(c2ccccc2F)=O)C1 C1(N(C(C2CCC2(C)C)=O)CC)CCCN(C(c2ccc(C(C)=O)cc2)=O)CC1 Cc1ccc(C)c(C(=O)NCCNC(=O)CO)n1.C1C(=O)NCCS1 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)NC1CCN(C(CCCOCCC)=O)C1 CC1(C)OCc2c1n[nH]c2C(=O)NC1CCC(NC(C2CCOC2(C)C)=O)CC1 c1(OCC)ccccc1C(N1CC2C(N(C(=O)CCNC(C)=O)C)C2C1)=O N1(C(C2(CC)CC(C)(C)C2)=O)C(C(=O)NCC(CO)OC)C2CC(O)C1C2 C1(C(=O)NCCSCCC=C)COC2(C1)CN(C(C1(C)CCC3CC3C1)=O)C2 O=C(CCCC(F)F)N1CCC(N(C(=O)C(c2ccccc2F)O)CCO)CC1 C1(NC(=O)CC2CCC(O)C2)CC2CC(NC(c3c[nH]nc3[N+](=O)[O-])=O)C2C1 N1(CC)CC(C(=O)NCC2CC3(C2)CN(C(=O)C=C(C)Cl)C3)CCC1=O C12C3CCC(C3)C1C(=O)N2.Cn1ccnc1SCCNC(=O)OC(C)(C)C N1(C(C(C)(C)C)=O)CC(C)CCC1CONC(=O)O.C(=O)(CCCn1ccnn1)NC CCC(F)(F)C(=O)NCC(=O)NCC1(CC)CC(C)(C)C1 C(C1CCCN1C(=O)Cn1ccccc1=O)=CC(=O)NC(CC=C)C CCC(C)C(C(=O)OCC1CC1)Nc1nnccc1C(F)(F)F C(=O)(CCC(C(=O)NCCN(C)C(c1cc(OC)ncn1)=O)N(C)C)OC c1(C(=O)NC2CC(C(C)NC(COCCCC)=O)C2)ccnc(F)c1O c1(NC(=O)NCC2C(OC)(OC)CC2)ccc(CC2CCC2)cc1C Cc1ccc2cc(C(=O)NCC3(C)CCN(C(=O)CC(F)(F)Cl)C3)[nH]c2c1 N1(C(CN(CC)CC)=O)C2CCC1CC(O)(CNC(c1csnn1)=O)C2 N(C(=NCCC1CCCC1)NC1CCC12CCCCC2)CC(N1CCOCC1)=O N1(C(C(C)OC(C)(C)C)=O)CC(CNC(=O)C2=CCCOCC2)OC2(CCC2)C1 N1(S(=O)(=O)C2CC2)CCC2(CCCN2c2ccncn2)C1 C(=O)(C1CCc2nccn21)N1CCC(CCCNC(=O)CC2CCC(=O)N2)CC1 C(=O)(C1CCOc2ccccc21)N1CCC(NC(Cc2c(C)nc[nH]2)=O)C(F)C1 CC(CC(=O)N1CCN(Cc2c[nH]c3cccnc23)C2CC12)CC(C)(C)C c1(CC)ocnc1C(=O)N(C1CCCC1)CCNC(C1CCOC1C(F)(F)F)=O C(=O)(C1CCCc2cncn21)N1CCCC(N(C(Cc2c(C)noc2C)=O)C)C1 C=CCC(C)(C)C(=O)N(C)CC1CN(C(=O)CSc2c(C)n[nH]c2C)CCO1 C(=O)(C1=NOC2(CCOC2)C1)NC1C(C)CCN(C(=O)C(C)(C)CS(N)(=O)=O)C1 CON(CCCO)C(=O)C1(C=C)CCN(C(=O)CC2CC=CCN2C)C1 c1(C(=O)NCCC(C)NC(c2c(C(C)C)nns2)=O)ccc(N)c([N+](=O)[O-])c1 C1(C(C)NC(c2ccco2)=O)CN(C(=O)Cc2nnc(O)s2)CCO1 CCCCCCC(C)(CC)C(=O)N(C)CCNC(=O)CC(c1ccc(F)cc1)C N1(C(C(C)CCO)=O)CCCC(C2CCN(C(=O)CCn3cccn3)C2)C1 Cc1nc(C(N2CCN(C(=O)C(N)=O)CC2)=O)c(C)n1C N(C(=NCCc1ccc(OC)cc1)N1CC(C)S(=O)(=O)C(C)C1)CC(CC)OC C(=O)(CC(C)CC(C)(C)C)N1CCOCC(CNC(CNC(CC)=O)=O)C1 N1(C(CCC=C)=O)CCC2C(CCN2C(c2ccc(NC(C)=O)o2)=O)C1 C(CCC(C)(C)NC(=O)C(C)Cn1cccn1)NC(Cc1c(C)nc[nH]1)=O c1(C(=O)NC2(CO)CN(C(C(CC)C)=O)C2)cccc(Br)c1 C1(NC(CCOCCOC)=O)CN(C(c2cc(C3CC3)cs2)=O)C2CCCC12 C(=O)(CCC(CF)CF)NCCCN(C(C1C(C)(C(F)F)C1)=O)CCO Cc1nn(C)c(C(=O)NCCC2CCCN(C(C3CC3CF)=O)CC2)c1Cl Cc1cncc(C(N2CC(CNC(c3cc(CCO)on3)=O)CC(C)C2)=O)c1C c1(OC)ccc(C)c(C(=O)NCCC(C)(C)NC(=O)C=CS(C)=O)n1 N1(C(C(CC)OC2CCCC2)=O)CC(NC(=O)CO[Si](C)(C)C)CC(F)C1 CCC1=NOC(CC(=O)NCC(C(=O)N(c2cscc2C)CC)OC)C1 C(=O)(C1=CCN(C(=O)C(C)n2ccnc2)CC1)NCCN(C)CC Cc1cc(C(=O)NC2(C3CN(C(=O)C=C4CCC(C)CC4)C3)CC2)ncc1C#N C(C1C(C(=O)NCCCC2(NC(=O)C(C)OCOC)CC2)C1(C)C)=C(C)C C1(NC(C2=CC(C)(CC)C2)=O)CC2CCC1CN(C(=O)C(C)COC)C2 c1(CCNC(=O)NCc2cc(C#N)cc(Br)c2)cccc2cnccc12 c1(C(=O)NC2CC(CNC(=O)C=C3CCCCC3)C2)cc(F)cc(F)c1 N1(CC2C(C)(C)C2C(F)F)CCOC2(CCS(=O)(=NC(=O)C3=CCCS3)CC2)C1 CC(C)CC(C(=O)NCCCCN(C(=O)Cc1csc(=N)[nH]1)C)C(C)C c1(C(CNC(c2cc(OC)ncc2)(C)C)O)ccc(Br)cc1F c1(C(=O)NC(C2CCOC2)CNC(c2cc(OC)no2)=O)cc(C)cc(F)c1N C1(C(N(C(CC)CC)CCC)=O)CCN(Cc2cccc(C#N)n2)CC1(C)C Cc1cnccc1C(C)C(=O)N1CC(NC(=O)CCC2CCCCN2C)C1 c1(C(N(C(CC(=O)NC(CCC=C)C)(C)C)C)=O)cnn2c1OCC2 c1(C)ccccc1Cl.C1(C)(ON(CC=O)OC(C2C(C)C2)=O)CC(C(F)(F)F)C1 C1(C(F)(F)C(=O)NCC2CCC2NC(C2CC2C(F)(F)F)=O)(OC)CCOCC1 CCN=c1[nH]cc(C(=O)NC2CCC(N(C(=O)COC(C)(C)CC)C)C2)s1 C1(C(=O)NC2C(NC(c3c(CN(S(C)(=O)=O)C)ccs3)=O)CC2)CCCNC1=O N1(C(C2(OCC)CCCC2)=O)CC2CCC1CN2C(c1csc(C(C)=O)n1)=O N1(C(Cn2nnc(=N)[nH]2)=O)CC(NC(=O)C=CC2CCC2)CC2(CC2)C1 c1(NC(C2N(C(CC(C)(C)F)=O)CCC2)=O)cc(-c2ccccc2)cnc1O C1(NC(c2ccc(C(C)C)o2)=O)CC(NC(c2cnns2)=O)C12CCC2 N1(C(C2(CC)CCOC2)=O)CCN(C(=O)CC(C2CC2)C2CC2)C(C2CCC2)C1 CC1c2ccccc2OC1CC(N1CCC(NC(=O)C(C)(C)C(F)(F)F)CC1)=O C1(c2cc(OC)c(C)cc2)CCCN(N2CCCC(C)(CO)CC2)C1 N1(C(C2CCN(C(C(CC=C)OC)=O)C2)=O)CCSCCC1C CC(C)CCCCC(=O)N1CCCC(C(=O)NCCc2ncnn2C)C1 C1(COC)CN(C(=O)Cc2ccco2)CCN1C(=O)CC1CCCC(C)(C)O1 c1(COC)ccoc1C(N1CCCC1CCC(=O)NC(c1n[nH]c(C)n1)C)=O C1(C(=O)NCCN(C(c2ncc(C(F)(F)F)cc2Cl)=O)CC)CC(=O)NC1(C)C N1(C(C(C(C)C)O)=O)CCCOC(CNC(=O)CC2(c3ccc(F)cc3)CC2)C1 C1(NC(C(C)(C)NS(C)(=O)=O)=O)CCCCCC1NC(=O)C(C)(C)C1CCCO1 C1(CCC)CN(C(=O)CN2CC=CC2)CC1NC(C1(C)CC=CC1)=O CC1CC(NC(=O)CC2CSC2)CCN1C(C1(C)CCN(C)C1=O)=O N1(C(C(C)SCC(C)C)=O)CC2C(NC(=O)C(CC)Sc3ccccc3)C2C1 c1(C(=O)NC(C(C)C)(C)CNC(C2CS(=O)(=O)C2)=O)ccc2nc(S)oc2c1 c1(C(N2CC(SC)C(NC(=O)Cc3cnn(C(C)C)c3)C2)=O)cc(Cl)cnc1O N12CC3(C(=O)O)CCC3(C1)C2.CN1CCOCC1C(=O)O c1(C(N2CCC(C(C(=O)N(CC(CC)CC)CCC)F)C2)=O)cnccc1C N1(S(CCC)(=O)=O)CCC(NC(=O)NC2CCN(CC(N)=O)CC2)CC1 C1(NC(CN2C(C)CCC2)=O)CC2CC(NC(=O)Cn3cnnc3)C1C2 N1(C(CCN(CC)CC)=O)CCC(CNC(=O)CC2OCCC2(C)C)C1(C)C Cc1ccc2oc(C(=O)NC(C)CC3CN(C(=O)C=C4CCCC4)C3)cc2n1 c1(C(N2CCCCC(N(C(CC)=O)C)C2)=O)nn2c(c1C)CCCC2 C(C)(C)(CCCC(=O)NCCCC1CCCC1O)NC(C(C(CC)C)=O)=O N1(C(Cc2c(C)nc[nH]2)=O)CCC(C)C1CNC(c1cccc(N(C)C)c1)=O N1(C(C=C(C)Cl)=O)CC2CCCN(C(=O)CN(C3CCCC3O)C)C2C1 Cc1cc(F)ncc1C(=O)NCC1CCCN1C(=O)CN(c1ccccc1)C c1(-c2ccc(C(=O)NC)cc2)cc(CN2CCCC(C(N)=O)C2)ccc1N(C)C C1(N(C(C(C2CCN(C(c3cn(CCO)nn3)=O)C2)C)=O)C)CCCC1(C)O C1(NC(C2C(=C)CC2)=O)CC2(CCN(C(c3nc(C)n(C)n3)=O)C2)C1 c1(-c2cc(CN(CCCC3CCOC3)CC)sc2)ccc(OC)cc1OC CC1(C)CC(NC(=O)CC2(O)CCOCC2)CN(C(=O)CC2(CO)CCC2)C1 C(=O)(CC(O)CN(C)C)NCCOCC(=O)N(C1CCCO1)CC#C C12(CNC(CN3CC(CC)C3)=O)CCCC1CCN2C(=O)CC1CCOCC1 C1(C(=O)NC2(CN(C(=O)CCCCCF)C)CC2)CCN(C)S1(=O)=O c1(C(N(C2CCN(C(C3CC3CCC)=O)CC2)CC#C)=O)cccc(F)c1CC C12(C(N3C(COC)CCCC3)=O)CC(C)(CN1C(=O)C(C)OCCN(C)C)C2 N1(C(COCC(=C)C)=O)CCC(C2CC2)C1CNC(=O)C=CCN(C)CC C1(C(N2CC3C(CNC(=O)CC4CCCOC4)C3C2)=O)CCc2ncncc2C1 N1(C(C(CCC)OC)=O)CC(NC(c2ncc(CC)s2)=O)C2CCCCC12 Cc1cc(-c2ccccc2)nc(N2CCOC(C(=O)Nc3cnn(CC)c3)C2)n1 CC(CC1CCC1)C(=O)NC1(C(=O)N(C2CCC2)C2CC2)CCCC1 N1(C(CCNC(CC(C)C)=O)=O)CCC(NC(c2ccc[n+]([O-])c2)=O)CC1C C#CC1(C(=O)Nc2cn(C)nc2OC)CCN(C(=O)CN2CCC(C)CC2)C1 C(=O)(CCC(C)CN(C)C)NCc1cccc(C(=O)NC2C(C(C)C)C2)n1 CCC(CC)(CCNC(c1nnn(C)c1C)=O)NC(=O)C=Cc1nccs1 Cc1noc2nc(C(=O)NC34CC(CNC(C5CSCCS5)=O)(C3)C4)ccc12 N1(C(c2c(C)noc2C)=O)C2CCC1CC(N(C(=O)C(C)P(C)(C)=O)C)C2 N1(C(C2(OC)CCC2)=O)CCC(NC(=O)C=Cc2cncc(C)c2)C2(CCC2)C1 c1(C(N2CC3C(C(=O)NCCN4CCNC4=O)(CC3)C2)=O)cnc2ccoc2c1 N1(C(C=CCCC)=O)CC(CCNC(c2ccc(C(N)=O)nc2)=O)OC(C)C1 C(=O)(C(CNC(c1cccc(F)c1C)=O)CC(C)C)NCc1ccc(C)c(F)c1 Cc1oc(C)c(C(=O)NCC(CC(C)C)NC(=O)C(F)C(F)(F)F)c1Br N1(C(C(=O)NCc2ccc(OC)cc2)C2CC2(Br)Br)CCC(S(N)(=O)=O)C1 CC1OC2(C)CC1(C(N1CC(NC(c3ccc(-c4ccco4)s3)=O)C(F)C1)=O)C2 C1(C(C(=O)N(CCC(C(=O)NC(C)(C)CC)C)CC)O)CC(F)(F)C1 C1(C(=O)NCCCOCCNC(Cn2ccc(C)c2)=O)COCC(C)O1 C(=O)(CC1c2ccccc2C=CN1C(C)=O)NC(CN(CCC)CC)C Cc1cc(OC(F)F)c(C(=O)NCCN(C2CCCCC2)C(C2CC2F)=O)s1 C1(C(=O)NCC(CNC(c2nnn(C)c2C)=O)OC)CC(c2ccncc2)=NO1 C1(N(C)C(C2CCO2)=O)CCCCN(C(=O)CN2CCOCC2=O)C1 c1(C(=O)NC2(CC(=O)OC)CCC2)ccc(Cl)c(Cl)c1N c1(COCC(=O)NCC2(C(=O)NC3CC(N(C)C)C3)CC2)ccnn1C N1(C(c2c(C)cc(CNC(CC(CC)O)=O)o2)=O)CCC2(CCCCO2)C1 CCCCCCCCC(=O)N1Cc2[nH]nc(C(N3CCOC(CCF)C3)=O)c2C1 C#Cc1ccc(C(=O)N(C(C)(C(N2CC3CCCCC23)=O)C2CC2)C)cn1 C1(NC(CC)=O)CN(C(=O)COc2ccc(OC)cc2)CCC1C(F)(F)F CCCC(CCNC(C12CC(CO1)N(C(c1nc(C)oc1C)=O)C2)=O)CCC c1(C(=O)NCC(=CC(=O)NCC2(CC=C)CCCC2)C)cnc(C)[nH]c1=N c1(C(=O)NCC(C)(C)NC(=O)CCCC2CCCO2)ccsc1Cl C1(N(c2ccc3nn[nH]c3n2)CCC)CCc2[nH]c(=N)sc2C1 N1(C(c2ncc(C)nc2)=O)CCC(C(=O)NCC2CCC2C)C(C)C1 C(=O)(C(C)(O)C(C)C)NCC(CCNC(c1cn(CC=C)nn1)=O)(C)C c1(N(CCO)Cc2cc(Cl)nc(Cl)c2)nc(O)c2ccc(Cl)cc2n1 CC1(C#CC(=O)N2CCC(CF)(NC(C3CC3C(F)F)=O)C2)CCCO1 C12(Cn3cc(CCON=C(C(=O)OCCOCC)C)nn3)COC(C1)C(O)C2 C=CC1(CC(=O)NC2CS(=O)(=O)CC2NC(C2CCC3(CC2)CC3)=O)CCOCC1 CCCC(CC)CC(=O)NC(CCNC(c1ccc(N(C)C)cn1)=O)C(C)C CC1(C)c2ccccc2CC1NCCS(=O)(=O)c1ccccc1 CC(C)S(=O)(=O)CC(=O)N1CCC(C(C)NC(c2[nH]ncc2C#N)=O)C1 n1(CCCOC)nnnc1C(C)(CCCl)NCCOC(C)C C1(CC)CCN(C(=O)CCN2CCOCC2)C1C(=O)NCCN1CCCCC1C N1(C(C2(C(C)(C)O)CC2)=O)CCC(NC(c2sccc2Cl)=O)C(CO)CC1 C(=O)(C1CCOc2ccccc21)NCC1(O)CN(C(c2nnc(C)s2)C)C1 C1(C(N(CC(O)CNC(=O)Cc2ccn(C(F)F)n2)C)=O)CCCCN1N=O c1(C(=O)NCC2CCCCN2C(=O)CN2CCC2)ncc2ccnc-2[nH]1 CCC(CN(C)C)CC(=O)NC(c1ccccc1)C(=O)NCC12CC(F)(C1)C2 c1(-c2n(CCSC)ccn2)cc(-c2ccc(CN(C)C)cc2)ccn1 C1(NC(c2nocc2Cl)=O)(CO)CCCN(C(=O)Cc2ccnc(O)c2)C1 C(=O)(C(CC)C(=O)N(C(C)C(=O)NCC1(CCCO)CC1)C1CC1)OCC c1(OC)cnnc(C(=O)NC2(C)CN(C(=O)CNC(c3ccoc3)=O)C2)c1 N1(C(c2cc(C)c(Cl)cc2)=O)C2CCC1CN(C(C1CN3CCCC3CO1)=O)C2 N1(C(c2scc(C)c2C)=O)CCCCC(CNC(=O)C2=CSCCO2)C1 C1(C(N2CC(CC)C(C(=O)NC(C)C(C)(C)C)C2)=O)CC2(CC2)CN1C N1(C(CCC2OCC(C)(C)C2)=O)CC2(CCC(CNC(=O)CCC3CCC3)O2)C1 C1(CCc2cn(CC(CCNC(=O)C=CC3CCCC3)F)nn2)CCS(=O)(=O)C1 C1(N(C2CCOC2)C(C2N(C)CCC2)=O)C2CCC1CNC2 C(=O)(C1=CCN(C(=O)CC2(C)CCOCC2)CC1)NCC1N(C)C(=O)COC1 C1(C(=O)NC(c2ccc(F)c(F)c2)C)CCCN(c2cnccc2C#N)CC1 C1(C(N2CC(CC)N(C(=O)CC3CCC(=O)C3C)CC2)=O)CCc2nn[nH]c2C1 C12(NC(C(C(C)C)NC(C)=O)=O)CCC(C(=O)NCCCC3CCOC3)(CC1)C2 C#CCCCC(=O)NC1CC2(C1)CC2NC(c1c[nH]cc1Br)=O CC1=NOC(CCNC(=O)C#CCNC(=O)CCn2ccnn2)C1 N1(C(C2N(C)CCOC2)=O)CCC(CNC(C2CC3CCC2O3)=O)C(F)(F)CC1 C(C(C(C)(C)C)NC(=O)CCc1ccc(O)nc1)NC(C1OCC(C)C1)=O C1(CNC(C(C)C=Cc2ccccc2)=O)CC(F)(F)CN1C(=O)Cc1cocn1 O=S(=O)(c1ccc(OC)c(Cl)c1Cl)N(CCCO)Cc1nccs1 C1(C(=O)NCC(C(F)(F)F)OC)CC12CCN(C(=O)C1=NOC(C)C1)CC2 C1(NC(C(=O)NCC)=O)CCCCC1NC(c1nncs1)=O C(=O)(C(C)(C)CCNC(C1CC1(F)Cl)=O)N1CC(C)C(F)C1 N1(C(c2ccc(CN(C)C)o2)=O)CCC2(CCN(C(c3cnn[nH]3)=O)C2)C1 C12(NC(c3ccncc3F)=O)CCC(NC(C3(O)CCSCC3)=O)(CC1)C2 c1(CC(=O)NC2C(NC(c3cccc(C)c3)=O)CC2)c(F)cncc1Cl C1(N(C(C(C)CO)=O)C)CCN(C(=O)CCc2ccccc2)CC1 Cc1sc(O)nc1C(=O)N(CC(C)C(=O)N(C)CCn1ccnc1C)C c1(OC)cc(C(=O)NCC(C)(C)CCNC(=O)CC(=O)NCC2CC2)ccc1F N1(C(CNC(CC)=O)=O)CC2CN(C(C3CC34CCCCCC4)=O)CC2C1 c1(OCC)cccc(C(=O)NC2CCCC2CNC(c2cnccn2)=O)c1N N1(C(c2ccc(CC)o2)=O)CCN(C)CC1CNC(c1ncsc1C(C)C)=O Cc1c(CNC(=O)NC2(NC(C)C)CCOCC2)cccc1F C(=O)(CCCCCCN(C)C)N(CC(C)NC(C12COCC(C1)OC2)=O)C C1(C2CN(C(c3nnc(Cl)cc3N)=O)C2)(NC(C(N2CCNC2=O)C)=O)CC1 Cn1cc(C(N)=O)cc1C(=O)NCC1COCC1NC(C1CC1(C)C)=O C1(NC(C(COCC)(C)C)=O)CC2CCC(C1)N2C(C1CC(CC(=O)OC)C1)=O Cc1ccc(C(=O)NC(C)CCNC(C2(C(C)N(C)Cc3ccco3)CC2)=O)s1 c1(CCC(=O)NC(CCNC(C2CCC(CC)C2)=O)(C)C)nnc(S)n1C c1(C(=O)NC2(c3cccc(OC(C)C)c3O)CCOCC2)cc(Cl)cc(F)c1F C1(C2CC2)(CNC(C(C)(C)F)=O)CCN(C(=O)CC2(O)CCCC2)C1 c1(C(=O)NC(C)CNC(=O)Cc2ccoc2)cccc(N2C(=O)CCC2=O)c1 N1(C(N)=O)CCCC1C(=O)NC1(CC(N2CCC(O)C2)=O)CCC1 C1(OC)COCCC1CC(=O)NCC(=C1CN(C(C2CCCO2)=O)C1)F c1(OC(C)C)ccc2[nH]c(C(=O)NNC(=O)c3cncnc3)cc2c1 N1(C(C(CC)OCC)=O)CCN(C(=O)C2=CC(C)(CC)C2)CC12CCC2 C1(C(N2C3C(CNC(C(C)C(C)O)=O)C(C3)C2)=O)CCc2n[nH]cc2C1 c1(C(=O)NCCOCCNC(c2c(CSC)cccn2)=O)cc2ccccc2o1 N1(C(C2CC2C(=O)OC)=O)CCC(C2CC2)C1C(=O)N(C1(C#N)CC1)C1CC1 CC1CC(NC(=O)C(C)(C)c2cnsc2)CCN1C(c1cc(Cl)c(Cl)[nH]1)=O c1(CC(=O)OCC)cc(S(=O)(=O)Nc2ncc(OC)c(C)n2)cn1C C1(C)(OCC)CCN(Cc2nc(CCO)c(C)s2)CC1 Cc1cc(C)c(C)c(C(N2CCN(C(=O)CCCN=[N+]=[N-])CC2)=O)c1C CCC(C)(CCC(C)C)C(=O)NCC1CN(C(=O)CC2CCOCC2)CCCO1 C(=O)(CC(C)c1ccco1)N(CC(C)NC(=O)CC(c1cccs1)NC(N)=O)C c1(C(N2C(C3CCN(C(c4c(CCC)n[nH]c4)=O)C3)CCC2)=O)cc(C)[nH]c1C c1(C(=O)NCC2(NC(c3c(C)nco3)=O)CCCCC2C)cc2cccnc2[nH]1 N1(C(C(C2(O)CCC2)NC(CC2(OC)CCC2)=O)=O)CCC(F)CC1 c1(C(N2CCCC(N(C)C(C3CCC(C)(C)O3)=O)C2)=O)ncn2c1COCC2 Nc1ccnc2c(C(N3CCCC3CNC(c3ccnnc3O)=O)=O)cnn12 C1(CCNC(CSCCC)=O)CCC(NC(=O)CSc2ccccc2)C1 c1(C(=O)NCC(CCNC(CC(CN(C)C)O)=O)O)cnc2n1CCS2 CON(CCCO)C(=O)c1cc(CNC(=O)CCOC2CCC2)no1 C1(NC(c2nc(OCC)oc2)=O)CCN(C(c2ccoc2CC)=O)CC1CO C1(CNC(C(C(C)(C)O)F)=O)CC12CCN(C(=O)C=Cc1cnccn1)CC2 c1(CCN(C(C)C(=O)OC)C(C2(NC(=O)CC3(C#N)CC3)CC2)=O)nnc(S)s1 c1(C(=O)NCC(CC(C)C)NC(c2c(C)n(C)nc2)=O)cc2ccc(O)cc2[nH]1 c1(CC(N2CCC(Cn3cc(C(C)(C)OC)nn3)C2)=O)csc2ccccc12 C(CC(F)F)(C(=O)N1CC(C)C1(C)C)NC(c1n(CC)ccc1)=O c1(C(N2CC(C)(C(=O)NCc3ccccn3)C2)=O)cc(Cl)cnc1F CN1N=C(C(=O)NCC2CCN2C(C2CCC=CO2)=O)CCC1=O c1(C(=O)NCCCOCCNC(C(C)CC2CCC2)=O)cn(C)c(=O)n1C c1(OC)cc(C(N2CC(CNC(=O)C(F)OC)C(O)C2)=O)cc(F)n1 C1(C2CCCC2)(C(=O)NC(CCNC(CN(CC)CC)=O)C)CCNC1=O Cc1coc(C=CC(=O)NC(C)CCCNC(=O)CCC2CCN(C)CC2)n1 C1(NC(C(CCC)NC(=O)COCCN(C)C)=O)CCC(=O)NC1(C)C c1(CN(C(CC2C(C)C2)=O)C)cccc(CNC(=O)COC2CCOCC2)c1 c1(CC(=O)OCC)ncccc1C(N1CC(NC(C2(C)CC2(C)C)=O)C1)=O C(=O)(C1CCCc2nncn21)NC1CN(C(c2c(Cl)cc(C)s2)=O)CC1O C1(Cn2cc(CN3C(c4nc(SCC)on4)CCCC3)nn2)CCCCN1N=O c1(CNC(=NC)NCCc2cccc([N+](=O)[O-])c2)nc(O)c2cc(Cl)ccc2n1 N1(C(c2cnn(C)c2Cl)=O)CCC(C)(C)C(NC(=O)Cc2ccns2)C1 c1(C(C(=O)NCC(C)(C)NC(C2(OC)CC2)=O)N(C)CC)ccccc1 c1(CC)c(C(=O)NCC(CCNC(=O)CN2CCCC2C)OC)cccc1C C12(C(=O)NCCC(C)(C)NC(COCC(=O)NC)=O)CCCN(CC1)S2(=O)=O C#CC1CC2(CC(C(=O)NC3CCCN(C(c4c(N)cc(C)cc4F)=O)C3)C2)C1 CC1CCC(CCNC(=O)CN(C2CCCC2)C(=O)Cc2ccnn2C)CC1 C(c1cccnc1)=CC(=O)NCC1CCC(NC(C2CCC(O)N2)=O)C1 N1(C(=O)OC(CC2N(c3cccc(C(=O)OC)n3)CCC2)=O)CC(C)CC(C)C1 Cc1cccc2c(C(=O)N(C(C)CNC(c3ccc(O)c(N)n3)=O)C)csc12 c1(OC)ccnc(OC)c1C(=O)NC(CNC(=O)Cn1ccc(C)c1)C(C)(C)C C(=O)(C(CC(C)C)N1CCCC1=O)OCC(CC)(C)CC n1(CC(=O)OC)cnc(C)c1C(=O)NC1COCC1NC(C1(O)CCC1)=O CCCCCC(=O)NCC(=O)NC1C=CCN(C(=O)Cc2ccc(C)s2)C1 N1(C(C23CCC(CC)(OC2)C3)=O)CCC2C(CCN2C(=O)Cc2cc[nH]c2)C1 N1(C(C(CCOCC)NC(c2cnc(C)cn2)=O)=O)CC(=O)NC(C)C1 C1(CNC(CSCC#C)=O)CN(C(=O)CC(c2ccccc2C)C)CCC1C C1(C(=O)NCCCOCCN(C(C2CCC(CC)CC2)=O)C)CC12CCOCC2 Cc1ccc(C(=O)NC2CCC(C)N(C(c3ccc(N)cc3)=O)C2)cc1F c1(C(=O)NC(C=C)C2CC2)ccc(C)cc1-n1cc(-c2ccncc2C(=O)O)nn1 CCCC(C(O)C(=O)N1CCC(CC(N)=O)CC1)NC(=O)CC(C)(C)C#N c1(CCC)cc(=NCCC(C)NC(c2c[nH]nc2C2CCCCC2)=O)[nH]c(Cl)n1 C1(C(=O)NC2(C(=O)OC)CC2)(Sc2cc(C)ccc2OC)CCCC(F)(F)C1 n1(CCC)cc(Cl)c(C(=O)NCC(C)CN(C(=O)Cc2cnnn2C)C)n1 c1(C(=O)NC2(CNC(C(CC#C)C)=O)CC2)ccc2cccnc2c1N N1(C(C(CC)OC)=O)CCC2CCCC(C1)N2C(=O)C(F)(F)CC(C)C C(C(C)(C)CC(=O)NC(C)CNC(=O)C(c1cccc(C)c1)F)OC N1(C(C(CC)n2ccnc2)=O)CCCC(NC(=O)CCC(=O)C2CCCCC2)C1 CCCCCOCC(=O)NC1CC1C(=O)NCCOCC(F)F N1(C(c2scc(OC)c2)=O)CCC=CC1C(=O)NCC(c1ccncc1)O C(=O)(C(O)CCCc1ccccc1)NC1CCN(C(C2CCC(=O)NC2)=O)CC1 c1(C(CNC(C(C)=CC2CC2)=O)NC(=O)C(O)c2cnc[nH]2)cc(F)cc(Cl)c1 C1(C)(C(=O)NC2C(CNC(c3c(COC)scc3)=O)C2)CCCNS1(=O)=O C(=O)(C(CC)CC(C)C)N1CCC(CC(C)NC(CC(C=C)(C)C)=O)CC1 c1(C(=O)NCC2(NC(CC3CCC(=O)CC3)=O)CCC2)ncc(F)cc1F c1(C(NNC(NCC)=S)=O)ccc(C(C)(C)C)c([N+](=O)[O-])c1 CC1(C(=O)NCC(C2CCOC2)NC(c2ncsc2Br)=O)CCCC1 c1(C(=O)NCCCCC(C)NC(C(CC#C)C)=O)c[nH]c2c(F)cccc12 N1(C(=O)NCC(COC)OC)CCCCCC1c1ccc(COC(C)=O)o1 N1(C(c2coc(C)n2)C(=O)NCC=C)CCOC2(CC1)CCS(=O)(=O)C2 CC1CC=C(C(=O)NCCCOCC(C)(C)NC(=O)C2=COCCC2)CC1 Cc1nc2n(c1C(=O)NCC1(C)CCOC1C1CC1)CC(C)CC2 n1(CC)ncc(C(N2CC(CCCCNC(=O)CCCn3ccnc3)C2)=O)c1C N1(C(c2cnc(CC)nc2)=O)CCN(C(=O)CNC(C2CCOCC2)=O)C(C)C1 c1(C(N(C2CCC(NC(c3occc3Br)=O)CC2)C)=O)ccc(P(C)(C)=O)cc1 C1(N(C)C(c2cc(Br)ncc2Cl)=O)CCc2ncccc2C1 C1(O)(CNC(=NCC=C)NC(C)COC(F)F)CCc2ccccc2C1 c1(OC)ccc(NC(=O)C(c2cccc(Cl)c2)N(CC(F)Cl)C)c(OC)c1 Cc1nsc(Br)c1C(=O)N(CCCCCNC(c1c[nH]cc1C1CC1)=O)C C1(C(=O)NC(COC)CC(=O)NCC2(O)CCC(C)C2)CC2(CCO1)CC2 Cc1cc2ccccc2nc1C(=O)NC(C)C(C(C)C)NC(=O)Cc1cc[nH]n1 C=CCCCCC(=O)NCC1(CNC(C2CC2C)=O)CCC1 CC1(NC(C2CC2(C)Br)=O)CCN(C(=O)C(F)=CC2CC2)CC1 C1(C)(CNC(C(CC)n2ccnc2)=O)CN(C(=O)CCn2ccnn2)CCO1 N1(C(C2(F)CN(C(C3CCC(CCCC)CC3)=O)C2)=O)CCCCC(C)(F)C1 C(=O)(N=S(C)(=O)c1cnn2c1CN(C(=O)CS(=O)(=O)c1cccs1)CC2)SC c1(CC)cc(C(=O)NCCn2cc(CNC(=O)CSc3cccs3)nn2)c(C)o1 C1(C(N2CCC(C)(CNC(=O)C(C3CC3)C3CC3)C2)=O)CCCC(F)(F)CC1 N1(C(c2c(OC)c(Cl)ccc2)=O)CC2C(NC(=O)CC(C)(C)O)CS(=O)(=O)C2C1 CCCCCC(O)C(C)C(=O)NCCCCCCN(C(=O)C(C1CCC1)OC)C C1(CNC(c2cc(OC)no2)=O)C2CCC1CN(C(C1(C(F)F)CCCC1)=O)C2 C1(NC(=O)NC(C(C)(C)CO)c2ccc(Cl)cc2)COCCC1(F)F N1(C(C(C)C(F)F)=O)CC2CCCC2(NC(=O)Cc2cccc(C(F)F)c2)C1 Cc1nsc(C(=O)NCC2CC(O)CN2C(=O)CCOCCOCCCO)c1N Cc1cc(=NCC2CC3(CC(NC(=O)Cn4ccnc4)C3)C2)[nH]cn1 c1(CNC(C(=O)NC(CSCC)CO)=O)ccc(Nn2cc(C)cn2)cc1 N1(C(C2(C)CS(=O)(=O)C2)=O)CC(CNC(C2CCCNC2=O)=O)C(F)(CO)C1 C1(C(=O)NCC2N(C(c3cc(CC)sn3)=O)CCC2CC)CC2CCCC(C1)C2 c1(C(=O)NC2CN(C(c3ccc(C)nc3C)=O)C(C)C2)ccc(S(N)(=O)=O)nc1 c1(CC(=O)N(C(C)CNC(=O)Cc2ncccc2F)C)cccc2nsnc12 CC1=NC(C(=O)NCCC2CCN2C(=O)OC(C)(C)C)CS1 C=C(Br)CC(C)(C)C(=O)N1CCC(O)(CNC(C2(C)CC2(C)C)=O)CC1 c1(C(=O)NC(CC)(CNC(C2(F)CCOC2)=O)CC)c[nH]c2cc(Cl)ccc12 CC(=O)CCCC(C)C(=O)N1CCSCC1C(=O)NCc1cc(C)ns1 N1(C(c2cc(OC)no2)=O)CC(CNC(=O)COCCF)C2(CC2)C1 C1(C(=O)Nc2cc(C(C)(C)C)no2)CCC(NC(=O)C#CC(=O)O)CC1 CON=C(C(=O)NC1(C)CCN(C(c2nnc(C)cc2O)=O)CC1)c1ccco1 C(=O)(C(NNC(=O)c1ccc(CCF)cc1)c1ccc(F)cc1)OC c1(C(N2C(CNC(C(C)N(C(C)=O)C)=O)CC2)=O)ccccc1C#N c1(C(=O)NC2CC(C)CN(C(=O)COc3ccsn3)C2)cccc2nnn(C)c12 N1(c2ccnc(C#N)n2)CC2CCC(NC(c3nc4ccccc4[nH]3)=O)CC2C1 C(=O)(CC(CC(=O)OC)C(F)F)NCCOCCC.N12C(=O)C(=O)N(C1=O)CC2 c1(C(N2CCCC2Cn2cc(-c3ccncc3)nn2)=O)conc1C(F)(F)F C(C(=O)N(C1CC(O)C1(C)C)C)(C(C)(C)C)NC(C(=O)NC(C)C)=O C1(CC=C)(C(=O)O)CCCN1CCN(C(C)(C)C)CCSc1cc[nH]c1 N1(C(C2C(C)C2)=O)CCOC2(CCN(C(=O)C=Cc3ccc(Cl)s3)C2)C1 C(CCCCC(=O)N1CCN(C(C2CCC(=O)O2)=O)CC1C1CCCC1)OCC C(=O)(C(C(C)CC)SC)N(CC(CC)NC(c1cccc(NC(C)=O)n1)=O)C c1(C(C)NC(C23CC(C(C)(F)F)(C2)C3)=O)ccnc(Cl)c1F N1(C(C2N(C(c3c(OC)csc3)=O)CCC2O)=O)CC(F)(F)C(F)(F)C1 Cc1nc(C2CCCOC2)sc1OCc1cn(CCCC2CCN(C=O)C2)nn1.SC N1(Cc2n(CC)nnc2C)CCCC1C1CCCCN1C(=O)C#CC1CC1 C(=O)(C(O)CCNC(=O)C(c1ccoc1)NC(=O)Cn1cc(C)cn1)OC Cn1cnc2sc(C(=O)NCCOCCNC(=O)CC3CCOCC3(C)C)cc12 C(CC(C(=O)NC1CCCCC1CO)NC(c1cc(OC)ns1)=O)OCC c1(OC)cc(C(=O)NC2(C(=O)NCC3CC3c3ccoc3)CC(O)C2)on1 C1(NC(Cc2c(C)ncs2)=O)CCC2(CCN(C(=O)CCc3ncnn3C)C2)C1 C1(C(=O)NCCC2CC(C(=O)NCC(N3CCOCC3)=O)C2)CCCCNC1=O c1(NC(C23CC(NS(CCOC)(=O)=O)(C2)C3)=O)ccccc1Cn1cccn1 C1(C(=O)NC2CCC(CNC(CC3CC(=O)C3)=O)C2)CC2CCCC(C1)C2 n1(CC)c(C(N2CC(N(C(=O)CSCC(C)C)C)C(F)C2)=O)cc2ccccc12 c1(CN2CCCNC2=O)cccc(C)c1.CC1=NC(C(=O)Nc2nccs2)CS1 C1(CC(=O)NCCCCCNC(=O)C(N2CCOCC2)C2CC2)CSCCS1 CC(C)CC(F)C(=O)N1CCC(O)(CN(C(=O)CCc2cnn(C)c2)C)C1 C=C(C)CC(C(=O)N1CCC(C#N)CC1)NC(=O)C(CC)SC N1(C(CCOCC(C)C)=O)CC2(COC(CNC(=O)C(=O)Nc3ncc[nH]3)C2)C1 C1(NC(C2C(CC)C2)=O)CCOC(CNC(c2c(C)nsc2N)=O)C1 c1(CN2CCC(C(=O)NC3CC(F)(CO)C3)C2)ccc(O)c(C2CCCCC2)c1 c1(C(=O)OC)oc(CNC(=O)CCc2nc(CCC3CCOCC3)no2)cc1C C1(NC(c2c[nH]nc2C)=O)CNC(=O)C12CC2.C1(OCC)CCOC(C(=O)N)C1 c1(CC)nonc1C(=O)NCCCC(=O)N(CC(C1CCC1)OC)C Cc1cn2c(=O)c(C(N3CC(NC(=O)CN4CC(C)(C)C4)C(O)C3)=O)cnc2s1 O=C(C1=CCSC1)NCC1CCN1C(c1ccnc(S)c1)=O.C12CN(C1)C2=O c1(CN(C)C(C2CCCN(c3ncc(I)cn3)C2)=O)ccc(Cl)cc1Cl N1(C(CC=CC=C)=O)CCC(CF)(NC(=O)C2CC2)C1 C(=O)(C1=C(C)CC1)N(C(CC)CNC(=O)CC1CC2CC2C1)C C1(NC(CC2(C=C)CC2)=O)CC(=O)N(C2CN(C(C3CC(C)=NO3)=O)C2)C1 C1(NC(C(C=C)O)=O)COC2C(NC(c3csc(C(C)OC)n3)=O)COC12 C12(NC(CS(C)(=O)=O)=O)CCC(CC1)N(C(c1csc3ccccc13)=O)C2 CC1(C(=O)NCC23CCC(CC2)C3)CCN(C(=O)CC23CCCC2C3)C1 c1(NCC)ccc([N+](=O)[O-])c(C)c1.C12CCCN(C1)C(=O)C1CC(C1)C(=O)NCC2 C1(CCNC(C2C(C(C)C)CCC2)=O)CCN(C(=O)CCN2CCCC2)CC1 c1(C(=O)NC(C2COC(C)(C)O2)CO)cc2n(c1)CCCC2 c1(C(=O)NC(CNC(CCSCCC)=O)CC(C)C)cc(OC)cc(OC)c1Cl S(=O)(=O)(c1cccc(Br)n1)NC1C(C(=O)Nc2nc3c(s2)CCC3)CCCC1 C(=O)(CC(COC)NC(c1nnn(C)c1N)=O)NC(c1n(CC)ccn1)C c1(C(=O)OCC)c(NC(=O)C(COC)CC)cnn1C1CCCC1 c1(NC(=O)NCC2OCC(CC(=O)OCC)C2)ncccc1Br C1(CNC(c2n(CCCSC)nnn2)c2ocnc2C)CCSC1(C)C c1(CN)nc(C)c(C(=O)NC2CN(CCCC3CCCOC3)C2)s1 CC(C)(C)CC(=O)N1CC(O)(CNC(C2(C(N)=O)CC2)=O)C1 CCCCC(C)CCC(=O)NCC(C)(C(C)C)NC(c1ccnn1CCCC)=O C(CCC(C)C(=O)N1CCC(CNC(=O)Cc2ccco2)C1)OC N1(CCC(=O)NCC(CNC(CC2(C=C)CCC2)=O)(C)O)CCN(C(C)C)CC1 C1(C(=O)NC2CN(S(CC)(=O)=O)C(CO)C2)CC12CCN(C(=O)C(C)C)CC2 N(C(=NCCc1ccccn1)NCC1CCOC(C)C1)CCOCC c1(C(=O)NC2C(NC(=O)CC3CC4(CC4)CO3)CCCC2)cc2ncccc2[nH]1 N1(C(C2(C)CC2(F)F)=O)CCN(S(=O)(=O)c2cn[nH]c2)C2(CC2)C1 C1(CC)CCCC1C(N1CC(CCCCNC(c2nocc2C)=O)C1)=O Nc1cc(Cl)nc(Cl)c1C(N1CC2(CCCC2NC(c2ccsc2)=O)C1)=O c1(C(=O)NC2CCC(CC(=O)NCc3c(C)nsc3)C2)cccc2c1CCC2 C(=O)(C1=C(c2cn(C)cn2)N(C2CC2)C(=O)NC1c1c(Br)cnn1C)OCC CC(C)C(C(=O)NCC(C(C)(C)C)NC(=O)Cc1ccns1)C1CCC1 c1(C(N2CC(CC(=O)Nc3cccc(O)c3Cl)OCC2)=O)cc(Cl)ncc1Br C(=O)(C(C)(C)CC(C)(C)C)N(C)CC1N(C(Cc2c(C)occ2)=O)CCC1 c1(C(=O)NC(C2CCN(C(CCCSC)=O)C2)(C)C)[nH]c2c(c1C)CCCC2 CC(C)CCC(C(=O)NCCC(=O)N(C)C1CC1)NC(C1CCSCC1)=O C#CCC(O)C(=O)N1CCC(OCCNC(=O)CC2CC(SC)C2)C1 C(C)(C(=O)NC(CO)C(C)NC(C1(CCN2CCCCC2)CC1)=O)(C(C)C)OC c1(-c2cn(C(CNCC)C(=O)NCC(O)(COC)CO)nn2)cc(=O)cc[nH]1 CC12CCCC1N(C(C1CCCOCC1)=O)CCN(C(C1SCCS1)=O)C2 c1(C(=O)NC2CC(C(C)NC(=O)CC3CCSCC3)C2)cc(CO)n(C)n1 C(=O)(CCN1C(=O)CSc2ccccc21)N(C(C)CN(C)C(c1cnn[nH]1)=O)C c1(C(=O)OC)ccn(CC(=O)NCC2(NC(C3CC=CCC3)=O)CCOC2)n1 c1(NC(N2C(Sc3cccc(C)c3)CCCCC2)=O)cc(Cl)c(Cl)cc1N C1(CC(=O)NCC(CCCC)NC(C2CCC(F)CC2)=O)CN2CCC1CC2 c1(CC(=O)Nc2cccc(CNC(C3C(C)N(C)CC3)=O)c2)cccc(F)c1F C1(C(=O)NC(CCC2(C)CC2)=O)CCSC12CN(c1nc3ccccc3s1)C2 C(=O)(C1=CCCC1(C)C)N(CCC(C(C)C)Nc1cc(-n2ccnc2)ncn1)C c1(C(=O)NCC2CN(C(c3scc(CC)c3)=O)C2)c(C(F)(F)F)ccc(F)c1F O=C(C1CCCn2c(O)nnc21)NCc1cccc2c1OCCCO2 c1(-c2cccc(C(C)=O)n2)cc(O)cc2ccccc12 Cc1cnc2cccc(C(=O)N(CC(C)O)CCNC(=O)CCC3CC3)c2c1 C1(CCNC(C=C(C)Cl)=O)CN(C(=O)C(c2ccccc2)F)CC1C n1(CC)nc(C)c(CC(=O)NC2CCC(NC(=O)C(O)CC(F)F)CC2)c1C C(=O)(CC(C)(C)CCC)NC(CC#C)C(=O)OC c1(C(N2CC(CNC(Cc3nc(C)oc3)=O)C3(C2)CC3)=O)cc2ccccc2[nH]1 CN1C(=O)C(NC(CC(N2CCCCc3ccccc32)=O)=O)c2ccccc21 Cn1cnc(S(N)(=O)=O)c1C(=O)NC1CCN(C(c2cn[nH]c2)=O)C1C1CC1 O=C1CC(CCn2cccn2)NC(=O)N1C1CC1.c1(C)nc(C2CC2)sc1Br N1(C(Cc2cn(CC)nc2)=O)CCc2c(C(=O)NC(c3ccsc3)C)n[nH]c2C1 c1(NCC)cccnc1C(N1CCC(NC(c2c(C3CC3)noc2C)=O)C1)=O CCC(CC)C(C)C(=O)NC(CO)CCCCNC(=O)CCCOC(C)C N1(C(c2ccc(N)cc2Cl)=O)CCC2(CCN(C(C3(N4CCCC4)CC3)=O)C2)C1 C(=O)(C(CC(C)C)n1ccnc1)N(C1CCN(C(CCCCOCC)=O)C1)CC C1(CC(=O)NC(C2CCCCC2)C(C)NC(c2csnn2)=O)CC2(CCC2)CO1 Cc1c(CC(N2CC(N)CC2C(=O)NCC(C)C)=O)cccc1[N+](=O)[O-] n1(CC)nccc1CNC(=O)C(=O)N(C(C)C)Cc1csc(-c2ccccc2)n1 C1(NC(C(CCC#C)O)=O)CCN(C(c2c[nH]nc2CCC)=O)CC1(C)C N1(C(C2N(C)CC(F)C2)=O)CC2=C(C1)CN(C(C1CC3C=CC1C3)=O)C2 Cc1csc(=NCC(=O)N(C(C)CCNC(c2nnn(C)c2C)=O)C)[nH]1 C(C)(CC(C)(C)OC)NC(CN(C(C1C(CC)CCO1)=O)CC1CC1)=O C1(NC(C(Cc2ccoc2)NC(=O)CCOC2CC2)=O)CCCCCC1F CC(C)C(O)(C(=O)NCC1(NC(C2CCCS2)=O)CCOCC1)C(F)(F)F CC(C)C(F)C(=O)NCC1CC(F)CN1C(c1ccc(C(N)=O)cn1)=O C1(F)(CNC(C2CCC(C)O2)=O)CCN(C(c2ncc(Br)cc2F)=O)CC1 Cc1cc(C)c(C(=O)NCC2CCN2C(c2cc(O)nc(N(C)C)n2)=O)c(Cl)n1 c1(C(=O)NCCC2CC(NC(C3CC3F)=O)C2)cc(-c2ccncc2)on1 C#CCCCC(C)C(=O)NCC1(CNC(c2cccc(O)c2Cl)=O)CCCCC1 C1(C(C)C)CN(C(=O)CCCCCF)CCN1C(c1cccc(C(C)(C)C)c1)=O c1(CNC(N2CCOC(c3nccs3)C2)=O)ccc(CO)cc1 Cc1cccc(C(=O)N(CC(C)NC(c2c(C)cnn2C)=O)C)c1[N+](=O)[O-] C(=O)(CCCCc1ccccc1)NCCN(C(=O)C(C)(CO)OC)CC N1(C(=O)OC(C)(C)C)CCCC2(C(=O)NCCc3ccc(F)c(Cl)c3)CC2CC1 Cc1nc(C)c(CNC(=O)C(C)(C)C2CCCN2C(=O)C(C)c2cc[nH]n2)s1 C1(C(=O)NCC2(C#C)CCCC2)C2CCC(C2)C1NC(=O)C(C)N=[N+]=[N-] C(=O)(CC1OCCc2ccsc21)N(C)CC1(O)CN(C(C(CC#C)O)=O)C1 c1(CCC)ccc(C(=O)N(CCCN(C(=O)C(O)CN2CCCC2)C)C)s1 c1(C(=O)NCc2ncc(-c3ccnn3-c3ccccc3)cn2)ncc(Br)cc1O N1(C(CC2CCC(C)(C)C2)=O)CC2COCC2(C(N2CC=CCC2)=O)C1 Cc1cc(S(=O)(=O)NC(c2cc3ccc(F)cc3s2)=O)c(C)o1 Cc1ccnc(C)c1C(N1CC(CNC(=O)CC2CCC(F)(F)CC2)C(O)C1)=O Cc1ccc(Br)c(C)c1C(N1CC2(CC2C(=O)NC(c2cccnc2)C)C1)=O N1(C(Cc2cc(C)[nH]n2)=O)CCN(C(c2ncc(N)cc2C)=O)C(C)C1C N1(C(CCN2CCN(CC)CC2)=O)CCCC(NC(C2(N(C)C)CCC2)=O)CC1 c1(C(=O)NC(CCNC(C2CC3(CC(OC)C3)C2)=O)C)ccc(S(C)(=O)=O)cc1 CC1CCC(C)N(C(C2CCCN(C(C3CC(CC4CC4)C3)=O)CC2)=O)C1 N1(C(C#CC2(C)CC2)=O)CCN(C(c2ccc(O)cc2)=O)CC2CCCCC12 Cc1nc2c(C)cc(C(=O)NCC3CCN3C(C3(C)C=CCC3)=O)cn2n1 C1(NC(c2ccc(OC)o2)=O)(CO)CCCN(C(c2ncccc2OC)=O)C1 c1(OC)ccc(Cl)cc1C(=O)NC1CC1NC(=O)CSC C1(CC(=O)NCC2C(NC(COC)=O)CC2)CCCCC1C(=O)OC(C)(C)C C#Cc1cc(F)c(C(N2CC(NC(=O)C(C)(C)c3cscn3)C(O)C2)=O)cc1F C(=O)(C(C)(C)CC(C)C)N1CC(CCC)C(NC(=O)CC(C)C2CCCO2)C1 c1(C(N(C2CCN(C(C3OCCC3CC)=O)C2)CCC)=O)ccc(F)cc1C c1(C(=O)Nc2cn(C3CN(Cc4n(C)ccc4)C3)nc2)nn(C)c(C2CC2)c1Cl Cc1cccc(Cl)c1OCC(N1CCC(NC(=O)CC2(C)CCC2)C(CO)C1)=O N1(C(CC(CC)OC)=O)CCC(CNC(C2CC(C)(C)C(C)(C)C2)=O)C(F)(F)C1 c1(-c2nc(CC)[nH]n2)ccc(C(=O)N(C)CCNC(C2CC2(C)C)=O)cc1 C(C(C(=O)NCC(O)C1CCC1)NC(=O)C=Cc1ccc[nH]1)OC C12(C(=O)NC3C(=O)NCC3)CC(CN1C(c1ocnc1C1CC1)=O)C2 C(=O)(C(F)CCC(C)(C)C)N1CC(CNC(=O)CCC2(C)CC2)CC(C)C1 N1(C(c2c(CC)noc2C)=O)CCC(N=c2nc(SC)[nH]s2)C(C)C1 C(=O)(C1=CCCC1C)N1CCCC(CCNC(CCc2ccc(C)o2)=O)C1 C1(NC(C2(OC)CC2)=O)CCC(C)(C)CC1CNC(=O)Cn1cnc(C(N)=O)n1 N1(C(C2(OC)CCC2)=O)CC2(C)CN(C(c3ccc(F)c(F)c3N)=O)CC2(C)C1 C1(NC(CCC#C)=O)CCCCC12CCN(C(c1cccc3nn[nH]c13)=O)CC2 C(CC(=O)NCc1cnc(F)cc1C)(CC(C)C)NC(Cc1ccn(CC)n1)=O c1(NC(C(N)=O)=O)ncc(CCNC(=O)C=CCn2cncn2)s1 c1(C(N2CC3CCN(C(C(C)SCC)=O)C3C2)=O)c(C)nn2c(C)cccc12 C1(CNC(CN(S(CC)(=O)=O)C)=O)CCCCN(C(C2(C)COC2)=O)CC1 C(=O)(C(C)(C)c1cnn(C)c1)NCC(=O)N(C1CN(C(=O)Cc2cscn2)C1)C C(CN=c1ccc2cccc(Cl)c2[nH]1)N1C(=O)c2ccccc2CC1 C(=O)(C1=COCCC1)NC1CCC(NC(=O)CCN2C(=O)CNC2=O)CC1 CCC(CC)(CN=c1[nH]c(=NCCc2ncccc2F)[nH]c2c1CSC2)OC C(=O)(C(C)C(O)C(C)C)N1CC(NC(=O)COC2(CCCC)CC2)C1 C1(NC(C2(F)CN(C(CN(C(C)C)C)=O)C2)=O)CC(C)OC1=O c1(C(=O)NCC(CN(C(C(C)C)=O)C)O)cnn2c1CC(C)CC2.C1(C)C(=O)N1 CC1(C(N2CCC(n3ccnn3)C2)=O)CCN(C(=O)Cn2cccnc2=O)C1 c1(C(C)OCC(=O)NC(C2CN(C(C3(CC)CC3)=O)C2)C)nccn1C c1(C(=O)NC2C(NC(C3N(CC)CCCC3)=O)C2)ccc2cc(F)c(F)cc2n1 c1(C(=O)NC(C(C)C)CNC(=O)CCC(C)(C)F)nc2cc(O)ccc2[nH]1 CN1CCC2(CCN2C(=O)C(CN(C)C)NC(C2CC(=O)CC(=O)N2)=O)C1 c1(-c2ccc(C)cc2O)cnc2c(C(=O)N(C)CCN(C)C)c[nH]c2c1 c1(CC)ccccc1C(=O)N(CCNC(=O)C(c1cnn(C)c1)O)C1CC1 CCC(CC)C(C(=O)NC(C(=O)NCC1(N(C)C)CCCC1)c1cccs1)OC c1(NC(C(C)NCCc2conc2Br)=O)ccc2c(c1)CCC2 C(C(C)CC(=O)N1CC(O)(C(C(=O)N2CC(CCC)C2)(C)OC)C1)O.OC c1(OC)ccc(-n2cc(O)c(NC(c3ccnc(CC(C)C)c3)=O)n2)cc1 Cc1nc(NCC2CCCC3(CC3)C2)cc(=NC(C)c2csc(C(F)(F)F)n2)[nH]1 C1(C(C)C)C(NC(=O)CS(=O)(=O)N(C)C)CCN1C(C1CC(F)C(=O)N1)=O N1(CC)CCC(C(=O)NCC(O)C(=O)N2CC(NC(C)=O)C2)C1 C12(NC(=O)NC)CC(CN1C(=O)Cc1ccc(NC(=O)C(F)(F)C(=O)OC)s1)C2 Cc1cccn2c(CC(=O)NCCNC(C3CCN(C(N)=O)CC3)=O)cnc12 n1(CC(=O)NC2CCN(C(CCCC#C)=O)C23CC3)cnc2ccccc12 Cc1cc(NC(C2CCN(C(c3ncc(Cl)cc3Br)=O)C2)=O)ccc1F C(C#Cc1cccnc1)NC(C1(C#C)CCN(C(=O)C(F)CCC)C1)=O c1(CC(=O)N(C)CC2CCN(C(C3CCOC3C)=O)CC2)cc(F)ccc1Cl N1(CC)CCN(CC(=O)NCC2(F)CCN(C(C3CNC(=O)C3)=O)C2)C(=O)C1=O c1(C(C)C)nnc2cc(N(CC(O)CN(C(=O)C(C)C3CCCC3)C)C)ncn12 CC1CN(C(C2CCCC23CNC3)=O)c2cccc(Br)c2O1 Cn1c(=O)oc2ccc(CNC(=O)NCc3noc4c3CCCCC4)cc12 C#Cc1ccccc1C(N1CC2(C1)CN(C(c1cccc(C)c1F)=O)C2)=O Cc1nc(C=CC(=O)NCC=CCNC(C2(c3ccccc3)CC2(Cl)Cl)=O)[nH]c1C C(CCC1CC1)(C(=O)N(C1CCCCC1)C)NC(C1N(CC)CCC1)=O C(=O)(CCCC(C)(C)C(=O)N1CCN(C(C2CCN(C)C(=O)O2)=O)CC1)OC c1(N2CCC(N(C)C(C3(Cl)CC3)=O)C2)ccc(C#N)cn1 c1(C(C(=O)NCc2ncc(-c3ccccc3)o2)O)cccc(Br)c1 C1(C(=O)NCCC(C)O)OCCC1NC(=O)C(C)C1CCCO1 C1(NC(C2C(OCC)COCC2)=O)CCN(C(C2CCC3(CCC3)O2)=O)CC1O c1(C(=O)NCC2CC(NC(c3c(C(C)C)cco3)=O)C2)cnc(S)n1C CC(C)CCCC(=O)N1CCC(O)C1C(=O)NC(CN(C)C)CCO Cc1cn2ccnc(C(=O)NCC(C)(C)NC(c3ccnn3C3CCC3)=O)c2n1 c1(CCC(N2C3CN(C)C(C3)C2)=O)cc(Br)ccc1[N+](=O)[O-].C12CCN1C2=O CCC(CC(=O)NC1CC=CCC1C(=O)NOCCOC(C)C)SC CC1=C(C(=O)N2CC(NC(c3ncc(Cl)cc3Cl)=O)CC(C)C2)CCO1 N1(C(C2CCCN(CCC)C2)=O)CCC(C)(CNC(c2sccc2F)=O)CC1 c1(NC(C(=O)Nc2c(C)n(C(C)C)nc2)=O)ccc(I)c(Cl)c1 Cc1cc(=NC2CC(F)(CNC(C34CCCC(CO3)C4)=O)C2)c(C#N)c[nH]1 CC(CCC(C)(C)C)C(=O)NC1CC1NC(c1ccc(Cl)c([N+](=O)[O-])c1)=O Cc1cccc(C(=O)NCC2(O)CCN(C(C3(O)CC3)=O)C2)c1O C=CC1(C(=O)NC(CC)C(=O)N(C)C)CCN(C(c2coc(CC)n2)=O)C1 C1(CC)CNC(=O)CN1C(=O)CCC(C)NC(=O)CNC(=O)OC CC1(C)CCc2c(C(=O)Nc3ccccc3C(=O)NCC(N)=O)csc2C1 C12(NC(=O)C=CCN3CCCC3)CCCN(C(=O)CC3CCS(=O)(=O)C3)CC1C2 N1(C(c2c(C)cnn2C)=O)CCCN(C(=O)CCc2ccccc2C(C)C)CC1 c1(NC(C(=O)NCC=CCNC(C2CCC(COC)C2)=O)=O)c(F)cccc1F Cc1ccc(Br)c(C(N2CCCCC2C2CCCN(C(=O)CC#N)C2)=O)c1 c1(C(=O)NCC2C(NC(c3cnn(CC)c3Cl)=O)CCCC2)ccnc(O)c1F C1(C(=O)NCCOCCNC(=O)CCC2CC(C)(C)CO2)(CC)CCC(=O)N1 N1(CC2(CC)CCC2)CCC2CC(N(C=O)Cc3ccnn3CCOC)C2C1 c1(CC(=O)NC(CN(C(c2cnoc2C)=O)CC)C)ccc(OC)cn1 c1(C(=O)NCC2(O)CC(NC(C(CC)=CCCC)=O)C2)nnn(C)c1C C(=O)(CCCC#N)N(C1CCCN(C(=O)C(N2CCOCC2)C2CC2)C1)C N1(C(C(CC)=CC)=O)CCC2(CC1)CN(C(C1CCCN(C(=O)OCC)C1)=O)C2 CCCC(C(=O)NC1CC(CNC(=O)CC2CCC(C)(C)C2)C1)OC Cc1cc(C)c(C(=O)NC2CC(C)N(C(c3ccncc3F)=O)C2)[nH]1 c1(C(=O)NC2C(NC(C3C(C(=O)OC)C3)=O)CC2)ccccc1Sc1ccco1 c1(NC2C=CCN(Cc3c(O)ccc(C#N)c3)C2)ncc2ccc(Br)cc2n1 CCC(CNC(c1cn[nH]c1)=O)(CC)NC(c1cnn(CC(F)(F)F)c1)=O c1(C(C)N(C)C(C(C)(C)C)=O)nc(-c2cc(O)n(C)n2)n(CC2CCCO2)n1 c1(C(=O)NCC(N(C(C=CC(CC)C)=O)C)C2CC2)c(C2CC2)nc2sccn12 c1(CC)cc(C(N2CCOCC2CNC(c2cncc(Br)c2)=O)=O)nn1C c1(OC)ncc(C)cc1NC(=O)CCC(C)(C)NC(c1cc(O)cs1)=O C1(NC(C2(F)CN(C(C(C)=CC(C)(C)C)=O)C2)=O)C2CCCCCC12 c1(OCC(C)C)ccc(C(=O)NC2(C)CCN(C(C3CN(C)CCO3)=O)C2)cn1 C1(C(=O)NCCC(C)SC)N(C(c2cc(C)cc(C)c2)=O)CCC1(C)C c1(NC(C2CC(F)(F)CN2Cc2cccc(Cl)c2O)=O)cnnc(O)c1Cl C(=O)(C1=NNC(C(F)(F)F)C1)NCC1(OC)CN(C(CCC(=C)C)=O)C1 CCC(C)C(C)C(=O)NC1C2CC1N(C(c1sc(-c3ccccc3)nc1C)=O)C2 CC1(C)CCC(NC(=O)C(F)C2CC(NC(=O)CCc3cccs3)C2)CC1 CCC(CC(C)C)C(=O)N1CCC(CO)(NC(c2cccc3oncc23)=O)C1 c1(CC)cccc(CC)c1C(=O)NC1CCCCC1CNC(c1ccsc1C)=O N1(C(c2c(C)nn(CCO)c2)=O)CC2CC1CN2C(=O)CCSC(F)(F)F c1(SC)ccc(CC(=O)Nc2ccc(CNC(c3ccc(C)cc3)=O)cc2)cc1 C(CC(=O)N1CC2CC(CO)C(C2)C1)(C(C)CC)NC(C(C=CC)O)=O c1(C(=O)NC(C2CCCN2C(=O)C(C#N)=CC2CC2)C)ccc(C(F)F)cc1 c1(C(C)C)ccc(C(=O)N(CC(C)CNC(=O)CC2CCC(F)(F)C2)C)c(O)n1 C1(C(N2CC(OCCNC(CC(=O)OC)=O)C2)=O)CC12CCOC2 N1(C(c2c(O)ncc(CC)c2)=O)CCC2(CCCN(C(=O)Cc3cn[nH]c3)C2)C1 c1(C(N2CCN(C(C3CC4(CCC4)C3)=O)CC(O)C2)=O)c(F)ccc2c1OCC2 c1(C(=O)NCC2N(C(c3n(C)nnc3)=O)CC2)c(C(F)(F)F)ncn1O C(=O)(C(O)CC(F)(F)F)N1C(C(=O)N(C(C)CC(C)C)C)(COC)C=CC1 C1(NC(c2c(CC)n[nH]c2)=O)CN(C(c2ccc(C(=O)OC)cn2)=O)CC1OC Cn1nc2c(c1C(N1CCN(CC3CCC3)CC1)=O)CN(C(=O)C(Cl)(Cl)Cl)CC2 C1(C)(C(=O)NCCCC2(NC(c3c(C)ccnn3)=O)CC2)CCCC1(F)F C1(NC(CCN(CC)CC)=O)CCN(C2CCc3c(F)cccc32)CC1O C12(CNC(C3CN(C)C3)=O)CCC(C1)N(C(=O)CCC1CCC(=O)C1)C2 C1(CN(C)C(c2cnsn2)=O)CCN(C(C2CC2(c2ccccc2)C)=O)C1 N1(C(C(C)=C2CCCC2)=O)CCCC1C(C)NC(C1CC1(Cl)Cl)=O N1(C(c2c(N)nc(Cl)cc2)=O)CCN(C(=O)C(O)CC2CCOCC2)CC12CC2 N1(C(C(COC)(F)F)=O)CCC(C)(NC(C23CC(F)(C2)C3)=O)CC1 N1(C(C(C)n2cccn2)=O)CCC2CN(C(=O)CC3CC4CCC3CC4)CC12 C1(C(N(C(CC)COC)C)=O)CCN(C(c2cc(=O)cc[nH]2)=O)CC1O c1(N2CC(C)N(CCC(C)(C)C)CC2)nc(N2CCSCC2)c2c(n1)CCCC2 C(=O)(C(C)(C)C(C)(F)F)N1CC(CCNC(C(c2cscn2)N(C)C)=O)C(C)C1 C(=O)(C1=NOC(CNC(=O)Cc2cscn2)C1)NCC(C#C)C(C)C N1(C(=O)Cn2cccnc2=O)CC2CC(NC(C3(Cl)CC3)=O)C2C1 c1(CC)cc(C(=O)NCC#CCNC(=O)CCc2cncc(C)c2)c(C)nn1 c1(C(=O)O)sc(CCC(=O)NC2C=CCN(C(=O)OC(C)(C)C)C2)nc1C.CCCC N1(C(c2ccc(N(C)C)c(F)c2)=O)CC(NC(c2coc(Cl)c2)=O)CC12CCC2 C1(C(N2CCC(N(C(=O)CCSc3ccccc3Cl)C)C2)=O)CCCCC(=O)N1 C1(C)(CNC(c2c(C)cnnc2O)=O)CN(C(=O)C(C)SC(C)C)C(C)(C)C1 Cc1cc(C(=O)N(C)CC2CC(F)CN2C(=O)Cn2nccn2)nc(N(C)C)n1 N1(C(CN(C(C)=O)C)=O)CC(NC(C2(C#N)CCOC2)=O)CC2(CCC2)C1 c1(C(N(CCNC(c2cccnc2Cl)=O)CC2CC2)=O)ccccc1C1CCC1 n1(C(C(=O)NCC(C)(C2CC2)NC(CC2CC(=C)C2)=O)CC)ncc2ccccc12 Cc1cc(C(=O)N(C(C)C(=O)NCC2(CO)CCCO2)C2CC2)cnn1 C(=O)(C(CC(C)C)OC(=O)C(c1nc(Cl)sc1Cl)N(C(C)C(=O)NC)C)NCC CC(C)C(C)C(C)CC(=O)NCCOCCCNC(=O)Cc1ccc(F)c(F)c1 C(=O)(C(C)CN(C)C(C1CCC(=O)C1)=O)NCC(c1ccncc1)C N1(C(C2=C(C)OCCC2)=O)CCCC(C2CC2NC(=O)COC2CCOC2)C1 C1(NC(c2ccn3cncc3c2)=O)CCN(C(=O)Cc2cc[nH]n2)C12CCCC2 N1(C(C=C(C)c2ccco2)=O)CC2(CCCC2NC(C2CC23CC3)=O)C1 C1(CNC(CNC(=O)OC)=O)C2CCC(C2)N1C(=O)Cc1cc(C(C)=O)n[nH]1 CC1CC1C1CC1NC(=O)CCN(C(=O)COC1CC1)CCO C1(CNC(c2ccon2)=O)CC(C(=O)NCC2(O)CC=CC2)=NO1 C(=O)(C(C)(C)CNC(=O)CC(C)CN(C)C)NCc1c(C)n[nH]c1 c1(NC(c2cn(C)nc2OCC(F)F)c2n(C(CC)C)nnn2)cnccc1C C=CCC(C)(CC)C(=O)NCC1CN(C(=O)CNC=O)C(C)(C)C1 c1(C(N2CC(CNC(C(C=C)(C)C)=O)N(C)CC2)=O)ccc(OC)c(OC)c1Cl C(=O)(CC(F)(F)Cl)NCC(CC=C)NC(c1cccn1C)=O C=CC1CCCCN1C(=O)C(O)CCCNC(=O)C1CC1 c1(OC)cc(C(=O)NC2CCN(C(c3cc(F)n[nH]3)=O)CC2O)nc(C)c1 C1(C(C)O)CCCCN1C(c1cc(CNC(c2ccc(C(F)F)o2)=O)cs1)=O C12(NC(=O)CC3COCCO3)CCCC1N(C(c1cc(F)c(Cl)cc1F)=O)CC2 Cc1ccc(C2(NC(=O)CC(C)(C)C3CC3)CCCCC2)cc1.c12ccnn1CC2 c12cccc(c1[N+](=O)[O-])N(C1CCN(C(=O)CN(C)C(C)=O)CC1)C2=O.CC.C(C)=C Cc1cc(NC(=O)NC(c2ccncc2)C)ccc1[N+](=O)[O-] C1(OC(=O)Nc2n(C)nc(C(F)(F)F)n2)CCC(F)(F)CC1.C1(=O)CO1 C#Cc1ccc(C(N2CC3CC(NC(c4nc(C)nn4C)=O)C2C3)=O)c(OC)c1 C1(C(N(CCCCCC)CCNC(C23CC(C)C2C3)=O)=O)CCCC(C)(C)O1 C1(COC)CC(N=c2nc(N(C)CCn3cnnc3)c3cc(F)cc(F)c3[nH]2)C1 c1(C(=O)NCC2CN(C(=O)Cc3cnoc3)CCO2)cc2ncc(Br)cn2n1 C1(C(N2CC(N(C)C)(CCNC(=O)OC(C)(C)C)C2)=O)CCC2CNCCN12 Cc1cc(CNC(C2(C)CN(C(c3cc([N+](=O)[O-])c[nH]3)=O)C2)=O)cc(F)c1 C(CCCCCC(=O)N1CC=CCC1C(=O)OC)NC(c1ccn(CC)c1C)=O C1(C(=O)NC(C2(O)CCN(C(c3c(SC)ccs3)=O)C2)C)CC1C1CCCCC1 CCCCC(CNC(c1ncccc1C(F)F)=O)NC(=O)CCC(N)=O C(CCCC(=O)NC(C)CNC(=O)Cc1ccc(COC)cc1)OCCC=C N1(C(CNC(CC)=O)=O)CC2CN(C(=O)CCC(N)=O)CCC2(CO)C1 C1(CNC(=O)CCC2CCCC2)CCC(C(=O)NCCc2nncs2)CC1 CC1CC(C(N2CCC(CCC(N3CC(C)(C)C3CO)=O)C2)=O)CN1C Cc1cc(OCC(=O)N(CC(C)CNC(c2cc(Cl)c[nH]2)=O)C)cc(C)c1Cl Cc1ccc(C=CCC(N2CC(NC(=O)Cc3c[nH]nc3C)CC(F)C2)=O)cc1 C(=O)(C(CCCC)NC(=O)CCc1cnco1)NC1(CC#C)CCOCC1 C12(C(=O)OC)COC(C(=O)N(CCCCN(C)C(C3CNC(=O)C3)=O)C)(C1)C2 C1(NC(Cc2c(C)scc2)=O)CCN(C(c2ccn(C)c2C2CCC2)=O)CC1C N(C1CCCc2c(O)cccc21)C(=O)N=c1nc(Cl)[nH]s1 CCCC(C(=O)NC1C=CCN(C(c2cnn[nH]2)=O)C1)c1ccccc1 N1(C(CCN(CC)CC)=O)CCC(C)C(NC(c2cc(Cl)no2)=O)C1 C1(C(=O)NC2CC(CNC(C(C)(Cl)Cl)=O)C2)CC(C2CCC2)C1 c1(CNC(C2COCCN2C(=O)CCOc2ccccc2)=O)ccc(F)cc1O C(N=c1[nH]c(N2CCC3CCCC3C2)nc2c1CSC2)c1cnc(SC)s1 c1(C(N2C(C)CCN(C(=O)CC3(C)CC3(F)F)CC2)=O)ccnc2c1nnn2C c1(C(C)C)cc(-c2cc(N)ccc2Cl)cc([N+](=O)[O-])c1 C1(CNC(C=CCOC)=O)CCN(C(=O)CCOCC2CCCO2)CC1C C(CN(C)C)(C(=O)N1CCC(OCC(C)C)C1)NC(CCC)=O C1(C(=O)NCc2c(C)n[nH]c2)CCN(C(C2CCN(C)C2)=O)C12CCC2 c1(OC)cc2c(cc1COC(c1cccc3c1CC(C)(C)O3)=O)OC(C)C2 C12(C(=O)NC3CCC(=O)NC3)CC(CO)(CN1C(=O)C(F)n1ccnc1)C2 C(C)(C(C(=O)NCCC1CCOCC1)C(C)C)NC(C(=O)NC(C)C)=O CCC(C(=O)NCC1C2CN(C(c3cnn(C)c3C)=O)CC12)C(C)(F)F CC1C(C=CC(N2CCC2CNC(=O)CC2(N(C)C)CCCC2)=O)C1(Cl)Cl c1(C(=O)NC2CC(OCC)C2)ccnc(C2(N3CCOCC3)CCC2)n1 C1(C(N(CC(O)CN(C)C(C2CC(F)(CO)C2)=O)C)=O)CCCN(CC(F)F)C1 C1(CC(N2CCC(NC(c3c(SC)nn(C)c3)=O)C2CO)=O)CCCCC(=O)N1 c1(CC(N2CC(CNC(=O)C(F)(F)c3cncs3)C(O)C2)=O)ccc(Cl)cn1 C(C(C)(C)C(C)(C)O)NC(C1CCN(C(CC2(OCC)CC2)=O)C1C1CC1)=O C1(CNC(=O)C=CC2CCOCC2)CN(C(c2snnc2C2CC2)=O)CC12CC2 N1(C(C2(CC#C)CC2)=O)CCC(O)(C2CCN(C(=O)CC(C)(C)C(F)F)CC2)C1 c1(CN(c2ccc(C(C)C)cn2)C(=O)NOCCCF)nc2c(s1)CCCC2 CC(C(F)C(=O)N1CCC(=O)N(CC(F)(F)F)CC1)C(F)(F)F C(C1CCCn2ncc(C(N)=O)c21)NC(=O)Nc1nc(C)n(-c2nc[nH]n2)n1 C(=O)(CC(O)CNC(C1CC(=O)CCO1)=O)N(C1CCC(C)(C)C1)C C1(NC(C2CCN(CC)C2)=O)CN(C(C2(C(C)C)CNC(=O)C2)=O)CC12CC2 c1(CSCC(N2CC(C)(NC(CN3CC(C)(C)C3)=O)C2)=O)ccc(O)cc1 N1(C(c2c(OC)ncc(F)c2)=O)CC(NC(C2(CO)CCC2)=O)CC12CCCC2 C1(NC(C(c2ccc(C#N)cc2)C)=O)CCCC12CCCC2 CC(O)C(C)CNC(c1ccoc1CNC(C1CCN1C(C)(C)C)=O)=O C1(CC)CCC(C)CN1C(=O)CC1CCCC1NC(c1csc(Cl)n1)=O N1(C(c2cccc(C(C)(C)C)c2)=O)CC2CCC(C1)N2C(C1(C)CCOC1)=O c1(C(N(CCCNC(c2ccncc2)=O)CC)=O)cnn2c1S(=O)(=O)NCC2 C(N=c1nc(C2CC2)[nH]s1)C1OCC(CNC(c2cc(-c3cccs3)[nH]n2)=O)C1 CCC(C)CC(=O)NC(C)CN(C(=O)CCN(C1CCCCCC1)C)CC N1(C(CCc2ccc(C)s2)=O)CCC(C)C(NC(=O)CC2CCCNC2=O)C1 C1(C(=O)NCC2(O)CCN(C(c3nnn(C)c3C)=O)C2)(SC)CCC(F)(F)CC1 C(C)(C)(CCCNC(c1ccc(CNC(c2cccnc2)=O)o1)=O)N(C)C N1(c2c(Br)cnc(OC)n2)CCC(C)(C)C(CNC(=O)CSc2nncn2C)C1 C(=O)(C1=COCCO1)NC(CC1CN(C(C2CCCC(C(=O)OCC)C2)=O)C1)C C(=O)(C1CCc2cc(F)ccc21)N1C(CNC(CC2(C#N)CC2)=O)CC(O)C1 CCC1=C(C(=O)NC2CCC(CCNC(c3cnn(C4CC4)c3)=O)C2)SCCO1 CCC(C(=O)c1ccccc1)C(=O)N=c1[nH][nH]cc1-c1ccc(F)cc1F C(C(C)(O)C(=O)N(CCC(=O)NCC1(CO)CC(C)(C)C1)C1CC1)OCC C1(S(C)(=O)=O)(C(=O)NC(C)CCCCNC(C2(Cl)CC2(F)F)=O)CCCC1 C1(=CC(=O)NC(CNC(C2C(C(C)=O)C2(C)C)=O)CO)CCC(C)CC1 c1(N(CC(CNC(C(C(C)C)(C)O)=O)C)C)ccc(S(=O)(=O)N(C)C)cn1 C=CCC(CC(C)C)C(=O)NC1(COC)CCN(C(=O)C(CC)C(C)C)CC1 CN1C(=O)CSC1=CC(=O)NC(c1ccccc1)CNC(=O)Cc1ccn(C)c1 Cc1ccc(C(N2CC3CC(CNC(=O)C=C4CCCC4)C3C2)=O)cc1C N1(C(=O)COc2cccnc2Cl)CC2CN(C(C3(CF)CCC3)=O)CC2C1 c1(NC(C2CC(=C)CN2Cc2c(C)cccc2C)=O)cnc2ccc(Cl)nn12 C1(NC(C(F)=CC)=O)CCN(C(=O)Cc2ccon2)C(C2CC2)C1 N1(C(COC)=O)CCC(C2CCCN(C(c3cc(S(C)(=O)=O)cs3)=O)C2)C1 C1(C(=O)NC2(CF)CCN(C(C34CCC(C)(OC3)C4)=O)C2)CCc2n[nH]cc2C1 c1(OC)ccc(NC(c2cnc(C#N)s2)=O)c(C)c1.N12CC(CC1C)C2=O N1(c2nnc(C)s2)CCC2(COC(CNC(C3CCn4ccnc4C3)=O)C2)C1 C1(C(=O)NCC(C#C)CC)CCN(C(C2CCCCC2O)=O)CCO1 c1(C(=O)NC(CNC(C2C(C(=O)OC)C2)=O)C(C)(C)C)ccnc(F)c1OC c1(C(=O)NC(CCC)CNC(=O)C(F)(F)C2CCC2)cc(=O)c(OC)c[nH]1 C1(C(=O)NC(C(=O)OCC)C)CN(C(=O)C2=NOCC2)CC(C)O1 N1(C(c2n3c(nn2)SC(=C)C3)=O)C2CCC1CN(C(c1nn(C)cc1C)=O)CC2 c1(OCC)ccc(NC(C2CSCN2C(c2ccc(O)cc2)=O)=O)cc1 Cc1c(C#N)c(O)nc(=O)n1NC(=O)C(C(C)(C)C)c1ccco1 c1(C(=O)NCC2CC(NC(=O)CCc3cncnc3)C2)cncc(F)n1 c1(C(=O)NCC2CCN(C(c3cncc(N(C)C)c3)=O)C2)c(N)cc(Cl)cc1F c1(C(=O)NCCCCCCN(C(=O)C=CCn2cncn2)C)cc(O)nc(Cl)c1 c1(N(C)C)ccc(F)c(C(=O)NCC2(C)CCCN(C(c3ncccc3Cl)=O)C2)c1 c1(C(=O)NC(CC)CN(C(C2CC2F)=O)CC)ccc(C(C)(C)C)cn1 c1(OC)cc(C(=O)Nc2cccc(NC(c3cnc(C(C)C)[nH]3)=O)c2)cc(F)n1 c1(C(=O)NC2CCN(C(c3c(CC)cco3)=O)CC2C)cnc2[nH]cncc1-2 c1(C(N2CC(C(=O)NCC3N(CC)CCC3)C(OC)C2)=O)ccc(C)c(CO)c1 c1(OC)ccc(C=NOCC(=O)NC2CC(NC(c3nc(Cl)sc3C)=O)C2)cc1 Cn1cncc(C(=O)NCCCC(N2CCOC3CC23)=O)c1=O c1(CC)sc(C(=O)NCCOCCNC(c2coc(C)c2)=O)cc1C C1(NC(c2cc(CNC(C3C(C(N)=O)COC3)=O)on2)=O)CCC(C#N)CC1 C(=O)(C1CCCc2ccnn21)NCC1CCN(C(C(C)=CC2CC2)=O)C12CCC2 Cc1cc(NC(c2c(Br)n[nH]c2C)=O)ccc1NC(c1ccnn1CCF)=O N1(C(C2(C)CNC(=O)C2)=O)CCc2[nH]nc(CNC(C3CC=CC3)=O)c2C1 CC1(C)NC(=O)CCC1NC(=O)CCOCCNC(=O)COC1CCOC1 N1(C(C(CC)C)=O)CCC(NC(=O)CCCc2ccccn2)C1CC c1(C(=O)NCC2C(CNC(C=CCCC)=O)C2)cnc2snc(C)c2c1 NC(=O)CCCC(=O)NCC(CO)NC(c1cn(C2CCCCC2)nn1)=O c1(C(=O)NC2(COC)CCCOC2)n[nH]c2c(C(=O)O)cccc12 C1(C(C)NC(COCC(C)C)=O)CCN(C(c2cnn(-c3cccnc3)c2)=O)C1 c1(CC)cc(C(=O)NCC(C)(CO)NC(=O)C(O)Cc2ccccn2)c(C)nn1 c1(C(N2CC(N(C(C(CC(C)C)NC(C)=O)=O)C)C2)=O)ccc2ccccc2n1 c1(C(=O)NCCC2CN(C(C3(SC)CC(O)C3)=O)C2)cccc(C#N)c1 CC1(C(=O)NCC(F)CNC(=O)Cn2nnc(C(C)(C)C)n2)CCCCC1(F)F c1(C(=O)NCCCC(C)NC(C2C(C)=C2)=O)ccccc1CS(C)(=O)=O Cc1ccc(F)cc1C(=O)NC1CCC(NS(=O)(=O)c2cccs2)C1.N12CC(C1)O2 C12(NC(CN(C3CCC3)C)=O)CCCC1N(C(C1CC13CC(C)(C)C3)=O)CC2 C(CC(CC)C(=O)N1CC(OC)CC1CC(=O)NCC(C(F)(F)F)OC)=CC CCC(C)C(=O)NC(Cn1cccn1)C(=O)N(C)CCn1cnnc1 O=C1CC(C(=O)NCC2CN(Cc3cccc4cccnc34)C2)C2CCCCC2N1 Cc1ccc2ncc(C(=O)NCCNC(C3COC(C)(C)O3)=O)cc2c1 c1(N2CCC(CN(C)CC)C2)nccc(=NCC2(C)OCCc3sccc32)[nH]1 CC(C)CS(=O)(=O)N1CCC(C)(C(=O)NCc2cccc(CO)c2)C1 C(=O)(C(C)CC(N)=O)NC(C(=O)NCC(C1CC1)SC)Cc1ccccc1Br C(=O)(CCCC(=O)C1=CC=CC=CN1)N1CCCC(C(=O)NC2CCC2CO)C1 N1(C(C=C)=O)CCCC(C(N2CCC(NC(c3cccnc3)=O)CC2)=O)C1 CC(C(=O)N1CCC(C(=O)NCc2cc(O)ncn2)O1)=C1CCCC1 c1(N(C)CC)ccc(C(=O)NCCCCC(C)NC(=O)CN(C)C2CC2)cc1 c1(C(=O)NC(C)C(C)NC(C2(F)CCCCCC2)=O)ccc(S(N)(=O)=O)cc1 c1(C(N2C(CN(C(CC(C)n3cccc3)=O)C)CCC2)=O)cc2sccc2s1 c1(C(N2CCC(C(=O)NC3CCCC3(C)OC)(CC)C2)=O)cc2cc[nH]c2cn1 N1(C(C)(C)CO)CCCN(C(c2cnn(CC(O)Cn3cccn3)c2)=O)CC1 N1CCCC(N(C)CC2(C=O)CC2)C1.c1(CC)cc(C)oc1C(F)(F)F C1(C(F)(F)F)(OC)CCCN(C(=NCC(C)C)NCc2nn(C(C)C)cc2Br)C1 C(=O)(CC(C(F)F)c1cccc(F)c1)NCC1(CCNC(CC(C)OC)=O)CC1 C1(CNC(c2cnc(OC)s2)=O)C(C)CCCN1C(=O)C(O)CC1CCCC1 C1(C(=O)NCCCCCNC(CC2CC(=O)C2)=O)CC12CCOc1ccccc12 N1(C(CCC#CC)=O)CC(N=[N+]=[N-])CC1C(=O)NC1C(C)CCC1C C1(C(=O)NCC(C)(C)NC(=O)CNC(c2ccoc2)=O)CCN(C2CC2)C1=O c1(CC(=O)NC2(C)CCN(c3cc(OC)nc(COC)n3)C2)ccc2nonc2c1 C(=O)(C(C)(F)C(F)(F)F)NC1CN(C(c2ccc(OC)c(Br)n2)=O)C1 C(=O)(C1=CCN(C(c2cccc(CC#N)c2)=O)C1)N(C(CC)COC)C C(=O)(CC(C)C(C)(C)C)NCC1C(NC(CCCCOCC)=O)C1 C1(NC(CN(C)C(N)=O)=O)COCC1CNC(C1CC1c1cncn1C)=O C#Cc1ccc(C(=O)NCC2(O)CCCN(C(=O)COCC(=O)NC)C2)c(F)c1 N1(C(C(C=C)CC)=O)CC(C)CN(C(c2cccc3c2CCO3)=O)CC1C C=CCC(CNC(=O)CC1CC2CC2C1)C(=O)NCCC1(C)CCCC1 c1(C2(CNC(=O)NC3(CF)CC3)CCC2)conc1C(F)(F)F N1(C(C2(OC)CC2)=O)CCCOC(CNC(C2(C)CCNC2=O)=O)C1 Cc1nc2[nH]c(C(N3CCC(NC(c4c[nH]cc4C)=O)CC3)=O)cc2s1 C1(C(N(C(C)C(=O)N(c2ccccc2)C)CC=C)=O)CCCC1NC(C)(C)C C1(CNC(c2cn(C)nc2)=O)CN(C(=O)C(C)(C)F)CCC1CC(C)(C)C N12CCCC(C1)C2=O.N1(C2CCN(Cc3ncsc3Br)C2)CCN(CCF)CC1 N1(c2ncnc3cc(OC)c(Cl)cc32)CCC2(CN(C(=O)CO)CC(C)O2)C1 c1(COC)nc(C(=O)NCC2CC(NC(c3c[nH]nc3C3CCCCC3)=O)C2)n[nH]1 N1(C(C(c2ccccc2)SC)=O)CC2CC1(CNC(C1(C)CCOC1C)=O)C2 N1(C(Cn2ncc(C)c2)=O)CCC(NC(C2NC(=O)C3CC23)=O)CC(C)(C)C1 Cc1cc(C(=O)NCC(C)(C)NC(=O)Cc2cscn2)cnn1 N1(C(C2C(NC(Cn3c(C)ccn3)=O)CCO2)=O)CCC(C2=NOCC2)C1 c1(CCNC(c2nccs2)=O)n[nH]cc1C(=O)NCCC1(CO)CCC1 C1(NC(C(COCC)C)=O)(CC)CCN(C(=O)CC2CCOC2(C)C)CC1 C(=O)(C(C)CC(F)F)N(CCNC(Cn1nc(C)c(Br)c1)=O)CC1CC1 CC1(NC(C2CN3CCC2CC3)=O)CCC(NC(=O)CC2CCCC2O)CC1 C(=O)(C1CCCc2nc(C)[nH]c21)NC1COCCN(C(CCC(=O)OC)=O)C1 O=C(C1CCCc2sccc21)NC(=O)CCNC1CCC2(CCC2)CCC1(C)C c1(N2CC3C(CC)(C3)C2)nc(NCC2CCS(=O)(=O)N2C)nc2ncn(C)c12 c1(C(=O)NC2CN(C(C3C(C)COCC3)=O)C2)c(-n2cnnn2)sc2c1CCC2 C1(NC(c2cc(F)cc(F)c2)=O)CCCCN(C(=O)Cc2csc(Cl)c2)CC1 N1(C(CSc2c(C)cccc2)=O)CCCC2(C1)CN(C(=O)C(O)C(C)C)CCO2 c1(CN=C(NC(C)C)NCC2(CN(C)C)CCCC2)ccc2c(c1)NC(=O)CO2 Cc1ccc(O)c(CNC(=O)CC2(C)CCN2C(c2c(C)cccc2F)=O)n1 N1(C(c2n(C)ncc2C2CC2)=O)CC2(CC(NC(C3(CF)CC(F)(F)C3)=O)C2)C1 N(C)(C[Si](C)(C)C)C(C1(NC(C(=O)NC(C)C)=O)CCSC1)=O C1(CC(=O)NC2CC(O)(CNC(c3csnn3)=O)C2)CCC12CCC2 Cc1coc(C(=O)N(C)CC2CCCCN2C(C2C(C)(C)C2(F)F)=O)c1C C(=O)(C(O)CC(C)(C)C)N(C)CC1CN(C(c2nnc(S)n2C)=O)CC12CC2 c1(OC)cncc(C(=O)N(C(C)CN(C(=O)CCCc2ccccc2Cl)C)C)c1 N1(C(CS(=O)(=O)NC)=O)CC2CCC1C(NC(=O)CCCCC1CC1)C2 N1(C(C2C=C(C)CS2)=O)CCC(C2CCN(C(=O)C(C)(C)n3cnnn3)CC2)C1 C(CCCCCNC(c1csc(CSC)n1)=O)NC(C1(COCC)COC1)=O C1(F)(CNC(C2CCN(C(CC)=O)C2)=O)CCN(C(c2[nH]cnc2C)=O)C1 C1(NC(CC2(OC)CCCC2)=O)CCC(N(C(=O)CNC2CCOC2C)C)CC1 C1(NC(C2CCCC2c2nc(S)n[nH]2)=O)CCCC2(C1)N=N2 CC1(NC(=O)CC2CN3CCN2CC3)CCCN(C(=O)CC2CCC(=O)O2)C1 c1(C(C)NC(CSC(C)=O)=O)ccc(NC(C2CN(C(C)C)C2)=O)cc1 CCCCS(=O)(=O)N1CCCC1C(=O)NC1C=CCN(C(=O)C=CS(C)=O)C1 c1(C(=O)NCC23C(CN(C(C(=O)c4ccco4)=O)C2)C3)ccc([N+](=O)[O-])cc1 c1(OC)cc(C#N)ccc1-c1ccc(COC(c2cc(F)c(C)cc2F)=O)nc1 CCC(C#N)C(=O)N1CCC(CCCNC(=O)CNC(=O)NCC2CC2)CC1 c1(C(N(C2CCN(C(=O)C(C(C)C)SC)C2)CC)=O)cnn2cccc(Cl)c12 CCC(CC)C(F)C(=O)NC12CCC(C(=O)NC3CSC(C)C3)(CC1)C2 C1(CC(=O)NC2C(NC(c3n(C)nnc3)=O)CCCC2)CCc2ccccc2C1 CC(C)C(C(=O)N1CC(O)CCC1C(=O)Nc1cncc(N(C)C)c1)C(C)C c1(CC)cccc2c(C(N3CC(CNC(C4CCCC(C#N)C4)=O)C3)=O)c[nH]c12 C1(NC(C2(S(N)(=O)=O)CC2)=O)CCCC2CN(C(=O)C(Cl)Cl)CC12 C(C1=CCN(CC(=O)Nc2ccccc2Br)CC1)C(C)(C)C c1(N(CCCOC2CCN(C)C2)CCO)ccnc(OCCOCCN)c1 N1(C(C(CC)=CC)=O)CCC(NC(c2cc(F)c(F)cc2Cl)=O)CC(O)C1 N1(Cc2cccc(OC)c2O)CCC2(CCN(C(c3ncnn3C)=O)CC2)CC1 N1(C(c2c(N)cn(C)n2)=O)CC(NC(c2cc(C3CC3)cs2)=O)CC(F)C1 Cc1cc(C(=O)NC2(CF)CCN(C(C3CCC(=O)N(C)C3)=O)C2)ncc1CO CC(CC(N)=O)C(=O)N1CCOCC1C(=O)N(C)Cc1cnnn1C c1(C(N2CC3CC2CN3C(C2CC3(CCCC3)C2)=O)=O)nccc2cccnc12 c1(CC)nocc1C(=O)N(CCC(=O)NC(C)Cc1cnccn1)C C1(C)(CC)CN(C(=O)C(CNC(C2CC2C#N)=O)OC)C1 C1(NC(C2C(C)CN(C(C3CC4CC3CC4O)=O)CC2)=O)CC(C)(C)OC1(C)C C(C)(CO)(C(=O)NCCCN(CCCNC(=O)C(=Cc1ccco1)C)C)OC C1(C(=O)NCCC(C)NC(=O)Cn2nc(C3CC3)cc2C(F)F)CCS(=O)(=O)C1 c1(COC)cc(-c2ccc(NC(c3ccns3)=O)nc2)ccc1F C1(O)(CNC(CSCC=C)=O)CN(C(=O)C(F)(F)C2CCCC2)C1 CCCC(C)(C)C(=O)NCCC1CCCN1C(=O)CSc1ccc(C)cc1 c1(C(N2C(C)(C)CC(NC(C3CCC3CF)=O)C2)=O)cc2ccccn2c1 Cc1cc(Br)c(CC(=O)NC(c2cn(CCCN3CCCC3)nn2)C)s1 C1(C(=O)NCC2CCN(C(C(c3cncnc3)C)=O)C2)CCC2CC1CO2 N1(C(CN(S(CC)(=O)=O)C)=O)CCC(COC)(NC(=O)CCc2cccn2C)C1 CC1CC(CNC(=O)Cn2ncnn2)CN1C(c1ccc(C(F)(F)CF)cc1)=O N1(C(C2(NC(C)=O)CCC2)=O)CC(NC(=O)CCC(F)(F)F)CC(C)(C)C1 CC(c1ccccc1)=CC(N1CCCC1C(=O)NOCCC(F)(F)F)=O CC(C)(CCCCNC(=O)C(O)C1CCCC1)C(=O)NNC(=O)c1n[nH]cc1Cl C(=O)(C(C)CS(C)(=O)=O)NC1C(NC(Cc2c(C)ncs2)=O)CC1 C1(C(=O)NCC(CN(C)C(C2C(C)(C)C2(C)C)=O)(C)C)Cc2ccc(F)cc2O1 C(=O)(C(C)C(C)S(C)(=O)=O)NCCC1=CCN(c2cc(C(C)=O)ncn2)CC1 Cn1ncc(C(=O)NC2CC=CCC2C(N2CCCC2)=O)c1N N1(C(CCC(CC)OC)=O)CCC2C(CCCN2C(c2cc[nH]c(=NC)c2)=O)C1 c1(COc2cn(C)c(C(N3CCn4nccc4C3)=O)c2)ccc(S(C)(=O)=O)cc1 C1(CC(=O)NCC2CCC(C(=O)NC3(C)CC4(CC4)C3)C2)(COC)CCOCC1 N1(C(C(c2ccccc2)OC(C)=O)=O)CCCC(N(C(=O)CS(C)(=O)=O)C)CC1 N(C1COCc2ccccc21)C(C)=O.c12ccc(c(F)c1)c(=O)o2 C(C(C)(C(=O)NC(C1CCCC1)C)NC(c1c[nH]c(C(N)=O)c1)=O)SC C1(C(=O)NCCCOCCCNC(C=C(C)C(F)F)=O)CCOC1C(F)(F)F c1(C(=O)NCC2N(C(C(C)C3CC3)=O)CCC2)cc2n(n1)CC(F)C2 N1(C(C2C(C)(C)CC2)=O)CC(CNC(c2cc(Cl)c(F)cc2O)=O)C2(CCC2)C1 c1(CCC(=O)NCC(C(C)C)NC(C(COC)NC(C)=O)=O)cc(C)nc(C)c1 CC1CN2CCN1C(C(N1CC(CN(C)C(c3ccc(C(C)(C)C)s3)=O)C1)=O)C2 CN1CCC(C(=O)NC2CCC(F)(CNC(c3nnn(C)c3N)=O)C2)CC1 n1(CC)ccc(C(=O)NC(C)CNC(=O)C=C(C)C(C)C)cc1=O c1(C(=O)NCCN(C(CN(C2CC2)CC)=O)C2CC2)ccc(F)cc1C#N N1(C(C2CCCC2)=O)CC2CCN(C(=O)Cc3ccc(Br)cc3Cl)C2C1 CC1(NC(=O)CC2(CO)CCOCC2)CCCN(C(C2(CO)CC2)=O)C1 c1(NC(CNC2CC(C#N)C2)=O)ccc(Cl)cc1 C1(C(=O)NC2CCC(CO)C2)CC2(CCN1C(=O)CCc1cnoc1)CC2 c1(C(=O)NCc2cccc(C(=O)NCCC3CCCC3O)n2)cc(F)cnc1O C#CCCCCC(c1nnnn1CCC)NCc1c(NC)cccc1F C(C(C(=O)NCc1ccccc1)N1CCC2CC12)(C1CCCC1)OCC CN(C)NC(=O)CCC(=O)NC1CC1C1CCN(C(=O)CC2CCCOC2)CC1 C(=O)(N=c1c(C)c[nH]cc1Br)C1C(NC(c2cc(OC)c(I)cc2)=O)C1 N1(C(C)=O)CCC2C(CCCN2C(C2CC(=O)N(CC(F)(F)F)C2)=O)C1 C(CC(C(C)C)NC(c1c[nH]nc1F)=O)N(C(C(CC)OCC)=O)C N1(C(C=C(C)CNC(=O)C(C)c2cccs2)=O)CC(F)CC1C CCC(CC)(CCNC(c1ccn(C2CC2)n1)=O)NC(c1nc(C)sc1C)=O c1(C(=O)NC2CC3CC(NC(C(C4CC4)SC)=O)CC32)cc(C)cc2nc[nH]c12 C=CCCCCCC(=O)N(CCC(C)NC(c1cnn(CC)c1Br)=O)C CCC(F)(F)C(=O)NC1CCC1NC(c1cnn(C(C)C)c1C1CC1)=O C(=O)(C#CC1(C)CC1)NCCC(CNC(C(C(C)C)NC(CC(C)C)=O)=O)(C)C c1(C(=O)NC(CC)CC(=O)N2CCOCC2)cc2occc2[nH]1 C(=O)(C(C)(C)c1cc[nH]n1)NCCC1(CNC(CC2(OC)CC2)=O)CC1 c1(CNC(=O)Nc2cn(C)c(NC(c3ccccc3)O)n2)c(F)ccc(F)c1F C1(CN=C(NC(COCC)C)NC2CN(S(=O)(=O)CC)C2)CCCS(=O)(=O)C1 N1(C(CN(C(C)=O)C)=O)CCCC2CN(C(c3cnc(N)c(O)c3)=O)CC12 C#CCC(C)(CC)C(=O)NCC(C)(C)CC1CN(C(c2ccncc2Cl)=O)C1 C#CCCCC(C)C(=O)NC(C1CCCC1)CNC(=O)Cc1cccs1 C1(CC)CN(C(=O)C=Cc2ccc[nH]2)CCN1C(=O)C(C)SCc1ccccc1 c1(C(N(C2CC=CC2)C)=O)ccc(CNC(C2CCCC(N(C)C)C2)=O)cc1 c1(CNCCCN(CCN(C)C)C(C2CC2c2cscn2)=O)cn(C(C)(C)C)nn1 C1(NC(C=C(CC)CC)=O)CC2(C1)CN(C(C1CCC(O)C1)=O)C2 N1(C(c2c(C)nc(C)[nH]2)=O)CC2CCC1CN2C(c1cc(Cl)c(F)cc1N)=O C1(C(=O)OC)CC(C)CN(C(c2nc(NC(=O)CCCCCl)cn2C)=O)C1 N1(C(c2nc(C(C)C)oc2)=O)CCC(C2CCCN(C(=O)C(O)C3CC3)C2)CC1 c1(C(=O)NCC(CC=C)NC(c2ccnc(CC)c2)=O)scc(C)c1Br c1(CC(=O)N(CC(C)NC(=O)C(C2CC2)N(C)C)CC)csc2nc(C)cn12 N1(C(C(C)(C)OC(C)=O)=O)CC2(CCN(C(=O)COC3CC(F)(F)C3)C2)C1 c1(C(=O)NC(C)C(C)(C)NC(c2cc(C(F)(F)F)cs2)=O)cc([N+](=O)[O-])n[nH]1 C1(C(=O)NCCN(C(Cc2c(C)ocn2)=O)C2CC2)CCCN(C(C)C)C1 c1(C(C)(C)C)no[nH]c1=NC(=O)Cc1ccc(CC(=O)NC(C)(CO)CO)cc1 C=CC1(CC(N2CC(N3CCCC3)C2)=O)CN(C(C2(C(C)=O)CC2)=O)C1 N1(C(c2c(OC)scc2)=O)CC2CCC2(CC(=O)NCC2CC(F)(F)C2)C1 c1(C(N(C)CC2OCCC2(C)C)=O)nc(=NCc2ccccc2)[nH]cc1Cl C(CNC(c1ccc(C(=O)N(C)CC)cc1)=O)(CC(C)C)CCNC(CC=C)=O C=CCC(CC(C)C)C(=O)NC(CNC(c1ccc(F)c(F)c1C)=O)C1CC1 C1(CNC(=O)C(F)n2ccnc2)CC(O)CN1C(=O)CCCc1ccccc1Cl C1(CC(C)NC(C(C)=C2CC2)=O)CC2CCC(C1)N2C(=O)C(C)(C)C(C)C CC1CCCC(C(N2CC(O)(C(F)C(=O)N3CCC3CC(C)(C)C)C2)=O)C1 C1(NC(C(C)(C)F)=O)CCN(C(c2cc(C(F)(F)F)ncn2)=O)C12CCC2 C1(NC(C2CCC(=O)NC2)=O)CC2CC(C1)N(C(=O)Cc1cc[nH]c1)C2 CN=c1[nH]c(C(N2CC(CNC(C3(F)CCOC3)=O)(COC)C2)=O)cs1 CC(CO)(CS(C)(=O)=O)NC(=O)NCCC(O)Cc1cccc(F)c1 C12(COC)CCC(C(=O)NC3CCC(CCNC(c4csnc4Cl)=O)C3)(CO1)C2 C=CCC(CC)C(=O)N(C1CCN(C(=O)CCOCC(F)(F)C(F)F)C1)C CC1CCCC(NC(=O)CN2CCN(C(=O)CCCn3cccn3)CC2)CC1 C#Cc1ccc(C(=O)NC2CCC(NC(c3sccc3CC#N)=O)C2)c(OC)c1 C1(C)(C(=O)NC2CCN(c3c(C)nccn3)C2)C2Cc3ccccc3C12 N1(C(C2C(C=C)C2)=O)CCN(C(=O)C=C2CCCCC2)C(CC(F)(F)F)C1 C1(NC(=O)Nc2ncc[nH]2)CCOC1.C12(CC1)C(=O)N(C)C2 C1(NC(C(C)NC(CC)=O)=O)CCC(N(C)C(c2cc(C(C)=O)on2)=O)CC1 C1(CNC(=O)COc2ccc(CO)cc2)CCN(C(c2cscn2)=O)CC1(F)F N1(C(C2CCCN(C(C(=Cc3ccccc3)C)=O)CC2)=O)CCC(C(N)=S)CC1 C1(C(=O)N(C2(C(=O)NC3CC3)CCC2)C2CC2)CCOC1=O C1(NC(c2ccncc2F)=O)CCC2CC1CN2C(c1cccc2cncn12)=O C12(NC(CCCC=C)=O)CCC(C(=O)N(C3CCC(C)CC3)C)(CC1)C2 N1(C(c2cc(C(C)C)on2)=O)CCCCCC(NC(C2(F)CCS(=O)(=O)C2)=O)C1 CCC(C)(C(=O)N1CC(NC(=O)OC(C)(C)C)C(c2ccccc2)C1)OC CCCCCCCC(=O)NCCCCCN(C)C(c1csc(C)c1C)=O c1(C(N2CC(NC(CC=CC=C)=O)C(F)CC2)=O)cc(Br)cc2c1OCC2 C1(CNC(C(C)(C)C2CCCO2)=O)CCCCCN1C(c1cn2c(n1)SCC2)=O c1(C(N(CC(CC)NC(=O)C(N2CCNC2=O)C)CC)=O)cn2cccnc2n1 N1(C(c2c(CC)scc2)=O)CCC(CNC(=O)C=CSCc2ccco2)C(C)C1 N1(C(CSCCOC)=O)CCC(C(C)C(=O)N(C)C(C2CCCC2)C)CC1 C12(CNC(c3ncc(CC)s3)=O)CCCCC1N(C(=O)CC(F)(F)C(F)F)CC2 C1(NC(c2cc[nH]n2)=O)(CNC(C2CC(=C3CC3)C2)=O)CC2CCC1C2 C1(N(C)C(C2CSCCS2)=O)CC2CC1N(C(c1cc(C(F)F)ccn1)=O)C2 c1(C(N(CC(C)(C)NC(C(C2CCC(=O)N2)C)=O)C)=O)cc2ccccc2s1 c1(C(C)C(=O)N2CC(CCNC(C34COCC(C3)C4)=O)C2)c(Cl)cccc1Cl C1(NC(c2ccnnc2)=O)CN(C(C2(F)CC23CCCCC3)=O)CC2(CCC2)C1 Cc1c(C)c(C)c(C(=O)OC(c2nc3ccc(Cl)cc3[nH]2)C)c(C)c1C c1(C(N2C(CNC(CC(C)C3CCCCC3)=O)CC(F)C2)=O)ccnc(O)c1F Cn1nccc(C(N2CC(O)(CNC(C3CCCCS3(=O)=O)=O)C2)=O)c1=O C1(CCNC(CS(CC)=O)=O)CCCN(C(c2ccc(F)nc2)=O)CC1 C(=O)(C(=O)CCC(C)(C)C)N1CC(C(=O)OC)(OC)C1.c1(CN)cn(C)nc1OC N1(C(c2ccc(OC)cc2)=O)CCCCCC(NC(c2ncoc2C)=O)C1 C1(NC(C2(COC)CC=CC2)=O)C2CC1N(C(c1ccc(OC)c(Cl)c1)=O)C2C c1(C(=O)NC2CCCC(NC(CCCCC)=O)C2)c(C)ccc(C)c1C(=O)OC c1(C(=O)NC(CCCNC(Cc2cn(CC)nn2)=O)C)cc(F)c(C)cc1N N1(C(CSCCC)=O)CCC(NC(=O)C=Cc2ccc(Cl)cc2)C12CC2 C1(NC(C(CC)NC(C)=O)=O)C2CCCN(C(=O)CCc3cnc(C)o3)C2C1(C)C C1(CC(=O)NCc2cc(C(=O)NC(c3cccnc3)CC)n[nH]2)CC(O)C1(C)C c1(C(=O)NCC2(F)CC(CNC(C=C(C)C(F)F)=O)C2)cnc2nccn2c1 c1(C(=O)NCC2(C)CCC(NC(=O)CCC(F)(F)F)C2)ccc2c(c1)CCO2 Cc1ccccc1CC(=O)NC(C)(C)CNC(C1CCC(=O)C1)=O N1(C(C(COC(C)=O)C)=O)C2CCC1CN(C(=O)C(O)c1ccco1)CC2 c1(C(N2CCC(C)(CNC(CSCCC)=O)C2)=O)ccc(S(C)(=O)=O)[nH]1 N1(C(CC2(N(C)C)CC2)=O)CCCC(CC(=O)NC2(C)CS(=O)(=O)C2)C1 C1(C(=O)OC)CN(C(=O)C(=O)N(C)C)C(C)(C)C1 C1(CNC(c2ccccn2)=O)CC2COCC2N1C(=O)COC1CC1(F)F c1(C(=O)NC2CCC(CNC(C3(OCC)CCC3)=O)C2)cc(F)cc(F)c1N n1(CC(=O)N(C2CCN(C(c3n[nH]cc3C(C)C)=O)C2)CC)nc(C)n(C)c1=O CC(C)(C(=O)NC1C=CCN(C(c2ccc(S(C)(=O)=O)[nH]2)=O)C1)S(=O)(=O)C1CC1 c1(C(N2CC(C(=O)NC(C3CC4(CCC4)C3)C)OCC2)=O)cc2cnccc2[nH]1 N1(C(C2C(CC)C2)=O)Cc2ccccc2C(NC(c2ccoc2Cl)=O)C1 c1(N(C(=O)NC2CCCN(C(C)C)C2)C)nc2c(s1)CN(NC(N)=O)CC2 Cc1cccc(OCCC(=O)NC(C)CC(C)NC(c2cc(F)c[nH]2)=O)c1C c1(NC(C2C(NC(C3CCC(O)C3)=O)CC2)=O)ccc2cccnc2c1 c1(C(=O)NCC(CNC(=O)C(CC(N)=O)NC(C)=O)OC)cnc(O)c(C)c1 c1(NC(C2N(Cc3ccc(C)c(C)c3)CCSC2)=O)cc2c[nH]nc2cc1Br N1(C(C2COCCO2)=O)CCCC1C1CCN(C(c2csc(CO)n2)=O)C1 Cn1cc(C=CC(=O)NCCCNC(C2(C)CCC(=O)C2)=O)c(=O)n(C)c1=O N1(C(Cc2c(C)non2)=O)CC2(C)CN(C(c3cc(O)ccc3Cl)=O)CC2(C)C1 CC1(C)C(C(=O)NC2CCN(C(=O)C(=O)OCCSCC(F)F)C2)C1C#N C1(CNC2CCCC(C=C)C2)CCCc2ccccc2C1 C1(CC(=O)N(C(C=C)C2CC2)C)CCCN1C(=O)C(C)CC c1(OC)nc(OC)nc(N2CCCC(C(C)NC(=O)C(F)(F)C3CC3)C2)n1 N1CCC2(CC(c3ccccc3)C2)C1.C1(C2(C)CCCN2C(c2ccccc2)=O)C2CCCCCC12 N1(C(C(N)Cc2cccs2)=O)CC(F)(F)CC1C(N1CCOCC1)=O N1(C(C)C)N=C(C(=O)NCCN(C)C(C2OC3CCC2CC3)=O)CCC1=O N1(C(C2CCN(CC)C2)=O)CC2CCN(C(c3cscn3)=O)CC(C2)C1 C(C(N=[N+]=[N-])C(=O)N(C)CC1CCN(C(c2ncc(C(N)=O)cc2Cl)=O)C1)OCC c1(CC)oc(C)cc1C(=O)NCC1(NC(c2nn(C(F)F)cc2Cl)=O)CCCC1 Cc1nc2c(o1)CCCC2CC(=O)N1CCC(CNC(c2ccc(C#N)o2)=O)C1 C1(C(=O)NCc2cccc(CNC(c3cc(Cl)no3)=O)c2)CCC2(CCCC2)C1 c1(OC)ccc(CNC(C2CN(Cc3c(O)cccc3Cl)C2)=O)c(C)c1OC c1(CC)ccc2cc(C(=O)NCCNC(=O)CSCC3CCCO3)ccc2c1 C1(NC(Cc2c(C)n[nH]c2)=O)CC2CCC1C(NC(=O)Cc1cccnc1O)C2 Cc1nc(O)nc(C)c1CC(=O)NC1CCCC(NC(c2ccon2)=O)CC1 C1(C(=O)NCc2cncc(C#N)c2)C2CC(O)C(C2)N1C(=O)Cn1[nH]cnc1=N CC(O)C(C(=O)N1CCC(CCNC(=O)CCc2ccc(Cl)s2)C1)N(C)C C1(CC)C(NC(=O)C(F)=C(C)C)CCN1C(C1C2CN(C)CC12)=O N1(C(C(C2CCC2)OC)=O)C2CCCC1CN(C(=O)COC1CCCC1)CC2 Cc1cc(C(=O)NCc2cccc(NC(=O)CC(C)C(F)F)c2)c2c(c1)CCO2 C1(NC(COCCOC)=O)CC2CC1CN(C(=O)CCCn1ccnn1)C2 c1(N(C(C)C)C)ccccc1CNC(c1nnnn1C1CC1)c1cc[nH]n1 Cc1cnccc1CNC(C1(NC(=O)C=Cc2ccoc2)CC1)=O c1(C(=O)NC2CC(O)(CNC(c3c(C(C)C)cco3)=O)C2)cc(F)cc(N)c1F c1(C(N2C(C)CC(NC(=O)C(C)(C)CF)C2)=O)ccc2nncn2c1 N1(C(c2c(C)n[nH]c2)=O)CC2C(CNC(c3cc(N)ccn3)=O)C2C1 c1(C(=O)NC2C(NC(c3nc(N(C)C)oc3)=O)COC2)ccc([N+](=O)[O-])c(Cl)c1 C1(C#N)(C(=O)NC(C2CN(C(C(CC)n3cncn3)=O)C2)C)CCOCC1 c1(C(=O)NC(COC)C(=O)NCCCC(=O)OCC2CC2)ccc(C)cc1 c1(C(N2CC3CC(CNC(C4(CC)CC4)=O)C3C2)=O)c(O)nnc2c1COCC2 C=CC(C)(CC)C(=O)NC1C2CCC(C2)C1C(=O)NCCc1cccs1 N1(C(C2C(COC)C2)=O)CC2CCC(C1)N2C(=O)Cc1cccc(Cl)c1 CN1CCC(C(=O)NC(CNC(=O)CN2CC(=O)NC2=O)C2CC2)C1=O C(=O)(C(C)(COC)CC)NC1CCC(CCC(N2C(CC)(CC)CC2)=O)C1 N1(C(CCC)=O)CC(NC(c2cc(-c3ccns3)on2)=O)C(C2CC2)C1 C1(C2CCN(C(c3cnc4c(c3)NCC(=O)N4)=O)CC2)(C(=O)OC)CCC1 C(=O)(CC1=CCCC1)OC.C12CC(n3cc(CC(C)O)nn3)CN1C2=O c1(C(=O)NC(C2CCN(C(c3ccncc3F)=O)CC2)C)ccn(C)c(=O)c1 N1(C(C)=O)CCOCC(C(=O)NCCC(C)n2cccn2)C1 N1(C(C2N(C(C)=O)CCC2)=O)CCCCC1CCC(=O)NCC(F)(F)Cl C(c1ccc(C)cc1)=CC(=O)NCC(CN(C(C(CCC)N(C)C)=O)C)C N#CC1CCC(NC(C2CN(C(C3(CNC(N)=O)CC3)=O)C2)=O)CC1 N1(C(C2(CC#C)CC=CCC2)=O)CC2CCC1C(CN=c1[nH]ccnc1F)C2 C1(C(N2C(C(=O)OC)CCC2)=O)CN(c2cc(C)[nH]c(=N)n2)CC(C)(C)O1 c1(C(N(CCNC(C2CCC2C2CCCO2)=O)CC)=O)ccc(C)c(C)c1 C12(NC(CCc3c(C)ncnc3O)=O)CCCC1N(C(=O)CCC(C)(F)F)CC2 Cc1nc2ccc(C(=O)NC(CNC(=O)C(C)S(C)(=O)=O)CO)cc2o1 Nc1cccc(F)c1C(=O)NC(CNC(=O)CC12COCC(C1)C2)CO C(=O)(C1CCCc2n[nH]cc21)N1CC(N(C(=O)C=Cc2ccc([N+](=O)[O-])s2)C)C1 c1(C(=O)NCC2(F)CN(C(c3ccc(NC)cn3)=O)C2)coc2c1C(O)CCC2 N1(C(CC(C=C)C)=O)CCCCC(NC(=O)Cc2cc(Cl)cs2)CC1 c1(OC)cc(N2CC(N3CCN(Cc4cc(C#N)ccn4)CC3)C2)c(OC)cn1 C1(OC)(CNC(c2cnn(-c3ccccc3)n2)=O)CN(C(C2(C)CCOC2)=O)C1 C(=O)(CCCCC(F)(F)F)NCC12CN(C(C(C)=C3CCCC3)=O)C(C1)CCO2 c1(C(N2CCCC(C)(C(=O)NCCCC=CCC)C2)=O)ccc(Cl)c(Cl)c1OC Cc1ccc(C(=O)NCC2CC(C)N(C(c3ccc(C(N)=O)o3)=O)C2)cc1C#N Cc1cc(C(=O)NC(C)CNC(c2ncc(Cl)nc2Cl)=O)c(O)nc1C N1(C(c2nccc(CC)c2)=O)CCCC(CC)(NC(=O)C2=NOCC2)C1 C(c1ccc(C)nc1)=CC(=O)NC(CNC(c1cncc(COC)c1)=O)(C)C N1(c2nccc(OCCC)n2)CCC2C(CCCN2C(C2COCCO2)=O)C1 C1(C(N(C2CCN(C(C3(CF)CCC3)=O)C2)CCC)=O)CC=CCC1 N1(C(c2c(CNC(=O)CNc3ncccn3)c[nH]n2)=O)CC2(CCCC2)C1 S(=O)(=O)(c1ccc(=NCc2cc(Cl)cc(Cl)c2F)[nH]c1)N1CC(C)SC1 N1(C(Cn2ccc(C)cc2=O)=O)CCCN(C(C2C=CCCC2)=O)C(C)C1 c1(CC)oc2ccccc2c1C(=O)NC(C1CCN(C(=O)Cc2ccsn2)C1)C CC1C=C(C(=O)NCC2CN(C(=O)C(c3c(F)cccc3F)N(C)C)C2)CC1 C(=O)(C1=COCCC1)N1CCCC(C(N2C(C)(C(C)C)CC2)=O)C1 C(CC(C)(C)C(=O)NCC1CC(F)(F)CN1C(=O)C(N1CCSCC1)C)SC NC(CCCCCC1OCCO1)C(=O)N1CCC1C1CCC1 N1(C(C2CCCCC23CCC3)=O)CC2OCCN(C(=O)CC3CC4(CC4)C3)C2C1 c1(NC(C(=O)NCC(CC)C)=O)cc(C)c(O)c(C)c1C C(=O)(CC(O)CNC(C1(CC)CCCC1)=O)Nc1cn(CCC#C)nc1 c1(CCC)cccc(C(c2ccc(Br)cc2)N(C(C)C(=O)OC)CCC(C)C)c1 c1(C(=O)NC2(C)CCN(C(Cc3nc(CC)sc3)=O)C2)nc(C)n(C)c1C CC1CC(CO)N1C(=O)CN(C(=O)CCc1nncn1C)C1CC1 C1(NC(CC2(COC)CC2)=O)CCC(CNC(C2(C(=O)NC)CCC2)=O)C1 CCC(C)(CO)C(=O)N1CCN(C2CN(C(=O)Cc3cnn(C4CC4)c3)C2)CC1 c1(NC(=O)Nc2c(C)nc(F)cc2)ccc(S(=O)(=O)NC(c2nc[nH]n2)C)cc1 C(C1CCCN1C(=O)CCc1ccncc1)=CC(=O)NC1C(C)(C)CC1 N1(C(CCCSC)=O)CC(CNC(c2cccnc2C2CC2)=O)C(C(F)(F)F)C1 CC(C)(C)CC(O)CC(=O)N1CC(O)(CCNC(c2cn[nH]c2)=O)C1 Cc1cc(C(N2CC(C(=O)NC3CCNC(=O)CC3)CC2(C)C)=O)cc(F)c1 c1(CC)cccc(-c2cn(CC(F)(F)CNC(=O)CC#N)nn2)c1 CC1(C)CC(C(=O)NCC2C=CCN2C(=O)CNC(c2ccccc2)=O)CCO1 N1(C(CC(=O)NCC)=O)CC2(CC(NC(=O)C(c3ccc(C(F)F)cc3)F)C2)C1 Cc1cc(C(F)(F)F)c2cc(C(N3CC(C)(NC(c4cncs4)=O)C3)=O)oc2n1 c1(C(=O)OC)ccc(CCN(C2CCCC2C(C)C)C)cc1OC(F)F c1(C(=O)OCC)nc(=NCCSC(C)C)cc(C)[nH]1 N1(C(c2n(CC)ncc2C)=O)CC2CC(C1)N2C(=O)CCc1nc(C)no1 c1(CC(=O)NC2CCC(CCNC(C(C)(Cl)Cl)=O)C2)cccnc1Cl C#CCCCCC(=O)N(CCCCN(C)C(C1CC(=O)N(C(C)C)C1)=O)C C1(C(N(CCC(N)=O)C)=O)CC2C=CC1N(C(=O)CC1(N(C)C)CCC1)C2 O=C(N1N=C(c2ccco2)CC1c1ccc(CO)cc1)N1CC(O)C(C2CC2)C1 CCCC(C)(C)CNC(=O)C(C)(CO)NC(=O)CCc1cncnc1 O=S(=O)(c1ccc2c(c1)OCCO2)NC1C2CN(Cc3ncc(Br)cc3Br)CC12 N1(C(CCCOC(C)C)=O)CC2(C1)CN(C(c1c(N)cc(Cl)cc1F)=O)CCO2 CC(CC(=O)N(CCCCCCNC(c1ccnn1CC(F)(F)F)=O)C)C(F)F N1(C(C(C)C)=O)CC2CN(C(c3ccccc3CC#N)=O)CC2C1 N1(C(CNc2cccc(OC)c2)=O)CCC2CN(C(=O)CC3(C)CC3(F)F)C2C1 C1(C)(OC)CCCN(C(=O)CNc2cccnc2)CC1.C12CCN(C1)C2=O C(C(C)(COC)C(=O)N1CCC(COC)(NC(=O)C(O)CC2CC2)C1)OC c1(NC(C)CC2CC2)[nH]c(=NCCC(=O)N(C)C)nc2sccc12.C1CS1 c1(CCC)ncoc1C(=O)NCC(C)NC(=O)Cn1nnc(=O)[nH]1 C1(C)(c2cn(C(C(=O)OC(C)(C)C)C)nn2)CCCN1C(C1(COC)CCC1)=O C1(NC(CC2CC(CC)C2)=O)CCC2(CCCN(C(=O)C(C)(F)F)C2)C1 C1(C(N2CCOC(CN(C(=O)CN(C)C3CC3)C)C2)=O)(CC)CCC(F)(F)CC1 C(=O)(CCCC(=O)NC)NC1C(CC)CN(C(=O)CSC(C)C)C1 C(CC(=O)NC(CC)CCCO)(C(F)F)NC(CC=C)=O c1(CCNC(C(C)Oc2ncccc2C(F)(F)F)=O)ccc2occc2c1 C(C)(C)(CC(=O)NCC(c1ccccc1)N(C)C(c1csc(C(N)=O)n1)=O)OC CC1=NNC(=O)C1CC(=O)NCC1CC1NC(=O)Cc1nn(C)cc1Cl C1(NC(c2ccnn2CC(F)(F)F)=O)CCN(C(=O)C2=NOCC2)C(C2CC2)C1 c1(NC(=O)Nc2c(C(=O)OC)cno2)nc(C)cc(C)n1 N1(C(C(CC)CC)=O)CC2CCN(C(c3ccc(C)c(F)c3)=O)CC12 Cc1nc(Br)sc1C(=O)NCC#CCNC(c1cn(C2CCC2)nn1)=O C1(CC#C)CCCCN1C(=O)C(C1CC=CCC1)NC(c1cc(CC)no1)=O C(=O)(C(C(C)(C)C)NC(C1C=CCC1)=O)N(C1CC(C)OCC1)C CCCC(CCCNC(=O)C(C)Oc1ccccn1)NC(C12CC(C#N)(C1)C2)=O c1(OC)cc(Cc2c(COC)n(C)nn2)cc(CNC(=O)Cn2ccccc2=O)c1 C1(NC(C2CC2c2ccc(F)cc2F)=O)CCCN(C(C2CCOC2)=O)CC1 C(=O)(C(C1CCC1C(F)(F)F)N(C(C1CCCC1)CC)C)NCC(=C)C C(=O)(C(C)(O)C1CCC1)N(CCNC(C1CC(C)(F)C1)=O)CC N1(C(C=NOC)=O)CCC2C(CCCN2C(c2ccc(F)c3[nH]ccc23)=O)C1 C1(NC(C(=O)NC2CC2)=O)CCCCCN(C(c2ccc(F)c(Cl)c2)=O)C1 C1(NC(c2c(C)sc(O)n2)=O)Cc2ccccc2N(C(C2CCCN2N=O)=O)C1 S(=O)(=O)(c1ccc(S(=O)(=O)NC2CCNC2(C)C)c([N+](=O)[O-])c1)N(C)C C1(N(C(CNC(C)=O)=O)C)CCN(C(=O)CNC(=O)OC(C)(C)C)CC1 C(=O)(C(C)(C)C(=O)N1CCCC1)NCC(CC(=O)N(C)C)OC C1(CNC(=O)CN2CCCC2)CCCC(CNC(c2csnn2)=O)C1 C#CCC(C)(C(=O)NC1CC2CSCC2C1)NC(=O)COCCCF N1(C(CCc2ccc(C)nc2)=O)CCN(C(=O)C(O)CC2CC2)C2(CCC2)C1 N1(C(c2c(CC)n[nH]c2)=O)CC2CCCC2(NC(C2CC23CC3)=O)C1 C(CC(=O)NCC(C)(C)NC(C1CC(C(C)(C)C)=NO1)=O)(C(F)(F)F)OC C1(NC(C2CC(CC)C2)=O)COC2(CCN(C(c3c[nH]ccc3=O)=O)CC2)C1 N1(C(c2cc(OC)no2)=O)CCN(C(c2ccc(CN(C)C)nc2)=O)C(CO)C1 c1(C(N2CCC(NC(COCCCOC)=O)C2)=O)cc2c(Cl)nccc2o1 c1(C(=O)NCC(C)N(C(c2c(COC)nn[nH]2)=O)CC)nccc(C(F)(F)F)n1 C1(N(CCc2ccc(C)cc2)C)CCCN(C(c2ccc(Cl)cc2)=O)C1=O CCC(CC(=O)NCC(O)CCNC(C1CC(N(C)C)C1)=O)SC C1(N(CCN(C)CCO)C)CCc2ccccc2NC1=O C(=O)(C1=C(Cl)CCCC1)NC1CC=C(C(=O)NC2CCN(CCF)C2)C1 CN1CC(O)CCC1C(N1CCC(C(C)(C)NC(=O)Cc2ccc(F)cc2)C1)=O C1(NC(C2C(C)N(C(=O)COC3(C)CCC3)CC2)=O)CCN(C)C(=O)C1 C1(NC(c2n(C3(CO)CC3)nnn2)C2CCC2)CCc2n[nH]cc2C1 n1(CC)nc(C(N2CCC(CNC(c3onc(Br)c3C)=O)C2)=O)cc1C C1(C(N2CCN(CC(C)(C)NC(=O)C(F)C3CCC3)CC2)=O)CC12CCCCC2 c1(NC(N2CCCN(C(c3c(C)nn(C)c3F)=O)CC2)=O)ccc(Cl)c(Cl)c1O c1(SC)ccc(Cl)c(C(=O)NCCCC(C)NC(C2(C)CNC(=O)C2)=O)c1 C(CCCC(=O)O)n1cc(CC2CC(C(N(C)Cn3cccnc3=O)=O)C2)nn1 N1(C(C2C3CC3CN2C(=O)CC2C=CCC2)=O)CC2C3C=CC(C3)C2C1 C(C(=O)NCC(O)CNC(=O)C(C)(C)c1cncnc1)(C(C)C)n1ncc(C)c1 C1(NC(=O)C(F)C2CCC2)CN(C(c2csc(-c3cccs3)n2)=O)CC2CC12 S(=O)(=O)(c1ccc(S(=O)(=O)NC2CC(=O)N(Cc3ccccc3)C2C)cc1)NC c12ccc(c(Cl)n1)CC2.N1(C(C2N(c3ccccc3)CC(F)C2)c2c(C)ncs2)CC2CC2C1C#N CC(C)C(CNC(c1nc(C(C)(F)F)cs1)=O)NC(=O)CCc1cncs1 c1(OC)cc(C(=O)NCc2ccc(C)cn2)c(NCc2cc(C#N)ccn2)cn1 c1(CN2C(C(=O)Nc3nccc(COC)c3)CCC2C)ccc2c(c1)CNC2=O N1(C(CN2CCCC(CC)C2)=O)CCCN(C(=O)C(Cl)=CCl)C(CO)C1 c1(CC)c(C(=O)NC(C2CN(C(c3ccc(CN(C)C)cc3)=O)C2)C)cnn1C N1(C(c2cccc(C)c2)=O)CC2CCC(N=c3nc(C4(CO)CC4)[nH]s3)C2C1 N1(C(c2cc(C(C)=O)on2)=O)CCN(C(=O)CC2CCCSC2)C(C(C)C)C1 C1(C(=O)NC2CC(C)(NC(CCCc3onc(CC)n3)=O)C2)CCC2(CCC2)O1 N1(C(c2c(C)non2)=O)CCC(C)(C)C(C(N2CCC(C)C2)=O)C1 Cc1nc(NCc2cn(C)nn2)cc(N2CCN(C(c3cn[nH]c3)C)CC2)n1 CC1=C(C(=O)NC(C)CCNC(=O)C(O)CC(N)=O)Cn2nnnc2N1C c1(C(=O)NC2CC(C)(NC(c3cnc(CCC)s3)=O)C2)cncc(C)n1 N1(C(C(C=C)OC)=O)CCN(C(=O)Cn2nnc(C)n2)C(c2ncc[nH]2)C1 N1(C(c2cn(CCC=C)nn2)=O)CCC(NC(=O)C(CC)(CO)OC)C(O)C1 CCC(C)C(C(=O)NC)NC(=O)NCCc1coc(-c2ccccc2)n1 c1(C(N2CC(CNC(C=CCC)=O)C(O)C2)=O)cc2cnccc2[nH]1 C1(C#CC(=O)NC(C)CCCNC(c2cnc(C3CCC3)nc2O)=O)(CC)CC1 CN1C2CCC1CC(C(=O)NCC1(F)CCC(NC(=O)CCc3cccs3)C1)C2 N1(C(C2C(=O)NCC2)=O)CCN(C(c2cnnc(O)c2)=O)CC1 c1(CC)cc(C(=O)N(CC(C)C(=O)NCCC2CCSC2)C)nn1C O=C(NNc1cccc(-c2nn[nH]n2)n1)c1cc(I)ccc1-n1cnnn1 CC1(C)CN(C(=O)Cc2ccoc2)CCN(C(C2(C#N)C(C#N)C2(C)C)=O)C1 c1(CC(C)C)nn(CN2CCC(Oc3ccccc3)CC2)c(=S)n1C Cc1sncc1CNC(=O)C(C)(C)C1CCCN1C(=O)COCC(C)(C)C c1(C(C(C)NC(c2cc(Br)co2)=O)NC(CC2(OCC)CC2)=O)ccccc1 CC1CN(C(c2cc(C(F)(F)F)ccn2)=O)CC1CNC(c1cncc(O)c1)=O C1(C(N(CC(=O)N(CC(F)F)C)CC#C)=O)CCCC1C C1(C(N2CC3C(NC(CCCc4[nH]c(=N)sc4)=O)C3C2)=O)CCn2cnnc2C1 c1(OC)ccc(F)c(C(=O)N(CCCNC(C2CCC3CC23)=O)CCO)c1 C(=O)(CCC(F)(F)C(F)(F)F)NC1C(NC(c2c(OC)ccc(F)c2)=O)C1 Cc1c(F)cc(-c2cc(F)c(N)cc2Cl)cc1F c1(CCC(c2onc(CC)n2)C)nccn1OC(C)C C1(CNC(c2c(CC)con2)=O)CCN(C(C2Cc3nncn3C2)=O)C1(C)C C1(F)(CNC(C2CC2C2CC2)=O)CCN(C(c2cn(C3CC3)cn2)=O)C1 c1(NC(C2CC23CCN(Cc2ccc(Cl)cn2)C3)=O)cc(Br)ccc1[N+](=O)[O-] c1(OC)ccccc1CNC(=O)C(CCN(C)C)NC(c1nc[nH]n1)=O NC1CC2CN(C(=O)C(c3cccc(Cl)c3)N)CCN2C1=O CC(C)(C)C(C(=O)NC1C2CCC1N(C(c1cccnc1O)=O)C2)n1ccnn1 c1(C(=O)NCC(C2(O)CN(C(=O)CS(N)(=O)=O)C2)(C)C)cnc2[nH]cncc1-2 C1(NC(c2cccc(C#C)c2)=O)CCN(c2ncc(C(F)F)cn2)C12CCC2 N1(C(C23CC2CN(Cc2c(F)ccc(O)c2F)C3)=O)CCC(O)C(F)(F)C1 N1(Cc2n(C)ncn2)CCC(NC(c2ccc(C(N)=O)[nH]2)=O)C(O)C1 C1(C(=O)NCc2oc(C(=O)NCCOCC(=O)OC)c(C)n2)CCC(O)CN1C c1(C(=O)NCCCCC(C)NC(=O)C(C)(C)F)cc2ncccc2cc1Cl C12(CNC(CC3(NC(C(CC=C)OC)=O)CCC3)=O)CCC(C1)C(=O)N2 N#CC1CN(C(C2(CNC(c3ccc(CC#N)cc3)=O)CC2)=O)CCO1 C1(CC)CN(C(=O)C(CN=[N+]=[N-])NC(c2ccoc2)=O)CCCO1 CCCC(CCC)C(=O)NC1CCCC1NC(c1ccc(Br)nc1OC)=O C1(CC(N2CC(OC)C(NC(C3(O)CCCCC3)=O)C2)=O)OCCCC1(C)C N1(C(c2c(C)con2)=O)CC2CCC(C1)N2C(c1ccn2c1CCCC2)=O n1(CC(=O)OC)cc(NC(C2CC(n3cc(C4(CO)CCC4)nn3)C2)=O)cn1 C=CCC(C(=O)N(C(C(=O)NC(c1nccs1)C)C1CC1)C)C(C)C CC1C2CN(C(=NCCSc3ccccc3)NCc3ccccc3)CC12 N1(C(CCC(=C)C)=O)CC(C)CN(C(=O)CN(c2ccccc2)C(C)=O)CC1C N1(C(c2nccc(C)c2)=O)CCN(C(=O)CN2CCCC2=O)CC(C)(F)C1 c1(N(C2CCCN(C(CC(CC)OC)=O)C2)C)cc(C)nc(C(C)(C)C)n1 N1(C(C(C2CC2)OC)=O)CC(NC(c2ccccn2)=O)C(c2nccn2C)C1 CC1CCC(NC(C2CC2(C)C)=O)CN1c1nnc(C(F)(F)F)s1 c1(C(=O)NCC2C(NC(C(CC3CCCCC3)OC)=O)CC2)ccc(Cl)nc1N c1(C(N2C(CCNC(C3CCN(C)C3)=O)CCC2)=O)cc(C(C)(C)C)ccn1 C(=O)(CC(C)(F)F)N(C1CCN(C(C2COCCN2C)=O)CC1)CC n1(CC)c(C)cc(C(=O)NC(C2CCCN2C(=O)C=CCCC(C)C)(C)C)c1C N=C1NC(=O)C(CC(=O)OCC2C=CCC2)S1 C=Cc1ccc(C(=O)N(CCCNC(=O)CCc2ccc(O)c(Cl)c2)C)cc1 C1(OCC)CN(C(=O)CCNC(C)=O)CC1CCCC.C12CC(=O)C1CNC2=O c1(C(N(C(CNC(=O)CCc2cscn2)C2CC2)C)=O)cccc(S(C)=O)c1 C(CCOCCO)(C(=O)N(C)Cc1cncnc1)NC(C(C1CCC(=O)N1)C)=O N1(C(C2N(C(C(C)S)=O)C3C(C2)C3)=O)CCC(C2CCOC2)C1 Cc1cc(C)c2c(C)c(C(=O)NCC3CCC3NC(C3CCCOC3)=O)sc2n1 C(=O)(C1CCCc2n[nH]cc21)N1CCC(CCCNC(C(C(C)C)F)=O)CC1 N1(C(c2c(CC)oc(C)c2)=O)CC(C(=O)N(CC)CC2CCCO2)CC1(C)C n1(C(C(=O)NC2C(NC(CSCCOC)=O)C2)C)cc2ccccc2n1 C1(C)(CNC(C2(C)CCC2)=O)COCCN(C(=O)CNS(=O)(=O)C2CC2)C1 c1(NC(=O)Nc2ncc(C)nc2C)ccc2c(c1)OC2C C(c1ccsc1)=CC(=O)NC(CC1CC1)C(=O)NCc1ncsn1 C(=O)(C[SH](=O)=O)NC(C)(C)C.CC(C(=O)NCC(C1CC1)=CC)c1ccco1 C1(OC)(CNC(c2ccc(C)o2)=O)CCN(C(=O)C(C)(C)COCC(F)F)C1 C1(NC(CC2CCN(CC)CC2)=O)CCN(C(c2cc(C#N)oc2C)=O)C12CC2 Cc1ncc(C(=O)NC2CCN(C(c3ccoc3Cl)=O)CC2C)cc1CC(C)C C1(N(C(C2(NC(C)=O)CCC2)=O)C)CCCN(C(C23COCC2C3)=O)CC1 Cc1c(C(=O)NCC(O)CCNC(=O)C2=COCC2)c[nH]c2nccc1-2 N1(C(CC(C=C)(C)C)=O)CCCN(C(c2cccc(OC)c2C)=O)CC1C C1(CC)(NC(c2ccc(C3CCOC3)cc2)=O)CCCN(C(=O)CCC2CC2)C1 c1(C(N2CCC(CCNC(CCC(C)SC)=O)C2)=O)cc(N)c(F)c(F)c1F C=CCC(CO)NC(c1occc1CNC(=O)C(n1nccc1C)C)=O C1(NC(c2cc(CC(=O)OC)on2)=O)CCCC12CN(C(C1CCCCC1)=O)C2 Cn1ncc2cc(C(=O)NCC3CCCC3NC(=O)Cc3ccsc3)cnc12 CCCC(CC)CCC(=O)NC(C(=O)NCC(C(C)C)C(C)C)C1CC1 c1(CN(C2CN(C(=O)C(C)(C)c3ccccc3)C2)C)ccnc2c(O)cccc12 Cc1ccc(F)cc1C(=O)NC1CCCC(C(N2CC3(CC3)C2)=O)C1 N1(c2c(C)cncn2)CCN(Cc2ccc3sccc3c2)CC1C#N C1(C(=O)NC2(CO)CCN(C(C(C)(C)OC)=O)C2)CC12CCC(F)(F)CC2 C(=O)(C(CNC(c1coc(C(F)F)c1)=O)CC(C)C)NC1(CSC)CC1 Cc1cn2cc(N(C3CCNCC34CC4)C(=O)CCCN(C)C)ccc2n1 c1(CNC(C2N(C(CSCC)=O)CC=C2)=O)ccnc(O)c1 c1(C(=O)NC2(CC)CN(C(=O)C(C(C)C)C3CC3)C2)cccc2[nH]ccc12 C1(C(N2CCCCC2CCN(C)C)C(=O)NCC(C)C)C(F)(F)C12CCC2 c1(C(=O)NCCC(C)N(C(c2ncn(CC)n2)=O)C)nc(C)ccc1O N12CCN(C(C)C1=O)CC2.C1(N(C2CNC2)C(C)=O)CCN(c2ccccc2)C1 n1(CC(C)O)cc(C(=O)NC(CNC(C2CCC(C)O2)=O)C(C)C)ccc1=O c1(NC(C(C)Nc2ccccc2CNC(=O)OC(C)(C)C)=O)ccc(Cl)c(Cl)c1 Cn1cnc2[nH]c(=NCC3(CNC(c4cc(Cl)no4)=O)CCC3)nc(O)c12 C1(NC(c2cccc(OCC(C)C)c2)=O)CC2CN(C(c3n[nH]cc3Cl)=O)CC12 c1(C(N2CC(NC(C3(C(C)(F)F)CCC3)=O)C2)=O)ccc(NC(=O)C=NO)cc1 CCC(CC(=O)NCC(Cc1ccccc1)NC(=O)C=C(C)C(C)C)OC CC(C)C(CC(=O)NCC(C)C1CC1)NC(c1cnn(C2CC2)c1)=O c1(C(=O)NCC=CCNC(C(C(C)OC)O)=O)nc(C)ccc1O c1(CC)cc(C(=O)NC2CC23CC(NC(=O)CCCC2CC2)C3)cn(C)c1=O C1(NC(C)=O)CCC(C(N2CC(NC(c3nnc(C(C)C)s3)=O)C(C)C2)=O)CC1 CC(C)CCC(F)C(=O)N1CCC(CF)(NC(=O)CC(C)n2ccnc2)C1 N1(C(C(=O)NC2CCN(c3cc(C)nn3C)C2)=O)CCC(C#N)CC12CC2 C1(NC(C2CCCC(OC)C2)=O)CC(F)CN(C(=O)C(C)(CO)NC(C)=O)C1 c1(NC(CC=C)=O)cccc(NC(C2CCN(Cc3ccnc(F)c3)C2)=O)c1 N1(C(=O)Nc2cc(C3CC(F)(F)C3)[nH]n2)CCC(N2CCCNC2=O)CC1 CC1CN(C(C2(Br)CC2)=O)CC2(CCN(C(=O)CCCCC3CC3)C2)O1 N1(C(C2(C(C)C)CCC2)=O)CC(C2CCN(C(=O)CC3CCOC3C)CC2)C1 C1(C(=O)NC)CC(C)CN1C(C1CCC(CNC2(C(=O)OC)CCCC2)CC1)=O c1(OC)cc(Cl)ccc1C(N1CC(CNC(=O)Cn2cccc2)CCC1C)=O C12(C(N(C(C)CO)CCO)=O)CC(C(=O)N(c3ccccn3)CC(C)O)(C1)C2 N1(C(C2C(C(=O)O)CC2)=O)CCNc2ccc(Br)cc21 C1(C)(CC)C=C(C(=O)N2CC=CCC2C(=O)NCC(C)(C)CC(F)F)C1 C1(C(=O)NCC(CC=C)NC(c2cnn(C)c2Cl)=O)CC(OC)C(OC)C1 CCCCC(CC)CC(=O)N1CCCC(CCC(=O)NC2CCCC(C)(C)C2)C1 c1(CC)cc(C(=O)NCCc2ocnc2CNC(=O)CC(O)CN(C)C)c(C)nn1 C1(C(=O)NC(C(C)(C)NC(CCC(=C)C)=O)C)CCc2nnc(Br)n2C1 c1(C(=O)OC)cc(C(=O)NC(C)CNC(c2cccc(-c3ncc[nH]3)c2)=O)ccn1 C(CCCCC(=O)N(C1CCCN(C)C1)C)N(C(c1cnc(C)o1)=O)C C1(C(=O)NC(C2CCN(C(c3ccnc(O)c3)=O)C2)C)CC2CCC1CC2 C12(NC(Cc3c(C)non3)=O)CC3CC(C1)CC(NC(C14CC(C)C1C4)=O)(C3)C2 N1(C(=O)C(c2cccc(F)c2Cl)(F)F)CC2(C1)CN(C(C13CCC1C3)=O)CCO2 N1(C(C2C(C)C2)=O)CCC(N2CCC(NC(C3CC4CC4C3)=O)C2)CC1 C1(CNC(=O)Cn2nnc(=O)[nH]2)CCCCCN1C(C1CCS(=O)(=O)CC1)=O c1(C(N2CCC(C(=O)Nc3ccc(C)nc3Br)CC2)=O)cc(F)c(CO)cc1F C(=O)(C(CC(F)F)N(C(=O)CC(C)C)C)NC(CCCC)C C1(CNC(C(C)C(F)(F)F)=O)CN(C(=O)C=CC=C(Cl)Cl)CC(C)(C)C1 c1(C(=O)NCCC(=C)CNC(=O)C=CCCC=C(C)C)cc(C)cc(Cl)c1 N1(C(CC(=O)OC)=O)CCN(C(=O)CC2COC3CC2C3)C2CCCCC12 N1(C(C(C)P(C)(C)=O)=O)CCN(C(C2CC2(C)C)=O)CC12CC2 C1(C(=O)NCc2ccc(CNC(c3cn(CC)nn3)=O)cc2)CCC2CC1CO2 N1(C(CN(C2CCOCC2)C)=O)CCC2CCC(NC(=O)C(F)CC3CC3)C1C2 c1(CNC(=O)NC(C2CCCO2)COC)ccccc1C#Cc1ccccc1 c1(NC(=O)NCC(=C)F)cc2c(s1)CCOC2 c1(C(N2CCC(CCNC(C(C)S(C)(=O)=O)=O)C2)=O)nc2cc(O)ccc2[nH]1 n1(CCC)ncc(C(=O)NCC2(F)CC(NC(=O)CCC3CCC(C)O3)C2)c1C N1(C(c2cnc(C)o2)=O)CC23CCCC2(C1)CN(C(=O)CC(C)CF)C3 n1(CCC)ccc(=NC(=O)C2N(C(=O)CC3CCCOC3)CC23CCCC3)[nH]1 C1(C(C)C)(C(=O)N(C(C)CC(N)=O)C)CCN(C(=O)C2CC2)C1 C#CCCCC(=O)NCC1CC(C(F)(F)F)CN1C(C1CC(Cl)(Cl)C1)=O c1(C(=O)NCCC(C)NC(C2(C#N)CCCOC2)=O)cc2cc(Cl)ccn2n1 C1(N(C(CCC)=O)C)CCCN(C(c2ccc(C(C)(F)F)nc2O)=O)CC1 C(=O)(C(C)CS(C)(=O)=O)N(CC(C)(C)CNC(c1cnc(C2CC2)o1)=O)CC N1(C(C(CC)CC)=O)CC(NC(c2ccn(C3CCC3)n2)=O)CC(O)C1 C(=O)(CC(CC)C1CCC1)NCC(CC=C)NC(c1cc(C2CC2)c(CC)s1)=O C1(CN(C(=O)C(=Cc2c[nH]cn2)F)C)CCCCN1C(c1ccn(C(F)F)n1)=O c1(NC(N(C)CCN2CCCCC2)=O)oc(C2CC2)nc1C#N c1(CCC(N2CCC(C)(NC(C3N(CC)CCC3)=O)C2)=O)n[nH]c2ccccc12 c1(CNC(C(C2CCCCC2)NC(C)=O)=O)cc(C)ccc1S(N)(=O)=O N1(C(C2(C#N)CC(C)C2)=O)CC2(C1)CN(C(=O)CN1CC3C=CC1C3)CC2CO C1(NC(c2coc(Cl)n2)=O)CCN(C(=O)CSc2nncn2C2CC2)C1 N1(C(C(N2CCNC2=O)C)=O)CC2CCCC2(NC(=O)COCC2(F)CC2)C1 C1(C(=O)NCC2(C)CCN(C(=O)COC3CCC3)C2)NC(=O)C2CCC12 c1(C(=O)NCCOC2CN(C(C3(C)C(C)C3)=O)C2)ccnn1C1CCCC1 N1(C(CCC=CC(C)C)=O)CCC(C)C(NC(c2ncsc2C(C)C)=O)C1 CCCCCC(CC)C(=O)NC(C)CCNC(C1CC(C)OC(C)C1)=O C(C(=O)NCC1C2CN(C(=O)CCCc3ccccc3)CC12)(C(C)C)OC n1(CC(=O)NSCCCNC(COCCOCCOCC#C)=O)ccccc1=O C(=O)(CCCCN(C)C1CC1)NC(CC)CN(C(=O)CNC(=O)C(F)(F)F)CC N1(C(CSCC#C)=O)CC2CCCC2(Nc2ncncc2Cl)C1 c1(C(=O)NC23COC(C(=O)NCCO)(C2)C3)cccc(-n2cc(CO)nn2)c1 c1(Cn2cc(C(N3C(C)C(c4ccccc4)CC3)=O)nn2)cc2scc(Cl)c2[nH]1 c1(C(N(CCNC(c2c(Cl)ccc(CC)c2)=O)C)=O)c[nH]nc1S(N)(=O)=O N1(C(C(CC#C)O)=O)CC23CCCC2(C1)CN(C(c1ccnn1CCCC)=O)C3 CC1CCN(C(=O)CC2CCOCC2)C1CNC(C12CC(C1)C2)=O c1(OCC)cc(C(N2CC3CC2CC3NC(=O)C=Cc2ncc[nH]2)=O)ccc1C CCC1=NOC(CC(=O)N(CC(CC)NC(c2cc(COC)cs2)=O)C)C1 C(=O)(C1=C(C#N)CCC1)N1CCC(C#C)(C(=O)NCc2cc(C)cc(C)c2)C1 CC(CCC(=O)N1CCCC1C(=O)Nc1ccccc1)NC(N)=O c1(C(=O)NC2C(CNC(c3c(C)ncs3)=O)CC2)cc2cc(Br)ccc2o1 C1(NC(C2N(CC)CC2)=O)CC2CCC1N(C(=O)Cn1cccn1)C2 C1(C(=O)NCc2csc(C(N3CC(CO)C3)=O)c2)(OCC)CCCC1 Cn1cnnc1CNC(C1CC(NC(=O)CCn2cccc2)C1)=O c1(CC(=O)NC2CCC2NC(C2CC(C(F)(F)F)C2)=O)c(Cl)cccc1Cl C(=O)(CC(C)(C)C(F)F)NC1C(CNC(c2c(N(C)C)cncc2)=O)CCC1 N1(C(C2CC(NCc3ccccc3F)C2)=O)CCC(F)(F)CC1 CC1(C)OCCC1C(N1CCCCC1CC(=O)NCCCOC(=N)O)=O n1(CCC)ccc(C(N2CC(C(C(=O)NC(COC)CC)OC)C2)=O)n1 c1(SC)sccc1C(=O)NC1CC(CNC(=O)CCOC2CCOC2)C1 c1(C(N2CC(NC(c3ccc(F)cc3)=O)C3C2C3)=O)cc2cccc(Cl)c2[nH]1 c1(C(=O)OC(c2cccc(C3COC3)c2)C(=O)OC)cc(Br)c(OC)cc1N C12(NC(C(c3cccc(Cl)c3)C)=O)CC1CN(C(=O)C=Cc1ccn(C)c1)C2 C1(C(=O)N(CCCNC(=O)C#CC2(C)CC2)C)(OC)CCCC(C)(C)C1 N1(C(CC(=O)OCC)=O)CCCCC(NC(=O)C(C)(c2cccs2)N(C)C)C1 C1(CC(=O)NC(c2cnc[nH]2)C)CN(C(c2cnccn2)=O)CCO1 c1(N(CCCC(CCCC)CC)C)ccc(S(=O)(=O)NCc2nccs2)cc1Br CC1CC(NC(=O)CN(CC(C)(C)C)C)CN1C(C1CC(N(C)C)C1)=O c1cccc(F)c1.c12cn(nn1)CCNC2=O.C(C(=O)NC)N(C)C.C1(=O)CN1 C(=O)(C1CCCc2nn[nH]c21)NCC(CNC(C1=NOC(C)C1C)=O)(C)C CC(C)CCC(=O)C(=O)NC(CO)C(N1CCC([N+](=O)[O-])CC1)=O N1(C(C2(F)CCC2)=O)CCC(C2CCN(c3ccc4nccnc4n3)CC2)CC1 N1(C(C2(CCOC)CC2)=O)CSCC1C(=O)NCc1ocnc1C C=CCC(CNC(c1c(C)cnn1CC)=O)C(=O)N(C)Cc1ncccn1 C1(CNC(CNC(Cc2c(C)n(C)nc2)=O)=O)CC2CCC(C1)N2C(=O)CCF C=CC(CC)CC(=O)NCC(=C)CCNC(=O)CCc1cccc(C#N)c1 N1(C(C2CC=CC(C(=O)NCc3cccnc3)C2)=O)CCC(O)C12CCCC2 C1(C(=O)NC2C(C#N)CN(C(=O)CC(F)(F)F)C2)CCc2ccccc2C1O C(=O)(CC(C)(C)C#N)N(CCOCCC(=O)NC(c1nccs1)CC)C c1(OC)ccc(S(=O)(=O)NC(=O)NNC(c2cc(Cl)nc3n[nH]cc23)=O)cc1C c1(CC(=O)N(C2CCN(C(=O)C=CC3CCOC3)C2)C)cccc2nonc12 N1(C(C(C(C)C)SC)=O)CC2(CC(NC(c3c(C)noc3N)=O)C2)C1 C=C=C(C)CC(=O)NCC(C)CN(C(=O)Cc1cccc(CC)c1)C C1(CC)C(C(=O)NC2(C)CN(C(=O)Cc3cnn(C(C)C)c3)C2)CCN1C CCCC(CCNC(=O)CC1CC1CNC(C1(C2CC2)CCCO1)=O)C1CC1 c1(OC)ccccc1S(=O)(=O)N1CCN(Cc2cc(Cl)cc(Cl)c2)CC1CC#N c1(C(N(CCCN(C(=O)CN=S(C)(C)=O)C)C)=O)ccc(C(F)(F)F)c(O)c1 CN1CCC(C2CCN(C(C3CC(c4ccc(C(C)(C)C)cc4)C3)=O)CC2)C1 c1(OC)cc(CN2CC(C)CC2C(=O)Nc2ccc(Br)cc2C)cc2c1OCO2 C1(N(C(c2nnn(C(C)(C)C)n2)C(=O)NCCC)C)CC2(CCC2)C1 N1(C(C(C)c2ccco2)=O)CC2CCC(NC(c3cccc(F)c3F)=O)CC2C1 CC1C(NC(C2CCC(F)(F)C2)=O)CCN1C(c1cc(=O)n(C)o1)=O c1(CNC2CCC(n3cc(CN)nn3)C2)nccc2c1[nH]c1ccccc21 N1(C(C(C)(C)SC)=O)CC2CC2(NC(=O)CC2CCCOCC2)C1 C#CCCCCCC(=O)N1CC(NC(c2cc(C)c(Cl)c(N)c2)=O)CC(C)(C)C1 c1(C(=O)NC2CC(CNC(C3C(C)CC3C)=O)C2)cc([N+](=O)[O-])nn1C C1(CC#C)(C(=O)NCc2ncn(CC)n2)CCN(C(C2CCNC2=O)=O)C1 N1(C(C(C)OCCOC)=O)CC2(CCN(C(=O)CCCc3ccncc3)CC2)C1 C1(NC(C(C)OC(F)F)=O)CC2COCC12 N1(C(c2cccnn2)=O)CCCC2(CCN(c3ncc4cccnc4n3)C2)C1 N(C(=NCCCCl)NCc1cc(C(=O)OC)ccn1)C1CCC(CC)CC1 Cc1cc(C)c(NC2CCN(CC(=O)NC3CCOC(C)C3)CC2)o1 c1(C(=O)NC(CCCCNC(CCCOC)=O)C)cn2c(C)cccc2n1 C1(CC)(CO)CCN(C(c2ccc(C)nn2)C(=O)NC(C)C(=O)OC)CC1 N1(C(C(C)CF)=O)CCC(CC(C)NC(c2cncc(C(F)F)c2)=O)CC1 N1(C(c2ncn(C(C)C)c2)=O)CCC(C)(C)C(C(=O)NCCN2CCCC2=O)C1 c1(C(c2n(CC=C)nnn2)NCc2ccn(C3CC3(F)F)n2)nc(C)sc1C N1(C(c2c(CCC)n[nH]c2)=O)C2CCC1C(C(=O)NCCCC(C)(C)C)C2 C(CO)(CO)(CO)NC(C1C(CNC(Cc2cc(C)on2)=O)C1(C)C)=O C1(CNC(c2ccc(N)cn2)=O)(CNC(c2csc(S)n2)=O)CC2CCCC2C1 c1(CC(C(=O)NCC2CN(C)C3CC23)OC)cnn(C)c1O C1(c2c(OCC)c(C)cc(C)c2)NC(=S)N(C(CC)CC)C2=C1C(=O)NC(C)C2 C(=O)(C(CC(C)C)CC(C)C)N1CCC(N(C(CNC(=O)OCC)=O)C)C1 c1(C(N2C(CNC(CC(=O)NCC#C)=O)CCC2)=O)cccc(F)c1O Cc1cc(C#N)ccc1-c1cnc(NC(C2CCCC2C)=O)s1 c1(CCC(N2CCN(C(C(CC)SC)=O)CC2)=O)csc2nc(C)cn12 C1(CC(=O)NCCN2CCC(NC(c3[nH]c(=N)sc3)=O)CC2)CCCCC1(F)F C1(OCCC)CCCN(C(=O)Nc2cc(C)n(C(F)F)n2)CC1 N1(C(C(C)(C)SC)=O)CCC(C)C(CC(=O)N(CC(=O)NC(C)C)C)C1 C(=O)(CCC(C)(C)C)NC(C(C)C)C(=O)NCC1C=CCOC1 C(CO)(C(=O)N(C)C)NC(C(SC)SC)=O.C12(CC1)CC(=O)NC2 C1(C(N2CCC(Nc3cc(C)no3)CC2)C(=O)NC)C2CCCCCC12 C(CC(C(=O)NCC(O)C(F)(F)F)OC)NC(c1c(OC)scc1)=O C12(C(=O)NC3C(NC(=O)COC4CCOC4)CCCC3)CCCC(CCC1)C2 n1(CC(=O)N(CCCCNC(C2CNC(=O)N2)=O)C)ccc(=O)c2ccccc12 N1(C(C2COCC(C)O2)=O)C2CCC(C2)C1C(N1CCC(F)(CF)C1)=O C1(C(=O)NC(Cc2cn[nH]c2)C(=O)NCc2nn[nH]n2)CCC2CC1CO2 c1(N(C(CC(COC)C)=O)CC(=O)NC2CCC2)c(C)cccc1Br C(=O)(C(C)(C)C(F)(F)F)NCC(CC(=O)Nc1c(OC)cccc1O)C C1(C2(O)CN(C(C3CCCCC3O)=O)C2)(CNC(c2cc(CC)nn2C)=O)CC1 Cn1cc(C(N2CCOCC(NC(c3cnc(OCF)cn3)=O)C2)=O)ncc1=O S(=O)(=O)(c1cnc(N2CCC3(CNC(=O)C3)C2)cc1C)NCC1(N(C)C)CC1 C(CCCC(C)NC(=O)OC(C)(C)C)NC(C1C(CC(=O)OCC)CCCS1)=O Cn1ccc(CN2C3(C)CN(C3)C2=O)c1.c1(CCCN(C)C)nonc1N c1(C(N2CC(CNC(C(C)=CC)=O)C(O)C2)=O)nccc(Br)c1C N1(C(CC2(C)OCCO2)=O)CC(NC(C2C=CCC2)=O)CC(O)C1 CC1(COC(C2CCC(=O)N(C(c3ccc(F)cc3F)=O)C2)=O)CC2CCC1C2 c1(N(C)CC2N(C(c3n(C(C)C)ncc3)=O)CCC2)ccc(Cl)cc1[N+](=O)[O-] c1(C(N2CCC(NC(CCS(C)=O)=O)CC(O)C2)=O)ccc([N+](=O)[O-])c(N)n1 CCCCCS(=O)(=O)CC(=O)NCCCNC(c1nnc(S)n1C)=O C1(NC(CN(C(=O)OC)C)=O)CN(C(=O)C(C)(F)CC2CCCC2)CC1(C)C C1(C(N(C)CCNC(=O)CCC2CCOCC2)=O)CCC2(C1)CC2(F)F N1(C(CCSCC(=O)OC)=O)CCCC(NC(=O)CC2CC2(C)C)C1C N(C1CN(C(=O)COCCCF)Cc2ccccc21)C(=O)CCC(F)F C1(CC(=O)N(C)Cc2ccsc2)CC(C)(C)CN1C(c1cncc2[nH]ccc12)=O C#CCCCC(C)(c1nnnn1CCSC)NCC(C)C(=O)OCC c1(C(C(=O)NCC2CC2)N(CC#CC)CC#C)nc(C(F)(F)F)n2c1CCCC2 c1(C(N2CCN(C(=O)CSC(F)(F)F)C(CC3CC3)C2)=O)nccc2occc12 C1(CNC(C2CC23CC3)=O)CN(C(c2scnc2C(F)(F)F)=O)CC1C(F)(F)F C1(C(=O)NC2C(NC(CCCC(OC)OC)=O)C2)CNC(=O)C(C)(C)C1 c1(CN(C(=O)C(Cc2ccccc2)n2cnnc2)C)ccc(F)cc1Cl C(=O)(CC(C)C(C)(C)C)NCC1(F)CC(NC(c2nc(C(=O)OC)sc2)=O)C1 C1(C(N2CCC(NC(CC(C)(C)O)=O)C(C)(C)C2)=O)CC2(CCCCC2)S1(=O)=O N1(C(C2CN(CCOC)C(=O)C2)=O)CCC2(C1)CN(C(=O)CC1C(C)C1(F)F)C2 C1(NC(c2n(CC)ccn2)=O)CCC2(CCCN(C(c3nnsc3N)=O)C2)C1 N(C1CN(c2ccc([N+](=O)[O-])cc2)CCc2ccccc21)C(C1CSCCS1)=O C1(NC(c2cn(-c3ccccc3)nn2)C)CCC(O)C(C)(C)C1 C12(C(N3CCC(NC(CCN(CCC)C)=O)C(F)C3)=O)CCC(N=[N+]=[N-])C1C2 C1(C(N(CCCSC)C)=O)CCCC(NC(=O)C(F)C2CCCC2)CC1 CCCC1c2ccccc2CCN1C(c1ccc(NCC)nn1)=O C1(C(N2CCC(CCN(C)C)C2)=O)CC(=O)CN1C(=O)C(O)CC1CCCC1 c1(C(=O)NC2(CNC(c3cncc(Cl)c3)=O)CCCC2)cc2c(s1)CCC2 c1(CN(C(C2C(C)C2)=O)C)cnn2c1CN(C(C13CCC(=O)N1CCS3)=O)CC2 c1(N2CCC3(CN(C)C(=O)O3)CC2)nc(=NCCCC(F)F)[nH]c2cc[nH]c12 C(=O)(CC(O)(C(F)(F)F)c1ncco1)NC1C(NC(CCCCCC)=O)COC1 c1(C(=O)OC)ccc(N2CCN(CC(F)(F)Br)CC2)c(F)c1 CC1CCC(NC(=O)C(C)(C)c2ccsc2)CN1C(=O)C=CCN1CCOCC1 C(=O)(CCCC(C)NC(=O)C(C)CCCC)NC(C#C)CC1CCCC1 C1(NC(C(N2CC3CCC3(C)C2)COC)=O)CC2(CO)COC1C2 N1(CC2OCC(C)C2)CCN(c2ccccc2)CC1.c1(CN2C(=O)C2)cccs1 Cc1nc(O)nc(C)c1CCC(=O)NCCC1(CNC(C2CC2Br)=O)CC1 C1(NS(c2c(C(C)(C)C)nns2)(=O)=O)COC2(CCCC2)OC1 CCC(CCC(=O)N1CC(C)=CC(C)C1)NC(c1cc(=N)[nH][nH]1)=O Cc1nnc(O)c(C(N2CC(CNC(C3CC(C(F)(F)F)CO3)=O)C2)=O)c1C CC1CN(C(C23CC(C)(CO2)C3)=O)CCC1CNC(C1(N2CCCC2)CCC1)=O C1(NC(c2nc(CCCC)sc2)=O)CC(O)CN(C(=O)C(C)C(C)(C)C)C1 c1(C(=O)NC(C)C(C)(C)NC(C2CCCCN2C)=O)cccc2c1ncn2C CC1Cc2cc(C(=O)N(C)CC3CN(C(C4CCOC4)=O)CCO3)ccc2O1 c1(N2C(CNC(=O)CCC3CC3(Cl)Cl)CCC2)ccc2c(n1)CCC2=O N1(C(CC(=O)NCC)=O)CCCCC1C1CCN(C(c2c[nH]nc2C(F)F)=O)C1 c1(C(=O)OC)ccc2c(c1)CCC(C)N2C(=O)C(c1nn(C)c(C)c1Br)(C)C N1(C(CC2C(OC)CC2)=O)CCN(CCNC(c2n[nH]c(C)c2Cl)=O)CC1 O(N(CC)S(=O)(=O)c1ccc(-c2ccccc2)cc1Cl)CC c1(C(=O)NCCCCN(C(=O)C(O)C2CC2)C)c[nH]c2cccc(Br)c12 c1(OC)cc(C)cnc1C(N1CC(NC(=O)C(C)(C)C2CCC2)C(O)C1)=O c1(OC)nccc(C(N2CCC(C(F)C(=O)N(C)CCc3cccs3)C2)=O)n1 CC1CC2(CCN(C(C3CCN(C(C4(C)CCCN4C)=O)C3)=O)C2)CO1 c1(C(C(=O)NCC(F)F)N(C(=O)COCC(F)(F)F)C)cc(C2CCC2)on1 CP(C)(=O)C(O)C(=O)NCC(C1CCN(C(C2(F)CC2)=O)CC1)F c1(C2(C(N3CC(C(C)NC(c4cnoc4C4CC4)=O)C3)=O)CC2)ccccc1C#N C=CCCC(C)(C)C(=O)NCC(F)(C(=O)NCCCN1CCOCC1)C(C)C N1(C(c2cc(CC)on2)=O)CCC(O)(CCNC(=O)CN2CCOCC2)CC1 c1(C(=O)NC(C(=O)NC(C(C)(C)OC)C)CC2CC2)ccc(O)nn1 N1(C(C2CCC(C(C)C)CC2)=O)CCOC2CN(C(=O)CNC=O)CC12 c1(C(=O)OC)c(F)ccc(NC(C2CC(F)CN(C(c3ccns3)=O)C2)=O)c1F c1(C(N(CCCCCNC(C=C(CC)CC)=O)C)=O)nn(C)c(Cl)c1C(F)(F)F CC(CC=Cc1ccccc1)C(=O)NCCCCCNC(C1CCC12CCC2)=O C1(C(C)=O)(N(C)Cc2cc(O)ncn2)CCCN(C(=O)OC(C)(C)C)C1 C1(NC(C(C#C)(C)C)=O)CN(C(=O)COCc2nc(C)no2)CC1N=[N+]=[N-] C1(NC(=O)NC2CCCCC2)CC(C#N)(c2nnc(-c3ccccc3F)o2)C1 c1(OC)ccc2[nH]cc([N+](=O)[O-])c(=NCCNC(=O)Cc3csc(NC=O)n3)c2c1 N1(CC(=O)C2CCC2)CCN(C(=O)NCC(=O)Sc2ccccc2)CC1 C1(C(N2CC3CC3(NC(c3ccncn3)=O)C2)=O)(COC)CC=CCC1 C1(C(N2CC3CC2C3NC(c2cnc(S)n2C)=O)=O)(COC)CCCNS1(=O)=O c1(OC)cc(I)c(CNC(=O)NCC2CCS2(=O)=O)cc1OC c1(OC)ccc2[nH]c(C(N3CCC3CNC(=O)C=CC=C(Cl)Cl)=O)cc2n1 N1(S(CCC)(=O)=O)CCN(CC(=O)N(C2CCS(=O)(=O)C2)CC[Si](C)(C)C)CC1 C(=O)(CC(CN(C)C)C(F)F)NCc1onc(C(C)NC(CSCC)=O)n1 C(=O)(NNc1cccc(Cl)c1Br)NC1C(NC(=O)OC(C)(C)C)C1 Cc1nc(C(N2CCC(C(C)(C)NC(=O)C(F)CC3CCCCC3)C2)=O)cs1 C#CC1(C(=O)NC2CCCN(C(=O)Cn3cccc3)CC2)CCCCC1 c1(C(=O)NC2CCN(C(c3cn[nH]c3)=O)C2)cc(Cl)cnc1Br c1(N(C(C2CCCC2)C)C)cc[nH]c(=NCCNC(=O)C(C)CC2CCCO2)n1 C(=O)(C(O)CC(C)C)N(CC(CC)NC(c1cnn(CCC)c1C)=O)CC c1(C(=O)NCC2C(NC(c3ccc4cnsc4c3)=O)C2)cncc2ccccc12 C1(CC)(NC(C2CCC(F)C2)=O)CCN(C(=O)CCCn2cncn2)CC1 C=CC(CC)CC(=O)NC1CCC(N(C(=O)Cc2n[nH]c(=N)s2)C)CC1 Cc1cc(=O)n(CCC(=O)NCC(CO)NC(=O)C2=CCOC2)cn1 C1(C(=O)NCC2CCN(C(c3cccc(C)c3)=O)CC2O)CCCCC(F)(F)C1 N1(C(c2c(C(N)=O)cccc2)=O)CCC2C(CCCN2C(=O)Cn2cccn2)C1 C1(C(N(C2CCN(C(C3SCCS3)=O)C2)CCC)=O)CC12CCC2 Cc1[nH]nc(C(=O)NCCC2CCCN2C(c2cccc(N)c2)=O)c1C c1(CC(=O)NC2CN(C(CC=CC=C)=O)C3C2C3)cccc(S(=O)(=O)CC)c1 c1(-n2c(C)cc(C(C)NC3CCNCC3)c2C)ccccc1[N+](=O)[O-] C12(CCNC(=O)COCc3nc[nH]n3)CCC(C1)N(C(C1CCOC1)=O)C2 C(=O)(NNC(=O)CC(N)c1ccccc1)c1c(C)nccc1 c1(C(N2C3C(NC(COCC#C)=O)CC(C3)C2)=O)ccc([N+](=O)[O-])n1C c1(C(=O)NC(C2(O)CN(C(c3ccc(CO)cn3)=O)C2)C)cc[n+]([O-])cc1 Cc1cn2c(CC(=O)NCc3ccccc3OC(C)(C)C)cnc2s1 CC(C)CCC(=O)NC1CCC(c2cn(Cc3ccoc3C(=O)O)nn2)CC1 c1(CNc2ccc(C#N)cn2)ccc2c(c1)CCCC2NC(=O)C1=CCCCO1 N1(C(c2c(C)csc2C)=O)C2CCC1CC(CNC(=O)CC1CCC(C)CC1)C2 C1(CNC(Cc2c(C)occ2)=O)CN(C(C2CC23CCOC3)=O)CCC1(F)F c1(OCC)ccccc1OCC(=O)NC1CCCCC1NC(=O)CC(C)(F)F Cc1cccnc1C=CC(=O)NCC1C(O)C(O)CN1C(C1CCCCC1O)=O c1(-c2cn(CCCC(=O)N(CCOCC3CC3)CC)nn2)ccc2nc(C)ccc2c1 C1(F)(C(=O)NC2CCC(C)(CNC(CCC=CC)=O)C2)CCCCCC1 C(=O)(CCC(=O)N(CC(C)NC(=O)C(C)n1ccnc1)C)Nc1nnc(C)s1 c1(C(N2CCCC(CNC(Cn3nnc(C)n3)=O)CC2)=O)ccnc2ccnn12 N1(C(c2c(SC)scc2)=O)CCOC(C(C)NC(=O)CC2CC(C)(C)C2)C1 N1(C(c2c[nH]c(=N)o2)=O)CCCN(C(=O)CC2CC=CC2)CC1c1ccccc1 C1(C(=O)OC)CN(C(=O)C(=O)NCCN2CCNCC2)CCN1CCO C(=O)(C1=Cc2ccccc2C1)N1C(CCNC(C(C)N(C)C)=O)CCCC1 C1(C)(NC(C=CC2N(C)CCC2)=O)CCCN(C(C2CCN2C)=O)C1 c1(C(=O)NCC(CNC(CC2N(CC)CCC2)=O)OC)cncc(OC)n1 c1(C(=O)NC2CN(C(c3c(C)n(C)nc3)=O)C(C)CC2)cccc2ccnn12 CC1CN(C(=O)CC2CCS(=O)(=O)C2)CC1NC(C1(C)CCOCC1)=O Cn1nnc(CNC(C2(F)CC2)=O)c1C(=O)NCCC1(C)CC1(F)F c1(NC(C2C3CC2N(C(C2CC4CCC2O4)=O)C3)=O)c(Cl)cc(Cl)cc1Br C=CCC(C)(CC)C(=O)NC1CCN(C(=O)COCc2ncc(C)o2)CC1CO C1(C(N(CCC)CC)=O)CC(C)CN(C(=O)C(C)NC(=O)C2CC2)C1 c1(C(=O)NCCN(C(C(CC)(CC)OC)=O)C2CC2)cc2c(nc1O)CCC2 CCC(C#N)(CC)C(=O)N1CCOC(CNC(C2CC=CCC2)=O)C1 Cc1ncc(C(=O)NC2(C(=O)NCC(c3cn(C)cn3)O)CC(O)C2)cn1 C1(C(=O)NCCCc2scnc2C)(CC)CN(C(=O)C(O)CN(C)C)C1 c1(CCCC)ccc(C(=O)NCCC(C)(C)NC(=O)C(CC)SCC)cc1 C(=O)(C(N)CCCS(C)(=O)=O)NC(C(=O)OC)(C)C1CCCC1 C=C(Cl)CC(C(=O)N1CC(F)(CF)C1)NC(=O)C(CC1CCC1)OC CC(C)(C)C(CO)C(=O)NC1CN(C(c2ccnn2C2CCC2)=O)CC1N=[N+]=[N-] c1(CNC(c2n(CCSC)nnn2)c2cn(C)nn2)cc(F)c(F)cc1F N1(C(C(C=C)(C)O)=O)CCC(C)(NC(=O)C(C)Oc2ccccc2)CC1 C1(NC(CC(C)OC)=O)CCN(C(c2cncn2-c2cnn(C)c2)=O)CC1CO C(=O)(C1CNC(=O)c2ccnn21)NCC(C)(C)NC(=O)C(O)C1CCC1 C1(C(N2C(Cn3cc(C(N4CCCC4)C)nn3)CC2)=O)CC(=O)NC1(C)C C1(NC(c2ccc(COC)o2)=O)CN(C(=O)Cc2ncc(C)o2)C2(CCC2)C1 N1(C(C2N(CC)CC2)=O)CC(NC(=O)CSc2cccc(Cl)c2)CC(F)C1 C1(C(N(CCCCCCNC(C2(C)CC2Br)=O)C)=O)Cc2ccccc2C1 C1(CC(=O)NC2CCN(OCC)CC2)N(C(=O)CCOC(C)=O)CCC1(C)C N1(C(C(C)NC(c2ccc(C(C)=O)o2)=O)=O)CC(N(C)C)CC1C N1(C(C2(F)C(C)C2)=O)CCC(CNC(c2ncccc2CO)=O)C(F)(F)C1 C(=O)(N1CCC(C(=O)NCC2(F)CC(CO)C2)O1)c1c(C)cncn1 C1(CC)CC(C)CN1C(C1(NC(c2cnn(CC)c2)=O)CCCC1C)=O C1(C(=O)NC2CC(c3ccccc3)(NC(c3n(CC)nnc3)=O)C2)CC=CCC1C N1(C(CCCOC)=O)CCN(C(c2cnc3c(ccn3C)c2)=O)C2COCC12 c1(C(=O)NC2CC3(C(NC(C4C(CCOC)C4)=O)C3)C2)ccc([N+](=O)[O-])nc1 C(C(C)(C)CC(=O)NCC1CC12CCCCC2)OC.C1(N)CC(N(C)C=O)C1 Cc1ncc(C=CC(=O)NCCC(C)(C)CNC(c2ncn(C)c2C)=O)s1 C#CC1(C(=O)NCC(CNC(C2(C)CCCCC2)=O)CO)CCCC1 N1(C(C2(C)C(C)(C)C2)=O)CCOC(C)(CNC(c2ccnc(OC(F)F)c2)=O)C1 C1(C(CNC(C2(CC=C)CCC2)=O)(C)O)CCN(C(c2csc(CC)n2)=O)CC1 C1(CC)CCCC(NC(C2(NC(=O)CCn3ccnc3C)CSC2)=O)C1 Cc1ccc(C(C)C(O)C(=O)N2CC(CNC(=O)C(F)(F)CO)C2)cc1 C(CCC(=O)NC(C)(C)CN(C)C(C1CCOC1C)=O)=C(C)C c1(C(c2n(C)nnn2)NCC2(CCCO)CCCC2)c2ccccc2nn1C c1(CC)cc([N+](=O)[O-])ccc1N1CCC(NC(c2ccnn2C(C)C)=O)C(O)C1 c1(C(N2CCCC(CCOC)C2)C(=O)NCCC)cc(-n2cccn2)ccn1 Cc1csc2ncc(C(=O)NCC3(C)CN(C(c4cscn4)=O)CCO3)c(=O)n12 C1(C(=O)NCC(C)(C)NC(C=Cc2cnc(C)s2)=O)CCCN1S(=N)(=O)N(C)C c1(C2(NC(c3cccc(F)n3)c3n(CC(=C)C)nnn3)CC2)ccc(F)cc1 C1(CC(=O)NC2CC(SC)C2)CCCC1CNC(=O)CCNC(=O)C(C)(C)C CCC(CC)(CCNC(=O)CCCc1cnn[nH]1)NC(=O)Cc1ccc(O)cc1 Cc1cccnc1CC(=O)NC1(C)CCN(C(=O)CCc2ccoc2)C1 CC1(C)CC(C(=O)NCCc2ncc[nH]2)CN1C(C1CCSC1)=O C1(NC(C(c2cccnc2)NC(C(C=C=C)C)=O)=O)CC=C(C(C)C)CC1 C(=O)(CS(=O)(=O)CC1CCCO1)NC(CNC(C=CCN(C)CC)=O)C C(=O)(C(CO)C(C)(C)C)N1CC(CNC(c2c(CC)ccs2)=O)C(C)C1 CC1CCC(C(N2CC(CNC(c3c[nH]cc3C(C)(C)C)=O)C2)=O)S1 C1(C(=O)NCC(C)CN(C)C(c2c[nH]nc2C2CCC2)=O)CCn2cnnc2C1 Cc1cc(-c2noc(CCC(=O)OCC(=O)NC(c3ccccc3)=O)n2)ccc1F c1(C(=O)NCC(CNC(C(CCC)C)=O)F)ccc2nc(C(F)F)[nH]c2c1 c1(C(=O)NC2CCN(C(c3cc(C4CC4)on3)=O)CC2)cccn(CCF)c1=O c1(C(N2CC(NC(CCSCC)=O)C(O)C2)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1C C1(NC(COC(CC)C)=O)COC2(CCN(C(C3CN4CCN3CC4)=O)C2)C1 c1(C(=O)NC2CN(C(C(C)n3cccn3)=O)C2)cncc2nnn(C)c12 c1(C(=O)NCC2(CNC(CC=C)=O)CCC2)cc2cc(Br)cn2c(O)n1 CC1CN(C(=O)CCn2cccnc2=O)CCCN1C(c1c[nH]cc(F)c1=O)=O CC1C(NC(c2cnc(C3CC3)o2)=O)CC2CCC1N2C(=O)C1=NNC(=O)CC1 CCC(C)(C)CC(=O)NC1CC(C)(NC(c2ncc(N)cc2Cl)=O)C1 C1(N(C(=O)Cc2cccs2)C(C)Cl)CCCN(C(=O)C=CC(C)NC(C)C)C1 Cc1csc2nc(CC(N3CCC(O)(CCNC(=O)CC4(C)CCC4)C3)=O)cn12 c1(CN(C)C)cccc(C(=O)NCCN(C(=O)CCc2cnccn2)C2CC2)c1 C(c1ccc(Br)s1)=CC(=O)N(C(C)CNC(=O)C(C)OCC1CC1)C N1(C(C)=O)CCC(N(C(=O)CN(c2ccccc2)C(C)=O)CC2CCCO2)C1 Cc1ccc(NC(C2CC3CCC2N(C(c2ccns2)=O)C3)=O)cc1C#N c1(CCN2C(=O)NCC(OCCCl)C2=O)cccc2ccccc12 c1(CC)c(C(=O)NCCC2(C)CCN(C(C3C4CC5C(C4)C35)=O)C2)cnn1C C1(CC)CN(C(C23CC(CC)(CO2)C3)=O)CCN1C(=O)Cc1ccn(C)n1 c1(N(C)C)cc(S(=O)(=O)N2CCCC(C(C)(F)F)C2)ccc1C#N c1(C(N2CCC(CNC(C3N(C)CCC3)=O)CC2)=O)ccc(F)nc1F c1(CN2C(C(=O)NC(CC)C(=O)OC)CC3CC32)cccc2nccnc12 c1(CC(=O)NC2CN(C(C3(C)C(C)(C)C3)=O)CC2O)nc2ncccn2n1 c1(NC(c2cc(-c3ccc4ccccc4n3)cnc2Cl)=O)nnc2ccc(Cl)nn12 Cc1c(CN(C(=O)CCC2CC(NC(C3(Cl)CC3C(C)=O)=O)C2)C)cnn1C c1(C(N2C(C(CNC(c3cc(C)[nH]n3)=O)(C)C)CCC2)=O)nn(C)nc1C CC1CCN(C(c2ccc(N(C)C)nn2)=O)CC1NC(c1cncn1C)=O C1(NC(C(C)OCc2ccccc2)=O)CN(C(=O)CCCCC#N)C2CCCC12 C(=O)(C(C)(O)CC(F)F)NC(CNC(c1ccc(COC)c(F)c1)=O)C(C)(C)C C1(C(N2CCC2C(=O)NCC)=O)(NC(c2cnn(CC)n2)=O)CCOC1 CCC(O)C(C)C(=O)NCCN(CCCN(C)C)C(=O)Cc1ccc(Br)cc1 c1(NC(C2CC2C(N2CCS(=O)(=O)CC2)=O)=O)c(Br)cc(Cl)cc1[N+](=O)[O-] C(=O)(CC(C)CC(C)C)NCC1(O)CCN(C(CCC(C)OCC)=O)C1 C12(C(=O)NC3(CCCNC(CC(=C=C)C)=O)CC3)CCC(CC1)C2(C)C C1(CNC(Cc2ccc(C)cc2)=O)CC(C(C)C)CCN1C(C1CC1F)=O N1(C(=O)Nc2cc(C(=O)OCC)[nH]c2)CC(C)C(C)C1 c1(-c2n(CC[SH](C)(C)=O)ccn2)cc(-c2ccccc2)nn1CC(=O)O C1(CNC(C2CCCCS2)=O)CN(c2cc(Cl)c(O)nn2)CCC12CCOCC2 C1(CNC(C(C2CCOCC2)C)=O)C2CCC(C2)N1C(=O)C(N)=O c1(C(=O)NC2(CC=C)CCN(C(C3CCCN3C=O)=O)C2)ccc(F)c(OC)c1 C1(F)(CNC(C2(COC)CCC2)=O)CCCN(C(c2cnc(C3CCC3)s2)=O)C1 C#Cc1cncc(N(C2CCNCCC2C)C(c2ccncc2F)=O)c1 N1(C(CCc2c(C)n(C)nc2)=O)CCC2CCN(C(=O)C(C)N(C)C)CC2C1 N1(C(C)C)CCCN(C(=O)NCc2nc(C(C)C)nn2C)CC1 C1(C(=O)NCCN(C(=O)CC=CCc2ccccc2)C)(CO)CC1(F)F C12(NC(C(C)SC)=O)COC(C1)C(NC(=O)Cn1nnnc1-c1ccsc1)C2 c1(-c2ccc(C3C(C(=O)NCc4cnco4)C3)c(F)c2)ccc2c(c1)NCCO2 C12(C(N(CCNC(C3(C)CC(=C)C3)=O)CCC)=O)COCC1C2(F)F c1(C(=O)NC2CC3CCC2N(C(C2CCCSC2)=O)C3)coc2cc(F)ccc12 c1(C(N2CCC(C(C)(C)NC(c3ccncn3)=O)CC2)=O)c(F)ccc(F)c1Cl C(=O)(C(CN=C(NCC(F)F)N1CCC(C(C)C)C1)C(F)(F)F)OCC N(C(=NCC1CCCC1(F)F)NC1CCS(=O)(=O)C1)CC1(N(C)C)CCC1 Cc1ccc(CCCNC(=O)C(N)CCOCCO)cc1 CC(C)C1C(=O)NC2N1CCCC2.C1(C(N(C)C(=O)OC(C)(C)C)C)CCCO1 CC(CCOC(F)(F)F)C(=O)N(c1cnn(C)c1)Cc1ccccc1 N1(C(CC(C)OC)=O)CCC(NC(=O)Cn2cnccc2=O)CC1C C1(N(C(C2C(C=C)C2)=O)C)CCCN(C(c2cc(C)c(Cl)cn2)=O)CC1 C1(C(=O)NC(C2N(C(CC(C)C)=O)CCC2)C)COc2ccc(Cl)cc2C1 c1(C(=O)NC2CN(C(=O)C3CC3)C2)c(Cl)ccnc1Cl C(CCSC)(C(=O)NCC1CCN1C(c1ncccc1NC(C)=O)=O)OC C(=O)(CC(C)CCc1ccccc1)NCCC(CNC(C(C=C)(C)C)=O)O Cc1cnc(F)cc1C(N1CC(C(C)NC(c2cnc(CC(C)C)s2)=O)C1)=O N(C1CN(C(=O)C(N2C(=O)CCC2=O)C)CCc2ccccc21)C(C(F)=CC)=O c1(C(=O)NC(CN(C(=O)C(C)Cc2cccc(Cl)c2)CC)C)nc(C)c(C)s1 Cc1cc(Cl)ccc1OCC(=O)NCC1CN(C)CCN1C(C1CC1(C)C)=O C1(C(=O)NC(CCCC)CNC(c2cccc(C)c2)=O)CCc2nc(C)cn2C1 CC1(C)CCC(C(=O)N(CC(F)F)C2CCC2)CN1C(C1CC1C1CC1)=O Cc1c(Br)ccc(C(=O)NC(C(C)NC(=O)CCC(C)C)C(C)C)c1N C(C(=O)N1CC(CC(C)NC(C2C=CCC2)=O)C1)(C1CC1)SC c1(C(N2CC(NC(C3C(C)COCC3)=O)C2)=O)ccc2c(c1)CCC=C2 C#Cc1ccc(F)c(C(=O)NCC2CC2NC(c2cnoc2C(C)C)=O)c1 C=CCCC(C(=O)NOCCOC)NC(=O)CCCC C(C)(CCC(=O)N1CCC(NC(=O)Cn2nnc(-c3ccco3)n2)C1C)OC C(N=c1[nH]cnc(Cl)c1F)C1(C)CCCCN(C(=O)C2=CCCCC2)C1 N1(C(CCC(=C)Cl)=O)CCC(NC(=O)Cc2cc(C)sc2C)C12CC2 c1(C(=O)OCc2cccc3[nH]ccc23)ccc2cc(Br)ccc2c1 c1(C(C(=O)OCCN(C)C(=O)OC2C=CC(=O)N=N2)(C)C)cc(Br)ccc1F c1(C(N2CC(CO)C(CCC)C2)C(=O)NCC=C)ccc2c(c1)CCO2 C1(C(=O)NCC(C(C)C)NC(=O)CN2CCCCC2=O)CN(C)CCN1C CCC(C)C(C(=O)N(CCN(C)C)Cc1nc(CC(C)C)cs1)NC N1(C(C(S(CCC)(=O)=O)C)=O)CCc2sccc2C1CNC(C12CC(F)(C1)C2)=O C12(C(=O)NC3CC(CNC(C4CN(C(C)(C)C)C(=O)C4)=O)C3)CCCC(C1)OC2 c1(C(=O)NC2C(C)(C)N(c3ncnc(O)c3Br)CC2)cc2n(n1)CC(F)C2 C(=O)(C(CC)C(=O)N1CCC2C(NC(C3CCC3)=O)CC12)OCC CCCC(O)CC(=O)NCC1CCCC(CNC(=O)CNc2ccc(Cl)cn2)C1 C1(N(C)C(c2cc(O)ncn2)=O)CCN(C(=O)CCC2CCC2)CC12CC2 C1(NC(c2ccco2)=O)CCC2CN(C(=O)CC3CC4(CC4)C3)CCC2C1 N1(C(c2c(COC)cco2)=O)CCC2CCC(C1)N2c1ncncc1Br c1(CC)sccc1C(=O)NC(C)(CNC(=O)CN(C)CCOC)CC c1(CN(c2nc(=N)nc(N3CCCCCC3)[nH]2)C)ccc2c(c1)CCCC2 c1(C(N2CCC3(C(NC(CC(=C=C)C)=O)C3)CC2)=O)cc2c(C)c(F)ccc2[nH]1 N1(C(C(CCCC)C)=O)CCC2(CC1)CC(NC(=O)CCn1nc(C)nc1C)C2 C(=O)(CCC(C)SC)NCC(C)(Cn1cccn1)NC(CC1CC(OCC)C1)=O c1(CC(=O)OC)ccc(N(C2CC3CNC2C3)C(=O)Cc2cc(C)on2)c(F)c1 N1(CC(C)NC(=O)C(F)C2CC(NC(=O)CCCC3CC3)C2)CCOCC1 C1(C(N2C(CC(N3CC=CC3)=O)CCC2)=O)CCCC1(F)F C1(CC)CN(C)CCN1C(=O)Nc1ccccc1CCN1CCOCC1=O C(=O)(CC1=CCOCC1)N1CC(CCNC(c2ccc(C(F)F)cc2)=O)(OC)C1 C=CCC(C)(C)C(=O)NCCN(C(=O)C(F)CC)CCOC C(CCC(=O)N1CCC(CCCO)C1)N(C)C(C1(CSC2CC2)CCC1)=O c1(CCC(=O)NCC(CNC(c2c(C(C)C)nns2)=O)F)nc2ccccc2[nH]1 C(=O)(C(C)C(O)C(C)C)NC(C(=O)NCc1c(OC)nsc1)COC C1(OCC)CC2CN(C(C3C=CCN3C(=O)CN3C(=O)CNC3=O)=O)CC12 C12(NC(C=CC=CC)=O)CCC(CN(C(=O)C(C)(C)c3ccn(C)n3)C1)C2 C1(C)(CNC(c2c(OC)cncc2)=O)CN(C(=O)CCSC(F)(F)F)CC1C C1(CC(=O)OC(c2cn(C3CC3)nn2)C(c2ccccc2)=O)CCCCC1(F)F CCC(O)C(C)(C)C(=O)NCCCCC(CO)NC(=O)C=Cc1ccco1 CC1CCN(C(=O)C(=O)NC2CN(C(C3CCCC3(C)C)=O)C2)CC1 C1(C)(CNC(C=CCOC)=O)CCC(NC(c2cc(CSC)cnc2O)=O)CC1 CC1CC(C)CN1C(c1cnc(C2CCC2)[nH]1)C(=O)Nc1ccccc1 Cc1nn(-c2ccc(F)cc2)nc1C(=O)NCC12CC1CN(C(=O)CN(C)C)C2 N1(C(C#CC(=O)N(C)C)=O)CC2CC1CC2NC(=O)C=Cc1cc[nH]n1 c1(C(=O)NCCN(C(=O)C(C)NC(N)=O)CCC)cc2cncn2c(O)n1 N(C)(C1CCc2c(C)cccc21)C(c1cc(CC)on1)=O c1(NCCCCC(C)NC(C(C)=C(CC)C)=O)ncc([N+](=O)[O-])cc1C CN1CC(=O)N(CC(N2CCOC(CNC(C3CCCCC3O)=O)C2)=O)C1=O N1(CC)CC(C(=O)NC2CC(N(C(=O)C(=Cc3c[nH]cn3)F)C)C2)NC1=O c1(C(=O)OCC)cc(C)[nH]c(=NCCCNC(C)CC(=O)c2ccccc2)n1 c1(C(N2CCCC(NC(=O)CC3=CCCC3)C2)=O)cc(F)cc2nc[nH]c12 Cn1c(=O)ccn(CC(N2CCC(NC(c3ccc[nH]3)=O)C(O)C2)=O)c1=O C1(OC(F)F)CC(CNC2CNC(c3ccc(C)cc3)C2)C(OC)O1 c1(OC)ncc(Br)c(=NC(=O)c2ccc3c(c2)CN(C(=O)CN(C)C(C)C)C3)[nH]1 CC1CCN(CC(c2ccccc2)(C)O)C1(C)C C1(NC(C(c2n(C)ncc2)O)=O)CCCC(Nc2ccc(C(C)=O)cn2)C1 c1(C(=O)NC(C(C)C)(C)CNC(=O)Cc2ccco2)ccc2cnoc2c1 CC(C)C(Cc1ccccc1)C(=O)NCCCC1CCCN1CC(Cl)=CCl C1(OCCC)CCCN(c2nnc(C(C)C)n2CCO)C1.C1CCCO1 C(=O)(C#CC1CCOCC1)NC(CC)(C)CNC(c1nc(C)ccc1Br)=O Cc1cnn(C2CN(C(=O)CCN(C(=O)CC3CC=CC3)C)C2)c1 C(CC(=O)NCC1=CCCC1)(C1CC1)NC(C(c1ccn(C)n1)C)=O c1(CC)cc(C(N2CC(CNC(c3cscc3CC)=O)C3(CC3)C2)=O)c(C)nn1 c1(C(=O)NCCN(CC(C)O)C(C2CN3CCC2CC3)=O)cccc2ccsc12 C1(CNC(CCCC)=O)COC(C(F)(F)F)CN1C(=O)Cn1nnc(=O)[nH]1 N1(C(C(CC(C)C)C)=O)CCC2(CNC(C3(C(=O)N(C)C)CC3)=O)CCCC12 C#CCC(CC#C)C(=O)NC1CCOCC1NC(c1nnc(O)nc1O)=O c1(C(=O)OC)c(C)[nH]c(C(N2CC(O)(C(C)NC(=O)CN3CCC3C)C2)=O)c1C c1(C(=O)NCC2C3N(C(C4CC(OC)C4)=O)C(CC3)C2)ccc(=O)n2c1CCC2 c1(N2CCC(N(CC#C)C(c3c(C4CC4)cnn3C)=O)CC2)ncc(Br)c(O)n1 C#CCC(C)(C(=O)NCC(C1CCCC1)C)NC(=O)CC1(OC)CCC1 C1(CNC(C(CCSC)O)=O)CN(C(=O)COc2ccc(F)cn2)C(C)(C)C1 C1(O)(CNC(c2c(C(=O)OC)coc2)=O)CCCN(C(=O)CC(C)(C)O)C1 C1(N(C)C)CC2CC1CN2c1ccc(Cl)c(C(F)(F)F)n1 C1(C(=O)N(C(C)C(C)SC)C)(N(C(c2ccc(C)nc2)=O)C)CCC(C)(C)C1 C12(CNC(C3CCN(CCC)CC3)=O)CCC1CN(C(c1occ(C)c1C)=O)C2 c1(C(=O)NCC2(OC)CN(C(=O)CS(N)(=O)=O)C2)cc(F)c(F)c(F)c1F C(C(C(=O)N(C1(C(=O)N(C)C)CC1)C)NC(C1CCC1C(N)=O)=O)N(C)C Cc1nc(C)n(CC(=O)NCc2ncccc2CNC(=O)C=CBr)n1 C1(N(C(c2scnc2C(C)C)=O)CC)CCCN(C(=O)C=Cc2cnc[nH]2)CC1 CC(C)(CS(C)(=O)=O)C(=O)NC1CC(F)(F)CC1NC(C1CCC(O)CC1)=O C(=O)(CCCC(F)(F)F)N1CC(CCCCNC(C(C)OCC(C)C)=O)C1 Cc1c(CC(N2CCC(C)(CNC(C3CSCCS3)=O)C2)=O)oc2ccccc12 C1(NC(c2cc(OC)c(Br)nc2)=O)CC2CC1CN(C(=O)C(C)C(C)C)C2 C1(CNC(C(C2CCC2)OCC)=O)CC(C)CN(C(=O)C(CC)C(C)C)C1 c1(C(=O)NCC(C2CCCCC2)NC(CCOCC)=O)nccc2ccn(C)c12 c1(CC)cc(C)c(C(=O)NC2(C)CC(NC(=O)C(C)CC3CCCCC3)C2)o1 c1(C(N2CCOCC(F)(CNC(C(F)=CCC)=O)C2)=O)cccn2c(C)nnc12 c1(C(N2CCC(NC(C3CCC(C)(C)C3)=O)C2(C)C)=O)nsc2ccccc12 O=C(C(O)Cn1cncn1)NCCC1CCCN1C(=O)COc1ccccc1 c1(CN(C)C(C2CCC3(C2)N=N3)=O)cccc(CNC(C2CCN2C)=O)c1 N12CCC(C(C)(C)C1)C(=O)NC1(CCC1)C2=O.C1(OC(C)C)(CN(C)C)CCC1 Cc1ccc(Br)c(C(N2CCCCC2C(=O)N)=O)c1F.c1(CC)cc(Br)cc(F)c1F c1(C(=O)NCc2ccc(CC(=O)OC)cc2)cc(C)nc(C#N)c1 N1(Cc2nc(C)c(C)[nH]2)CC(NC(=O)C(C)(C)C)CCC1C c1(N2CC(CC)SCC2)nc(=NCC2CCOC(C)(C)C2)[nH]c2ncn(CC)c12 N1(c2n(Cc3ccc(Cl)cc3I)nnn2)CCCC12CCOC2 c1(C(=O)NC(C(C)C)CCN(C)C(c2ccns2)=O)ccc(F)c(S(C)(=O)=O)c1 Nc1cncc(C(N2CCNC(=O)C2)OCc2ccccc2)c1.c12cccc(c1)N2 c1(OC)cc(C)c(CN2CCOC(C(C)C)(CN(C)C)C2)cc1OC c1(C(=O)NC2CCN(C(=O)CC3CCC(O)C3)CC2)cncc([N+](=O)[O-])c1 c1(C(N(CC(O)CN(C)C(C2CC2[N+](=O)[O-])=O)C)=O)ncc[nH]c1=O C1(C)(C(=O)NCC(=O)NCC(=O)NCC(CCC)C)CCC(=O)C1 C1(CNC(C(CN(CC)CC)F)=O)C2CCCC1N(C(C1CSC1)=O)C2 C1(NC(=O)OC(C)(C)C)CCC(C(=O)NCC2CC(NS(=O)(=O)CCOC)C2)C1 C#CCCN=c1scc(-c2occc2C)n1CC1CCC(C(N)=O)O1 CC(C)C(CC(=O)NC1CC(CC(C)(C)C)C1)NC(c1cnn(C)n1)=O c1(CC)ccc(CCN(CCNC(CC2OCCN(CCOC)C2)=O)CC)c(F)c1 C1(CNC(C(C)N(C)C)=O)CCC12CCN(C(=O)Cn1cnc([N+](=O)[O-])n1)CC2 Cc1noc(C)c1C(=O)NC1CN(C(=O)CCN(C)C)C2CC12 C(C(C)NC(=O)CCNC(c1ccncc1)=O)(C(C)C)NC(CC=CC)=O c1(OC)ccc2c(C(=O)NCC3CC(NC(c4c(C)[nH][nH]c4=N)=O)C3)csc2c1 C1(CC#C)CN(C(C)=O)CCO1.C12(CNC(=O)OC)CN(C1)C2=O Cc1nc2nc(=S)[nH]n2c(C)c1CCC(=O)NC1CC1CNC(=O)C(F)(F)CO C1(C(=O)NC(C2CCCN2C(=O)Cc2sccc2Cl)C)C(C(F)(F)F)C1[N+](=O)[O-] c1(C(N2C(C)CC(CNC(=O)COC3COC3)C2)=O)cc2nn[nH]c2cc1F C(=O)(CCCCCCC(=O)NC(C(=O)OC1(C)CC1)c1ccsc1)OC C1(NC(c2cccc(C)c2)=O)CCN(C(=O)CC(C)N(C)C)CC1C CC(C)C(C(=O)N1CCC1C(=O)NCCOCCCF)NC=O C(=O)(C1Cc2ccccc21)NCCn1cc(C(=O)NC(c2c(C)n(C)nc2)C)nn1 C1(CC)CCCC(NC(c2cc(CNC(c3cc(C)c[nH]3)=O)nn2C)=O)C1 C(C1CN(C(=O)C=CC(C)(C)SC)CC1C(=O)NCc1cccc(CO)n1)=CC C1(C(C)C)C(=O)NCCN1Cc1nc(CN(C)C)no1 CCC(CC)C(=O)NCCCCNC(=O)CCc1cnn(-c2ccccc2)c1 C1(C(N2CCC(O)C2)=O)CC(F)(F)CN1Cc1cc(C(F)(F)F)cnc1Br Cc1n[nH]c(C)c1SCC(=O)NC1CCCN(C(=O)Cn2ncn(C)c2=O)C1 O=C(C1=CCCN(C(=O)CC2CC2)C1)NCCCc1ccc(Br)cc1 N1(C(n2cc(OC)nn2)=O)CCC(C(=O)NOCCN(C)C)C12CC2 C(=O)(C(CC(C)C)N(C)C)NC1C(NC(COCC(=O)NC)=O)CC1 C1(NC(c2ccc[n+]([O-])c2)=O)CCC2CC1CN2c1nnc(C(F)F)o1 c1(C(=O)NC2CCC(NC(CC3(OC)CCC3)=O)C2)cc2c([nH]1)CCC(C)C2 NC(=O)CC(O)C(=O)NCC12CC1CN(C(=O)CCCC(=O)NCC(F)(F)F)C2 CC(CCCNC(=O)CSC(F)F)NC(C1CCCSC1)=O C(=O)(C1=NOC(CNC(c2cnns2)=O)C1)N(c1cccc(F)c1)C C1(NC(=O)C=CCn2cncn2)CN(C(c2ccc(F)cn2)=O)C2CC12 N1(C(C2C(NCCOC)C2)=O)CCCC1(C)c1ccccc1 c1(C(=O)NCC(C)(CO)NC(C2CC2C#N)=O)cc(F)cc2nc[nH]c12 CCC(CC(C)C)C(=O)NC1CN(C(C23CC(C2)CS(=O)(=O)C3)=O)CC12CC2 C1(C(=O)NCCCN(C(C(C)SC)=O)C)C2CCC1(C)C2(C)C C(=O)(C1=C(C)CCOC1)N1CC(C=C)(CC(N2CCC(OC(C)=O)CC2)=O)C1 n1(CC)ncc(C(=O)NCCC(N2CCCC2CF)=O)c1C CCC(CC)CC(F)C(=O)N1CCCC1CCC(=O)NC1(CO)CC(O)C1 CC(C)CC(C)(O)C(=O)NCC1CC(C(N2CCC(O)(C(F)F)C2)=O)C1 N1(C(C2N(C(=O)OC)CCC2)=O)CC2CC(NC(=O)Cn3cnnn3)C1C2 C1(CC)CCN(C(c2cnc(O)o2)=O)C(C(=O)NCC=CBr)C1 N1(C(C(CCC)NC(=O)CC2CCCN2C)=O)CCOCC(C)(O)C1 c1(C(N(CC(C)NC(c2cnnn2C)=O)CC)=O)cccc(OCCF)c1 c1(C(C)O)ccc(NC(=O)NC2C3CN(C(=O)OC(C)(C)C)CC23)cc1 N1(C(C2(C)ON=C(C)C2)=O)CCC(C)(CNC(c2ccc(C)nc2N)=O)CC1 Cc1c(C(=O)N(C2CCN(C(=O)CC3OCCCC3(C)C)C2)C)cncc1N CCCCC(C)C(=O)N1CCCC(CN(C(=O)CN(CC(=O)NC(C)C)C)C)C1 C1(CCC)(NC(=O)C(CC)C2CC2)CCN(C(C2CN3CCN2CC3)=O)CC1 N1(C(C(C#C)(C)C)=O)CC(N=c2[nH]c3c(cc2C#N)CN(C)CC3)CC(C)(C)C1 C(C)(CN=c1cc(C)[nH]c(=NCCc2cnc(C)cn2)[nH]1)OCC=C N1(C(c2ccn(C)n2)=O)CC2CN(C(c3ncn(C(C)(C)C)n3)=O)CC2(C)C1 C1(C)(OC)CC(N(C)C(c2ccc(C(F)(F)F)cc2Br)=O)C1(C)C C1(CNC(Cc2ccc(CC)c(F)c2)=O)COC(C)(C)CN1C(c1cnn[nH]1)=O C#CC1(C(N2CCCCCC2)=O)CCN(C(c2cc(OC)cnn2)=O)C1 c1(C(=O)NC(C(=O)NCc2ncn(C)n2)Cc2cn[nH]c2)ccc(O)nn1 C1(C(N(C2CCN(C3CC3)C2)C)=O)CN(C(=O)C#CC2CCOC2)C2(CCC2)C1 c1(C(N2CC(O)(CNC(COCCOCC#C)=O)C2)=O)cc(F)cc2ccoc12 C(c1ccccc1Cl)=CC(N1C(CN(C(c2cc(CO)on2)=O)CC)CCC1)=O N1(C(c2snnc2C2CCC2)=O)CC2CCN(C(c3cc4n(n3)CCC4)=O)C2C1 C(c1cncnc1O)=CC(=O)NCC1(F)CCN(C(C2ON=C(C)C2)=O)C1 C1(C)(C(=O)N(CCCN(C(=O)CN(S(C)(=O)=O)C)CC)CC)CC=C(C)CC1 n1(CC)cc(Cl)c(C(=O)NCCCN(CCCNC(C2(O)CCOC2)=O)C)n1 CCC(C)(C(=O)NC1CCN(C(=O)COCc2nc[nH]n2)CCC1CO)C(F)F C1(C(=O)NCC(CCNC(=O)C=Cc2ccco2)O)CCOC(=O)CC1 N1(C(C(C)OC)=O)CC2CC(NC(=O)C=CCN3CCC3)C(C2)C1 c1(C(N2CC3C(NC(=O)C(C4CC4)N(C)C)C3C2)=O)ccc2c(c1O)CCCC2 Cc1cc(-c2nc(C(=O)NC3CCCN(C(=O)C(C)CN(C)C)C3)co2)ccn1 C(N=c1[nH]cc(Cl)c2nccnc12)C1C(N)CCC1 C1(NC(=O)CC2CCC(O)C2)CN(C(C23CCC(F)(CC2)C3)=O)C2CCCCC12 CCCC(C)(CC)C(=O)NC1CC(NC(=O)C(CO)C(C)(C)C)C1 N1(C(COC)=O)CCc2ccccc2C1CNC(=O)C(C)CC(F)F C1(CNC(C2(CC)CCC2)=O)CC(C)CN(C(c2ncoc2C(C)C)=O)C1 C=CCCCCC(=O)N1CCC(N(C(=O)C(CCOC)OC)CCC)CC1 C1(C(=O)NC2(C(=O)NCCN3CC(=O)NCC3)CC(F)(F)C2)CCC2(CCC2)C1 C1(NC(N2C(CN(C)C)CCC2)=O)CCN(c2cnn(C)c2)C1=O C(CCC(CO)NC(c1cnn(CCO)c1)=O)NC(C=CSC)=O N1(C(N(CCNC(C23CC(OC)C2C3)=O)C)=O)CCC(C(N)=O)CC1 c1(OC)nc(C)c(S(=O)(=O)N2CCCC(O)C2C)s1 c1(C(=O)NC(C2CCN(C(=O)Cn3cnnn3)CC2)C)cncc(CN(C)C)c1 c1(C(=O)NC(C2(O)CCCCC2)C(=O)NCCn2c(C)ncc2)cc(CO)n(C)n1 Cc1cc(C(=O)NC(C(C)NC(=O)CCc2ccn(C)n2)C(C)C)oc1C C(CC(C(C)(C)C)NC(c1cc(Cl)ccc1N)=O)N(C)C(c1cscc1F)=O C1(C)(CNC(c2c(C(C)C)c[nH]n2)=O)CCN(C(=O)CCc2cc(Cl)no2)CC1 c1(OC)c[nH]c(C(=O)NCC2CC2NC(c2cc(C)n(C)n2)=O)cc1=O Cc1nc(CC(N2CCC(C)(NC(C3CCCN3C(C)C)=O)C2)=O)[nH]c1C C1(NC(COCC(C)(C)C)=O)CN(C(=O)CC2CCCOC2)CC1CC(C)(C)C C(=O)(C(C)(C)C(F)(F)F)N1CCC(C)(CNC(c2c(C(C)C)ncs2)=O)C1 CC1(C(N2CCC(NC(C3(F)CC=CC3)=O)C(CO)C2)=O)CCCCCCC1 c1(OC)ccccc1C(N1CCC(C(=O)NC(C)C)C1)C(=O)NCCC#N CCCCC(C)C(=O)NC1(C)CC(NC(C2OCCO2)=O)C1 Cc1ccc(CC(=O)NCC(O)CNC(c2ncc(C(F)F)s2)=O)c(C)c1 N1(C(C2CCC(C3CC3)O2)=O)CCC12CC(CNC(=O)C(F)(F)F)C2 N1(C(C(C(CCC)NC(C=C(CCC)CCC)=O)O)=O)CCC2(COC(=O)N2)C1 O=[N+]([O-])c1cc(Br)cnc1CNc1cc(Cl)cc(Br)c1F c1(NC(C2C(C(=O)NCC(F)F)C2)=O)cnc2ccc(Br)cc2c1 N1(C(C2CC(C#C)(O)C2)=O)CCN(C(c2ccnc(COC)c2)=O)C(C)C1C c1(C(C(=O)NCC23CC(NC(CC4CC(C)(C)C4)=O)(C2)C3)O)ccc(Cl)cc1Cl C1(N(C(c2cc(CC)no2)=O)C)CC2CC1N(C(=O)Cc1cccc(OC)c1)C2 c1(OC)ccc(CC(N2CCC(NC(C3CCCN3C=O)=O)C2)=O)c(F)c1 c1(C(=O)NC2CN(C(C(CC)C#N)=O)CC(C)C2)c[nH]c2c(Cl)cccc12 C1(C(=O)NCc2scc(CNC(CN3CC(C)(C)C3)=O)n2)OCCC1(C)C c1(C(=O)NC(CNC(C(C)N(C(C)=O)C)=O)C(C)(C)C)ccc2nnn(C)c2n1 c1(C(=O)NCCC2N(C(Cc3cncc(C)c3)=O)CCC2)cc2sc(C)cc2[nH]1 C(=O)(C1CCCc2cccnc21)NC1CC2CN(C(CSCC#C)=O)C(C1)C2 c1(C(CC)C)nc(C)cc(=NC2CC(CNC(=O)C(C)NC(=O)NC)C2)[nH]1 c1(NC(C2C3CN(Cc4c(C#N)cc(F)cc4)CC32)=O)ccc2c(c1)CCC2=O c1(C(=O)NC(C2CCCN2C(=O)C(C)Cc2ccccc2)C)coc(CN(C)C)n1 CCCCC(O)C(=O)c1ccc(CN2CCCC(N)C2)cc1 C(CC(C)(C)C)(C(=O)NC(c1ccc(C)cc1)CNC(C1CS(=O)C1)=O)OC c1(NC(C2N(C(Cc3ccn(C)n3)=O)CCC2O)=O)ccc2c(c1)C(=O)NC2 CC1CCOCC1C(N1CC2CC2(CNC(=O)Cn2cnnc2O)C1)=O N1(C(=O)Cc2cccnc2)CCC2CN(C(=O)C=Cc3ncco3)C2C1 S(=O)(=O)(C1CCCCC1)N1CC(C)C(NCc2cc(F)c(OC(F)F)c(F)c2)C1 N1(C(c2cc(COC)no2)=O)CC2CC1CN(C(c1cncc(C)n1)=O)C2 CN1CCN(C(=O)CN2CCSCC2)CC1CNC(=O)CC1OCCCO1 Cc1ccccc1SCC(N1CCCC1(C)CNC(=O)C(=Cc1c[nH]cn1)F)=O CC(F)(F)C(C)(C)C(=O)NC1COCCC1C(N1CCCC(O)CC1)=O S(=O)(=O)(c1ccc(NC2CCSC(C)C2)nc1)N(CCCC=C)C CC(C)C(O)CC(=O)N1CCCC1CNC(c1cc(-c2cccc(F)c2)on1)=O N1(Cc2c(C)c(O)ccc2)CCc2[nH]nc(C(=O)Nc3cccc(I)c3)c2C1 C1(CN(C)C(c2cnn(C(C)(C)C)c2I)=O)CCCC12CCC2 C1(NC(=O)C(F)Cl)CCCCC12CN(C(C1CCCCO1)=O)CCO2 Cc1c(NCC2(CC(N)=O)CC2)ncnc1N1CCC(CCN(C)C)C1 CC(C)C(O)CCNC(=O)C(Cn1cccn1)NC(=O)CC1CC=CC1 Cc1cc(C(=O)NCC2CCN2C(=O)C(C)Cc2cnn(C)c2)oc1C c1(NC(C2C(O)CCN2C(c2ccc(O)cn2)=O)=O)cc([N+](=O)[O-])ccn1 c1(CCNC(=O)NCc2c(F)cncc2F)cc(C(F)(F)F)cc(C(F)(F)F)c1 c1(OCC)nccc(C(N2CC=CC2CNC(=O)CC2(OC)CC2)=O)c1F N1(C(c2c(C)ccc(O)c2)=O)CC2(CCN(C(=O)CCC3CCCN(C)C3)C2)C1 Cn1nc2c(c1COc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)CS(=O)(=O)CC2 C1(OC)CCCC1C(N1CC(C)C1C(NC[Si](C)(C)C)=O)=O N1(CCC)CCC2(CC1)CC2NC(=O)CCC(C)(F)F C1(C(=O)NC(CSCC)CO)CC=CC(NC(c2ccc(OC)nc2)=O)C1 C1(CC)CCN(C(=O)CC2CCCO2)C(C(N2CC3CCC2CC3)=O)C1 c1(CC)nc(C(=O)NCCNC(C2CN(C(C3CC4(CC4)C3)=O)C2)=O)cs1 N1(C(C(=O)NC(CN(C(C(F)OC)=O)C)(C)C)C)CCCCCC1 c1(C(=O)NCC(CC)NC(=O)C=C(Cl)Cl)ncccc1OC C(CCCC(=O)N(C1CCN(C)CC1)C)NC(C(CC1CCC1)OC)=O N1(C(C(c2ccoc2)N(c2cccnc2)C(C2CCC2)=O)=O)CCCC1CF c1(C(=O)NCC=CCNC(CCCc2ccc(C)s2)=O)c(C)ccc2nsnc12 C1(c2nnnn2CC2CCOCC2)(NC(C=C)C)CCC(C)(C)CC1C C1(C(=O)NCCCc2onc(C)n2)CCN(C(c2ncncc2N)=O)C1C(C)C Cc1cc(Cl)c(C(=O)NC2CC3C2CCN3C(C2CNC(=O)N2C)=O)cn1 C(C(C)(C)S(C)(=O)=O)c1nnc(N(CCOC(C)(C)C)C(=O)C2CC2)o1 O(NC(=O)CCC1CCCCN1C(=O)CCc1cnccn1)C(C(=O)OC)C C(C(=O)NCc1ccsc1C(=O)NCCC1CCC(C)CC1)(C(C)(C)C)OC N1(C(c2cnns2)=O)CCC2CC2(C(=O)Nc2cc(CO)cc(F)c2)CC1 N1(C(CCC(=C)Br)=O)CCC2(CCC(NC(C3(C)CCCS3)=O)CC2)C1 C1(NC(CCC2CC(NC(CC=CCC)=O)C2)=O)CCCC1(C)O N1(C(C2=CCC(NC(CC=CC)=O)C2)=O)CCC2(CCOC2=O)C1 C(C(O)C(CC)CC)NC(C1CCC(CNC(C2(C=C)CCC2)=O)CC1)=O C1(CNC(CCC(C)NC(CN2CCC(C)CC2)=O)=O)CCC(C)(C)CO1 CCCCCCCC(C(=O)NC(c1ccccc1)CC)N1CCC2CCCCC12 CC(C)CC(C)(C)C(=O)NC(C)C(C)NC(c1ccn(-c2ccncc2)n1)=O c1(C(=O)NCC(CNC(C(C2CCOCC2)OC)=O)O)cc2nc(C)ccc2o1 Cc1nc(C(N2CCC(NC(=O)Cn3ccccc3=O)CC2C)=O)c(C)n1C C1(NC(CCSCCC)=O)CCCC(N(C)C(c2nc(C3CC3)oc2C)=O)C1 N1(C(C(c2ccc(C)cc2)(C)C)=O)CC2CCCC(NC(C3CSC3)=O)C2C1 CC(C)CCC(O)C(=O)NC1CCC(N(C)C(c2ccc(OCF)cc2)=O)CC1 N1(C(CC)=O)CCCN(C(C2COCCN2C(=O)C(CSC)OC)=O)CC1 N1(C(C(C)(C2CC2)OC)=O)CCC=CC1C(N1CCCC(CC(N)=O)C1)=O C#CCC(C)(C(=O)NCC1(CO)CCN(C)C1)NC(c1cc(C)ncn1)=O c1(C(=O)NCCCN(C)C(C2NC(=O)CC2C(F)(F)F)=O)cn(C)nc1O c1(C(=O)NCC2CN(C(C(C)SC)=O)CC23CCC3)n[nH]c2cc(C)ccc12 C1(c2n(Cc3ccc(C)cc3)nnn2)(C(N)=O)CCN(C2CCCNC2=O)CC1 C1(NC(C=CCC)=O)CC2CN(C(c3ccc(C(F)F)o3)=O)CC12 C(C(O)(C1CC1)C1CC1)OCC(=O)C(C1(C(=O)OCC)CC1)=O c12ccc(cc1O)[nH]c2=O.C(C(C)(C)CS(C)(=O)=O)NC(C1C(OCC)C1)=O c1(CC(=O)NCC2C(NC(c3cc(CCC)ncc3)=O)C2)c(C)ncnc1C C1(C)(NC(C(C2CCC2)OCC)=O)CCN(C(=O)COCc2ccccn2)C1 N1(C(=O)CCC2CC(NC(C3(n4nccn4)CC3)=O)C2)CCOCC(CO)C1 C1(CCOC)(C(=O)NC(C)CC(C)NC(c2cc(C(C)=O)on2)=O)CCN(C)CC1 C1(N(C)C(c2cn(CCF)nn2)=O)CC2CC1N(C(=O)C(C1CC1)C1CC1)C2 C1(O)(CCNC(CN2CCC(C)(O)C2)=O)CCN(C(=O)C=CC2CCCO2)CC1 c1(-c2nc(CC)nn2C(c2ccc(Cl)cc2)C)ccc2c(c1)CCCS2(=O)=O C(=O)(CC(CNC(=O)CC1CCSC1)OC)NC1(CCOC)CC1 C(=O)(C(C)(C)CCC#N)N(C1CC(n2cc(C3(S(=O)(=O)N(C)C)CC3)nn2)C1)C CCC(C)(COC)CNC(c1ccc(C(F)(F)F)cn1)c1nnnn1C(C)(C)C N1(C(c2ncn(C)n2)=O)CC(NC(c2cc(O)n(C)n2)=O)C2CCCC12 c1(C(N(C2CCN(C(=O)CC3CCC3)C2)CC)=O)nccc(Br)c1O S(=O)(=O)(CC(=O)N1CCCC1C1CCN(C(C2CC(n3cnnc3)C2)=O)C1)NC c1(C(N2CCC3(NC(CN(CCC)C)=O)C(CC2)C3)=O)cc(O)cc([N+](=O)[O-])c1 CCCCCCCC(=O)N1CC2CN(Cc3cnn(CC)c3)C2C1 CC(C)(C)CC(O)CC(=O)NCCC1(C(=O)NC2CSC2)CCCC1 c1(SCC(=O)NCC2(NC(C=C(CCC)C)=O)CCC2)ccccc1O C1(C(=O)NCCC2CCN(C(c3n(CC)ccn3)=O)C2)CC2OC(C)(C)OC2C1 O(N1CCC(CC(N2CCC(CNC(=O)C3=CCCSC3)C(C)C2)=O)CC1)CC CC1CC(N(C)C(c2ncoc2CNC(C2CCCC2C2CC2)=O)=O)CC(C)O1 C(=O)(C1CCCc2ccccc21)N1CC(C2N(C(CS(N)(=O)=O)=O)CCC2)(O)C1 C1(CNC(CCCOC)=O)CCC2(CN(C(C3COC4(CCC4)C3)=O)C2)O1 C1(COCN(C(=O)C(C#N)=CC2CC2)C)CCn2cc(C(F)(F)F)nc2C1 C1(OC)CC(CCNC(=O)CCSC)N(C(=O)CCCOc2ccc(C)cc2)C1 C(=O)(N=c1ccn(CCF)[nH]1)N(CC[Si](C)(C)C)C(c1cc2c(s1)CCCC2)C c1(C(=O)NC(C(=O)N(CC#C)CC2CC2)CC2CC2)c(C)[nH]c(C)c1C c1(C(=O)NC2(C3N(C(C(C)n4cccn4)=O)CCCC3)CC2)cncc(Cl)c1Cl c1(NC(C)=O)ccc(F)c(C(N2CCC(NC(C3CCC3C(F)F)=O)C2)=O)c1 C=C(C)CCC(=O)NC1COCCC1NC(=O)C(O)c1ccco1 c1(C(=O)NCCC(C)N(C)C(c2ccc(OCCO)cc2)=O)ccc(C#N)[nH]1 Cc1ccc(C(=O)NCC23CC2CN(C(=O)CCC2CCOCC2)C3)c(F)c1Cl C1(C(=O)NC(C)Cc2ccncc2)C2CCCC2CN1C(C1OC2CCC1C2)=O N1(C(C2(COC)CCCO2)=O)CC(NC(=O)CSC2CCOCC2)CC(F)C1 N#Cc1cnc2c(F)cc(F)cc2c1N(CCNC(c1ncccc1F)=O)C1CC1 C1(CNC(c2cn(C)nn2)=O)CN(C(=O)C(C)(C)C2CCCO2)CCC1(F)F c1(OC)cc(O)ncc1C(N1CC2CCC1(CNC(=O)C(C)(C)F)C2)=O C1(C(=O)NCC(C2CC2)NC(c2ncccc2C(F)F)=O)CCC2CC1CO2 N12CCCC1(C(=O)NOC1N(C(CC)=O)CC=C1)C2=O.OC S(=O)(=O)(c1ccc(CN(C(C2CCC(C(=O)O)S2)=O)CCO)cc1)N1CCCC(C)C1 C1(NC(C2(CNC(=O)Cc3nonc3C)CC(=C)C2)=O)CCC(F)(F)C1 C1(C(=O)NC(c2cc[nH]n2)C)CCN(C(c2ccncc2F)=O)CC1O N1(C(C(=O)NCCC#N)C2CC2c2cccs2)CCCC1c1ccco1 N1(CC(N2CC(O)(C(C)NC(=O)CN(C)C3CC3)C2)=O)CCC(C)(O)C1 C1(NC(c2cnc(CNC(c3ccc(C(F)F)o3)=O)nc2)=O)C2CCCC1CC2 c1(C(=O)Nc2n(C)nc3c2CCCC3)cnc2c(c1)CCN(C(=O)C(C)(F)F)C2 N1(C(c2ccc(C)cc2Br)C)CCCC2C1CCN2Cc1c[nH]nc1C CN(C)S(=O)(=O)NCC(=O)NC1(CO)CN(C(c2ncc[nH]c2=O)=O)C1 C1(CNC(CNS(NC)(=O)=O)=O)CN(C(c2cc(N)ccn2)=O)CC(C)(C)C1 c1(N2CCC(N(C)CC)C2)nc2ccsc2c(=NCc2ccc(SC)o2)[nH]1 C1(C(N(CCCOCCNC(C(CC)c2cccnc2)=O)C)=O)CC2CCC1O2 C1(C(N(CCOCCNC(C(C(CC)C)=O)=O)C)=O)Cc2ccccc2C1 C1(C(N2CCC(C(=O)NCCc3cn(C)cn3)(CC)C2)=O)CCCC(=O)CC1 CCC(CC(=O)N1CCOCC1C(C)(C)C)NC(=O)CCc1cnn(C)c1C c1(CN2C(C(N3CC(C(=O)OC)C(O)CC3)=O)CCCC2)nc2ccccc2[nH]1 c1(CSC)cccnc1C(=O)NCC1(CCNC(c2cc(C)on2)=O)CC1 C(C(=O)N1CC(O)CO1)(c1ccccc1F)NC(C1C(C(=O)O)CCC1)=O Cc1c(C(=O)N(CC(C)NC(C2CCCS(=O)(=O)C2)=O)C)oc2ccccc12 C1(C)(NC(C(CC)NC(C2CCOC(C)(C)C2)=O)=O)CCC2(CC1)CC2 N1(C(CCSC)=O)CC2CC(NC(=O)C=CCn3cncn3)C(C2)C1 CC(C(C)(C)C)N(C)C(c1c[nH]nc1CCNC(=O)CCc1cnco1)=O C1(C(=O)NCCN(C(c2n(CC)ncc2C)=O)C2CC2)CCC2CC1CO2 N1(C(C(C)N(C(C)=O)C)=O)CCC(CCCNC(C2CC(C)C2)=O)CC1 c1(CNC(COC)(C)C)ccc(-n2nc(C)cc2C)nc1 C1(C(=O)Nc2c(OC)nc(Br)cc2)CN(Cc2cc(Cl)ccc2Br)CC(F)(F)C1 c1(SC)cccc(NC(N2CCC2(C)CNC(=O)CN2CC3CC3C2)=O)c1 C#CCCC(O)C(=O)NC1(C2CN(C(=O)CNC(=O)CCCCO)C2)CC1 O=C(C#CC1CCOCC1)NC1C2CC1N(C(=O)CCc1cnc(C3CC3)o1)C2 n1(-c2cn(CC)nc2)nc(-c2cc[nH]n2)nc1CCC1CC2CCC1C2 C=C=CC(C)C(=O)NC1(CCOC)CCN(C(C2(CCOC)CCCC2)=O)C1 N1(C(C2CN(C)C2)=O)CC2CC(NC(C3(C)CCOCC3)=O)C(C2)C1 N1(C(CCc2c(C)ncs2)=O)CCCC2C1CCCN2C(=O)CNC(N)=O Cc1cc(C)n2nc(C)c(C(N3CCC(CNC(=O)CC(C)C)C3)=O)c2n1 Cc1cc2sc(C(=O)NC3CC(NC(=O)CCc4ccoc4)C3)c(C)c2cc1C C1(OC)CN(C(c2ccc(Cl)o2)=O)CC1NC(C1CC1c1ccccc1F)=O C1(C(=O)NCC2CC(CC)C2)CN(C(=O)Cn2[nH]cnc2=N)CC1C N1(C(C2CN(c3nc(CCC)c(C)s3)C2)=O)C2CCC1CN(CC)C2 C1(C(N2C(C)CC(N3CCC3)C2)=O)Cc2ccccc2N1C c1(C(=O)NC2CCCC(C)C2)ccc(NC(C2CCN(C(N)=O)CC2)=O)c(O)c1 N1(CC(N2CCC(O)(C(C)CNC(C3CC(F)(F)C3)=O)C2)=O)CCP(C)(=O)CC1 c1(OC)cc(C(=O)NCC2CN(C(c3ccc(OC4CC4)cn3)=O)C2)ccc1Cl c12cn(nn1)C1CCC(C1)C(=O)N(CCCCO)CCC2.CC(=O)OCCO C(=O)(CC(CC1CC1)NC(c1ccc(CF)cc1)=O)N(CC(CC)(C)OC)C C#Cc1cc(F)ccc1CNC1CCCC(C(=O)Nc2ccc(Br)c(C)c2C)C1 CC1(C(N2CC(CCO)(NC(=O)C(=O)NCCO)C2)=O)CC2(CC2)C1 C1(=O)C(C(C)C)N1.N1(C2CC(N(C(=O)OC(C)(C)C)CC)C2)CCCCC1 C1(NC(CC2(N(C(C(CC)(CC)OC)=O)C)CC2)=O)CCCC(C2CC2)C1 Cc1ccc2oc(C(=O)NC3CCN(C(c4cn5cccnc5n4)=O)C3)cc2c1 Cc1cc(Cl)nc(NC(=O)CN2CCN(c3cnn(C)c3)S2(=O)=O)n1 C1(NC(c2ccc(CC)s2)=O)CC2(CCN(C(=O)CC3CC=CCC3)CC2)C1 C1(OC)CC(C(=O)NCc2nc(CNC(=O)C(O)C(C)C)cs2)CC1OC C(CC(C)C)(C(=O)NC(C)C(C)NC(=O)Cc1cc(C)cc(F)c1)NC(C)=O C(=O)(CCCN=[N+]=[N-])NC(C(C)C)C(=O)NCCCC(C)(C)CO c1(C(=O)NCC(CC=C)NC(=O)CS(=O)(=O)NC2CC2)cc2c(nn1)CCOC2 CC1(C)CCC(C(=O)NCc2nc(CNC(C3CC=CC3)=O)cs2)C1 C1(C(=O)NC2CCCC(NC(CN(S(C)(=O)=O)C)=O)C2)CSC2(C)CCC(=O)N12 C1(C)(NC(c2nc(CNC(C(CN(C)C)O)=O)oc2)=O)CCOC1=O CC1(C(=O)NCCC2CCCCC2)CC(O)CN1C(=O)C1=CCCCC1 N1(C(C=CC(=O)OCC)=O)CCC(NC(c2n[nH]c(C)c2Cl)=O)C12CC2 c1(C(=O)NCCCCCNC(C2CC(CC)(CC)C2)=O)ccnc(CO)c1 N1(C(c2ocnc2C(F)F)=O)CC2CN(C(C3CC4(CCC4)CO3)=O)CC2C1 N1(C(CC2N(C)CCOC2)=O)CC(NC(c2cccnc2O)=O)C2CCCC2C1 N1(C(C23N(C(c4nccc(COC)c4)=O)CCC2C3)=O)C2CCC1COC2 N1(C(=O)COC2CCC2)CCC2OCCN(C(=O)C=CCc3ccccc3)C2C1 n1(CC)ccc(C(=O)NC2CCCCC2CNC(=O)CC(=O)NC)cc1=O c1(C(=O)NC2C3(CC(NC(c4nn(C)c(CO)c4)=O)C3)C2)n[nH]c2c1CCCC2 c1(C(N2C(CC(=O)NC3CN(C)C(CO)C3)CC2)=O)c[nH]c2ccncc12 C1(O)(C(C)NC(=O)CCc2cnco2)CCN(C(c2ccc(C3CC3)cc2)=O)C1 N1(C(C(N)=O)=O)CC2(CC(CNC(=O)CCOc3cccc(Cl)c3)C2)C1 c1(NC(C(CCNC(C(c2ccccc2)C)=O)O)=O)ccc2cnccc2c1 N12CCC(CC1)N(CC)C(CC)C2=O.c12ocnc1C(=O)N1CC2C1.OC N1(C(c2c(C)nns2)=O)CC2CCC1CC2NC(c1cnn2cccc(Cl)c12)=O C1(O)(CNC(=O)C=CC=C(Cl)Cl)CCN(C(C2CC(O)C2)=O)C1 c1(NC(N2CC(c3cc(C)no3)C2)=O)ncn(C)c1C(F)(F)F N1(C(C2(Br)CC2)=O)CCCN(C(C2(Sc3ccccc3)CC2)=O)CCC1 c1(C(c2n(CCC(=O)OC)nnn2)NCC2(CC3CC3)CCC2)cc(C)c(Br)s1 n1(CC)cc(C(=O)C(N2CCCC2C2(NC(C3CCC(=O)N3)=O)CC2)=O)cn1 C1(CNc2cncc(C#N)n2)CCC2(CCOCC2)CO1 CC(C)CC(O)C(=O)N1CC2CCC2(CNC(=O)CSc2nncn2C)C1 c1(CC(=O)NCCNC(C2CCC(F)C2)=O)ccc(F)cn1 C1(F)(CNC(CCC)=O)CC(NC(c2scnc2Br)=O)C1 C=Cc1cccc(-c2cscc2C(=O)Nc2ncccc2Oc2ccccc2)c1 C1(C(N(C)Cc2cnn(C)c2)=O)COC2(CCCC2)C1 C(=O)(C1=CCCNCC1)Nc1ccc(N(C)C)c(C(F)(F)F)c1 C12(N(C(C(CC)N(C(=O)CN3CCSCC3)C(C)=O)=O)C)COC(C)(OC1)OC2 CCC1(C(=O)NC(C)CNC(c2nccnc2O)=O)CCCc2ccccc21 CC(=O)CCCCC(=O)NC1CCCCCN(C(c2ocnc2C)=O)C1 Cc1ncc2ccc(C(=O)NCC3C4CCC3CN(C(=O)CCC(N)=O)C4)cn12 N1(C(c2c(CC)cno2)=O)CCC(C)N(C(C2CCCC23CCC3)=O)CC1 C=CCCCC(=O)NC(C)(CSC)C(=O)N1CCC1(C)CCC Cc1cc(Br)cc(F)c1C(=O)NCCCCN(C(=O)Cc1ccno1)C C=CCCCC(C)NC(c1ccc(CNC(=O)C(C)(C)C2CCCO2)o1)=O CCCC(CNC(=O)C(CC1CCCC1)NC(C1CCC2(CC1)CC2)=O)CCC c1(OCCN(C(C(=O)NCC(c2cccnc2)C)=O)C)ccccc1Br C1(CC(=O)NC2CCN(CCC)C2)CCCN(C(=O)C=Cc2cscn2)C1 C1(C(=O)NCC(C)(C)NC(=O)C(O)C2CC2)CCc2nnc(-c3ccsc3)n2C1 N1(C(CC2(CSC)CC2)=O)CC(NC(=O)CSCCC(C)C)CC12CCCCC2 c1(C(=O)NCCC2(O)CCN(C(CCCN(C)C)=O)C2)cnn2c1OCC(F)C2 CCC(CC(C)C)C(=O)NCC1(C)CCCN(C(c2cccn3cnnc23)=O)C1 Cc1ccc(C(N2CCC(N(C)C(c3ccnc(CO)c3)=O)C(C)C2)=O)nc1C CC(C)(C)C(C(=O)NCC1CCCCCC1)NC(c1cc(O)cc(F)c1)=O c1(CC)cc(C)c(C(=O)NC2CCC(NC(=O)C(c3ccccc3F)O)CC2)o1 c1(NC(=O)NCC(C)CCCO)cccn(C2CC2)c1=O CC(C(=O)N1CCC(CNC(c2ccnc(OC(F)F)c2)=O)C1(C)C)S(N)(=O)=O CC(C)(C)C#CC(=O)N1CCN(C(c2ccncc2F)=O)C(CF)C1 Cc1cc(C)c(C(=O)NCC(C)(C2CCC2)NC(=O)CCC2CCCCO2)o1 CC1(C(N2CCN(C(=O)CCCCCF)C(C(F)F)C2)=O)CCCS1(=O)=O Cc1ccc(NC(C2CNCCN2Cc2csc3ccccc23)=O)c(C)c1Cl c1(-n2ncc(C(=O)NCC3(F)CC(NC(=O)CSC4CC4)C3)c2)cccc(F)c1 c1(-c2ccc(CN3CC(C)NC(=O)C3)c(F)c2)c[nH]c2ccccc12 C1(CNC(c2n[nH]c(C)c2F)=O)(NC(=O)CCCn2ccnc2)CCCCC1C C=CC(C)(C)CC(=O)NCCC(C)N(C(=O)CCCSC)C N1(C(C(C)=C2CC2)=O)CCC(NC(C2CCCN(CC(C)C)C2)=O)C(O)C1 N1(CCN(C(c2cccc(OCCC)c2)=O)C)c2ccccc2CC1C c1(C(C)C)cccc(C(N2CC(NC(=O)C(F)CC3CCC3)C(C)C2)=O)c1 c1(-c2cn(CC(c3ccc4c(c3)OCCO4)(C)C)nn2)cccc2c1CCCC2 N1(C(c2ccc(COC)o2)=O)CC(NC(c2ccnn2CCN(C)C)=O)C2CC12 CCC(Cc1ccccc1C)C(=O)N1CCC(N(C)Cc2cscc2Br)C1 N12CC(C3(C1)CN(C(=O)OC(C)(C)C)C3)CNC2=O.C1(OCC)CCC1CO C12(C(=O)NC3C(NC(C4CCOCC45CCC5)=O)C3)CCCN(CCC1)C2 C1(CNC(=O)CSCc2ccccn2)CCC(NC(=O)CC2CCOC2)CC1 CC#CCCC(=O)NCC1C2CN(C(=O)C(N)=O)CC12 N1(C(C2(CC)N(C(C3CC(CC)C3)=O)CCC2)=O)CCCC2COCC12 N1(C(COCCCN(C)C)=O)CCC(NC(C2CC3CC3C2)=O)C(CO)C1 c1(C(=O)NCC2C(NC(C(C)=C(CC)C)=O)CC2)ccc(OC)c(Cl)c1OC N1(C(CSCC#C)=O)CCCN(C(=O)C(C(C)C)N2CCC(C)CC2)CCC1 Cc1ccc(C(N2CCC(NC(=O)CC34CCCC3C4)C(C(N)=O)C2)=O)nc1C C(N=c1[nH]c2c(c(=NC(C)C)[nH]1)CCCC2)c1n(CCC)nnn1 c1(N2CC(CC)N(C)CC2)nc(NCC(c2ccccc2)F)c2ncsc2n1 CN1CCN(N2CCCC2(C)C2CCC(F)(F)CC2)CC12CCOC2 C1(NC(c2ccc(C(C)(F)F)nc2)=O)CCN(C(C2CC2F)=O)CC1F C1(CC(C)NC(c2ccc(C)o2)=O)CC2CCC(C1)N2C(=O)C(C)C1CCCC1 N1(C(c2c(C)onc2)=O)CCOCC1CN(C(=O)CC1CCC2CC12)C CCC(C)(C)CC(=O)NCC1C=CCN1C(=O)Cc1ccnn1C C(=O)(CN=S(C)(C)=O)NCC(c1ccc(N(C)C)cc1)NC(Cc1c(C)n[nH]c1)=O c1(N2CCCC(C)(C)C2)ncccc1S(=O)(=O)NC1CCC(F)CC1 N1(C(C(C(CC)C)O)=O)CCC(C2CCCN(C(=O)C3=CCC3)C2)CC1 Cc1c(Br)c(C(N2CCC(O)C(C(=O)N(C)CC3CCC3)C2)=O)nn1C c1(C(=O)NCc2n(C)ncc2CO)cc(OC(F)F)ncc1-c1cnn(C2CC2)c1 Cn1nc(C2CCN(C(=O)NCC3CCCOC3c3ccccc3)CC2)cc1N C(=O)(CC(C)CC)N1CC(OCCNC(CCSCC)=O)C1 c1(CC(=O)N(CC(O)CNC(=O)COC2CC2)C)c(F)cccc1Br C1(O)(CN(C(=O)CO)C)CCCN(C(=O)CC2CC(O)C23CCC3)C1 N1(C(c2n(CCOC)ncc2)=O)CCC2CN(C(=O)CS(=O)(=O)CC)CCC2C1 N1(C(c2nc(CCC)oc2)=O)CCC(C(F)(F)F)C(CNC(=O)C(C)(F)F)C1 c1(C(C(N2CCC(C(C)C)C2)=O)N)cccc(I)c1 C1CCC(C2CCN(C(=NCc3ccnn3CC3CCOC3)NC3CC3)C2)CC1 C=CCC(CNC(C1(CNC(=O)COC2CCOC2)CCCC1)=O)CC(C)C C1(C(=O)NCC=CCNC(C(C)=CC)=O)CC(C(F)(F)F)CO1 c1(C(=O)NCC2N(C(C(C)CC(F)F)=O)CC2)ccc2cnccc2c1 C1(N(C(C(CCC)NC(=O)NC)=O)c2c(C)csc2C)CCC12CCNCC2 C(CC(=O)NCC1CC2(CCC2)C1)(C(F)F)NC(C(C)N(CC)CC)=O C=Cn1nccc1C(=O)NCC1CCCN1C(c1ccnc(OC2CC2)c1)=O c1(CN(C(c2csc(Br)n2)C(=O)Nc2c(SC)cccc2)C)ccc(C#N)cc1 n1(CC(=O)N(C2CC3CCC2C3)CC(=O)OC)cc(I)c(-c2nn[nH]n2)n1 CCCCC(C)CCC(=O)NC12CCC(CNC(=O)CC(=O)OC)(C1)OC2 Cc1cc(C(=O)NCC(O)CN(C(=O)C(C)(C)CO)C)ncc1C(N)=O c1(OCCC)ccc(C(=O)NC2(CNC(c3cn(C(F)F)c(C)n3)=O)CC2)cc1 CCC(C(=O)NCCCCCN(C)C(c1cnoc1C(C)C)=O)C(C)C c1(NC(c2c(-n3ncc(C)c3)cncn2)=O)ccc(N2CCOCC2)cc1F C1(CCCC)CN(C(=O)C(CC)CCC)CCN1C(c1cc(C)c(C)cn1)=O O=C(C(F)CC1CCCC1)NC1CCN(C(=O)C(F)C2CCOC2)C1 C(=O)(C(=O)C(C)(C)C)NC1(C(=O)NCC(CCC)(C)O)CCOCC1 c1(C(N2C(C(C(=O)OC)C)CCC2)=O)cc(C=O)ccc1F c1(C(=O)NC2C(CC)CN(C(=O)C=CC(=O)OCC)CC2)c(C)cc(C)cc1N c1(C(=O)Nc2cc(C)c(C(F)(F)F)nc2)cccc(Cl)c1N=[N+]=[N-] C1(C(N(CCCCC)C)=O)C=CCN(C(=O)C(F)C(=O)OCC)C1 C(C(CC1CCCC1)C(=O)N1CCC(CC(F)F)C1)NC(CSC)=O CCC(C)CC(C(=O)NCC1(CC(=O)OC)CC1)NC(c1sccc1C)=O C12(NC(c3ccc(NC)cc3)=O)CCC1CN(C(c1ccc(CCF)cc1)=O)C2 c1(C(NNC(=O)Cc2cc[nH]n2)=O)cc2ccc(F)cc2nc1O N1(C(c2c(CC)csc2)=O)CC(CNC(c2coc(C(C)C)n2)=O)CC1(C)C C1(CCNC(CCc2c(C)ncs2)=O)CN(C(=O)CC23CCC(CC2)C3)CCO1 N1(C(C(CCOC)C)=O)CCN(C(c2cnn(CC(F)(F)F)c2N)=O)C(CF)C1 C(=O)(CCCCC(C)(C)C)NC1(CCNC(c2cc(C(CC)C)c(C)o2)=O)CC1 c1(N2C(CNC(C(C3CCC(=O)N3)C)=O)C(C)CC2)nc2ccccc2s1 N1(C(CCSCC(C)C)=O)CCC2(CC1)COCC(CNC(=O)C(O)CN(C)C)O2 Cc1cc(Br)cnc1C(=O)NC(CO)C(C)NC(C1(NC(N)=O)CC1)=O C12(C(c3ccccc3)NC(=O)OC(C)(C)C)CC(C(=O)O)(C1)C2 C(c1ccc([N+](=O)[O-])s1)=CC(N1C(CCNC(CSCC#C)=O)CCCC1)=O CC1CN(C(=O)CSc2cnn(C)c2)CC(C)C1NC(=O)CC1(O)CCC1 N1(C(C(N2CCC(CC(C)O)CC2)=O)=O)CC(=O)NC2CCCC2(C)C1 c1(C(N2C(CNC(CC(=C=C)C)=O)C(C)CC2)=O)ccnc2cc(OC)ccc12 C=C1CCN(C(=O)CCOCC2CC2)C(C(=O)NC(CC2CC2)COC)C1 c1(Oc2ccc(C(C)NC(C(C=C)(F)F)=O)cc2)ccc(Cl)c(Cl)c1 C1(C(=O)NCC2CC(COC)C2)CC(F)CCN1C(=O)CC(O)CN(C)C C(=O)(CCCC(F)(F)F)N1C2C(NC(C(C3CC3)OCC)=O)C(C2)C1 C1(n2c(-c3ccc(-c4cnn(C)c4)o3)nc(C(C)OCC)n2)CCCS(=O)(=O)C1 N1(C(Cc2ccc(C)c(O)c2)=O)CC2C=CC1C(C(=O)NCc1nc(=O)o[nH]1)C2 c1(C(N2CC(OC)(CNC(=O)CCCC3CC3C)C2)=O)cc(C)cc(C#N)c1 CC1OC2CCC1(C(N1C(C(=O)N(CC(C)(C)N(C)C)C)CC3CC13)=O)C2 N1(C(=O)C=CC2CCCC2)CC2(CCC2)CC1CNC(C12COC(CCO1)C2)=O c1(N(C(C2CCCCC2CC)C(=O)NCC=C)C)ccc(C#N)c(C)n1 C1(CNC(=O)COCC(F)(F)F)CC2CCC1N2C(C1CC2CCC1CC2)=O C1(C(=O)NCC2(Nc3nc(OCC)c(Cl)cn3)COC2)CCC2(C1)CC2(F)F Cc1oc(C2CC2)nc1C(N1CC(CNC(=O)C=Cc2ccc(Cl)s2)C(C)C1)=O CN1CCCC(CN(C)Cc2cccc(C(=O)NCCCN3CCCC3=O)c2)C1 N1(C(c2c(SC)ccc(Br)c2)=O)CCCCC12CCCNC2 c1(CC)nn(C)c(NCC(C2CC2)N(C)C(c2ccc(Br)o2)=O)c1[N+](=O)[O-] C(=O)(CCC#Cc1ccccc1)N1CCN(CC(C)NC(CSCC)=O)CC1 Cc1nnc2c(C(=O)NC3(CN(C)C(C4CCCNS4(=O)=O)=O)CC3)nccn12 c1(NC(=O)C=CCNC(C2CC23CCC3)=O)ccc2c(c1)CCO2 C1(NC(C2CNC(=O)N2)=O)(CO)CCN(C(c2ccc(C(F)(F)F)[nH]2)=O)C1 c1(C(N2CCCC(O)(CNC(C(C)C(F)F)=O)C2)=O)nc2ccccc2nc1O C(=O)(C1=CC2C=CC1C2)NC(C(CC)C)C(=O)N1CC2CC1CN2CC N#Cc1ccc(CCC(N2CCOCC2CCNC(C2C=CCC2)=O)=O)c(F)c1 CC1(C)CCN(C(=O)C=Cc2ccco2)C1CNC(=O)CCc1ccncn1 c1(C(=O)NCC2OCCN(Cc3ccc(CC)s3)C2)cc(C)c(Cl)cc1OC c1(C(N2CCC(CNC(C(CC)SC)=O)CC2)=O)nnc2c(F)cccc2c1O Cc1nc(C)c(CNC(=O)CCN(C(=O)CNC=O)CCO)[nH]1 N=c1ccc(C(N2CC(O)(CNC(=O)CC(O)c3ccccc3)C2)=O)n[nH]1 C#CCCCCC(=O)N1CCOC(CN(C)C(c2cccc(F)c2)=O)C1 CC(CC(=O)NCC(C1CCC1)NC(=O)CCc1cc[nH]n1)C(F)F Cc1nc(C(=O)NCCC2CCN(C(C3CCN3C3CCCC3)=O)C2)c(C)n1C N1(C(c2c(OC)c[nH]n2)=O)CCC(C(C)(C)CNC(=O)CCc2cn[nH]c2)CC1 c1(C(=O)NCC2(NC(C3C=C(C)CS3)=O)CCCCC2C)ccc2c(c1)NCC2 C1(CCO)CCCCC1N=c1ccnc(N(C2CC2)CC2(CO)CCCCO2)[nH]1 C1(C(=O)NCC(C)(C2CC2)OC)CC(C(=O)O)C12CCOCC2 c1(CC(=O)NCCN(CC(C)C)C2CC2)cncs1 N1(C(C(COC)O)=O)CC2(CCCC(CNC(c3cnc(C(C)(C)C)[nH]3)=O)O2)C1 n1(CCC=C)nc(-c2ccco2)nc1-c1ccc(OC(F)F)cn1 c1(C(N2C3C(NC(c4c(C)c[nH]n4)=O)CC(CC3)C2)=O)cn2cccc(F)c2n1 C1(NC(C2CCN(OC)CC2)=O)CC1C1CCCN(C(c2ccc(O)nn2)=O)C1 C=CC(C)(CC)C(=O)N(CC(C)NC(c1cc(-c2ccncc2)[nH]n1)=O)C c1(NCCCOCC=C)[nH]c(=NCC(C2CC2)C2CC2)nc2c1cnn2C CCCS(=O)(=O)CC(=O)NC1CCN(C(C2CCN2CC)=O)CC(O)C1 Cc1cccc(OCCCCC(=O)NC2CCCC(CNC(=O)C=CCO)C2)c1 C1(C(=O)NCC(C)CNC(=O)CNC(C2CCCC2)=O)(OC)CCCOC1 c1(CCC)occc1C(=O)NC(C)(C)CN(C(=O)C(C)C1CCCO1)C c1(C(=O)NCC(CC)NC(c2ccc(COC)o2)=O)ccn2ccsc12 c1(C(CC(=O)NCCCN(C(=O)CC2(C)CC2(F)F)C)C)c[nH]c2ccccc12 c1(OC23C(F)(F)C2CCC3)ncc(Cl)cc1Cl c1(C(=O)NCC(CC)NC(c2ccnc(C)n2)=O)csc2cc(OC)ccc12 O(NC(=O)C(O)C1CCCN1C(C1CCC(=O)N1CC)=O)CCC=C N1(C(C2CC=CCO2)=O)CCC(C2CCCCN2C(=O)Cn2cncn2)CC1 CCC(CCOC)C(=O)NCCC1(C(N2CCC2C(=O)N(C)C)=O)CCC1 S(=O)(=O)(c1c[nH]c(C(=O)NC(C)CN(C)C(C2(C(C)(C)O)CCC2)=O)c1)NC CC(C)C(N=[N+]=[N-])C(=O)NCC1CCC(C)N(C(=O)C(F)C(F)(F)F)C1 N1(C(c2c(CC)nn[nH]2)=O)CCCN(C(=O)CC(C)O)C(CO)C1 N1(C(C#CC2(CC)COC2)=O)CCCC2(C1)CN(C(=O)C=CS(C)(=O)=O)CCO2 c1(OC)cnc(Br)cc1C(c1nnnn1C1(C)CC1)NC1CCCNC1=O c1(OC)ccc(C(=O)NC2CN(C(C3(C(=O)O)CCCOC3)=O)CC2F)cc1 C1(NC(c2c(N)c(Cl)ncc2)=O)CC2CCC1N(C(=O)Cc1ccccc1O)C2 CN1CC(C(=O)NCC#CC(=O)NC2CC3CCC(C2)C3)CCC1=O C1(C(=O)NCc2cccc(C3(F)CNC3)c2)CCCC12OCCO2 C(c1cncnc1O)=CC(=O)NC(CNC(C(=Cc1ccccc1)OC)=O)CO N1(C(c2c(C)con2)=O)CCN(C)CC1CNC(c1cccc(N)c1O)=O N1(C(CCc2cnc(C)o2)=O)CCC=CC1C(=O)NCC(C1CC1)C1CC1 c1(C(N2CC(C(=O)NCCCC(C)O)CC2(C)C)=O)c[nH]c2ccncc12 c1(OC)cnnc(C(N2CC3CC2C3C(=O)NCc2csc(C)c2C)=O)c1 C1(NC(C(C)CN(C)C)=O)CN(C(C2(c3cccnc3)CC2)=O)CC(C)(C)C1 C1(C(N(C2CCN(C3CC3)C2)C)=O)CCN(C(=O)CC2CCSC2)C1 c1(C(=O)NCC(C2CC2)NC(c2nc(C)oc2)=O)cc2n(n1)CCCC2O c1(-c2[nH]c(=N)sc2)cccc(CN2CCC(=CC(=O)OC(C)(C)C)CC2)c1 C=C(C)CC(=O)NC(C)CC1CN(C(=O)C(N2CCSCC2)C)C1 N1(C(C2CCCC(NC(c3ccccc3)=O)CC2)=O)CC2CC(O)CC2C1 C(C1(C)OCCc2sccc21)NC(c1cc(C)cc(OC)c1O)=O CCCC(CC)CCC(=O)NC(C1CCN(C2CC2)C1)C(=O)OC.C1(C2SO2)CC12CCC2 Cc1c(NC(C2(C)CCN2S(=O)(=O)c2ccc(O)cc2)=O)ccc(C#N)c1F c1(CN2C(C(C)C)CN(C(c3cnsn3)=O)CC2)ccc(O)c2ccccc12 C1(NC(c2cc(CCO)on2)=O)CCCC(NC(c2scnc2C(F)(F)F)=O)C1 Cc1cc(CN(C(=O)C=C(Cl)CCN(C)C)Cc2ccco2)cnc1F N1(C(CC(C=C)CC)=O)CC2CCC(C1)N2C(=O)CCCCCF C1(CCC)CCCN(C(C2CCN(C(C3(N(C)C)CC3)=O)CC2)=O)C1 c1(C(=O)NC2CC(NC(C3CCC4CC34)=O)CC2O)cc2n(n1)CCCC2 C1(CC(N2CCCC(N(CCF)C(C3CC(F)(F)C3)=O)C2)=O)CN2CCC1CC2 C#CCC(CC#C)C(=O)NC1CC(C)CN(C(=O)Cc2nocc2C(C)C)C1 Cc1ccc(O)cc1NC(C1(C)CCN1C(c1c(I)ccnc1Cl)=O)=O Cc1ocnc1C(=O)N(CC(=O)O)Cc1cn(Cc2cccs2)nn1 Cc1ccc(C=CC(N2CC(O)CC2c2ccc(Br)cc2)=O)cc1 c1(NC(C(C)Oc2cccc(C(C)=O)c2)=O)cc(F)c(O)c(Cl)c1 CC1(C(=O)NCC23CCC2CN(C(=O)CCC2CCCO2)C3)CCC(=O)NC1 c1(OC)cc(C)cc(C(=O)NCC2CN(C(=O)CNC(=O)CCC3CC3)C2)c1O C(=O)(C1=CCCC1(C)C)N1CC(C(C)C)N(C(=O)C(F)C2CCC2)CC1 C12(CNC(CCCOCC)=O)CCC(CC1)N2C(C1CC1c1ccccn1)=O C12(NC(Cc3ccc(OC)c(O)c3)=O)CCCC1CN(C(=O)CN1CC(C)C1)C2 C1(NC(CN(C(COC)=O)C)=O)CC(F)CN(C(C2(C)CCC(=O)NC2)=O)C1 C(=O)(C(C)(C)CC(F)(F)F)N1CC(NC(C2(C)CCOC2)=O)CC(C)(C)C1 C(CCCC(=O)NCC1CCCCN1C(=O)CCCN(C)C(C)=O)OC Cc1nc(-c2ccc(COC(C)C)cc2)n(CCC(=O)NC2CCC2)n1 N1(CCNC(CN(C(C)=O)C)=O)CCCN(C(C2CC2C2(C)COC2)=O)CC1 N1(C(C2CC(C)C2)=O)CCC=CC1C(=O)Nc1ccc(N2CCCC2)cc1 c1(NC(CCCSC)=O)ccc(NC(=O)CCCc2ncco2)cc1C Cc1c(C(=O)NC2(CNC(c3ccc(=N)[nH]c3)=O)CC2)cnn1CC(F)F C(=O)(CS(=O)(=O)C(C)(C)C)N1CC(CCNC(c2ccn(C)n2)=O)S(=O)(=O)CC1 N1(C(c2ccc(CO)cc2)=O)CC(CO)C2(C1)CN(C(C1CC3(CC3)C1)=O)C2 C(C(Cc1ccccc1)N=c1[nH]c2c(c(=NCC3CC(F)C3)[nH]1)CCCC2)OC C1(NC(c2coc(-c3ccccc3Cl)n2)=O)CC2CC1N(C(c1csnn1)=O)C2 c1(CC)nc(C)cc(=NC2CC3CN(C(=O)C(C)COC)CC23)[nH]1 c1(C(N2CC(C)(C)C(NC(=O)C(O)C3CCC3)C2)=O)cc(F)cc(N)c1N c1(CC)ccc(C)c(NC(=O)C(CN=[N+]=[N-])NC(c2n[nH]c(C)c2O)=O)c1 CCC(C)(COC)C(=O)NC1CC(F)CN(C(c2cc(C)ncn2)=O)C1 N1(C(C(CC)SC)=O)CC(CNC(=O)C(=O)NCC2CC2)C2(CCC2)C1 C1(NC(c2[nH]cc(C)c2)=O)CC(NC(c2occc2C2CC2)=O)C(O)C1 c1(C(=O)NC(CNC(CNC(=O)OC)=O)CO)cccc(-n2cccn2)n1 N1(C(Cc2c(C)con2)=O)CCN2CCN(C(=O)C=Cc3cn(C)nn3)CC2C1 C1(NC(C(c2cccc(F)c2)(C)C)=O)CCCC12CN(C(C1C=CCC1)=O)C2 c1(C(=O)NCCC2CC(C(=O)NC(CC=C)C)C2)cc(CO)ccn1 c1(-n2ccc(C(=O)NCC(C)NC(=O)C(C)CC3CCCC3)n2)ccc(F)cc1 C1(C(NOSC)=O)CN(C(=O)CC(C)(C)C(C)=O)CC1C1CC1.C1CCCCCCN1 C#Cc1cccc(C(=O)NCC2CN(C(=O)CC3OCCC3C)C2)c1F C(CCC(O)C(=O)N(C1CC2CCC1O2)C)NC(c1n[nH]c(C)c1Cl)=O C(=O)(CC(C)C(F)(F)F)N1CCC(C(N(C(C)CC2CC2)C)=O)(CF)C1 C1(CC=C)(C(=O)NCC23CC2CN(C(=O)Cc2ccn(C)n2)C3)CCOCC1 N1(C(C(CC)=CCCC)=O)CCN(C(=O)CC(C)(C)CCOC)CC(C)(F)C1 CC1C(NC(C2CN3CCN2CC3)=O)CC2CCC1N2C(=O)C1=COCCC1 C1(NC(c2nccc(C(N)=O)c2)=O)CN(C(c2cc3sccc3s2)=O)CCC1F Cc1cc(C(=O)NCC(C)CC(=O)NCCC2COCC2O)n(C)n1 CC1C(C(=O)NCC(=O)NCc2csnn2)CCN1C CCC(C)CCCCC(=O)N1CC2CC1CN(C(=O)CC1CC=CC1)C2 N1(C(CCCC)=O)CC(NC(=O)Cc2ccc(OC)cn2)CC12CCOC2 CC1CN(C(C2CC2C(C)(F)F)=O)CC1(C)CNC(c1ncccc1N)=O C1(NC(c2cnc(SC)[nH]2)=O)CC(NC(c2ccnc(O)c2)=O)C12CCC2 C1(NC(CCC(C)SC)=O)CN(C(c2cccc(Cl)c2F)=O)CC2CCCC12 Cc1cnc(NC(C(C)C)C2CC2)c(S(=O)(=O)NCc2cc(C(F)F)no2)c1 c1(C(=O)NCC)cccc(-c2cnc(Nc3c(C)ccnc3Cl)s2)c1F c1(N(CC(=C)C)C)nc2cc(Cl)c(S(=O)(=O)N3CCCC(C#N)C3)cc2s1 Cc1cccc(NC(=O)NCCOc2ccccc2C(=O)N(C)C)c1 C1(C(N(C2CCN(C(c3cnoc3CC)=O)C2)CCC)=O)CC(=O)N(C2CC2)C1 c1(C(=O)NCCC2(NC(CCc3cnc(C)s3)=O)CCC2)ccc2nncn2c1 c1(C(CNC(C2(CO)CCOC2)=O)NC(C=C(CCC)C)=O)ccc(OC)cc1 C1(C(N(C(CC)C)CC)=O)C2CCC(C2)N1C(=O)C(C)NC(=O)C1CC1 N1(C(C(C)OCC)=O)CCN(C(c2csc(C(F)F)n2)=O)CC1CS(C)(=O)=O C1(C(N(CCCNC(COCCCCCC)=O)C)=O)CCCC(SCC)C1 c1(C(N2CCC(NC(C(C)(C3CCOCC3)OC)=O)C2)=O)c(C)cc(=O)oc1C Cc1nc(O)nc(O)c1CCC(N1CC(NC(c2cnco2)=O)C(O)C1)=O N1(C(=O)CCC2CC2(Cl)Cl)CCCCC1C1(NC(=O)CC2(O)CCOC2)CC1 c1(C(=O)NC2C3(NC(C4CC(CC)C4)=O)CCC(C2)C3)ccc(S(C)(=O)=O)s1 C1(C(=O)NCCN(C)C(c2cncn2C2CC2)=O)OC(C)(C)OC1(C)C CC(C)CC(C)CC(=O)N1CCC=C(C(=O)N2CCOCC(C)(C)C2)C1 C(=O)(CCCC(=O)N(CC(C)CNC(=O)CCc1ccncc1)C)N(CC)CC C(=O)(C(C(C)CC(C)C)N1CC2CCC2(C)C1)Nc1c(C)cc(F)cc1 c1(C(=O)NC2CCC(C(=O)NC3CCCOC3)OC2)cccc([N+](=O)[O-])c1Br N1(C(CCC=CC(C)C)=O)CCCC(CNC(c2cc(F)cnc2O)=O)CC1 C12(CNC(c3ccncc3)C3CCC3)COCC(C1)C2 c1(C(N(C2CCN(C(CCC(=C)Cl)=O)CC2C)C)=O)ccc(OC)c(Cl)c1F N1(C(C=NOC)=O)CC2CCCCC2(C(=O)Nc2cc(Cl)ccc2OC(C)C)C1 N1(C(C2(NC(c3c(C)occ3)=O)CCSC2)=O)CCc2nnnn2CC1 Cc1nc(=NCC2C3CN(C(=O)CCOCC4CCCO4)CC23)[nH]cc1[N+](=O)[O-] c1(NC(C)=O)ccc(NCC2CNC(=O)C2)cc1F C1(NC(CC=C(C)C)=O)CCC(NC(c2ccnn2C(F)F)=O)CC1 N1(C(CNC(CNC(C)=O)=O)=O)CCC2(CCCC2NC(=O)CCC(C)(C)C)C1 C12(CNC(CN3C(C)CCC3C)=O)CCC(CN(C(=O)CCC(N)=O)C1)C2 N1(C(c2c(C)ccc(C)c2O)=O)CC(C)CN(C(=O)C#CC(C)C)C(C)C1 C(=O)(C(F)(CN1CCCC(CNC(C)=O)CC1)C(=O)OC)OCC C1(C(=O)NCCC(=C)CNC(=O)CCC)CCc2cnn(C)c2C1 c1(C(N2C3C(C(N4C(C#N)CCCC4)=O)C(C3)C2)=O)ccc2sncc2c1 C(=O)(C(C)(C)CO)N1CC(CCO)(NC(C=C(C)C(C)(C)C)=O)C1 C1(C(=O)NCC(C)CC2CCCC2)(CC)CN(C(=O)Cc2nocc2C)C1 N1(C(c2c(CC)ncs2)=O)CCC2(CC2)CC1C(=O)N(C)CC1(C)CCCC1 Cc1nc2c(o1)CCCC2CC(=O)NCC1C=CCN1C(=O)C1CC1 C1(C(=O)NC(C)Cn2cnnc2)CC(N=[N+]=[N-])CN1C(=O)CCn1cncn1 C(C(C)(C)C(=O)NC1CN(C(C2CC23CCC3)=O)CC1c1cnn(C)c1)N(C)C c1(CC(N2C(C3CCN(C(CC=CC)=O)C3)CCCC2)=O)cnn2c1CCCC2 C(c1cccc(F)c1)=CCC(=O)NC1CN(C(=O)CSC2CC2)CC12CC2 Cc1cc(C(N2CCC(CO)(NC(C3CCC=CCC3)=O)C2)=O)nnc1C C1(C(=O)NC2CCN(C(CCC)=O)CC2O)OC2CCCCC2C1C c1(C(N(CC(CNC(CCN(CCC)C)=O)O)C)=O)nc(Cl)c(Cl)s1 O=C1CCC(C(=O)NC2CCCCC2CNC(C2(C3CCC3)CC2)=O)=NN1 c1(N(C(c2c(C(C)C)occ2)=O)C(C)C)cccc(C(N)=O)c1 c1(NC(C2CCN(C(C(c3ccnn3C)C)=O)CC2)=O)cccc(C#N)c1 c1(OC)cccc(C(N2CCC(C)(C(=O)NC(CO)C(C)O)C2)=O)c1F c1(N(C)CCO)ccc(S(=O)(=O)NCc2ccc(C(C)(F)F)cc2)cc1F C(CC(=O)C(C)(C)C)c1cn(C(C(=O)N(C(CCCC)C)CCO)C)nn1 C1(C(N(C(C=C)C)C)=O)CC(NC(=O)Cn2ccnc2C)C1(C)C c1(C(C(=O)NCCOCC)N(C)CC2CCOC2)ccnn1CC(F)F c1(C(N2CC(N(C)C(C3CCCS3)=O)C2)=O)ccc2c[nH]nc2n1 S(=O)(=O)(c1ccc(NCC2CCCCCC2)c(Br)c1)NC(CC(=C)C)CO N1(C(C(CC=CCC)C)=O)CCC2CN(C(C3CC3C(F)(F)F)=O)C(C)C12 C(=O)(C1=NOC(c2ccccc2)C1)N(CC(C)NC(c1ccc(COC)o1)=O)C C(CCCCC(=O)NC1CC2CC1N(C(=O)C(C)N=[N+]=[N-])C2)OC CCCC(C(=O)N(CCNC(c1cccn1C)=O)CC)c1cccc(Cl)c1 c1(CC)c(C(=O)NCC(C(C)C)NC(C2CC(S(C)(=O)=O)C2)=O)cccc1F C12(COC)COC(C(=O)NCc3ccccc3SC(F)(F)F)(C1)C2 O=C1CCC(CC(N2CCC(F)(c3cccc(Br)c3)C2)=O)C(=O)N1 c1(C(N2CC(C(C(=O)N(CCCCCO)C)OC)C2)=O)cccc(C)c1F Cc1cccc(C(N2CC(C(N3CCCCC3CF)=O)C(C)C2)=O)n1 Cc1ncc(N)cc1C(N1CC2CC1CN2C(c1ncoc1C1CCCO1)=O)=O C(=O)(CC(C)(C)CC(F)(F)F)N1CC(O)(CN(C(=O)CCn2ccc(=N)[nH]2)C)C1 C1(C(N(CCCC)CCO)=O)(NC(=O)Cc2cn[nH]c2)CCSC1 C1(C(=O)NCC(C)NC(C2(CC=C)CC2)=O)CCC2C(C1)C2(F)F C12(NC(C(=O)NC(C)C)=O)COC(C1)C(NC(C1CC1(Cl)Cl)=O)C2 N1(C(=O)CCc2ccncn2)CCCC2(CNC(=O)C(F)(F)C(F)F)CCCC12 N1(C(c2c(C)c(C#N)ccc2)=O)CCC2CCN(C(=O)C(O)C(C)C)C2C1 Cc1[nH]c(C#N)cc1C(N1CCN(C(=O)CC(C)c2cccnc2)CC1)=O N1(C(C(CCC)CC)=O)CCC2(CCCN2C(c2cc(C)c(C)nn2)=O)C1 Cc1c(C(=O)NCC2CN(C(=O)C(F)C(C)C)CC2(C)C)sc2cncn12 N1(C(c2c(C)cnnc2)=O)CCC(NC(C2CC(N(C)C)C2)=O)C(O)C1 c1(C(=O)NC)nc(O)nc(O)c1OC(C)C.c12ccc(cc1)CNC2=O c1(CC)cccc(CC(=O)NCC(c2n[nH]c(C)n2)(C)C)c1 N1(C(C(C)(C)SC)=O)CC2CCCC2(CNC(=O)CCc2ccccc2C#N)C1 CC1(CNC(C2CCC3(CC2)CC3)=O)CCCN(C(=O)COC(F)(F)F)C1 c1(C(=O)NCCC(C)NC(=O)C=Cc2ccc(Cl)s2)ccn2ccnc2n1 c1(C(=O)NCC(C(C)C)NC(C2(CCOC)CC2)=O)ccc(N)c(C(F)(F)F)c1 C1(C(=O)OC)C(O)CCN1C(=O)C(F)C1CC(NC(=O)CC2CCCC3CC23)C1 C(CC(C)C)(C(=O)Nc1ccccn1)Oc1ccc(C)nc1 C(CO)(C(=O)NC(C1CCCN1C(c1cn(CCO)nn1)=O)C)NC(C(C)C)=O C1(C(=O)NC2CCC(C(C)C)CC2)CC2(CC2)CN1C(=O)CN1CCCCC1C C(C(C(=O)NNC(N)=S)Cn1cncn1)c1n(C)c(-c2ccccc2)nn1 N1(C(CC(C)(C)N(C)C(=O)NC2CCOCC2(C)C)=O)CC(O)CC1(C)CO c1(SC)c(C(=O)NC2CN(C(=O)CCCc3nncn3C)CC2C)cccc1F C1(CSC)(O)CCCC1.C1(C(=O)NC)CCC1C.C12CC1CN(C)C2=O CC12CN(C(=O)CCN3CCOCC3)CC1CN(C(C1CC13CCSCC3)=O)C2 C(CCC(=O)NCC(C)NC(c1[nH]nnc1-c1ccccc1)=O)OC(C)C CCC(CC)(CO)C(=O)N(C1CCN(C(c2cn(CCO)nn2)=O)CC1)C C(=O)(CS(=O)(=O)C(C)C)NC(C1CCN(C(c2c(C#N)cnn2C)=O)CC1)C c1(C(=O)NCCC2CCN(C(c3[nH]n(C)c(=O)n3)=O)CC2)ccc(F)c(CO)c1 C(C)(C(=O)N(CCCO)OC)N(C(c1c(CCC)con1)=O)CC c1(OC)ccc2ncccc2c1C(=O)NCC1CC1CNC(c1csc(O)n1)=O C1(C(N2CC(C(C)NC(=O)C(C)(C)N3CCCCC3)C2)=O)CCN(CCF)CC1 C(CCC(N)=O)(C(=O)NC1CN(C(C2CC2F)=O)CC1F)NC(=O)OC(C)(C)C C(=O)(C(CC)CC)NC(CNC(CC=CCC)=O)C(C)C c1(C(=O)NC2(CCNC(CNS(CC)(=O)=O)=O)CC2)ccc2c(c1)nc(C)n2C c1(CC(=O)NC(CNC(C2CC(C)(O)C2)=O)CO)cc(C(F)(F)F)c(O)nn1 C(c1ccc(F)cc1)=C(C)C(=O)NC1(CCNC(=O)CSC(F)(F)F)CC1 C(=O)(C1=CCCOC1)NCC(C)(CNC(C1CC(C)(C)CO1)=O)OC CCC1=C(C(=O)OC(C)(C)C)C(c2ccc([Si](C)(C)C)o2)NC(=S)N1CC(C)C C(C)(CC(=O)N1CCC(CCNC(C2CC(C)(C)C2)=O)C1)(C1CCC1)N(C)C C12COCCN(C1)C(=O)NC2.C1(CC=C)(Sc2ccccc2)CCCN1 CP(C)(=O)C(O)C(=O)NCCc1ocnc1CNC(C1C=CCC1)=O c1(C(=O)NC(CNC(C(=O)NCCCCCCCC)=O)C)cc(C)c(O)c(N)c1 C(CCC1CCC1)(C(=O)NCCOC(c1ccccc1)=O)N1CCC(OCC=C)C1 N1(C(C=C(C)CNC(C2C=CCS2)=O)=O)CC(N(C)CCO)C1 c1(C(C(=O)N(CCC#N)C)NC(C(C)OCC(C)C)=O)cccc(C(F)(F)F)c1 C12(c3nnc(N4CC(C)C(C)C4)n3CC(N3CCCCC3)C3CC3)CCC(CC1)CO2 c1(OC)cccc(CC(N2CC(NC(=O)CC3CCC(=O)C3)CC2C)=O)c1 C1(CN(C(C(=O)OC)C)C)CCCC2CCCN12.c1(C2C(=O)N2)cc(SC)cs1 C1(CCNC(CCn2c(C)ncc2)=O)C(C)CCCN1C(=O)CC(C)(C)F N1(C(C2C(CCC)C2)=O)CC(CNC(C2(c3cncnc3)CCCC2)=O)C(C)C1 CC1(C)CCC=C(C(=O)N2CC(n3cc(COc4ccc(O)cc4)nn3)C2)C1 c1(NC(C2CCCN2C(c2cc(I)ccc2F)=O)=O)cc(Cl)ccc1O c1(CC#N)cccc(C(=O)NCC(O)CNC(=O)CSc2nnc(S)s2)c1 C1(CNC(c2n(C)ccc2)=O)CC2(CC2)CN1C(c1cccn(C)c1=O)=O CCC(O)C(C)(C)C(=O)NC(CNC(c1ccc(=O)n(C)n1)=O)C(C)C CC(C)(CN=c1[nH]c(=NCC2CCCC(F)(F)C2)[nH]c2c1CCC2)CC(F)(F)F c1(CC(=O)NC2C(NC(Cc3cc(C)sc3)=O)CCC2)nc(F)c(F)cc1F c1(OC)cccc(C(=O)NC(CNC(C2CC2c2cnc[nH]2)=O)C2CCC2)c1 C1(C(=O)N(c2cccc(OC(F)(F)F)c2)Cc2cscn2)CC(=O)C1C1CCC1 C(c1cc(Cl)ccc1Br)=CC(=O)Nc1ccc(OC)c(-n2cnnn2)c1 CN1CC2CC1(CN(C(=O)C(Cl)Cl)C1CCCC1)C2 CC1(NC(C2C3COCC23)=O)CN(C(=O)C(C)(F)c2ccccc2)C1 c1(C(=O)NC)ccc(CC(=O)NCCCN(CCCNC(=O)CS(=O)CC)C)cc1 C1(NC(CCC(C)OC)=O)CC2CCC1C(NC(=O)C1=CCSC1)C2 c1(C(=O)NCC(C2CCOC2)NC(C2(COC)CC2)=O)cnc2sc(C)nc2c1 C1(CCOC)(C(=O)NC(C)(C)CNC(C2CN(C(=O)OC)C2)=O)CCCC1 N1(C(C(CCC)CC)=O)CCCC2(CCN(C(C34CC(CSC)(CO3)C4)=O)C2)C1 c12ccc(cc1)C(=O)N(CC)C2.C1(C(=O)O)CCC(CCc2noc(C)n2)CC1 N1(C(Cc2ccc(OCC)cc2)=O)CCN(C(c2cnsc2C)=O)C2CC12 N1(C(C=C(CC)C)=O)CC2OCCN(C(c3oc(C(=O)OC)cc3C)=O)C2C1 c1(C(N2CCCN(C(c3c(C)cncc3)=O)CC2)=O)ccc(F)c2cccnc12 C1(C(=O)NC2CCCN(C(C=C3CCC(C)CC3)=O)C2)CCc2ncccc2C1 Nc1cc(C(N2CC3CC2CN3C(C2CCc3nccn3C2)=O)=O)cc(F)c1O c1(C(=O)NC(CCNC(c2cc(OC)nc(F)c2)=O)C)ccc2nc(O)sc2c1 C=CCCCC(C(=O)NC(C)CCCO)NC(=O)C=Cc1ccncn1 c1(C(=O)NCC2(COC)CCCN2C(c2csc(Cl)c2)=O)ccc([N+](=O)[O-])[nH]1 N1(C(CCc2c(C)ncs2)=O)CCC2CC(C1)CN(C(C1C(C)C1(F)F)=O)C2 C1(NC(CCn2c(C)csc2=O)=O)C2CC1CN(C(C1(O)CCC1)=O)C2 N1(C(C2CC=C(C)CC2)=O)CCCC(CC(N2CC(F)(F)CC2C)=O)CC1 C(=O)(C1CCc2cccnc21)N1C(CN(C(C(CCCCC)CC)=O)C)CCC1 Cc1ccc(Cl)c(C(N2CC(CNC(c3onc(Br)c3C)=O)C2)=O)c1O c1(CC(=O)NCCCC2CCCN2C(c2ccncc2)=O)ccnc(F)c1 c1(C(=O)NC(C2N(C(c3c(CC)n(C)nc3)=O)CCC2)C)cc(S(N)(=O)=O)cs1 C(=O)(CCS(=O)(=O)c1ccccc1Cl)N1CCC(C)C1c1cn(C(C)CO)nn1 C1(F)(CNC(=O)CC2CC2)CC(NC(=O)CCOC2CCOC2)C1 C(=O)(C#CC1CCCC1)N1CCC(NC(c2cc(CC(C)C)on2)=O)C1C N1(C(c2ccc(C(=O)OC)n2C)=O)CCCCCC1CNC(=O)C=CC1CCC1 O=C(N=c1cc[nH]c2cccnc12)N1CCC2(CCCOC2)C1 C1(CCNC(=O)COC2CC(F)(F)C2)CCCN(C(=O)CSc2nncs2)C1 C1(CC=C)(C(=O)NCCC2CC2C2CC2)CCN(C(=O)CC=CC)C1 c1(OC)ccccc1C(C(N)=O)NC(=O)CCC(=O)c1ccc(Cl)s1 [N-]=[N+]=NC1CN(C(c2cccc3ccnn23)=O)CC1NC(C1CC1F)=O c1(C(=O)NCCCOCCNC(C2C(C)C2C)=O)csc(CS(C)(=O)=O)n1 c1(CC(=O)NCC2CCCCC2NC(=O)CCc2cnco2)cc(F)ccc1O c1(COCC)ccc(N)c(C(=O)NCC=CCNC(=O)C(C)CC2CCCO2)c1 C1(CNC(c2c(C)coc2C)=O)CC2(CCC2)CN1C(=O)C=CC1CCOCC1 C(=O)(CC(O)C(=O)N1CCN(C(C2CCCS2)=O)CC1C1CCC1)OC(C)(C)C N1(CC(=O)NC23CC(Nc4ncc(C(=O)OC)s4)(C2)C3)C(=O)CSC1=S N1(C(CC=C)=O)CCN(C(=O)CCCC(C)=O)C(C2CC2)C1 c1(C(=O)NC(C)CCNC(c2cc3c(s2)CCC3)=O)cccn2[nH]c(=N)nc12 c1(C(=O)NC(CC=C)CNC(c2ccc(C#N)cc2)=O)nc2cnccc2s1 C1(C(=O)NCC(COC)C(C)C)C2CCCC2CN1C(=O)C=C(C)C(F)F C=C(C)CCCC(=O)N1CCC(NC(=O)CC(C)F)C1(C)C C1(N(C(CC(=C)C)=O)C)CCC(NC(c2cn(C)c(C(F)F)n2)=O)CC1 C1(CNC(c2c(C)noc2)=O)(CO)CCN(C(c2cc(C3CC3)cs2)=O)CC1 c1(C(=O)NC2C(CC)CN(C(=O)CSC(C)(C)C)CC2)cc2nccnc2[nH]1 CC(C)C(C(=O)NCC1CCC(NC(C2C=CCC2)=O)CC1)C1CCC1 C12(CCC)CN(CCSc3ccc(Br)cc3C)CC(CO)(C1)C2 C1(NC(C(OC)OC)=O)CCC(CNC(C23CC(C(F)F)(C2)C3)=O)CC1 c1(C(N2CC(NC(CN(C3CCC3)C)=O)C(O)C2)=O)n[nH]c2c1CCC(C)(C)C2 C(C1=CCN(C(C2CCCO2)=O)CC1)NC(c1ccccc1F)=O c1(C(N2CC3CN(Cc4cccc(C)c4)C3C2)=O)cnc2[nH]ncc2c1 N1(C(Cc2cc(C)[nH]n2)=O)CC2(C1)SCCC2NC(C1CCn2nnnc2C1)=O c1(NC(C2C=CCN2)=O)cccc2c1C1CN(C(=O)CC3CCC3)CC1O2 c1(SCC)cnc(O)c(C(=O)NC2COCC2NC(=O)Cc2ccc(O)cn2)c1 c1(NCc2cc(OC)cc(OC)c2)ccc2c(c1)CCCC(=O)N2 N1(C(Cc2cc(COC)no2)=O)CC2CC1CCC2NC(=O)CCc1ncc[nH]1 C1(NC(C2CN(CC)C(=O)C2)=O)CC2CC(C1)N(C(c1cc(O)cs1)=O)C2 C1(C(=O)NC2CC(CNC(c3c(OC)cc(C)cn3)=O)C2)CN2CCN1CC2C C1(NC(c2ccnc3ncsc23)=O)CN(C(C2CC2(F)F)=O)CC2(CC2)C1 CN1CCn2nc(C(N3CCC(CC(C)(C)NC(=O)CC4CC4)CC3)=O)cc2C1 C12(C(N3CC(O)(CCNC(CC4CC(CC)C4)=O)C3)=O)CC1Cc1c[nH]nc12 C1(C(=O)NC(C(C)=O)(C)Cc2ccccc2)C2Cc3cc(Br)ccc3C12 C1(C(=O)NCC2C(NC(CCC3C(C)C3)=O)CCCC2)CCCC12OCCO2 c1(C(=O)OC)cccc(C=C2CCN(CCC(CO)CO)CC2)c1 C1(CNC(c2cnc(SC)nc2O)=O)CC2(CO1)CN(C(C1(C)CC1(F)Cl)=O)C2 C1(C(N(C2CCOC2)C)=O)C=CCN(C(C2CCN2C(C)(C)C)=O)C1 N1(C(c2ccc(CN(C)C)o2)=O)CCC(NC(c2cn(C)c(O)n2)=O)C(C)(C)C1 N1(C(C(C=C)(F)F)=O)CCCC(N(C)C(c2ccn(C)c2C2CCC2)=O)CC1 C#CCC(C)C(=O)N1CCCC(N2CC(NC(=O)NC(C)(C)C)CC2=O)C1 c1(NC(C2C(CNCc3cc(OC)ncc3)C2)=O)cc(C#N)cn1C(C)C C1(N(C(CCN(CCC)C)=O)CCC)CCN(C(=O)CC2CCC2OC)C1 c1(C(N2C(C(C)C)C(NC(=O)C(C3CCOCC3)F)CC2)=O)cc(N)ccc1O C(=O)(C(O)(C(F)(F)F)C1CC1)NC(C)CNC(c1cccnc1S)=O C(C(C)C(C)C(=O)NC1CC(C)(NC(C2(CCN(C)C)CC2)=O)C1)OC N1(C(c2c(OCC)ccc(Cl)n2)=O)CC(NC(=O)CC(F)F)C2(CCOCC2)C1 C1(NC(Cc2nc(NC=O)sc2)=O)C2CCN(C(=O)C=CSc3ccccc3)C12 c1(C(N2C(C(CNC(COCC#C)=O)(C)C)CCC2)=O)ccc(C(F)F)c(F)c1 c1(CC)ncccc1C(=O)NCC1C(C)CCN1C(=O)CCSc1nnnn1C C12(CNC(c3ccc(Cl)s3)=O)CCC1CCN2C(c1csnn1)=O c1(C(=O)NC2C(NC(=O)CCN3C(=O)CCC3=O)CC2)cc2c([nH]1)CCOC2 Cc1noc(C)c1CC(=O)NCC1COCC1NC(=O)C(C(C)C)NC(N)=O C(=O)(C(C)CCCC)N1CCC(N(C(=O)CCF)CC#C)CC1 c1(C(=O)NCC2CN(C(CC=CC=C)=O)C3(C2)CCC3)cnc(O)c2cncn12 C(=O)(C(C)(C)c1cnn(C)c1)N(CC(C)NC(C1C(C(=O)OC)CC1)=O)C N1(C(C2C(C)(C)C2c2ccccc2)=O)CCCC(CNC(C23CC(C2)C3)=O)CC1 N1(C(CC2(COC)CCCC2)=O)CCC(C(C)(C)NC(=O)CN2CCC2C)CC1 Cc1c[nH]nc1C(N1CC(C)(NC(=O)C(C)N(CC(F)(F)F)C)C1)=O Cc1c(C(=O)NCC2CCN2C(C2CCCCC(=O)C2)=O)cnc2nncn12 CC1CC=C(C(=O)NCC2(NC(=O)C(CO)N(C)C)CCCCC2)CC1 C1(C2CCN(C(=O)CSc3n[nH]c(O)n3)CC2)(Nc2snc(SC)n2)CCC1 C1(NC(C=CC(=O)OC)=O)CCN(C(=O)CCC2(C)CC2)CC1C C(CC)(C(=O)NC1(C(=O)NCCSCC(C)C)CSC1)=CCCC C1(CNC(=O)COC(F)F)CCN(C(C23CCCC2OCC3)=O)CC1(F)F C1(CC(=O)NC2C(C(=O)OC)CC2)CCCN(C(=O)CN2CC(C)(C)C2)CC1 c1(C(=O)NCC2(F)CCN(C(CC3ON=C(C)C3)=O)C2)cc2cccc(C)c2s1 C1(C(=O)NCC2(C(=O)NCc3cc[nH]n3)CCC2)CC2CCC(C1)O2 CC1CN(C(=O)CSCc2cccnc2)CCC1NC(=O)Cn1cnc(C#N)n1 N1(C(c2cc(Cl)ns2)=O)CCC2CN(C(c3cc(CO)ccc3Cl)=O)C2C1 C(C(CC1CCCC1)C(=O)NCC(CO)N(C)C)NC(C1(CCC)CC(=O)C1)=O C1(C(=O)NC2CC(NC(=O)C(c3ccc(Cl)c(Cl)c3)O)C2)CCN2CCOCC12 CCCC(C(=O)N1CCC(NC(c2cccc(OC(F)F)n2)=O)C(O)C1)C(C)C c1(C(N(CC(C)C)Cc2ncn(CC(=O)O)n2)=O)cnn2c1CC(C(C)C)CC2 CC(C)CC(O)C(=O)NCC(N1CCN(C(c2cncc(N(C)C)c2)=O)CC1)=O CN=c1cc(C(=O)NCC2(F)CC(NC(=O)Cc3ccc(Cl)c(F)c3)C2)cc[nH]1 c1(C(=O)NCC(C)(C(C)C)NC(C=C(C)c2cccs2)=O)cnc(C)c(C)c1 N1(C(C2C(NC(c3n(C)cc(Cl)c3)=O)CCOC2)=O)CC(O)CC(O)C1 O=S(=O)(c1cnc(NCCc2c(Cl)cncc2Cl)c(Cl)c1)NCC1CSCCS1 Cc1cc(C(=O)NC2CN(C(C3(C(C)(C)O)CC3)=O)CC2C)n(C)n1 C12(CNC(C3CCC(CC)O3)=O)CC1CN(C(=O)COCCCF)C2 N1(C(c2cc(C(N)=O)no2)=O)CC2CC(NC(=O)C3=CCCCC3)C1C2 CCCCCC(O)CC(=O)NC1(CO)CCC(C(F)(F)F)C1.C(COCCOC)N C1(OC)C(N=c2[nH]c(=N)[nH]c(=NCCc3ccc(F)c(Cl)c3)[nH]2)CC12CCC2 Cc1ccc(C(=O)NC(C)C(C)NC(c2c[nH]cc2-c2cnn(C)c2)=O)s1 C1(C(N2C(CNC(CC3CC(OCC)C3)=O)CC2)=O)CCCN1C(=O)C(F)(F)F c1(C(=O)NC2(C#N)CCN(S(C(C)C)(=O)=O)C2)cccc2cnccc12 C1(C(c2ccccc2)C)NC(=O)N(Cc2nccn2CC(F)(F)F)C1=O c1(OC)nccc(C(=O)NC(C)C(C)NC(c2csnc2OC)=O)n1 N1(C(=O)Nc2cc(C)nn2-c2ccccc2)CCCC#CCCCCC1 c1(C(N(CC(O)CNC(=O)CSS(C)(=O)=O)C)=O)cc(=O)cc(Cl)[nH]1 Cc1cccc(C(=O)NC2CCCC(CNC(C34CC(C)(CCO3)C4)=O)C2)c1Cl C1(F)(C(=O)NC2C(CNC(CCOC)=O)C2)CS(=O)(=O)CC12CCC2 c1(CN2C(CN3CCCC3)CCC(C(F)(F)F)C2)cccc2ncoc12 c1(C(=O)NC(C(C)NC(Cn2nc(C)c(Cl)c2)=O)C)ccc2c(c1)CNC(=O)N2 C1(CC)CCCCC1C(=O)NCC1(CNC(=O)CNc2cnn(C)c2)CCC1 C1(CC(N(c2nn[nH]n2)C(C=C(C)C)=O)C2CC2)CN(C(=O)OC(C)(C)C)C1 c1(CC)[nH]nc(Cl)c1C(=O)NC1CC1CNC(=O)Cn1cnccc1=O c1(CN)ccc2c(c1)N(C(=O)CC1SC3=NCCN3C1=O)CCC2 C1(OCC)(CNC(=O)OCCCn2cc(CO)nn2)CCCOC1 C(CN=C(NCC1CCCSC1)NCC(C)(O)c1ccco1)OC Cc1nc2ccc(F)c(CNC3CCC4C5CCC(C5)C34)c2[nH]1 CC1=C(C)CN(C(C2CCN(C(=O)c3cc(C)ncc3C)O2)=O)CC1 C(C(c1nnnn1C(C)C)NCc1cn(C)nc1C(C)C)(C(C)C)OC Fc1ccc(CNCc2ccccc2)cn1.OCC c1(N2CCC(N(CCC)C(C3(C)CCC3)=O)C2)nc2cccnc2s1 C(C(CC(F)(F)F)NC(=O)C(F)C1CCC1)NC(=O)CCc1ncco1 C(C)(CO)(C(=O)NCCCN(C(=O)CCCc1cc(C)no1)CCO)NC(C)=O C1(C)(C(N2CC(NC(=O)OC)C2)=O)CCN(C(c2c(C)ncn2O)=O)C1 CCC(F)(F)C(C)(C)C(=O)NC1CN(C(c2cc(CF)on2)=O)CC1F C(C)(C)(CCC(=O)NC1CC1CNC(c1cn(CC(=O)OC)nn1)=O)OC CCC(C(=O)N1CCCCC1CCNC(C1CCCC1OC)=O)C(C)O C1(NC(C(C)P(C)(C)=O)=O)CN(C(=O)COc2cccc(Cl)c2)CC1C1CC1 C#CCC(C)C(=O)N(CCCNC(=O)C(C)NC(C1CCOCC1)=O)C(C)C C(=O)(C1=C(C)OCC1)NCC1CC(NC(CNC=O)=O)C1 C(=O)(CC1=CCCCC1)NC1CC(C(C(=O)N(CC(CC)CC)CC)F)C1 C(=O)(C(C)(C)CN(C)C(c1ccnc(O)c1)=O)NCC1(COC)CC1 C=CCCC(C)(C)C(=O)NCC1CCC1C(=O)NC(c1ccccc1)CO c1(CN(C(C=CCNC(C(C)=CC(C)(C)C)=O)=O)C(C)C)ncccn1 Cc1nn(C)c(Cl)c1C(=O)NCC1CCCN1C(C1OCC2CCCC12)=O C(=O)(C1=C(C)C(C)(C)OC1=O)NCC(CC)NC(COC1(C#C)COC1)=O C(=O)(C1CCCc2sc(=N)[nH]c21)NCCC(C)NC(c1c(C)nc(C)o1)=O N1(C(C2(CC#C)CCCC2)=O)CCCC(C(=O)NCCC2CC(F)C2)C1 NC(=O)C(CCC(F)F)NC(=O)Cn1c(=O)ccn(Cc2ccccc2)c1=O C(N=c1[nH]cnc2c1COC2)C1CN(C(C2CCC(C)C2)=O)CC1C CC(C)(CCC(=O)N1CC(NC(C2(C)CCCCO2)=O)C(C2CC2)C1)[N+](=O)[O-] C#CC1(C)CCCN(C(=O)C(C)N(CCC)C(c2nonc2C)=O)C1 N1(C(C(C)=C2CC2)=O)CCC(C2CC2)(CNC(c2ccnc(Cl)c2)=O)C1 c1(C(N2C(C(=O)NCCOC(F)(F)F)C3CCC2C3)=O)n[nH]c2c1CS(=O)(=O)C2 CC1CCN(c2nnc(-c3cn(-c4ccccc4)nn3)n2CC2CC2)CC1O c1(C(N2CC(CNC(c3c(C)snn3)=O)C2)=O)coc2cc(F)ccc12 CC1CCC(C(=O)NCC2CN(C(C)C)C2)CN1C(=O)CCc1ccc(F)nc1 C#Cc1ccc(C(N2CCC(NC(=O)CCNCCCCOC)C(C)C2)=O)cc1 C1(NC(C(CO)N(C)C)=O)CCCN(C(c2cnc(-c3ccccn3)nc2)=O)C1 N1(C(C(CCOC)C)=O)CC(C2(NC(c3ccc(C)nc3OC)=O)CC2)C1 C#CC1(C(=O)Nc2cnc(Cl)nc2C)CCN(C(c2ccn(C)c2)=O)C1 C1(C(=O)NCCCN(C(C2(CSC)CC(F)(F)C2)=O)C)CC2(COCCO2)C1 N1(C(CNC(=O)NCC2CC2)=O)CCC2(NC(C3CC=CC3)=O)CCCC12 Cc1c(C(=O)N(C(C)CCNC(=O)CNC(C2CCC2)=O)C)ccn1CC1CC1 O(N=C1CCCCCC1)CC(=O)NCCC1CC(NC(=O)COC2CC=CC2)C1 C1(C(N2CC(O)(CNC(COc3cc(C)on3)=O)C2)=O)CN(C)CC1C(F)(F)F N1(C(C(C)OCCCCCC)=O)CCC2CN(C(=O)Cc3cnn(C)c3C)C2C1 c1(C(N2CC(OC)C(NC(=O)C(C)C(F)(F)F)C2)=O)ccc2oc(=O)oc2c1 c1(OC)cc(CN2CCN(C(C3CCS(=O)(=O)C3)=O)CC2)ccc1-n1ccnc1 c1(C(=O)NCC2C(NC(c3ccc(C)cc3)=O)CCC2)ccc2c(n1)NCC2 C(=O)(C1=C(C)OCC1)N(C1C2CN(C(C3C(CC)OCC3)=O)CC21)C S(=O)(=O)(c1cc(C)cnc1NCc1csc(CC)n1)N(C)CC1(OCC)CCC1 C1(C2CC2)(CNC(c2cc(C)n(C)c2)=O)CCN(C(=O)CC2(O)CCOCC2)C1 C1(C(=O)NCc2cc(CC)on2)N(C(=O)CN2CCSCC2)CCCC1(C)C Cc1c(C(=O)N(C2(C(C)C)CC2)C)sc2ncn(C)c(=O)c12 CCC(CC(=O)NCC1CN(C(=O)CCOC2CCOCC2)CCCO1)C(C)C N=c1[nH]c2ccc(C(=O)NC3CCN(C(C4CC(=O)N(C5CC5)C4)=O)C3)cc2[nH]1 c1(C(=O)NC(CC(C)NC(c2c(C)ccn2C)=O)C)cc2c(nc1O)CCSC2 N(C(=NCCC(C)(F)F)NCc1ccc(C(C)C)cc1)C(COC)C C(C)(C)(CCCNC(C1CC(C)C1)=O)NC(C=CC=CC)=O C(=O)(C1=CCCC1)N(CCCOCCN(C)C(c1cnn(C)n1)=O)C N1(C(C2CC(=C)C2)=O)CC2CCCC2(NC(c2csc(CO)n2)=O)C1 CC(C)(F)CCC(=O)N1CC(NC(=O)C(O)Cc2cc(Cl)cc(Cl)c2)C2(CC2)C1 C(=O)(Nn1cnn(CC)c1=O)C1(CC=C)CCN(C(=O)Cc2cnns2)C1 N1(C(c2cnc(OC)s2)=O)CC2CCOC2(CNC(c2cc(Cl)nnc2O)=O)C1 CC#CCCC(=O)N1CCC(N(CC(C)C)C(C2COCCO2)=O)CC1 c1(CC)cc(C(=O)N(CC(=O)NCCC(C)c2nc[nH]n2)C)ccn1 c1(C(=O)NC(CNC(C2C(CCC)C2)=O)(C)C2CCC2)c(C)nn(C2CC2)c1Cl C#CCC(CC#C)C(=O)N1CCOCC1(C)c1cn(CC2CC2C(F)(F)F)nn1 c1(C(=O)NC2CC(c3ccccc3)(CNC(C3C(C)C3)=O)C2)cc(F)c(F)cc1N C12(C(=O)NC(C)CC3CN(C(=O)CCc4cn[nH]c4)C3)CC1COC21CCC1 C1(CC)(CNC(c2coc(CNC(C3CC=CCO3)=O)n2)=O)CCCC1 c1(C(=O)NC(CN(C(c2c(CC)cno2)=O)C)C)cc2c(OC)ccc(F)c2[nH]1 c1(C(N2C(CNC(C(c3ccccc3)C)=O)CCC2)=O)cnc2scnc2c1 C1(C(C)C)CC(C(=O)NC(C)CCCNC(=O)CSS(C)(=O)=O)CCO1 N1(C(c2cc(CCC)c(C)s2)=O)CC2CCCC2(NC(c2ccncn2)=O)C1 c1(CC(=O)NCCC(CNC(c2ccc(CCCCC)[nH]2)=O)O)cc(C)ccc1C N1(C(C2(C)CCC2)=O)CCCC(CO)(NC(=O)Cn2cnnc2O)C1 C1(NC(C(C)Sc2ccccn2)=O)CN(c2cc(Cl)nc(C3CC3)n2)CC1(C)C Cc1ccc(N)c(C(=O)NCC=CCNC(c2csc(-c3ncccn3)n2)=O)c1 CC1CN(C(=O)C(C)OCCN(C)C)CC1CN=c1[nH]ncs1 C(=O)(C1=CCC(C)(C)CC1)N1CCC(CNC(C(CCOC)OC)=O)(OC)C1 CC1CCN(CC(=O)N(C)CCNC(C2C(c3ccccc3)C2(C)C)=O)C1 c1(OC)cc(CN(C)CC2(OC3CCC3)CCC2)ccc1Cl C1(C(N(CC(=O)NCc2ccc[nH]2)C)=O)CC(CO)CO1 N1(C(c2ccc(OCCC)cc2)C(=O)NCC)Cc2ccccc2C(CO)C1 N1(C(C(C)NC(=O)NC)=O)CCCC(NC(=O)CC2(C(F)(F)F)CC2)CC1 Cc1ccc(C)c(OCC(=O)NC2CN(C(=O)CC3OCCCC3(C)C)C2)c1 c1(C(N(c2nc(OC)c(C)cn2)C2CNCC2(F)F)=O)cnc2cccnn12 CC1CC(CNC(=O)CC2OCCO2)CN1C(c1ccc(C(F)F)s1)=O C1(CNC(C(C(C)C)n2cnnn2)=O)CN(C(=O)C=Cc2cnc[nH]2)CCCO1 Cc1nc2ncc(C(=O)NCC=CCNC(c3c(C)nc(C)n3O)=O)cc2o1 c1(C(N2C(C)CN(C(=O)Cn3cccc3)CC2)=O)cc2ncccc2s1 c1(OC)cc([N+](=O)[O-])c(C(N2CC(C)N(Cc3ccccc3)CC2C)=O)cc1O C1(C(=O)NCCC(=O)NC(c2cccnc2C)C)(COC)CCCCO1 c1(C(N2CC(NC(c3c(C)cco3)=O)C(F)C2)=O)cnc2ccnn2c1 N1(C(CCOC(C)C)=O)CCC2C(CCN2C(c2ccccc2Br)=O)C1 CC1(C)CC(C(=O)NC2(C3CC3)CCN(C(c3cc4sccc4[nH]3)=O)C2)=NO1 CCCC(C(=O)OCC)NC(=O)NC12CC(C1)C(C)O2 n1(CCC)ccc(C(=O)NCC(O)CN(C(=O)C=CC2CCCC2)C)n1 c1(C(=O)NCC2(F)CC(NC(C(C=C=C)C)=O)C2)cccc(Cl)c1Br Cc1ccc(F)c(C(=O)NCC23CC(NC(=O)CCc4cncn4C)(C2)C3)c1Cl C1(NC(c2cnc(CC)[nH]2)=O)CCC(C)N(C(=O)CN(C)C(C)C)C1 c1(C(N2CCC(N(C(=O)CCc3ncccn3)CC3CC3)C2)=O)ncccc1O C(C)(CC(=O)NC(C)CCNC(c1c[nH]nc1-c1ccccc1)=O)OC c1(OC)nccnc1C(=O)NC(C1CCCN(Cc2cnn(C3CC3)c2)C1)C Cc1ncncc1C(=O)NCCCC(C)(C)NC(c1cnc(CC2CC2)s1)=O Cc1cc(C(N2CCOC(C(N3CCC(CO)C(O)C3)=O)C2)=O)c2cc[nH]c2c1 c1(CC)cc([N+](=O)[O-])ccc1NC(=O)NCC1CS(=O)(=O)CCO1 C1(F)(CNC(c2c(CC)nc[nH]2)=O)CCCN(C(C2CC2(C)C)=O)C1 Cc1ncccc1CN(c1c(NC(C2CCCO2)=O)[nH]cn1)c1ccccc1 N=S1(=O)CCN(C(C2Cc3cccc(F)c3O2)=O)CC12CCC2 CC1CCC(=CC(=O)NC2(CCNC(=O)C(=C3CCCCC3)F)CCC2)C1 c1(C(=O)NC(CC=C)CNC(=O)Cc2[nH]cnc2C)cc2cc(C)ccc2o1 c1(C(CNC(N2CCC(c3ccc(C)nc3)C2)=O)(C)C)cccc(Cl)c1F C1(C(=O)NCC(CC)NC(=O)CCc2ccn(C)n2)Cc2ccc(C)cc2S1 N1(C(c2cc(C)on2)=O)CCC2(CCN(C(c3cnccn3)=O)C2)C1 Cc1c(C(N2CCCC(NC(=O)CCc3ccc(=N)[nH]c3)C2)=O)cnn1C(C)C c1(C(=O)NCC23CC2CN(C(C2CCCSC2)=O)C3)cc2ncccc2[nH]1 c1(C(=O)NCCOC2CCN(C(Cc3c(C)scc3)=O)CC2)cc2occc2[nH]1 c1(C(=O)NCC(CNC(c2cccc(C)n2)=O)(C)C)cc(S(N)(=O)=O)cs1 CC1(C)CCC=C1C(=O)NC12CCCC1CN(C(=O)Cn1nnnc1C1CC1)C2 c1(C(=O)NC2C(CNC(C(c3scc(C)n3)C)=O)C2)cnc2ncnn2c1C Cc1cc(C(N2CC(NC(c3cscc3F)=O)C(C)C2)=O)c2cc(F)ccc2n1 C1(C(C(C)C)NC(CSC)=O)CCN(C(=O)C(C)Oc2ccccc2)CC1 CC1CC2CN1C2=O.c1(NC(=O)CC2(OCCC3CN(C)C3)CC2)ccccc1 C1(C(=O)NCCCN(C(c2ccc(C=C)cc2)=O)C)CCC2CCC(=O)N12 c1(C(=O)NCC(CC)NC(=O)Cn2cc(CO)nn2)nc(C(C)C)c(C)s1 n1(CC)ncc(CN(C(=O)CC(C)(C)F)C(=O)OC(C)(C)C)c1C c1(C(=O)NCC(CNC(C2NC(=O)OC2C)=O)OC)[nH]nc([N+](=O)[O-])c1Cl C12(NC(C3CCCCC3)=O)CCCC1N(C(=O)C=CC=Cc1ccccc1)CC2 C12(C(N(CC(=O)NOCC(=O)N(C)C)C(C)C)=O)CC(C)(CCO1)C2 Cc1ccnc(C)c1C(=O)NC1(C2CCCN2C(C2CCC(=O)N(C)C2)=O)CC1 C(=O)(C1=CCN(C(=O)CSC2CC2)CC1)NCCn1c(C)nnc1 c1(CC(N2CCC3(NC(=O)COCCF)C(C2)C3)=O)cccc2ccoc12 c1(CC)ccc(C(=O)NCC2CCN2C(C2CCSCC2)=O)c(C)c1 N(C)(S(N)(=O)=O)CC(=O)NCCN(C(=O)CCc1cnoc1)C c1(C(N2CC(O)(CNC(C3C(SC)CCC3)=O)C2)=O)ncc(N(C)C)cn1 C1(C(=O)NC2CCN(C(C34CC(C)(C3)C4)=O)C2)CCc2ccc(Br)cc2O1 C1(C(COC)N(C)C)CCCC12CCCN(C(=O)COCCCF)C2 c1(SCC)cccnc1C(=O)NCC1(NC(=O)CCC2CCCN(C)C2)CC1 N1(C(c2c(CC)nc[nH]2)=O)CCOCC(CNC(C2CCSC2)=O)C1 CCCC(O)C(=O)N1CC(NC(C2(CC(=O)NC)CCCCC2)=O)C(CCC)C1 CC1CC(NC(=O)C(C)n2ccnn2)CN(C(=O)COC(F)F)C1 C1(CNC(CSCC=C)=O)(NC(C2CC2OCC)=O)CCCC1 N1(C(Cn2cccc(N)c2=O)=O)CC2(CCN(C(C3CCC3CF)=O)C2)C1 CCCC(CC(=O)NCC1(OC(C)C)CCC1)NC(c1cccnc1S)=O O=[N+]([O-])c1cc(S(=O)(=O)NC2CC(CNc3c(Cl)cc(Cl)cc3I)C2)ccc1F C(CC1CC1)(C(=O)NC1CC(CN(C(=O)C2CC2)C2CC2)C1)OC C(=O)(CCC(=O)C(C)(C)C)N1CCC(C(=O)NCC(O)C(N)=O)(CC)C1 c1(CNC(CN(C(COCCCC#C)=O)C(C)C)=O)c(F)cncc1F N1(c2[nH]c(=NCc3c[nH]c(=N)s3)[nH]c(=N)n2)CC23CCCCC2(C1)CS(=O)(=O)C3 c1(C(=O)NCC(C(C)(C)C)NC(C2CC(C)(C)OCC2)=O)cccn2ccnc12 N1(C(C2N(CC)CC2)=O)CCC(CNC(c2nocc2C(=O)OCC)=O)CC1 C1(CC(=O)NCCC2N(C(CCCOC)=O)CCOC2)CCCCC12CC2 c1(C(C(=O)NC2CCN(C(CC3CC(OCC)C3)=O)C2)(F)F)cccc(C)n1 C(CSC)(C(=O)NCC(C1CCC1)NC(=O)Cc1csc(C)n1)NS(CC)(=O)=O N1(C(CC)=O)CC2C(CNC(c3cn(C4CCOCC4)nn3)=O)C2C1 O=C1Nc2cc(Cl)ccc2CC1NC(C1CN(C(c2ccncc2)=O)CCN1)=O C(=O)(CCCC(C)(C)C)NC(CCN(C(C=C(C)Cl)=O)C)C C=C(C)CCCC(=O)NCC1CN(C(=O)CCOc2cccnc2)C(C)(C)C1 N1(C(CSC(C)C)=O)CCc2ccccc2C1CCNC(C1(F)CCOC1C)=O C1(C(N(CCCNC(C2(CC=C)CC2)=O)C(C)C)=O)Cc2nccnc2C1 Cn1nc(Br)cc1CCNC(=O)CCC1CCNC1 C1(NC(=O)Cc2nncs2)CCCN(C(C2(C(F)(F)F)CC=CCO2)=O)CC1 N1(CCC(=O)OC2C(C(N)=O)CC2)CSCCSC1 C1(NC(Cc2cn(CC)nc2)=O)CCN(C(C2CC(C)(C)C2)=O)C12CCCC2 c1(C(=O)NC2CN(C(CC3CCC(C)O3)=O)C2)cc(F)c(Cl)cc1F N1(C(CCN(C)CC)=O)CCC(C)C(NC(C2CSC(C)=N2)=O)C1C N1(C(c2cc(CC)c(C)s2)=O)CC(NC(c2cc(CCOC)on2)=O)CC(O)C1 Cc1cccn2cc(C(=O)NC3CC4CCC3C4)nc12 c1(OC)cc(CNC2CCC(C(=O)Nc3cscn3)C2)c(Cl)cn1 c1(C(=O)NC2CCC(C(=O)Nc3ccc(C)c(Br)c3)CC2)c(Cl)cnc(Cl)c1Cl c1(C(C(=O)NCCN(C)C(C2NC(=O)C3CC23)=O)=O)c[nH]c2ccc(F)cc12 C(=O)(C1=CC2C=CC(C1)C2)N1C(C(C)C)(C(=O)NCc2cnns2)CCC1 C(c1c(C)nn(C)c1Cl)=CC(=O)N(C(CCNC(C=Cc1cnc(C)s1)=O)C)C C1(CCCNC(c2ccoc2Cl)=O)CCCN1C(=O)CC1COC(=O)C1 O=C(C#CC1CCC1)NC1CCN(C(=O)C(O)C(F)F)C1 CCCC(CC(C)C)C(=O)NCC1(NC(=O)C(c2ccc(F)cc2F)C)CC1 c1(OC)cc(F)ccc1-n1ccc(C(=O)OCc2nc(C(C)C)n(C)n2)n1 c1(C(=O)NCCOc2ccccc2)cc(F)ccc1[N+](=O)[O-] C12(NC(C(C3CCOCC3)OCC)=O)CCCC1N(C(=O)CCC(C)(F)F)CC2 Cc1ccc(C(=O)N(CC(C)CNC(=O)C2=CC(C)CC2)C)c(C)n1 c1(C(C#C)NC(=O)N(CC(c2nccn2C)O)C)ccc(F)cc1 CS(=O)(=O)c1ccc(C=CC(=O)NC2CN(C(C3CC34CC4(F)F)=O)C2)o1 C1(C(=O)NC(C(=O)NC)C2CC2)CCCC(NC(c2ccnn2C)=O)CC1 N1(C(COc2ccn(C)n2)=O)CC(NC(C2CC3CC2CO3)=O)C(CC2CC2)C1 CC1CCOC(C(N2CC(CNC(C3(O)CCC3)=O)C(C)C2)=O)C1 N1(C(c2cc(C)c(C)nn2)=O)CCC(N=[N+]=[N-])(C(N2CC3COCC3(C)C2)=O)C1 C12(C(=O)NCC(CC)OC3CCOCC3)CC(C1)C(C)O2 N1(C(CC=C(C)C)=O)CCC(C2CC2)C1C(=O)NC1CC2CC1CC21CC1 [N-]=[N+]=NCC(C(=O)NCC(O)C(F)(F)F)NC(=O)CN1CCCC1=O N1(CC(C2CC=CCC2)(C)C)CCC(C(=O)NOCCCCC2CC2)=C(F)C1 C(=O)(CCC(=O)NCC(C1CC1)NC(=O)Cc1ccc(O)nc1)OC C1(C(=O)NCCCCCCNC(C(C)C(F)F)=O)Cc2nccnc2C1 c1(C(N2CCC(N(C(=O)CCCc3nccs3)C)C2)=O)nnc(O)nc1O n1(CCNC(c2c(C)con2)c2nnnn2C)cc(C(F)(F)F)ccc1=O N12CC3(CCN(C3)CC3(CC3)C1=O)C2.CC(=O)CSC1CC1 C1(C)(C(N2CC(NC(c3cnc(C)[nH]3)=O)C(C(F)(F)F)C2)=O)CC(C(C)C)=NO1 c1(C(=O)NCC(CCOC)NC(=O)COC2CCOC2)ccc2ncccc2c1 Cc1cc(C(=O)NC2CCN(Cc3ccc(F)nc3C)C2)cc(C)c1O C1(CC(=O)NC(C(=O)NCCCC=CC)(C)C)NC(=O)NC1=O c1(C(N2CCC(CN(C)C(C3CCC(O)CC3)=O)C2)=O)ccc2nonc2c1 C(CC(=O)NNC(=O)NC1CC2(CC2)C1)c1ccc(C)s1 C(C(CC(=O)N1CC=C(CNC(=O)Cc2cc[nH]n2)CC1)C(F)(F)F)N(C)C c1(CC)ccsc1C(=O)NCC1CCC(C(=O)NCCc2ncc[nH]2)C1 C#CC1CC2CCC1N(C(C1CC=CCN1C(=O)CC1COCC1O)=O)C2 Cc1c(C(=O)NCC2CCC(NC(=O)CC3CCCO3)CC2)cnc2[nH]ccc12 C(c1c(C)nn(CC)c1C)=CC(=O)OC(CCCC#C)C C(C(=O)NCC1(O)CCN(C(=O)CC2CC=CC2)C1)(C(C)C)OCC c1(C(=O)NC2CN(C(CCCCC)=O)CC2(C)C)cccc2c1C1CCC2CC1 C(C)(CC(C)(C)C)NC(C(c1cnn(C)c1)NC(c1cc(C)sc1)=O)=O C1(NC(C(C2CCOCC2)OCC)=O)CN(C(=O)Cc2ncc(C)[nH]2)C(C)(C)C1 C=CCC(C(=O)NCC1CCCCN1C(=O)Cc1cncn1C)N(C)C c1(NC(C2(O)CCN(C(CC)=O)C2)=O)c(C(C)=O)cc(Cl)nc1Cl C1(C(=O)NC(C(N2C(C)(CCO)CC2)=O)(C)C2CC2)CC2(CCO1)CC2 c1(OC)ccc(C(=O)NC(C)CCCNC(=O)C(C)(C)OC)nc1 C1(CNC(C2CC(C)(c3ccccc3)C2)=O)CCCCCN1C(C12CCC1C2)=O c1(CC)sc(=N)[nH]c1C(=O)NCC1CCCCN1C(c1c(OC)noc1C)=O c1(C(N(CCCNC(CCOC(C)C)=O)CCO)=O)cnc2occc2c1 C1(CNc2c(C(=O)OC)cc(F)c(C)c2)CCCC2(CCC2)C1O c1(C(CNCC(=O)NC(C)(C)C)N(CC)CC)ccc(Br)cc1.c1(C)ccccc1 c1(C(C)C)ncc(C(=O)NCC2CCCC2NC(c2coc(Cl)c2)=O)s1 c1(C(=O)NCC(CNC(c2cnc(OC)nc2C)=O)F)cccc2cnsc12 C(=O)(C(O)CC(N)=O)N1C(CNC(c2c(C)cc(C)s2)=O)CCC1 c1(C(=O)NCCOCCN(C(C(C)OCCC(C)C)=O)C)cccc2ccoc12 C1(O)(C(=O)NCC2C(C(=O)NC3(CCCCSC)CC3)CCC2)CCOC1(C)C CC(CC(=O)NCC1(NC(c2nnn(-c3ccccc3)n2)=O)CC1)C1CCCO1 c1(CC)cccc(C(=O)NC2CN(C(c3oc(C)nc3C(F)(F)F)=O)CC2O)n1 N1(C(CC=CC(C)(C)C)=O)CCC(C)(NC(=O)Cc2ccc(O)cc2)C1 C1(c2c(C(=O)OCC)nco2)CCN(C(C2CC2c2ccccc2)=O)CC1 c1(C(=O)Nc2ccc(C(=O)NC)nc2)cc(F)ncc1Br C(CCC(C)(C)C(=O)N1CC(C)CCC12CC2)NC(c1c(CC)nns1)=O C1(N(C(=O)Cn2ncnn2)CCC)CCN(C(=O)CSC(F)F)CC1 C(=O)(C1=CC2(CCOC2)C1)N1CC(NC(c2ncc(C)c(C)c2)=O)C(C)C1 c1(OC)cc(OC)cc(S(=O)(=O)N2CCCN(c3cccc(C)c3)CC2)c1 c1(C(=O)O)cc(S(=O)(=O)N2CCN(Cc3nccn3C)CC2)oc1Cl c1(C(=O)NC(C(C)NC(c2c(C)nsc2)=O)C)ccc2c(c1)CCCS2(=O)=O c1(N(C2CN(C(c3cc([N+](=O)[O-])cs3)=O)C2)C)ncnc2c(Br)csc12 Cn1cnc2cc(C(N3CCC(NC(C4CCC(=O)N4)=O)CC3)=O)ccc2c1=O CCC(CC(F)(F)F)C(=O)N(CC(C)NC(c1c(C)ccc2n[nH]cc12)=O)C NS(=O)(=O)c1ccc(C(=O)NC2CCCC(NC(C34CC(CCO3)C4)=O)C2)s1 Cn1ncc(C(=O)NC2(C3CCCCN3C(C3CNC(=O)N3)=O)CC2)c1Cl c1(C(C(=O)NCCCSC)N(C)CCc2cccc(F)c2)ccc2n[nH]cc2c1 c1(C(=O)NCC2C(NC(c3cnc(C4CC4)nc3)=O)CC2)cc2cn[nH]c2cn1 c1(C(N(CC(CC)NC(c2ccnc(C3CC3)c2)=O)C)=O)nc2ccccc2[nH]1 c1(C(=O)NC(CCNC(C23CC(CCC)(C2)C3)=O)C(C)C)cc(OC)nc(Cl)c1 c1(C(N2CC(OCC(N3CCN4CCC3CC4)=O)C2)=O)cccc2occc12 CC1(C)C(NC(=O)CN2CCC(CO)CC2)CCN1C(=O)CCn1cncn1 Cc1ccc([N+](=O)[O-])cc1-c1noc(N2C(=O)CCC2=O)n1 c1(C(=O)OC)ccc(CCC(N2CC(O)(C(C)NC(=O)CCF)C2)=O)cc1 c1(C(N2C3(CNC(CC4(C)CC4F)=O)CC(C2)C3)=O)ccc(N)c(CC(C)C)c1 C1(CNC(C2(C)CC=CCO2)=O)CN(C(=O)COCC2CCC2)CC1(F)F c1(CC)ccc(F)c(C(N2CCOC(CNC(=O)CC3SC(=N)NC3=O)C2)=O)c1 C(=O)(CS(=O)(=O)c1ccccc1F)NC1CC(C)(NC(c2cccnc2O)=O)C1 c1(C(N2CCCN(C(CC(C=C)CC)=O)C(CO)C2)=O)nc2nccc(C)n2n1 c1(CC(=O)NCC2CN(C(C(C)C(C)(C)C)=O)C(C)CC2)ccc2c(c1)COC2 C1(C(N2CCCC2CC(=O)CC23CC(C2)C3)C)CCCCN1CC1CCOC1C S(=O)(=O)(c1cc(F)cc([N+](=O)[O-])c1)N1C(C)CC(Cc2ccccc2)CC1 Cc1cccc(CC(=O)NC(C)CCCNC(C2CC2CN(C)C)=O)c1 N1(C(CCOC)=O)CCCC(C)C1CCNC(c1cnc(O)c(F)c1)=O C12(CC(=O)NC(CNC(C(CC)C)=O)(C)C)CCC(CC1)N2C(=O)OC(C)(C)C n1(C2(C(=O)NC3CN(C(c4ncncc4Cl)=O)C3)CC2)cnc2ccccc12 CC(C)S(=O)(=O)CCN=C(NCc1ccc2ccccc2c1)NCc1ccco1 Cn1[nH]nnc1=NCCNC(=O)C=CC1CCCC1 c1(C(N(C(CNC(c2cc(C(C)=O)sc2)=O)C2CC2)C)=O)ncn2ccccc12 C#CCCC(=O)NC(C)(C)C(C)NC(=O)COCC(C)(C)C N1C(=NCCC2CC(=O)N(C)C2)NCC1.c1(CC(C)C)c[nH]nc1C(F)(F)F c1(-c2nc(C)sc2)cccc(C(=O)NCC=C2CCOCC2)c1 c1(OC)cc(C(=O)NC2(CO)CN(Cc3ccc(F)cc3Br)C2)ccc1I C1(C(C#C)C)CCN(C(=O)CCC2(C)CCCN2C(=O)C=CC2CCCC2)CC1 C1(C(=O)Nc2c(C)ccnc2)CN(C(c2ncccc2Cl)=O)CCN1C N(C(=NCC1CC1)NCC1CCN1C(=O)OC(C)(C)C)C(C1CCOCC1)COC C1(C(=O)NCC2CCN(C(c3n[nH]c4c3CCC4)=O)C2)CCc2ncnn2C1 CC1CCC(CNC(c2cccc(C3CC3)c2)=O)CN1C(C1CC=CCC1C)=O CCCC(CCC)C(=O)N1CCCC(C(=O)NC(c2csnn2)C)(CC)C1 C1(NC(CCC)=O)CCCOC12CCN(C(C1COC(=O)O1)=O)CC2 C1(NC(C2(NC(CC(C)O)=O)CCSC2)=O)(CO)CC(C)(C)C1 n1(CC)ncc(C(=O)N(C)Cc2cccc(CNC(=O)CC34CC(C3)C4)c2)c1C Cn1cc(C(=O)NCC(F)CNC(C2CCCC(F)(F)CC2)=O)c2ccccc12 C1(CN(C(c2cc(COC)[nH]n2)=O)CC)CCN(C(c2ccccn2)=O)C1 N1(C(CCc2c(C)ncs2)=O)CCC(NC(=O)Cc2n[nH]c(=N)s2)C2(CCC2)C1 CCC(CC)C(F)C(=O)NC1CC12CCN(C(=O)C(C)c1ccco1)C2 C(=O)(C1=C(C#N)CCC1)NCCC1C(C)CCCN1C(=O)CN1CC(=O)NC1=O C(=O)(CCCCC(=O)N1CC(CCO)(OC)C1)OCC CC1=CCC(C(=O)N(C2CCCCC2N(C)C(c2sccc2F)=O)C)CC1 CC1CCCCC1(CNC(=O)Cc1ccccc1)NC(=O)COC1CCCOC1 Cc1cc(Cl)ccc1OCC(=O)NCCC(C)N(C(=O)C(C1CCCCC1)F)C C1(NC(COc2cn(C)nc2)=O)CCCN(C(=O)CSC(F)F)C1 N1(C(c2cc(C(=O)OC)on2)C(=O)NC2COC2)CC2CCCC(O)C2C1 CC(C)CC(C(=O)N(C(C)(CO)C1CCC1)C1CC1)ONC(=O)CC1CC1 N1(C(C(C)OCc2ccc(C)cc2)=O)CCN(C(c2ocnc2C)=O)C(CF)C1 CC1(C)CC(C)(CNC(C2(CO)CCOCC2)=O)CN1C(C1CC12CC2)=O c1(C(C)C(=O)NCCCOCCNC(=O)C=Cc2cc[nH]c2)nc(F)ccc1Cl Cc1nncc(C(=O)NC2C=CCN(C(=O)CCCF)C2)c1C C1(CNC(CCn2cc(-c3c(C)ncs3)nn2)=O)(CO)CCCCC1 c1(CCC)nc(C(=O)NC(C2(O)CN(C(=O)Cc3cnn(C)c3)C2)C)cs1 Cc1cc(C(=O)NC2(C)CCCN(C(=O)C(F)(F)c3cscn3)C2)cc(C)c1 c1(C(C(C)O)NC(=O)N(C)CCS(=O)(=O)c2ccccc2)nnc2ccccn12 C=CC(CCC)CC(=O)N1CC(CNC(c2csc(O)n2)=O)C(F)(F)C1 CC1c2sccc2CCN1C(c1cc2cc(F)ccc2o1)=O C(=O)(CCC(C)(C)NC(c1csnn1)=O)NC(C1CCCC1)C C1(NC(CC2(C)CCCO2)=O)CC12CCN(C(=O)COCCCF)C2 C1(CNC(c2cc(CC)[nH]n2)=O)(NC(c2cn(CC)cn2)=O)CCC(F)(F)CC1 c1(NC(C)=O)ccc(N(C)C(N2CCN(C(c3cnc(O)o3)=O)CC2)=O)cc1 O=C(Cc1ccc(I)cc1)NNC(=O)c1ccnc(-c2cc[nH]n2)c1 CC1CN(C(C2CC(F)(CO)C2)=O)CC(CCNC(c2cccc[n+]2[O-])=O)O1 c1(C(C(=O)NC(C)(C)C)N(C(C#C)C(C)(C)OC)C)cn2cc(Br)ccc2n1 c1(OC)cc(C(=O)NC2CN(C(=O)CCCn3cccn3)C2)cc2cccnc12 C1(CCOC)CN(C(=O)CC2=CCCC2)CCN1C(c1ncn(C)c1C)=O C(CC(C(C)C)NC(=O)Cn1cc(Br)c(C)n1)N(C(CCC)=O)C c1(C(C(=O)NCC(C)C)N(C2CC2)CC2CCOC2)ncc(Cl)cc1Br CCC(F)(F)CC(=O)NCC1(C)CCCN(C(=O)CCN2CCC(F)C2)C1 N1(C(=O)OCc2ccncc2)CCC(Nc2ccccn2)C2CC12 C1(NC(C2(COC)CC2(F)F)=O)CCCC(CNC(=O)CNC=O)C1 C1(C2CCN(C(C3CC3c3ccccc3F)=O)C2)(NC(C(F)=CCC)=O)CC1 N1(C=O)CCC12CC(O)C2.N1(C(C2CN(C3COC3)C2)=O)CCC(C(F)(F)F)C1 O=C1CCCN(CC2(c3ccccc3)COCCO2)CC1 N1(CCC=CCC)CCC(NC(C2(c3cccs3)CCCC2)=O)C(O)C1 Cc1cc(C(=O)NCc2cc(C)c(C(=O)NC3(CF)CCCC3)o2)ncc1F C1(C(N(CC)Cc2occc2C)=O)CC2C=CC1N(C(c1ccn(C)c1C)=O)C2 C1(NC(c2ccc(C)n2C)=O)CC2CCC1N2C(=O)C(n1ccc(C2CC2)n1)C Cc1ccc(Br)c(F)c1C(N1CCC(F)(F)C(NCc2ccc(F)c(F)c2)C1)=O n1(C(CC)C)nnnc1C(C1CCC1)NCC(=O)OCCc1nccs1 CC#Cc1ccc(C(C(=O)NCCCF)N(C2CC2)C(C)C2CC2)cc1 N1(C(CCC(=O)NCCC)=O)CCC(NC(c2ncc(C)cc2F)=O)C(O)C1 c1(OC)ccc(Cn2cc(C(C)NC(c3[nH]ncc3C#N)=O)nn2)cc1 CC#CCCC(CO)NC(=O)C(C)CSC1CCCCC1 CC1(C)C=C(C(=O)NC(C2CCOC2)CNC(=O)Cn2ccc(O)nc2=O)C1 CC(C)C(=O)C(=O)N(C)CC1CCCN1C(C1CC2CCC2C1)=O N1(C(C(CC)=O)=O)CC2CN(Cc3cc(Cl)cc(Cl)c3O)CC2C1 CC1(C)C(=O)NC(=O)N1CC(N1CCN(C(=O)C2=CCCS2)C(CC(F)F)C1)=O C1(CNC(C(C)C)=O)CCC12CN(C(=O)CC1CCCN1C(=O)OC(C)(C)C)C2 c1(C(=O)NCC(C)(C)NC(c2ccc(CC)[nH]2)=O)ccc(S(=O)(=O)CCO)cc1 c1(CC(N2C(CN(CC(=C)Br)C)CCCC2)=O)ccc2nc(O)[nH]c2c1 N1(C(CN(C)CC)=O)CCN(C(c2cc(Cl)c(F)cc2OC)=O)CC12CCC2 Cc1ccc(F)c(CC(=O)NC(C)CCNC(C2CC(F)C(=O)N2C)=O)c1 C1(C(C)NC(C2OCCOC2C)=O)CCCN(C(=O)C=CCN(C)C)C1 c1(C(=O)NC2C=CC(CNC(Cc3cnc(C)[nH]3)=O)C2)cc(N)c(O)c(F)c1 c1(CN2C(C(=O)NCCCN3C(=O)C=CC3=O)CCC2)cc(Br)ncc1F CC1CCCN(C(=O)C(C)n2ccnc2)C1CNC(c1cc(O)ccc1Cl)=O C1(CNC(CCC=C)=O)CN(C(=O)CCc2cncnc2)CCC1(C)C C(=O)(C(C)C1=CCCC1)NCC(C(C)C)NC(c1c(OC)cnc(Cl)c1)=O C1(CNC(CSCC#C)=O)CC(NC(=O)CCC2CC2)CO1 C1(CN(C)C(c2cn(C3CC3)cn2)=O)CN(C(C2C(C)(C)C2(F)F)=O)CCO1 CC(CC(C)(C)C)C(=O)NC1(CO)CCCN(C(=O)CC2CCCSC2)C1 c1(C(=O)NCCN(C(c2[nH]cc3c2CCC3)=O)C2CC2)c(Cl)cccc1[N+](=O)[O-] C1(C2(O)CN(C(c3cc(C(N)=O)no3)=O)C2)(CNC(C2C(COC)C2)=O)CC1 CC1(C)CN(C(c2cc(C#N)ccc2O)=O)CC(CNC(C2(Br)CC2)=O)O1 c1(C(N2CC(CNC(C3=C(C)CCCC3)=O)C2)=O)cc(C)c(F)c(S(C)(=O)=O)c1 c1(N2CCC(=CC(N3CCOC4CC34)=O)CC2)ccnc2cc(Br)nn12 CC(C(=O)N1CCN(C(c2sccc2-n2ccnn2)=O)CC1CCO)C(C)(F)F Cc1cc(=NCC(C2CCCC2)NC(C2(O)CC3CCC2C3)=O)[nH]c(CO)n1 CC1(C)CN(C(=O)CN2CCS(=O)(=O)CC2)CC1CNC(c1cc(F)c[nH]1)=O c1(SC)cc(Br)ccc1C(N1CC(NC(C2(O)CCC2)=O)CC(C)C1)=O c1(C(=O)NCCC2(C)CCN(C(C(CC)(C)O)=O)C2)cc(C)cc([N+](=O)[O-])c1 c1(C(=O)NCCC(C)NC(c2cccc(F)c2Cl)=O)c2c(nn1C)CCSC2 N1(C(C(C)C)=O)CCC(C(=O)NCC(C)(F)CNC(=O)CC(C)(C)O)CC1 C1(NC(C(C)NC(=O)OCC)=O)CCCCC1NC(c1cnc[nH]1)=O C(=O)(CCCC(C)(C)NC(c1ccc(Cl)cn1)=O)N(C1CC(SC)C1)C C1(CNC(c2csc(C(F)(F)F)n2)=O)CN(C(C2CC3(CCC3)C2)=O)CCO1 C(N=c1[nH]c(=NC(C)c2cn[nH]c2)[nH]c2c(F)cccc12)c1c(C)ccc(Br)c1 c1(C(N2C(C(C)NC(=O)CNC=O)CCC2)=O)cccc2c1ccn2C N1(C(C(n2ncc(C)c2)C)=O)CCC2(CC(C(=O)N(CC(C3CC3)N(C)C)C)C2)C1 CN1CC(NC(=O)C(C)(C)CN(C)C(c2ccc3c(c2)CC3)=O)CCC1=O C1(C(=O)NCCCC2N(C(CNC(C(C)(C)C)=O)=O)CCC2)CCCCN1N=O c1(OC)ccc(C(=O)NC2(CO)CCN(C(C3(S(N)(=O)=O)CC3)=O)CC2)c(F)n1 CCC(O)C(C)C(=O)NCCC1CCCN1C(=O)COc1ccccn1 c1(C(=O)NC2C(CNC(c3[nH]c(=N)sc3)=O)C2)cccc(C2CCC2)c1 C1(C(=O)ON2CC(C(C)(C)C)C2)CCCC(C(=O)Nc2sccc2C#N)C1 N1(C(C2(COCC)CCC2)=O)CCCC(F)(CNC(C2CC(F)(F)CS2)=O)CC1 C1(C(=O)Nc2ccc(OCC)nc2)CCC2CCCCC2N1 c1(C(C(=O)NCC(=O)NCC(=O)N(CCC(C)C)CC)C)ccc(F)cc1 C1(NC(C2C(C=C)OCC2)=O)CC2CCC(C1)N2C(=O)CN1CCNC1=N c1(CC)cc(C(N2CCC(CC)C2CNC(c2nn(C)nc2C)=O)=O)cc(Cl)c1 CC1CCCc2c(C(N3CCC(N(C)C(c4sc(F)cc4Cl)=O)C3)=O)cnn21 C(=O)(CS(F)(F)(F)(F)F)N(C1CCCN(C(=O)CCN(C)CCO)C1)C O=C1NCCC2(CN(C(=O)C3=CCN(C(c4ncccc4O)=O)CC3)C2)O1 Cn1cc(Br)c(C(N2CCCC(N3CCNC(=O)C3)C2)C(=O)NC2CCCC2)n1 c1(OC)cc(F)ccc1C(=O)NCC1(CNC(=O)Cn2nc(C)nc2C)CC1 CCCC(CC(C)C)C(=O)NC1CCC(COC(=O)CCN2CCC(OC)C2)C1 Cc1c[nH]c2ncc(C(=O)NC(C)(CNC(=O)C=Cc3ccco3)C3CC3)cc12 C1(F)(CNC(c2scc(C)c2)=O)CC2CCC(C1)N2C(c1nc(=O)n(C)[nH]1)=O c1(C(=O)NC(C2(O)CN(C(=O)CN(S(C)(=O)=O)C)C2)C)cc2ccsc2c(O)n1 c1(C(=O)NCC(C2CCCCC2)NC(c2c(OC)scc2)=O)cccc(N)c1N C12(C(=O)NCC3(C)CCCOC3)CC(CO1)N(C(=O)CN1CCCNC1=O)C2 N1(C(c2ncc(C)cn2)=O)CCC(N(C)C(c2cncc(C(C)C)c2)=O)C(C)C1 C1(C(=O)NC(c2nc(CC)[nH]n2)C2CC2)CCN(CC2CCOC2C)CC1 CCC(C)(C)C(=O)NCC(C)N(C(c1oc(Br)nc1C)=O)CC CC1CCCN(C(=O)CCC2CC(NC(=O)C(=O)NC3CCCC3)C2)C1CO c1(C(N(CC(CNC(C(CC=C)NC(C)=O)=O)C)C)=O)cnc2scc(C)n12 c1(OC(C(N2CC(CNC(c3cc(C)no3)=O)C2)=O)C)ccc(Cl)cc1C C1(CC(=O)NC(CCC)C2CC2)CCCN(C(C2(C3(O)CCC3)CC2)=O)CC1 C1(NC(C2C(C=C)CC2)=O)CC12CCN(C(c1cc(OCC)cc(=O)o1)=O)CC2 c1(C(N(CCCNC(=O)CN2CCCCC2=O)CC)=O)cccc(C#N)c1 CC(C)CCCCC(=O)NCC(C(C)(C)C)NC(C1(O)CC(C)(C)C1)=O C(CC(O)C(=O)NCCC(C)N(C(=O)CN(C)C(c1ccccc1)=O)C)SC CCC(CN(C)C)CC(=O)NCCN(C1CC1)CC.n12cc(cn1)c(=O)[nH]2 c1(CC)ccc(F)c(C(N2CCC(CF)(NC(=O)C(C)OCCC(C)C)C2)=O)c1 N1(C(C2C(C)C2C)=O)CC2(CC(NC(c3ncc([N+](=O)[O-])n3C)=O)CO2)C1 Cc1sc(C(=O)NC(C)C(CO)NC(=O)Cc2ccc(F)cn2)cc1S(N)(=O)=O N1(C(c2n(C)cnc2)C(=O)NC(C)(C)C)CCCC(O)C1 c1(NC(C)=O)cccc(C(N2CC3CC3(CNC(=O)CC3CCCO3)C2)=O)c1C CC(C(=O)NCC1CC1C(=O)NC1CCCCCC1C)S(C)(=O)=O C12COCCN1C(=O)C(=O)NCCn1ccnc12.C(C)(CN(S(C)(=O)=O)C)N.CC CC(CCCCO)NC(c1coc(CNC(C2CCC2C#N)=O)n1)=O c1(C(=O)NC2C(NC(C3C(OC)CC3)=O)CCC2)cc2cc(Cl)c(Cl)cc2[nH]1 C(C(COC)CC(=O)N(CC(C)NC(=O)Cc1cccc(NC(N)=O)c1)C)OC N1(C(C(C(=O)OCC)C(C)C)=O)CCC2(CC1)CCN(C(=O)CC(C)C(F)F)C2 C1(C)(C(=O)OC)CC12CCN(C(C1C3CCCC13)=O)CC2.C12CCCN(C1)C2=O N1(C(c2c(OC)c(F)ccc2)=O)CCC2(CCCN2C(c2cccc(=O)o2)=O)C1 c12cc(no1)CC(C)C1CN(C1)C2=O.C(=O)(C(CN(C)C)N(C)C)N.CSC CCCCC(CNC(=O)C(C)Cc1cccc(Cl)c1)NC(=O)Cc1cccnc1 N1(C(C2CN(C(=O)Nc3c(C)ccc(C)c3)C(CO)C2)=O)CC2CCCCC2C1 c1(C(=O)NCC2C3CC2N(C(=O)CCCC2CCC2)C3)cnc2ccccc2c1 c1(CC(=O)NC(CN(C(c2cc(C(F)F)[nH]n2)=O)CC)C)cn(C)nn1 CCC(CO)(C(=O)NC1CCC(NC(=O)C(O)C(C)(C)C)CC1)OC Cc1cnc(C(N2CCC23CN(C(c2cn[nH]c2)=O)C3)=O)c[n+]1[O-] CC1(F)CCCN(C(=O)C(CC(N)=O)NC(=O)CCOC2COC2)C1 C12(C(=O)OC(C)(C)C)CCC(C(=O)NCCc3ccccn3)(CC1)O2 C1(NC(c2ccccc2)=O)CCCCC12CN(C(=O)CN1CCCC1=O)CCO2 CC(C)CC(O)C(=O)N(CC(C)C(N1CCn2ccnc21)=O)C c1(-c2n(C)ncc2)cnc(Cl)c(C(=O)NCC2(O)COC2)c1 Cc1[nH]nc2cc(C(=O)NC3CN(C(c4ccc(N)c(F)n4)=O)CC3O)ccc12 N1(C(c2cc(C(C)C)on2)=O)CCCCC(C(N2CCCCC(N(C)C)C2)=O)C1 C(=O)(CCC(C)S(C)(=O)=O)N1CCN(C(C(CCC)CC)=O)C(C)C1 c1(C(=O)Nc2nnc(C(C)N)s2)ccc(N)c(OC(F)(F)F)c1 N1(C(COCC)=O)CCC2(CCN(C(c3c(C)oc(C)c3C)=O)CC2)C(C)C1 N1(C(c2c(OCCC)cccn2)=O)CC(C2(NC(c3nc(C)sc3C)=O)CC2)C1 C12(CNC(=O)CN3CC(=O)NC3=O)CCCC1N(C(=O)Cn1nccn1)CCC2 c1(OCC(=O)NCC2CCC2NC(=O)CN2C(=O)CNC2=O)cccc(O)c1 N1(C(C2C(CC(C)(C)C)C2)=O)Cc2n[nH]cc2C1C(=O)N1CCCC12CCCC2 C1(NC(c2nc(C(N)=O)sc2)=O)CCN(C(=O)CCn2cccn2)CCC1(F)F C(=O)(C(F)C(F)(F)C(F)(F)F)NC(C1(O)CCN(C(c2cnc(Cl)[nH]2)=O)CC1)C Cc1cc(C(=O)NCC(C)CNC(C2CC(N(C)C)C2)=O)nc2ccccc12 CN=c1cc(C(N2CC(NC(c3ccc[n+]([O-])c3)=O)C(C)(C)C2)=O)cc[nH]1 CN1CCN(c2ccccc2-n2cc(CN3CCCCC3C(=O)O)nn2)CC1 O=C(C#Cc1ccc(Cl)cc1)N1CCc2cc(C3CCC(=O)CC3)ccc2C1 N1(CC(=O)N(C(C)C(=O)NCc2ncco2)CCC)C(=O)CCC1=O c1(OC)cccc(I)c1NC(=O)CC1CC(Nc2ncc(-c3nn[nH]n3)cn2)C1 c1(C(=O)NCCC2CCN(C(=O)C=C3CCCC3)CC2)cccn2c(O)nnc12 C1(NC(C(C)NC(=O)C(n2cc(CCN(C)C)nn2)C)=O)CCCCN1C CC1c2ccccc2OC1C(=O)NCC1C=CCN1C(c1cnc(N(C)C)s1)=O C(=O)(C(C)CC(C)C(C)=O)NCC.c12cncc(c1)NSC2.N12CCN(CC1)C2=O N#Cc1cc(Cl)c(C(=O)NCC2(NC(=O)Cc3nc[nH]n3)CCOCC2)s1 c1(C(=O)NC(c2nc(NC(c3ncccn3)C)cs2)C)ccc(F)cc1 c1(C(N2CC(N(C(C(C)NC(CC)(C)C)=O)C)C2)=O)c(C)nn2c1CCCC2C c1(OC(C)C(=O)N(CCCN(C(=O)C(C)(C)C(N)=O)C)C)ccc2c(c1)CCC2 N1(c2cc(N3CCCC(C(=O)NC)C3)ncn2)CCCc2[nH]ccc2C1 Cc1cccc(NC(=O)C(C)N(CCNc2cncc(C(F)F)c2)CCO)c1 C1(N(C(C=CC)=O)CCCNC(c2ccc(CO)o2)=O)CCS(=O)(=O)C1 C1(C(N2CCC(CNC(C3CCC(C(=O)OC)CC3)=O)C2)=O)CCCCN1N=O C(=O)(C(C)CC(C)(C)C)N(C(C(=O)NCC1(C#C)CCOCC1)C1CC1)C C1(CNC(c2ccn(CC(F)F)n2)=O)CCN(C(=O)C2=NOCC2)CCC1(F)F N1(C(c2c(Cl)cn(C)n2)=O)CC(NC(=O)CNC(=O)NC2CC2)C2(CCC2)C1 C12(NC(CSCC(=O)OCC)=O)CCCOC1CCN(C(=O)CC)C2 CC1CCN(CC(=O)NCC(O)CCN(C(=O)C(F)(F)CO)C2CCCC2)CC1 C1(C(N2CCCC2CNC(c2cccc(COC)n2)=O)=O)C2CC3C(C2=O)C13 N1(C(CCCCC#C)=O)CCC(C(=O)NC2CC(C)(C(=O)OC)C2)CC1(C)C c1(C(=O)NC2CC(CNC(C=CCOC)=O)C2(C)C)cc(Cl)c(F)cc1Cl N1(C(c2c(C)cccn2)=O)CC(NC(=O)C(C)(C)c2cc[nH]n2)CC(C)C1 CC1(NC(C23CC(CO)(C2)C3)=O)CCN(C(c2cocn2)=O)CC1 Cc1c(Cl)ccc(C(=O)NC2(C3CN(C(=O)Cc4c[nH]ccc4=O)C3)CC2)c1O C1(OC)CC(NC(=O)CCCN2C(=O)CCC2=O)CN(C(C2CNC(=O)C2)=O)C1 CCCCCC(C)(CC)C(=O)N1CCC(=O)N(C)CC1.C1(CCN)NC(=O)NC1=O c1(C(N2CC(CNC(C(C)n3cccn3)=O)C(C)C2)=O)ccc(F)c2ccsc12 C1(C(=O)NCCC(C)(C)NC(=O)CNC(C2CCCC2)=O)CCS(=O)CC1 c1(C(N(C)CC2(CC(C)C)CC2)=O)c[nH]nc1CNC(=O)CC1CCC(C)O1 N1(C(c2ccon2)=O)CCN(C(=O)C(F)n2ccnc2)C(CC(F)(F)F)C1 C1(NC(c2c(C)noc2)=O)C=CCN(C(=O)CCN(CC(C)C(C)C)C)C1 C1(C(N(C)Cc2ccon2)=O)CCN(C2CCCNC2)C1 CCC(CN(C)C)C(=O)NCCC1(C)CCN(C(=O)C=CC(C)(C)NC(C)=O)C1 C(=O)(C(C)(C)c1cnco1)N(CC(C)O)CC(F)F n1(CC=C)cc(C(=O)N(C2CCC(NC(=O)C=CBr)C2)C)nn1 Cn1ncc(Cl)c1CNCCC1CCCN(C(=O)OC(C)(C)C)C1 c1(C(=O)NC(CNC(c2c(C)ccnc2O)=O)C2CC2)cc2ccsc2c(O)n1 N1(C(C(C)CC2CCCC2)=O)CC(NC(=O)CC2(CO)CCOCC2)CC1(C)C c1(OC)nc(C)ncc1C(N1CCCC1CNC(c1cc(C)[nH]c1C)=O)=O CCC(C)(C)C(O)C(=O)N1CCC(C)N(C(C23CCC(C2)OC3)=O)CC1 N1(C(C(C=CCCC)O)=O)CC(C)C(N=c2nc(C)[nH]s2)C(C)C1 c1(C(C)C)ccc2c(Cl)c(C(N3CCCC3CN(C(=O)CC(C)F)C)=O)sc2c1 CCC1=C(C(=O)NC2CC3CCCC(C2)N3C(=O)CCCCO)CCCO1 C1(O)(C(N(C)Cc2ccccc2)=O)CCN(C(C2CCCCC2N)=O)CC1 C1(NC(COCCCOC)=O)CC2(CCN(C(=O)C(C)(C)CC3CC3)C2)C1 N1(c2ncnc(-c3cc4cn[nH]c4cn3)n2)CCC2(CCCc3ccccc32)C1 C1(OC)CC(C(=O)NCC(CO)NC(=O)CCc2nc(C)cs2)CC1OC N1(CC)CC(NC(=O)CC=CCNC(C2COCCN2C)=O)CC1=O C1(C(=O)NC(c2cn(C)nn2)C(=O)NC(c2nnc(C)o2)C)COCCC1C C1(C(=O)NCc2c(C(=O)NC(C=C)(C)C)c[nH]n2)C2CCC(F)C12 N1(C(C#C)=O)CCC2C(CCN2C(c2ccnc(OC)c2Cl)=O)C1 Cc1ccc(C(=O)NCC2(F)CCCN(C(c3cnsc3)=O)C2)c(C)c1 C(C(=O)NC1CCOCC1)(C(C)CC1CC1)N(CCC)CC1CCCOC1 c1(OCC(=O)OC)ccnc(NC2CN(C3CCC3)C2)n1 Oc1ncnc(SCOCC(F)(F)C(F)(F)F)c1I c1(C(=O)NCC2N(C(C(CC)OC)=O)CCCC2)ccc2c(n1)CCCC2 N(C(=NCc1ccc(F)c(Br)c1)N(C)CC1CCCN1CC)C(CC)C Cc1cnc(C(=O)OC2CC(C3=CCOC3)C2)cc1C C(C(C)C(=O)N1CCCC1CN(C(=O)COCc1ccnn1C)C)OCC CCCCS(=O)(=O)CC(=O)NC1CCN(C(=O)C(F)(F)CCn2cccn2)C(C)C1 C(=O)(C(C)(C)CC(=O)N1CC(NC(=O)CCc2cccn2C)CC(O)C1)OCC N1(C(C(CC)F)=O)CCCC(CCNC(c2ccc(N)c(F)n2)=O)CC1 C1(C)(NC(CCc2nc(C)c(C)[nH]2)=O)CCN(CCc2cnccn2)CC1 c1(C(N2C(C)CC(NC(c3cc(CC)no3)=O)C2)=O)ccc2nn[nH]c2c1 c1(-c2nc(CNC(=O)CCCCNC(N3CCCCC3)=O)[nH]n2)cc(O)ccc1F n1(C(C)C)cc(C2CC2C(=O)NC2(C)CN(C(=O)C(C)CO)C2)cn1 N1(CCC)CCCCC1C(=O)NC1CCCCC1CNC(=O)CCc1cnn[nH]1 c1(SCCC(=O)NC(C(C)NC(c2c(CC)cno2)=O)CO)ccc(Cl)cc1 c1(C(=O)NCCC2(C(N3CC(OCCC)C3)=O)CCC2)scnc1C CCC(CC)C(=O)N(C)CCOCCN(C(=O)C(C)(C)n1cnnn1)C c1(CC(=O)NC2(CC)CCCN(C(=O)CC3CC3)C2)ccc2cnccc2c1 C1(NC(CCNC(=O)C=CCl)=O)CC(NC(c2cc(Cl)ns2)=O)C12CCC2 CC1(C)CCCC1(C)NC(C1C2CC3C(C2NC(c2cc(CO)on2)=O)C13)=O CCCC(C)C(C(=O)NCC)N(C1CCN(C2CC2)C1)CC(C)(C)C c1(OC)ccc(NC(c2ncccc2CN)=O)cc1CSc1ccc(C#N)cn1 C1(CC(N2C(C(=O)NCC3(N(C)C)CCC3)CC2)=O)CCC(=O)C1 C(=O)(C1CCCc2sccc21)N1C(CC)(CC)CC(NC(C2CS(=O)(=O)C2)=O)C1 C1(C2(O)CN(C(=O)CCC(N)=O)C2)(CNC(c2nc(C)sc2C)=O)CC1 c1(C(=O)NC2C(NC(c3ccc(C(C)=O)cc3)=O)CC2)cnc2n1CCCC2C c1(CC(C(=O)OCc2sccc2I)O)cc(Cl)ccc1Cl CCCCCC(CC)C(=O)NCC(C)N(C)C(c1cc(C)nc(C(F)(F)F)n1)=O c1(C(=O)NC2COCC2n2cc(CNC3CCCO3)nn2)nc2c(s1)CCCC2 c1(C(N2CCC(C)C2)C(=O)NCC(C)C)cccc(C#N)c1.C1(NC)CCOCC1 N1(C(COCC)=O)CCOCC(NC(c2cnoc2C2CC2)=O)C1 c1(N2CCC(C)S(=O)CC2)nc(=N)[nH]c(=NCc2nnc(C(F)F)s2)[nH]1 N1(C(C(C)(C)c2ccns2)=O)CCC(NC(c2ccc(F)c(N)c2)=O)C(CO)C1 N1(C(c2ccc3c(c2)N(C(C)=O)CCC3)=O)CCc2nc(C#N)ccc2C1 N#Cc1ccc(CNC23CC(NC(=O)C(=O)C4CC4)(C2)C3)cn1 CC1(C)CN(C(c2cocn2)=O)C(CNC(c2nccnc2C(N)=O)=O)CO1 C(C)(CCC(=O)NC(C)CC1CN(C(=O)C(C)CN(C)C)C1)OC C=CC1(C(=O)NCCCn2nccn2)CCN(C(C)=O)C1 c1(OCC(C)(C)C)ccc2c(c1)CCN(C(=O)C(C1CCCOC1)N)C2 c1(CC)cnc(-c2nc(-c3ccc(N)cc3)nn2CCCO)cn1 N1(C(CCC2C(C)=NOC2=O)=O)CC2CCC1C2NC(c1cc[nH]c1C)=O CCC(CC)(C(=O)N1CCC(OCCNC(C2(CC(F)F)CCC2)=O)C1)C(C)C N1(C(c2ccncc2Cl)=O)CC2CCC(C1)N2C(=O)C(F)(F)c1nccs1 N1(C(C2(C=C)CCC2)=O)CC(NC(=O)CCc2ncc(F)cn2)C(O)C1 C1(CNC(=O)Cc2csc(-c3ccoc3)n2)CN(C(c2cncnc2)=O)CCO1 c1(C(N2CC3CC3C2)=O)cnc2c(-c3cccc4ncccc34)cnn2c1 N1(C(c2n[nH]c(C)c2O)=O)CC(Nc2ncc3c(n2)CCOC3)CC2(CCC2)C1 C(=O)(C1=C(Cl)CCOC1)NCCC1N(C(C2(C)C(C)(C)C2)=O)CCCC1 c1(CC)c(Cl)nc(C(C)(C)C)[nH]c1=NCC1CCCN1C(=O)C(C)SC O=S(=O)(c1ccc(NC2CC23CCCC3)c(F)c1)NC1CC(CF)C1 N1(C(=O)COCC(F)F)CCCC2C1CCN2C(C1CC1F)=O n1(CC(=O)NC(CCNC(CCC(C)OC)=O)C)c(C)cc2ccccc12 c1(-n2cc(C(=O)NC(c3cc(CO)on3)C)nn2)cccc(Cl)n1 C(=O)(C(F)C(C)(C)O)NCCC1CC(C(=O)NC(c2ccc(C)s2)C)C1 CCCC(C(=O)NCc1nocc1C(=O)NCCC1CC2CCC1O2)OC CCC(C)C(C(=O)NC1(CC)CCOCC1)N(C)C(c1nonc1N)=O C1(NC(c2c(NC(CC)=O)cccc2)=O)CCN(C(c2occc2C)=O)CC1O C1(NC(C2NC3CC2C3)=O)CCC(C(N2CCCC2)=O)CC1 Cc1cc(C(=O)NCCN2CCN(C(c3nc(=N)cc[nH]3)=O)CC2)nn1C(C)C C(CC(C)C(=O)NCC1(OC)CCN(C(C2C=CCC2)=O)C1)=CCC C(C(C(C)C(C)C)NC(=O)Cn1cnccc1=O)NC(c1cccc(SC)c1)=O c1(C(=O)NC(C(C)NC(C2CCCN2C(=O)C2CC2)=O)CO)c[nH]ccc1=N N1(C(CCC(=O)OC)=O)CCC(NC(=O)Cc2cccc(OC)c2Cl)C(O)C1 N1(C(Cc2c(C)n[nH]c2)=O)CC(C(=O)NC2(C(O)CO)CC2)CC12CCC2 N1(C(C2C3CC(=O)CC32)=O)C2CCC1CN(C(C1Cc3cccnc3C1)=O)C2 CC(C)C(=O)C(=O)N1CCOC(CC(=O)Nc2ccc(CO)nc2)C1 Cc1n[nH]c(C)c1C(C)C(=O)NCC(C)(C)NC(=O)Cc1ccoc1 c1(OCC)ccccc1-c1nc(Cc2cn[nH]c2)n(C2CCSC2)n1 N1(C(C(C)C(F)F)=O)CCC(O)C(NC(c2c(NC(N)=O)cccc2F)=O)C1 C(=O)(C1=CCC(C)CC1)N(CCC(C(C)C)NC(=O)Cc1ccoc1)C N1(C(C(CC)=O)=O)Cc2cccn2CC(C(=O)NCc2ccc(C#N)c(C)c2)C1 CC(CNC(=O)CCn1cnnn1)C(=O)N(C)CC1CC1C CCC(C)C(C(=O)NCc1ncc(CO)[nH]1)N(C(=O)C=Cc1cc(C)no1)C Cc1cccc(CC(=O)Nc2ccc(-c3nn[nH]n3)cc2C)c1C Cc1ccnc(O)c1C(N1CCC=C(CNC(C2CS(=O)(=O)C2)=O)C1)=O CC1CC2CN(C(c3cn(CCNC(c4cccnc4)=O)cn3)=O)CC12 c1(C(N2CCNCC2c2ccc(Br)cc2)=O)cccc(O)c1O c1(CNC(c2ccc(N3CCCCCC3)cc2)=O)cccc(-c2ccccc2)n1 N1(CC(C)NC(c2c(C)cc[nH]2)=O)CCN(c2ccccc2)CC1 c1(CNC(c2ncn(C)n2)=O)cccnc1CNC(C1C(C#N)C1(C)C)=O CC(F)(C(=O)N1CCCC(N2CCN(C(C3(C#N)CC3)=O)CC2=O)C1)C(F)(F)F c1(CN(C(C2CC(=C)C2)C(=O)NCCC2(C)CC2)C)csc(C)n1 c1(C(=O)NCC(CNC(c2c(C)ccn2C)=O)CO)cccc2c1C(=O)CC2 N1(C(C2(CCC)CC2)=O)CCCCC(NC(C2(C(=O)NC)CC2)=O)C1 c1(OC)cnc(F)cc1C(=O)NC1CCCCC1NC(=O)Cc1cnsc1 C1(O)(CNC(C(CO)NC(COCC=C)=O)=O)CC(C)(C)C1 C1(C(=O)NCc2cnccc2Cl)CCC2CCC1N2C(=O)C1=C(Cl)CCC1 N1(C(C2CC(SC)C2)=O)CC2(CCN(C(c3cc(C)n(C(C)C)n3)=O)CC2)C1 C(=O)(CCC(=O)NCC1CC1)NCC1C(NC(C=CC(=O)OCC)=O)C1 C(=O)(CCC(C)CN(C)C)NC1CCC(CNC(Cc2c(C)con2)=O)CC1 S(=O)(=O)(C1CCOCC1)N1CC2C(CNC(c3ccnnc3)=O)(C2)C1 c1(C(=O)NCC(CNC(CNC(N)=O)=O)CO)cc2cc(Cl)ccc2[nH]1 c1(OC)ncccc1NC(=O)CC1(OC)CN(C(C2CC(C)CO2)=O)C1 C(=O)(C1CCCn2cncc21)NC1(COC)CCN(C(=O)CCc2cnco2)C1 CCC(C)(COC)C(=O)Nc1cncc(CNC(=O)CCc2ncnn2C)c1 C1(CNC(CCc2cc(C)no2)=O)CC(NC(=O)C=Cc2cocn2)CCO1 Fc1ccc(OCCN=C(NCC(F)(F)C2CC2)NCC2CCCCC2)cc1Cl C(=O)(C1(C)CCn2c(C)nnc21)NC(CCCNC(C1(CCOC)CC1)=O)C Cc1ccc(O)cc1CN1CCC(C(N2CCCC(N(C)C)C2)=O)C(O)C1 C(=O)(C1=NOC2(CCOC2)C1)NC1CC2(CC(NC(CCCC#CC)=O)C2)C1 N1(C2Cc3n(-c4ccc(OC)cc4)ncc3CC2)CCOC2(CCS(=O)(=O)C2)C1 CC1(C(=O)NCC2CCCN2C(=O)C(=O)NCC2CC2)CCC(=O)NC1 N1(C(C(C)(N(C)C(c2cncc(CO)c2)=O)C2CC2)=O)CCC2=C(CCCC2)C1 C1(C)(NC(C2OCCN(C)C2)=O)CCCN(C(=O)CNC(C2CCCN2)=O)C1 C1(N(S(=O)(=O)CC2CCCNCC2)C)CC2CC1C1CCCC21 N#Cc1cc(CNC(=O)Cn2cc(CNC(=O)COCC(F)F)nn2)cs1 c1(C(=O)NCC2(O)CN(C(c3cccc(NC)n3)=O)C2)cnc2ccccc2n1 N1(C(C(=O)N(CCCNC(c2cc(Cl)n[nH]2)=O)CC)C)CCCCCC1 CCC(N=c1[nH]c(=NCC2C3CCC(F)(F)C23)[nH]c2c1CSC2)c1ccc(C)o1 C1(C(=O)NCc2c(C(C)C)noc2)CCC2(CC2)N1C(C1CCC(O)C1)=O c1(C(N(CC(C)NC(=O)Cc2cnc(C)[nH]2)CC)=O)onc2c1CCCC2 c1(C(=O)NC(COCC)C)n[nH]c2c1CN(C(c1c[nH]c3ncccc13)=O)C2 N1(CCC)CCCC1C(=O)NC(C)CN(C)C(C1CC12CC2)=O N1(C(C=CCC)=O)CCC(C(N2CCC(CCN(C)C)C2)=O)(CF)C1 C#Cc1cnn(CC(=O)NCC(C2CCOC2)NC(C2(CF)CC2)=O)c1 c1(OC)ccc(S(=O)(=O)NC2CCCC(O)CC2)c(C(F)F)c1 Cc1cc(S(C)(=O)=O)ccc1CNC1CCC2(C1)CN(C(c1ncsc1C)=O)C2 N1(C(CCCCCC=C)=O)CCN(C(=O)CCCCC(C)=O)C2COCC12 c1(C(=O)NCC(CNC(C(C)OC)=O)O)csc(C)c1C C1(CSC)CCN(C(C2CCCN2C(=O)C(=O)NC2CC2)=O)C1 c1(C(=O)NCC(CNC(c2c(CC)con2)=O)OC)ccc(-n2ccnn2)cc1 c1(OCC)ccc(N)c(C(=O)N(C2CCN(C(=O)CC3COCCO3)CC2)C)c1 C(C)(CCCC(=O)NCCC(F)F)NC(C=Cc1cc(C)no1)=O C(=O)(CC(C)(C)CN(C)C(C1CCOC(C)C1)=O)NCc1n(CC)cnn1 c1(C(=O)NCC(CC)(C)NC(=O)CCCCSC)ncncc1Br C1(C(N(CC(O)CNC(c2nsnc2O)=O)C)=O)CCS(=O)(=O)C12CCC2 N1(C(CC2CN(C)C2)=O)CC(N(C(=O)CCN2CCC(C(N)=O)CC2)C)C(O)C1 C(CC(C)(O)CNC(=O)CCn1cc(CCOC(C)=O)nn1)OC CC(C)=C=CC(=O)N(C)CCC1CCN(C(=O)C=CC2CC2)CC1 N1(C(CC=CCC)=O)CCC(NC(=O)Cc2ccno2)C2(CCC2)C1 Cc1cc(F)c(C(=O)NC2CCC2NC(C2(C)CC=CC2)=O)cc1F CC1CC(NC(=O)CC2CCCCC2O)CN(C(=O)CCc2cnccn2)C1 CC(c1ccco1)=CC(=O)NCC1CCCC(CNC(c2cc(O)nn2C)=O)C1 Cc1ccc(NC(C2CC3CC2N(C(=O)C(C2CCCCC2)O)C3)=O)c(C)c1 C(C(CO)C(F)(F)F)NC(CCC1(C)CN(C(c2cn(C)nc2)=O)C1)=O c1(C(N2CCC(CNC(c3cc(C)sc3)=O)C2)=O)cc2ccccc2c(=O)n1C N1(C(C=Cc2cn(C)nc2)=O)CCCOC(CNC(=O)CCN2CCOC2=O)C1 c1(C(N(C2CCN(C(C(C)Cc3ccnn3C)=O)C2)C)=O)cc2n(n1)CCCO2 C(=O)(C(C(F)(F)F)C(F)(F)F)NC(CN(C(CCc1onc(C(C)C)n1)=O)C)C c1(N2CCC(OCCC)CC2)nc2c(c(=NCc3cccc(C)c3F)[nH]1)SCC2 C(CC(C(=O)N1CCCC(CSC)C1)NC(=O)C(C)OCC1CC1)SC N1(C(c2[nH]cc(CC)c2)=O)CC2(CCCC2NC(c2cn(C)nc2C)=O)C1 C=Cn1nncc1C(=O)NC(C1(O)CCN(C(=O)CCC(=O)c2cccs2)C1)C C1(CC)CCc2sc(C(N3CC(CCNC(=O)C(C(C)(C)C)OC)C3)=O)cc2C1 C(=O)(CCC(=O)N(CCCN(C)C)CCC)NC(c1cnc(C2CCCO2)s1)=O C(=O)(C(C)(C1CCC1)NC(=O)CC1C=CCCC1)N(CCOC)CCOC C1(O)(CC(=O)NCC2CCC2CO)CN(C(c2cc(CO)on2)=O)C1 Cc1cc(Cl)cc(N)c1C(=O)NC(C)CNC(=O)CCOc1ccccc1Cl N1(C(C(CC)OC)=O)CCCC2(C1)CC2.C(=O)(CC(C)C1CC1)NC N1(C(C(=O)OCCCC(=O)NCCN(C)C)=O)CCCC(N(C(C)=O)CC)C1 CON1CC(C(N2CCC(C(=O)NCC(=O)NC3CCC3)C2)=O)CC1=O C(=O)(C#CC1CC(F)(F)C1)NC1CCN(C(c2c(N)c(Cl)ccc2F)=O)CC1F CN1CC(C)(NC(C2CCOC2CNC(c2cnc(N)cn2)=O)=O)CCC1=O N1(C(c2ccc(C)o2)=O)CCN(C(=O)CCC2CC2CC2CC2)CC1CF C1(CC(=O)OC(C(C)c2ccsn2)=O)CC2CCC1N(CCOC(C)(C)C)C2 c1(CNC(C(OCC)OCC)=O)occc1C(N1CCC(CF)C1)=O c1(C(=O)NC2(C)CCCN(C(C3CCCC3C(F)F)=O)C2)ccnc2ncnn12 CC1CCn2cc(C(=O)NC3CC(CCNC(=O)CNS(N)(=O)=O)C3)nc2C1 N1(C(c2c(C)oc(CO)c2)=O)CC2CC(NC(c3cc(CO)oc3C)=O)C2C1 C1(CC)CC(C(N2CC(NC(c3c[nH]nc3[N+](=O)[O-])=O)CC2C)=O)CCC1=O c1(OC)ccc(NC(c2ncccc2C)c2nnnn2CC2CCOC2)cc1C c1(CN2C(C(N(C)C)=O)CC3CC32)ccc(F)c(C#N)c1 C=CCCC(C)(C)C(=O)NC1CC2C(C(=O)NC3C4CCCCCC34)C2C1 N1(C(c2c(C)cc(C)o2)=O)CCC(NC(c2ccc(C(C)C)c(F)c2)=O)C(F)C1 c1(C(N2CCCC(N(C)C(C3CC4(C3)CC43CC3)=O)C2)=O)c(F)cc(F)cc1Cl Cc1sc(=O)n(CC(N2CCC(O)(CNC(=O)C(C)(C)C#N)C2)=O)c1C CC1CN2CCN1CC2C(N1CC2C(CNC(C3(c4cccs4)CC3)=O)C2C1)=O C(C(C)(C)CC(=O)N1CCOC(CNC(=O)CC2CSCCS2)C1)OC c1(C(N2C(C3CCN(C(=O)C=CC=C(Cl)Cl)C3)CCCC2)=O)nnc(O)nc1O C1(C(=O)NCC2C(C(N3CCCC3COCCO)=O)C2)CC12CCCC2 Cc1cc(C)n2c(CNC(=O)NC3CCOC(c4cccc(Cl)c4)C3)nnc2n1 C=C(C)C(CC(=O)N1CC2CC2(CNC(c2ccnn(C)c2=O)=O)C1)OCC C=C(C)C(C)(C)C(=O)N(C)CC1CN(C(=O)CN(c2ccncc2)C)CC12CC2 C=C(C)CC(=O)NC1CN(C(=O)C(C)CSCc2ccccc2)C1 N1(C(c2nc(CCC)oc2)=O)CCN(C(C2SCCS2)=O)C(C)CC1C C(=O)(C(C)(C)C1=CCN(C(c2ccc(C#N)s2)=O)C1)NC1CC(C)(C)OC1 c1(C(=O)NCCN(C(=O)C(Cl)=CCl)CCC)cccc(-n2cccn2)c1 C(C(CC(C)C)C(=O)N1CC(CC(=O)N(CC(O)C2CCC2)C)(OC)C1)OC CCCCC(O)C(=O)NC1CC(CNC(c2cnc(Cl)n2C(C)C)=O)C(O)C1 N1(C(c2c(C(=O)OC)scc2)=O)CC2CC(NC(=O)C#CC3CC3)C1C2 N1(C(C=Cc2n(C)ccc2)=O)CCC2(CCN(C(C3CCCC(C)(C)C3)=O)C2)C1 C1(NC(C2(SC)CN(C(C3CCN(C)C3)=O)C2)=O)CCCCCC1F c1(C(N2C(C(=O)NCCCCCC)(CC)CCC2)=O)ccc2cncn2c1 C1(C(=O)NC2CC(C)N(C(C3CCS(=O)(=O)CC3)=O)C2)CCCCS1(=O)=O N1(C(C(C(C)(C)C)OC)=O)CCC2(CC1)C(NC(=O)CN1CC=CC1)CS2(=O)=O C1(CNC(C(CC)(F)F)=O)CC2COCC2N1C(=O)C(CC)CCOC c1(C(=O)NCC(CO)NC(c2c(C)[nH]c(C)c2C)=O)coc2c(F)cc(F)cc12 c1(CC(=O)NC)ccc(C(N2CCN(C(=O)C(C)O)CC2)=O)cc1 C1(CNC(CCCC(N)=O)=O)CC2CCC(C1)N2C(C1CCCCC1O)=O c1(C(N2C(C(=O)Nc3ccccc3)CCC2C2CC2)=O)cc2ncccc2[nH]1 C(Cc1cnsn1)(C(=O)O)NC(c1cncn1-c1ccccc1)=O c1(C(N2CC(NC(c3n(CC)ccc3)=O)C2)=O)ccc(-c2cscn2)cc1 C#CCCC(=O)NCC(CC)NC(c1ccc(C2CCOC2)s1)=O c1(C(N(CCCNC(=O)Cn2cncn2)CCC)=O)cc[n+]([O-])cc1 C1(NC(C(C)=CC)=O)CCCC(CNC(=O)COC)C1 C1(C(N)=O)(CNC(CCOCCC)=O)CN(C(=O)C(C)CC2CC2)C1 C12(C(=O)Nc3c(CC)nsc3)CC(CN(C(=O)C(C)NC=O)C1)C2 c1(C(=O)NCC2(C)CC(NC(c3ccsn3)=O)C2)ccc2ccccc2c1F N1(C(C2(CCOC)CCC2)=O)CCC2CCN(C(=O)CSC3CC3)C2C1 C12(C(N(C)CC3CCN(C(c4ccc(SC)s4)=O)C3)=O)CCC(C1)C(C)(C)O2 C(C)(CCC(=O)NC1CC2(CC2)C1)NC(C(C1CCCC1)OC)=O C(=O)(N=c1[nH][nH]c2ncccc12)C1N(C)CCCC1.N12CC(CC(F)C1)C2=O CCC(CC)CC(=O)NCC1(CNC(=O)C(c2cc(F)cc(F)c2)C)CC1(F)F N1(C(C(C)CO)=O)C2CCCC1CC(NC(c1coc(C(N)=O)c1)=O)C2 Cc1cccc(F)c1C(N1CCC(CNC(=O)CCCC(C)C)C1)=O CC(O)(CC(F)F)C(=O)N1CCCN(C(c2ccc(O)nc2)=O)CC1 N1(C(C2N(C(C(C)N(C)C)=O)CC=CC2)=O)CCOCC(C)(O)C1 c1(NC(=O)NCC(c2ccccc2C(F)(F)F)O)ccc(NC2CC2)cc1 N1(C(C2N(C)CCC2)=O)CC(CO)C2(C1)CN(C(=O)CSc1cn[nH]c1)C2 c1(C(=O)NCC2C3CN(C(C(CC)=CC)=O)CC32)cc(=O)c(OC)cn1C C1(CNC(CN(C)C2CC2)=O)(NC(C2CCCC2N(C)C)=O)CCCCC1 CCCS(=O)(=O)CC(=O)NCC1(C2CC2)CCN(C(c2nc(C)sc2C)=O)C1 N1(C(c2cc(SC)c(C)o2)=O)CCCC12CCN(C(C1CCC(C)(C)O1)=O)C2 c1(C(=O)NCC2N(C(C=C(C)C3CC3)=O)CCC2C)cccc2cncn12 C1(C(=O)NC(C=C)C(F)(F)F)CN(C(=O)C(C)(C)CO)CC(C)O1 N#Cc1cccc(NC(=O)CN2CC3CC2CN3C(C2CC23CCSCC3)=O)c1 c1(C(=O)NCC2C(NC(C(COC)COC)=O)CCC2)c(O)nnc2c1CCCC2 c1(N(c2cc(-c3c(SC)ccnc3)[nH]n2)C(=O)C(C)(C)C)ccc2c(c1)OCO2 C1(NC(C2CC(CC)OCC2)=O)CCN(C(c2nn[nH]c2C(F)(F)F)=O)C(C)C1 O=C(CS(=O)(=O)CC(F)(F)F)NCC1CCCN(C(c2cnnn2C2CC2)=O)C1 N1(C(C2(Cc3ccccc3)CC2)=O)CCCC2CN(c3ncnc(Cl)c3F)CCC12 c1(C(=O)NC2CCOCC2NC(C2(F)CC=CC2)=O)cccc(C#CC2CC2)c1 CC(C)CC(O)C(C)C(=O)NCC#CCNC(c1cccnc1N(C)C)=O c1(OC)ccncc1C(=O)NC1(C)CCN(C(C2C=CCC2)=O)C1 CC1(CCNC(c2n[nH]c(C3CC3)n2)=O)CCN(C(c2csc(C3CC3)n2)=O)C1 CC1(C)CCN(C(=O)Cn2ncccc2=O)C(C(N2CCC(F)(F)CC2)=O)C1 C1(C(=O)NC(C2(O)CN(C(c3ccc(F)c(F)c3)=O)C2)C)CC2CCCC(C1)C2 N1(C(CSCC#C)=O)CCC(C)(C)C(C(=O)NCC2(C)CCOC2)C1 C#CCC(CC(F)F)C(=O)NC(COC)CNC(c1c(Cl)cnn1C)=O c1(OC)ccc(CC(N2CC3CC2(C(=O)O)CO3)=O)c2ccccc12 c1(C(N2C(C(N(C(C3CCOCC3)C)C)=O)C(C)C2)=O)ccc(O)c(F)c1 C1(CNC(c2cccc(SC)c2)=O)CN(C(=O)CC2CC(N(C)C)C2)CCCO1 N1(C(C2CC(NC(C3CCN(C)C(=O)C3)=O)C2)=O)CC2(C1)NC(=O)NC2=O c1(OCC(=O)NCC(C2CC2)NC(C2CCCCO2)=O)ccc(F)cc1 N1(C(c2c(C)nns2)=O)CCC(NC(C2(Cl)CC2C(=O)O)=O)CC1 CC1(C)OCC2CC12C(=O)NCC#CCNC(c1cc(-c2ccncc2)[nH]n1)=O C(=O)(CS(=O)(=O)C(C)C)NCCCN(C(C1Cc2nncn2C1)=O)CC c1(CC(=O)NCCN(C(C2(n3cccn3)CCC2)=O)CC)cnn(CC)c1 c1(NCC(=O)NCCC2CCN(C(c3cc(C(F)(F)F)no3)=O)C2)ccccn1 c1(CC)cc(C(=O)NC2C=CC(CNC(=O)C(O)CSC)C2)c(C)nn1 C1(C(=O)NCCC2CCN(C(C(CCCC)C)=O)CC2)C2CCC3C(C2)CC13 C#Cc1ccc(N)c(C(=O)NCC2(C)CCCN(C(c3nccc(C)n3)=O)C2)c1 C1(NC(=O)C(O)CN2CCCC2)CN(C(c2nn[nH]c2Cl)=O)CC2(CC2)C1 C12(C(=O)NCCN(C(=O)C(F)(F)c3nc(C)cs3)CC)CCC(OC)C1C2 CC(C)C(C(=O)NC(c1nc(C2CC2)cs1)C(=O)NCC(F)F)N1CCCCC1 C1(C(N2CCC(CO)(NC(C3CCCN3C(=O)OC)=O)C2)=O)(CC)CCCCC1 N1(C(c2c(Cl)cn(CC)n2)=O)CCN(C(c2ccc(C)s2)=O)CC1C1CCC1 c1(OC)cncc(NC(C2CCN(Cc3cccc(-c4nn[nH]n4)c3)C2)=O)c1 CCCCS(=O)(=O)NCC(N1CCC(C(C)(C)C)(CNC(=O)CC(C)F)C1)=O C1(C(=O)NCC2SCCS2)(CNC(C2CCC(=O)C2)=O)CC12CCC2 C(=O)(CCCC(=O)N1CC(C(N2CCC(F)C(F)C2)=O)C(C)(C)C1)OCC S(=O)(=O)(c1ccc(N2CC3COCC(C3)C2)cc1Cl)N1CCC(C)C(C)(C)C1 n1(CC)ncc(C(N2CCCC(NC(c3ccc(CCO)cc3)=O)C2)=O)c1Cl N1(CC(=O)NCCCC)CCC(OCCCNc2cnn(C)c2)C1 CC(CC(=O)NC(C(=O)NCC1CSC1)C1CCC1)n1cccc1 N1(C(c2cc(O)cc(F)c2)=O)CCCC2(C1)CN(C(C1(CF)CC(F)(F)C1)=O)C2 C(=O)(CCC[N+](=O)[O-])N1CCC(CC(=O)NC)C1 c1(SCC)ccc(NC(=O)CC2(NC)CCC2)cc1[N+](=O)[O-].N12CCC(C1)C2=O c1(C(=O)NCC2(O)CCN(C(c3cc(Cl)c(Cl)s3)=O)C2)cccn2ccnc12 C(=O)(CS(=O)(=O)CCOC)N1CCC(N(CCC)C(c2nccc(C)n2)=O)C1 c1(C(=O)NCC(O)(C(F)(F)F)c2ccc(Cl)cc2)ccc(N2CCOCC2)c([N+](=O)[O-])c1 Cc1cc(C(=O)NC2(C)CCN(C(=O)CN3CCC(F)(F)C3)CC2)cc(C)c1N n1(CCC)cc(C(C(=O)Nc2ccccc2)N(C2C3CCCC23)C)cn1 N1(C(C(C)OCC=C)=O)CC2CC(C1)C2NC(=O)C(F)C1CC1 Cn1nnc2c(C(=O)Nc3cncc(C(C)(F)F)c3)cccc12 C1(C(N2CCC(NC(C3CCN(C)C3)=O)C2)=O)CC12CCOCC2 c1(CCNC(C2CCN(C(C3(C)C(C)CCC3)=O)CC2)=O)c[nH]c2ccccc12 CC(CNC(=O)C(C1CC1)C1CC1)C(=O)N1CC(O)(c2cc[nH]n2)C1 Cc1cnn(CC(=O)NCC2(O)CC(C(=O)NCc3ncc(C)o3)C2)c1 N1(C(c2nc(C)on2)C)CCC2(CN(C(=O)Cn3nccc3C)CC(C)O2)C1 N1(C(C2=NOC(CNC(=O)CSC3CC3)C2)=O)CC2CCCC(O)C2C1 c1(C(N2CCOCC2c2nnc(C)o2)C(=O)NCCCSC)nc(Br)cn1C N1(C(CSCCC=C)=O)CCC(C2CC2)C1C(=O)NOC(C)(C)C N1(C(c2nccc(C#C)c2)=O)CCC(NC(C2CC(C)(C)CO2)=O)C12CCC2 C(CCC(=O)NC1CCCCC1)N(C)C(C1C=CCC1)=O C(CO)(C(=O)N(CC(C)(C)NC(=O)CCOc1ccccc1)C)OC CC1CCC(=CC(N2CCC2OCCCN(C(=O)C(N2CCC(C)C2)=O)C)=O)C1 c1(C(C)OC)nc(C(=O)NCC2(NC(=O)CN(C)C(=O)C3CC3)CCCC2)cs1 CN(C(=NCCCN1CCCCCC1)NC1CCCC1)CCC(C)(C)C C#CCC(CC(F)F)C(=O)N1CCCC(CCNC(=O)C(F)(F)CC)CC1 C(c1cnc(C)nc1O)=CC(CN1CCN(C(C(C(C)C)NC(C)=O)=O)CC1)=O C=C(Cl)C(C)(C)C(=O)N1CCC(C)C(NC(=O)Cc2ccoc2)C1 CC1CCc2[nH]c(C(=O)NCC3CC3NC(c3cc(Cl)ccc3O)=O)cc2C1 N1(C(CCC(=C)Cl)=O)CCN(C(=O)C(F)(F)c2nccn2C)CC1CO N1(C(C(F)=CC)=O)CC2CCOC2(CNC(c2cn3ccccc3n2)=O)C1 c1(C(N2CCC(F)(C(=O)NCC(=O)N(CC)CC)C2)=O)ccc2sccc2c1O c1(C(=O)NCCN(C)C(c2ccc(Br)cc2Cl)=O)ccc(O)c(N)n1 O=C(Cc1ccc(NCc2cc(Br)cc(Br)c2O)cc1)N=c1ccnc(Br)[nH]1 N1(C(CCNS(CC)(=O)=O)=O)CCC(O)(C(C)CNC(=O)C=CC(F)(F)F)C1 C1(O)(CCNC(C2C(=C)C2)=O)CCCN(C(=O)Cc2ccccc2C#N)C1 C12(NC(C=CCOC)=O)CCCCC1CN(C(c1cccn3nnnc13)=O)C2 Cc1oncc1C(=O)NCC(=O)NC(C)CCCNC(c1ccc(F)o1)=O N#Cc1cnn(CC(=O)NCc2cccc(NC(C3CC(F)C(=O)N3)=O)c2)c1N C(=O)(C(O)CNC(c1occc1C1CC1)=O)N(CCC1CC1)CC c1(N(CC=C)C(=O)NCCC(C)C(F)F)cccc(F)c1F C#Cc1ccc(C(N2CC(CNC(c3cncc(Cl)c3)=O)C(O)C2)=O)c(C)c1 C1(NC(Cc2c(C)n[nH]c2)=O)CC2C(NC(=O)C(C(C)C)n3ccnc3)C2C1 Cc1ccc(C#N)cc1C(N1CCC1CC(=O)NC(C)(C)CCN(C)C)=O CCCCC(=O)NC(C)C(=O)NC1CCC(N(C)C)C1 CCC(C(=O)NCCCSCCO)NC(c1cc(CCO)on1)=O c1(NC(CC2CC(C(C)C)OCC2)=O)ccc(C(=O)O)c(P(C)(C)=O)c1 C1(CC(=O)NC2CNC2)CCC(NC(C2CNCO2)=O)C1 c1(C(=O)NC(CNC(c2c(C)onc2Cl)=O)(CC)CC)cc2c(Cl)nccc2o1 C12(NC(=O)C(F)(F)F)CCOCC1CN(C(N(c1cnc(=N)[nH]c1)CC)=O)C2 N1(C(c2c(C)nc(C(C)C)o2)=O)CCC2CC2(NC(=O)COC(F)F)CC1 Cn1cnc(C(=O)NC2CCCN(C(=O)OC(C)(C)C)CC2)cc1=O c1(CN2C(CCC)CCCC2)ccc(OC)c(-c2cnc(C)c(C)c2)c1 c1(CC=C)cccc(C(=O)NC2CCOC2C(=O)NC2(C)CC(O)C2)c1 Fc1cc(-c2nc(-c3cccnc3)nn2CC(F)(F)F)cc(-c2ccncc2)c1 c1(OCC(=O)NC2C(NC(CC(C)(C)O)=O)COCC2)ccc(Cl)cc1[N+](=O)[O-] Cc1noc(C)c1C(=O)NCCC1CC(C(=O)NC2(CCO)CCC2)C1 c1(OC)cc(F)ccc1C(=O)NC(C)CCCNC(=O)Cc1cccc(SC)c1 CCCC(C(=O)NCCC1(C)CCN(C(C2(CC(C)C)CC2)=O)C1)N(C)C C1(CC)(NC(c2nc(C)cs2)=O)CCN(C(C2C3COCC23)=O)CC1 C(=O)(C(F)(F)C(O)CC)OCC(=O)NC1CCCN(c2cccc(OC)c2)C1=O c1(CN2C(=O)CN(CC3CC(F)(F)CO3)C2=O)cc(C(F)(F)F)c2n1CCCC2 CC(C)(CCNC(=O)C=CI)NC(c1ccccn1)=O c1(CC(N2CC(NC(=O)Cc3ccnc(Br)c3)C(O)C2)=O)cc(F)c(F)cc1F CCCS(=O)(=O)C(C)C(=O)NCCN(C(=O)CCNC(=O)C=Cc1ccco1)C c1(C(N2C(C)C(NC(=O)C=C(C3CC3)C3CC3)CCC2)=O)ccc2c(c1)CCO2 n1(CC=C)nnnc1C(c1ccncc1)NCc1ncc(CO)o1 C(C(N=[N+]=[N-])C(=O)N1CCC(NC(C2CCCO2)=O)C1(C)C)OCC C(C(=O)N(CC(C)(C)CNC(=O)CCn1ccc(C)n1)C)(C(C)(C)C)SC c1(C(=O)NC(CN(C(C(=C(C)C2CC2)F)=O)C)(C)C)ccccc1F CC1C(NC(c2n[nH]c(O)n2)=O)CC2CCC1N2C(c1ccc2c(c1)CC2)=O c1(C(=O)NCCOCCNC(C2N(C(C)=O)CCOC2)=O)cc(C)ccc1Cl C1(NC(c2cscn2)=O)Cc2ccccc2C1NC(c1cccc(F)c1O)=O C1(NC(C(C)(C2CC2)OC)=O)CCN(C(=O)CC2CCCN(C)C2)CCC1CO N1(Cc2[nH]nc(C(=O)OCC)n2)CCc2nc(Cl)cc(Cl)c2C1 C1(CNC(CS(CC)=O)=O)CN(C(c2cnn(C(F)F)c2)=O)CC1(C)C N1(C(CCOCCC)=O)CCN(C)C(CNC(=O)C(C)(CC)CO)C1 N1(C(c2cc(SC)oc2C)=O)CC2CC1CC2NC(c1sccc1Cl)=O CCCC(CCC)CCCC(=O)N1CCOCC1C C12(C(=O)NCC(C)(C)NC(C3CCOCC3)=O)CCCC1OCC2 c1(C(N2CC(CNC(C(CC)C)=O)C(C)(C)CC2)=O)cc(F)c2ncccc2c1 CC(C)CC(C(=O)N1CC(O)(CNC(C2CC3CCC2CC3)=O)C1)n1ccnc1 O=C(C1=NN(CCO)C(=O)CC1)NC1CC2CC1CN(C(c1ccncc1)=O)C2 c1(CCC(N2CC3C(CNC(=O)CCCF)C3C2)=O)ccc2c(c1)OC(F)(F)O2 C1(C(=O)N(C(CF)CF)C)(OC)CCN(C(C2CC(O)C(F)C2)=O)C1 C1(CNC(C(n2ncc(C)c2)C)=O)CCCN(C(c2cnc(N)c(Cl)c2)=O)CC1 C1(C(N2C3(C(=O)NCCCCC(=O)OC)CC3CC2)=O)CCC2(CCC2)O1 c1(C(=O)NC2CN(C(CN(C(COC)=O)C)=O)CC2C)c(F)ccc(F)c1O N1(C(CC(CC)C2CC2)=O)CC2(CO)CC1(C(N1CCC1(C)COC)=O)C2 c1(C(=O)NC2CCN(C(CNC(=O)NC)=O)C2)ccc(C(F)(F)F)cc1O C(=O)(CCC(C)(C)C)NC(CNC(COC(CC)CC)=O)C(C)C Cc1nccc(C(=O)NC(C)(C)C(C)NC(=O)CCc2cc(F)cc(F)c2)c1C c1(N(C(=O)Nc2cncc(Nc3ncccn3)c2)CC)ccc2c(c1)CCO2 Cc1cc(C(=O)NCC2C3CN(C(=O)CCC(N)=O)CC23)cc2ccsc12 c1(SC)ccc(N)cc1C(=O)NC(CNC(c1occc1F)=O)C1CC1 CC1CCCC(CC(=O)NCC(O)CNC(=O)C(O)C2CCC2)O1 C#Cc1cc(F)c(C(=O)NCC2CN(C(c3onc4c3CCCC4)=O)C2)cc1F CCCC(C(=O)N1CC2(C)CC1(C(=O)NCCC1(C)CCOCC1)C2)C(C)C C1(NC(=O)NC2C(C)(CC)C2)CCN(c2cccc(C)c2)C1=O C1(NC(c2cc(CCC)on2)=O)CN(C(c2c(C)ccn2C)=O)CC1N=[N+]=[N-] CC(C)(C)C(O)C(=O)N1CCCC(F)(C(N2CCCC(CCCO)C2)=O)C1 C1(NC(C2(CC)CCNC2=O)=O)CCC2(CC1)CN(C(c1ccsc1C#N)=O)C2 C1(C(N(C)Cc2ccnn2C)=O)CCN(C(C2CC=CC(O)C2)=O)CCO1 n1(CC=C)nnnc1C(c1csc(C(F)(F)F)n1)NC1CCC=C1Br C(=O)(CCCC(=O)NCC1C(C)CCN1C(=O)CN(c1ncccn1)C)NCC C1(O)(CNC(CC=CC)=O)CC(NC(=O)C(C)(C)OC(C)=O)C1 c1(OCC)ccc(OC)c(C=CC(=O)NC2CN(C(=O)C3CC3)CC3(CC3)C2)c1 c1(CC)c[nH]c2nc[nH]c(=NCC(C)NC(=O)CCc3cnoc3)c12 N1(C(C(C)OCC(C)C)=O)CCC(OCCNC(C2(S(N)(=O)=O)CC2)=O)CC1 Cc1ccc(F)c(C(N2CCCC2CNC(C2(C(F)(F)F)CCCCO2)=O)=O)c1 C1(C(C)NC(c2cnn(CC)n2)=O)CCCCN1C(c1occc1C)=O c1ccc2c(c1)OC1(CCOC1)CC2NCc1cn(C2CCNC2)nn1 Nc1cc(F)c(Cl)cc1C(=O)NC1CCCC(NC(=O)CC2CC2)CC1 C1(C(=O)NCCCNC(=O)C(F)F)(OC)CC(C)CC(C)C1 N1(C(C(C#C)(C)C)=O)CCC(C2CCN(C(C34CC(O)C3C4)=O)C2)CC1 CCC(Cc1ccccc1)C(=O)N1CC2CC2(NC(c2ccn(C)c2C)=O)C1 c1(C(N2CCN(C(CNC(C(CC)C(C)O)=O)C)CC2)=O)nc2ncccn2n1 Cc1cc(C(=O)NC(CC2CC2)C(=O)NCCOCCN=[N+]=[N-])nc(O)n1 N1(C(C=CC(=O)OCC)=O)CC(NC(=O)CC(C)CN(C)C)CC12CCCCC2 CN1CC2(CC2)CC1C(N1CCCC1C(C)(C)C(=O)N1CCC(C(C)(C)C)C1)=O CC1CN(c2nccc(C(F)(F)F)n2)CCC1NC(=O)Cc1c(O)ncnc1O N1(C(C(C)O)=O)CC(NC(=O)C(C)(C)O)Cc2ccccc21 C=CCC(CC(F)F)C(=O)NCC1C2CN(C(c3ncc(N)cc3Cl)=O)CC12 C(=O)(C#CC1(C)COC1)N1C(CC(=O)NC2(CC)CCCCC2)CCCC1 CN1CC(N(C)C(C2COCCC2NC(=O)C(O)C(F)(F)F)=O)CCC1=O N1(C(C=Cc2c(C)cncc2)=O)CCC2(CCC2NC(c2nccn2C)=O)CC1 c1(NC(C(C)(CC2CCC2)CO)=O)ccc(-n2cc(C3C4COCC34)nn2)cc1 N1(C(CC(c2cc(F)ccc2F)NC(C)=O)=O)CCC(S(=O)(=O)N(C)C)CC1 N1(C(C(CC(=C)C)C)=O)CCCN(C(c2ccc(F)cc2NC(C)=O)=O)CC1C c1(C(=O)NCc2cccc(NC(CC3CC(SC)C3)=O)c2)cncc2c1CCC2 N1(C(C2CCOC2)=O)CCC(O)(Cn2cc(COc3ncccn3)nn2)C1 N1(C(CC=CCC)=O)CCC2CCN(C(=O)C(C)N(C)C)CC2C1 c1(NC(C(C)CNC(c2cncn2C)=O)=O)cccc([N+](=O)[O-])c1 N1(C(C(C(C)C)(C)O)=O)CC(NC(c2cccnc2OC(F)F)=O)CCC(O)C1 Cc1sc(-c2nc(C3CCN(C)C3=O)no2)cc1Br c1(C(N(C(CN(C(c2ccc(COC)o2)=O)C)C)C)=O)cnc(SC)nc1O N1(C(CCCCNC(=O)Cn2cnnn2)=O)CCN2CC(O)CC2C1 c1(SCC(=O)NC2CN(C(C(C)O)=O)CC2C)ccc2ccccc2c1 c1(CC)oc(C)cc1C(=O)NCC(O)CCNC(c1cn(C)nc1Br)=O C1(C(=O)NC2CN(C(c3cn(CCCOC)nc3)=O)CC2F)CC2CCC(C1)O2 c1(C(=O)NCC2N(C(C3(OC)CC3)=O)CC2)c(Br)ccc(F)c1C N1(C(C(CC)(C)O)=O)CCC2(CCCN2C(c2cnn(C3CC3(F)F)c2)=O)CC1 Cc1ccc2c(C(N3CCC(CNC(C4(F)CC4C)=O)C34CCC4)=O)csc2c1 C1(C(N2C(CN(C)C(C3(C#N)CC3(C)C)=O)CCC2)=O)CC2(CCCC2)CO1 c1(CC(=O)NCCCCCNC(CN(CCC#C)C)=O)cccc(Br)c1F CCC(C(=O)NCCCN(C(=O)CCOC1CCCCC1)C(C)C)OC N1(C(c2ccc(N(C)C)nn2)=O)CC(C2CCCN(C(c3n[nH]cc3Br)=O)C2)C1 Cc1cc(C(=O)NCC2CN(C(C3CSCN3C)=O)CCO2)c(C)n1NC(N)=O C1(C(N(c2n(CC(=O)OC(C)(C)C)ncc2)CC2CC2)=O)CCCC2C1C2(F)F N1(C(C2CC(CCC)C2)=O)CCC2(CCC2CNC(=O)C=CCOC)CC1 C1(NC(CCN(C)C(C2CC3(CCC3)CO2)=O)=O)CCCCCC1F c1(C(c2nc(CC(F)C3CCC3)on2)C2CCC2)ccc(Cl)cc1Br Cc1sc(C)c(C(=O)NC2CC(O)(CNC(=O)C(=O)N(C)C)C2)c1C#N C1(NC(c2scc(OC)c2OC)=O)CCN(c2nc(OC)cc(C)n2)C12CCCC2 c1(C(N2CCC(C)(CNC(CC3C(C)(C)C3)=O)C2)=O)cccc2ccc(O)nc12 c1(OC)ncc(C(=O)NC(C2CCCN(C(c3cc(C)cs3)=O)C2)C)cc1F C12(CNC(c3ccc4ncnn4n3)=O)CCC(CC1)N(C(C1C=CCCC1)=O)C2 C(N=c1cc(C(C)C)nc[nH]1)C1CCN(C(c2c(C)nc(C)[nH]2)=O)CC1C CCC(CC(C)C)C(=O)NC(C)(CNC(=O)CCc1csnn1)Cn1cccn1 N#Cc1ccc(CC(N2CCC3(C2)CN(C(=O)Cc2cnc[nH]2)C3)=O)c(F)c1 c1(C(=O)NC2(CNC(CCc3cc(C)on3)=O)CCOCC2)ncc(Cl)nc1Cl c1(C(N(C)CCOCCNC(C2(C)CC=CCC2)=O)=O)cc(F)cc2nn[nH]c12 C(C(C)(C)C(C)(C)C)NC(C1CCN(C(CCn2c(C)ncc2)=O)C1)=O N1(C(C23CC(C)(C2)C(C(F)(F)F)O3)=O)CCC2(CCOCC2)CC1 c1(NC(=O)NCc2cc(C(=O)OCC)no2)cccc(CN(C)C)c1 c1(NC(C(CCCOC)NC(=O)CC=C(Cl)Cl)=O)cccc2cnc(Cl)cc12 C(=O)(C(C)(C)S(C)(=O)=O)NC(C)C(CO)NC(=O)CCc1cnn[nH]1 C1(NC(C(CCC)NC(C)=O)=O)CC2CCCC(C1)N2C(=O)C(Cl)=CCl C1(C(=O)OC)CN(C(=O)NCc2cncc(Cl)n2)CC1C(C)C C1(CNC(CN(CCCCCC)C)=O)COCCN(C(=O)C(C)(C)O)C1 C1(C(=O)NC2CCN(C(c3cc(CO)on3)=O)C2C)(OC)CCCOC1 N1(C(c2c(C(C)(C)C)n[nH]c2)=O)CCC2(CC1)CC2NC(=O)CCc1cncs1 N1(C(c2c(C)nc(COC)s2)=O)CC=C(C(=O)O)CC1 CN1CC(O)CC1C(=O)NC(C)(C)CC(=O)NCc1ncc[nH]1 c1(C(N(C(C)CNC(c2cnnn2C)=O)C)=O)cnn2c1CC(C)CC2 Cc1cccc(NC(c2ccc(NC(C3CC4CCC3N4)=O)cc2)C)n1 Cc1cn2c(n1)CN(C(=O)CCCC(C)(C)NC(=O)CC1COCC(C)O1)CC2 N1(C(C=COCC)=O)CCC(NC(=O)CC(CC)SC)C(C)C1 CCCCC(CNC(c1ccoc1Cl)=O)NC(=O)COc1ccccc1C CC(C)CC(C(=O)N1CCC(O)(C(C)NC(=O)CC(C)(C)C2CC2)C1)C(N)=O CC1CN(C(=NCC2CC2)NCC2CC3(CCC3)C2)CC1C c1(C(N2CC(C)N(C(C3CC(=O)C34CCC4)=O)CC2)=O)c(N)cc(Cl)nc1Cl C1(C(=O)NCC(C)N(C(=O)Cc2ccsc2C)CC)CCN(C(=O)NC)CC1 Cc1nc(Cl)cc(=NCC2CCCC(NC(c3ccc(-c4ccco4)s3)=O)C2)[nH]1 N1(C(c2c(C(C)C)nns2)=O)CCC(O)(C(C)CNC(=O)Cc2ccno2)C1 C(c1cn(C2CC(NC(c3ccc(C4CCC4)cc3)=O)C2)nn1)=C(C)O C1(C2CC2)(NC(C=CC(=O)NC2CC2)=O)CCN(C(=O)C(c2cccnc2)O)C1 c1(C(=O)OC)cc(F)cc(C)c1NC(N1CCCCC1CSC1CCC1)=O N1(C(C2(SC)CC(O)C2)=O)CCC(C)N(C(=O)CN2CC(C)C2)CC1 CN1C(=O)CCCC1C(=O)NCC1(CC(=O)NC2(COC)CC3CCCC23)CC1 C1(OC)CC(NC(C2CCCS2)=O)CN(C(=O)C(C)(C)CC2CCOCC2)C1 N1(C(C2OCCN(C(CN3CC(C)(OC)C3)=O)CC2)=O)CC2CCOC(=O)C2C1 Cc1cc(C(=O)NC2CCN(C(=O)CN3CCSCC3)C2)c2cnn(C)c2n1 C=C1CC(C)(C(=O)NC(C2CCCCC2)CNC(=O)CC2CC2CC)C1 c1(C(N2C(C(=O)Nc3cc(CC)no3)CC2)=O)c[nH]c2ncc(C(F)(F)F)cc12 C12(CNC(CCC=C)=O)CCC(CC1)N2C(=O)Cc1c(C)nn(C(F)F)c1C C1(CC(=O)N(CC(C)NC(c2ncccc2Br)=O)C)CCC(F)(F)CO1 C(=O)(CCCC(N)=O)N1CC(NC(CCc2cn(C)nc2)=O)C(O)C1 C1(C(=O)NCC2N(C(C(C3CC(C)(C)C3)OC)=O)CCC2)CC12CCOC2 C(=O)(CCC(F)(F)Cn1cc(CN2CC3CC3C2)nn1)Nc1cc(=N)[nH]c(Cl)n1 N1(C(C(C)OCC#C)=O)CC2(C)CC1(C(=O)N(C(C)COC)C)C2 C=CCCCCCC(=O)N(CC(N1CCCC(NC(C)=O)C1)=O)CC CN1CCC(C)(C(=O)NCCC2CCN(C(C3(C(N)=O)CCC3)=O)C2)C1=O Cc1sc(C(=O)NC(C)CCN(C)C(c2cc(CO)on2)=O)cc1Br N1(CC(=O)N(CC(C(=O)N(C(C)C(C)C)CC)C)C)CCC(=O)CC1 C(CC(C)(C)C(=O)NCCC1COCCN1C(=O)C(O)C1CCC1)SC N1(C(c2c(C)cncc2C)=O)CCC(C(=O)NC2CCCCCC2)C(C)(C)C1 c1(C(c2n(C(c3ccccc3)C)nnn2)NC2CC(NCCCF)C2)ccccc1 c1(CC)cc(C(N2CCC(C(C)NC(=O)C3CC3)C2)=O)on1 c1(C(C)NCC#CCCO)ccc(F)c([N+](=O)[O-])c1 C1(C)(CC)CCN(C(=NCC(O)c2cccc(OC)c2)NC(CC)CC)C1 c1(C(=O)NCC2CC(F)(CNC(c3c(CC)nns3)=O)C2)cc(C#N)ccc1F c1(OC)cc2c(cc1C(N1CCCCC1CN(C(=O)CCS(C)=O)C)=O)OCO2 C1(CC)CCCC(c2nnnn2CCSC)(NCCCCF)C1 c1(C(C)C)cccc(C(=O)NCC2CCN2C(c2cc(C(N)=O)co2)=O)c1 C(CCCO)N(C(=O)C(C)N(C(C1CC(CC2CC2)C1)=O)C1CC1)CC C(=O)(CC(CC)C(C)C)NCC(CC)NC(=O)CCN(S(C)(=O)=O)C c1(C(N(CC(CN(C(=O)CC2CCCCC2)C)O)C)=O)cc([N+](=O)[O-])n[nH]1 C1(SCC(=O)NCC=CCNC(=O)CCc2cocn2)CCOC1=O C1(NC(c2ccns2)=O)CN(C(=O)Cc2cnns2)CC1c1ccccc1 N1(C(COC(CC)CC)=O)CCOCC1CNC(=O)CCc1cccnc1 N1(C(c2c(CNC(COc3cc(C)on3)=O)nccc2)=O)CC2C3CCC(C3)C12 C(=O)(C1=C(C)OCC1)NCC(CCOC)NC(C1CCCN(S(C)(=O)=O)C1)=O c1(CC2N(Cn3c(-c4c(C)scc4)ncc3)CCCC2)nn(C)c(Br)c1C CC(C)(C)CCCCC(=O)N1CC2CC2(CNC(C2(C)COC(=O)OC2)=O)C1 c1(N2CCC(CC)C2)ncc(S(=O)(=O)N(C)CC2(CC)CCCC2)cc1Cl CCC(C)C(C(=O)NC(C)CCCCNC(=O)CCC(=O)c1ccc[nH]1)NC(C)=O CC1(C)CCCCC1CNC(=O)CCNC(c1cc(Cl)no1)=O c1(C(=O)OC)cc(C(=O)NCC2(O)CC(NC(=O)C=Cc3ncc[nH]3)C2)c[nH]1 N1(CC(CNC)(C)C)CC=C(c2c(C)[nH]c3ccccc23)CC1 C=CCC(CNC(=O)CCc1cnc(C)o1)NC(c1cc(C2CCOC2)[nH]n1)=O N1(C(CSS(C)(=O)=O)=O)CC2CC(Nc3ncnc4[nH]ccc34)CC1C2 N1(C(c2n(C)ncc2)=O)CCCC2CN(C(=O)CC3(C)CC(F)(F)C3)CCC12 C(=O)(C(CO)C(C)(C)C)N(CC(CNC(C1(C(=O)OC)C(=C)CC1)=O)(C)C)C c1(C(=O)NC2CCC(F)(CNC(c3c(C)nc(O)[nH]3)=O)C2)ccc2ccoc2c1 CCC(CC(=O)N1CC2C(N(C)C)C2C1)N(C(=O)CCC(C)SC)C c1(C(=O)NC2CC(NC(Cc3c(C)con3)=O)C23CCC3)cncc([N+](=O)[O-])c1 c1(CNC(CCCOCC=C)=O)cnn(C)c1C(=O)NCC1CC(CO)CO1 N1(C(Cc2c(C)nn(C)c2C)=O)CC(C)CN(C(C2CCC2)=O)C(C)C1 c1(NC(c2ccc(C)s2)C)cc(=NC2C=CCCC2)[nH]c(CCC#N)n1 C1(C)(CCNC(C(CC)F)=O)CCN(C(c2ccc(C(C)C)cn2)=O)CC1 c1(C(=O)NCC(C)(C2CC2)NC(c2cscn2)=O)ccc(C2COC2)cc1 C1(CCNC(C(C)NC(CC)=O)=O)(OC)CN(C(=O)CC(C)n2ccc(C)n2)C1 CC1(C)CC1(C#N)C(=O)NCC1(C)CCCN1C(=O)CCn1cnnn1 C1(CNC(c2ccc(F)cc2F)=O)CC2CCC1N2C(=O)COCC(F)(F)F C#CC1(C(=O)NCCc2nccn2C)CCN(C(=O)C(C)SC)C1 N1(C(c2cc(C)cc(O)c2)=O)CCC(C)N(C(=O)CC(=O)N(C)C)CC1 S(=O)(=O)(c1ccc(NC(C2CCCCC2)C)nc1)NCCOc1cccc(C)c1 CC1CNCC(CC(=O)N(c2nccs2)C)O1 N1(c2snc(C(C)NC)n2)CCCC(C(=O)OC)C1 CC1(O)CCN(C(=O)CC2CCC(NC(C3C4CC5C(C4)C35)=O)C2)CC1 c1(NC(C=CC(=O)NCC2(F)CN(C(C3CCC3)=O)C2)=O)cccc(O)c1 CCCC(CCC)C(=O)NCc1ccc(C(N2CC(CO)C(O)C2)=O)cc1 C#CC1(C(=O)NCCSCCF)CCN(C(=O)C(O)CSC)C1 c1(C(N2CC3(CC(CNC(=O)C4=COCCC4)C3)C2)=O)cnc2c(c1)CCCO2 C(=O)(C1=Cc2cccc(Br)c2OC1)NCC(C)(C)OCCNC(=O)C1=CCC1 O=C1NCc2cc(C(N3CCCN(C(C4C=CCC4)=O)C(CO)C3)=O)ccc21 c1(C(=O)NC2CC(NC(C=CC(CC)C)=O)C(O)C2)ccc2nc[nH]c2n1 c1(C(N2C(C)CC(NC(CC=CC=C)=O)C2)=O)cccc2c1COC2 C1(NC2CCC(C(=O)OC)(CBr)CC2)CCOC2(CCOCC2)C1 C1(CC)(NC(C2CCSC2)=O)CCCN(C(c2ccc(C(=O)OC)nc2)=O)C1 C(=O)(CCCC(=O)N(C)C)N1CCC(NC(COCc2c(C)ncs2)=O)C1C c1(C(N(C)C)=O)ccc(NC(C2CCC3CC23)=O)cn1 N1(C(C(C)n2ccnc2)=O)CC(O)CC1C(=O)NOCCCN(C)C Cc1c[nH]c2ncnc(N3CC4CN(C(c5ccc[n+]([O-])c5)=O)CC34)c12 c1(C(=O)NCC(C)NC(CCOCCCOC)=O)ccc2c(c1)OCCNC2=O N1(C(C(C)NC(=O)OC)=O)CC2CC1(C(=O)NCCC1CCCN(C)C1)C2 Cc1nc2c(o1)CCN(N1CC(C)S(=O)C(C)C1)C2c1ccccc1 C(C)(C(C(=O)NC1CCOCC1C(=O)NCCCP(C)(C)=O)N(C)C)OC C(=O)(CC(C(C)C)NC(=O)OC(C)(C)C)NCC1CN(C(CCC=CCC=C)=O)C1 CCCCC(CCCC)C(=O)NCC1C(CC)CCN1C(C1CC1C1CC1)=O Cc1cc(C(=O)NC2CN(S(=O)(=O)CC3CC3)CC2(F)F)ccc1F c1(C(N2C(C)(n3cc(C4(OC)CCOC4)nn3)CCC2)=O)cccc(Cl)c1C C(=O)(C1(C)CCCc2ccccc21)NCCC(C)(C)NC(C(F)=CCC)=O C(CCCCC(=O)N1CCC(c2nn[nH]n2)C1)NC(c1cc(C)ncc1)=O C1(F)(CNC(C(CC)(C)O)=O)CCCN(C(=O)COc2ccc(C)c(C)c2)C1 Cc1ccc2oc(C(=O)NC3CCCN(C(C4CCCCC4)=O)C3)cc2c1 c1(CNC(CCc2cc(C)cc(C)c2)=O)nc2c(c(O)nc(=O)n2C)n1C c1(C(=O)NC23CCC(CN(C(CSCC(N)=O)=O)C2)C3)ccc(F)cc1[N+](=O)[O-] C(=O)(C(C)(C)CC(=O)N(CC(C)CNC(=O)CC(C(F)F)n1cccn1)C)OC C12CCCCN1C(=O)C(CC)N(CC)CCC2.C(C(=O)NCC)OCC#C C1(N(C(=O)CCCCCF)C)CCC2CN(C(c3csc(F)c3)=O)CC12 C(F)(c1ccccc1)=CC(=O)N(CCCNC(CCSCC(C)C)=O)CCO c1(CC)cc(C(=O)NC(CNC(=O)CCCCN2CCCC2)CO)ccc1C O=C(N=c1nc2cc(Br)ccn2[nH]1)N1CCN2C(=O)CCC2C1 C1(CC)C(NC(C23CSCC2C3)=O)CCCN1C(c1ccn(CC)n1)=O N(C1c2ccccc2CC1NC(c1cc(C(F)F)cs1)=O)C(c1cc(C)no1)=O C1(CNC(C2(CCC=C)CN(C(C3CCN3CC)=O)C2)=O)CN2CCN1CC2 c1(C(=O)OC)nc(Cl)[nH]c(=NCCN(C(=O)CC2CC3CC3C2)C)c1OC N1(C(C2C(C)(CC)C2)=O)CCC2CCN(C(=O)COC3CCCC3)C2C1 c1(C(C)C)ccc(C(C)C(=O)NCc2csc(-c3ccccc3)n2)cc1 N1(C(CN(C)C(N)=O)=O)CCCC1C(C)(C)NC(C1CCC1(C)C)=O C1(N(C(=O)C(C)(C)C)C)CCC2(CC1)CC2NC(=O)CSC(C)(C)C c1(C(=O)NC2CCC(C(=O)Nc3ccnc(C)n3)CC2)cc2[nH]ccc2cc1Cl c1(C(N2C(Cn3cc(-c4ccn(C)n4)nn3)CC2)=O)ccc(S(N)(=O)=O)o1 c1(CNC(C2CC2Cl)=O)n[nH]c2c1CN(C(c1c[nH]c3cccnc13)=O)CC2 N1(CCC)C(=S)NC(c2cnc(Cl)cc2N)C2=C1CC1(CCC1)NC2=O N1(CCC(=O)NC(C)CC2CN(C(=O)C=CC3CCC3)C2)CCCCC1 C(CCC(CCC)NC(c1ccc(N(C)C(C)=O)cc1)=O)NC(CCCC#C)=O N1(C(C2(CC(C)C)CC2)=O)CC(CNC(=O)CC2CN(C(C)=O)C2)C1 Cc1ccc(Cl)c(C(=O)NC(CNC(c2ccnn2C)=O)CC(F)(F)F)c1N C(CC(C(=O)NCC(CSC)OC)NC(=O)C(n1ccc(C)n1)C)=CC N1(C(C2(COC)CCCO2)=O)CCN(C(=O)C(C)(C)C(C)C)C(C)C1 N1(C(c2c(C)ccs2)=O)CCC2C1CCN2C(=O)Cc1noc(C(C)C)n1 O=C(CC(F)(F)C(F)(F)F)N1CCCC(n2cc(CO)nn2)C1 c1(NC(C2CC2NCc2ccc([N+](=O)[O-])cn2)=O)ccc(I)cc1[N+](=O)[O-] c1(NC(N2C(CNC(CSc3n[nH]c(=N)s3)=O)CCCC2)=O)cc(F)cc(F)c1 c1(C(CNC(N(C(c2ccccn2)CCC)C)=O)(C)C)c(C)noc1C c1(CNC(C2(OC)CCNCC2)=O)ccc2nc(O)oc2c1 N1(C(C2CCN(CC)C2)=O)CCC2(CCN(C(=O)CCCC(F)(F)F)C2)C1 C(CC(=O)NCC1(NC(C2CC(C)(C)CN2C)=O)CC1)(C(N)=O)NC(C)=O c1(CC(=O)NCC(CC)(C)NC(C2NC(=O)OC2C)=O)ccc(Cl)nc1 C1(C(=O)NC(c2cccnc2)C)(NC(C2C(C)=CCS2)=O)CCCC1C c1(C(=O)NCC2C(NC(c3c(C)nc(C)[nH]3)=O)COC2)cncc([N+](=O)[O-])c1 C1(C(N2C(C(=O)NC(C)(C)CCF)CCC2)=O)CC2(CC2)CN1C(N)=O C1(NC(CN(CCC#C)C)=O)CCCN(C(=O)CCOC)CCC1 C(=O)(CC(C)(C)CC(F)(F)F)NC1(C)CCC(NC(C(C(C)C)C)=O)CC1 C1(C(=O)NC(CCO)C2CCC2)CCN(C(c2c[nH]ccc2=O)=O)C12CCC2 C1(NC(c2c(CC)ccs2)=O)CCN(C(=O)C(C)(C)C(=O)N(C)C)CC1C c1(CC)ncc(Cl)c(C(=O)NC(C)CC(C)NC(c2[nH]cnc2C)=O)n1 C1(C(=O)NC2CCCCN(C(CCC(=O)NC)=O)C2)CCc2c(n[nH]c2C)C1 c1(C(N2CCC(C(C)NC(=O)C=CC(F)(F)F)C2)=O)cc2cccnc2s1 C=CCCC(F)(F)C(=O)N(CCCCN(C(=O)CNS(=O)(=O)CC)C)C C1(CNC(C2CC2c2cccnc2)=O)C2CN(C(c3csc(CO)n3)=O)CC12 N1(C(c2ncc(CC)s2)=O)CCC(CC(C)NC(=O)C(F)(F)c2cscn2)CC1 Cc1csc(C(c2nnnn2C2CC2)NCCc2ncccn2)n1 N1(C(=O)CCn2cc(Cc3ccnc(CO)c3)nn2)CCC2(CCCC2)CC1 N1(C(c2ccc(C(C)=O)o2)=O)CCOCC1CC(N1CCN(CC(=O)NC)CC1)=O c1(C(N2CC(CC)(CO)C2)=O)ccc2c(n1)CN(C(C1CC1(C)C(F)F)=O)CC2 N1(C(C(C)(C)C)=O)CCC2COC(CNC(c3ccc(C4CC4)s3)=O)C2C1 Cc1ccc(C)c(CCNC(=O)Cc2ccccc2OCC(F)F)c1 c1(C(N2C(COC)CN(C(=O)CN(C)C(C)C)CC2)=O)cc2cccnn2n1 C1(C(=O)NCC2(CNC(C(COCC)(C)C)=O)CC2(F)F)CC2(C1)CC21CC1 Cc1c(NC(=O)C(C2CCN(c3ncc(C(F)(F)F)cn3)CC2)C)ccnc1Br c1(C(=O)NCC2N(C(C(C)C#N)=O)CCC2)cccn2ccnc12 N1(C(Cc2c(C)occ2)=O)CCN(C(C2CCCN2C=O)=O)CC1C c1(C(N(C2CCN(C(C3CC4(CC4)C3)=O)C2)C)=O)cc(O)ncc1Br CCC(C)(CNC(=O)C(Cc1ccccc1)OC)NC(C1(N(C)C)CC1)=O c1(C(=O)Nc2ccc(OC)cc2Cl)n[nH]c2c1CN(Cc1ccc(Br)cn1)CC2 C(C(O)CC(F)(F)F)N(C1CCCC1)C(=O)NC1CCCN(CCCOC)C1 N1(C(CC(CC)(F)F)=O)CC2CC(NC(=O)CSc3ccncc3)CC(C2)C1 CC(CC(=O)N(C)CC1CCCN1C(=O)CCOC1CCC1)C(F)(F)F Cc1ccccc1NC(=O)C(C)OC(c1ccoc1I)=O C1(C(=O)NC(C)CC2CCCCC2)CCN(C(C2CC(F)CN2C)=O)C(C)(C)C1 Cc1cccn2c(C(N3CCC(C)(CCNC(=O)C(C)O)C3)=O)cnc12 C1(NC(c2cnco2)=O)CN(C(=O)Cn2ncc(O)nc2=O)C2(CCC2)C1 c1(C(=O)NC2CCCC2C(=O)NCCCOCCOCCO)ccc[n+]([O-])c1 CCC(CC)C(=O)N(CCNC(=O)CC1CC1(Cl)Cl)CC1CC1 O=C(CS(=O)(=O)CCO)NC1CC12CCN(C(c1ccnc3ccsc13)=O)CC2 N1(C(C2CC(OC)C2)=O)CCC2CN(C(c3sccc3-n3cccc3)=O)CC2C1 N1(C(c2nnn(CC)c2C)=O)CC2CC(NC(c3ccc(C(C)C)o3)=O)C(C2)C1 C12CCC(NC1=O)C(=O)N2.c1(-n2cc(-c3nc(C)sc3)nn2)ccncc1F C12(NCCCCCOC)CCC(n3cc(-c4nccn4C)nn3)C1C2 CCCCS(=O)(=O)CC(=O)N1CCN(C(=O)CSC(C)(C)C)C(CO)C1 N1(C(CC2(OC)CCC2)=O)C(CNC(=O)CCc2cnc(C)s2)CC2COCC12 C=CC1CN(C(=O)C(F)C2CC(NC(=O)C#CC(C)C)C2)CCO1 C(O)(CCN=c1[nH]nc(-c2ccc(Cl)cc2)o1)(C(F)(F)F)c1n(C)ccn1 C(N=C(NCC1CCCOC1)NCC1CCCCO1)c1nnn(C)n1 c1(C(=O)NC2CN(C(c3nc(OCC)sn3)=O)CC2F)cc2c(cn1)COCC2 N1(C(Cn2c(C)ccn2)=O)CC2CC1CN2C(=O)C(C)(O)c1ccccc1 n1(C(C)C)cccc1C(=O)N(CC(C)NC(=O)C=CC1CCOC1)C CC(C)(C)C(CC(=O)NCC1CCCCN1Cc1ccc(Br)s1)C(F)F N1(C(CCc2cccc(OCC)c2)=O)CC2CCC(N)(C2)C1 N1(C(COC(CC)C)=O)CC(C2CC2C(=O)NC2(CO)CCC(C)C2)C1 c1(C(N(C2CCN(C(=O)CC3CC=CCC3)C2)CCC)=O)ccccc1OC N1(C(C(C)C2CCCC2)=O)CC(CNC(=O)CC(=O)NC2CC2)CC1(C)C CCCC(C)(CCC)C(=O)NCC1CN(C(=O)C2=C(Cl)CCCC2)CCC1(C)C N1(CC)C(=O)COC(C(N2CC(NC(=O)C3CC3)C(F)C2)=O)C1c1cccnc1 C1(CC)CCCCC1C(=O)NCC1(COC)CN(C(=O)CC2CCSC2)C1 CC1CN(CCC(=O)N2CCCC2)Cc2c[nH]nc21 O=C1CC(C2CC2)(C(N2CC3CC2CN3C(=O)C=Cc2ccc(O)cc2)=O)C1 Cc1cccc(F)c1CC(=O)NC1CC(CNC(C2CCC(C)CC2)=O)C1(C)C N1(C(C(CCCOC)C)=O)CC2CCC(C1)N2C(C1CCC1C(C)(C)C)=O C(=O)(C(CNC(C1CC1OC(C)=O)=O)C(C)(C)C)NC(C#CC)(C)C C12(NC(c3nc(O)nc(O)c3F)=O)CCCCC1CN(C(C1CCCO1)=O)C2 C1(C(=O)NC2CN(C(C(CC)C3CCC(=O)N3)=O)C2)CCCN(C(C)=O)C1 c1(N2CC(C)C(NC(c3cc(C(F)(F)F)n[nH]3)=O)C2)ncccc1S(C)(=O)=O CC(C)CCCCCC(=O)NC(C)(C)C(N1CCC(N=[N+]=[N-])C1)=O CC1(C)CC1(C(=O)NCC1CC1[N+](=O)[O-])NC(=O)CCCn1ccnc1 C1(NC(c2c(CC)scc2)=O)C(CNC(=O)C2=CCC2)CCC12CCC2 CCC(CC)C(C)(c1nnnn1-c1ccccc1)NCC1CC(=O)N(OCC)C1 C1(C(=O)N(C(C)CC2CC2)C)(CNC(C(OC)OC)=O)CC12CCC2 c1(NC(N2CC3(OCC(C)C3)C2)=O)cccc2c(=O)c3ccccc3[nH]c12 N1(C(c2nn(CC)c(O)c2)=O)CC(CO)C2(C1)CN(C(c1cc(Cl)cnn1)=O)C2 c1(C(N2CCCC(CN(C(=O)C3=CCC3)C)C2)=O)ccc(N)c(F)c1 N1(C(C(c2ccccc2)C)=O)CCCCCCC1C(N1CCC1c1nc[nH]n1)=O C1(NC(C=CCOC)=O)CC(C(=O)N(C2CC2)Cc2ccc(Cl)nc2)C12CCC2 c1(C(=O)NCC2(C)CCN(C(C(C)=C(CC)C)=O)CC2)ccc2nnn(O)c2c1 c1(NC2CCCN(C(COC)=O)C2)ccc([N+](=O)[O-])cc1Br Cc1ccccc1OCC(N1CCC(CN(C)C(c2csc(C3CC3)n2)=O)C1)=O c1(CCC(=O)NCC(=C)CCNC(=O)CCC(C)N(C)C)nnc(S)nc1O C1(C(=O)NCC(=C)CC(F)(F)F)CC12CCC1(CC2)OCCO1 C12(C(N3C(CC=C)CCCC3)=O)C(NC(c3nc[nH]n3)=O)C3CC1C2C3 Cc1cc(C(=O)NCC(F)CNC(=O)C(C)C(F)F)n(C)n1 N#Cc1cc(Cl)c(C(=O)NCC(Cc2ccco2)CO)c(Cl)c1 c1(NC(C=CC(=O)OCC)=O)cc(C)cc(C)c1.c12ccc(o1)C(=O)NOC2 C1(OC2CN(C(C(CC)n3cncn3)=O)C2)CCN(C(C2CC2C(N)=O)=O)CC1 CCCC(C)CC(C(=O)NCCCF)N1CC(C(=O)OC(C)(C)C)C2(CC2)C1 C12(CNC(CN3CC(C)C3)=O)CCCC1CN(C(C13CC1COC31CCC1)=O)C2 C=CC(CCC)CC(=O)N1CC=CC1CNC(c1ccc(C(F)(F)F)s1)=O c1(-n2c(SC)ncc2)ccc(OC(Cc2cnc[nH]2)C(=O)O)cc1C.C1CO1 N(C(=NCCC1(C)CC1)N1CCc2cc(C)ccc21)C(CC)C c1(C(N(CC(CC)NC(C2CCCCS2)=O)C)=O)[nH]ccc(=O)c1C Cn1cc(C=CC(=O)NC(C)(CNC(c2cc(C(N)=O)co2)=O)CO)nn1 C(CCCC(CO)NC(C12CC(C)C1C2)=O)NC(c1c(Br)cn(CC)n1)=O C(CN=C(NCCc1ccccc1)NCC12CCCCC1C2)C1(C)CC1 N1(C(C(=O)c2ccco2)=O)CC2OCC(NC(c3cc(Br)co3)=O)C2C1 C1(NC(C(=C(C)C2CC2)F)=O)CC12CC(NC(C1CC(=O)N(C3CC3)C1)=O)C2 c1(C(=O)OC)ccc2ccccc2c1N.c1(CC(=O)N(C)C)csc(CN)n1 c1(OCc2cn(C3CCCN(C(C=NOC)=O)C3)nn2)cc(CO)n(C)n1 N1(C(CCC(C)N(C)C)=O)CCN(C(C23COC(CF)(C2)C3)=O)CC1C C(=O)(C1=NOC(C(C)(C)C)C1)NC1CC(N(C(=O)CNC(=O)C2CC2)C)C1 C(=O)(CCCCC(C)C)N1CC(CNC(c2cnc(OC)nc2C)=O)(OC)C1 C=C1CC2CCC(C1)N2C(C1(C)CC(C(=O)NC(C)(C)C)C1)=O c1(N2CCC(NC(C(C)C3CCOC3)=O)C(CO)CC2)ncc2ncn(C)c2n1 C12(CC(=O)N(C)CCNC(=O)Cn3cnc(-c4ccccc4)n3)COCC(C1)C2 C1(C2CCN(C(=O)CNC(=O)NC3CC3)CC2)(NC(CC2C(C)C2)=O)CC1 N1(C(c2c(C)cccc2Cl)=O)CCC2(CCCC2NC(=O)C=CS(C)(=O)=O)CC1 N1(C(C#C)C)CCN(C(=O)CC2(COCCOC)CCC2)CC1.C12CN(C1)C2=O C(c1ccncc1)=C(C)C(=O)NCC1(O)CCN(C(=O)Cn2c(C)ccc2C)C1 Cc1cc(C(N2CCN(C(=O)CN(C)C(N)=O)C(C3CC3)C2)=O)cc(O)c1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCCN(C(C(CC(C)C)C)=O)C(C)C O=C(C1CCCc2sccc21)NCC1CC(NC(C2CCCC23OCCO3)=O)C1 C(=O)(CC(C)C(F)(F)F)NCC1N(C(C2CCN(C(N)=O)CC2)=O)CCC(C)C1 CN1CC(=O)N(CC(N2CC(CO)(NC(C3CCCO3)=O)C2)=O)C1=O c1(NC(C(N2CCC(C(=O)OCC)C2)c2cnc(Br)s2)=O)ccc(F)cc1 C12(CNC(c3c(CC)n(CC)nn3)=O)CN(C(C3CCCCS3)=O)CC(F)(C1)C2 CCC(CC(=O)NC(C1(O)CN(C(=O)C(F)(F)c2cnn(C)c2)C1)C)C1CC1 C(CC)(C(O)C(C)C)NCC(CC1CCCO1)OC CC(C)CCC(O)C(=O)OCCCSc1cc(NC(=O)OC(C)(C)C)cn1C CC1CC(CSCC(=O)NCCCCCCN=[N+]=[N-])CCC1=O c1(C(=O)NC2(C(N3C(C(=O)OC)CC=CC3)=O)CC2)cc(=O)n(C)cn1 N1(C(C(=Cc2ccc(F)cc2)C)=O)CCCN(C(C2CC2(C)C(F)F)=O)CCC1 C(=O)(CCN1CCCO1)N1CCC(C(=O)NCC2COCCO2)CC1 C1(NC(C(c2ccc(F)cc2)(C)N(C)C)=O)CCCCC1NC(=O)CCC1CC1 C=CC(C)(C)C(=O)N1CCC(C(N2CCS(=O)(=O)CC2)=O)O1 N#Cc1ccc(CN2CCNCC2C(=O)N(C2CC2)Cc2ccncc2)c(Cl)c1 c1(C(=O)OC)cc(OC)cc(OC)c1CN1CC(C(C)C)CCC1C C(CCC1CCC1)(C(=O)N1CC2C=CC2C1)NC(C1C(=C)C1)=O c1(NCC(=O)NCCN(C(c2nc(F)ccc2Cl)=O)C2CC2)ccc([N+](=O)[O-])cc1 c1(N2CCCC(NC(C(C(C)C)C)=O)C2)ncnc2c1cnn2C CC(CNC(C1CC(C)(C)CO1)=O)CC(=O)NCC(C)CC1CC1 C1(C(=O)NCCC2(NC(=O)CSC3CC3)CCCC2)CCc2ccc(F)cc2O1 C(c1ccc(F)c(F)c1)=CC(N1C(CC)C(NC(C2CC(OC)C2)=O)CC1)=O CCC(C)C(C)CNC(C1(NC(=O)Cc2ncoc2C)CCCCC1)=O c1(SC(C(=O)NCC2(O)CN(C(COCCCC(C)C)=O)C2)C)ccccc1Cl N1(C(C2N(C(C)C)CCC2)=O)Cc2occ(C(=O)NC(C)(C)CC3CCC3)c2C1 C1(C(N2C(CC)CC(C)C2)=O)CN(C(c2cnn(C(F)F)c2)=O)CC12CCC2 C(=O)(CC(CNC(=O)C(C)N=[N+]=[N-])C1CCC1)NCCC(=O)NCC#C Cc1ccc(Br)nc1NC(C1CCN1Cc1ccc(O)cn1)=O c1(C(N(C)CC2N(C(CC3N(C(C)C)CCC3)=O)CCC2)=O)cc(F)cnc1O C1(NC(c2[nH]nc3ncccc23)=O)CN(C(C2CCCS2(=O)=O)=O)CC2(CC2)C1 C1(C(N(CCCCCNC(c2c(OC)n(C)nc2)=O)C)=O)Cc2nnc(C)n2C1 C(=O)(C1=C(Cl)CCOC1)N(CC)CC1CCCN(C(=O)CS(N)(=O)=O)C1 c1(C(N2C(CNC(C(C(C)C)O)=O)C(C)CCC2)=O)cc2c(cc1N)OCCO2 Cc1ccc(COCC(=O)NCCC2(NC(=O)CC3CNC(=O)O3)CC2)cc1 C1(NC(=O)C=CC2CC2)CC2CCC(C1)N2C(c1n[nH]cc1I)=O Cc1cc2c(cnn2C)c(N(C)C(c2ccc(C(F)(F)C(F)(F)F)cn2)=O)c1C Cc1cc(Cl)ccc1-n1cc(-c2cn(C)nc2NC(=O)OC(C)(C)C)nn1 N1(C(CN(C(COC)=O)C)=O)CCC(C2CC2)C1C(=O)NCC1(C)CCC(=O)N1 c1(COCC)nc(C)c(C(=O)NC(CCNC(C2CC(N(C)C)C2)=O)CO)s1 c1(C(=O)NC2C(NC(c3ccc(CC)nc3)=O)CCC2)nn(C)c2c1COCC2 CC(CCNC(C1(C(=O)OC(C)(C)C)CCC1)=O)NC(C1CC(CC2CC2)C1)=O c1(COC(=O)CC2CC2c2ccc(Br)cc2)cc2cc(Br)ccc2o1 N1(C(c2cc(Cl)cs2)=O)CC(C2(NC(C34CCCC3CC4)=O)CC2)C1 N#Cc1ccc(CCCC(N2CC(CNC(=O)Cc3cn[nH]c3)C3CC23)=O)cc1 C=C(C)CCCC(=O)N1CC2CC(NC(c3ncccc3F)=O)C2C1 N1(CC(=O)NCCN=[N+]=[N-])CCN(CC2CCOC2)CC1 C1(NC(C=CC(=O)N(C)C)=O)CCN(C(=O)CCC2CC(C)(C)CO2)C12CC2 c1(N2CCC(C)(COC)CC2)nc(C)cc(=NC(C)c2ccc(C)c(C)c2)[nH]1 c1(C(=O)NCC2CC(C(C(=O)C(F)=CC3CC3)C)C2)sccc1CC#N C1(C(=O)NCCC(CNC(CCC=CC)=O)(C)C)CCCC(F)(F)C1 C1(C(C)NC(c2cc(CC)on2)=O)CN(C(C2(CO)CCC2)=O)CCO1 C1(NC(=O)C=Cc2ccsc2)CCCN(C(c2cnn(C3CCOC3)n2)=O)CC1 C(=O)(C(=O)C(C)(C)C)NC1(C)CC(C(N2CC(S(C)=O)C2)=O)C1 c1(NC)cc(Cl)ccc1C(=O)NCC(C)NC(=O)CC1CC2(CCC2)C1 C1(C(=O)NC(c2ncc(F)cn2)C)CCN(C(=O)C2=NOC(C)(C)C2)O1 c1(NC(C)=O)cnc(C)c(C(=O)NC2C=CCN(C(c3ccc(F)o3)=O)C2)c1 N1(C(COCCCCCC)=O)CCCC2CN(C(C3CCC(C)O3)=O)CC12 C1(C(=O)NC2(CCCC(=O)NCC3(CCC)CCC3)CCC2)CC(C)(C)CCO1 CCC(CC)C(C)C(=O)NC(C(=O)N(CCO)CCN(C)C)C(C)C n1(CC)nc(CN=C(NCC2(c3ccccc3C)CCCC2)NC2CC2)c(C)n1 c1(N(C(C)=O)C(C)=O)ccc(N(N2CCCC2)CCN2CCC2C(C)C)cc1.CC c1(C(=O)NC2CC3N(C(C(C)(O)C(F)(F)F)=O)C(CC3)C2)cc2[nH]ccc2cc1Cl c1(CNc2cccc(N3CCN(C)CC3)n2)ccc(N2CCOCC2)cc1OC c1(CNC2C(C(N3CCOCC3)=O)CCCC2)cccc(O)c1F Cc1nn(C(C)C)cc1C(c1nnnn1C1CCOC1)NCC(C)(C)F C1(CC)(NC(c2cc(N(C)C)ccn2)=O)CCCN(C(c2cccn2C)=O)C1 C(=O)(CCC(C)(C)C)N1C(C)C(NC(=O)C(C)(C)c2ccno2)CC1 C(CC(O)C(=O)N1CCSCC1CO)NC(c1csnc1Cl)=O c1(C(=O)NCC2(O)CN(C(C(C)SCCCC)=O)C2)cc2c(ccn2C)[nH]1 c1(N2CCC(Oc3ccccc3)CC2)nc(N2CCOC(CF)C2)nc2c1CCC2 C1(C2CCN(C)CC2)(C(N2CC(N(C(C3N(C)C(=O)OC3)=O)C)C2)=O)CC1 CS(=O)(=O)c1ccc(C(=O)NC2CC3CC2CC3O)c(N)c1 C(=O)(CC(F)(F)Cl)NCCC1CCC(NC(C2(CC)COC2)=O)C1 C1(C(C)NC(CC=CC=C)=O)CCCCN1C(=O)CC1(C(=C)F)CCC1 c1(C(CC(=O)NC(C)CCCNC(c2cnc(Cl)[nH]2)=O)O)ccc(F)cc1 C1(NC(C2CC3(CCC3)C2)=O)CCCC12CN(C(c1ccco1)=O)C2 C1(C(N2C(C(=O)NC3(C(=O)NCC)CC3)CCC2)=O)CC12CCCCC2 N1(C(COCC#C)=O)CCC(C)(NC(c2cnn(C(C)(C)C)c2N)=O)C1 N1(SC)CCC2(CCC2)C(CO)C1.C(=O)(C1=C(C)OCC1)c1n2c(nn1)C1CCCCC12 C1(OC)CN(C(C2CCN(C(C)=O)C2)=O)CC1NC(c1c(C)cnn1C)=O c1(OC)cc(OC)c(C(N2CC=CC(NC(=O)CCCC(C)C)C2)=O)c(N)c1 c1(C(N(C(C)C(=O)O)CC)=O)cccc(-c2cn(CC(C3CCCO3)O)nn2)c1 CCCC(O)CC(=O)N1CCN(C(c2ncc(Br)cc2C)=O)C(C)C1 c1(C(=O)NCC(=O)NCC(N2CCC(c3cc[nH]n3)C2)=O)cncc(O)c1 N1(C(c2c(C)ccc(C)n2)=O)CCN(C(=O)CCCC(=O)NC(C)C)CC(O)C1 c1(OC)cccc2[nH]cc(CCNS(=O)(=O)c3cc(OC(F)F)ccn3)c12 C(=O)(CCCS(N)(=O)=O)NC1(C)CN(C(C2(C)CC(=C)C2)=O)C1 C1(C(N(C(CC(CC)C)C)C)=O)CCN(C(=O)C#CC(C)(C)C)CC1(C)C N1(C(CCCCC)=O)CC2CCCN(C(C3CCN(C4CC4)C3=O)=O)C2C1 N1(C(C(CCC)C)=O)CC2(CO)CC1(C(N1CCC3CC13)=O)C2 C#Cc1ccc(C(=O)N(CCC(C(C)(C)C)NC(C2CCC3(CC3)C2)=O)C)cc1 c1(C(C(N2C(C)(C)CC(C(=O)C3CC3)C2)=O)=O)cc(F)c(F)cc1F C1(NC(c2ccc(CCC)[nH]2)=O)CCCCC1NC(c1ccccc1C(C)=O)=O Cc1c(F)ccc(C(=O)NC(CNC(c2ccc(C(C)C)s2)=O)CC(C)C)c1N C(N=c1ncc(Cl)c[nH]1)c1c(NCNC(C(C(C)(C)O)F)=O)cccc1 N1(C(C(C=CC)O)=O)CCN(C(c2ncccc2N)=O)CC1C(C)(C)C C(CS(=O)c1ccccc1F)N1C(=O)NC(C)(C)C1=O C1(NC(C=C(C)Cl)=O)CCN(C(=O)CSCC2CCCCO2)C1C N1(C(C2(OC)CCOC2)=O)CCC(C2(O)CN(C(c3cncs3)=O)C2)CC1 N1(C(CC)=O)CC(C2CCN(C(c3ccc4c(c3)CN(C)CC4)=O)CC2)C1 C(C)(CO)(C(=O)N1CCC(OCC(N)=O)C1)NC(CSCCCC)=O C=CC(O)C(=O)NCC1(CCCNC(=O)Cc2ccc(C)s2)CCCC1 C12(CNC(=O)CCn3cccn3)CCCN(C(c3ccccc3F)=O)C1C2 C1(NC(c2nnc(C)s2)=O)COC2(CCN(C(c3cnc(C)nc3C)=O)CC2)C1 C1(C(N(CCCCCNC(C(CC)NC(N)=O)=O)C)=O)CC(F)(F)CCC1(C)C N1(C(c2scc(C)c2Br)=O)CCC2CCN(C(=O)CN(C)C3CC3)CC12 c1(C(=O)NCc2c(C(=O)NC(CN(C)C)CO)occ2)ncccc1F N1(C(CNC(=O)OCC)=O)CCCC2CN(C(C3C4CCCCC34)=O)CC12 N1(C(c2c(C)ccc(C)n2)=O)CCC2CC2(NC(C2CC3C=CC2CC3)=O)CC1 N1(C(CCCCOC)=O)CCN(C(C2CCc3c(nnn3C)C2)=O)C2(CCC2)C1 C(=O)(C1=CCCCCC1)N1CCC(N(C(c2cc(C)nc(C)n2)=O)C)CC1 c1(Cc2cc(C)sc2)nnc(N2CCC(Cc3ccc(C)s3)C2)n1C C(=O)(C(CC(C)CCC)N1CCOC(C(C)C)C1)NCCC C1(C(=O)N(C2CC2)CC2CCN(C(C3COC3)=O)C2)CCCCCC1 Cn1ccc(C(=O)NC(c2cccnc2)C(=O)NCC(O)C2(Cl)CC2)n1 c1(OC(C(=O)NCC2(CNC(=O)CCC3CCOC3)CCC2)F)ccccc1F C1(CC)CN(Cc2cc[nH]c2)CCN1C(c1cc(C(F)(F)F)cc(Cl)c1)=O C1(C(N2CC3(CN(C(c4c(NC(N)=O)cccc4)=O)C3)C2)=O)CCc2nn[nH]c2C1 C1(CC(=O)NCC2CN(C(C(C)O)=O)C2)COCCO1 C(CC(=O)Nc1csc(Cl)c1)(C(F)(F)F)NC(=O)Cn1cc(C2CC2)nn1 Cc1noc(CCNC(C2C(NC(C3CCO3)=O)CC2O)=O)n1 c1(OC(C)C)ccc(NC(C2CCC(NC(=O)C(C)NS(C)(=O)=O)C2)=O)cc1 c1(C(=O)NCC2CC(C)N(C(=O)Cc3sc(O)nc3O)C2)cncc2[nH]ccc12 N1(C(c2nc(CNC(c3ccc(C)nc3)=O)oc2)=O)CCC2(CNC(=O)C2)C1 C1(C(=O)NCC(N(C(CSC(C)C)=O)C)C2CC2)CCCN1C1CCCC1 N1(C(CC(C)C2CC2)=O)CC2CC(NC(=O)COCCc3cccs3)CC1C2 c1(SCC(=O)N(C)CC2(NC(=O)Cc3ccoc3)CC2)ccc2ccccc2c1 N1(CC(=O)NCCC(C)NC(c2c[nH]c(C(N)=O)c2)=O)CCCC1=O C(=O)(C(CC(C)C)NCc1nc(C)n(C)n1)N(CC(O)CN(C(C)(C)C)C)C c1(C(=O)NC(C(C)(C)NC(CCN(CCCCC)C)=O)C)oc(C2CC2)nc1C C(=O)(C(O)CCSC)N(C(C)CNC(c1cc(Cl)n[nH]1)=O)CC C=CC(C)(C)C(=O)NC1CCCN(CCNC(c2ccsc2C(C)=O)=O)C1 O=C(CCS(=O)(=O)N1CCOCC1)NC12CC(NC(=O)C(O)CC3CC3)(C1)C2 c1(COC(C2C(CCCc3cccc(C)c3)C2)=O)cc(C)ccc1N(C)C c1(C(N2CCC(C(F)C(N)=O)CC2)C(=O)NCCSC)cccc(C(C)(F)F)n1 C1(C(=O)NC2CC(F)(CNC(=O)Cc3cnn(C)c3)C2)(CC)CCOCC1 N1(C(c2cccc(C)n2)=O)CCC(NC(=O)CC2OCCC2(C)C)C(O)C1 c1(CC(N2CCCC3(CCOC3)C2)=O)ncc(C2=CCSCC2)cn1 C1(C(=O)O)(CO)CCCN1C(=O)CC1(c2cn(CCN(C)C)nn2)CC1 C1(C)(C(N2C(C#C)CCC2)=O)CC(O)CN1C(C1CC1OC(C)=O)=O N1(C(CCOCCOC(C)(C)C)=O)CC2CCC2(CNC(c2sccc2Cl)=O)C1 Cc1cccc(Cl)c1CC(=O)N(CCCNC(c1cnn(CC(F)F)c1C)=O)C S(=O)(=O)(c1cnn(Nc2cncc(Br)c2)c1)C(C1CC2(CNC2)C1)=O.C1CC1 S(=O)(=O)(c1cccs1)NCC(N1CC(C2N(C(C(CC=C)C)=O)CCC2)(O)C1)=O CCC(C)(C#N)C(=O)NCCCOCCNC(=O)C(C)(C)C1CCOC1 CC1=C(C)CN(C(=O)CCN(CCCO)C(C2CCCC(N(C)C)C2)=O)CC1 C1(C(C)C)(C(=O)NC(C)Cn2cncn2)CCCN1C(C12CSCC1C2)=O CCC(C)C(CC(=O)NC(COC)C(=O)OC)NC(=O)Cc1ccc(F)cc1 C(C(CC(C)C)NC(=O)Cc1csc(C)c1)NC(C(CN(CC)CC)F)=O CC1(NC(=O)CC2CC(=O)NC(=O)C2)CCCN(C(=O)CC2CCCCC2O)C1 Cc1nccc(C(=O)N(C)CC2CCCCN2C(=O)C(C)NC(N)=O)c1N c1(C(=O)NC(CC=C)CNC(=O)CCn2cnnn2)ccc(N(C)C(C)=O)cc1 C1(C(=O)NC2(CC=C)CC2)CCC2CC1CN2C(=O)CC1(CO)CCCC1 N1(C(C2C(CC(C)C)C2)=O)CCN(C2CCN(C(=O)C=C(Cl)Cl)CC2)CC1 c1(C(=O)NC2CCN(C(c3nc(C)nn3C)=O)C2)cnn2c1OCCCC2 C1(NC(CC(=C)C)=O)CN(C(=O)CC2CSCN2C(=O)OC(C)(C)C)C(C)(C)C1 CC(C)C1=NOC(C(=O)NC(C2CN(C(=O)C(C)(C)OC(C)C)C2)C)C1 N1(C(C2C(C(=O)OC)C2)=O)CC2(CCN(C(=O)Cn3ccccc3=O)CC2)C1 CCCCC(C(=O)N(CC(C)C(F)(F)F)C)NC(=O)CN1CCCCC1C c1(C(=O)NCC(C)NC(C2CCC2c2nc[nH]n2)=O)cccc(Cl)c1O N1(C(CC2CC(=C)C2)=O)CCC(CNC(c2csc(C(N)=O)n2)=O)(OC)C1 N1(CC2(C)CCC(C)C2)CCN(C)C(c2cn(Cc3ccc(F)c(Cl)c3)nn2)C1 N1(C(c2cc(CC)no2)=O)CC=C(C(C)(C)C(=O)N2Cc3ccc(O)cc3C2)C1 C=C(C)CC(C(=O)N1CCC(O)(CC)C1)NC(C1CC(O)C(F)C1)=O c1(C(=O)NCC2(F)CCC(NC(C(C)C(F)(F)F)=O)C2)noc2c1CCCCC2 c1(NC(C2C(C(C)NC(c3c(C)cnn3C)=O)C2)=O)cc(Cl)cnc1O CCC(C)CC(=O)C(=O)NC1CCC(CCC(N2CCNC(=O)C2C)=O)C1 N1(C(C(C)OCCC=C)=O)CC(CO)(NC(=O)C(C)NC(N)=O)C1 c1(C(=O)OCC)cc(C(C(=O)NC(CC)C2CC2)N(CC(=O)OC)C)ccc1O c1(CC)c2ccc-2c1F.N12CCCC(C1)OC(=O)C1CC1C2=O.C(C)(C)(C)O.OC C(=O)(N=c1cc(-c2cccc(F)c2)[nH][nH]1)c1ccc(-n2c(C)cc(C)n2)cc1 c1(C(N2C3CC(CNC(C(CCCC)C)=O)(OC3)C2)=O)cc2c(C)cccc2o1 C1(C(N(CC)CC)=O)CC12CCN(Cc1ccc(NC3CCN(C)C3)cc1)CC2 c1(C(=O)NC2C(CNC(C(C3CC3)SC)=O)CC2)ccnn1C C1(C2(O)CCN(C(C3CC3F)=O)CC2)(NC(C(C(C)C)N(C)C)=O)CC1 N1(C(C(CC)OC)=O)CCN(C(=O)Cn2nccc2C)C(c2cccc(Cl)c2)C1 c1(C(N2CCN(C(CS(=O)(=O)NC)=O)C(C)C2)=O)cc(F)c(F)c(O)c1F C(=O)(C(C)(C)CC(=O)N1CCC(C(=O)Nc2cnn(C(F)F)c2)C1)OC C1(C)(C(=O)NCC2(C)CCN(C(CCCC=C)=O)C2)CC(C(F)(F)F)=NO1 c1(OC)cc(C(=O)N(C2CN(C(C3CC(C)C3)=O)CCC2C)C)ccc1F c1(CC(=O)NCCC2CC(NC(C3CC4CC4C3)=O)C2)ccc(Cl)cn1 c1(CNC(c2coc3c2COC3)=O)c(F)cc(F)c(F)c1F C12(C(=O)NCC3(C)CCCN(C(c4ccco4)=O)C3)CCCCC1CS(=O)(=O)C2 N1(CC)CCCCC1C(N1CCCC(C(=O)NCC2OCCC2(C)C)C1)=O C(=O)(C1COc2ccccc21)N1CC2(OCC(NC(CCC(C)(C)C)=O)C2)C1 C1(CNC(CNC(C(CC)C)=O)=O)CN(C(C2COCCN2C=O)=O)CCN1C N1(CC)CCC(O)CC1.c12noc(n1)C(C)NC(=O)NCCN2 C1(NC(CCCC=C)=O)CCCN(C(=O)Cc2ncn(C)c2C)C1C N1(C(CSc2c(C)n[nH]c2C)=O)CCN(C(c2ccc(=N)[nH]c2)=O)C(C)C1C C1(C(=O)NC2CN(C(c3nnc(O)nc3O)=O)C3CC23)COC2(CCC2)C1 C(=O)(CC(CC(C)C)NC(C1CC(C)CC(=O)N1)=O)N(CC(F)F)CC N1(C(C=Cc2c(C)ccnc2)=O)C2CC1CN(C(=O)C(CCO)N(C)C)C2 CN1C(=O)CCCC1C(=O)N(CC(Cl)=CCl)C(CC(C)(C)C)=O c1(C(=O)NCC(=C2CN(C(C3CC=CCO3)=O)C2)F)c(Cl)nc2ccccn12 C(=O)(CCCN=[N+]=[N-])NCC1N(C(C2CCCC(C)O2)=O)CC(O)C1 CCCC(C(=O)NCCCC(N1CCOC(CF)C1)=O)NC(=O)OC(C)(C)C C=CCC(CC(C)C)C(=O)NCC1CN(C(=O)CC2CC(=O)C2)CC1O c1(C(N(C(CCNC(C(CC)(C)CO)=O)C)C)=O)cc2cnc(Cl)cc2s1 c1(C2CCN(C(=O)NC3CCC(SC)C3)CC2)ccc([N+](=O)[O-])cc1 N1(C(C2(C=C)CCC2)=O)CC(NC(=O)Cc2ccc([N+](=O)[O-])cc2)C(N=[N+]=[N-])C1 C#Cc1ccc(C2CC2C(=O)NC2(CNC(=O)C(C)(C)C(=C)C)CCOC2)cc1 C1(C(C(=O)N(CCCCCNC(Cn2c(C)nnn2)=O)C)C)CCC(=O)N1C Cc1ccc(OCC(=O)NC(C)(CNC(=O)Cn2cc(CO)nn2)CO)c(F)c1 C(CCCCCNC(C1CCC1c1nc(S)n[nH]1)=O)NC(=O)C(Cl)=CCl c1(NC(=O)CCn2cncn2)c(C2CC2)nc2ccccn12 CS(=O)(=O)c1sccc1CNC(C1CC2CC12)=O C(=O)(CC(C)(C)C)NC(C(=O)NCCCC1N(C(c2c(C)con2)=O)CCC1)C Cc1nc(C)c(CNC(=O)C(C2CCCC2)NC(c2cnn(C)c2N)=O)[nH]1 C1(NC(CCC#CC)=O)CN(C(=O)COC(F)(F)C(F)(F)F)CC1(C)C C1(C)(CNC(C=C(CCC)C)=O)CCCN1C(c1cc(C)c[nH]1)=O C1(CNC(C(CC)(F)F)=O)CCCC2(CN(C(C3(CCOC)CCCC3)=O)C2)O1 C1(C(=O)NC(CCOC)CNC(=O)C(C)=CC2CC2)CCS(=O)(=O)C1 c1(CCNC(N2CC(c3ccccc3)CC(C)C2)=O)cc(Cl)c2c(c1)OCCO2 c1(C2(C(N(CC(C)CNC(=O)Cc3cscn3)C)=O)CC2)cccc(C#N)c1 c1(NC(N2CC(C(=O)OC)C(F)(F)C2)=O)cncc2nncn12 C1(C(N2C3(CN(C(CSC)=O)C3)CC2)=O)C(C)OCC(=O)N1Cc1ccccc1 C1(C(N2CCC(OCc3cn(CCCC)nn3)CC2)=O)CC(C)(C)OC1(C)C C12(C(=O)NCC(NOCC)=O)CCC(NC(C3CC(=O)CO3)=O)(CC1)C2 CCC(C)(C)CC(=O)N1CCC(c2ccccc2)C(NC(=O)C(C)CF)C1 c1(C(N(C2C(C)CN(C(=O)Cc3csc(S)n3)CC2)C)=O)nc2ncccn2n1 c1(NC(C2C(NC(=O)CCCCCl)CCC2)=O)ccnc(F)c1Br C(CN=c1[nH]cncc1I)C1CCC(NC(c2cncc(OC)c2C)=O)C1 c1(C(C(=O)NC(C)CCCCNC(c2nnn(C)c2N)=O)C)ccc(F)c(F)c1 c1(OC)cccnc1C(=O)NC(CCN(C(=O)C(C)CO)C)c1cccs1 CCC(O)(CC)CCNC(=O)C(C(C)(C)O)NC(=O)Cn1cc(Cl)cn1 C#CCCC(C)(c1nnnn1-c1ccccc1Cl)NCC1CCS(=O)(=O)N1 N1(C(=O)CC2CCCCC2F)CCn2ncc(O)c2C1 C(=O)(C1=CC(C)(C)C1)N(C1CCN(C(C2C(CC)CCO2)=O)C1)C CC(C)C(F)(CNC(=O)C=Cc1ccc[nH]1)C(=O)NCC12CC(CO)(CO1)C2 CCC[SH](=O)=O.n1(CC(=O)O)cc(CNC(c2cn(-c3ccncc3)nn2)=O)nn1 CCC(C)C(CNC(c1cc(CNC(=O)C(O)CSC)[nH]n1)=O)CO c1(OCC)ccccc1C=CC(=O)NC(C)C(C)Oc1ccc(F)cc1 Cc1cc(C(N2CCCCC(NC(=O)COC3CCCC3)C2)=O)nc(O)n1 C=CC(C)(C)CC(=O)NC1CC(CNC(c2ccnc(C)c2)=O)C1(C)C Cc1noc(C)c1C=CC(=O)N(C(CNC(=O)C=C1CCC(C)C1)C1CC1)C C(=O)(C(CC(C)(C)C)OC)N1CC(CC(C)NC(CCN(CC)CC)=O)C1 c1(N(C)CC2N(C(C(C)=C(CC)C)=O)CC=C2)ccc(C)c(C(=O)OC)c1 c1(C(=O)NCC2(C)CCC(NC(CN(CC)CC)=O)CC2)cc2n(c1)CCOC2 N1(C(C=CC)=O)CC2C3CCC(C3)C12.C(=O)(CC(C)C)N1CC1=O CC(C)C(C(=O)NCC(C)(C)NC(=O)CCn1ccnn1)N(C)C C#Cc1cc(C(N2CC(CC=C)(NC(c3ccoc3Cl)=O)C2)=O)cc(F)c1 C=CCC(C)(C)CC(=O)N1CCC2CN(OC(C3CCC(C)NC3=O)=O)C2C1 Cc1cc(Cl)ccc1C(=O)N(C1CCN(C(c2coc(C#N)c2)=O)CC1C)C C(=O)(CCC(C)(F)F)NC1CCC(CCNC(c2ccc(C(=O)OC)s2)=O)C1 C1(NC(c2c(C)nccn2)=O)CN(C(c2cc(C(F)(F)F)ns2)=O)CC12CC2 Cc1cc(C(N2C3CN(C(c4ccc(F)c(F)c4O)=O)CC23)=O)ccc1[N+](=O)[O-] c1(C(=O)NCC2C(CNC(c3c(CCC)[nH]cc3)=O)C2)c(C(C)C)cccc1C Cn1ccc(-c2cn(Cc3ccc(C(N4CCC4)=O)o3)nn2)n1 C(C(C)C)(C(O)C(=O)NCC12CC(CO1)N(C(C1C3CC(=O)CC13)=O)C2)OC CCCCCCC(CC)C(=O)N1CCCCC1CNC(C1CC(=O)C1)=O CS(=O)(=O)c1ccc(CNC(=O)NCCCc2ccon2)nc1 c1(CCC(N2CC(Cc3cn(CC=C)nn3)OCC2)=O)ccc2[nH]ccc2c1 C#CCCC(=O)N(C)CCOCCCNC(=O)C(c1ccn(C)c1)C c1(C(N(C)CC2N(C(c3c(C)c[nH]n3)=O)CCC2)=O)cc(C#N)c2n1CCCC2 C#Cc1cnn(C)c1C(=O)NCc1cc(C(=O)NCC2CC[Si](C)(C)C2)no1 CC(CO)(C(=O)N1CCC(O)C1)NC(=O)COCCCF.C(=O)N(C)C C(=O)(C(CCSC)NC(=O)NCCc1cncc(Br)c1)OC C1(C(=O)NC2(C)CN(C(C3CC(OC)C3)=O)C2)CCCCN1C(C)C N1(C(C2C(CNC(COCC=C)=O)CCC2)=O)CCN(C2CC2)C(C)C1 C(=O)(C1CCCc2c[nH]nc21)NC1CC(CNC(CNC(CC)=O)=O)C(O)C1 C=Cc1ccc(C(=O)N(CC(C)N(C)C(c2cc(CC(C)C)[nH]n2)=O)C)cc1 C(=O)(C(C)(C)CC(=O)N(CCCOCCNC(C1CC(C(F)F)C1)=O)C)OC C(c1c(F)cccc1F)=CC(N1CCC(CNC(c2c(C)cc(C)o2)=O)C1)=O N1(C(=O)CCC2CC2(F)F)C(CNC(=O)C(F)(F)C(O)C2CC2)CC2COCC12 Cc1ccc(NC(C=CO)=O)c(F)c1.C1(=O)C=CC(=O)OCCN1C.C(C)(C)(C)O c1(C(N2CCC(NC(c3cc(CC)nn3C)=O)C2)=O)cc(C)n(C)c1C C12(NC(CSCCCC)=O)CCCC(NC(=O)C(F)=C3CCCC3)(C1)C2 Cc1ccc(N)cn1.C12(C(N(CC(=O)NCCC)C)=O)CC(C(=O)N(C)CCF)(C1)C2 Nc1cccc(C(=O)NCC2CCN2C(C2CC3(C2)CC32CC2)=O)c1Br c1(CC(=O)NCC(C)N(C(=O)CSCCC#N)C)ccc(-c2nc[nH]n2)cc1 Cc1c(N)ccc(C(=O)NC2CCCCC2CNC(=O)Cc2cnsc2)c1Cl C1(CC=C)(NC(c2cc(OCC)ns2)=O)CCN(C(=O)CC=C(Cl)Cl)CC1 N1(C(C(=O)OC)CC(C)C)CCC2(CCCN2S(=O)(=O)C2CC(SC)C2)CC1 C1(C(=O)NC2C(CNC(c3cnc(O)s3)=O)CC2)CCc2nc[nH]c2C1 C1(CC(=O)NCC(C)N(C)C(c2n[nH]cc2-c2ccncc2)=O)CCS(=O)(=O)C1 CC1(C(=O)O)CCN(C(=O)CN2CCN(C(=O)CC#N)CC2)C1 Cc1cc(Br)ncc1CO.C1(c2nnnn2C(C)C)C(C)(CC)N1 C(CCC(F)(F)F)N(C(=O)C=CC1CCCN1C(c1cccc(F)c1)=O)C N1(C(CC(COC)C)=O)CC(NC(c2ccc(SCCCO)cc2)=O)CC(C)C1 C(c1cc(Cl)c2c(c1)OCO2)=CC(N1CCC(C(C)NC(c2cc(Cl)no2)=O)C1)=O c1(C(=O)NCC(C)N(C(=O)CCc2ccccc2F)C)cccc2nnn(C)c12 c1(-c2c(C(c3nnnn3C3COC3)NCC(=C)Br)c[nH]n2)ccc(Br)cc1 C1(CC(=O)NCCCc2cn[nH]c2)CN(C(=O)CSCC(F)F)CCO1 c1(COCCN2CCN(C(C=CC=CC)=O)CC2)c(F)ccc2occc12 Cc1c(NC(=O)NC(C)CN2CCCC(C)C2)[nH]c2cc(Cl)ccc12 C#Cc1ccnc(C(=O)NCC2CC(NC(=O)Cc3ncc(Cl)s3)C2)c1 N1(C(CSC)=O)CC2CC(CNC(=O)COc3ccc(F)c(Cl)c3)CC1C2 c1(CC(C)C)ccc(-n2ccnc2)cc1.C1(C2C(=O)N2CC(C)C)CCOCC1 c1(C(=O)NC2CCC(CNC(Cc3cccc(C)c3)=O)C2)sc2nccn2c1C c1(C(=O)OCC)cc(C(N2CCC(N(C)C(C3CC34CCC4)=O)C2)=O)[nH]c1C O(NC(=O)C(c1ccco1)NC(=O)C(CSC)OC)CC(=O)OCC N1(C(c2ccc(CCC)s2)=O)CCC(CNC(c2c(C)ncn2C)=O)C12CCC2 C1(NC(C2CC23CCOC3)=O)CCCC(NC(C2CCCO2)=O)C1 C1(CCNC(CN(CCC)C(c2sccc2C)=O)=O)OCCC1C N1(C(c2ncn(CC)n2)=O)CCCC(CO)(NC(C2COCCO2)=O)C1 C=C(C)COCC(=O)NCC=CC(=O)NC1(C(C)O)CC1 N1(C(CCOC)=O)CCC2CCN(C(=O)C(c3cc(C)cc(F)c3)C)CC2C1 C1(NC(C=C(C)C)=O)CCN(C(=O)Cc2cc(C)cs2)CC1C(C)C C1(CNC(C2N(C(C)(C)C)CC2)=O)CCC(F)(CNC(C2CCC(=O)N2)=O)CC1 Cc1nn[nH]c1SCC(=O)NCC#CC(=O)N(C)C c1(C(=O)NCC2(C(C)NC(C(C)c3cccs3)=O)CC2)ccnc(S(N)(=O)=O)c1 CC1CC2CN(C(C3CCC3)=O)CC2N1C(C1CCN(C(c2cccs2)=O)CC1)=O C1(NC(C(CC)c2ccccc2)=O)CCC(NC(=O)CCS(C)=O)CC1 C1(C2CC2)(CNC(CC2(NC(C(c3ccn(C)n3)C)=O)CCC2)=O)CC1 n1(CC=C)cc(C(=O)NCC(C)N(C)C(c2cn(CC3CC3)nn2)=O)cn1 C#Cc1ccc(C(=O)NC(CCOCC)C(=O)NC2CC(OC)C2(C)C)cc1C C(=O)(CCC(=O)C1CC1)N1C(CC2C(C(C)C)OCC2)CCC1 c1(SCC(=O)NCC(C)NC(=O)CS(=O)(=O)NC2CC2)ccsc1[N+](=O)[O-] c1(N2CC(CC=C)(NC(c3cnn(C)n3)=O)C2)ncc(OCCOC)cn1 c1(C(=O)NCCC2N(C(C=COCC)=O)CC(F)(F)C2)ccc2sccc2c1 C(=O)(C(O)C(F)(F)F)NCC=CCNC(c1cc(C)no1)=O N1(C(c2ccc(OC)s2)=O)CCC2(NC(C3CN(C(C)=O)C3)=O)CC2C1 c1(N(C(=O)CNC(=O)CCc2cnccn2)CC)ccc(Cl)cc1 c1(SC)cccc(CCNC(=O)CC2CNCC23CC3)c1 N1(C(C2CCN(C(C3C(COC)CC3)=O)C23CC3)=O)CCC(O)(C2CC2)CC1 c1(C(=O)OC)ccc(C(=O)NCCCN(C)C(C2CC3CCC23)=O)cc1Cl CC(C)C(C(=O)N(C)C)NC(=O)C(CNC(C1CCS1(=O)=O)=O)CC1CC1 n1(CC(=O)NCC=CCNC(C2CCC3CCC23)=O)nc(O)ccc1=O n1(C(CC(N2CCCCC(OC)C2)=O)C)cnc2ccccc12 CC1CC(NC(c2nc(C3CC3)no2)=O)CN1C(=O)CC1(C)CC1(F)Cl c1(-c2ccc(SC)cc2F)cc(C(=O)NC2(C)CC2)c2cn[nH]c2c1 N1(C(C(C(CNC(Cn2c(C)cc(C)n2)=O)C)F)=O)CCC2(CCOC2)CC1 N1(C(C(C)c2cc[nH]n2)=O)CC2CCC1CN2C(=O)C(c1cnn(C)c1)O C1(c2nnnn2CC2CC2)(Nc2ccc(OC)cc2)CCCC(CC#N)C1 C1(C(=O)NC2C(NC(CC3(OC)CCC3)=O)CCC2)CCC2(CCCCC2)C1 N1(C(C(CCCC)(F)F)=O)CC2CCCC(C1)N2C(C1CC1(C)C(F)F)=O C1(C(=O)NC(CCC=C)C2CC2)CCCCCC1NC(c1cc(O)nn1C)=O C(=O)(C1=CC(O)C(O)C(O)C1)N1CC2CCN(C(c3c(C)nn(C)c3)=O)CC2C1 CCC(C(=O)NC(C(=O)N1CC(C2CCCOC2)C1)C1(O)CCC1)OC C1(NC(CN(C)CC2CCCC2)=O)C2CCC1CC(NC(=O)C(N)=O)C2 c1(NC(C2(SC)CCNC2)=O)ccc(OCCC(C)C)cc1 C1(C(=O)NC(C2CN(C(C3(S(N)(=O)=O)CC3)=O)C2)C)CC2COCC(C1)C2 C(c1ccc(Cl)cc1F)=CC(=O)NC1CCCN(Cc2cnn(C3CC3)c2)C1 N1(C(CCCOCC)=O)CCC2CCN(C(=O)C(F)Cc3ccccc3)CC2C1 Cc1cc(OCCC(=O)NCC2(C)CCCN2C(=O)C2=CCOC2)cc(C)c1 c1(C(=O)NCC2CCCC(CNC(C3C(C=C)C3)=O)C2)cncc(C#N)c1 n1(CC)cnc2[nH]c(=NCc3ccoc3)nc(N3CCCC(C(F)(F)F)CC3)c12 C1(C)(CNC(c2cc(C(C)C)nn2C)=O)CN(C(C2CSCCS2)=O)CCO1 c1(CC(=O)NC2CCN(c3ccccc3Cl)C2=O)cccc2c1[nH]c1ccccc21 N1(C(c2c(C)ccc(OC)n2)=O)CC2CCC1CC2NC(=O)C(F)=C(C)C c1(C(N2C(C(=O)NC)CC(O)C2)C(=O)NC(C)(C)C)cc(C)cc(Br)c1 c1(C(=O)NC2CCN(C(CC(C)F)=O)C23CC3)cc2cnccc2o1 N1(C(c2cn(C)cc2C(F)(F)F)=O)CC(NC(=O)C(=O)c2ccco2)CC2(CC2)C1 c1(COCCCN2CCC(NC(=O)CCCc3ccsc3)C2)cccc(Cl)c1 C1(C)(CNC(CC2CC(CC)C2)=O)COCCN(C(=O)CCn2cncn2)C1 N1(C(c2ccc(C(=O)OC)o2)=O)CCC(NC(=O)C(F)(F)CF)CC1C1CC1 c1(CC(=O)NCCOC(CNC(CC2CCN(C)C2)=O)(C)C)ncc(F)cc1F C(=O)(C1CCCn2cc(C(C)(C)C)nc21)NCc1cc(OC)c(OC(F)F)cc1 c1(C(=O)NCC(C)N(C(c2c(C)nc(C)[nH]2)=O)C)ccnc2ccc(O)cc12 C1(CNC(Cc2c(C)n[nH]c2C)=O)CCN(C(=O)CC(O)C2CC2)C1(C)C c1(-n2cc(C(N(C(C(C3CCC3)OC)=O)C)C)nn2)cccnc1C(=O)O c1(OCC(=O)NC2CCN(C(COCC#C)=O)C2)cccc(C(N)=O)c1 C1(C(N(CCCNC(=O)Cc2cscn2)CC)=O)CCCSC1 c1(C(=O)NC2CCCN(C(CC3CCN(C)C3)=O)CC2)ccc(F)c2ccsc12 c1(C(=O)NC(CN(C(C(C=C)O)=O)CC)C)c(C(C)=O)cnc2ccccc12 N1(CC)CCC(NC(C2CC3CC3N2C(=O)CC2CCCC(=O)C2)=O)CC1 CCC(C)CC(C)C(=O)NCCC(C)(C)CNC(=O)CCNC(C)=O c1(C(=O)NC2CCC(NC(c3c(C)ccs3)=O)C2)cc(Br)c(Cl)cc1F C1(CNC(C2C(Cl)(Cl)C23CC3)=O)COCCN(C(=O)C(F)F)C1 C(C)(CC(C)NC(=O)CSc1cn[nH]c1)NC(C(C)NC(C)=O)=O C1(C(N2C(C(CNC(CC(C)(F)F)=O)(C)C)CCC2)=O)C(F)(F)C12CCC2 C1(N(C(C(c2c(C)noc2C)CC)=O)C)C2CN(C(c3ccnc(C)c3)=O)CC12 C1(NC(CCCOCCC)=O)CCC(CN(C(=O)Cc2conc2C)C)CC1 C12(C(=O)NC(C(=O)NC3(CCOC)CCC3)Cn3cccn3)CCCC1C2(F)F C1(c2nnc(C)o2)CN(C(=O)N(CCCn2ccnc2C)CCO)CCO1 C1(C(=O)NC2C(C(N(C)Cc3nnc(CC)o3)=O)C2(C)C)CC2CCC(C1)O2 N1(C(C2(F)CCN(C(c3cc(SC)oc3)=O)C2)=O)CC(C#N)C2(CCC2)C1 c1(OCC(=O)NC2C(NC(CS(CC)=O)=O)CC2)cccc(C)c1C c1(CC)cccnc1C(=O)N(C1CC(NC(C2CCSC2)=O)C1)C c1(CC)nc(C)c(C(N2CC3CC2C3CNC(=O)CCc2ccc(F)nc2)=O)s1 C1(NC(CNC(C(CC)CC)=O)=O)CCCN(C(c2onc(Br)c2C)=O)CC1 C1(C(=O)NCCCCN(C(C2(CCC)CCC2)=O)C)COc2ccc(F)cc2C1 C1(C)(C(N(CC(C)O)C)=O)CCN(C(C2CC2Cl)=O)CC1 c1(C(N(C(CNC(C2(OC)CCOCC2)=O)C)C)=O)[nH]nc2c1CCC2(C)C c1(COC(C2C(C(F)(F)F)CC(=O)NC2)=O)nnc(O)c2ccccc12 CCC(C)CC(C(=O)NC1CC(CO)C1)NC(=O)Cc1cncn1C C(=O)(C(=O)CCC(C)C)N1C(CC(=O)NCc2c(C)nn(C)c2)CC(C)(C)C1 c1(C(=O)NC(CNC(Cc2c(C)nc(S)s2)=O)C)nccc2c(Br)cccc12 Cc1nnn(CC(N2CC(Cn3cc(C4CCCCC4)nn3)C2)=O)n1 c1(OC(C)C(=O)NCC2CCCN2C(=O)CC2CCC2)ccccc1F N1(C(C(CC=C)(C)C)=O)CCOC2CCN(C(=O)CSC(=N)N)CC12 C1(CC)CN(C(c2ccn(C(C)(C)C)n2)=O)CCN1C(c1ncn2c1CCC2)=O C(=O)(CCC(=O)NCC(O)CCNC(=O)C(C)NC(=O)COC)NCC C(C1CCN(C(=O)C=CC2CCCC2)CC1)=CC(=O)N(CCC)CCO c1(CC)ccc(C(=O)NCC(C)NC(=O)CCN2CCCC2=O)cc1C(F)(F)F Cc1sc(C(=O)NC(C)CNC(c2ccc(N)cc2Cl)=O)cc1[N+](=O)[O-] c1(C(N2C(C)CC(CC(=O)NCCC(C)(C)F)C2)=O)ccc(F)cc1F N1(C(N2CCC(CN=c3[nH]ncc(C)c3)C2)=O)CCC2OC(=O)NC2C1 C12(NC(C(CCC)CC)=O)CCC(CNC(C3CCCC(C)C3)=O)(CC1)OC2 c1(C(C)N(C(=O)NCCOCc2cncc(Cl)c2)C2CC2)cccc(S(N)(=O)=O)c1 C1(C2(O)CN(C(=O)CCC3CC3)C2)(CNC(c2c(C)[nH]nc2C(C)C)=O)CC1 C1(CNC(=O)NCC2C(C)C2)CCN(CCC(F)(F)F)CC1 c1(C(=O)NC2CC3CN(C(C(C)C(F)(F)F)=O)C2C3)n[nH]c2c1CSCC2 N1(C(CCC(CC)OC)=O)C(C)CC2CN(C(=O)CCCC(N)=O)CC12 c1(OC)cccc(CC(=O)NC(C)(CNC(c2csc(C)c2)=O)C2CC2)c1Cl N#Cc1cc([N+](=O)[O-])cnc1NCC1CC(NC(=O)CCc2nccs2)C1 CCCC(C(C(=O)NCc1ccccc1Br)N1CCCC12CCC2)OC C(=O)(C(C#N)CC)NC1(C(=O)NCC(C#C)CC)CCC1 c1(OC)cccc(NC(=O)CN2CCN(C(=O)CCc3ccco3)CC2)c1 C1(CC(=O)NC2CCC2CNC(c2csc(C(F)F)n2)=O)C=CCCC1 C(CC(=O)NCc1nccc(OC)n1)(C(C)C)NC(C(CC)CN(C)C)=O c1(C(N2CCC(CNC(C(c3c(C)noc3C)C)=O)C2)=O)ccc(Cl)c(F)c1N c1(CC)c(C(N2CC(C(=O)NCc3[nH]nnc3C)C(CC)C2)=O)cnn1C C1(C(=O)NCCCN(C(C2CC(OC)C(OC)C2)=O)CC)CCn2nccc2C1 C1(C(=O)NC2CCC(NC(CCc3cc(C)on3)=O)CC2)CCc2nn[nH]c2C1 c1(C(N2CC(N(C(C=COCC)=O)C)C(F)C2)=O)c(Cl)cc(Cl)c2ncccc12 N1(C(C(C=C=C)C)=O)CC(NC(c2c(C)nsc2Br)=O)CC2(CCC2)C1 c1(CCC)ncc(C(N2CC(CC(C)NC(C3(n4nccn4)CC3)=O)C2)=O)s1 N(C1CCOc2c(C)cc(F)cc21)(C(=O)CCCCCCc1nn[nH]n1)CC Nc1c(C(N2CCCCC2CCNC(C2CCCC2(F)F)=O)=O)nc(O)nc1O c1(CC)cnc(C(=O)NCC(CNC(=O)CCc2ccc(C(=O)OC)[nH]2)C)nc1 C1(NC(=O)COc2ccsn2)CN(C(C2SCCS2)=O)C2(CCC2)C1 C1(NC(C2C(C)=CCS2)=O)C2CC(NC(c3c(C)ccn3C)=O)CC12 CCCCCC(c1nnnn1C1CC1CC)Nc1cn[nH]c1 CCS(=O)CC(=O)NCC12CC(CNC(=O)C(C3CCCC3)OC)(CO1)C2 C(CN=c1nc2scnc2c(NC2CCC3(C2)CC3(F)F)[nH]1)N(C)C N1(C(CCc2ccn(C)n2)=O)CCOCC(NC(=O)COC2CCCCCC2)C1 c1(CNC(=O)Cc2ccc(F)nc2)ccnc(C(N2CC3CCC3C2)=O)c1 C1(OC(C#CC(C)C)=O)CC(F)(F)CC1OC(C1(C(F)(F)CO)CCOCC1)=O CC(CNC(c1ccsc1C#N)=O)C(F)C(=O)N(CCCc1ccco1)C N1(C(c2c(=N)cc[nH]c2)=O)CC2CC1CC2NC(c1cc2n(c1)CCC2)=O N1(C(C2CN(C(C)C)C2)=O)CCCC(C)(NC(C23CC2CCC3(F)F)=O)C1 C1(C(=O)NCC(=O)OCC)(COC)C=CCN1C(C1CCCSC1C)=O N1(C(CC2(OCC)CC2)=O)CC(CNC(c2cn(CC)nc2C)=O)C(C)(C)C1 C12(CNC(c3c(CC)nn[nH]3)=O)CCCC1CCN2C(=O)Cc1ccsn1 c1(CCC)n[nH]c(=NC(C)CC(C)NC(c2cc(OC)ns2)=O)s1 C1(CN(C)Cc2cccc(F)c2OCCO)CCCCC1C1CCCCC1 c1(C(N(C)CC2(O)CN(C(C3(OCC)CCC3)=O)C2)=O)ccc(C)nc1 C1(CNC(C(c2cnn(C)c2)OC)=O)CCN(C(=O)CC2(C#N)CCC2)C12CC2 C(C(O)C(C)(C)C)N(C)C(C1CCC(NC(C2(O)CCSC2)=O)C1)=O C(=O)(C(C)CC(F)(F)F)N1C(C(C)NC(CCNC(COC)=O)=O)CCC1 CCCCC(C(=O)N1CCCC(O)(CNC(=O)C(=Cc2ccco2)C)C1)N(C)C C=CCC(CNC(=O)C(F)C(C)(F)F)C(=O)NCCN1CCCOCC1 C1(C(=O)NC(CCNC(c2n[nH]c(C)c2C)=O)(C)C)OCCN(C)C1=O C(N=c1[nH]c2ccc(Br)cc2o1)C1(O)CCN(C(CC(COC)(C)C)=O)CC1 C1(NC(C(N2CCCCCC2)C)=O)CC2CCC1(NS(C)(=O)=O)C2 N1(C(CC(=O)OC)=O)CCC2(CNC(c3cn4ccnc4cn3)=O)CCCCC12 Cc1ccc(C(=O)NCc2csc(C(=O)NC(CN(C)C)C(C)C)c2)cc1F C(=O)(CCCCCNC(N)=O)N1C(CCNC(C(CCC)C)=O)COCC1 C=C(Cl)CCC(=O)NC(CCC1CCC1)C(=O)NCC1(CO)CCCO1 N1(C(c2cc(C(C)C)n(C)n2)=O)CC2(CCCC2NC(=O)C2=CCC2)C1 N1(C(CCOCCC)=O)CCN(C(=O)C=Cc2ncco2)CC1c1ccccc1 N1(CC)CCCC1CC(=O)NC1CC(NC(=O)C(F)(F)c2ccnn2C)C1 c1(OC)ccc(C)c(C(N2CCC(NC(=O)C3=CCS(=O)(=O)C3)C2)=O)c1N C1(NC(=O)CCC2CC(F)(F)C2)C2CC3CN(C(=O)C4=CCCCC4)C1C3C2 C1(C(=O)NCC(CC=C)NC(=O)Cn2cccn2)CC2(CCC2)CCO1 c1(C(=O)NCC=CCNC(C2CC23CC(O)C3)=O)cccc(C2CCOC2)c1 C(=O)(N1OC2CCC1C2)C1(NC(c2c(C)nns2)=O)CCCC1C C1(NC(Cc2c(C)occ2)=O)CN(C(=O)C(C)(C)C2CCC2)CCC12CCC2 CCC(C)CC(=O)C(=O)NC1CC2(C1)CC(C(N1CC(C)=CC(C)C1)=O)C2 C1(CC(=O)N(CCC(=O)NCCc2cscn2)CC#C)CCC2CC12 n1(CC(=O)NC2CC(F)(CNC(C34CC(F)(C3)C4)=O)C2)[nH]cc2c(=O)ncnc1-2 c1(CC(C)C)ccc(C(C)NCC2CCC(C(C)(C)C)CC2)cc1 N1(C(c2cccc(CCC)c2)=O)CC(OC)CC(NC(C2(CO)CC2(F)F)=O)C1 c1(CC)cccc(C(N2CCCC(NC(c3cncc(N(C)C)c3)=O)C2)=O)n1 N1(C(C2C(OCC)CCCC2)=O)CCN(C(=O)CN(C)C)C(CC)C1 c1(C(=O)NCCN(C(CC2C(OC)CC2)=O)CC2CC2)cnc2cc(C)ccn12 O=C(CN=c1cc[nH]cc1)N1CC2CC2(C(N2CCCC(O)(CO)C2)=O)C1 CC1(C)CCC(CO)N(C(=O)CSCc2ccccc2Br)C1 C(C)(C)(CC(=O)N(C(C)C(F)F)C)N(C(CC(C)C)=O)C C(=O)(C1CCCc2c[nH]nc21)NC(C)CCNC(=O)C=Cc1ccccc1F c1(C(C)NC(c2n[nH]cc2CNC(C2CC(C)(C)C2)=O)=O)nccc(O)n1 Cc1ccc2ncc(C(N3CC4(CC(NC(C5CCC(C)S5)=O)C4)C3)=O)n2c1 N1(C(CC(CNC(C2CC3(CCC3)C2)=O)O)=O)CC2CC1CC2CF c1(OC)cc(Br)c(Cl)cc1NC(c1cc(OC)ncc1NCc1ccc(Br)[nH]1)=O Cc1cc(CN2CCN(c3nccc(N4CCCC4)n3)C(C#N)C2)c(C)cc1O C(CCC(O)C(=O)N1CCC(N2CCC2)CC1)NC(C1(C)CCC(=O)N1)=O O=C1NC(Cc2ccc(Cl)cc2Cl)C(=O)N1CCSC1CCCC1 CC(C)(C)C(C(=O)N=C1C=C2C=CC(Cl)=CN12)n1cc(CC2(O)CCC2)nn1 Cc1cc(C(=O)NCCC(O)CNC(=O)CCN2CCCC2=O)cc2nc[nH]c12 C(=O)(C(F)(F)CC1CCCO1)N(C1CCN(C(=O)CSC2CC2)C1)C C(=O)(CCP(C)(C)=O)NC1(COC)CN(C(=O)CC2C(=O)N(C)N=C2C)C1 Cc1c(C(N2CC3(CCCC3NC(=O)C(CO)C(C)C)C2)=O)sc2cncn12 N1(C(C=CSC)=O)CCC2C(NC(=O)C(C)(O)C3CCC3)CC12 C1(COC)(NC(c2nccc(NC)n2)=O)CCCN(C(=O)COC(F)F)C1 C(CC(=O)NC1CCCCCC1)(C(C)CC)NC(CC(C(=C)C)OCC)=O c1(C(N2CCCC2CNC(=O)C(F)(F)C(O)C2CC2)=O)cccc(C#CCO)c1 C(=O)(C1=CCC(C)CC1)NCC1C2CN(C(c3c(Cl)ncc(C)c3)=O)CC21 c1(C(N(CCN(C(C=C(C)C2CC2)=O)C)C(C)C)=O)cnn(CC2CCC2)c1 c1(C(=O)NCC(CO)NC(C(F)=CCC)=O)cc2cc(OC)c(F)cc2[nH]1 C1(NC(C=C(C)C)=O)C2COCC1CC(NC(=O)CC1CCC1(C)C)C2 C1(C(N2C(CNC(C(CC)CC)=O)CC(C)CC2)=O)COc2cc(F)ccc2O1 C1(CCNC(c2cncc(F)c2)=O)CCCN(C(C2CCCC2C(F)F)=O)C1 c1(C(=O)NCC2CN(C(C3N(C)CCOC3)=O)CC2(C)C)ccc2sccc2c1 N1(C(C2CN(C)C(=O)CC2)=O)CCCC2(C1)CN(C(C1OCCC1(C)C)=O)C2 C1(C(N2CCC(F)(C(C)C)C2)=O)C(C)OCCN1C(C1CCCS1(=O)=O)=O C(=O)(CC1=CCN(C)CC1)N1C(C(=O)NC(C(=O)NCC)C)(C(C)C)CCC1 N1(C(CC2CC(C)N(C(c3ccn4ccccc34)=O)C2)=O)CCc2c[nH]nc2C1 C1(C(=O)NC2CCC2C(=O)OC)CCN(C(=O)CC(=O)N(C)C)CC1(C)C C=C(C)c1ccccc1NC(=O)CC1CN(C(c2nc(C)cnc2C)=O)CCO1 Cc1cc(C(=O)N(C2CN(C(c3cc(C#N)no3)=O)CC2(C)C)C)cc(Cl)c1 N(C1c2ccccc2CC1NC(C12CCCC1C2(F)F)=O)C(C(C(=O)OC)C)=O c1(N2CC(OCC)(CNC(c3cnn(C)c3CC(C)C)=O)C2)snc(C)c1C#N C(=O)(CC(C)(C)C)N(CC)CC1CCN(C(C2CCCN2CC(F)(F)F)=O)C1 Cc1cc(=O)oc(C)c1C(=O)NC(C)CCNC(C1CCCC2C1C2(F)F)=O c1(C(=O)NC2CC3CC(NC(=O)CC45CCCC4C5)C3C2)ccn2nnnc2c1 N1(C(C2C(C)CCC2)=O)CC2CCC1CN2Cc1csc(C2CC2)n1 CC(=O)CCCC(=O)N1CCN(C(c2nn(C)c(C)c2Br)=O)C2CC12 C1(NC(=O)CN2CCSCC2)CC2CCC1N(C(c1nc(Cl)cs1)=O)C2 N1(C(c2cccc(Oc3cnc(-c4ccccc4)s3)c2)=O)CCCCCC1CO N1(C(=O)Nc2cccc(CN(c3ccc(Cl)cc3F)C)c2)CCCC(F)(F)CC1 c1(C(N2C(Cn3cc(C(COC)O)nn3)C(C)(C)C2)=O)ccnc2c1ncn2C N1(C(c2c(OCC)ccs2)=O)CC(C)C(C)(CNC(=O)C(C)(CO)OC)C1 N1(C(Cc2ccc(OC)cn2)=O)CCN(C(C2CC23CC(O)C3)=O)C2(CCC2)C1 C1(NC(CSCC#C)=O)CCN(C(=O)C(C#N)C2CC2)C1CC c1(CCNC(c2nnnn2CC(F)F)CCOCC=C)ccnn1C c1(CCC)cc(=NC(=O)N2CCCC2C)[nH]o1 C1(C(=O)NC(c2ccco2)C)(CO)CCCCC1C.C1(NC(=O)CO)CCCNC1 C1(NC(c2c(CC)occ2)=O)CCN(C(c2cscc2C(F)F)=O)CC1F c1(CCC)[nH]nc2ccc(C(N3CC(NC(C4(SC)CC4)=O)CC(C)C3)=O)cc12 C(=O)(C(CC(F)F)NC(c1cc(CO)n(C)n1)=O)NC(CC)CO c1(C(N(c2nccc(Br)n2)C2CC(N)C2)=O)cnc2ccccc2n1 C12(CNC(C=CC(=O)OCC)=O)CC(CC)(CN1C(C1CCC(C#N)CC1)=O)C2 c1(OC)cc(C(=O)NC2CCC2NC(c2ccc(CS(C)(=O)=O)o2)=O)cc(C)n1 C1(NC(C(COC)C)=O)CN(C(c2nnc(O)cc2O)=O)CC12CC2 C(C)(C)(CC(F)C(=O)N1CCCC1C1(C)CC1)NC(Cc1c(C)n(C)cn1)=O C=CC(C)C(C(=O)NS(=O)(=O)Cc1ccc(F)c(F)c1)c1ccccc1 C1(C(N2CC3C(CNC(CC4CC(=C)C4)=O)(C3)C2)=O)CCN(OC)CC1 N1(C(CCCc2ccc(C)s2)=O)CC(NC(=O)C(C2CC2)N(C)C)CC1(C)C c1(C(C(=O)NCCN(C2CCCC2)C(CC2CC(NC)C2)=O)C)c(C)noc1C c1(C(=O)NC2C(C)CC2)ccoc1CNC(C1CC(=O)C1)=O c1(OC)ncc(C=CC(=O)NC2CCN(C(C3C(C)CC3C)=O)CC2)cn1 N1(CC)CC(C(=O)NC2CC(NC(c3ccncc3Br)=O)CC2O)CC1=O c1(C(N2CC(C(=O)NCC3(O)CC(C)(C)C3)C(F)C2)=O)ccc2[nH]ccc2c1 Cc1[nH]c(=N)ccc1C=CC(=O)NC(C)CNC(=O)C=CCOc1ccccc1 c1(C(N2CC3C(NC(C(CC(C)C)C)=O)(C3)C2)=O)cnn2c1OCCCC2 c1(C(N2CCC(N(C(=O)Cc3cocn3)CCO)C2)C)cccc(Cl)c1 C1(C(N2CCC(NC(c3c(C)cns3)=O)C2C)=O)CCC(C#N)CC1 N1(CC(C2CCCCO2)(C)C)C(=O)CCN(CC2CCCCC2)C1=O C(CC(F)(F)C(=O)N1CCC(CC2CCC2)C1)n1cc(C2CCC(C)C2)nn1 c1(C(C)=O)ccc(NC2CN(CC(F)(F)F)C2)nc1.c12ccc(nc1)[nH]c2=O C1(CC)CCC(C)CN1C(=O)CCN(C(=O)CCC1CC1(F)F)CC N1(C(C2C(C#C)C2)=O)CCCC2(CCCN2C(c2ccnc3ccnn23)=O)C1 c1(C(N2C(CC)CC(C)C2)C(=O)NC)ccc(C(F)(F)F)cc1Cl C(=O)(C(C)CC(=O)OC)NCC1CCCN(C(Cc2ccc(OCC)cc2)=O)C1 c1(C2(C(=O)NC(C(C)C)CNC(=O)CC3(CO)CC3)CC2)cccc(F)c1F c1(C(=O)NCCC(C)(C)NC(C2CC3C=CC2O3)=O)nccc2c1CNC2=O C1(C(=O)NCCC(=O)NC)CN(C(c2cc(C)nc(O)n2)=O)CC1(C)C C1(NC(Cc2c(C)ncs2)=O)(CNC(=O)C(C)(C)O)CC2CCC1CC2 Cn1c(O)nc2cccc(C(=O)NC3CC(NC(=O)C(C)(C)C(F)(F)F)C3)c12 Cc1nc2sccn2c1C(=O)NCCC1(NC(C2CC3(C2)CC(O)C3)=O)CCC1 Cc1cc(=O)c(C(=O)NCCCN(CCCNC(=O)Cc2cccs2)C)cn1C Cc1cnc(CCNC(=O)CC(C)CNC(c2cnn(C3CC3)c2)=O)nc1 C(=O)(C#CC1CCCOC1)N1C(CN(C)C(c2ccc(C(N)=O)o2)=O)CCCC1 c1(OCC)cc(CNc2cc(F)cc(F)c2O)cc(Br)c1OCC c1(C(=O)NC2CCC(C(=O)NCC3CCO3)C2)ccc(C(F)(F)F)c(Br)c1 Cc1cnc(C=CC(N2CC=CC2CNC(=O)CC2CCC(F)(F)C2)=O)[nH]1 c1(N2CCCC(CC=C)(NC(=O)C(F)C(F)(F)F)C2)nc2ccc(C)nc2s1 CC1CC(NC(=O)CC2CCCC(C)C2)CCN1CCCC1CCS(=O)(=O)CC1 OC1CCCCC1CNC(c1nnnn1CCC1CC1)c1ccno1 C1(C(N2CCC(NC(CCCCC)=O)C2C)=O)CCCCC1C1CC1 C1(C(=O)OC)(CNC(c2cc(C(CC)CC)no2)=O)CCCS1(=O)=O c1(C(C(=O)NC(C)(C)C)N(C)CC2CCCN(C)C2)cnc(N(C)C)nc1 c1(C(=O)NCC23N(C(Cc4cn(CC)nn4)=O)CC(C2)C3)ccc(F)cc1Cl c1(C(N2CCN(CC(C)NC(C(C)OC)=O)CC2)=O)ccc2c(c1)C=CCC2 C(=O)(C(C)(F)C(C)(C)F)NCc1cn(CCNC(CN(C)CC)=O)nn1 CC1CCCc2nc(C(N3CCC(C)(CNC(C4(CO)CC4)=O)C3)=O)cn21 c1(CC)c(NC(C2CSCCN2C(C23COCC2C3)=O)=O)cnn1CC N1(C(C(C#C)(C)C)=O)CC2CCC1C(NC(c1ccc(Cl)c(C(F)(F)F)c1)=O)C2 C1(C(=O)NC(C2CCOC2)C#C)CCCCN(C(c2c[nH]cc2CC)=O)C1 C1(COCC)CC1(C)C(=O)CCN(C(=O)COC(C)=O)C.C(C)(C)(C)O c1(CC)ccc(CC(=O)NC2CCCC2NC(=O)C(C)(COC)OC)cc1F Cn1cc(C(N2CCC(CNC(=O)CCc3cnn[nH]3)CC2)=O)c(C2CCC2)n1 c1(CC(=O)NC(C(C)C)(C)CNC(=O)Cc2ccc(O)nc2)cccc(Cl)c1F C1(C(=O)OC(C)(C)C)CCCC2(CC2)C1.N12CCCC1C1(CC1)C(=O)NCC2=O N1(C(c2occ(C)c2)=O)CCSCC1C(=O)NCC1(CC2CC2)CCC1 Cc1cc(NC2CC(NC(c3cc(O)nn3C)=O)C23CCC3)ccc1[N+](=O)[O-] c1(N(C2CN(C(c3ccc(C)c(C)c3)=O)C2)C)ncnc2sccc12 CC1C(C)N(C(=O)CCOC2CC2)CCN1C(=O)CCCF C1(C(=O)NCCCOC(C)C)CN(C)CCN1C(=O)Cn1cccn1 c1(NCc2cccc(OC(C)C)c2)cc(N2CCC(F)(CF)C2)nc(C(C)C)n1 C1(O)(C(=O)NCC2(CNC(C(C)Cn3cccn3)=O)CCCC2)CCCCCC1 CCC(C)(C(=O)O)N(C)C(c1ccc(-n2cncn2)cc1)=O C1(NC(COC)Cc2ccccc2)CCCN(S(=O)(=O)Cc2ccccc2)C1 c1(C(N(C)CC2CCCN(C(C3(C)CC(C#N)C3)=O)C2)=O)cc2c[nH]cnc-2n1 C1(CC)CN(C(C2CN(Cc3cccc(OC(C)C)c3)CCO2)=O)CCO1 c1(C(N2CCC(CCNC(=O)C(F)OC(F)(F)F)C2)=O)cc2ccccc2cn1 C1(NC(CCNC(N)=O)=O)CC12CCN(C(C1CC(=O)N(C(=O)O)C1)=O)CC2 CC1(C(=O)NCC2CC(F)(CNC(c3csc(CO)n3)=O)C2)CC(F)(F)C1 c1(CCNC(c2n(CCCC)nnn2)CC2CCCCO2)cc(Br)ccc1F c1(OC(c2c(OC)cc(NCC(N)=O)cc2)=O)ccc(Br)c2ccccc12 C(C)(C(=O)N(C(C)C(=O)NC(COCC)C(C)C)C)OCC#C c1(CNC(c2c(NC(c3cc(Cl)ccc3Cl)=O)c[nH]n2)=O)cccc([N+](=O)[O-])c1 C(=O)(CCCC(=O)N1CCCC(NC(=O)Cc2[nH]cnc2C)C1C)NCCC Cc1cc(CN(C)C(c2cn(CCNC(=O)Cn3ccnc3)nn2)=O)no1 C(=O)(C(CCF)NC(c1n[nH]c(O)n1)=O)NCCNC(N)=O C1(O)(C(C(=O)NC(C)C(C)n2cccn2)NC(Cc2nc(C)sc2)=O)CCCCC1 N1(C(C(C=C)O)=O)CCOC2CN(C(c3ccn4cncc4c3)=O)CC12 C1(OC)C(OC)CN(C(=O)CN(C)S(N)(=O)=O)C1CNC(C1CCCCO1)=O C(C(O)CCCS(N)(=O)=O)N(C1CCCC(C)C1)CC Cc1ncnc(C(=O)NCC2CC2CNC(C2(c3ccccc3)CCC2)=O)c1C C(C)(C(=O)NNc1cccc2c1OC(F)(F)O2)(C(C)C)OC C(=O)(CC(O)(C(F)(F)F)c1ccccc1)NCC(CC(C)C)NC(C1CC1F)=O C1(NC(C2(C=C)CC2)=O)CC2(CCCCN2C(c2oc(C3CC3)nc2C)=O)C1 c1(N(C)CC2CC2CO)nc(Cc2ccccc2F)c2c(F)cccc2n1 C1(C2CN(C(=O)CNS(=O)(=O)C(F)(F)F)C2)(CC)CC1.CC1CC(C(=O)NC)C(=O)O1 c1(C(N2CC3C(CN(C(=O)CCC4CC4)C)C3C2)=O)ccsc1S(C)(=O)=O c1(NCC2C(C(=O)NCC34CC(C(F)F)(CO3)C4)C2)ccc(F)cc1F NS(=O)(=O)CCNC(C1CCN(C(C2(C3CC3)CC2)=O)C1)=O c1(C(N2CCCC(NS(=O)(=O)CC3CCC3)C2)C)ccc(Cl)cc1 N1(C(C2(C)CCCCC2)=O)CC2CC(NC(C3CCCC3C3CC3)=O)CC1C2 C#CCC(C)(CNC(c1cc(CNC(=O)CC(C=C)CC)nn1C)=O)CO CC1CN(C(c2sccc2F)=O)CCC1N(C(=O)Cc1cncn1C1CC1)C CC(c1cccs1)=CC(=O)NC1CCCC1CNC(c1ccc(C(F)F)s1)=O C12(C(=O)NC(C(OC)OC)C)CCC(NC(=O)NCC3(C)CCOC3)(CC1)C2 Cc1nn(C2CC2)c(Cl)c1CNC(N1CCC(C)(CN)C1)=O n1(CC)ncc(C(=O)NC23CC(CNC(=O)CC4COC(=O)C4)(C2)C3)n1 c1(C(N2CCCC(NC(c3nnc(C)s3)=O)C2C)=O)cccn2c(C)cnc12 C1(CNC(C(C)S(N)(=O)=O)=O)CC2(CO1)CN(C(=O)COC(F)(F)F)C2 C=CCC(C(=O)N1CCC(CC=C)(NC(=O)COC)CC1)C(C)C C1(NC(c2cn(CC)nc2)=O)CC(NC(c2ccc(C(C)(C)C)cn2)=O)CC1O N1(C(c2ccc(C)c(Cl)c2)=O)CC(NC(=O)C(O)Cc2cnc[nH]2)CCC(O)C1 c1(C(=O)NC(O)C2CN2)cc(C(N)=O)ccc1CC1(C(C)C(c2ccc(CO)nc2)=O)CC1 N1(CC)CC(C(N2CCC(OCCNC(=O)C=CC(C)C)C2)=O)CCC1=O N1(C(C2(COC)CC2)=O)CCC2CC(C1)CN(C(C1CN3CCN1C(C)C3)=O)C2 C1(C)(OCC)CCN(C(=O)C(CC)N(C(=O)C(F)F)C)CC1 CC(C)C1=CCC(C(N2CCCC(N(C)C(C3CC(F)(F)C3)=O)CC2)=O)CC1 CCC(CNC(=O)C(F)CNC(=O)OC(C)(C)C)C(C)C c1(OC(C(N2CC(O)(CNC(C(CSC)O)=O)C2)=O)C)cccc(CO)c1 CC(C)C(C)(O)C(=O)N(CC(C)NC(C1CC1C(N)=O)=O)C c1(OCCC)ccc(Cl)cc1C(=O)NCC1(C)CCC(NC(c2cn[nH]c2)=O)C1 C1(NC(CNC(=O)OCC)=O)CS(=O)(=O)CC1NC(=O)Cn1ncnn1 C(C)(CCC(=O)NC1C2CCN(C(c3cccnc3O)=O)C12)OCC N1(C(CSCCSC(C)C(F)(F)F)=O)CCC(N2CCOCC2)CC1 CC1CC(C)(C)CC1NCc1ncnn1C1CC1 C(=O)(C(CO)NC(=O)OC(C)(C)C)N(CC(C)N(C(C=C(C)C(C)C)=O)C)C Cn1cc(S(N)(=O)=O)cc1C(N1CC(NC(c2ccc(N)cc2O)=O)CC1C)=O C1(C2CC2)(NC(CCC(=C)Cl)=O)CCN(C(c2cnc(OC(C)C)cn2)=O)C1 N1(C(c2c(NSCC)cccc2)=O)CCNC(C)C1C CN1CC2(CN(C(C3CCOC3(C)C)=O)C2)OC1=O C(=O)(C(F)(CC)C(=O)OC)NCC(C)(C(C)C)NC(c1cc(CC)oc1C)=O C(CC(C(N)=O)NC(=O)C(F)C1CC(NC(=O)C(=O)N(C)C)C1)OC C(CCCCC(=O)N1CCC(C)(CNC(c2[nH]cnc2C)=O)C1)=CC CCC(C)C(C(=O)NC)NC(=O)CCCNC(=O)CC(C)COC N1(CCC(=O)NCC)CCCC(C(=O)N(C)CCc2ccc(Cl)cc2)CC1 C1(C2CC2)(NC(C2OCCN(C(c3ccc(N)cn3)=O)C2)=O)CCOC1 CC1(C)CCC(=CC(=O)NCC2CN(C(c3cc(C4(C)CC4)n[nH]3)=O)C2)CC1 c1(C(=O)NC(CC(C)C)CNC(=O)C(C)(C)Br)cccc2ccn(C)c12 C1(CC)CN(C(c2cc(CC(C)C)on2)=O)CCC(C)O1 c1(NC(C2CCN(C(C(C)OC)=O)CC2)C)cccc(C)c1C C1(CC(=O)NCC(CC)NC(c2ccc(C(C)C)o2)=O)CCCC2(CCC2)O1 Cc1cc(=O)ccn1CC(=O)NC1CC1NC(C1C2CCC1(c1cscn1)C2)=O c1(OCCC(N2CCC(C(=O)NCCCC)C2)=O)ccc(Cl)c(C)c1 N1(C(C2(C)COC2)=O)CCn2ncc(CNC(c3nocc3Br)=O)c2C1 c1(C(C)OC)cn(C2COCC2NC(c2sccc2C(C)=O)=O)nn1 C1(C)(C(=O)NCC2C(NC(C(c3c(C)noc3C)(C)C)=O)CC2)CCCS1(=O)=O c1(C(N2CC(C(C(=O)NCCCC(=O)OCC)O)C2)=O)ccccc1F C1(CC(N2CCC(c3cnn[nH]3)C2)=O)C2CCC(C2)N1C(C1CCC(O)CC1)=O C1(CC=C)(NC(=O)COCC(F)(F)F)CCCN(C(C2CC3(CSC3)C2)=O)C1 C1(CC(=O)NCC2CCN(C(C3CC(C)SCC3)=O)CC2)CS(=O)(=O)CCN1C C(=O)(C(F)(F)CCn1cccn1)NC1CCC(NC(C2CC(C)C2)=O)CC1 Cn1cc(N)c(C(=O)NC2CN(C(=O)COc3cccc(Cl)c3)CC2C(F)F)n1 Cc1nc2cc(C(N3CC4CC(C3)C4NC(c3ncccn3)=O)=O)ccc2o1 N1(C(c2c(NC)nccc2)=O)CCC(C(=O)NC2CCCC2C2CC2)C(C)(C)C1 c1(SC)nc(=NCC2CC(NC(C34CC(CN3C3CCCCC3)C4)=O)C2)s[nH]1 c1(-c2n(CCC=C)c(N3CCS(=O)(=O)CC3)nn2)sc2ccccc2c1Br Cn1nc(C(N2CC3CCN(C(=O)C(C)(C)C)CCC3C2)=O)c2cc(F)ccc12 c1(C(N2C(CCNC(C(C)(C)OC)=O)COCC2)=O)[nH]c(=N)ccc1C C1(C(=O)NCC(CN(C(=O)Cc2ccon2)C)(C)C)CCC2(CC1)CC2(F)F C1(NC(CC(C)OC)=O)CC(OC)CN(C(c2nn(C)cc2C)=O)C1 C(=O)(CCCC(=O)N(C)C)NC1CC(C=C)C1.C12CC(C(O)C1)C(=O)N2 C1(NC(c2c(NC(C)=O)cncc2)=O)CN(C(=O)CCC(N)=O)C2(CCOC2)C1 c1(C(N(CC(C)NC(=O)C(O)CC2CCCC2)C)=O)coc(C(C)(C)C)n1 N1(C(C(CC)C(C)O)=O)CCN(C(c2cccc(C(F)(F)F)c2N)=O)C2(CC2)C1 c1(C(N(C2CN(C(C3CC3F)=O)CC2(C)C)C)=O)cc(Cl)ccc1Br N1(C(C(N2CC(OCCNC(C3CC(CCC)C3)=O)C2)=O)C)CCCCCC1 Cc1ncccc1CN1CCN(C(c2cc(C3CCNCC3)on2)=O)CC1 C1(NC(C(COC)NC(c2ncc(F)cc2F)=O)=O)CCC(=O)N(C)C1 c1(C(=O)NCC2CCN(C(c3cnc(C(C)=O)s3)=O)C2)cccc2c1SCCC2 C1(C(=O)NCC(C)(C)n2ccnc2)CN(C(c2cc[nH]c2)=O)CC1C1CC1 c1(C(N(CC(=O)Nc2c(CC)noc2)CC2CC2)=O)nn(C)cc1C N#Cc1cccc(N(C(=O)CNC(=O)CCC(N)=O)CC=Cc2ccco2)c1 c1(C(=O)NC2CCN(C(C(CC)SC)=O)C2)c(C)c2cnccn2c1C N1(C(C2C(OC(C)=O)C2)=O)CCCC(C)(NCc2cnn(-c3ccccc3)c2)C1 C1(C)(CNC(C2CC(C)C2)=O)CCCN(C(=O)CCOC2CC2)C1 S(=O)(=O)(c1cnc(NCC(c2nncn2C)C)c(Cl)c1)NC(CCSC)COC Cc1c(CC(=O)N(C)CC2CN(C(=O)C=CC3CCOCC3)C2)cnn1C C1(C(N(C(CNC(CC(=O)NCC)=O)C)CC)=O)CCOC(=O)CC1 c1(CCC)nnc(S)n1CC(N1CCCC(c2ccc(OC(C)C)cc2)C1)=O S(=O)(=O)(c1ccc(Cl)c(NC(C2(C)CCC2)=O)c1)NC(C)C CC1CC(NC(=O)C#CC2CC2)CN(C(c2nc(C3CC3)ncc2Br)=O)C1 S(=O)(=O)(c1ccc(Cl)cc1F)N1C2CN(C(C(CCC)C)=O)CC21 c1(CNC(C2(C)CC(C)C2)=O)ccccc1CNC(=O)Cc1cocn1 C(=O)(CCCCCNC(C1CCOCC1)=O)N1C(C(N)=O)CCC1 C(c1ccc(S)cc1)=CCC(=O)NC1C(CNC(=O)C=C)C1.n1(C2CC2)nccn1 C1(NC(c2cc(C)nc(O)c2)=O)CC2CCCC(C1)N2C(=O)C(C)O c1(NC(C2C3CN(C(C4N(C)CCCC4)=O)CC32)=O)cc(Br)cc([N+](=O)[O-])c1 c1(C(=O)NC(C)CN(C)C)n[nH]c2c1CCN(Cc1cc(F)c(F)cc1O)C2 C(C(C)N(C(=O)COCC(F)F)C)(OC)OC c1(C(=O)OC)cc(C(=O)NC(C)(CNC(c2ncc[nH]c2=O)=O)CO)ccc1C c1(-c2cn(C3CC(NC(c4n(CC=C)ccc4)=O)C3)nn2)cccc(N)n1 N1(C(c2cc(CC)nn2C)=O)CCC12CN(C(C1(C)CCCC1)=O)C2 c1(C(=O)NCC2(C(C)NC(c3cscc3C(F)F)=O)CC2)nnc(O)cc1O CN1CC(C)(C(=O)NCC2(F)CCN(C(C3CC3C(F)F)=O)CC2)CCC1=O c1(COC(c2c(C(C)=O)n(C)nc2)=O)ccc(Oc2cccc(F)c2)c(Cl)c1 C#Cc1cccc(C(=O)N(C(C)CNC(c2cc(F)cc(C#C)c2)=O)C)c1Cl c1(C(=O)NCC(C)C(=O)NCC23CCCN(CC2)C3)cccc(F)c1N N1(CC#CCC)CCCC(COC(=O)CC2CCCCC2)C1 CC1OCCOC1C(=O)N(CCCCNC(C1(n2cccn2)CCOCC1)=O)C Cc1nc(CC(=O)N(C)CCNC(c2coc(Cl)c2)=O)co1 c1(NC(C2N(Cc3c(C)cc(Cl)c(Cl)c3)CC2)=O)c(C#N)ccc(F)c1F c1(CC(=O)NCCCCC(C)NC(COCCC#C)=O)cccc(C)c1Br C(CC(C(=O)N(C1CCCC1)C)NC(=O)CCc1nc[nH]n1)=CC c1(C(=O)NC2CN(C(C=COCC)=O)CC2C)ncc(Br)cc1OC C1(NC(C(C)Cn2ccnc2)=O)CCN(C(c2ccc(N)cc2F)=O)C12CC2 c1(OC)ccc2[nH]nc(C(=O)NCC3CCN3C(C3C(Cl)(Cl)C34CC4)=O)c2c1 C(=O)(C(C)C(O)C(C)C)N1C(C(C)NC(c2cc(OC)c(C)cc2)=O)CCC1 N1(C(C2CC(C)(C)N(C(=O)CCCC#N)C2)=O)CCOC2COCC2C1 c1(N2C3CC(CNC(c4n(CCC)ccc4)=O)(OC3)C2)nc(C)nc(C)c1F c1(SC)cncc(C(N2CC(CNC(c3ocnc3C(F)(F)F)=O)C(C)C2)=O)c1 CC(C)CC(F)(F)C(=O)NCCN(C(=O)CN1CCCOC1=O)C1CC1 C1(C(N2CC(=C(CNC(C(C)NC(CC)=O)=O)F)C2)=O)CC(C(=O)OC)=NO1 N1(C(CCCCOCCC=C)=O)CC(CNC(c2ccc(SC)o2)=O)C2(CC2)C1 C1(CC(C)NCCn2cc(-c3ccccn3)nn2)CCN(C(C(C)(C)C)=O)CC1 C#Cc1ccc(C(N2CC(OC)C(C(=O)NC3CC(CC(N)=O)C3)C2)=O)cn1 C1(OC)CN(C(c2cnn(CCO)c2)=O)CC1NC(=O)CCN1CCCCC1C C(C(=O)NCC(O)CCNC(C1(CC(F)F)CCC1)=O)(C(C)C)SCC C1(COC)(NC(C2CCCC3(CC3)C2)=O)CCN(C(=O)CCC(C)OC)CC1 c1(C(=O)OC)ccc(C)c(C(=O)NCC(C)CNC(C2CC3(C2)CC(C)C3)=O)c1 N1(C(c2c(SCC)nccn2)=O)CCC(NC(C2(C(=O)N(C)C)CC2)=O)C(C)C1 C(=O)(CC(C)(C)C(=O)NC(C)CCCNC(C12CCCC1C2(F)F)=O)OC N1(C(Cn2c(C)csc2=O)=O)CCN(C(=O)COc2ccsn2)C(C)C1 n1(CC)cc(CC(=O)N(CCCNC(=O)C(C)c2ccco2)CCO)nn1 c1(C(N(CCOC)CCNC(C2CNC(=O)C2)=O)=O)cc(F)cc([N+](=O)[O-])c1N Cc1ccc2cccc(-n3cc(Cc4cncc(O)c4)nn3)c2n1 CC1CN(C(=O)C=CCF)CCC1NC(=O)CCc1ccc(C(N)=O)cc1 c1(CC(=O)OCC(=O)NCCCOCC)ccc2ncnn2c1 C(CN=C(NCCC1CC1)NCc1cccc(Cl)c1)c1c(C)noc1C CC(C)CCCC(C)C(=O)NCC1(C)CCC(NC(=O)CCc2nc[nH]n2)C1 C(=O)(CCCN=c1nccc[nH]1)NCC1(F)CC(CNC(C2CC(OC)C2)=O)C1 c1(C(=O)NC(C2(O)CCN(C(=O)C=CC3CCOC3)C2)C)cc2c[nH]nc2s1 C1(C(=O)NC(c2ccccc2)C#C)C2CC1N(C(C1CCCSC1)=O)C2 N1(C(c2cc(C)c(O)nn2)=O)CCC(NC(=O)C(C)OC2CCOC2)C12CCC2 C1(C(=O)NCC(CCC)NC(=O)Cc2ccnc(O)c2)CCC(O)CN1C CC(C)CC(C(=O)NCC1CC(CF)C1)NC(c1cccn(C)c1=O)=O C1(C(=O)NC2C=CCN(C(c3cc[nH]c3)=O)C2)CCCCCS1(=O)=O c1(C(=O)NCCC2CCN(C(C3CCCN3C3CC3)=O)C2)cc2cccn2cn1 C(C(=O)N1CC(CC(C)(C)CNC(c2nncs2)=O)C1)(C(C)C)OC c1(SCCNC(C2CC(NC(c3sccc3Br)=O)C2)=O)cccc(F)c1 C#CCCCC(C)C(=O)N1CCN(C)CC1C(=O)N(C)Cc1ccc(O)cc1 c1(C(N(CC(C)CNC(=O)C(C)N(C2CCCCC2)C)C)=O)nn[nH]c1Cl C1(C(N(C)CC2CCCCCC2)=O)CC12CCN(Cc1ccncc1F)CC2 C1(C(=O)NCC2CCNC(=O)C2)CCOCCN1C(C1CC2CC(=O)C1C2)=O O=C1COC(CNC(C2CCC2NC(c2cn(C3CC3)nn2)=O)=O)CN1 C(=O)(C1=NOC(C)(C)C1)NC(C)C(C)(C)C(=O)NCC1CC2(CCO1)CC2 Cn1cnc(C(=O)NCCCNC(C2CC(O)(CCC(C)(C)C)C2)=O)c1 C1(C(C)C(=O)N(CCCNC(=O)Cn2cccn2)C)CCOCC1 C#Cc1ccc(C(=O)NCC2CN(C(c3oc(CC)nc3C)=O)CCO2)c(C)c1 N1(C(c2cc(CC)[nH]n2)=O)CCC(C(N2CCC3(CC3)C2)=O)(CF)C1 C1(C(CNC(C2C(C)C2C)=O)(C)C)CCN(C(C2CCCC2)=O)CC1 C(C(C)C)(C(O)C(=O)NC1(CN(C)C(C2CC(F)C(=O)N2)=O)CC1)OC CCC(CCC(=O)NCCC1CC(F)C1)NC(=O)C(O)C1CCC1 CC1C(NC(c2scnc2C(F)F)=O)CCCN1C(C1CC12CCOC2)=O c1(OC)cc(C(=O)NC(C)(C)CCN(C)C(C2OCCN(C)C2=O)=O)cnc1O C=CC(CC)C(=O)NC1CC(NC(=O)CSc2ccncc2)CC1O c1(C(=O)NC(CNC(C(CSC)(C)C)=O)C(C)C(C)C)cncc([N+](=O)[O-])c1 C(C)(CC(C)C)(C(N)=O)NC(C(=Cc1cn[nH]c1)C)=O CCCN=C(NCC(C)(F)C(C)(C)F)NC1CC(C(=O)OC)c2ccccc21 CC(O)C(C(=O)N1CC(CO)(NC(=O)C=CC2CCC2)C1)NC(=O)C1CC1 C1(OC)CCCN(C(c2cccc(-c3ccccc3)c2)C(=O)NC(C)C)CC1 C1(CCC)CN(C(=O)CC2CC3(CC3)CO2)CCN1C(c1cc(C(C)C)[nH]n1)=O c1(C(=O)NC23CC(NC(C4N(C(C)=O)CCCC4)=O)(C2)C3)cnc2ccnn2c1 C(C)(CCC(=O)NCC(C)NC(=O)C(C1CCCCCC1)F)OC c1(C(=O)NCCCC2N(C(COCC(=O)NC)=O)CCC2)nc2c(s1)CCCC2 Cc1cc(NC(=O)COC2CCN(C(C3CCCN3C)=O)C2)cc(F)c1 Cc1ncnc(C)c1C(N1CCN(CC2(O)CN(C(c3ccco3)=O)C2)CC1)=O C(=O)(C1OCCn2ccnc21)N1CC(C)CN(CC(F)(F)F)CC1 C=C(C)C(C)(C)C(=O)NCC1CCN1C(=O)C=Cc1cncc(F)c1 c1(C(CC)(C)C)cn(CCCNC(C2CC2C(c2ccccc2)=O)=O)nn1 c1(C(N2CC(F)(CNC(CCCOCCOCCOC)=O)C2)=O)cc(N)cc(O)n1 N1(C(c2c(CC)ccc(N)c2)=O)CCC(C2CC2)(NC(C2(CN(C)C)CC2)=O)C1 C1(C(n2c(-c3cn(C(C)C)nc3)ncc2)=O)CCC(O)CN1C C1(OC)CN(C(=O)CCN2CCOCC2)CCC1NC(=O)CCC(C)(C)F n1(CC)ncc(C(=O)NCCC2(O)CCN(C(c3ccnc(SC)c3)=O)C2)c1Cl C(C1=NOC2(CCC2)C1)NC(C(C1CCCO1)NC(C1CN(C)CC(C)O1)=O)=O CC1(C(=O)NCCCN(C(=O)C(N)=O)CCO)CCNC1=O c1(C(=O)NC(C2N(C(C(C(=O)OC)C)=O)CCC2)C)cc2n(n1)CCNS2(=O)=O C=CCC(C(=O)NOCC1CCOC1)NC(=O)C(C)COCC N1(C(c2cn(C)nc2)=O)CCC(C2(NC(c3nc(O)[nH]c(=O)n3)=O)CC2)C1 C1(Cl)(C(N2CCC(CN(C(Cc3nnc(C)o3)=O)C)C2)=O)CC12CCC2 C1(C(N(C)Cc2n(C(C)C)ncc2)=O)CC12CCC2=O c1(CC)c(OC)cccc1C(=O)NC1CN(C(C2CC3C=CC2C3)=O)C(C)(C)C1 N#Cc1sccc1C(N1CCC(CCNC(=O)C(C2CCOCC2)F)CC1)=O O=C(C#CC1CCCOC1)NC1CCN(C(c2cnc3n2CCOC3)=O)CC1F C1(NC(C2(C)CC2(Cl)Cl)=O)CC2(C1)CC(NC(C1COCCC1(F)F)=O)C2 Nc1c(C(=O)NC2(CO)CCN(C(=O)CC3CC34CC4)C2)ccnc1Cl N1(C(CC2(NC(C)=O)CC2)=O)CCN(C(C2CCCN2N=O)=O)C2(CCC2)C1 c1(C(N(C2CCCN(C(CNC(C)=O)=O)C2)C)=O)ccc(Br)c(Cl)c1 C1(C(=O)NC2(CNC(c3nccnc3N)=O)CC(OC)C2)CCC2C(C1)C2(F)F S(=O)(=O)(C1(C(c2nnnn2CCOC)NCc2[nH]cnc2C)CC1)NC c1(C(N2CCOC(c3ccccc3C(F)(F)F)C2)=O)ncccc1Cl C(CCC(O)C(=O)N1CCC(CC2CCC2)C1)NC(CCC(C)OCC)=O CCC(CC(=O)N(C(C)CNC(c1cc(C)n(C(C)C)n1)=O)C)C(F)F N1(C(C=NOC)=O)CC(C)OC2(CCN(C(=O)C(C)CS(C)(=O)=O)C2)C1 C1(C(=O)NCC(C(=O)NC2(C(=O)NC(C)C)CC2)CC2CC2)CCCN(C)C1=O C#CCC(C(=O)N(C)CC)NC(=O)C(C)C=C N1(C(CNC(=O)OC)=O)CCN(C(=O)Cc2cccc(C(=O)OC)c2)CC(O)C1 C1(COC)(CNC(=O)CC(C)NC(=O)CNC(=O)OC(C)(C)C)CN(C(C)=O)C1 n1(CC(N2CCCOCC2)=O)ccc(=NCc2c(Cl)cc(Cl)cc2Cl)nc1O CCCCCC(C)(C)C(=O)NC1CC1CNC(c1cnn2ccc(C)cc12)=O Cc1cc(C(=O)NC2(CN3CCN(C(=O)C4=CC(C)CC4)CC3)CC2)ccc1Cl n1(C(C)C(N2CCCN(C(C3CC34CC4)=O)CC2)=O)cnc2ccccc12 N1(C(C(C)=C2CCCC2)=O)CCN(C(=O)CC2CCCCC2)CC1CC(F)F C(=O)(C#CC(C)C)NCCOCCCNC(C(C=C)O)=O c1(C(=O)OC(C(=O)NCC)Cc2ccc(F)cc2)cc2ccc(O)cc2[nH]1 c1(C(=O)NCCNC(Cc2cccc(C)c2Cl)=O)cc2cccnc2[nH]1 C(=O)(C(C)CS(C)(=O)=O)N1CCC(C)(CNC(c2cncc(C#C)c2)=O)C1 C1(C)(CNC(Cc2c(C)occ2)=O)CCC(NC(c2coc(O)n2)=O)CC1 c1(SC)ccc(O)c(C(=O)NC2CCCCC2N(C(=O)C(C)P(C)(C)=O)C)c1 C12(C(=O)NC(CC(C)C)CNC(=O)CSc3n[nH]c(=N)s3)CC(C1)S(=O)(=O)C2 c1(C(=O)NC2(C)CC(NC(c3ccsc3Cl)=O)C2)coc2c1C(O)CCC2 N1(C(c2c(OC)scc2)=O)CC2(CNC(=O)CCCC3CCC3)CCC1CC2 C1(CNC(C(C2CCC2)OC)=O)CCN(C(=O)C(=Cc2cccnc2)F)CC1C C(C(N=c1[nH]c(Cl)ncc1C(N)=O)C(C)C)NC(COCc1cc(C)on1)=O N1(C(c2cc(C)c(C)s2)=O)CCC(C)CC1C(=O)NC1CN(c2ncco2)C1 C1(C(=O)NC2C3CN(C(CC(COC)(C)C)=O)C2CC3)CSc2ccccc2O1 CC(CC(=O)Nc1cnn(CC2CC2)c1)C(F)(F)C(F)(F)F Cn1cnc2nc(=NCCC3CCC(NC(c4cc5n(n4)CCC5)=O)C3)[nH]cc12 C1(CNC(C(CC)OCC)=O)CCC12CCN(C(C1(SC)CCC1)=O)CC2 Cc1cccnc1CCC(=O)NCC1COCCO1 C(=O)(CC(C(C)C)NC(c1ccc(C)cc1C)=O)N(C(CC)C)C N1(C(C(CC)N(C)C)=O)CCCC(CO)(NC(=O)COc2cccc(Cl)c2)C1 Cn1cnc2nc(N3CCCCC(CNC(C4CC(N(C)C)C4)=O)C3)ncc12 C1(C2CCC2)(C(=O)NC(CC(C)NC(c2n(COC)ncc2)=O)C)CCC1 CC1(C)CC(NC(=O)CC2CC3(CCC3)C2)CN(C(c2cnc(N)c(Cl)c2)=O)C1 Cc1cn2c(n1)CCC(C(=O)NCC1(CNC(c3cn4c(n3)CCC4)=O)CC1)C2 N1(C(c2nc(C)n(C)c2)=O)CCC(O)C(N(C(=O)CC2CC(F)C2)C)C1 C1(C2CCOCC2)(CNC(C(CSC)C)=O)CCN(C(=O)CCCN(C)C)C1 C(=O)(C1CCc2cccnc21)NCC1(C)C(C)CN(C(c2c(C)c[nH]n2)=O)C1 CS(C)(=O)=NC(=O)C(=O)N1CCCCC1C1(NC(c2cc3cccnc3o2)=O)CC1 N1(C(C2CCC3(CC3)C2)=O)CCN(C(C2CC(C3CC3)=NO2)=O)C2(CC2)C1 c1(C(=O)NCCN(C(c2ccc(C#C)cc2)=O)C)cc2cc(OC)c(F)cc2[nH]1 c1(CC)ncsc1C(=O)NCC1CC(NC(C2CCC2c2nc[nH]n2)=O)C1 c1(C(=O)NC(CC)(C)CNC(C2C3CC4C(C3)C24)=O)cc(C)n(C(C)C)c1C N1(C(CC(CCC)C)=O)CCC(C2CCCN(C(C3CC4CCCC34)=O)C2)C1 N#Cc1cnc(NC2CCC3CN(C(c4ncccn4)=O)CC23)c(Br)c1 C1(C(=O)NC(CC2CN(C(C3(C)CC(=C)C3)=O)C2)C)CCCN(C(C)=O)C1 Cc1ccc(C)c(C(=O)NCC2(NC(C3CC(C)OC3=O)=O)CC2)c1C CON(C)CC(O)Cn1cc(NC(=O)NCCCn2cc(Cl)cn2)cn1 C(=O)(C1=Cc2ccccc2C1O)NC(CC1CN(C(CNS(CC)(=O)=O)=O)C1)C c1(OC(C(=O)N(CCCNC(CC(=O)NCC)=O)C(C)C)CC)ccccc1F C(=O)(CCCCC(N)=O)NC1CN(C(c2cc(OCC)n[nH]2)=O)CC(C)C1 C(=O)(CC(C)C(F)(F)F)N1CCC(OC)(CNC(=O)C2=CC(C)(C)C2)C1 c1(C(N2C(CNC(c3c(COC)cco3)=O)C(C)CC2)=O)cnnc(C)c1C Cc1ccc(C(=O)NCC(=O)NC2CC2NC(=O)CSc2cn[nH]c2)cc1C c1(C(=O)NCCC(C)Nc2ncccn2)ccsc1C(=O)O C1(NC(c2c(CC)cco2)=O)CCC2CC1CN2C(c1oc(C)cc1C)=O C1(C(N2C3CN(C(=O)CSC4CCCCO4)C(C3)C2)=O)CC2COCC(C1)C2 N1(C(C(CSC)OC)=O)CC(C(=O)NC(c2csc(C)n2)C)C2(CC2)C1 C(CCCC(C)(C)C(=O)NNC(=O)c1cc(O)cs1)NC(C1C(C)OCC1)=O c1(OC)cc(-c2cn(C3CC(NC(c4nocc4Cl)=O)C3)nn2)ccc1Br C1(CNC(CC2CC(=C)C2)=O)CC2(CC2)CN1C(c1cccc(CS(C)=O)c1)=O N1(C(CC(C)O)=O)CC(C)CN(C(c2ccccc2OCCF)=O)C(C)C1 C1(C(=O)NC(CC2CC2)C(N2CCC(C(F)F)(CO)C2)=O)CCC(F)(F)CC1 c1(C(=O)NCC(C)N(C(C(CC#C)C2CC2)=O)CC)cc(F)ccc1CC N1(C(CCc2ccn(C)n2)=O)CCCCCC1C(=O)Nc1cccc(C#N)c1 O=C(C1=CC2(CCOC2)C1)N1CCCC(CNC(C2(CC(F)F)CC(F)(F)C2)=O)C1 c1(C(N2CC(C=C)OCC2)=O)ccc2c(n1)CN(C(=O)C(N)=O)CC2 c1(NC(CCNC)(C)C)nc2c(F)cccc2c(=NC(C)c2[nH]c(C)nc2C)[nH]1 C1(C(C)NC(=O)CCN2CCC2)CN(C(=O)CC2CCCN(C)C2)CCO1 Clc1cccc2nc(CN(c3nc(-c4cccnc4)cs3)CCO)sc12 C(CCC1CCC1)(C(=O)NC(c1ncccn1)CC)NC(c1c(CC)occ1)=O Cc1cc(C(=O)NCC2CCCN2C(=O)Cc2n[nH]cc2Br)ncc1F c1(COCC2N(C(C3C(C)(C)CCC3)=O)CCC2)c(F)cccc1F c1(N(CC(CCC)C)C)nc2ccsc2c(=NC2CC3CCCCCC23)[nH]1 c1(C(=O)NCC2C3CN(C(C4C(C)(C)C4)=O)C(C3)C2)cscc1S(C)(=O)=O C1(O)(CCNC(c2conc2C2CCC2)=O)CCCN(C(=O)COC2CC2)C1 C(=O)(C1=CCN(C)C1)N1CC=CC(NC(C(C)(C)SC)=O)C1 C1(CC(N2CCC(OCC(N)=O)C2)=O)COCCN1C(c1cnsc1)=O C(CC(C(=O)NCCc1cscn1)NC(=O)Cc1cnco1)=CC C12(CNC(=O)Cc3ccccn3)CCC1CN(C(=O)CCCCc1cnc[nH]1)C2 C1(C(=O)NCCC(C)NC(C=C(CCC)C)=O)C(C(=O)OC)CC(=O)N1C c1(C(=O)NCCCNC(C2CC3COCC3C2)=O)cc2cc(F)ccc2[nH]c1=O c1(CN(CC(C)NC(C2(C)CCNC2=O)=O)C)ccc2ccccc2c1 c1(C(N2C(CC)COCC2)C(=O)NCC(F)F)c(C)nn(CCCl)c1Cl C(c1cn(C)c2ccccc12)=CC(=O)NCC(C(C)C)NC(C1N(CC)CC1)=O c1(C(N2C(CNC(c3nc(COC)oc3)=O)CC(OC)C2)=O)ccc(C#N)cn1 CCCC(C#N)C(=O)N1CC(NC(c2cc(O)ncc2Br)=O)C2(CC2)C1 C12(NC(C3CC(C)C3)=O)CCCC1(F)CN(C(c1cc3n(n1)CCC3)=O)C2 N1(C(CCc2ccc(C)c(C)c2)=O)CC(NC(C2CC=CCO2)=O)CC12CCC2 C1(CCCCC)CCC(C(=O)N(CCCNC(=O)C(C2CC2)SC)C)O1 n1(CC(N2CC(F)(CNC(C3(COC)CC=CC3)=O)C2)=O)ccc(=O)c(O)c1C c1(C(N2CCCC(CNC(c3cncc(C)c3Cl)=O)C2)=O)cc2n(c1)CCSC2 Cc1cc(C(=O)Nc2nnc(CC(C)(C)C)s2)co1 C1(CC(=O)NCC(C(=O)OCC)C)CC2(C1)CN(C(C1(O)CCCCCC1)=O)C2 C1(C(=O)NCC(C)(C)OCCNC(c2c(C)csc2)=O)C2CCC(C2)C1(C)C C1(C(=O)NC(COC)C(=O)N2CC(N3CCOC3=O)C2)(CC)CNC(=O)C1 C(CN=C(NCCSC)NC1CCCCC1F)=CCC(=O)OC C1(C(N2CCC(O)(C(C)CNC(c3ccc(O)nn3)=O)C2)=O)(CC)CCCCC1 CN(CC(F)(F)F)NC(=O)c1ccn(-c2ccc(F)c(F)c2)n1 c1(C(N2CCN(C)C(CO)C2)C(=O)NC(C(=O)OC)C)ccc(Cl)c(Cl)c1C C12(C(N3CCC(=CCNC(C4(C)CCCC4)=O)CC3)=O)CCCC1OCC2 C1(NC(C2CCCCN2c2ncccn2)=O)CN(C(C2(O)CC2)=O)CC12CC2 C(=O)(C(O)CC[S+](C)C)N1CCCC(O)(CNC(CCN(C)CCO)=O)C1 c1(OC)cnc(F)c(C(=O)N(CCCCNC(=O)C(F)C(C)(C)O)C)c1 c1(C(=O)NCCCC2N(C(CCC(C)OC)=O)CCC2)ccc2c(c1)CCCO2 N1(C(C2N(C(c3cc(C)oc3C)=O)CC(C)(C)C2)=O)C2CCC1CC(C)C2 C1(C(=O)NC2(C)CCCC2NC(=O)C(O)Cn2cncn2)CC2(CCC2=O)C1 C1(CC(N2CCC(N(C(=O)COCCN(C)C)CCC)C2)=O)COC(C)(C)C1 N#CC1(C(N2CCC2CNC(=O)CCNC(=O)C=CCl)=O)CC1C(F)(F)F CC1(C)C(NC(C23CC(CO)(C2)C3)=O)C2CCCN(C(=O)CCc3ccoc3)C12 N1(C(CCCNC(C(CCCC)(C)F)=O)=O)CCCC2(CCCC2)C1 C1(CNC2C(CNC(=O)CNS(N)(=O)=O)C2)CCN(C(c2nc[nH]n2)=O)CC1 c1(C(N(C)CC2CCCN(C(C(CC)=CC)=O)C2)=O)cc(F)ccc1C1CC1 C(CC(C)(C)C(c1nnnn1C1COC1)NC1(CF)COC1)OC Cc1cnc(C(N2CC(F)CC2C(=O)NCC2CN(C(N)=O)C2)=O)cn1 C1(CC(=O)N(CCC#C)C)CCN(C(c2ccsc2)=O)C1 C1(CNC(C=CCCC=C(C)C)=O)CN(C(=O)Cc2ccns2)CCC1(F)F N1(C(CN(C)CC)=O)CCCC(N2CCN(C(c3c[nH]nc3F)=O)CC2)C1 C1(OC)CN2CCCC2(C(N2C3CCC2CN(C(=O)CN2CC4CC4C2)C3)=O)C1 Cc1ccc(C(N2CC(CC(=O)NCCc3cc(C)n(C)n3)CC2C)=O)cc1O C1(C(=O)NCCCN(C(C2CCC(C)S2)=O)C2CC2)CCC(C(F)(F)F)CC1 C1(NC(c2cc(C)no2)=O)C2CCCN(C(=O)C(F)CC3CCOC3)C2C1(C)C c1(CC(=O)NCC(C2CCC2)NC(=O)COC(F)F)cccc2ccccc12 C(=O)(C(C)(C)C(O)C(C)C)N(CC(CC)NC(=O)CCC(C)(C)[N+](=O)[O-])C CCC(CC)CCC(=O)N1CCN(Cc2cnc(N3CCOCC3)nc2)CC1C N1(C(C)C)N=C(C(=O)NCCC(C)NC(C2(CO)CCOC2)=O)CCC1=O c1(OC)ccc(C(=O)NCC2CC(NC(=O)COc3ccccc3O)C2)cc1F C(=O)(CCCC(=O)N(C(C)(C(=O)N1CC(C(C)(C)C#N)C1)C1CC1)C)N(C)C C1(C(N2C(CC(=O)NCc3ccncn3)CC2)=O)CC2CCC(C1)C2 S(=O)(=O)(c1cnc(N2CCn3[nH]c(=N)nc3C2)cc1C)NC(CC)C(C)O N1(C(CCOCCN(C)C)=O)CCC(CCNC(C2CCC(O)C2)=O)CC1 c1(OCC)ccc(-c2nc(CC(c3ccc(Cl)cc3)O)n(C(C)CC)n2)cc1 N1(C(C(c2cccc(F)c2)(C)O)=O)C2CCC1CN(C(=O)C1=CS(=O)CCC1)C2 CC1(C(=O)NCC(CNC(=O)Cc2cccc(O)c2)CO)CCCNC1=O C12(NC(c3c(C)cccc3)=O)CCN(C(c3cc[nH]c(=N)c3)=O)CC1C2 c1(NC2(c3nnnn3C3CCCCCC3)CSC2)ccc(C)c(SC)n1 n1(CC(=O)NC2C3CC(NC(C(CC=C)NC(C)=O)=O)CC32)ncc(C)cc1=O C12(CC)CC(C1)C(C(=O)NC13CC(C(N4CC5CC5C4)=O)(C1)C3)CC(=O)N2 C1(C(N2CCC(C(C(=O)NCc3c(C)n[nH]c3C)C)C2)=O)CC12CCOCC2 O=C(C(CO)C(F)(F)F)NCC1CCN1C(c1cnccc1C(F)F)=O C1(CCNC(CSC(C)C)=O)CN(C(C2CC2(Cl)Cl)=O)CC1C N1(C(C2CCN(C(C3C(C)(C(F)F)C3)=O)CC2)=O)CCC2(C=CCO2)C1 C12(NC(=O)C3CC3)CCN(C(=O)CCc3cc(Br)cs3)CC1C2 Cc1ncc(Cl)cc1C(N1CCN(C(=O)C(C)Cc2c(C)noc2C)CC1C)=O c1(C(N(CCCN(C(C2(C#N)C(C)C2)=O)C)C)=O)ccnc2cc[nH]c12 CN1CC(O)CCC1C(=O)NC(CCF)C(=O)N1CC(CO)C1 C1(C#N)(C(N2CC3(CN(C(c4c(C)[nH]nc4Cl)=O)C3)C2)=O)C(C#N)C1(C)C c1(C(=O)OC)ccccc1CCC(=O)NCC(C)NC(C1CN(C)C1)=O C(CCCC(=O)N(CC(=O)NC(c1nn[nH]n1)C1CC1)CO)(OC)OC C=CC1(C(N2CCn3cnnc3C2)=O)CCN(C(C2CC(C)CO2)=O)CC1 C1(NC(c2csc(Br)n2)=O)CCCCN(C(=O)Cc2ccccn2)C1 N1(C(C=CC(C)NC(C2CC(CF)C2)=O)=O)CCN2C(=O)CCC2C1 CON1CCC(CC(=O)NCCOCCN(C(=O)CC2CCOC2=O)C)CC1 C1(C(=O)OC(C)(C)C)(NC(=O)OCC2(CC)CCCCO2)CCCCC1 c1(C(N2CC(OC)C(NC(c3cnc(C4CC4)s3)=O)C2)=O)ccc(F)c(C)c1 N1(C(CC(CC)C2CC2)=O)CCN(C(=O)Cc2cc(F)cc(Cl)c2)CC1C CCC(C)C(=O)NCC(C1(O)CN(C(=O)CSCc2ccccn2)C1)(C)C CC1=NNC(=O)C1CC(=O)NC(C1CN(C(=O)C(F)=CC2CC2)C1)C C1(C(CNC(C2C(C)C2)=O)O)CCN(C(=O)CN2CCS(=O)CC2)CC1 Cn1nnc2c1CC(C(=O)NC(CNC(C1CCS1(=O)=O)=O)C(C)(C)C)CC2 N1(C(c2c(COC)cco2)=O)CCCCCCC1C(=O)Nc1ccc(C)cc1C c1(N(C2CC3CCC(C2)N3)C(CCc2n(CC)ccn2)=O)cnc(C)c(OC)c1 N1(C(c2c(C)ocn2)=O)CCC(c2nnc(CNC(c3cnc(O)o3)=O)s2)CC1 c1(C(N2CC(NC(C3(F)CCCN(C)C3)=O)CC2(C)C)=O)cccc2nn[nH]c12 Cc1ccc(=O)n(CC(=O)NCCC(C)NC(=O)C(O)CN2CCOCC2)n1 C1(NC(c2c(CNC(c3ocnc3C3CC3)=O)n[nH]c2)=O)CCOCC1F c1(C(=O)NC2(CN(C)C(c3cnn4ccsc34)=O)CC2)ccc(Cl)c(O)c1 C(=O)(C(C)(C)CC(C)C)NC1C(NC(c2ccc(CC)c(C(F)(F)F)c2)=O)CC1 C12(C(N3CCCC(NC(c4ccnc(C)c4N)=O)C3)=O)CCCCN1CCC2 C1(NC(C2C3CCC2(c2ccco2)C3)=O)CCNCC1C1CC1 CC(CCC(C)(C)C)C(=O)NC1CCCCN(C(=O)CSC(F)F)C1 C1(CC(C)C)CCCCN1C(=O)CN(C)C(C1(NC(N)=O)CC1)=O C(CCC(C(=O)N(C(C)CO)C)NC(=O)CCn1cnc(=N)[nH]1)OC CCC(CNC(=O)CC1CCCC(NC(=O)CCC(C)OC)C1)(CC)CC c1(NC(c2cnc(OC)c(-c3ccccn3)c2)=O)ccc2c(c1)CCC2=O c1(C(N2CCN(C(c3nc(Cl)sc3Cl)=O)C(CF)C2)=O)cnc(O)cc1O C1(NC(C2(C#C)CC2)=O)Cc2cc(C)c(C)cc2O1.C12CN(CCO1)CCS2 c1(NC2COCCN(C(c3c(OCCC)cccc3)=O)C2)ncc2c(n1)CCC2 c1(C(=O)NC2CC(CNC(C(Br)=C(C)C)=O)C2)ccc2nn(C)cc2c1 n1(CC(=O)NC2C(NC(c3c(CC)nc[nH]3)=O)CC2)ncc(C#N)c1N c1(C(=O)NC2CCN(C(CN(C(C)C)C)=O)C2C)cnn2c1OCC1(CC1)C2 Cc1cc(CC(=O)NCC2CC(F)(CNC(C3(C)CC3C(F)(F)F)=O)C2)c(C)s1 C1(OC)CC(CNC(=O)C(O)CN(C)C)N(C(=O)CC2(CO)CCOCC2)C1 N1(C(c2oc(CC)c(C)c2)=O)C(C(=O)NC2CCOC2C2CC2)CCC12CC2 c1(-c2cncc(NCc3cccc(OCC(=C)C)c3)c2)ccc(F)cc1CO N1(C(COC(CC)C)=O)CCCC(n2cc(COCC)nn2)C1 C(=O)(CCCC(=O)C1CC1)N1CC2C(C(N3CCC(CC(=O)OC)CC3)=O)(C2)C1 Cc1cccc(CC(N2CCOCC2CC(=O)Nc2cc(C(N)=O)ncn2)=O)n1 C1(NC(CCN(C2CC2)CC)=O)CCCCC1NC(=O)Cc1cnnn1C C1(C#N)(C(=O)NC(C)CCC(=O)NCCS(C)(=N)=O)CC12CCC2 C=CCCCCCC(=O)NC(C1(O)CCCN(C(C2(n3cccn3)CC2)=O)C1)C C1(CNC(C2CN(C(C)=O)C2)=O)CN(C(=O)CC2(O)CCCC2)CC1C C1(C(=O)NCC=CCNC(CC=C(C)C)=O)C2CCC1(c1cccs1)C2 C1(C(N2CCOCC(NC(CC(C)OC)=O)C2)=O)CC2(C1)CC1(CC1)C2 c1(C(C)C)ccccc1N(C(=O)CN1CCN(C(=O)OC(C)(C)C)CC1)C CS(=O)(=O)c1ccc(N2CCC(CNc3ccccn3)C2)c([N+](=O)[O-])c1 c1(N(C(CC2CC2)Cc2cccc(F)c2)CC)nc2c(C)cccc2s1 O(N=Cc1ccc2c(c1)OCO2)CCOC(CCCC#C)=O N1(CC(=O)NCCCn2cc(C3(C)CC(F)(F)C3)nn2)CCS(=O)(=O)CC1 CN=c1[nH]c(C(=O)NC(c2ccc(C)cc2)CNC(=O)C(C)(C)CC2CC2)cs1 N1(C(c2n[nH]c(=N)s2)=O)CCCCC(NC(c2c[nH]nc2C(F)F)=O)C1 C#CCCCCC(=O)NCC1(F)CC(NC(C2COC(C)C2)=O)C1 C1(NC(=O)NCC23CCCCCC2OCC3)CC2(C1)CC1CCC2C1 CC(C(=O)N(CCCN(C(=O)CC1(CO)CC1)C)C)OC(C)(C)C CC1C2C(CCN2C(C23CSCC2C3)=O)CN1C(=O)CCCC(=O)N(C)C C1(C(=O)NC(CNC(c2cn(CC(=O)OCC)nn2)=O)C)COC2COCC12 c1(C(=O)NCC(C)NC(=O)C(F)=CCCF)cc(O)cc(F)c1 C1(C(N(CCCCNC(c2c(C)ncc(C)c2)=O)C)=O)CCCCC12CCC2 C1(NC(c2n(CC)nc(C)c2)=O)CN(C(=O)CC2(CO)CC2)C2CCCC12 c1(C(=O)NCC(CCNC(CN(C2CCSC2)C)=O)O)ccc2cccnc2n1 C1(C(N(CC(CC)C)C)=O)C=CCN1C(C1CCCC1OC)=O c1(N(C2(N(C)C)CCCC2)CCCCOCCO)ccc(Cl)c(F)c1 C(=O)(C=CS(C)=O)N(C(C)CNC(=O)CNC(c1ccccn1)=O)CC N1(C(CCCC(=O)N(C)C)=O)CCC2CCCN(C(=O)COCC(F)F)C2C1 CC(C)(C)CC(C(=O)NCCC1CCOC1(C)C)NC(c1ccncn1)=O C(=O)(CCCC(=O)NC(C1CCN(C(=O)C(F)(F)CO)C1)C)NCC N1(C(C2(CC(C)=O)CCC2)=O)C2CCC1CC(NC(=O)C(C)N1CCC1)C2 C(C(C)(O)C(=O)N1CCC(C(C)CNC(c2ccoc2C2CC2)=O)CC1)OC c1(N2C3CC(CNC(=O)CN4CC5CC5C4)CC2CC3)ncnc2scc(Br)c12 C1(CNC(c2c(NC(=O)CSc3ccccn3)c[nH]n2)=O)CCC(O)CC1 N1(CC(=O)NC2C=CCN(C(C34CCC(CC3O)C4)=O)C2)Cc2ccccc2C1 C=CCC(CC)C(=O)NC(CNC(c1ccc(Br)c(F)c1)=O)C(C)(C)C CC1(C)CCCC(C(N2CCN(CC(=O)NCC(C)(F)C(C)(C)F)CC2)=O)C1 N1(C(c2c(CC)noc2C)=O)CC2(C)CC1(C(N1CCOC(CC3CC3)C1)=O)C2 N1(C(c2c(C)c[nH]c2)=O)CCC(CO)C(NC(c2nc(C)c(C)s2)=O)C1 C1(F)(C(=O)NC(CC)CCOC)CCN(C(=O)C(C)(C)CCF)CC1 C1(CC)(CC)CCCCCC1.c12ccc(C)cc1O2.C1(=O)NCCO1 CC1C(=O)Nc2ccccc2N1C(c1cc(C(C)(C)C)nn1C)=O N1(C(CC(CC=C)NC(=O)CCC(F)(F)F)=O)CCc2cccc(C)c21 CCCCC(C(=O)N1CC(n2cc(C)cn2)C1)N(C)C.C(C(=O)OCC)(NC)C1CC1 C1(NS(CC)(=O)=O)CCN(C(=O)C(N2CC3CC3C2)C)C1 C1(C)(CC(=O)NCCC(C)N(C(=O)C(Cl)=CCl)C)CC(F)(F)C1 n1(C(C)C)ncc(F)c1C(=O)NCC(C)CNC(=O)C(C(C)C)N1CCCCC1 c1(C(N2C(C)(CNC(c3cnc(O)o3)=O)CCC2)=O)cc(F)c(Cl)cc1Cl C1(NC(c2[nH]c(=NCC)sc2)=O)CCN(C(=O)C(C)OC2CCCC2)CC1(C)C c1(NCc2occ(C)c2)nc(C)cc(=NC2CCS(=O)(=O)C(C)C2)[nH]1 N1(C(c2occ(C)c2)=O)CCC(C(=O)NCCC2CCC(C)(C)C2)(CF)C1 Cn1nc2c(c1N)CN(CC(=O)NCC1CC3CCC1C3)CC2 C1(C(N(C(CC(CC)C)C)C)=O)CCN(C(c2cnccc2OC)=O)C12CC2 C(CCC(=O)N(C(C)Cc1cc(C)[nH]n1)C(C)CO)OC CC(O)CC(=O)N(C(c1ccccc1)CNC(=O)C(C)(C)c1nncn1C)C c1(C(=O)NCC(CC(C)C)NC(=O)C2=COCCC2)cc2c(s1)CCSC2 C1(NC(c2cnc(C)[nH]2)=O)C2CCCC1CC(NC(=O)CCCS(C)(=O)=O)C2 Cc1cccc(NC(=O)CCC2CCCN2c2cc(C#N)ncn2)c1F C12(NC(CCNC(=O)C=CCl)=O)CC1CC1CN(C2)C(=O)CC1(C1CC1)CC N1(C(C=CC(=O)NC)=O)CCC(C)C(NC(=O)CC2C=CCC2)C1C n1(CC)cc(S(=O)(=O)N2CCCC(C(=O)NCc3cc4ccccc4s3)C2)cn1 C12(C(=O)NC3(C(N(OC)C)=O)CCN(C)C3)CC1COC2(C)C c1(C(=O)NCC2N(S(CC(C)C)(=O)=O)CCC2)c[nH]c2ccc(C#N)cc12 c1(C(=O)NC2C(NC(=O)CCN3CCOCC3)COCC2)ccc2ccsc2c1 c1(N2CC(C)=C(C)C2)ccc(C(C)C)cc1S(=O)(=O)NCC1COC2(CCC2)C1 n1(CC(N2CC(C(C(=O)NCC(C)N(CC)CC)O)C2)=O)c(O)nnc1O CC1=NOC(C)(CNC(C2CCC(NC(=O)CCCC3CC3)CC2)=O)C1 Cc1ccc(NC(=O)CC2CCN(C(c3cncn3C(C)C)=O)C2)c(C)n1 n1(CC(=O)NC2CC(CCNC(C3CCC3(F)F)=O)C2)cnc2sccc2c1=O c1(OC(C(=O)NCC(CC=C)NC(=O)CCC(=C)Cl)C)ccc(Cl)cc1C c1(CC(=O)NCCC2CCN(C(c3cn(CC)nc3)=O)C2)c(C)nn(C)c1Cl c1(CC(=O)NCC2CC2NC(C2CCc3nc[nH]c3C2)=O)ccc2c(c1)CCC2 C1(C(=O)NC2CCN(C(=O)C3CC3)CC2F)CCn2c(C(F)(F)F)nnc2C1 c1(NC2C(C)C2(F)F)cc(N2CCOC(C3CCCCC3)C2)ncn1 N1(C(C(C)NC(CC)=O)=O)CCC2C(CCCN2C(C2SCC=C2C)=O)C1 CCCC(C(=O)NC)NC(=O)NC1CCCCC1C(N1CCCC(CO)C1)=O c1(C(N2CCC(N(C(COCCOC)=O)C)CC2)=O)cc(F)cc2ccncc12 N1(C(C=CC=C(c2ncon2)C)=O)CCN(C(=O)Cn2cc(Cl)cn2)CC1 c1(C(=O)NC(CNC(CC(C)=C(C)C)=O)(C)CO)ncccc1C C(C(N=[N+]=[N-])C(=O)NCCCOCCNC(=O)CCN1CCC1)OCC N1(C(C(C)S(N)(=O)=O)=O)CCC2CCN(C(c3ccnc(C(N)=O)c3)=O)CC12 CC1C(NC(c2cnns2)=O)CC2CCC1N2C(c1cnoc1C1CC1)=O C(=O)(C(CC(F)F)NC(c1csc(O)n1)=O)NC(c1cncs1)C C1(C(C)C)CN(C(=O)C=Cc2cccs2)CCN1C(=O)CSCC1CCCCO1 N1(C(c2cccc(C(=O)OC)n2)=O)CCN(Cc2ccc(I)c(F)c2)CC1C#N N1(C(C23CC(C(C)(C)C)(C2)C3)=O)CCCN(C(c2nc(Cl)sc2Cl)=O)CC1 c1(N2CC(NC(c3cc(OC)c(Br)cc3)=O)(CO)C2)ncnc2c1CCCC2 Fc1ccc(OC(F)F)c(Oc2ccc(-c3nc[nH]n3)cc2)c1 N1(C(c2cnc(C)[nH]2)=O)CC(NC(C2CC2c2ccccc2F)=O)C(C)C1 c1(C(=O)NC2(CNC(c3cnn4c3OCC4)=O)CCC2)cc(F)c2cn[nH]c2c1 c1(C(N2CCC(CO)C(NC(=O)C(F)(F)CC3CC3)C2)=O)[nH]cc2c1CCCC2 N1(C(C2N(C(CCC(=O)NC)=O)CC(O)CC2)=O)CCOC2C(O)CC12 C1(CNC(CCOCCC)=O)C2CN(C(c3cncc(NS(C)(=O)=O)c3)=O)CC12 C1(C(=O)NCCCCCS(C)(=O)=O)C2Cc3c(Br)cccc3C12 n1(CCC(N2CC3CC2CS3=O)=O)sc2ccccc2c1=O CN1CC2CCCC(NC(=O)N=c3[nH][nH]cc3C(N)=O)C2C1 c1(NC(c2ccc(-c3cc(C)nnc3)cn2)=O)cc(NC(C)C)ccc1Cl C1(CCC)(NC(c2sncc2CC)=O)CCCN(C(=O)C(C)=C2CCC2)C1 N1(C(C2CCOC2=O)=O)CCC2CCN(C(c3[nH]cc4c3CCS4(=O)=O)=O)C2C1 C1(C(N2CC(n3cc(CC4(O)COC4)nn3)C2)=O)CCN(c2cc(O)ncn2)CC1 C1(C(=O)NCC(C)CNC(c2conc2C(F)(F)F)=O)CCCCC1O C(=O)(CCC(=O)NCC1CC1)N1C(CN(C(CSCC)=O)CC)CCC1 C12(NC(c3[nH]cc(SC(C)(C)C)c3)=O)CCC(CC1CNC(C1CC1(C)C)=O)C2 CC1CCC(C)(C(N2CC(O)(CNC(=O)Cc3cccnc3O)C2)=O)C1 Cn1nnc2c(C(=O)NC3(C)CCN(C(c4cc[nH]c(=N)c4N)=O)C3)ccnc12 C1(C(=O)NCC(O)C(C)(C)C)(CC)CCN(C(c2cccc(O)c2)=O)C1 C12(NC(C(C(C)(C)O)F)=O)CCCC1N(C(c1cc3c(s1)CCC3)=O)CCC2 c1(C2(C(=O)NC(C(C)NC(CN(S(CC)(=O)=O)C)=O)C)CCC2)ccc(O)nc1 C=CCN=C(NCCCC1CCCCO1)NC1CCOC(C)(C)C1 N1(C(CCCC#C)=O)C(CNC(c2ccc(F)cn2)=O)CC2CCCC12 c1(COC)cc(C(=O)NCC2(NC(=O)C(c3ccccc3)F)CC2)c(C)o1 c1(CN(CCOC)C)ccnc(SCc2ccccc2N(C)C)c1 c1(C(N(C(CCNC(CN(C(C(C)C)=O)C)=O)C)C)=O)cnn(C(C)C)c1F C#CC1(NC(C2C3CN(C(=O)C(C)OCOC)CC23)=O)CC2CCCC12 C(CNC(C1C=CCC1)=O)(CC(F)(F)F)NC(C(c1cccc(OC)c1)(F)F)=O N1(C(CCC)=O)CC2CC1C2NC(=O)C(O)Cc1cc(Cl)sc1Cl N1(C(C2COCC(C)O2)=O)CCC2CCCC12C(=O)Nc1cn(C)nc1O c1(NC(C2CCN(Cc3nc(Br)ccc3F)CC2O)=O)cc([N+](=O)[O-])ccc1Cl C(=O)(NNC(=O)C(=O)N1CCCC1)C1SCC(C(=O)OC)C1 CCCC(C)C(c1nnnn1C(C)(C)C)NCc1ccc(Cl)o1 c1(C(N(CCOC)CCNC(=O)CSCCC(C)C)=O)c[nH]nc1Cl c1(C(=O)NC(CN(C(c2cnc(C)[nH]2)=O)C)C)ccccc1-n1cccn1 c1(C(N2C(CNc3ccc(NC(C)=O)s3)CCC2)=O)cccc(C(=O)C2CC2)c1 S1(=O)(=O)c2ccc(s2)C(=O)N1C.N1(CC#N)CCS(=N)(=O)CC1.Cc1cccc(N)c1 C(c1ccc(Br)cc1)=CC(=O)NCC(CO)NC(C1CCCCC1)=O c1(NC(C2N(C(CCN(C)C)=O)C3C(C2)C3)=O)ccc2c(c1)CCOC2 CC1CCCC=C1C(=O)Nc1c(Sc2ccc(Cl)cc2)cccc1F C1(O)(C(=O)NCC2C3CN(C(CCCCOC)=O)C2C3)CCc2ccccc2C1 C(c1ccc(Br)c(C)c1)=CC(N1CC2C(NC(COC(C)=O)=O)(CC2)C1)=O c1(C(N(CCOC)CCNC(=O)C=Cc2cccs2)=O)ccncc1O C1(CNC(CC(C)C2CC2)=O)C2CC3CC(C2)CC1C3 N1(C(C2C(OCC)C2)=O)C2CCC1CN(C(=O)CC(O)CCSC)C2 CCCC(C)C(=O)NC(C1(O)CCN(C(C2CSCCS2)=O)C1)C CONC(=O)C(=O)NCCC(=O)NCCC(C)N1CCCC1 C1(CC(=O)NCCN)C=CS(=O)(=O)C1.N1(N(CCC)C(C2(C=O)CC2)=O)CCCC1 S(=O)(=O)(c1ccc(NCCCC(C)CO)c(Br)c1)NC1(CC=C)CCN(C)CC1 N1(C(=O)C2=NOCC2)CCCC(O)(CCNC(C2(C(F)(F)F)CCCCC2)=O)C1 C1(C(=O)NCC(n2cccn2)C)CC(C)(NC(C2CC(CF)C2)=O)C1 CC1(C)CC(C(=O)NCc2nccn2C(C)C)CN(C(=O)C(O)C(F)(F)F)C1 Cc1cccc2c(C(=O)NC3(C)CCCN(C(=O)C(O)C4CCC4)C3)n[nH]c12 c1(N2C(CNC(C(c3ccc(C)cc3)(F)F)=O)C(C)CC2)cc(O)nc(C)n1 C12(C(=O)NCC(C(C)C)Nc3cc(=O)n(C)c(O)n3)CC3CC(C(=O)N1)C2C3 CC1CN(C(=O)CCCNC(=O)C(N2CCNC2=O)C)CC(C(N)=O)O1 c1(C(=O)NCC(C)C(=O)NCC2CC2[N+](=O)[O-])cccc2occc12 c1(NC(C2(F)CCN(c3nccc(OC)n3)C2)=O)ccc(Br)c(C(C)=O)c1 N1(C(C(C)OC)=O)CC(NC(=O)CNC(=O)CCC(C)C)C(C(F)(F)F)C1 c1(C(=O)NCC2CN(C(c3c(CC)nns3)=O)C3C2C3)ccc(C(F)F)c(F)c1 c1(CCC(=O)NC2C(NC(C=Cc3ccc(C)o3)=O)CC2)c[nH]c2ccccc12 C1(C(=O)NC(CCOCC)C(=O)NCC2CCSC2)CC2CCCC2C1 C1(CNC(CS(CC)=O)=O)CC(C(C)C)CCN1C(=O)CCc1cccnc1Cl CS(=O)(=O)c1cc(CN2CCC(CC(=O)Nc3ccc(O)cn3)C2)ccc1F c1(OC)ccnc(C(N2CCCC(CCNC(C3C(C)C3C)=O)C2)=O)c1F c1(C(=O)NC2CCC(NC(C(CC)=CCCC)=O)CC2)ccc(Cl)nc1N c1(C(N2C(C(=O)NCCC(C(C)C)OC)C(C)(C)C2)=O)ccnc2cc[nH]c12 CC1C(C(=O)N2CCC(CNC(=O)CCCn3cccn3)C2)=Cc2ccccc21 c1(C(N2CC3(CN(C(C(CC)(CC)CO)=O)C3)C2)=O)cc(N)c2ccccc2n1 C(=O)(CCN(OC)C(=O)C12CC1CCN2C(=O)CC(C)C1CCCC1)OC C1(CNC(C2CC(CC(=O)OC)C2)=O)COC(CNC(c2csc(O)n2)=O)C1 C1(CCNC(=O)CC2CCCCC2)(OC)CN(C(C2C(C)CC2C)=O)C1 C1(CNC(=O)NC(c2cn(C3CC3)nn2)CC)CC2CC(OC)C2C1 N1(C(C(=O)NC(c2ncccc2Cl)C)=O)CC2COCCC2(N)C1 N1(C(C(c2ccc(C)o2)C)=O)CCC(C)(C(=O)NCC2CN(C3CC3)C2)C1 c1(C(=O)NCC2(O)CN(C(C=C(C)C)=O)C2)cccc2c(O)ncnc12 C1(CC)CN(C(=O)C(Cc2ccsc2)NC=O)CCC1NC(c1sccc1C)=O N1(C(c2c(C#C)c[nH]n2)=O)CCCN(CCNC(C2CN(C(N)=O)C2)=O)CC1 C1(CNC(C(=O)NCC2C(c3ccccc3)(C)C2)=O)C(F)(F)C12CC2 C(=O)(C1=CC2(CCOCC2)C1)NC1CCC2CN(C(C(C3CC3)OC)=O)CC2C1 Cc1ncc(C(=O)NCC=CC(=O)NCCCC2CC2C)s1 N1(C(CC(C)(C)O)=O)CCC(NC(=O)Cc2ccc(F)c(F)c2)C2CC12 C1(NC(CCC)=O)(CF)CCN(C(c2cnn(-c3ccccc3)c2)=O)C1 C12(C(=O)NC3CN(C(=O)COc4ccccc4)CC3F)CCCC(CCC1)C2O CC1CN(C(=O)CSc2ccccn2)CCCN1C(=O)CC1CCCC(F)(F)C1 CCCC(CNC(c1ccn(C)c(=O)c1)=O)C(=O)Nc1cccc(Cl)c1O c1(C(=O)OCC)cnccc1N1CCC(C)(NC(=O)C(=Cc2cccs2)C)C1 C1(NC(c2ccc(CN=[N+]=[N-])o2)=O)CN(C(C2CCCC(F)(F)C2)=O)CCC1F C=CCC(C(=O)NCC(F)(C(=O)NCc1ccc(Cl)o1)C(C)C)C(C)C C(C(CO)C(C)C)NC(C(c1cn(C)nn1)NC(CCC=CC)=O)=O C(CC(CNC(c1ccnn1CCF)=O)NC(C1OCC1(C)C)=O)OC Cc1cc(C(=O)NC2CCCCC2CNC(C2CC2(C)C)=O)ccc1F C#CC(CNC(=O)C(CCF)NC(=O)Cn1[nH]cnc1=N)C(C)C c1(C(=O)NC2CC(C)(NC(Cc3ncc(CC)[nH]3)=O)C2)cn(C)nc1C(C)C c1(SC)nc(Cl)c(CN2CC(C)(CC(N3CCOC(C(F)(F)F)C3)=O)C2)c(Cl)n1 C1(NC(C=CCC)=O)CC2(CCC(CNC(C34CCC(CC3)C4(C)C)=O)OC2)C1 C#CC1(C(N2CC(CCCCNC(C3(C)CCCC3C)=O)C2)=O)CCCC1 c1(CCC)ccccc1NC(C1CC(F)CN1C(c1cnn(C(C)C)c1)=O)=O CCC(CC)C(C(=O)NC1CCC(C(N2CCCCC2COC)=O)C1)OC Cc1cnc(C(=O)NCC2CN(C(=O)CC3CCN(C)CC3)CCC2C)c(C)c1 n1(C(C)C)cc(C(=O)NC2CN(C(=O)CNC(N)=O)CC3CC23)ccc1=O CCCCCCC(CC)C(=O)NCC1(O)CN(C(c2ccnn2C)=O)C1 C(=O)(CCS(N)(=O)=O)N1CCN(CC(C)(C)NC(=O)Cn2cncn2)CC1 Cc1cccc(C2(CNCCC3OCCC3C)CCCCC2)c1 C1(C(=O)NC2CN(C(CCc3nc(C)c(C)o3)=O)C2)CCCC2(CCOC2)O1 C1C2=CN(CC2)C(=O)CNC(=O)C(C)N1C.C(C)(C)(C)O.C1CC1 c1(OC)cc(C(N2CC(NC(c3cc(C)ncc3Cl)=O)C2)=O)nc(C)c1 N=c1[nH][nH]c(=NC2CCCN(C(c3cc4c(s3)CCSC4)=O)CC2)[nH]1 c1(C(=O)NC2CN(C(CC(c3ccc(C)cc3)C)=O)CC2C)ccc(F)c(C)c1 C1(NC(=O)COCC2CC2)CC(F)CN(C(C2C(F)(F)C23CC3)=O)C1 C(CC(C(=O)NCc1ncoc1C1CC1)NC(=O)Cn1ncccc1=O)OC N1(C(CCC(=O)OC)=O)CCC2CCN(C(c3cc(OC)c(Br)s3)=O)C2C1 N1(C(C(COC)COC)=O)CCCC(N(C)C(c2cccn2C)=O)CC1 N1(C(c2cc(C(C)C)on2)=O)CCC(F)(F)C(NCc2cc(Cl)ccn2)C1 N1(C(C(C(C)C)F)=O)CCC2CCCC(C1)N2C(=O)Cn1ncc(O)nc1=O N1(C(c2cncc(CNC(C3(F)CCC3)=O)c2)=O)Cc2ccccc2C1 C(C1=CCN(C(=O)C(c2ccccc2)F)CC1)NC(c1cc(C)c(C)[nH]1)=O O=C(C1=CC2CCCCCC12)NCC1CCCN1c1ccc([N+](=O)[O-])c(C)c1 Cc1nc(C(=O)NCCCC(C)NC(=O)CCC2CC2C(F)F)cn1C(F)F c1(NC(C2C=CC(NCc3n(C)ncc3)C2)=O)ccc2c(O)nc(O)nc2c1 Cc1nccc(CNC(=O)Cn2cc(C(=O)O)nn2)c1C c1(-c2ccc(C(NOC)=O)cc2)cnc(C(=O)NCc2ccccc2C)cc1C C(=O)(C1=COCCO1)N1CCC(N(C(C(CC)OCC)=O)CC2CC2)C1 C1(NC(c2[nH]n(C)c(=O)n2)=O)CCN(C(=O)CNC(N2CCCC2)=O)C1(C)C N1(C(c2ccc(C(C)C)s2)=O)CCN(C)C(C2COC2)C1 N1(C(c2cnc(C(C)OC)s2)=O)CCN(C(c2cc(C)cc(N)c2)=O)C2CCC12 Cc1ccc(OC(C)CNC(C2CC2c2[nH]cnc2C)=O)c(C)c1 c1(CC(=O)NCCCCC(C)NC(c2nccc(C)n2)=O)ccc2c(c1)CCO2 c1(C(=O)NC(C(=O)N(C)Cc2cc(OC)no2)C2(C)CC2)scc(C)c1C N1(C(Cc2c(C)nc[nH]2)=O)CCN(C(C2(C)CCCCCC2)=O)CC1CF N1(C(CN(CCC)C)=O)CCCC(C)C1CCNC(=O)CC1CCN(C)CC1 N1(C(c2ccc(OC)c(N)n2)=O)CCC2CN(C(=O)C=CS(C)=O)C2C1 N1(C(c2cc(C)[nH]c2)=O)CCCC(C(=O)NCC(C)(C)C(C)O)C1 CN1CCCC(CC(=O)NCC(C2CC2)N(C(=O)CCc2cn[nH]c2)C)C1 CC1CN(C(c2cc(Cl)c(Cl)[nH]2)=O)CC1NC(c1coc(Br)n1)=O C1(NC(=O)C(O)C(F)F)CN(C(c2cc(C3CC3)no2)=O)CC2(CCOCC2)C1 N1(C(C2(CC=C)CCN(C(C3CC(OC)C3)=O)C2)=O)CCc2c[nH]nc2C1 C1(NC(C2C(C)=C2)=O)CN(C(c2coc(C3CCC3)n2)=O)CC1(C)C C1(CNC(c2ccc(NC)cc2)=O)CN(C(=O)C(c2ccccn2)O)CCCO1 c1(C(N2CCN(C(CCCOCCC)=O)CC2C)=O)ccc2c(c1)C(C)CN2 C1(C2CCCN(C(c3ccnc(C#N)c3)=O)C2)(NC(C(C(C)C)O)=O)CC1 c1(CCNC(C2CC(=O)N(Cc3ncccc3O)C2)=O)coc2ccccc12 Cc1cccc(C(=O)NCCC(O)CNC(c2nnc(O)cc2O)=O)c1O c1(C(=O)NC2CN(C(c3c(C)nns3)=O)CC3C2C3)c(N)cccc1[N+](=O)[O-] CSC=CC(=O)NC(C)(CNC(=O)C(C1CCOCC1)F)Cn1cccn1 N1(C(C(C)C2(O)CCC2)=O)CCC2CCN(C(=O)CC3(O)CCC3)C2C1 C1(CN(C(C(C)OCC2CC2)=O)C)CCCN(C(=O)CN2CCC(C)(C)C2)C1 N1(C(Cc2c(SCC)cccc2)=O)CCC(NC(=O)CC#N)C(C)C1 c1(C(N2CCC(C(=O)NCCN(C)C)CC2)=O)ncc(Br)cc1Br c12cccc(c1)CNC(=O)N2.c1(C(C2CC2)SC)ccccc1-c1cccnc1 N(C(=NCC(C)C)NCC1(C)NC(=O)NC1=O)CC(C1CCCCC1)OCC c1(C(=O)NC(c2ncccn2)C(C)C)csc(-c2ccccn2)n1 c1(C(=O)NC2CC(C(=O)NCC#N)C2)ccc(Br)cc1 c1(C(=O)NCC(=O)N(CC(=O)OC)C)oc2ccc(F)cc2c1-c1ccccc1 C#CC1(O)CC(C(N2CC(NC(c3scc(C)c3OC)=O)C(F)C2)=O)C1 Cc1ncc(C=CC(=O)NC(C2CCCN2C(=O)C(C)(F)F)(C)C)c(O)n1 C(=O)(C(C)CCCOC)NCC1(C)CCN(C(CN(CCC)C)=O)C1 c1(C(=O)NC2C3CN(C(c4ccc(C)s4)=O)C(C3)CC2)cn2ncnc2nc1C N1(CC(=O)NC(C(C)C)C)CCC(C)C(NC(c2cc(F)cnc2O)=O)C1 CC1=C(C)CC(C(=O)NCC2(C(N3CCC=CC3CO)=O)CC3(CC3)C2)CC1 CN1CC(NCCC23CCC2CN(C(=O)OC(C)(C)C)C3)CCCC1=O C1(C(=O)NCC(CC)CC)CC(F)CCN1C(=O)CC1CC(OC)C1 Cc1nc2cc(C(N3CCCC(C)C3CCN=c3cc(F)nc[nH]3)=O)ccc2o1 C1(C)(CC)CCCN(C(C2CC3CN(C(c4ccsn4)=O)CC3C2)=O)CC1 C12(C(=O)NCC(COCC)C)CC(CN(C(c3c[nH]nc3CC)=O)C1)C2 c1(N(CCN(C(C)=O)Cc2cccc(C)c2)C(C2CC(Cl)C2)=O)cc(C)oc1C C1(F)(CNC(CC)=O)CCN(C(c2ccc(CC(C)(C)O)cc2)=O)C1 CCC1=NOC(CC(=O)NCC2CC(NC(c3c[nH]nc3Br)=O)C2)C1 CCC(CCC(=O)NCc1nc(=O)o[nH]1)NC(=O)C(C)(C#N)CC c1(OC)ccc(F)c2[nH]c(C(=O)NCC(C)NC(=O)CC(C)P(C)(C)=O)cc12 c1(C(=O)NCC(=C)CCNC(=O)CCNC(=O)CO)cc(CO)n(C)n1 CC(C)C(C(=O)NCC1CCC(C(=O)NOCCCCC2CC2)C1)C(C)C Cc1nc(C)n(O)c1NC(C1CCC(CN(C2CCN(S(C)(=O)=O)C2)C)CC1)=O C1(NC(C(C2CN(C(=O)C(C)(C)CCF)C2)OC)=O)CCn2nccc2C1 c1(C(=O)NCC2C(NC(c3cc(F)cnc3O)=O)CCC2)cnc2[nH]nnc2c1 n1(CC(N2CC(C)C(C)(CNC(=O)C(C)(C)C)C2)=O)cc2ncccc2n1 c1(CNC(CC2OCCN(c3nc(C)c(Br)cn3)C2)=O)ccc2ncnn2c1 C1(C(=O)NC(C2CCCCC2)C(=O)NCCC(C(=O)OC)C)CCC(C)=C(C)C1 Cc1c(O)c(=O)ccn1CC(=O)OCC(=O)NCCCc1ccccc1F c1(C(=O)OC)cccc2cc(COCCC3(C(=O)O)CCOCC3)c(=O)oc12 C1(NC(C2CCOCCN2C(=O)C=Cc2ccoc2)=O)CC2CCCCCC12 C1(C(N(CC(C)CNC(C2CC2c2ccsc2)=O)C)=O)CS(=O)(=O)CC(=O)N1 N1(C(C2CC(OCC)C2)=O)CC=CC1C(=O)NCC(C)(C)CO CC(CC(F)F)C(=O)NCC1CCN(C(=O)C=CC2CCCCCC2)CC1O c1(C(=O)NC2CC3CC(NC(C(F)=CC)=O)CC32)cc(Br)c(F)cc1F N1(C(=O)NCc2ccn(C)n2)CCOC(c2nc[nH]n2)C1 c1(C(N(C2CC(CNC(C3(O)CC(CF)C3)=O)C(O)C2)C)=O)cccc(CO)n1 Cc1ccnc(CNC(=O)C(O)CNC(=O)C=Cc2ccco2)n1 C1(CNC(C(C)NC(CC)=O)=O)CC(NC(c2ccccc2C(C)C)=O)CCO1 c1(C(N(CC(C)CNC(=O)CCS(N)(=O)=O)C)=O)ccc2c(c1)CC(=O)N2 N1(C(C2CCSCC2)=O)CCC(C2CN(C(C3CCC(C4CC4)C3)=O)C2)CC1 C#Cc1ccc(C(=O)NCC(F)CNC(=O)CCOCC(C)C)cc1 N1(C(CN(C2CCCC2)C)=O)C2CCC1C(CNC(C13CCCC1CCC3)=O)C2 c1(ONC(C2N(C(C(COC(C)=O)C)=O)CC=C2)=O)cccc2[nH]ccc12 C1(C(=O)NCCCCN(C)C(c2ccncn2)=O)CCC(C(F)(F)F)O1 CCCCCCC(=O)NCC(O)CN(C)C(c1cc(F)c[nH]1)=O CC1CN(C(C2CCCCS2)=O)CC(C(=O)NCC2(F)CN(C)C2)O1 CCC(CN(C)C)CC(=O)N1CC(CNC(=O)CCN2CCC(N(C)C)CC2)C1 CN1N=CC(CC(=O)NC(CNC(=O)C(c2cccc(Cl)c2)(F)F)C2CC2)C1=O N1(C(=O)OC(C)(C)C)CCCC2(CCN(CCN3CCOC4(CCC4)C3)C2)C1 C1(COCC)(CNC(=O)C(C)OC)CCN(C(=O)COC2CC(F)(F)C2)C1 C(=O)(CCC(C(=O)N1CCCC(C(O)C(F)F)C1)NC(=O)OC(C)(C)C)OC N1(C(C)C(=O)Nc2ccn(C)n2)CCCC2C(NC(=O)NC3CC3)C(C)(C)C12 C1(C(N2CCC(c3ccon3)C2)=O)CCN(C(=O)CCCC2CCC2)C12CC2 c1(-n2ccc(C(=O)NCCOC3CCN(C(C4C(C)C4)=O)C3)n2)cncc(F)c1 C12(CCCNC(=O)NCCc3cc(C(=O)OC)no3)CC3CC(C1)CC(Cl)(C3)C2 C1(CC=C)(C(=O)NCCCC)C=CCN1C(=O)C(C)COc1ccccn1.C1CO1 C(CC(O)C(=O)NCC(C(F)(F)F)N1CCN(C(=O)C(C(C)C)OC)CC1)SC CC(C)(CO)CCNC(C1CCCN1C(c1cnnc(O)c1)=O)=O Cc1cc(C(=O)NCC2CCC2NC(c2nnn(C)c2C)=O)ncc1F C1(NC(c2cc(CC)[nH]n2)=O)CC2CC(NC(c3cncc(NC)c3)=O)C2C1 N1(C(CC(C)(C)SC)=O)CCC2(CCN(C(=O)CN3CCn4ccnc4C3)C2)C1 c1(OC)ccc(C(=O)NCCN(C(C2CCC(N(C)C)CC2)=O)C(C)C)nn1 Cc1c(NC(C2C3CN(S(=O)(=O)CC4CCCCC4(F)F)CC23)=O)cccc1Cl C1(NC(CC2(CNC(CSCC#C)=O)CC2)=O)(CO)CCOCC1 CCCC(CC1CCCC1)C(=O)NC1CCC1Cc1cccs1 C=C1CCC1(C(=O)NC(C)CC(C)NC(=O)CC(C)c1ccco1)C(=O)OC c1(OC)ccc(F)c2cc(C(=O)NCC=CCNC(C3(C)CC3)=O)[nH]c12 c1(C(=O)NC2COCCN(Cc3cnc(CCC)s3)C2)cc(O)c(O)c(O)c1 c1(C(=O)NC2CN(C(C(COC)O)=O)CC2O)c(C)nc(C2CC2)nc1O Cc1ccc(C(=O)NC2CC(CNC(c3scnc3C)=O)C2)c(Cl)c1 C#Cc1c[nH]nc1C(=O)NC(C1(O)CCCCC1)C(N1CC(C)(C#N)C1)=O C12(CC(=O)NCCCCO)CCC1CN(C(c1nccs1)=O)C2 N#CCCCC(=O)NCC1CCC(CNC(C2(C(F)(F)F)CCOCC2)=O)CC1 N1(C(CC)C(=O)NC2CC(F)(CNC(=O)C(F)=C3CCCC3)C2)C(=O)CCC1=O c1(C(=O)NC(C)CCNC(C2CCCN(C)C2)=O)cc2c(F)ccc(Cl)c2[nH]1 CCCC(CCNC(C1(CC)CN(C(c2sccc2OC)=O)C1)=O)CCC c1(CC(N2CC(NC(C3C(CCC)CCC3)=O)C2)=O)n[nH]c2ccccc12 c1(C(N(CCC#C)CC)=O)cnn(CCNC(C2CC(F)C2)=O)c1 C1(C(=O)NCC(C(C)C)O)CCN(C(=O)C(C)C#N)O1 N1(C(Cc2cc(C)no2)=O)CCC2CCCC12CNC(c1cc(N)nc(Cl)c1)=O c1(C(=O)NC2C(OC)CN(C(=O)CCC(=O)c3ccc[nH]3)C2)cc(C)nc(C)c1 C1(NC(C2CC(O)C23CCC3)=O)COC2(C1)CN(C(c1nc(Cl)c(Cl)s1)=O)C2 C1(NC(C(CN(C)C)N(C)C)=O)CCCC(CNC(=O)CCc2cscn2)C1 Cc1csc2ncnc(N3CCC(CNC(=O)C(O)C4CC4)C34CC4)c12 c1(CCNCc2n(C)cc(Cl)c2)ccc2c(c1)CCCO2 Cc1cnc(CCCC(=O)OCC(=O)CCC2CC2(C)C)[nH]1 C1(NC(C2CCN(C)C2)=O)CN(C(C2(F)CCCCC2)=O)CC2(CCC2)C1 S(=O)(=O)(CCC(=O)NCCC(F)Cn1cc(C2CCOCC2)nn1)N(C)C C1(S(C)(=O)=O)(C(N2CC(CCNC(C(C(C)C)NC(C)=O)=O)OCC2)=O)CCC1 N1(C(C2CC(SC)C2)=O)CCC(CCCNC(c2nc(C)c(C)s2)=O)CC1 C(C)(C(C(=O)NC1(CCNC(=O)CC(=O)N(C)C)CC1)N(C)C)OC N1(C(C(C)OCC(C)C)=O)CC(C2CN(C(=O)C(CC3CC3)CC3CC3)C2)C1 c1(C(=O)NCC2(O)CN(C(C(c3ccccc3)C)=O)C2)cccc(F)c1N C1(NC(C(N2CCNC2=O)C)=O)CC(NC(=O)C(C)(C)c2cnn(C)c2)CC1O c1(CC)ccc(C(=O)NC2(C3CCCN3C(c3cnc[nH]3)=O)CC2)c(C)n1 N1(C(C=CC=CCC)=O)CCC(CN(c2ncncc2C)C)CC1 c1(C(=O)OC)cc(S(=O)(=O)NCc2ccc(F)c(C#N)c2)c(C)cc1C C(=O)(C(CC(F)F)NC(C1CC(C)C1)=O)NCCC(C(=O)OC)O c1(C(=O)NC2CCC(CNC(C3C(C)=C3)=O)C2)cccc2nc(C)sc12 C12(CCOCC1)c1onc(n1)CCCN(C)C2C.c1(CO)ccccc1.C(C)(C)(C)N=O S(=O)(=O)(c1ccccc1)Nc1ccc(C(=O)NC(C)CNC(=O)C(C)(C)F)cc1 N#CC1(C(=O)NCC2CC(C(=O)NCc3cnccc3Cl)CO2)CCCO1 S(=O)(=O)(c1ccc2c(c1)CCC2)N1CCC2(CN(C(C3C(C)=CCC=C3)=O)C2)C1 N1(C(c2cn(-c3ncccn3)cn2)=O)CCC12CN(C(C1(O)CC1)=O)C2 Cc1ncc(CCC(N2CCSCC2CCNC(c2conc2C)=O)=O)c(O)n1 c1(C(N2CCCC(CNC(c3ccn(CC)n3)=O)CC2)=O)nn(C)c2c1CCC2 CCCC(C)(C)CC(=O)N(C1CCCN(C(c2sc(C)nc2C)=O)C1)CCO c1(OC)c(C(=O)NC(C)(C)CCNC(c2cnc(C(C)C)s2)=O)csc1Cl N1(C(C(CC)(C)COC)=O)CCN2CCN(C(=O)CCc3csnn3)CC2C1 c1(CN2C(C(=O)Nc3c(OC)ccc(Cl)c3)CC3CC32)ccc2cnn(C)c2c1 c1(C(=O)NCCN(CC(C)O)C(C2CC2F)=O)cnc(Cl)cc1N C=CC1CN(C(=O)C(O)C2CCCC2)CC1NC(=O)CC1CC2(CC2)C1 c1(C(N2C(C)CCC(NC(c3c(C)nn(C)c3C)=O)C2)=O)cc(Cl)c(F)cc1O N1(C(C(C)OC)=O)CC(CNC(c2ccc(Br)c(F)c2)=O)C(C)(C)C1 n1(CC)nnnc1C(c1cc(C)no1)NCc1nocc1C(C)(C)C c1(C(=O)NCC2(F)CCC(NC(c3cc(C)[nH]n3)=O)C2)cccc2c1CCC2=O c1(CNC2CCCC(C(=O)Nc3cnc(C(=O)OCC)s3)C2)c(Cl)cccc1Cl CCC(O)C(C)(C)C(=O)NC1C2CC(NC(=O)C(C)C(F)(F)F)CC12 N1(C(c2c(C(C)(C)C)con2)=O)CCC2CCN(C(=O)CC3CC34CC4)C2C1 Cc1cccn2cc(C(=O)NCCNC(c3csc(=N)[nH]3)c3ccccc3)nc12 O=C1OC2CC(C(=O)NCCC3CCCCN3C(c3ccc(F)cn3)=O)CC2O1 N1(CCc2cn(CCC3CC(CC)C3)nn2)CCC2(CC1)OCC(C)(C)CO2 N1(C(C(C(=O)OCC)CC)=O)CCCN(C(c2cn(C(C)(C)C)nn2)=O)CCC1 C=CCC(CNC(=O)C(C)NC(c1cccs1)=O)NC(c1ccco1)=O CCCC(CNC(C1(C#N)CCOCC1)=O)C(=O)NC1(C(O)COC)CC1 N12CC3C(C3C1)C2=O.C1(C(=O)OC)CC(F)(C2CCCN2C(C)C(=O)N(C)C)C1 N1(C(C(C2CCN(C(c3n[nH]c(C)c3C)=O)C2)F)=O)CC(F)(C2CC2)C1 c1(CC)nn(C)cc1CNC(C1CN(C(c2cncc(OC)n2)=O)CC1C)=O C(CC(C(C)C)NC(c1ccccc1SC)=O)N(C(C1(CC)CC1(F)F)=O)C c1(C(=O)NC(C(C)(C)NC(c2c(COC)nn[nH]2)=O)C)nn(C(F)F)cc1Cl C1(F)(CNC(c2ccc(C(F)F)o2)=O)CCCN(C(c2ccccn2)=O)C1 N1(C(CCC2CCC(C)NC2=O)=O)CC2CN(C34OCC(CF)(C3)C4)CC2C1 C(=O)(CCCC(=O)N1CCOCC(CNC(=O)CC(O)C2CC2)C1)N(CC)CC Cc1nc(CNC(c2cnn[nH]2)C)n[nH]1 CC1CN2CCN1CC2C(=O)NCCCN(C)C(c1ccoc1)=O C1(NC(C2N(C(CN(CC)CC)=O)CCCCC2)=O)CCn2ccnc2C1 c1(C(=O)NCCC(C)(CC)NC(C(CC)OC)=O)ccnc2c1CCO2 c1(C(=O)NC(C2CCN(C(c3scc(C)c3)=O)C2)C)sc2nccnc2c1N C1(C(=O)NCC(C(C)C)NC(=O)CC2CCCCC2)COCCC1(F)F N1(C(C(OCC)OCC(=O)NCC2CC(Cl)(Cl)C2)=O)CCC(OC)C1 C1(C(=O)NC2C3COCC23)C2CC(CC2F)N1C(C1(F)CCCCC1(F)F)=O C(CN=C(NCCC(=O)OC(C)(C)C)NCC1CCC(=O)N1)c1c(C)cccc1 N1(c2n(C)nnn2)CCC(C(N)=O)CC1.N12CCC(CC1)NC2=O c1(OC)cnccc1C(=O)NC1CN(C(c2ccnnc2O)=O)CC1O Cc1cc(C)c(C(=O)NC(C2CCCCC2)CNC(=O)CC2CC(C(F)F)C2)s1 N1(C(C(=O)N(C(Cc2c(OC)cccc2)C)C)=O)CCCCC(S(C)(=O)=O)C1 C(=O)(C(CC)CC)N1C(CCCSCCNC(C(C)OCC#C)=O)CCC1 c1(OCC(=O)NC23CCC2CN(C(C2CC4CC4C2)=O)C3)cccc(Cl)c1Cl c1(C2N(C(c3cc(Br)no3)C(=O)NC3CCC3)CCC2)ccc(F)cc1 c1(C(N2CCN(C)CC2CNC(=O)CC(F)(F)F)=O)ccc(=O)n2c1CCCC2 N1(C(C2N(C(c3cc(CC)oc3C)=O)CC(O)C2)=O)CCN(C2CC2)C(C)C1 c1(CNC(N(CCC)C2CC2)=O)ccc(Oc2cccc(C(F)(F)F)c2)nc1 C1(SC)COCC1N=c1nc2sccc2c(N(CCCNCC(C)(C)C)C)[nH]1 CC1CCCN(C(=O)Cc2ccn(C)n2)C1CCN=c1[nH]ncs1 C1(NC(C(C)=CC2CC2)=O)CC(NC(=O)Cc2sccc2C)CC1O C1(CNC(=O)C(F)CC2CC2)CC12CCN(C(c1ccccc1O)=O)CC2 c1(C(=O)NCC(C)N(C)Cc2ccccc2C(F)(F)F)cn2c(n1)COCC2 N1(CC)CC(C(N2CCC(O)(C(C)NC(=O)CCOC)CC2)=O)CCC1=O C1(OC)(CNC(C2COC3(CCC3)C2)=O)CCN(C(=O)C(C)(C)CC#N)CC1 c1(CNC(C(OC)OC)=O)nocc1C(=O)NC(CO)CCO Cc1c(C)c2c(c(C)c1O)CCC(C)(C(N1CCC(C(N)=O)CC13CC3)=O)O2 c1(C(=O)NCC2C(NC(CC(C)C)=O)CCC2)ccc(OC(F)(F)F)cc1 CC(C)C#CC(=O)NCCSCCn1cc(CCN(C)CCO)nn1 c1(C(N2CCN(C(C(CC=CCC)C)=O)C(CCO)C2)=O)cc([N+](=O)[O-])c(C)s1 C(CC(C)(C)CO)NC(C(C)CNC(c1ccc(Cl)s1)=O)=O C1(C(=O)NC(c2cccnc2)CC)CCN(C(=O)CN2CCCC2)C12CCC2 C(=O)(C(C)S(C)(=O)=O)NCCSCC(=O)NCC(C)CCN(C)C c1(C(=O)OC)cc(-n2cc(CNC(=O)CC3(C(=O)OC(C)C)CC3)nn2)ccn1 CC1CCC(Cc2nc(-c3ccccc3)no2)C1.N1(C)C(=O)N1C c1(C2(C(=O)N(CCNC(C(C)n3cncn3)=O)C)CC2)nocc1Br.C(C)(C)(C)O c1(C(=O)NC2C(C(N(CC(C)C)CCN(C)C)=O)CCC2)cc2cnccc2[nH]1 c1(COC(=O)CSCC#C)ccc(NC(=O)OC(C)(C)C)cc1 c1(C(=O)N(CC(=O)NCCN2CCCC(CCCCl)C2)CCO)cc(F)ccc1Cl c1ccc2c(c1)CC1(CC1)C2NCCc1ccco1 c1(C(N2CC(NC(C3(CCCC)CCCC3)=O)C3C2C3)=O)c(C)nn(C)c1C CC#CCC(C(=O)NCc1cccc(Cl)c1)NC(=O)Cc1ccc(C)s1 CC1(C)CCN(CCC(N2CCOC(c3ccncc3)C2)=O)C1 c1(C(N(OC)C)=O)c(ONC(=O)OCOC(C)(C)C)cnn1C Cc1nn(CC(=O)NC(CO)C(C)(C)C)c(C)c1C.c1(OCC(=O)O)ccccc1Cl C(CCCCC(=O)N1CCCC1CCC(N1CC2C(CO)C2C1)=O)OCC Cc1cc(C(N2CCCCC(CNC(=O)COC(C)C)C2)=O)ncc1CO C1(NC(C(=Cc2ccncc2)C)=O)CCC2CCN(c3cc(F)ncn3)C1C2 C1(O)(C(C)NC(=O)CC(C)C2CCCO2)CCN(C(C2(O)CCSC2)=O)CC1 N1(C(c2cn(C)nn2)=O)CCC(C)(CNC(C2C=CCS2)=O)C1 C1(C2CN(C(C3CC3[N+](=O)[O-])=O)C2)(NC(CCc2cccc(N(C)C)c2)=O)CC1 C1(C(N(CCC)CCNC(=O)CC2COC3CC2C3)=O)CSc2ccccc2O1 C(=O)(CCC(=O)N(C)CC1COCCN1C(=O)Cc1ccoc1)NCC C1(C(=O)NCC(C)=CC(N2CC(CN=[N+]=[N-])C2)=O)CC2CC(=O)C1C2 c1(CC(=O)NCC(C2CCOC2)NC(CC=C)=O)cnc(C)nc1O CC(O)CCCCCC(=O)N(CC(C)NC(=O)CCCC(N)=O)C c1(NC(C2CC(CSc3ccccc3)CN2)=O)ccc(C2CCOCC2)cc1F C1(CC)CCC(C(N2CCC(C)(C(=O)NCC(O)C(C)C)C2)=O)CC1 CC1OCCCC1C(=O)N(c1cnn(C)c1)CC1CC1 CC(N=c1nc(C2CCCC2)[nH]s1)C1CCN(C(=O)COCC(F)F)C1 C(CC(O)C(=O)N(C1CC(C(=O)NCC(C)(O)CO)C1)C)N(C)C C1(CCNC(c2c(C)nsc2Br)=O)CC(=O)NC1(C)C.C12CN(C1)C2=O c1(C(N(CCC(C(C)C)NC(C2CCCN2N=O)=O)C)=O)ccc([N+](=O)[O-])n1C Cc1cc(F)c2cc(C(N3CCC(C)C(CNC(=O)C=CCF)C3)=O)[nH]c2c1 c1(C(=O)NCc2c(C(=O)NC(C)C(C)n3cccn3)occ2)ccc([N+](=O)[O-])o1 C(=O)(C(CC(C)C)C(C)C)NCC(CC(C)C)NC(c1cc2c(nn1)CCC2)=O c1(-n2c(C(CCC)CC)nc(Cc3ccccc3OC)n2)ccc(C)c(F)c1 c1(C(CNC(=O)Cc2cnnn2C)NC(CC=C=C)=O)ccc(CN(C)C)cc1 Cc1cc(=O)c(C(=O)NC2CN(C(=O)C(C)n3cccn3)CCC2C)cn1C C1(C(=O)NCCC(C(C)C)O)CCC(C)(C)N(C(=O)COCCCF)C1 N1(C(c2ccc(CNC(C)=O)o2)=O)CCOCC1CNC(=O)COC(F)F CCCCC(C(=O)N1CCC(C)(C)C(C(=O)N(CC(OC(C)=O)OC)C)C1)C(C)C Cc1ncc2ccccc2c1C(=O)NCC1CN(C(C)C)C1 CCCS(=O)(=O)C(C)C(=O)NCC=C1CCN(C(=O)CCn2cc(Cl)cn2)CC1 C=CC(C(=O)NCC(CCC)NC(C1C(C)C1C)=O)OC c1(NC(=O)NC2C(C=C)CNC2)cc(C)nc(C)n1 CCC(F)(F)C(C)(C)C(=O)N(CC(C)(C)CNC(c1cc(C(=O)OC)cs1)=O)C c1(C(N2CCSC(C(N3CCc4ccsc4C3)=O)C2)=O)sc(Br)c2c1OCCO2 N1(C(C2(C)CCCC2)=O)CCC(NC(=O)CCc2ccc(O)nc2)C(F)(F)CC1 c1(C(=O)NCc2csc(-c3cc(Br)cs3)n2)ccc(OC2CC2)cc1 Cc1cc(C(=O)N(CC(C)O)CCNC(=O)Cn2cc(Cl)cn2)cc(C)c1Cl N1(C(C2C(C(C)O)C2)=O)C2CCC1CC(NC(=O)CCCn1ccnc1)C2 C(=O)(C1CCc2nccn21)N(C1CC(C)(C)C1)C1CC1.C1(=O)CN1 N1(CC(=O)N(CCC)CCC)CC2(CN(C(c3scnc3C)=O)CCO2)C1 C1(C(=O)NCc2c(CC)nc(C)s2)CC2CCN(C(=O)C(C)C3CCC3)CC12 C=CC(O)C(=O)NC(CCN(C(=O)C(CC)=CC)C)c1cccs1 CC1CN(C(=O)CC2CCSCC2)CC1NC(C1OCCC1Cn1ccnc1)=O c1(OC)cnc(F)c(C(=O)NCC(C)CN(C)C(C2(c3cc[nH]n3)CCC2)=O)c1 CCCCC(O)CC(=O)N(C)CC1(O)CCN(C(=O)CCc2cc(Cl)no2)C1 Cc1cnc(N2CCC=C(Cl)C2)c(S(=O)(=O)NC(C(C)C)C2CC2)c1 Cc1csc(C(=O)NC2CCCC2C(=O)NC(C)CN2CCCC2)c1 C(=O)(C(F)CC(C)(C)NC(C1CC(F)(F)C1(C)C)=O)N(C)C C1(n2cc(CCOC(CCSC)=O)nn2)CCN(Cc2ccc(Cl)cc2)CC1.C1CCC(C)N1 C12(C(=O)NC3CC(NC(C4(CC)CCOCC4)=O)C3)C3C4C1C1C2C3C41CO N1(C(C(CC)(C)O)=O)CCCC2(CC(NC(c3ccc(OC)c(C)c3)=O)C2)C1 C(=O)(CCC1=CCCCC1)N1C(CC(=O)NC2(C(=O)NC(C)C)CC2)CCC1 N1(C(c2cn(C)c(=O)cc2)=O)CC(NC(C2CC2(C)Br)=O)CC12CCOCC2 c1(C(N(C2CCN(C(=O)C(C)(C)OC(C)=O)C2)CCC)=O)ccnc2ncccc12 C=CCC(CC)C(=O)NCC(C)(C)NC(=O)CC(O)Cc1ccccc1 C1(O)(C(N(CCCN(C(c2c(CCC)n(C)nc2)=O)C)C)=O)CCCC(C)CC1 c1(NCC(COCCCC)O)ccccc1-c1ccccc1 c1(C(=O)NC2CCC(NC(Cc3c(C)noc3Cl)=O)CC2)cc(N)c(O)c(F)c1 N1(C(CCC2CC(N(C(C(C)C)=O)CC(C)C)C2)=O)CCCCCC1CO C(CN=c1[nH]c(=NCc2ncc(C)s2)[nH]c2ccsc12)N(CCO)CC C1(NC(C(n2ncc(C)c2)C)=O)CC(N=c2nc3[nH][nH]cc-3c(O)n2)C12CCC2 CCC(C)C(C)C(=O)NCCCN(C(=O)Cc1cncc(C#N)c1)C C(=O)(CCCCC(N)=O)NC(C(=O)Nc1ccc(C)c(C)c1)(C)CO c1(-c2ccc(OC)cc2)ccc(S(=O)(=O)OC2CC2)cc1C C(=O)(C(C)(O)C(C)C)NCC12CC(NC(Cc3c(C)ncs3)=O)(C1)C2 C1(NC(c2n(C(C)C)ncc2)=O)C2CCC1N(C(C1CC(=O)N(O)C1)=O)C2 N1(C(C(C(C)C)=O)=O)CCC(NC(C2CCC(=O)NC2)=O)C(F)C1 C(=O)(CC1OB(O)c2ccccc21)N1CC(C)(NC(C2CCc3nccn3C2)=O)C1 C(C)(CC1=CCCCC1)NC(C1(CC)CCN(C(C2C(=C)C2)=O)CC1)=O c1(C(N2CC(C#C)N(C(=O)C(O)CC)CC2)=O)cn(C)c2ccccc12 Cn1ncc(C#N)c1OC1CCN(C(N2CCC2C(=O)OCCCl)=O)C1 C1(CNC(c2cnc(OCC)s2)=O)CCCCC1NC(C1CCCN1C1CC1)=O c1(C(N2CC(NC(C3(CCC)CC3)=O)C3C2C3)=O)ccc([N+](=O)[O-])c(Cl)c1 CC1=C(c2ccc3ccn(CNCc4cc(C)c(Cl)c(C)c4)c3c2)CCCC1 C#Cc1cccc(C(=O)NC2CC(F)CN(C(=O)C(C)(C)C#N)C2)c1Cl N1(C(c2c(C(N)=O)coc2)=O)CC(NC(C2CN(S(=O)(=O)C(F)F)C2)=O)C2(CC2)C1 Cc1cc(C(=O)NCc2cncc(C(N3CC(C)C3CO)=O)c2)ccn1 C(=O)(C(CCC)C(C)C)NC(C(=O)NC(c1ccccc1)C#C)C(C)(C)O CCC(C)(F)C(=O)NC(c1cccc(Br)c1)CNC(C12CCC(C1)C2)=O C1(C(=O)NCC2CCC(C(=O)NCCC3(OC)CCC3)C2)CC2CC(=O)C1O2 N1(C(CCSCCC)=O)CCCC(COC)(NC(C2CC(=O)NC(C)C2)=O)C1 C1(C(=O)NC2CCN(C(CCC=CC(C)C)=O)C2)CCN(C(=O)CC2CC2)CC1 C1(C(=O)NC2CN(C(c3ccc(C)cc3N)=O)CC2O)Cc2cc(Cl)ccc2O1 S(=O)(=O)(c1cccc(Cl)c1F)N1C(C)(C(=O)Nc2c(C(=O)OC)cccc2)CC1 N1(C(C2(C)CCN(C(CC(C)C(F)F)=O)CC2)=O)CCC2(C1)CC2(F)F c1(COC)cc(=NCC(C)CNC(=O)CCCCCF)[nH]cn1 c1(C(=O)NC(CN(C)C(c2noc3ncccc23)=O)(C)C)cnc([N+](=O)[O-])n1C S(=O)(=O)(c1cccc(-c2ccsc2)c1)CN(C1(CCc2ccccc2F)CC1)C C(=O)(CC(C)(C)C(=O)N1CCCC2(NC(c3cc(C)no3)=O)CC2C1)OC c1(C(N(CC(C)O)CCNC(CC(C=C)C)=O)=O)cc(S(N)(=O)=O)cc(Cl)c1F Cc1noc(C)c1CC(=O)N(CCCNC(=O)COC1CCCCC1C)C O=C(CCC(CF)CF)NC1CC2(C1)CC2C(=O)NCCN1CC=CCC1 O(N1CCC(NC(C2(F)CCN(C(=O)C(C3CCCC3)OC)C2)=O)CC1)OCC N1(C(CSC(C)C)=O)CCN(C(C2OCCOC2(C)C)=O)CC1c1ccccc1 c1(NC(C(C)CNC(c2nc[nH]n2)=O)=O)ccc[n+]([O-])c1 N1(C(C2(OCC)CC2)=O)CCOC2(C1)CN(C(=O)C(F)(F)CO)C2 c1(NC(c2n(CCCC)nnn2)(C)CCC)cccc(C(OC)OC)c1 C(=O)(C(C)(CC)CCC(C)C)N1CCC(O)(CNC(C(C(CC)(C)C)O)=O)CC1 N1(C(c2scc(COC)c2)=O)CCN(C(=O)CC2(OC)CCC2)CC1C(C)(C)C C(=O)(CCCCCNC(N)=O)NCC1N(C(c2c(C)ocn2)=O)CCC1C c1(NC(C)=O)ccc(O)c(C(N2CC(NC(c3cncnc3C)=O)CC2C)=O)c1 C1(C(=O)NC2CCC(C(N3CCC3CCc3ccccc3)=O)C2)CCCCC1O c1(CCC)nc(=NC(CNC(C2CCSC2)=O)C2CC2)s[nH]1 O=C(C(O)CC(F)(F)F)N1C2CC1CN(C(C1(c3cc[nH]n3)CC1)=O)C2 C1(COC)CN(C(=O)C(Cn2ccnn2)NC(=O)C(C)CC2CCCO2)C1(C)C C1(C(=O)NC2CCN(C(c3ccns3)=O)C23CC3)CC12CCC(F)(F)CC2 c1(C(=O)Nc2cccc(CNC(CC3(COC)CC3)=O)c2)ccc(S(N)(=O)=O)o1 CC1(C)CC(C(N2CC(O)CC2CNC(C2CCC(C)(C)C2)=O)=O)CC(C)(C)O1 C1(CC(=O)NCC(COC)NC(c2nc(Cl)oc2C)=O)C(=O)NN=C1C Cc1cc(=O)n(C)cc1C(=O)NC(C)CC(C)NC(=O)CCCCNC(N)=O CC1(C)C(NC(=O)C(O)Cc2ccccc2)C1C(=O)NCC(N1CCCCC1)=O C(C(O)C(=O)N1CCCC1c1ncc[nH]1)N(C(C(C)c1ccsc1)=O)C1CCC1 C1(NC(CC2(C(=O)OC)CC2)=O)CCCCN(C(c2nc[nH]c2C(F)(F)F)=O)C1 c1(OC)cc(C(=O)OC(=O)C(C)C(=O)NCC)cc(F)c1.C1(C)CS1.C(C)(C)(C)O N1(C(C(C)n2cccn2)=O)CC2COCC2(C(=O)N(C)CC2COCCO2)C1 C(c1ccc(C)cn1)=CC(=O)NC1C(NC(CC(=O)OC)=O)COC1 c1(OCC(=O)N(CC(C)(C)NC(=O)CC2(C)CCOC2)C)ccc(F)cn1 c1(C(=O)NC(C=CC(=O)N(CCC)C)(C)C)cnc(O)o1 c1(NCCCCOC(=O)Sc2ccccc2-n2ccnc2)ccc([N+](=O)[O-])cc1 N1(C(C(C)SCC)=O)CCN(c2ccccc2CNC(=O)COCCF)CC1 C(CC(C(C)C)NC(=O)CC1CCC(=O)N1)N(C(C=C(C)C)=O)C c1(NC(C23C(CN(C(c4scc(C)c4Cl)=O)C2)C3)=O)cn(C)c(=O)nc1O c1(CC(=O)NC(C2OCCN(C(COCC#C)=O)C2)C)sc2ccccc2c1C c1(C(N2C(C)CC(NC(c3nonc3N)=O)CC2)=O)cc2ccccc2cc1F CCC(C(=O)NC1CC(CNC(=O)C(C)(C)Oc2ccccc2)C1)C(C)O CC1(C)CCCC(CC(=O)NC2CCCC2CNC(c2csc(C3CC3)n2)=O)C1 C12(NC(c3cccc(N)c3)=O)CCCC1CN(C(c1coc(Br)n1)=O)C2 C1(C(=O)NC(CNC(CN2CC(C)C2)=O)C)CCCN1c1ccccc1 C1(C(C)NC(c2ccc(Br)o2)=O)COCCN1C(c1ccc(OCF)cn1)=O c1(CC)c(Cl)nc(C)[nH]c1=NCC1CC(NC(c2c(C)cccc2Cl)=O)C1 C1(COC)(NC(c2nnc(S)n2C)=O)CCN(C(C2CCC2(OC)OC)=O)CC1 N1(C(c2ccc(CC)o2)=O)CCC(C)(C)C1C(=O)N(C)Cc1ncnn1C C1(C)(NC(c2ccc(C(C)=O)[nH]2)=O)CCN(C(=O)CCC(C)N(C)C)C1 C1(NC(c2nn(CC)nc2C)=O)CN(C(=O)C(F)n2cccn2)CC1S(C)(=O)=O c1(CCC)cc(C(N2CC(NC(=O)C(C)=C3CC3)C2)=O)cc(O)n1 C1(C(=O)OC(C)(C)C)CCCC1CNC(=O)NC(=O)CCCc1ccccn1 N1(C(C=CC)=O)CC(O)(C(F)CCCOCCOCC)C1.C12CC(C1)NC(=O)C2 C1(NC(c2nc(SC)sc2)=O)CN(C(C2C3(CC3)C23CC3)=O)CC1C C1(C(=O)NC(CC=C)CNC(=O)C=C(C)C(C)C)CCC(=O)N1C(C)C n1(CC(N2CCCC(F)(CNC(C=C(C)C)=O)C2)=O)ccc2c(C)cccc12 C1(CCCC)CCCN1C(=O)C(C1CC1)N(C)C(c1cscn1)=O c1(C2(C(N3CCn4nc(Br)nc4C3)=O)CC2)nccc2ccccc12 C=CCC(C)(C)CNC(=O)C(Cc1cc[nH]n1)NC(=O)C(CO)NC(N)=O N1(C(CNC(=O)NC23CCN(CC2)CC3)=O)CCc2ccccc2C1 N1(C(CN(CCC)C(c2n[nH]cc2C)=O)=O)CCC(F)(CC)C1 C1(C)(C(=O)Nc2c(C)nccc2)COC(C)CO1 C1(C(=O)NOCC(=O)N(C)C)(NC(C(C)C2CC2)=O)CC1(C)C CCCC(C(=O)N1CCN(C2CCC2)CC1)NC(C1CCCC(=O)N1)=O c1(OC)ncnc(OC)c1C(=O)NCC1CC2CN(C(=O)CC3CC34CC4)CC12 N1(C(CC(C(C)C)C)=O)CC2=C(C1)CN(C(C1CN(CP(C)(C)=O)C1)=O)C2 N1(C(C2=CC(O)C(C(C)(C)C)C2)=O)CCc2cc(Br)c(Br)cc2C1 N1(C(c2nc(OC)oc2)=O)CCN(C(C2CCCNC2=O)=O)C(C2CCCC2)C1 CCC(C)C(C)(O)CNC(C1CN(C(=O)CCC2OCCO2)CC1(C)C)=O C1(OC)CN(C(c2cc(C)sn2)=O)CC1NC(c1ccon1)=O C1(CNC(C(n2cc(-c3ccc(N(C)C)cc3)nn2)C)=O)CCC(C)(C)C1 n1(CC)ncc(C(=O)NCC2CC2CNC(=O)CCc2cccc(F)c2)c1C C1(CNC(=O)NCCCCCCC=C)(CF)CC12CCOCC2 c1(C(=O)NCC2CC3CN(C(CC=CC=C)=O)CC32)c(Cl)nc2sc(C)cn12 C1(c2c(C(C)=O)c[nH]n2)CCCN(C(=O)C(C)(C)Cc2ccccc2)C1 C1(CC)(NC(c2ccc(OC)nn2)=O)CCCN(C(C2CCCC23CCC3)=O)C1 C(=O)(CCC(F)(F)C(F)F)NC1(C)CC(NC(=O)C(C)(C)n2cnnn2)C1 C1(C(=O)NCC(C)(C)CNC(=O)Cc2cncnc2O)CC2(C1)CC1(CCC1)C2 C1(CCC)CN(C(c2ccc(C)nn2)=O)CC1C(=O)NOCc1cn(C)nn1 Cc1cc(C(N2CC3CC3(CNC(=O)C(C)(C)C)C2)=O)c(Br)s1 C1(NC(CCC(=O)N(C(C)C)C)=O)CCCN(C(=O)CC(F)(F)F)CCC1 N1(C(c2c(C)c(Br)no2)=O)CCC2C(C1)CN2C(C1CC2(C1)CC(C)C2)=O C1(CNC(c2cc(C)ncc2)=O)CCCN(C(c2cc[nH]c2)=O)CC1 C=CCC(C)C(=O)N1CCC(N2CCN(C(C3CCC3C(F)(F)F)=O)CC2)CC1 CCC(C)CCC(=O)NCC(O)CNC(c1csc(Br)c1)=O C(=O)(C1=Cc2cc(Cl)ccc2OC1)N1CCCN(C(COC)=O)C(CO)C1 C(=O)(C1c2ccccc2C(=O)N1C)NCC(C)CNC(=O)C#CC1CC1 c1(NCc2ccc(CNC(C3C(C(=O)OCC)C3)=O)o2)nccnc1O CC(C)(C(=O)N1CCCC(CNC(C2(C(O)C(F)(F)F)CCC2)=O)C1)S(C)(=O)=O C(=O)(C(N=[N+]=[N-])C(C)C)NC(CN(C(C1CC2OC1C1CC21)=O)CC)C c1(C(N2CCC(n3ccnn3)C2)C(=O)NCC=C)ccc(Cl)c(Br)c1F CC(C)CC(C)(O)C(=O)NC1CCCC1NC(=O)CCc1cnn(C)c1 C1(NC(=O)CCc2nncs2)CCOC(C(=O)NCC2CCC2)C1 N1(C(C2CN(CC)C(=O)C2)=O)CC(NC(=O)CSCC(F)F)C(C2CC2)C1 c1(C(C)C)nc(N2CCCC3(NC(=O)CSC(F)(F)F)CC3C2)c2cc[nH]c2n1 C1(CC=C)(NC(c2ccccn2)=O)CCN(C(c2cnsn2)=O)C1 c1(OC)cc(CNC(c2cccnc2)c2nc[nH]n2)ccc1Br c1(C(=O)NC2CN(C(CCCC=C)=O)CC2CC)nc(C)ncc1Cl C(C1CCCCCC1)=CC(=O)NCC(CNC(Cc1c(C)noc1C)=O)C N1(c2[nH]c(=NCc3nn(C)c(Br)n3)[nH]c(=N)n2)CCc2[nH]c(=N)nc(O)c2C1 C1(NC(COC)=O)CCCC(CNC(C2CC(Sc3ccccc3)C2)=O)C1 Cc1ccc(CC(N2CC(NC(=O)CC(C)c3cccnc3)C(O)C2)=O)cc1C c1(CC)sccc1C(=O)NCCCN(C(=O)CC1(C)CC1(Cl)Cl)CC c1(OC(C)C)ccc(Cl)cc1.N12CC3(CC1C3)NC(=O)C=CCOC1(CC1)C2=O CC1=C(C(=O)NC2CN(C(c3ccc(C(N)=O)[nH]3)=O)CC2(C)C)CCC1 c1(C(=O)NCC2C(C)CN(C(=O)CC(C)(F)F)C2)ccnc2[nH]cnc12 N1(C(CC2N(CC)CCC2)=O)CCOCC1CN(C(=O)CNC(=O)CC)C c1(C(=O)NCC(C)(CNC(=O)C(c2ccn(C)n2)C)OC)cncc(C(=O)OC)n1 c1(C(N2CCC(C(=O)NC(c3ncc(C)[nH]3)CC)C2)CC)cn2ccsc2n1 Cc1c(C(N2CC3CN(C(c4cc(C)n(C)n4)=O)CCC23)=O)cc(F)cc1Br c1(C(=O)NCC2(NC(c3ccc(O)c(F)c3)=O)CCC2)cnc2[nH]cncc1-2 Cc1cc(C(=O)N(C(CC(F)F)C(=O)N(C)C)C)ccc1F C1(NC(CC2CC(=C)C2)=O)CCCC(NC(=O)C(c2cccc(C)c2)O)C1 c1(C(=O)NC(CCN(C(C(CCC)OC)=O)C)C)c(OC)cccc1OC N1(C(C(=O)N(CC(=C)C)CC)C)CCC(N(CCC)C(c2occc2C)=O)C1 CC(C)CC(O)CC(=O)N1CCC(O)(CNC(=O)C(F)=CCCF)C1 c1(NC(C2CCC(NCc3c(Cl)ccc(C)c3F)C2)=O)c(Cl)cc(Br)c(Cl)c1Br Cc1c(C(=O)NCC2CN(C(=O)C3=CC(C)CC3)C2)[nH]c2ccccc12 c1(C(=O)NC2CN(C(CC(C)(C)OC)=O)C(C)C2)c(N)c(F)cc(F)c1F CC1(C)CC=C(C(=O)NCc2csc(C(=O)NC3CC3c3ccsc3)c2)CC1 C1(NC(=NC)NCc2ccccc2)CCC(C(C)C)CC1 c1(CCC(=O)NC2(C)CCN(C(C3CC3c3ccco3)=O)C2)ccc(C#N)cc1 N1(c2c(NC(COCCOCC)=O)cno2)CCCC1CC(=O)NCC c1(C(=O)NC2COCCC2NC(C23CCCC2C3)=O)ccc(Cl)cc1F C(CC(C)C(=O)N1CCC(C(=O)NC2(C(F)F)CCC2)C1)=CCC CC(C)CC(C(=O)NCC1CC1N=[N+]=[N-])N1CCCCC1=O C(=O)(C(C)(C)C(C)(F)F)N(CCNC(c1snc(-c2ccccc2)c1N)=O)CC Cc1c(C(N2CC3CCN(C(C4COC(=O)N4)=O)CC23)=O)sc2[nH]cnc(=O)c12 c1(CC(C(=O)C(C)C)O)cccc(Cl)c1.C12(CC1)C(=O)N(C(C)C)CCN2 C1(C(N(CCN(C(C(C(CC)C)O)=O)C(C)C)C)=O)COc2cc(F)ccc2O1 N1(C(CC(CC)SC)=O)CC(NC(c2cnc(O)cc2C)=O)CC1(CC)CC C(CC(C(C)C)NC(C1(C(F)(F)F)CC(F)(F)C1)=O)N(C(C(C=CC)O)=O)C C1(CNC(CC=CC=C)=O)C(C)CCN1C(=O)CCCNC(N)=O Cc1[nH]c2ccc(CNC(=O)C(N3CC4CC5CC4C3C5)=O)cc2c1C C1(NC(C2(OC)CCC2)=O)CCCCCN(C(=O)Cc2cnns2)C1 N1(C(CCCCCSC)=O)CCCC2(CCCCC2NC(=O)CNC2CCC2)C1 C(=O)(CC(C(C)C)C(C)C)NCC1(C)C(C)CN(C(C(C(C)C)NC(C)=O)=O)C1 CCCCCC(CC)C(=O)NCC1CN(CC2CCS(=O)(=O)C2)CCC1(F)F C1(O)(CNC(CCCOC)=O)CCCN(C(=O)Cc2ccn(CC(F)(F)F)n2)C1 N1(C(c2cc(C3(OC)CC3)cc(F)c2)=O)CCCC2CN(C(C34CCC3C4)=O)CC12 C1(C(=O)NC(C2CN(C(c3cc(C4CC4)ns3)=O)C2)C)OCCN(C)C1=O c1(SC)cc(C)c(C(=O)NC2CC2NC(c2cc(-c3ccccc3F)no2)=O)o1 Cc1sc2ncc(C(=O)NC3CC(F)CN(C(C4CCOC4=O)=O)C3)n2c1C N1(C(C(n2c(C)ncc2)C)=O)CC(C)(C)CC1C(=O)NC1CCSC1C N1(C(CNC(c2c(C)con2)=O)=O)CCCCC1CCC(N1CCOCC1)=O N1(C(CN(C2CCC2)C)=O)CC2(CCCC2NC(C2CCC(N(C)C)CC2)=O)C1 C1(N(C(=O)C=Cc2cncn2C)CC)CCC(NC(=O)C(F)OC(F)(F)F)CC1 Cc1nc(C)c(C(=O)NC2(CO)CCN(C(=O)C(O)Cc3[nH]cnc3C)C2)o1 c1(C(N2C(C)(CNC(C3(O)CCOCC3)=O)CCC2)=O)cc(F)cc(F)c1O N1(C(CSCC=C)=O)CC(NC(c2ccc(F)cn2)=O)C(C)C1 N1(C(c2n(C)ncc2)=O)CCC(CO)(NC(=O)Cc2cnoc2)C1 C1(C2CN(C(C3CCNC(=O)C3)=O)C2)(NC(C(c2c(C)n[nH]c2C)C)=O)CC1 CCC(CC(=O)NC1CN(C(=O)Cc2ccoc2C)CC1OC)SC Cc1cn(CC(=O)N(C2CCN(C(=O)C(O)C(C)C)C2)C)nc1C(F)(F)F C(=O)(CS(N)(=O)=O)N(C(C)CNC(C1(CF)CCC1)=O)CC N1(C(c2c(CNC(c3nccc(C)c3N)=O)ocn2)=O)CCC12CCN(C)C2 c1(C(=O)NCCN(C(CSCCCC)=O)C2CC2)oncc1C c1(C(=O)NCC(CO)NC(c2c(C)nc(CO)o2)=O)cc(C(N)=O)ccc1F S(=O)(=O)(CC(=O)NCc1ccccc1F)N1CC(C(C)(C)O)(Cc2cccs2)C1 c1(C(N(CCCNC(=O)C(O)CC(F)(F)F)C)=O)ccc2nc(S)oc2c1 CC#CCCCC(=O)NC(COCC)C(=O)NCC1(CC)CCOC1 c1(C(N(C(C)C)CCN(C(=O)CC2(C)CC2F)C)=O)cnc(O)c(C(F)(F)F)c1 C1(C(=O)NC2CN(C(CCC#N)=O)C3(C2)CCC3)CCc2nnc(O)cc2C1 CC(C)C#CC(=O)N1CC(O)CC1CNC(c1cc(Cl)ccn1)=O CCC(C)CCCC(=O)NCC(=O)NCC(=O)N(C)Cc1csc(C)n1 c1(NCCN(C(C(CC)OCC)=O)CC)cc(C)ncc1C#N N1(c2n(CC=C)c(CC(c3ccc(Cl)cc3)(C)O)nn2)CCC2(CCC(=O)N2)C1 N1(C(c2nn(CC)c(C)c2)=O)CCN(C(c2ccnc(Br)c2)=O)C2CC12 c1(C(=O)NCC2CC(NC(C3(CCC)CC3)=O)C2)cnn2c1OCC(O)C2 Cc1ncc(Cl)cc1NC(C1CC(O)CN1C(c1cnon1)=O)=O c1(C(=O)NCC2CC(CNC(CC=C)=O)OC2)ccc(C(F)F)nc1 C=CCC(C)(O)C(=O)N1CCC(C(=O)NCCC2(OCC)CCC2)C1 c1(C(=O)NC)ccc(C(c2nnnn2C)NC(c2ccncc2)c2cccs2)cc1 C1(CNC(c2c(C)n(C)nn2)=O)COC(C)(C)CN1C(=O)C(C1CC1)N(C)C CC1(C)CC(CNC(C2(C)C(C)(C)C2(C)C)=O)N(C(=O)CN2CCOCC2)C1 C(=O)(C(C)CC(=O)NC1CCCC1C(=O)NC1(C)CCC(C)(C)C1)OC C(=O)(C1=CC2C=CC1C2)N(C1CCCN(C(Cc2ccn(C)n2)=O)C1)CCO N1(C(C(CC)C)C(=O)NC2CC(F)(F)C2)CCC=C(c2ccccc2O)C1 c1(C(=O)NCC(C)NC(C(c2ccccc2)NC(C)=O)=O)cc2c(ccn2C)s1 Cc1cc(C(N2CCN(C(c3ccccc3)=O)C3CC23)=O)cc(C)c1 c1(C(=O)NCCN(C(=O)CCC2CCCN2C)C)ccc2ncnn2n1 c1(C(=O)OC)cc(C)c(F)c(S(=O)(=O)N2CCC(C)CC2C(N)=O)c1 N1(C(C(c2ccccc2)OC)=O)CCCC(C)C1CNC(C1COC(=O)O1)=O c1(C(=O)NCC2CC(NC(CSCC)=O)C2)cn(C)nc1C c1(CNC(c2c(CC)cno2)=O)nnc2n1CCN(C(=O)CCC(O)C(C)(C)C)C2 N1(C(C(C(C)C)C)=O)C2CCC1CN(C(=O)CCc1nnc(S)nc1O)C2 N1(c2nc(C)nc(O)c2)CC(NC(C2(OC(C)C)CCC2)=O)CC(C)(C)C1 N1(C(CCCSC)=O)CC2CCN(C(c3cccc(-c4ccncc4)c3)=O)C2C1 c1(CNC(C2C(C(=O)OC)C2)=O)ncoc1C1CN(C(=O)Cc2cscn2)C1 CC1CCCn2ncc(C(=O)NCCC(C)CCNC(=O)CC3CC3)c21 N1(C(CC(=O)NCC)=O)CCCC(F)(C(=O)NC(CC2CC2)C(=O)NC)C1 C12(CNC(c3c(C(C)C)ccs3)=O)CN(C(C3(C#N)CCC3)=O)CC1CCO2 CCCCC(C)(F)C(=O)N(C)CC1CCCN(C(c2nscc2C)=O)C1 c1(CC(=O)NC2CC(NC(CCc3cc(C)no3)=O)C2)ccc(C)c(Cl)c1 c1(C(=O)NC(C(C)(C)C)CNC(c2c[nH]c(=N)nc2O)=O)cccc2sncc12 C(=O)(C1=Cc2cc(Cl)ccc2OC1)NC1CN(C(C(F)=CCC)=O)C2C1C2 C#CC1COCCN1C(=O)CCn1cc(C(C)(C)CCN2CCN(C)CC2)nn1 N1(C(CC(=C)C)=O)CCC(C(C(C)C)NC(c2cc(OC)n[nH]2)=O)CC1 C1(CC(=O)N(C(CC(CC)C)C)C)CC2(C1)CN(C(c1c[nH]nc1C(F)F)=O)C2 N1(C(CNC(=O)OCC)=O)CC(=O)NCC1C(=O)NCC1CC2CCC(C1)C2 c1(NC(=O)COCCCF)ccccc1NC(=O)COC(=O)Cc1cccc(F)c1 C1(CCOC)(C(=O)NC(C)C(O)C(C)C)CCN(C(=O)Cn2cnnc2O)CC1 Cc1c(O)cc(C(=O)Nc2cccc(C(=O)NC3CCCCC3)c2)cc1O C(C(C)CCC)(c1nnnn1C(C)C)NC(CC)(C)CC C#Cc1nc(C(=O)NCCC(C)N(C)C(C2CCOC2=O)=O)cs1 C(CCC(N)=O)(C(=O)N1CCC(NC(C)=O)CC1)OC(c1ccoc1CF)=O CC(C)CC(F)C(=O)NC1CN(C(c2ccc(O)c(C(C)(C)C)c2)=O)C(C)(C)C1 C1(C(=O)NCCC(C)N(C(=O)CC(C)(F)F)C)CN(C(N)=O)CCO1 CC1CC(CNC(=O)CCC2CCOCC2)CCN1C(c1cc(Cl)n(C)n1)=O C1(NC(CCN(CCCCC)C)=O)C=CC(CNC(=O)C(C2CC2)OC)C1 Cc1c(C(N)=O)cccc1C(N1CCC(NC(=O)Cc2cc(F)cc(F)c2)C1)=O C(=O)(C1CCc2nccn21)N1CC2(CCC(CNC(=O)Cc3ccccc3)O2)C1 CCC(C(=O)NCC1(CCNC(=O)C=C2CCC(C)C2)CC1)C1CCOCC1 C1(OCC)CC2CN(C(C3C(C)CN3C(=O)CC3CC=CC3)=O)CC12 C1(CC=C)(NC(C2CCCN2C)=O)CCN(C(=O)C(C)S(C)(=O)=O)CC1 n1(CC(=O)NCC2N(C(c3n(CC=C)ccc3)=O)CC2)nc(C2CC2)n(C)c1=O n1(CCCC)cc(C(=O)NCC(C)NC(c2cscc2CC)=O)nn1 Cc1nc(C)c(C(N2CCCOC(CCNC(C3COC(=O)C3)=O)C2)=O)c(C)n1 C(=O)(C1CCc2ccc(Cl)nc21)NC1CN(C(c2ccc3ccn(C)c3c2)=O)C1 C1(C#N)(C(=O)NC(CN(C(C(CCC)N(C)C)=O)C)C)CCSCC1 n1(SCC)cc(CNC(=O)CCN(C)C(C2CCN2C)=O)nn1 c1(C(=O)NC2CN(C(CC(=C)C)=O)C(C)CC2)cnc2n(c1=O)CCS2 c1(C(=O)OC)ccc(C(=O)NC(CO)C(C)NC(=O)Cc2ccsc2C)o1 C(=O)(C(=O)C(C)(C)C)N1CCC(OCCNC(c2c(CC)cns2)=O)C1 CCC(C)CCCC(=O)NCCCC1(NC(=O)C#CC2CCC2)CC1 C1(C)(CNC(Cc2scc(CC)n2)=O)CCCN(C(c2ccc(O)cn2)=O)C1 C1(NC(C(C(C)C)O)=O)CC2CCCC(C1)N2C(=O)C=CC1CC1 c1(C(=O)NCC2C3CN(C(c4c(CC)noc4C)=O)CC32)ccc(C)c(F)c1N C1(C)(C(=O)NC(c2nccn2C)CC)CCCN(CS(=O)(=O)N2CCCCC2)C1 c1(NC(C=CC2N(C(CCCC)=O)CCC2)=O)c(OC)cccc1O c1(C(C)(C)NC(=O)COc2ccncc2)ccc(O)cc1F C1(C(N(CCOCC)C)=O)(COC)C=CCN1C(c1c[nH]nc1Cl)=O C1(C(=O)OC)C(C)CCN1C(c1cccc(-c2nc(=O)o[nH]2)c1)=O N1(C(CCCN(C(=O)OC)C)=O)CCC2CN(C(=O)C=CS(C)=O)CC2C1 Cc1noc(C)c1S(=O)(=O)Nc1ccc(CNC(C2CC(C)CN2)=O)cc1 c1(OC)ccc(C(N2CCCC(C3CCCN3C(c3cc(F)c[nH]3)=O)C2)=O)cn1 CC1CC(NC(C2CCC(=O)N2C)=O)N(Cc2cccc(-c3ccccn3)n2)C1 Cc1cc2c(CC(=O)NCC(CNC(c3cnc[nH]c3=N)=O)CO)csc2s1 N1(C(C=C(C)C(F)F)=O)CCN(C(C2(C(C)C)CCC2)=O)CC1CC1CC1 N1(Cc2n(CC)ccc2)CCC(C(=O)NOCCOC(C)C)C(O)C1 N1(C(=O)NCC2CCCN(CC)C2)CCc2cc(C#N)ccc2C1 N1(C(C(=O)N(CC(F)Cl)CC)=O)CCCC1(C)C N1(C(CC(=O)OCC)=O)CC2CCCC(NC(=O)C=C3CCCC3)C2C1 C1(N(C(C2CC(=C)C2)=O)C)CCN(C(=O)CSc2cnn(C)c2)C1 c1(CC)cnc(Cl)nc1N1CCC(F)(CNC(=O)Cc2c(C)nn(C)c2C)CC1 N1(C(C(C(=C)Cl)(C)C)=O)CC(C2CCN(C(c3cc(O)ncn3)=O)CC2)C1 c1(C(CNC(c2cccc(N)c2)=O)NC(C2(SCC)CC2)=O)ccc(F)cc1F C1(C(N(CC(CNC(CC=CC)=O)C)C)=O)CC(=O)N(C(C)(C)C)C1 Cc1nn(C)c2nc(C(=O)NCC(F)CNC(=O)C(C)(O)C(C)(C)C)cc(O)c12 N1(C(c2c(C)n(CC(F)F)nc2)=O)CCC(C)(NC(C2CNC(=O)N2C)=O)CC1 Cc1nc(C(=O)NCCC(C)N(C)C(C2CCOC2(C)C)=O)sc1C c1(SC)nn(C)cc1C(=O)NC1(C)CC(NC(=O)Cc2ncc(C)s2)C1 C1(C(=O)NC2C(NC(C34CC(C(C)C)(C3)C4)=O)CC2)CC2CCC(C1)O2 CN(C)S(=O)(=O)N1CCC(N2CCC(OC(=O)C(C)(C)c3cccs3)C2=O)CC1 N1(C(c2n(C)c(Cl)nc2Cl)C(=O)NCCC2CC2)CC2COC(C)(C)OCC2C1 S(=O)(=O)(c1ccc(NCc2sncc2Br)c(C#N)c1)NC(C)CC1CCCC1 c1(C(=O)NC2(C)CN(C(=O)C=Cc3ncco3)C2)cc(C#N)c(F)cc1F CCCC(C#N)C(=O)NCC1CC(NC(c2nc(Br)sc2C)=O)CCO1 C12(C(N(CCCNC(c3c(OC)cc(O)nc3)=O)C)=O)OCCCC1C2(F)F c1(OC)cccc(Cl)c1C(=O)NCC1(C)CCCN(C(=O)CCN(C)C(C)=O)C1 N1(S(C(CC(C)C)c2ccccc2)(=O)=O)CC23CCCC2(COC3)C1 C1(NC(=O)C=C(C2CC2)C2CC2)CC1C1CCCN(C(=O)Cn2cc(Cl)cn2)C1 C1(NC(c2c[nH]nc2F)=O)CN(C(c2ccc(=O)n(CCF)n2)=O)CCC1CO C(CC(O)C(=O)N1CCC(NC(=O)C(F)CC2CCOCC2)CC1)SC c1(C(=O)NC2CN(C(c3c(SC)csc3)=O)CC2C)noc2c1CCCC2 c1(CC(=O)NC2CC(CCNC(c3[nH]cc(C)c3)=O)C2)ccc2c(c1)CCCO2 C#Cc1ccc(-c2cnc(C(=O)NCCCCO)c(C(F)(F)F)c2)cc1 Nc1ccc2nc(C(=O)NCCc3ncccc3F)ccc2c1 C1(CNC(c2cccc(N(C)C)c2)=O)CCN(C(c2snc(C)c2N)=O)C(C)C1 C1(NC(C(C)N(C)C)=O)CCCC(NC(c2ncccc2-c2ccccn2)=O)C1 N1(C(C)C)CCC(CC(=O)NC2CC(C)(NC(=O)CC3CCC(=O)N3C)C2)CC1 n1(CC)ncc(NC(=O)N(C)CCc2ccccc2-c2nn[nH]n2)c1C(F)(F)F C1(CCNC(c2c(CC)cno2)=O)COCCN1C(c1cc(C)sn1)=O c1(OCCN(C)C)ccccc1NC(N1CC(c2ncc(Br)cn2)(O)C1)=O C(CCCC(=O)NC1CCC(NC(c2ccoc2)=O)CC1)NC(=O)OCC=C C(=O)(C1=C(C#N)CCC1)N1CCC(C(C(=O)NCC2(C(=O)OC)CC2)F)C1 c1(C(N2CC3C(NC(C4(CO)CC4(F)F)=O)C3C2)=O)ccc(NC2CCC2)cc1 C=CC1CCN(C(C2(O)CCN(C(c3ccnc(C(C)C)c3)=O)C2)=O)C1 C1(C(=O)NCC(c2ccccc2)C)COC2CN(C(=O)C(O)c3ccco3)CC12 Cc1ccc2ncc(C(N3CC4(CCN(C(=O)CCC(C)(C)O)CC4)C3)=O)n2c1 CC(C)C(CC(=O)N(C)CCN1CCOCC1)NC(C1CCOC1(C)C)=O C1(NC(CC)=O)CCN(C(=O)C(c2ccc(Cl)cc2)=O)CC12CCC2 C1(CC(=O)NCCCN(C(=O)C=C2CCOCC2)C)COC(C)(C)CO1 C(=O)(C1CCCc2nccn21)NCCCN(C(C(COC)C)=O)C(C)C C1(NC(C2C(C)(C)C2)=O)CC(NC(C2(n3cc(Cl)cn3)CC2)=O)C(O)C1 C(C(=O)NCCCC1CCCN1C(c1cc(C#N)cn1C)=O)(C(C)(C)C)SC c1(C(CC)NC(=O)C(=O)N(C2CCCC2)C(C)C)cccc(C)n1 C1(NC(CCSC)=O)CN(C(=O)C(C)Oc2cccc(CO)c2)C(C)(C)C1 Cc1ccc(C)c(CCCC(=O)N2CCCC2c2cn(-c3cccnc3F)nn2)c1 C(=O)(CCCC(C)(C)NC(=O)CC1(NC(C)=O)CC1)NCC1(CC)CCCCC1 c1(-c2ncn(C)n2)ccccc1C(=O)NCCC1CN(C(=O)C2=CCC2)CCO1 N1(CC)CCCN(C(C2CCN2C(c2ccccc2NS(C)(=O)=O)=O)=O)CC1 CCC(Cc1ccccc1OC)N=c1[nH]c2c(c(=NC(C)CCCO)[nH]1)CCC2 O=C(C1=CCOC1)NCCCOCCNC(C1CCS(=O)(=O)N1)=O C1(C(=O)Nc2c(C)cccc2)CCC(C)N(C(=O)C(C)Nc2ccccn2)C1 CN1CCN(C(=O)Cc2cnn(C)c2)CC1C(=O)NCc1cc(C(N)=O)no1 C1(CC)CCCC(N=c2[nH]c3c(c(=NC4CCN(C(=O)CC)CC4)[nH]2)CC3)C1 c1(C(=O)NC23CC(C2)N(C(=O)CSCC2CCCO2)C3)cn2c(n1)CCCC2 C(CCO)(C(F)(F)F)NC(C1CC(C)N1C(=O)CNC(=O)C1CC1)=O CC(C)(C)CCC(F)C(=O)N1CC2CC1C2C(N1CCC(N2CCCC2)C1)=O CCCC(CCC)C(=O)NCC1CCN(C(=O)Cc2ccc(N)cc2)C1(C)C N1(C(CC2(OCC)CCCC2)=O)CC(NC(C2C3CCC2CC3)=O)CC1CO N1(C(C2C(NC(c3c(C)nsc3)=O)CCC2)=O)CCC(C)(CO)C(O)C1 c1(C(=O)NC2CC(NC(C3N(C)C(=O)CC3)=O)C2)ccc(Cl)c(Br)c1F N1(C(CCC2(C)CCN(C(Cc3n(C)cnc3)=O)C2)=O)Cc2cncnc2C1 c1(C(=O)NCCC2(NC(C3CCC(C)NC3=O)=O)CCC2)ccc2nnnn2c1 c1(C(C(=O)NC(C(=O)OC)C)N(C2CC2)CC2CC2C)cc(C2CCC2)on1 c1(CNC(C2N(C(CN(CCC#C)C)=O)CC=C2)=O)ccccc1F c1(C(C)=O)ccc(C(=O)NC2CCCN(C(C3CCCSC3)=O)C2)cc1 c1(C(=O)NCCOCCNC(CC(c2scc(C)c2)O)=O)nc(C(C)C)oc1C CC(C)C(C(=O)NCCC(C)CCNC(c1cccnc1OCCO)=O)C(C)C CC1OC2CCC1(C(=O)NCCOCCC(=O)N(C1CCOC(C)C1)C)C2 N1(C(c2cn(C)nc2C)C(=O)NCCCC(=O)OCC)CCOC(C)(C(F)F)C1 N(C1CCCc2cccnc21)(C(COCCOC)C)Cc1ccccc1 c1(C(=O)NC2CC(C)N(C(c3cnn(CC(F)(F)F)c3)=O)C2)cnc(O)c(Cl)c1 CC1C(NC(=O)CN2CCC(O)CC2)CCN1C.c12cc(ccn1)-n1cc-2nn1 Cc1oc2cc(C(=O)NCCCC(C)NC(=O)CC(C)n3ccnc3)[nH]c2c1C c1(N2CC(C)NC(=O)C2)nc(N2CCCC(CC(F)F)C2)c2c(n1)CCCCC2 c1(C(N(C(C)C(=O)NCC(CC)(CC)C(N)=O)CC)=O)c[nH]c2ncccc12 N1(C(C2(CC)CCOC2)=O)CCN(C(=O)C=Cc2cn(C)nn2)CC1C Cc1ccn(CC(C)C(=O)NC2(CNC(=O)CCc3ccc[nH]3)CCOC2)n1 C1(NC(C2CC2C2CC2)=O)CN(C(=O)Cc2cscn2)Cc2nccn2C1 C#CCC(CC(F)F)C(=O)NCC(C)(CC)C(=O)NC(C)CCN1CCCC1 C#CCC(CC#C)C(=O)NC1CC1CNC(=O)Cc1cccc(OCC#N)c1 CC1CN(C(c2cccnn2)=O)CCCN1C(c1cccc(C2CCOC2)c1)=O c1(C(=O)NC(CCC)CCCNC(=O)CC(C)(C)O)scc2c1OCCO2 C1(CNC(CCN(CCC(C)(C)C)C)=O)CCC(F)(CNC(C2CC23CC3)=O)CC1 C1(C2CC2)(C(=O)OCC)CCN(c2c(F)cccc2C#N)C1 C(=O)(C(C)CC(C)(F)F)NCCC(C)NC(C1C2CN(C)CC12)=O C1(CNC(=O)CC2COCC2O)CC(C(=O)N2CCCN(C3CC3)CC2)=NO1 c1(CCC(=O)NC2CCCN(C(c3cncc(C(N)=O)c3)=O)C2)cccc(F)c1 C(=O)(CNC(=O)CN(C(C1CC1C(C)(F)F)=O)C1CC1)NC(C)C C1(CC)OCCCC1C(=O)NCCCCN(C(=O)COc1ccc(Cl)cc1)C C(O)(CNC(=O)CNC1CNCCC1(C)C)(C(F)(F)F)c1ncc(C)o1 N1(C(=O)CCN(C(C2CCC(F)(F)C2)=O)C2CC2)CCC12CCCSC2 C1(NC(C(C)OC)=O)CN(C(c2cc(C(F)(F)F)ncc2N)=O)C(C)(C)C1 c1(OC)ccc2cnc(N3CC(NCc4ccc(Br)c(C#N)c4)C(C)C3)nc2c1 C1(NC(CC2CCN(C)CC2)=O)CN(C(=O)CC2CCN(C)C2=O)CCN1C c1(C(=O)NC2CCN(C(Cc3cc(CC)no3)=O)C23CC3)cc2ccccn2c1 C=CC1(C(N2CC(OC)C2)=O)CCN(C(=O)C(F)=CC)CC1 CCC(CNC(=O)C(O)C(C)SC)(CC)NC(c1cnn(C)c1C)=O c1(C(=O)NC2C(CC)CN(C(=O)C(C)(C)O)C2)cccc2c1CCCC2 CCN(OC)C(=O)CNC(=O)C=CC(C)(C)NC(C1CN(C)CCN1C)=O N1(C(CNC(C(CC)C)=O)=O)CC(C(=O)NCc2cnc(C)cn2)C2(CC2)C1 Cc1c(C(N2CC(CNC(=O)C(C)(C)N(C)C)CCC2C)=O)oc2ccccc12 C1(NC(c2cnccn2)=O)CC12CCC(NC(C1CN3CCC1CC3)=O)CC2 C1(C(=O)NCC2(C(C)NC(C3CN(CC(C)C)C3)=O)CC2)CCC(=O)N1 C1(CC(N2CC(CNC(CC3CC(=C)C3)=O)C2)=O)COCC(C)O1 CC(C)CC(C(=O)N1CCOCC1CCO)N(C(=O)C(=O)NCC(F)F)C CC(C)(C)CC(O)C(=O)N1CCCC(CNC(c2ccn3c2CCCC3)=O)CC1 c1(C(N2C(CN(C)C(C3(F)CCOC3)=O)CCC2)=O)cncc(Cl)c1Cl c1(C(N2CC3(C(C(=O)Nc4c(OCC)ncnc4)C3)C2)=O)cc(Br)ccc1F C(c1cccc([N+](=O)[O-])c1)=CCC(C)(C)NC(=O)NCC1N(C)C(C)(C)CC1 N1(C(c2c(CC)n[nH]c2)=O)CC(C2CC2C(=O)NC(C)(COC)CC)C1 C1(NC(CNC(CCCCC)=O)=O)CC2(CCN(C(=O)C(C)(C)C3CCC3)C2)C1 CCC(C)(C)C(C)CC(=O)N(C1CCC(NC(=O)C(C2CCCCC2)O)CC1)C C1(NC(c2cnoc2)=O)CCCC2CN(C(=O)C3=COCCO3)CC12 C1(CC(=O)NCC(C)(C)NC(CC(=C)C)=O)CCCCCO1 c1(C(=O)NCCCCNC(c2cncc(OC(C)C)c2)=O)cscc1S(C)(=O)=O n1(CC(=O)NC2C(NC(C(C(C)C)OC)=O)C2)cnc2cc(C)c(C)cc12 C(=O)(CC(O)CC(C)(C)C)N1C(C(=O)NCC(c2ncc[nH]2)C)CC(C)C1 C(CCC(C)(C)NC(C1CSCCS1)=O)NC(Cc1nc(COC)sc1)=O N1(C(C2C=CC(NC(CCC3CC(OC)C3)=O)C2)=O)CCC(N=[N+]=[N-])C1 c1(CC(=O)NCC2C(NC(C(c3cncnc3)C)=O)C2)ccc(Br)s1 C1(CC)CN(CCCCOc2cccc(C)c2C)CC(C(F)(F)F)O1 c1(C(=O)NC2C(CNC(C3(CC#C)CC3)=O)C2)cn(C)nc1-c1ccoc1 C(=O)(CCC(=O)NC(C1CCN(C(c2cc(C(F)(F)F)cs2)=O)CC1)C)OC N1(C(C(=O)NC2CCC(F)(F)CC2)C2C(C)C2)CCCC2CC1C2(C)C CC(C)CC(O)C(=O)NCC1C2CN(C(c3[nH][nH]c(=N)c3Br)=O)CC12 N1(C(C(C=CC)O)=O)CC2(CCC(CNC(C3CC3(F)F)=O)O2)C1 c1(C(N(C)CC2(NC(C(C(CC)C)O)=O)CC2)=O)ccc2c(c1)CCCO2 c1(NCCC(C)NC(Cc2nc(CC)sc2)=O)ncnc(O)c1Br C=CCCC(F)(F)C(=O)NC1CC(NC(=O)CC2CC(C)=NO2)CC1O C(c1ccc(F)cc1)=CC(=O)NCC1CCN1C(C1CC2(CC2)CO1)=O Cc1c(C(=O)NC(CC(=O)O)C2CC2)cc(C2CCCC2)n1C C12(C(N(C3CCN(C(c4cc(Cl)cn4CC)=O)C3)CCC)=O)COCC1C2(F)F Cc1cc(Br)c(CN(C)CCC2(O)CCNC2)s1 c1(SCC)ccc(C(=O)NCC2CC(C)N(C(c3ncccn3)=O)C2)cn1 C1(NC(C(C(C)C)n2ccnc2)=O)CC2CC(NC(C3(CC4CC4)CC3)=O)C2C1 n1(CC(N2C(C)CCC(CNC(=O)CO)C2)=O)ncc2cc(Br)cnc12 N1(C2CCCN(C(CN(CCC)C)=O)C2)CCN(C(=O)C(F)=C2CCC2)CC1=O Cn1cnc2nc(=NCc3noc4ccccc34)[nH]c(NCC3(F)CC3)c12 c1(OCCCC(=O)N(CCCNC(=O)C(C)c2cncs2)CC)ccc(F)cc1 C1(C(=O)NC2CCN(Cc3c(C)ccc(Br)c3)C2)CCc2nc[nH]c2C1 C1(CNC(Cc2nc(=N)[nH][nH]2)=O)CN(C(=O)C(F)(F)C2(O)CCC2)CC12CC2 N1(C(Cc2nc(C)sc2)=O)CCN(C(c2cccc(Cl)c2F)=O)CC1CO C(=O)(CCCS(N)(=O)=O)N1C(CNC(c2c(C)n(C3CC3)nc2)=O)CC2(CC2)C1 Cc1cc(C)c(C(=O)NCCC(C)CCNC(C2CCCN(C)C2)=O)c(N)c1 N1(C(CN(CC)CC)=O)CCC(C)(CCNC(=O)COc2cc(C)on2)C1 c1(OC)c(Cl)cc(NC(c2cnnn2C)c2nnnn2CC2CCOC2)cc1Cl C(c1ccc(S(C)(=O)=O)o1)=CC(=O)NC1C(NC(C2CC(=C)C2)=O)CS(=O)(=O)C1 C1(C)(C(=O)NCCCC2CCN(C)CC2)COCCN(C(=O)OCC(C)(C)C)C1 Cc1cccc2c1CCC2N(C)C(=O)NC1CCCCC1S(C)(=O)=O C(=O)(CCC1=NNC(=O)CC1)N1CCC(CCOC)(NC(C=CC=CC)=O)CC1 C1(C(=O)NC2CC(NC=O)C2)CCC(n2ccnn2)CC1.C1(C)CC(CF)C1 N1(C(CCSCC)=O)CCN2CCN(C(C3CCNC(=O)C3)=O)CC2C1 c1(N2Cc3c(nn(C)c3CO)CC2)nc(=NC2CCSC2)[nH]c2c1SCC2 C1(C(N(C)Cc2onc(C)n2)=O)CCN(C(c2ccc(C3CC3)o2)=O)CC1(C)C C1(NC(C)=O)CCCN(C(=O)CCOCCOC)C1.CCSCC N1(C(c2c(C)ocn2)=O)CC(C)CN(C(=O)CCOCC(F)(F)F)CC1C C1(C(=O)NC2CCCN(C(c3cnc(OC)s3)=O)C2)CCc2cnn(C)c2C1 O=C(CC(O)Cc1ccccc1)NCC1(F)CC(CNC(=O)COC2CC2)C1 c1(C(N(CC=CC(=O)NCc2c(C)cc(C)s2)C)=O)c[nH]c2ncccc12 C(=O)(CC(C)C(F)F)N(C(CC(N1CCCC(COC)C1)=O)(C)C)C Cc1cc(CNC(C2CC(NC(C3CC(F)(CF)C3)=O)C2(C)C)=O)cnc1F c1(OC(C2C(=C)C2C(=O)NCC(C)(O)CNC(=O)C(C)(C)OC)=O)cccc(Cl)c1 c1(CS(N2CCCC(C3CCO3)C2)(=O)=O)cc2c([nH]1)CCCC2 Cc1oc(C#N)cc1C(N1CCC(NC(=O)Cc2cscn2)C12CC2)=O c1(COC(C)C(=O)NCC(C)(O)CNC(C23COCC2C3)=O)ccccn1 c1(-c2n(-c3ccn(CC)n3)nc(C3CC=CCC3)n2)cc(C)c(C)cc1Cl c1(OCCNC(C2(O)CC2)=O)ccc(C(F)(F)F)cc1-c1nn[nH]n1 C1(COC)C2CCN(C(=O)CCN(CCO)C(c3cc(C)n(C)n3)=O)CC12 C1(OC)CCCC(C(N2CCCC(CNC(c3ccc(=N)[nH]c3)=O)C2)=O)C1 C1(CNC(CCSC)=O)CN(C(c2conc2-c2ccccc2)=O)CC12CCC2 c1(C(=O)NCC2N(C(C(C(C)C)C)=O)CCCC2)ccc2nc[nH]c2c1F C(=O)(C1=NN(C)C(=O)CC1)N1CC(C)C(NC(C23C4C5C2C2C3C4C52C#N)=O)C1 c1(CC=C)cc(OC)c(O)c(CN2CCCC(C)(C(=O)NCC(=C)C)C2)c1 N1(C(C2C(c3c(C)occ3)C2)=O)CCC(F)(C(=O)Nc2ccc(C(C)C)cc2)C1 C#CC1CC2(CC(C(N3CCCC(N(CCF)C(c4ncsc4C)=O)C3)=O)C2)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)NC1CN(C(C23CC(C)C2C3)=O)CC(O)C1 c1(CN(CC(C)(C)C)C(c2c(CC)cno2)=O)ccc(N(C)C)cc1 C(CC1=CCN(C(C2CN(C)CCN(C)C2)=O)CC1)NC(c1c(CC)nc[nH]1)=O C1(C(=O)O)CC12CCN(C(C1CCN1Cc1ccccc1)=O)CC2 c1(OC)nscc1CNC(=O)C=CC(C)NC(c1ccoc1C1CC1)=O C(C)(C)(CCCNC(=O)C(c1ccc(Cl)s1)=O)NC(CC1(C)CC1)=O c1(CN(CCCC2CCOC2)C)cc(Cl)sc1Cl Cc1cc(C(=O)NCC(C)CN(C(=O)CCN2CCC(C)CC2)C)cc(F)c1C S(=O)(=O)(CC(=O)NCCCC1CCCCN1C(C1CC(C)=NO1)=O)NC N1(C(c2cn(C)c(=O)cc2)=O)CC(NC(C2CC2CC(C)(C)C)=O)CCC(O)C1 N1(C(N=c2ccn(C)[nH]2)=O)CC2OCc3cnnn3C2C1 C1(NC(c2cnn(C(C)(C)C)n2)=O)CCC(C)(CNCC2CCS(=O)(=O)C2)C1 CC1(C(=O)NC2CN(C(=O)CCc3cnn[nH]3)CC2CC2CC2)CC2CC2C1 C(C(C(=O)NC1CC1)N(C(C)C(C)C)C(C)C(C)C)C1CC(C(=O)OC)C1 C(CC(C(=O)N(CC(=O)NC)C)NC(=O)CC1CCSCC1)=CC N1(C(=O)Cn2cccn2)CCN(C2CCN(C(c3coc(Cl)c3)=O)C2)CC1 c1(C(C)C)ccc(NC(=O)N(C(c2ccccc2)CO)C)nc1 C(=O)(CCCF)NC1(CN(C(=O)Cc2ccsc2)C)CC1 c1(C(N(C2CN(C(C3CC(F)C(=O)N3)=O)C2)C)=O)cccc(Cl)c1[N+](=O)[O-] N1(C(Cn2c(C)nnn2)=O)CCC(C(=O)NCC2(C)CCCO2)C(O)C1 c1(N(C(C)CNC(c2ccnc(O)c2)=O)C)ncccc1[N+](=O)[O-] c1(C(=O)NC2C(OC)CN(C(c3ncn(CC)n3)=O)C2)nnn2c1CSCC2 Cc1ccc(F)cc1NC(N1CCC(C)C(C(F)C(=O)Nc2ccccc2O)C1)=O c1(OC)cc(C(N2CCOCC(NC(=O)C3=CCOC3)C2)=O)c(Cl)cn1 N1(C(C(=O)NC2CCC(CC)C2)=O)CCc2nc(C)sc2C1 CC1CCN(C(c2cc(CC3CC3)c[nH]2)=O)CC1CNc1cc(C(F)F)ncn1 C(=O)(C(CC)C(=O)NCc1nc(C(=O)NCc2cc(OC)ns2)co1)OCC C(=O)(C1=CCCOCC1)NC1(C(N2CC(C)(C)CCC2CO)=O)CCN(C)C1 c1(N2CCCC(N(C)C(C3(C(F)(F)F)CC3)=O)CC2)nc2cc(F)ccc2o1 c1(CCC(N2C(CNC(C3(C)C(C)C3)=O)C(O)C(O)C2)=O)c[nH]c2ccccc12 c1(C(=O)NCC2(OC)CCN(C(=O)Cc3c[nH]nc3C)C2)nc[nH]c2nccc1-2 c1(OC)cc(Cl)cc(CN2CCN(C(c3ccc(OC)cn3)=O)C3CC23)c1O C1(NC(C2CCCC(F)C2)=O)CCC2CN(C(=O)CCCCC3CC3)CC2C1 C(=O)(C1=CCCN(C(c2cccn(C)c2=O)=O)C1)NCC#C C1(NC(c2c(C)con2)=O)CCN(C(C2CC(C)(F)C2)=O)C(C)C1 CC1(C)CCC(C(=O)N2CCCC2C(=O)Nc2ccccc2O)c2ccccc21 N1(C(C2CCOC2)=O)CCOC2(CCN(C(C34CC5CC3(CO)CC5C4)=O)C2)C1 N1(C(c2cc(CC)[nH]n2)=O)CCC2CC2(NC(c2ccnnc2C)=O)CC1 N1(C(C2CC(=C)C2)=O)CCC(C)C1CNC(c1cnc(Cl)s1)=O C1(C(=O)NCCOCCC(N2C(CC=C)CCCC2)=O)CC2C(C1)C2(C)C C(=O)(C1CCc2nccn21)N1CC(O)(CNC(c2c(C(C)(C)C)ncs2)=O)C1 Cc1c(C(N2CCC3CC23C(=O)NCc2cccnc2)=O)[nH]ccc1=O C1(NC(C(C)C2CCOC2)=O)CC2(CCN(C(=O)C3=CCCC3)C2)C1 c1(C(N2C(C)C(NC(=O)C(Cl)=CCl)CCC2)=O)cc2c(F)cc(F)cc2[nH]1 N1(C(c2c(C)cc(CO)o2)=O)CC(NC(C2COCCC2C)=O)C2(CCCC2)C1 C12(C(N3CCC(C)(NC(C)=O)C3)=O)CC(CO)(CN1C(=O)CN1CCCCC1)C2 c1(OC)ccc(C(=O)NC2CCC(NC(C3SCCS3)=O)C2)cc1C(C)C C#CC1CCCCN1C(C1CCCN(C(=O)OC)C1)C(=O)NCSc1ccccc1 C1(NC(CCOC)=O)CN(C(c2ccc(C(C)C)cc2O)=O)CCC1C C#CCC(C)(C(=O)N1CCCN(C(N)=O)CC1)NC(=O)CN1CCC(C)C1 C1(C(N(CCCNC(C(C(C)C)NS(N)(=O)=O)=O)C)=O)CCc2nn(C)cc2C1 N1(C(CC2C(C)(C)C2(C)C)=O)CC2(C1)CN(C(C1CC3(CCC3O)C1)=O)C2 CC1CCc2onc(C(=O)NCC3CC34CCCCCC4)c2C1 c1(C(=O)NC(CNC(c2c(SC)cc(C)cc2)=O)C)cnn2c1CCCC2C C1(CCNC(CCC2CC(OC)C2)=O)CCC(NC(=O)Cc2cncs2)C1 c1(OCC)ccc(C(=O)NCC2(F)CC(NC(C3(O)CCOC3)=O)C2)cc1 c1(C(=O)NC(CCNC(C(C)Oc2ccc(SC)cc2)=O)C)c(C)cccc1C CC(C)C(C#N)C(=O)N(C1C2CN(C(=O)Cc3nc(C4CC4)cs3)CC12)C c1(-c2ccc(NC(CCOc3cc(C)c(Cl)cc3)=O)cc2)nn(C)c2c1CCC2 Cc1ncccc1C=CC(=O)NCC(C)(C(C)C)NC(=O)CN1CCC(C)C1 c1(CNC(C(=O)N(CC)Cc2ccc(Br)s2)=O)ccc2c(c1F)CCC2 C1(C(=O)NCc2c(C(=O)NC3CN(C(=O)OC)C3)[nH]cc2)CCC(C)(C)CC1 CC(C(=O)N1CCCC(N(CCF)C(C2CN(S(C)(=O)=O)C2)=O)C1)P(C)(C)=O Cc1ccc(SCC(=O)NCCCN(C)C(C2CC3(C2)CC3F)=O)cc1C C1(C(N2CCC(C(C)NC(C3CC(C)OCC3)=O)CC2)=O)CCC2(CCC2)CC1 C(C(O)CCNC(c1cn(CCOC)nn1)=O)NC(CSCC#C)=O c1(C(=O)NC(CC)CN(C(=O)C(c2cccnc2)O)C)ccc2nn[nH]c2c1 C(CC(=O)NCCCOCC(F)F)(C(C)C)NC(c1cc(C)oc1C)=O C1(NC(=O)C=CC2CC2)CC12CCC(NC(c1ccc(C(F)F)cc1F)=O)CC2 C(C(=O)NCC(C)CCCO)(C(C)C)NC(Cc1c(C)n[nH]c1)=O c1(N(C(CC=CC=C)=O)CCC2CN(C(=O)CCC)C2)ncc(Br)cn1 c1(C(=O)NC23CC(NC(Cc4c(C)cccc4C)=O)(C2)C3)ccc2nc[nH]c2c1 CC1(C)NC(=O)CC1C(N1CCCC(CCNC(c2cccc(O)c2Cl)=O)C1)=O CCC(C)(CNC(C1CCN(C(C2(CO)CCCCC2)=O)CC1C)=O)C(N)=O N1(C(CCCCC)=O)CCN(C(c2cnn(C3CC3)c2)=O)CC1C(C)C C1(NC(=O)OC(CCC(C)c2ccc(Br)cc2)=O)CCC(O)CN(C(C)(C)C)C1 C1(C(=O)NC(C)CN(C)C(c2cc(C(C)(C)C)ccn2)=O)COC2COCC12 N1(C(CCC=CCC=C)=O)CCC(F)(C(N2CC(C)CC(C)C2)=O)CC1 c1(C(=O)NCC(CNC(C(C2CC2)OC)=O)CO)cccc(OCC=C(C)C)c1 c1(C(=O)NC2(CNC(=O)C=Cc3cncs3)CC(OC)C2)ccc(CCF)cc1 N1(C(Cn2ccc(C)cc2=O)=O)CCCN(C(=O)Cn2c(C)ccc2C)CCC1 c1(CC)nc(C(=O)NCC2CCN2C(C2CCCC2OC)=O)cs1 c1(C(=O)NCC(C2CC2)NC(c2ccc(C(=O)OC)s2)=O)cc(Cl)nnc1O N1(C(C(C)NOC(C)(C)C)=O)CCCC2(CCCCO2)C1.C1(=O)CCN(C)C1=O C1(CNC(c2c(CC)cno2)=O)C(C)CCN1C(c1cc[nH]c(=N)n1)=O Cc1ccc(C(=O)NCCSCC(=O)NCC2CCCN2C(C)C)n1C N1(C(C2(OC)CCCOC2)=O)CC(C2CCN(C(C3C=C(C)CS3)=O)CC2)C1 C1(CNC(C2(NC(c3ccc(CC)[nH]3)=O)CC(F)(F)C2)=O)CC(C(N)=O)=NO1 N(C1CCCn2ccnc21)C(=O)C(F)C1CC(NC(=O)C(O)CN2CCCC2)C1 C#Cc1ccc(F)c(C(N2CC3CCC2(CNC(=O)CC(C)CCC)C3)=O)c1 N1(C(c2ccc(C)s2)C)C(=O)NC(CC2(C)CC2)C1=O CC12CN(C(=O)Cn3cc(Cl)cn3)C(C(=O)NCC3CC3c3ccoc3)(C1)C2 c1(OC)ncc(C(=O)NC2(CNC(C3CCCOC3)=O)CC(F)(F)C2)cn1 N1(C(C)=O)CCC2CN(C(c3cc(-c4ccccn4)[nH]n3)=O)CCC12 c1(C(=O)OCC)cc(C(=O)N(C2CC(NC(C3(C)COCCO3)=O)C2)C)nn1C N1(C(Cc2ccc(Cl)c(C)c2Cl)=O)CC2(C1)CN(C)C(=O)C2(F)F C1(OCC)CC2(C1)CC2C(=O)NCC1CC(C)N(C(c2cnn(CC)c2)=O)C1 CC1=CCC(C(=O)NC2CCCCC2CNC(=O)CC(O)C2CCCC2)CC1 C1(C(C)C)CN(C(=O)C(O)C(C)C)CCN1C(c1cc(C(N)=O)cn1C)=O Cc1cnncc1C(=O)NCC(C)(C)CNC(c1ccc(NCC(C)C)nc1)=O O=S(=O)(c1cccc(=NCC23CCCC2C3)[nH]1)NCC1CC(O)C1 Cc1cc(=NCc2ccnc(C#N)c2)[nH]c(NCCN2CCC(N(C)C)C2)n1 CC(O)(C(=O)N1CCOCC(F)(CNC(=O)CCC(N)=O)C1)C(F)(F)F N1(C(CN2C(C)CCC2)=O)CC(C2CN(C(=O)C(F)n3ccnc3)C2)C1 Cc1cccc2c1CC(C(=O)NC1COCC1NC(c1ccn(C(F)F)n1)=O)O2 C1(N(C(C(C)OCCC=C)=O)C)CCN(C(=O)C=Cc2ccco2)C1 c1(C(N(CCNC(C(CC)N(C)C)=O)CC2CC2)=O)cc(C)cc(OCC)c1N c1(CN=c2scc(C(N3CCCC4(CCC4)C3)=O)[nH]2)ccc2c(=O)cc[nH]c2c1 Cc1cc(C(=O)NCC(C)(C)OCCNC(c2cncnc2C2CC2)=O)c(C)s1 CCC(CNC(=O)C=Cc1cnc(C)s1)(CC)NC(C1OCCC1COC)=O c1(NC(N2CC(C(=O)NCc3ccccc3)OCC2)=O)cc(Cl)c2cc[nH]c2c1 N1(C(c2cc(C(=O)OCC)n[nH]2)=O)CCC(NC(=O)CC(C)C(C)C)C(O)C1 c1(C(=O)NC(CNC(c2c(CC)ccs2)=O)CO)cc(C)ncn1 N1(C(c2c(CC)onc2)=O)CC2(CCN(C(=O)CCCOC(C)=O)CC2)C1 c1(C(=O)NCC2(F)CCC(CNC(c3ccncn3)=O)C2)ccc2sccc2c1 c1(C(=O)NCCC2(CNC(C(C)Cc3cnc[nH]3)=O)CC2)csc2cccnc12 c1(C(N2CC(NC(c3cncc(C)c3)=O)C(F)C2)=O)ccc([N+](=O)[O-])cc1Br c1(CNC(COC(CC(n2c(CC)ncc2)C)=O)=O)[nH]c(C)nc1C C1(C(=O)NC23CC(NC(C4CC(F)(F)C4)=O)(C2)C3)CCCS(=O)(=O)C1 N1(C(Cn2ccc(C)n2)=O)CCN(C(=O)C(O)CC[S+](C)C)CCC1C N1(C(C2(CC=C)CC2)=O)CCC(N(C(=O)CCCCN2C(=O)CCC2=O)C)CC1 C1(CNC(C(=O)NCC)=O)C(C)(C)C(NC(=O)C=CCN2CCOCC2)C1(C)C C1(CC(=O)NC(CNC(C(CC)C)=O)(C)C)CCN(C)C1=O n1(CNC(C2C(C)C2C)=O)cc(C(N2CC(CCN(C)C)C2)=O)cn1 C(C)(CC(=O)NC(C1CCN(C(c2cc(C3CCC3)[nH]n2)=O)C1)(C)C)SC Cc1ccn2ncc(C(=O)NCC(C)(C3CCC3)NC(=O)Cn3cnnn3)c2c1 C1(CNC(Cn2c(C)nc(C)n2)=O)C2CCC1CN(C(c1sncc1C)=O)C2 CCCCCCC(=O)NCCN(C(C1CCCN1Cc1ccccc1)=O)CC Cc1cc(O)c(C(=O)NCC(CC(C)C)NC(C2CC(=C3CC3)C2)=O)nn1 C(CC(C)C(=O)NCC1CN(C(c2nc(C3CNC3)oc2C)=O)CCO1)=CC C#CC1(C(=O)NCC(C)C(C)(C)C)CCN(C(=O)C(=O)C2CCCC2)C1 N1(C(CNC(CC)=O)=O)CC2(C1)CN(C(C1CN(C(c3ccncc3)=O)C1)=O)C2 C(=O)(C(C)CCCC(C)=O)N1CCC(NC(c2ccc(OC)nn2)=O)C1C1CC1 C1(CC(=O)NC(C2CCN(C(=O)CC3(C#N)CC3)C2)C)SC2=NCCN2C1=O Cc1o[nH]c(=NC(=O)NCC2CCC(=O)NC2=O)c1C C1(NC(C(CCC)CC)=O)CCCCCN(C(=O)CSc2cn[nH]c2)C1 c1(CN2CC3C(C(=O)NC4CCCC(O)C4)(C3)C2)c(Br)ccc2c1OCO2 CC1CN(C(c2ccccc2O)=O)CC1NC(=O)Cc1nc(C2CC2)cs1 CCS(=O)(=O)CC(=O)N1CCCC(O)(CN(C(=O)C=CBr)CC)C1 c1(C(=O)NCC2(O)CN(C(C(C3CC3)OCC)=O)C2)c(C)n[nH]c1C c1(N(CCCSC)C)nc(=NC2CCCn3nccc32)[nH]c2c1COC2 N1(CCNC(C2CCCCS2)=O)CCCN(C(=O)C=C2CCOCC2)CC1 c1(OC)ccc(OC)c(C(=O)NCCC2CCC(NC(=O)C(C)=C3CCC3)C2)c1 N1(C(=O)NC2CC(c3ccc(C)cc3)C2)CC2(CCOCC2)C1C(C)C C=CC(CCC)CC(=O)NC1CCC(CC(=O)N(c2ccccc2C)C)C1 C=CCCC(F)(F)C(=O)NCC(C1CCN(C(=O)C(F)CN(CC)CC)CC1)O C(C(C)(C(C)C)NC(c1cccc(NC(=O)OC)c1)=O)NC(C1C(=C)CC1)=O c1(OC)cc(C(=O)Nc2ccc(F)c(F)c2)c(NC(c2ccc(Cl)nc2)=O)cn1 C1(C(=O)NC2CC3(CN(C(C=CCC)=O)C3)C2)CC2CCCCC2O1 c1(NC(C2CCN(C(C3(C)CCCO3)=O)CC2)C)nccn2nnnc12 N1(C(C(CCC)=CCC)=O)CC23CCCC2(C1)CN(C(C1CCOC1CC)=O)C3 C(=O)(C1=NOC2COCC12)NC1(C)CCN(C(c2cc3cccnc3cn2)=O)C1 c1(C(=O)NCC(C2CC2)NC(C(C)Cc2cnc[nH]2)=O)cc(N)cc(O)c1F c1(C(=O)NC(CNC(Cc2cc(C)on2)=O)C)noc(C)c1I Cc1c(C(N2CCN(S(=O)(=O)CCCl)C(C)C2)=O)cc(F)cc1Cl c1(OC)cc(C=CC(=O)NC2CCC(CNC(=O)CSCC(C)C)C2)sn1 CN1CC=C(C(=O)NC2CCC(CCNC(=O)COCc3nc[nH]n3)C2)C1 C1(C2CN(C(=O)Cc3cncs3)C2)(NC(C(C)OCc2ccc(C)cc2)=O)CC1 N1(C(C(C(CC)O)C)=O)CC(NC(=O)Cn2cnc(C(F)(F)F)c2)C2(CCC2)C1 c1(SC)ccccc1C(N1CC2C(CNC(=O)C(C)OCOC)C2C1)=O C(=O)(CCCC(C)(C)C#N)NCC(C(C(=O)NCCNC(CC)=O)F)C c1(C(N2CCN(C(C3CC(C)N(C)C3)=O)CC2C)=O)cn(C)c2c(Cl)cccc12 N1(NC(C2C(C)C2)=O)CCN(CC2CCN2C(c2coc(C(C)(C)C)n2)=O)CC1 C12(CC(=O)NC3C4CN(C(C5CC(N(C)C)C5)=O)C3C4)CCC(C)(C1)OC2 C1(C(C(=O)N(C(C(N)=O)=O)Cc2[nH]ccc2-c2cccs2)F)(OC)CCOCC1 c1(C(N2CCC(NC(CN3CC(CC)C3)=O)C(O)C2)=O)cc2oc(C)cc2[nH]1 C1(C(=O)NC(CN(c2ncc(C(=O)OCC)cn2)CC)C)CC(=O)NC(=O)N1 C(=O)(C(C(CC)CC)OCC)N1CCN(CC)CC1.C1(=O)C(=O)NC2(CC2)CN1 C1(C(N(C)CC2CCCCN2C(=O)Cc2cc(Cl)cs2)=O)CCc2nnnn2C1 CCC(CC)CCC(=O)NC1CC(C)N(C(c2ccc(S(C)(=O)=O)[nH]2)=O)C1 C1(OCC(=O)OC)CCN(C(c2csc(C)c2)=O)C1 Cc1c(C2OCCC2C(=O)NC(C)CCNC(c2cc(CO)[nH]n2)=O)cnn1C N1(C(C(C=C)O)=O)CCC2CCN(C(=O)C=Cc3cncc(O)c3)C2C1 c1(C(c2nnnn2CC(F)F)NCc2cncc(C)c2)cc(Cl)cc(Br)c1 N1(C(C2C(C)OCCN2C(=O)CC2CCCSC2)=O)CCC(O)C(C)(C)C1 N1(C(CC2CC(NC(c3ccccn3)=O)C2)=O)CCn2nc(CO)cc2C1 c1(CC)ccc(C(=O)NCC(CC)NC(=O)C2=CCCCO2)cc1CC N1(C(=O)C(C2(O)CCCCC2)(F)F)CCOC(c2cn(Cc3cnns3)nn2)C1 CC1CC(NC(=O)CCc2cn[nH]c2)CN1C(=O)COC1CC1 C1(C(=O)NC2CN(C(C(C3CCCCC3)C)=O)C2)CCC2CC1C2(C)C N1(c2n(CC3N(C)C(=O)CC3)nnn2)CC2(CCCCC2)CC1CO C1(CCNC(=O)C(O)Cc2cnc[nH]2)CCCN(C(=O)CC2CC3CC3C2)CC1 N1(C(C(CC)(CC)OC)=O)C2CCC1CN(C(C1CN(C(C)=O)CCO1)=O)C2 C1(C(=O)NCCC(C(=O)NC(COC)(C)CO)OC)CCC2(CC1)CC2 C1(C)(C(=O)NCCC2(C)CCC2)CCCN(C(c2ccccc2C(F)(F)F)=O)C1 C1(CC(=O)NC2C=CC(NC(C=C(CC)CC)=O)C2)(CN(C)C)CCOCC1 N1(C(CCSC)=O)CCC2(CCC2NC(c2cc3ccccc3cn2)=O)CC1 C#CCCC(O)C(=O)NC1COCC1CNC(c1c[nH]c(=O)cn1)=O c1(OC)ccccc1-n1cc(C2(C)CN(C(=O)COc3ccc(Cl)cc3)C2)nn1 N1(C(C(=Cc2cccs2)C)=O)CCC(C(C)(C)NC(C2COC(C)C2)=O)CC1 C1(CNC(Cc2c(C)con2)=O)C(C)CCN1C(c1ccnc(O)c1)=O S(=O)(=O)(c1cccc(Cl)c1C)N1C2CCN(Cc3scc(C)c3)C2CCC1 N1(C(CC(C)C)=O)CCC2CC2(C(=O)N(C)Cc2nc[nH]n2)CC1 Cc1cc(=N)[nH]cc1C(N1CC(CNC(=O)C(F)=CC2CC2)CC1C)=O c1(N(C2CCNCC2O)C(c2nc(C)oc2)=O)ncnc2n[nH]cc12 C(=O)(CCN(OC)C(=O)CN(C)CCOC)CC.O1P(C)(=O)CN1.C=CC N1(C(c2n(CC)cnn2)=O)CCC(C)C(NC(C2CCN(CC3CC3)CC2)=O)C1 c1(C(=O)NCC(CO)NC(c2ncn(-c3ccccc3)n2)=O)cn2c(n1)CCC2 N1(C(c2nccc(C)c2)=O)CC(NC(c2cc(CO)on2)=O)CC12CCCCC2 c1(C(=O)NCC2(NC(c3c(CC)oc(C)c3)=O)CC2)cc2ccc(Br)cc2[nH]1 c1(N2CC(CCC)C(COC)C2)cc(C)c(S(=O)(=O)NC(C)CCOC)cn1 S(=O)(=O)(c1ccc(N2CC3CCC(C2)N3C)c(F)c1)NCC1CC(C)SCC1 C1(NC(c2ccc(OCC)cc2)C(=O)OC)CC2(C1)CC(C(=O)O)C2 C1(CNC(c2cn(C)nn2)=O)CCCCCN1C(C1CCOC(=O)N1)=O C1(C2CN(C(C3CC34CCC4)=O)C2)(NC(C(=O)NCC(F)F)=O)CC1 c1(C(=O)NC(c2cnn(C)c2)C(N2CC(CC(=O)OC)C2)=O)ccoc1Cl c1(CNC(C)=O)ccc(C(=O)NC2CCC(CNC(C3(C)CC3C)=O)C2)s1 C1(C(=O)NC)CC(F)CN(C(c2c(C)oc(C)c2C)=O)C1 C(C(CC=C)C(=O)NCC1=C(C)CCOC1)NC(c1n(CC#C)ccc1)=O c1(C(=O)NCCN2CCNC2=O)nc(-c2cccnc2F)c2ccccn12 C1(NC(C2(COC)CCC2)=O)CN(C(c2ncc(C)cn2)=O)CC1O C12(C(=O)NCC(C)NC(=O)CNC=O)CCCN1S(=O)(=O)CC2 C(N=c1ccnc(C2CCC2)[nH]1)C1CC(NC(Cc2ccn(CC)n2)=O)C1 N1(C(CC2(OC)CCCC2)=O)CCC2(C1)CN(C(c1oc(Br)cc1C)=O)C2 c1(-n2c(C(C3=CCSC3)C(n3cc(Cl)cn3)C)nnn2)ccc2c(c1)CCC2.N Cc1cccc(C(=O)NCC2(C(=O)NCCCC(N)=O)CC(C)(C)C2)c1N C1(CNC(C(C(C)C)SCC)=O)CC2CCC1N2C(c1cc(F)cc(F)c1)=O c1(C(N2CCC(N(C(=O)C(SC)SC)CC)C2)=O)c(C)ccc(F)c1N C(CC(=O)N1CCC(OCC(N)=O)C1)(C(F)(F)F)NC(c1c(C)non1)=O C(Cn1cncn1)(C(=O)NC1COCC1O)NC(c1sccc1F)=O C12(C(=O)NCCCN(C(CCCN(C(C)=O)C)=O)C)CCCC(=O)N1CCC2 C1(c2nnc(COC(CC)CN(C)Cc3ccccc3)n2C)CCNC(=O)CC1 C(c1ccco1)=CC(=O)N(CC(CC)NC(c1ccc(C(=O)OC)s1)=O)CC Cn1cccc1C=CC(N1CCC(NC(=O)C=Cc2ccc(C(F)F)o2)CC1)=O N1(C(C(F)=CCC)=O)CCC2(CC2)CC1C(=O)Nc1ccc(F)cc1O c1(C(=O)OC(CSC)C)ccnc(OCC(F)(F)F)c1 c1(C(=O)NC2CCC(CNC(c3c(C)oc(CO)c3)=O)C2)cc2scc(Cl)c2[nH]1 C1(C(N(CC)CC2CCCOC2)=O)CN(C(=O)C(C)OC(C)(C)C)CC1(F)F CC(C(=O)NCC1(CO)CC=CC1)(C1CCC1)NC(c1cc(C2CC2)on1)=O Cc1ccccc1C=CC(=O)NC1CCN(C2CC2)C1 c1(OC(C)(C)C)cccc(OC2(C(=O)NCC#N)CCCOC2)c1 CC1CC(NCC2(F)CCC(C(=O)N(C)C)C2)CCC1O c1(COC)ccnc(CNC(=O)C(C)(C2CC2)N(C)C(c2ccc(C#N)[nH]2)=O)c1 c1(CN(C(=O)C=CC=C(Cl)Cl)C)cnn2c1CN(C(C1CC3C=CC1C3)=O)CC2 C1(C(=O)NC2(C)CCN(c3nccc(N4CCCC4)n3)C2)CCCC2(CCC2)O1 C(=O)(CC(CC)CC)NCCC1N(C(c2cc(CC)on2)=O)CC(OC)C1 c1(OC)ccc(C)c(-c2nc(Cn3cc(Br)cn3)nn2C2CCCSC2)n1 N1(C(CNC(CN(C)C)=O)=O)CC2CCC1C(NC(c1cc(Cl)ccc1N)=O)C2 N1(C(c2c(OC)c(C)sc2)=O)CCC2(C1)CN(C(=O)Cn1nnc(=O)[nH]1)CCO2 C(=O)(C1=CC2(CCN(C(C3(C)CCCCC3O)=O)C2)C1)NC1C(O)CCN(C)C1 c1(NC2CN(C)C(=O)C2)cc(=NC2CCC2C2CC2)[nH]c(C(F)(F)F)n1 c1(OC)ccc(C(N2CCC(CO)(NC(=O)C(O)C3CCCC3)C2)=O)cn1 c1(C(N(C2CCN(C(=O)CCOC)CC2)CC)=O)cccc(-c2ccncc2)n1 CCCC(C(=O)N1CCCCCC(NC(c2cc(Cl)cn2C)=O)C1)S(N)(=O)=O N1(C(C(C)OCCOCC)=O)CC(C(=O)NCc2cccc(F)c2C)CC1(C)C N1(C(C(C)CC(N)=O)=O)CCCCCCC1C(=O)NCCN=S(C)(C)=O C(C)(CC(C)N=c1cc(C2CC2)nc(C2CC2)[nH]1)NC(C(C(C)C)F)=O c1(C(=O)NC(C(C(C)C)NC(c2ncccn2)=O)C)cc2ccnn2cn1 C1(CS(=O)(=O)NCC2(c3c(OC)nccc3)CC2)CS(=O)(=O)CCO1 c1(C(CC)C)nc(N2CCN(C(C3CC3C)=O)CC2)cc(C)n1 N1(C(C(C)(C)OC(C)C)=O)CCC2CCN(C(=O)CC3(C)CC3)CC2C1 C12(CNC(C3(NC(CC4N(C)CC=CC4)=O)CCOCC3)=O)CCCN(CC1)C2 S(=O)(=O)(CCC(=O)NC12CC(C1)N(C(c1cnc[nH]1)=O)C2)N(C)C c1(C(=O)NCC2(NC(c3cnc(COC)s3)=O)CCOC2)ncc(F)cn1 C12(CN(C(=O)CCCOCCOC)C1)C(=O)N2.C1(CC)C(CO)C1(C)C C12(CNC(c3ccc(NC(C)=O)cc3)=O)CC(C1)C(NC(c1cnc[nH]1)=O)CO2 c1(C(N(CC(C)NC(C(n2ncc(C)c2)C)=O)C)=O)c(C)nc(C2CC2)nc1S C1(NC(CC(=C)C)=O)CCC(C)(C)CC1CNC(c1cnc(NC2CC2)s1)=O c1(C(N2CC(C)(NC(C34CCN(CC3)CC4)=O)C2)=O)ncnc2c1CCC2 C1(N(C(=O)CN(C)C(C)C)CCC)CCN(C(=O)C(C)C2CCC2)CC1 CONCCC(=O)N1CCN(C(=O)C(C)C2CCC2)CC1 N=c1nc(N2CCOC(c3ccccc3)C2)[nH]c(=NC2CCNC3(CCC3)C2)[nH]1 C1(CC)CN(C(=O)CC2(C)CCCCC2)CCN1C(c1cc(Br)n(C)c1)=O Cc1nsc(C(=O)NC(Cc2ccoc2)C(=O)NC(C)CCN(C)C)c1N c1(C(N2CC(C)(NC(c3cc(C)sn3)=O)C2)=O)ccc2ccccc2c1 C(CC(C(=O)NCCN1CCCOC1=O)NC(C1CCC1C)=O)OC C#CCC(CC#C)C(=O)NC1CCN(C(c2cn(C(C)C)nn2)=O)CC1CO C1(CC)CN(C(c2sccc2Br)=O)CCC1NC(=O)Cn1cnc(=N)[nH]1 C(CC)(CCCC(=O)NCC1(F)CCC1)NC(c1c(CC=C)cccc1)=O c1(C2C(C(=O)OCC3OCCN(C(=O)OC(C)(C)C)C3)CCC2)ccc(F)c(F)c1 c1(C(=O)NCc2ncc(C)o2)cc2c(C)cc(C)c(C)c2[nH]1 C12(CNC(c3c(OC)csc3)=O)CN(C(=O)C(C)(C)OC)C(COC)(C1)C2 C1(C(N2CC(CC(C)NC(c3sc(C)c(O)n3)=O)C2)=O)CCOC(C)(C)C1 c1(C(N2CCCC(C(F)F)C2)C(=O)NCC=C)nc(C)c(C)n1C C(=O)(CC(C(F)(F)F)N1CCOCC1)N1CC(C)(NC(CCNC(=O)OC)=O)C1 N1(C(CN(CCC)C)=O)CC=CC1(C(=O)NCC=CCOC)COC N1(C(CC2CC(=C)C2)=O)CCN(C(=O)CC2CCOC2=O)C2CCCC12 CCCC(C)(C)CC(=O)NC(C)(CNC(=O)COC(=O)CO)CC(C)C c1(C(=O)NCC2(CNC(c3c(CC)n[nH]c3)=O)CCC2)cnccc1C(F)F C1(NC(CNC(CCNC(C)=O)=O)=O)CN(C(c2nnc(S)n2C)=O)CCC1C C1(C(C)C)CCC(C(N2CCC2CNC(=O)CSc2ccccc2)=O)C(=O)N1 C1(NC(N2CCC(O)(COCCO)C2)=O)CCCOC1c1ccc(F)cc1 CC(C)C(O)C(=O)N1CCC(CN(C)C(c2cccc(-c3ccoc3)c2)=O)C1 N(C1c2ccccc2CC1NCCOC)C(C(=O)NC(CC)C)=O C(=O)(CC(C)CC(C)C)N1CC(C(=O)NC(C)Cn2cc(C)cn2)(SC)C1 C1(CNC(CN(CCOC)C)=O)CCN(C(=O)Cc2nc(=N)[nH][nH]2)CCC1(F)F n1(CCC)cc(C(=O)NCc2cc(C(N3CCC(N4CC(O)C4)C3)=O)n[nH]2)cn1 C(=O)(C1CCCc2ncccc21)N(CCCNC(Cc1nc(C)oc1)=O)CCO C1(OC)CN(C(=O)C=CC2CCC2)C(C)(CNC(=O)CCCCSC)C1 n1(C(C(=O)N(CC(CC)NC(C2(n3cccn3)CCC2)=O)C)C)cc(C)cn1 c1(NC(C2CCN(C(C(CCC)CCC)=O)C2)=O)ncc([N+](=O)[O-])cc1F CC1CNc2c(C(=O)NC3CC(NC(c4nccc5occc45)=O)C3)cnn2C1 c1(C(=O)NC(CC)C2CCC2)cn(C2CC(C(=O)NC(C)C3CC3)C2)nn1 C1(NC(C2CCc3cnnn3C2)=O)CN(C(=O)Cn2cccn2)C2(CCCC2)C1 c1(C(N2CC(C)(O)C2)=O)noc2c1CC(NC(=O)CN1C(=O)CSC1=S)CC2 c1(N(CC(=O)NC(C(=O)N(C)C)Cc2ccccc2)C)ccc(S(C)=O)cc1 CC1(C)C2(C(=O)NCCSCCCc3cn(C4CC4)nn3)CCC1(C)C(=O)O2 N1(C(CCC(CC)CC)=O)CCc2sccc2C1CNC(C1C=CCC1)=O C1(C(=O)NCC=CC(N2CC(NC(=O)NC)C2)=O)CCCCNC1=O Cn1cc(C(=O)NCC2(CNC(=O)Cc3nccn3C)CC2(F)F)c(=N)[nH]1 C1(C(N(CCCNC(c2cnc(OC)nc2)=O)CCO)=O)CN2CCN1CC2 c1(C(=O)NCC(C)NC(=O)CSCCC(F)(F)F)c[nH]c(=O)c2ccnn12 Cn1cc(C(C(=O)NCC(=O)OCC2CC2)NC(=O)Cn2cnnn2)nn1 C#CC1(C)CCCN(C(C2CCN(C(=O)CCC3CCCCO3)C23CC3)=O)C1 N1(C(C)=O)CCCC(CC(N2CCCC2(C)CNC(=O)C(F)=C(C)C)=O)C1 N1(C(C2(C#N)CCOC2)=O)CC2OCCN(C(=O)C3CC3)C2C1 C(C1c2ccccc2CCN1C(c1cnn(C)c1F)=O)NC(C1(COC)CC1)=O N1(C(c2cc(CC)n(C)n2)=O)CC2CC(C1)C2NC(c1cc(C2CCC2)[nH]n1)=O C(CC(=O)OC)(C(C)C)CCOC(CC=CCCCCC)=O O=C(CC(C(F)(F)F)NC(=O)CN1C(=O)CNC1=O)NCC1CCC=CO1 n1(C(C)C)ncc(C(C(=O)NC2CCCC2)N(C2CCCC2)CCC#N)c1F c1(C(N(C)CC2CCCC(NC(COCC=C)=O)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(NC(C(CNC(c2nncc(CCC)c2)=O)O)=O)CCN2CCC1C2 C(=O)(C(C)(F)C(=O)N1CCCC(N(C(=O)C=CC2CCOCC2)CCF)C1)OC N1(C(CS(CC)(=O)=O)=O)CCCN(C(=O)C(F)C(C)(C)O)C(C)C1 c1(CC(N2CC(=C(F)CNC(C3(CO)CCC3)=O)C2)=O)cnsc1 CCC(C)C(C(=O)NC(c1ccc(F)cn1)(C)C)N(C(=O)C=CC1CC1)C C1(OC)CC(C(=O)NC(C(=O)N(C(C)CSC)C)C2CC2)C1 C1(C(=O)NC2C(NC(c3cc(C)on3)=O)COCC2)CCC2(CCC2)O1 N1(C(C(CC)SC)=O)CCC(NC(=O)C=CCN(CC)CC)C(CC)C1 c1(NC(C(CC2CC2)NC(=O)C=Cc2cncs2)=O)cc(F)ccc1F N1(C2C3(CC(OCC(=O)OC)C3)C2)CC2CCCC(C1)N2C c1(C(N(CC)CC2CCCCN2C(=O)COC)=O)cccc(Cl)c1[N+](=O)[O-] N1(C(c2ccc(C)nc2)=O)CCC(F)(C(=O)NCC(Cl)C(C)(F)F)CC1 CN1CCCc2cc(CNC(=O)C(C3CCCCN3)O)ccc21 N1(C(CN(C(=O)OC)C)=O)CCC(CCNC(=O)C(F)(F)c2ccnn2C)C1 CCC1(C(=O)N2CCOC(COC)CC2)CCCc2ccccc21 C12(C(N3C(CCN(C(c4cnc(C)nc4)=O)C)CCCC3)=O)CCC(F)C1CC2 N1(C2N(CCC3CC(C(=O)O)C3)CCCC2)Cc2ccccc2C1 N1(C(c2nc(C)oc2)=O)CC2(COC(CNC(c3cc4c(nn3)CCC4)=O)C2)C1 c1(C(N(C2CCS(=O)(=O)C2)CCN(CC)CC)=O)ccnc(C2CCC2)c1 c1(OC)ccc(C(=O)NCC2C(C)CCN2C(C2CN(S(N)(=O)=O)C2)=O)c(Cl)c1 C12(C(=O)NCCN(C(C(C3CC3)OC)=O)C)CCC(CO1)C2.C1CC1 C1(NC(c2c(F)ccnc2F)=O)CC2CCC(C1)N2C(C1CC=CC1)=O N1(C(C2(COC)CC2)=O)CC(C(=O)NCCN(C)C)CC2OCCC12 N1(C(CCC=CC(C)C)=O)C2CCC1CC(F)(CNC(c1ccncn1)=O)C2 CCC(O)C(C)(C)C(=O)NCC(C)N(C(=O)Cc1ccccc1Cl)C c1(CC)ccc(C(C)C(=O)NCC23CC2CN(C(=O)CCCC2CCC2)C3)cc1 C1(C(=O)NCC(N2CCN(C(C3CC(S(C)(=O)=O)C3)=O)CC2)C)CC(=O)OC1(C)C n1(CC(=O)NCC(C)N(C(C(C)NC(CC)=O)=O)C)ccc(=O)cc1C C1(C(=O)NCC2N(C(C(C)C3CC3)=O)CCC2)CC(=O)C12CCC2 Cc1cccc(-c2ccccc2C(=O)NCC(F)CNC(C23CCC2C3)=O)c1 N1(C(CC(=O)NCC)=O)CC2CC(NC(c3nc(C)ccc3OC)=O)C2C1 C1(C(N2C(C)(CNC(C(C(=C)C)(C)C)=O)CCC2)=O)CCC(=O)CC1(C)C N1(C(C(CNC(=O)OC(C)(C)C)OC)=O)CCC(O)C(N(C(=O)C(Cl)=CCl)C)C1 N1(C(CC(C)C2CCCC2)=O)CCCC12CCCN(C(C1CCCO1)=O)C2 CC1CCCC(C(=O)NCc2cc(C(=O)NCc3cn(C4CC4)cn3)n[nH]2)C1 C=C=CC(C)C(=O)NCc1ccc(CNC2CC2CNC(c2csc(=NC)[nH]2)=O)o1 C1(n2c(C(c3cccc(Cl)c3C)C)nc(-c3cccnc3)n2)C(C)CCCC1C C1(C)(NC(COCC)=O)CC(C(=O)NCC2CCOC2=O)C1 C(CCF)(C(=O)NCCc1nc(C)cs1)NC(C(C)SCC)=O CCCCC(O)CC(=O)NC1CN(C(c2ccc(C(C)C)nc2O)=O)CC1C c1(SC)ccccc1C(=O)NCC(C1CC1)NC(=O)CSC.c1(N)ccccn1 CC1=NOC(C)(c2nc(-c3ccccc3N(C)C)no2)C1 C(=O)(C(=O)N=S(C)(C)=O)N1CC(COC)N(C(=O)CC(C)OC)CC1 CC(CS(C)(=O)=O)C(=O)N1CC(C)(C)CC1CNC(c1ccnn1C)=O C(=O)(CCCS(C)(=O)=O)NC1(C(=O)OC)CCCN(C(=O)C(C)O)C1 N1(C(CSCCN(C)C)=O)CC(NC(C2CCN2S(C)(=O)=O)=O)C2CC2C1 CC(C)C(C(=O)N1CCC(O)(CCNC(c2ncncc2Cl)=O)C1)NC(N)=O C(C(C)(Cn1cccn1)NC(c1occc1Cl)=O)NC(COC(CC)C)=O NC(CCF)C(=O)NC(c1ccccc1)COCc1ccccc1 CC(Cc1ccccc1)CC(=O)NCC(C)(C)CC1CN(C(C2CC2(F)F)=O)C1 C(=O)(CCCCCF)N1C(CCNC(C=Cc2ccc(C)o2)=O)CCC1 CN1CCCCC1CCC(=O)NCCC1CCN(C(c2cc(Cl)sc2Cl)=O)C1 N(C1c2cc(Br)ccc2SCC1C)C(CSc1ccc(C)cc1)=O c1(CC)ccc(CN(C(C2CCC(n3cc(C(C)(C)O)nn3)C2)=O)C2CC2)nc1 C(C1=Nc2ccccc2S(=O)(=O)N1)CNCc1c(C)nn(C2CC2)c1 CC1CC(CCNC(c2c(F)cncc2F)=O)CC(C)O1 c1(OC)ccc(C(=O)NC2CC(CNC(c3cn(C4CCC4)nn3)=O)C2)c(F)n1 C1(C(=O)NCC2C(C)CCCN2C(C2CCCN2C=O)=O)CCc2n[nH]cc2C1 c1(C(=O)NCC2OCC(C(N3CC(NC(=O)NC)C3)=O)C2)ccncc1Cl c1(N(C(C)(C)C)C(C2CC2(F)Cl)=O)ccc(F)cc1 C1(NC(CCC(C)C)=O)CN(C(c2ccc(C(F)(F)F)nc2Cl)=O)CC1N=[N+]=[N-] N1(C(C(C)OCC(C)C)=O)CCCN(C(c2ccnn2C(F)F)=O)CC1 CS(=O)(=O)CCC(=O)N1CCC2(NC(=O)CSCc3cccc(Cl)c3)CC2C1 N1(C(c2ncn(C)n2)=O)CCC2(NC(c3cncc(F)c3)=O)CCCCC12 CC1(C)CC(=O)N(CC(N2CCCC2CNC(C2CC3(CCC3)CO2)=O)=O)C1=O Cc1cc(C)c(C(=O)NC2CCCC2NC(C2CC3(CCO2)CC3)=O)c(C)c1 c1(CC(=O)NCCCC(C)NC(CN(CCOC)C)=O)ccncc1Cl Cc1cccn2ncc(C(N3CCC(C)(CNC(c4cnc(Cl)s4)=O)C3)=O)c12 N1(C(CC=CC)=O)CC2CC(NC(c3ccnc(C)n3)=O)CC1C2 CC(C)(C(=O)NCCCC1CCCN1C(c1cccc[n+]1[O-])=O)S(C)(=O)=O C(N=c1ccc2nnnn2[nH]1)C1CCC(NC(C(C)OCCC=C)=O)CC1 c1(OCC=C)cccnc1C(=O)NC1CCC(CNC(=O)Cc2ccc(Cl)s2)C1 c1(C(C)(C)C)cc(CO)nc(=NCC2CC23CC3(F)F)[nH]1 CCCC(C)CC(=O)NCC(c1ccccc1)N(C(=O)C#CC1CC1)C c1(C(C(=O)NC2C(C(C)NC(c3ccn(C4CC4)n3)=O)C2)O)cnn(C)c1 N1(C(c2cc(C)nc(O)c2)=O)CC=C(CC(=O)NCc2cnn(CCO)c2)CC1 N1(C(CC2(CNC(c3cnc(O)c(F)c3)=O)CC2)=O)CC2CC3CC2C1C3 CC1CC(CNC(C2CC3(CCC3)C2)=O)CN(C(=O)Cn2cncn2)C1 c1(CNC(C(CCCC#C)C)=O)nnc2n1CCN(C(=O)CC(C)SC)C2 C12(CNC(CCC=CC(C)C)=O)CC(NC(=O)COC3CCCOC3)(C1)C(C)O2 N1(C(C2C(OC)(OC)CC2)=O)CC(F)CC1C(N1CC(O)(C(=O)N(C)C)C1)=O C1(OC)CC2N(C1)C(=O)C=CC(=O)NCC2.C(C1CCOC1)=CC(=O)NC1CC1 c1(OCCC)cccnc1C(=O)NCC1(O)CCN(C(C2(O)CCSCC2)=O)C1 C1(NC(COCC=C)=O)CCN(C(c2cnc(SC)nc2O)=O)CC(C)(C)C1 n1(CC)nc(C(=O)NCC2CN(C(=O)CCc3cn(C)cn3)C3CC23)cc1O N(C(=NCC1CC1)N1CCC2=C(CCCC2)C1)Cc1cn(CC(F)(F)F)nc1 N1(C(Cc2n(C)nnc2)=O)CCC2(CCN(C(c3cc(Br)cn3C)=O)C2)C1 Cc1cc(C(N2C(C)CC(Nc3ccccc3C)CC2C)=O)c2c(C)noc2n1 N1(C(=O)CCc2cn[nH]c2)CCCC(CC(N2CCC2CF)=O)C1 c1(C(=O)NC(C)CC2CN(c3ncc(Cl)cn3)C2)cnc(C2CC2)nc1 N1(C(c2n(CC=C)ccn2)=O)CCC2CCN(C(=O)C(C)C#N)CC2C1 N1(C(CCCC=C)=O)CC(C)CN(C(=O)CNC(c2ccc(Cl)cc2)=O)C(C)C1 c1(C(=O)NC2C(C)CN(C(=O)CC3CCN(C)C3=O)C2)nc2c(s1)COCC2 C(CCCN=c1[nH]c2c(c(=NCCC3CC3)[nH]1)CCCCC2)OC.C1CS1 C(=O)(C(C(C)(C)C)OC)N1C(C(=O)N(C2CCC3CC23)C)(CC)CCC1 Cc1cccc(C(c2ccccn2)NC(c2snnc2C2CCC2)=O)c1 N1(C(CC2(C)CC2(Cl)Cl)=O)CC2CCC1C1CN(C(C3CC3C#N)=O)CC21 c1(OC(C(=O)NC2CCCC(NC(C(F)=CCC)=O)C2)C)ccc(F)c(F)c1 C1(CC)CC2CCC(C1)N2N(CC=CC(=O)SC1CCC1)C.C1(C=O)(CCOC)CC1 C(C(F)(F)C(F)(F)F)N(S(CC1(C(=O)OCC#N)CCCC1)(=O)=O)C(C)(C)C c1(C(=O)NC2C(NC(c3c(C)cc(SC)o3)=O)CCC2)cnc2cccnc2c1 CN1CC(O)CCC1C(N1CC(NC(=O)Cc2ccc(C3CC3)cc2)C(O)C1)=O C(CC(F)F)(C(=O)NCC(O)C1CC1)NC(c1csnc1Cl)=O C=C(C)CCC(C)N=c1[nH]c(=NC(C)c2cc(OC)no2)[nH]c2cccc(F)c12 N1(C(c2cnc(C)o2)=O)CCC(N(C(=O)CN2CCCNC2=O)C)CC1 C1(NC(C2N(C)C(=O)CC2)=O)CCN(C(c2c[nH]ccc2=O)=O)C12CC2 N1(C(c2cncc(OCC)c2)=O)CCC2CCC(NC(=O)C=CCF)C1C2 C(=O)(C(C)(COC)CC)NC(CCCC)CNC(c1cncc(C(F)(F)F)c1)=O N1(C(CCN(C(C)=O)C)=O)CCCCC(C2CN(C(=O)C(C)C(C)C)C2)C1 c1(CN2C(=O)CN(CC(COC)C(C)C)C2=O)cc(F)nc(F)c1F c1(C(N2C(CNC(CSCC(=O)OC)=O)CC(OC)C2)=O)cc2n(n1)CCCO2 n1(CC)cc(Cl)c(C(=O)NC(C)C(C)(C)NC(c2cn(C)nc2OC)=O)n1 c1(C(N2C(C)CC(CNC(CN(C(C(C)C)=O)C)=O)C2)=O)ccc2c(c1)NC(=O)C2 C(=O)(CCCC(F)(F)F)N(CCC(=O)Nc1c(CC)n(C)nc1)CCCO CCCCC(O)CC(=O)N1CC2(C1)SCCC2NC(c1cnn(C2CCC2)c1)=O CC1CC=C(C(=O)NC23CC2CN(C(c2coc(-c4ccsc4)c2)=O)C3)CC1 N1(C(C(CC=CCC)C)=O)CCC(F)(F)C(CNC(C2(CF)CCOCC2)=O)C1 c1(NC(C2SCCN(Cc3ccc(C)cn3)C2)=O)cnc(C#N)c(C(F)(F)F)c1 Cc1ccnc(C(N2CCC(F)(C(=O)NCCOC(=N)O)CC2)=O)c1F c1(N2C(C(=O)Nc3ncnc4[nH]ccc34)CC(O)C2)ncnc2ncc(Br)cc12 O(NC(=O)C(C)(C)C1CCCNC1)C(C1CCCC1)C.c12cccc(c1C)C(=O)N2 Cc1cc(F)c(F)cc1C(=O)NCCCc1cn(-c2cccc([N+](=O)[O-])c2)nn1 Cc1ccnn1CC(=O)NC(CNC(=O)CCc1cn[nH]c1)C1CC1 c1(C(=O)OC2COCC2N2CCCCC2)cnccc1N(C)C C(CC1CC1)CN=c1[nH]c(=NCC23CC(CCO2)C3)[nH]c2c1COC2 C1(N(C(=O)CC2CCC2)C)CCCCC1NC(C12CCC1C2)=O CS(=O)(=O)c1cccc(C(CO)NC(c2cc(O)cc(O)n2)=O)c1 c1(C(C(=O)NCCCOC)N(C)Cc2ccn(C(C)(C)C)c2)cc(Br)ccn1 c1(CNC(N2CCCC2c2ccccc2Br)=O)cnn2c1OCCC2 C(c1cncc(O)c1)=CC(=O)NC(CN(C(=O)CCC=C(C)C)CC)C FC1(c2ccccc2)CCN(c2cc(CN3CCCC3)ncn2)CC1 n1(CCC(=O)NCC2CC(CNC(C3(CC(F)F)CC3)=O)CO2)cccnc1=O c1(NC(C(CC)Br)=O)cc(-c2ccn(C(C)C)n2)cnc1OC C1(NC(C(=O)NCc2c(CNC)nn[nH]2)=O)CCCN(C(C)(C)C)C1=O Cc1ccc2c(n1)N(C(=O)NC(c1ccc(Br)cc1)C(N)=O)CCO2 C12(C(N3CCCC(CNC(c4c(OC)nccc4)=O)C3)=O)CCCC1C2(F)F N1(C(=O)CC2CCC2)CCCC(N(CCO)C(C2(Cl)CC2(F)F)=O)C1 CC1(C)CCCC(C(N2CCC3CC23C(N2CC(NC(=O)C3CC3)C2)=O)=O)C1 c1(C(=O)NCc2ccc(CC(=O)OCC)cc2)cc(C2CC2)cc(F)c1 Cc1noc(C)c1S(=O)(=O)NC1CC(Nc2cc(C(F)(F)F)ncn2)C1 CC1CN(C(=O)CC2CCN2C(=O)CCn2cccn2)CCC1N(C)C Cc1nc(CO)ncc1C(=O)NCC1(O)CCN(C(=O)C(=O)NCCC(N)=O)C1 CN1CCC(C(=O)NC2(C)CCCN(C(c3cccnc3N(C)C)=O)C2)CC1=O C12(C(=O)NCC3C(C)CCN(C(C4(SC)CCC4)=O)C3)CCCCC1C2(F)F C1(CNC(Cc2nc(COC)sc2)=O)CC(OC)CN1C(=O)CC1(O)CC1 N1(C(COCC)=O)CCC(C(F)(F)F)C(NC(=O)CCC2CC(F)(F)C2)C1 C1(C(C(=O)N(CCN(C(C)C)C)CC#N)C)CCCN(C(=O)OC(C)(C)C)C1 C(=O)(C(C(C)C1CC1)N1CCC(CN(C)C)CC1)NCC C(C(C)(C)C(=O)NCC(C)CN(C)C)N(C(c1ccc(C)s1)=O)C C1(C2CCN(C(=O)CN(C(=O)C(C)C)C)C2)(NC(C(C)OCC)=O)CC1 c1(C(=O)NC(C2N(C(C(COC)OC)=O)CCC2)C)ccn2ccccc12 CCCC(C)(O)CC(=O)N1CCC(CNC(C2CCC2)=O)C1 C(=O)(C(C)(C)CC(=O)N(C1CN(C(=O)C(C)C2CCC2)CC12CC2)C)OC C1(C)(NC(c2cnc(COC)s2)=O)CCN(C(=O)C(F)OC(F)(F)F)CC1 c1(C(C)C)ccc(C(C)CC(=O)NC2CCCC2Oc2ccccc2)cc1 c1(C(=O)NCCC2CCCCN2C(C2CCCO2)=O)ccn2c1CCC2 c1(C(=O)NCC2(NC(c3cnsn3)=O)CC2)cc(Br)ccn1 CCCCCC(C)CC(=O)NC(C)CC(C)NC(C1CCN(C)CC1)=O c1(OCC(=O)NCC(C)N(C(=O)CC#N)CC)ccc(F)nc1 C1(OC)(CNC(c2conc2C(C)NC(C2CCC(C)O2)=O)=O)CCOCC1 C1(CC(=O)NC(C)C(C)(C)O)CN(C(c2coc(C(F)F)c2)=O)CC12CC2 CCC(CC(=O)NCC#CC(=O)NC1CC12CCCC2)C1CC1 CC1CC(CNC(=O)CCCN2CCCCC2)CN1C(c1cc(C#N)c[nH]1)=O CS(=O)(=O)CC(=O)NCC(O)CCNC(=O)CC(c1cccs1)NC(N)=O c1(CN(C)C(C2CCNC2=O)=O)ccc(CNC(C2(n3cnnn3)CC2)=O)cc1 N1(C(CN(C(C)=O)C)=O)CC2CC(NC(c3ccc(F)cn3)=O)CC1C2 CCCCCC(O)C(=O)NC(C(=O)N1CC(F)C(F)C1)C(C)(C)O C1(S(C)(=O)=O)(C(=O)NCC2CN(C(C3N(CC)CC3)=O)C2)CCCC1 C1(CCC(=O)NC(c2cccnc2)C(=O)N(C2CCCOC2)C)CCCCCC1 N1(C(N2CCC(OC(F)(F)F)CC2)=O)CC(C2CC2)C(F)(CO)C1 C=C(Cl)C(C)(C)C(=O)N1CCC(CCNC(=O)Cc2n[nH]c(=N)s2)CC1 C1(N(C(CN(CC)CC)C)C)CCC1NC(=O)N(C)C C(C)(CCC(=O)N1CC(C2CCN(C(=O)C(Cl)=CCl)CC2)C1)OCC c1(OC)cc(C(N2CCCC2C=CC(=O)NCCNS(N)(=O)=O)=O)nn1C CC(C)CCC(C(=O)Nc1csnc1C1CC1)NC(c1cc(=O)n(C)cn1)=O CCC(C)CCNC(=O)CCNC1CN(C(C2(CC3CC3)CCC2)=O)C1 C(CCCCCC(=O)N1CCC(O)C1C)NC(CCCCCOC)=O N1(C(c2cc(C(F)(F)F)n[nH]2)=O)CCCC(N=c2ccnc(C3CCC3)[nH]2)CC1 C(CC1CC1)(CC(=O)NC1CCN(C)C1)NC(C(CC)=CC)=O C=CCCCCCCC(=O)NC(C(=O)NC(C)CC1(O)CCC1)C(C)C c1(CC(=O)N(CC(C)CNC(=O)CCc2cn[nH]c2)C)ccnn1C1CCCC1 C1(C(=O)NCC(C)(C)N(C)C)CCCCN(C(C2CCC3CC2CO3)=O)C1 c1(OCCC(=O)O)ccc(C(N2CC3C(NC(=O)CC4CC4)C3C2)=O)cc1 N1(C(C(C)N=[N+]=[N-])=O)CCN(C)C(CNC(C2CCC(O)CC2)=O)C1 CC1(C)CC(NC(=O)CC2CC3(C2)CN(C(C)(C)C)C3)CC(C)(C)S1 N1(CC=C)CCN(C(=O)CC(COC)NC(=O)CC2CC3CCC2O3)CC1 C1(NC(C2N(C(c3c(CC)cc[nH]3)=O)C(C(C)C)CC2)=O)CC2CC1C(O)C2O Cc1cc(O)c(CN2CCC(C(=O)Nc3cc(Cl)ncn3)CC2)cc1Cl C#Cc1cccc(C(=O)N(c2ncncc2C#N)CC2(C)CCNCC2)c1 C1(CC(C)C)(C(N(CCNC(=O)C(F)C2CCOC2)CC)=O)CCNC1=O CC1CN(C(c2cc3ccccn3n2)=O)CC(C)C1NC(=O)CC=CC(C)(C)C C1(NC(c2ccc(CSCC)cc2)=O)CCC2CN(C(C3CC3F)=O)CC2C1 N1(C(CCC(=C)Cl)=O)CC2CCC(CNC(c3ccn(CC)n3)=O)(C2)C1 c1(C(=O)NCC(CC=C)NC(=O)C(O)CSC)nccc2ncncc12 c1(CNC(C2(C)CCCN2C(c2ccn(CCF)n2)=O)=O)cccc(C#N)n1 c1(OC)cccc(Cl)c1C(=O)NCC(C1CC1)NC(c1cc2n(n1)CCC2)=O N1(C(c2ccc(-n3cccn3)cc2)=O)CC2CN(Cc3ccc(F)cn3)C2C1 C12(CNC(=O)C=C3CCCC3)CCCC1CN(C(=O)CCN1CCCC1=O)C2 c1(NCc2ccc(C(=O)OC)o2)ccccc1NC(=O)COC1COC1 C1(NC(C2(N3CCOCC3)CC2)=O)CC2CC1CN2Cc1cc[nH]n1 N1(C(C2CC3CC3N2Cc2cccc(Br)c2Br)=O)CCCC2(CCOC2)C1 C(CC(=O)N1CCCC(C)CC1)(C(F)F)NC(C(C1CC1)OCC)=O C1(CC=C)(C(=O)N(C(C(N)=O)C2CC2)C)CCN(C(=O)CCCC#N)C1 C(=O)(CCC(=O)N(CC(O)CNC(C1CC=CCC1)=O)C)Nc1nnc(CC)s1 c1(C(=O)OCC)cccnc1N1CCC(CF)(NC(=O)C(C)CC)C1 C(=O)(CC(O)CC(C)(C)C)N(CC(=O)OC)CC#C.C1CC(=O)NCCO1 c1(C(N2C(CNC(C(C)NS(CC)(=O)=O)=O)COCC2)=O)ccc(F)c(F)c1F CCC(CC(=O)NCCOCCOC)NC(C1CCCC(CF)C1)=O C(=O)(C(O)CC(N)=O)N1C(C(=O)NC(C#CCC)(C)C)C=CC1 CC1(C)C(CC(N2CC=C(CO)CC2)=O)CCN1C(C1CCCOC1)=O c1(C(N(C2CCN(C(=O)C(COC)NCC)C2)CC)=O)cc2nnn(C)c2s1 c1(C(N(C2CCC(NC(C3CN(C)C3)=O)C2)C)=O)cccc(-c2cnn(C)c2)n1 C=C(Cl)CC(C(=O)Nc1ccc(CO)nc1)NC(=O)CCC(N)=O C(=O)(C1=CCCS1)NCCOC1CCN(C(C(C)(C)N(C)C)=O)C1 C1(C(N(CCOCC=C)C)=O)COC2(C1)CN(C(=O)C(F)C(CC)CC)C2 N1(C(=O)N(c2nccc(C(F)(F)F)n2)C(=O)C2CC2)CCc2c(ccnc2O)C1 C1(CCC=C)(C(=O)N(C2COCC2O)C)CN(C(c2ccoc2C)=O)C1 c1(CC)[nH]nc(C(=O)NC2CCC(C)(CNC(C3C=C(C)CS3)=O)C2)c1C Cc1c(C(N2CC(C(N)=O)(CNC(C3CCCOCC3)=O)C2)=O)cccc1O c1(C(=O)NC2CCC(NC(C(COC)NC(C)=O)=O)CC2)ccnc2[nH]cnc12 N1(C(=O)Nc2c(SC)cnn2C)CCC(F)(C(F)(F)F)CC1 N1(C(CCN(C(=O)CC2CC3CCC2O3)CC=C)=O)CCC2CC1C(=O)O2 c1(C(=O)NCC2(NC(C=CS(C)=O)=O)CCCC2)ccn2nncc2c1 C1(C)(C(=O)NCC(CNC(C2C(OCC)C2)=O)O)CC(C(F)(F)F)C1 c1(C(=O)NCC(CNC(C2(CC)CC2(F)F)=O)CO)ccc2nsnc2c1 C(=O)(C(CCC(N)=O)NC(N)=O)NC12CC(NC(c3c(C)occ3)=O)(C1)C2 c1(C(CNC(CN(CC#C)C(C2CN(CC(C)C)C2)=O)=O)O)cccc(C)c1 N1(C(CC(=O)OCC)=O)CC2CC2(NC(c2ccoc2Cl)=O)C1 C(C(=O)NCC1(O)CCC(C)C1)(C(C)(C)C)NC(CC1CCC(C)CC1)=O CCC(C(=O)N(C)Cc1nc(CC(=O)O)cs1)N(C)C C1(C(N2CCN(C(=O)C#CC3CC3)C(CO)C2)=O)OCC2CCCC12 Cc1c(C(=O)NCCN(C(=O)Cc2cn[nH]c2)Cc2ccccc2)[nH]ccc1=O Cc1conc1C(=O)NCC1CC1CNC(c1cccn1C)=O N1(C(C(CC=C)(C)C)=O)CCC2(NC(c3cccn3C)=O)CCCC12 c1(-c2cc(OC)cc(F)c2F)nc2c(s1)CCN(C(c1cccc(Cl)c1F)=O)C2 N1(C(C2CC3(C2)CC3F)=O)CC2CN(c3cc(Cl)ncn3)CC2C1 C1(C(=O)NC2(CC=C)CN(C(C3CC(OCC)C3)=O)C2)CCCC(O)C1 C1(NC(C2(C(F)F)CC(=C)C2)=O)CN(C(c2cccc(NC(C)C)c2)=O)C2CC12 CC1CN(C(=O)COC(c2cn(C3CCOC3)cn2)=O)C(C)(C)C1 Cc1oc(CO)nc1C(=O)NC1CC2CC2C1.C12CCC(CC1)CNC2=O c1(C(=O)NCC(CC(C)C)NC(C(C(C)C)SC)=O)ncc(Br)cc1O c1(CN2C(CNC(=O)Cn3cccn3)CCC2)nc(Br)ccc1F N1(C(C2CCC(C)CC2)=O)CC2CC3CC2C1C3NC(c1cc(F)n[nH]1)=O C(=O)(C(C)(C)C1CCOC1)NC(C1CN(C(C2C(C)C2C)=O)C1)C c1(C(N2CC(NC(c3cc(OCC)n[nH]3)=O)C2)=O)cc(C(F)(F)F)ccc1O C1(NC(C=COCC)=O)CC2CN(c3ncnc(Cl)c3C(C)=O)CC2C1 C(=O)(C1CCCn2nccc21)NCC1(CNC(C2C(C)C2)=O)CCC1 C=C(Cl)C(C)(C)C(=O)NC1CN(C(c2sc(-c3ccc(C)o3)nc2C)=O)C2CC12 c1(C(=O)NCC(N(C(C(C=C)(F)F)=O)C)C2CC2)cnc(O)c(C(F)(F)F)c1 c1(C(=O)NC(c2cn(-c3cccc(CC)c3)nn2)C)c(C)ccc2ccccc12 c1(CNC(c2scc(CNC(C(C3CC3)SC)=O)c2)=O)nn(C)c(=O)n1C c1(N2CCCC(C)(CC)CC2)nc(=NCc2cc(OC)no2)[nH]c2cc[nH]c12 C=C1CCN(C(=O)C(C)CC2CCC2)C(C(=O)NC2CCCC2F)C1 c1(C(N2CCC(NC(C(CC)CC(C)C)=O)C2)=O)cc(F)cc([N+](=O)[O-])c1N S(=O)(=O)(c1cccs1)NC(C(=O)N(CC(CC)NC(C(C=C)(C)C)=O)C)C c1(C(=O)NC2(CC)CCCN(C(C3CCNC3=O)=O)C2)[nH]c2ccccc2c1C C1(NC(CC(C)C2CC2)=O)Cc2ccccc2N(C(C2C(C)(C)C2(C)C)=O)C1 C1(CC(=O)NCC2CC(NC(Cc3n(C)ccn3)=O)CC2O)CCOCC1(C)C c1(C(C(=O)NCCN(C(=O)COc2ccn(C)n2)C)OC)ccc(F)cc1 c1(C(C)=O)ccc(NC(c2ncc(Cc3ccccc3)s2)=O)nc1 c1(OC)nccc(C(N2CCC(N(C(=O)C3=NOC(C)C3)C)C2)=O)c1Br N1(C(C(C)Nc2nccs2)=O)C2CCC1C(NC(=O)CC1SC(=N)NC1=O)C2 C(CCN=c1[nH]c(C)cc(=NCCNC(=O)Nc2c(C)cccc2C)[nH]1)OC C1(NC(CCc2ccc(C)s2)=O)CC2CC(NC(=O)CC(C)c3ccco3)C1C2 c1(CC(=O)NC2(C)CC(NC(=O)C(C3CCCO3)F)C2)ccc(C(F)(F)F)cc1 C1(CCC)CN(C(=O)C(C)(C)SC)CC1NC(=O)COCC(=O)NCC Cc1ccc(F)c(C(=O)NCC2(F)CCC(CNC(=O)C(C)C3CCC3)CC2)c1 C1(C(=O)NCCCNC(c2cc(C)nn2C(F)F)=O)COc2cc(F)ccc2C1 c1(C(N2CCC(c3ccc(C#N)s3)C2)=O)cccc2c1CNCC2 c1(C(N2CC(CNC(C3C(C)C3)=O)C(C)(C)C2)=O)cncc2cc(Cl)ccc12 C(N=c1[nH]c(=NCCC#CCO)[nH]c2c1CCCCC2)C1(OCCO)CCC1 c1ccc2c(c1)CCN(CCSC1CC3CCC(C1)C3)C2.C1CO1 C1(CC)CN(C(C2CCC3(CCC3)C2)=O)CCN1C(=O)CNS(=O)(=O)N(C)C CC1(C)CN(C(C2CCC23CCC3)=O)CCC1NC(c1n[nH]cc1Br)=O c1(CNC(CCC#C)=O)ccc2c(c1)CCCC2NC(=O)CC1CCC12CCC2 N1(C(c2c(C(N)=O)nccn2)=O)CCC2CCCN(C(C3CSC3)=O)C2C1 C(=O)(C1CCCc2scnc21)N1CC2=C(CN(C(CSCC(=O)OC)=O)C2)C1 N1(C(=O)OC(C)(C)C)CC(CNC(C2(n3nccn3)CC2)=O)CC1(C)C N1(C(C=CC(=O)NC2CC2)=O)CCC(NC(C2(O)CCCC2)=O)C(CO)CC1 C1(C(N2C(CNC(CCC(=O)NCC)=O)CC2)=O)CCN(C)C(=O)C1 N1(C(C)=O)CCC(OC(c2nc(C)oc2N(C)C)=O)CC1 CC(N=c1cc[nH]cc1)C(=O)N1CC(CNC(=O)C=Cc2ncc[nH]2)CC1C CC1(C)C(NCc2cn[nH]c2)CC1CC(=O)Nc1ncccn1 N1(C(CC(CC(C)C)C)=O)CCN(CCNC(C2CC(C)(C)C2)=O)C2(CCC2)C1 N1(C(C2(COC)CC2(F)F)=O)CCC(O)(CS(C)(=N)=O)CC1 N1(C(CCC#CC)=O)CCCC12CCCN(C(C1CCCN1CC(F)(F)F)=O)C2 CC1(C)CCCC(NC(C2(NC(c3cnn4c3CCC4)=O)CC2)=O)C1 CC1CCC(NC(c2cc(O)nc(Cl)c2)=O)CN1C(c1ccc(C(F)F)nc1)=O C1(C(=O)Nc2cc(C)c(NC(=O)CCS(C)=O)cc2)Cc2ccc(F)cc2C1 CC(S(=O)(=O)c1ccc(CCS(C)(=N)=O)cc1)c1c(F)cccc1F C(=O)(C(C(C)(C)O)NC(=O)C(N)=O)Nc1cc(C)sc1 CC1CN(C(=O)C(C2CCCO2)C2CC2)CCN1C(=O)C=CC1CCOC1 N1(C(c2c(COC)cccn2)=O)CCN(C(=O)C2=COCCO2)C2(CCC2)C1 C=CCC(CNC(c1ccnnc1C)=O)C(=O)Nc1ccc(F)cc1O N1(C(C2(CNC(c3csnc3C)=O)CC2)=O)CCCCC1C(C(C)C)OCC c1ccc(CNC(c2ccc(C3CCCO3)s2)c2nnnn2-c2ccccc2)cc1 N1(C(CCC)=O)CC(NC(=O)Cc2cc(Br)ccc2O)C2(CC2)C1 C(C(C)(C(=O)NCCCCC(C)C)NC(=O)Cc1cc(C)cs1)SC C1(N(C(CC=CCNC(=O)CC2CCCCO2)=O)C2CC2)CCCCC1F CCC(C)(C(=O)N1CCCC(O)(CN(C)C(c2cc(C(C)C)on2)=O)C1)C(N)=O C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(C)C(CNC(=O)CSC(C)(C)C)C1 c1(C(=O)NCC2CCN(C(c3cc(C)c(Cl)s3)=O)CC2)cccc2ccnn12 C1(CC)CN(C(=O)C=CS(C)=O)CCC1CNC(c1cnc(C2CC2)nc1O)=O c1(C(N(CC(C)NC(C2(C(F)(F)F)CC(F)(F)C2)=O)C)=O)cc(F)cc(F)c1 C1(C(N2CCC(C)(NC(CC(c3ccc(C)cc3)C)=O)C2)=O)CC12CCSCC2 N1(C(C=C(C)C2CC2)=O)CCC(O)(C(C)NC(=O)Cn2cnc([N+](=O)[O-])n2)CC1 C(C(CC(=O)NCCc1ccc(F)nc1)OC)NC(C1CC(C(=O)OC)C1)=O Cc1ccc(C(=O)NCC2CC2CNC(=O)COc2ccc(F)cc2F)c(=O)n1C c1(C(=O)NCC(O)CC2CCCO2)ccc2nnc(-c3ccccc3)n2c1 C12(NC(C(C)C#N)=O)COC(CNC(=O)C(=O)NCc3ccc(F)cc3)(C1)C2 C(CNC(C1CCCN1Cc1cccc(OC(C)C)c1)=O)(C(C)(C)C)NC(C)=O C(CC(C)CC)(C(=O)NCc1nccc(C)c1F)NC(c1c(CC)nc(C)o1)=O C1(NC(C2CC(OCC)C2)=O)CC2CC(NC(=O)C(CC)NC(N)=O)CC12 c1(C(=O)NC(CNC(CCSCC)=O)(C)CC)cncc(O)c1 C(=O)(CCCCCCCC1CC1)N1CC(NC(c2c(CC)cco2)=O)C1 C(C(CN=c1[nH]n(C)cc1[N+](=O)[O-])C(F)(F)F)NC(C1CCN(C(C)C)CC1)=O CCC(CN=c1nc(N2CCC(C)(C(N)=O)C2)c2ccc(OC)cc2[nH]1)C(C)C c1(N2CCC(C#CC)C2)ccc(S(=O)(=O)NC(C)(C)C(C)O)cc1C#N C(=O)(CC(C(F)F)NC(C1CCNC(=O)C1)=O)NCCOCC(C)C N1(C(C23C(=O)CC(CC2)C3)=O)CCOCCC12CC2 c1(OC)ccc(CN(C(CCN2CCC(Cc3nccs3)C2)=O)C)cc1Cl C1(NC(CN(C)C(N)=O)=O)CCN(C(C23CC4CC2C3C4O)=O)CC1O c1(C(=O)NCC(C)CN(C(=O)C2=CCCS2)C)cc2scnc2[nH]1 C1(C(=O)NCCNC(C(C)(C)C)=O)CN(C(=O)CCNC(=O)CO)C2(CCC2)C1 Cc1ccc2cc(C(=O)N(CC(C)CNC(c3c(C)ncn3O)=O)C)nn2c1 c1(CC(N2C(CNC(CC)=O)CCCCC2)=O)cc(F)c(OC)c(S(N)(=O)=O)c1 C1(C(=O)NCC(C)NC(C2COC(=O)O2)=O)CCC(=O)N1 CCC(CC1CCCCC1)C(=O)NCCN(C(=O)C(c1cccc(Cl)c1)OC)C N1(C(Cc2c(C)n[nH]c2C)=O)CCCCC(CNC(=O)CSc2nnnn2C)C1 N1(C(COC)=O)CCC=C(C(=O)NC(CCO)C(F)F)C1 c1(C(=O)NCCOC2CCN(C(c3c(C)cn(C)c3)=O)C2)ncc(Cl)cc1O N1(C(C2CCC(=O)N2)=O)CC(C2CCCN(C(=O)C(F)(F)c3ccccn3)C2)C1 c1(C(=O)NCCN(CCOC)C(C2CC(F)C2)=O)cnn2c1C(C)CCC2 C1(C(=O)NCCC2CN(C(C(CC)(F)F)=O)C2)CCC(C)(C)OC1 c1(OC)ccc(C(=O)NCCNC(C2(OC)CCSCC2)=O)nc1N C1(CNC(C=C(C)C(C)(C)C)=O)CC(O)CN1C(=O)C(=Cc1c[nH]cn1)F c1(C(=O)NCCC2CCCN(C(C3(C)COC3)=O)C2)ccc2cc(F)ccc2n1 O=S1(=O)CCN(CCc2nnc3n2CCS3)C(c2ccccc2)C1 C(C(C)(C)C=C=C(C)C)(c1nnnn1Cc1cccs1)NCc1n(CC)ncn1 c1(CC)cc(NC(=O)C(CN(C)C)NC(=O)CC2CC(N(C)C)C2)cnc1C C(=O)(C(CC)(CO)OC)NC(CN(C(C(CCC)NC(N)=O)=O)C)C CC(CC(=O)NCCCN(C1CCCC1)C(c1cc2occc2[nH]1)=O)C(F)F C1(CC=C)CCCCN1C(=O)CC1CCN1C(C1CC2C=CC1O2)=O Cn1cc2c(C(=O)NC(CNC(=O)COC(F)F)C3CC3)cccc2n1 n1(CC)cc([N+](=O)[O-])c(C(=O)NC2CCCCC2NC(C2(C(F)(F)F)CC2)=O)n1 c1(C(=O)NC2(CNC(c3c(C)cc(N)s3)=O)CCCC2)cc2c(=O)[nH]ccn2n1 C(=O)(CCCC(=O)NC1CC(CNC(=O)CNC(=O)C2CC2)C12CCC2)N(C)C Cc1cnn2cc(C(=O)NCC3CN(C(C4COCCOC4)=O)CC3O)cnc12 C(c1cn(CC(F)(F)CC)nn1)=CCN(C)C(C1CCCN1CC(C)C)=O.CC=CC c1(CCC(=O)NC2CCN(C(C3(CCC=C)CC3)=O)C2)nncnc1O CCC(CC)(CC)C(=O)N1CC2CCC1C2NC(=O)C(C)SC c1(CN2CC(NC(=O)Cc3ccc(Br)cc3)C(F)C2)ccc(I)c(F)c1F c1(C(N2CC(C)(C)C(NC(=O)CC3CCOC3)C2)=O)cc2c(cc1N)OCO2 N#CC1(CC(N2CC=C(CNC(c3cnc(C(F)F)s3)=O)CC2)=O)CCOCC1 c1(C(=O)OC)cc(C)cnc1N1CCC(CNC(=O)CC2COCCO2)C1 N1(C(C2(CNC(C(CSC)O)=O)CCC2)=O)CCCC(C(N)=O)C1 C1(C(N(CCCNC(c2nc(=O)n(C)[nH]2)=O)C(C)C)=O)CN2CCN1C(C)C2 c1(C(=O)NC2(CNC(COCCCC)=O)CCCCC2)cccc(C2CC2)c1F CC1=C(C(=O)NCC2(C)CC(NC(C3(F)CCC(C)CC3)=O)C2)S(=O)(=O)CCO1 CCCCCC(CC)C(=O)N1CCCN(C(c2cnn3ncccc23)=O)C(C)C1 N1(C(=O)Nc2c(N(C)C)ncc(C(F)(F)F)c2)CCC(C)(CO)C(O)C1 C(C(CNC(=O)C(F)(F)C1(O)CCCC1)C(F)(F)F)NC(C1CCCCS1)=O CCCC(C#N)C(=O)N1CCC(NC(C2CC3(CCO2)CC3)=O)CC1C N1(C(C=CSC)=O)CCC2CN(C(=O)Cc3ncoc3C)CC2C1 N1(C(CC2CC(C)C2)=O)CC(C(N2CCCC2C2CC2)=O)C(C)(C)C1 N1(C(CC(C)CN(C)C)=O)CCC2(CC1)CCN(C(=O)CC(C)F)C2 c1(C(C(=O)NCCCOC)N(C(C)CS(C)=O)C)cc(I)ccc1F N1(C(C(C)C2CC2)=O)Cc2[nH]nc(C(=O)NCC(=O)NC(C)(C)C)c2C1 c1(NC(CC2CN(C(C(C)=O)=O)C2)=O)cccc(-c2ccn(C)c2)c1 C12(C(=O)NC(C(=O)OCC)(C)C)CC(CO)(CN1C(C1CCC1C)=O)C2 C(=O)(C1Cc2c(Cl)cccc21)N(CCCNC(C1C=CC=CC=C1)=O)CCO c1(C(=O)NCCC(=C)CNC(c2nccnc2C)=O)cc(=N)[nH]cc1Br N1(Cc2c(C)onc2)CCCOC(CNC(c2cnccc2C(F)(F)F)=O)C1 n1(CC)nc(C(N2CCCC2CN(C(=O)CC2CC(N(C)C)C2)CC)=O)c(C)n1 C(=O)(CC1=CCN(C(=O)C(C)NC=O)CC1)N(C)Cc1onc(CC)n1 N1(C(c2[nH]cc(C#N)c2)=O)CC2CCCCC2(NC(=O)C=CC2CCCO2)C1 c1(C(N(C2CCC(NC(=O)C(C)(F)F)CC2)C)=O)cnn2c1OCC2 C1(NC(=O)CCCN2CCCC2)CC2CC1CN2C(=O)CC1(O)CCOCC1 Cc1ccc(C(C)NC(=O)C(C)(C)C2CCCN2C(=O)CCc2nccs2)s1 CC(N=c1[nH]c(=NCC2(C)CC2(Cl)Cl)[nH]c2c1COC2)c1cccc(O)n1 c1(OCC(=O)NCCCNC(C(CC(=C)C)C)=O)cnc2ccccc2n1 c1(CNCCc2ccc(C)o2)nnc(-c2ccc(Cl)cc2)n1N C1(C(=O)NCC2COCCO2)CCCN1C(=O)CN1CCCC1 C1(C(=O)NCC2(O)CC(NC(C3(CC(C)C)CCC3)=O)C2)CCCCC1O C(C1CCCN1C(=O)CC(O)CN(C)C)=CC(=O)NC(c1cc[nH]n1)C n1(CC#C)c(C)cc(C(=O)NCCCCNC(c2ccc(Cl)cc2CC)=O)c1C N1(C(c2cc(OC)c(Cl)cc2)=O)CC2CCN(C(C3CCS3(=O)=O)=O)CC2C1 Cc1noc(C)c1C(C)CC(=O)NCCC(C)(C)NC(=O)CCc1ncco1 N1(C(C(C)(C2CC2)OC)=O)CC(C(=O)N2CCCO2)CCC1(C)C C1(NC(Cc2ccc(CC)cc2)=O)CC(O)CN(C(c2cnc(O)o2)=O)C1 C1(C(C)(C)C)CN(C(=O)C(O)CC2CCCC2)CCN1C(C1CC=CCC1)=O Fc1cccc(Cl)c1Cc1nc(-c2cccs2)nn1Cc1ccccn1 C1(CNC(CCc2cc(C)[nH]n2)=O)CCCC(NC(c2c[nH]cc2C(C)C)=O)C1 N1(C(CCC2(C)N=N2)=O)CCC2CCCC12C(N1CCC(C)(F)C1)=O C1(CC(=O)NC2(CCCNC(c3n(CC)nnc3)=O)CC2)CCCCC1C N1(CC=C)C(=S)NC(c2cccc(C)c2I)C(C(=O)OCC)=C1CC(F)(F)F C12(NC(CC3C(CC)C3(F)F)=O)CCCC1N(C(c1csc(C)c1)=O)CC2 c1(C(N2CCN(C(C=C(C)C)=O)C3C2COC3)=O)n[nH]c2c1CC(C)(C)CC2 c1(CN=C(NC2CC(OCC)C2)NC(C)CC)ccc(OC)c(F)c1 C1(N(C(C=COCC)=O)C)CC2CCC(C1)N2C(c1cnn2ccsc12)=O N1(C(C(CC)(C)C(N)=O)=O)CCC2(CC1)OCCC2NC(c1cnco1)=O c1(C2CCN(C(C(=O)NCC(F)F)CCCC3CC3)C2)ccc([N+](=O)[O-])c(O)c1 N1(C(c2cc(C(=O)OC)no2)=O)CC2CCCC(NC(=O)CCNC(C)=O)C2C1 c1(C(C)=O)cc(N2CCCC2(C)CNC(c2cc(C(F)F)nn2C)=O)nc(Cl)n1 C1(NC(C(CCC)NC(C)=O)=O)C2CCC1CN(Cc1cc(C)ccc1Br)C2 C1(C(=O)NC2CC2NC(C2(Br)CC2)=O)CCC(CSc2ccccc2)C1 N1(C(CCOCCOCC)=O)CCCC1C(=O)N(CCO)CCO.C1CC1 c1(C(N(CC(C)NC(C(CC(C)C)C)=O)C)=O)cc2ccccc2cc1F c1(C(C(=O)NC(C#C)CC)NC(C2CC2CC(C)(C)C)=O)cccnc1 C1(C(C)NC(C2CC(CF)C2)=O)CCN(C(c2cnn(C(F)(F)F)c2)=O)CC1 c1(NC(C2(C)N(C(c3cccc(N(C)C)c3)=O)CCC2)=O)cc(F)c(O)c(F)c1 C1(C(=O)NCC2C(NC(=O)C3=C(Cl)CCC3)COC2)CCc2cncn2C1 n1(CC(=O)NC2C(CNC(c3c(C(C)=O)cccc3)=O)C2)ccc(=O)n(C)c1=O C1(C(=O)NCC(c2c(CC)cccc2)NC(=O)C#CC2CC2)CCC(C)(O)CC1 c1(-c2cn(C(C(=O)NCCCCC)C)nn2)ccc2c(c1)NC(=O)C2 C1(C(=O)NC(C)C)CN(C(=O)CCc2nccn2C)CC1C c1(C(C)C)ccc(C(N2CC3CC2C3NC(=O)CC2CCC(C3CC3)O2)=O)nc1 c1(SC)nc(O)c(C(=O)NC2CCC(N(C(=O)C3=CCC3)C)C2)cc1C#N c1(C(N2C(CC(=O)NC)CCCCC2)=O)cc2nc(C)cc(C(F)(F)F)n2n1 c1(NC(C2(C)CCN2C(c2cc(C#N)cs2)=O)=O)ccc(CO)c(Cl)c1 C1(C(=O)NCc2snc(CC)n2)CCN(C(c2cc(C)n(C)n2)=O)C(CC)C1 C1(C)(C(N2CCC(CNC(C=C(C)C3CC3)=O)(CO)CC2)=O)CCCCC1(F)F C1(NC2C(C)SCCC2)CC2(CCNCC2)C1 c1(CNCC(C2CCCCC2)N(C)C)cc(F)c(F)c(Cl)c1F C1(C(=O)NCC2CCC(O)(c3ccccc3)C2)CC(c2ccccc2F)=NO1 C1(CC)(NC(=O)C=CC2CCOC2)CCN(C(c2ccc(O)cc2OC)=O)CC1 c1(C(N2C3(CNC(c4cc(OC)ncc4)=O)CC(C2)C3)=O)cc(OC)cc(C)n1 c1(NC(C(C(C)C)C)CNC(C2(C)CCCCC2)=O)c(C#N)cccc1[N+](=O)[O-] c1(C(N2CCOC(CN3CCCC3)C2)C(=O)NCCC)c2c(nn1C)CCSC2 N1(C(C2(C#N)CC=CC2)=O)CC2CCOC2(CNC(C2CCCSC2)=O)C1 C1(C(=O)NCCC2CN(C(=O)CC3COCC(C)O3)C2)(CC)CCCCCC1 c1(C(=O)NC2(CC)CN(C(C3CCCCC3O)=O)C2)c[nH]c2c(C#N)cccc12 C(=O)(CC(CC)C(C)(C)C)NC1(CC=C)CCN(C(c2ccc(O)cc2F)=O)C1 c1(C(N2C(C)CC(NC(=O)C=CCN3CCCC3)C2)=O)ccc(=O)n(CCF)n1 N1(C(C(C)(O)C2CCC2)=O)CCC2(CC1)CC(CNC(=O)C1=CC(O)CCC1)C2 c1(OCC)nc(C)ccc1C(=O)NCC1CCN(C(c2ncc(N)cc2Cl)=O)C1 C(CC(C(C)(C)C)NC(C1C(C(C)=O)C1(C)C)=O)N(C(C(COCC)(C)C)=O)C C(=O)(C(CCS(C)=O)N(C)C)NC(CC)CNC(c1ccn(CC)c(=O)c1)=O Cc1ccc(F)c(C(=O)NCC2(C(N3CCC3CF)=O)CC23CCC3)n1 C=CC1(CC(=O)NC(C)CCCC)CN(C(=O)CC2(C)CCOC2)C1 c1(C(=O)NCC(CCOC)NC(c2ccc(CC)s2)=O)ccccc1C1CCC1 C1(CNC(c2coc(C(F)F)c2)=O)CC(O)CN1C(C1CCCC1C(F)F)=O Cc1noc(C2CC2)c1C(=O)NCC1(NC(=O)CC2(C)CCOC2)CCC1 C1(NC(c2c(CC)n(C)cc2)=O)COC2C(NC(=O)CC3CCOC3C)COC12 Cc1nn(C)c(C)c1CCC(=O)NC(C)(CNC(C1CCCC(F)C1)=O)C1CC1 C1(CCNC(C2C(=C)C2)=O)CN(C(=O)Cc2cccc(O)c2)CCS1(=O)=O C1(CC(=O)NCC(CC)NC(=O)CN(C)C(c2cccs2)=O)CCCCN1C c1(OC)cc(CN2CCCC(CNC(c3cccnc3O)=O)C2)ccn1 Cc1nc(NC(CCNC(=O)Cn2cnnn2)C(C)C)cc(SC(C)C)n1 c1(C(C)C)cc(Cl)ccc1NCC(CNCc1cccs1)C(C)C N1(C(CC(CNC(CSCCC(C)C)=O)C)=O)CCn2c(C)nnc2C1 C1(NC(C(C(C)C)C2CCC2)=O)CC2CCCC(C1)N2C(C1CC(O)(C#N)C1)=O c1(NC(C(CC#C)N(C)C(C)=O)=O)cccn(CCOC)c1=O c1(C(C)N(C)Cc2cn(C(c3ccc(Cl)cc3)C)nn2)nnc2n1CCCC2 c1(OC)ncc(NC(c2cnc(CNC(=O)CC3CCCC3)nc2)=O)cc1C C1(CNC(c2ccc(N(C(C)=O)C)cc2)=O)CN(C(=O)CCF)C2COCC2O1 N1(C(C(C2CN(C(=O)CNC=O)C2)OC)=O)CC2CCC(C1)O2 S(=O)(=O)(c1ccc(NCC2CCCCN2CCO)cc1Cl)NC1C(C)CCC1 CC(C)C(C)C(CNC(=O)CN1CC(C)(C)C1)NC(C1(c2ccnn2C)CC1)=O C1(NC(CC2C(C)CCO2)=O)CCN(C(c2cnsc2)=O)CCC1CO C1(C(N2CC(N(CCOC)C)C2)=O)(CNC(=O)C(C)c2ccco2)CC(C)(C)C1 C(C(C(C)(C)C)NC(=O)CCC1CC1)NC(C1CC(C(F)(F)F)(OC)C1)=O CCCC(C)(C)CC(=O)NC(C)(C)COCCCNC(C1CCN(C)C1CC)=O N1(C(c2nc(COC)oc2)=O)Cc2[nH]nc(C(=O)N(C3CCSC3)C)c2C1 N1(C(C(=O)NC(c2ccc(C(C)C)cc2)C)=O)CCC2(CC1)CC(=O)NCC2O C(=O)(C(C(=O)N(C(C)(C(=O)Nc1cccnc1C)C1CC1)C)OC)OC C1(C(=O)NC2CCC(C)N(C(=O)Cn3nccn3)C2)CCc2ccnn2C1 C1(CC=C)(NC(c2n[nH]c(=N)s2)=O)CCN(C(=O)COc2ccccc2OC)C1 C1(c2nnnn2CCSC2CCCC2)(NCCSC(C)C)CSCCSC1 CC1CCN(C(=O)C(C)CCO)CC1NC(C1CCCN1C1CCCC1)=O N1(C(Cn2c(C)nnn2)=O)CCCCC1CCC(N1CC(C)(N(C)C)C1)=O C1(C(N2CC(CC(C)NC(c3occ(C)c3)=O)C2)=O)C2CCC(C2)C1(C)C C(C(C(C)C)C(C)C)(c1n(-c2c(CC)cccc2)nnn1)NCCc1ccns1 C1(CNC(=O)CN2CCOCC2)CC2(CCC2)CN1C(c1ccc(CO)cc1)=O N1(C(CC(C)SC)=O)CCOCC(CNC(c2cc(SC)oc2C)=O)C1 n1(CC(=O)NCCN(C(c2[nH]ccc2C2CC2)=O)CC)ccc(O)nc1=O N(C(=NCCCCC(F)(F)F)NN(C)C(=O)C1CC1)Cc1ccc(CC)cc1 C1(CC(=O)N(CCCNC(c2ncccc2F)=O)CCO)CCN(CCF)CC1 c1(C(=O)NCCCNC(C2CC2C(F)F)=O)c[nH]cc1-c1ccc(Cl)s1 CC1CC(C(N2CCCC(CC3CC3)C2)=O)CN(C(C2(Cl)CCCCC2)=O)C1 c1(C(=O)NC2CC(C)(NC(C=C3CCC(C)C3)=O)C2)c(C(F)(F)F)ncn1O C1(CC)CN(C(C2CC(O)C2)=O)CC1C(=O)Nc1ccc(F)cc1 C(CN=C(NCC(c1cccs1)OC)NC(C)C1CC1)c1onc(CC)n1 C1(C(=O)NC2C(NC(c3ccnc(OC(F)(F)F)c3)=O)CC2)C(F)(F)C12CCC2 Cn1cnc2c1CCCC2C(=O)NCCCCNC(=O)C(C)(C)C1CCOC1 C(F)(c1ccccc1)=CC(=O)NC(CCN(C)C(C1CC1(C)C(F)(F)F)=O)(C)C c1(OCCCNC(C)=O)ccc([N+](=O)[O-])c(C)c1.C1(C)(C(F)F)C(=O)N1 c1(N2CCCC(O)(CNC(c3cncc(OC)c3)=O)C2)[nH]cnc2nc(Br)cc1-2 c1(C(N(C2CCN(C(c3ccncc3)=O)C2)CCC)=O)nnsc1C c1(C(=O)NCC2C(NC(c3c(OC)cccn3)=O)CCC2)cc2ccncc2[nH]1 c1(CC(N2CC(O)(CNc3nccc(CC#N)n3)C2)=O)ccc2n[nH]cc2c1 c1(OC(C)C)ncc(NC(C2CCCN2Cc2c(Cl)cccc2I)=O)cc1Cl Cc1cc(CN(C)Cc2ccn(CCc3cccs3)n2)nc(C)c1 N1(C(c2ccoc2C)C(=O)NCCOCC)CCCC(c2ccccc2)C1 C1(CNC(c2c(CCC)nco2)=O)CCC2(CCN(C(=O)C(C)(F)F)CC2)O1 C1(C#N)(C(N2CC=CC(C(N3CC(N(C)CC)C3)=O)C2)=O)CCCCC1 C1(C(C)N(C(CCC=CC)=O)CC)CCN(C(c2sccc2-n2cccc2)=O)CC1 CCC(C)(C(=O)OC)NC(C1CC=CCN1C(C1C(C)(C)C1(C)C)=O)=O C(=O)(C(=O)NCCOCCN1CCCC1)NCCC1C(C)C1 CC1CCC(=CC(=O)NCC=CC(=O)NC2(CCF)CC(O)C2)CC1 CC1(C)C(C(=O)NCC(=C2CN(C(c3cncnc3)=O)C2)F)CCS1(=O)=O N1(C(CN(C2CCC2)C)=O)CCC(F)C(NC(c2c(Cl)nsc2Cl)=O)C1 C1(N(c2ncnc(=N)[nH]2)CCO)CS(=O)(=O)CC1NC(=O)CCOC1CCCCC1 Cc1[nH]c(=N)nc(O)c1CCC(=O)NCC(C)(O)CNC(C1(C)CC1(F)F)=O O(NC(=O)C(C)N(C(c1ccc(O)cc1)=O)CC)CC(=C)Cl C1(CNC(C(C2CCOC2)OC)=O)CN(C(C2CC(F)(CO)C2)=O)CCN1C C1(NC(C(CCC)C)=O)CC2(CCN(C(c3ccc4c(n3)NCC4)=O)C2)C1 C1(Cn2cc(COCC)nn2)CCCCN1C(=O)Cc1cn(OC(I)Br)nn1 c1(C(=O)NCC2CN(C(C(C)=CC)=O)C2)cc(F)cc(C)c1I c1(C(=O)NC2(C)CN(C(C(CC)O)=O)C2)ccc(-c2nc[nH]n2)nc1 N1(C(C(c2ccc(OC)cc2)CC)=O)CC2OCCN(C(c3cc[nH]c3)=O)C2C1 c1(OCC2COC(C(=O)OC)C2)cc(=O)n(C)cn1 C12(CNC(CCSCCC)=O)CC1CN(C(=O)COc1ccc(C)cc1)C2 c1(C(=O)NC2C(CC(=O)N(CCC(F)(F)F)C)C(O)C2)cn(C)ccc1=O C(=O)(C#CC(C)(C)CNC(=O)C(C)OCC1CC1)N1C(CC)CCCC1 C1(NC(C2(CCNC(C3C(C)C3C)=O)CC2)=O)(CO)CCOCC1 C12(C(=O)NC(C(C)S(N)(=O)=O)=O)CC3CC(CC(C3)C1CO)C2 C1(C(=O)NC2CN(C)C(CO)C2)CC(N=[N+]=[N-])CN1C(c1ccc(O)cn1)=O Cc1cc(=O)n(C)nc1C(=O)NC(C)CCCNC(c1n[nH]cc1C(F)(F)F)=O c1(C(=O)OC)cc2c(nc1NC1CN(C(c3c[nH]cc(C)c3=O)=O)C1)CCC2 Cn1nc(C(=O)NC2(CNC(=O)CC3CC(=O)C3)CC2)c2c1CCSC2 N1(C(c2ccn(C(F)(F)F)n2)=O)CC2CCOC2(CNC(=O)C(F)(F)C2CC2)C1 n1(CCC)cc(C(=O)NCCCNC(=O)C(O)C(C)c2ccccc2F)c(C)n1 c1(CC)oc(C(=O)NC(C)(CNC(=O)Cc2ccc(Br)cc2)CC)cc1C CN1CCN(C(C2COCCN2CC(F)F)=O)C(CNCC2CC3(CC3)C2)C1 n1(C2(C)CC2)nnnc1C(C)(C1CC1)NCc1nc(C2CCC2)no1.C1(C)CCCO1 N1(C(C2CN(C(CC#N)=O)C2)=O)CCCCC1CO C1(NC(CC2(NC(C)=O)CC2)=O)C2CC(O)C1N(C(=O)CC13CCCC1C3)C2 C1(C(N2CCC(CN(C(=O)CCN3C(=O)CCC3=O)C)C2)=O)CC(C2CCC2)C1 CCCC(CNC(=O)CCCCNC(C)=O)C(=O)N(C1CCCNC1=O)C N1(C(C)=O)CC2CC2(C(=O)NC(C)CN(C(=O)CCc2nc(O)n[nH]2)C)C1 N1(C(C=CCN(C)C)=O)CCCC(Cn2cc(C3(C)CCCO3)nn2)C1 C1(C(=O)OC)CCCCN1CCN(C)C(=O)OC(C)(C)C.c1ncccn1 C1(C(=O)OCC)CCCCCN1C(=O)CSC12CCCC1C2Br C(C)(C)(CCC(=O)NC)NC(CC(CC)N)=O c1(CC(N2CCC(C3N(C(c4nc(C)sc4)=O)CCC3)C2)=O)sc(C)nc1C C(=O)(CCC(C)(C)C#N)N1C(CCNC(C(C(C)C)CN(C)C)=O)CCC1 C1(NC(c2cn(C)nn2)=O)C=CCN(C(=O)CC(c2cccs2)NC(N)=O)C1 N1(c2cccc(C(=O)NCCn3c(C)cnn3)c2)CC(C)OC(C)C1 C1(NC(C(Cc2cn[nH]c2)NC(=O)CCc2cccs2)=O)C2CCCC1COC2 C1(NC(C2C(=C)CC2)=O)CCCCC12CCN(C(c1n[nH]cc1[N+](=O)[O-])=O)CC2 C(=O)(C1CCCc2sccc21)NCCC(C)NC(C(C(=O)OC)OC)=O c1(NC(C2CCC2Cc2ccccc2)=O)cncc(OCC(F)F)n1 c1(C(C(=O)N(CC(C)N(C)C(c2cscc2F)=O)C)SC)ccccc1 CCCC(CCCNC(=O)CCCF)NC(=O)CC1(C)CCCC1 Cn1c(C(N2CC3CCCC3(NC(C3CCC(O)CC3)=O)C2)=O)cc2sccc12 C(=O)(C1=CCC2CCC1N2C(c1ccc(C)nn1)=O)NC(CC)C(C)(C)C c1(C(=O)NC2CC(CNC(C3(CC#C)CCC3)=O)C2)ccc(C)c(C)c1O N=c1[nH]nc(CCNCc2ccoc2C(F)(F)F)s1 C1(CNC(C(CCSC)OC)=O)CN(C(=O)Cc2cc(C)ccc2F)CC1(C)C c1(C(N2CCCC(N(C(C(C)C#N)=O)CCO)C2)=O)cc(F)cc2c1NCCC2 c1(SC)nccc(C(=O)NCC2(C(C)(C)O)CN(C(=O)CCNC(N)=O)C2)n1 C(CN1CCOCC1)(CC(F)(F)F)NC(CCCC)(C)C.C1(=O)NO1 N1(C(CCCCCC)=O)CCC(C=C)(C(=O)NC(C2CCOC2)CC)CC1 c1(OC)cc(CC(C)NCC(c2ccc(Cl)cc2)C)cc(OC)c1OC CC(CS(C)(=O)=O)C(=O)N=c1cc(C2CCOCC2)[nH][nH]1 C1(C)(C(N(C2CC(NC(c3cn(CC)nc3C)=O)C2)C)=O)CCCN(C)C1 c1(C(N2CCN(C(N(C)C)=O)CC2)=O)c(-c2ccc(I)cc2)ccc2c1OCO2 N1(C(c2c(OC)cc(F)cc2)=O)CCCC(C2(NC(=O)C(C)=C(C)C)CC2)C1 CC(C)C(C(=O)NCC12CCC(CC1)N2C(c1ncccc1N)=O)C(C)C C=C(Br)CC(=O)NCCOCCNC(=O)Cn1ccnn1 N1(C(C2(CC(C)=O)CC2)=O)CC(C(=O)NC2CCN(C(C)C)CC2C)CC(C)C1 c1(C(=O)NC2CC3(CC(NC(c4cc(C)nnc4)=O)C3)C2)c(N)ccc(C)c1F C(=O)(CCCCCCCC1CC1)NC1CCN(C(c2cnc(C)s2)=O)C1C1CC1 N1(C(Cn2c(C)ccn2)=O)CC2CCC(C1)N2C(C1CC(F)C1)=O CC1CC(CC(=O)NCCN(C)C(c2cc3cnn(C)c3s2)=O)CC(C)(C)C1 C(=O)(C(C)(C(F)F)c1ccccc1)NC1C(C)CN(C(c2cc(O)nn2C)=O)C1 C1(C)(NC(c2ccnc(C)n2)=O)CCCN(C(c2ccc(C)c(F)n2)=O)C1 Cc1ccc2[nH]c(C(N3CC(NC(=O)CCC(C)C)CC34CCCC4)=O)cc2c1 C(=O)(C1(C)CCn2ccnc21)N1CCCC(NC(C(C)n2cnnn2)=O)C1 C1(C(N(C2CC3CC3C2)C)=O)CN(C(c2cc(C3CC3)[nH]n2)=O)CC1(F)F N1(C(C2N(CC)CC2)=O)CCC(F)C(NC(C2CN(C)C2)=O)C1 c1(C(N(C2CCC2(C)C)C)=O)c(F)ccc2ccoc12 C(=O)(C(CC(C)C)C(N)=O)NC1CCC(CC(=O)N(CCOC(C)=O)CCO)CC1 C1(CNC(CC2(C)CC2)=O)CC2(CCN(C(C3(F)C(C)(C)C3(C)C)=O)CC2)C1 CC(CC(C)(C)C)C(F)C(=O)N(C)CCN(C)C(c1ccnc2[nH]ncc12)=O C1(C(N(CCCNC(c2ccc(Cl)o2)=O)C2CC2)=O)C2Cc3ccccc3C12 C(N=c1[nH]c(N2CCc3[nH]nc(O)c3CC2)nc2ccsc12)c1c(O)nccc1 C1(N(C)C)CN(N2CC3(CC=CC3)C2C2CC2)CC1F c1(OCC(C)C)cccc(-c2ncsc2C(=O)NCCc2ccncc2Br)c1 c1(OC(C)C(=O)NC2C3CCN(C(=O)CCc4n[nH]c(=N)s4)C23)ccc(F)cc1 C(=O)(CC(CC)C(C)C)N1C(C(=O)Nc2cnc(CCC)nc2)C2CCC1C2 N1(C(c2n[nH]cc2F)=O)CCCc2ccccc2CC1 C1(C(=O)NCCOCCC)CC(F)CN1C.c1(C(=O)OC)nc(OCCOC)co1 c1(OC)ccc(CN2CCC(C(N3CCOCC3)=O)C2)c(Cl)n1 Cc1nc2cccc(C(=O)NC3CCN(C(C4CCCO4)=O)CC(O)C3)c2s1 c1(OC)cccc(SCC(=O)NC2CCC(NC(C3(C)CC3F)=O)CC2)c1 C1(CNC(C2CC(OC)CC2C(F)F)=O)COC2(CCC(C)CC2)O1 c1(C(=O)NC(CCNC(C(C)=C2CC2)=O)C)cccc(C2CNC(=O)C2)c1 N1(Cc2cccc(CC)n2)CC(C)Oc2cc(C)ccc21 c1(C(=O)NCC(C)N(C(c2cccnn2)=O)CC)cc(Br)cnc1O C1(CC)CC(O)CCN1C(C1CCN(C(c2c[nH]cc2C2CC2)=O)C1)=O C(=O)(CC(F)(F)C(F)F)NC(C(C)(C)NC(c1scc(C)c1Br)=O)C CN1CCC(CC(=O)NCC2CN(C(=O)CN3CCCC3=O)CC2O)CC1 O=C1CCC(CCC(N2CCC(C(F)CNC(=O)CCCC3CC3)CC2)=O)CN1 c1(CC)cc(N2CCOCC2C(C)C)nc(C(C)(C)C)n1 S(=O)(=O)(c1cnn(C(C)C)c1)N1CCCC(CC(C)C)C1 N1(C(CC2CN(C)C2)=O)C2CCC1CC(NC(C1COC3(CO)CC1C3)=O)C2 c1(OC)ccc(C(N2CCN(C(=O)C(C)n3cncn3)C(C)C2)=O)cc1Br Cc1cccc(CN(C(=O)C(C2CC=CCC2)NC(C2CCC(=O)NC2)=O)C)c1 C12(C(=O)NCCC(CC)C)CCC(CN(C(=O)C=Cc3cnn(C)c3)C1)C2 c1(C(N2CCCC(N(C(C(C=C)(C)O)=O)CC)CC2)=O)cc2ccsc2n1C C(=O)(C(O)CC1CCCCC1)NC1CC(NC(=O)CCNC(c2ccco2)=O)C1 N#Cc1ccc(N2CCCC(CCNC(=O)C3=COCC3)C2)c([N+](=O)[O-])c1 CC(C)CC(C(=O)NC(c1ccco1)CO)ONC(C12CCCN(CC1)C2)=O C12(C(N(CC(CNC(CC3(C=C)CCOCC3)=O)C)C)=O)C3CC(CC13)C2(F)F C1(CNC(CC=CC=C)=O)CC(NC(c2cc(C)nc(O)n2)=O)C12CCC2 Cc1nc(NCc2ncc(C(C)C)o2)cc(N(CCC(F)(F)F)C)n1 c1(-c2c(C(=O)NC3(CCNC(C4CC4CF)=O)CCC3)nco2)cccc(F)c1 CC(CS(C)(=O)=O)C(=O)N1CC(C)C(C)(C(=O)NCC(N2CCCCC2)=O)C1 N1(CC(=O)NC(C)CN(C(=O)C(c2cnccn2)C)C)CCC(=O)NC1=O C1(C(=O)NCC(CCOC)NC(=O)CC(C)CN(C)C)CCCCCC1 N1(C(C2C(C)C2)=O)CC2OCCN(C(=O)C=C3CCC3)C2C1 Cc1cc(C)c(C(=O)NC2CCN(C(c3cc(C)c(Cl)s3)=O)CC2C)c(C)n1 C1(CC=C)(NC(=O)C(CC(C)C)OC)CCCN(C(=O)C(O)COC)C1 N1(C(C2C=CCN(C(c3ccc[nH]3)=O)C2)=O)C(CO)CCC12CCC2 C(CNC(c1c(C)oc(C)c1C)=O)(C(C)C(C)C)NC(COCCCCC)=O Cc1c[nH]c(C(N2CCCC(N(C(=O)CSCc3ccccn3)C)C2)=O)cc1=O NS(=O)(=O)c1csc(C(C(=O)Nc2ccccc2Cl)N(C)CC2CC2(F)F)c1 c1(C(=O)NC(C)C(C)NC(c2cccs2)=O)sc2sccc2c1Cl C(C(C(=O)NCC(C)C(F)F)n1cc(Cn2cccn2)nn1)OCC C1(CNC(C(C(C)C)SCC)=O)CCN(C(c2sncc2CC)=O)C1(C)C c1(OC)cc(C(=O)NC2CCOCC2NC(C23CCC(CC2)C3)=O)ccn1 c1(CC)cc(C(=O)N(C)CCc2ccccc2O)c(C)o1 c1(C(=O)NCC(C)(O)CNC(C2CC(F)C2)=O)cc(C#N)cs1 c1(OCC)cc(C(=O)N(CC(C)CNC(=O)C(C)(C)C2CC2)C)oc(=O)c1 N1(C(CCC(C)(F)F)=O)CC2CCC(CNC(=O)CC3CN4CCC3C4)C2C1 c1(C(=O)NC(C(C)NC(CC=C)=O)(C)C)cc(C#N)n(C)n1 C1(CCNC(C(c2cnn(C)c2)C)=O)CCCCN1C(=O)CCN1CCOCC1 c1(C(=O)NC(C)CN(C)C(C2CCCOC2CC(F)(F)F)=O)cc(N)cc(F)c1 c1(CC)noc(CCCC(=O)NC(C2CCN(C(=O)CCCC3CC3)C2)C)n1 N1(c2cn(C)nc2)CC(NC(=NCCC2CC3CCC2O3)NC2CCC2)CC1=O C1(CC(N2CCC23CC(F)C3)=O)CCCC2(CCC2)O1 CC1CN(C(c2ncoc2-c2cnn(C)c2)=O)CCC1N(C(=O)CCC(N)=O)C C1(C(=O)NC2C(NC(C3(C)CCN(C)C3)=O)CCCC2)CC2(CCCCC2)C1 c1(C(CC(=O)N2CCC(CCCO)C2)CC2CCC2)c(F)cccc1Br N1(C(C(c2ccc(CC)s2)=O)=O)CCC(CCNC(=O)C2=NOCC2)C(F)(F)C1 C1(C)(NC(c2n(C)ncc2)=O)CCN(C(=O)C=Cc2nccs2)CC1 C1(C(=O)NCc2c(C)nccc2)CC2CCC1N2C(c1cnco1)=O C=CCC(C(=O)NCCCCC(=O)NC(CN(C)C)CCO)NC(C)=O c1(CC(=O)NCCO)cccc(C2CC2)c1.CC1C(C(C)NCCC2CC2)C1C C(C(C(=O)NC(C)CCCN(C)C)C(C)C)NC(CC1CC(=C)C1)=O N1(C(CN(C2CCS(=O)(=O)CC2)C)=O)CC2CCC1C(C(=O)N(C)C1CC1)C2 CCC(F)(F)C(C)(C)C(=O)N1CCCC2(C1)CN(C(=O)C=Cc1cnc(C)s1)C2 C1(C)(NC(c2c(NC)nc(C)nc2C)=O)CCOC12CC2(F)F c1(C(=O)NCC2CN(C(C3CCC3)=O)CC23CCC3)cccc2cc(F)ccc12 C1(NC(C(CC)(CC)CO)=O)CCC2CN(C(=O)Cn3cc(N)cn3)CCC2C1 N1(C(C2C(C)C2C)=O)CCC2(C1)CN(C(c1cc[nH]c(=N)n1)=O)CCO2 CC(C)CC(C)CC(=O)NC1CN(C(C2CCS(=O)(=O)CC2)=O)CC1C c1(C(=O)OC)ccc(CN(C(C2CCC(Nc3cc(C)on3)CC2)=O)C)c(F)c1 C1(CCNC(Cn2c(C)ncc2)=O)CN(C(C2CC=CC2)=O)CCCO1 O=C(C#CCNC(C1C2CCCC(=O)C12)=O)NOCCCO C1(C(N(CCCC(=O)NCc2[nH]nc(CC)n2)C(C)C)=O)CCCN(C)C1 C1(NC(C2CCN(C(C)=O)C2)=O)CCN(C(c2cn(C)[nH]c2=N)=O)CC1 C1(NC(c2c(SC)cnn2C)=O)CCN(C(c2cncc(C3CC3)c2)=O)CC1C c1(C(N2CC3(CC(NC(C4CCC(OC)C4)=O)C3)C2)=O)cc2c(Cl)cncc2s1 C1(NC(CC(CC)C)=O)CCC(C)N(C(=O)CC(C)C(F)F)C1 C1(NC(CCC(=O)NCC)=O)CCN(C(=O)CC2COCC(C)(C)O2)C1(C)C c1(N(C(C(=O)N(C)Cc2onc(C(C)C)n2)=O)C)cccc(NCCCCO)c1 Cc1cccc2cc(C(N3CC(CNC(=O)C(C)(C)C4CCCCO4)C3)=O)[nH]c12 N1(C(C(CCSC)N(C)C)=O)CC2(C1)CN(C(=O)Cn1cnc(C(N)=O)n1)C2 C=CCC(C)(O)C(=O)N1CCC(F)(C(=O)NCC(N)=O)CC1 CC(C)CCCOCC(N1CCC1(C)CC(=O)N(CC(F)F)CC(C)O)=O C1(C(N(CC(C)NC(=O)C(C)(F)F)C)=O)CCc2cc(Br)ccc2O1 c1(OC2CC(C3CCN(C(=O)OC(C)(C)C)CC3)C2)ccc2nccnc2c1 C1(NC(C)=O)CN(C(=O)Cc2cncc(F)c2)C2(CCC2)C1 CC12CCCC1N(C(=O)NCCC(=O)NCCc1cccnc1)CCC2 n1(CCC(=O)NCC(C)NC(=O)CCC(=O)c2ccc[nH]2)ncn(C)c1=O c1(C(=O)NCC2N(C(C3COC(=O)C3)=O)CCN(C)C2)cc(F)cc2ccoc12 Cc1c2c(nn1C)CC(NC(=O)NCCc1nnc(Br)n1C)CC2 C1(C(=O)NCC(CCC)NC(c2cc(C)ccc2O)=O)CCc2n[nH]cc2C1 N1(C(c2cnc(C)o2)=O)CC(NC(=O)CCNC(c2ccncc2)=O)C(C)C1 C1(COC)C(O)C(O)CCN1C(C1CCN(S(=O)(=O)C(F)F)C1)=O c1(CCN(CCC)C)nc(-c2cccnc2)nn1CC1CC(F)(F)C1 C(CCCCCCO)NC(C1C(O)CCN1C(=O)Cc1ccon1)=O Cn1ncc2ncc(C(=O)N(c3ccccn3)CC3CC3)cc12 C1(NC(C2(CCOC)CCCC2)=O)CN(C(C23COC(CCO2)C3)=O)CCC1C C1(NC(C2CC=CCC2)=O)CCCC1CNC(C1(C(F)F)CCCC1)=O C(CC(CC)C(=O)NCC(O)CNC(c1ccnc(OCCO)c1)=O)=CC c1(C(N(C2CCCN(C(C3(C)CCSCC3)=O)CC2)CC)=O)cc(Cl)ccc1F N1(C(C2C(C)OCC2)=O)CCC2(CCCN(C(c3ccc4c(c3)OCC4)=O)C2)C1 CCCCCCCCCC(C)CC(=O)N1CC2(CCN(C(=O)CCS(C)=O)C2)C1 n1(CC(=O)NC2C(CNC(C(c3[nH]c(=N)sc3)=O)=O)CC2)cnc([N+](=O)[O-])n1 C1(NC(C(CC)SC)=O)CC2CC(C1)N(C(c1cc(C3CC3)ncn1)=O)C2 c1(NCC(C)CNC(C2CCS2(=O)=O)=O)ncnn2cccc12 c1(NC(=O)NC)cccc(C(=O)NCCNC(C2CN(C(=O)C(O)CC)C2)=O)c1 O=C(C1=CS(=O)CCC1)NC1(CNC(c2cc(C3CC3)ccc2F)=O)CCOC1 Cc1nc2cc(C(=O)NC3CC(C)(NC(C4CC4C)=O)C3)[nH]c2s1 C1(C)(NC(C(C)N(C(c2cccnc2O)=O)C2CC2)=O)CCC(=O)N(C)C1 C1(C(=O)N(CCCSC2CCCC2)CCO)(NCCCC(=O)C(C)C)CCOC1 N1(C(CC(=O)OCC)=O)CCC(O)C1C(N1CCC=C(C)C1)=O c1(CC)ccccc1CNC(C1(CC(F)F)CCC1)=O c1(C(N2C(CNC(c3cc(CO)ccc3Cl)=O)C=CC2)=O)cc2ccccc2s1 c1(CNC(CCN(C(=O)CCc2ccc(C3CC3C)o2)CC=C)C)ccccc1Cl C1(NC(c2c(C)scc2)=O)C2CC(CN(C(=O)C(F)CC3CC3)C2)C1CO C1(CNC(CCC=C)=O)CC2CCC1N2C(=O)C(C)Sc1ccccn1 C1(C(=O)NC(CC)C(C)CN(C)C)CC2CC1CN(C(c1n[nH]c(C)c1O)=O)C2 C(=O)(CCN=C(NC1CCCC1)N1CCC=C(c2ccncc2)C1)OC C1(NC(c2c(C)cc(CC)o2)=O)CC(O)CN(C(c2c(C)cncc2C)=O)C1 C12(CC(=O)NC3CCN(C(c4[nH]cc(C#N)c4)=O)CC3)CCCCC1C2(F)F c1(O)ccc(F)cc1F.C1(C(=O)O)CCN(C)CC1.c12cn(nn1)C1CCN(C1)C2 N1(C(c2cc(SC)ncc2)=O)CCC(F)(CNC(C2CC23CCOCC3)=O)CC1 N1(C(C(c2ccc(F)cc2F)OC)=O)CC2CN(C(=O)C3=CCCCC3)CC2C1 c1(C(=O)NCC2CN(C(c3cn(C)nc3)=O)C3C2C3)cc2sc(Cl)cc2s1 C1(C(=O)NC2CCCC23CN(C(c2ccncn2)=O)C3)CC2CC1C1C2C1(F)F CCC(C)CCC(=O)N1CC2(CC(NC(=O)Cc3cccc(C)c3C)C2)C1 C1(NC(C=CCCC)=O)CN(C(C2CC2c2cnc(C)[nH]2)=O)CC1F C(C)(C)(C(c1nnnn1C(C)C)NC1(CC)CCOC1)OCC N1(C(C=COCC)=O)CCCC(CO)(NC(C2CC3(C2)CC3(F)F)=O)C1 c1(C(=O)NC(Cc2cccc(C)c2)C(=O)O)csc(=NCc2cc(CO)on2)[nH]1 N1(C(C(C)OCC(C)C)=O)CCC(C)(CC(=O)N(C2CCNC2=O)C(C)C)C1 N1(C(C=CCCC)=O)CC2CCC(NC(=O)C(c3ccc(F)cc3)C3CC3)(C2)C1 c1(C(=O)NCC2(C)CCN(C(C(COC)OC)=O)CC2)ccc(S(N)(=O)=O)s1 C1(Cn2cc(C(C=C)(C)O)nn2)CCCN(C(C2(C(F)F)CC2)=O)C1 N1(C(C2CC(C)S(=O)(=O)CC2)=O)CCN(C(=O)C2=CS(=O)CCC2)C2(CCC2)C1 C1(CCOC)(NC(C2CC=CCO2)=O)CCN(C(=O)COc2cccc(Cl)c2)C1 C12(C(N(CC(O)CNC(c3ccc(Br)cn3)=O)C)=O)CC=CCN1CCC2 CC1CCN(C(=O)CCc2cccn2C)CC1CNC(=O)CCC1CCOCC1 N1(C(c2ccnc(S(C)(=O)=O)c2)C(=O)NCCOC)CC2C3CCC(CC3)C2C1 c1(C(N2CCC(C(C(C)C)NC(CCC)=O)CC2)=O)nccc2ccsc12 C1(NC(CC(CC)Cc2ccccc2)=O)CN(c2ncc(Br)c(O)n2)CC2(CC2)C1 C(C(C)(O)CC(=O)N(C)CCNC(=O)CC1CCC(C)(O)CC1)OC C(=O)(C(C)(C)C)NC(C(=O)NC(c1ccccc1)C)C1CCC1 c1(C(=O)NC2CCCN(C(C(C#C)(C)C)=O)CC2)[nH]nc2ncccc12 CC1=C(C(=O)NC2(C)CC(NC(c3ccnnc3)=O)C2)C(C)(C)CCC1 C1(C(C(C)C)NC(=O)C(n2cc(CC(O)C3CC3)nn2)C)CCOCC1 C1(NC(CCCCOCCC=C)=O)CCN(C(C2CC2CF)=O)CC12CCC2 CC(C)C(F)(F)CCNC(=O)NCC1(C(=O)O)CC1 C1(CC)CC(C)CN(C(c2cnn(C)c2C#N)=O)C1.C12(C)CCN1C2=O Cc1ccc(C(N2CCC(Sc3cc(F)ccc3F)CC2)=O)c(O)c1 c1(CNC(C2C(C)(C)C(NC(=O)C(F)(F)F)C2)=O)cscc1S(C)(=O)=O c1(C(C(=O)NCC(n2ccnn2)C)NC2CC2c2cn[nH]c2)cccnc1 N1(C(C2C(OC)CCC2)=O)C2CC1CN(C(c1ncc(F)cn1)=O)C2 C=CCC(CC)C(=O)NC(CC(=C)Cl)C(=O)N(CC)CC1CC1(C)C N1(C(C(C)C2CC2)=O)CC2ON=C(CNC(C34CC5CC(C(=O)N3)C4C5)=O)C2C1 c1(C(=O)NCCC(CC)C)cccc2cc(O)ncc12 Cc1cc(C(N2CC3CC2CC3NC(c2sccc2C2CC2)=O)=O)nc(O)c1 c1(C(C(=O)NC2CC2)N(C2CSC2)C(c2ccccc2)C)sc(Cl)cc1Br c1(NC(=O)NC2C(SC)CCC2)cnc(C)nc1C C1(NC(CCC2CC(NC(CNC(C3C(C)C3)=O)=O)C2)=O)CN2CCCC1C2 c1(CCC)ccccc1C(=O)NCC(C)NC(C1(C(F)(F)F)CC(O)C1)=O C1(c2n(CC)nnn2)(NC(c2cn(C)cn2)C)COCCOC1 N1(C(C2OCCC(C)C2)=O)CC(C(=O)NC(CCO)C2CCC2)CC1(C)C N1(C(CCCOC(C)=O)=O)C2CCC1CN(C(=O)C(F)CC1CCCCC1)C2 c1(N(C)C)ccc(N(C(=O)C(=C2CCNCC2)F)CCO)nn1 N1(C(C2=C(C)CCC2)=O)Cc2ccccc2C(CNC(c2c(Br)cnn2C)=O)C1 C(=O)(C(C)CC(C)(C)C)NCC1CC(NC(CCCN(C(=O)OCC)C)=O)C1 C(C)(CCCCNC(c1cncc(C(F)(F)F)c1)=O)NC(C1CC(C)C1)=O C1(NC(CCCC2C(C)C2)=O)CN(C(=O)Cn2cc(CO)nn2)CC1C c1(C(N2CCC(CC)(NC(=O)C3=CCCC3)CC2)=O)cccc2ncsc12 c1(C(=O)NCC(CC=C)NC(C2CC(CCO)C2)=O)c(C2CC2)nc2sccn12 N1(C(c2cc(C)[nH]n2)=O)CCCCC(NC(c2cnn(CC3CC3)c2)=O)C1 N1(C(c2ccc(SC)o2)=O)CCC(C(=O)NCC2CCC(=O)N2C)C1(C)C C1(C(NOC)=O)CCCCCCN1C(=O)C(n1cnc(C#N)n1)C C1(N(C(=O)CCC2CCCN2C)C)CCCN(C(c2cn(C)c(C(F)F)n2)=O)C1 O=CCC(C(F)(F)F)N.C1(C(=O)N(C2CC2)Cc2ccoc2)CCS1(=O)=O c1(C(=O)NCC(CNC(CCC#CC)=O)(C)O)nccc(OC)c1C N1(C(c2nc(C)nn2C)=O)CCC(CNC(=O)Cn2nnnc2C)C(F)(F)CC1 C12(C(=O)NCCN(C)C)CC3CC(C(=O)N1)C2C3.C12CCC(CC1)C(=O)N2 c1(CC)cc(C(=O)NCC2(C)CCN(C(C3CC(CC)(CC)C3)=O)C2)cc(O)n1 N1(c2scc(C(c3cccs3)CNC(c3ccccc3)O)n2)CCS(=O)(=O)CC1 c1(C(N2C(C)CN(C(C3CC4CC3C3CC43)=O)CC2)=O)ccc2ncn(C)c2n1 C1(N(C(=O)CSC(C)C)CC)CCCN(C(c2cccnc2NC(C)C)=O)C1 CC1(C)CC(=O)N(CC(=O)NC2C3CN(C(C4CC5(CCC5)CO4)=O)CC23)C1=O C1(C#N)(C(=O)NCC(CC=C)NC(C2(n3cncn3)CC2)=O)CC12CCOCC2 c1(C(N2CCSC(CC)(CC)C2C(=O)O)=O)ccc(Cl)c2c1OCCO2 CN=c1nc(N2CCNC(=O)CC2)[nH]c(=NC(C)C2CCN(C)C2)[nH]1 c1(C(=O)NCC(C)N(c2cc(OC(C)C)ncn2)C)coc2ccc(F)cc12 N1(C(CC(C)c2cccs2)=O)CCCC(CCC2CCN(C(=O)C3CC3)CC2)C1 CCCC(C)CC(=O)N(C)CC1CN(C(=O)C(c2ccccc2F)(F)F)CCO1 n1(CC(=O)NC2C3(CC(NC(C(CC)C(C)C)=O)C3)C2)ccc(=O)c([N+](=O)[O-])c1 CC1CCC(C)N1CC(=O)NCCC1(NC(C2CC=CC2)=O)CC1 C1(NC(=O)Cn2cncn2)CN(C(=O)Cc2cnc(C3CC3)[nH]2)C2(CCCC2)C1 Cc1cc(NCC2CCC3(CN(C(C4(O)CC4)=O)C3)O2)n2nc(C)cc2n1 Cc1ccc(C(=O)NC(C)(C)CC(=O)NC2CCOCC2C)cn1 C1(NC(c2c(CC)nns2)=O)CCCC2CN(C(c3sccc3C3CC3)=O)CC12 Cc1nccc(C(=O)NC2(CF)CCN(C(=O)C=Cc3cnc[nH]3)C2)n1 c1(OC)cc(C(=O)N(C(C)C(F)(F)F)C)ncc1Cl CCC(C)C(CNC(C1CCCN1C(=O)CC1CC(O)C1(C)C)=O)CO C12(C(=O)NCC(C)NC(C3(CS(C)(=O)=O)COC3)=O)CC(C1)Oc1ccccc12 N1(Cc2nc(C)nn2C)CCC2CCCNC2C1 C1(NC(c2cc(Br)co2)=O)CN(C(c2ccc3nncn3c2)=O)C2CCCCC12 CC1C=C(C(=O)N(CCNC(C2CCCOCC2)=O)C2CC2)CC1 C(=O)(CCC(C)C)NC(C1CCCN(Cc2ccc(C(N)=O)cc2)C1)CC C(C(=O)NCCC#N)(C1=CCSC1)N(C(C)CS(=O)(=O)CC)CC C1(CNC(C23CC(CCC)(C2)C3)=O)CCCN(C(C2CCCC2SC)=O)C1 C1(C)(NC(c2c(CC)[nH]cc2)=O)CCCN(C(=O)CCS(=O)(=O)N(C)C)C1 C1(O)(CNC(C(C)(c2ccccc2)SC)=O)CCN(C(c2ccc(C)n2C)=O)C1 C1(NC(CCN(S(C)(=O)=O)CCC)=O)CCC(C)N(C(=O)NCC#N)C1 C1(C(N2CCN(CC(=O)NCC3CNC(=O)O3)CC2)=O)CCC(F)(F)CC1 Cc1cc(N2CCCC(c3cnco3)C2)nc(=NCCc2cccc(F)c2F)[nH]1 C(=O)(C1=CC2(CCOC2)C1)N(CCNC(C(CN(CC)CC)F)=O)CCOC C(=O)(C(CN=[N+]=[N-])NC(c1cc(C)c(N)cn1)=O)NC1C(CC=C)CCCC1 CC1(C)Cc2ccc(C(=O)NC3CN(C(C4(C5(C)OCCO5)CC4)=O)C3)cc2C1 C(=O)(CC(C)C(C)(C)NC(C1CC(F)C(=O)N1)=O)NC(CCC)C1CCC1 N1(C(C2C(C)C2)=O)CCCC(C)(CNC(c2ccc(-c3cnn(C)c3)o2)=O)C1 c1(CC(=O)NCCNC(=O)C2=CCCC2)ccc(-n2cccc2)cc1 n1(CC)ncc2cc(C(=O)NCC(c3ccc(OC)c(Br)n3)=O)cnc12 S(=O)(=O)(c1cccs1)N(CC(N1CCN(C(C2(CCN(C)C)CC2)=O)CC1)=O)C C(CC(C(=O)N1CC(F)(C(=O)NCC2(F)CCOCC2)C1)OC)OC C(C)(CNC(=O)C(C(C)C)N1CCCC1=O)(CC(C)C)NC(CSCC=C)=O C1(O)(C(C)NC(=O)CCCOC(C)(C)C)CCN(C(C2CC2c2ccnn2C)=O)C1 c1(C(=O)NC(C(C(C)C)NC(=O)C=Cc2cn(C)nn2)C)cc(Cl)c(Cl)n1C c1(SCC2=CCCC2)cccc(NC(c2nnnn2C2CCOC2)C2CC2)c1 C=CC(C)(CC)C(=O)NCCCC1CCCN1C(=O)C(c1cc(F)ccc1F)=O CCC(CNC(=O)CCCOc1ccc(F)cc1)N=c1[nH]c(Cl)c(C#N)s1 c1(C(=O)NC2CN(C(CC(C=C)C)=O)CC23CCC3)cc2cccnc2cc1F N1(C(CC(CC)(C)C)=O)CC2CC(NC(=O)CC3(O)CCOC3)C(C2)C1 C(=O)(C1=Cc2ccccc2C1)NC1CC2N(C(C3C(=C)C3)=O)C(CCC2)C1 c1(C2(C(=O)NC3(CO)CN(C(c4ccccc4O)=O)C3)CCC2)ncccc1F c1(CN(c2ncc(C3CC3)cn2)C(C2CCCNC2)C)sc2ccccc2c1C CC(C)C(O)C(C)C(=O)NCCC1CN(C(c2c[nH]nc2-c2cnn(C)c2)=O)C1 C1(C2CCN(C(=O)C=C(CC)CC)CC2)(NC(C(CC)OCC)=O)CC1 N1(C(C(N2CCOCC2)C)=O)CC(=O)CC1C(=O)Nc1ccc(O)cc1 N1(C(C(C)=C(CC)C)=O)CCC(CNC(=O)C(c2cccnc2F)(C)C)(OC)C1 C1(C(N2CCCC(CCC=C)C2)=O)CCN(C(=O)C(C2CCCCC2)=O)C(C)C1 CC1CCC(C)N1C(C)C(=O)NCCN(C(c1ccc(C(N)=O)s1)=O)C1CC1 N1(C(C(C)NC(=O)NC)=O)CCCCC(CNC(c2coc(Br)c2)=O)C1 C(=O)(CC(C)CNC(=O)CN1CCC(F)CC1)N(C(C(CC)C)C)C1CC1 c1(COC)ncc(C(N2CC3CC2CC3NC(C23CC4CC2C3C4)=O)=O)c(=N)[nH]1 C1(NC(C2CC2C(F)(F)F)=O)CC2CCC(C1)N2C(c1nc(Cl)sc1Cl)=O c1(C(=O)NCCC(CNC(C2(C(N(C)C)=O)CC2)=O)O)coc2c1CCCC2 C(C)(C(O)C(F)F)NC(CC1N(C(c2ccc(C)[nH]2)=O)CCC1)=O n1(CC(=O)N(C)CCOc2ccccc2F)ncc2cc(Br)cnc12 c1(C(=O)NC2(COCC)CCOC2)c(C(F)(F)F)coc1C(C)C C1(C(=O)NCCCC(=C)C)C(C2CC2)CCN1C(c1cn(C)c(C)n1)=O N1(C(c2c(C)nc(O)cc2)=O)CC2CC(NC(=O)CCc3cc(Cl)no3)C(C2)C1 N1(CCNC(=O)C=Cc2c[nH]cn2)CCC(NC(=O)Cn2cncn2)CC1 c1(OC)ccc(Cl)cc1CC(N1CC(CNC(=O)CSc2ccccc2C)C1)=O N1(C(C2CN(C(c3c(CC)ncnc3)=O)CC2CC)=O)CC2(C1)CN(C)CCO2 c1(C(=O)NC(CC)CNC(C2(Cc3ccc(O)cc3)CC2)=O)cc2cn[nH]c2cn1 C1(OC)CN(C(=O)CN2CCCS2(=O)=O)CC1NC(c1ccc(CCO)cc1)=O Cc1[nH]c(-c2ccccc2)c(C)c1CNC1(C)CN(C(=O)C(F)C(F)(F)F)C1 N1(C(=O)COc2ccsc2)CCC(n2cc(CC3CCOCC3)nn2)C1 c1(C(C)NC(c2ncoc2CNC(C2CC2(F)Cl)=O)=O)ccccc1O C(=O)(C(CCN(C)C)NC(=O)C(C)=CCC)N(CC#C)CCF C(=O)(C1COc2ccccc21)NC1CN(C(C2C(C)C(=O)C2)=O)C2C1CCC2 C=C(Cl)CC(C(=O)N1CCN(CCO)C(=O)C1)NC(=O)CN1CCCCC1C Cc1[nH]c(C(N2CC=C(CNC(C3(C)CC(O)CN3C)=O)CC2)=O)c(C)c1C Cc1cccc(Oc2ccccc2C(=O)NC(=O)C(CC#N)c2nn[nH]n2)c1 N1(C(C23CC(C#N)(C2)C3)=O)CCC2CC2(C(=O)NC2CN3CCC2CC3)CC1 C1(CNC(C(C)Cn2ccnc2)=O)CN(C(c2ccnn(C)c2=O)=O)C(C)(C)C1 c1(C(=O)NC2CC(CCNC(C3(C(N)=O)CC3)=O)C2)cn(CC(F)F)nn1 C(=O)(CCCC(=O)NCCN(C(C1SC2C=CC1C2)=O)CC1CC1)N(C)C N1(C(C(C(C)NC(c2ccnnc2O)=O)C)=O)CC2(CCOCC2)C1 c1(OC(COC(c2ccco2)COC2CC(COC)C2)=O)cnc(Cl)s1 c1(OCCN(CCCOC)C)ccccc1OC(=O)Cc1cccc(C(F)(F)F)n1 C1(C#C)(NC(CCC2(NC(CCCC#C)=O)CCCC2)=O)CC2CCCC12 c1(C(=O)NCCNC(C(CN(C)C)O)=O)cccc2ccoc12 C1(SCCCOC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)CC(C)(C)C(=O)O1 C1(NC(CCc2ccc(C)s2)=O)CN(C(c2cc(CO)[nH]n2)=O)CC12CCC2 C(c1ncc(C)[nH]1)=CC(=O)NC(CC=C)CNC(=O)CNS(C)(=O)=O O=C(N=c1cnn(C2CCC2)[nH]1)C1CCOC1 c1(SC)cnn(C)c1C(N1CCC(O)(CN(C)C(C2CCCCC2)=O)C1)=O n1(C(C)C)nccc1C1OCCC1C(=O)NC(C1CCCC1O)c1nn[nH]n1 c1(OC)ccc(C(C)C)c(C(N2CCC(O)C(NC(=O)CC(C)CSC)C2)=O)c1 C1(OC)CN(C(=O)CC(O)CN(C)C)CC1NC(c1cncc(C2CC2)c1)=O N1(C(c2cn(CC=C)nn2)=O)CCC2(CCC(NC(=O)C(C)CC)CC2)C1 c1(OC)ccc(C(F)(F)F)cc1C(=O)NC(C)CCNC(=O)C=C(C)C(F)F CC(C)C(CCNC(c1cc[n+]([O-])cc1)=O)NC(c1cocc1Br)=O Cc1cccc(C(=O)NC(C2CC=CCC2)C(=O)Nc2cccc(CCF)c2)n1 c1(C(N2CC(CC)N(C(=O)CC(C)(C)CC)CC2)=O)cn2c(n1)COCC2 N(C1CCCn2ccnc21)C(C(CC#CC)NC(=O)Cc1c(C)noc1C)=O C1(NC(c2ccc(C)o2)=O)CN(C(C2CC3(C2)CC3(F)F)=O)CC1S(C)(=O)=O CN1CCC(C#N)(C(=O)NCC2CCCN(C(C3CCC3(C)C)=O)C2)CC1 C(=O)(C(=O)CCC(C)C)NCC(CC(=O)NC(CC)CC)O Cc1cccc(C)c1NC(=O)C(N1CCC(CNCC(=O)O)C1)=O C12(C(N3CCN(C(C(C(C)OC)O)=O)CC3C)=O)CC3CC(C(=O)N1)C2C3 N1(C(C2C(C(C)(C)C)CC2)=O)CC2C(NC(=O)C(O)CC3CCCCC3)C2C1 N1(C(C2C(NC(c3ccc(OC)nc3)=O)CCC2)=O)Cc2ccc(C#N)cc2C1 C(=O)(C(O)CC(F)(F)F)NCCCN(C(C1CN(C)C(=O)C1)=O)C1CC1 N1(C(C(c2cnn(C)c2Br)C)=O)CC(c2ccccc2)(CO)C(c2ccccc2)C1 N1(C(C(C)NC(C)=O)=O)CCC(F)C(NC(c2c(Br)sc(C)c2C)=O)C1 C1(CNC(c2cc(CCC)[nH]n2)=O)CCCN(C(=O)OC(C)(C)C)CC1 CC(C)CCC(O)C(=O)N1CC(O)CC1(C)C(=O)NCC(C)(C)C(N)=O CC(C(=O)NC(=O)CCc1nc(-c2ccoc2)no1)C(F)F c1(CC)onc(C)c1NC(C1C2CN(C(c3ccc(CO)cn3)=O)CC12)=O CC(C)(CC(=O)N1CCCC12CCN(C(C13CCCC1C3(F)F)=O)C2)CC(F)F Cc1ccc([N+](=O)[O-])c(C(N2CC(NC(=O)C(F)C(C)(C)O)C(O)C2)=O)c1 c1(SCCCC)ccc(NC(=O)N(c2cccnc2S)C(C2CCOC2)=O)cc1 C(C(O)CN(C)OC)c1nc(-c2c(C(=O)NCCC)cccc2)on1 C1(CCC)(NC(=O)C2=CCOC2)CCN(C(=O)C=C2CCCC2)CC1 c1(C(N2CCCC(C(C)NC(=O)C3=COCC3)C2)=O)cnc2[nH]ncc2c1 c1(OC)ccc(C(=O)NC2(C3CCCCN3C(c3cnns3)=O)CC2)cc1 N(C(=NCCCOCC)NCc1cc(C)nc(C)c1)CC(C=C)C c1(C(=O)NCC2C(C)(C)CN(C(c3ccccc3)=O)C2)cc(F)c(N)c(F)c1 CC1(C)C(CC(=O)NC2CC(NC(c3ccc(C4OCCO4)cc3)=O)C2)C1(C)C Cc1ccc(C)c(C(N2CCC(C(C)NC(=O)CN3CC(=O)N(C)C3=O)C2)=O)c1 CC(CC1=CCCCC1)NC(C1C=CCCN1C(c1c[nH]c(=O)cn1)=O)=O c1(C(N2CCCCC2c2cn(N3CC4CC3(C(F)F)C4)nn2)=O)ccc(O)cc1 c1(NC(C2C3(CCN(S(CC#N)(=O)=O)C3)C2)=O)cccc2nc(O)ccc12 N1(C(CC(C(F)F)NC(C2(C(=O)NC)CCC2)=O)=O)CCOC(C)(C)CC1 CCC(C)(CNC(=O)C=C1CCOCC1)C(=O)N(CCC(C)(C)C)C Cc1cc(C(C(=O)NCc2cccs2)N(C)Cc2cc[nH]n2)ccc1I N1(C(COc2cccc(C)c2)=O)CCN(C(=O)C2CC2)CC1C1CC1 C12(NC(c3nccc(C)c3)=O)CCOCC1CN(C(c1ccc(C(F)F)s1)=O)C2 CC(C(=O)NCC1(F)CCC(CNC(c2coc(CO)c2)=O)CC1)C(C)C(C)(C)C C1(NC(CC2ON=C(CC)C2)=O)(CNC(C2(C3CCC3)CC2)=O)CCCCCC1 O=C(C1=NNC(C(F)(F)F)C1)OCCSC1CC2CCC1O2 Cc1cccc(C2CCCCC2C(=O)NC2CC(N(C(=O)C(=O)N(C)C)C)C2)c1 c1(C(=O)OCC)[nH]cc(CNC(C)Cc2nn[nH]n2)c1C c1(C(CF)NC(=O)NC2C3CCOCC23)ccccc1Br CCCC(C(=O)NC(C1(O)CCN(C(c2c[nH]nc2CC)=O)CC1)C)S(N)(=O)=O Cc1noc(C)c1Cc1nc(-c2ccn(C)n2)nn1CC1CCCCO1 C(=O)(C#CC1CCCO1)NC1(C2CN(C(CCc3ccc(C)nc3)=O)C2)CC1 C1(C(=O)NCc2c(C)cccc2)CN(C(=O)C(F)CC2CCOC2)CC(C)(C)C1 c1(C(N(CCCN(C(=O)C(F)C2CCOC2)C)C)=O)cc(F)cc2nc(S)[nH]c12 c1(C(N(CCCNC(C2CSCCS2)=O)C(C)C)=O)cc2c(=O)[nH]ccn2c1 C(C1CCCN1C(C1CCCCC1O)=O)=CC(=O)NC(Cc1cc(C)[nH]n1)C C(=O)(C(CNC(C1(C#N)CC(F)(F)C1)=O)CC=C)NC1(C(=O)NCC#C)CC1 N1(C(CCC2(C)N=N2)=O)CC2CCCC1C2CNC(C1(C)CCCCCCC1)=O N1(C(C2(C)C(C)OCC2)=O)CC2CCC(NC(=O)COC3CC3)(C2)C1 C(CC(C(=O)N1CCC1CNC(=O)Cc1cccnc1Cl)NC=O)SC N1(C(N2C(COC)CCOCC2)=O)CC2COCC2(C)C1 CC1(C)CCN(C(=O)CCOC2CC2)C1CNC(C1CCC(=O)N1)=O C1(CNC(C(CC)O)=O)CN(C(=O)C(c2cncnc2)C)CC1(F)F c1(OC)c(C(=O)NC(C)CC(C)NC(c2cc(C#N)cs2)=O)ccc(Cl)c1C c1(C(=O)OCC)cnn(CCNC=O)c1C.c1(CCOCCOCC)ncsc1 CC1(C)OCCC1CC(=O)NCC1(CO)CCN(C(C23CSCC2C3)=O)C1 C(CCC)(C(=O)N1CCC(O)(CCNC(=O)COc2cc(C)on2)C1)=CCC C=CCC(C(=O)N1CCOCC1CNC(=O)CC1CCCSC1)NC(C)=O S(=O)(=O)(c1ccc(NCC(C)C)c(Cl)c1)N(C1(SCC(C)C)CC1)C c1(C(=O)NC2(CNC(=O)Cc3ccc(Cl)c(F)c3)CC2)cc(F)cc2nn[nH]c12 N1(C(CC#C)=O)CCCC2CN(CCc3csc(C)n3)CCC12 N1(C(c2cc(C)nn2C)=O)CCC(F)(CNC(C2(C)CCCC2O)=O)CC1 Cc1cncc(C(=O)NC2CCN(C(c3ccc(C)n3C)=O)C(C3CC3)C2)c1Cl C1(OC)CN(C(=O)Cn2ccnn2)CC1NC(=O)Cn1cc(C2CCOC2)cn1 c1(CNC(COCCC=C)=O)cnn(C)c1C(=O)NC12CC(CCCC)(C1)C2 N1(C(C(CC)n2ccc(C3CC3)n2)=O)CCCC(CNC(C2(CF)COC2)=O)C1 c1(C(=O)NCC2(CNC(=O)Cc3ccsn3)CCC2)cnn(C(F)F)c1 Cc1cc(N2CCCC(NC(=O)Cn3cc([N+](=O)[O-])cn3)C2)nc(S(C)(=O)=O)n1 c1(C(N2C(C)(CNC(c3cccc(C)c3F)=O)CCC2)=O)ccc(F)c(C)c1C c1(C(N(CC(C)(C)NC(C(C(C)SC)O)=O)C)=O)ccc(Br)c(C)n1 CC1CN(C(=O)C=Cc2ccnn2C)CCN1C(=O)C(=O)Nc1ncc[nH]1 C1(C(N2C(C)(CNC(c3cn(CCC=C)nn3)=O)CCC2)=O)C(F)(F)C12CCC2 N1(C(C(C2CCCN(C(=O)CC3CCC(=O)C3)C2)(C)C)=O)CCOCC2(CC2)C1 C(=O)(C1=C(C)CCOC1)NCC(CCCC)NC(c1cscc1Cl)=O CON(CCC(=O)NCC1Cc2nccn2C1)C(=O)c1c[nH]c(=N)o1 C=Cc1cnn(C)c1C(=O)NCCC1(O)CN(C(C2CCCNS2(=O)=O)=O)C1 C1(C)(CCC)CCN(C(C2(NC(=O)CC3C=NN(C)C3=O)CC2C)=O)C1 C1(O)(C(C)NC(C2CC2c2nc(C(F)(F)F)no2)=O)CN(C(C2CCC2C)=O)C1 N1(C(C(CNC(C2(C#N)CCOCC2)=O)N(C)C)=O)CC2COC(=O)C2C1 N1(C(c2c(C)ocn2)=O)CC(CNC(=O)C=Cc2ncc[nH]2)OC2CCCC12 C1(NC(c2c(CC)cco2)=O)C2CC1N(C(c1ncc(Cl)cc1F)=O)C2C C(c1c(C)nn(C)c1Cl)=CC(=O)NCC(C)NC(CCc1ccc(C)o1)=O C(=O)(CC(CC(N)=O)CC(C)C)NCC1(C)OCCN(C(c2cc(CC)[nH]n2)=O)C1 c1(C(=O)NCC(C)CN(C)C(C2CCC(N(C)C)CC2)=O)ccc2nc[nH]c2c1 CC(C(=O)N1CCC(C)(CC(=O)NC(C)C(=O)NO)C1)S(C)(=O)=O c1(C(CO)NC(C(C2CC=CCC2)NC(COC2(C)CCC2)=O)=O)ccccc1 C1(N(C)C)CCCN(CCNC(=O)NC2CCC(OC)C2)C1=O c1(NC(C2C(NC(c3ccn(C)n3)=O)CC2)=O)ccc2cnn(C)c2c1 c1(C(=O)NC2CC(CNC(C3(CC=C)CCC3)=O)C2)ncoc1C c1(CCCC(=O)N(CC(CNC(C(C)CF)=O)(C)C)C)c[nH]c2ccccc12 C#Cc1cccc(NC(=O)C(N2CCCC(NCC3CCCC(N)C3)CC2)=O)c1 N1(Cc2c(OC)c(C)ccc2)CCC2(CCCC2C(N2CCCCC2CO)=O)C1 C=CC(CC)CC(=O)N1CC2CC1CN2C(C1CC2(C1)CC2F)=O Cc1cc(C(=O)NC2CCCCC2N(C)C(c2cn(C3CC3)nn2)=O)cnn1 N1(C(C2(C#C)CN(C(=O)CSCC)C2)=O)CC2CC(C1)C2(C)C N1(C(=O)CO)CC2CCN(C(c3ccc(C4CC4)c(Br)c3)=O)CC2C1 C1(C(=O)NCC(C2CCC2)OC)CCN(C(=O)c2ccc(C)nc2)O1 N1(C(C2(C)CC=CC2)=O)CCC(C)(CNC(=O)Cn2cnnn2)C1 c1(OCC)c(OC)cc(C(=O)NC2(CO)CN(C(=O)Cc3cnc[nH]3)C2)cc1Cl n1(CC=C)nc(-c2ccc(SC(C)C)nc2)nc1-c1cnc(OC(C)(C)C)cn1 N1(CC)CCN(CCC(=O)N(CC(=O)CC2CCOC2)C2CC2)CC1 N1(C(C2(C)ON=C(C)C2)=O)CCC2(CC1)CN(C(c1nnc(C(C)C)s1)=O)C2 N1(C(CCSC)=O)CC(F)CC1CC(=O)NCC(=O)NC(C)(C)C c1(C(=O)NCc2occ(C(=O)NC(c3cccnc3)C)c2)ccc2cncn2c1 C1(C(=O)Nc2c(C)ncs2)CCC(C)N1Cc1ccc(N2CCCC2)cc1 c1(CNC(C(C2CCC2)OCC)=O)ccc(C(=O)NCCCN=[N+]=[N-])nc1 c1(C(C2CC2)NC(CC)=O)cn(C(C)CNC2CC(C(C)C)C2)nn1 c1(C(N2CCC(OCC(C)C)C2)=O)coc(CNC(C2CC3(CC3)C2)=O)n1 c1(C(=O)NC2(C)CCN(C(c3cc(F)cc(F)c3)=O)C2)ccc2ncncc2c1 N12CC3CC(C(C3)C1)C2.c1(SCC)cnc(Br)cn1 c1(NC(C2C(O)CCN2Cc2ccnc(O)c2)=O)nc(Cl)c2ccnc-2[nH]1 N1(C(CC2CC(CC)C2)=O)CCC(NC(=O)C(C)(C)O)C(C)C1 CCC(CC(=O)NC1CC(OCC(N2CC(c3cc[nH]n3)C2)=O)C1)C1CCC1 c1(C(C(=O)NCC)N(C(CCC)C#N)CC)ccc2c(c1)CCC2 CCC(CC(=O)N(C)CCC1CCN(C(=O)C(C2CCOCC2)F)CC1)OC C1(CNC(=O)CCc2ccon2)CCCCC1NC(=O)CC1CCC1 c1(CC)c(C(=O)NCC(CNC(c2cc(CC)on2)=O)OC)oc2ccccc12 N1(C(C2(SC)CCC2)=O)CCC(CNC(=O)CCC2OCCO2)C(O)C1 C(=O)(C1=C(C)CCOC1)NC(CCCC)C(=O)NC1CCCC1C#N C(=O)(CS(=O)(=O)C(C)(C)C)NCCN(C(=O)CN1CCP(C)(=O)CC1)CCOC CC1(CNC(C2CC2F)=O)CCCN1C(c1nc(Cl)c(Cl)s1)=O C(=O)(C1=NOC(CNC(=O)CN2CSCC2=O)C1)NCC1(C)ON=C(C)C1 N1(C(C2C(C(=O)OC)CCO2)=O)CCC(NC(=O)CCCC(N)=O)C(CO)C1 C1(CCNC(C2(CCCC)CC2)=O)C(C)CCCN1C(c1cnc(C(C)C)s1)=O C1(NC(C=CCN(CC(F)(F)F)C)=O)CC2(CCCN(C(C3CC3(F)F)=O)C2)C1 C1(N(C(CN(CCC)C(c2conc2C)=O)=O)C)CCOCC1C Cc1ccc(NC(C2CCN(C(c3cnsn3)=O)CC2O)=O)c(Br)n1 N1(C(C2C(=C)C2)=O)CCC12CN(C(=O)C(C)(C)CF)C2 CC1CCc2c(Cl)cccc2C1NC1CCc2ccccc2OC1 C123CCC(CC1)(C2)CNC3=O.NC(=O)C(O)CNC(c1ccoc1C1CC1)=O c1(OCC)nc(N2CC(O)CC2C(=O)NC2CCCN(C)C2=O)ncc1Cl c1(C(=O)NCCCN(C(C2C(C)(CC)C2)=O)C)c(O)cnc2ccccc12 N1(C(C(C=CC)O)=O)CCOC(C)(CNC(=O)Cn2nc(C)c(Br)c2C)C1 c1(NC(N2CC(OC(F)F)C2)=O)ccc2c(Cl)csc2c1 CC(CN=C(NCC1CCCCC1)N(C)Cc1ncc(Cl)n1C)C(C)(C)C Cc1nc2c(o1)CCCC2CC(=O)NC1(C)CN(C(c2ncc(N)cc2Cl)=O)C1 N1(C(C=CC(C)=O)=O)CCC(C)C(CNC(c2ncccc2C2CC2)=O)C1 C1(C(=O)NC2CCC(C(N(C)Cc3c(C)ccnc3)=O)C2)CC(C)CC(=O)N1 C12(C(N3CC(OCCCC#N)C3)=O)CN(Cc3ccccc3)CC1CS(=O)(=O)C2 c1(OC)ccc(CN2CCC(CCNC(=O)C(O)C(C)(C)C)CC2)c(OC)c1 CCCCCC(C)CC(=O)N(C(C)(C)CC(=O)N(C(C)CCC)C)C C1(C(N(C)CC2CCCN2C(=O)CC(F)(F)F)=O)CC(C2CC2)=NO1 c1(NC(=O)NC(CC=C)C(=O)OCC(F)(F)F)nc(OC)cc(C)n1 C(C1=CCN(C(c2cc(Cl)cc(Cl)c2)=O)CC1)OC.c12nn(C)cc1C(=O)NC2 c1(OC(C)C)c(CNC23CC(C(NNC(=O)OC(C)(C)C)=O)(OC2)C3)cccc1F C1(COC)CN(C(C2CC=CCC2)=O)CCN1C(=O)COCc1cc(C)no1 c1(C(=O)NCC(CN(C(c2ccc(C#C)cc2)=O)C)O)cc2nc[nH]c2cc1N c1(N(C)C)ccc(C(=O)NCCc2c[nH]c3cnccc23)cc1[N+](=O)[O-] c1(C(N2CCC(C)C2CNC(c2nn(C)cc2Cl)=O)=O)ccc(F)c(C#N)c1 N1(C(C2CN(CC3=NCCO3)CCO2)=O)CC2C3CCC(O3)C2C1 N1(C(C(C(C)C)OCC)=O)CCC2CCN(C(c3cnc(S)n3C)=O)CC2C1 N#Cc1cc(C(N2CCC(NC(c3c[nH]nc3F)=O)C(O)C2)=O)cc(O)c1 c1(OCC(=O)NCCCNC(Cc2cc(C)[nH]n2)=O)ccc(Br)c(C)c1 N1(C(C(C)=C(C)C)=O)CCCC(O)(CCNC(c2ccn(C(F)(F)F)n2)=O)C1 CCCC(CCCNC(=O)C(C)NC=O)NC(=O)Cn1cnnn1 C1(C(=O)NCCCN(CCO)C(c2coc(Br)n2)=O)(CC)CCOC1 C(=O)(CS(=O)(=O)N(C)C(C)=O)NC(C(C)NC(C=CC=CCC)=O)CO CN=C(NCCC1CCCS1(=O)=O)N1CCC(n2ccc(C)n2)CC1 S(=O)(=O)(CC(=O)NC1CN(C(=O)CCc2ccccc2O)CC1C)NC CC1CCN(CC(N2CCCCC2CCCNC(C2COCCOC2)=O)=O)CC1 C1(C(N(C2CCN(C(c3sc(CC)c(C)c3)=O)C2)CC)=O)Cc2cccnc2C1 C1(NC(=O)Cc2cncnc2)CC2CCC1C(NC(c1c[nH]cc(Cl)c1=O)=O)C2 CC1(O)CCC(C(=O)NCC(O)C(=O)NCCC(=O)N(C)C)CC1 CC(C)(CC(=O)NC1CC1NC(=O)C1=C(Cl)CC1)CC(=O)c1ccccc1 c1(CC(=O)N(CCCNC(CNC(C)=O)=O)C(C)C)c(F)cncc1Cl c1(C(C)C)ncc(C(=O)NCCOC(C)C)o1.C1C(=O)N(C)CC(C)N1 c1(C(=O)NC23CC(C(=O)NC(c4csc(C#N)c4)C)(C2)C3)cc(I)ccc1[N+](=O)[O-] CC1CCC(NC(=O)C(C)(C)Cc2ccc(O)cc2)CN1C(c1cnsn1)=O N1(C(CCNC(=O)NC)=O)CCC2CCC12CNC(=O)CN1CCCCS1(=O)=O c12nccc(n1)N2C(C)C.c1(CC(=O)NC(C2CCCNC2)C)ccc(Cl)cn1 N1(C(C2N(C)CCCC2)=O)CCC(NC(=O)CCC2CCOC2)C(C)(C)C1 CC1CC(C)N(C(C2CC(C(=O)Oc3ccccc3)C2)=O)c2ncnn21 N1(C(C2(C(=O)OC)CC2)=O)CCC(NC(=O)CC2COCC(C)(C)O2)CC(O)C1 c1(C(=O)NCCN(C(CCN(C)CC)=O)CC)cc(C#N)no1 CCS(=O)(=O)CC(=O)NC1CCN(C(c2cn(C(C)C)nn2)=O)C1C1CC1 C(C(COC)C(C)C)NC(C1C(NC(C(CC)C)=O)CCO1)=O c1(NC(C2C(C(=O)Nc3cccc(CCOC)c3)C2)=O)ccc(Br)nc1Cl C1(C(=O)NC2C3CN(C(C(C(=O)OC)(C)F)=O)C2C3)CCC2(CCOCC2)C1 C(C)(C)(C(=O)NC(C)CC(C)NC(c1cscc1F)=O)OC c1(OC)cc(Br)c(F)cc1NCC1CC12CC2(F)F C1(NC(c2cc(CC)on2)=O)CCCC12CN(c1nnc(CC(F)(F)F)s1)C2 c1(COC)nc(NCCN2CCOC2=O)cc(=NC2CCCC2C#N)[nH]1 CCCCC(F)C(=O)Nc1cc(C2CCCN2C(=O)OC(C)(C)C)nn1C CN1CC(C)(C)CC1C(=O)NCC1(C(C)(C)O)CN(C(C2(C)CNC(=O)C2)=O)C1 N1(C(CCCCCNC(C)=O)=O)CCC2CCN(C(=O)C=Cc3cnc[nH]3)C2C1 C1(CC(=O)NCCCCc2cn(C3CCCC3O)nn2)Cc2ccccc2CN1 N1(C(C2=C(C)S(=O)(=O)CC2)=O)CCCC12CCCN(C(C1(F)CC1)=O)C2 c1(C(=O)NC2C3CN(C(c4ccc(SC)s4)=O)C2C3)cc2cccnn2c1 c1(OCC(=O)NC2CCN(C(C3C(C=C)CC3)=O)C2C)ccc(Cl)c(C)c1 N1(C(c2c(C(C)C)ocn2)=O)CC2(CCC(CNC(C3CC3C(C)O)=O)O2)C1 N1(C(C2CCCN(C)C2)=O)CCC(C2CCN(C(c3coc(Cl)n3)=O)CC2)CC1 c1(C(=O)NCCC=CC=C)ccoc1CNC(c1cc[nH]n1)=O C1(CNCCCc2cccc(C(F)(F)F)c2)Cc2ccccc2C1 Cc1cc(C(N2CC(CCNC(C3CS(=O)C3)=O)C2)=O)ncc1Cl n1(CC(N2CC(CC)C2)=O)cc(C2CCN(C(c3occc3C)=O)C2)nn1 C1(C2CN(C(C3CC3C3CCC3)=O)C2)(NC(C(C)=CC)=O)CC1 c1(OC)cccc(NCC(O)CNC(c2cc(C)cc(O)n2)=O)c1[N+](=O)[O-] c1(OCC(=O)NCC2(F)CN(C(Cc3nc(C)oc3)=O)C2)ccc(C)c(C)c1 C1(CN(C(C)C)C)CCN(CC2CSCCS2)CC1 C1(C(N(CC(=C)C)CC)=O)CCOC1CNC(=O)CCCSC(C)(C)C C(C(C)(C)C(=O)NC1CC(N(C(=O)CCOc2cccnc2Cl)C)C1)OC(C)C C=CC(CCC)CC(=O)NCCCCNC(=O)CC1CCS(=O)(=O)C1 c1(C(=O)NCC2(CNC(C3C(C=C)C3)=O)CCC2)cc(N)ccc1F CN1CCCC1C=CC(=O)NC(CCOCCO)C(=O)Nc1cnn(CCO)c1 c1(CC)nc(NC2CC(CNC(c3ccnc(C(N)=O)c3)=O)C2)c(C)c(Cl)n1 C(C#Cc1ccc(F)cc1)NCC(=O)Nc1cc(OC)c(C(F)(F)F)cc1 c1(CC(N2CC(C(C)(C)O)(CNC(C(CCOC)C)=O)C2)=O)c(F)cncc1Cl C12(CNC(c3cc(OCC)n[nH]3)=O)CC1CN(C(=O)CCC(=O)NC)C2 c1(C(CCN(C(=O)C(=O)NCc2cnsc2)C)O)ccccc1 N1(c2ncc(CCC)cn2)CCC2CN(C(c3ocnc3C)=O)CC12 S(=O)(=O)(c1cccs1)NCC(c1cn(C)nc1)NC1COCC1n1ccnc1 N1(C(CCN(CCC(C)(C)C)C)=O)CCC(C)(NC(=O)C(O)c2ccco2)C1 C1(C(N(CCNC(CCOC)=O)CCc2ccccc2)=O)CCCC12CC2 N1(C(C=C(COC)C)=O)CCC(O)(CNC(c2nocc2Br)=O)CC1 N(C(=NCCF)N1CCC(Cc2ccnn2C)C1)CC(C)C(F)F C1(C(=O)NCCC2CC(F)(F)CN2c2nnc(CO)s2)CCc2nnnn2CC1 O=C1NCCCCC1C(N1CC(O)C1)=O.C(CC(=O)Nc1ccsc1)OC=O N1(C(C=CC)=O)CC2(C1)SCCC2NC(=O)C(CC(C)(C)C)c1ccccc1 N1(c2n(CC(=O)N(C)C)ncc2)CC2CCCCCCC12 C#CCCCCC(=O)NCC(C)(C)NC(=O)CCc1c(F)cccc1Cl C1(C(C)NC(C2CC(CC)C2)=O)CCCN1C(=O)CC1(C)CCC1 c1(NC(C2(CNC(c3cnn(CCF)c3)=O)CC2)=O)ncccc1O C1(NC(C(=O)NC(C)C)=O)CCCC12CN(C(C13COCC1C3(F)F)=O)C2 C1(CNC(c2ccc(CC)o2)=O)CCN(C(=O)CSCc2ccncc2)C1(C)C CC(O)CN(C(=O)COCC1COC1)CCNC(=O)CN(S(C)(=O)=O)C C1(NC(c2cc(C)c(F)cn2)=O)CN(C(C2CNC(=O)N2)=O)CC(F)(F)C1 Cn1cc(S(C)(=O)=O)c(C(N2CC(CNC(C3(C)CCCCO3)=O)C(O)C2)=O)n1 C=CCC(CC(C)C)C(=O)NC1C=CC(C(=O)N(C)Cc2ccon2)C1 CC1(C(N2CCC(C(F)F)C2)=O)CCN(C(=O)C=Cc2ccncn2)C1 C1(OC)(CN)CCN(C(=O)Cc2ccc(F)cc2C(F)(F)F)CC1 CC1(NC(c2sc(F)cc2Cl)=O)CCCN(C(C23CCCC2C3)=O)C1 c1(OC)ccc(C(=O)NC2CCCC(CNC(=O)CN3CCCC3)C2)cc1Cl C=CCCCCCC(=O)N1C(C(=O)NC(C)(C)C(O)CO)CC1C CCCCC(CNC(=O)C(C)(O)CSC)NC(c1ccc(C(N)=O)nc1)=O C(c1ccc([N+](=O)[O-])cc1)=CC(=O)OC.c12cc(C#N)ccc1NC2=O c1(NC2C3(CCC(NC(c4ccn(C)c4)=O)CC3)C2)ncnc2c1c(Br)nn2C c1(CC)ccc(NC(=O)CCN(C)C(c2ccc(F)cc2)=O)cn1 C1(C(=O)NCCN(C(=O)CCc2cccc(C)c2)CC)CCCOC1C n1(CCC=C)cc(C(=O)N(C)CC2CCCC2NC(=O)COCP(C)(C)=O)nn1 c1(C(N2CC(C3C(C(=O)NC4(COC)CC=CC4)C3)C2)=O)ccn2cncc2c1 C(=O)(C(C)S(N)(=O)=O)N1C(C(N(CCN(CC=C)C)CC)=O)C(CC)CC1 C1(NCc2nnc(C)o2)CC2CCCC2N1C(=O)OCc1ccccc1 C1(C2CN(C(C3CC3F)=O)C2)(NC(CNc2nccc(OC)n2)=O)CC1 c1(C(=O)NC(C)CCCCNC(C2C(C)C2(F)F)=O)ccc(S(C)(=O)=O)cc1 N1(C(c2cc(C)no2)=O)CC2CCC1CN(C(=O)COC(C)(C)C)C2 N1(C(CCC(C)N(C)C)=O)C2CCC1CN(C(c1cccc(=O)o1)=O)C2 Cc1ccc(C(=O)NCCNC(=O)C(C)COC(C)C)c2c1CCCN2 C1(CNC(c2[nH]cc(C#N)c2)=O)CC12CCN(C(=O)CCCN1CCCC1)CC2 C1(C(=O)NCc2cnccn2)CCC2CCCCN12 N1(C(C(C(C)C)SCC)=O)CCN(c2ccccn2)C(=O)C1 c1(C(N(C)C)=O)cn(CC(=O)N(CCc2cn(C3CCCC3)nn2)CCS)nn1 n1(CCCOC)nnnc1C(c1ccc(C(C)C)s1)NCC(CC1CC1)OC c1(C(=O)NC(C(N2C(CC)COCC2)=O)C(C)C)cc2ncccc2[nH]1 c1(C(N2CC(O)(C(C)NC(c3nnc(CC)s3)=O)C2)=O)cc(O)ccc1OC Cc1cnc(C(=O)NCCC(C)(C)CNC(C2(F)CC2)=O)c(F)c1 c1(CCC(=O)N(CC(C)NC(C(C)SCC)=O)CC)cc(Cl)no1 N1(C(C2=CC(C)(CC)C2)=O)CC2=C(C1)CN(C(=O)COC1CC=CC1)C2 N1(C(c2nc(CCC)sc2)=O)CCC2CN(C(c3ccn(C(C)C)c3C)=O)CC12 C1(C(=O)O)(CSC)CCCN(C(C2CCC(Oc3ccncc3)C2)=O)C1 N1(C(c2cc(C)cc(Cl)c2)=O)CCC2C(C1)CN2C(c1ncc(Cl)cc1F)=O Cc1ccc(O)c(C(=O)NCc2cc(C(N3C4CSCC3C4)=O)on2)c1 N1(C(Cc2nc(C)sc2)=O)CC2CC(C1)CN(C(=O)CCC1(C)CC1(F)F)C2 CCCC(C)CC(C)(c1nnnn1C1CC1)Nc1cc(F)c(C(=O)OC)cc1F c1(C(C)C)ccc(CN(CCCN(C)C)C(=O)CN2CCOCC2=O)c(F)c1 C(=O)(CC1OCc2ccccc21)NC(CCOC)C(C)C C1(C(NOCCCC)=O)(NC(c2n[nH]cc2Cl)=O)CCCC1C c1(OC(C)C(=O)NC2CCC(NC(=O)C(C)(C)C)C2)ccccc1Cl C1(CNC(C(CO)NC(N)=O)=O)CCC(CNC(C2(C3CC3)CC2)=O)CC1 Cc1cc(CC(=O)NCc2ncoc2CCNC(=O)C(Cl)=CCl)cc(O)n1 c1(OC)cc2ccc(C(=O)NCC(F)CNC(c3ccccc3)=O)nc2cc1F N#Cc1cc(C(=O)NCc2cc(C(=O)NCCCc3ccco3)on2)cs1 N1(C(C2N(C(Cc3ccc(C)s3)=O)CCC2C)=O)CC(=O)NC(=O)C1 C1(C(=O)NCCC2CN(C(c3ccc([N+](=O)[O-])s3)=O)C2)CCc2ccccc2O1 c1(C(N2CCC(CN(C(C(CC)(CC)CO)=O)C)C2)=O)csc2cc(Cl)cnc12 O=C1CC(C(=O)NCC2(C(=O)NCC3CCOC3)CC=CC2)NC(=O)N1 c1(CN2CCCN(CCC(=O)OC)CC2)ccc(N(C)C)cc1Cl C(=O)(C1=CCCC1C)NCC1C(C(F)(F)F)CN(C(C2CC(OCC)C2)=O)C1 C1(C(=O)NC2(C(=O)NCC(CC=C)(F)F)CCSC2)CN2CCC1CC2 CC1CN(C(c2ccc(CO)s2)=O)CCC1NC(c1cc(C(F)(F)F)on1)=O N1(C(C(C)Cn2ccnc2)=O)CCN(C(c2ccc(N(C)C)c(F)c2)=O)C(C)C1 c1(C(N2CC3C(NC(c4ccn(CC)c(=O)c4)=O)C3C2)=O)ccc(C#N)nc1O c1(C(=O)NC2(C)CC(NC(=O)C3=COCCC3)C2)ccc([N+](=O)[O-])cn1 CCC(C)C(O)CC(=O)NC12CCC(C(N3CCCN(CC)CC3C)=O)(CC1)C2 C1(C(N2CC=CC2CF)=O)CN(C(c2ccc(O)cn2)=O)CC12CC2 c1(OC)nc(=NC2CC(CNC(C3(C)C=CCCC3)=O)C2)[nH]c2[nH]cnc12 C1(N(C)C)CN(C(C2(CF)CCN(C(C3CCCN3C)=O)C2)=O)CC12CC2 c1(C(C)NC(=O)Nc2cnccc2C(F)(F)F)nnc2ccc(=N)[nH]n12 C(C)(C)(C(=O)NCCCN(C)C(c1cc[nH]c1C1CCC1)=O)OC(C)C c1(C(=O)NCCCNC(c2c(C)c(Br)ccn2)=O)[nH]nc2ncccc12 N1(C(C(c2[nH]c(=N)sc2)=O)=O)CCCCC(CNC(=O)CCCCCF)C1 C(=O)(CC(C(C)C)NC(c1cc(O)cc(=O)o1)=O)N(CC(C)O)CCOC c1(C(=O)NCCN(CC(C)O)C(c2c(C)csc2)=O)cccc(CF)c1 C1(C(=O)NC(CNC(c2cc(C3CC3)ns2)=O)C2CC2)CC(=C(F)F)C1 c1(OC)ccc2nc(C(F)(F)F)[nH]c(=NCC(CO)OC)c2c1 C(=O)(CC(C)C(F)(F)F)NC(CC#CC)C(=O)NCC1(C)CCC(=O)N1C C1(NC(C2(C)CC(C)(C)C2)=O)CCC2CCN(C(=O)CS(=O)(=O)C3CC3)C1C2 C1(OC)CC2CC1CN(C(c1ccc(CNC(=O)C(C)(C)C(F)F)o1)=O)C2 CCCC(C)CC(=O)N(C(C)CNC(=O)C(CC)n1cncn1)CC S(=O)(=O)(c1ccc(C(N)=O)cc1)N(c1cc(OC(C)C)ncn1)C1CCNCC1 O=C(C1=NN(C2CC2)C(=O)CC1)NC1CC(NC(=O)C2CC2)C1 C1(CNC(c2cc3c[nH]cnc-3n2)=O)CCN(C(c2cnccn2)=O)C12CCC2 C1(OC)CCC(NC(=O)CCn2cc(-c3cc[nH]n3)nn2)C1 C(C(=O)N1CCCO1)NC(C(CC1CCC1)OC)=O CC1(NC(=O)CCc2ncco2)CCN(C(c2c[nH]c(Br)c2)=O)CC1 c1(-c2c(CC)cns2)nc(CSc2ccc(OC)cc2)nn1CC1CCCO1 C(=O)(C(COC)CC(C)C)NC(C(=O)N(C(CC)C(=O)OC)C)CO c1(C(N(C)CC2N(C(CCOC)=O)CCOC2)=O)ccc2ncsc2c1 C(CCCC(CO)NC(=O)C(c1ccc(F)cc1)F)NC(COC)=O.C1C(=O)N1 N1(c2cc(C)ncn2)CCCCC(NC(=O)CCC(=O)N2CCOCC2)C1 CC(C)(C(=O)NC1CC1CNC(=O)CC1CC1)S(C)(=O)=O C1(CC(C)C)CCCC1C(=O)N(CCO)Cc1ccc(C(N)=O)s1 N1(C(CCc2cn(-c3c(C(=O)O)cccc3)nn2)=O)CCCC2(CC2)C1 N1(C(c2nc(OC)c(C)s2)=O)CC(NC(C2(C)CC(C(F)(F)F)C2)=O)CC1(C)C c1(C(=O)NC2(CNC(CC)=O)CCOC2)cc2cc(C)c(Cl)cc2[nH]1 c1(CC(=O)N(C2CC2)Cc2c(OC)cccc2)cc2ccccc2cc1O C(=O)(C(CC(C)C)C(N)=O)NC1CC2(CC(NC(Cc3cn(CC)nn3)=O)C2)C1 c1(C(=O)NCCN(CCC)C(c2c(C)nn(C)c2C)=O)cccc2ncn(C)c12 C1(N(CCC)C(c2coc(SC)c2)=O)CCN(C(c2cccc(=O)o2)=O)CC1 c1(C(=O)NC(CCNC(C2CCN(C(CC)=O)C2)=O)C)ccc(N)c(F)c1 c1(C(N2CCC(CN(C(c3cnc(C)s3)=O)C)C2)=O)cc(O)nc2c1CCCN2 Cc1nc(C)c(C(=O)NCC2(CCNC(=O)C(C)N3CC(C)C3)CC2)nc1C c1(C(=O)Nc2cnc(Br)o2)cccc(-n2ccnc2)c1 c1(C(=O)NC2CCC(C)(CNC(c3n(C)cnc3)=O)CC2)cc(F)cc(F)c1O CC1CN(C(=O)CC(O)C2CCCC2)CCC1CNC(=O)C(c1ccccn1)O c1(C(N2CC3CN(C(C4C(CC)OCC4)=O)CC3C2)=O)cc2oc(C)c(C)c2[nH]1 C12CC(F)CN1C2=O.C1(C)(CNC(CNC(=O)OC(C)(C)C)=O)CC(C)(C)C1 N1(C(C2CN(C(=O)NC)C2)=O)CCN(C(=O)Cc2ccsn2)CC2(CC2)C1 C(CC(CC)C(=O)NCC1CCC1C(N1CCC(OCC(N)=O)C1)=O)=CC C1(CCNC(CC(C)CN(C)C)=O)CN(C(=O)CCC#N)CCS1(=O)=O C1(C(=O)NC(C=C)(C)C)CN(C(=O)C(C)(C)C(N)=O)CCC1(C)C N1(C(C(c2ccc(C)s2)C)=O)CC2CC(N(C(=O)COC3(C)CCC3)C)C1C2 Cc1cc(C)c(NC(=O)C(C)N(C)C(c2occc2C)=O)cc1C c1(CC)cc(C)c(C(=O)NCC2CCN2C(=O)CS(=O)(=O)NC2CC2)o1 c1(OC)cnc(Cl)nc1N1CC2(CN(C(=O)C(C)CC(C)C)C2)C1 C(C1CCCCCC1)=CC(=O)NC(C1OCCN(C(C(CCSC)O)=O)C1)C C=CC1(COC)COCCN1C(c1cc(-c2nn[nH]n2)ncc1F)=O C1(c2n(CC)nnn2)(NCC2(c3ccccn3)CC2)CCOC1C N1(C(C2CCN(C(=O)CCC3CC3)CC2O)=O)CCC12CCCOCC2 c1(C(N(CC(C)NC(=O)CCc2cc(C)on2)CC)=O)ccc(OC(F)F)cc1 CC1CC2(CCC2)CN1C(C1CN(C(=O)C2=CC3C=CC2C3)CC1(C)C)=O C=Cc1cc(C(N2CC(CNC(=O)C(C)(C)C)CC23CCC3)=O)cc(F)c1 C1(NC(CCCC=C)=O)CN(C(c2c(C)coc2C)=O)CC12CC2 N1(C(CCSCCCC)=O)CC(C)(C)CC1CN1CC(C)(C(=O)NCC)OCC1 Cc1cc(C(=O)NC2C3CN(C(=O)CC(C)(C)F)CC23)c(O)nc1C CC(C)(C)CC(O)C(=O)NCC1CCCC1NC(=O)CN1CCN(S(C)(=O)=O)CC1 C1(C)(C(N(CC(C)CNC(=O)C(c2ccc(Cl)cc2)CO)C)=O)CC2(CCC2)C1 C1(NC(c2cc[nH]n2)=O)CS(=O)(=O)C2CN(C(=O)C(c3cccnc3)O)CC12 N1(C(c2c(OC)csc2)=O)CCN(c2ccccc2C(F)(F)F)CC1 C(=O)(C#CC(C)(C)O)NC(C1CCCN(C(c2cc(F)cnc2O)=O)C1)C C1(N(C)C(C2CC(F)C2)=O)CCCN(C(=O)CCc2n[nH]c(=N)s2)CC1 c1(C(=O)NCCC2(NC(CC3C(C)C3)=O)CCC2)cncn(C)c1=O C1(C(=O)NC2C(NC(c3c(CC)ncs3)=O)CCCC2)CCCNS1(=O)=O C=CC(C(=O)NC(C(N1C=CCCC1)=O)C1(C)CC1)OC N1(C(c2ccccc2Cl)C(=O)NCCCSC)CCC12CCC(CO)CC2 C12(CNC(C3N(CC)CC3)=O)CCC(CN(C(c3ccnc4c3CCC4)=O)C1)C2 c1(C(=O)NCCC2CSCCN2C(=O)CCC2CCCO2)ccc2ncnn2n1 c1(C(N2CC(O)C(O)C2)=O)cc2ccc(Br)c(Cl)c2s1 C(=O)(C1=NOC(C)(C)C1)N.C1(NC(CN(CCOC)CC=C(C)C)=O)CNCCC1C C(=O)(C(C)N=[N+]=[N-])N(C1CC(C(=O)NC(C(=O)NC(C)C)C)C1)C Cc1cc(Cl)cc(C)c1C(N1CC(CNC(=O)CCC2CCCOC2)C(O)C1)=O c1(C(=O)NC(CNC(c2nc(C)n(C)c2)=O)C(C)C(C)C)c[nH]c(C)c(Cl)c1=O N1(C(C(C)CN2CCOCC2)=O)CCC(NC(=O)C(N2CCC(O)CC2)C)C1C Cc1nnc2ccc(C(N3CCCN(C(=O)CC(F)(F)F)CC3)=O)cn12 C(=O)(CC(C)CCC)N(CC1CC(NC(c2ccc(CCC)o2)=O)C1)CC c1(C(=O)NCCOC2CCN(C(CC(C)c3cnn(C)c3)=O)C2)cn(C)[nH]c1=N C1(C(=O)OCC)Cc2nnc(C(=O)NNC(=O)NCC(c3ccccc3)C)n2C1 N1(C(CNS(CC)(=O)=O)=O)CCCN(C(=O)C=Cc2cscn2)CC1C(C)C c1(C(=O)NC2(CN(C(CS(CC)(=O)=O)=O)C)CC2)ccc2c(c1)CCCO2 O=C(C1=CCS(=O)(=O)C1)N1CCN(C(c2ccc(F)cc2O)=O)CC1 N1(CC(=O)NCC2C3CN(C(c4cc(C)oc4C)=O)CC32)CCn2ccnc2C1 c1(C(=O)NC2CC(O)(CNC(C(CC=C)(C)C)=O)C2)nc2ccccn2c1F C(=O)(N1OC2CCC1CC2)C1C2N(C(c3c(CC)nc(C)o3)=O)CC(C=C2)C1 CCCC(C(O)C(=O)NC1CC2C=CC1C2)NC(C1(OC)CCCOC1)=O C1(NC(c2n[nH]c(C)c2C)=O)CN(C(c2ccc3c(c2)CCO3)=O)CC(C)(C)C1 C1(NC(c2cc(C)c(C)nn2)=O)CN(C(=O)CSC(F)F)C2(CCOC2)C1 CC1CC(C(=O)N(CCF)C2CC2)CN(C(=O)CCc2ccnn2C)C1 C1(C2CC2)(C(=O)NCC2C3CN(C(CC4(C)CCCO4)=O)CC32)CCOCC1 c1(N(C)C2CC2)ncc(-c2cn(CCC(N3CCC(c4ccco4)C3)=O)nn2)cn1 c1(C(=O)OC(C=CCC)C)ccc(C)nc1OC c1(CC(=O)NC(C(=O)N(C)Cc2scc(C)c2)(C)C)ccccc1C c1(OC)ccc(I)c(C(=O)NCCN2CCN(C(=O)CCC(C)=O)CC2)c1 c1(CNC(C2C(NCc3cc(C)ncc3)CCC2)=O)ccc2c(c1)CCCO2 C#Cc1ccccc1CC(N1CCCC(CN(C(=O)C(C(C)C)SC)C)C1)=O C1(CN=c2nc(NC(=O)OC(C)(C)C)s[nH]2)CC2(C1)CC1(CCC1)C2 Cn1nc(CNC(=O)CNC(=O)CCc2cnn[nH]2)oc1=O N1(C(C2CC2[N+](=O)[O-])=O)CCCC(C2CN(C(C34CCN(CC3)CC4)=O)C2)C1 CCC(C)C(O)C(=O)NCC(=O)NCCCNC(N)=O N1(C(c2cc(C)on2)=O)CCC(O)C(C(=O)NCCCN2C(=O)C=CC2=O)C1 c1(C(=O)NCCOC2CN(C(CNC(=O)OC)=O)C2)cnc(O)n(C)c1=O CC1CCOCC1C(N1CCOCC1CC(=O)N(CCCCCO)C)=O CCCS(=O)(=O)CC(=O)NCCC1CCCCN1C(=O)C1=CCCC1 N#Cc1cc(CN2C(C(=O)NCc3ccc4c[nH]nc4c3)CC2)cc(F)c1 CCCC(CNC(C1(Br)CC1)=O)NC(=O)C=CC1CC1 C1(C(=O)NC(C(=O)NCC(=O)NCCOC)C(C)C)CCCCC1(C)C c1(NC)c(C(N2CCC2CNC(=O)CC2CCCCC(=O)N2)=O)sc2nccnc12 N1(C(=O)CC2C=CC(NC(C3(CO)COC3)=O)C2)CCOC2CCC12 N1(C(C2(C#C)CCCC2)=O)CCC2(CCN(C(C3(C(F)F)CC(=C)C3)=O)CC2)C1 C=C(C)C(CC(=O)N1CC2CC2C1C(N1C(CC)CCC1C)=O)OCC N1(C(C(C=C)(C)C)=O)CCCCCC(NC(=O)CSc2nncn2C(C)C)C1 N1(C(C2(C)C(C)C2)=O)CCCC2(CCCN2C(=O)C=CC2CCOCC2)C1 C(C(=O)NOC1CCCC1)(c1cccnc1)NC(C1C(C(=O)OCC)C1)=O c1(C(N(C)CC)=O)ccc2c(c1)C1(CCCC1)CN2C(c1ncc[nH]1)=O c1(C(N(C2CC3CN(C(C=CC=CC)=O)C2C3)C)=O)cncc2cnccc12 C#Cc1cnn(CC(=O)NCCC2(C(=O)NC3CCOC(C)C3)CC2)c1 N1(C(C(C=CC)O)=O)CCC2(CCCC2CNC(=O)COc2ccsc2)CC1 C(=O)(CC(C(F)F)NC(C1C2CCCC12)=O)N(C)CCO N1(C(c2c(CC)non2)=O)CCC2(CC2NC(c2cc(O)ncc2F)=O)C1 CCC(C(=O)NCC1CN(C(=O)CCc2cccc(O)n2)CCCO1)C(F)(F)F CN1CC(=O)NC(CC(=O)NC2CN(C(=O)CCS(C)=O)CCC2F)C1=O c1(C(=O)NCC(CNC(CC(CC)C)=O)C(F)(F)F)cccc2ncnn12 N1(C(COC(CC)C)=O)CCN(C(=O)C=C(Cl)Cl)CC1CCO N1(C(C2C(CC)OCC2)=O)CC2CCC1CN2C(c1cccnc1OC)=O C(=O)(CS(=O)(=O)C1CC1)NC1C(CNC(C23OC(C)(C)C(C2)C3)=O)CCCC1 c1(C(=O)Nc2cccc(OC)c2)cc(O)ccc1Br N1(C(C2ON=C(C)C2)=O)CCC(C)(NC(=O)C(=O)Nc2ccccc2)CC1 C(CO)(C(O)C1CCCCC1)NC(CCNC(C=C)=O)=O c1(OC)cc(OC)c(C(=O)NCCCNC(C2CC(C)(C)CO2)=O)cc1OC C1(NC(CC(=O)Nc2ccccc2)C(F)F)CCc2ncccc2C1 C1(NC(C(C)OCC#C)=O)CCCCCC1C(=O)NC(c1c[nH]ccc1=O)C c1(C(N2CCN(C(CC3CC(=O)C3)=O)C3C2C3)=O)[nH]c2ccc(F)cc2c1Cl c1(C(N2CCC(O)(C(C)NC(c3ccc(C)nn3)=O)C2)=O)nnn2c1COCC2 CC(C)(C)CCC(F)C(=O)N1CCC(CCC(=O)NC2CC(C(F)F)C2)C1 CC1(C)COCC1C(=O)NC(C1CCN(C(C2(c3ccccc3)CC2)=O)C1)(C)C CC1CCCN(C(=O)C(=O)NCCN(C2CCCC2)C(=O)CC2CC2(Cl)Cl)C1 CCC(C)C(=O)C(=O)N1CCCC(F)(CNC(c2ccc(F)s2)=O)C1 CN1CCc2ccc(NC(C3CCCN(S(=O)(=O)C(F)(F)F)C3)=O)cc2C1=O N1(C(c2c(C)n(C)nn2)=O)CC2(CCN(C(=O)CC3CCCCC3F)C2)C1 C1(C(=O)NN2C(C3CC3)C2)CCCCCC1.C(C)(C(=O)C1CC1)C(CC)=O.OC C(=O)(CCCCCN=[N+]=[N-])NCC(C)(C1CC1)NC(=O)CC1CC1(C)C CC1CCN(C(=O)CN2CCN(C(C3(n4cnnn4)CC3)=O)CC2)CC1CO c1(OC)cc(C2(C(=O)N(CCCCCNC(c3cnc[nH]3)=O)C)CC2)ccc1C C1(NC(CN2C(=O)CCC2=O)=O)C2CC3C1C3C2C(=O)N1CCCCO1 CCC(CC(=O)N1CCCCC(CCC(=O)NCCCc2nncs2)C1)C(C)C O=C(CCC(F)(F)C(F)F)NCC(C1CC1)NC(C1CC1F)=O C1(NC(C(CN(C)C)NC(C#CC(C)C)=O)=O)CCCCC12CC2 C1(CNC(C(C)OCC=C)=O)(COC)CCCN1C(c1cnn(C)c1N)=O CC(C)(CO)C(=O)NCC1CN(C(C2CCC(F)C2)=O)CCO1 c1(CNc2nc(-c3c(OC)cc(I)cc3)sc2)c(Br)cc(Br)c(O)c1Br CC(C)(C)C(=O)CCCC(=O)O.C1(C)CC2CC(c3ccccc3)CC12 C(=O)(C(F)C(C)C(F)(F)F)N1C(CNC(c2c(C)ncs2)=O)CCCC1 N1(C(=O)NC(C(C(F)(F)F)OC)C)CC2(CCC(=O)N2)C1 c1(C(=O)NCCC(C)NC(=O)CCC2CC2)nc[nH]c2nccc1-2 N1(C(C(C)=CC)=O)CCC2(CCC2NC(=O)CCc2cccnc2C)CC1 Cc1c(C(N2CC3CCC(C2)N3C(C2CCCC23CC3)=O)=O)cnc2ncnn12 CN1C(=O)CSC1=CC(=O)NCC(O)CCNC(c1ccc(C2CCOC2)s1)=O C1(C(N(C)Cc2cn(CC)nn2)=O)CCC=CC1NC(C1CCCOCC1)=O c1(CC)nc(-n2cccc2)sc1C(=O)NC1CCN(C(=O)C(C)(CO)OC)C1 C1(NC(C(C)OCCOC)=O)CCCCC1CC(=O)NCC(C)C(=O)NC N1(C(C2CC(O)(CNC(Cc3n(C)ccn3)=O)C2)=O)CCC(C)(CCO)C1 C=CC(CC)CC(=O)N(CC(=O)NC1CCCNC1=O)C(C)C c1(N2C(C(=O)Nc3c(Cl)cc(F)cc3Cl)CC2)ncnc2cnccc12 c1(C(c2cn(CCNC(C3CN(C(C)=O)C3)=O)nn2)=O)cc(Cl)ccc1Cl Cc1ccc(S(=O)(=O)CC(C)NC(C2(c3nnnn3C)CC(C)N(C)C2)=O)cc1 N1(C(CC(C)c2ccccc2)=O)CCN(C(=O)CC(C)O)C(C#N)C1 c1(NC2CCCC(NC(c3occ(C)c3)=O)C2)cc(O)nc(=O)n1C c1(CC(=O)NC(CNC(C2(CC)CCNC2=O)=O)(C)C(C)C)c(C)nn(C)c1C c1(CC)nnc(CNC(c2ccn(C3CC3)n2)c2nnnn2C2COC2)o1 CCC(C(=O)N(CC)CC1CCCN1C(C1CC2(CC(=O)N2)C1)=O)C(C)O S(=O)(=O)(c1cccc(Br)c1F)N(C1CCCN(C(CC=C)=O)C1)C c1(C(=O)NCC(CC=C)NC(=O)CC2CCS(=O)(=O)C2)[nH]c(C)c([N+](=O)[O-])c1C Cc1cnc(C(N2CC3C(c4cn(C(C)C(=O)O)nn4)C3C2)=O)c(C(F)(F)F)c1 C(CC(=O)NOCC(=O)OC)N(CC#C)C(c1ccc(C(N)=O)o1)=O Cc1c(Cl)c[nH]c(=NCC2CN(C(C34CC3C4)=O)CC23CCOCC3)c1C#N C1(C)(C(=O)NCC2(CO)CCN(C(CC=C)=O)C2)C2Cc3ccccc3C12 C1(CNC(Cn2c(C)ccn2)=O)CC2CCC(C1)N2C(=O)Cc1cc[nH]c1 C(CC(O)CC(=O)NCC(C)(C)CC1CN(C(=O)CC2CC2)C1)SC c1(NC(CC2(NC(c3ccc(OC)c(Br)c3)=O)CCC2)=O)cccc(Br)c1C#N c1(C(=O)NC2(COC)CCN(C(=O)CC3CN(C(C)=O)C3)C2)cccc(C)c1F C1(NC(c2ccc(CCC)s2)=O)CCN(C(c2snnc2C)=O)CC1C(C)C c1(OC)cc(CN(C(c2ccccc2)CCO)C)cc(C(C)C)c1OC Cc1ccc(C(=O)NCC(N2CCN(C(c3ccsn3)=O)CC2)C(F)F)c(C)c1 C1(C(N(C)CC2(CO)CC2)=O)CC2CCC(C1)N2C(=O)C(C1(O)CCCC1)F c1(OC)cc(OC)c(C(=O)NCC(O)CN(C)C(c2ccccc2)=O)c(F)c1 c1(C(=O)NC(CNC(C(=O)NCC)=O)(C)C2CCC2)cnc(C(F)F)c(Cl)c1 CC1CN(C(c2n[nH]cc2Cl)=O)CC(CCNC(c2cnc(Cl)[nH]2)=O)O1 C1(NC(CC=C=C)=O)CCC12CN(C(=O)CC1CC(F)(F)C1)C2 C1(CNC(c2[nH]cc(C#N)c2)=O)CCC2(CN(C(=O)COC3CCCOC3)C2)O1 CC1(C(=O)NC2C3CN(C(=O)Cn4cc(C5CC5)nn4)CC23)CC=CCO1 N1(C(CN(S(C)(=O)=O)C)=O)CCC2(CC1)CC2NC(c1c(O)cc(Cl)cc1F)=O C(CCC(=O)NC1(C(=O)NCCC(F)(F)Cl)CC1(C)C)OCCC C1(C(=O)NC(C#C)CC)CCN(C(c2cnn(C(C)C)n2)=O)CC1 N1(C(C2C(C)(C)COCC2)=O)CCC(C2CCN(C(=O)Cc3cc[nH]c3)C2)CC1 CC1(C(=O)NC2CC2NC(=O)Cn2cnnn2)CCc2ccccc2C1 c1(N(C)C)noc(CNC(=O)C(CNC(=O)CCC2CCCO2)N(C)C)n1 C#CCN(OC)C(=O)C1CN(C(C2COCCC2C)=O)CCO1 C1(Cn2cc(CN(C)C(C3CN4CCN3CC4)=O)nn2)Cc2ccccc2O1 C1(CNC(c2cnn(CC(F)F)c2)=O)CCCN1c1ncns1 C1(NC(CCCCCC)=O)CCSC12CN(C(=O)C(C(C)(C)C)NC(C)=O)C2 N1(C(C=C(CCC)C)=O)CCN(C)CC1C(=O)NC(c1noc(C)n1)CC C1(CNC(N(CC(CC=C)O)C)=O)COCCC1(F)F C1(NC(C(C)=CC2CC2)=O)CCN(C(C23CCC(C)(CO2)C3)=O)CC1(C)C N1(C(c2n(CC)ccn2)=O)CCSCC1CCNC(C1C(C=C(C)C)C1(C)C)=O N1(C(C=C(C)CNC(C2CCCCO2)=O)=O)CC2CC2C2CC12 C1(NC(CN(C)C(c2ccoc2)=O)=O)CCCC1NC(C1(Br)CC1(C)C)=O N1(C(c2[nH]cc(CC(C)C)c2)=O)CC2CC(NC(C3CC(O)C3)=O)C1C2 N1(C(C2N(C(CCC=C(C)C)=O)CCC=C2)=O)CC2(C1)NC(=O)NC2=O CC(C)(C)C(C#N)C(=O)NC1C2CC3C1C3C2C(=O)NCC1CCC2(CC2)C1 C(=O)(C(C)C(=O)NCC(c1ccccc1)N(C(=O)Cc1c(Cl)cnn1C)C)OC c1(C(=O)NC2CC(OCC)C2OC)cnc2c(c1)S(=O)(=O)NC=N2 c1(OC)cccc(CC(O)C(=O)N2CCC(NC(c3ccc(C)o3)=O)C2)c1 CCCCCCC(CC)(CC)C(=O)N(CC(C)NC(c1[nH]nnc1COC)=O)C C=CCCCC(C1CC1)NC(c1nnnn1CC(=C)C)(CC)C1CC1 CCS(=O)(=O)c1ccc(CC(=O)N(C2CC3CCC(C2)N3C(=O)C(C)O)C)cc1 CC(CCN(C)C)N=c1[nH]c(=NCCc2csc(O)n2)[nH]c2c(F)cccc12 Cc1cc(F)c(NC(=O)C(O)CCCNC(=O)Cn2cnc(=N)[nH]2)cc1F c1(C(N2CCCC(C(=O)OCC)C2C)C(=O)NCCSC)cnc2ccccn12 C(=O)(CC(C)C(F)F)N1CCC(N(C(C(c2cnn(C)c2)C)=O)CCO)CC1 C(=O)(CCCCCCCC1CC1)NC12C(CN(C(C(CC)n3ccnc3)=O)C1)C2 C(=O)(CC(C)(C)C)NCC(=O)NCC1CCC(NC(C(C)NC(N)=O)=O)C1 C(=O)(CCC(=O)N1CCCC(NC(=O)C=CC2CC2)C1)N(C)C C1(NC(C(CC)(C)C)=O)CN(C(=O)Cc2n[nH]c(C)n2)C(C)(CC)C1 n1(CC(=O)NCCCCCNC(C2CC2(F)F)=O)nnn(C2CC2)c1=O Cn1cnc2c1CCCC2C(=O)NCC1CN(C(c2n[nH]cc2F)=O)C1 C12(CNC(c3c(C)ccnc3)=O)CCCC1CCN2C(=O)CCc1nccn1C n1(CC(=O)NC23CCC2CN(C(=O)CC24CCCC2C4)C3)nc(O)ccc1=O C1(C(N(CCOCCNC(C2CC(C)(CC)C2)=O)C)=O)OC(C)(C)OC1(C)C C12(C(N3CCCC3(C)CNC(CN(C)C(c3cccs3)=O)=O)=O)CC1COC2(C)C N1(Cc2c(C)ccc(F)c2)CCc2oc(CO)cc2C1 CC(CC1CC1)C(=O)NCC1(F)CC(NC(c2cnn(C3CCC3)c2)=O)C1 n1(CC(=O)N(C(CC)CNC(=O)CCCN2CCCC2)C)cc(Cl)cn1 C(=O)(C(C)(C)S(C)(=O)=O)N1C(Cn2cc(CCCC)nn2)CCC1 C12(C(=O)NC3CC(OCC)C3)CC(C)(CN1C(C1(CO)CCCCC1)=O)C2 c1(-c2cn(C)nc2)cncc(NC(c2cc(C(C)(C)F)on2)=O)c1 C1(NC(c2cc(CC)on2)=O)CCC(C(=O)NCCC2CCCCO2)CC1 CC(C)C1=NOC(C)(C(=O)NCC2CC2CNC(c2cnc(O)s2)=O)C1 C1(C(=O)NC(CNC(C2N(C(C)=O)CCC2)=O)CO)CCC2(CCC2)CC1 c1(SCS(=O)(=O)CCNC(CCO)C2CC2)ccc(F)c(F)c1 N1(C(C2C(CC)CCO2)=O)CCCN(C(c2ccc(F)c(F)c2C)=O)C(C)C1 N1(C(C(C(C)OC)NC(c2cn(CC=C)nn2)=O)=O)CCn2cc(C)nc2C1 C12CN(CC1C)C(=O)c1ccccc1OC(=O)c1noc(n1)CC2.CCOC C1(C(=O)NCc2ccns2)(CNC(C(CC)N(C)C)=O)CCCCC1 c1(CC)nc(C)cc(=NCCCCC(C)NC(c2ccc(Cl)cc2C)=O)[nH]1 C1(OC)(CNC(=O)C=C(C)C2CC2)CCN(C(=O)C(C(C)C)C2CCC2)CC1 C1(C(=O)NCC2N(C(C3CC(OCC)C3)=O)CC(C)(C)C2)CC(C2CCCC2)C1 N1(C(C(=O)OC)C2CC2Cl)CC2COCC2(CCN)C1.N1(CC2CCCO2)CCOCC1 N1(C(c2c(CC)cccc2)=O)CC2C=CC1C(C(=O)NCc1cccc(C)n1)C2 C1(C(=O)Nc2c(NCCc3c(C)n[nH]c3C)cccc2)CCc2ncccc2C1 c1(C(N(CCCCNC(CC2CC(CC)C2)=O)C)=O)sc(Cl)c(Cl)c1N C(C(C)(C)C(=O)NCC=CCNC(c1sc(NC2CC2)nc1C)=O)OCC CCC(C)(C)C(C)CC(=O)NCC1CC(OC)CN1C(c1cc(F)ccc1N)=O c1(C(=O)NC2C(CNC(c3cccc(C#C)c3F)=O)C2)ccc2cccnc2n1 c1(NC(C2CC(CCNC(CC(C)OC)=O)C2)=O)cc(C)c(O)cc1C C(=O)(C1=CCCOC1)NC(CNC(C1(C(F)F)CC(=C)C1)=O)C C1(C(=O)NC(C=C)COC)CCC(CNC(=O)CC2CCCCC2C)CC1 N1(C(c2c(CCC)n(CCO)nc2)=O)CC(NC(=O)C(O)C2CC2)CC(F)(F)C1 c1(C(=O)OCc2nnc(C)n2C)ccc2c(c1)nc(O)n2C c1(CNCc2cnn(C)n2)cncc(F)c1.c12nnnn1C2C1CC1 c1(C(=O)NCC2CCN(C(C3N(C)CC3)=O)CC2O)ccc2cnoc2c1 N1(C(C(CCCCC)O)=O)CC(NC(=O)Cc2cn(CC)nn2)CC12CCCC2 CCCCCC(C)(C)C(=O)NCC1CN(C(C2CCCN2C)=O)CC1C C1(OC)CN(C(=O)CCn2ccnn2)CC1NC(=O)C(CCN(C)C)N(C)C C1(n2cc(C(C)(C)OC)nn2)CCC(C(=O)NCc2cscn2)CC1 Cc1ncc(C(N2CCCC(n3ccc(C(F)(F)F)n3)C2)=O)cc1C1CC1 N1(C(C=Cc2c(C)n[nH]c2)=O)CCC(NC(C2CC2(F)F)=O)C12CCC2 N1(C(C23CC(C)C2C3)=O)CCCC2(C1)CN(C(c1c[nH]nc1[N+](=O)[O-])=O)CCO2 C1(OCC(=O)OCC2(C(=O)OCC(=O)C3CC3)CC2)CCCO1 N1(C(C(C(C)C)NC=O)=O)CC2CCC(C(=O)NC(c3cn(C)cn3)C)(C2)C1 Cc1cc(C(=O)NC2CCCC(NC(=O)Cc3csc(C(C)C)n3)C2)cnc1O c1(N(C)C)ccc(Br)c(C(=O)NC2CCCC2CNC(=O)COC(F)F)c1 N1(C(C(CC)C)=O)CCC(F)(C(=O)NC(c2ccc(Cl)cc2)CO)CC1 c1(C(=O)NCC(C)NC(C2CC(N(C)C)C2)=O)cc2c(C(F)(F)F)cccc2s1 c1(N2CC(C)NC(=O)C2)nc(NCCCSC(F)F)c2c(n1)CCS2 C(c1cnc(O)nc1O)=CC(N1CCC(O)(C(C)NC(c2nc(C)[nH]n2)=O)C1)=O c1(CCC)[nH]nc(C(N2CC3(C2)CN(C(C2(CC4CC4)CC2)=O)C3)=O)c1[N+](=O)[O-] C(C)(C(=O)OC)NC(=O)NCCNCCC c1(-n2cc(COCC(=O)NC3CN(C(=O)C(Cl)=CCl)C3)nn2)ccccc1Br c1(C(=O)NCC2C(NC(Cc3cc(CC)no3)=O)C2)cc(Cl)cc(Cl)c1OC N1(C(CS(CC)=O)=O)C(CNC(=O)C=CC(N2CCOCC2)=O)CC2CCCC12 C1(C(N2CCCCCC2)=O)COCCN(N2CCc3c(O)cccc3C2)C1 n1(CC(=O)NCCC2CSCCN2C(=O)CCCCF)cc([N+](=O)[O-])cn1 C(=O)(C1=C(Cl)CCC1)N(C1CCCN(C(=O)C(C2CCOCC2)O)CC1)CC C12(OC)CCCC(C(=O)NC3CC(NC(=O)C=CSc4nc[nH]n4)C3)(CC1)C2 c1(C(C)C)csc(CCNC(c2cc(Br)cs2)c2nnnn2CC2CCCO2)n1 C(=O)(CC(C)(O)c1ccccc1)NCC(C)NC(=O)C(C1CCCCCC1)O C1(C(C)C)C(NC(c2cc(C3CCC3)[nH]n2)=O)CCN1C(C1(C(F)(F)F)CC1)=O c1(C(C(=O)OC)NCC(C)OC(c2ccc(F)cc2)=O)cccc(OC2CC2)c1 Cc1cccc2c1OCC2C(=O)N1CCC(O)(CNC(=O)CN2CC(C)C2)C1 c1(OCC(=O)NC2CCCN(C(c3c(C#C)c[nH]n3)=O)C2)cccc(SC)c1Cl C1(NC(c2cc(C)c(F)cc2)=O)CN(C(=O)CC(=O)OC(C)(C)C)CC12COC2 C1(CC(=O)NCC(CNC(=O)CC2CCC(=O)CC2)OC)CCOCC1(C)C c1(C(=O)NC(C2(CNC(C3COC(=O)C3)=O)CC2)C)cn(CC2CCCO2)nn1 c1(OC)ccc(CC(=O)NC2CC2C(=O)NCc2ccc(F)c(OC)c2)cc1F c1(OC)ccc(C(C)CC(N2CCN(C(C3CC(CC4CC4)C3)=O)CC2)=O)cc1 Cc1ccccc1-n1nccc1C(=O)NCC(C)NC(=O)C=Cc1cnccn1 N1(C(C2OCCN(C)C2=O)=O)CC2CCCC(NC(C3CCC(=O)C3)=O)C2C1 c1(C(N(CCCNC(c2cnn(CC)c2C)=O)CCO)=O)cnc2sccc2c1 n1(CC(=O)NC2C(C)CN(C(c3ccsc3)=O)C2)c(=O)nc(O)c2ccccc12 C1(C(=O)NC2(C)CC(NC(C3(C(C)(F)F)CCC3)=O)C2)CC2CCC1C2 C(C(C)CCCC(C)C)NC(CC1(C)CCN(C(C(CC)n2ccnc2)=O)C1)=O C#CCC(C(=O)N1CCCC(=C)C1)NC(=O)C(O)CC CC(C)C(O)C(=O)N(CC(O)CNC(c1cc(C#N)on1)=O)C C(=O)(C(C)(C)CCF)N(CC(C)(C)CNC(=O)C=CC(F)F)CC Cn1nc(C(=O)NC2(CCNC(C3(C)CCCS3)=O)CCC2)c2cc(F)ccc12 N1(C(COCCCC#C)=O)CCN(C2CCN(C(c3ccc(O)nn3)=O)C2)CC1 C1(C(N2CCC(NC(C(CC)CN(C)C)=O)(CF)C2)=O)CCCCC(=O)N1 c1(CC)cc(C(=O)NC(C)(CNC(=O)CCCC2CCCC2)CO)on1 c1(C(N2C(C)CC(CNC(=O)CNC=O)CC2)=O)nn(C)c2ccccc2c1=O N1(C(C(N2CCOC2=O)C)=O)CC(NC(=O)Cc2ccco2)C(O)C1 CC1(C)CC(CNC(c2cncc(Cl)c2Cl)=O)N(C(=O)Cn2cnnn2)C1 c1(C(=O)NCCCN(C(=O)CC2C=CCCC2)C2CC2)ccc(S(C)(=O)=O)o1 CC(C)(CC(=O)N1CC2CC2(CNC(C2CCCCC2(C)C)=O)C1)C(F)(F)F C=CC(C)(CC)C(=O)NCCC1(NC(=O)CCN2CCN(CC)CC2)CCC1 c1(CC)nc(N2CCCC(NC(c3cc(C(N)=O)[nH]n3)=O)C2C)cc(C)n1 C=CCC(C)(C)C(=O)N(C)CC1CCCN(C(c2c(C(F)F)n[nH]c2C)=O)C1 Cc1cc(C(=O)N(CC(=O)NOCC2CCC2)C(C)C)c(C)[nH]1 N1(C(C2(C=C)CCC2)=O)CCC2CCC(C1)N2C(c1ccc2c(c1)CC(C)O2)=O C1(C(=O)NCC(CN(C(=O)C=CC=C(Cl)Cl)C)O)CCc2nc(C(F)(F)F)cn2C1 Cc1cc(C)c(C(N2CCCC3OCCC23)C(=O)Nc2ccccc2Cl)cc1C N1(C(c2c(OC)nn(C)c2)=O)C2CCC1CC(CNC(=O)C(F)C(C)(C)O)C2 N1(C(c2cc(C(C)C)no2)=O)CC(NC(=O)CSc2nncs2)C2CC12 c1(CC)cccc(C(N2CCCCC2c2nccs2)C(=O)NC2CCCC2)c1F C1(C(N2CC3(C(C(=O)OC)C3)C2)=O)CC(O)CCN1C(C1CC1C(N)=O)=O c1(C(=O)NC(CNC(CCCC)=O)(C)CO)cnc2c(=O)[nH]ccc2c1 c1(C(N2CCC(NC(c3cc4occc4s3)=O)(CF)C2)=O)cc(=O)cc(Cl)[nH]1 N1(C(CC(=C=C)C)=O)CC2C=CC1C(C(=O)NCC(C1CC1)N(C)C)C2 C1(O)(CNC(C(Cc2cc[nH]n2)NC(C(C)=C(CC)C)=O)=O)CCN(C)C1 N1(Cc2ccc(C(=O)NC(C)C)cc2)CCC2C(CCN2C(=O)C(F)Cl)C1 c1(C(=O)NCCCN(C(=O)CC23COCC(C2)C3)CC)cccnc1SC(C)C C1(NC(COCC(C)(C)C)=O)CC12CCN(C(c1cc(C(C)(C)C)no1)=O)C2 C(=O)(C1=C(Cl)CCC1)NCC1(C)C(NC(C(C2CCCCCC2)OC)=O)CCC1 c1(C(N2CC(NC(CN(C(C)=O)C)=O)C3C2C3)=O)cccc(Cl)c1Br C1(C)(CNC(c2cn(C)nc2)=O)CC(F)(F)CN1C(c1nccc(N)c1Cl)=O c1(COC)ncc(C(N2CC(NC(C3OCCO3)=O)C(O)C2)=O)c(O)n1 CC1CCC(Cl)=C(C(=O)NCCCOCCNC(c2cc(C(N)=O)cs2)=O)C1 C1(CC(=O)N(CC(C)O)C(C)C)CN(C(C2CCCC(O)C2)=O)CC1C c12ccc(cc1)C(C(=O)NC1CC1)OC2=O.c1(CCNCC)ncc[nH]1 N1(C(C(C)SCC)=O)CCC(C2CCCN(C(c3cnc(Cl)n3C)=O)C2)CC1 C1(CC(=O)N(CCCNC(=O)C(F)n2ccnc2)C)(C(F)(F)F)CCC(=O)NC1 N1(CC(=O)N(C2CCN(C(=O)C(O)CC3CCCCC3)C2)CCC)CC(C)(C)C1 C1(C(=O)NCCCOCC)C(C2CC2)CCN1C(C1CCCCC1)=O N1(C(CCCN(C(c2ccc(C#C)cc2)=O)C)=O)CCC(F)(F)CC1C C(C)(CNC(=O)C(Cl)=CCl)(CNC(c1nccn1C)=O)OC C(CN=c1[nH]cc(C#N)c2ccsc12)N(C(C(c1ccc(F)cc1F)C)=O)C C1(NC(CC2C(C(=O)OC)C2(C)C)=O)CCOCC1NC(=O)Cc1n[nH]c(C)n1 Cc1cnc(C(=O)NCC2CC(NC(c3n[nH]c(C)c3Cl)=O)C2(C)C)cc1Cl C1(CC)CCCN(C(c2cncnc2)=O)C1C(=O)NC1CC2OCCCC12 c1(NC(c2cc(C)cc(Br)c2)c2nnnn2C2CCCC2)cnc(C)c(C#N)c1 CC1CCCc2c(C(=O)N(C)CCNC(=O)CCc3cccc(Br)c3)cnn21 C1(CNC(COCCOCC)=O)CC12CCN(C(c1cscc1OC)=O)CC2 c1(COC)nc(NCC2(C)CSC2)cc(=NC2CCc3ccc(C)cc32)[nH]1 C1(CC(N2CC(NC(c3c(CC)nco3)=O)C(C)C2)=O)CCOCC1(C)C c1(NC(C2N(Cc3n(CC)ccn3)CC(O)C2)=O)cccc(C)c1C c1(CNCC2N(C(C(C)S)=O)CCCC2)cccc(Br)c1O N1(C(C(c2ccc(F)cc2)C)=O)CCN(C(C2CCC(=O)O2)=O)C(CC(F)F)C1 Cc1cc(O)ncc1C(=O)N(C1CN(C(=O)C(N2CCC(C)C2)=O)CCC1O)C C1(C(C)NC(C2(N(C)C)CC2)=O)CCCN1C(c1ccc(Cl)[nH]1)=O O=C(C1=CCCOC1)NC1CN(C(C2CCCO2)=O)CCC1F C1(C(N2CCC(CNC(=O)CCC3(C)CCC(=O)N3)C2)=O)(OC)CCC(C)CC1 C1(C(N2CCN(C(c3cnc(O)o3)=O)CC2C2CC2)=O)CCc2nn[nH]c2C1 c1(CC(=O)C2CC2)ccc(=NC2C3CCC(O3)C2c2ccccc2)[nH]n1 C1(C(N2C(CN(C(c3nnc(C)o3)C)C)CCCC2)=O)CC(C(C)C)=NO1 C1(C)(C(=O)NC(CC(=O)NCC(NOC)=O)CC2CC2)CC2CCC1C2 CCC(C)(CC)C(=O)NCCC1(O)CCN(C(c2cccc(NC(N)=O)c2)=O)C1 C12(NC(C3N(CCC)CCCC3)=O)CCC(NC(c3cscc3OC)=O)(CC1)C2 c1(N2CC(C(C)NC(C(C)OCCOCC)=O)C2)ncnc2cc(Br)sc12 N1(C(c2c(SC)nn(C)c2)=O)CCOCC1(C)c1cn(C2CCCC2)nn1 C1(NC(CC(C)C2CCCO2)=O)CC2(CCN(C(C34CC5CC3C4C5)=O)C2)C1 c1(N2CCC(F)(C(=O)Nc3c(OC)ccc(Cl)c3)C2)ncnc2ccc(F)cc12 C1(NC(C(CCO)OC)=O)CN(C(c2cccc(F)c2C)=O)CC1(C)C CN1CCN(CC(=O)NC2CCCC2NC(=O)C=CSCc2ccco2)CC1=O C12(C)CN(CC1(F)F)C2=O.C1(C)(NC)CC(NC(=O)OC(C)(C)C)C1 C1(CCC)(NC(=O)C=Cc2cn[nH]c2)CCCN(C(=O)Cc2csc(C)c2)C1 C1(C)(CC)C=C(C(=O)N2CCN(C(c3ccc(C4CC4)cn3)=O)C(C(C)C)C2)C1 CC1C(C(=O)N2CC(N(C)C)C(CNC(=O)CN3CCCCC3C)C2)=NOC1C c1(NC2CCCN(C(=O)OCC=C)C2)nccc(=NC(C)CC2CC2)[nH]1 C(=O)(C1=CC2(CCN(C(=O)C=Cc3cc[nH]c3)C2)C1)NC(C)CCC(C)(C)C C1(NCc2cccc(OC)c2Br)CCCCCCC1(F)F CC1CC(C(N2CC(C(c3ccccc3)C3CC3)C2)=O)C12CCC2 c1(C(N2CC(C)(NC(CC3C(CC)C3)=O)C2)=O)cc2c(OC)ccc(C)c2[nH]1 c1(C(=O)NC2C(C)(C)N(C(=O)CCc3nccs3)CC2)cccc2oc(O)nc12 N1(C(C(C)CO)=O)C2CCC1CC(NC(=O)Cc1nc(CN(C)C)nn1C)C2 c1(C(=O)NC2C(CC)CN(C(=O)C(C)=C3CC3)CC2)cn2cccc(Cl)c2n1 CC1CC(NC(C2(C)CCC(F)(F)C2)=O)CCN1C(=O)CCN1CCCC1 CC(=O)CCCC(=O)NC1CCC1CNC(=O)C(S(C)(=O)=O)C1CC1 c1(C(=O)NCC2(COC)CN(C(=O)CC3OCCC3C)C2)ccc(SC)cc1C CC(CSc1ccccc1)C(=O)NCCN(C(=O)C=CCl)Cc1ccccc1 C(=O)(C(CO)C(C)(C)C)NCC(CNC(c1c(C)cco1)=O)CO C(=O)(C(C)C(=O)N1CCN(CC2CN(C(=O)COc3cccnc3)C2)CC1)OC C1(C)(CC)CC(NC(=O)CSCCOC)CN1C(=O)CCc1nncs1 c1(C(=O)NCC2CCCN2C(c2ccsc2)=O)ccc2oc3ccccc3c2c1 c1(C(N2CCC(=CC(=O)NC(C3CCOCC3)C)CC2)=O)n[nH]c2c(Cl)cccc12 N1(C(CCOCCCNC(CC2CC(N(C)C)C2)=O)=O)CCCOC(CCO)C1 N1(c2nnc(C)s2)CCC(NC(c2ccnc(CN(C)C)c2)=O)C(CO)CC1 N1(C(c2c(C)csc2)=O)CC=CCC1C(=O)N(C)CC1COC(=O)N1 c1(C(=O)NC2CCN(C(C(C=CC)O)=O)CC2O)c(C)c(C)c(C)c(C)c1C C1(CN(C)C(c2ccc(OCCN)cc2N)=O)CCn2ccnc2C1 c1(C(N(CC(C)NC(C(C)SC)=O)C)=O)cccc2c(C)ccnc12 Cc1cc(C)c(C(=O)N(CCCCN(C)C(C2(C#N)CC3CC3C2)=O)C)c(S)n1 N1(C(CCCN(C)C)=O)CCN(C2CCC(NC(c3cc(O)nn3C)=O)C2)CC1 C(=O)(CCC1CCc2ccccc21)N1C(CN(C)C(c2cn(C)cn2)=O)CCC1 S(=O)(=O)(c1ccc(NCC(c2ccccc2)F)c(Br)c1)NC(c1cnn(C)c1)C n1(CCCC)cc(CNC(=NCC2CCC2)NCC2CCCS2(=O)=O)c(C)n1 CC(C)CC(C)C(=O)NC1CCCCCC1NC(=O)Cc1ccnn1C c1(CCC(=O)NC(CC(C)NC(c2c(CC)[nH]cc2)=O)C)ccc(Br)nc1 c1(CNC(C(CCC)O)=O)ncc(-c2cn(-c3ccn(C)n3)nn2)cc1C Cc1c(C(=O)NCCC2CCC(NC(c3cnsn3)=O)C2)sc(Cl)c1Cl c1(CNC2CCN(C(C3(O)CC3)=O)C2)c(F)cc(Cl)cc1Br CC1=NS(=O)(=O)N(C)C=C1C(=O)NC1(CF)CCN(C(c2ccncc2C)=O)C1 c1(C(=O)NC2(CNC(C3CC(C)(C)O3)=O)CCOC2)ccc(Cl)cc1Cl N1(C(C2CN(S(N)(=O)=O)C2)=O)C2CCC1CN(C(C1CCN3CCOCC13)=O)C2 C#CC1(NC(C2(NC(=O)CCC=C)CC2C)=O)CC(F)(F)C1 c1(C(=O)NC2CC(C)(CNC(c3ccc(C#C)cc3)=O)C2)cc([N+](=O)[O-])nn1C C1(C2(O)CCOC2)(C(=O)NCCCCC(=O)OC)CCC1 N1(C(C(CC2CC2)OC)=O)CC(C)C(C)(CNC(=O)COCCC(C)C)C1 c1(NCc2ccc(NC(C)=O)cc2)nc(N(CC(F)(F)Br)C)nc2scnc12 C(=O)(C1=CCCOCC1)N1CC(C(=O)Nc2cnc(CC)nc2)C2(C1)CC2 C1(C2(O)CN(C(=O)CC(n3nc(C)cc3C)C)C2)(CNC(CCC(=C)Cl)=O)CC1 n1(CCCC)ncc(C(=O)NCCC2CC(NC(C34CCCC3C4)=O)C2)c1C CC1C(NC(=O)C2=CCOC2)CCN1C(C1CCN(C(=O)N(C)C)CC1)=O C1(NC(Cc2c(C)n[nH]c2)=O)CCN(C(c2cnc(C(C)C)[nH]2)=O)CC12CCC2 c1(OC)cc(F)c(F)cc1-c1csc(C(=O)Nc2cccc(-c3nn[nH]n3)c2)n1 c1(CNC(CCC)(c2nnnn2C(C)C)C2CC2)ccc(F)c(OC)c1 N1(C(C2CCC(CC)C2)=O)CC2(CCN(C(c3cc4n(n3)CCCN4)=O)CC2)C1 N1(C(CCCCC)=O)CCCN(C(=O)CCc2nc3ncccn3n2)CC1C CCC(C(=O)NC1COCCC1C(=O)NC(C)C(C)C(=O)OC)C(C)C C1(CC(N)=O)(NC(c2cc(CC)c(C)s2)=O)CCN(C(=O)CSC2CC2)CC1 C#CCC(CC(=O)OC)NC(=O)CN(C(c1c[nH]c(=NC)o1)=O)C(C)C C1(C(N(C)CC2CCCN2C(c2coc(N(C)C)n2)=O)=O)CCC(F)(F)C1 Cc1cc(C(=O)NCC=CC(=O)NC2CC(CN(C)C)C2)ns1 Cc1cc(C)c(CNC(=O)CCOCCCNC(=O)C(C)(C)N=[N+]=[N-])cn1 c1(C(N(C(C)CCNC(C2(C)CS(=O)(=O)C2)=O)C)=O)ccc2c(c1)CCO2 c1(NC(CCCc2cccc(C(C)=O)c2)=O)ccc(F)c(Cl)c1.C1(=O)C(C)O1 Cc1cc(=NC(=O)C(=O)N2CCC(C(C)NC(C3(O)CC(F)(F)C3)=O)CC2)[nH]o1 c1(CC(=O)NC(CCN(C(c2ccc(CC)cc2)=O)C)C)csc2nc(C)cn12 C(=O)(C1=CCCC(C)(C)C1)NCC(=C)CCNC(c1ccc(CS(C)(=O)=O)o1)=O c1(C(=O)NC2C(CNC(=O)CCOC3CCC3)CC2)ccn(-c2ccccc2)n1 c1(CC#N)cccc(C(=O)N(C2CCN(C(C3(CCCF)CC3)=O)CC2)CC#N)c1 N1(c2nccc(C(=O)OC)n2)CC2(C1)C(NC(C1CCOCC1)=O)CCS2(=O)=O C1(C(C(=O)NCC2(NC(c3cnc(C(=O)OC)s3)=O)CCC2)C)CCC(=O)N1C C1(NC(C(CC)N(C)C)=O)CCC(O)CN(C(c2cc(Cl)no2)=O)C1 c1(C(N(CCNC(C2OCCN(CC)C2)=O)C2CC2)=O)cc2sccc2s1 C1(NC(CCc2c(C)cccc2)=O)C(C)(C)C(NC(c2ccon2)=O)C1(C)C n1(CC(=O)NCC(C)NC(c2cccc(S(C)=O)c2)=O)ncc2cccnc12 c1(CC)ccsc1C(N1CCCC1CNC(c1cc(Cn2cccn2)on1)=O)=O c1(CC(=O)NC(CC2CC=CCC2)C(=O)O)cc(F)c(Br)cc1F N1(CC)CCCCC1C(=O)NCC(C1CCC1)NC(=O)CCC1CCCC1 N1(C(=O)OC(C)(C)C)CC2CCCC1C2c1ccc(NC(=O)C2CC2)cc1 C=CCC(CC(F)F)NC(C1CC(C)CCN1C(=O)C=Cc1cncs1)=O N1(CC)CCC(NC(C2C=CCCN2C(=O)CC(=O)OC(C)(C)C)=O)C(C)C1 C1(NC(c2c(OC)nn(C)c2)=O)CC1C1CCCN(C(=O)C=Cc2cc[nH]n2)C1 c1(C(N(C2CN(C(C3(C)COCCO3)=O)CC2O)C)=O)ccn2c1CSCC2 c1(C(=O)NCCNC(C(C)c2cccs2)=O)cc(-c2ccccc2)nn1C C1(CNC(CC=C=C)=O)CCCCN1C(C1CCCN(C(N2CCCC2)=O)C1)=O C1(C(N(C2C(C)COCC2)C)=O)CCCCN(C(=O)CC2CC=CC2)C1 c1(C(=O)NCC2N(C(c3cc(C)c(C)nc3)=O)CCC2C)cccc2c1CC(=O)N2 N1(C(c2cc(C)sc2C)=O)CC2CCCN(C(C3CC4CC(O)C(C3)C4)=O)C2C1 c1(SCC)ccc(C(=O)NC23CC(NC(c4sncc4C)=O)(C2)C3)cn1 C1(C(N(C(C#C)C)C)=O)CC(O)CN1C(=O)C(CC1CC1)OC N1(C(=O)CO)CCCCC1n1cc(CCC(C)(C)CO)nn1.C(C)(CN)(OCC)OC c1(NC(C2CCCN2Cc2cnc(Cl)c(Cl)c2)=O)ncc2cc(F)c(F)cc2n1 n1(C(C)C)ccc(C(=O)N(CCCN(C(=O)C(C)(O)C2CCC2)C)C)n1 OC1CCCC(NC(c2ccc(Cl)cc2Cl)c2ccccc2)CC1 C(=O)(C1=CCC(C)CC1)NCCC(C(C)C)NC(c1cc(C(C)(C)C)nn1C)=O C12(CNC(c3cc(CC)ncc3)=O)CCC(CC1)N2C(c1cnc(Cl)[nH]1)=O C1(C(=O)NC2CC3CC3C2)CCN(C(=O)CCOCCCOC2CC2)CC1 N1(C(c2cc(COC)cn2C)=O)CC(CNC(=O)C(F)OC)C2(CCOCC2)C1 C#Cc1cnn(C)c1C(=O)NC1CCN(C(=O)CCc2ccccc2O)CC1O C(C)(CCC(=O)NCC(C)(C)OCC(=O)NCCc1cc(O)ncn1)OCC N1(C(c2ccn(C)c2)=O)CCOC(C2CN(C(=O)Nc3cccc(CO)c3)C2)C1 c1(NC(C=C2CCN(C(c3cc(C)nn3C)=O)CC2)=O)cc(Br)cc(Cl)n1 N1(C(C(c2n(C)ncc2)O)=O)CCC2(CCCN2C(=O)C=C2CCC2)C1 C1(CC(=O)NCC2CN(C(C(C)Oc3ccccn3)=O)CC2O)CC2CCC1CC2 C1(C(=O)NC(C#N)C(N)=O)CCCC12CCN(C(c1cccc(Cl)c1Br)=O)C2 c1(CC)ccsc1C(=O)N(C1CC(NC(c2cnc(CC(C)C)s2)=O)C1)C C(=O)(CC(C)C(C)C)N1CC(CNC(CCSCC)=O)OCC1 c1(C(=O)OC)nc(Cl)ccc1NC(C1(C)CN(Cc2ccc(Br)s2)C1)=O c1(C(=O)NC2CC3CN(C(CCC(C)=O)=O)CC32)cc([N+](=O)[O-])cc(C)n1 C12(NC(C(=Cc3cn[nH]c3)C)=O)CCN(C(=O)CC3=CCCC3)CC1C2 c1(C(N2CC(NC(C3C4CCC3(c3ccccn3)C4)=O)C2)=O)c[nH]c(=O)cn1 c1(C(N(C(C)CNC(=O)CN(S(C)(=O)=O)C)CC)=O)cc2c[nH]nc2cc1C C1(C)(NC(C(CC=CC)NC(c2c(CC)n(C)nn2)=O)=O)CCC(C)(C)C1 N1(C(c2ccc(C#C)o2)=O)CCCC2CN(C(C3(F)CCOC3)=O)CC12 c1(-c2cn(CN(C(C)C(=O)O)CCCC)nn2)ccc2cccnc2c1 CCC(C(=O)NCC1COCC1NC(=O)OC(C)(C)C)NC(C1CCCO1)=O Cc1cc(C(N2CCC(C)C2CNC(=O)CCc2cn(C)nc2C)=O)[nH]c1C N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CC(CNC(C23CCC2C3)=O)C(O)C1 C1(C(=O)NCC(CNC(=O)CN2CCC(C)(C)C2)OC)CCOCC12CCC2 c1(C(=O)NC2C(OC)CN(C(c3cn(CC=C)nc3)=O)C2)ncnc2ccsc12 c1(C(=O)Nc2c(C)cc(OC)c(OC)c2)ccc(F)cc1[N+](=O)[O-] N1(C(CN(C(COC)=O)C)=O)CC2CC2(CNC(=O)CC(C)(C)OCO)C1 N1(C(C(C)CSC(F)(F)F)=O)CC(NC(C2(F)CCOC2C)=O)C(C)C1 C1(NC(C2C(CC)C2)=O)CCN(C(C2SCCCS2)=O)C(C)C1 C=Cc1cncc(C(N2CCN(C(c3ccn(CCO)c3C)=O)CC2)=O)c1 N1(C(C(N2CC(C(C)C)C2NC(C2CCCCC2)=O)=O)=O)CC(CO)C(C)C1 c1(SC)cc(C(=O)NCC2(NC(C3CC3c3cccs3)=O)CC2)c(C)o1 CCC(C)C(O)C(=O)N1CCCCC1CCNC(c1n[nH]cc1F)=O C(=O)(C(C)CNC(=O)C(CO)NC(=O)Cc1nc(=N)[nH][nH]1)OCC C1(CN(C)C(C2C3(CC3)C23CC3)=O)CCN(C(c2cn(C3CCC3)nn2)=O)CC1 Cc1cc(=O)c(NC(C2COCCC2NC(=O)C2=CC3C=CC2C3)=O)c(C)[nH]1 N1(C(Cc2nc(C)[nH]n2)=O)CCC2CC2(C(=O)N(CC2CCC2)CC2CC2)CC1 CCC(C)(CNC(C1(CC)CCN(C(c2ncccn2)=O)C1)=O)CC S(=O)(=O)(c1ccc(S(=O)(=O)NC2CCC(N)CC2)cc1)NC(C(C)C)C#N C=CCC(C)(C)CCNC(C1CC(C)(NC(C2CC(C3CC3)=NO2)=O)C1)=O c1(C(=O)NCC2N(C(C(C)(O)C3CCC3)=O)CC2)ccc(Br)nc1 c1(CNC(C=CCOC)=O)ccc(C(N2CCC(CN=[N+]=[N-])C2)=O)cc1 N1(C(C(C2(O)CN(C(c3cc(C(C)=O)sc3)=O)C2)F)=O)CC2CC=CC1C2 C1(NC(c2cc(C(F)F)on2)=O)CCCN(C2CC2)C1 C1(CCC(=O)N(C)CC2COCCO2)CCN(C(=O)CC#N)C1 O=C1CC(C(=O)NCCSCc2cn(-c3ccncc3)nn2)NC(=O)N1 c1(OC)ccc(Br)c(F)c1CNc1cc(F)cnc1C Cc1cccn2c(C(=O)N(C(c3ccccc3)CNC(=O)C(C)(F)F)C)cnc12 C1(NC(C2CN(CCC)C2)=O)CCC(=O)N(C2CC2)C1c1ccnn1C CC1CCCN(C(=O)C=Cc2cscn2)C1CCNC(c1occc1Cl)=O C1(O)(C(C)NC(CNC(C)=O)=O)CCN(C(C2(c3ccno3)CCOCC2)=O)C1 C1(N(C(CN(C)C(N)=O)=O)C)CCC(NC(c2ccsc2C(F)(F)F)=O)CC1 N1(C(c2[nH]cc(C)c2)=O)CCN(C(c2cc(C(C)C)n(C)n2)=O)C2CC12 C#Cc1ccc(C(=O)NCCC(C)N(C(=O)CC23COC(C)(C2)C3)C)c(F)c1 Cn1ccc(CCC(=O)NCC2CC2CNC(=O)CC2CSCCS2)c1 c1(CC)ccc(C(=O)NCC(C)N(C)C(c2cccc(C)c2C)=O)c(OC)c1 Cc1cc(C)c(C)c(C(=O)NC2CCCC(N(C(=O)Cn3nccn3)C)C2)c1C c1(OC)ccc(NC(=O)CC(CSC)c2ccc(Cl)cc2)cn1 C1(CCNC(Cc2ccc(C(C)=O)s2)=O)CCCCN1C(C1CCC(=O)O1)=O c1(OC)ccc2[nH]cc(C#N)c(=NCC3C(C)CCCN3C(=O)C=C(C)Cl)c2c1 C1(OCC)CCCC(C(N2CCC2CNC(=O)COc2ccccn2)=O)C1 C(=O)(C(N=[N+]=[N-])C(C)C)NC(C(C)C)CC(=O)NC(C)(CO)C(C)C C1(NC(c2nnn(C)n2)(c2nnnn2-c2ccccc2)CCSC)CCCC=C1Br C1(NC(COCCOCC#C)=O)CCN(C(=O)CSc2c(C)noc2C)CC1C C1(C(=O)NC2CC(C)N(C(c3cccc(C(F)F)n3)=O)C2)CC2(C1)CC(F)C2 C=C1CN2C(=O)CCC2(C(=O)NCC(O)CCNC(C2CC(=O)CC(=O)N2)=O)C1 N1(Cc2nccc(C)c2)CC2(CCC(Nc3ncc(C)c(C)n3)CC2)C1 c1(C(=O)NC2CC2NCCn2cnc([N+](=O)[O-])c2)cc2cc[nH]c(=O)c2s1 N1(c2nnc(-c3ccc(C)c(F)c3)n2Cc2cnn(C)c2)CCn2cncc2C1 C=CCC(CC(F)F)C(=O)N1CCC(NC(=O)Cc2cc[nH]n2)CC1C C1(C(N(CC(O)CO)C(C)C)=O)CN(C(=O)CN2CCCC2)CCC1(F)F c1(C(=O)NC2CN(C(c3c4nnc(C)n4ccc3)=O)C2)c[nH]c2ncnc(O)c12 C1(NC(CCC2(NC(c3c(C)snn3)=O)CCCC2)=O)CCN(C)C1C C1(CNC(C(C)n2cnnn2)=O)CCC(C(=O)NOCC2CCOCC2)C1 CC1(C)C(C(N2CC(CC(=O)NC3CCN(C4CCC4)C3)(OC)C2)=O)CC1(F)F C(C(C)C(C)C(=O)NCCN(C(=O)CCc1ncccc1C)CCOC)OC c1(CC(=O)NCC2(CCNC(c3cc(F)n[nH]3)=O)CC2)ccn(CC(F)(F)F)n1 c1(CC(N2C(C(C)NC(CCC(C)SC)=O)CCC2)=O)cc2ccccc2s1 c1(NC(c2c(OC)cccc2OC(F)(F)F)=O)cc(Cl)nc(C#N)n1 c1(N2C3C(CNC(C4C(C)CC5CC5C4)=O)C(C3)C2)ncn(C)c(=O)c1Br CCCC(C)(C)C(=O)NCC1CN(C(=O)CCNC(c2ccccc2)=O)CC1O C1(NC(C2(C(=O)NC)CC2)=O)CC2CN(C(c3ccc(C)cc3F)=O)CC2C1 N(C(=NCC(C)(C)C(C)(C)O)NC1CC1)Cc1c(OC)ccnc1O CCC(C)C(C(=O)NC1COCC1N=[N+]=[N-])NC(c1cccn1CC)=O C1(CC#C)(C(=O)N(CC=C)CCO)CCN(C(c2coc(SC)c2)=O)C1 CC1COCC(C(=O)NCc2cn(-c3cccc(CCCOCCO)c3)nn2)O1 Cc1nn(C)c(N)c1C(=O)NC1(C)CCC(NC(=O)CNC(N)=O)CC1 N1(C(c2cnc(C)o2)=O)CCOC(C)(CNC(C2CC23CC(C)(C)C3)=O)C1 c1(OC)ccc2cccnc2c1C(=O)NCCC(C)NC(=O)CCN1CCC(F)C1 N1(C(C(CC)CC)=O)CCCC2(C1)CN(C(=O)CC1CCC1C(=O)OC)C2 c1(C(=O)NC(CN(C(=O)C(C)(C)C2CC2)CC)C)ccc(C(C)=O)c(F)c1 c1(C(N2C(CNC(C3(C)CC(C#N)C3)=O)CCC2)=O)ccc2nc(O)[nH]c2c1 c1(C(N(CC(C)NC(c2ncc(OC)nc2)=O)C)=O)c(N)ccc(C)c1F c1(CC)ncc(C(=O)NC2CCC(NC(=O)CCNC(=O)OC)C2)s1 C1(C(=O)Nc2c(C(=O)OCC)cno2)CC2CC2N1C(=O)Cc1cccnc1Br N1(C(c2nnsc2C2CC2)=O)CCN(C(C2(F)CCC2)=O)C2CC12 C(=O)(C1CCCc2cncn21)NC1C(SC)CN(C(=O)C2=CCCCC2)C1 N1(C(CCCOCCOCC)=O)CC2CC1C2NC(C1CCC(F)CC1)=O c1(C(=O)OC)cc(NS(=O)(=O)CCC2CCS(=O)(=O)C2)c(O)cc1F C(CCCC(=O)N(C1CCN(C(c2ncn(C(C)C)n2)=O)CC1)C)OC c1(OC)ccc(Cc2cn(C(C3CCOC3(C)C)C)nn2)cc1C C(CCC(=O)NC(C(=O)NCCCO)c1ccco1)OCCOC C1(O)(CCNC(=O)C(O)C2CCC2)CCN(C(=O)C=CC(F)F)C1 C(=O)(C(F)(F)CN1CCCC1)NC1(C)CN(CC(F)(F)F)C1 c1(CCC=C)ccc(C(=O)NC2C3CC(NC(=O)C=CC4CC4)CC23)cc1 N1(C(CCc2c(C)nccn2)=O)CCN(C(c2cc(C(N)=O)[nH]n2)=O)C2(CC2)C1 CN1CC(C)(C)CC1C(=O)Nc1cccc(NC(c2cnc(C3CC3)s2)=O)c1 Cc1nn(C)c(I)c1Cn1nnnc1NC1(C2CCCC2)CC1 C1(C(=O)NC(C2CCN(C(c3cnns3)=O)C2)C)(N(C)C)CCCC1 n1(CC)cnc2c(NCc3cnco3)[nH]c(=NC3CCOC(C4CC4)C3)nc12 C1(NC(CCC=CC(C)C)=O)CN(C(=O)CC2CCC(F)(F)C2)CCC1CO c1(OCC=C)ccc(C=CC(=O)NCCC(=O)NC)cc1OCCCC C12(CC)CN(C(c3ccnn3C(C)C)=O)C(CNC(C3(C)CCOCC3)=O)(C1)C2 C1(C(=O)NC(C2(CSC)CCC2)=O)CN(C(=O)C(C)(C)OC(=O)C2CC2)CCO1 Cc1nnc(CCC(=O)N(C(C)CCNC(c2cncc(Br)c2)=O)C)n1C C1(C)(C(N2CCC(N(C)C(c3ccncc3Br)=O)C2)=O)CC(C2CC2)=NO1 N1(C(C(C)N(C(=O)COc2cc(C)on2)CC)=O)CCCC(C(=O)OC)C1 N1(C(C(C)NC(CC)(C)C)=O)CC2CCC1C(CNC(=O)C(C)O)C2 C(=O)(C(CC(C)C)n1ccnc1)N1C(CN(C(C(C)OCC)=O)CC)CCCC1 c1(C(=O)NCC(CCNC(c2n(CC)ncc2)=O)O)c(Cl)c(C)nn1C N1(C(C(C)N(C(CSCC#C)=O)C2CC2)=O)CCC(C)(O)C1 c1(CC(=O)NC(C)C(C)NC(=O)CCCCC(N)=O)cn2c(n1)CCCC2 C1(C(C2=CCOCC2)NCc2sccc2Cl)CCc2c[nH]nc2C1 N1(C(CN(C)CC)=O)CCCC12CCN(C(C1CCC3CC3C1)=O)C2 C#CCC(C)C(=O)NCCNC1CC(OC)C1(C)C C1(N(C(=O)OC)C)CCCC1=C1CC1C c1(N(CCCN(C(C(c2ccc(Cl)cc2)C)=O)C)C)nccnc1F N1(C(CN(c2cccc(C=O)c2)C)=O)C2CCC1CC(O)(CO)C2 Cc1cc(=NC(=O)C(=O)NC2CCN(C(=O)C(C)(C)c3cccs3)CC2O)[nH]o1 C1(CCCC)CN(C(=O)C(C)CSC)CCN1C(=O)C(c1nc(F)ccc1Cl)C CSC1=C(C(=O)N2CC3(C2)CN(C(c2cccc(C)c2)=O)C3)CCCC1 C(C(CO)C(F)(F)F)NC(=O)CN(C(=O)C1=CCOCC1)CC1CC1 C1(C)(NC(C(C)(C2CCC2)NC(CC=C)=O)=O)CC(O)(CO)C1 N1(C(C2C(C(C)C)CCO2)=O)CCCC(NC(=O)CC2(C)CCCCC2)C1C CC1CC(NC(c2ccc(C3CC3)nc2O)=O)CCN1C(C1CCSCC1)=O C1(CNC(c2ccc(COC)s2)=O)COCCN1C(c1cc(CF)on1)=O c1(C(=O)NC(c2ccccc2)CNC(C2C(=C)C2)=O)ccc2cc(C)oc2c1 c1(C(=O)NC2CCCN(C(C34COC(CO)(C3)C4)=O)CC2)cn2cccnc2n1 Cc1nn(CC(F)F)c(C)c1C(=O)NCC(C)(C)NC(=O)C(C)C1CCCO1 Cc1ccc(CC(=O)NC(C(=O)NCC(C)CC2CC2)c2ccoc2)s1 CC(CC(=O)N(CCC(C)(C)NC(c1cnc(CC2CC2)s1)=O)C)CC(C)(C)C C#CC1(C(N2CCS(=O)(=O)CC2)=O)CCN(C(C2CCCCCN2C)=O)C1 C1(CC(=O)N)CCC(C)(O)CC1.c1(C(N2C3(CC3)C2)=O)coc(C)c1.CC c1(OC)ccc(C(=O)NC(C2CN(C(c3nc(C)n(C)n3)=O)C2)C)cc1F C1(C(=O)NCCc2ncn(CC)c2)N(C(=O)C(C)SC)CC12CCCC2 Cc1cc(C)c(C(=O)NC(C)CCCNC(c2cccc(C(F)F)c2)=O)o1 C#Cc1cn(C)nc1C(=O)NC1CCN(C(=O)CCN(CC)CC)C(C)C1 CCCCCCCCNCC.c12ccc(nc1)N1CCN(CC1)CCOC2=O.O CN1CCN(c2ccc(CNC(N3CC4(CC4NC4(C)CC4)C3)=O)cc2)CC1 c1(N2CC=C(CNC(c3ccc4ocnc4c3)=O)CC2)nc2cccc(Br)c2o1 Cc1nc(NC(C2CCN(C(c3ncc(Br)cc3Cl)=O)C2)=O)ccc1Br N1(C(C2(C)CCCN(C(=O)Cc3ccc(F)cc3F)C2)=O)CC2CC(O)CC1C2 c1(C(C)NC(=O)CSCCNC(=O)C(F)C2CCOC2)ccn(C)n1 N1(C(CCC=C)=O)CC2CCC(C1CO)N2C(=O)Cc1c(C)cc(OC)cc1C C1(C(N(CCCN(C(=O)CC2CCC2)C)C)=O)CCCC12CC2 c1(C(=O)NCC2C=CC(NC(CCOCC)=O)C2)ccc2c(c1)NC(=O)NC2 c1(C(=O)NC(c2cccc(F)c2F)CO)nc(Br)n2c1CNCC2 c1(NCC23CCC(NC(CC(C)C4CC4)=O)(C2)CO3)cnc2ccccc2n1 Cn1c(O)nc2cccc(C(=O)NCC3CCCN3C(=O)CC3CC4(CC4)C3)c12 C1(C(N(CCCOCCNC(=O)Cc2ccns2)C)=O)COCCO1 C1(C(=O)NCC2(O)CC(NC(=O)CSc3ccncc3)C2)CCCC(F)(F)C1 c1(CC)cc(C(=O)NCc2cc(C(=O)NC3CSCC3C)n[nH]2)ns1 c1(C(C(=O)N(CC#CC)CC#C)N)ccncc1C C12(C(N3CCN(C(c4n(C)c(C#N)cc4)=O)CC3)=O)CC3CC(C(=O)N1)C2C3 C(=O)(CCC(=O)N(C)C)N1CC(C(N)=O)(CNC(c2n(CCC)ccc2)=O)C1 c1(C(=O)NC2(C)CC(NC(COCCC)=O)C2)nccn2nccc12 C12(C(=O)NCc3nc(C4CC4)n[nH]3)CCCC1CN(C(=O)C(O)C1CC1)C2 C1(NC(c2cnc3n2CCC3)=O)CN(C(C2CC3(CCCC3)C2)=O)C2(CCC2)C1 C1(NC(CC2(OCC)CCC2)=O)CC12CCN(C(c1csc(CC)c1)=O)C2 C1(C(=O)NCC2(C(N3CC(OCC(C)C)C3)=O)CCC2)CCCC(C)(C)C1 c1(C(N2C(C(C)(C)CNC(c3cnn[nH]3)=O)CCC2)=O)ccc(N)cc1Br N1(C(C2N(C(c3cccnn3)=O)CCN(C)C2)=O)CCC2(CNC(=O)C2)C1 c1(C(=O)NC2CC(C(=O)Nc3c(C)nsc3)C2)c(C)ccn1C CC(C(=O)NCC(=O)NC1CCC1)NC(=O)C(N)=O N1(C(C2ON=C(C)C2)=O)CC(C)N(C(C2CCCC2)=O)CC1C c1(C(=O)NCCN(C2CCCC2)C(C2CCCN(C)C2)=O)cc2ccsc2n1C C(C(C)(O)C(=O)NCCCC1(NC(C2(C)CC2(F)F)=O)CC1)OC C(CC(CC)C(=O)N(CC(C)CNC(c1cccc(C)n1)=O)C)=CC C=CC(C)(O)C(=O)NC(c1cccnc1)C(=O)NC1CCC(C(C)O)CC1 Cc1cc(Cl)nc(Cl)c1C(=O)NCc1ccc(-c2cccc3ccoc23)cn1 C(=O)(C(C)C(C)C(C)(C)C)NCCC1(OC)CN(C(C2(C(=O)NC)CCC2)=O)C1 C(=O)(C1=Cc2cccc(Br)c2OC1)N1CC(N(C)C(C23CCC(CC2)O3)=O)C1 c1(OC)ccccc1CN(C(=O)CCc1nc(C)no1)C.c12cccc(c1)NC2 CC1OC2(CNC(C34CCCN3CCC4)=O)CC1(NC(=O)C(Cl)=CCl)C2 C1(C(=O)NC2CN(C(COCCC=C)=O)CC(C)(C)C2)Cc2ccc(C)cc2S1 c1(NC2CC(CNC(Cc3cc(COC)on3)=O)C2)cc(=O)n2oc(C)cc2n1 c1(C(=O)NC(c2cccc(N3CCCC3=O)c2)C)cc(O)nc2c(Br)cccc12 N1(C(c2c(C(C)(C)C)noc2)=O)CCC(n2cc(-c3cccc(F)c3)nn2)CC1 C1(NC(C2CC(C)CN2C(c2c(F)cncc2F)=O)=O)CNC(=O)C1(C)C C(c1ccc(SC)cc1)=CC(N1CC(COC)(CNC(C2CC2(F)Cl)=O)C1)=O c1(C(=O)NC(Cn2cc(-c3cccc(OC)c3F)nn2)C)ccc([N+](=O)[O-])cc1 n1(CC)cc(C(=O)NC2CC(CNC(C3CCN(C)C3=O)=O)C2)c2ccccc12 c1(CC)cc(Cl)ncc1NCc1ccc(F)cc1OC.c12ncccc1NC2=O Cc1cc(C(=O)NCC2CC(C(=O)NCCc3cncs3)=NO2)cc(F)c1 CCC(C)(C(=O)NCCC1(NC(=O)CCOCc2ccccc2)CCC1)C(N)=O C1(O)(CNC(N(CC(C)C#N)CC)=O)CCOC(C)(C)C1.O N1(C(CCCC(=C)C)=O)CCCCC(C2CN(C(C3CCOC3CC)=O)C2)C1 C1(C(=O)NC(C2(C(=O)NC3CCC(F)(F)C3)CC2)C)COCC1(C)C C(=O)(C(O)CCS(C)=O)N(CCCNC(C12CCC(C(=O)OC)(CC1)C2)=O)C C=CCC(C(=O)OC)NC(=O)C(Cc1ccoc1)NC(c1cc(COC)[nH]n1)=O C1(CNC(C2CCC(COC)C2)=O)CC(C)(C)CN1C(c1cc(F)ccc1N)=O C1(NC(NC(C=C)C)=NCC(C)F)CCc2cc(OC)ccc2C1 Cc1ncc(C(=O)NCC2CCC2NC(=O)C(N2CCC(C)C2)=O)o1 N1(C(C(CC)N(C)C)=O)CCN(C(=O)C(C)=Cn2ccnn2)CC(C)(C)C1 C1(NC(C2(F)CN(C(CC3CN(C(C)=O)C3)=O)C2)=O)CCCN(CCO)C1 c1(C(=O)NCC(c2cccnc2)NC(CSCC=C)=O)ccc2c(c1)CC2 N1(C(C2(C)CCCN2C(=O)CC2CC3C=CC2C3)=O)CCC2CCC(C1)S2 C1(F)(CNC(c2cc(OC)ns2)=O)CCN(C(=O)C(C)=C(C)C)C1 c1(C(=O)NCC2C(CNC(c3c(C(C)C)onc3)=O)C2)noc2c1COCC2 C(C(O)C(=O)NCC(C1CC1)NC(=O)CCc1csc(Br)c1)=CCCC CCC(CC)CC(=O)N(C1CCC(NC(C2CSCCS2)=O)CC1)C N#CC1CCCN(C(C2CCN(C(c3ccc(C(F)(F)F)c(Cl)c3)=O)CC2)=O)C1 Cc1ccc(F)c(NC(=S)NNC(=O)C2(CC(C)C)CCNC2=O)c1 C1(C(N2C3CN(C(C(C=CC)O)=O)CC2C3)=O)CN=C2N=CNN2C1 c1(-n2cc(C3N(C(C)=O)CCCC3)nn2)c(C)cccc1Br.C=CC1C(=O)O1 Cn1cncc1C(N1CCC(CNC(C2CCN(c3ccccc3)C2)=O)C1)=O c1(CC)cc(CC)[nH]c(=NC2CN(C(=O)CC(F)F)CC23CCOCC3)n1 N1(C(C(c2n(C)ncc2)O)=O)CCN(C(=O)CSc2nc[nH]n2)C(C2CCC2)C1 c1(C(=O)NC2CCCCN(C(CCC(=O)OC)=O)CC2)cnc2c(n1)CCCC2 CN1CC2CCCN(C(C3CCOCC3NC(C3CS(=O)(=O)C3)=O)=O)C2C1 C(=O)(CC(C)(C)C)NCC1C(CNC(C(C)NC(N)=O)=O)C1 Cc1ccc(C(CC(=O)OCC(=O)NC(=O)OC(C)(C)C)NC(N)=O)cc1 c1(C(=O)NCC(C2CCCC2)NC(CSCCC(C)C)=O)cc(N)ccc1F CC1(C)CCCC(C(N2CC(NC(C3CCN(CCO)C(=O)C3)=O)C(O)C2)=O)C1 C(=O)(C1=Cc2ccccc2C1O)NCCCNC(C(CC(C)C)C(C)C)=O N1(C(C(Cn2cncn2)NC(C=C(C)C)=O)=O)CCCCC1CF N1(CCCSC)CCCCC12CCN(C)C2 C1(C(N(CC(C)NC(c2ccn(C3CC3)n2)=O)CC)=O)CCC(CN(C)C)CC1 N1(C(CN(C)C(N)=O)=O)CCN2CCN(C(=O)CCCc3cnn[nH]3)CC2C1 c1(C(=O)NCC2C=CC(NC(C(c3ccc(C)cc3)C)=O)C2)cnn2ccsc12 C(CN=c1[nH]c2c(C)cccc2o1)N(C(C12CCCN1CCC2)=O)CC c1(CC)sccc1C=CC(c1ccnnc1)=O C(=O)(C1=CC2(CCOC2)C1)N1CCN(C(C(C)(C)c2cccs2)=O)CC1CF N1(C(C(c2ccn(C)n2)C)=O)CCC(NC(C2(C)CCOC2)=O)C1 Cc1ccc(C(=O)NCC2CC3CCCC3N2C(=O)CC(F)(F)Cl)c2c1CCC2 N1(C(C(C2CCCC2)OC)=O)CC(O)(CNC(=O)C(C2CCOCC2)C)C1 C#CC1CCCC(CNC(C2(C#C)CCN(C(=O)CCC(F)(F)F)C2)=O)C1 C1(CC(=O)OCC(C2C(C)C2)=O)CN(C(C2(c3cccc(Br)c3)CC2)=O)CC1(C)C c1(CC)cc(C(=O)NCC(CC)(CC)NC(=O)CCCc2ccccc2)n(C)n1 Cc1c(C(F)(F)F)n[nH]c1C(=O)NCC1CCC(NC(=O)Cn2cc(Cl)cn2)C1 C(=O)(CCCCCCC(C)C)N1CC(O)(C(C)NC(C2C(CC)N(C)CC2)=O)C1 N1(C(Cn2c(C(C)C)ncc2)=O)CC2(CC2)CC1CNC(=O)C(F)C(F)(F)F C(C1CCc2nccn21)NCCC1C(O)CCC1 c1(C(=O)NCC(CNC(c2ccc(F)cc2)=O)O)cnc2[nH]ncc2c1 c1(CC(=O)NCC2CCCCN2C(C2(F)CC2(F)F)=O)ccc(Cl)cc1Cl CCS(=O)CC(=O)N1CC(O)CC1CNC(=O)C=CC(=O)OC(C)(C)C C1(NC(C(C=CC)O)=O)CC2CCC(C1C)N2C(c1cc(O)ccc1[N+](=O)[O-])=O C1(CNC(=O)CC2CC(CF)C2)CC2CCC(C1)N2C(=O)Cc1sccc1Cl N1(C(C(CC2CCC2)NC(C23CCC(OC)C2C3)=O)=O)CCc2nccnc2C1 c1(N2CCC(NS(CCC)(=O)=O)CC2)cc(NC2CCCCC2O)nc(C)n1 c1(C(N(CCNC(C23CC(COC)(OC2)C3)=O)CCOC)=O)cc(F)ccc1Cl CCCC(O)CC(=O)NC(C)CCNC(=O)CCCOc1ccc(Cl)cc1 CC1(C)CC(=O)NC1CNC(=O)C(N1CCC12CCC2)=O N1(C(CC2C(C)(C)C2(C)C)=O)CC2CCCC(C1)N2CCN1C(=O)CNC1=O CC1CC(NC(C2CC3(CCCC3)C2)=O)CN(C(=O)Cn2cnc(C(N)=O)n2)C1 CC(C(=O)NC(CN(C(=O)C=Cc1ccoc1)C)(CO)CO)S(N)(=O)=O Cc1sc(NC(=O)C(=O)NCCc2cccc(O)c2)nc1-c1ccccc1 C(C)(C)(CC(=O)N(CCCCO)C)N(C(C1OCC(C)C1)=O)C C(C)(CNC(=O)C(N)Cc1cc(Br)sc1Br)(C(F)(F)F)OC C1(C(N2CCC(O)(CCNC(CCCC#C)=O)C2)=O)CCCC2(CCOCC2)O1 CC1(C)CCc2c(C(=O)NCC3C=CCN3C(c3ccc(CO)o3)=O)n[nH]c2C1 C1(N(CC#C)C(c2nccn2C(C)C)=O)CCN(C(c2ccncc2Cl)=O)CC1 c1(C(=O)NCc2c(C(=O)NCCOCC(C)C)cco2)ccnc2cc[nH]c12 Cc1nccc(C(=O)NCCN2CCN(C(C3CC3Br)=O)CC2)c1C c1(C(N2CC(C(C)NC(=O)CCC(=O)N(C)C)C2)=O)ccc2nccnc2c1 Cc1cc(C(=O)NC(CNC(=O)C(C(C)O)N(C)C)C(C)C)[nH]c1C c1(C(=O)NCC2CCCC(NC(c3ccon3)=O)C2)ccc2sccc2c1 Cn1nc2ccccc2c1C(N1CCC(C)(NC(=O)C2=C(Cl)CCOC2)CC1)=O CC1(C(=O)NCCNC(N)=O)CCCN1C(=O)Cn1cnnc1O Cc1cnc(COC(C)(C)CNC(=O)CSCc2cccnc2)nc1 C1(NC(C2N(C)CCOC2)=O)CC=C(C(=O)N2CC(C)(O)CO2)C1 C12(NC(C3COCCOC3)=O)CC3CC(C1)CC(NC(C1CCCOC1)=O)(C3)C2 N1(C(c2c(C)csc2)=O)CCOC2CN(C(c3ccc(N)c(Cl)n3)=O)CC12 N1(C(c2c(NC)cccc2)=O)CCC2(CC1)CC(NC(=O)CCCCC(N)=O)C2 N1(C(CNC(C=CC(C)C)=O)C(F)F)CCN(C(=O)C(C)O)CC1 N1(C(C(COC)OC)=O)CC2(NC(=O)CC(Cl)Cl)CCCC2(F)C1 CCCCC(C(=O)N1CC(NC(c2ccc(C)c(Cl)c2Cl)=O)CC(F)C1)C(C)C N1(C(CC(C)SC)=O)CCN(C)C(C(=O)Nc2cnc(C)c(Cl)c2)C1 CC(C)CCC(F)C(=O)NCC1CCC(C(=O)NC(CO)C(C)(C)CO)C1 N1(C(c2n(C)cnc2)=O)CCCC2(CNC(=O)Cc3ccc(Cl)cc3)CC12 C(=O)(CCCCCS(N)(=O)=O)N1CC(CNC(Cc2c(C)noc2)=O)N(C)CC1 c1(OC)cccc(C(=O)NC(C)(C)C(C)NC(=O)Cn2cnc(C(N)=O)n2)c1 C1(OC)CCC(C)(C(=O)NC2CC3C2CCN3C(c2ccc(O)nc2)=O)CC1 C1(C(=O)NCCc2ncn(CC)c2)(CO)CCN(C(=O)C(CO)N(C)C)C1 C(=O)(C(C)(C)C1(O)CCC1)N(CCCNC(CCOCC=C)=O)C1CC1 CC(C)C(C)(O)C(=O)NC1CC1NC(c1csc(C2CC2)n1)=O C(=O)(C(C)C(F)(F)F)N1CCC(N(C(C(C=C=C)C)=O)CCO)CC1 c1(C(=O)NCCCC(C)NC(CCOCCOC)=O)ccnc(Br)c1N C(=O)(CC(O)C(C)(C)C)N(C(CNC(c1c(CC)nc(-n2cccc2)s1)=O)C)C CC1CC2(CCN(C(=O)CCOC3CC3)CC2)CN1C(C1CCN(C)C1=O)=O N1(C(C(CCC)NC(C2CCCOCC2)=O)=O)CCC12CC(O)C2 C(=O)(CCP(C)(C)=O)N1C(C(=O)OC)CC(n2cc(Cn3ccnc3C)nn2)C1 Cc1c(Cl)ccnc1C(=O)NC1CCC(C)(CNC(c2[nH]cnc2C#N)=O)C1 n1(CC)ncc2cc(-c3nc(C4CC4(C)C)nn3C3CCSC3)c(C)nc12 c1(C(C)=O)cc(C(=O)N(CC(C)N(C)C(c2csc(C(F)(F)F)c2)=O)C)no1 N1(C(C(CC)=CC)=O)CCC(C)(CNC(c2ccn(C)n2)=O)C1 N1(C(c2ccc(Cl)cn2)C(=O)NCCC)CCSC(C)C1C C(CCC)(C(=O)NC1(C2CCC2)CC1)NC(COCC#C)=O C(=O)(C1=COCCC1)N(c1ccncc1)CCCC1(N(C(C)=O)CCC)CC1 CC1(NC(C2CCCCO2)=O)CC(C(N2CC(c3ccon3)C2)=O)C1 N#CC1CN(Cc2occc2Br)CC1N=c1ncnc2[nH][nH]cc1-2 C(=O)(C(C)CC(F)F)NC1C(NC(c2nc(C)n(-c3nc[nH]n3)n2)=O)C1 N1(C(C2CCC(C)C2)=O)CC(C2(NC(=O)CCN3CCCC3=O)CC2)C1 c1(NC(C2C(C(=O)OC)C2)=O)ncccc1OC1CCCCC1 C12(CNC(C3CC(CC)C3)=O)CC(CC)(CN1C(C1CC(=O)N(CC3CC3)C1)=O)C2 Cc1ccc(C(C)CC(=O)N(CCNC(=O)CSC(F)F)CCOCCO)cc1 C(=O)(C(C)C(C)c1ccc(F)cc1)NCCC1(NC(CSCC#C)=O)CCCC1 c1(C(N(CCCN(C(C(C(CC)O)(C)C)=O)C)C)=O)cc2c(cc1F)OCO2 C1(c2cn(CC)nn2)CCCCN1N1CC2CC2C1.c1(C=O)ccc(-n2ccnn2)o1 C(=O)(CC1=CCCC1)NC1C(NC(CC(C)N2CCCC2=O)=O)COC1 C1(CNC(CCC(=C)Cl)=O)CN(C(=O)Cc2csc(C(C)C)n2)CCC1C N1(C(CCC=CC)=O)C(CNC(=O)CC(C)CCCCC)CC2CCCCC12 O=C1CCC(OCC2CCOCC2)C(=O)N1.c12ccc(cc1)OC(=O)N2 C1(NC(C(CSC)C)=O)CN(C(=O)CCCCCN(C)C)Cc2ccnn2C1 C1(C(N(CCCN(C(CCCOC)=O)C)C)=O)CCCN2CCCC12 N1(C(c2cc(OC)ncn2)=O)CCCCC(CCC(=O)N(C(C)CO)C)C1 Cc1cc(C(=O)NC(C2(O)CN(C(c3cccc(CF)c3)=O)C2)C)nc(C)c1 c1(OC)ccccc1C(C)CC(=O)NC(CO)C(C)NC(=O)CN1CCOCC1 c1(C(=O)N(CCNC(c2ccsc2)=O)Cc2ccccc2)ccc(C2CC2)cc1 c1(C(=O)NC2C(NC(c3c(SC)scc3)=O)C2)cc(Cl)c(Cl)cc1C c1(C(=O)NC2CC(CNC(C34CCCN(CC3)C4)=O)C2)cc2ccnc(Cl)c2s1 C(=O)(CC(C)C(C)(C)C)NC1C(C=C)CN(C(=O)COc2ccccc2)C1 CCCCC(C)(F)C(=O)N1CC(CNC(=O)COC(F)F)C(C(F)(F)F)C1 C(=O)(C1=CC2(CCOCC2)C1)N1CCC2CCN(C(C(CCC(C)C)O)=O)CC21 N1(C(CCC#C)=O)CCCC(O)(CNC(=O)COc2ccccc2C(C)(C)C)C1 C1(NC(C(=O)N(C2CC(C)C2)CC(F)F)=O)CCCC12CCC2 c1(C(=O)NCC2CN(C(CCCC=C)=O)CC2O)cc(C)ccc1[N+](=O)[O-] N1(C(CNC(=O)OCC=C)=O)CCN(C(=O)C2=C(Cl)CCC2)C2CCCCC12 N1(CCC)CCCC(CNC(=O)C(=O)NC2CCCCC2OC)C1 O=C1OCCC1NC(c1nnnn1-c1ccccc1)C1CCCCC1 C(=O)(C(C(=O)N1CCC(NC(C2CC(N(C)C)C2)=O)C1)C(C)(C)C)OCC c1(NC(=O)COC(=O)CC(C(F)F)c2cccc(F)c2)ncc(Cl)cc1[N+](=O)[O-] N1(C(CC)=O)CSCC1C(=O)NC1CC1NC(C1(C)CC1)=O C(=O)(CCCCN(C(=O)C(C)c1ccco1)C)N(C(C)COC)CC N1(c2ccc(C(C)=O)cn2)CCN(C(c2c(C)ccnc2Cl)=O)CC(C)(F)C1 C(=O)(C1=COCCC1)N(CCCN(C)C)CCNC(C1(C(C)(F)F)CCOCC1)=O c1(C(N(C(C)C(=O)N(C(C)CC(N)=O)C)CC)=O)nc(O)sc1C N1(C(c2c[nH]c(=NCC)s2)=O)CC(C2CCCN(C(C3(C)C=CCCC3)=O)C2)C1 CN1CCC2(CCN2C(=O)C2=CC(O)C(NC(c3ccc(CO)nc3)=O)C2)C1 CCCCC(O)CC(=O)NC1(C)CCN(C(c2cc(C#N)no2)=O)CC1 C1(C(=O)NCCNC(c2cnnn2-c2ccccc2)=O)C2CCC1(C(F)F)C2 C(c1ccc[nH]1)=CC(=O)NCC1(CNC(C2(COC3CC3)CC2)=O)CCC1 N1(C(CC(=C=C)C)=O)CCN(C(=O)CSc2cc(F)ccc2F)C(C)CC1C C1(C(N2CC(OC(C)C)C2)=O)CCN(C(C2CCCCC2)=O)CC1O C1(CNC(c2cc(C)no2)=O)CCCC2CN(C(=O)CCSC(=N)N)CC12 C=C(C)CC(C)C(=O)NCC1N(C(c2cccc(CN(C)C)c2)=O)CCC1(C)C Cc1cc(C(=O)NCC2(C)CCCN2C(=O)CCC=CBr)c(O)c(C)n1 c1(C(C)(C)C)ncc(C(=O)NCCC2CC(NC(=O)CCNC(=O)CO)C2)[nH]1 c1(C(CNC(=O)NC2CN(C(C(C)OC)=O)C2)O)cccc(OC)c1 C(=O)(C#CC1(C)CCCO1)N(CCC)CCNC(c1cc(C(N)=O)c[nH]1)=O Cc1cccc(CC(=O)NCCc2cn(CCOCCO)nn2)c1 N(C(=NCCOCc1cccc(Br)c1)NC(C)C1CC1)C1C(C=C)C1 N1(C(=O)CC2CC=CCC2)CC2CN(C(=O)C(c3ccccc3F)F)CC(C1)O2 c1(C(=O)NC(C2CCN(C(c3cc(N)ccc3O)=O)C2)C)cncc(Cl)c1Cl c1(C(=O)NC2CN(C(CCCCC=C)=O)CC2(C)C)ccc(F)c(C)c1Cl N#Cc1cn[nH]c1C(N1CCCC(N(C(=O)C=CSc2ccccc2)CCF)C1)=O C1(N(C2CN(N(CCN(C(COC)=O)CC)CC)C2)C)C(C(=O)C2CC2)C1(F)F CC1OC(=O)NC1C(=O)NCC(O)CN(C)C(c1nnn(C(C)(C)C)n1)=O Cc1cc(C(N2CCOCC2CNC(c2cnn3c2CCC3)=O)=O)cc(C)c1N c1(C(N2C(CCNC(CCN(C)CC)=O)CCCC2)=O)ncc(F)cc1N C(=O)(C(CC)C(=O)OC)N1CC(C=C)(CC(=O)NCC2CC(SC)C2)C1 c1(CC)ccc(OCCN2CC(NC(c3csc(C(=O)O)n3)=O)OCC2)cc1 Cc1cc(C(=O)NC2CC3(C2)CN(C(C2CC2(C)C(C)C)=O)C3)ccc1O N1(C(C(CCCCC)C)=O)CCc2ncc(NC(=O)CC3CCC3)cc2C1 C(C(CC)(CC)C(=O)NCCC(C)c1cn[nH]c1)NC(C(CCC)C)=O N1(CC)CC(C(=O)NCC2CCCN(C(C3CNC(=O)N3)=O)C2)CCC1=O N1(C(C(=O)NCCCCCNC(c2nn(CC)c(O)c2)=O)C)CCP(C)(=O)CC1 C(c1ccccc1)=CCC(=O)NC1CCN(C(c2cccc(CO)c2)=O)C1 c1(C(N(C(C)CNC(=O)CCC(F)(F)F)CC)=O)cc(C#N)cc(C)n1 c1(C(=O)NCC(CNC(CC=CC)=O)F)cc(C2CC2)nn1C C1(CCC)CN(C(=O)C#CC(C)(C)C)CCN1C(=O)C(C)P(C)(C)=O c1(CC)cccc(CC)c1CC(=O)NC1CCN(C(=O)CC2CC3(CC3)C2)C1C CC(C)(CO)C(=O)NCc1ccc(C(=O)NC2CCC2O)cc1 N1(C(C2(c3ccc(OC)cc3)CC2)=O)CC2CCC(C1)N2C(c1cncs1)=O Cc1ccc(F)cc1NC(=O)C(C)(C)NC(=O)CCc1ccccn1 N1(C(CC2CCCN(C(CN(C3CC3)CC)=O)C2)=O)CCCC(CO)CC1 C1(CNC(c2ccnc(Cl)c2F)=O)CC2(CCN(C(=O)CSC3CC3)CC2)CO1 C12(CNC(c3cnc(C)s3)=O)CCCCC1N(C(=O)CCC1(O)CCC1)CC2 C(=O)(C1SCCc2sccc21)NCCCOCCN(C(C(CC)(C)CC)=O)C N1(C(C(C)OCC#C)=O)CCCC(C2CC2NC(c2ccccc2OCC)=O)C1 N1(C(C2C(=C)CC2)=O)CC2CCC1CN2C(=O)CCCOc1ccc(Cl)c(C)c1 c1(C(N2CC(NC(C(CC)C)=O)CC(F)(F)C2)=O)c[nH]c2nccc-2c1C C1(NCC(=O)Nc2cc(C)no2)CCN(C(c2cc(C)n(C(F)F)n2)=O)CC1C N1(C(c2cc(CNC(Cc3c(C)n(C)cn3)=O)no2)=O)CC2C3C=CC(O3)C2C1 N1(C(C2OCCC(C)C2)=O)CC(NC(c2csc(C3CC3)n2)=O)CC(F)C1 C(=O)(C#CC1(C(F)(F)F)CC1)NCC(C(C)C)NC(C(C)(C1CC1)NC(C)=O)=O c1(C(=O)NCCc2cnc(NC(c3c(C)nc(Cl)cc3)=O)s2)c(F)cc(Br)cc1Br c1(C(=O)Nc2c(C(N)=O)nccc2)cc([N+](=O)[O-])cnc1O C(C(C)(C)C(=O)NCCCCCCN(C)C(c1nc(C)sc1C)=O)NC(C)=O c1(OC)ccc(C)cc1-n1cc(CC2CCCN2C(=O)NCC(C)(C)C)nn1 S(=O)(=O)(c1[nH]c(=NCc2ccc(C#N)o2)ccc1Br)NCc1c(C(C)C)con1 c1(C(=O)NC2CC(NC(CCCC=C)=O)C2)cc(N2CCCC2=O)ccc1Cl C1(c2nnnn2CC(F)F)(NCCCC(CC)O)CCCSCC1 C(=O)(CC(C)(C)C#N)N1C(Cn2cc(C3(S(=O)(=O)N(C)C)CC3)nn2)CCC1 CC1CC(CNC(=O)C(C2(O)CCCC2)F)CN1C(C1(O)CC1)=O Cc1nc(-c2nn[nH]n2)ccc1CNC(C1(C)COCCO1)=O c1(C(C)C)cc(C(N2CC(O)(CNC(=O)CC3CC4CC4C3)C2)=O)ns1 CC(C)CC(C(=O)Nc1cccc(Cl)c1)ONC(C1(C)CCCN(C)C1)=O Cn1cc(C(N2CCCC(CNC(c3nn[nH]c3Cl)=O)C2)=O)c(-c2ccco2)n1 N1(C(C(C(C)C)SCC)=O)CC2CC1CC2CNC(c1cccc(Cl)c1O)=O CC1CN(C(=O)Cc2cnccc2Cl)CCN1C(=O)C(C)OCCN(C)C c1(OC)ccc(C)c(C(=O)NCCN(C(=O)C(C(C)(C)C)OC)C)c1N Cc1cnc(C(=O)NC(C)C(CO)NC(c2ccnc(C(C)(F)F)c2)=O)c(C)c1 Cc1ccc(C(=O)NC(CNC(=O)Cc2cccnc2C)C(C)C(C)C)nc1C c1(C(=O)NCCN(C(c2ccccc2C)=O)CC)cnncc1C(F)(F)F c1(C(=O)NC(c2ccccc2)C(C)NC(C2CCC(C)O2)=O)ccc2cnoc2c1 CCC(C)C(C(=O)N1CCCC1(C(N1CC(C(N)=O)C(C)C1)=O)CC)N(C)C C(=O)(CCCC(=O)NCC1CC(C(=O)NCC23CC(CO)(CO2)C3)C1)OCC C=CC(C)(C)CC(=O)N1CC(CNC(=O)CNS(=O)(=O)NC)CC1C C1(C(=O)NC2(C)CCC(NC(=O)CN3CCOCC3)CC2)CC1C1CC(F)(F)C1 N1(C(c2ccc(CNC(C(C)N3CCCC3)=O)o2)=O)CCOC(C)(C)C1 C#CC1(O)CCN(C(=O)NCCN2C3CCC2COC3)C1 N1(C(C2(C)CC(C)(C)C2)=O)CC2CCCC(C1)N2C(=O)C(C)(C)c1cncnc1 Cn1nccc1CC(=O)NC(CNC(C1(CC(F)F)CC1)=O)C1CC1 CC(C)CC(O)C(=O)NCCCCn1ccnc1C N1(C(CCOCCCOC)=O)CCCC(C2CCN(C(=O)C(C)O)CC2)C1 CC1(C)C(CNC(=O)COC2CN(C(=O)C#CC3CC3)C2)CC1O N1(C(c2cncc(C)c2)=O)CCC2(CCCN2C(c2sccc2C(F)F)=O)C1 Cc1ccc(NC(C2COCCN2C(=O)Nc2cc(O)no2)=O)nc1 c1(C(=O)NC2(CO)CC(C)C2)cncc(CNC(C2(C)CNC(=O)C2)=O)c1 c1(C(C)C(F)(F)F)cccc(NC(C2CCCN2Cc2cccs2)=O)c1 c1(SC(C)C(=O)Nc2cc(Br)ccc2Br)ccc(S(=O)(=O)N2CCCCC2)cc1 c1(NC2(c3nnnn3C)CC(CC(C)C)OCC2)cccc(N=[N+]=[N-])c1 N1(C(c2c[nH]c(=NC)o2)=O)CC2(CC(NC(=O)CCOCCC(C)(C)C)CO2)C1 c1(C2C(C(=O)NCC(C)(C)NC(=O)CSC3COCCO3)C2)ccc(C#N)cc1 N1(C(c2c(C)cnnc2)=O)CCC(NC(=O)C2=COCCO2)C(CO)CC1 C1(C(=O)NC(C2CCCCC2)C#C)(NC(C2C(C)(C)C2(C)C)=O)CCN(C)C1 c1(OCC(=O)NCC23CCC2CN(C(=O)C(Cl)=CCl)C3)c(F)c(F)cc(F)c1F c1(C(=O)NCc2c(C)cccn2)cc2n(n1)CCN(C(C1CCOCC1)=O)C2 c1(OC)cc(F)cc(C(=O)N(CC(C)CNC(C2CCCCN2N=O)=O)C)c1N N1(C(C(COC)(F)F)=O)CCCN(Cc2cn(C3CC(O)C3)nn2)CC1 C1(C(=O)OC)CN(Cc2cccnc2OCc2ccccc2)C(CN)CO1 CCCC(F)C(=O)N1C(C(=O)N(C(C)C(C)(C)O)C)CCC1C1CC1 N(C1CCCOc2c(F)cccc21)C(c1snnc1OC)C.c1(C)ccccc1 c1(C(N2CC3CCN(C(c4nc(Br)cs4)=O)CC3C2)=O)cc(Cl)cc2cc[nH]c12 c1(NC2C(NC(c3n(C(C)C)ccn3)=O)CCCC2)nc(Cl)nc2c1ncn2C c1(SCC)ccc(CC(N2CCOC(CCNC(c3cncnc3)=O)C2)=O)cc1 C(CC(C)C(=O)N1CCC(C(C)NC(=O)C(C)Cc2ccco2)CC1)OC C1(NC(C(=O)N(CCCNC(C(C)OC2CCOC2)=O)C)C)(CO)CCCC1 C(c1ccc(S(C)(=O)=O)o1)=CC(=O)NCCCNC(CCC(CC)OC)=O C1(CCC)CN(C(=O)Cc2ccc(Cl)s2)CCN1C(=O)C(C)Cc1ccnn1C CC1CN(C(=O)Cc2cccnc2Cl)CC2(CCN(C(=O)CO)CC2)O1 N1(C(C2C(=C)C2)=O)CC(OC)CC1CCNC(c1ccc(OC)nc1)=O C1(CNC(C(C)SCC)=O)C(C2CC2)CCN1C(=O)COCC(F)F C(N=c1ccn(C2CCSCC2)[nH]1)c1c(N)n(C2CC2)nc1 CC(C)CC(C(=O)NC1CCOC1)ONC(c1cnn(C(F)F)c1)=O N1(C(c2cn(C3CCC3)nn2)=O)CC2CCC1CN2C(=O)C(O)CC(F)F CC(C)C(F)(F)CNC(=O)CCOCCNC(=O)CCC1CC1(F)F C(=O)(CCCCN(C(=O)C(O)CNC(C1(C)CCOC1)=O)C)NC C(=O)(CC(C(F)F)n1ccnc1)NCCCC(C)(C)NC(CN(CCC)C)=O c1(C(N2CC(C3(NC(CCc4n[nH]c(=N)s4)=O)CC3)C2)=O)ccc2cncn2c1 c1(C(=O)NC2CCCC(NC(c3scc(C)c3Cl)=O)C2)ccc2c(n1)CCOC2 c1(COC)cccnc1C(=O)NCC1(NC(C2CCC23CCC3)=O)CCOC1 C1(N=[N+]=[N-])(C(=O)NCC2(CSC)CC2)CCN(C(=O)C(C)OC2CCCC2)C1 N1(C(C2(N(C)C)CC2)=O)CC2CC(C(=O)NC3CC34CCC4)(C2)C1 C(=O)(CCCc1ccccn1)NCC(C)N(C(C(C)OCC#C)=O)C c1(CC(=O)NC(C)C(C)NC(C2CCSCC2)=O)cccc2c1SCCC2 N1(C(C2C(COC)C2)=O)CC2(CCC(CNC(c3nc(C)c(C)[nH]c3=O)=O)O2)C1 N1(C(C2(Br)C(C)(C)C2(C)C)=O)CC2CC(CNC(=O)CC#N)CC1C2 CC1OC2(CN=c3[nH]nc(CO)s3)CC1(NC(=O)Cn1ncn(C)c1=O)C2 C1(C(N2CC(NC(c3cn(CC(=O)OC)nn3)=O)C(C)C2)=O)CN=C2N=CNN2C1 CS(=O)(=O)c1ncc(C(=O)NCC2(F)CCC(NC(=O)C#CC3CC3)C2)s1 c1(C(=O)NC2CCCC2NC(C2CCOC2)=O)ccc(C2CC2)nc1 CCCCCC(O)CC(=O)NCc1nc(C(=O)N(C2CCCC(C)C2)C2CC2)co1 C1(NC(C2(CC)CCOCC2)=O)CCN(C(=O)C=Cc2ccncc2)C(C)C1 c1(C(C(=O)Nc2cccc(C(C)F)c2)NC(C2CC2(Cl)Cl)=O)c(C)cccc1Br N1(C(c2cc(CCC)oc2C)=O)CCC(NC(=O)CC2(C)OCCO2)C(CC)C1 N1(C(C2CC3(CSC3)C2)=O)CCCC2(CCN(c3ccc4nccnc4n3)C2)C1 C1(C(=O)NC2CC(CCNC(c3ccc(C(N)=O)[nH]3)=O)C2)CCc2nncn2C1 C(CCCC(=O)N(CC(O)C1CCC1)C)N(C(C1C(C(=O)OC)CC1)=O)C C(=O)(C1CCN(C)c2ccccc21)N(C)Cc1cncc(C)c1 C12(C(=O)NCCCN(C(C)C)C(c3c[nH]nc3Br)=O)CC1COC2(C)C c1(C(=O)NCC(CN(C(c2cnc(C)nc2)=O)C)(C)C)cc([N+](=O)[O-])oc1C C1(CC)CN(C(=O)C(C)(C)CN(C)C)CCN1C(=O)C(F)=CC1CC1 C(CC(C)(C)C(=O)NCC1CC1c1ccco1)NC(CC1(C)CCOCC1)=O C(=O)(C#CC1CCCC1)N(C)CC1CN(C(=O)COCC2CCCO2)CCO1 C(=O)(CC(C(F)(F)F)OC)N1CCC(N2CCN(C(CCC=CC)=O)CC2)C1 N(C(=NCc1ccc(Br)cn1)NCCC1CC1)C1C(C)C1 C1(C(=O)NCC2C(NC(c3ccn(CC)n3)=O)CC2)CCCC12CCC2 Cn1cncc1C=CC(=O)NC1CCCN(C(c2c[nH]nc2C2CCOC2)=O)C1 c1(OCCC)ccccc1C(=O)NCCN(C(=O)C(C)(C)C)C N1(C(=O)NC(C(=O)OC)C)CCSC(C(N2CCCC(O)C2)=O)C1 c1(OC)c(C(=O)N(C2CCN(C(C3CCC3F)=O)CC2)C)cccc1C(F)F Cc1[nH]nc(C(=O)NC2CC(n3cc(C4CCCN(C)C4)nn3)C2)c1Br S(=O)(=O)(c1cc(C(F)(F)F)ccc1N1CCn2ncnc2C1)N(C)CC1C(C)C1 C(=O)(C#CC1CCCO1)NC1CCN(C(c2c(Cl)sc(C)c2C)=O)C1 C1(C(C)NC(=O)C(c2ccnn2C)NC(=O)CNC(=O)C(F)(F)F)CCCCC1 N(C1CC(C)(C)CCc2ccccc21)C(C)C(c1ccccc1)O Cc1ncnc(O)c1CCC(=O)NCC(C)CNC(=O)C=Cc1cccs1 c1(C(=O)NCC(CCC)NC(C2CCS(=O)(=O)C2)=O)ccc2nn[nH]c2n1 Cc1cccc(C(NC(=NCc2nnc(CO)s2)NCC2CCCO2)C)c1C N1(C(c2ccc(C)cn2)=O)CC2CC1CN(C(=O)C(C)(O)C1CCC1)C2 C1(CC=C)COCC1NC(C1CCC(NC(C2CC(C)C2)=O)C1)=O C(C#Cc1ccccc1Cl)N1CCC(N(C(=O)C(O)C(C)(C)CC)CCC)C1 c1(C(N2CC=CC(NC(c3oc(C)c(CO)c3)=O)C2)=O)ccc2cccnn12 Cc1cc(F)c(C(N2CCCC(C(N3CCCC(C(C)C)C3)=O)CC2)=O)c(Br)c1 c1(C(=O)NC(CCF)C(=O)N2CCC(CSC3CC3)CC2)cc(Cl)ccc1F c1(CN=C(NC(C)C)NCc2cccc(CN(C)C)c2)nn(C)c2ccccc12 c1(C(=O)NCC2CCN2C(=O)C(O)CC2CCCCC2)nc2cccnc2s1 CC(CNC(c1csc(Cl)c1)=O)CC(=O)N1CC([N+](=O)[O-])C1 C1(CNC(c2scc(OC)c2)=O)CCN(C(=O)Cn2cnnc2O)CC1(F)F N1(C(=O)NC2C(C)C2)CCSC(C(F)(F)F)C1 Cc1cc(NC(C2(F)CC=CCC2)=O)cc(C(C)C)c1 N1(C(c2ccc(C#C)nc2)=O)CC2CC1CN(C(=O)C1=CCCO1)C2 C12(NC(CN(CCC)C)=O)CCCC(CN(C(c3ccc(C(N)=O)o3)=O)C1)C2 C1(CCCC)CN(C(C2CCSCC2)=O)CCN1C(=O)C(C)C(C)C c1(C(CC(N(C)C(C2CCCN2CCO)=O)=O)(C)C)ccc(C(F)(F)F)cc1 c1(CNC(C(CNC(C)=O)(C)C)=O)nnc2n1CCC2.C12OCCC1NC2=O N1(C(CC(CCC)C)=O)CC2CCCC1(CNC(c1ccc(C)cn1)=O)C2 C1(C(=O)NCC(CNC(C2(C(C)C)CNC(=O)C2)=O)(C)C)CC(C2CC2)=NO1 c1(COC(CC=C)CNCc2ccc(C)o2)ccc(F)cc1 N1(CC(=O)NCC2N(C(c3c(C)ncnc3)=O)CC2)OC(C)(C)CC1=O C1(CN(C(CC#C)=O)C)CCCN(C(C2CC2C(F)F)=O)C1 C1(C#N)(C(=O)NCCCOCCN(C)C(c2cn(C3CC3)nn2)=O)CCCO1 c1(C(=O)NCC(Cn2cc(C(C)N(C)C)nn2)OC)snnc1C1CC1 N1(C(C(CC)OCC)=O)CCCC12CCCN(C(=O)C1=C(Cl)CCCC1)C2 C1(C(N(CCCCNC(C2C(C)OC(=O)N2)=O)C)=O)C(F)(F)C12CCC2 CCCCC(CC)CC(=O)N(C)CCOCCNC(c1cc(C#N)ccc1O)=O C(CCC(F)(F)F)(S(CC1CCC(C)CC1)(=O)=O)c1cccnc1 C(=O)(CC(C)(C)CN(C)C)N1C(C(=O)NC2(CCOC)CC2)CC(F)C1 c1(CSCCNC(C2CC(F)(F)CN2NCc2ccco2)=O)cc(O)ccc1Cl c1(OC)ccc(C(N2CCC(C(CO)NC(C3CCOC3C)=O)CC2)=O)nc1 N1(C(c2c(C)con2)=O)CCC2(CCCCN(C(C3CC3C3CC3C)=O)C2)C1 C(N=c1ccnc(NCc2nn(C)c(C3CC3)c2C)[nH]1)C1(COC)CCCO1 C1(CC(=O)NCCn2ccc(C(=O)NC34CCCC3C4)c2)NC(=O)NC1=O C1(COC)(NC(=O)CN(C)CC2(F)CC2)CCN(C(=O)CC(C)CN(C)C)C1 N1(C(C2(F)CN(C(c3c(C)snn3)=O)C2)=O)CC(C(N)=O)C(C)C1 c1(-c2cn(CC(=O)CC3(CC)CCNC3=O)nn2)ccc2cnccc2c1 C(CC(C)S(C)(=O)=O)NC(C(=O)NCCOC)=O.c12cccc(c1)C(=O)N2 c1(C(=O)NCCC2(NC(C(C)OCC3CCCO3)=O)CC2)cn2c(n1)CCCC2 N1(C(C2CC3CN(C(CC(C)F)=O)CC3C2)=O)CC2C3CCC(O3)C2C1 C(C(=O)NC1CCCCC1)(C(C)CC(C)(C)C)N(C1CCCCC1)CC C1(C)(CC)C=C(C(=O)Nc2cccc(NC(=O)CC3(C(=O)OC(C)=O)CC3)c2)C1 C12(NC(c3cccnc3O)=O)CCCN(C(C3CCOCC3)=O)CC1C2 c1(C(N(CCCNC(=O)CN2CC(C)C2)CC)=O)cnn2ccc(Cl)c(F)c12 C1(C(N(C2CCC2)CC#C)=O)CC2C=CC1N(C(=O)CN1CC(=O)NC1=O)C2 n1(CC(=O)NCC2(C)N(C(CC(C)C3CC3)=O)CCC2)cnc([N+](=O)[O-])n1 N1(C(C)=O)CCn2ncc(CNC(=O)CCNC(C3CCCCC3)=O)c2C1 C1(C(=O)NCCC(=C)CNC(=O)CN2CCCCC2=O)CCCC(C#N)C1 C1(NC(c2c[nH]nc2C2CC2)=O)CCN(c2cc(C3CCC3)ncn2)CC1F c1(C(=O)NC2CCN(C(C3C(C)CCO3)=O)CC2CO)c2c(nn1C)CCSC2 c1(C(N2CCC(C)(NC(=O)C(c3ccccc3)F)C2)=O)cccn2ncnc12 c1(-n2c(C)ncc2)ncccc1C(=O)OC1CC(OCc2ccccc2)C1 CC(C)CC(C(=O)NC1CC(C)(C)C12CC2)NC(c1cccc(O)n1)=O C1(C(N(CCNC(=O)CC2CCCC2)CC)=O)CC2CC1CC2(F)F CC(C)C(F)(CNC(C1CCN(C)C(=O)C1)=O)C(=O)NCCC1(C)CCOCC1 C(=O)(CS(N)(=O)=O)N1C(CN(C(CNC(CNC(C)=O)=O)=O)C)CCC1 N1(C(C(C=C)OC)=O)CCC(O)CC1C(=O)NCC1(C2CC2)CC1 C(CCC(C)(C)C(=O)N1CC(C)=C(C)C1)NC(C1CN(CC)C(=O)C1)=O c1(C(=O)NC2C(CNC(CCCCCC)=O)C2)cnc2c(Cl)cccn12 Cc1n[nH]c(C)c1C1CC(C(N2CC(CCF)C2)=O)C1 C1(CNC(c2c(CC)nc[nH]2)=O)CC2(CCC2)CN1C(C1CC1[N+](=O)[O-])=O C(C)(c1ccccc1C)=CC(=O)NC(CNC(C(CCSC)O)=O)CC(F)(F)F N1(C(c2c(C(C)(C)C)ccs2)=O)CC(NC(C2(C)CCCO2)=O)C2CCCCC12 C(=O)(CC(C(F)(F)F)NC(C1(SC)CC1)=O)NCC(C(=O)NC)O C1(C(=O)NCC2(CNC(C(CC)O)=O)CC2)CCCCN1C(C)C C1(CC(N2CCC(N3CCC3)CC2)=O)CCCN(C(c2ccc(Br)s2)=O)C1 C(C(CC1CC1)C(=O)NC(CO)CCF)NC(COCCN(C)C)=O C1(C(C)C)C(NC(=O)COCCF)CCN1C(=O)CCN1CCNC(=O)C1 N1(C(C(C)=NOCC#N)=O)CC=C(C(=O)NCC(C)(C)CCCO)C1 CCCC(C)(CC)C(=O)NCC1CCN(C(c2cc(C)no2)=O)C(C)C1 C(CC(C(=O)O)N(C(=O)CC1CC2CC2C1)C)SC c1(OC)cc(C)c(C(=O)NCC=CCNC(C2CCCC(F)C2)=O)c(C)c1 C(=O)(C(O)C(C)C)N1C(CN(C(C2CCC(C(N)=O)CC2)=O)CC)CCC1 C(CC(C(=O)NCC1CSCCO1)NC(c1cc(C)[nH]c1C)=O)SC N1(C(C2CCN(CC)C2)=O)CCCCC(C(=O)NCCCC(C)C)C1 N1(C(C=C(C)C)=O)CCCC(CCC(=O)NCC2(CO)CCCO2)C1 N1(C(CCCC2C(C)C2)=O)CC(C2CN(C(c3ccc([N+](=O)[O-])cc3)=O)C2)C1 C1(C(N(CC(N2CCN(C(CC(C)C3CC3)=O)CC2)=O)C)=O)CC(=O)NC(=O)N1 CC1CCCCN1CC(=O)NC(c1ccccc1)C(=O)NCC=CC(C)(C)C C1(NC(CCC(C)SC)=O)CN(C(=O)C(c2cc(C)oc2C)C)CCC1O c1(C(=O)NC2CN(C(CCC(C)C)=O)C(C)CC2)cnc2c(F)cccc2c1 C(C(C)(C)CC(C)C)NC(C1CCN(C(CCC(C)=O)=O)C1C(C)C)=O c1(NC(C(=O)N(CC)Cc2cccc([N+](=O)[O-])c2)=O)ccc2oc(O)nc2c1 c1(C(=O)NC2CC(CC(NOCC(=O)N(C)C)=O)C2)ccc(Cl)cc1 C1(CNC(C(CC)NC(C)=O)=O)C2CN(C(=O)CCn3ccnc3)CC12 C(c1cc(F)c(F)c(F)c1)=CC(N1CC(CCNC(C(C)SC)=O)OCCC1)=O N1(C(C2CCC(NC(=O)C=CC3CC3)C2)=O)CCCc2occc2C1 CC1C(NC(C2CCCN2C)=O)CC2CCC1N2C(C1(c2ccccc2)CC1)=O N1(C(COCCC(C)C)=O)CC2CCCC2(NC(C2CC(CCO)C2)=O)C1 C1(NC(c2cc(F)c[nH]2)=O)CCN(C(c2ccc(CO)cc2)=O)CC1 CC1=NN(C)C(=O)C1CC(N1CC(C)C1CNC(=O)CC12CCC(CC1)C2)=O S(=O)(=O)(c1c[nH]ccc1=NC1CCCC(C)C1)NC(CC)(CC)CCO C(N(C)N1CCCC1C(F)F)c1sc(C)c(C2CCCO2)n1 N1(CC)CCCN(C(C2CC2C(C)NC(c2cc(C)n(C)c2C)=O)=O)CC1 CCC(C)(C)CCNC(C1CCN(C(=O)C(C)n2cncn2)CC1)=O C(=O)(NNC(=O)C(N)C(C)(C)C)c1ccc(OC)c(Cl)c1 S(=O)(=O)(c1ccc(N(C)C2CC2)c(Br)c1)NCCNC(=O)OCC c1(C(=O)NCC2N(C(C3CN(CC)C(=O)C3)=O)CC(F)C2)ccn2ccnc2c1 c1(C(=O)NCC2N(C(C3C(=O)NCC3)=O)CCC2)cc2c(Cl)nccc2o1 CCCC(C)(CC)C(=O)N1CCC(N(c2cc(CC)nc(C)n2)C)C1 N1(C(c2ccc(C(C)(C)C)nc2)=O)CC(NC(c2cc(Br)c[nH]2)=O)CC(O)C1 C(C)(C(CC(=O)N1CCCCC1C1(O)CC1)NC(c1c[nH]c(=N)c(C)c1)=O)OC C1(NC(CC2CC(C)(C)OCC2)=O)CC2CC(C1)N(C(=O)CCC[N+](=O)[O-])C2 C1(CC#N)CN(C(c2cc(O)nc(O)c2)=O)CCN1C(c1cc(Cl)c(Cl)s1)=O C1(C(=O)NCC(C)NC(C2(c3c(C)cno3)CC2)=O)COc2ccccc2C1 N1(C(C(CC)CO)=O)CCCC2CN(C(c3ccc(OC)cc3O)=O)CC12 C=CCC(C)(CC)C(=O)NC(C1CCCN1C(c1ccc(Cl)cc1N)=O)C c1(C(=O)NCC2(C)N(C(C=CC=CC)=O)CCC2)ccc2c(c1)nc(O)n2CC N1(C(c2c(CCC)[nH]nc2)=O)CCCC2(C1)CN(C(c1conc1C)=O)CCO2 c1(CNC(=O)NCc2csnn2)ccccc1CC1CCCCC1 c1(C(N(C2CCCN(C(=O)C=CC(C)(C)C)C2)CC)=O)[nH]nc([N+](=O)[O-])c1Cl c1(C(N)=O)nc(C(=O)NCCCCCNC(c2cc(C(F)F)no2)=O)cs1 C(=O)(C1Cc2c(Cl)cccc21)N1CC(NC(c2csc(C3CC3)n2)=O)C(O)C1 N1(C(C2(NC(C)=O)CCCC2)=O)CCC(NC(=O)CC2CC2(C)C)C(O)C1 C1(NC(c2onc(C)n2)=O)CN(C(C2CCC2(C)C)=O)Cc2nccn2C1 c1(OC)cccc2c1OCCC2N=c1cc[nH]c(=NCCC2CCCO2)[nH]1 Cc1cc(C(=O)NCC(C)CC(=O)N2CC(C)(F)C2)c(C)[nH]1 S(=O)(=O)(c1ccc([N+](=O)[O-])c(F)c1)N(CC(N1CCC2CCOCC2C1)=O)C C1(C)(C(=O)NCC2(CC)CC(C)(C)C2)CN(C(C2CC(C)(C)C2)=O)CC1C CC1(NC(=O)CCC2CC(F)(F)C2)CC(NC(=O)CCC2CCC(=O)N2)C1 C1(N(C(C2N(CC)CC2)=O)CC)CCCN(C(=O)C(C)O)C1 c1(C(=O)NC2C(CNC(CS(=O)(=O)NCC)=O)CC2)cnn2c1OCC(C)C2 N1(C(c2ccc[n+]([O-])c2)=O)CC2CCN(C(c3n[nH]cc3Cl)=O)C2C1 C1(NC(c2cc3oc(Cl)cc3[nH]2)=O)CCC2CN(C(=O)CCC3CCC3)CC2C1 CCCCCC(C)CC(=O)NCC(C)(CO)NC(=O)C(c1cccn1C)=O Cc1cc(C(=O)NC2CN(C(c3ccoc3Br)=O)CC3(CC3)C2)c(O)nc1C C(=O)(C(C)CCC)NCCOC1CCN(C(c2nc(CCCC)sc2)=O)C1 CC1C(C(=O)N2CC3(CCCC3)C2C(N2CCCC3(C2)N=N3)=O)=NOC1C N(C1CCCc2ccoc21)C(=O)NCC1CCN(CCOC)CC1 Cc1cc(C(=O)N(C2CCCN(C(C3CCCN3C3CC3)=O)C2)C)cc(C)c1N CS(=O)(=O)c1cc(C(N2CC3CC(NC(C4CCOC4)=O)CC2C3)=O)ccc1F c1(OC)cn(CC(=O)N(CC(O)CNC(c2ncc(F)cn2)=O)C)c(C)cc1=O C1(COC)(CNC(=O)C(C)CO)CCN(C(C2CCCN2C2CC2)=O)CC1 N1(C(C(CCC)CC)=O)CC(NC(=O)COCCOCCO)CC12CCCC2 N1(C(c2c(CC)[nH]cc2)=O)CCC(C)(C)C1C(N1CCC(CC2CC2)CC1)=O c1(C(=O)NCC2(O)CN(C(C(C)C(C)(F)F)=O)C2)ccc2c(c1)C(=O)N(C)C2=O n1(CCC)nccc1C(C)NC(c1cnc(C2CCCCC2)s1)c1nnnn1C c1(CC)cc(C(N2CC(NC(=O)C(C)(F)F)C(F)C2)=O)ccc1Cl N1(C(C(=O)NCCCCCC)C2CC=CC2)CCCC2(C1)NC(=O)NC2=O C1(C(N2C(CC(=O)NCC(O)C3(Cl)CC3)CC2)=O)CC2(CCC2)C1 c1(CC(=O)NC2CC(n3cc(CSCC)nn3)C2)ncc2c(n1)CCC2 C1(NC(=O)C=Cc2ccoc2)CC(NC(=O)CCCN2CCCCC2)CC1O C1(C)(NC(C(C)N(C)C)=O)CN(C(=O)C(C)(C)c2ncco2)C1 C1(OCC)CCN(C(C2CC2C(=O)Nc2cc(OC)nn2C)=O)CC1 C1(C(N(CCOCCNC(c2c(CCC)cccc2)=O)C)=O)CN2CCN1CC2 C1(CNC(=O)CSc2nncs2)C=CCN1C(=O)C(n1ccc(C2CC2)n1)C C1(OC)CCC2(C(N3CC(F)(CNC(C4CC4Cl)=O)C3)=O)CC12 CCC(CC)C(=O)NC(CN(C)C(C12CC(CO1)C2)=O)Cc1ccccc1 C1(c2n(C(C)(C)C)nnn2)(Nc2cccc(O)c2)CCC2(CCCOC2)C1 C(CC)(C(=O)NCC1(COC)CN(C(c2ccc(C(C)=O)[nH]2)=O)C1)=CC C=CCC(C)C(=O)NC(C(=O)NCc1ccncc1CC)c1ccoc1 CS(=O)(=O)CC(=O)NCC1(C(N)=O)CN(C(c2cnn[nH]2)=O)C1 C(C(C(C)(C)C)NC(=O)Cc1nccs1)NC(C1(C(=O)OC)C(=C)CC1)=O c1(C(N2CC3CC3(CNC(C3CC(F)C3)=O)C2)=O)ccc(Cl)cc1Cl c1(C(N(C2CCCCC2NC(C2(C3CC3)CCOCC2)=O)C)=O)cn(C)[nH]c1=N C1(NC(Cc2c(C)nc[nH]2)=O)CN(C(c2cc3ncccc3s2)=O)CCC1(C)C CC1CCC(C(=O)N(CC(C)O)CCNC(c2csc(Br)c2)=O)CC1 N1(CC(=O)N(CC(CC)NC(=O)C(C)n2cccn2)C)CCNC(=O)C1 c1(C(C)=O)cc(Br)c(C(=O)NCCC2CCCCN2C(=O)OC(C)(C)C)s1 C1(NC(c2cc(CCC)on2)=O)CC2CCC1CN2C(C1CCC(C)C1)=O c1(OC)cccc(C(=O)NC2CC(NC(C3(CC(F)F)CC3)=O)C2)c1 C#Cc1cccc(C(N2CCOCC2CNC(=O)CCOc2ccccc2)=O)c1 NS(=O)(=O)c1csc(C(=O)NCC2CN(C(=O)COc3ccc(F)nc3)C2)c1 Cc1ncc([N+](=O)[O-])n1Cc1cccc(CS(=O)CCC(=O)N2CCOCC2)c1 c1(C(=O)NC(C(C)NC(c2cc(CCOC)on2)=O)C)ccc(Cl)c(C)c1OC C1(NC(C(C)(C)c2cscn2)=O)CC2CCC1N(C(c1ccc(C#N)cc1)=O)C2 N1(C(C2(CCC)CCNC2=O)=O)CCCN(C(c2occc2COC)=O)CC1 Cc1cc(C(=O)N(C2CN(C(=O)CCCc3cnccn3)CC2F)C)c(C)cn1 C1(C(=O)NC2CCC(NC(c3cccnc3)=O)CC2)(COC)CCC(=O)N1 Cc1nc(C(=O)NC2CC(NC(C3CCC(=O)NC3)=O)C2)nn1C c1(C(=O)NCC(C)N(C(C2C(C=C)C2)=O)C)ccc(C)c2cccnc12 Cn1cc2c(C(N3CCC4(C3)CN(C(=O)CC(F)F)CCO4)=O)cc(F)cc2n1 C1(NC(C2(OC)CC2)=O)C2CCN(C(=O)C(C)CC3CCCC3)CC12 C1(NC(CC2C(C)OC(C)C2)=O)CCC2CC1CN2C(c1ocnc1C1CC1)=O C1(N(C)C(c2cn(C(F)F)cn2)=O)CCCCC1NC(=O)C1=NOCC1 CCC(C(=O)NCCN(C(C1CC1C(F)(F)F)=O)C(C)C)SC CN1CC(C)(C)CC1C(=O)NC1(CF)CCN(C(=O)C=Cc2ccn(C)c2)C1 CC(C)CC(CNC(c1ccnnc1)=O)C(=O)NC1CCCC12CC2 C1(C(N2CCN(C(C=Cc3c(C)cccc3F)=O)CC2)=O)Cc2c(F)cccc2O1 c1(CNC(C2CCC(COC)C2)=O)ccc2c(c1)CN(C(=O)CCOC(C)=O)C2 C=CCCCC(C(=O)NCCN(C)C(=O)C1CC1)NC(=O)C(F)C(C)(F)F C=C(Cl)CC(C(=O)N1CC2CSCC2C1)NC(c1cnc(C)c(C)c1)=O C1(C(N(CCCCN(N2CCCC2)C(=O)C=C2CC2)C)=O)(C(C)=O)CCOCC1 C1(C(N2CCCC(NC(c3n(C(C)C)ccn3)=O)C2)=O)CCCC12CCOCC2 c1(C(=O)NC(CN(C(=O)CC2CCN(C)C2=O)C)(C)C)cccc(P(C)(C)=O)c1 C1(CN(C(C(n2c(C)ccn2)C)=O)C)CCCN(C(=O)Cc2ncsc2Cl)C1 N1(C(CC2(CSC)CC2)=O)CCC2(C1)CN(C(C1CC1C)=O)C2 Cn1ncc(C(=O)Nc2ccc(O)cc2)c1C(N)=O S(=O)(=O)(c1ccc2[nH]c(=NC3CCN(C(C)=O)C3)ccc2c1)NC1C(CC)C1 c1(N2CC(C(=O)Nc3c(C)cccc3Cl)C(O)CC2)ncc2c(n1)NC(=O)C2 C1(NC(N(CCC)CC=C(C)Cl)=O)CCC(c2ccccc2)O1 N1(c2nnc(C)s2)CCCC(CNC(c2coc(Cc3ccccc3)n2)=O)CC1 C1(C(=O)NCC(C)(C)CC2CCOCC2)CNCC12CCS(=O)(=O)CC2 Cc1cccc(CC(=O)NC2CCCC2NC(C2(C3CCCCO3)CC2)=O)c1F c1(C(N(CCOCCNC(CC2CC(=C)C2)=O)C)=O)cc(Cl)nnc1O C1(NC(C(CC=C)OC)=O)CCC12CCN(C(=O)CC(C)F)CC2 C(=O)(CCCC(C)NC(=O)CC1CCCN1C)NC(C(=O)OC)CO C1(NC(C2(C)CN(C(c3ncc(NC)nc3)=O)C2)=O)CCCN(O)C1=O C#Cc1cccc(C(=O)NCC(CC=C)C(=O)N2CCC(SC)CC2)c1 c1(C(C)NCc2cnc(C(F)(F)F)o2)ccncc1Cl c1(N2CC(CNC(C3(C)C=CCC3)=O)C(C)(C)CC2)ncnc2ccc(O)cc12 C(=O)(C1CCc2ccc(OC)cc21)N(CCN(C(C(CCC)C)=O)C(C)C)C CC1(C)CC(CNC(=O)CSCc2cccs2)CN1C(=O)C1=CCOC1 N1(C(CCSCCCC)=O)CC(C(=O)N(CC)Cc2ccsc2)CC(C)C1 c1(C(=O)NC2C(CNC(C3CC(OCC)C3)=O)C2)ccc(F)cc1Br N1(C(C2(C)CCCN(C(c3cn(C)nc3)=O)C2)=O)CCC2(CC1)CNC(=O)C2 C1(C(N(CC(C(=O)NC2C(CC(C)C)C2)C)C)=O)COCCN1C C(=O)(C1=CC2CCCC12)NCC1N(C(C2(C)CCN(C(C)=O)CC2)=O)CCCC1 c1(NC(CCN(CC=C)C(C2CCOCC2C)=O)=O)ncc(C#N)cc1C c1(NCC(N2CC(C(C)NC(C3(C)C(CC)CCC3)=O)C2)=O)cccc(C#N)c1 c1(C(=O)NCC(C)N(C(=O)C(F)C(C)(C)O)CC)cc(C)c2c(O)n[nH]c2n1 c1(C(C)C)ccc(OC(C)C(=O)NC2CCCN(C(=O)C(C)(C)C#N)C2)cc1 c1(C(=O)NC(C)C(CO)NC(C2CNC(=O)C2)=O)nc(Br)c2ccccn12 n1(CC)ccc(C(=O)NCC(C)N(C)C(C2CCN(C3CC3)C2=O)=O)cc1=O C1(CC(=O)NC(C)CCCNC(c2ccsc2Cl)=O)CC2CCC1O2 C1(C(=O)OCC)Cc2c(ccc(F)c2F)CN1CC(=O)NCCC1CC1(Cl)Cl c1(C(N2CCC(CNC(C=C(C)Cl)=O)C23CCC3)=O)cc2ccccc2nc1O C(=O)(C#CC1CC1)NCC1(OCC)CN(C(c2cnn(C)c2)=O)C1 CC1C(NC(C2C3CCCC23)=O)CCN1C(C1CC12CCC2)=O C(=O)(CCCNC(=O)NC)NCC(CC)NC(c1cnc(OC(C)(C)C)s1)=O c1(C(=O)NC(CC)C(=O)NC(c2nccc(O)n2)C)c(C)cccc1C N1(C(C(CNC(C2CN(C)CCO2)=O)OC)=O)CCc2cccc(O)c21 c1(C(=O)NCC2C(OCC)CN(C(C3CCSCC3)=O)C2)cc(Cl)ccc1N C(=O)(CC(C)CCCCC)NCC(C(N1CC(C=C)N(C)CC1)=O)N(C)C C(=O)(C1=CCCCCC1)NC(C)(CNC(C1CC2CCC1O2)=O)C1CCC1 C=CC(CC)CC(=O)N1CC2C(N(C)C(c3ccc(C(C)(F)F)nc3O)=O)C2C1 CCCCCC(C)(CC)C(=O)NCC(C(C)C)NC(c1nncs1)=O C(CC(F)(F)CO)n1cc(C(C)(C)NCC(=O)NC2CCCCC2)nn1 C1(CNC(=O)CCOCC2CC2)(NC(=O)CC2CCOC2=O)CCCC1 N1(C(c2cnn(CC)c2Cl)=O)CCC(O)C(NC(=O)Cc2nonc2C)C1 N1(C(C2(N(C(CN3CC(=O)NC3=O)=O)C3CC3)CCC2)=O)CC2(CCCC2)C1 CC(C)CCC(F)C(=O)N1CCCCC1C(=O)NCCCCCCF N1(C(c2cccc(CC)n2)=O)CCN(C(C2SCC=C2C)=O)CC1CCO CCCS(=O)(=O)C(C)C(=O)NC1CCC1CNC(c1ccc2c(c1)OCC2)=O N1(C(CC#N)=O)CCC(NC(C2CCC(F)C2)=O)CC1 C12CC3CCCC3N1C2=O.C12(N)C3C4C5C3C1C5C24.C1(C=O)CC2C=CC1C2 Nc1cccc(Cl)c1C(=O)NC1CC1NC(c1ncoc1C1CC1)=O c1(C(=O)NC2C(NC(c3cn(CCC)nc3)=O)COC2)nccnc1N N1(C(C23C(CN(C(C)=O)C2)C3)=O)CCOC2CN(C(=O)CCCNC(N)=O)CC12 N1(C(CCCCCC)=O)CCC=C(C(=O)N2CC3(C2)CC3(F)F)C1 c1(C(N2C(C(N3CC(CC(=O)OC)C3)=O)CC(O)CC2)=O)cccc2c1CCC2 C12(CNC(=O)Cn3cccn3)CC(C1)C(NC(=O)C(F)(F)C1CC1)CO2 CC1CCC(C(=O)NCc2nnn(C)c2C(=O)N(C)CC2COC(=O)N2)CC1 C1(NC(CN(CC(C)(C)C)C)=O)COCCN(C(=O)C(F)(F)c2ccccn2)C1 c1(OC)cc(C(=O)NC(C)CCNC(=O)C(C)n2cccn2)ncn1 c1(C(=O)NCC2(C)CCN(C(C3(CCOCC)CC3)=O)C2)cnn(C)c1C(C)=O C(=O)(CC(C)(C(F)F)N(C)C)NC1CCC(NC(c2c(C)cc(F)cn2)=O)C1 Cc1[nH]c2ncnc(NCC(C)NC(=O)CSc3n[nH]c(O)n3)c2c1C C(=O)(CC1CC(=O)Nc2ccccc21)N1C2CN(C(COCC#C)=O)C(C2)C1 C1(C(N2C(CNC(c3ccsc3Br)=O)CCC2)=O)CC12CCOC2 N1(C(C(C)NC(N)=O)=O)CCC(NC(c2cc(F)cnc2O)=O)C(O)C1 N1(C(C2CC(OC)(OC)C2)=O)CCC(NC(=O)C(C)Cc2ccco2)C12CCC2 N1(C(C(C(CC)C)C)=O)CC2CCCC(C1)N2C(C)C(N1CCN(C)CC1)=O N1(C(c2c(C)c(Cl)ccn2)=O)CC2CC(C)N(C(C3CC(C(F)(F)F)C3)=O)C2C1 c1(-n2c(C)c(C(=O)NC3(C)CC(NC)C3)nn2)cccc2cccnc12.C1(=O)CN1 c1(OC)ccc(C(N2CC(O)(CNC(C3CC34CCC4)=O)C2)=O)c(O)c1 C1(CNC(C2C(C(C)C)CCC2)=O)CCC2(CN(C(c3cc(N)ccn3)=O)C2)O1 N1(C(C(COCC)C)=O)CCCC(CNC(c2csc3nccn23)=O)CC1 C(=O)(C(CNC(c1ccc(C)c(O)c1)=O)C(C)(C)C)NC1C(CC=C)COC1 CCCCC(F)C(=O)N1CCN(C(c2cccc(C=C(F)F)c2)=O)C(CO)C1 C=C(C)CCC(=O)NCCC1CC(NC(c2ccnn2-c2ccccc2)=O)C1 N1(C(CC2CCN(C)C2=O)=O)CC2(CC2)CC1CNC(c1csnc1Cl)=O N1(C(c2c(C)ccnc2)=O)CCC2(CC(NC(=O)C(C)O)C2)C1 C=C1CCC(C(=O)NCC2CC(F)CN2C(C2CCCCN2CCCC)=O)CC1 CCC(C)CC(C(=O)N1CC(CO)C2(CC2)C1)NC(=O)CCC(N)=O Cn1cc(NCc2ccccc2C(F)(F)F)cc1CNC(C12CC3CC1C2C3)=O CC(c1ccc(F)cc1)=CC(=O)NCC1(C)CCN(C(=O)Cc2cnccn2)C1 C(C(C(C)C(C)C)NC(=O)CC12CCC(CC1)OC2)NC(COCC(=O)NC)=O c1(C(N2C(C(N3CC(C(=O)OC)N(C)CC3)=O)CC2)=O)ccc2[nH][nH]c(=N)c2c1 C(CCO)(C(=O)NCC(O)CNC(=O)Cn1ccc(Br)n1)N(C)C C(=O)(C1CCc2c(Cl)cccc21)N1CC(NC(c2ccc[nH]2)=O)(CO)C1 c1(C(=O)NC2C(CNC(C(COC)(C)O)=O)C2)cc(Cl)c(Cl)c(Cl)c1 CCC(C)CC(C(=O)O)NC(=O)Nc1ccc(Oc2ccccn2)cc1 c1(C(=O)OC)nnc(-c2ccc(Cl)cc2)cc1C(F)(F)F.C12OCCC1C2 NS(=O)(=O)N1CCC(C(=O)NCCC(O)CNC(C2CC3CCCCC23)=O)CC1 c1(CC)ccc2cc(C(=O)NC3CCC(N4CCCC4)CC3)ccc2c1 c1(C(=O)NC(C)CN(c2ncc(C#N)cc2F)C)ccc2nc[nH]c2c1 c1(C(N2C(C(C)NC(C3CC4C=CC3C4)=O)CCC2)=O)ccc(O)cc1F Cc1cc(C(N2CC3CC3(CNC(C3CCCC(O)C3)=O)C2)=O)cnc1C(F)F O(NC(=O)CN=c1nc(N2CCC(CC(=O)N(C)C)CC2)c2sccc2[nH]1)CC CC(C(F)C(=O)NC1CC2(CCCN(C(=O)CC(C)(C)C(F)F)C2)C1)C(F)(F)F C1(NC(CC2OCC(C)(C)C2)=O)CC2CCC(C1)N2C(=O)C(C)(C)C#N c1(C(=O)NCC2C(C)CCN(C(CCCCSC)=O)C2)ccnc2c1cnn2C c1(C(=O)NC2(CC=C)CN(C(=O)C=CS(C)=O)C2)cn(CC)c(C)cc1=O C1(NC(C2CCC(CC(=O)OC)C2)=O)CCCCCN1C(=O)COCC(C)C c1(C(=O)NC(CCNC(C(C)OCCC#C)=O)C)ccnn1CC(F)(F)F C1(NC(c2ccc(C(F)F)nc2)=O)CCN(C(=O)C(F)=CC2CC2)CC1CO C(c1ccc(F)cc1[N+](=O)[O-])=CC(=O)NC1CCCC(NC(C2(C#N)CC2)=O)C1 CC#CCCCC(=O)NCC1CCC(NC(=O)CC2(n3ccnc3)CC2)C1 c1(C(N2CC(O)(CNC(Cc3n(C)ncc3)=O)C2)=O)c(C(F)(F)F)cncc1F C1(OC)(CNC(C2(NC(=O)C=C(C)C(C)(C)C)CC2)=O)CCCCC1 c1(CCN(CCC(=O)N(C(C)C)CC2CC2)C)nc(O)c2ccccc2n1 C(=O)(CC(F)(F)C(F)(F)F)NCC1N(C(=O)COC(F)F)CCC1C1CC1 c1(C(=O)NCCCN(CC)Cc2cncnc2)ccccc1C(C)C C(=O)(CCS(=O)(=O)c1cc(Cl)ccc1Cl)N1CCC(C)CC1C(F)(F)F C1(CNC(C2(CC=C)COC2)=O)(COC)CCCN1C(=O)Cc1c[nH]nc1O C1(C)(CC)CC(NC(c2ccn(CCNC(=O)C(O)C(C)(C)C)c2)=O)CCO1 c1(OC)nc(C)cnc1C(N1CC(O)(CNC(C2COC(=O)N2)=O)C1)=O c1(NCCCc2c(C)cccc2)ncccc1S(=O)(=O)NC1CN(C)CC1C c1(C(=O)NCc2cc(C)cc(Br)c2)cc2cc(-c3cccc(C)c3O)ccc2[nH]1 Cc1[nH]c(C)c(C(N2CCC(CF)(NC(C3CC=CCC3)=O)C2)=O)c1C N1(CC(C)C)N=C(C(=O)NCC2(C)CCN(C(C3CNC(=O)N3)=O)C2)CCC1=O N1(C(C=CC=CCC)=O)CC(N(C(=O)CCC2CC2(F)F)C)C(C)(C)C1 CC1CC(NC(=O)C(C2CC2)C2CC2)CN(C(c2ccccc2O)=O)C1 C(CCCCC(=O)NC(C1CC1)C1CC1)N(C(C1C(C)CCC1)=O)C CCC(CC)C(=O)NCC1CN(C(c2ccc(N)cn2)=O)C2CC12 C1(C(N(CC)CC)=O)CCC(NC(C2CCCN(NCC3CCCC3)C2)=O)CC1 C(=O)(C1=NOC(C)(C)C1)N1CCC(NC(c2cn(C(C)C)nc2)=O)C(O)C1 c1(C(=O)NC2CCN(C(c3ccc(CC)[nH]3)=O)C2)cc(Cl)c(Br)[nH]1 c1(C(=O)NC(CN(C(=O)C(C)c2cccs2)CC)C)cc(C(N)=O)n(C)n1 C(=O)(C(CNC(=O)COCC1CC1)CC(C)C)N1CCC(N(CC)CC)C1 N1(C(CN(CCOC)C)=O)CCC(C)(C)C1C(N1CCN(CCO)C(=O)C1)=O c1(C(N2CCCC(CN(CC)CC)C2)C(=O)NCC)nc(Cl)ccc1Cl Cc1cc(C(C2CC2)NC(=O)C(=O)NC(C)CCc2ccccc2)cc(C)c1 c1(C(=O)NC2CCN(C(c3cc(OC)n[nH]3)=O)CC2O)cn2cc(C)ccc2n1 c1(N2CCN(CC)C(C)(C)C2)nc2cc[nH]c2c(=NCc2c(C)noc2C)[nH]1 c1(C(N2CC(NC(CC(C)C(F)(F)F)=O)C(C)C2)=O)cc2n(c1)CCS(=O)(=O)C2 Cc1c(C(=O)NC2CCCC(NC(=O)C=CBr)C2)cnn1C1CCC1 C(=O)(C1=CCOCC1)N1CC(C#C)(C(=O)NCC(C)C(=O)OCC)C1 c1(C(N2CCC(NC(CC(C=C)(C)C)=O)C(C)C2)=O)cccc2c1CCOC2 c1(CC(=O)NC23CCC(NC(CC(C)CF)=O)(CC2)C3)ccc(S(N)(=O)=O)cc1 c1(C(N2CC=C(CNC(c3ccc(F)o3)=O)CC2)=O)c[nH]c2ccccc12 N1(CCNC(CCOCC)=O)CCN(C(c2ccc(C3CC3(F)F)cc2)=O)CC1 c1(CC)ncnc(N(C2CCC3(CC2)CC3)CC2(F)CCCNC2)c1F C=CCC(CC)N=c1nc(N2CCC(C)(CCO)C2)c2sccc2[nH]1 c1(COC(=O)Nc2ccccc2F)nnc2n1CCC(C1CC1)C2 N1(c2cc(C(C)=O)ncn2)C2CCC1CC(CNC(=O)Cc1c(C)noc1C)C2 c1(CN(C)CCOc2ccc(C(F)(F)F)cc2)ccc2sccc2c1 CC1(C)CCCC1CCNC(=O)C(C1CC1)NC(C1OC2CCC1C2)=O N1(C(c2c(C)nccc2Cl)=O)CC2(C1)SCCC2NC(=O)CC12CCCC1C2 C1(NC(C2CC(Cl)(Cl)C2)=O)CC1C1CCN(C(c2cccc3c2OCO3)=O)CC1 C12(C(=O)OC)CCC(CNC(=O)CCc3ccncc3C)(CC1)OC2 CCC(CCCC(=O)NC1CCSC1)NC(c1ccc(N)cn1)=O C#CC(C)(C)C(=O)NCC(C1CCCN(C(c2sc(CC)nc2C)=O)C1)(C)O C=C(C)CCC(=O)N(C1CCN(C(C2(CO)CCCO2)=O)C1)CC N1(c2nccc(OCC)n2)CCC2(CCCC2CNC(c2ccc(Br)o2)=O)CC1 c1(C(=O)NCC2CCN(C(C3N(CC)CCCC3)=O)C2)c2c(nn1C)CCC2 N1(C(c2c(OC)csc2)=O)CCC(CNC(c2n[nH]cc2[N+](=O)[O-])=O)C(F)(F)C1 Cc1ccnc(CNC(C2CCC(CNC(=O)Cc3ccc(F)cc3)CC2)=O)n1 n1(CCC(N2C(CNC(c3c(Cl)cn(CC)n3)=O)CCC2)=O)cc([N+](=O)[O-])cn1 C1(NC(c2c(CC)scc2)=O)CCN(C(c2[nH]cnc2COC)=O)CC(C)(C)C1 C1(C(N2CCC(NC(c3c(SC)csc3)=O)CC2)=O)CCCC(C#N)C1 C(=O)(CCC(C)C)NC(C(=O)NC(CC(=O)OC)C1CC1)c1ccco1 c1(C(N(C)CCNC(C2CCCOC2C2CC2)=O)=O)c(Cl)ccc2ncccc12 N1(C(c2cn(C)nc2C)C(=O)NCCCCCC)CCc2ccc(OCC)cc21 CC(CCNC(=O)C(C)CNC(=O)CNC=O)C(C)(C)C N1(C(CC(=O)NC)=O)CCCC(C2(NC(c3cnc(F)c(F)c3)=O)CC2)C1 CCC(C)C(=O)C(=O)NCC#CC(=O)NCC1(C)CCCC1O c1(N2CC(CN(C(C(CC)=CC)=O)C)OCC2)nc(Cl)nc2c1ncn2C C1(C(=O)NCCOC2CCCC2)CC=CCN1C(=O)CCC1CCCOC1 N1(C(=O)CSc2ccccn2)CC2CC1CN2C(C12CC3CC1C2C3O)=O N1(C(C(C=CC)O)=O)CCOCC(C(=O)NC(c2ccc(O)nc2)C)C1 CCC(CC)CCCC(=O)N1CCC(C)(NC(=O)C(c2ccc(Cl)cc2)CO)C1 C(=O)(C1=CC2CCCC12)N1CCC(C(C)NC(c2c(N)cnn2C)=O)CC1 C1(CCC)CCCN1C(=O)CC1C(NC(c2cnn(C(C)C)n2)=O)CC1O c1(C(N2CCCC(NC(c3c(N)cn(C)n3)=O)C2)=O)cccc2c1C(=O)NC2=O C1(C(=O)NCC2(C(C)(C)C)CCN(C(C3CN(C)C3)=O)C2)CN2CCCN1CC2 C(C(C(C)C(C)C)NC(c1csc(Br)c1)=O)NC(CCOC)=O c1(C(N2CCC3(NC(C(CC)CC)=O)C(CC2)C3)=O)cnc2ccccc2c1 C(C(C)(C)C#CC(=O)NC1CC(O)C1(C)C)NC(c1nc(N(C)C)oc1)=O CC1CN(C(C2CC(F)C2)=O)CC1CCNC(=O)CCC1CCCCC1 C1(CC)CCCN(C(c2cnc(CNC(=O)C=CC(=O)N(C)C)nc2)=O)CC1 C1(NC(CCNC(C)=O)=O)CCCC(NC(=O)C(C2CC2)C2CC2)C1 Cc1coc(C)c1NC(=O)CN1CCCC1CNC(c1nc(C2CC2)oc1C)=O C1(CNC(=O)Cc2cccs2)CC2(CCC2)CN1C(C1C2CCCOC12)=O c1(OC(CC)C)cc(C(N2CCOC(CNC(=O)CC3CC3C)C2)=O)ccn1 CN1CC2CC1CN2C(=O)CC1CCCN(C(=O)CCn2ccnn2)C1 c1(OC)c(C(=O)NC2CC23CC(NC(c2ccncc2)=O)C3)cccc1Br C1(C(=O)NCC(N(C(CCC(=O)N(C)C)=O)C)C2CC2)CCCS(=O)(=O)N1 C12CC(C13CCC3)CCC(=O)N2.C(=O)(C(=O)NC1CC1)N.C(C=O)NC(C)=O C1(CNC(c2c(CC)cc[nH]2)=O)CN(C(c2ccc(F)s2)=O)CC(C(F)(F)F)O1 CCCCC(C(=O)N1CCC(C)(C(=O)NC2CN(C(C)C)C2)CC1)C(C)C N1(C(C23N(C(C4ON=C(CC)C4)=O)CCC2C3)=O)CCOCC2(CC2)C1 c1(OC)ccc(C(=O)NC(C)CNC(=O)C(C2CC2)C2CC2)c(OC)c1Cl N1(C(Cn2c(C)cnc2)=O)CCC(NC(C2CC3CC2C2CC32)=O)C2(CCC2)C1 C1(CNC(c2csc(F)c2)=O)C(CNC(C2CCS2(=O)=O)=O)C1(F)F C1(C(=O)NCCC2N(C(c3cc(C)nn3C)=O)CCC2)CC2CCCCN2C1 N1(C(C(C)OCCOCC)=O)CCC(NC(=O)CCCC(C)=O)CC(C)(C)C1 c1(SC)cccc(CC(=O)NCC23CC2CN(C(C2(F)CCOCC2)=O)C3)c1 c1(OC)ccnc(C(N2CC(NC(=O)CCC3CCCCC3)C(O)C2)=O)c1OC C(=O)(CCS(C)(=O)=O)N1CC(C(C)NC(C2CC2c2ccnn2C)=O)OCC1 c1(OC)c(C(=O)NC2CN(C(=O)C#CC3(C)CC3)CC23CC3)ccnc1Cl N1(C(CCN(C(C(CSC)O)=O)CC2CC2)=O)CCC(C)(C2CC2)C1 c1(OC)ncc(C(=O)NCC2CC(F)(F)CN2C(c2cc(C)sn2)=O)cc1C N1(C(C23CC(C4CC4C(=O)OC(C)(C)C)(C2)C3)=O)CC=C(CC2CC2)CC1 c1(C(N(CC(O)C(=O)NCC(F)(F)CC2CC2)C)=O)ccc(C2CC2)cc1 C1(CNC(CCC)(C)c2nnnn2CC)CCC2(CCCC2)C1 c1(C(C)NC(=O)C2CC2)ccc(NC(c2cn(CSC3CC3)nn2)=O)cc1 N1(C(CCCN(C(=O)OCC)C)=O)CCC(C)(C)C(CNC(C2(F)CC2C)=O)C1 C12(NC(C=CSC)=O)CCCCCC1N(C(c1ccc3ccnn3c1)=O)CC2 C=Cn1nccc1C(=O)NC(CCCNC(=O)CCSC1CC1)c1ccccc1 C1(OC)C=CCN(C(=O)OC(C)(C)C)C1.c1(C2C3(CC3)N2)nnnn1C Cn1cccc1C(=O)Nc1cccc(CNC(=O)C(c2cccc(F)c2)O)c1 CCC(COC)C(=O)N(CCCCCCNC(C1CCCCC1)=O)C C(=O)(C1CCOc2c(F)cccc21)N1CCC(NC(C2(CSC)CC2)=O)C(O)C1 CC1CCN(C(C23CCC(C2)OC3)=O)CC1CNC(c1ccncc1Cl)=O C(=O)(C1=COCC1)NCc1cc(C(=O)NCC2(CC)CCCC2)no1 N1(C(CC2(NC(C)=O)CC2)=O)CCCN(C(C2CC3CCCCC23)=O)C(C)C1 c1(C(=O)NCCN(C(C2C3CCCC23)=O)CC2CC2)coc2ccc(Br)cc12 c1(C(N2CC(C)C(NC(=O)CC3CCCOC3)C2)=O)ccc(S(N)(=O)=O)cc1F N1(C(C(C(CC)C)O)=O)CCCN(C(=O)CCCCCNC(C)=O)CC1C N1(C(C2(NC(C)=O)CCC2)=O)CCCC1C(=O)NCc1nnc(CO)s1 c1(C(N2CCC(C)(NC(C3OCC4CCCC34)=O)C2)=O)cnc2c(F)cccn12 C1(NC(c2nn(CC)c(C)c2)=O)CC(C)CN(C(=O)C(C2CCOCC2)F)C1 N1(C(C2(C)CCCO2)=O)CCC2CCC(C1)N2C(=O)C(c1ccccc1)O c1(C(N(CCCCCC)CCNC(C2CCCS2)=O)=O)ccc(OC)nc1 N1(C(CC(n2c(CC)ncc2)C)=O)CC(NC(=O)CC2(CSC)CC2)C(C)C1 c1(C(=O)NC2C(CNC(c3c(OC)cc(C)cn3)=O)C2)scc2c1CCCC2 Cc1oc(C(=O)NCC(C)NC(=O)Cn2cnc(C(F)(F)F)n2)cc1Br N1(C(c2cc(C)cc(O)c2)=O)CCC2CCN(C(c3n[nH]c(C)c3O)=O)CC2C1 c1(NC(C(N2C(CC)CCC2)CC2C=CCC2)=O)ccc(OC)cc1C c1(CCCC(=O)NC2(CNC(C3CCC(CC)C3)=O)CCC2)cc(F)ccc1F N1(C(C2C(C)C2)=O)CCC2CN(C(c3ccc4cccnc4n3)=O)CC2C1 Cc1cc(O)ncc1C(=O)NCc1cc(C(=O)N(C2CCOC2)CCF)n[nH]1 CC(C)CC(O)C(C)C(=O)NCCOC1CN(C(c2ncccc2C2CC2)=O)C1 Cc1ccn2c(=O)c(C(=O)NCC(C(C)C)NC(c3cnsc3C)=O)cnc2c1 c1(C(=O)NCCCC(C)NC(c2cc(OCC)n[nH]2)=O)sc(CO)nc1C N1(C(CCN(C)CCO)=O)CC(NC(c2ccc([N+](=O)[O-])s2)=O)CC(O)C1 N1(C(C(C)OC)=O)C2CCC1(CNC(=O)Cc1cc(C)ccc1Br)CC2 N1(C(CCC(C)OCC)=O)CCN(C(=O)Cc2ccnn2CC)C(C2CCC2)C1 N1(C(c2c(OCC)cncc2)=O)CCOC(C)(CNC(C23CCCC2C3(F)F)=O)C1 N1(C(C2(C#C)CCC2)=O)CCCC(C2CCN(C(c3ncccn3)=O)C2)C1 c1(C(=O)NC(C(C)NC(C(C)N(C)C)=O)CO)cccc2c1CCO2 C1(CNC(CCC)=O)CN(C(=O)Cn2nc(C(F)(F)F)cc2Cl)CCCO1 CC(CCCCNC(=O)CCCc1cnn[nH]1)NC(=O)CCC1CC1 C1(C(N(CC(CNC(C2(CCOC)CC2)=O)(C)C)C)=O)CC2CC(O)C(C1)C2 c1(C(=O)NCC2CCC2CF)nc2nc(C(F)(F)F)ccn2n1.C12COCC1N2 N1(C(Cn2c(C)c(Cl)cn2)=O)CCN(C(C2CCn3nnnc3C2)=O)C2CCC12 c1(OCC)ccc(C)cc1C(N1CC2CC(NC(=O)CCn3cccn3)C2C1)=O N1(C(c2c(C)n(C(C)C)cc2)=O)CC(NC(C23CCCC2C3)=O)CC(C)C1 Cc1cn2nc(C(=O)NC3CCN(C(c4sncc4C)=O)CC3F)cc2c(=O)[nH]1 CCC(N=c1nc(N2CC3OC(=O)OC3C2)c2ncn(C)c2[nH]1)c1ncc(C)[nH]1 C1(CC)C(=O)NCCN1C(=O)CCCCNC(C1OCCC1(C)C)=O c1(C(=O)NC2CCC(NC(CSCCC)=O)C2)ccc2c(c1)CC(C)(C)C2 N1(C(C(C)OCc2ccccc2)=O)CC(C2CN(C(C3CCCC34CC4)=O)C2)C1 C1(NC(c2ncc(CC)s2)=O)C(C)CCN(C(=O)CCCN2CCCC2)C1C C12(CNC(C(COC)C)=O)CCCC1N(C(c1ccnc(C(F)(F)F)n1)=O)CC2 CC(CN(C)C)CCC(=O)NCC1CC2CC1CN2C(c1c[nH]c(C(N)=O)c1)=O c1(NC2C(OC)COCC2)nccc(=NCCC2CCS(=O)(=O)CC2)[nH]1 c1(OC)c(CC(=O)NC2CC2CNC(=O)C(C)(C)CF)cccc1F c1(C(=O)NC(C)CNC(c2nncn2C)=O)ccc2c(c1O)CCCC2 c1(SC)cc(C(N2CCC(NC(c3cncc(N)c3)=O)C2)=O)ccc1Br C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC2C(NC(C3CCCN(CCC)C3)=O)C(C2)C1 C(=O)(C1=CCCCC1C)N(CC(=O)NCC(C)S(C)(=O)=O)CC N1(C(=O)OC(C)(C)C)CCC1CNC(C1CC(C(C)(F)F)C1)=O c1(C(=O)NC(C2CCCC2)CNC(CC(=O)NCC)=O)cscc1S(C)(=O)=O C(=O)(CCCC(=O)OCC)NC1(C(N2CC(=CCC)C2)=O)CC(F)C1 CCC(CC)CCCC(=O)NCC1CC2(CO1)CN(C(=O)CN(C1CCCC1)C)C2 C1(C(=O)NCC(CNC(c2c(C)nccn2)=O)F)CC2C(C1)C2(C)C c1cc(CSCCCNC(C(C)OCCOCC)=O)c(C(=O)OC)c(Cl)c1.OC Cc1ccccc1C(C)CC(=O)NCCNC(c1c(Cl)n[nH]c1C)=O CCC(C)CCCCC(=O)NCC(C)NC(C1(C(F)(F)F)CCCCO1)=O c1(C(=O)NC(C2CCCN2C(=O)CC2CC2)C)ccc(Br)cc1 c1(CC)ccccc1C(CNC(=O)C(C)CCOC)NC(=O)CC(C)(C)C c1(C(N2CCCC(CN(C(=O)CC3C=CCC3)C)C2)=O)ccc(=O)n(CCO)c1 N1(C(c2cc(C)c(Cl)cn2)=O)CC(NC(C23CSCC2C3)=O)CC12CCCCC2 c1(OCCOC)ccc(C(=O)NCCC(O)CNC(C2CC3CC3C2)=O)c(Cl)c1 C1(SCc2nc(C(C(C)(F)F)NC(=O)OC(C)(C)C)on2)CCc2nnnn2C1 N1(CC(=O)OC)CCCN(C(c2cnc(O)cc2C)C(=O)NCC2(C)CC2)CC1 N1(C(Cc2ncn(C)c2)=O)CC2(C(=O)NC3CCC4CC34)CC1CCO2 c1(NC(C2OCCN(Cc3ccc(C)c(O)c3)C2)=O)c(F)cc(Br)cc1F CN1CCCC1CC(=O)NC(C)(CNC(=O)C=Cc1ncc[nH]1)C1CCC1 C(=O)(C1CNC(=O)c2ccccc21)NC1CN(C(c2cnn(C(C)C)c2N)=O)C1 C1(CNC(C(C2CCCC2)OCC)=O)CC2CCC1N2C(=O)CCCCC#N C(=O)(C1CSc2ccccc21)N(CC(C)O)CCNC(c1ncccc1N)=O CC(C)(C)C(=O)C(=O)N1CC2C(CNC(c3cccc(N4CCCC4)n3)=O)C2C1 C1(CNC(C2CC(CCNC(C3CCSC3)=O)C2)=O)CCCC(CO)C1 N1(C(C2(C)CCCN2C(C23CC(C#N)(C2)C3)=O)=O)CCC2(CCCC2)C1 N1(C(c2cc(OC)cc(Cl)c2)=O)CC2CCN(C(c3cc(F)cc(I)c3)=O)C2C1 N1(C(C(C2CN(C(C(CC)O)=O)C2)O)=O)CCC(O)(CC(C)C)C1 C12(NC(C3C(CNC(CCCNC(=O)OC)=O)OCC3)=O)CCC(CO)(CC1)C2 C(C(F)(F)CCC(=O)NC1CCC1)n1cc(C(C)NC(CCOC)=O)nn1 Cc1ocnc1CC(=O)NC1CC(CCNC(=O)C(n2ccc(Br)n2)C)C1 C1(C(N2CC(C(N)=O)(CNC(c3n(CC)ccc3)=O)C2)=O)NC(=O)OC1C C1(NC(c2cc[nH]c2)=O)CN(C(C2CC3CC2C3)=O)CC12CCC2 C1(NC(C2C=CCC2)=O)CC2CCC(C1)N2C(=O)C(c1ccc(F)c(F)c1)(F)F C=CCC(CC)C(=O)NCCCC1CCCN1C(C1CCC(C)(C)CC1)=O O=C(C1=CS(=O)CCC1)NC1CC2(C1)CC(NC(C1CCn3ncnc3C1)=O)C2 C1(F)(CNC(C(CC)n2cccn2)=O)CCC(CNC(=O)C=CC2CCOC2)CC1 Cc1cn2c(=O)c(C(=O)NC(C)CNC(c3ccn4ncccc34)=O)cnc2s1 CCC(CN(C)C)CC(=O)NCC1CCCCN(C(=O)C=Cc2cn[nH]c2)C1 Cc1nonc1C(=O)NOCC(=O)NCc1occc1C1CC1 c1(C(=O)NC(C(C(C)C)C)CNC(=O)CSC(C)(C)C)ncnc2ccsc12 c1(CNC(C(C)OC)=O)cncc(C(N2CCC(n3cnnn3)C2)=O)c1 Cc1coc(C)c1C=CC(=O)NCCC1CCC(NC(c2c(Cl)n[nH]c2C)=O)C1 c1(NC(C)=O)sc(Cl)cc1NC1CCN(C(=O)CN(C)C(C)=O)CC1 c1(C(N(C)CCNC(c2cc(Cl)c([N+](=O)[O-])[nH]2)=O)=O)cc2n(c1)CCCNC2=O C=CCCCCCCC(=O)N(C(C)C(=O)NOCCC(C)O)CCN(C)C c1(C(c2nnnn2C(C)C)NCCCCSC)c(C)cnn1COC c1(-c2onc(Cc3ccc(Cl)cc3)n2)ccc2sccc2c1 N1(CC)CCN(c2ccc(NC(=O)CC3CCCCCO3)cc2)CC1 C1(C(N2CC(C)C(NC(=O)C3=CCCOC3)C2)=O)CC2(CCCC2)CO1 C(=O)(C(CC)(CC)Nc1ccccc1)NCC1CCN(C(C(C#C)(C)C)=O)CC1 C1(NC(C(CC=C)OC)=O)CCCN(C(=O)Cc2ccon2)C1CC N1(CCC)C(=O)CCC1C(=O)N(C(CNC(c1scnc1Cl)=O)C1CC1)C Cc1nc(C)n(CC(=O)NC2CCC(C(F)C(=O)NCc3cnn(C)c3C)C2)n1 n1(CCOC)cccc(C(=O)NCC2CC(C)N(C(=O)C(C(C)C)SC)C2)c1=O C(=O)(CC(CC(C)C)NC(=O)CCN1CCCC1=O)N1CC(c2nc(C)on2)C1 C1(C(C)C)(CO)CCN(C(=O)C(C2CCCC2)NC(c2cc[nH]c(=N)n2)=O)C1 CCCC(C(=O)NCC1(CNC(C2(CO)CCCO2)=O)CC1(F)F)NC(N)=O C(C(=O)NCCCF)(C1=NOC2CC12)N(C)Cc1cccc(C(F)(F)F)c1 N1(C(C2(CNC(C3CCC4(CCC4)C3)=O)CCCO2)=O)CC2CC3CC2C1C3 CC1CN(C(=O)CC(CC2CC2)NC(=O)COC(C)(C)C)CCO1 C(CC(CNC(c1cnco1)=O)NC(=O)C(C)CSCc1ccccc1)OC CC1(C(=O)NCCN2CCN(C(c3c[nH]c(=S)cn3)=O)CC2)CCNC1=O c1(C(N(C)Cc2cn(-c3nonc3C(=O)O)nn2)=O)nccc2ccccc12 Cc1cc(C)c(NC(=O)NCCS(=O)(=O)C2CC2)c(C)c1 N1(C(C#CC(C)C)=O)CCC(N(C(=O)CCSc2nccn2C)C)C2(CC2)C1 N1(C(C2CC3(C(OC)CC3)C2)=O)C2CCC1CC(NC(=O)Cc1nonc1C)C2 Cc1ccc(-c2cn(C3CC(C(=O)NC4CC(CN5CCCC5)C4)C3)nn2)nc1 N1(C(CN2CCC(C)(O)C2)=O)CCCC2(CCCN2C(=O)Cc2cn[nH]c2)C1 c1(NC2CN(C(CC3(C)CC3(Cl)Cl)=O)CC23CCC3)cc(=O)n2ccccc2n1 CC1CCC(CNC(C2NC(=O)OC2C)=O)CN1C(c1cocn1)=O n1(CCC(=O)NCCN(c2nnc(C3CC3)o2)CC)ccc(O)nc1=O C1(C(=O)NC)CC(O)CN1C(=O)C(C1CCCN(C(=O)CCCCN(C)C)C1)C CC1CC(Nc2nccc(-n3ccnc3)n2)CCN1C(=O)CC1CCC(O)C1 C1(CC=C)(C(=O)N(C)CC2CCCC3CC23)CCN(C(C2CC(N=[N+]=[N-])C2)=O)C1 C1(CNC(c2cc(COC)sc2)=O)CCC(NC(c2cc(F)n(C)n2)=O)CC1 CC1(C)CC(NC(=O)C2=CCSC2)CN1C(c1cnn(C2CC2(F)F)c1)=O CC1(C)CC(CC(N2CCOC(CNCC3CC34CC4)C2)=O)CO1 C1(C(=O)NCC2OCCN(C(COCCCN(C)C)=O)C2)CC(C(C)(C)C)=NO1 O=C1CCC(CCC(N2CC(O)(CNC(=O)CC3CSC3)C2)=O)N1 Cc1cc(C)c(NC(=O)C(CCC2CCC2)N(C)CCN2CCOCC2)c(C)c1 c1(CC)cc(C(N2CCC(CNC(c3nnccc3C)=O)CC2C)=O)c(C)nn1 N1(C(c2c(C)ccs2)=O)CCC(NC(C2CCCN(C(N)=O)C2)=O)CC(C)(C)C1 CCC(C)CC(C)C(=O)NC1(CC=CC(=O)NC2CC3CC2CC32CC2)CCC1 N1(C(C=CC(=O)N(C)C)=O)CC23CCCC2(C1)CN(C(c1c(C)coc1C)=O)C3 c1(C(c2n(CCSC)nnn2)NCC2(C)COC2)cc(SC)ccc1Br N1(C(c2ccc(C)c(F)c2)=O)CC(NC(C2CC(F)C2)=O)CC12CCCCCC2 Cc1ccc2oc(C(N3CC4CC(C3)C4(F)F)C(=O)NCC3CC3)cc2c1 CCC(C)(CCNC(=O)C(C)C(F)F)NC(C1SCCS1)=O c1(C(=O)NCCC(C)F)cccc(-n2cc(CNC(c3ccnnc3)=O)nn2)c1 c1(C(=O)NCC(C(C)C)NC(Cn2ccc(C)n2)=O)cn(C)c(C)n1 C1(SC)CN(C(=O)C(F)(F)c2cn[nH]c2)CC1NC(=O)C(N)=O C(=O)(CC(F)(F)c1ccc(Br)nc1)NC(C)CCN1CCCC1=O Cc1ccc(C(N2CCCCCC2C(=O)NCC(C)(C)C2CC2)=O)c(F)c1 c1(C(=O)NC2(C)CN(C(c3cncc(SCC)n3)=O)C2)nc(C)ccc1F C1(CC(=O)NC(CNC(C(CCOC)C)=O)(C)C)CSc2ccccc2O1 C1(O)(CN(C)C)CCN(C(=O)CCNCC(C)(C)n2ccnc2)CC1 c1(OCC(N2CC(CCNC(C(CC)COC)=O)OCC2)=O)ccc(Cl)cc1Cl N1(C(C(c2cccnc2)C)=O)CC2CCC(C1)N2C(c1cnc(O)n(C)c1=O)=O C1(CNC(COC)=O)CCC(C)N(C(=O)CC(C)n2cccn2)C1 N1(CC(=O)NCCCn2cc(C(c3ccccn3)O)nn2)CCCS1(=O)=O Cc1c(C(=O)NC2CCNCC2C2CC2)sc2cc(Cl)ccc12 c1(C(N2CC=CC2)C(=O)NC2CCC(CNC(=O)CO)C2)cc(Cl)cc(Cl)c1 Cn1cc(OCC(=O)NC2(CO)CN(C(C3CCCN3CC3CC3)=O)C2)cn1 N1(C(CNC(=O)NC)=O)CCCCC(CCC(=O)NC(c2ncc[nH]2)C)C1 Cc1ccc(C(=O)NCC2CN(C(=O)Cc3cc[nH]c3)CCN2C)cc1C Cn1cnc2sc(C(N3CC(F)(CNC(C4CCCN4C(N)=O)=O)C3)=O)cc12 C(=O)(CCCCCN(C)C)NC1CC(N(C(C2(OCC)CCC2)=O)C)C1 N1(C(=O)Cc2cnns2)CC(NC(C2(CO)CCCO2)=O)CC(F)(F)C1 C1(CNC(c2c(C)ocn2)=O)CC(C)(C)CN1C(C12CCCCC1C2)=O C1(C(N(C2CN(C(=O)C(C)(O)C(F)(F)F)CC2(C)C)C)=O)CCC2(CCC2)CC1 C1(O)(CNC(CN2C(C)CC2)=O)CCCN(C(=O)CSCc2ccc(F)cc2)C1 Cc1cc(C(N2CCOC(C3(C)CC3)C2)C(=O)NC2CC2)cc(C)c1 c1(C(=O)NC2CC2CNC(c2cc(Cl)ccn2)=O)ccc(F)c(C2CCC2)c1 C(=O)(CC(C)(C)C(F)(F)F)NC1C(CNC(CN2CC(C)(C)C2)=O)CCC1 c1(C(=O)NCC2N(C(CCOCCOC)=O)CCN(C)C2)ccccc1N=[N+]=[N-] C12CCC(CC1)Cc1cn(nn1)C2.CC1CCC(CC(=O)NCN)C1 c1(C2CCN(C(c3cccc(CCC)c3)=O)C2)ccc(OC)c(OC)c1 c1(CN(C(=O)NC(c2noc(C(F)(F)F)n2)C)C)nnn(C)n1 CC(C)CC(O)C(C)C(=O)NCC1(NC(=O)C=CC2CCOCC2)CCC1 c1(C(N2CC(NC(C(C)CC3CCCCC3)=O)C(O)C2)=O)cccc(F)c1Cl C(=O)(CCCCCN=[N+]=[N-])N1C(C(=O)NC(C=C)(C)C)CN(C)CC1 N1(C(C(COC(C)C)NC(=O)CC(C)CN(C)C)=O)CCC2(CCCCC2)C1 Cc1cc(C(N2CC(C(=O)NCC3(C)NC(=O)NC3=O)C3(CC3)C2)=O)c(O)nn1 C1(CNC(=NCCC=C)NCc2ncccc2Cl)COc2ccccc2O1 N1(C(Cc2nnc(C)o2)=O)CC2CC1C2NC(c1ccsc1Cl)=O c1(NC(CC2(C=C)CN(C(=O)CCCCCCC)C2)=O)ccc2ccncc2c1 c1(C(=O)NCC2C3CN(C(C(C4CC4)OCC)=O)CC32)cc(OC)cnc1F c1(C(C)=O)ccc(-c2csc(C(=O)Nc3cc(O)nc(Cl)n3)n2)cc1F N1(C(c2cc(OCC)n[nH]2)=O)CCCCC(NC(C2CC2(C)C(F)(F)F)=O)C1 Cc1cccc(C(O)C(=O)NCCCN(C(c2ccc(Cl)s2)=O)C2CC2)c1 c1(CC2CN(C(C(C(C)C)Cc3ccccc3)=O)CC2(C)C)cccc2cc[nH]c12 c1(CC(N2CC(C)C(N(C(=O)C3=CCCSC3)C)CC2)=O)ccn2cncc2c1 C12(CNc3cnc(SC)nc3C)COCCN1C(=O)OC2 c1(C(N2CCC(CCNC(C3NC(=O)OC3)=O)C2)=O)cccc2c1COCCN2 c1(C(=O)NCC2C(NC(c3n(C)nc(C4CCC4)c3)=O)CC2)cn(C)c(=O)n1C N#Cc1ccc(NNC(=O)NC(c2cccc(F)c2)CO)cc1F c1(NC(N(C(C(=O)OC)C2CC2)C)=O)nc(CCl)c(C)cc1C#N c1(C(N(CC(CC)NC(=O)C(COC)OC)C)=O)ccccc1Br Cc1sc2ncnc(NC(CN(C(=O)CC(C)C(F)F)C3CCCC3)CO)c2c1C N1(C(CCOC(C)C)=O)CCN(C(c2ccc(C(C)(F)F)nc2)=O)C(C(F)F)C1 Nc1cccc(F)c1C1CC1N1CCC(N2CCC(c3ccccc3)CC2)CC1 C1(CC)(NC(c2ccc(C3CC3(F)F)cc2)=O)CCN(C(=O)C(O)C2CC2)CC1 Cc1ccc(C(=O)NC23CC(NC(=O)CC4CC(N(C)C)C4)(C2)C3)c(F)c1F c1(C(=O)NC(CC)CNC(=O)C(C)C2CCCC2)cc2cc(Cl)ccc2[nH]1 CCCC(C(=O)N1CC=CC1CNC(=O)Cn1cc(C)cn1)N(C)C C1(NC(C(CC(C)C)OC)=O)CCC2CN(c3ccnc(CO)n3)CC2C1 N1(C(Cc2c(C)ccnc2)=O)CCN(C(c2cccnn2)=O)C2CCCCC12 CC1CN(C(=O)Cn2cccnc2=O)CC1CNC(=O)CCc1ccon1 c1(-c2scc(C(=O)NC3CC(CNC(c4cc(O)ns4)=O)C3)n2)cccc(F)c1 Cc1cc(C#N)cnc1C(=O)N(CC(C)(C)C(=O)NCC1CCN(C)CC1)C C=Cc1cncc(C(N2CC3CC2C3C(N2CCCCCC2CC)=O)=O)c1 C(CN=c1nc(N2CCC3(CCOC3)C2)c2sccc2[nH]1)NC(C1CCC1)=O C1(OC)(CNC(=O)C(C)S(N)(=O)=O)CCN(C(=O)Cc2ccnc(C)c2)CC1 C(=O)(CCC(CC)OC)NC(CCC)CNC(c1cnn(C)n1)=O C(CCC)(CCCNC(=O)C1=COCCO1)NC(C(C)OCC#C)=O Nc1ncccc1CC(N1CCCC(NC(=O)CC2CNC(=O)C2)C1)=O C(CCCCC(=O)NCC1CC2CCC1C2)NC(C(F)=CCC)=O N1(C(CCSCCC)=O)CCC(NC(c2ccnc(NC(C)C)c2)=O)C1C C1(CC(=O)NC2CN(C(C(C(C)C)O)=O)CC2(C)C)CC(C)(C)OC(C)(C)C1 c1(C(=O)NCC2(F)CC(NC(C=C(C)Cl)=O)C2)ccc2c(c1)NC(=O)C2(C)C C1(CC(=O)NCCCCNC(C2(C)C(C)(C)C2)=O)COCC1(C)C c1(C(N2C(CNC(c3c(CC)occ3)=O)COCC2)=O)cc(F)c(N)cc1OC c1(C(N2CC(C(=O)Nc3c(C#N)cc(CC)s3)C2)=O)ccc([N+](=O)[O-])c(C)c1 c1(OC)ccc(Cl)c(C(=O)NC2CCC2NC(=O)CC2COCCN2C)c1 c1(OC)nc(C(=O)NC(C)CC(C)NC(=O)C=Cc2ncc[nH]2)ncc1F c1(NC(=O)C(N2CC3CC(F)CC3C2)=O)cccc(S(=O)(=O)NC2CCCC2)c1 c1(C(=O)NC2(C)CCN(C(C3(c4ccccc4)CC3)=O)C2)[nH]nc2ncccc12 C(=O)(C1=CCCC(C)(C)C1)NCC(C(C)C)NC(c1cc(CO)n(C)n1)=O c1(C(=O)NCC23CC(NC(C4CC5CC5C4)=O)(CCO2)C3)cc2cccnc2s1 C1(C(=O)NCC(N(OC)C)=O)(NC(=O)CCOC(C)=O)CCC(C)(C)C1 c1(C(=O)NC(CC)(CNC(=O)C=Cc2nccs2)CC)cc2oc(C)cc2[nH]1 CC(C)CCOC(C)C(=O)NCC(C1CC1)NC(C12CC(C1)C2)=O c1(C(=O)NC(C2N(C(C(C)SCC)=O)CCC2)(C)C)cnc(O)c(C(F)(F)F)c1 C1(NC(C(C)Cc2ccccc2)=O)CC(C)N(C(=O)C(C)(C)c2nccs2)C1 C(=O)(C1CCCc2ccccc21)NCC1CC(NC(c2csc(Cl)n2)=O)C1 c1(C(N2CCC3CN(C(C(COCC)C)=O)CC32)=O)coc2ccc(OC)cc12 c1(SC)cc(C(=O)N(C)CCN(C(=O)Cc2cnn(C)c2C)C(C)C)c(C)o1 C1(C(=O)NCC2CCC(C(=O)NCCN(CCC)C(C)C)C2)CCOCC1C C(CCCCC(=O)N(CC(C)(C)O)C)N(C(c1c(OC)scc1)=O)C CC(C)C(CC(=O)NCc1nc(CO)n[nH]1)NC(=O)CCC(C)(C)F c1(C(N2CCCC(C(=O)NCCOC)C2)C(=O)NC(CC)C)sc(=O)n(C)c1Cl N1(C(CNC(C(CC)C)=O)=O)CC2CCC(N(C)C(C3CCN3CC)=O)C2C1 C12(C(N(CCCCN(C(C(CC)NC(N)=O)=O)C)C)=O)CCCN(CC1)C2 C1(C(C2(F)CC(CO)C2)NC(=O)CNC(=O)CCSC2CC2)CCCCO1 C=CCC(CNC(C1(C)CC2(CCC2)C1)=O)C(=O)N(c1cnn(CC)c1)C c1(OC)cc(CC(=O)NC(C)Cn2cc(C3(O)CCCCC3)nn2)ccc1Cl Cn1ccc2c(-c3nc(CCN(C)C)nn3C3CCS(=O)(=O)C3)ccnc12 c1(C(c2n(CC)nnn2)NCCCn2cc(CO)nn2)cnc2n1CCC2 c1(CCC(=O)NC(c2cn(CC3CCOC3)nn2)CCC)cccc(I)c1 N1(C(C2CC(=C)C2)=O)CCN(C(=O)CNS(=O)(=O)CC)C(CCC)C1 c1(C(=O)NC2CC(NC(c3ccc(C(F)(F)F)[nH]3)=O)C2)ncoc1Br c1(CC)ccc(C#CC(=O)NCc2ccc([Si](C)(C)C)s2)cc1 Cc1cc(NC(=O)NC(C)C(c2cccc(F)c2)O)cc(Br)c1 CC(C)(CO)C(=O)NC1CCN(C(=O)CCc2ccsc2Br)C1 CC1(CC(=O)NC2CC(NC(=O)CC3CCCOC3)C2)CCCCC1 CC1CCN(C(=O)CCOC2CCC2)CCN1C(c1coc(C(F)F)c1)=O n1(CC)c(CNC(C2(CO)CCN(C(C3C4COCC34)=O)C2)=O)nnc1O Cc1nc2cc(CC(N3CC(CN=c4ncc(I)c[nH]4)C(C)C3)=O)ccc2o1 CCCC(C(=O)NC12CC(CNC(C3(C)CCCOC3)=O)(C1)C2)N(C)C C(N=c1[nH]c2ccc(O)cc2s1)C1C(NC(c2cnc(C3CC3)[nH]2)=O)CCC1 N1(Cc2ccc(-c3c[nH]c(=N)s3)cc2)CCCC2(COCCN2)C1 C1(C(=O)NCC(=C)Br)CCC(CNC(=O)CCc2cnoc2)C1 c1(CC)ccnc(CNC(C2C3CN(C(c4cnncc4C)=O)CC23)=O)c1 N1(C(CC(CC)C)=O)CCN(C(=O)COCCF)CC1CF c1(C(=O)NCCCC2CCCCN2C(c2ccc(Cl)cn2)=O)csc2nnsc12 CCCC(=O)C(=O)N1CCCC(C(=O)Nc2onc(C)c2C)C1 c1(COC)nc(C)cc(=NCCCC(C)NC(=O)Cc2cccc(F)c2)[nH]1 C1(O)(CC#N)CCN(C(c2cn(C3CC3)cn2)C(=O)NCCCC2CC2)C1 C1(CNC(CNC(C)=O)=O)CN(C(c2ccc(-n3nnnc3C)cc2)=O)C2CC12 Cc1nnc2n1C(C(=O)N1CCN(C(=O)C(C3CC3)C3CC3)CCC1C)CC2 Cc1noc(C)c1CCNC(C1(NC(=O)CCc2nncn2C)CC1C)=O CC(CN(C)C)CCC(=O)NCCCC1CCCN1C(=O)COC1CCC1 C1(N(C(CCC2C(C)(C)C2)=O)CCF)CCCN(C(c2c[nH]c(=N)s2)=O)C1 C1(CCC(=O)NC(c2cn(C)nc2)C(=O)NCCCC2CCC2)CC(C)(C)CO1 C(=O)(C(F)(F)C(F)F)N1CC(CN(C(=O)COCC2CCOCC2)C)OCC1 Cc1cccc(C(=O)NC(C)CC(C)NC(C2CCC=CCC2)=O)c1[N+](=O)[O-] C=CC(CCC)CC(=O)N(CCC(=O)Nc1ccc(O)cc1CC)CCO c1(C(N2CC(NC(C3N(CC)CCOC3)=O)C(C(F)F)C2)=O)nn(C)c(C)c1Cl c1(OC)cc([N+](=O)[O-])ccc1C(N1CC2CCN(C(=O)CC3(C)CC3)CC2C1)=O N(C1CCCn2ccnc21)C(C(=O)Nc1ccc(C(=O)OC)cc1N(C)C)=O C1(C(=O)NC2CCCN(C(CCC(=O)NCC)=O)C2)CCCC2CCCN12 C1(C(N(C)CC2N(C(C(CCCC)O)=O)CCC2)=O)CCN2CCOCC12 c1(NCC(=C)Br)nc[nH]c(=NCc2ccccc2C(C)C)c1C CCCCCC(O)CC(=O)N1CC2OCC(NC(=O)CC(C)O)C2C1 N1(C(C2C=C(C)CS2)=O)CC2(C(N3CCC4(CSC4)C3)=O)CC1CCO2 C1(C)(NC(C(C2CC2)OC)=O)CCCN(C(c2cc(C(F)F)[nH]n2)=O)C1 c1(CC)ccc(C(=O)NCCCN(C(c2occc2C)=O)C2CC2)c(C)n1 c1(C(N2CCCC(N(C(c3n(CC)ccn3)=O)C)C2)=O)ccc(O)cc1C c1(CNC(C(CC)C)=O)cccc2c1CN(C(C1(C)CC=CCC1)=O)C2 c1(OC)cc(C(=O)NC2CC(CO)N(C(c3cc(O)n(C)n3)=O)C2)c(Cl)cn1 c1(C(=O)NCCCN(C(=O)CCCCN(C)C)CC)ccccc1[N+](=O)[O-] c1(C(N2CC(n3cc(C(CC)O)nn3)C(C)C2)=O)c(F)ccc2c1OCO2 c1(CN2CCC(NC(=O)Cc3ccccc3O)C(O)C2)c(Cl)cc(O)cc1Cl N1(C(c2ccc(C#C)cn2)=O)CC2(CCCC2NC(C2(CCF)CC2)=O)C1 c1(OCC)ccc(CC(N2CCSCC2CCNC(c2cnns2)=O)=O)nc1 C1(CNC(CC(CC)SC)=O)CC2CCC1N2C(C12CC(F)(C1)C2)=O N1(C(CC2(OC)CCC2)=O)CCC(C)C1CNC(=O)CNC(=O)Cn1cncn1 C1(C(=O)NCCCN(C(C(COC)(C)O)=O)C)CCOCC12CCCC2 C1(C(=O)NCn2ncc(C(C)N(C)C)c2)CCC2CN(C(=O)OC(C)(C)C)CC2O1 C(=O)(CCS(C)(=O)=O)NC1(CC=C)CCN(C(C2CCCC(C)C2)=O)C1 c1(C(N2CCC(C)(CNC(CC=CC=C)=O)C2)=O)ccc2c(c1O)CCCC2 c1(OC2CCN(C(c3c(CC)cccc3)=O)C2)cc(C(N)=O)ccc1OC N1(C(c2cccc(C)c2)=O)CCN(C(=O)Cn2nnnc2C2CC2)CC(CO)C1 Cc1cc(C)c(C(N2CC3(NC(C4CC5CC5C4)=O)CCC2CC3)=O)c(C)n1 Cc1ncncc1CC1(c2ccc(-c3cccs3)s2)CC1.C12CC(F)CN1C2=O C1(C(=O)NC(C)(C)CC=CC(=O)NC2CCCC2C(C)(C)C)(OC)CCOCC1 CN=c1ccc(C(N2CCC(O)(CNC(=O)CC(C)SCC(F)(F)F)C2)=O)c[nH]1 C1(NC(CC)=O)CCN(C(C2(CCN3CCCC3)CCCCC2)=O)CC12CCC2 C1(CNC(CC(C)C2CC2)=O)CCC12CCN(C(c1ccc[nH]1)=O)CC2 c1(CC)ncc(C(=O)NCCCC(C)NC(=O)C(F)(F)c2cnn(C)c2)o1 N1(C(c2n(C)ncc2Br)C(=O)NC2CCOCC2)CC23CCCC2(C1)C(=O)NC3=O C1(CO)CCC2(CCN(Cc3ccccc3Oc3cccc(Cl)c3Cl)C2)C1 Cc1ncc(C)c(NC(CNC(=O)CCn2cc([N+](=O)[O-])cn2)C(C)C(C)C)n1 C(=O)(C(CO)C(F)(F)F)N1CCCN(C(Cc2c(C)n(C)nc2)=O)CC1 c1(C(=O)NCc2oc(C)c(C(N3CC(c4nncs4)C3)=O)n2)cc(O)ccc1F c1(C(=O)NC2C(NC(C(C)OCC#C)=O)CCC2)cnn2c(=O)cc[nH]c12 C(C1(C)CC(=O)Nc2ccccc21)N(C1CCSC1)C C(CO)(C(=O)NC1CC(F)(CNC(=O)CCn2cc(Cl)cn2)C1)N(C)C CC(CCNC(C1C(C)C1C)=O)NC(C1CC1c1ccsc1)=O C1(C)(COC)CC1C(=O)NCC1(C(=O)NC2CC(SC)C2)CC1 CC(CC(F)F)C(=O)N1C2CCC(C2)C1CNC(c1cnn(CC2CC2)c1)=O C12(CNC(CCCCSC)=O)CCCCC1CN(C(=O)CCOC1CC1)C2 N1(C(C2C(C(=O)OC)C2)=O)CCCC1CN(C)C(C1(F)CC1C)=O c1(C(=O)NC2C(C)CN(C(C3CC(F)(CO)C3)=O)C2)cnc(N)c(Br)c1 c1(NCCS(CC)=O)ncc(S(=O)(=O)N2C3CCC2CC2(CC2)C3)cc1Cl C(C(C)(CC(C)C)NC(=O)CCn1cnccc1=O)NC(C=NOC)=O c1(C(N(C(C)CNC(=O)C=CC2CCOCC2)CC)=O)ccnnc1C C1(C(=O)NCCC=C=C)CC(C)CN(C(=O)CSc2nc[nH]n2)C1 N1(C(C(CCSC)O)=O)Cc2ccnn2CC(NC(=O)Cc2ccccc2C)C1 c1(CCC(N2CCC(O)(c3cn(CC(=O)OC)nn3)C2)=O)cc(F)ccc1Br CC1CC(C(=O)NCCN(C(=O)CC2CCC(C)(C)O2)C(N)=O)CCO1 CCC(C)CCCC(=O)NCC1CC(O)CN1C(c1nccc(Cl)c1F)=O N1(C(CCN(C(=O)CSC(F)F)CC#C)=O)CCC(C(C)(C)O)CC1 c1(NS(C2C(c3cccc(OC)c3)CCC2)(=O)=O)cc(F)c(Cl)c(F)c1 c1(C(=O)NCC(CO)NC(C2(COC)CC2)=O)csc2cc(Cl)ccc12 Cc1cccnc1C(N1CC(NC(c2ccc(-c3cc[nH]n3)s2)=O)C2CC12)=O C1(NC(CC(C)(C)O)=O)CC2CN(C(c3cnc(Cl)s3)=O)CCN2C1=O N1(C(CCc2c(C(=O)O)ccc(Br)c2)=O)CCn2c(CC(F)(F)F)nnc2C1 C12(CNC(=O)CC=CC(=O)NCCOc3ncccn3)CCCCC1C2 C=CCCCCC(=O)N1CC(CNC(=O)C(C)(C)c2ccsc2)C2(CC2)C1 C12(CNC(C3(NC(N)=O)CC3)=O)CCCC1CCN2C(c1cnc(C(F)F)s1)=O N1(C(C(c2cccc(N)c2)(C)C)=O)CCC2(CCCN2C(C2CCCC2)=O)CC1 N1(CC(=C)Br)CCN(C2CCN(C(C3CCCCN3C(C)C)=O)C2)CC1 N1(Cc2c(NCC)c(F)cc(Br)c2)CCN(S(=O)(=O)NCCN(C)C)CC1 N1(C(c2cc(OC)no2)=O)CCC2C(C1)CN2C(C1CCN(CC(F)(F)F)C1)=O N1(C(C2CCCN(C)C2)=O)CCN2CCN(C(C3CC4CC4C3)=O)CC2C1 C12(CNC(c3ccc(C)nc3O)=O)CCCC1N(C(c1cccnc1C)=O)CC2 C(=O)(C1CCc2cccnc21)C(=O)CCn1ccc2cccnc12.C1(N)CNC1 C1(CNC(c2n(CCC)ccc2)=O)CCC2CN(C(=O)Cc3ncoc3C)CC12 c1(C(=O)NCCN(C2CC2)C2CC2)ccc(CO)c(F)c1.C(=O)(CCCc1cccs1)N C1(NC(c2c(CC)ccs2)=O)CCC(N(C)C(c2cnc(Cl)n2C)=O)CC1 c1(CNC(C(C)OCCCC)=O)nc2c(s1)CN(C(=O)Cc1c[nH]nc1C)CC2 N1(C(c2cccc(C)c2)=O)CC2C3CCC(C2C1)N(C(=O)CN1CCCC1=O)C3 Cc1ccc(C(=O)N(C2CCCN(C(C3CC3(F)F)=O)C2)CCF)c(C)n1 N1(C(c2c(CC)con2)=O)CC(NC(c2coc(C)c2)=O)C(C)C1 N1(C(c2cnc(CC)s2)=O)CC(CNC(=O)CCc2ccoc2)C(O)C1 c1(C(=O)NCCN(CCC)C(c2ccc(OC)c(F)c2)=O)nc(C)c(C)nc1C c1(NC)cc(C(=O)NCC(O)CNC(c2c(C)cccc2C)=O)cc(Cl)n1 C=C(C)CC(C(=O)N1CCN(C(C)=O)C(C)C1)NC(c1ncccn1)=O CC1(C)CCCC(C(=O)NCC2COCCN(C(C3(C(F)F)CCCO3)=O)C2)C1 C12CCCN(C1)C2.CC(C)(C(=O)O)NS(C)(=O)=O.c12cn(nn1)C2.c1ccncc1 c1(C(=O)NCCC(C)NC(c2cc(C(C)=O)c(C)o2)=O)ccc2c(c1)CCCS2 N1(C(c2c(C)nn(CCO)c2)=O)CC(NC(=O)Cc2c(Cl)cnn2C)CC(C)C1 c1(C(=O)NCCCC2CCCN2C(C2(C(F)(F)F)CCC2)=O)ncc(F)cn1 CC(C)CC(C)(C(=O)NCC1CC(C(C)(C)C)=NO1)NC(=O)OC(C)(C)C C(C(=O)N=c1cc[nH]cc1)C1CC2(N(C(C(C)(C)c3cccs3)=O)CC2)C1 Oc1ccc(-c2nc(C3CCC3)nn2-c2ccc(CN3CCOCC3)cc2)nn1 N1(CCNC(c2c(CC)nc(C)[nH]2)=O)C(=O)NC(c2ccccc2)(C2CC2)C1=O C#Cc1ccc(CC(=O)NCC23CCC(NC(=O)C(O)CCCC)(CO2)C3)cc1 N1(C(CC(CC)C2CC2)=O)CCC(C(=O)N(CC(C)C#N)C)C(C)(C)C1 CC1CN(C(C2(CO)CC2)=O)CC1CCNC(=O)CN1CC(=O)NC1=O C(=O)(C1=C(C#N)CCC1)NCC(=O)NCC(=O)NCC1(CC)CC(C)(C)C1 N1(S(CC2CCC(C)O2)(=O)=O)CCc2c(ncn2C2CCCCC2)C1 Cc1ccc2c(C(N3CCCC4(C3)CN(C(C3COC(=O)O3)=O)C4)=O)c[nH]c2c1 CC(CC(=O)N(C)CCc1ncon1)C(C)(C)NC(=O)CCCC#N C1(NC(c2c(Cl)ccc(C)c2)=O)CC2CC(C1)N(C(C1CCCN1C=O)=O)C2 CC1=NS(=O)(=O)N(C)C=C1C(=O)NCC1(NC(=O)C=C2CCC(C)(C)CC2)CC1 C1(C(N2CC(C3N(C(C4COCCN4C)=O)CCC3)(O)C2)=O)(CSC)CC(F)(F)C1 Cc1cc(C(=O)NCC(C)(C(C)C)NC(c2cc(C(C)C)no2)=O)c(C)o1 c1(C(N(CC(C)NC(=O)C(C)CF)C)=O)cccc2c1OCCC2 CCC(CC)C(F)C(=O)N1CCC(O)(CN(C)C(c2cccc(CO)c2)=O)C1 CC(C)(C)CC(=O)NC1(CO)CN(C(C2CN(C3COC3)C2)=O)C1 c1(CC(=O)NCCOC2CCN(C(Cc3ccc(C)s3)=O)C2)cnccc1C N1(C(=O)COc2ccc(CN3CCOC3=O)cc2)CCC(F)(F)C(O)C1 n1(CCCC(=O)NC2(CO)CN(C(C(OC)OC)=O)C2)nc(C)nc1C C(C(C)(F)C(C)(C)F)(c1nnnn1C(C)(C)CC)NCc1cccc(OCC)c1 N1(C(c2scc(C)c2Br)=O)CCN(C(=O)CCCCC(C)C)CCC1C c1(OCC)ccc(C(=O)NC23CC(NC(=O)CC4OCCC4(C)C)(C2)C3)cc1C C(=O)(CC1CCc2ccccc21)NC(C)CN(C)C(c1cnc2c(c1)NCC2)=O c1(OC)ccc(CCC(C)C(=O)NCC2CCCC(CO)C2)cc1 O=C1CC(C(=O)N2CCN(C(C3CCCN3CC(F)(F)F)=O)CC2C(F)F)=NN1 c1(CNC(C2(CCCC)CCC2)=O)csc(C(=O)NCc2cnc(C)s2)c1 c1(C(N2CC(NC(C3(C4CCCO4)CCCC3)=O)C2)=O)cc2c(nn1)CCOC2 c1(NCCCCCN(C)C)ncccc1S(=O)(=O)NC1CCC12CCC2 c1(C(=O)NCC(Cn2cc(C(C=C)N)nn2)(C)C)c(C)cnnc1O C=CCC(CC(=O)NCC(C)N=[N+]=[N-])NC(C1(C#N)CC(=O)N1)=O C(CNC(=O)C=Cc1cccc(OC)c1)(CC(F)(F)F)NC(C(C=CC)O)=O Cn1ccc2nc(NC3(C#N)CCN(Cc4cccc(CO)c4)C3)nc(Cl)c12 N1(C(c2ccc(C)cn2)=O)CCC(C(=O)NC2C3COCC23)C12CC2 c1(OCCOC)cccc(C(=O)NC2CCC2CNC(c2cc(=O)cc[nH]2)=O)c1 C1(NC(CCC#N)=O)CC2(NC(=O)Cn3cc(Br)cn3)COC1C2 N1(C(c2cc(OCC)n[nH]2)=O)CCC(C(=O)NCc2noc(C3CC3)n2)(CF)C1 N1(C(c2c(-c3ccc(CCCCCC)s3)c[nH]n2)=O)CCC(C)(F)CC1 C1(CNC(C2(CCCC)CCC2)=O)CCC(NC(=O)CC2CCCCO2)C1 CC1CN(C(C2(CO)CC2)=O)CCN1Cc1ccc(F)cc1.N12CCCC1C2 C1(C(N(CC)Cc2ncc(C)[nH]2)=O)CC=CCN1C(=O)C(O)C1CCCC1 c1(OC)ccnc(Cl)c1CNC1CCCC(C(=O)NCC(C)(C)C(N)=O)C1 CCC(CC)(CCNC(=O)CCn1ccc(C)n1)NC(c1cc(C)no1)=O C1(NC(C23CCC(OC)C2C3)=O)CC2CCC1CN2C(=O)C(C)(C)Br CC1CC(CNC(=O)CCc2cnoc2)CCN1C(=O)CC1CCCC(F)(F)C1 CCC(C)CC(=O)C(=O)NC1(C(N2CCCC(N3CCC3)C2)=O)CCCCC1 N1(C(C(c2ccc(C)cc2)C2CC2)=O)CCC2CCC(C1)N2C(=O)CN(C)C C1(CNC(C(C2CC2)SC)=O)(NC(c2cc(C#N)c[nH]2)=O)CCCCC1 C1(NC(C2CC23CCC3)=O)CC12CCN(C(c1cnn[nH]1)=O)CC2 C1(NC(c2c(CC)nco2)=O)CC12CCN(C(c1scnc1COC)=O)CC2 C12(NC(c3cn4c(n3)SCC4)=O)CCOCC1CN(C(C1CCCCO1)=O)C2 n1(COCC(CC#N)O)ccc2cc(C(=O)O)ccc12 C#Cc1ccc(CC(=O)NC(CNC(=O)Cc2cnnn2C)CCCC)c(F)c1 C1(C(=O)NCCNC(=O)OCC)CCCCN1C(=O)Cc1nc(C#N)cs1 c1(C(=O)NC2(C)CC(NC(C34COCC(C3)C4)=O)C2)nc2ccccn2c1F c1(C(=O)NC2CC(NC(C(n3ncc(C)c3)C)=O)C2)cccc(CCO)c1 c1(C(=O)NC2(C3N(C(C(C(C)C)C#N)=O)CCC3)CC2)ccc2nnn(C)c2n1 C1(C2(NC(C3C(O)CCN3C(c3cscc3C)=O)=O)CC2)(OC)CCC1 c1(C(N2CCN(C3CCN(C(C4(SC)CC4)=O)CC3)CC2)=O)c(C)cccc1N c1(C(=O)Nc2ccns2)ccc(-n2cc(CNCCO)nn2)cc1 CCC(C(=O)NCC(C)N(C(C12CC(C(=O)OC(C)(C)C)(C1)C2)=O)CC)C(C)C N1(C(c2cc(C#N)no2)=O)CCCC2CN(C(=O)CC3CC4(CC4)CO3)CCC12 c1(C(=O)NC2CCC(N(C(CC)=O)C)C2)cc([N+](=O)[O-])cnc1N C(=O)(CCCCC(F)(F)F)NCC1CCN(C(Cc2cnc(C)[nH]2)=O)CC1CO c1(OC)c(Cl)nc[nH]c1=NCC(C1CC1)NC(c1ccc(C(F)F)o1)=O C(=O)(C1=CCCCCC1)N1CCCC(C(=O)NCc2ncsc2C)(CC)C1 Cc1ccc(C(=O)NCC2CCCC2NC(=O)CCc2ccon2)c([N+](=O)[O-])c1 CCCCC(CC(=O)NCCCC(=O)NO)NC(=O)CN(C)CC c1(C(N2CC(CC)C(C(=O)OC(C)(C)C)CC2)=O)ccc2ncn(C3CC3)c2c1 c1(C(=O)NC(C(CO)NC(CCNC(C)=O)=O)C)ccc([N+](=O)[O-])cc1Cl C=CC(CCC)CC(=O)NC1CCC(C)N(C(=O)CCc2cnc(C3CC3)o2)C1 CC(C)(C#N)CCC(=O)N1CCCC1C(=O)NCC1(c2ccccc2)CC1(C)C N1(C(=O)Cc2cn3ccccc3n2)CCC2CN(C(C3CCS3(=O)=O)=O)CC2C1 N1(C(CCn2cnc(=N)[nH]2)=O)CC(NC(=O)CCC2CCOCC2)C(C2CC2)C1 CN1CCC2CCN(C(=O)CCN(C(C3CCCCO3)=O)C3CC3)C2C1 c1(OC)cncc(C(=O)NCC2CN(C(=O)COCc3nc[nH]n3)CC2O)c1 N1(C(CCOC)=O)CCC(C)(C)C(C(N2CC3CCC(C(=O)OC)(C3)C2)=O)C1 C(C(CNC(=O)OC)C(=O)NCC(C1CC2CCC1C2)=O)OCC Cc1ccc2c(c1C(=O)N(C)CC1CCCN1C(=O)Cc1ccco1)CCCN2 c1(C(=O)NC(C(C)NC(C(CC#C)CC#C)=O)C)ccc2nnc(C)n2c1 C=CCC(CC(=O)NOCC1CC1)NC(=O)C1=NOC2COCC12 C1(NC(=O)NC(CCCC)CN)C2CCC1CC(CO)C2 C1(CNC(c2c(C)noc2)=O)CC2(CCC2)CN1C(C1CCS1(=O)=O)=O N1(C(C2N(C(CC=CC)=O)CCOC2)=O)CC2(CCCO2)C1 CC1(C)CC(CC(N2CC(F)(F)C2C2CC2)=O)CN1C(=O)C(=O)NC1CC1 N1(C(C2(C)CC(C)C2)=O)CCN(C(=O)CCc2cccc(O)c2)C(C(F)F)C1 CCCC(CCC)=CC(N1CCCC1C(C)NC(=O)CCCCOC)=O C1(C(=O)NC2(C(N3CCCCCCC3)=O)C(C)C2)CCCC12CCC2 C(=O)(C(C)(C)C1=CCN(C(=O)C2=COCC2)C1)NC1C(C=C)CC1 C(=O)(CCCCC#N)NC(CCC)C(=O)N1CCC(N2CC(O)C2)C1 CC1(C)CN(C(=O)C=Cc2ccccc2)CC1NC(=O)COCC(F)F CC(C(=O)N1CC2CC1C2CNC(c1ccc(Cl)s1)=O)C(C)(C)C c1(NC(C2C(C)N(C(C3(O)CCOC3(C)C)=O)CC2)=O)cccc(Cl)c1O c1(C(N(C2CCN(C(C3CCCN3C)=O)C2)CC)=O)oc(Br)cc1C Cc1nc(CNC(=O)OC(C)(C)C)ncc1C(=O)NCC1COC(=O)N1 Cc1nc2c(C(=O)NCC(C)(CC(C)C)NC(c3nn[nH]c3Cl)=O)ccnc2[nH]1 N1(Cn2nnc(C(C)(C)C)n2)CCC2CCC(C1)N2C(c1cc2n(n1)CCO2)=O C1(C(=O)NC(C#C)(C)C2CCC2)CCOCC1NC(C1CCCN1C=O)=O C(C(=O)NCC1CCN(C(c2ncoc2-c2ccco2)=O)C1)(C(C)C)SC N1(C(c2ccc(C)c(C#N)c2)C(=O)NC(CC)C)CCC2(CC1)COC(=N)N2 c1(C(N(C2CCN(c3ncc(OCC)cn3)C2)C)=O)cccc(F)c1Br C(=O)(C1=CCC(F)(F)CC1)NC(C(C)C)(C)CNC(=O)C(C)N(C)C C1(NC(C(CC)N(CC)CC)=O)COC2(C1)CN(C(c1ncnc(C)c1C)=O)C2 N1(C(C(C)C)=O)CC(C(=O)N(C)CCC2CCCO2)C(C)(C)C1 C(CC(=O)NCC=CCNC(C1CC1(Cl)Cl)=O)=CCC Cc1cc(C(=O)NCCC2(O)CCN(C(=O)CCc3cccc(O)c3)C2)nn1C c12cccc(c1)NC2=O.C1(SC)C=CCN(C(=O)CCCCN(C)C)C1 N1(C(CC(COC)(C)C)=O)CCC(N=[N+]=[N-])(C(=O)N(C)Cc2ccsc2)C1 C(=O)(CCC(CF)CF)N(C1CCN(C(C2(C(F)(F)CC)CC2)=O)C1)CC#C N1(CCC(N2CC(NC(CCC#C)=O)(COC)C2)=O)C(C)CCCC1C C1(NC(c2ccc(C#C)nc2)=O)CN(C(=O)C(O)CCC(C)C)CC(C)(C)C1 C(=O)(CS(=O)(=O)CCOC)NC(CCC)CC(=O)NCCS(C)(=N)=O N1(CC(=O)NCC(CC)NC(c2c(C)ncn(C)c2=O)=O)C(=O)C(C)C(C)C1=O c1(CCC(=O)NCC(C)(C2CC2)NC(=O)CCCF)ccc(F)c2c1CCCC2 c1ccc(CCC(c2nnnn2C2CCC2)NC2(C3CCCO3)CC2)cc1 N1(C(C(Cc2ccco2)NC(C(C)OC)=O)=O)CC(OC)CC(C)C1 c1(C(=O)NC(CN(C(C=Cc2n(CC)ccn2)=O)C)C)ccc(C)nc1O CP(C)(=O)c1csc(C(=O)NCC2C3CNCC23)c1 N1(C(C(CC)OC2CCCC2)=O)CCC2(CC(NC(C3CCC=CO3)=O)CO2)C1 c1(C(C)C)c(NC(=O)N(C)Cc2ccnnc2)cnn1-c1ccccc1 c1(C(C)OC(CN(CCC)CCC)=O)cc(Cl)c(Cl)cc1O C1(NC(CCCC2C(C)C2)=O)CN(C(c2cc(C)n(CCO)n2)=O)CC1C1CC1 c1(C(N(CC(O)CNC(c2c[nH]ccc2=N)=O)C)=O)nc2n(c1Br)CCC2 c1(CC(N2C(CNC(C(F)=CCC)=O)C(C)CC2)=O)cccc(Br)c1C Cc1cccc2c(C(N3CCC(C)N(c4cncc(C#N)n4)CC3)=O)c[nH]c12 CC1=NN(CCC(C)C)C(=O)C1CC(=O)NCCNC(C12CC(C)C1C2)=O c1(OC(C)C)cc(C(=O)NC(CNC(c2ccon2)=O)CO)ccn1 CCC(CC(=O)N1CC2(CC2)CC1C(=O)NC1CCCSCC1)C(F)F c1(C(N2CC(C)(NC(c3cc(C)n(C(C)C)c3)=O)C2)=O)ncc2ccccn12 c1(OC)ccc(N)cc1C(N1CCCOCC1C)=O N1(C(C(N2CCOCC2)C)=O)CC2CCN(C(c3ncc[nH]c3=O)=O)C2C1 c1(C(=O)NCC2(O)CCN(C(CC3(C)OCCO3)=O)C2)sc2cccnc2c1Cl C(CN=[N+]=[N-])(C(=O)NCC(C)(O)C1CCC1)NC(C(CC)SC)=O N1(CC=C)C(=S)NC(c2cc(C)ccn2)C(C(=O)OCC)=C1C(C)F Cc1[nH]nc2c1CC(C(N1CC3CN(C(c4ccsc4Cl)=O)CC3(C)C1)=O)CC2 C1(C2(NC(=O)Cc3ccsn3)CC2)CCCN1C(C1CCSCC1)=O C1(C(N2C(COC)(CNC(=O)CC(=O)NC3CC3)CCC2)=O)CC12CC(C)(C)C2 CC1CCCN(C(C2CC3CCCC23)=O)C1CNC(=O)COCC1CCOC1 c1(C(C(=O)NCC2C(NC(COCC(=C)C)=O)CC2)C)ccccc1F C1(C(C)NC(C2CC(CC(F)F)C2)=O)C2CN(C(=O)COCCF)CC12 C(=O)(CC(C(=O)NC(C)CCN(C)C(c1ccnc(C2CC2)c1)=O)N(C)C)OC C1(NC(C=CC)=O)CN(C(=O)CCCn2cccc2)CC12CC2 CC1(C)C(CNCCCOC2CCC2)C1(C)C.C1CCCC1 C1(O)(C(N2CCC(N(C)C(c3ccnn(C)c3=O)=O)C2)=O)CCCC(C)(C)CC1 N1(C(C(CC)N(C)C)=O)CC(NC(=O)Cc2nc(C)sc2C)C(C2CC2)C1 c1(C(=O)NCC(CC(=O)Nc2ccc(NC(C)=O)cc2)OC)cc2cccnc2[nH]1 Cc1cccn(CC(=O)NCCCOCCN(C)C(C2CCC3(CC3)C2)=O)c1=O C12(C(=O)NC(C3CCCN3C(=O)C(CO)N(C)C)C)CC(C)(C1)OC2(C)C C(=O)(CCC(=O)c1cccs1)NC(C)CNC(=O)CCc1cnn(C)c1 c1(CN2C(C(=O)NCc3cnc(CCC)o3)CC2)cnc(Cl)cc1Br Cc1cnn(C)c1-c1cn(CC2CN(C(C3C4CC(=O)CC34)=O)CCO2)nn1 c1(-c2nc(C3C4CC(O)C43)n(-c3ccncc3)n2)ccc(Cl)cc1O N1(C(c2c(C)non2)=O)CCC(CO)(CNC(c2cnn(CC3CC3)c2)=O)C1 C1(CC)CN(C(c2cc(CNC(=O)C(C)C3(O)CCC3)cs2)=O)CC(=O)N1 C1(CC)OCCCC1C(=O)NCCCOCCNC(=O)CCCN(C)C CN1N=C(CC(=O)NC2CC3(C2)CC(CNC(c2cc(C#N)c[nH]2)=O)C3)CC1=O N1(C(C2CC(O)(CC#C)C2)=O)CCCC(CC=C)(NC(c2sccc2OC)=O)C1 C#CC1(O)CCCN(C(C2C(C)CCN2C(=O)CNC(C2CC2C)=O)=O)C1 c1(OC(F)(F)F)cccc(CNC2CC2C(F)(F)F)n1 C1(NC(=O)NCC(c2ccccc2C)(C)OC)CCOC12CCCCC2 Cc1ncc(C(=O)NCCC2CSCCN2C(c2csc(Cl)n2)=O)n1C O=C(C1=NOC2COCC12)NC1CCCC(C(N2CC(C3CC3(F)F)C2)=O)CC1 S(=O)(=O)(CC(=O)NCCC1(NC(=O)CCn2cc(C)cn2)CC1)N(CC)CC c1(NC2(CCC)CCN(C(c3cccc(CF)c3)=O)CC2)ncn(C)c(=O)c1Br c1(C(N2CC3C(CNC(Cc4cc(C)no4)=O)(C3)C2)=O)c[nH]c2ncc(F)cc12 N1(C(c2c(C)noc2)=O)CCOC2(CCN(C(c3cnn(C)c3N)=O)C2)C1 c1(C(=O)NCC=CCNC(C(C(CC)O)(C)C)=O)c[nH]c2ccc(C#N)cc12 N1(C(CCC)=O)CCC(OCCNC(C2CCCCC2C(=O)O)=O)CC1 C1(NC(C(C)=C2CCC2)=O)CCN(C(=O)C(F)C(F)(F)F)CC1(C)C C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(C)N(C(C2CC(OC(F)(F)F)C2)=O)CC1 C1(C(N2C(C)CN(C)CC2)=O)CCC2(CN(Cc3cccc(O)c3F)C2)O1 Cc1cc2nccnc2cc1C(=O)NCC(C)CNC(C1CCOCC1)=O c1(C(=O)NC2CCC(CNC(c3cccc(N4CCC4)c3)=O)C2)nccnc1Cl c1(NC(CC)C2CCC2)ncc(C)cc1S(=O)(=O)NCC1CCS(=O)(=O)C1 c1(C(=O)NC(C(C)(C)NC(C2C(C(=O)OC)CC2)=O)C)cc2ccccc2cn1 Cc1ccc(C)c(C(=O)CCC(=O)NC2CCC2NC(c2nnsc2C)=O)c1 N1(C(C=COCC)=O)CCC2CN(C(c3ccc4c(c3)CN(C)C4)=O)CC2C1 C(C(C)(O)CC(=O)NC1(C)CC(C(N2CCCC(O)C2)=O)C1)OC C(=O)(C(C)(C)C(F)(F)F)N(CC1(c2ccc(C)cn2)CCC1)C(C)C c1(NC(C2OCCN(C(c3cn(CCC)nc3C)=O)C2)C)cc(=O)n(C)cn1 Cc1oc(C(N2CCC(F)(CNC(c3csnc3Cl)=O)C2)=O)cc1CO c1(CCC(=O)NCC(CNC(COCCOCC#C)=O)F)nccn1C Cc1ccc(Sc2ccc(C(=O)N(CC(C)CNC(=O)CO)C)cc2)c(C)c1 c1(C(=O)NCCSCc2ccccc2)cc2c(cc1F)NCCC2 C(=O)(C1=CCC(C)(C)CC1)NCC(C(C)C(C)C)NC(C1CC(OC)C1)=O N1(C(C=C(COC)C)=O)CCCC(CC(N2CCC(CC3CCC3)C2)=O)CC1 c1(C(C(C)C)=O)ccc(NC(=O)Cc2cncnc2)cc1 N1(C(C=NOC)=O)CCCC1C=CC(=O)NC1CC2C=CC1C2 CN1C(=O)NCC1C(=O)NC1CC(F)(CNC(C2CCCC2)=O)C1 c1(OC)cccc(Cl)c1CC(N1C(CNC(=O)C(C)C2CC2)CC2CC12)=O C1(NC(c2ccc(OC)o2)=O)CC2(C1)CN(C(=O)C(CO)N(C)C)C2 c1(CN(C(c2cc(C)on2)=O)C)cnn2c1CN(C(c1cccnc1)=O)CC2 c1(C(N2C(CNC(C(COC)OC)=O)CCCC2)=O)cccc(Cl)c1F c1(CN(C(COC)=O)C)cccc(NC(C2(Nc3cccnc3)CCC2)=O)n1 Cc1cc(NC2CN(C(c3csc(CC(C)C)n3)=O)C2)n2ncnc2n1 C12(NC(C3CCN(C(C4(CO)COC4)=O)C3)=O)CC(C3CCCC3)(C1)C2 c1(C(N(CC(C)CNC(C2CC2C)=O)C)=O)ccc([N+](=O)[O-])cc1Br C(CC(C)C)(C(=O)NC1(C(=O)OC)COC1)NC(=O)NCCC c1(C(=O)Nc2c(C)ccc(OC)c2)cc2cc(-c3cncn3C)ccn2n1 c1(CC(N2CCC(N(C(C3C(C=C)C3)=O)CC)C2)=O)ncccc1F N1(C(c2c(OC)n[nH]c2)=O)CCC(C)C1CNC(=O)CC1(C(F)(F)F)CC1 N1(C(C(c2ccc(Cl)s2)C)=O)CCN(C(c2ccc(CF)cc2)=O)C(C)C1C C1(NC(N2CCCC(C(N)=O)C2)=O)CCS(=O)(=O)C2(CCOCC2)C1 c1(C(N(CC(C)(C)CNC)CC)=O)nc(COC)cs1.C1(=O)COCC(=O)N1 C(=O)(C1c2c[nH]nc2CN1C(c1ccc(C(N)=O)o1)=O)N1C(C(C)O)CC1 C1(C(=O)NCC(O)CNC(=O)Cn2ncc(Cl)c2C)(OCC)CCCCCC1 c1(C(=O)NC2(C)CN(C(c3ncn(CC)c3)=O)C2)cn2nc(OC)ccc2n1 C(CC(C)(C)F)SC1CC1CC(=O)N(CC(C)C)NC(C=CC(=O)OCC)=O C(=O)(C(F)C(C)(C)O)NC(C(=O)NCC(C)C#N)(C)C c1(OC)ccc(CN2CCC(C(=O)NCCN3CC(C)OC(C)C3)CC2)cc1Br CCCCCC(O)C(=O)N1CC2CC(NC(=O)CCC3CCCCO3)CC1C2 C(=O)(C(F)(F)CC1CC1)NCC(C)(CO)NC(C(COC)N(C)C)=O n1(CC)cnc2c(N(CCCNC(=O)CCc3cncn3C)C)ncnc12 CC1CN(C(c2cnc(S)nc2)=O)CCN1C(=O)CCC1CC(C)(C)CO1 c1(C(=O)NC2C(NC(c3c(OC)cc(C)cn3)=O)CCC2)cc2nnn(C)c2s1 Cn1nc(C(=O)NCC2C3CN(C(C4CN(C(N)=O)C4)=O)CC23)cc1C1(Cl)CC1 C1(CC)C(NC(=O)C(C)Cc2cccnc2)CCCN1C(C1CCC2(CC2)C1)=O c1(OC)c(C(C(=O)NC2CCCC2C#N)NCCN2CCOCC2)cccc1Br C(=O)(C1=CS(=O)(=O)CCC1)NC1CC(CNC(C=C(C)c2ccco2)=O)CC1O c1(C(CNC(NC(C=C)C)=NCc2ccccc2)OC)ccc2c(c1)C(=O)N(C)C2 CC1(C)CCCC(C(=O)NCCCCCNC(=O)COc2cccc(O)c2)CC1 Cc1cccc(CC(=O)NCC2CC(NC(C3(N=[N+]=[N-])CC3)=O)C2)c1 Cc1cncc(C(=O)N(CCNC(=O)C2=CCCC2)C(c2ccccc2)C(C)C)c1C CCCC(C#N)C(=O)NC(C)(C)CNC(=O)CSCC(C1CCCCC1)=O CC(C)CCC(C(=O)N1CC(O)(CO)C1)NC(=O)CCN(C)C N1(C(CCCCC)=O)CC(C(N2CC(n3ccnc3)C2)=O)CC12CCC2 C1(C(C)NC(c2c(CC)nc(C)s2)=O)COc2ccccc2O1 c1(C(N2CCC(NC(C3C(C)C3)=O)C2)=O)ccnc(Cl)c1Cl Cc1nn(C)c(C(F)F)c1C(=O)NCC1(O)CN(C(=O)C(C)CC2CC2)C1 c1(C(C(N2CCC(N(C(=O)CCC3CC3(C)C)CC)C2)=O)O)ccccc1CC CCCCCCCCC(=O)N1CCC2CCN(C(=O)CCCCOCCC)C2C1 c1(C(N(CC(C)NC(c2nn(CC)c(C)c2)=O)C)=O)cc(Cl)cnc1OC CC(C(c1nnnn1C(c1ccccc1)C)NC1CCS(=O)CC1)C(C)(C)C N1(C(CC2C(CC)C2(F)F)=O)CC(NC(=O)Cc2c(F)cncc2Cl)CCC(O)C1 C(C(Cl)C(C)(F)F)NC(C(C1(O)CCCCC1)NC(C(CSC)C)=O)=O N1(C(c2cc(OCC)ncc2)=O)CC2CCN(C(C3CC4(CC4)C3)=O)C(C2)C1 c1(N2CCC(NC(CC)=O)CC2)cc(NCC2(C)CC(C)C2)nc(C(C)C)n1 Cc1nn(C)c(C(=O)NC2CCN(C(c3cnc(=N)[nH]c3)=O)C(C)C2)c1Br N(C(=NCCF)N(C)CC12CCC(CO1)C2)C(c1cnn(C)c1)C(=O)NC(C)C CCCCCC(F)C(=O)NC(C)C(=O)N(C1CC(CO)C1)C c1(OC(C)=O)ccc2c(CN3CCn4c(C5CCCCC5)nnc4C3)c[nH]c2c1 N#Cc1c[nH]c2ncnc(N3CCC(NS(=O)(=O)CCBr)C(O)C3)c12 C12(C(=O)OC)CCN(C(=O)C(N3CCC(CC(F)F)(CO)CC3)=O)CC1C2(F)F c1(C(=O)Nc2c(C)cnc(F)c2)ccc2[nH]cc(-c3cccc(C(C)O)c3)c2c1 Cc1cc(F)c(CC(N2CC3CCC3(NC(=O)C#CC(C)(C)O)C2)=O)cc1F c1(C(N(CCCNC(=O)C(C)NS(=O)(=O)CC)CC)=O)c[nH]nc1COC c1(C(=O)NCCN(C(=O)C(C)(O)c2ccccc2)CC)ccnc(O)c1 CC1CC2C(CC(C(=O)Nc3nc4c(s3)CCC4C#N)N2C(=O)OC(C)(C)C)O1 CC1(C)Cc2cccc(C(=O)NC3CCCC3CNC(=O)Cc3ccsc3)c2O1 Cc1ccccc1S(C)(=O)=NC(=O)c1sc(Cl)cc1C(F)F c1(CNC(c2n(CC=C)nnn2)(C)CC2CCCC2)cc(S(C)(=O)=O)ccc1F c1(CNC(C(C)NS(CC)(=O)=O)=O)nc(NC(C2CCCN2C(C)C)=O)cs1 Cn1ccc2cccc(CN3CCC3C(=O)Nc3ncc(Cl)nc3C(N)=O)c12 C1(SC)CN(C(=O)C2CC2)C2(CCC2)C1.C(C(=O)NC(C)(C)C)N1CCOC1=O C1(Cl)(C(N(CCNC(=O)C(O)c2ccco2)CC)=O)CC12CCOCC2 N1(C(c2ncn(C(C)C)c2)=O)CCCN(C(C2CNC(=O)N2C)=O)C(C)C1 N1(C(c2c(C)scc2)=O)Cc2n[nH]cc2C1C(=O)NC(c1nn[nH]n1)C1CC1 c1(C(=O)NC2CCN(C(c3c[nH]cc(C)c3=O)=O)C2)cc(S(C)(=O)=O)cnc1O N1(C(CC(C)(C)C)=O)CC(C(=O)NCCNC(N)=O)C2(CC2)C1 c1(C(=O)NCC2CN(C(C3(C=C)CCC3)=O)CC2C)cc(Cl)ccc1F c1(C(=O)NC2CCN(C(=O)C(F)(F)CO)CC2F)cccc2cncn12 C1(C(N2CCC(C(C)C(=O)NCc3cc(CO)ccn3)C2)=O)CN(C)CCN1C CC(C(=O)NOCc1cn(-c2ccc(F)cc2F)nn1)C(C)(C)C C1(C(=O)NCCC2N(C(c3c(C)oc(Cl)n3)=O)CCOC2)C2(CCC2)C12CCC2 C(=O)(N=c1cc(Cl)n(C)[nH]1)C1N(Cc2c(C(=O)OCC)cccc2)CC1 C(=O)(CC(C(F)F)NC(=O)C1CC1)NCC(C1COC(C)(C)O1)O Cc1ccc(C=CCC(N2CC3CC3(CNC(C3CC3C)=O)C2)=O)cc1 N1(C(c2c(O)ncc(CC(=O)OC(C)(C)C)c2)=O)CCC(O)CC12CC2 c1(C(N2CCC(N(C)C(C3CCC(C)(C)C3)=O)CC2)=O)nc2cc(O)ccc2[nH]1 Cc1ccc(F)c(CNC(c2nnnn2C(C)(C)C)C2(C)CCCO2)c1F C1(CC(=O)NC(C=CC(=O)N(C(CC)C)C)C)CN(C(=O)NC)C1 N1(C(=O)C2=CCCC2)CC2(CCN2C(c2cc(O)ccc2Br)=O)C1 c1(C(=O)NC2CCN(C(c3c(OC)ccs3)=O)C2C)ccc2nc(O)oc2c1 C1(c2n(C)cnc2)CN(C(C2(F)CC2)=O)CC1NC(=O)CC1CCC=CCC1 CC1C2C(CCN2C(=O)CC2CCCSC2)CN1C(c1cc([N+](=O)[O-])sn1)=O C#CCC(C)C(=O)NCC1C2CN(C(C3CCC(C(C)C)CC3)=O)CC12 Cc1cc[nH]c1C(=O)NCC(=O)NC1CC(N(C)C)C1.C12CC(C1)N2 N1(C(CN(CCC#C)C)=O)C2CCC1C(F)C(NC(=O)C(C)(COC)CC)C2 C1(C(=O)NCC2N(C(CNS(CC)(=O)=O)=O)CC2)COC2(CCC2)CO1 c1(NCC2CC(OC)CN2C)cc(N2CCC(Nc3nccs3)CC2)nc(C)n1 N1(C(C2C(CC(C)(C)C)C2)=O)CC2CC(NC(=O)COCC3CC3)CC2C1 c1(C(N(CCCNC(c2nn(C)c(Cl)c2Cl)=O)C)=O)coc2c(F)c(Cl)ccc12 C1(O)(C(C)NC(C2CCCO2)=O)CCN(C(C2CS(=O)(=O)C2)=O)CC1 c1(CN(c2ccc(C)cc2Cl)CC)cc(C)nc2c1CCCC2 CC12CN(C(=O)CCF)CC1CN(C(=O)C=CCF)C2 c1(CC(=O)N(CC(CNC(C(C)CN(C)C)=O)O)C)cc2cc(Cl)ccc2[nH]1 c1(N(CCC(N2CC(CCC(=O)OCC)C(=O)CC2)=O)C)nccn2cnnc12 C1(N(C)C)CCC(CNC(C23CC2CCN3C(c2cc(C(N)=O)c[nH]2)=O)=O)CC1 C(C)(C)(CCCNC(c1cnn(CC2CC2)c1)=O)NC(C(F)=C(C)C)=O C1(C(=O)OCC)CCN(C(c2cn(C(C)(C)C)nc2C)=O)CC1(C)C CC1(C)C2CCC1(C(=O)NC1(CC=CC(=O)NCC3CC3(Cl)Cl)CCC1)C2 c1(OCC=C)cccc(C(N2CCCC(CC=C)C2)C(=O)NCC(F)F)c1 N1(C(C2(CC#C)CCC2)=O)CCC(NC(c2ncsc2C)=O)C(CO)CC1 c1(CNC(C(C)N(C(=O)CCc2nncn2C)CC)=O)nnc2n1CCC2 c1(CC)cccc(C(N2CC3CCC3(CNC(=O)C(C)(COC)OC)C2)=O)c1O C1(C(=O)NCCCCOCC)CCCC1NC(=O)CC(=O)N(C)C C1(CNC(CCC(C)OC)=O)CCCC12CCN(c1ccnc(C#N)n1)CC2 C12(C(=O)NC(CC)Cn3cncn3)CCCC1CCN2C(C1(F)CCOC1)=O Cc1ncc([N+](=O)[O-])n1CC(N1CCCC(C)(C)C1CNC(c1ccsn1)=O)=O C1(NC(C(CC)N2CCCC2=O)=O)CN(C(C2CC(C)C2)=O)C2(CCOCC2)C1 C1(C)(CNC(c2occ(NC(C3CC(C(C)C)C3)=O)c2)=O)CC2(CC2)C1 c1(N2CCN(C(C(=O)OC)COC(C)(C)C)CC2)nc(F)c(F)cc1F c1(CN2C(CC)CN(C(=O)C(C)(C)CC)CC2)cc2nc(OC)ccc2[nH]1 CC1(C)CC(CNC(=O)C=CCO)N(c2cncc(C#N)n2)C1 c1(C(N2CC(NC(C(C)C3CCOC3)=O)C(C)(C)C2)=O)cc(Cl)c(N)cc1F c1(CN2C(C(=O)Nc3ccc(Cl)nc3I)COCC2)cc(F)c(I)c(F)c1 CS(=O)c1cccc(C(=O)NCC2CCCN2C(c2nccc3cc[nH]c23)=O)c1 c1(OC)ccc(CN2CC3(CC(CC(N4CCC(C#N)CC4)=O)C3)C2)cc1C C1(C2CCN(C(c3ncc(Cl)cc3Cl)=O)C2)(NC(CCC(C)O)=O)CC1 c1(C(N(C)CC2N(C(C3(CC)COC3)=O)CCC2)=O)cc(NC(C)=O)ccc1F c1(CC)ncc(C(=O)NC(CCN(C)C(c2nn(C)cc2C)=O)C(C)C)c(O)n1 CC1CN(C(=O)CC(c2cccc(F)c2)N(C)C)CC(C)N1CCO c1(NC(COCC=C)=O)cccc(NC(=O)CC2CCOCC2OCC)c1 c1(C(=O)NCC2(OC)CCN(C(C3CC=CCO3)=O)C2)cc(C)cc(C)c1O CCC1=C(C(=O)NCC2CN(C(=O)CCC(C)SC)CCO2)SCCO1 c1(OC)ccc(CNC2CCCCN2C(=O)Nc2ccccn2)c(C(F)(F)F)c1 C1(NC(c2c(CC)oc(C)c2)=O)CCCN(C(=O)Cc2c(C)cccc2F)CC1 c1(CC)ccc(C(=O)NCCC(O)CNC(C2CCOC2)=O)cc1Br C(=O)(C(CC(C)(C)C)OC)N1CC(CC)N(C(c2cc(C3CC3)on2)=O)CC1 C1(CCNC(C(CC)=CCCC)=O)CN(C(C2(C(N)=O)CCC2)=O)CC1C C1(N(C(=O)CC2(C)CCC2)C)CN(C(c2ncnc(O)c2F)=O)CCC1O N1(C(c2c(N)cn(C)n2)=O)CCC(CNC(=O)CN2C(=O)CCC2=O)C(F)(F)C1 CN1CC2C(CCCN2C2CC(n3cc(-c4ccc([N+](=O)[O-])cc4)nn3)C2)C1=O C1(C2(NC(c3ccc(N4CCCC4=O)s3)=O)CC2)CCCN1C(c1cn[nH]c1)=O C=CC1CCCCN1C(=O)CC1CC(C)(C)CN1C(=O)CS(C)(=O)=O c1(CC(=O)NC2CCC(CCNC(C(F)=CCC)=O)C2)cccc(C2CC2)c1 C(=O)(C(C)(C)n1cc(Br)cn1)NC(C1CN(C(C2(C(C)=O)CCC2)=O)C1)C c1(N(C(C)C)C)ccc(C(=O)N(CC(O)CNC(=O)C(C)C2CC2)C)cc1 C1(CNC(C=CCC)=O)CN(C(=O)CC(c2nc(-c3ccsc3)no2)C)CCO1 c1(NC(c2cncs2)=O)cnn2c(-c3ccc(N4CCC(O)CC4)cc3)ccnc12 c1(CC(=O)NC(CNc2ccc(CC(=O)OC)s2)C(=O)OC)ccc(C)c(C)c1 N1(C(C=COCC)=O)CCN(C(C2(C)CCC2(C)C(=O)OC)=O)C2(CC2)C1 N1(C(C(CO)NC(N)=O)=O)CC(NC(C2(F)CC2)=O)C2CCCCC12 C1(C(=O)NCC2CC(NC(C(CCC=C)(C)C)=O)C2)CCOC2(CCOCC2)C1 C(CN=C(NCC1CC1C1CC1)NC1CCS(=O)(=O)C1)c1c(C)nn(C)c1 N1(C(C(CCSC)NC=O)=O)CCC(C)(NC(c2ccncc2F)=O)CC1 C[Si](C)(C)C1(CNC(C2C(O)CCN2C(c2csc(Cl)c2)=O)=O)CC1 c1(C(N2CC(C(N)=O)OCC2)=O)nn2c(c1-c1ccc3nccn3n1)CCCC2 C1(C(=O)NCC2CCN(C(C(c3cccc(Cl)c3)C)=O)CC2)CCCNS1(=O)=O C1(C)(C(=O)NCc2cc(C(N(C)Cc3nnc(C)s3)=O)n[nH]2)CCCC1O CC(C)(CNC(C1C(C(F)(F)F)C1[N+](=O)[O-])=O)CCNC(C1(C)CCC1)=O c1(C(=O)NCC(C)SC)cccc(CNC(=O)CC2C=CCCC2)n1 C1(C(=O)NC2CC3(CC(NC(C4CC(=C)C4)=O)C3)C2)OC(C)(C)OC1(C)C C1(C(N2CC(NC(C(C(=O)OC)C)=O)(CF)C2)=O)CCCC(C)(C)CC1 C1(NC(c2c(C)oc(C(C)(C)C)c2)=O)CCN(C(=O)CSC(F)(F)F)C(C)C1 c1(C(C)=O)cc(C(=O)NC2COCCC2NC(=O)CCC2CCOC2)ccc1O n1(C(C)C)ncc(C(=O)NCC2C=CC(NC(C3CCC3(F)F)=O)C2)n1 C(=O)(C1c2ccccc2C2CC1C2)NC1C2CN(C(CC=CC=C)=O)C(C2)C1 C(=O)(CC(C)C(C)(C)NC(c1cc(O)ccc1F)=O)N1CC(CC)C1 C#CCCCCCCC(=O)N(C(C)CNC(c1cccc(-n2cccn2)n1)=O)C C1(C(=O)NC2CN(C(CC3(C)CC3)=O)CC2F)COCCN1C=O N(C1CCCc2ncc(C(F)(F)F)cc21)C(c1c(Cl)cccc1[N+](=O)[O-])=O c1(C(N2CCC(N(C(=O)Cc3ccccc3)CC)C2)=O)ccc(S(C)(=O)=O)c(C)c1 N1(C(c2c(CNC(CCCn3cnnn3)=O)cc[nH]2)=O)CCOCC1CO N1(C(c2cncc(OC(C)C)c2)=O)CC(NC(=O)CCn2ccnn2)CC1(C)C C(N=c1nc2c(ncn2C(C)C)c(NCc2cccc(N)c2F)[nH]1)c1c(C)ccs1 C#CCCCCCCNC(C1(CCNC(=O)C2=CC(C)(CC)C2)CCCC1)=O c1(C(=O)NC2CCCC2CNC(C2CC3(CC3)C2)=O)ccc2ncncc2c1 CCCCC(F)C(=O)N1C2CCC1C(CNC(=O)C(C)(C)n1cccn1)C2 c1(OC)ccc(C)c(C(=O)N(C)CCNC(=O)C(C)C2CCCO2)n1 Cc1nc2c(N3CC(CCCCNC(=O)C(CO)NC(N)=O)C3)ncnc2s1 c1(C(N2CC(COC)(NC(c3ccc(O)cn3)=O)C2)=O)ccc(C)c(Cl)c1Cl C(CC(C(=O)N1CC2CC1(CNC(=O)Cc1ccco1)C2)NC(N)=O)SC c1(NC2CN(C(=O)OC(C)(C)C)CC2C#N)cccc(P(C)(C)=O)c1 c1(C(=O)NCC(C)NC(C2CN(C)C(=O)N2)=O)cccc(C(=O)C2CC2)c1 C(=O)(CCCC(F)(F)F)NCCCCC(C)NC(C1(F)CCCCC1)=O C1(N(C(CCC)C(=O)NCCN=[N+]=[N-])CC(=O)OC)CCC(F)(F)CC1 N1(C(c2c(C)nn(C)c2)=O)CCC12CN(C(c1cncc(F)c1)=O)C2 N1(C(Cc2ncc(OC)nc2)=O)CCC(CCNC(=O)COC(C)C)CC1C c1(C(=O)NC(C)(C)CNC(C2(C3CCCO3)CCCC2)=O)cnn2ncccc12 Cc1cccc(C(N2CCCC(CNC(C34CC(CN3C3CC3)C4)=O)C2)=O)c1Cl N1(C(c2cncc(C)n2)=O)C2CCC1C(NC(C1(C)CCN(C)C1)=O)C2 C(CC(C(C)C)NC(c1cnc(C(=O)OC)cn1)=O)NC(COC)=O N1(C(CCC(C)C)=O)C2CCC1CC(CNC(c1ccc([N+](=O)[O-])s1)=O)C2 C=C(C)C1OCCC1C(=O)NCC1(C)CCN(C(=O)Cc2nnc(S)n2C)CC1 c1(CC)cc(C(=O)NCC(CO)NC(c2cc(Br)c(C)o2)=O)c(C)nn1 C1(C(N(CC#C)Cc2ccco2)=O)CC(C)CN1C(c1nscc1C)=O c1(NC(C2N(Cc3c(OCC)nccc3)CC(F)C2)=O)cccc(Cl)c1O C(c1ccccn1)=CC(=O)NCCCC(C)NC(c1n(COC)ncc1)=O C=CCC(C)(C)C(=O)NCC(C1CCC1)NC(c1ccc(C(F)(F)F)s1)=O c1(OCC)ccccc1NC(=O)C(C1CCN(C(c2cccnc2C)C)CC1)C c1(C(N(CCCNC(C2(C)CCCNC2=O)=O)CC)=O)ccc(C#N)cc1O c1(CN(C)C(=O)NCCC2(F)CCC2)ccc(N2CCCS2(=O)=O)cc1 C1(C(=O)OC)C2=CC(CC2)C1C(=O)N(c1cnc(OC)c(F)c1)C C1(CNC(CCc2onc(C)n2)=O)CN(C)CCN1C(C1OCCN(C)C1=O)=O c1(C(=O)NCC2CN(C(C(CCC)C)=O)CC2(C)C)ccc2nc[nH]c2c1 C(=O)(C(CC(F)F)N(C)C(C1CC2(CC2)CO1)=O)NCc1occ(C)n1 C(C)(CCN=c1[nH]c(=NC2CCn3nnnc3C2)[nH]c2cc[nH]c12)OC c1(C(=O)NCC(C)N(C(c2c(C)nns2)=O)C)cc2c(cc1F)NCCC2 N1(C(C(CC)CC)=O)CCOCC(CNC(c2cnn(CC3CC3)c2)=O)C1 CC(CC(C)(c1nnnn1C1CCCC1)NCC1CC(C(=O)N(C)C)C1)C(F)F C1(N(C(C)(C)C)C(C2C(C)C2)=O)CN(C(=O)NC2CCC(F)(F)CC2)CCC1(C)C C1(CCC(=O)NC2(C)CN(C(c3cnn(CC)n3)=O)C2)CCCC(O)C1 c1(COC(c2nn(-c3ccc(OC)cc3)c(C)c2)=O)cc(Br)cnc1CCN N1(C(C(C)Oc2ccn(C)n2)=O)CC2(C1)CC(C)(C)C2 C1(CCC)(NC(=O)C=CC2CCCO2)CCN(C(=O)CC2CCCS2(=O)=O)CC1 c1(CNC(C2CNCC2F)=O)cc2cnccc2[nH]1 c1(OC2CCN(C(C(=O)Nc3cccc(OC)c3)C3CC3)C2)ccc(F)cc1C c1(C(N(C(C)C2CC2)C2CC2)=O)coc(CNC(=O)C(C)(C)C2CCOC2)c1 Cc1cc(C(=O)N(C)CC2CCN(C(=O)C(C)P(C)(C)=O)C2)ccc1O N1(C(c2c(OC)scc2)=O)CC(NC(C2CCCOC2C)=O)C(C)C1 Cc1ccc(C(CN(C)C)NC(c2csc(-c3ccc(Cl)cc3)c2)=O)cc1 C(=O)(CCS(=O)(=O)C(F)(F)F)NCC(CNC(C1CC(CC)OCC1)=O)(C)O N1(C(c2ccc(SC)s2)=O)CC(C(=O)NCc2ccc(C)cc2O)CC(F)C1 c1(C(N(C(C)CCNC(=O)Cc2ccco2)C)=O)nccc2cnn(C)c12 C1(CNC(C=CCCC(C)C)=O)CCCN(C(=O)C(C(C)C)c2cnn(C)c2)C1 Cc1cc(C(=O)C(C)NC=O)c(C)n1-c1nccs1.c1(C)nc(C2CC2)nn1C c1(C(=O)NC2CC(CNC(C3C=CCCC3)=O)C2)ccc2c(Br)cnn2c1 N1(C(c2[nH]c(=NC)sc2)=O)CCC2(CC1)C(OC)CC2NC(=O)CC1(OC)CC1 N1(C(=O)NCCC(C)N2CCC2)CCC(NC(=O)C(F)(F)F)CC1 Cc1nn(C)c2c(NCC=CCl)nc(=NC3COc4c(F)cc(F)cc4C3)[nH]c12 N1(C(CC)=O)CCC(CNC(=O)CC2(O)CCCC2)(COC)CC1 C1(CNC(C=C=C(C)C)=O)CCN(C(=O)CC2CC=CCN2C)CC1O C(CNC(=O)NC(CC)C(=O)O)(C(C)(C)C)SC C#CC1(C(=O)NCC2CCC(NC(c3sccc3Cl)=O)CC2)CCCC1 CCC(C(=O)NC(C)(C)C1CC1)n1ccc(C2CC2)n1 Cc1nn(CCO)c2nc(C3CC3)cc(C(=O)NC3(C)CC(O)C3)c12 c1(C2(NC(c3nnnn3C3CCC3)C3(CS(C)(=O)=O)CC3)CC2)ccc(Br)cc1 C1(NC(C23C(C)(C)C(CC2)CC3)=O)CCC(N=c2ccnc(CO)[nH]2)CC1 C(C(C)C(=O)NCCN(C)CCN(C)C)NC(CCN(C(CCC)C)C)=O C1(C(=O)NCC(CSC)(C)O)C=CCN(C(=O)CC23CCC(CC2)C3)C1 N1(C(CC(CC)C)=O)CCN(C(=O)Cn2nc(C)c(Br)c2C)CC(O)C1 c1(CNc2cccc(-c3c(C)nc(C)s3)c2)cc(O)ccc1Br N1(C(CN(CCC)C(C2CCOC2(C)C)=O)=O)CCC(F)(F)C(F)C1 C1(C(=O)NCC#CCNC(CCC(c2cc(C)sc2C)=O)=O)CCC2C1C2(F)F Cc1nc2cc(C(=O)N(C3CC4CNC3C4)CC3CC3)ccc2s1 C1(NC(CC(=O)NCC#C)=O)CCC12CCN(C(c1cnn(C)c1N)=O)CC2 c1(CC)nnc2n1CCCC2C(=O)NC1CN(C(C2(OC)CCCCC2)=O)C1 C1(C(=O)NCC2(C(=O)NC(C)CF)CC23CCC3)CC2CC(=O)C1C2 N#Cc1ccc(SCCC(N2CC3(CNC(C4C5CCC45)=O)CCC2C3)=O)cc1 C1(C(N2CCC(COC)C2)=O)(CC)CCCN(C(C2CCN2CC)=O)C1 C1(C)(NC(c2scc(CNC(CCC3CC(C)C3)=O)c2)=O)CCCCC1 N1(C(C(c2ccccc2)=O)=O)CCN(C(C2CC(F)C2)=O)CC1CCO C1(NC(c2c(CC)[nH]cc2)=O)CCCC(NC(=O)CCc2cn(C)nc2C)C1 c1(C(N(C)CCOCCCN(C)C(C2(N=[N+]=[N-])CC2)=O)=O)cccc(CO)c1 C1(n2cc(C(COC)(C)O)nn2)CCN(CC(C2CC23CCCC3)=O)CC1 N1(C(C2CC(CC)C2)=O)CCN(C(c2ccc(C)c(C)n2)=O)CC1CO c1(C(N2CCN(C(c3cnc(CC)s3)=O)CC2CO)=O)cnn2c1CC(C)CC2 Cc1ccnc(C(F)(F)C(=O)NCC(C(C)(C)C)NC(=O)CC2CCCC2)c1 C1(C(=O)NCC2CN3CCC2C3)C=CCN(C(c2ccc(Cl)o2)=O)C1 CN1CCC(CCC(=O)NCC2(CNC(C3CC3)=O)CCCC2)C1.C(=O)NC1CC1 C=C(Cl)CCC(=O)NCCN(C(=O)CC=Cc1ccccc1)Cc1ccccc1 Cc1ccnc(C(=O)NC(C)(C)CCN(C)C(c2cncn2C)=O)c1F N1(c2c(OC)cncn2)CC(C2CCCN(C(c3nc(C(C)C)cs3)=O)C2)C1 N1(C(C2N(C)CCC2)=O)CC2CC(NC(=O)Cc3cccc(F)c3)CC2C1 N1(C(c2n(CC)ncn2)=O)CC2CCC2(CNC(c2sc(CO)nc2C)=O)C1 c1(C(N(CC(CNC(CCCCCC)=O)C)C)=O)ccc(F)c(N)c1F C(N=c1[nH]c(=NC2CCC(OC)C2)c2c(ncn2C)[nH]1)C1(OCC)CCCCC1 N1(C(COCc2ccc(OC)cc2)=O)CCC(NC(=O)COC(F)F)C(O)C1 c1(C(c2cccc(SC(CC=CC)C(=O)O)c2)=O)ccc2cncn2c1 N1(C(C(C)OCCOCC)=O)CCC(N2CCN(C(=O)C)CC2)CC1.C1(O)CC1 C1(CCC)(NC(=O)CCC2CC2CC2CC2)CCCN(C(=O)CCS(N)(=O)=O)C1 c1(CC(N2CC(CN=c3nc(SC)[nH]s3)C(C)(C)C2)=O)nsc2ccccc12 C1(C(=O)NCCCN(C(c2n[nH]c(C)c2Cl)=O)CCO)COCC(C)(C)O1 c1(C(=O)NCC(CCNC(CSC)=O)O)ccc(C2CNC(=O)C2)cc1.C1CS1 Cc1cnc(CCCC(=O)N(C)CCN(C(=O)C(C)NS(C)(=O)=O)C(C)C)o1 CCC(CC)CC(=O)N1CCOCC(NC(=O)CCc2ccc(C)c(Cl)c2)C1 n1(CC(C)C)nccc1C(N1CC(O)(CCNC(=O)C=CC=C(Cl)Cl)C1)=O Cc1scnc1C(N1CC(C)(CCC(=O)N(CCN(C)C)C(C)C)C1)=O CCCCC(CCC)N=c1[nH]c(=NCc2nc(CO)n[nH]2)[nH]c2ccsc12 CCC(C(=O)N1CCC1C(=O)NCC(C)COCC1CC1)OC C1(C(=O)NCCN(CCO)CC)CN(C(c2cc(C(C)C)[nH]n2)=O)CC(C)O1 N1(C(=O)C#CC2CC2)CC2CCN(C(c3ccc4ncnn4c3)=O)C2C1 N1(C(C2CC(SC)C2)=O)CC2(CCC(NC(=O)CC3CC(=O)NC(=O)C3)CC2)C1 CCC(F)(F)CC(=O)NC1CCCN(C(c2[nH]c(C)c(C)c2C)=O)CC1 N(C1CCCc2c[nH]nc21)C(CCN(C(C(CC)n1ccnc1)=O)C1CC1)=O C1(CN(C(C(=O)NCCC2CC2)C2CC=CC2)C)CC(F)(CO)C1 CCC(C(=O)N(CC(C)(C)CNC(C1(OC)CC(C)C1)=O)CC)N1CCCC1=O.OC Cc1ccnc2nc(C(=O)NCC3CCC3NC(=O)CC(C)C)nn12 C1(C(=O)NCCN(C(C2CN3CCN2C(C)C3)=O)CC)CC12CCOC(C)C2 Cc1cc(Cl)cc(C)c1C(=O)NCCC1CN(C(=O)C(N2C(=O)CCC2=O)C)C1 c1(C(N2CC(CC(C)NC(=O)C(N3CCCCCC3)C)C2)=O)cccc(F)c1F C(=O)(CC(O)C(C)C)N(C1CCN(C(=O)CN(C(=O)C(C)C)C)CC1)CCCC Cc1nn(CC(F)F)cc1C(=O)NC1CC(C)(NC(=O)C=Cc2nccs2)C1 N1(C(CCSC)=O)CCC(C)(CNC(C2(C3CCCO3)CCOCC2)=O)CC1 C(=O)(C1=C(Cl)CCOC1)NC(C(=O)NCCOCC(=C)C)c1ccco1 c1(CC(=O)NCC2(NC(C(C(C)OC)N(C)C)=O)CC2)cncc2ccccc12 c1(C(N(C2CCN(C(C3OCCN(C(C)C)C3)=O)CC2)C)=O)cc2sccc2s1 N1(C(C(COC)C)=O)CCCCC12CC(NC(c1cccc(C#CCO)c1)=O)C2 CC(C)CC(C(=O)N1CCC(C(C)(C)NC(=O)C(CN(C)C)N(C)C)CC1)N(C)C Cc1cc(N2CCC(NC(c3sc(CC4CC4)nc3C)=O)C(F)C2)nc(Cl)n1 Cc1cc(Br)cc(Cl)c1NC(=O)C(C)OC(=O)Cc1ccc(N(C)C)cc1 C1(N(C(C)C)C)CCN(c2nnc(C(=O)NC3CC3)n2CCCSCCO)CC1 c1(C(=O)OCC)cc(N2CCC(NC(=O)CCC(F)(F)F)CC2C)nc(CC)n1 c1(CC(N2CCCCC(CNC(CSCCCC)=O)C2)=O)ccc([N+](=O)[O-])cc1 C1(NC(c2c(C)c(C3CC3)on2)=O)CCCCN(C(c2cnoc2C(C)C)=O)C1 N1(CC)CC(C(=O)NC2CCCC2NC(c2ccn(CCOC)n2)=O)NC1=O c1(OC)ccc(CC(=O)NC2CCCN(C(=O)COC3CC(F)(F)C3)C2)c(F)c1 C(=O)(C1=Cc2ccccc2C1O)NCC1(CNC(CC(CCCCC)C)=O)CC1 c1(CC#N)ccccc1CC(N1CC(CNC(=O)C=Cc2ncco2)C1)=O c1(C(N(CCOCCCN(C(CC=CC=C)=O)C)C)=O)cncc(C(=O)OC)c1 C1(NC(CCCOc2ccc(C(C)=O)cc2)=O)CCCCCN(C(=O)C(C)C)C1 N1(C(CCOCCN(C)C)=O)CCCC(C(=O)NCCN2CCC(C)(C)C2)C1 c1(C(=O)NCCCCNC(C2(c3c(C)cno3)CC2)=O)cc2c(ccn2C)[nH]1 c1(C(=O)NC2(CO)CCCN(C(C3CC(=C)C3)=O)C2)ccccc1N=[N+]=[N-] N1(C(CCC(N)=O)=O)CCC(CNC(c2ccc(O)nc2)=O)C(F)(F)C1 C12(C(=O)NC3CC4CC(NC(C5(C)CCCCC5)=O)C4C3)CCCCN1CCC2 C1(NC(c2cc(C(F)F)ncn2)=O)C=CCN(C(C2(C(O)C(F)(F)F)CCC2)=O)C1 N#Cc1ccc(S(=O)(=O)N2CCCC2CNC(c2ccc(CCO)cc2)=O)cc1 c1(CC(=O)N(CC(CNC(c2c(C)snc2)=O)O)C)cnn2c1OCCC2 C(C(=O)NCC(CO)NC(=O)CCCc1ccncc1)(C(C)C)SCC c1(COC)cccc(CC(=O)NCC2CCCN(C(c3c(C)ccn3C)=O)C2)c1 CC1COCC(C(=O)N(CCCNC(c2coc(Cl)c2)=O)Cc2ccccc2)O1 c1(C(=O)NCC(CNC(c2c(CC)onc2C)=O)C)csc2nnsc12 C1(C(N(CC(CC)NC(C23CC(CF)(CO2)C3)=O)C)=O)CCCCC1F c1(C(=O)NCC2(OC)CN(C(c3cc(CC)c(C)s3)=O)C2)n[nH]c2c1CCSC2 c1(COC)nsc(CNC(C2C(C)CC2C)=O)n1 C1(CNC(CCOCCOCC)=O)CC2CCCC2N1C(=O)CC1CCC2CC2C1 C1(NC(c2ccc(CN(C)C)[nH]2)=O)(C)CCC(F)(F)CC1.C(C)(C)(C)OC(=O)N c1(NCC(N(C(Cc2c(C)nc(C)s2)=O)C)C2CC2)cnc(C#N)cn1 N=c1ncc(C(=O)NC2COCCC2NC(c2ccsc2Br)=O)c[nH]1 C1(NC(CC=C=C)=O)CCCCN(C(c2ccc(NCCS(C)(=O)=O)s2)=O)C1 CCC(CNC(C1CC12CCC2)=O)(CC)NC(=O)Cc1nonc1C C1(NC(C(=O)NCC2CC2)=O)CC2(CCN(C(=O)CC3CC4CC4C3)C2)C1 C1(NC(C(CC)NC(C)=O)=O)COCCC1C(=O)N(CC(C)(F)F)C C1(CNC(c2cc(C)ncc2)=O)CC2CN(C(=O)C(C(C)C)OCC(C)C)CC12 c1(OCC(=O)NC(CNC(C2C(C)=C2)=O)(C)CO)cc(C)ccc1Cl N1(C(=O)Cc2cn[nH]c2)CC2C(c3ccc(Br)cc3)(C1)CS2(=O)=O S(=O)(=O)(c1ccc(NCc2cn(CCO)nc2Cl)nc1)NCC(C(C)O)C N1(C(C(C)CN(C)C)=O)C(CNC(c2cc3cccnc3s2)=O)CC2CCCC12 CC1CN(C(C2CC2(C)C)=O)CCCN1C(=O)CCCc1c(F)cccc1F C1(CC=C)(NC(c2cncc(Cl)c2)=O)CCN(C(C2CCC(F)C2)=O)CC1 c1(C(N(C2CN(C(c3n[nH]c(C)c3C)=O)C2)C)=O)cnc2cccc(C)n12 N1(C(Cc2cccc(SCC)c2)=O)CC(NC(=O)C(C)C2CCC2)CCC(O)C1 C1(C)(NC(C)=O)CCN(C(C2CCC2NC(=O)Cc2ccnc(O)c2)=O)C1 c1(C(=O)NCC(CNC(c2cc(SC)oc2)=O)(C)F)cc2c([nH]1)CCCC2 C(=O)(CC(C)C(F)(F)F)NC1CCC(CCC(=O)NC(C)Cn2ccnc2)C1 c1(C(N2CC(O)(CCNC(C(C)NC(C)(C)C)=O)C2)=O)ccc2c(c1)N(C)CC2 C1(CC(N2CC(CNC(C(C)(C3CC3)NC(C)=O)=O)C2)=O)OCCOC1(C)C C12(C(N3CCC(N(C)C(c4ccc(CO)s4)=O)C3)=O)CCC(N=[N+]=[N-])C1C2 C(C(C)C(C)C(=O)NCC(C)(C1CC1)NC(=O)Cc1cncc(C)c1)OC Cc1cc(C(=O)NC2(C)CN(C(C3C=CC=CC=C3)=O)C2)nn1C(C)(C)C C1(C(=O)NCCCC2(NC(CCSCCC)=O)CC2)CC(C#N)C1 CN1CC2C(C(=O)NC3CCCC(CC(=O)NCCC4CC=CC4)C3)C2C1 Cc1nn(C)cc1CC(=O)NC1CC1CNC(=O)C(C)NC(=O)C(C)(C)C C(=O)(C(O)C(C)c1ccccc1F)NCC1(CNC(CCOCC)=O)CCC1 CC1(C(N2CC(CO)(NC(=O)CN3CC(C(F)(F)F)CCC3)C2)=O)CCCC1O n1(C(C)(C)C)cc(C#N)cc1NC(c1c(NC(=O)CCC(N)=O)cccc1F)=O Cc1nnc(O)c(C(N2CCC(NC(c3ccnnc3O)=O)C(F)C2)=O)c1C C1(CNC(=O)C(O)C(F)F)CCCCN(C(=O)Cc2ccc(O)cc2)C1 Cc1c(F)cc(C(N2CCOCC2C(=O)Nc2c(F)cc(Cl)cc2Br)=O)cc1F C1(n2cc(COC)nn2)CN(C(C2CCN(C(=O)OC)C2)=O)CC1CO C1(C(N(C)CC2CCCN2C(C2(F)CCC2)=O)=O)CC(C)(C)CO1 N1(C(CCCOCC=C)=O)CCC2(COCCN2C(=O)Cc2cc[nH]n2)C1 N1(C(COCCC=C)=O)CC2CC1CN(C(c1c(Cl)sc(C)c1C)=O)C2 c1(C(=O)NCC23CC2CN(C(=O)Cc2ccc(F)cc2F)C3)cc(F)ccc1I C1(CNC(C(C)Sc2ncccn2)=O)CC2CCC1N2C(=O)CCN1CCCC1 c1(N(C)Cc2ccc(C)o2)nc(=NCCc2nncs2)[nH]c2c(C)nn(C)c12 C1(NC(CCNC(C)=O)=O)CC(NC(c2n[nH]cc2Br)=O)C12CCC2 C1(CC)(NC(=O)C(F)C(C)C)CCN(C(c2ccc(C)[nH]2)=O)CC1 c1(C(N2CC(N(C(CC(C)n3cccn3)=O)C)C2)=O)cn(C)c(C(F)F)n1 C(CNC(C1CC1[N+](=O)[O-])=O)(CC(=O)Nc1cccnc1N(C)C)OC C=CCC(C(=O)NC(C)C(C)(C)CO)NC(=O)CCNC(=O)NC C1(NC(C(C=C)O)=O)C2CC1CN(C(C1CC(=O)N(C3CC3)C1)=O)C2 C1(NCC(C(=O)OC)NCCCOC)CCCN(C(=O)OC(C)(C)C)C1 c1(C(=O)NC2CC(CNC(C3CC(C)C3)=O)C2)cccc2cccc(O)c12 c1(C(=O)NCC(C2CC2)NC(C2CC23CCCC3)=O)ccc(COC2CC2)cc1 Cc1cc(C(N2CC(CCNC(c3cn[nH]c3)=O)C(C)C2)=O)ccc1Br N1(C(C(C)n2cccn2)=O)CCC2(CC1)CC2CNC(C1CC2C=CC1C2)=O C1(C(=O)NC(C)CCCCNC(=O)C(=O)CC2CC2)CC2(C1)CC1(CCC1)C2 c1(OCC)ccc(C)nc1C(N1CCC(NC(=O)C=CC2CC2)C1)=O c1(C(=O)NC(CC)(CNC(=O)CC2CC(C)(C)C2)CC)cc(F)c2[nH]nnc2c1 C1(CC(N2CC(CNC(C3(CC4CC4)CC3)=O)C2)=O)CCC2CC2C1 C1(NC(CCN(c2ccccc2)C)=O)CC2CC1N(C(C1(C)CCC(=O)N1)=O)C2 c1(C(=O)NC2(COC)CCCN(C(=O)CC(C)SC)C2)ccc2c(c1)CCO2 C1(C(N(C2C(C)CC2)C)=O)CC1C1CN(C(c2coc(C(N)=O)c2)=O)C1 C#CCC(C(=O)N1CCC(C(C)C)CC1)NC(=O)CC(C)c1ccco1 C(=O)(C(C)(C)n1ccc(C2CC2)n1)NCCCN(C(C1C(C)CC1)=O)CCO n1(CC(N2CC(N(C(C(C)C(C)(C)C)=O)C)C3(C2)CC3)=O)ncc2ncccc12 CC(C)C(C)(O)C(=O)N1CC(NC(c2cnc(S)n2C)=O)C1 C(=O)(CCCCCNC(=O)C(O)C1CC1)NCCCCCC C(=O)(C(C)(C)S(C)(=O)=O)N1CC(O)(C(C)NC(c2cncc(OC)n2)=O)C1 N1(C(C(CC)COC)=O)CCC2CCN(C(=O)C#CC3(C)CC3)C2C1 C1(CNC(C(C=C)O)=O)CN(C(=O)CCC2NC(=O)NC2=O)CCC12CCC2 C12(NC(CC(=O)NCC#C)=O)CCN(C(c3c(C)nn(CC)c3Cl)=O)CCC1C2 C1(NC(c2c(C)noc2)=O)CC2(CCCN(C(c3cc(C4CC4)nn3C)=O)C2)C1 n1(-c2ccn(CCOC)n2)nc(CC(C)(C)C)nc1CCC(C)(C)C c1(C(=O)NCC(C)N(C)C(c2cc(C(C)(F)F)on2)=O)ccn(C2CCCC2)n1 N1(C(COCC)=O)CCC2(CC1)CC(NC(=O)CC1COC(=O)C1)CCO2 CCC(C)(C)CC(=O)N1CC2CCC1C2NC(c1ccc(F)c(C)c1)=O c1(C(=O)NC2(C)CCN(CCC(=C)C)C2)cc(C)nc(O)c1 c1(C(=O)NC(C(C)NC(c2c(CC)nccc2)=O)C)ccc(CSC)c(Cl)c1 c1(CCC(=O)NC(CC=C)CNC(C2CCC3(CC3)C2)=O)csc2nc(C)cn12 N1(C(C2C(CCC)C2)=O)CCC2CN(C(c3cc(O)cs3)=O)CC2CC1 N1(C(C2CCCN(C(C)C)C2)=O)CCC(O)(C(C)NC(C2CCCCC2)=O)CC1 C1(CNC(Cn2c(CCC)ncc2)=O)CC(C)CN(C(C2CC2(Cl)Cl)=O)C1 C1(CN(CC(=O)NC(C2CC=CCC2)CO)C(C2CC2)=O)COC(=O)N1 C(C)(C)(C(=O)NCCCO)NS(C)(=O)=O.c12cn(nn1)C2.C1(SCC)CC2CC2C1 C12(NC(=O)CCCCN3CCOCC3)CCC1CN(C(=O)C1=CSCCO1)C2 c1(C(N2CC(CNC(C(C)C)=O)C(C(F)(F)F)CC2)=O)ccc([N+](=O)[O-])cc1 N1(Cc2ccc(OCCC)cc2C)C(=O)CCN(CC2CCC(=O)N2)C1=O c1(C(=O)NCC2(OC)CN(C(=O)C(F)n3cccn3)C2)cc2cccc(C)c2[nH]1 Cc1cc(C(=O)NC2(CO)CCN(C(=O)C(C)(C)C(F)F)C2)c(Cl)cc1Cl C(c1nc(C)c(C)[nH]1)=CC(=O)NCC(CC)NC(=O)Cc1ccc(Cl)nc1 c1(CN(C)C(c2sc3c(c2Br)CNC3)=O)cc(I)c(F)cc1F N1(C(CCCOCCC)=O)CCN(C(N2CCN(C(=O)C(C)CO)CC2)=O)CC1 N1(C(C(C)=C(C)C)=O)CCCCCC1C(=O)NCC1CCCC1 c1(C(=O)NC2C(C(=O)NCC(C#C)CC)C2(C)C)ccncc1OC C(CCCN=c1cc(C)c(S(=O)(=O)NC2COC(C)(C)C2)c[nH]1)=CC c1(N2CC(CC3CCN(C(C=CC)=O)CC3)(OC)C2)nc(OCC)nc(OC)n1 N1(C(C2(CC(C)C)COC2)=O)C2CCC1CC(N(C)C(C1CC(N(C)C)C1)=O)C2 c1(C(=O)NCCN(C(=O)CC2OCCO2)CCC)ccc2c(c1)nc(C)n2C C(C(N=[N+]=[N-])C(=O)N1CCC(NC(C2(OC)CCC2)=O)C1)OCC c1(C(=O)NCC2C3(CCN(Cc4c(C)nn(C)c4Cl)C3)C2)cccc([N+](=O)[O-])c1 c1(OC)cc(C(=O)NC(C)C(CO)NC(C2CCC2C#N)=O)[nH]n1 N1(C(Cn2ccc(C)n2)=O)CCC(C(O)CNC(c2oc(C)nc2C)=O)CC1 C1(Nc2cccc(Nc3c(OCC)cnnc3)c2)CCC(C)(C)CC1 C1(NC(c2c(SC)ccs2)=O)CCCC(NC(=O)CC(C)n2ccnc2)C1 CC1(CO)CC(O)CN1C(c1ccoc1CNC(=O)CN1CC2CC2C1)=O CCC(CC(=O)NCCCCNC(c1cnn(CC)c1Br)=O)C(C)(C)C C1(NC(COCc2onc(CC)n2)=O)CC2CC(C1)N(c1cc(O)ncn1)C2 C1(CCNC(C2C(OC)CC2)=O)CN(C(C2CN(C(C)C)C2)=O)CC(C)O1 Cn1cc(C(=O)NC2CCC2CNC(c2ccccc2F)=O)n2cncc2c1=O C1(C(C)NC(c2c(CC)ocn2)=O)CCCCN1C(=O)CCc1csnn1 C1(C2CCN(C(C3CN(C4COC4)C3)=O)CC2)(NC(c2cc(CO)[nH]n2)=O)CC1 N1(C(c2c(C)ncn2C)=O)CCN(C(=O)CN=S(C)(C)=O)C(C)C1 N1(C(c2ccc(CC)o2)=O)CCC(F)(C(=O)NC2(C)CCC(O)CC2)CC1 c1(CC(C)NCc2cn(-c3ccccc3N)nn2)ccc(Br)cc1F c1(C(=O)NC(CNC(CCc2ccc(=N)[nH]c2)=O)CO)cccc2c1OCC2 CC1CCC(CNC(c2sc(F)cc2Cl)=O)CN1C(=O)CNC=O c1(C(=O)NC2(C(N3CC(C(C)OC)C3)=O)CCCC2)cnn(C)c(=O)c1 Cc1ccc(CC(N2CC(NC(=O)C(c3cccnc3)C)CC2C)=O)cc1Cl N1(C(=O)CCC2CC2)C2CCC1C(NC(C1(c3cncc(Br)c3)CC1)=O)C2 N1(C(C=C(COC)C)=O)CCCOC(CNC(=O)Cc2cc(OC)ccc2F)C1 C(C)(CN=c1[nH]c(Cl)nc(N2CCCCC2)c1C)Oc1ccc(C)cc1C c1(C2(c3cc[nH]n3)CC2)nc(Cl)sc1Cl.C1C(C2CCC2)NC(=O)N1 Cc1cc(=NCC2CCC2C(=O)OC(C)(C)C)nc(O)n1-c1ccccc1 C1(CC(=O)NC(CC)(C)CC)C2CCC(C2)N1C(c1ccc(=N)[nH]c1)=O N1(C(C2(CC)CCC2)=O)CC2CCN(C(c3cn(C4COCC4F)nn3)=O)C2C1 C(=O)(CCC(C)(C)C#N)N1CCCCC(CNC(CC2ON=C(C)C2)=O)C1 C1(C(=O)N(C)CC2CCN(C(c3cccc(N)c3)=O)C2)(OCC)CCOCC1 c1(NC(=O)Nc2cccnc2C2COc3ccccc3O2)nc2cc(Cl)ccn2n1 C(CC(C(F)F)N1CCC1)NC(=O)C(c1cccnc1)C1CCCCN1 c1(NC(=O)OCCC)ccccc1NC(C)(CCCC)c1nnnn1CC(F)F CC(CC(=O)NC1CCN(CCCNC(=O)C=CC2(C)CCOCC2)C1)C(F)(F)F C(CC(=O)NC1(C)CC=CC1)(C(F)(F)F)NC(c1cc(CCC)[nH]n1)=O c1(SC)cc(C)ccc1C(=O)NCC1CCCN(CC#N)C1 C1(C(=O)NC2(CF)CCN(C(C(C)NC(CC)=O)=O)C2)CCCC2C1C2(F)F N1(C(c2cncc(SCC)n2)=O)CCN(C(C2(OC)CC2)=O)CC1CCO N1(C(CCc2cnc(C)o2)=O)CCC(C(N2CCC2C(N)=O)=O)C(C)(C)C1 CC(C)(CC(=O)NCC(C1CCCCC1)O)n1cc(CNS(N)(=O)=O)nn1 C=C(C)CC(C(=O)NCCN1CCCCC1)NC(=O)CCOCC(=O)OC CC1CN(C(c2cc[nH]c(=N)c2)=O)CCC1NC(c1cc(Cl)nnc1O)=O C1(NC(c2sc(CCC)c(CC)c2)=O)CCN(C(c2cc(C#N)on2)=O)CC1C c1(C(=O)NCC2N(c3nnc(C)s3)CCC2)cc(F)c(F)cc1F S(=O)(=O)(CC(=O)NC12CC(NC(c3cncs3)=O)(C1)C2)N(C)C C=C(C)CC(C(=O)NCCCOCC(=O)NCC(C)(C)SC)OC C1(F)(CNC(c2ncccc2Cl)=O)COCCN(C(c2cn(CCF)nn2)=O)C1 C1(C)(CNC(c2c(C(C)C)ocn2)=O)CN(C(=O)CN(C2CCSC2)C)CCO1 C1(NC(C2(CC=C)CCC2)=O)CC(O)CN(C(c2c[nH]nc2CC2CCC2)=O)C1 CN1CCN(C(=O)CC(=O)N(C)C)C(CNC(C2CC23CCSCC3)=O)C1 N1(C(CC(=O)NCC)=O)CC(NC(c2c(Cl)nn(C)c2Cl)=O)C(C)(C)C1 C1(C(=O)NC)C2CC(O)C(C2)N1C(c1ccc(N2CCCC2)nn1)=O N1(C(=O)Cc2ccc(O)c(O)c2)C2CCC1CN(C(C1(F)CCCC=C1F)=O)C2 Cc1c(C(=O)NC(C2CCOC2)CNC(c2ccoc2C2CC2)=O)cncc1F N1(c2cc(N(C)Cc3ncc(Br)cn3)nc(C(C)C)n2)CCC2CN(C)CC2C1 N1(C(c2c(SCC)cncc2)=O)CCC(NC(c2ccon2)=O)C(F)C1 c1(C(C(=O)NC(CCCC)C(=O)OC)Sc2nnnn2C)cc2ccncc2s1 Cc1nnnn1CC(=O)NC1CC(C(=O)NCC2CCOC2C)C1 c1(C(=O)NC2N(CC)CCNC2=O)cccc2nc(-c3ccccc3)[nH]c12 N1(C(C2N(C)CCCC2)=O)CC2CC1CCC2NC(c1ncc(Cl)nc1Cl)=O c1(C(N(CC(CNC(CCN(CC)CC)=O)O)C)=O)ccc(OC)nc1 N1(C(CNC(CC(C)OC)=O)=O)CCCC(C)(F)C1 C(=O)(CC(F)(F)CS(C)(=O)=O)NC1CCCN(C(C=C(C)C)=O)C1 C1(C(N2CCC(CCNC(c3nnc(O)cc3O)=O)C2)=O)Cc2ccccc2S1 n1(CN(C)C)cc(CC(=O)NCCC2CCC(NC(C3(C#N)CC3)=O)C2)cn1 C(CC(C)C(=O)N1CCN(C(C2CC(C)(C)O2)=O)CC1)OC C1(C)(CNC(c2c(OC)nsc2)=O)CN(C(c2scnc2C(C)(C)C)=O)CCO1 c1(C(N2C(CN(C(CCCCCOC)=O)C)CCC2)=O)nc2cc(O)ccc2[nH]1 C1(C(=O)NCCC2(CNC(CC3CCN(C)C3)=O)CC2)CC2(CC2)CO1 C1(CNC(c2cc(C)nn2C)=O)CCC(C)(C)CN1C(=O)C(O)CC(N)=O c1(C(=O)NCC(CC2CN(C(C(C)OCC)=O)C2)(C)C)cc2ccc(Cl)cc2o1 c1(NC(c2cnsc2)C)ccc(S(=O)(=O)N2CCCC2C2CCCOC2)c(Cl)c1 Cc1cc(F)sc1C(N1CC(CNC(=O)CNCc2cccc(O)c2)C(C)C1)=O N1(C(C2(CC)COC2)=O)CCCC(C(N2CCN(CCF)CC2)=O)CC1 C1(C(N2CC(CNC(c3cn(C)nc3C3CCC3)=O)C2)=O)(OC)CCC12CCC2 c1(OC)cnc(C(=O)NCCC(O)CNC(c2cccc(Cl)c2Cl)=O)c(F)c1 N1(CC(=O)NC2CC(CN)C2)CCOC(c2n[nH]c(CO)n2)C1 C12(C(=O)NCC(C)N(C(=O)CC3CCCO3)C)CCCC1C2Br c1(OC)nc(C)cc(=NCC2CCCN(C(c3cncn3C)=O)C2)[nH]1 N1(C(CC=C)=O)CCC(N(C(=O)CCc2cnc3ccccc3c2)C)C2(CC2)C1 c1(OC)cnc(Cl)[nH]c1=NC1CS(=O)(=O)CC1NC(c1ccc(C2CC2)nc1)=O N1(C(C)(C)C)CCN(C(c2sccc2NC(c2n[nH]cc2I)=O)=O)CC1 c1(C(N2CCCC(O)(CCNC(COC)=O)C2)=O)cc2c(F)cc(C)cc2[nH]1 c1nc(NCC23CCC(CN2)C3)cc(NCC2CCOCC2)n1 c1(C(CC)=O)cc(C(=O)NCC2=CCN(C(=O)CCCNC(N)=O)CC2)ccc1F CCC(CC(=O)NC(CNC(=O)CC(COC)COC)CC(C)C)CC(F)(F)F c1(C(N2CCC(NC(C(n3cnc(C#N)n3)C)=O)C2C)=O)cc2occc2n1C C1(C(N(C2CC3(CC3)C2)C)=O)CCN(C(=O)c2cnnc(O)c2)O1 C1(CNC(c2n(CCC)ncc2)=O)CC(C)CN(C(c2ccc(=N)[nH]c2C)=O)C1 CC1(C)C2CCC(C(=O)NC3CC3CNC(c3cnc(O)c(F)c3)=O)C1C2 c1(C(N2CCCC(N(CC(C)CO)CCO)C2)=O)cccc(S(=O)(=O)N)c1.C(C)=O C1(NC(=O)CC2CC2)CC2CCC1(NC(=O)Cc1ccc(Cl)cc1)C2 C(=O)(C1=NOC(C)(C)C1)NCC1(F)CCC(NC(c2c(C)nc(C(C)C)s2)=O)C1 O(NC(=O)C(Cc1ccccc1Br)NC(=O)CC1COC(=O)C1)CC=C(C)C n1(CCNC(C(=O)NC2CC(COC)C2)=O)cc(-c2ccccc2)nn1 c1(CC(CN(C(=O)Cc2cncn2C)C)NC(C2CC2C(N)=O)=O)ccccc1 CCCC(C)(CC)C(=O)N1CC2(COC(CNC(=O)C(F)(F)C3(O)CCC3)C2)C1 c1(CC)cnccc1C(=O)NC1(CC(=O)NCC(F)Cl)CC1 [N-]=[N+]=NCCCCCCC(=O)NCC(CNC(c1cnn2cnnc2c1)=O)CO N1(C(C=CCC)=O)CC2CCC(NC(c3coc(C(F)F)c3)=O)CC2C1 c1(C(=O)NCC23CC(CNC(CSCC)=O)(OC2)C3)ccc2ccccc2c1O C(C1CCCC1)=CC(=O)NCC(=O)N(C1CCC1)CC1CC1Cc1cn[nH]c1 Cc1ccsc1CC(=O)NC(C1CCCC1)CNC(=O)Cn1nnnc1C N1(C(C2CC(OC)C2)=O)CCC(N(C)C(c2cnc(C)[nH]2)=O)C1 C1(C(=O)NCC(C)CC(C)C)(CC)CCN(C(=O)Cc2cccc(C)c2)C1 c1(CC(=O)NC2(CNC(c3c(C)cnnc3O)=O)CC2)ccc(O)c([N+](=O)[O-])c1 CCS(=O)(=O)c1ccc(CNC(=NCC2CCOC2)NC2CCSC2)s1 N1(C(C=CC=CC)=O)CC2CCOC2(CNC(C2CC2c2cnccc2C)=O)C1 C1(C(=O)NCCC(C)NC(CCCNC(=O)NCC#C)=O)CCOC(C)C1 c1(C(=O)OC)cccc(Cl)c1NC(CCc1ccc(NCc2csc(C)n2)[nH]1)=O C1(C(=O)NC(CO)C(=O)NCC2CCOC2)C2CCCC12 C(C(C)C)(C(O)C(=O)NCC1CN(C(=O)CCOC2CCC2)CCC1(C)C)OC C1(CC(=O)NCC(C)(C)CNC(=O)COc2ccccc2)CCC(=O)NC1 Cc1cccc2cc(C(=O)NCCC3(CNC(c4n[nH]c(=N)s4)=O)CC3)oc12 C1(CNC(C2CCS(=O)(=O)CC2)=O)CCCCN(C(=O)CCc2ccc(O)nn2)C1 c1(OCCN2CCC(COC(CCCSC)=O)CC2)cccc2ccccc12 C(=O)(C(C)(C)C(C)(C)O)N1CC(NC(c2c(F)ccc(C)n2)=O)C(C)C1 Cc1cc(C)c(C(=O)NC2(CNC(C3CCC(C)CC3)=O)CCCCCC2)cn1 N12CCC(CC1)C2C(=O)NCC(F)F.c1(N(c2ccccc2)C)ncccn1 c1(OC)cccnc1C(=O)NC1CN(C(C2CCS2(=O)=O)=O)C1 C(=O)(C#CC1(C)CCCO1)N1CCC(C(N2CCC(C(N)=O)C(C)C2)=O)(CC)C1 c1(C(=O)Nc2ccc(COC)cc2)cccc2c1OCCN2 N1(C(C(C)=CC)=O)CCC2(CC1)C(NC(c1ccnnc1Cl)=O)CS(=O)(=O)N2C C1(C)(C(N2CCN(C(C(C)(C)C)=O)CC2)=O)CC2CCC1O2 C(=O)(C(O)CC(C)C)NCCCN1CCC(NC(CCC=C=C)=O)C1 N1(CC)CC(NC(c2ccc(C(=O)OC)[nH]2)=O)CC1=O.C12CC(C1)CCNC2=O c1(C(=O)OCC)ccsc1COC1CCCC1NC(C1OCCC1CC)=O C(=O)(C(C)(C)CCC#N)NC1C(CO)CCN(C(CCSc2n(C)ccn2)=O)C1 c1(-c2cc(C)c(F)c(C)c2)ncn2c1CN(C(=O)C(C)(C)CCl)CC2 CC1C(C(N2CCN(C(=O)CS(C)(=O)=O)CC23CCC3)=O)OC2CCCCC12 Cc1cc(C(=O)N(C)CC2(O)CN(C(C3(CC(F)F)CCC3)=O)C2)c[nH]c1=N c1(C(N(S(=O)(=O)CC2(CCCl)CCC2)C)=O)cccc(C(F)F)c1 c1(NC(=O)NC)ccc(C(=O)NC(C)C(CO)NC(c2cc(C#N)no2)=O)nc1 CCCCCC(F)C(=O)NC(Cn1ccnn1)C(=O)N1CC(CO)(OC)C1 N1(C(C(C(C)O)C)=O)CCC2(CCN(C(=O)C=Cc3ncc[nH]3)CC2)C1 C1(CC(=O)NC(=O)CSC2CC2)CC(C2CC2)C1.C12(CC1)C(C)NC2=O N1(C(C(C)OCCCC)=O)CCN(C(c2cccnc2-n2cccn2)=O)CC1 c1(OC)ccc(Cl)c(C(N2CC(NC(=O)C3=CCCSC3)CCC2C)=O)n1 Cc1cc(C=CC(=O)NC2CCN(C(=O)CC3CC(F)(F)C3)CC2)on1 C1(C)(CNC(C2CCC(CC)O2)=O)CN(Cc2cccc(C)c2Cl)CCO1 C(=O)(C(C)S(C)(=O)=O)NCC(C1CCCC1)NC(Cc1c(C)n(C)cn1)=O C(=O)(CC1=CCOCC1)N1CCC(CNC(C(C)OCCCC)=O)C1 CCC(CC(=O)NC1(C(=O)NC(c2ccccn2)CO)CCOCC1)C1CC1 c1(CC(=O)N(C)CCC2CCN(C(=O)CNC=O)CC2)cc(Cl)c2c(c1)OCCO2 C1(O)(CCC)CCN(C(C23CC2CN(C(=O)C(C)(C)CCSC)C3)=O)CC1 C1(C(=O)NCC(C(CC)C)C)CN(C)CCN1C(=O)C(C1CC1)SC N1(C(CC2CCC(OC)CC2)=O)CCCCC(CNC(C2CCCC2C)=O)C1 C=Cn1cc(C(=O)NC2CCN(C(=O)COCC(=O)OC)C2)cn1.C1COO1 C(=O)(C1=CCCCO1)NCC(C)N(C(=O)CSC(F)(F)F)CC c1(C(N2C(C(N(CC(O)CO)C(C)C)=O)CC(O)C2)=O)cc(F)cc(Br)c1 C1(NC(C2(N=[N+]=[N-])CC2)=O)CC(O)CN(C(=O)CCc2cncs2)C1 c1(C(=O)NCCOCCNC(C2CN(OC)C(=O)C2)=O)cc2c(C#N)cccc2[nH]1 C1(C(=O)OCCn2cc(-c3ccccc3)cn2)C2CNC(=O)C12 c1(OC)ccc(OC)c(CC(=O)N(C)CCOCCNC(=O)CC2CC(C)C2)c1 C1(c2ccccc2F)(NC(C2(C(=O)OCC)CC(=O)C2)=O)CCCCC1 CC(C)CC(CNC(c1cnc(C2CC2)s1)=O)NC(=O)COCC(C)(C)C c1(C(=O)NC(CC)CNC(c2cnc(S)n2C)=O)cccc(OC)c1OC C(=O)(CCN=c1[nH]c2ccccc2s1)NC(CCNC(C(CC)SC)=O)C C1(CC(=O)NCC(C)CN(C)C(c2ccnc(NCCO)c2)=O)NC(=O)NC1=O Cc1cnnc(O)c1C(N1CC(C(O)C(=O)NCC2OC3CCC2C3)C1)=O CCCCCC(O)C(=O)N1CCN(CC(=O)NCC2CCC2)CC1C C1(NC(COCC(=C)C)=O)CCCN(C(C2C(C)C2C)=O)CC1 C1(CC)CCCCCN1C(=O)Nc1ccc(-c2ccc(C)c(N)c2)cc1 C1(c2c(C(=O)NCCNC(C)=O)c[nH]n2)CCCCN1C(=O)C=C(C1CC1)C1CC1 CN1CC(=O)N(CC(=O)NCCN(C(=O)CN(C2CCCC2O)C)C)C1=O C1(C(N(C2CCN(c3nnc(O)s3)C2)C)=O)CC(c2ccccc2)=NO1 C1(C(N(C)CC2CCN(C(c3n[nH]cc3Cl)=O)CC2)=O)CCC(F)(F)CC1(C)C c1(CNC(C2C(F)(F)C23CC3)=O)ccc(C(N2CCCC2(CO)CO)=O)cn1 N1(C(C=C(CC)C)=O)CC(NC(c2ccccc2)=O)C(C)C1 c1(CC)nc(O)c(C(=O)N(C2CCC(NC(=O)CCOC3CCC3)C2)C)cc1C N1(C(C2(OC)CCC2)=O)CCN(C(=O)C(CC(C)C)NC(N)=O)C2(CC2)C1 C(C(CC(F)(F)F)NC(C1CC(C(C)C)C1)=O)NC(CSCCOC)=O C(C)(CCN=c1nc(C(F)(F)F)[nH]s1)NC(c1c(C)ccc(C)c1)=O C1(c2c(OC(F)F)ccc(C)c2)NC(=S)N(CCC#N)C2=C1C(=O)OC2 C1(N(C(C)C(=O)OC(C)(C)C)c2ccsc2)CCCCC1.C1C(=O)N1 c1(SC(C)C)ccc(CNC(=O)NC2CCCC(CO)C2)cc1 C1(CC(=O)NCCOc2c(OCCN(CC)CC)cccc2)CCC(C)(C)CO1 CN=c1nc(N(C)Cc2ccc(OC(F)(F)F)cc2)[nH]c(=NCCS(C)(=O)=O)[nH]1 C(=O)(CN=c1ccc(C#N)c[nH]1)N1CCC(O)(C(CNC(CCCC=C)=O)C)C1 CC(C)CC(C(=O)NCC(O)CNC(c1cn(C2CC2)cn1)=O)C(C)C N1(CC)N=C(C(=O)NCC2(COC)CCCN2C(=O)CNC(C)=O)CCC1=O c1(C(N2CCC(NC(c3n(CC)nc(C)c3)=O)C2C)=O)nc(Cl)ccc1N c1(NC(C2CC3(CC3)CN2Cc2ccc([N+](=O)[O-])s2)=O)nc(O)nc(O)n1 Cc1[nH]nc(C(N2CCOCC2CN(C(=O)CCCNS(C)(=O)=O)C)=O)c1N N1(C(c2cn(C=C)nc2)C(=O)NC2CCC2)CCN(C)C(=O)C1CCCC S(=O)(=O)(c1cnccc1N1CCCC(N(C)C)C1)N1CCC(NC(C(C)C)=O)C1 C(=O)(C(Cc1ccoc1)NC(=O)C(C)CC1CC1)OC.C12CC(C1)CNC(=O)C2 c1(NC(c2ccc(-n3cccn3)cc2)=O)cccc(Cl)c1-n1cccn1 C1(CNC(=O)CCc2cccs2)CC2CC(C1)N(C(=O)Cn1cnnc1)C2 C1(C(=O)NC(CNC(c2ccc(-c3ccccc3)[nH]2)=O)C2CC2)CC2CC2C1 C(=O)(C1=CCCN(C(C2CCC(=O)CC2)=O)C1)Nc1c(OC)nccc1 c1(C(=O)NC2C3N(C(C4C(C)(C)C4)=O)CC(CC3)C2)cc2cccc(F)c2o1 c1(C(=O)NC2CN(C(C=CCOC)=O)CC2C2CC2)cc2cccc(F)c2s1 c1(NCC(C2CCCCC2)NC(c2c(C)nn(C)c2)=O)ccc([N+](=O)[O-])cc1Br C12(CNC(c3ccncc3O)=O)CCC(C1)N(C(=O)C1=COCCO1)C2 Cc1ncc(C(=O)NCC#CC(=O)NCC(C)(O)C2CC2)c(C)n1 C1(C(N2CCN(C(c3c(CC)scn3)=O)CC2CC)=O)CCn2c(O)nnc2C1 N1(C(C(C)Cc2cnn(C)c2)=O)CC2(CCN(C(=O)CC3(C4CC4)CC3)CC2)C1 C12(C(N3CCCC(N(C)C(c4ccncc4F)=O)C3)=O)C3C4C1C1C2C3C41C#N C1(NC(C(C)CNC(C2C3COCC23)=O)=O)CNC(=O)C1(C)C C12(NC(c3c(C(C)C)sc(Cl)n3)=O)CCCN(C(=O)CSC3CC3)CC1C2 c1(CCC(=O)NC(C)CN(C(=O)C=CCn2cncn2)CC)ccc2c(c1)CCO2 Cc1nc(NCCN2CCOCC2C)cc(N2CCCC(C#N)C2)n1 CC1CCN(C(=O)CC(Cl)Cl)C(C(=O)NCCOCC(C)(C)O)C1 c1(C2C(C(N(C)CC3(O)CN(C(C4CC4C(F)F)=O)C3)=O)C2)ccc(Cl)cc1 C1(NC(C(F)=C(C)C)=O)(CNC(C2CCN(C3COC3)C2)=O)CCCCCC1 C1(C(F)(F)F)(NC(c2cn(C3CCNCC3)nn2)=O)CCNCC1 c1(OC)ccc(C(=O)NC2CCCN(C(c3csc([N+](=O)[O-])c3)=O)C2C)cc1F C1(CNC(C(C)CC(N)=O)=O)CN(C(C2(CC(F)F)CC2)=O)CC12CCOCC2 c1(C(=O)N(CC2N(C(C3C(OCC)C3)=O)CCC2)CC)ccc(C)c2c1NCCC2 N1(C(CC(C)C2CC2)=O)CCCC(C2CC2NC(=O)COC(F)F)C1 c1(C(=O)OC(C)C)ccc(NC(C2CCCN2C(c2ccc(Br)o2)=O)=O)cc1 Cc1n[nH]c(C)c1C(=O)NC1CCCC1CC(=O)NC1CCC(C(N)=O)CC1 N1(C(c2c(SC)scc2)=O)CCC(N(C)C(c2ccc(C)o2)=O)CC1 c1(C(=O)NC2C(C=C)CN(C(=O)CNC(=O)C3CC3)C2)cnn2ccnc(C)c12 c1(C(=O)N(CCCc2cn(C3(C(=O)O)CC3)nn2)CC2CCC2)ocnc1CO c1(C(=O)NCC2C(NC(CNC(CCCCC)=O)=O)CC2)cc(O)nc(C)n1 N1(C(C2N(C)CCC2)=O)CCC2(CNC(=O)CC3CC4CCC3O4)CCCC12 Cc1ncc(C(N2CCC(N(CC(=O)Nc3ccco3)C(=O)OC(C)(C)C)C2)=O)[nH]1 C1(C(=O)NC2(CNC(C(C)CC3CCCC3)=O)CCCC2)CC2CC1CC2(F)F c1(C(N(CC(F)(F)F)C(C)C2CC2)=O)ccc(N2CCCC(O)C2)nc1 C1(C(=O)NC2CCC2CNC(C2(Br)CC2)=O)CC2CCC(C1)S2 c1(C(C)(C)C)ccc(C(N2CCCC2CN(C(c2csc(Cl)c2)=O)C2CC2)=O)cn1 CN1CCCC1C=CC(N1CCCCC1CCC(=O)NCCN1CCCC1=O)=O C(=O)(C(C)C(C)NC(=O)CCc1ccccc1Br)NC(CC(=O)OC)C1CC1 c1(CC)nc(C(C)C)ccc1NC(C1C(F)(F)C12CC2)=O C=CC(F)(F)C(=O)NCC(c1ccccc1F)NC(c1nccn1C(C)C)=O c1(C(C(=O)NCC(C)(C2CCC2)NC(Cc2ccn(C)n2)=O)O)ccc(F)cc1 c1(C(C(=O)NC(CC)C)N2CCC2C(C)C)cnc(N(C)C)c(F)c1Cl c1(NC(C2N(C(CCCC(C)C)=O)CC(O)C2)=O)cccc2occc12 N1(C(C2C(=C)C2)=O)CC2CCC1CN2C(=O)CN(C)C1CC1 C1(COC)CN(C(C2CC2(C)C)=O)CCN1C(=O)CCc1nc(C(C)OC)no1 N1(C(C2(F)C(C)OCC2)=O)CCCC2(C1)CN(C(c1ccccc1F)=O)CCO2 C1(C(=O)NCC(C)N(C(c2n(COC)ncc2)=O)C)CC=CCC1C(F)(F)F N1(C(c2cc(C)sc2)=O)CC2CC(NC(C34CC(C)(CO3)C4)=O)CC1C2 CCC(C)CCN=c1[nH]c(=NCc2ccnc(C(N)=O)c2)c2ncccc2[nH]1 C1(O)(C(N2CCC(O)(CCNC(C=C(CC)C)=O)CC2)=O)CCCC(C)(C)CC1 N1(C(C2(N(C)C)CCC2)=O)CCC2CN(C(c3nocc3Cl)=O)CCC2C1 N1(C(c2c(C)oc(C(C)C)n2)=O)CCCC12CCN(C(=O)C(C)CF)C2 C(=O)(C1=CS(=O)CCC1)N1CC=CC(NC(CCCc2nnc(C)n2C)=O)C1 C(=O)(C(CNC(c1ccc([N+](=O)[O-])[nH]1)=O)C(C)C)NCCNS(CC)(=O)=O C1(NC(C(CNC(C=C(C)C)=O)C(C)C)=O)CC(C)N(C)CC1C CC1CC2(CC2)CN1C(=O)C(O)C1CN(C(c2ccccc2C2CC2)=O)C1 C(C(CN=c1[nH]c2ncc(Cl)cc2s1)C(F)(F)F)NC(C12CC(C)(OCC1)C2)=O C12(C(N(CC(C)NC(c3cnn(C)c3C(F)(F)F)=O)C)=O)CCCCC1C2(F)F N1(C(c2cc(CC)on2)=O)CC2CCC1C1CN(C(=O)C(F)=CCCF)CC21 C(=O)(CS(=O)(=O)CC)NCC(=O)NCC1CC(CC)C1(C)C.n1(C)cc(CO)nn1 C1(C(=O)NCCCC(C)NC(=O)CC2CCC(=O)NC2)CN2CCN1CC2C CCC(CCC(=O)Oc1cccc(Br)c1)NC(c1cc(C2CC2)on1)=O CCCCCCC(CC)C(=O)N1CC2C(c3cn(-c4c(F)cccc4Br)nn3)C2C1 C(=O)(CCCC(F)(F)F)NC(C)CN(C)C(c1ccc(O)cc1O)=O CN1CCCC(C(N2CCC(C(C)(O)CNC(C3CCC3)=O)CC2)=O)C1 C1(C(N2CCC(CCCO)C2)=O)(COC)C=CCN1C(c1sc(O)nc1C)=O CCCCCCCC(=O)NC1(C(=O)O)CCC(C)C1.C12CCC(O1)C(=O)NC2 C(C(=O)N1CCC(C(=O)NOC2CCC(O)C2O)O1)=C1ON=C(CC)C1 C1(NC(c2c(SC)cn(C)n2)=O)CC12CCN(C(c1[nH]c(C)cc1C)=O)CC2 C(CC(C)C(=O)NC(CNC(=O)CSCC1CCCCO1)CC(C)C)=CCC C(=O)(CS(=O)(=O)CC(=O)NC(CNC(=O)CC1CC2(CC2)C1)C1CC1)OC C1(C(N2CC(CCNC(C3(C#N)CCCC3)=O)(OC)C2)=O)CCCCC1(F)F N1(C(COCC(C)C)=O)CC2(CCCC2)C1C(=O)NCCOC(F)F CCC(C)CCCC(=O)N1CC(O)(CCNC(c2[nH]nnc2COC)=O)C1 c1(OCC)cc(-c2ncccc2NC(c2cc(C(C)C)on2)=O)cc(C)c1 C1(NC(C=CCCC(C)C)=O)CC12CCN(C(=O)CCC1CC1C)C2 NS(=O)(=O)c1ccc(C(N2CC=CC(NC(c3cncn3C3CC3)=O)C2)=O)cc1 C(=O)(C(C)CCC(C)(C)C)N1CC(CC=C)(NC(=O)C2=C(C)CC2)C1 N12CCC3(CCN(C3)C(=O)C3(COC3)C1=O)C2.c1(CC)cnncc1C c1(C(=O)NC(C(=O)N(CCCO)CC)C2(O)CCC2)cscc1C(N)=O C1(NC(Cc2scc(C)n2)=O)CCCCN(C(=O)CC(=O)NCC(F)(F)F)C1 C12(CNC(C3CC(C)(O)C3)=O)CCC1CN(C(c1cccc(F)c1Br)=O)C2 CCS(=O)CC(=O)N(CCC(=O)NCC1COCC1(C)C)OC C(=O)(C1=CC2C=CC(C1)C2)N1CCN(C(c2c(C)occ2)=O)CC12CC2 c1(C(=O)NCC(C(N2CC(C#N)(COC)C2)=O)(C)C)cccn2cncc12 c1(NCC(c2ccsc2)C)nccc(=NCC(CO)c2cccc(Cl)c2)[nH]1 c1(C(=O)NC2(CCNC(C3CCC(C)S3)=O)CCC2)cc2cccc(Cl)c2o1 CCC1CCN(C(c2cnc(C)c3c2CCC3)=O)c2cc([N+](=O)[O-])ccc21 c1(CC)ccc(C(N2CCC(CN(C)C(c3ccc(N)c(O)c3)=O)C2)=O)cc1F C(CCC(O)C(=O)NC1CC1C(C)(C)C)NC(c1c(C)n[nH]c1C)=O Cc1ccnc(C(F)(F)C(=O)NCCCNC(=O)CN(C(=O)C(C)C)C2CC2)c1 c1(N2C3CC(N(C)C)CC2CC3)nc(=NCCCCCN(C)C)[nH]c2c1COC2 C1(CC(=O)N(CCC(C(C)C)NC(C(CCC)C)=O)C)CCn2cncc2C1 C12(C(=O)NCC3(NC(c4ncccc4F)=O)CCCC3)CCCN(CC1)C2 c1(N2CC(C)(NC(C3CC4CCCC34)=O)C2)ccncc1C#N C(=O)(C(C)CS(C)(=O)=O)N1CCC(NC(C2CCC(C#C)CC2)=O)C(O)C1 Cc1ncc(C(=O)NCCC2(O)CN(C(=O)CC3CCCC(C)C3)C2)c(C)n1 C(=O)(CCCCCOC)N(C1CCN(C(c2ccc(OC)cc2F)=O)CC1)CC C1(NC(CCCOCC)=O)CCN(C(c2c(OC(F)F)cccc2Cl)=O)CC1C CN1CCN(C(C2C=CCN(C(C3(C)CCCCC3)=O)C2)=O)CC1=O C(=O)(CC(C)C(=O)N1CCC(CF)(NC(=O)CS(N)(=O)=O)C1)OC c1(CC(=O)NC2C(NC(c3cc(C(=O)OC)sc3)=O)C2)c(Cl)cncc1Cl c1(C(C)C)ccc(C(N2CCC(NC(=O)C(C)C(C)(C)C)C(CO)C2)=O)cc1F N1(C(CCC(=O)OC)=O)CC2CCC(C(=O)Nc3cccc(OC)c3C)C2C1 C1(C(N(C2CCCN(C(C(CCC)N(C)C)=O)C2)CCO)=O)CC(=O)C12CCC2 Cc1nc2ccccc2nc1C(=O)NC1CN(C(c2ccccn2)=O)CC1O C1(NC(=O)Cc2ccno2)(CO)CCN(C(=O)CSCC(N2CCCC2)=O)CC1 c1(C(=O)NC2C(COCCCNC(C)=O)C2)cc(CS(C)(=O)=O)c(C)s1 C1(NC(C=CC(N)=O)=O)CCN(C(=O)C=Cc2ccc[nH]2)CC12CCC2 Cc1ccc(C(N2CCOCC2CN(C(=O)C2=NOCC2)C)=O)cc1N CC1=C(C(=O)N2CCCC2CN(C)C(c2ccc(C(F)F)cc2Cl)=O)CCCC1 C#Cc1cccc(CC(=O)NC(Cc2ccccc2)CCNC(=O)CN(C)C)c1 c1(N)cnc(OC2CN(C(COc3cn(C)nc3)=O)C2)cn1.c1(N)cccc(F)c1 C(C(C)(C)CNC(C1CC1c1ccccc1)=O)N(C(=O)COC(C)=O)CC c1(CNC(=O)NCc2ccc(C#N)nc2)ccc2oc(O)nc2c1 C(C(=O)N(C1CCN(C(=O)CCCCc2cnn[nH]2)C1)CCO)(C(C)(C)C)SC N1(C(=O)NCc2cc(C)sc2Cl)CCNC(=O)C1c1ccc(Br)cc1 C(=O)(CCCCCOC(C)=O)NC1CCN(C(c2c(CC)cco2)=O)C1 c1(CN2C(C(N3C(CC(C)C)COCC3)=O)CC(F)(F)C2)ccc2nc[nH]c2c1 CCC(CC(=O)NC1CC(OCC(N2CCN(C)CC(O)C2)=O)C1)C(F)F N1(C(c2n(CCOC)ncc2)=O)CC(NC(C2OCCC2COC)=O)C(O)C1 C(C(=O)NCCOC(C)(C)CNC(=O)Cc1ccn(C)n1)(C(C)C)OC C1(NC(c2n(C)c(=O)ccc2)=O)CCC2(CC1)CCN(C(=O)CC1CC(F)C1)C2 CCC(C)C(C(=O)NCCOC1CCN(C(=O)C#CC(C)C)C1)N(C)C C1(NC(c2ccc(C(C)=O)o2)=O)COCCC1NC(=O)C(C)=C1CCCC1 c1(OC)ccc(C)c(NC(=O)C(Cc2cn[nH]c2)NC(=O)CN2CCC(C)C2)c1 Cc1ccc(C(N2CCC(O)(CN(C(=O)C(C)c3cncs3)C)C2)=O)n1C N1(C(Cc2c(C)nc[nH]2)=O)CCN(C)CC1CNC(c1cc(N)cnc1Cl)=O Cc1cc(N)cc(C(=O)NCC(CNC(c2nc(Cl)oc2C)=O)S(C)(=O)=O)c1F COn1cnc(C)c1C(=O)NCC12CCCCC1C2 C(=O)(C1Cc2ccccc21)NC1CCC(C)(NC(c2onc(C)c2C)=O)CC1 C1(CNC(C=NOC)=O)CCCCC1C(=O)NOCC1CCOCC1 C[Si](C)(C)c1cccc(-c2cccc3c2CN(C(c2ccc(F)cc2)=O)CC3)c1 c1(C(=O)NCCCC(C)NC(C2CSCCS2)=O)c(Cl)c2ccccc2n1C C1(C(=O)NC2CCC(NC(COc3c(C)cccc3)=O)CC2)CC2CCC(C1)C2 c1(CN2C(C(=O)Nc3ccc(CO)nc3)CNCC2)c(F)cc(Cl)cc1Cl C#CCCCCCCC(=O)NC1CCC(C)N(C(=O)CCc2cnn(C)c2)C1 C(=O)(CCC(C)(C)C)N(C1CCCN(C(C2C(F)(F)C23CC3)=O)CC1)CC CC1CCC=C1C(=O)NC1(CNC(c2cn(CCO)nn2)=O)CCCCCC1 N1(Cc2cn(C3CC(N(C(c4cc(Br)co4)=O)CCO)C3)nn2)CCCCCC1 c1(C(=O)NCC2CC(COC)CN2C(=O)CCn2cnnn2)ncc(F)cc1C C1(C)(CNC(C(C=C)(C)C)=O)CN(c2nc(C3CC3)ns2)CCO1 C1(N(C(C2(CC)CC2)=O)C)CCN(C(=O)C(c2ccc(C)cc2)F)CC1 c1(C(C)C)cc(C(N2CC3C(CNC(C4CCOC4)=O)C3C2)=O)n(C)n1 N1(C(C2(CC#C)CCOC2)=O)CC2CCC1C(CNC(c1occc1C)=O)C2 c1(C(=O)NC(c2ccccc2)C(=O)NC2C(C)CCCCC2)cccn2cncc12 c1(NC(C2CC(NC(c3ccc(Br)cc3O)=O)C2)=O)cc(Cl)ccc1CO c1(C(=O)OC)cccc(C(=O)NC(C)(C)CCCNC(C23COCC(C2)C3)=O)n1 O(NC(=O)C(C)NC(c1ccc(C(C)=O)o1)=O)CCCC=C c1(C2(CC)CC2)ccc(C(=O)NCCC(C)NC(=O)CC2CCC(F)(F)C2)cc1 C1(NC(C2C(C)OCC2)=O)CCCN(CCc2cc(Cl)cc(Cl)c2)C1C CC1CCCCN(CC(C2CCNC2=O)=O)C1 c1(C(N(CC(C)N(C(C(C)COc2ccccc2)=O)C)C)=O)nccc(N)c1Cl C12(OC)CCC(C(=O)NC3CC3NC(=O)CC(C)c3ccccc3)(CC1)C(=O)C2 C1(O)(CN(C(Cc2cc(C)no2)=O)C)CCN(C(c2ccccc2Cl)=O)C1 C1(CNC(c2nn(C)c(F)c2)=O)CN(C(c2ccc[nH]2)=O)C2CCN1C2 C1(CNC(COCc2ncc(C)o2)=O)CC2(CC2)CN1C(C1CCC1C(F)F)=O C1(C(=O)NC(C2CCOC2)C#C)CCCCCN1C(c1[nH]ccc1COC)=O C1(C(=O)NCCCCNC(Cn2cc(C(C)O)nn2)=O)CC12CCCCC2 C1(C(=O)NCC(CN(C(c2c(CCC)occ2)=O)CC)(C)C)CCCNS1(=O)=O N1(C(c2cc(F)cs2)=O)CC(NC(C2(CO)CC2(F)F)=O)C(O)C1 c1(CNC(CNC(c2c(C)nc(NC3CC3)s2)=O)C)ccc2c(c1)CCC(=O)N2 C(=O)(C1=CC(C)(CC)C1)NC1C2CN(C(c3c(OC)csc3)=O)C1C2 c1(C(N(C(C)CCNC(c2ccc(C(F)F)o2)=O)C)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NC(CC)CN(C(=O)CNS(N)(=O)=O)CC)cc(C)n(C(C)C)n1 N1(C(C(C)(C)CO)=O)CCOCC(CNC(=O)CN2CCCCCC2)C1 c1(CC(=O)Nc2cc(C)c(-c3ccccc3)cn2)cnc2ccccc2n1 CC1(C)CC(C)(CNC(c2cnc(O)c(F)c2)=O)CN1C(=O)CC1CS(=O)(=O)C1 CC1CCCn2ncc(C(=O)NC3CCN(C(C4(C)CCCCO4)=O)CC3O)c21 C1(CNC(C=C(CCC)C)=O)CN(C)CCN1C(C1CC1CCOC)=O C1C(=O)N=S2(=O)CCC3(CCCN3CC2)CCC(C)C2CCN1CC2 C(=O)(CCC(C)S(C)(=O)=O)N(C(C=C(C)c1cccc(Br)c1)=O)C(C)C C(C1CCCC1)=C(C)C(=O)NC(C1(O)CN(C(=O)C(C)OCC2CCCO2)C1)C C1(NC(c2ccc(C#N)[nH]2)=O)C2CC3C1C3C2C(=O)NCCc1nccc(O)n1 N1(CC(=O)NCCCNC(C2CCC(CC)O2)=O)CCCCC1=O Cc1cc(CNC2CC(N3CCOCC3)C23CCC3)c(Br)cc1F C1(NCc2c(O)cc(Cl)cc2)CCCC12CCCO2 C(C(=O)NC1CC(C)(NC(=O)C(F)OC(F)(F)F)C1)(C(C)C)(C(C)C)NC(C)=O c1(C(N2CCC(C(C)C(=O)NCCC(=O)N(C)C(C)C)C2)=O)c[nH]nc1[N+](=O)[O-] c1(C(N2CCCC(C(=O)Nc3cc(C)cc(C)n3)C2)=O)cccc([N+](=O)[O-])c1F C(=O)(CCCCCCN=[N+]=[N-])NCC(CC(C)C)NC(=O)C(C)CCN(C)C C(CN=c1[nH]n2cc(C)nc2s1)N(C(CCCOCC)=O)C N1(C(CS(CC)=O)=O)CC2(C1)CN(C(c1c[nH]cc1C(F)(F)F)=O)CC2CO Cc1cc(Cl)nc(Cl)c1C(=O)NCC1CN(C(c2cnnc(O)c2)=O)C1 C#Cc1cncc(C(=O)N(CC(C)NC(c2cnc(-c3ccncc3)s2)=O)C)c1 CC(C)(C)CCC(F)C(=O)NC(C)(C)C(NC1CCCn2ncnc21)=O c1(C2(C(CCn3ccnn3)=O)CC2)ccc(Cl)cc1.C1(C(=O)N)CC1 c1(C(=O)NCCC2CCCN2C(=O)CSCc2ncc[nH]2)cn2c(n1)SCC2 C1(NC(CCCc2scc(C)n2)=O)CCN(C(=O)COC2CCCC2)CC1O Fc1ccc2c(c1)CCC(CNC1CCCCNC1)O2 N1(CC(=O)NC2CC2)CCOC(CNC(CNC(CC2(OCC)CCC2)=O)=O)C1 c1(NC(C2(F)CCN(c3cc(C(=O)O)ncn3)C2)=O)ccc(Br)cc1 CC1(CC(=O)NCc2cnc(C3CC3)[nH]2)CCN(C(C2(F)CCOC2)=O)C1 c1(C(n2cc(C(C)(C)NC(Cc3c(C)nn[nH]3)=O)nn2)C)ccc(Cl)cc1 n1(CC)ncc(C(=O)NCC2CC(CC(F)F)C2)n1 C(=O)(C(C)CS(C)(=O)=O)NC(CN(C(C(C)CC1CC1)=O)C)(C)C C(=O)(C1=NOC2(CCC2)C1)NCC(C(C)(C)C)NC(C(CC=C)CC)=O CC1CCOCC1C(N1CCCC1(C)CCC(=O)Nc1ccccc1)=O N1(CC(=O)N(C(C)C(=O)N(C2CN(C)CC2O)C)CC)CCCCC1=O CN1CC(C)(C(N2CCCCC(N(C)C(C3CS(=O)(=O)C3)=O)C2)=O)CCC1=O c1(OC)cc(NC(=O)C(c2ccc(CC(C)CO)cc2)C)c(Br)cn1 Cc1cccc(C)c1NC(=O)C(=O)N(CCC(C)NC(=O)C=CC1CCOC1)C N1(C(C2N(C)CC(O)C2)=O)CC(NC(=O)CCc2ccc(F)cc2Cl)C(C)(C)C1 c1(NC(C2CCN(C(CCNC(C)=O)=O)C2)=O)ccc(Br)c(F)c1 N1(C(c2cc3n(n2)CCC3)C(=O)NCc2nnn(C)n2)CCC2(CCSC2)C1 C1(C(=O)NC(c2ccc(C(C)C)cc2)CNC(C(CC)C)=O)CCCC1(C)C c1(CC(=O)NC(C)CCN(C(=O)C(C)C2CCC2)C)cccc(Br)c1F CCCC(C(O)C(=O)N1CCCC1)NC(C1CCCN1CC)=O Cc1cc(CNC)cc(C)n1.C1(CNC(=O)CC2(n3ccnn3)CC2)CC(C)CO1 C#Cc1ccc(C(N2CC(OC)C(NC(C3CCCC(C)(C)C3)=O)C2)=O)c(F)c1 CCC1=NOC(CC(=O)NC(C2CCN(C(=O)C=CCOC(C)=O)CC2)CO)C1 c1(C(N2CC3C(CNC(c4c(C)cco4)=O)(C3)C2)=O)cc(Br)cnc1F C1(CC(=O)NCC2C(C(=O)NCc3nnc(CC)o3)CCO2)CCCC2CC12 N1(C(CCOCC)=O)CCN2C(=O)C(NC(c3nccc(Cl)c3F)=O)CC2C1 C1(c2nnnn2C2COC2)(NCc2cc(C)nn2C)CCN(C)C1C C1(CNC(CN(C(C)C)C(C23CCCCC2C3)=O)=O)Cc2nccn2C1 C1(CNC(C2C(CCC)C2)=O)CCCCN(C(=O)Cc2cccnc2)C1 N1(CCC)CCC2CCC(NC(=N)NC3CCC(C(=O)OC(C)(C)C)CC3)C12 C1(C(=O)NC(c2ccc(Cl)cc2)C)CN(C(c2ccc(Br)cc2)=O)CC(F)(F)C1 N1(C(CC(CC(C)C)C)=O)CC23CCCC2(C1)CN(C(=O)CCc1nc[nH]n1)C3 N1(C(c2cc(C)on2)=O)CC2CCCC(N(C(=O)CC(C)C(F)F)C)C2C1 CCCC(O)CC(=O)N(CCNC(c1ccc(CSC)o1)=O)CC1CC1 c1(-n2cc(C3N(C(c4c(CC)oc(C)c4)=O)CCC3)nn2)ccc(Cl)c(Cl)c1 C12(C(=O)NCC3(C)C(C)CN(C(CN(C(C)C)C)=O)C3)C3C4C1C1C2C3C41C C#CCCCCC(=O)NC1CCCCCC1NC(c1cnn(C(F)F)c1)=O N1(C(CCC(N)=O)=O)CC2OCCN(C(c3cc(F)cc(F)c3Br)=O)C2C1 c1(C(N2C(CNC(C3C(CN(C)C)C3)=O)CC2)=O)cn(C)c(=O)nc1O CCCCC(=O)NCC1(O)CC(CNC(C2CCN(c3nccn3C)C2)=O)C1 C(C)(C)(CCC(=O)NCC(c1ccc(F)cc1F)NC(=O)Cc1ccsn1)OC C1(C(N2CCCC(NC(=O)C3=C(Cl)CCOC3)CC2)=O)CCc2nncn2CC1 C1(C(N(C2CCCN(C(C=CC3N(C)CCC3)=O)C2)C)=O)Cc2cscc2C1 Cc1onc(-c2ccsc2)c1C(=O)NC(CNC(C1CNC(=O)N1)=O)C1CCC1 c1(N(C)C)cccc(C(=O)NCC(C(C)(C)C)NC(C2(CS(N)(=O)=O)COC2)=O)c1 C1(NC(c2c(Br)cn(C)n2)=O)CCN(C(c2ns[nH]c2=O)=O)CC1CO N1(C(COCCC(C)C)=O)CCC(CNC(=O)Cc2csc(NC=O)n2)C(C)C1 C1(CC(=O)NC(C(C)C)CNC(=O)C2=CCOCC2)CC(C)(C)OC(C)(C)C1 Cc1c(C(=O)NCCC(F)Cn2cc(-c3cnccn3)nn2)sc2nccn12 c1(C(=O)NCCC(CNC(C2(C=C)CCOCC2)=O)=C)ccc2ccncc2c1 C1(C(=O)NC2CC(CCOC)C2)CCOCC1NC(c1cc(F)n(C)n1)=O c1(OC)cncc(C(N2CCC(C(=O)NCCN(C)C)C2C(C)C)=O)n1 N1(C(c2cc(CC)on2)=O)CCCC(N(C(=O)CCc2cc(C)nn2C)C)C1 c1(OCC)ccccc1NC(=O)NCC(C)CNC(c1c[nH]c(C(F)(F)F)c1)=O C=CC(C)(O)C(=O)NCCN(C(c1cn(-c2ccccc2)nn1)=O)CC CC(C(C)(C)NC(=O)CCOc1ccccc1)NC(c1cc(C2CC2)cs1)=O c1(CNC(c2cccc(CC)n2)=O)ccc(CNC(=O)C(F)C(C)(C)O)c(F)c1 C#CC(CC(C)(C)C)NC(c1ccncc1OC)C c1(CC(=O)N(C(C)C)CCNC(=O)C(O)C(F)(F)F)ccc2ccoc2c1 N1(C(C(C)=C2CC2)=O)CCC2(CC1)CC2CNC(=O)CCc1cccnc1F c1(C(=O)NCC2CCCC(F)C2)ccccc1C1(C(F)F)CC1 Cc1nnc(NC2CCN(C(C3CNC(=O)CC3C)=O)C2)c(C#N)c1C O=C(CC1OCCc2sccc21)NCC1CC2CCC(C1)N2C(c1csnn1)=O C12(C)CN(C1)C2.c1(C(N(C)CC2CCCO2)=O)ccn(CCn2cccn2)n1 C=CCN=C(NCC(C)C(F)(F)F)NC1CC(OC(=O)N(C)C)C1 c1(OCC(=O)N(CCNC(CSCCOC)=O)C)cccnc1 C1(OC)CN(C(=O)NC2CC(F)(F)C2C)CCC1(CO)OC c1(OC)cc(C)c(CC(=O)NC(C)CC(C)NC(c2ccccn2)=O)c(C)c1 CCC(CC)C(C(=O)NCC(C(=O)N1CC(C(C)OC)C1)N(C)C)OC C12(CNC(C3(CCCC)CC3)=O)CCC(CN1C(c1cc(C)ccc1F)=O)C2 C12(C(N(C(C)CNC(=O)CCCOC(C)(C)C)C)=O)CC1COC2(C)C Cc1ccc2ncc(C(=O)NCC(F)CNC(C3CCCN(C)C3)=O)n2c1 Cc1cncc(C(=O)NC(CNC(=O)Cc2ccc(C(N)=O)cc2)C(C)C)c1C C(=O)(C(C)(C)C1=CCSCC1)N1CC(CC(CNC(n2ncc(C)c2)=O)(C)C)C1 c1(C(=O)NC2CCN(C(C3(C)CNC(=O)C3)=O)C2)nnc(O)c(Br)c1O Cc1cc(-c2cn(C(C)CNC(c3cc(F)ccc3N)=O)nn2)c[nH]c1=N C1(NC(CCC#C)=O)COC2C(NC(C3(CS(C)(=O)=O)COC3)=O)COC12 Cn1ncc(NC(c2cn[nH]c2)=O)c1-c1cn(CC2CCC(=O)O2)nn1 N1(CC2(C)CCOCC2)CC(=O)N(Cc2csc(Cc3ccccc3)n2)C1=O N(C1CCc2cccnc21)C(C1CN(C(c2ccc(C)nc2C)=O)CC(F)C1)=O C(C(C)(O)C(F)F)NC(c1cc(CNC(c2c(C)non2)=O)oc1)=O Cn1nncc1CNc1ccsc1CNC(=O)OC(C)(C)C C(CCC(C)C)(C(=O)NC1CCC12CCC2)NC(C(=O)OCC)=O N1(C(CNC(c2cc(OC)ncc2)=O)=O)CC2CN(C(c3ccco3)=O)CCC12 N1(C(C2CCN(C(CC)=O)C2)=O)CCC(F)(CNC(C2CCOC2(C)C)=O)CC1 N1(C(CC2(C)CC2)=O)CCN(C(c2ccc[nH]2)=O)C(c2ccccn2)C1 Cc1cc(C(N2CCC(CC(=O)NCc3cccc(O)c3)C2)=O)ncc1C(F)F c1(C(=O)NC(CN(C(C(CCC)CC(C)C)=O)C)C)cc[nH]c(=NC)c1[N+](=O)[O-] c1(C(N2C(CNC(=O)CNC(c3ccco3)=O)CCC2)=O)ccn2cccc2c1 Cc1cc(C(=O)NCCC2CN(C(c3c[nH]cc3C(C)(C)C)=O)C2)cnn1 CC1(CNC(=O)CCc2ncccn2)CCN(C(=O)C(F)(F)C2CC2)CC1 C1(C(=O)NCCC(C)(C)NC(c2cnn(C(C)C)c2F)=O)C2CCCCCCC12 c1(C(=O)NC(CC)CNC(c2ccc([N+](=O)[O-])s2)=O)cc2cc(F)ccc2o1 CC1(C)CCC(C(=O)NCCNC(C2C(c3ccncc3)C2(C)C)=O)C1 C1(C(N(C)Cc2ccc(C)cc2)=O)CCCN(C(c2cc(Br)cnc2F)=O)CC1 N1(C(C2N(C)C(=O)NC2)=O)C2CCC1C(CNC(c1ccnc(Cl)c1Cl)=O)C2 C(c1cscn1)=CC(=O)NC1CC(CCNC(C(C)NC(C2CCCC2)=O)=O)C1 O=C(CCC1CCc2ccccc21)NCC1(CNC(C23CC(F)C2C3)=O)CCC1 c1(C(=O)NCCCC(C)NC(=O)C=Cc2cncn2C)cc2cccn2c(O)n1 c1(CC)ccccc1-n1cc(O)c(C(N2CC3(CCC3)C2)=O)n1 CC1(C#CC(=O)NC2CCC(NC(=O)CCCC(N)=O)CC2)CC1 c1(OC)ccc([N+](=O)[O-])c(NCC2(NC(c3csc(C)n3)=O)COC2)n1 CCCCC(O)CC(=O)NCCN1CCC(NC(=O)CC2(C)CCCC2)CC1 N1(C(c2nc(C(C)C)oc2)=O)CCC(NC(c2coc(CO)c2)=O)C1C(C)C c1(C(N(CCNC(C2CC2COC)=O)CC)=O)cccc(OCCF)c1 c1(C(=O)NC2(CCNC(c3nncn3C3CC3)=O)CC2)cc(-c2ccco2)c[nH]1 C(C1=CCCN(C(=O)COCC(C)(C)C)C1)NC(C(=Cc1ccco1)C)=O C1(CNC(c2cc(SC)c(C)o2)=O)CC2(CC(NC(c3cnn(C)c3Cl)=O)C2)C1 C1(C(=O)NCC(=O)NC)CCCCC1NC(=O)CC1CCC(C)CO1 C(N=c1[nH]c(=NCCc2ccc(CO)cc2)[nH]c2c1CCC2)C1(C)CCCC1O C1(NC(C(c2ccncc2)C)=O)COCCN(C(=O)CCC(C)N(C)C)C1 C1(C(=O)NC(C(C)NC(=O)CN2CSCC2=O)C)CC(F)(F)C1(C)C C(CC(C)C(=O)NC1CN(C(C2(CC(c3cnn[nH]3)=O)CCC2)=O)CC1C)=CC C(=O)(C(C)C(C)S(C)(=O)=O)NC(C1OCCN(C(c2cccc(C)n2)=O)C1)C N1(C(c2c(CC)nc(C)[nH]2)=O)CC2N(C(c3nc(C)ccc3F)=O)CCC2(C)C1 c1(NC(C)=O)ccc(C(N2CC(CNC(c3ccon3)=O)C(C)(C)C2)=O)cc1F Cn1cnc(NC(C2(C)CCN2C(c2cncn2-c2ccncc2)=O)=O)c1 C1(CC(=O)NC2C(C)CCN(C(C3CCC4CC4C3)=O)C2)Cc2ccccc2N1 C1(NC(C(CCSC)(C)C)=O)CC2CC1CN(C(c1cc3cn[nH]c3cn1)=O)C2 N1(C(CCC(C)C)=O)CCC(CNC(C2CCCS2(=O)=O)=O)C(O)C1 C1(CC=C)(C(=O)NCCOCCC(C)C)CN(C(C2CCOC2C(C)C)=O)C1 Cc1nc2cc(C(N3CC(NC(c4[nH]cnc4C)=O)C(F)(F)C3)=O)ccc2o1 c1(C(=O)NC2CCN(C(C3C(C)(C)C3)=O)C2C2CC2)cnc2cc[nH]c2c1 CCCCC(=O)NCC=CC(=O)NCC1(CC)CC1 N1(C(c2c(OC)scc2)=O)CCC2(CC1)CC2NC(C1(C)CC1C)=O N1(C(CC(CC)(F)F)=O)CCN(C(=O)C(C)c2ccsc2)CC2CCCCC12 c1(C(=O)NC2(C(=O)NC(CC#CC)CO)CC2)ccc(C)c(O)n1 O(N1CCC(CC(=O)NCCC(F)Cn2cc(-c3cccnn3)nn2)CC1)CC n1(CC)ncc(C(=O)NCC2CCN2C(C2(C)CC(C)C2)=O)n1 C1(C(=O)NC2CCN(C(Cn3c(C)ncc3)=O)C2C)CCn2c(C)nnc2C1 CC#CCC(C(=O)NC)NC(=O)CC1(OCC)CCC1 N1(C(C(=O)NC)=O)CCC2CCN(C(C3CCc4nc(C)cn4C3)=O)CC2C1 N#CC12CC(C(N3CC(NC(c4cc(C5CCOCC5)on4)=O)C4CC34)=O)(C1)C2 CS(=O)(=O)CCCNC(c1nnnn1CCCSCCO)(C)C1CC1 c1(C(=O)NC2CCCCN(C(c3cc(F)c[nH]3)=O)C2)ccn2ccccc12 c1(OC(c2ccnn2C)C(=O)N(CCNC(C(C)NC(N)=O)=O)C)cnn(C)c1 c1(OCC(=O)NCC(C)N(C)C(C2CCCN2C=O)=O)ccc(S(N)(=O)=O)cc1 c1(NC(c2c(CC)[nH]c(=N)s2)=O)ccc(NC(C2CC(C)CCO2)=O)c(C)c1 Cc1ccc(O)cc1NC(c1cncc(-c2cn(C)nc2C)n1)=O c1(CNC(Cc2cc(C)sc2)=O)cccnc1CNC(=O)CC1COCCN1C Cc1nccnc1NC(=O)NC(CCO)c1nccs1 c1(CC(=O)NC23COC(CNC(c4csc(S)n4)=O)(C2)C3)ccccc1F N1(C2CCN(C(C3C(C)C3)=O)C2)CCC(NC(=O)COc2cnn(C)c2)CC1 CCC(CNC(C1(NC(c2c[nH]c(=N)o2)=O)CC(O)C1)=O)CC(C)C c1(C(=O)NCC2(F)CCC(CNC(=O)Cc3cncnc3)C2)cc2sccc2s1 N1(Cc2ccn(CCC)n2)CCOC(C)(CNC(=O)C(c2cnn(C)c2)C)C1 CCCC(C(=O)NCC1(F)CC(NC(=O)CC(C)OC)C1)OCC C(=O)(C(CC(C)C)OC)NCCCC(=O)NC.O1NC(=O)CC2(CC2)C1 C(C1=CCN(C(=O)C(F)CC2CC2)CC1)NC(c1c(Br)cn(CC)n1)=O CCC(C)C(C(=O)NCCC1(NC(=O)Cc2ccc(C)nc2)CC1)N(C)C C(C(C(=O)NCCCNC(C)C)NC(=O)C(CC)OC)OCC O=C(CCCCCCn1cc(CNC2CC2(F)F)nn1)NC1CCN(C2CC2)C1 c1(CC)cc(Cl)ccc1C(=O)NCCCC1(NC(c2cnc(C)o2)=O)CC1 Cc1noc(N)c1C(=O)NCC1CCCC1NC(=O)Cc1ccnc(O)c1 C1(CC=C)(NC(=O)CSc2nncs2)CCN(C(=O)Cc2cccnc2F)C1 N1(C(C(C)(C)O)=O)CCCC(O)(CCNC(c2cncc(-n3cccc3)c2)=O)C1 c1(C(C)C(=O)N(C2CC(NC(c3cnns3)=O)C2)C)cccc(O)c1 CC(C)(C(=O)NCC1CC1NC(c1ccc(SC(F)(F)F)s1)=O)C(F)(F)F Cc1nc(O)[nH]c1C(=O)NCCCOCCNC(c1oc(CC(C)C)nc1C)=O N1(C(C23CC(C2)C3)=O)CCN(C(C2(c3ccc(F)cc3)CCC2)=O)C(CO)C1 CC(C)(C)CC(CO)NC(C1CCC1NC(=O)C#CC1CC1)=O Cc1cc(CCC(=O)NC(C2CCN(c3ncns3)C2)C)no1 c1(C(=O)NC2C(C)(C)C(CNC(C3COCCOC3)=O)C2)cn2cccnc2n1 C1(CC)CCN(C(c2nnc(S)n2C)=O)C1C(=O)NCCCC(N)=O c1(C(=O)NC(c2c(OCCC)cccc2)C)cc(Br)cnc1O C(c1ncccc1C)=CC(=O)NC(CNC(C1N(C(C)=O)CCCC1)=O)C(C)C C1(C(=O)NC2(C(=O)OC)CCCC2)CN(C(c2ncc(Cl)cc2C)=O)CCN1C C1(C)(CNC(C2(CC)CC2(F)F)=O)CCCN1C(c1sc(C)nc1C)=O CC(C)(F)CCC(=O)N1CCC(C)(CCNC(c2ccnc(S)c2)=O)C1 CCC(CC)C(CNC(c1cn(CC2CCCO2)nn1)=O)N1CCOCC1 c1(C(c2n(Cc3sccc3)nnn2)NCC2COC(=O)C2)cc2c(Cl)nccc2s1 Cc1cc(CC(=O)NC2CCCN(C(c3cc(C)nc(O)c3)=O)C2)c(N)c(C)c1 N1(C(CC(CCC)CC)=O)CCC2(CCC2)C(CNC(=O)C(C)N2CCC2)C1 c1(C(=O)NC2C(NC(c3ccc(C)o3)=O)CC2)cccc(C2CC2)c1Cl C1(C(N2CC3(C(NC(CCCC(=C)C)=O)CCS3)C2)=O)CCC(C2CCCO2)O1 Cc1nc(C)c(CC(=O)NCCc2cn(CC3CCC(=O)O3)nn2)s1 C1(C(=O)NC(C2CCCN2C(=O)CN2CSCC2=O)(C)C)CCS(=O)(=O)N1 c1(C(=O)NCC(=C)CCNC(C2CC2F)=O)cnc2n1CCOC2 C1(COC)CN(C(c2ccnn2C(C)(C)C)=O)CCN1C(=O)Cc1cnns1 C1(N(C(CCC(=O)NCCC)=O)C)CCN(C(=O)CCC(C)OCC)CC12CC2 c1(C(N2C(CNC(c3n[nH]c(CC)c3F)=O)CCC2)=O)c(Br)ccc2c1OCO2 C1(CC)CCCC(C(=O)NCCN(C)CCS)N1 C1(CNC(CCCCSC)=O)CC(C)(C)CN1C(=O)Cc1sccc1Cl C(=O)(C(CC(C)SC)N(C1(C#N)CCC1)C)NC(CC)(C)C c1(CCNC(=O)NCc2c(C(=O)OC)n[nH]c2)ccc2ccccc2c1 c1(C(=O)NCC(C)N(C(c2c[nH]c(=NCC)s2)=O)C)cccc(S(N)(=O)=O)c1 Cc1ccc(C(C)C)c(C(N2CCCC(NC(c3ccsc3C#N)=O)C2)=O)c1 Cc1cc(F)cnc1C(N1CCC2(NC(=O)CC3(N(C)C)CCCC3)CC2C1)=O Cc1ccc(O)nc1CNC(=O)C(C1CCCO1)NC(c1ncn(C)n1)=O c1(C(=O)NCC(CC(C)C)(C)NC(=O)C(CO)C(C)(C)C)cc(Cl)c(N)cc1F N1(C(C=Cc2c(C)nccc2)=O)CCCC2C1CCCN2C(=O)CSCCN(C)C Cc1c(Cl)ccc(C(N2CCC(F)(CNC(=O)CC(O)CN(C)C)C2)=O)c1O CC1CC(NC(=O)CC2(O)CCCC2)CN(C(C23CC(C2)C(C(F)(F)F)O3)=O)C1 c1(N2CCC(CCCCNC(COC)=O)CC2)nc(Cl)nc2nc(Cl)n(C)c12 Cc1c(C(N2CCCC2CN(C(=O)C(F)(F)C(C)O)C)=O)cccc1O C12(C(=O)NC(CC)C(F)(F)F)CCC1CN(C(c1cnc(C)s1)=O)C2 c1(C(=O)NC2CC(C)(NC(c3c(C)nc[nH]3)=O)C2)ccc(C(F)(F)F)c(O)c1 N1(C(c2nnc(C)s2)C)CC(NC(c2sc(C)nc2C)=O)C(C)(C)C1 c1(C(=O)NC2CCC(NC(C3CNC(=O)N3)=O)C2)cc2nn[nH]c2cc1F c1(NC(N(C(C)(C)C)CCOCCCN)=O)c(C#N)cnc2c(Cl)cccc12 n1(C(C)C)cnc(C(N2CCC2CC(=O)NCC2CC=CCC2)=O)c1 CC1CC(CNC(=O)C(F)(F)c2nccn2C)CN1c1ccc(C(F)(F)F)nn1 c1(C(=O)NCC(C)NC(C2(SC)CCC2)=O)ccc(CN2CCCCC2)o1 S(=O)(=O)(c1ccc(CC(=O)NCCOCCOCCOC)s1)NC C12(C(N(C3C=CC(NC(C(N4CC(C)C4)C)=O)C3)C)=O)CCC(CO)(CC1)C2 CCCC(C(=O)N(CC(CC)NC(C1(CF)CC(F)(F)C1)=O)C)N(C)C C1(NC(C(=O)NCCOC)=O)CN(C(c2cc(Br)cs2)=O)CCC1F c1(NC(C2CC(NC(C(C)Oc3ccc(F)cc3)=O)C2)=O)snc(Cl)c1C#N n1(CC(N2CC(O)(CCNC(C3(CC)CCCC3O)=O)C2)=O)ccc(O)nc1=O C(CCC)(C(=O)NCC(c1ccc(F)cc1)NC(=O)C=Cc1ncco1)=CCC C1(C(N2CC(C=C)C(NC(c3cccn3C3CC3)=O)C2)=O)CCCC(C)(C)CC1 N1(C(C2(c3ccc(OC)cc3)CC2)=O)CCC(O)(CCNC(=O)CCC#N)CC1 c1(C(=O)NCC2N(C(c3cc(C)ns3)=O)CCN(C)C2)cccc(C#CCO)c1 C1(NC(C(=Cc2cccs2)C)=O)CC(F)CN(C(=O)Cn2cnnc2O)C1 CCCCCCCCC(c1nnnn1C(C)(C)CC)NCc1ccc(F)cc1Br c1(CC)nn(C)cc1S(=O)(=O)NC1(CO)CC(OC)C1.c1(C)ccccc1 c1(OCC(=O)NCC2(C)N(C(COCCC)=O)CCC2)cc(F)cc(Br)c1 c1(C(N2C3CC(NC(C(CCC)OC)=O)(C3)C2)=O)c(F)cc(C#N)cc1F C(=O)(CC(O)C(Cl)(Cl)Cl)N(CC(C)CNC(c1cnn(C)c1C(F)F)=O)C NS(=O)(=O)c1cccc(CNC(C2CCCC2C2CCCC2)=O)c1 C(=O)(CC(C=C)CC)N(CCCC(=O)NC(CNC(N)=O)(CC)CC)CC=C C1(N(C(C2N(CC)CCC2)=O)Cc2ccc(N(CC)CC)o2)CCNC(=O)CC1 N1(C(C(CCC)(C)CC)=O)CC2CCC(NC(=O)C(CC)N(C)C)CC2C1 C(=O)(CC1CCc2ccccc21)N(CCNC(c1ccc(F)c(C)c1N)=O)CC N1(C(C(=O)NCC)=O)CC2CN(C(=O)C3=NOC(C4(O)COC4)C3)CC2C1 c1(CC(=O)NC(CCNC(C(C)OCC)=O)(C)C)cn2cccc(C)c2n1 CC1(C)OCCC1C(=O)NC1CC(NC(c2cc(C#N)c[nH]2)=O)C(O)C1 CC1(C)CCCOC1C(N1CCCCCC1C(=O)NC(CCO)C(F)(F)F)=O C1(CC(=O)N(CC(CC)(C)OC)C)CCCCN1C(=O)CCn1ccnc1 c1(C(=O)NC(CC)(CNC(c2cccc(N)c2)=O)CC)cc2nc(Cl)ccc2s1 N1(C(c2cncc(NCC)c2)=O)CC(O)C(O)C1CNC(c1ccnnc1)=O S(=O)(=O)(CC(=O)NC(C)C(C(C)C)SC)NCC.c12cc([nH]n1)CN2 c1(CC)cnc(C(N2CCC(C)C2C(=O)N(C)Cc2ncccn2)=O)nc1 N1(C(C(C)SCC)=O)CC2(C(=O)NCCCc3nc(C)no3)CC1CO2 c1(C(N2C(C)CC(NC(C3(CC#C)CCCC3)=O)C2)=O)cc(Cl)cc(F)c1N CCCCC(CNC(=O)COCC(C)C)NC(c1ccnn1C(C)(C)C)=O c1(NC(N(CCC)CCN(C)C)=O)ccc(OC(C)CC)c(Cl)c1 c1(C(N(CCNC(=O)C(C(C)O)NC(N)=O)CC)=O)ncc(Br)cc1N C1(C(C(N2CC(=CCC)C2)=O)NC(=O)CSc2cn[nH]c2)CC=CCC1 N1(C(C(CC)n2nccc2C)=O)CCN(C(=O)C(N)=O)CC1CC1CC1 c1(C(N2CC(C)CC(NC(c3ccc(CC)s3)=O)C2)=O)cccc2[nH]ncc12 C=CCC(C(=O)NC1CCCN(CC(O)C2CC2)C1)NC(=O)OC(C)(C)C C12(CNC(c3ccsn3)=O)CCC(CNC(c3nc(C4CC4)cs3)=O)(CC1)CO2 c1(NC2CC(CC(C)(C)C)C2)nccc(=NCc2cccc3[nH]ncc23)[nH]1 Cc1c(C(=O)NC2CC2NC(=O)CC2(O)CCCOC2)oc2ccc(Cl)cc12 c1(C(=O)NCC2C(NC(c3c(C)cn(C)n3)=O)C2)cc(F)cc2cccnc12 c1(OCC)cccc(CC(=O)N(CC(O)CN(C)C(C2CSC2)=O)C)n1 CC1CN(Cc2ccccc2)CC1COC(c1c[nH]cc1-c1ccc(Cl)s1)=O C1(N(C(=O)CC2(C)CNC(=O)C2)C)CCCN(C(C2CCCC2)=O)CC1 Cc1ccn2ncc(C(=O)NC3(C4CCN(C(C5CC5F)=O)C4)CC3)c2c1 c1(C(N2C(CCC(=O)Nc3n(C)cc(Br)n3)CCC2)=O)ccc2[nH][nH]c(=N)c2c1 Cc1cc(NC(=O)C(C)OC(=O)Cc2cscn2)ccc1C(C)C C(=O)(C(CC(C)C)NC)OCC1CCCC(c2nccn2Cc2ccc(F)cc2)O1 C(c1ccc(Cl)s1)=CC(N1CCC(N(C(=O)CCNC(=O)NC)CCC)C1)=O N1(C(C(C2CN(C(CC(C)(C)C3CC3)=O)C2)O)=O)CC2CCC(C1)C(=O)N2 C1(N(C(=O)NC(COC)CO)C)CC(=O)N(C(C)(C)C)C1=O C1(NC(c2cc3cccnn3n2)=O)C2CC3CN(C(c4ccsc4)=O)C1C3C2 c1(OC)ccc(C)cc1C=CC(=O)NC(CCN(C)C(C1(C)CC1)=O)C(C)(C)C c1(C(CC)=O)ccc(N(C2CC2OC)Cc2ccccc2)c([N+](=O)[O-])c1 C(=O)(C(CC#CC)NC(c1cc(C)c[nH]1)=O)NCC1(CCC=C)CC1 C(=O)(C(C(C)C)c1ccn(C)n1)N1CC(F)(CNC(COCCCC#C)=O)C1 C1(NC(c2nccc(C)c2)=O)CC2CN(C(=O)C(C)C3CCOC3)CC12 C(=O)(N=c1[nH][nH]c(C)c1Cl)c1c(-c2cc(OC)c(C(F)F)cc2)ncs1 c1ccc(C(C)O)cc1.C1(C(=O)NCCOCCN(C=O)C)CCCN1N=O C(C1=CCN(c2ncccc2F)CC1)NC(c1ccc(CC)s1)=O c1(C(=O)NC2CC2)cccc(-c2ccccc2F)c1.O=C1C(=O)NCC2C(C2)CN1 N1(C(C=CC)=O)CCC2(CCCCN(C(=O)COCC3CCCCO3)C2)C1 C1(NC(C2N(C)C(=O)OC2)=O)CN(C(c2ccc(Cl)s2)=O)C2(CCCCCC2)C1 C1(CNC(C=CC(=O)OC(C)(C)C)=O)CN(C(=O)CC2(C)CC2(C)C)CCCO1 CC1C(=O)N(CC(N2CC(CCCCNC(c3cccnn3)=O)C2)=O)C(=O)C1C C12(C3CN3)CCC(CC1)C2.c1(C(C)NC(=O)C(N)=O)ccn(C2CCC2)n1 Cc1cccc2[nH]c(C(N3CC(NC(=O)C=Cc4cccnc4)C3)=O)cc12 C(CNC(=O)C(C(C)C)OC)(C(C)(C)C)NC(c1c(COC)cc[nH]1)=O C1(C(N2CCOCC(CNC(C(C(COC)C)C)=O)C2)=O)CCC2(C1)CC2(F)F CCCCC(C)C(=O)NCc1ocnc1C(=O)NCc1nn(CC)cc1Cl N1(C(c2c(CCC)nns2)=O)CCCC(C)C1CNC(=O)CC=CC(C)(C)C C(=O)(C(C)(C)C1=CCN(C(c2c[nH]nc2C)=O)C1)NC(CCN(CC)CC)C C(CCCC(C)NC(c1ccc(-c2cccnc2)cc1)=O)NC(C(CC)SC)=O c1(C(=O)NCCN(C(=O)CNC(N)=O)C(C)C)cc(C(F)(F)F)cnc1N C1(C(N2CC(C)C(CNC(=O)CCS(N)(=O)=O)C2)=O)CCC(C2CCCO2)O1 c1(CNC2CC(C(=O)NC3CC3(F)F)C2)cc(Cl)cc(Cl)c1O c1(NCc2cc(C(C)(C)C)sc2)ccc2c(=O)cc[nH]c2c1 c1(C(N2CCN(C(c3c(C)n(C)cn3)=O)CC2CCO)=O)ccn2ccnc2c1 N1(C(Cn2cnc(C#N)n2)=O)CCCC(NC(C2(O)CCCCCC2)=O)CC1 c1(C(OC)OC)ccc(C#N)c([N+](=O)[O-])c1.c12oc(C)nc1C=Cc1nc-2no1 C1(SCC(C(=O)OCC=C)NC(=O)C2CC2)CCCC(C(F)(F)F)O1 N1(C(C(C)CC(F)F)=O)CC2(CC(C(=O)NCC3(CO)CCC3)CO2)C1 C1(C(=O)NC2(C)CC(NC(C=Cc3ccc(C)cn3)=O)C2)Cc2ccccc2C1 C1(CN(C(C(CC)N(C)C)=O)C)CCCCN1C(=O)CN(C)C(=O)OC(C)(C)C c1(C(=O)NCC(CC)NC(C(CCC)CC)=O)c[nH]c2ccncc2c1=O N1(C(CC(C)C2CC2)=O)CCC(C)CC1CNC(=O)C(F)(F)c1cnn(C)c1 C1(NC(c2c(C)[nH]cc2)=O)CN(C(C23CCC(CC2F)C3)=O)CC1C1CC1 CCC(CC(=O)NC1CC(NC(c2cc(Cl)c(Cl)[nH]2)=O)C1)C1CC1 n1(CC)nc(C)cc1C(N1CC(C)(NC(c2ccc(C(C)C)s2)=O)C1)=O c1(C(C(=O)NCC)N(CCOC)CC2CC2)nc(Cl)cs1 c1(NC(C2C(C(=O)NCCCN3C(C)CCCC3)C2)=O)ccc(Cl)c(C#N)c1 C#CC1(NC(C23CC(C)(CN2C(=O)C(C#N)C(C)(C)C)C3)=O)CC2CCCC12 C1(C(=O)NCCN(C(=O)C(F)=CCCF)C2CCCC2)CCCN1c1ncccn1 c1(C(N2CC(F)(CNC(C=CC(=O)N(C)C)=O)C2)=O)cccc(CO)n1 c1(NC(C(c2ccccn2)C)=O)ccc2c(c1)OCC(=O)N2 C=CCC(CC(=O)NCC1CCCCS1)NC(C12CC(C)(CCO1)C2)=O C(=O)(N=c1[nH]nc(-c2cccc(C)c2)s1)N(CC(C(=O)NC)(C)C)C1CC1 N1(C(c2c(C(C)=O)csc2)=O)CCC2(CCOCC2)C(CNC(=O)CNC=O)C1 C1(CCNC(C2(OC)CCC2)=O)CCCN1C(=O)C(C)CC1CCCCC1 Cc1ccc(CC(N2CCCC2CNC(C2CCC3CC23)=O)=O)cc1[N+](=O)[O-] c1(CC(C)NC(c2n(CC=C)nnn2)c2cnccn2)ccc(Br)cc1 c1(OCC)ccc(C(=O)NC(C)C(C)NC(=O)C=CC2CCCC2)cc1Cl C(=O)(CC(CC(N)=O)CC(C)C)N1CC2C(CNC(CC3CC(=C)C3)=O)(CC2)C1 C1(C(=O)NC2CCCN(C(C(C)n3cnnn3)=O)C2)CCn2cnnc2C1 N1(C(C2C(C)C2C)=O)CC(NC(c2cn(CC3CC3)nn2)=O)CC1(C)C C1(NC(C2(OC(C)=O)CC2)=O)CCOCC1C(=O)N(C1(CCO)CC1)C N1(C(CC)=O)CCc2ccc(S(=O)(=O)N3CC(Oc4ccc(O)cc4)C3)cc21 C(=O)(C(N=[N+]=[N-])C(C)C)N(C1(C(=O)NC(C(=O)NC)C)CC1)C c1(OC)cc(CCC(=O)NC(C)(CNC(c2cccs2)=O)C2CC2)ccc1Cl C(CNC(c1cc(C2CCC2)nn1C)=O)(C(C)C(C)C)NC(CSC)=O C(c1cn(CC2CCN(C(=O)Cc3cscc3Br)CC2)nn1)=CC c1(C(=O)OC(C(C)=O)C(C)C)cc(F)c(C)c([N+](=O)[O-])c1 C1(N(C)C(c2ccc[nH]2)=O)CN(C(c2ccnc(NC3CCC3)c2)=O)CC12CC2 Cc1cccc2oc(C(=O)NC(C3CCN(C(C4(C)CNC(=O)C4)=O)C3)C)cc12 N1(C(C=Cc2ccn(C)c2)=O)CCCCC(NC(c2cc(Cl)ccc2Cl)=O)CC1 c1(CN(c2cc(CO)sn2)C(=O)CC2(SC)CCCO2)cccc2cccnc12 c1(C(N2CC(OC)(CNC(C3(C4CCCCO4)CC3)=O)C2)=O)cc(C)ccc1C N12CCn3cc(nc3C1)C(=O)CC2=O.C1(NC(C=C)=O)CCN(S(C)(=O)=O)CC1 C1(C(=O)NCCC(COC)(C)O)CN(C(c2cc(C(C)=O)[nH]n2)=O)CC12CC2 N1(C(c2c(C)nsc2N)=O)CCCC(F)(CNC(=O)C(F)CC2CCC2)C1 C1(CC(N2CCC(OCC#C)C2)=O)CN(C(c2cc(F)c[nH]2)=O)CCC1C c1(NC(=O)NCc2c(CC)cccc2F)ccc2c(c1)C(=O)OC2(C)C N1(C(c2c(N)cncn2)=O)CC2CC(C1)N2C(=O)C1=CCOCC1 c1(C(=O)NCC2(C(=O)Nc3cc(O)cc(O)c3)CC2)cc2c(F)cc(F)cc2[nH]1 C(=O)(C1=CC2CCCC12)N1C(CNC(c2c(C)occ2)=O)CC(F)(F)C1 CN1CC2OCCN(C(C3CCN(C(C4C5CCCC45)=O)CCO3)=O)C2C1 C1(NC(CN(C)C(=O)C2CC2)=O)CC2CC(NC(C3(C(F)F)CCCC3)=O)CC12 C1(O)(C(C)NC(=O)C2=CCC2)CCN(C(=O)C(=O)Nc2ccccc2)C1 C1(C(=O)NCC(N(C(c2cccc(C)n2)=O)C)C2CC2)CC2(CCCCC2)C1 CS(=O)CCC(O)C(=O)NCC1(c2nnnn2CCCC2CC2)CC2CCCC12 c1(C(=O)NCCc2ccc(C(=O)NCC3(O)COC3)cc2)cc(F)c(Cl)nc1Cl C(CCCCNC(c1cnc(C(C)C)[nH]1)=O)NC(C(C)OCC=C)=O C(=O)(CCCC(=O)NC1CC(CNC(=O)COc2cnn(C)c2)C1(C)C)N(C)C CCC(C(=O)NCC(C(C)C)NC(=O)Cc1nc[nH]n1)C1CCOCC1 C1(C)(C(=O)NCC2(C)CCN(C(=O)CCCCC3CC3)C2)CC(C2CC2)=NO1 c1(CNC2CCC(C(=O)Nc3ccc(CC)cc3O)C2)c(O)ccc(F)c1F c1(NC(CNC(c2n(C(CC)CC)ncc2)=O)C2CC2)nc(C)nc2sccc12 C12(C(N(CCC(N)=O)C)=O)CCC(NC(=O)CN3CC4CC4C3)(CC1)C2 c1(C(N2CCC(NC(c3c(C)cnnc3)=O)C2)=O)csc2c1CCC(C)C2 c1(C(N2CCCC(O)(C(=O)Nc3cnn(CC(F)F)c3)C2)=O)cnc(O)c(Br)c1 CC1(C)CC(C(=O)NCC2CNC(=O)O2)CCN1C(c1c[nH]c2cnccc12)=O c1(CC(=O)NCC(O)CNC(=O)C(O)CC2CC2)cc2nc[nH]c2cc1Br C1(N(C)C(c2ncccn2)=O)CN(C(C2CC(=O)C2C(C)(C)C)=O)CC12CC2 N1(C(C(C)CC2CC2)=O)CCC(NC(=O)CSc2ccc(O)cc2)C(C)(C)C1 c1(C(=O)NC(CNC(C2C(=C)C2)=O)CCCC)cc(NC)cc(F)c1 c1(C(=O)NC(C(=O)NC(c2nnc(O)o2)C)(C)C2CCC2)ncc(F)cn1 c1(C(=O)NCC(C)N(C(CCC#C)=O)C)ccc2c(n1)NCC2 Cc1cc(F)c(C(N2CC3CC2CCN3C(=O)C=CC2CCCCC2)=O)c(F)c1 C(=O)(N=c1cc(OC)n(C)[nH]1)C1C(CC)CN(C(C2CC3(CCC3)C2)=O)C1 C1(CNC(C(C)OCC)=O)CCCC(NC(=O)C=CC2(C)COC2)C1 N1(C(COCC(C)C)=O)CC(F)(F)CC1CCNC(=O)CC(O)CN(C)C c1(CCC(=O)NCC(C)NC(C2CCc3ccnn3C2)=O)ccc(F)c(F)c1F N1(C(C(C)C#N)=O)CCC(F)(F)C(NC(=O)COc2cccc(F)n2)C1 C#Cc1ccc(C(N2CC(NC(c3csc(=N)[nH]3)=O)C(CC3CC3)C2)=O)cc1 CC1CN(C(=O)CCCOc2ccccc2Br)CCN1C(C1CC1C)=O S(=O)(=O)(c1cc(C(=O)NC(C)C(C)NC(c2ccc(SC)o2)=O)co1)NC c1(C2(C(=O)NCC(CO)NC(=O)CC3(O)CCC3)CC2)ncco1 CC1CCN(C(=O)Cn2cnc(=N)[nH]2)CC1C(=O)N(c1cccc(Cl)c1)C C(=O)(C(Cc1ccccc1C)CC)NCCCC1(NC(C(C)OCC)=O)CC1 c1(C(N(C)CC2CCCN(C(C=CSC)=O)C2)=O)c(Cl)cccc1[N+](=O)[O-] C=CC(C)(C)CC(=O)N1CCC(CNC(=O)C=C(C)CN2CCOCC2)C12CC2 c1(C2(NCC(C)CCc3ccccc3)CCC2)cccc(NS(C)(=O)=O)c1 c1(C(=O)NCC(C)NC(C(COC)OC)=O)ccc2[nH]ccc2n1 N1(C(C(C=C)OC)=O)CCCC(CCNC(c2ocnc2C(C)C)=O)C1 CC1(C)CN(C(=O)CC2CCC(=O)NC2)CC1CNC(=O)C(=O)NCC(F)F N1(C(C(C=C)(C)O)=O)CCCOC(CNC(c2ccc(Br)c(O)n2)=O)C1 N1(C(c2c(COC)nn[nH]2)=O)CCC(CNC(C2CCC(C)(C)OC2)=O)C12CC2 N1(C(C(C)NC(CC)=O)=O)CCCC2(CC(NC(=O)CCC3CCOC3)C2)C1 N1(C(c2cc(CC)on2)=O)C2CCC1CC(N(C(=O)C=Cc1cccn1C)C)C2 c1(CNC(C2(CC#C)CC2)=O)cccc(C(=O)NCc2cncn2C)n1 CCC(CC)C(C)C(=O)N1CCCC(C)(C(N2CCC(F)(F)C2)=O)C1 CC1(C)C2CCC1(C(=O)NC1CN(C(c3conc3C3CCC3)=O)CC1F)C2 N1(C(C(CC)Cl)=O)CC2(CCN(C(C3C4C=CSC34)=O)CC2)c2ccccc21 N#Cc1cc(NC(=O)NCC23CC4CC2C3C4)ccc1N1CCCC1 c1(OC)ccccc1C(=O)NC1COCCC1C(=O)N(C)Cc1cccc(O)c1 CC1(C)CC(Nc2ncnc3ccsc23)CN(C(=O)C(Cc2ccccc2)S(C)(=O)=O)C1 C1(CNC(C(c2ccccc2)C)=O)CC(O)(CNC(=O)CN2CCOCC2)C1 CC1CCN(C(=O)Cc2ccsn2)C(C(=O)NC2(C3CCCCO3)CC2)C1 C1(CNC(=O)COCC(F)F)CC2(CC2)CN1C(c1ccc(C(F)F)cn1)=O C1(NC(CN(CC#C)C(C2C3(CC3)C23CC3)=O)=O)(CO)CCC(C)(C)C1 C(=O)(CC(C)(C)OC)N1CCC(CCC(=O)N(C(CC)C)C)C1 C(=O)(CCCCCNC(C1CCCC(=O)C1)=O)NC(CC#C)C(N)=O c1(SCC(N2C(C(N(CC=C)Cc3ccccc3)=O)CCC2)=O)ccccc1C c1(C(=O)NC(CNC(C(C#C)(C)C)=O)(C)C(C)C)nn(C)c2c(=O)[nH]cnc12 N1(CCCOCC)CCN(c2ccnc(NC3CCCN(CCCO)C3)n2)CC1 Cc1cc(CC(=O)NCC2CCC2NC(c2ncncc2F)=O)cc(F)c1 N1(C(C(CCCNC(CNC(C2C(C)C2)=O)=O)O)=O)CCCC2(CC(O)C2)C1 C1(C(N2C(CC)(CC)CC2)=O)CCN(C(c2ccoc2Cl)=O)CCO1 C(=O)(C1=CC2C=CC1C2)N1CCCCC(N(C(C(CCCC)C)=O)C)C1 N1(C(C2N(C)CCC2)=O)CC2CC1CN2C(=O)C(c1cccnc1)O CCCCCC(O)CC(=O)NC(C)CCCC(=O)NCC=CCl N1(C(CNC(=O)OC)=O)CCC(NC(C2CCOC2(C)C)=O)C2(CCC2)C1 Cc1oc(CNC(=O)C(F)C2CCOC2)nc1C(N1CCCC(C(N)=O)C1)=O c1(CC)c(C(=O)NCC2(C)CCN(C(=O)CN3CCCC3CO)C2)nnn1CC C1(NC(c2ncc(C)nc2)=O)CN(C(=O)CCc2nccs2)CCC1C C(=O)(C1CN(C(=O)OC(C)(C)C)Cc2ccccc21)OCC#C N1(CC(N2CC(CC(=O)NCc3cc[nH]c3)C2)=O)CCC(C(=O)OC)C1 C(=O)(C1=CCC2(COC2)OC1)N(C(C)CNC(=O)C(C)(C)C(F)(F)CC)CC C1(C)(NC(CSCC(=O)NCC(C)(C)CNC(C)(C)C)=O)CC2CC2C1 C1(CNC(c2cn(C)nc2C2CC2)=O)CC2CCC1N(C(=O)CC1OCCO1)C2 C1(CNC(CN(C(COC)=O)C)=O)CCN(C(=O)CN2CCC2)C12CC2 CC1(C)CCN(C(C2CC3(CCC3=O)C2)=O)C1C(=O)NCc1ccnc(CO)c1 C(C1=NOC2CN(C(c3cc(C(=O)OC)sc3C)=O)CC12)NC(CC=CCC)=O c1(OC)cc(CNC(=O)NC(COC(F)F)CO)c(F)cc1Br C1(=CC(=O)NC(C)C(CO)NC(c2cnc(N(C)C)o2)=O)CCCCC1(C)C N1(C(C2(n3cc(CCCCCCC)nn3)CC2)=O)CC(CC(=O)O)OCC1(C)C c1(C(N2C(CC)C(NC(=O)COC3(C)CCC3)CC2)=O)ccc(F)c(C(F)F)c1 c1(C(N2CCC(NC(C(COC)OC)=O)(COC)C2)=O)cn2c(n1)CCC2 C1(C(=O)NCCC(C)N(C(c2ccc(CC)[nH]2)=O)C)CCOC(C)(C)C1 C1(C(=O)OCC)Cc2ccccc2N1C(C1CCC(C(=O)NC2CC2)CC1)=O C=CCCCCCC(=O)NCCCC1(NC(c2ccccc2)=O)CC1 N1(C(COCCCC)=O)CCCC(C)C1CCNC(=O)CC(F)(F)F C1(CC)CC(CC(=O)OC(c2ccc(Br)cc2)C(C)(F)F)CCO1 Cc1cc(NCC2C3CN(C(C4(O)CCC(C)CC4)=O)CC23)ncc1[N+](=O)[O-] C12(OC)CCCCC(C(N3CC(N(C(=O)C(c4ccc(C)cc4)C)C)C3)=O)(C1)C2 C1(C(=O)NCC(CC)(CC)NC(=O)CC(C)C(=O)OC)CCc2nnnn2C1 C1(C(COC(CCC(c2ccc(OCCC)cc2)=O)=O)=O)CCCC(F)(F)C1 N1(C(C2C=CCN2Cc2ccc(Br)cc2Cl)=O)C2CCC1CC(O)C2 C=CCCCC(=O)NC(C)C(c1ccc(OC)cc1)NC(c1ccc(CO)o1)=O C12(CC)CN(C(c3cnccc3C)=O)C(CNC(=O)C(F)C3CCOC3)(C1)C2 N1(C(CCn2cc(-c3c(N)ccc(OC)c3)nn2)=O)CCC2(CCC2)C(O)C1 c1(C(=O)NCC(C(C)(C)C)NC(CC(C)(C)C)=O)cc(S(=O)(=O)N(C)C)c[nH]1 C1(CCNC(C(C)N(C(=O)Cc2ccsn2)CCC)=O)CC(=O)N(C)C1 O=C(C1=CS(=O)(=O)CCC1)NCC1CCCC1NC(c1cc2sccc2cn1)=O Cc1ccnc2sc(C(=O)NCC(C)NC(=O)C(F)(F)C(O)C(C)C)c(C)c12 Cc1cc(N)ccc1C(N1CCCC1C1CCCN(C(=O)Cc2cnoc2)C1)=O c1(C(=O)NC(CCNC(C2N(C(C)C)C(=O)CC2)=O)C)nnn2c1CCCCC2 N1(C(C=CCOCCOC)=O)CCC(O)(CN(C)C(C2CCC(C)C2)=O)CC1 CCCC(F)C(=O)NCCC(CNC(C1CC(C)(CC)C1)=O)OC CCCC(C)(c1nnnn1C1CC(F)(F)C1)NC(C1CSC1)C c1(C(=O)NC(CC)(C)CNC(=O)Cc2nc(C)c(C)[nH]2)cc(Cl)cnc1O C1(C(=O)NCc2occ(C(=O)NC3(CO)CCCC3)n2)CCC=CCC1 c1(OC)ncc(C(=O)NCC(C2CCCN2C(=O)CSC(C)C)(C)C)cc1Br c1(OC)cccnc1C(F)(F)C(N1CCC(O)(C(N)=O)C1)=O N1(C(C(C)(C)OCCC)=O)CC2C(C(N3CCC(C(F)(F)F)CC3)=O)C2C1 c1(C(C(=O)Nc2c(C)cccc2C)N(CC=C)C(C)C)cc(C(F)F)cc(C)c1 C(C)(CCCCNC(c1csc(COC)c1)=O)NC(c1n(CC)ccc1)=O C(N=c1[nH]c2c(c(=NCCCC(C)CO)[nH]1)CCC2)c1c(C)nc(CC)o1 c1(OC)ccc(OC)c([N+](=O)[O-])c1C(=O)NC1CC1C(=O)Nc1ccsc1 C(C)(CCC(=O)N1CCCC1C(=O)NC(C)CC(C)C)OC c1(NC(C2(NC(C3CCCN(C)C3)=O)CCOCC2)=O)cc2n(n1)CCNC2=O c1(CC)nc(=NCc2cccc(CNC(C3CC3C3CC3C)=O)c2)s[nH]1 c1(NC(C(C(CC)CC)C)=O)nccc2c(C)cccc12.C12C3CN(CC13)C2=O C1(CNC(C2C=C(C)CS2)=O)(NC(=O)CC2CCCC(O)C2)CCCCC1 C(c1ccc(C)cc1)=CCC(=O)NC1C(NC(c2c(CC)noc2)=O)CCCC1 c1(C(N(C2CCC(NC(C3(CC#C)CC3)=O)C2)C)=O)cccc2c1CCCC2 C12(NC(COCCC=C)=O)CCCCCC1N(C(c1nn(C)c(Cl)c1Cl)=O)CC2 C1(NC(CC(C)C2CC2)=O)CC2(CCN(C(=O)Cc3ccc(O)nc3)CC2)C1 c1(C(=O)NCC(C)(C)NC(C2C(C(C)C)OCC2)=O)ccnc2ccnn12 C(=O)(CC(=O)NC1CC1)NCC(C)(C1CC1)NC(C12COCC1C2)=O c1(C(N(CC(C)N(C(C2CCC(C)O2)=O)C)C)=O)nn(C)cc1S(N)(=O)=O c1(Cc2cn(CC3N(C(C4(C5CC5)CCCO4)=O)CC=C3)nn2)ccc(F)cc1 N1(C(c2ccn(COC)n2)=O)CC=CCC1C(N1CCC=C(C)C1)=O C1(NC(=O)COCCF)CC2CN(C(c3ncccc3SCCO)=O)CCN2C1=O c1(NC(=O)CCCn2ccnc2C)cnc(C)[nH]c1=N.C12(COC)CN(C1)C2=O CC(C)C1=NOC(C(=O)N(C2CN(C(=O)C=CBr)CC2(C)C)C)C1 c1(C(N(CC(C)CNC(=O)CCC2CCCO2)C)=O)cccc(OCC2CC2)c1 Cc1cccc(C(O)C(N2CC(CNC(=O)Cc3cn(C)cn3)C(O)C2)=O)c1F C1(C(=O)NCC=CCNC(c2c[nH]c3cccnc23)=O)CCc2nnnn2CC1 N1(C(c2sc(C)c(O)n2)=O)CC2CN(C(c3c[nH]nc3C(C)(F)F)=O)CC2(C)C1 C(=O)(CC(O)CN(C)C)NC(CN(C(c1cn(CC=C)nn1)=O)CC)CC OC1(c2ccccc2Nc2nccnc2F)CCNCC1 C(CCCCC(=O)NC1CCCCN(C(C2C3CCC2CC3)=O)C1)N(C)C CCC(CC(C)C)C(=O)N1CCN(C(C2(F)CCN(C)CC2)=O)CC1C1CC1 CC(CCC(=O)NC1(CF)CCN(C(=O)C(C2CC2)C2CC2)C1)N(C)C CC1CN(C(c2cc(C3(C)CC3)n[nH]2)=O)CC(C)C1NC(c1coc(CO)c1)=O C=CC1(c2cn(C(C)CO)nn2)COCCN1Cc1cccc(CC(=O)OC)c1 C1(O)(C(C(=O)N(CCN(C(=O)CC2CC(N(C)C)C2)CC)CC)F)CCCC1 C1(CC(=O)NCC2CC(CNC(CC(=O)NCC#C)=O)C2)CC(=O)NC1=O c1(C(N(C(C)CCNC(C2(C(C)(F)F)CC2)=O)C)=O)ccn2nnnc2c1 C(=O)(CC(C(F)(F)F)OC)N1CCN(C(CS(=O)(=O)NC)=O)CC1c1cn[nH]c1 c1(C(=O)O)cccc(S(=O)(=O)N2CC3C(C(=O)NC(c4cccs4)C4CC4)C3C2)c1 C1(C)(C(=O)OCC)CN(C(=O)NCC2CCC2)C(C)(C)C1.C(CCC(=O)N)NCCO CC(C)C(C)(F)CNC(=O)C(Cn1cncn1)NC(=O)COCC(F)F c1(CNC(c2c(C)n3c(s2)cnc3)=O)ccc(F)c2c1CCC2 C1(NC(c2coc(C3CCOCC3)n2)=O)COCC1CNC(C1(CO)CC1)=O C1(C(=O)NC(CCO)C(F)F)(CC)CCCN(C(=O)COCCC(C)C)C1 C1(CCNC(COCCN(CC)CC)=O)(NC(=O)CCC(=O)OC)CCOCC1 C(CCCC(=O)NCC1(C)CCCOC1)N(C(COC)=O)C C(C(C)(C)CNC(=O)CN1CCOCC1)C1CN(C(COC(CC)C)=O)C1 C1(C(=O)NCC(C)(O)CNC(=O)CC2CCOCC2)CCOC(=O)N1 Cn1c(C(N2CCN(C(=O)C3=CC4CCCC34)CC2CO)=O)cc2ccccc12 c1(CC(=O)NC(CCNC(CN(CCNS(CC)(=O)=O)C)=O)C)cc(C)[nH]n1 N1(C(CCNC(=O)OCC)=O)CC(C(=O)NCC2C(CO)C2(F)F)CC1(C)C c1(CNC(C(CSCC)NC(=O)CC(C)O)=O)ccnc(C)n1 C1(C(=O)NCCOC)CCC(CNC(=O)C(c2c(C)n[nH]c2C)C)CC1 CC1(C)COC(CC(=O)NCCN(C(=O)Cc2csc(Cl)n2)C2CC2)C1 C(=O)(C1=Cc2ccccc2C1)NCC1N(C(C2C(C#N)C2)=O)CC2(CCC2)CC1 C1(O)(CC(=O)NCC2(CCNC(C3CC4CC3C4)=O)CC2)CCCC1 C12C3CCCN(C3C1(C)C)C(=O)N2.Cc1nnc(Cn2cc(CN(C)C)nn2)o1 N1(C(C2C(C)=CCC=C2)=O)CCc2sc(C(N3CCC(C)C(O)CC3)=O)cc2C1 CCC(C)(C)C(=O)NC1CCC(NC(c2nc(C(F)(F)F)cn2C)=O)CC1 C(=O)(C(F)(F)C(O)C(C)C)NC1CN(C(CCCCOCC)=O)C(C)CC1 c1(C2C(C(NOCC(CC)C)=O)C2)ccc(C(=O)OC)nn1 N1(CC#C)CCC(N(C(c2cc(CC)[nH]n2)=O)CC)C1 N1(C(C(C)F)=O)CCCCC1Cn1cc(-c2cccnc2Br)nn1 CC(Cn1cccn1)C(=O)N1CCC(CCNC(C2CC(C(F)(F)F)C2)=O)C1 N1(C(C(CCC)O)=O)CCN(Cc2ccccc2)C(CNC(c2cnn[nH]2)=O)C1 C#CCCCC(C)C(=O)NC(CCN(C)C)C(=O)NC(C=C)COC c1(C(=O)N)cccc2cc[nH]c12.c1(CC)nc(C)c(CNC(c2ccc(C)s2)=O)o1 CC1CN2CCN1C(C(=O)NCCN(C(C1CC(C)(C(C)(C)C)C1)=O)C1CC1)C2 C#CCCCCC(=O)NCCCOCCNC(C1CCN(CC(F)(F)F)C1)=O C(=O)(CC(CC)N(C)C(c1ccc(C#N)s1)=O)NC(C1CCCO1)CC C1(CC)CCN(C(=O)CCOCCCOC)C1CNC(=O)CS(C)(=O)=O N1(C(c2nnn(C(C)(C)C)n2)=O)CCCCCC1CNC(c1coc(Cl)c1)=O N1(C(C(=O)NCC)=O)CCCC(C)C1CNC(=O)C(C)(C)c1ccccc1 C1(C)(C(=O)NC(C)CCNC(c2ccc(-c3ccncc3)o2)=O)CC(C#N)C1 N1(C(C2C(C=C)CC2)=O)CCCN(C(c2cccc(Cl)c2C(F)(F)F)=O)CC1C n1(CC)cc(C(c2nnnn2Cc2ccccc2)NCCn2cc(Cl)cn2)cn1 C12(C(=O)NCC(C)(CNC(C3(C)CCCCC3C)=O)OC)CC3CC1C2C3(F)F c1(C(N2CCN(C(Cn3ccc(C)n3)=O)C3C2CC3)=O)cnc2nccnc2c1 C(=O)(C1CCCc2c1ncn2C)N1CCC2(CCN(C(C(OC)OC)=O)C2)CC1 CCCC(C(=O)NCC=C1CCN(C(c2nnsc2C)=O)CC1)NC(C)=O C1(NC(COCCC=C)=O)CCCC12CCN(C(C1CCCC(C)C1)=O)CC2 c1(C(=O)NCC(CNC(C(CC)n2cncn2)=O)(C)O)ncc2n1CCCC2 N1(C(C2C3C=CSC23)=O)CCC2(CCC(C(N3CCCSCC3)=O)O2)CC1 c1(C(=O)NCC2CC(NC(C3C(=C)CC3)=O)C2)cnoc1C(C)C C1(C(N2C(C)(C(N3CCC(OC(C)=O)C3)=O)CCC2)=O)CC(C(C)C)=NO1 CC(C)(C)CC(O)CC(=O)NCC1CCN1C(c1ccc(Cl)cc1OC(F)F)=O c1(SC)ccc(NC(=O)CC2CCCC2NC(c2cnc(C3CC3)o2)=O)cn1 N1(C(CC)=O)CSCC1C(N1CC(COC)(NC(=O)COC2CCCC2)C1)=O C(CCN(C)C(C1(C)CC2CCC(C1)S2)=O)(C(C)(C)C)NC(CNC(CC)=O)=O c1(CC(=O)N(C2CC(C(NOC(CC)C)=O)C2)C)ncccc1C N1(C(c2c(C)cc(C)o2)=O)Cc2ccnn2CC(NC(=O)C(C)CF)C1 n1(CC(N2CC3CC(C2)C3NC(C2CC2F)=O)=O)nc(C(F)(F)F)c2c1CCC2 C(=O)(CCCCCSC)NCC1(C(C)(C)C)CCN(C(C(C)NC(CC)=O)=O)C1 c1(C(N2CCC(O)(CCNC(C3CC34CC(O)C4)=O)C2)=O)nccc2[nH]ccc12 CC(C)C(C(=O)NC(C)(C(=O)NCc1noc(C(N)=O)n1)C1CCC1)C1CCC1 CC(C)C(C(=O)N(C)CCN(C)C(C1CCCC12CC2)=O)C1CCC1 N1(C(CCCOCCC)=O)CCC2OCCN(C(=O)CN3CCC(C)C3)C2C1 C12(CNC(C(C)OCC)=O)CCC(CC1)N2C(c1cc(N)nc(Cl)c1)=O Cc1ccc(CC(=O)NC2CC(C)CN(C(=O)CN(C)C3CC3)C2)cc1C C(CC1=CCN(C(=O)CC(C(F)(F)F)N2CCCC2)CC1)NC(C(C)OCC)=O c1(C(N(CCCCCNC(=O)Cc2cnc[nH]2)C)=O)nc2ccccc2cc1Cl C1(NC(CC2(OC)CC2)=O)CCCCN(C(C2CN(C)CCO2)=O)C1 C1(C(=O)NC2(C)CN(C(CN(C3CCC3)C)=O)C2)C(F)(F)C12CCC2 CC1CN(C(c2c[nH]nc2C2CC2)=O)CC(C)N(C(=O)C(F)=C2CCCC2)C1 C(c1nc2ccccc2s1)=CC(=O)N(CC1N(C(C(C(C)C)F)=O)CCC1)CC CN1CCC(C)(C(N2CC=C(CNC(C3CC4CCCCC34)=O)CC2)=O)C1=O N1(C(c2c(C#N)cc(F)cc2)=O)CCC2C1CCCN2C(C1CCC(O)CC1)=O c1(CC)ccccc1C(F)(F)C(=O)N(CCNC(=O)C=CCO)C(C)C C1(CNC(C2(C)CSC2)=O)CN(C(c2c[nH]c(=N)s2)=O)CCO1 c1(C(=O)NC2CN(C(c3c(C)cc(C)nc3)=O)CC23CC3)ccc2cc[nH]c2c1 C1(CNC(C2(CNC(c3n(C=C)nnc3)=O)CC2)=O)CCCCC1(C)C CC(C)C(C)CN(CCC(=O)N(C(c1ccccc1)CNC(C1(O)CC1)=O)C)C CC1(NC(c2ccoc2C2CC2)=O)CCCCC1C(=O)NOCCN(C)C C(=O)(C1=CC2(CCOC2)C1)NCC(CNC(c1cnc(CC)nc1C)=O)(C)OC C#CCC(C)C(=O)N1CCCC(N(CCO)C(c2cnnc(O)c2)=O)C1 N1(C(C(C=C)(C)O)=O)C2CCC1CC(CNC(=O)CC1CCOC(C(C)C)C1)C2 C1(CC)CCCCC1C(=O)NCC1(CCNC(=O)CCN2CCOCC2=O)CC1 C1(NC(C(CNC(C2(OC)CCC(C)C2)=O)OC)=O)COCCC1(F)F c1(C(=O)NCC(=C)CCNC(C2CCCC2O)=O)coc2c(OC)cccc12 c1(CC(=O)NCC2(O)CN(C(CC(C)C3CCCO3)=O)C2)ccc(Br)cc1 c1(C(=O)NC2CCCC(CNC(C3(N(C)C)CC3)=O)C2)cc2occc2[nH]1 C1(c2n(C)nnn2)CCN(C(C2CC(Oc3ccccc3)C2(C)C)=O)CC1 c1(NC(=O)NCCC2(C)N=N2)ccc([N+](=O)[O-])c(OCc2ccccc2)c1 N1(C(C(COCC)C)=O)CCC(C)(C)C(C(N2CC(N(C)C)C(C)(C)C2)=O)C1 c1(CC)ccc(F)cc1NC(=O)CCNC(=O)Cc1cncc(C)c1 c1(C(=O)NCCC(O)CNC(C2CC2CF)=O)ccc(OCC(F)(F)F)nc1 Cc1nc(C2CC2)sc1C(=O)NC(C)CCNC(C1(C)CC1C)=O c1(C(=O)NCC2(C(C)NC(=O)Cn3cnnn3)CC2)cc(O)nc2c1CCCC2 C1(C)(CNC(C(C)CN(C)C)=O)CCC(NC(=O)Cn2ccc(C3CC3)n2)CC1 CCC(CC)C(F)C(=O)NC1CN(C(=O)C(C2CCCCC2)OC)C1 c1(CCCN=C(NCC(C=C)C)NCC(C)C)ccc2c(c1)OCCO2 C1(CNC(C(CC)(F)F)=O)CN(C(=O)C(C)(C)N(C)C)CCC12CCC2 C(C(O)C(C)c1ccccc1)NC1CC(NC(C(C)OCCOCC)=O)C1 N1(C(C(C)O)=O)CC(C)N(C(C2CN(C3CCOCC3)C2)=O)CC1C c1(N2CCC(C)(NC(CC(CC)CN(C)C)=O)C2)nc2ccccc2o1 c1(C(=O)O)ccc(Cl)cc1O.C123CC1CN(C2)C(=O)c1ccc(o1)CNC3 C1(CC)(NC(c2cc(C(F)F)[nH]n2)=O)CCCN(C(c2cncc(OC)n2)=O)C1 c1(C(=O)NC2CN(C(CCc3ncc(C)[nH]3)=O)CC23CC3)c[nH]c2ccccc12 C(=O)(C1SCc2cccnc21)N1CC(C)C(n2cc(-c3cnsc3)nn2)C1 c1(C(=O)OCc2ccc(C(=O)OC)c(C)n2)noc2c1COCC2 c1(C(N(C(c2ccccc2)CNC(CNC(CCC)=O)=O)C)=O)cc(C#N)no1 C1(NC(C2CC(C3C(C)C3)C2)=O)CCCC(NCc2ccccc2N2CCCC2)C1 c1(CCOCC(=O)NC2CCN(C(=O)CCc3ncco3)C2)ccccc1 C#CCC(C)(CC)C(=O)N1CCN(C2CCN(C(=O)Cc3cccn3C)C2)CC1 N(C(=NCCCF)N1CCC(OC)C(C)(C)C1)CC1CCC(CC)O1 CCCC(CC)C(C(=O)NC1CC1)N1CCCC(Cn2ccnn2)C1 c1(C(N(C(C(C2CN(C(C(C)=CCC)=O)C2)O)=O)C)C)cnn(C)c1 c1(C(N2C(CCNC(C3CCC3)=O)CCCC2)=O)ccc2nc(O)[nH]c2n1 C1(NC(c2n(CC)nc(C3CC3)c2)=O)CN(C(=O)CSC(F)(F)F)CC1C1CC1 CCC(CC(=O)NC1CC(CF)C1)N(C)C(c1cn(C)nc1C)=O C(CCCC(C)C)N(C(C1N(C(C(COCC)C)=O)CSC1)=O)C c1(CNC(C(C(CNC(C2CN(C(C)=O)C2)=O)C)F)=O)nn(C)c(=O)n1C c1(C(=O)NC2C3(CC(NC(C)=O)C3)C2)ccc(C)nc1Cl N1(C(CCC(C)SC)=O)CCCC2C1CCN2C(=O)CN1CCC(N(C)C)CC1 N1(C(C(C)NC=O)=O)CC(C)(C)CC1CC(=O)NCCCc1ncn(C)n1 c1(CN2C(C(=O)Nc3ccc(F)nc3)C(O)CC2)ccc(F)c(C(=O)O)c1F C1(C(N2CCN(C(CC)=O)CC2)=O)CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCN1C c1(C(N2CC(CC(=O)NCc3cn[nH]c3)OCC2)=O)cc2n(n1)CCCC2 C(=O)(C(CCC1CCC1)NC(c1cn(C(C)C)nn1)=O)NCCC=CC=C N1(C(C(C)Cn2ccnc2)=O)CC2(CC(CC(=O)N(CCCF)C)C2)C1 c1(NC(C2OCCN(C(Cn3ccc(C)n3)=O)C2)=O)ccc2nnsc2c1 c1(C(=O)NCC2C(F)(F)CCN(C(C3(C#C)CC3)=O)C2)cc2cccc(F)c2s1 C1(NC(c2cnc(COC)s2)=O)CC(F)CN(C(=O)C=Cc2ccccc2)C1 CCC(CC)CCC(=O)N1CCCC1C1(C(=O)NCCc2cnc(C)[nH]2)CC1 CCCCCCC(C)C(=O)NC1CC2CN(C(=O)COC3CCCOC3)CC2C1 c1(C(N(CCCN(C)C)CCNC(C2(C)COC2)=O)=O)ccc(O)nc1 C(=O)(CCCC(=O)NC(c1ccc(F)cc1F)CNC(C1CC1(Cl)Cl)=O)OCC c1(SC(C)C(N2CCOC(CNC(C3CC3(C)C)=O)C2)=O)ccc(F)cc1 C12(NC(CC3C(C(C)C)CNCC3)=O)CCCN(CC1)C2 C(CCCCCNC(C1CC(C)(O)C1)=O)NC(c1n(C)cnc1)=O CCCCC(CC)CCC(Cn1c(N(C)C)nnc1-c1ccccc1CO)CC C(=O)(CCCC(F)(F)F)NC1C(NC(CCCC(=O)OCC)=O)COC1(C)C c1(C(N(C2(CC(=O)N(C(C)CS(C)=O)C)CC2)C)=O)ncccc1O C1(NC(c2cncc(C#C)c2)=O)CCN(C(C2COC3(CO)CC2C3)=O)CC1(C)C N1(C(c2cc(C)on2)=O)CC2(CCOCC2C(=O)NCc2cnccn2)C1 c1(C(=O)NCCCN(C(=O)C=Cc2ccc(Br)o2)C)cc(N)cc(O)c1 C1(NC(C2OCCN(CC)C2)=O)CN(C(=O)CS(=O)(=O)CC)C2(CCOCC2)C1 C1(C(=O)NCC2C(CNC(c3cccc(OC)n3)=O)C2)CC2(CCOCC2)CO1 N1(C(C(CC=CC)C)=O)CCCC2CN(C(c3cccc4c[nH]nc34)=O)CC12 C1(CCC(=O)Nc2ccccn2)CCCCN1C(=O)CNCCCCO c1(NC(C23C(CN(C(C=COCC)=O)C2)CC3)=O)c([N+](=O)[O-])ncn1C C1(O)(C(C)NC(c2nc(C)[nH]n2)=O)CCN(C(c2ccc(CO)cn2)=O)CC1 c1(NCC2(CNC(C3CCC(C)(CC)O3)=O)CC2)nnc(C)c(C)c1C#N c1(CN2C(CC(=O)Nc3cccc(F)c3)CCC2)ccc(CO)cc1 C(c1cccc(O)c1)=CC(N1C2C(CNC(C(N3CCOCC3)C)=O)C(C2)C1)=O N1(C(c2c(C#N)scc2)=O)CC2CC(C1)N(C(C1CC3(CSC3)C1)=O)C2 N1(C(Cc2c(C)ccs2)=O)CCOCC(CNC(=O)CCCC2CCCC2)C1 CC1(C)CCC(NC(C2C3CCC(C3)N2C(c2cccc(C3CC3)c2)=O)=O)CC1 N1(C(CSc2n(C(C)C)cnn2)=O)CC2CC2(CNC(=O)COC(F)(F)F)C1 C#CC(CC(C)(C)C)NC(C1CN(C(C2(C)CNC(=O)C2)=O)CC1(C)C)=O c1(CN(C(C2CC(CC)C2)=O)C)ccccc1CNC(c1nnc(C)s1)=O CC1CN(C(c2cnc(C3CC3)o2)=O)CC1CCNC(C1CS(=O)C1)=O C1(NC(c2cc(CC)on2)=O)CN(C(c2cccc(OCCO)c2)=O)CC1F C(=O)(CCC(=O)N1CCOC(CN(C)C(c2cnn(C)c2)=O)C1)c1ccc(C)s1 O=C(N=c1c(Br)c[nH]cc1I)C1CC(NC(=O)CCc2ncc[nH]2)C1 c1(C(N2CC(N(C(=O)C#CC3CC3)C)C3(C2)CC3)=O)cccc(Cl)c1[N+](=O)[O-] C1(NC(CC2(NC(C=CCOC)=O)CC2)=O)CCCC1CSC1CCC1 N1(C(c2c(NC)snc2C)=O)CCC2(CCC2)C(NC(=O)CC2CC2(Cl)Cl)C1 c1(C(=O)NCC2C(c3n(C)ncc3)C2)c(Cl)ccnc1Br c1(CC)c(C(=O)N(C)CCOCCC(=O)NCCCCCOC)cnn1C C1(NC(C(=O)NC(CC)COC(F)(F)F)=O)CSCCC1(OC)OC CC(C)CC(O)CNC(c1ncco1)Cc1ccccc1 Cc1nc(CNC(c2nccnc2N)=O)oc1C(=O)NCC1CNC(=O)O1 C1(CCC)CCN(C(C2(CNC(C3CCCN3)=O)CCCC2)=O)CC1 Cn1nccc1CNC(C1CCCC1NC(=O)CC1COCC1O)=O c1(C(N2CC3C(N(C(=O)Cc4ccc(F)cn4)C)C3C2)=O)cc(F)cc(Cl)c1N CC1(C)CCC2(CC1)CC2C(=O)NCC1CCN(C(c2cc(Cl)ncc2O)=O)C1 c1(CNC(C2CC2NCc2cc3cc[nH]c3cn2)=O)ccc(OC)c([N+](=O)[O-])c1 C1(CNC(c2cnn[nH]2)=O)CCCN1C(=O)C(F)OC(F)(F)F c1(CC(=O)NCC(CC)NC(c2cc3n(c2)CCC3)=O)ccc(OC)cc1Cl c1(OCCNC(c2n(CCSC)nnn2)c2ncco2)ccc2ccccc2c1 N1(C(C=CC2N(C(CCC(N)=O)=O)CCC2)=O)CCCC(F)(F)C1 c1(C(=O)OCC)ccc(S(=O)(=O)NC(COC)C2CCC2)o1 C(C)(CNC(=O)CCc1ccc(C)o1)(CNC(c1cscn1)=O)OC N1(C(Cc2ccc(C)cc2)=O)CCCC(NC(c2c(C)ncnc2O)=O)CCC1 CCCCC(C)(F)C(=O)NCC1CN(C(=O)C(C)(C)C(C)(F)F)CC1(C)C c1(NC(=O)NC2(CN3CCCCC3)CCOC2)cc(-c2ccncc2)ccc1F N1(C(C2(CC)CCNC2=O)=O)CC(NC(=O)NC)CC2(CCC2)C1 CCC(CC(C)C)C(=O)N1CCC(OCC(=O)NC(C)(C)C(C)(C)C)C1 c1(CC(=O)NC2CCC(NC(C(C)(C)c3cccnc3)=O)C2)cc(O)nc(O)n1 N1(C(C2(N)CCS(=O)(=O)C2)=O)CCc2c(F)cc(C(=O)O)cc2C1 C1(C(N2CCC(C(C)NC(CCCOC)=O)C2)=O)CC(=O)N(C2CCCC2)C1 CN1CCC(=O)Nc2cc(C(N3CCN(C(=O)C(F)F)CC(C)(F)C3)=O)ccc21 N1(C(CN2C(=O)CNCC2)=O)CCC(C(C)C)C1.C(=O)(C(C)(C)C)OC C(=O)(CC(C)CCC(=O)N1CCN(CCN(C(=O)CCF)C)CC1)OC c1(OCC)cccc2c1OCC(NC(=O)C(=O)NNC(=O)C1CCS(=O)(=O)C1)C2 c1(C(N2C3(C(N4CC(CC)SCC4)=O)CC(C)(C2)C3)=O)cccn2ccnc12 C1(NC(CSC)=O)CCC2(CC1)CN(C(=O)CNC(N1CCCC1)=O)CCO2 Cc1nncn1CCNC(=O)C(Cc1cc[nH]n1)NC(c1csnc1Cl)=O N1(C(CCCOCC=C)=O)CCC2C(C1)CN2C(=O)C(F)C1CC1 Cc1ccc(NC(=O)Cc2c[nH]c(=NCc3csc(Br)c3)s2)cc1O N1(C(Cc2scc(CC)n2)=O)CCC(C)(NC(c2cc(Cl)cn2C)=O)CC1 c1(CNC(C2C(CCC)C2)=O)ccccc1CNC(=O)Cc1c[nH]nc1O C12(C(=O)NCC(C(=O)NCC(=O)OC)N(C)C)CC(C#N)(C1)C2 c1(C(=O)NCC(CC(=O)NCC(CCC)(C)O)C2CCC2)ccc(C)c(C)n1 C1(CNC(C2CCC(C)CC2)=O)C2CCCC1N(C(C1CCS(=O)CC1)=O)C2 Cc1nc(O)nc(O)c1CCC(=O)NC12CC(NC(C3CC(O)C3)=O)(C1)C2 Cc1cc(C)c(C(=O)NCC(CO)NC(C2CCC(C)(C)CC2)=O)cc1Br c1(OC)cc(C)cc(C(N2CC3(CC3)CC2CNC(=O)CCCC(C)C)=O)c1C c1(C(=O)NC(C)CCCCNC(=O)CCC2OCCO2)cnc2[nH]ccc2n1 N1(C(C2(CC)CCNC2=O)=O)CC=C(CCNC(=O)CC2CCSCC2)CC1 c1(N2CCN(C)C(=O)C2)nc(NCC2C(=O)NCCC2C)c2ncsc2n1 c1(C(=O)NCC#CCNC(C=CC(CC)C)=O)cnnc2ccccc12 Cc1ccc(F)c(C(=O)N(C(C)C(=O)NCCc2cn(C)cn2)C2CC2)n1 c1(C(N(CC(CNC(C(Cn2ccc(C)n2)C)=O)(C)C)C)=O)cc(F)cnc1O N(C(=NCCSC)NCC(c1ccc(C)o1)O)Cc1ccc(OC)nc1 C12(CNC(C=CCN(C)CC)=O)CC(CC)(CN1C(c1sccc1OC)=O)C2 CC(C(=O)NCc1ccoc1C(=O)NCCc1ccccc1F)C(C)S(C)(=O)=O Cc1ccc(C(N2CCN(C(C3CC(O)CN3C(N)=O)=O)CC2)=O)cc1O c1(SC)cc(=NC(=O)CC2CCN(C(C3CCCCN3C)=O)C2)[nH]n1C C1(C(N2CC(c3cn(-c4ccccc4)nn3)C2)=O)C2Cc3ccccc3C12 N1(C(=O)COC2CC=CC2)CC2(C1)CN(C(c1ccc(Cl)nc1Cl)=O)C2 C(c1ccccn1)=CC(N1CCC(CNC(C2(CCOC)CCC2)=O)C1)=O N1(C(c2c(C)nsc2)=O)CCN(C(c2cc(C(C)C)cc(F)c2)=O)C(C)CC1C c1(CC(=O)NCC2CN(C(=O)CCF)C2)cn(C(F)F)cn1 N1(C(CN(C(=O)NC)C)=O)CCOC(CNC(c2cc(C(=O)OC)on2)=O)C1 N1(C(c2c(CCC)nns2)=O)CCN(C(c2ncnn2CC)=O)CC(O)C1 N1(C(Cc2ccc(C)cc2)=O)CCc2nc(C(=O)NC(C)(C)C)cn2CC1 C1(CNC(CCCC2(NC(c3cn(CC)nc3)=O)CCC2)=O)CCC(C)(C)CO1 c1(OC)coc(C(=O)NCC(C)(O)CNC(C2CC(CC(C)(C)C)C2)=O)cc1=O Cc1cc(C(=O)NC2(CF)CCN(C(c3cc(C#N)ccn3)=O)C2)cc(C)n1 C(=O)(CC(C)C(=O)OC)NC(CSCC)C(N1CCOCC(CC)C1)=O C(CCCCCNC(C1(CC)CC1(F)F)=O)N(C(C=CC=CC)=O)C O(NC(=O)C(CC(C)C)ONC(=O)CC#N)C(C)C C1(CC(=O)NC2C3CC(CNC(CCCCC)=O)(C3)OC2)CCN(OC)CC1 C1(C2CC2)(COC)CN(C(=O)C=CC2CCCN2C(=O)C(C)OC)C1 C1(C(N2C3C(CNC(CCCOC)=O)CC(CC3)C2)=O)CC(C)(C)OC(C)(C)C1 Cc1ccc(NCCC(=O)NCCC2(O)CCCNC2)c(Cl)c1 N1(C(CN(CCC#C)C)=O)CC2CCN(C(c3nc4ccccc4[nH]3)=O)CC2C1 C(=O)(CCC(=O)NCCCC(C)NC(=O)C(c1ccc(C(F)F)cc1)C)OCC Cc1cccc(C(=O)NCC(C)(C)NC(C2CCC(O)C2)=O)c1 c1(C(=O)NC2CN(C(CCOCC#C)=O)CC2C)ccc(F)c(COC(C)C)c1 Cc1ncnc(C)c1CC(=O)NC1CC(C)CN(C(C2(C)CC(F)(F)C2)=O)C1 c12nnn(c1C(F)(F)F)C1CCN(CC1)CC(=O)OC2=O.N1(CC)CC(C)CC1 C(=O)(C(C(C)C)Nc1ccc(Cl)cn1)N(CC(=O)NCC(C)C)CC c1(C(N(C)Cc2ccncn2)=O)cncc(CNC(C2C=CCC2)=O)c1 Cc1nc(C(=O)NCC2(NC(=O)Cn3nnnc3C(C)C)CC2)ccc1C#N C(CCC(O)CO)N(C(=O)CC(O)CNC(=O)CNC1CC1C)CC C1(CNC(COC)=O)CCC12CCN(C(=O)C=Cc1ccc(O)c(O)c1)CC2 c1(NC2CC(C(=O)Nc3c(C(=O)OC)scc3)C2)ncnc2c1ncn2C C(C)(C)(C(C)CC(=O)NCc1cnc(COC)[nH]1)NC(c1n(CC)ccn1)=O c1(C(N2CC(NCc3ccc(C)nc3Br)C(F)CC2)=O)ccc(O)c([N+](=O)[O-])c1 CC1CCC=C1C(=O)N1CCC(CC(N2CCCC2c2ccon2)=O)CC1 c1(NC(c2ccc(CNC(Cc3c(C)ncs3)=O)s2)=O)cnc(N(C)C)nc1 N1(C(c2c(C)nc(CC)o2)=O)CCC(C2CC2NC(=O)C(C)C2(O)CCC2)CC1 c1(C(=O)NCC(C(C)C)NC(C2CCCN2N=O)=O)cccc(CCCCO)c1 C1(NC(c2c(-c3c(C)nn(CC)c3C)nccc2)=O)CS(=O)(=O)C12CCOCC2 n1(CC(=O)N(CCNC(=O)CC2C=CCCC2)C2CC2)ccc([N+](=O)[O-])n1 C1(CNC(C2(CNC(c3c(C)ccs3)=O)CCC2)=O)CC2CCC1CC2 N(C(=NCC1COCCOC1)N1CCC2OCCC2C1)C(C=C)C N1(C(C(n2cc(C)nc2)(C)C)=O)CCC(NC(=O)C=CC2CC2)C(O)C1 CCCN=C(NCC(CO)C(C)(C)C)NCC1CC1COC c1(OC)cc(OC)ccc1C(=O)NC1CN(C(=O)CCC(C)OC)CC1C(F)F [N-]=[N+]=NC1(C(=O)NCc2[nH]ccc(=O)c2O)CCN(C(=O)CC23CCCC2C3)C1 c1(OC)cccc(C(C)CC(=O)NCC(C)NC(=O)C(C)(C)OC(C)=O)c1 c1(C(N(CCNC(C(C)=C2CC2)=O)CC2CC2)=O)ccc(-c2ccncc2)nc1 c1(OC)sccc1C(N1C(C(=O)NC2CC(C)(C)C2)CC1C)=O c1(OC)cccc(OC(F)(F)F)c1C(=O)NC(C)(C)CC1CCCCC1 C12(NC(CCCOCC)=O)CCCC1N(C(C1CC1c1ccccc1Cl)=O)CC2 c1(C(N2CC(NC(Cc3c(C)cccc3)=O)C(F)CC2)=O)cc(C#N)ccc1Br C1(NC(CN2CCC(C)C2)=O)CC(F)CN(C(c2cc(CO)ccn2)=O)C1 c1(C(C)NC(=O)CC(C)(C)CNC(c2cn(C)nn2)=O)coc2ccccc12 c1(C(N2CC(CN(C(c3cc(C)nc(Cl)c3)=O)C)C2)=O)nccc2ccsc12 c1(C2C(C(=O)NC3(N4CCCC4)CC3)CC2)nc(S)n[nH]1 c1(C(=O)NC2CC(CNC(CC(C)(C)C)=O)C2)cc([N+](=O)[O-])ccc1Br c1(COC)nc(C)ncc1C(N1CC2(NC(C3CCOC3)=O)CCC1C2)=O C(=O)(C1=CCCN(C(c2cnn(C3CC3)c2)C(=O)NCCC#N)C1)OCC C12(C(=O)NCCc3ccc(OC)c(Cl)c3)CCC(C(F)(F)F)(CC1)CC2 N1(C(=O)Nc2cccc(Br)c2)CCCCNCC(F)(F)C1 C(=O)(C(F)C(C)C)N(CC(C)NC(Cc1nc(C(=O)OC(C)(C)C)sc1)=O)CC C1(C2(C(=O)OC)CCC2)CCCN1C(c1ccnn1C1CCCCO1)=O CN(CCOc1ccc(Cl)cc1Cl)N1CCn2c(-c3cccnc3)nnc2C1 N1(C(c2c(C)nccc2)=O)CCC(F)(F)C(NC(c2cc(F)c(F)cc2F)=O)C1 C(=O)(C(CC1CC1)CC1CC1)N(CC(CC)NC(=O)C(C)(C)c1ccnn1C)C N1(C(C(C)NC(COC)=O)=O)CCCC(NC(=O)C=CC=C(Cl)Cl)C1C C1(NC(c2cc(C)nc(O)n2)=O)CCC2CN(C(=O)C(C)S(N)(=O)=O)CC2C1 N1(CC)C(=O)CCC1CC(=O)NC1CC(CNC(=O)CSc2ccncc2)C1 c1(C(=O)NCC2(F)CCN(C(C3(SC)CCC3)=O)CC2)ccc2c(c1)nnn2C c1(C(=O)NCC2(C)N(C(CNC(CC)=O)=O)CC(F)(F)C2)cc(S(C)(=O)=O)oc1C CN1CCC(CC(=O)NCC2CC(NC(C3COCC3(C)C)=O)C2)CC1 c1(C(=O)NC)ccc(C(=O)N(C2CN(C(=O)CSC3CC3)CC2(C)C)C)cc1F CN1CCN(C(=O)C(C2(CC3CC3)CCC2)NC(C2CC=CCC2)=O)CC(O)C1 n1(CC(N2CCN(C(CCC)=O)C(CO)C2)=O)ccc2ccccc12 N1(C(C)CCC2CNc3ccccc3C(=O)O2)CCC2C(C1)NC(=O)CCN2C N(C(=NCC(C)C1CCCCC1)NCC(c1cccnc1)O)C(C=C)C C(=O)(N=c1nc[nH]n1C)C1N(Cc2c(OC)cc(Br)cn2)C2C(C1)C2 C1(C(=O)NCCC=CCCC)CC(NC(c2cc3n(n2)CCC3)=O)C12CCC2 Cc1ccc2cccc(C(=O)NCCC3CCCCN3C(=O)C=CS(C)=O)c2n1 CC1CN(C(=O)COc2ccc(O)cc2)C(C)CN1C(=O)CCC(F)F c1(C(=O)OC)cc2c(Br)cccc2c(N2CCOC(C3CC3)C2)n1 C1(COC)(CNC(c2nnn(C)c2C)=O)CCN(C(C2CC(C3CC3)C2)=O)C1 c1(C(C)(C)C)conc1C(=O)NC1CCC1NC(c1cncn1C1CC1)=O C12(CNC(c3n[nH]cc3C3CCC3)=O)CCC(CC1)N2C(=O)C(F)F S(=O)(=O)(c1cccnc1)NCCC(=O)NC1(C)CCCC1.C1(C(=O)N)COC(=O)O1 C1(NC(C(CCC)OCC)=O)CCCN(C(=O)C(C)=CC(C)(C)C)C1C N1(c2nnn(C)n2)CCC(C2CCCN(C(C3CCC4CC4CC3)=O)C2)CC1 Cc1cc(C)c(NC(=O)C(N2CCC(N(C)CCO)CC2)=O)c(C)c1 C#CC1CN(C(C2C(CC)CCN2C(=O)Cc2cnsc2)=O)CCO1 N1(C(c2cncc(SCC)n2)=O)CCN(C(=O)Cn2cccnc2=O)C(CO)C1 C1(NC(CCCNC(=O)OCC)=O)CC2(C1)CC(NC(=O)Cc1cnoc1)C2 C1(COC)(CNC(C2C(C(=O)OC)C2)=O)CCN(C(C2(S(C)(=O)=O)CC2)=O)CC1 C1(CC(=O)NCC(Cn2cc(C(N(C(C)=O)C)C3CC3)nn2)C)COCC(C)(C)O1 C1(C)(OCC(N2CC(CNC(c3ccc(CC)s3)=O)C2)=O)CCOCC1 N1(C(C2(N3CCN(C(C)=O)CC3)CC2)=O)CC(=O)NC(c2cn[nH]c2)C1 N1(C(=O)NC(C2COC3(CCCOC3)C2)C)C2CCC1CC(c1ccnn1C)C2 N1(C(C(CCC)OCC)=O)CCC(F)(C(=O)NCCN2CCC(OC)C2)CC1 c1(CN(C(=O)NCC(Cc2ccccc2Cl)C(N)=O)CC)cc(C)ccc1C C(=O)(CN=c1ccc(C#N)c[nH]1)NCC1(NC(CC(C)N(C)C)=O)CC1 c1(C(CC(N2CC3(C2)NC(=O)N3)=O)C)ccc(C(N)=O)cc1.C(C)(SC)SC C1(CNC(C2(C)C=CCC2)=O)CCCCN1C(c1sccc1SC(F)F)=O Cc1c(C)c(CC(N2CCC3C2CCCN3C)=O)c(C)c(C)c1Br N1(C(Cc2cnn(C)n2)=O)CCCC(CO)(NC(=O)COC2(C)CCCC2)C1 C12(C(N3CC(CCC)C(CO)C3)=O)CC(C)(CN1C(c1ccoc1Cl)=O)C2 C(=O)(CCC(C)c1ccccc1)N1CC(CC(C)NC(CC2CCC(C)C2)=O)C1 N1(C(C(C)NC(c2ccoc2)=O)=O)CC2CC(NC(c3ccn(C)c3)=O)C1C2 c1(C(N(C2CCCN(CC3(C#N)CCNC3)C2)CC)=O)ccc(Cl)cc1OC C1(CC(=O)N(CC(=O)OCC)CC2CC2)OCCO1 CC(CCO)CN=c1nc(N2CCCC3(CCCC3)C2)c2sccc2[nH]1 C(CC(C)N=c1nc(C#N)[nH]cc1C)NC(C1CCCN(CC)C1)=O c1(-n2cc(CN(C)C(c3cccs3)=O)nn2)cc(F)ccc1Cl C1(NC(c2cncc(OC)c2C)=O)CN(C(=O)CC(F)F)CC(C)(C)C1 C=CCCCCCCC(=O)NC1CCC2CC1CN2C(=O)CSC(C)(C)C CCCC(CC(=O)NCC1CCC(O)CC1)NC(=O)C(O)C(C)C N1(C(C2C(C)N(C)CC2)=O)CCCCC(CN=[N+]=[N-])C1 c1(OC)cnc[nH]c1=NCCc1cc(C(C)(C)C)no1 Cc1cc(F)cc(NC(C2CCC(CNCc3c(O)cccc3F)CC2)=O)c1O c12nc(ncc1Br)N2.N1(C(CN(CCOC)C)=O)CC2C(C(=O)O)C2C1 n1(CCC)ncc(CNC(=O)CSC2CCCOC2)c1C.N12CCCCC1C2.C C1(NC(CC(C)(C)OC)=O)CN(C(C2(O)CN(c3ccccc3)C2)=O)CC12CC2 N1(C(c2cc(CCC)ncc2)=O)CC2=C(C1)CN(C(=O)COC1CCC1)C2 Cc1cc(C(=O)NCC2(CNC(c3cncn(C)c3=O)=O)CCC2)ncc1Cl C1(COC)CC(CNC(=O)C(C)Cc2cccc(Cl)c2)N(C(=O)CCF)C1 C1(C2CC2)(NC(C2C(OC)C2)=O)CCN(C(c2cnc3n2CCS3)=O)C1 c1(C(C(=O)NCCC#N)N(C)CC2CCCS2)cc(Br)ccc1Cl c1(C(N(C(C)CNC(C2COC(=O)N2C)=O)C)=O)oc2ccccc2c1CO C1(C(=O)NC2C(NC(c3nc(COC)sc3)=O)CCC2)CCCN(CC(C)C)C1 C1(NC(CC(C)c2ccco2)=O)(CNC(=O)C(O)Cn2cncn2)CCOCC1 c1(C(=O)NC2CN(C(C=C(CC)C)=O)CC2C)cnc(OC)c(C(F)(F)F)c1 c1(C(N(CC(C)NC(C2(F)CC=CCC2)=O)CC)=O)coc2c(F)cccc12 C(CC(C)CC)(C(=O)NOCc1ccccc1)NC(c1cc(CC)on1)=O C1(C(=O)NC2CCCC(c3ccc(Cl)cc3)C2)CCCC1C1CC1 N12C3CCC1(CC3)C2.O=C1CCCC(CNn2cc(C3(O)CCCCC3)nn2)O1 C(CCc1ccccc1)(C(C)NC(=O)C=CC1CC1)NC(C=C1CCC(C)C1)=O N1(C(c2c(COC)cco2)=O)CCOC(C(=O)NC2CCCC2OC)C1 Cc1cc(=NCC(=O)NC(CCc2ccccc2)CC(F)(F)F)[nH]c(CO)n1 CCS(=O)CC(=O)NC(CCF)C(=O)NCCc1ccncc1 c1(N(C(=O)C(C)Cc2ccco2)CCN)ncnc2n[nH]c(C)c12.CO N1(C(=O)Cc2ccnc(Br)c2)CC2(CCCCN(C(C3COCCO3)=O)C2)C1 Cc1cc(C=CC(=O)NCC2CC(F)(F)CN2C2CC2)ccc1C(F)(F)F c1(C(=O)NC(CN(C(C(=O)NCC)=O)C)(C)C)cc(C)cc2ccncc12 C#CCCCC(C)C(=O)N1CCC(CCCNC(c2c(C)cccc2Cl)=O)CC1 c1(CC)ccc(NC(=O)NCC2CCN(C(=O)C(N3CCCCC3)=O)C2)cc1 Cc1nc(O)[nH]c1C(=O)NC(C1CCCCN1C(C1CCCCC1)=O)C C(=O)(CS(=O)(=O)C(C)C)N1CC(n2cc(CNC(C3CC(=C)C3)=O)nn2)C1 C=CCC(CNC(c1cc(C)cc(C)n1)=O)C(=O)NCC(Cl)C(C)(F)F c1(C(=O)NC2CCN(C(=O)C=CC3CC3)CC2)cncc(Br)c1Cl c1(C(N2CCC(NC(CCC(=O)NCC#C)=O)CC2)=O)cc(F)ccc1C(C)=O N1(C(C(C)c2cncs2)=O)CCCC2(CCCN2C(=O)CCCF)C1 C(C(C)CC(=O)NC(Cn1cncn1)C(N1CCCOCC1)=O)OC C1(C(N2CC(c3cn(CC(C)C)nn3)N(C)CC2)=O)CCc2nccn2C1 c1(CC(N2CCC(NC(=O)CC3CC3C3CC3)C2)=O)cccc(Cl)c1 CCCCC(F)C(=O)N1CC(CNC(C2(C(F)F)CCCO2)=O)C2(CC2)C1 c1(C(N2C(CN(C(C3OCCN(CC)C3)=O)C)CCC2)=O)cnc2scc(C)n12 CC(C)(C)CCCCC(=O)N1C2CCC1CC(O)(CNC(c1cc(F)n[nH]1)=O)C2 O=C(N=c1ncnc2[nH][nH]cc1-2)C1CC2(C1)CN(Cc1cc(F)c(F)c(F)c1)C2 CN=c1cc(C(=O)NC23CCN(C(c4oc(SC)cc4C)=O)CC2C3)cc[nH]1 c1(C(N2CCN(C(CCCC=C)=O)C(C(F)F)C2)=O)nc2ccccc2o1 c1(N2CCN(C(C)C(N)=O)CC2)ncnc2c1ncn2CC(O)CO C(=O)(C(C(C)C)NC(C1CC12CC2)=O)N(C(c1ccccn1)C)CC c1(C(=O)NCC(=O)OCCCC)ccc(CNC(=O)C(C)n2cnnn2)cn1 N1(C(c2c(C)cc(Cl)cc2)=O)CC(N=c2[nH]c3cccc(C)c3o2)C1 C1(CCO)(NC(C2CC2C)=O)CC2CCC(C1)N2c1nnc(C(F)F)s1 CCCC(CNC(=O)CSc1ccccc1Cl)CCC c1(C(=O)Nc2ccc(NC(C3CC=CCC3)=O)nc2)cc(Cl)ccc1Cl c1(CNC(N)=O)ccc(C(N2CC(NC(C3CCCCC3)=O)C3CC23)=O)cc1 C(C(C)C)(C(O)C(=O)N1CCOCC(NC(C2CCC(O)CN2C)=O)C1)OC C1(CNC(=O)NC(c2cnc(N3CCOCC3)s2)C)CC(C)OC1C Cc1noc(CCCC(=O)NCC2CCCC2NC(=O)C=Cc2cc[nH]c2)n1 c1(CC)c(C(=O)NCCCN(C(=O)Cc2cccc(C)c2)C)cnn1C(C)(C)C Cc1ccc(C#N)cc1C(=O)NC1CC2CC1CC2C(=O)N(C)Cc1ccns1 CC1=C(C(=O)N2CC(NC(c3ccc(C4CCC4)nc3)=O)CC2C)CCO1 C1(C(=O)OC)C=CC(C(=O)NC2CC(N(C(=O)C=CC3CCCC3)C)C2)C1 N1(c2c(C(N3CCC(n4c(=N)nc(C)[nH]4)CC3)=O)cccc2)CCOCC1(C)C C(CC(C(C)(C)C)NC(C1(C)CCOCC1)=O)N(C)C(c1cc(=O)cc[nH]1)=O C(CC(C)C(=O)N(C)CC1CN(C(c2cc(Br)cn2C)=O)CCO1)=CC c1(N(C)C)ccc(C(=O)NCCN(C(=O)CCn2ccnc2)CC2CC2)cc1F C1(NC(c2ccc(F)o2)=O)CC2CC1CN2C(=O)CCc1ccccc1Cl C(C(=O)N1OC2CCC1C2)C1C(NC(CSC(C)C)=O)CC1O N1(C(c2cc(CC)[nH]n2)=O)CCC2(CCC(NC(=O)CSS(C)(=O)=O)CC2)CC1 Cc1cc(C(=O)NCC(CC2CC2)C(=O)NCc2ncc[nH]2)nc(O)n1 CCCC(CCCNC(=O)CCc1ncc[nH]1)NC(C1(CN(C)C)CC1)=O N1(C(CCOCC)=O)CCN(C(C2CC(F)(COC)C2)=O)C(C)C1.C(=O)OC Cc1cc(NC(C2CCCCC2NC(=O)Cc2nc(Cl)cs2)=O)cc(O)c1 C1(C(N2CC3CC(NC(CC(C(C)C)C)=O)C3C2)=O)CC2(C1)CC(F)(F)C2 c1(CC(=O)NC(CNC(C2CCCO2)=O)CO)csc2cc(Cl)ccc12 C12(C(=O)NC(c3noc(C)n3)CC)CC1CN(C(c1cc(Cl)c[nH]1)=O)C2 C1(C(N(CCNC(C2CCC(=O)C2)=O)C2CC2)=O)CCc2ncc(Br)n2C1 c1(OC)noc(C)c1C(N1CCCC(CNC(=O)CC2CCCN2C)C1)=O c1(C(N)=O)csc(C(N2CC(NC(C3COC(=O)C3)=O)C2)=O)c1 CCCC(C(=O)NCc1ccc(CN(C(=O)CC2C=CCC2)C)cc1)NC(N)=O N1(C(C2CN(C(C)=O)C2)=O)CC2CCN(C(C3CC(C#N)C3)=O)C2C1 c1(C(N2CCC(C(C)NC(CC(CCC)C)=O)C2)=O)ccc2nc(C)cn2c1 C1(C(=O)NC2CCN(CCC)C2)CC2CN(C(C3CCCC(OC)C3)=O)CC2C1 c1(C(N2CCC(N(C(C3C(F)(C(=O)OCC)C3)=O)CC)C2)=O)cc(SC)oc1C C1(NC(C(C(C)(C)C)NC(C2N(CC)CCOC2)=O)=O)CN2CCC1(C)CC2 N1(C(c2cc(C(=O)OC)on2)=O)CC2CC(NC(=O)C3=NOCC3)C2C1 N1(Cc2nc(C(=O)OC)c(Br)s2)CC2(C(=O)OCO)CC1(CO)C2.C(C)(C)C N1(C(CCn2c(C)ccc2C)=O)CCC(CNC(=O)CC(C)C2CC2)CC1C C1(F)(C(N(C)CC2OCCN(C(C3CC(SC)C3)=O)C2)=O)CCS(=O)(=O)C1 C1(CNC(C(N2CCC(C)C2)=O)=O)C2CC1N(C(=O)Cc1ccccc1Br)C2 N1(C(CCN(CCCCOC)C)=O)CCCC(C(N2CCC(O)C2C)=O)C1 c1(OC)cc(N)ccc1C(=O)NCC1CCCC1NC(=O)CC(C)C1CC1 N1(C(C(C)Oc2ccc(OC)cc2)=O)CCN2CCN(C(=O)CC3CC3)CC2C1 N(C(=NCC1CCC1)NC1CCOc2ccc(F)cc21)CC1(SC)CCOCC1 c1(NC(C(C)Cc2ccncc2)=O)ccc2nnc(C(F)F)n2c1 N1(C(C2(CC)CC(C)(C)C2)=O)CCCC(CCNC(c2nnc(S)n2C)=O)CC1 C1(NC(c2nc(COC)oc2)=O)CC2CC(NC(=O)CC(C)SC)CC2C1 N1(C(Cn2cnc(C(N)=O)n2)=O)CC(C2CN(C(c3cscc3F)=O)C2)C1 Cc1cnc(C(=O)NC(C2CCCCC2)C(=O)NCCn2ccnc2C)c(F)c1 n1(CC(=O)NCC2C(C(=O)NC3CC(C(C)(C)C)C3)CCO2)cccnc1=O C1(CCOC)(NC(C2OCCN(C)C2=O)=O)CCN(C(C2CCCO2)=O)CC1 N1(C(COCCOC)=O)C2CCC1C(NC(=O)CCc1ncccc1C)C2 N1(C(c2cc(C)n(C(F)F)n2)=O)CC2CN(C(C3CC3(F)F)=O)CC2(C)C1 c1(NCCN(CCCNC(c2coc(O)n2)=O)CC)ccccc1NS(C)(=O)=O c1(-c2ccc(OC)cc2)cc(CN2CC=CCO2)cc(F)c1F C1(C2CC2)(NC(CC(=C)C)=O)CCN(C(c2cnc(C)nc2CC)=O)C1 n1(-c2ccc(SC)cc2)nc(C2CSC2)nc1C1COc2ccccc21 C(=O)(C1CC(=O)Nc2ccc(Br)cc21)NC1C(NC(CCC)=O)CCC1 N1(Cc2ccc(C(=O)OCCC3CC3(Br)Br)cn2)C(=O)c2ccccc2C1=O c1(C(N(C(C)CNC(c2cnc(OC)s2)=O)CC)=O)cn2cc(Cl)cc(Cl)c2n1 C1(CNC(c2nc(C(C)OC)oc2)=O)CCCCCN1C(c1ccnc(O)c1)=O C1(C(=O)NC(C(CC)C)CO)C2CC(O)C(C2)N1C(c1ccsc1C#N)=O CC1CN(C(C2CC3(C2)CC(C)(C)C3)=O)CC(C)C1NC(=O)C1=COCCC1 C(=O)(C(C)(C)CNC(C1(C#N)CC(C)C1)=O)N1CCC(OCC#C)C1 c1(C(=O)NC(CNC(CCCC=C)=O)(C)C(C)C)ccc(C2CC2)nc1O CC1=C(C(=O)Oc2ccc(Br)cc2)C(c2ccnn2C)NC(=S)N1CC1CC1 c1(C(=O)NC2CCC(NC(c3c(C)nn(C)c3)=O)C2)c[nH]cc(F)c1=O C(C1c2ccccc2CCN1C(C1CC1F)=O)NC(c1c(C(N)=O)nccn1)=O CN1CCC(NC(=O)CCC2CCCCN2C(c2ccccc2C#N)=O)CC1=O N1(C(C2(C)N(C(c3n(CCC)ncc3)=O)CC=C2)=O)CCC(C)OC(C)C1 N1(C(C(CC)(CC)c2ccc(Cl)cc2)=O)CCCC12CCOC2=O CON(CCO)C(=O)C1CC=CC(NC(=O)Cc2ccnc(O)c2)C1 C(C(C)(C)CCNC(C1CCOC1C(F)(F)F)=O)NC(CCNC(C)=O)=O N1(C(C(CC)CCc2ccccc2)=O)CCc2nncn2CC1.c12cn(nn1)C2 c1(CCCC)ccc(C(=O)OCC2(F)CC(OCOC(C3(F)CC3C)=O)C2)cc1 N1(C(C2OCCN(CC)C2)=O)CCCOC(CCNC(C2CCCC2)=O)C1 CCC(C)(CC)CN=c1nc2scnc2c(NCC2(C)CCCCO2)[nH]1 N1(C(C(CC)F)=O)CCC(C(C)(C)CNC(C2CCCN2N=O)=O)CC1 C1(C(N(CCNC(C2C=CCCC2)=O)CC)=O)CC2CCC(C1)O2 C(=O)(C1=CC2(CCOC2)C1)NCC(CC)(CC)C(=O)NC1CN(C)CCC1O N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)CC(C)C2CCCCC2)CC(CO)C1 C1(NC(c2c(CC)c[nH]c2)=O)CCCC2CN(C(c3cncc(NC)c3)=O)CC12 c1(NC(N)=O)cc(COCC2CC(OC(C3OC4CCC3C4)C)C2)ccc1[N+](=O)[O-] C1(NC(C2N(C(C)=O)CCCC2)=O)CN(C(=O)Cc2ccns2)CC(C)(C)C1 c1(C(=O)NCC(CN(C)C(C2COCCOC2)=O)O)cn2c(n1)CCC2 CCCCC(C)(F)C(=O)N1CCCC(CN(C)C(c2cc(C)nc(O)c2)=O)C1 Cc1cc(C(N2CCCC2c2cn(C3(C(N)=O)CC3)nn2)=O)cc(C)c1C O=C(NNc1ncc(I)cn1)C1CCCN(CC2CCCO2)C1 c1(N(C)CC2CCN(C(Cc3c(C)ccc(Br)c3)=O)C2)cc2nncn2c(C)n1 c1(OC)ccccc1C1CNCCN1C(N1CCC(C(C)(C)O)C1)=O C1(NC(c2ccnc(C)n2)=O)CCC2(C1)CN(C(=O)CCC(F)(F)F)C2 N1(C(c2c(C)n(C3CC3)nc2)=O)CCC(CNC(=O)C(F)CC2CC2)C(F)(F)C1 c1(C(C(=O)NCC)N(C(C)C(=O)N(C)C)C)nncn1C CC1CCCC(C)N1C(=O)C(=O)NCCC1CN(C(=O)CCc2cccnc2)C1 C1(C(=O)NC(C2CCC2)C)(NC(Cc2c(C)occ2)=O)CCN(C)C1 Cc1ncc(C(=O)NCC2(C(C)(C)O)CN(C(C3(C)CC3(F)F)=O)C2)s1 c1(C(N2C(C)CN(C(C3C4CN(C)CC34)=O)C(C)C2)=O)cccc2nc(O)oc12 N1(C(c2c(N)ccc(C)c2)=O)C(C)CC2CN(C(C3(C)CC3(F)F)=O)CC12 C1(CC(=O)N(CCN(C(=O)C=CC2CCOC2)CC)CC)CCCC2CC12 C(=O)(CCCCCN(C)C(C1C2COCC12)=O)N1CC(=CC)C1 C1(NC(C(=O)NC(C)C)=O)CCN(C(c2cc3nnn(C)c3s2)=O)CC(O)C1 CC#CCCCC(=O)N1CC(C(N)=O)(CNC(=O)C(C)(F)F)C1 C1(NC(=O)C(F)C2CC2)CCN(C(C2CC2(F)F)=O)CC1 C1(C)(C(=O)NCCC2N(C(Cc3n(C)nnc3)=O)CCC2)CCCC(F)(F)C1 c1(C(=O)NC(CNC(C(C)=C(C)C)=O)CO)cc(F)ccc1Br c1(C(N(CCCCNC(C2C(CC)CCCC2)=O)C)=O)ccc(Cl)c(O)c1 CCCCCC(O)C(=O)NCC1(NC(c2cnn[nH]2)=O)CC(OC)C1 C1(NC(CC)=O)(CNC(C2(c3ccccc3)CC(O)C2)=O)CCCCC1C CC1(C(=O)NC(CNC(c2ccc(-n3ccnc3O)cc2)=O)CO)CCCCC1 C1(C(N(C(C(N2CCC(C(F)F)C2)=O)C2CC2)C)=O)C2(CC2)C12CC2 N1(C(C(CC)=CCCC)=O)CCCC(C)C1CCNC(c1nccnc1C)=O CC1C(NC(=O)OC(C)(C)C)CCCN1CCCN1CCCC1=O C1(CC#C)(C(=O)NC(C)C(CO)NC(C2C3CCCC23)=O)CCCCO1 C(=O)(CC(C)C(=O)c1ccccc1)N(C(CNC(c1c(OC)ccs1)=O)C)C C1(C(C)C)CC(C(=O)NCc2cccc(OCc3cccnc3)c2)CCO1 CCCCC(C)C(=O)N1CCC1CNC(=O)C(C)Cc1c(C)noc1C Cc1ccc(C(N2CCN(C(=O)Cc3sc(O)nc3O)C3CC23)=O)c(=O)n1C S(=O)(=O)(c1nc(N2CCCC(C(F)(F)F)CC2)ccc1Br)NCC(C)(C)C1CC1 c1(C(=O)OCC)nsc(NCC2CC(CNC(=O)C(C)OC)CO2)n1 N1(C(c2cnn(CC(F)F)c2)C(=O)NCCOC)CCC2(CCOCC2)C1 C1(CCNC(C2CCC(C)O2)=O)CN(c2ncnc3c2CCO3)CCS1(=O)=O c1(NC(C2N(C(CNC(c3ccccc3Cl)=O)=O)CCC2)=O)nccc(Br)c1O C(=O)(CC(O)CC(C)(C)C)N1CCC(C(C)C(=O)Nc2ccccc2Br)CC1 N1(C(=O)Nc2ccc(C(C)C)cc2)CCCC(C)(C(=O)NCc2cscc2Br)C1 C1(CNC(C(CCC)=CCC)=O)CC(C)(C)CCC1NC(C1CC(=C2CC2)C1)=O CN1CCN(c2ccnc(C(=O)NCC3CN(C(c4nonc4N)=O)C3)c2)CC1 CC(C)C(N=[N+]=[N-])C(=O)NC1CC1CNC(C1CCOC1c1ccnn1C)=O C1(NC(=O)C(Cl)=CCl)CCCCC12CCN(C(=O)Cn1cccn1)C2 C1(N(C(CCCc2cc(C)no2)=O)C)CCN(C(=O)COCC2CCC2)CC1C N1(C(C)=O)CCC(C2CCCN(C(c3ncoc3-c3cccs3)=O)C2)C1 CCC(C)(CCNC(=O)Cc1cn[nH]c1)NC(=O)C(O)Cn1cncn1 CC1CC(C(N2CC(C3(NC(=O)C#CC4CC4)CC3)C2)=O)CCS1(=O)=O C1(C(=O)NCCC2(OC)CN(C(=O)C3=NNC(=O)C3)C2)CCCC(F)(F)C1 N1(C(=O)NCc2cc(CO)cc(C(F)(F)F)c2)CCCC(C2CC2)CC1 C1(CCC)CCN(C(C2CC(CNC(=O)CCN3CCOCC3)C2)=O)C1 C1(C(=O)NC2CC(CNC(Cc3nc(C(C)C)sc3)=O)C2)CC(=O)N(C(C)C)C1 N1(C(C(CCC)CC)=O)CCCC(C)(C)C1CNC(C1CCN(OC)CC1)=O c1(C(=O)NC2CC3N(C(C(CCOC)C)=O)C(CC3)C2)ccc2oc(O)nc2c1 N1(CCC)C(=O)CCC1C(=O)N(C(C)CNC(C1CC(C#N)C1)=O)C C1(CN(C)C(c2cocc2Br)=O)CCN(C(c2scnc2C2CC2)=O)C1 S(=O)(=O)(CC(=O)NCC1CN(C(=O)COC2CCOCC2)C2CC12)NC c1(C(=O)NC)ccc(C(=O)NCC2CCC2NC(=O)C(C)SC(F)(F)F)cn1 c1(C(=O)NCC(C)NC(c2c(OC)n[nH]c2)=O)noc(C)c1I c1(CNC(=NC)NC(CCOC)C(C)C)cccc(C(F)(F)C(F)(F)F)c1 CCC(C(=O)NCC1C(C)CCN1C(=O)C(c1n[nH]c(C)n1)NC(C)=O)C(C)O C(=O)(C(C)(C)COCC(F)F)NC1(CNC(c2c(C)con2)=O)CCOC1 c1(C(N2CCN(C(=O)C=C(Cl)Cl)CC2c2ccncc2)=O)cc2cccnn2n1 c1(NC(=O)NC2CCC(OC)CC2)cc(=O)n(C(C)C)c(O)n1 N1(C(C2NC(=O)OC2)=O)CCN2CCN(C(c3ccc4nonc4c3)=O)CC2C1 N1(C(C(C)O)=O)CCCC2C1CCN2C(c1cccc(NC(N)=O)c1)=O C1(C(=O)NCC(CNC(COCCC)=O)C)CCc2nccn2CC1 C1(NC(C(C(CC)C)C)=O)CC2(CCC(NC(C3CC(=O)CCO3)=O)CC2)C1 N1(C(C2C(=C)C2)=O)CCCC(N(CCO)C(c2cncc(O)c2)=O)C1 n1(CC(N2CC(C)N(C(c3ncccn3)=O)CC2)=O)sc2ccccc2c1=O N(C(=NCCOCC1CCCCC1)N1CN(C)C(=O)C1C)C(C=C)C C1(NC(COCCCCC)=O)CC(F)CN(C(=O)CNC(c2ccc(C)cc2)=O)C1 N1(C(C(C)NS(CC)(=O)=O)=O)CCCN(C(c2ccc(N)cc2F)=O)CC1C Cc1ccc(C=CC(=O)NCC2(C(N)=O)CN(C(C34CCC3C4)=O)C2)cc1Cl C1(CNC(c2cc(C)on2)=O)CCN(C(=O)C(c2ccc(CO)cc2)(C)C)CC1 N1(C(C(C(C=C)C)C)=O)CCC2(CC1)CN(C(=O)CC1COC3CC1C3)CCO2 N1(C(C)=O)CC2CCC1C(N=c1[nH]c(=NCCC3CC3)[nH]c3ccccc13)C2 C1(CNC(c2ccc(Cl)c(Br)c2)=O)CC2(CCN(Cc3ccn(CCF)n3)CC2)C1 c1(NC)ccc(C(N2CC3(CCC3NC(=O)C(C)SC)C2)=O)c(Cl)c1 N1(C(Cc2cn(CC)nc2)=O)CCCC(C)(CCNC(=O)C(SC)SC)C1 c1(N2CC=CC(NC(CC(=C)C)=O)C2)c(F)cc([N+](=O)[O-])cc1F N1(C(=O)Cc2ccc(Cl)s2)CC(NC(C2CC(F)(CO)C2)=O)C(C2CC2)C1 c1(CCC(=O)NCC(CN(C(C(C(C)C)C)=O)C)C)ccc2c(c1)CCCO2 C(CC(C)C(=O)N1CC(CNC(c2cnsn2)=O)(OC)C1)=CC C1(C(CNC(C(C)(C)C)=O)F)CCN(C(c2cc(-c3ccccn3)c[nH]2)=O)CC1 C(=O)(C1=CC2(CCOC2)C1)N1C(CNC(CCC(=C)Br)=O)COC(C)(C)C1 S(=O)(=O)(c1nc(N2CCC(N3CCC3)C2)ccc1Br)N(CC(N1CCCC1)C)C O=C(N=c1cc(C2CCOC2)[nH][nH]1)C1CCC2(CN(Cc3nccs3)C2)O1 C(=O)(C1=CCC(F)(F)CC1)NC1CCC(CNC(C2=C(C)OCC2)=O)C1 C1(C(=O)NC(C2CC2C(=O)O)C)COCCN(C(C2(C)CNC(=O)N2)=O)C1 C1(CNC(CN(C)C)=O)(CNc2nccc(-c3cnccn3)n2)CCOCC1 CCCC(C)CC(=O)NCC1(C(=O)NC(c2nnc(C)o2)C)CC2(CC2)C1 N1(C(=O)C(c2cc(Cl)cc(Cl)c2)O)CCCN(C(=O)CC2CC2)C(CO)C1 c1(C(=O)NC(C)C)nc(NC(=O)Nc2nc(-c3ccccc3)cs2)co1 c1(CNC(C)COc2ccc(F)cc2)c(-n2cccn2)cccc1F CCCCS(=O)(=O)N1CCC(C(=O)NC2CC3(C2)CC3NC(=O)CC(F)F)CC1 C1(C(N(CC(C)NC(c2ccsc2OC)=O)CC)=O)CN2CCCN1CC2 C1(NC(=O)C=Cc2ccco2)CC2(C1)CC2C(=O)NC1CCC(F)CC1 C1(c2cn(C(C)(C)C)nn2)CC(NCCCS(=O)(=O)N2CCCC2)CCS1 CC(C)(C)C(CNC(=O)CC1(C)CC1(Cl)Cl)NC(c1cn(C2COC2)nn1)=O c1(N2C(C(=O)OCC)CC(F)C2)ncc(F)c2c([N+](=O)[O-])cccc12 C1(C(=O)NC(CC)CN(C)C(c2ccc(Cl)cc2OC)=O)CC2C=CC1CCC2 C1(C(=O)OC)CC=CCN1C(c1ccccc1OC)C(=O)NC1CCOC1 c1(C(=O)NC(C(C)C)CNC(=O)CN2CCC(C)(O)C2)cccc(F)c1Br C(=O)(C1=C(C2CCC2)N(CC2CC2)C(=S)NC1c1ncsc1C)OCC c1(C(=O)NC(C2CCN(C(=O)CSc3nncn3C)C2)C)ccn2ccnc2n1 c1(C(=O)NCCN(C(Cc2c(C)ncs2)=O)CC(C)O)c[nH]c(C#N)c1 c1(C(C)O)ccc(-c2csc(NC(C3CNCC(C(=O)O)C3)=O)n2)cc1 n1(CCC)nnnc1C(c1sccc1C)NCC=CCl c1(C(C(=O)OC)C)cc(Cl)cc(N2CCC(OC)CC2)n1 CCCC(C(=O)NCc1nc(C(=O)NCC(C2CCC2)OCC)co1)OC c1(C(=O)NCCCCCCN(C(C(C(C)C)OCC)=O)C)c(C)nn(C)c1OC C1(CCC)(NC(CCCC=C)=O)CCCN(C(=O)C(CC)n2ccnc2)C1 C(=O)(CCCC(F)(F)CO)N1CC2C(CNC(c3cn(CC(C)C)nc3)=O)C2C1 CC1(C)CN(CC(=O)NCC(C)(O)CN(C)C)C1.c12cc(n[nH]1)C(=O)NC2 n1(CCOC)cc(C(=O)NC(c2ccc(C(=O)O)cc2)C)c(C)n1 Cc1ccsc1C(=O)NCC(C1CC1)NC(=O)CSc1nccn1C C#CCCCC(C)C(=O)N1CCOC(C(N2CCN(C(C)CC)CC2)=O)C1 C1(COC)(CN(C(C2CCCC2O)=O)C2CC2)CN(C(C)=O)C1 C1(CNC(CC2CC(=C)C2)=O)CCC2(CCN(C(c3ccsc3C#N)=O)CC2)O1 C(=O)(CCCCc1ccc(Cl)cc1)N(C(C)CNC(C1CC1CN(C)C)=O)C C1(C(=O)NCCCNC(c2cccs2)=O)CCCCN1C(=O)C(O)CN1CCCC1 c1(C(=O)NC2CCC(NC(c3cccc(OCC)c3)=O)C2)cncc(C)c1C C(C(C(=O)N(CCNC(=O)CC(C)CC)CCOCCO)C(C)(C)C)OCC=C N1(C(CCCCCC)=O)CCC2(CC2)CC1C(=O)NC1CCCOC12CCC2 N1(C(C2C(OCC)CC2)=O)CC2C(CC(=O)N(C3(COC)CCC3)C)C2C1 c1(CC)ccc(CN(C)C(C2CCC2CNC(=O)C(C2CC2)SC)=O)o1 C(C)(CCC(=O)NC(C)CCN(C(=O)C(=O)NC(C)C)C)SC CC(CCCNC(=O)CC1CCCCO1)NC(=O)C(C)NC(c1ccncc1)=O N1(C(C2C(C=C)CC2)=O)CC2CCCC2(NC(c2c(NC(C)=O)c[nH]c2C)=O)C1 C12(C(N3CCC4C(NC(CCn5ccc(C)n5)=O)C43)=O)CCCC1C2(F)F C=CCC(CC=C)NC(=O)CC(CC)NC(c1occc1C)=O N1(C(C2C(NC(c3cn(C4CC4)nn3)=O)CCC2)=O)CCN(C2CC2)C(=O)C1 CCCN=C(NCC1CCCC(O)C1)N1CCN(c2cccc(F)n2)CC1 N1(CC(C)C)N=C(C(=O)N2CC(NC(c3cnc4[nH]ccc4n3)=O)C2)CCC1=O N1(C(C(C)N(C(C)=O)C)=O)CCCC1C1(C(=O)NC(C)CC(C)C)CC1 C(C(=O)NOCC=CCl)(c1cn(C)nn1)NC(C(C)C)=O c1(NC(CCN(C)C)=O)ccc2c(c1)CCN(C(c1cccc(F)c1I)=O)C2 N1(C(c2c(C)n(C)cn2)=O)CCN(C(C2CC2C2CC2)=O)CC1CF c1(C(N2CCN(C(C(CC)F)=O)C(C(C)C)C2)=O)ccnc2c1CCC2 N1(C(c2c(F)ccc(NS(C)(=O)=O)c2)=O)CCOC2(CCC2)CC1 CCC(C)(C(=O)NC1CCCN(C(c2cc(C)c(C)[nH]2)=O)CC1)C(N)=O c1(C(N(C2CCOCC2)CC#C)=O)cnc(CNC(=O)CC2COC(=O)C2)nc1 c1(OC)ccc(C(=O)NC2(C)CC(NC(C3CN(CP(C)(C)=O)C3)=O)C2)c(F)c1 C1(CNC(C2N(C(Cc3nnc(C)o3)=O)CC(O)C2)=O)CCCCC1(F)F c1(C(N2C(CNC(c3ccccc3C(F)(F)F)=O)CC2)=O)nnc2ccccn12 C12(C(=O)NC3CC(NC(C(N4CCC(O)CC4)C)=O)C3)CC=CC(C1)OC2 Cc1ncc(C(N2CC(NC(c3sccc3OC(F)F)=O)C(O)C2)=O)cc1N C1(NC(C(CC)OC2CCCC2)=O)CCCCC1NC(c1ccnnc1)=O C(C(C(=O)N1CC(O)CCO1)NC(=O)Cc1cccc(C#N)c1)OC(C)C c1(C(=O)NC(CNC(C2CCCS2)=O)CO)cc2c(s1)CCC2=O N1(C(c2c(CC)cco2)=O)CCC2CC2(NC(=O)COCc2ccccc2C)CC1 C1(NC(C(C)OCCC=C)=O)CN(C(c2nc[nH]c2C(F)(F)F)=O)CC12CC2 N1(Cc2c(-n3c(C)nc(C(=O)O)n3)cccc2)CCCC(c2ccccc2)CC1 C1(CC)CCN(C(c2cnnc(O)c2)=O)C1C(=O)NCc1nncn1C C1(CNC(C(C)OCC(C)C)=O)CC2CCC1N2c1nnn(C)n1 C1(NC(C2C(CCC)CN(C(=O)CC(C)n3ccnc3)C2)=O)C2CCCCCC12 c1(CC)cc(C)c(C(=O)NC2CCCC2C(=O)NC2(CSC)CC2)o1 C1(C(=O)NC(CNC(c2cc(C3CCC3)no2)=O)C2CC2)CCc2cncn2C1 CC1C(C)N(C(=O)CCC#N)CCN1C(=O)C=Cc1cc(Cl)cc(Cl)c1 C1(c2n(C)ccn2)CC(C(=O)NCCS(=O)(=O)CC2CC2)CCO1 C12(NC(c3ccncc3)=O)CCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)CC1C2 c1(C(=O)NCCC2CCN(C(C(COC)(F)F)=O)C2)cc2c(C)nn(C)c2s1 CC1(C)CCC(NC(=O)NCc2ccc(Oc3ccc(F)cc3)cc2)O1 c1(C(=O)NC(CC(C)NC(C2(SC)CCC2)=O)C)snc(C)c1N C1(NC(C=C(CC)CC)=O)C2CC1CN(C(=O)CCc1nnc(C(C)C)o1)C2 C1(CN(C(c2c(NC)nccc2)=O)C)CN(C(C2CC3CCC2O3)=O)CC12CC2 C1(C(=O)NCCCN(C(=O)CCC2CCOC2)C)CCCN(CC(F)F)C1 C1(C(C)C)N(C(=O)C(n2cc(CCNS(C)(=O)=O)nn2)C)CC12CCC2 CCC(CCCO)NC(C1C2CC1N(C(C1(OC)CCC(C)C1)=O)C2)=O C1(C2CCC2C2CC(Cl)CN2)Cc2ccccc2NC1=O CC(C)CCC(=O)NCC1(F)CC(CNC(c2conc2C(C)C)=O)C1 c1(CCCC(=O)Nc2cccc(NC(CCC(C)SC)=O)c2)ccc(C)c(C)c1 N1(C(=O)Cc2cscn2)CCC2CCCC12C(=O)NC1CC2(CCCCO2)C1 c1(CC)cccc(F)c1C(=O)NC1CCN(C(c2nncn2C2CC2)=O)CC1C C1(NCC2(C(N)=O)CN(C(CSCC)=O)C2)C(C)OC(C)C1C C(C(C(=O)N1CCOCCC1CNC(=O)CC1CC(C2CC2)C1)C(F)(F)F)OC N1(CC#C)CCN(C(=O)C(C)C(C)NC(c2occc2COC)=O)CC1=O C(=O)(CC(C)(C)C(F)F)N1C(C)CC(CC(N2CC3CCC3(CO)C2)=O)C1 C1(NC(CCS(=O)(=O)NC)=O)CC2CC(C1)N(C(c1cc(C)c(C)s1)=O)C2 C12(NC(c3c(C)oc(C)c3C)=O)CCCC1N(C(=O)CCOCC(F)(F)F)CC2 C(=O)(C(CCC(=O)O)NC)N1CC(C)(CNC(CSC)=O)C1 C=CCCC(C)C(C(=O)NCCC#N)N(C(C)(C)CC)C C1(C(=O)NC(C)(CNC(C2(C(F)(F)F)CC(O)C2)=O)C2CC2)OCC2CCCC12 N(C1c2ccccc2OCC1O)Cc1c(C)nn(CC(C)C)c1C c1(C(N2C(C)(C)CC(NC(C3CC4(CC4)CO3)=O)C2)=O)ccc2c(c1)COC2 CC1C(C(=O)NC2CCCC(F)(F)C2)CCCN1C(c1cc(Cl)ns1)=O C(=O)(C1=NN2CCC(C)N=C2N1)NCC(CN(C(Cc1cc(C)sc1C)=O)C)O C(CCC(=O)NC1(C(=O)Nc2ccncc2)CC1)OCC c1(C(=O)NC2(C(C)C)CCNCC2)ccc2c(c1)ncn2C C(=O)(C(F)C(C)CNC(=O)Cc1cnnn1C)N1CC(C#CC)C1 C1(CNC(C(C(C)C)N(C)C)=O)(NC(c2csc(CO)n2)=O)CCCCC1C C1(C(N2C(C)CN(C(c3n[nH]c(C4CC4)c3Cl)=O)CC2)=O)CCc2nn[nH]c2C1 C(=O)(C(=O)C(C)(C)C)NCc1ccc(C(=O)NC(C#C)C(C)C)cc1 Cc1ccc(C=CC(=O)NCC2COCCN2C(C2CCCN2C(C)C)=O)nc1 c1(C(=O)NCC2(F)CCCN(C(c3coc(O)n3)=O)C2)nccc2ccsc12 n1(CC(N2CCC(NC(CCC)=O)C2(C)C)=O)ccc2cc(F)ccc12 C(=O)(CCCC1(NC(=O)C(C)C2CCOC2)CCC1)NC1(CC=C)CCC1 C1(OC(C)C(=O)N(C)CCNC(c2cc(C(N)=O)co2)=O)CCCCCC1 C1(CC(=O)NCC2(NC(c3ccoc3Cl)=O)CC2)CCC(O)C1 C1(CCCC)(C(=O)NCC(CC)NC(=O)CC2CCCO2)CCCCC1 C1(C(=O)NC2CCC(CNC(=O)CC(C)n3cccn3)CC2)(CC)CNC(=O)C1 C1(c2ccccc2)(CO)CN(N2CC3(CCC3)C2c2ccccc2)C1 C1(C(C)C)CN(C(=O)C(C(C)O)NC(C2CC(=O)NC(=O)N2)=O)CC(=O)N1 Cc1ccc(C(=O)NC(C)CCCCNC(c2c(N)cnn2C)=O)c([N+](=O)[O-])c1 C1(C(=O)NC(C(C)(C)NC(C(C)=CC)=O)C)CCc2cc(C)ccc2O1 N1(C(c2ccnc(OC)n2)=O)CC(NC(c2cnc(OC)nc2)=O)C2CCCC12 CCC(C)(COC)C(=O)NCC(C)(C1CCC1)NC(=O)CCCCCN(C)C c1(C(=O)NCC2(C(N)=O)CN(C(C34CC(C)C3C4)=O)C2)ccccc1S(C)=O CC(C)(F)C(C)(F)C(=O)NC(C)(CNC(=O)CCNS(C)(=O)=O)CO C1(NC(C2(C#C)CCC2)=O)CCC(N(C(=O)COC2CCC(C)CC2)CC)CC1 C(=O)(CCCCCc1ccccc1)N1CC2C(CNC(C(C(C)C)SC)=O)(C2)C1 c1(C(=O)NCC(CNC(c2cccc(C(C)C)n2)=O)F)cnc(O)c([N+](=O)[O-])c1 C12(CNC(CCOC)=O)CCCCCC1N(C(=O)COc1ccc(Cl)nc1)CC2 c1(CC(=O)NCC2CC2C(=O)NCCCCC2CCCC2)ccccc1F c1(C(C(=O)NCCOC)N(C)CCn2ccnc2)cnn(C2CCC2)c1 C1(C(=O)Nc2cccc(CCCC)c2)CCN(C(=O)COC(C)=O)CC1C c1(C(N2CCCC(NC(=O)CCC(F)F)C2)=O)ccc(=O)n(C2CC2)c1 N1(C(C2C(C(=O)NCCNCCO)C2)=O)CCc2cc(F)ccc2C1 C(C(C)(O)CC(=O)N(C1CCCN(C(C2CC(SC)C2)=O)C1)CCO)OC C(CCC(C)C(=O)NCC1(C(N)=O)CN(C(c2n[nH]cc2[N+](=O)[O-])=O)C1)OC N1(C(CC(C=C)(C)C)=O)CCC2CN(C(c3nnn(C)c3C(F)F)=O)CCC2C1 Cc1nnc2c(C(=O)NC3CC(NC(=O)Cn4cnnn4)C34CCC4)nccn12 C(=O)(CCC(=O)NC1CC2(C1)CC2NC(=O)OC)NCC.C1(=O)CC2CC2N1 C(=O)(C(F)(F)CO)Nc1c(C(=O)NC(CCOC)COC)con1 C1(NC(=O)CC2CCC(O)C2)CN(C(=O)COCCCF)CC1CO N1(C(c2cnc(C)n2C)=O)CCC(CO)CC1C(=O)NC1CC1(C)C(F)F C1(C2CCCOC2)(NC(C2N(C(c3cc(C)[nH]c3C)=O)CCC=C2)=O)CC1 N1(C(c2c(CC)onc2)=O)CCC(C2(NC(=O)CC3(C#N)CCC3)CCC2)CC1 C1(NC(C2CC(C)CN2C(C2CC3C=CC2O3)=O)=O)CC(CO)C12CCC2 C(CC(=O)NN1CCCC1CNC(=O)CN1CCC2(CC2)C1)C1C(C)C1 Cc1cnccc1CC(N1CC(C)(C)C1c1cnn(C)c1)=O C1(C(=O)NC2CC2NC(C2CC(F)(CO)C2)=O)(OC)CCCCCCC1 c1(CC)ccc(F)cc1C(N1CC(F)CC1CNC(C1CCCC12CCC2)=O)=O C1(C(=O)NCCC(CNC(=O)CCNS(C)(=O)=O)OC)CC2C(C1)C2(F)F c1(NC2CC(CNC(c3c(CC)onc3)=O)C2)nc2ccc(N)cc2s1 C1(C(=O)NC2C(NC(C(C(=O)OC)C)=O)CCCC2)COc2cc(F)ccc2O1 C1(NC(c2nc(C)sc2C)=O)CCCC(C(=O)NCC2CC2[N+](=O)[O-])CC1 C1(NC(COCCCCC)=O)CC2CCC(C1)N2c1ncns1 N1(C(CC2(OCC)CC2)=O)CCC(C=CC(=O)NC(C)Cc2ncn(C)n2)CC1 N1(C(C(COC)COC)=O)CCOC2CN(C(=O)CNC(=O)CN(C)C)CC12 c1(C(N(CCCCCNC(c2cnnc(O)c2)=O)C)=O)ccc(C2CC2)nc1O N1(C(C(CCC)c2ccccc2)=O)CCCN(C(c2ccoc2C)=O)C(CO)C1 c1(C(=O)NCC(CN(C(C2N(C(=O)OC)CCC2)=O)C)C)ccc(C(N)=O)cc1 Cc1nc(-c2ccc(Cl)cc2)sc1C(=O)OCC1COC(C)(C)C1 c1(C2C(C(=O)OC)C2)ncc(C(=O)N(C)CC)[nH]1.C(=O)(CCC(=O)OCCN)NC S(=O)(=O)(c1cccc(F)c1)NCC(=O)N(CCNC(c1c(C)ncnc1)=O)C N1(C(CC(C)CNC(C2(F)CCCCC2)=O)=O)CC(O)(C2CC2)C1 c1(C(N2CC(NC(=O)Cc3nc[nH]n3)(CO)C2)=O)csc2nccn12 Cn1ccc(C(=O)NCC2OCCC2C(=O)N(C2CCCC2F)CCO)c1 C(=O)(C(C(C)(C)C)c1ccccc1)OCC(c1c(C)[nH]c(C(C)(C)C)c1)=O N1(C(C(C)=C(C)C)=O)CC2(CCC2NC(C2CCCN2C(c2cccs2)=O)=O)C1 C(=O)(CCCC(=O)C(C)(C)C)NCC(CC)NC(C1CC2CCC1O2)=O C(=O)(C(CNC(C1CS(=O)C1)=O)C(C)C)NCC(C#C)CC1CC1 N1(C(c2ccc(CC)nc2)=O)CC2(CC2)CC1C(=O)N(C)Cc1nnc(O)o1 CCCCCCCC(=O)Nc1cnc(Cl)cc1C(=O)Nc1cnc(F)nc1 N1(C(C2(C=C)CCC2)=O)CC2CC(NC(=O)C(c3cnn(C)c3)C)CC2C1 C1(NC(CCOCC)=O)CC(CNC(c2ccnc(C(C)(C)C)n2)=O)C(O)C1 c1(OC)ccc2c(C(=O)Oc3cccc(F)c3O)csc2c1 C(=O)(CCC=C(C)C)N(CCC(=O)N(CCCC)CC)C1CCCC1 C1(c2ccccc2)(C(=O)NC(C(C)C)CNC(=O)C(C)CF)CC(F)(F)C1 C1(C(=O)NCCF)(COC)C=CCN1C(=O)CC1CCC(C)(C)C1 N1(C(C(C)CC(F)(F)F)=O)CC2CN(C(=O)CCCCc3cnc[nH]3)CC2(C)C1 c1(C(=O)NC(CNC(c2c(CC)cco2)=O)C(C)C(C)C)ccc2c(c1)OCC2 C12(C(=O)NCC(C)OCC#C)CC(CN(C(C3(C#N)CC3C)=O)C1)C2 C(=O)(C1CCc2c[nH]nc21)NCC(C)(C)OCC(=O)NC1CC2CCC1C2 c1(C(N2C(CC)C(NC(C3CCCN3N=O)=O)CC2)=O)cc(Cl)cc(Cl)c1Cl C1(CNC(C(C)(C)n2cc(Br)cn2)=O)CCN(C(=O)CC(F)F)CC1O c1(C(=O)NCC2CC(O)(CNC(CS(N)(=O)=O)=O)C2)ccc([N+](=O)[O-])cc1 Cc1nc2cc(C(=O)NC3CCC3NC(=O)CCCS(N)(=O)=O)cnc2s1 O=C(N(O)Cc1cn(Cc2nc(C(=O)O)cs2)nn1)C(O)C1CCCCC1 CC1(C)CCC(c2nc(-c3sccc3S(N)(=O)=O)no2)CC1 O=S(=O)(c1cccnc1NC1CC(N2CCCC2)C1)NC1CCN2CCCCC12 C(=O)(C1SCCc2ccccc21)NCCC1(NC(C2CC3COCC3C2)=O)CC1 CN(C1c2cc(Cl)cc(Cl)c2CC1O)C(=O)NCc1ccoc1 C1(OCCNC(CC=CC)=O)CCN(C(=O)C(F)C2CC2)CC1 Cc1c(Br)ccc(F)c1C(N1CC(N(C)C(c2cc(F)c(F)cc2I)=O)C1)=O c1(CC)ccc(N)c(C(N2CCCN(C(c3nn(C)nc3Br)=O)CC2)=O)c1 C1(C(F)(F)F)(C(N(CC(CC)NC(c2snc(O)c2Cl)=O)C)=O)CCCCO1 c1(OC)nc(C(=O)NC(C)(CNC(=O)CCC2CC2(F)F)CO)ncc1F CCC(C)(C)C(O)C(=O)N1CCCCC(CNC(C2(N=[N+]=[N-])CC2)=O)C1 C1(C(N2CC(CC)N(C(=O)CCC(C)(C)N(C)C)CC2)=O)CCC(N=[N+]=[N-])CC1 Cc1ccc(C(=O)OCc2ccc3ccccc3n2)cc1S(=O)(=O)NCC#N C1(C(=O)NCC(C)C(C)(F)F)CCN(C(c2ccccc2CC#N)=O)CCO1 N1(C(c2ccc(OC)o2)=O)CCN(C(C2CC(=O)N(OC)C2)=O)CC(C)C1 C(N=c1[nH]c2ccc(F)cc2o1)C1OCC(CNC(C(CC#C)(C)C)=O)C1 C1(C)(NC(=O)NCC(CC(C)C)(C)Cc2ccccc2)COc2ccccc2O1 C(=O)(N(CC1CC(F)(F)C1)NS(=O)(=O)c1cc(Br)ccc1Cl)OC(C)(C)C CC1=CC(C)C(c2cn(CCCC(=O)N3CC(c4ncc[nH]4)C3)nn2)CC1 Cc1cc(NC(C2CCN2C(C2(C#N)CC23CCC3)=O)=O)cc(C)c1C c1(C(=O)NC(CCCNC(C2(COC)CC2)=O)CO)cc([N+](=O)[O-])cn1C N1(C(C(c2c(F)cccc2F)NC(=O)OC(C)(C)C)=O)CC2CC1CS(=O)(=O)C2 C=CC1(C(=O)NCCC2CC(CNC(=O)C3=CCOCC3)CO2)CCCCC1 Cc1cc(C(=O)NC2C3CC2N(C(=O)C=Cc2ccc(Cl)cc2)C3)c(O)nn1 N=c1nc(SCC2CCOC3(CCC3)C2)c2nc[nH]c2[nH]1 N1(C(C=CC=CCC)=O)CC(NC(=O)C(=C2CCCCC2)F)CC(C)C1 c1(C(=O)NC2C3CN(C(C(C)(C)OC)=O)CC32)cnc2c(=O)[nH]ccc2c1 CCC(C)(C)C(C)CC(=O)N(C(C)CNC(=O)C=Cc1ccco1)C c1(NC2CC3(CN(C(CSCC)=O)C3)C2)cccn2nc(C)nc12 Cn1cc(C2CC2NC(C2CCN2C(C2(n3nccn3)CC2)=O)=O)cn1 N1(C(C2CCC(C(C)C)CC2)=O)CCCC(C)(CNC(=O)CCc2ccsc2)C1 S(=O)(=O)(c1cccs1)N(C1COCC1O)Cc1c(C(=O)O)cccc1 CC1(C(=O)NCCC2CN(C(C3CC4CCC4C3)=O)C2)CCC2(CC1)CC2 N1(C(c2c(CC)nc(Br)s2)=O)C(C)CC2CN(C(C)=O)CC12 N1(C(C(C)c2ccco2)=O)CCC(CNC(=O)CC2CC3(CCC3)CO2)C(O)C1 c1(C(N2C(CN(C(C3C(CC)C3)=O)C)CCC2)=O)cncc(Cl)c1 c1(OC)ccc(C(N2CC3CN(C(=O)Cn4nc(Cl)ccc4=O)C3C2)=O)cc1Br N1(S(CC(=O)OC)(=O)=O)CC2(CN(C(c3cc(F)ccc3F)=O)C2)C1 N1(CC2C(C)(C)C(O)C2)CCC(=O)N(Cc2cccnc2-n2cccn2)C1=O Cc1ccnc(Cl)c1C(=O)NCC1=CCN(C(C2CC2(C)C(C)C)=O)CC1 c1(C(N2CC(C)C(NC(CCC#C)=O)C(C)C2)=O)cc2c(Cl)nccc2o1 c1(C(=O)OC)ccc(C(N2CCC(CF)(NC(=O)Cc3ccco3)C2)=O)cc1C C1(C(N(CCNC(C2(CO)CC(F)(F)C2)=O)CC)=O)CCC2(CCC2)CO1 CC12CCC(C(N3CCCC(C)(NC(=O)CC4CCS(=O)(=O)C4)C3)=O)(CC1)CO2 C(=O)(N1OC2CCC1C2)c1c(NCc2c(C)c(Cl)ccc2)ccc(Cl)c1 C12(C(N3CCCC(CCCCC)C3)=O)COCC1CN(C(=O)C(F)C(C)(F)F)C2 C=CC(C)CC(=O)N(CCCNC(c1cc(CC2CCC2)c[nH]1)=O)CC c1(C(=O)NC(CNC(COCC=C)=O)CO)cc(COc2ccccc2)on1 Cc1nc2nccc(C(=O)NCCC3CCCN(C(=O)C=CCO)CC3)n2n1 C1(NC(C(CN(C(C2=CCN(C)C2)=O)C)(C)C)=O)CCC2(CCCC2)C1 Cc1cccc2cc(C(=O)NCC(O)CN(C)C(C34CCCC3C4(F)F)=O)oc12 c1(OC(C)C)nccc(C(=O)NC2CCC(NC(C3CC(C(F)F)C3)=O)C2)c1F C1(C(=O)NCc2snc(C)n2)CN(C(C2CC(=O)NC2=O)=O)CC12CCC2 C(C(C)(C)CN=c1nc2sccc2c(NCC2CC2(Cl)Cl)[nH]1)SC C(=O)(C1=CC2CCC1C2)NCCOCCN(C)C(C1CCC(=O)NC1)=O C1(O)(C(C)C)CCCN(C(=O)C(=O)NCCN2CCS(=O)CC2)C1 C1(C(=O)NCCCN(C(c2nccc(C(F)F)n2)=O)CC)CC12CCCC2 N(C(=NCCc1ccc(Cl)cc1)NC(C)CCc1ccco1)C(C)C CC(C)C(CC(=O)N1CCC=C(F)C1)NC(=O)CS(C)(=O)=O c1(NC(NNC(c2c(C#N)cc(Cl)cc2)=O)=O)ccc2c(c1)C(=O)CC2 N1(C(c2cn(CC)nn2)=O)CCN(C(=O)C(F)(F)C2CCOCC2)CC1COC CCC(C)CCCC(=O)N1CCCC1C1(C(=O)NCCOC(F)F)CC1 c1(OC)ccccc1CC(=O)NC(CO)C(C)NC(=O)CCSc1nnnn1C N1(C(C(F)=CC)=O)C2CCC1CC(NC(c1ccc(-c3ccncc3)o1)=O)C2 C1(C2C(NC(CCSCC)=O)C2)COCCN1C(=O)C(C)NS(=O)(=O)CC c1(C(=O)NC(C)CN(C)C(C2CCCCN2N=O)=O)cc2ccccc2[nH]c1=N C12(CNC(c3c(C)n(CCC(C)C)nc3)=O)CCC1CCN2C(=O)CN(C)C C1(NC(CSCCCC)=O)CN(C(c2ccc(O)nn2)=O)C2(CCC2)C1 N1(C(C2(C=C)CCC2)=O)CCC2CN(C(c3c(S(C)(=O)=O)cnn3C)=O)CC2C1 N1(C(C(CC)CC)=O)CC(NC(=O)CS(=O)(=O)N2CCOCC2)CC2(CCC2)C1 Cc1ccn(C)c1C(=O)N(CCC(C)NC(=O)C(c1cnn(C)c1)O)C C(=O)(CCCCCC(C)O)NCC(CCNC(c1c(C)nc(CC)o1)=O)O C(=O)(CC1=CCOCC1)NC(CNC(=O)Cc1cc(Cl)ccc1O)Cl CCC(C(=O)N(CCCCNC(=O)CC1CC(C)=NO1)C)OC N1(C(C(=O)O)=O)CC(O)CCC1C.C1(NC(=O)OC(C)(C)C)CCC(OC)C1 c1(C(N2CCCN(C(C(C(C)(C)C)C#N)=O)CCC2)=O)cc(Cl)cc2c1OCC2 Cc1oc(C)c(C(=O)NCc2csc(C(N3C(CO)CC3CO)=O)c2)c1C c1(C(=O)NC(CC)CNC(C2(n3cccn3)CCCC2)=O)c[nH]c2ccccc12 C1(NC(CC2(OC)CC2)=O)CCC2CCN(C(=O)CN3CC4CC4C3)C1C2 c1(CC(=O)NCCN(C(C(CC#C)O)=O)C(C)C)c(Cl)cccc1Br CON(CCC(=O)NCc1cn(C)nn1)C(=O)C(F)(F)CO c1(OC)cc(C(=O)NCCN(C(=O)C(C#N)CC2CC2)C)cnc1C(F)(F)F Cc1nc(C)c(C(=O)N(C(CNC(C2CCOC(=O)N2)=O)C2CC2)C)nc1C N1(CC(N2C(C(CCC)C)CCC2)=O)CCN(C(c2cc(CC)ncn2)=O)CC1 c1(OC)ccccc1C(C(C)(C)C)NCCc1ccn(C(C)C)n1 CCCCC(CNC(=O)CCC1CCN(C(C2(C3CC3)CC2)=O)C1)CC C=CCCC(=O)NC(C1CC(n2cc(C3(OC)CCCC3)nn2)C1)=O c1(CC(=O)NC(CNC(C2ON=C(C)C2)=O)C2CC2)ccc(F)cc1Br c1(CCNC(C(N2CC(C(C)=O)C2)=O)=O)c(C)[nH]c2ccccc12 N1(C(C(c2ccccc2)OC)=O)CCCC(N(C)C(c2cc(C)co2)=O)C1 CC1CC(CNC(=O)CCN(C(=O)CCC2CCC(=O)C2)C)=NO1 Cc1cccc(C(=O)NC2CC2NC(=O)CSCc2ccccc2)c1Br C(C)(CNC(=O)CN1CCCCC1)(CC(C)C)NC(c1cncc(C)n1)=O c1(OC)cc(-c2ccc(-c3nccn3CCC3CCCC(C)C3)cn2)ccc1C Cc1cc(O)ccc1-c1cncc(C(=O)Nc2ccccc2C2CC2)n1 Cc1nn(C)c2ncc(C(=O)NC3C(C)CN(C(=O)CC(C)(C)F)CC3C)cc12 N(C1CCc2cc(CNC(=O)C(O)CSC)ccc21)C(Cc1scc(CC)n1)=O N1(C(C(CCF)NC(c2ncc(OC)nc2)=O)=O)CC(S(C)(=N)=O)C1 c1(C(N(CCNC(C2(C)C(C)C2)=O)C)=O)ccnc(OC(C)(C)C)c1 C1(NC(CSc2cccc(C)c2)=O)CCC12CN(C(C1CCCC3(CC3)C1)=O)C2 N1(C(C(CC(C)(C)C)O)=O)CC=C(C(C)(C)C(=O)N2CCCC2CF)C1 C(C)(N=c1cc(Cl)nc(S(C)(=O)=O)[nH]1)C1CCN(C(c2cc(C)nc(C)n2)=O)C1 C(=O)(C(C)(C)C(F)(F)CC)NCC(CC=C)NC(=O)C(C(C)C)SC C12(C(N3CCNCC(F)(F)C3)=O)CCCC1CC(F)(F)CC2 C1(N(CCCC)C(C2CC2C2CCCO2)=O)CCN(C(c2ccc(C)o2)=O)CC1 C1(C(=O)NCCCCC2C(C)C2)CC2CCC1N2C(=O)CN1CC=CC1 n1(CC)cc(C(=O)NCCC(O)CNC(=O)C(=O)NC2CC2)c(C2CC2)n1 N1(C(c2cccc(CC)c2F)=O)CCN(C(c2nn(CC)cc2Cl)=O)CCC1C c1(C(=O)NCC(C2CCCC2)NC(C(c2cncnc2)C)=O)ccncc1Cl N1(C(Cn2nnc(C)n2)=O)CCC2(C=C(C(=O)NCC3CC34CC4(F)F)C2)C1 N1(C(C2CCN(C(C34CCC(CC3)C4)=O)C2)=O)CCCC(Cc2ncon2)CC1 O=C1CCC(CC(N2CCC(C(=O)NC(CO)C3CC3)(CO)C2)=O)CN1 C1(C(=O)NCc2cc(C(N3CC(OC(N)=O)C3)=O)on2)CC12CCOCC2 Cc1sc2ccccc2c1C(=O)NCC(C)CN(C(=O)C(=O)NC(C)C)C C1(C(=O)NCC=CCC(=O)N2CC(CCO)C2)CCCC1C1CC1 Cc1c(F)ccc(C(N2CCC2CNc2cccc(-c3ccccc3)n2)=O)c1Cl c1(C(=O)OC)cnc(N2CC(F)CC2CNC(=O)CC23COC(C)(C2)C3)cc1C c1(OC)c(F)cc2nc(N(C)Cc3ccc(F)cc3C)sc2c1F Cc1oc(C)c(C(N2CC3CC(NC(c4ncoc4C(C)(C)C)=O)C2C3)=O)c1C c1(C(=O)NC2CN(C(C3(C(C)C)CCC3)=O)CC2F)cc(Cl)c(Cl)nc1Cl c1(C(=O)OC)cc(S(=O)(=O)N2CCCC3NC(=O)CC23)cnc1C C1(CN(C(=O)CCc2ccc(Cl)s2)C)CCCCN1C(=O)CO c1(OC)nccc(C)c1C(N1CCCC1)=O.N1(CC(=O)N2CCC2)CCC(C)CC1 n1(CC(N2C(C)(CNC(C3CC3C(F)F)=O)CCC2)=O)cc(S(C)(=O)=O)cn1 c1(CC(N2CC3C(CN(C(C4C(OC)CCC4)=O)C)C3C2)=O)ccc(C)c(C)c1 c1(CC(=O)NCCC(CCNC(C=CC(C)C)=O)C)cccc(Cl)c1F N1(C(Cc2c(SC)cccc2)=O)CC2CC1CCN2C(c1csc(NC=O)n1)=O CC1(C)C(CO)CCN1C(=O)CONC(c1ccccn1)=O C1(O)(c2cn(CCC3CN(C(c4ccn(CC(C)C)n4)=O)C3)nn2)CCOCC1 C1(NC(C(C)SC(F)(F)F)=O)COC2(C1)CN(C(C13C4C5C1C1C3C4C51C)=O)C2 C1(CC(=O)Nc2ccc(-c3ncon3)cc2)CCc2sccc2C1=O C1(C(=O)NCCC(C)(C)NC(CCNC(COC)=O)=O)CN2CCC1(C)CC2 CC1CC2CN(C(=O)OC(C)(C)C)CC2N1C(=O)COc1cc2ccccc2o1 c1(C(N(C(C(OC)OC)C)C)=O)cc(C)n(-c2ccc(Cl)cc2)c1C C1(C(N(C)CC2CCC(NC(CC3C(OC)CC3)=O)CC2)=O)CC12CCSCC2 C1(CCC)CN(C(c2ccsc2C)=O)CCN1C(c1ccc(Cl)c(OC)c1)=O C(=O)(C(F)C(C)(F)F)NC1C(C(=O)NC(c2cn[nH]c2)C)C1(C)C c1(C(=O)NC(CNC(C(C(CC)O)(C)C)=O)CO)cc(C)c2c(O)n[nH]c2n1 c1(SC)nc(N2CCN(CCNC(=O)C(C)(C)CSC)CC2)cc(Cl)n1 C(CCCCCC(=O)N1CCOC(C2CC2)C1)NC(CCC(C)OCC)=O CC(C)C(C)(C)C(c1nnnn1C1CCCC1)NC(C1CCC1)C c1(NC(C2CCN(C(C3CCC4(CC3)CC4)=O)CC2O)=O)cnc(F)c(Br)c1 C12(C(=O)OC)CCCC(C(=O)NCCCNC(=O)CC3CCCCCC3)(CC1)C2 c1(OC)ccc(CCC(N2CCC(NC(=O)C3=NOCC3)C2C)=O)cc1Br N1(C(c2c(C)cco2)=O)CC(C(=O)NCc2cc(Cl)cc(Br)c2)CC(F)C1 C1(C)(C(=O)NCC23CN(C(C(C)(C)C4CCCO4)=O)C(C2)CO3)CCCCNC1=O C1(C(N(C(C)CNC(c2ccn(CF)n2)=O)C)=O)CCc2n[nH]cc2C1C c1(C(=O)NC2CC(NC(c3cnn(C)c3Br)=O)C2)cnc2n1CCCC2 c1(C(CC(=O)NCC2(F)C(C)C2)=O)ccoc1C(=O)NCCOCCOCCO n1(CC)cc(Cl)c(C(=O)NCC(C2CCCN2C(C2(F)CCCCC2)=O)(C)C)n1 c1(C(=O)NCC(CO)NC(C(C=C)(C)O)=O)cccc(OC)c1C Cc1oc2ncnc(O)c2c1C(=O)NCC1CN(Cc2ccccc2C(=O)O)C1 C1(C(=O)O)CN(C(c2[nH]c3ccccc3c2C(F)(F)F)=O)CC12CCCC2 C#CCCC(=O)N1CC(O)(C(F)C(=O)N(CC(C2CC2)OC)C)C1 C1(C(=O)NOCCc2ccccc2)CC=CCN1C(C1CCCOCC1)=O CCC(CC(C)C)C(=O)NCC1CCC2(CN(C(=O)Cn3nnc(=N)[nH]3)C2)O1 C#CCC(C)C(=O)NC(C)CNC(=O)C(N1CCN(c2ccccc2)CC1)C C(C)(CO)(C(=O)NCc1ocnc1C(=O)NC1CC(O)C(F)C1)OC c1(OC)ccc2c(CCC(=O)N(CC(C)NC(=O)C#CC3CC3)C)c[nH]c2c1 Cc1cccc(C(c2cc(Cl)cnc2-c2cncc(F)c2)=O)c1O CC(C)(CNC(=O)CCc1nc2ccc(Cl)cc2[nH]1)C#C[Si](C)(C)C c1(C(=O)NCC(CO)NC(=O)CCc2cnoc2)cc2n(n1)CCCC2O C(CS(=O)(=O)Cc1cccc(NC(=O)C(=O)N2CCC2c2ccc(Cl)cc2)c1)OC C1(C(C)C)(C(=O)NCCCOCCC(=O)NC(C(C)C)c2ncc[nH]2)COC1 CN=c1[nH]c(C(=O)NCC2CN(C(C3CC(F)(CO)C3)=O)CC2C)cs1 N1(C(=O)C(Cl)=CCl)CCC(C2CCN(C(=O)CCCOc3cccnc3)C2)C1 N1(C(COCCC(C)C)=O)CCC(C2CC2)(CNC(=O)CCN2CCCC2)C1 CC(C)(CCN=c1ccn2ccnc2[nH]1)NC(=O)CC1(O)CCC1 CC1OCCN(C(=O)CCN(C)CCO)C1C(=O)NC1CCCC1C#N C1(C(=O)NCC(C)N(C(C(CC(=O)OC)C)=O)C)CC2CCCCCCC12 CCC(C)(C)C(O)C(=O)N1CCCCCC(NC(C2CC(=C3CC3)C2)=O)C1 c1(N2CC=C(CNC(C3N(C)C(=O)NC3)=O)CC2)nc(Cl)nc2c1CCOC2 CCC(CC(=O)N1CC=CCC1C(=O)NC(CCOC)C(C)C)C(F)F Cc1cc(CC(N2CCC(CO)(NC(=O)C3=CCCC3)C2)=O)cc(F)c1 N1(C(Cn2ccc(C)n2)=O)CCCC(C)(CNC(=O)CCN2CCC(F)C2)C1 Cc1ccc(C(C)NC(C2(C(C)NC(=O)COCC(C)(C)C)CC2)=O)o1 C(CCC(c1nnnn1CCCOCC)NCCc1noc(C)n1)OCC CC1(C(=O)NCC(c2ccccc2F)NC(C2CCOC2)=O)CC2(CC2)C1 n1(CCC)ccnc1C(C)NC1(c2nnnn2CCOC)CC1 CC#CCC(C(=O)NCC(C)CC1CC1)NC(c1cncc(OC)n1)=O Cc1ccc2cc(C(N3CCC(CC(=O)N=c4cnn(C)[nH]4)(O)CC3)=O)[nH]c2c1 N1(C(C(CC2CC2)OC)=O)CCC(C)(CCNC(=O)C(F)CC2CCOC2)CC1 N1(C(Cc2cccc(OC)n2)=O)CCC(NC(C2COC(=O)O2)=O)C2(CCC2)C1 C1(C(N2CC(C)(NC(C(CC)NC(C)=O)=O)C2)=O)COc2ccc(F)cc2C1 c1(C(N(CCC)CC)=O)coc(C(C)NC(=O)C(n2cc(C)cn2)C)n1 c1(CNC(C(C)SCCCC)=O)cccc(C(=O)NCc2cncn2C2CC2)n1 c1(C(=O)NCC2C(CNC(=O)CO)C2)cc2cc(Br)sc2[nH]1 Cc1ncc(C(=O)NC2CCC(CNC(C3(O)COC3)=O)C2)n1C C1(C)(CC)CN(C(c2ccc(C)cc2F)C(=O)NC2CCCC2)CCO1 c1(C(=O)NCCC(C)NC(=O)C(C)Cn2ccnc2)cnccc1C#N n1(CC)ccc(=NC(=O)CC2(CN(C(c3cnn(C)c3Cl)=O)C3CC3)CC2)[nH]1 c1(SCCS(Cc2scc(C(=O)OC)n2)=O)cnn2c1OCCC2 C1(CNC(CC=CC=C)=O)CCCC(NC(=O)CN2CC(C)C2)C1 n1(C(C)C)cc(Br)cc1C(=O)NCC1CC(NC(c2ncccc2N)=O)C1 CCC1=NOC(CC(=O)NC2(CCC(=O)N3CC(C(=O)NC)C3)CCCC2)C1 CC(C)C(CNC(=O)CC=CCc1ccccc1)NC(=O)C(C)(Cl)Cl C1(C(N(C2CC3CC2N(C(=O)CNS(C)(=O)=O)C3)C)=O)CC(C2CC2)=NO1 N1(C(CNC(C)=O)=O)CCC2(NCC(=O)NCC(C)(C)C)CCCC12 N(C(=NCCC1Cc2ccccc2O1)N1CCC(OC(F)(F)F)CC1)C1C(C)C1 C1(C(=O)Nc2cccc(C(C)=O)c2)CN(C(C2(Br)CC2)=O)CC(C)(C)C1 N1(C(CSC)=O)CCCC2(CCCCC2CNC(=O)C(C)Nc2cccnc2)C1 C(C(=O)NCCN(C(c1cnc(CC2CC2)s1)=O)CC)(C(C)C)SCC c1(C(=O)NCC(=CC(=O)NC(COCC)C)C)ccc(O)cc1 C1(NC(C(CC(C)C)NC(CC=CC)=O)=O)CN(C)C(=O)C12CC2 N1(C(CC(C=C)CC)=O)CCC2CCC(C1)N2C(C1CCC(C(=O)OC)CC1)=O c1(C(=O)NCCN(C(C2C(OC)CCC2)=O)CC2CC2)cc2cccc(C)n2n1 c1(C(N2C3CN(Cc4cc(F)cc(C)c4O)CC32)=O)cc(Cl)c2cc[nH]c2c1 c1(C(C)=O)ccc(C(=O)NCc2cc[nH]c2C(=O)NC(C)C2CC2)[nH]1 c1(C(=O)NC2CCCN(C(=O)CO)CC2)ccc2nncn2c1 N1(C(C(CC)N(C)C)=O)CCc2ccccc2C(NC(=O)CSC(=N)N)C1 c1(C(=O)NC(CC)CN(C)C(c2ccc(CO)s2)=O)c(C)cccc1Cl c1(N(C)C)cc(C(=O)NC2CCCC(CNC(=O)C3=NOCC3)C2)ccn1 CC(C(C)(C)C(=O)NOCCCO)NC(=O)CCc1ccn(C)c1 C1(CC)CN(C(C2CCC2)=O)CCC1NC(=O)C(O)Cc1ccccc1 c1(NC(C2(C)CCN(Cc3ccc(C)nc3)C2)=O)cccc2c1OCCO2 c1(OC)ccc(S(=O)(=O)N2CCCC(NC(c3cccc(C(F)F)c3)=O)C2)cc1 CCCCC(C(=O)N(CCCC(N1CC2CC1(C(F)F)C2)=O)C)C(C)C n1(CC)nc(C(=O)NC2(C(=O)N(C)CC3CCCCC3O)CC(O)C2)cc1C C(=O)(C#CC1(C)COC1)NC(CC(C)C)C(=O)N(CC(F)Cl)C C=CCC(C)(CC)C(=O)NC1CCOC1C(=O)NC(C(=O)OC)C1CC1 CCCCC(C(=O)N1CCC(NC(c2sncc2Br)=O)C1(C)C)N(C)C c1(CN(C(C)(C)C)CC2CCCO2)cnc(-c2ccco2)s1 CC1(C)CCC(C)(NC(=O)CC(CNC(c2ncc[nH]2)=O)C2CCC2)CC1 C1(C(=O)NCc2noc(C3CC3)n2)CCCCN(C(C2C=CC=CC=C2)=O)C1 C(=O)(C(C)C(=O)NCC1CC(C(=O)NCC#CCCO)CO1)OC C#CCCC(C(=O)NC(COC)C(C)C)NC(c1ccc(O)c(C)c1)=O C1(NC(=O)C(C)Oc2ccc(F)cc2Cl)CC(CNC(C)=O)C12CCC2 CCCCC(C(=O)N(CCNC(=O)Cc1nc2c([nH]1)CCCC2)CC)C(C)C CC(C)P(=O)(CC(=O)NCC#CCNC(C1CCS(=O)(=O)C1)=O)C(C)C N1(C(CCCC)CCC)C(=O)C2N(CCCC2(C)C)C1=O c1(CC)ccc(N=c2scc(-c3cnn(C)n3)n2C2CC2(C)C(F)F)nc1 c1(C(N(C2CCC(NC(=O)COc3ccccc3)C2)C)=O)cccc2nonc12 Cc1csc2ncc(C(=O)NC3CCCC3NC(=O)CSCc3ccncc3)n12 c1(C(=O)OC)cc(C)c(CN)cn1.C1(CO)C2CCC(C2)C1OC c1(NC(N(CCC(C)(O)c2ccccc2)C2CC2)=O)cccc2c1CCS2(=O)=O C(=O)(C1CCCc2cccnc21)N1CC2CN(C(CSCC#C)=O)CC(C1)O2 c1(C(N(C(CC)C)CC(=O)O)=O)ccc(C(C)(C)C)c(I)c1 N1(C(C(=O)NC(C)C)=O)CC2(C1)CN(C(C1CC(C(F)(F)F)C1)=O)CC2CO N1(C(C2(C)CCOC2)=O)CCOC(C(=O)NCC(c2ccco2)O)CC1 CN1CCc2ccc(C(=O)NCC3(NC(=O)CC(C)(C)C4CC4)CCOC3)cc21 N1(C(c2cccc(C)n2)=O)CCC(C)C(NC(=O)COCC(C)C)C1 Cc1ncc(C(=O)NCC2=CCNCC2)c(Br)c1Cl C1(C(N(C(C(C)C)C)C2CC2)=O)CN(C(=O)Cc2cnsc2)CCC1(C)C C(=O)(C(F)C(C)CNC(=O)CCNC(N)=O)N(C1CCC(C)CC1)C C(C(C)CC(=O)NC1CCCC1NC(C1CCOC1(C)C)=O)OC C12(CCNC(C(C(C)O)C)=O)CCC(CC1)N(C(=O)CCNS(C)(=O)=O)C2 C1(N(C)C)(C(=O)NCC2CCCN(C(=O)C=CS(C)=O)C2)Cc2ccccc2C1 Cc1cc(CNC(C23CC(CO2)N(C(c2ccsc2C)=O)C3)=O)cnc1C C(=O)(C(F)C(F)(F)F)NC(CN(C(C1OCCC1C(C)C)=O)CC)C N1(C(CCC(N)=O)=O)CC(CNC(c2nscc2Br)=O)C2(CC2)C1 c1(C(=O)NC2(CNC(=O)CCC(=O)c3cccnc3)CC2)ccn2cncc2c1 Cc1ccc2c(c1)CN(C(c1cccc(NCc3cccc(O)c3F)c1)=O)CC2 c1(C(=O)NCC2(F)CN(C(CC(=O)OCC)=O)C2)ccn2cncc2c1 C1(NC(CC=C(C)C)=O)CN(C(=O)CCc2cnc[nH]2)CCC1C(F)(F)F Cc1cc(C(=O)NC(CNC(C2CC(=C3CC3)C2)=O)C2CCC2)c(F)cc1Cl CC1(C)C(NC(=O)C(C2CCCCCC2)F)C2CCCN(C(c3ccsn3)=O)C12 CN1CC2C(C(=O)NCC=C3CCN(C(=O)CC4COC(=O)C4)CC3)C2C1 C1(CCC)CCC(C(N2CCCC2CCNC(C2CC2(F)F)=O)=O)CC1 C1(NC(CC(C)(C)C)=O)CN(C(=O)C(C2CCOCC2)O)CC1(C)C C1(NC(C2=CCC(C)CC2)=O)CC2(CCCCN2C(=O)CC2CC(=O)NC2=O)C1 c1(N2CCC(C)C(NC(c3c(CC)ccs3)=O)C2C)ncc2ncn(C)c2n1 N1(C(C2(C(C)C)N(C(CNC(CCC#C)=O)=O)CCC2)=O)CCC(C#CC)C1 CCCCC(CC)C(=O)NC(CNC(=O)C(C(C)C)c1cnc(C)s1)(CC)CC c1(C(=O)NCC(=O)NCC(=O)NCC2CCCC2)ccc2n[nH]cc2c1 CCCCC(C)C(=O)N1CCCC1(C(=O)NCc1n[nH]cc1CC)C(C)C CC(C)(C(=O)NCC1CC1CNC(=O)CCc1cncnc1O)S(C)(=O)=O CCC(C)C(=O)NCC(N1CCC(C(C)(C)NC(=O)C(C)(C)C2CCC2)C1)=O c1(CC)nc2sc(C)cn2c1C(=O)NC(C)CNC(=O)CC1(CS(C)(=O)=O)CC1 C1(CNCc2cc(F)cc(C(F)F)c2)COc2ccccc2C1 N1(C(CC(=C)C)=O)CCCCC1CCN(C)C(c1ccc(NC(C)C)cc1)=O CCC(CNC(=O)C(F)Cc1ccccc1)(CC)NC(=O)CN1CSCC1=O O=C(C1=COCC1)NC1CCC(NC(=O)CCSCc2ccccc2)CC1 S(=O)(=O)(c1ccc(Cl)cc1)NCC(=O)NCCC1(NC(C(C=C)O)=O)CCCC1 c1(-c2cncc(C(=O)Nc3ccc(C(C)=O)o3)n2)ccc2nc(C)ccc2c1 c1(C(=O)NCC2(C)CC(NC(=O)C=CCN3CCCC3)C2)c(Cl)nc2ccccn12 C(=O)(C1CCCn2ccnc21)NCC1CN(C(c2ccnc(C)c2C)=O)CC1C C=C(C)CC(C(=O)N1CCC(O)C1C(=O)N(C1COCC1O)C)OC N1(C(c2cn(C)nc2)=O)CCOCC1CCNC(c1cnc(C(=O)OC)cn1)=O c1(C(=O)OCC)cnc(C)[nH]c1=NCC1CCN1C(=O)CCCN1CCCCC1 C(=O)(CC(O)CC(C)(C)C)NC(CC(C)NC(C(=O)NCCOC)=O)C N1(C(CC(CC)O)=O)CCCN(C(c2cccc(F)c2OC)=O)CCC1 C(CCCC)(C(=O)NCCS(=O)(=O)NC)NC(CCC=C)=O C(=O)(CCN=C(NCc1cccc(OC)c1C)NC1CCS(=O)(=O)C1)NC c1(C(c2cc(C(C)=O)sc2)=O)ccccc1F.c12cn(nn1)CC(O)COCC2 N1(C(CC(=O)N(C)C)=O)CCCC2(CCC(NC(c3cnc(S)[nH]3)=O)C2)C1 C(CN=[N+]=[N-])(C(=O)N(C)CCn1ccnc1)NC(c1n[nH]c(C)c1C)=O C1(C(C)O)CC(NC(=O)CC2CC(NC(C3CC3C3CCCO3)=O)C2)C1 c1(CC(=O)N(C2CCCN(C(c3snnc3C)=O)C2)CC)ccc(F)cc1C C#CC1(C(=O)NCC(C)(C)C)CN(C(=O)COCC2CCN(CCCO)C2)C1 Cc1nc2c([nH]1)C(C(=O)N1CCN(C(=O)CC3CCC3)CC1CC1CC1)CCC2 C1(CNC(C2(C)COC2)=O)CC2(CC(NC(C3CC4(CCCC4)C3)=O)C2)C1 C1(CNC(c2cnc(C(C)C)[nH]2)=O)CCCCCN1C(C1CCCOC1)=O C(N=c1[nH]cnc(Cl)c1CO)C1CCC(CNC(C(C)OCC)=O)CC1 c1(C(=O)NCCCN(C)C(C2CNC(=O)N2)=O)cc2n(c1)CCSC2 C1(O)(CN(C(CNS(C)(=O)=O)=O)C2CC2)CCN(C(C2CCC(CO)CC2)=O)C1 c1(CCC)ccc(C(=O)NCC(O)CNC(=O)Cc2cc(C)on2)s1 N1(C(C2(C)CCN(C)C2)=O)CC2(C)CN(C(=O)CCc3ccn(C)c3)CC2(C)C1 Cc1csc(C(c2nnnn2C2CCOC2)NCCCC2CC2C)n1 c1(C(=O)OCC)cccc2c(C(N3CC4CCCN4CC3C(=O)O)=O)[nH]nc12 c1(NC(C(NOC)C)=O)ccccc1S(=O)(=O)C(F)F N1(C(CCOCCNC(C2(C(C)C)COC2)=O)=O)CC(C)C(C)C1C CON(C)CCCNC(C1CC(C)(NC(=O)CC2(O)CCOC2)C1)=O c1(OC)ccncc1CNC(C1(C(C)NC(C2CCC(=O)C2)=O)CC1)=O c1(OCCOC)cnc(NC(c2nccn2C)C(C)C)nc1 c1(OC)cccc(CN2CC(CCCNC(c3cccc(OC)c3)=O)C2)c1 C1(NC(c2cc(CNC(=O)CCOC3COC3)no2)=O)CCOC12CCCC2 Cc1csc2ncnc(N3CC(NC(C45CC=CCN4CCC5)=O)CCC3C)c12 CC(CC(=O)Nc1ccc(NC(C2(C)COC2)=O)cn1)CC(C)(C)C C=CC1CN(C(=O)C(C)(C)CO)CC1NC(=O)C(c1ccc(F)cc1F)(C)C C1(C(=O)Nc2cn(CC(=O)NOCC3CCOC3)nn2)(COC)CCCC1 c1(CC#N)ccc(S(=O)(=O)NC(C2CC2F)=O)cc1 N12CCCCC1CNC(=O)C2=O.N1(C(C(C)C)C)CCOCC1 c1(C(=O)NC(C(=O)NC(CC)C2CC2)CC2CCCC2)cc(C)c(F)cn1 N1(C(CCC(=C)C)=O)Cc2ccnn2CC(NC(=O)C(C)OC2CCCCC2)C1 C(Cc1cnc[nH]1)(C(=O)NCc1c[nH]nc1C1CC1)NC(C=C(C)C)=O C(=O)(C(CC(F)F)C1CCC1)N1CC(NC(CCOC(C)C)=O)C(C)C1 CC1(C#CC(=O)NC(CO)C(N2CC3CC(N(C)C)C2C3)=O)COC1 Cc1cc(C(=O)NC(CNC(c2cc3[nH]ccc3s2)=O)C(C)(C)C)cc(C)c1F C1(CCC=C)(CNC(c2ccc(CCN)s2)=O)CCCC1 c1(C(=O)NC(CC)CNC(=O)C(c2ccc(Cl)cc2)CO)ccc2nc[nH]c2n1 S(=O)(=O)(c1cc(F)ccc1C)N(CC(=O)NC1C(OC)CN(C(C)=O)CC1)CCO C(=O)(C(O)CCNC(=O)C(C)(C)C1CC1)N(CCCC)CCOC CON=CC(=O)NC(c1cnn(C)c1)C(=O)NCCn1cnnn1 c1(C(=O)NC(CNC(c2ccc(C)s2)=O)(C)CO)ccc(OCF)nn1 C1(CNC(C)=O)CC2CCC(C1)N2N1CCC(OCc2ccccc2)C1 c1(C(C)C)ccc(C(N2CCCCC(NC(=O)C=Cc3ncco3)C2)=O)c(F)c1 N1(C(C2(CC)CC2(F)F)=O)CC2CC(Nc3cncc(Cl)n3)CC1C2 S(=O)(=O)(c1ccc(I)cc1)N1C(C(N2CCN(C)C(=O)CC2)=O)CCCC1 c1(C(=O)NC(c2ccccc2)CNC(COC(CC)CC)=O)csc(O)n1 c1(CSC)noc(CCC(=O)NCCCCCNC(=O)Cc2cnns2)n1 c1(C(=O)NCCCCCNC(C2CCC(N(C)C)C2)=O)cccc2c1CCOC2 CC(CC(F)(F)F)C(=O)NC1CCCN(C(c2nccc(C(F)F)n2)=O)C1 c1(C(N(C2CCC(NC(c3cc(F)n[nH]3)=O)C2)C)=O)c2c(nn1C)CCSC2 Cc1nc2cnn(C)c2cc1C(=O)NCC1COCCN1C(c1c[nH]c(=N)s1)=O C(=O)(C1=Cc2ccccc2C1)N1CCCC(C(N2Cc3c(nc(C)s3)CC2)=O)C1 C12(C(=O)NC3CC(CNC(C(C)SC(F)(F)F)=O)OCC3)CCC(CC1)C(C)O2 CC(C)CC(O)C(=O)NCCCCNC(=O)CC(C(F)F)N1CCOCC1 N1(C(C(CCCOC)NC(c2cc[nH]n2)=O)=O)CCOCC2(CCC2)C1 c1(CC)cc(C)[nH]c(=NCC2CN(C(C3(c4ccccc4)CCCC3)=O)CCO2)n1 N1(C(CC2(C=C)CC2)=O)CCN(C(=O)C(C)NC(C)=O)CC1c1ccnn1C C(=O)(CCC(C)C)NC(c1ccccc1)CNC(c1c(CC)[nH]cc1)=O C(c1ccc2c(c1)OCO2)=CC(=O)NC(C)CNC(C1CS(=O)(=O)CC12CC2)=O C(C(F)(F)CC(=O)O)NCc1c(OCC)cccc1.c1(CC)cc(CC)nc(CC)n1 N#Cc1ccc(CNCC23C=CC(=CC2CC)N3)cc1.C(=O)(C1=NOCC1)NC Cc1ccc(F)c(-n2cc(CNC3CC34CC(O)C4)nn2)c1 c1(CC)nn(C)c(Cl)c1C(=O)NC(C)CC1CN(C(=O)C=CI)C1 C1(C(=O)NCC2CC(C(N3C(CSC)CCC3)=O)C2)CC(F)CN1C C(=O)(C1=CC(O)CCC1)NCC1(F)CCC(CNC(=O)CCc2cccnc2)C1 c1(CC)nc(C(=O)N(C(C)CN(C(=O)CCC2CCOC2)C)C)c2ccccn12 CC1CCN(C(=O)CN(C2CCCC2)C)CCN1C(=O)Cn1cccn1 C(=O)(C(C)N(OC)C(=O)CCCNC(=O)CCCC(=O)NC)OC c1(C(C)=O)ccc(C(=O)NC(C)CNC(C2CC2C)=O)[nH]1 CC1(C(=O)NCC(O)C(=O)NO)Oc2ccccc2NC1=O C1(C(=O)NCC2(C(N)=O)CN(C(CCOC(C)=O)=O)C2)CCCOCC1 N1(C(C(C2CN(C(=O)Cc3ncccc3F)C2)OC)=O)CCCCC(CO)C1 C(c1c(Cl)cccc1Cl)=CC(=O)NCCN(C(CSCCC#N)=O)C1CC1 C(=O)(CC(F)(F)C(C)C)N1CCC(C(C)(C)NC(c2nc(C)n(C)c2C)=O)CC1 CS(C)(=O)=NCC(=O)N1CCCC1CNC(c1ccnn1C1CCCCC1)=O N1(C(C23N(CC(=C)C2)C(=O)CC3)=O)CCN(C(=O)CCSC)C2CCCC2(C)C1 c12cnc(C(F)(F)F)cc1OC2=O.CNC(CC=C)C Cc1ccncc1CC(=O)NC1CC(CNC(=O)CCCN(C)C)C1 N1(C(c2n(C)c(O)nc2)=O)CCCC12CCN(C(=O)Cc1ccsc1)C2 C1(C(=O)NC2(C)CCCN(C(=O)CCc3nc(=N)[nH][nH]3)C2)CCn2cncc2C1 c1(C(=O)OCC(F)F)sc(C(C)NC(=O)CCO)nc1C.N(CC)CC1CC1.CC C1(NC(=O)CCC2CCN(C(c3ccnn3C3CC3)=O)C2)C2CCCOC12 C1(COC)(CNC(C)(CCOC)c2nnnn2C2CCCCC2)CCCCO1 C(CCS(C)=O)(C(=O)NC(CNC(c1ccnnc1)=O)CC(F)(F)F)N(C)C CC(C)(CCCCNC(=O)C#CC1CCC1)NC(c1coc(CO)c1)=O Cc1cc(N)c(C)nc1C(N1CCC(NC(C2CCN(C)C(=O)C2)=O)C(O)C1)=O C#CC1(C)CCCN(C(C2(CC)CCCN2C(=O)C(C)OCCN(C)C)=O)C1 C1(NC(Cc2scc(C)c2)=O)CC2CCC(C1F)N2C(=O)CCCN1CCCC1 C1(CN)CCCC(c2cn(CC(=O)NCc3ccc(=O)oc3)nn2)C1 Cc1cc(Br)cc2cc(C(=O)Nc3cc(Br)cc(Br)c3O)oc12 N1(C(CCCCC(C)=O)=O)CCCC2NC(=O)CC12 Cc1conc1C(=O)NCCOCCCNC(=O)C(c1ccnn1C)C c1(C(=O)NC2C(NC(C(COC)N(C)C)=O)CCCC2)cc(Cl)cc(F)c1N c1(COC)cc(C(=O)NCCCOCCN(C(=O)Cc2ncoc2C)C)sc1C N1(C(C2=CCCCC2C)=O)CC(C)N(C(=O)C(F)CC(C)(C)C)CC1C N1(C(C2C(CC)C2)=O)CCC2(CCN(C(=O)CN3CCC(F)C3)C2)C1 c1(OCC=C)ccc(C(=O)NCC2CC(NC(C3C=CCC3)=O)C2)cc1 C1(C(=O)NCCCNC(CC2(C=C)CC2)=O)CC12CCCc1ccccc12 c1(OC)cccc2c1OCC(C(=O)N1CC(NC(=O)C(C(C)C)N(C)C)C1)=C2 Cc1c(C(=O)NC2CCC2NC(c2ccsc2)=O)cnc2c(Cl)cccc12 CC(C)C(CN(C)C)C(=O)N1CCN(C(c2cnn(C(C)C)c2)=O)CC1C(C)C C1(C(=O)NCCCN(C)C(C23CCCC(C2)C(=O)N3)=O)CCC2(CC1)OCCO2 Cc1nn(CC(N2CCCC(O)(CNC(C3CC3C)=O)CC2)=O)c(C)c1C=NO CCC(C(=O)N(CCCNC(=O)Cc1nncn1C)C)N(C)C Cc1cccn2cc(C(=O)NC34CC3CN(C(=O)CCN(C)C)C4)nc12 C1(N=[N+]=[N-])(C(N2CC(C#C)C2)=O)CCN(C(c2cc(C)n(C)c2)=O)C1 C(=O)(C1CCCc2scnc21)NC(CNC(c1cnc(C)s1)=O)CC(C)C c1(C(N(C(c2ccco2)CNC(c2cccs2)=O)C)=O)cc(CC2CC2)on1 Cc1sc2cc(F)ccc2c1CCNC(c1cccc2cncn12)=O C(=O)(C(C)(C)CCCNC(c1cc2cccn2cn1)=O)N1C(COC)C=CC1 C(=O)(C(C(C)(C)C)NC(C1CC(C)(C)CN1C)=O)N(CC1=CCCOC1)C c1(C(=O)NC(C(C)C)C(C)NC(=O)CN2CCCCC2)ccc2nccnc2n1 CCCC(CCC)C(=O)N(C)CC1COCCN1C(c1csc(C(F)F)c1)=O c1(OC(CC)CNC(=NC)NC(C)CC)ccc(F)cc1F C1(SCCN2C(=O)OCC2)CCCCN(C(=O)C2=COCC2)C1=O CC1CN2CCN1C2=O.N1(C(=O)OC2CC2)CCN(C)CC1c1ccccc1 Cc1nc(N2CC(NC(c3cccc(F)n3)=O)C(C)C2)c2cc(Br)ccc2n1 c1(C(N(CC(C)NC(CN2CC(CC)C2)=O)CC)=O)cc(C)c(Cl)cc1C C(=O)(C1=CC2CC=CCC12)NC1(CC=C)CN(C(C2CCS(=O)(=O)CC2)=O)C1 c1(CC)cc(C(=O)NC2(C(=O)NCC3(F)CCOC3)CCCCC2)ncn1 Cc1oc(S(N)(=O)=O)cc1C(N1CCC(C(C)NC(=O)CCNC(=O)CO)C1)=O C1(C(N2C(C)(C(=O)NC3C=CC(C(=O)OC)C3)CCC2)=O)CCOCC1(C)C Cc1nc(C)n(CCCC(N2CC(NC(=O)Cc3c(C)noc3Cl)CC2C)=O)n1 N1(C(c2cccc(SC)c2)=O)CCC(CNC(=O)C(C2CC2)N(C)C)CC1C C12(CNC(CCNC(CCCCC)=O)=O)CC(C)(CCO1)C2 C1(NC(CC2C(C)CCO2)=O)CCCC2CN(c3cc(Cl)nc(C4CC4)n3)CC12 C1(C(=O)NC2CC(CNC(CC(C)CN(C)C)=O)C2)CCc2cnn(C)c2C1 N1(C(CCC2(C)CN(C(c3ccc(C)nc3)=O)C2)=O)CCC2(CCC2)C(O)C1 c1(NC(C2C(NC(CC(=C)C)=O)C2)=O)cncnc1C1CC1 C(N=c1[nH]c(C(F)F)nc(=N)[nH]1)C1CCC(NC(Cn2ncc(C(N)=O)c2)=O)C1 c1(C(N2C(COC)COCC2)=O)cnc2n[nH]c(-c3ccc(F)c(F)c3)c2c1 c1(C(N(CC(=O)OC)CCOC)=O)cccc(OC(C)C)c1Cl N#Cc1cc(S(=O)(=O)N2CCC3CC3C2)ccc1NCc1csc(C(F)F)n1 c1(C(=O)NCCCOC)ccc(NC(c2cncn2C)=O)nc1 N1(C(CC)C(=O)NCC(CC)NC(C2(C(C)C)COC2)=O)CCc2ccccc21 N1(C(c2cc(C)c(N)cc2Cl)=O)CC2CCC(C1)N(C(=O)CC1(C(F)F)CC1)C2 N1(C(c2nc(OC)nc(O)c2)=O)CC2CC1CN(C(C1CCOC(C)C1)=O)C2 C1(C(=O)NCCCN(C(C(CC#C)C)=O)C(C)C)CCC2(CC1)CC(O)C2 c1(CNC(C2(C)CCN(C)C2)=O)cc2n(n1)CCN(C(=O)CC1CCCOC1)C2 N1(C(c2nc(C)nn2C)=O)CCC2CN(C(c3cnn(C4CC4)c3)=O)CCC2C1 CC(=O)C(C)CC(C)C(=O)NC(C(=O)NCC(O)C(C)(C)O)C1CC1 c1(C(N(CC(CNC(C(CC)C2CCC2)=O)C)C)=O)cccc(C(F)F)c1OC N1(C(c2c(C(C)=O)ccs2)=O)CCN(C(c2noc(C3CC3)c2C)=O)C(CO)C1 CCC(C)CC(C(=O)N(CCCOC)C)NC(c1nnccc1C)=O C1(NC(c2nc(N(C)C)oc2)=O)CS(=O)(=O)C12CCN(C(C1CC13CC3)=O)CC2 N1(C(=O)C2=CC3C=CC2C3)CCC2C(CCCN2C(=O)Cc2csc(Cl)c2)C1 n1(C(C=C)C)nc(C2CC2)nc1CN1CC(C)CO1 C1(O)(CNC(c2[nH]c(=NC)sc2)=O)CCN(C(c2ccc(C(N)=O)[nH]2)=O)CC1 C1(CC)COC(C)(C)CN1C(C1(CNC(=O)C(O)CC(N)=O)CC(C)(C)C1)=O C12(CNC(CCOCCC)=O)CC(CO1)N(C(=O)Cc1nnc(S)n1C)C2 C#CC1(O)CC(C(=O)N(CC(C)CNC(=O)CCn2ncn(C)c2=O)C)C1 c1(CC)cc(NC(=O)C(Cn2cncn2)NC(=O)C(F)F)ccc1F c1(CC)c[nH]cc1C(=O)NC1CCN(CC)C1.c12cn(nn1)C21CC1 N1(C(c2c(SC)snn2)=O)CCN(C(=O)Cc2ccoc2C)C2CCCCC2C1 N1(C(c2ccccc2C=O)=O)CCC(NC(=O)Cc2cccc(O)c2)CC1C c1(OC)c(F)ccc(Br)c1C(=O)NCC(C)(C)CC(F)(F)F C1(NC(C(C)=C2CC2)=O)CCN(C(=O)C(C#N)Cc2ccc(C#N)cc2)CC1F C(C)(CCCCNC(=O)CCN1CCCC1=O)NC(C(C)Cc1ccccc1)=O CCCC(C(=O)N1CCCC1CNC(c1cnn(C(F)(F)F)c1)=O)S(N)(=O)=O C(C1=CCN(C(C2CCOC2)=O)CC1)NC(C(CCN(C)C)O)=O C1(CC(=O)NCC2CSC2)CCN(C(C2CCCOC2)=O)CC1 N#CC1CCCCC1N=c1[nH]c(=NCCN2CCCOCC2)[nH]c2cc[nH]c12 C(=O)(CCC(C)(F)F)NC(C1CCCN1C(c1ccc(=O)oc1)=O)C C1(CC=C)(C(=O)NC2CCCC2NC(C2(CC(C)C)CCCC2)=O)CCOC1 N1(C(=O)OCC)CCC(NC(=O)COC(c2ncccc2Cl)=O)CC1.NCC N1(C(C2CC3CC2(C(=O)O)C3)=O)CCC(O)C(O)C1 N1(C(CCCN(C)C)=O)CC2CC(N=c3ccc4ncc[nH]c-4n3)C2C1 CCCC(CCC)CC(=O)NCC1(CNC(=O)C(O)C(C)C)CCCC1 CC(CNC(=O)NCC(Cc1cccc(F)c1)C(=O)O)CC(F)F C1(C(=O)NCCCN(C(C(F)=CC)=O)CCO)C(c2ccncc2)C1(C)C c1(C(N2CC(NC(=O)CC(C3CC3)C3CC3)C(O)C2)=O)cc(C(F)F)cc(F)c1 C1(C(=O)NCCCNC(C2(C)CS(=O)(=O)C2)=O)COc2cc(F)ccc2O1 C1(F)(CNC(c2ccc(Br)o2)=O)CC(NC(C2CC(CCF)C2)=O)C1 N1(C(CCOCC(C)(C)C)=O)CC(O)CC1(C)C(=O)NC1CC(O)C(O)C1 c1(CC(=O)NC2CCN(C(c3cncc(C)c3)=O)C2)ccc2sccc2c1 CC1(NC(C2CCCCC2)=O)CCN(CC=Cc2ccccc2)CC1 CC1(O)CCCN(C(C2CC(=O)NC3CNCC23)=O)CC1.c12cccc(c1)CO2 N1(C(c2nc(C(F)(F)F)nn2C)C(=O)NCCOC)CCOCC12CCSC2 CC1CN(C(C2CCC(NC(C3CC34CC4)=O)C2)=O)CCC1(F)F C1(C(N2C(C)CN(C(c3nc(C(F)(F)F)cs3)=O)CC2)=O)CC2CC1CC2(F)F C1(C(=O)NCC(c2cnn(C)c2)C)CC2CN(C(=O)CCCNC(N)=O)CC2C1 CCC(F)(F)CC(=O)NCC(C1CCCCN1C(=O)C(O)Cc1cnc[nH]1)(C)C O=S(=O)(Oc1cnc(Br)c(F)c1)c1cccc2ncccc12 c1(SC)ccc(C(=O)NC(C)C(C)NC(c2sc(-c3ncc[nH]3)nc2C)=O)cc1 C12(C(=O)NC3C(C)(C)OCC3)CC(CO1)N(C(=O)CC1CCCC(=O)C1)C2 C(=O)(C(CCOCCOC)NC(=O)NCCO)NCc1ccc(C#N)o1 Cc1nn(C)cc1C(O)C(=O)NCCCN(CCO)C(c1ccc(Cl)s1)=O N1(C(Cn2c(C)nnn2)=O)CC(C)N(C(=O)CCCS(N)(=O)=O)CC1C C=CCC(CC(C)C)C(=O)NCC=CCC(N1CCOCC(C)(C)C1)=O Cn1cc2c(n1)CC(C(=O)NC(CNC(=O)C1=CC(C)(C)C1)CO)CC2 C1(C)(CC)CCN1C(=O)CC1(NC(=O)CC(C)C2CC2)CC1 C1(NC(C2CC2c2ccccc2)=O)CCN(C(=O)Cc2ncc(Cl)s2)CC1F c1(C(=O)NC2CC(CNC(C=CC)=O)C(O)C2)cccc2c1OC(F)(F)O2 C1(C(C)NCC2(C(=O)OCC)CCCOC2)CC2(C1)CC2(F)F c1(NC(C2CCN(C(c3cnc(O)cc3O)=O)C2)=O)ccc(Cl)nc1Br Cc1cc(C=CC(=O)NCC2CCN(C(=O)CCc3scnc3C)C2)on1 c1(NC(C2CC(=C)CN2C(c2cc(Cl)ccn2)=O)=O)cccc2nsnc12 C(c1csc2ccccc12)=CC(=O)NCC(CC(C)C)NC(C(C=C)(C)C)=O N1(C(c2cc(CC)on2)=O)CCN(C(=O)CCc2cc(C)cc(C)c2)CC(O)C1 c1(C(=O)OC)cc(S(=O)(=O)Nc2ccc(OC(F)F)c(C#N)c2)cn1C C1(C(C)(O)CNC(C2(n3nccn3)CC2)=O)CCN(C(=O)Cn2cncn2)CC1 c1(CNC(c2csc(-c3ncc[nH]3)n2)=O)cc(OC2CCOCC2)ccn1.O Clc1ccc(Br)c2c1CN(C(c1ccccc1)Cc1ccccc1)CC2 C#Cc1ccc(CC(N2CC(NC(C3(C=C)CCCC3)=O)CC(F)C2)=O)cc1 N1(C(CC=CCC)=O)CCOCC(F)(CNC(C2C(C)C2C)=O)C1 N1(C(c2[nH]cc(CC)c2)=O)CC(OC)CC(NC(=O)C(C)CSC)C1 CC1=C(C(=O)NCC(C)NC(c2cccc(-n3cnnn3)c2)=O)C(C)(C)CCC1 C1(NC(Cc2ccc(C)s2)=O)CCCN(C(=O)Cn2cc(C#N)cn2)CC1 C1(C(N2CCC(n3ccnn3)C2)=O)C(O)CCN1C(=O)CN1CCCC1 C1(C(=O)NCC2(NC(C3CC(CF)C3)=O)CCOC2)CCS(=O)(=O)C1 c1(CC)c(C)sc(NC(=O)C(=O)N(C)CC2COCCO2)c1C(N)=O N1(C(CC2C(CC)C2)=O)CCC(C(C)(C)C)(CNC(c2ncsc2NC)=O)C1 C1(C(C)C)CC(O)CN1C(c1c[nH]nc1CNC(C1COCOC1)=O)=O C#Cc1ccc(C(=O)NC2CCC(C)N(C(=O)C=C3CCOCC3)C2)c(F)c1 C1(OC)CC2(C(=O)N(CCCN(C(=O)CCC3CCOCC3)C)C)CC12 CC1CN(C(=O)C(C)(Cl)Cl)CC1NC(c1ccc(CN(C)C)s1)=O N1(C(c2cnc(C(C)C)[nH]2)=O)CCC(C)C1CNC(c1ccccn1)=O Cc1ncc2c(n1)CCC(C(=O)NC1CN(C(c3nc(C)n(C)n3)=O)CC1C)C2 c1(C(=O)NCC2C(NC(C3(F)C(C)OCC3)=O)CCC2)ccc2[nH]c(=N)[nH]c2c1 c1(CC)c(C(N2CCC(C)(CNC(C3(O)CC3(C)C)=O)C2)=O)cnn1CC(C)C C1(C(=O)NC2CC(CNC(Cn3nc(C)oc3=O)=O)C2)COC2(CO)CC1C2 C(C)(C(O)C(=O)NCCCCCNC(=O)Cn1nc(-c2cccs2)oc1=O)SC c1(NC(C2CC2C(F)(F)F)=O)cnncc1O.c12ccc(cc1)-c1cn(nn1)C2 C1(C(=O)NCCCC2(C)N=N2)(CNC(C(C)OCCCC)=O)CCCO1 n1(CC)ccc(C(=O)NC(C)(CNC(=O)CC2CCC(C)(C)O2)C2CC2)cc1=O C#CC1(C(=O)N(C2CC(C)(C)C2)C)CCN(C(=O)C(N)=O)CC1 Cc1cc(Cl)c([N+](=O)[O-])cc1C(=O)OC(c1ccc2ccccc2c1)C C#Cc1cccc(C(N2CC(NC(=O)CC3CC34CC4)C3(CCC3)C2)=O)c1F C1(O)(C(C(=O)N(C2CCOCC2)CC#C)F)CN(C(=O)CC2CC(=O)C2)C1 CCCCCCCCC(=O)NCC(C)CC(=O)N(C1CCCC1C#N)C c1(C(N2C3CCC(NC(C4C(=C)C4)=O)(CC3)C2)=O)ccc2ccn(C(C)C)c2c1 c1(-c2n(CCC#C)c(N(C)Cc3cnc(C)s3)nn2)cnc2n1CCC2 CC1(C)CCC2(CC1)CC2C(=O)NC1CN(C(=O)CN2CCC(O)CC2)CC1O C(=O)(C1Cc2ccccc21)N1C(C(N2CC(NC(N)=O)C2)=O)CC(C)(C)C1 S(=O)(=O)(c1cc(C)ccc1C)NC1CCCN(C(c2cc(C)[nH]c2)=O)C1 C1(NC(CCOCCNC(C2OCC(C)C2)=O)=O)CC2CC3C(C2)C13 C1(C(C)NC(C2(OCC)CCC2)=O)CCN(C(=O)Cc2cc[nH]c2)CC1 C1(CC)(NC(=O)CC2CC=CCC2)CCN(C(c2cc(C)cnc2N)=O)CC1 N1(C(COCC(C)C)=O)CC2CC(NC(=O)CC3(C)CCOC3)CC2C1 Cc1cc(CC(=O)NCCC2CN(C(=O)CSCCN(C)C)C2)n(C)n1 C12(NC(C(CC)COC)=O)CCCC1(F)CN(C(c1cnc(OC)c(C)c1)=O)C2 c1(C(=O)NC(CCN(C(CC(C=C)(C)C)=O)C)C)n[nH]c(CC)c1[N+](=O)[O-] N1(C(CC=C=C)=O)CCC(C(C)CNC(c2ccccc2)=O)CC1 C1(C(=O)OCC)(C(=O)N(C)CCNC(c2cc(C(C)C)[nH]n2)=O)CCN(C)CC1 c1(C(=O)NCC2(F)CC(NC(C3CC(C)C3)=O)C2)sc2cccnc2c1Cl C(C1=NOC2CN(C(=O)Cc3cccnc3Cl)CC12)NC(C(C#C)(C)C)=O C1(C(=O)NCC2(NC(c3cnc(C4CC4)s3)=O)CCCCC2)CCC2(CCC2)O1 Cc1cc(C(=O)NCC(c2ccccc2)CN)n2ncc(C#N)c2n1 Cc1nccn1C(C)C(=O)NCc1nc(CNC(=O)C(C)O)cs1 N1(C2(C(=O)NCCNC(C3CC(O)C3)=O)CC2)CCOCC1 N1(C(CN(C(C)C)C(c2ccc(CO)o2)=O)=O)CCCCCC1C c1(C(N2CCC(C(F)F)(OC)C2)C(=O)NC2CCOC2)nn(C)c2c1COCC2 C1(C(N(C2CCCN(C(c3cc(C(C)C)oc3C)=O)C2)CC)=O)CCCN1C=O c1(CC(=O)NC(CC#C)C(=O)NCc2cnn(C(C)C)c2)ccc(C#N)cc1 N1(C(C2C(C(=O)OC)C2)=O)CCN(C(=O)C2=CC3CCCC23)CC(C)(F)C1 c1(CCC(=O)NCC2C(NC(CC(CC)O)=O)COC2)cccc([N+](=O)[O-])c1 C=C1CC2CCC(C1)N2C(=O)C(C)C(C)NC(c1ccc2occc2c1)=O Cc1nc2c(CCC(=O)NCC(C)NC(C3(CO)CCOCC3)=O)cccc2o1 C(C(=O)N(C)Cc1sccc1C)(C(C)(C)C)NC(C1C(CC)C1)=O N1(C(CN(C2CCC2)C)=O)CC(C2(NC(C3CCN(C)S3(=O)=O)=O)CC2)C1 c1(C(N(CCNC(=O)C(C)Sc2ccccc2)CC)=O)cc(OC)c(F)c(F)c1 CC(CNC(=O)CC=CCNC(=O)CN1CCCCC1=O)C(C)(C)C c1(C(N(CCN(C(C2(C)COCCO2)=O)CC)CC)=O)cnc(O)c(C)c1 C1(C(N2CCCN(CCNC(c3c[nH]c(=N)s3)=O)CC2)=O)CCC2CCCCN12 N1(C(C2CC(OCC)C2)=O)CC(C2CCCCN(C(=O)CCCNC(C)=O)C2)C1 C1(NC(CCSC)=O)CN(C(c2ccsc2Br)=O)C2(CCOCC2)C1 c1(C(N2CC(O)(C(C)NC(=O)CSc3nc[nH]n3)C2)=O)c(F)ccc(F)c1N C1(CC(=O)N(CC(CNC(C(C)OC)=O)C)C)CCCC(F)(F)C1 C1(NC(C(c2cn(C)nc2)O)=O)CCOCC1NC(C1(C(C)(C)O)CC1)=O c1(C(=O)NCC23OCCC(NC(C(CCCC)O)=O)(C2)C3)cc(OC)cc(Cl)c1F c1(OC)cc(F)c(CNCCC2CC(C(=O)O)C2)cc1Br C1(CNC(C(C=C)c2ccccc2)=O)CC2CCC1N2C(c1[nH]nnc1C)=O C1(C(=O)NCC2=CCN(C(C(C(=O)OC)C)=O)CC2)CCC2(CC1)CC(OC)C2 N1(C(C=CCC2(NC(=O)CCCCC3CC3)CCC2)=O)CC2C3CCC(C3)C12 C(C(F)C(=O)N1CC(n2cc(CN(C(=O)CC(C3CC3)SC)CC)nn2)C1)SC c1(C(=O)NCCCCCCNC(C2(CC)CCNC2=O)=O)ccc2nsnc2c1 N1(C(Cc2cccc(OC)n2)=O)CCCC2CCN(C(c3cnoc3C)=O)CC12 N1(C(C2CN(C(Cn3c(C)cc(C)n3)=O)C(C)(C)CC2)=O)CCCC(C2CC2)CC1 C1(C(=O)NCCC(C)(C)F)C(C2CC2)CCN1C(=O)C(F)C1CCCC1 C12(OC)CCCC1CN(c1nc(-c3ccc(OC(C)=O)cc3)no1)C2 c1(OC)ncnc(C(N2CCN(C)CC2CNC(=O)CN2CC=CC2)=O)c1F O=C1CCC(C(N2CC(CCCCNC(c3snnc3C3CCC3)=O)C2)=O)C1 c1(CC(=O)NCC(CO)NC(C2(C)CCCCCC2)=O)ccc(C#N)cc1F c1(CNC(C=C(C)C(F)F)=O)ccc(CN(C)C(c2cncnc2O)=O)cc1 C1(N(C(=O)C(F)CC2CC2)C)CCCN(C(=O)CCc2ncco2)C1 c1(C(N2CCCCC2C(N2CC(F)C(F)C2)=O)=O)ccc(CO)cn1 N1(C(C2ON=C(C)C2)=O)CCCC(NC(C2CC3(C2)CC3F)=O)C1 c1(CCCC)nc(C(=O)NCCC2CC(NC(C3CCS3(=O)=O)=O)C2)cs1 N1(C(COc2c(C#N)cccc2)=O)CCN(C(C2CCCCS2)=O)C2COCC12 C1(CN(C(C2CC(F)C2)=O)C2CC2)CCCN1C(C1CCCO1)=O C12(NC(COC(C)C)=O)CC1CN(C(=O)C(C)NC(=O)Cn1cnnn1)C2 c1(C(N2CC(OC)(CNC(=O)CCC(C)SC)C2)=O)csc2c1CCCC2 c1(C(N2CCN(C(C3CCOC3)=O)CC2C(F)F)=O)[nH]c2ccc(F)cc2c1Cl C(CCCCC1CC1)(c1n(CCCSC)nnn1)Nc1cnn(C2CC2)c1 C1(NC(C2CN(C(N)=O)C2)=O)Cc2ccccc2N(C(=O)CCC2(O)CCC2)C1 C1(CNC(c2cnco2)=O)CCN(C(C2CC2c2ccccc2)=O)CC1O N(C1CC2(CCN(C(=O)CCF)C2)Oc2ccccc21)C(C(=O)NC(C)C)=O Cc1cc(C(=O)NCCOc2ccc([N+](=O)[O-])cc2)c(N)c(C)c1 C1(NC(c2nc(C)nn2C)=O)COC2(CCN(C(c3cccn3C)=O)C2)C1 CC1c2nccn2CCN1C(c1cccc(-c2ccc(S)cc2)c1)=O N1(C(=O)NC2(C(C)(C)C)CC2)CCC2CC(c3ccc(F)cc3)C2C1 c1(C(=O)NC(CCC#C)C(=O)OCC)cc(C)nc2ccc(Cl)cc12 C1(CC)C(NC(c2ccc(=N)[nH]n2)=O)CCCN1C(=O)CC1CCCC1O c1(Cn2cc(C(N3CCC(C(=O)NC)C3)=O)nn2)ccc(Cl)cc1 Cc1nc(C(=O)NC(CNC(C2(CO)CC2(F)F)=O)C2CC2)c(C)o1 C(=O)(CCS(=O)(=O)C1CCCC1)N(C1CC(NC(=O)C(O)C2CC2)C1)C C#CCC(C)(C)CNC(=O)C(O)CCNC(C1(C)CNC(=O)N1)=O CC1CN(C(=O)CC#N)CCC1CNC(C1CC(=O)N(C(C)C2CC2)C1)=O C1(=CC(=O)NCCN(C(C2CC(F)(CF)C2)=O)Cc2ccccc2)CCCCC1 C1(CNC(=O)NCCNS(NC)(=O)=O)CCC2COCC2O1 N1(C(C(C)C(C)(F)F)=O)CCN(C(c2ncn(C)n2)=O)C2CCCC12 CC(C)C(CNC(c1n[nH]c(O)n1)=O)NC(C1(F)CCCC1)=O N1(CC(N2CC3CC2C3CNC(=O)Cn2cc(CO)nn2)=O)CCS(=O)CC1 C1(NC(C2(C)CCN(C(C)=O)C2)=O)CC2CCC(C1)N2CCCC1CCC1 C(=O)(C(F)CC(C)(C)C)NCC(CCCC)NC(c1ccc(C)cn1)=O C(=O)(CCCC(=O)NOC(C)(C)C)NCC1CC(NC(C=CSC)=O)C1 c1(C(=O)NCC2C3N(C(C=C(C)Cl)=O)C(CC3)C2)c(F)ccc(O)c1F Cc1onc(-c2ccncc2)c1C(N1CCC1CNC(=O)C(O)CC1CC1)=O c1(N2CC(C)S(=O)CC2)nc2ccc(S(=O)(=O)NCCSCCO)cc2s1 c1(C(=O)NC2CN(C(CCCCSC)=O)CC3C2C3)cncc2ccccc12 c1(-n2ncc(C(=O)NCC(CNC(C3C(CC(C)C)C3)=O)O)c2)ccccc1F C(=O)(CC(C)(O)C(F)(F)F)N1CCC(NC(C(COCC)(C)C)=O)C(O)C1 N1(C(C2C(c3c(C)cc(F)cc3)C2)=O)CC2CCC1CN2C(=O)C1=CCCOC1 Cc1nc(NCc2cnc(C(C)C)s2)cc(=NCC2CC3CCCCC3O2)[nH]1 C(CS(=O)(=O)CC(=O)NCC1COCC1NC(C1CCC(=C(F)F)CC1)=O)OC C1(C(N2C(C)CN(C(c3ccsc3)=O)CC2)=O)CC12C1CC3CC(C1)CC2C3 C(=O)(CCCCCF)N(CCCCN(C)C)CCNC(C(CC)NC(C)=O)=O c1(C(N2CC(C)C(NC(c3cnc(S)[nH]3)=O)C2)=O)ccc2nc(O)nc(O)c2c1 C1(NC(c2n(COC)ncc2)=O)CC(NC(=O)CN2CCC(C)C2)CC1O c1(C(=O)OC)ccc(Br)cc1NC(c1cc(-c2ccc(Cl)nc2)cs1)=O Cc1cc([N+](=O)[O-])cc(Br)c1NC(C1CC1C(=O)NC1CCS(=O)(=O)C1)=O CC1CCc2[nH]nc(C(=O)NCC34CCCC3CN(C(=O)CSC3CC3)C4)c2C1 C1(NC(c2cc(=O)cc[nH]2)=O)CN(c2nc(Cl)ncc2Br)CC2(CCC2)C1 CCC(CC)C(C)C(=O)N(c1cc(C(F)(F)F)ncn1)C1CCNCC1F C1(CC)(CC)CC(NC(=O)C(C)c2ccsc2)CN1C(c1cc(OCC)no1)=O CC1Cc2ccc(F)c(Br)c2CN1C(C1CN(CC(F)(F)F)C1)=O CC1=C(C(=O)N2CCC(CO)C(NC(=O)C(C)(C)N(C)C)CC2)C(C)(C)CCC1 C(CC(C)C)(C(=O)N1CC2CC2(CNC(=O)C(C)(C)N(C)C)C1)NC(=O)OC N1(C(C=CCCC)=O)CCC2(CCCN(C(=O)Cc3cc(OC)ncn3)C2)CC1 c1(C(CC)=O)ccccc1C(=O)NCCN(C(=O)C(c1c(C)noc1C)C)C N1(C(=O)CCc2ncccn2)CC2CCN(C(c3ccc4c(c3)CC4)=O)C2C1 C1(C)(C(=O)NCCn2ncc(C(N(CCCOC(C)C)C)=O)c2)CCCCC1 CC1(C)Cc2cc(C(=O)NC3C4CC3N(C(C3CC(C(F)(F)F)C3)=O)C4)sc2C1 C1(C(N2C(CNC(c3cnn(C)c3N)=O)CCC2)=O)CCc2nnc(O)cc2C1 c1(OCC)cc(NC2CCC(CNC(c3ccnc(F)c3Cl)=O)CC2)ccc1O c1(C2(C(N(CC(C)(C)CNC(C3CC3Cl)=O)C)=O)CCC2)ncccc1F C(=O)(CCCS(=O)(=O)N1CCCC1)NCC1N(C(C(CC)O)=O)CCC(C)C1 N1(C(COCCSC)=O)CC(=O)NC2CN(C(=O)CC3CC3C(F)(F)F)CCC12 CC(CCC(C)(C)C)C(=O)NC(CC(=O)N1CC(C)(F)C1)C(F)(F)F C1(C(=O)NC2CC(CCNC(c3cc[n+]([O-])cc3)=O)C2)C(F)(F)C12CC2 C1(NC(c2csnc2C2CC2)=O)CCCCN(C(C2C=CCCC2)=O)C1 Cc1cccc(F)c1CC(=O)NCC(CC(F)(F)F)NC(=O)C=CC(C)C C1(CNC(C(C)CCO)=O)CN(C(c2cn3cccnc3n2)=O)CCC1(C)C C(=O)(NN1CCc2ccccc21)c1c(Cl)ccc(CC(=O)OC)c1 C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC1(C)CCC(NC(C=CCCC)=O)CC1 c1(C(=O)NCc2ccc[nH]2)cccc(C(=O)NC(CNC)C)n1 Cc1noc(Cl)c1CCC(=O)NCC1(NC(=O)CCCCO)CCCCC1 C1(C)(CC)CC(N=c2nc(N3CC(C)(C)OC4(CCOC4)C3)c3c([nH]2)CSC3)C1 C1(CC=C)(NC(=O)C(C)N(C)C)CCN(C(c2c[nH]cc2CC)=O)C1 n1(C(C(C)C)C)nc(-c2ccc(Br)cc2)nc1CCc1ccc(F)cc1 N(C(=NCc1cc(Cl)n(C)n1)NC1CCCC(OC(F)F)C1)Cc1cnn(C)n1 Cn1c(C(=O)NCC2CCCN(Cc3ccc(O)c(Cl)c3)C2)cccc1=O CCC(CC)(C(=O)NCCN(C(=O)Cn1ccc(=O)cc1C)C)c1ccccc1 C1(C(=O)Nc2cccc(OC)n2)C2CCC(C2)N1Cc1ccccc1OC(F)F c1(C(=O)NCC(=O)NCCCCN(C(=O)C(F)C2CCC2)C)ccccc1 Cc1nc(CNC(c2ccc(O)nn2)=O)oc1C(=O)NCc1nc(C#N)cs1 C1(CNC(C(COC)NC(C)=O)=O)CCCCCN1C(=O)C(C)=C1CC1 C1(c2nnnn2CC2CC2)(NC(C2CCOC(CSC)C2)=O)COC2(CCCC2)C1 CCCCCCC(C(=O)NC(C)C)N(C)CCN1CCOCC1 CCC(CCC(=O)NC(C)COC)NCCCC1(C)CC1 C=CC(C)(CCOC)C(=O)NCC(CCOC)NC(c1nc(C)ccc1C)=O CC(C)CCC(=O)C(=O)NC1CCCCC1CNC(=O)Cc1nccs1 c1(C(N(C2CCN(C(c3ccoc3C3CC3)=O)CC2)C)=O)nc2ccccc2o1 c1(C(=O)NCc2ncoc2C2CN(C(C3CCC3(F)F)=O)C2)ccc(CO)cn1 N12CCC(O)(C1)C(Cl)OCC2=O.C(=O)(CCCc1cccs1)NC(C)(C)C c1(OC)cccc(Cl)c1CN1CC(C(O)CO)C1 n1(CC(=O)NCCC2CCCN2C(=O)CC2CCCC2O)cc2ccccc2n1 c1(CC)ncc(C(N2CC(CNC(C3CC3CC(C)C)=O)C(C)C2)=O)c(C)n1 N1(C(CCC=CC(C)C)=O)CCOC(C(C)NC(=O)COC2CC2)C1 CCCCCCC(C)C(=O)N1CCC(N(CCO)Cc2cc(F)ccc2F)CC1 CCC(C)(O)C(=O)NC1CCC(CNC(c2cncc(N3CCCC3)n2)=O)C1 CC(C)(C)CCCC(=O)N1CC(C(C)(C)O)(CNC(=O)C(c2ccccc2)O)C1 c1(C2(C(N(C(C)CNC(c3nsnc3O)=O)C)=O)CCC2)cccc(F)c1 N1(C(CC(CC)(C)C)=O)CCCC2(CCCN2C(=O)C#CC2CCOC2)C1 N1(C(CN(C2CC2)CC)=O)CC(C(N2CC[Si](C)(C)C2)=O)C(C)C1 c1(NCC(C)CNC(c2cc(S(N)(=O)=O)c[nH]2)=O)nc(Cl)nc2c1ncn2C N1(C(CSc2c(C)n[nH]c2C)=O)CCOCC(NC(C2(C)CC2(F)Cl)=O)C1 c1(C(N2C(CNC(c3ccn(C)n3)=O)C=CC2)=O)cc([N+](=O)[O-])c(Cl)cc1Cl C1(C(=O)NCC(CNC(C(C)(C)C(N)=O)=O)O)CC2COCC(C1)C2 CC1CC(NC(c2ccccc2C2CCC2)=O)CN1C(C1CC(C#N)C1)=O c1(C(=O)NC2C(NC(c3ccc(Cl)cc3O)=O)CCOC2)onc2ccccc12 O=C(CCC(F)F)NC1CC(CCNC(c2cccc(N3CCOC3=O)c2)=O)C1 CC1=CCC(C(C)CC(N2CCCC(CNC3CCCCN3)C2)=O)CC1 C1(NC(=O)CNC(=O)C2CC2)CCN(C(=O)Cc2cnns2)CC1O C(=O)(C(F)(F)CCn1cccn1)N1CC(NC(C2N(C)C(=O)NC2)=O)C(O)C1 c1(C(=O)NCCOCC2CCC2)coc(CNC(C2(C(F)(F)F)CC2)=O)n1 N1(C(CCC(=O)OC)=O)CCCOC(CNC(=O)C(C)(C)n2cccn2)C1 Cc1ccc(C#N)c(NC2CN(C(C3CC4CCC3O4)=O)CC2C)n1 c1(C(C(C)NC(c2cccc(-c3n[nH]c(C)n3)c2)=O)OC)ccc(F)cc1 N1(C(C2CC(C)C2)=O)C2CCCC1CC(NC(=O)Cn1cnnn1)C2 CC1CCc2c(F)cccc2C1NCC1CCCCC1CC(F)(F)F C1(CNC(c2ccc(OCCF)cn2)=O)CCC(F)(CNC(C2(F)CCC2)=O)C1 CCCC(C(=O)NCCc1cc(C(N2CCC(O)(C(C)C)C2)=O)no1)OC C1(CN(C(=O)Cn2cc(Cl)cn2)C)CCCN(C(C2CCC(N(C)C)C2)=O)C1 c1(N(C)C)ccc2c(c1)NC(=O)C2NC(=O)C(N)Cc1ccc(Cl)s1 c1(C(=O)NC(CC)CNC(=O)CC2CC(F)(F)C2)cccc2ncc(Br)n12 C(=O)(C1=CCCOCC1)N1C(CNC(=O)Cc2ccn3cncc3c2)CC(F)C1 C=CCC(CC=C)C(=O)NC1CC2CCC1(C(=O)NCCN(C)CC)C2 C1(C(N2CCCC(NC(C3(O)CCC3)=O)C2)=O)Cc2cc(Br)ccc2O1 c1(C(N2C(C)CCC(NC(C3(CC=C)CC=CC3)=O)C2)=O)cc2n(n1)CCNC2=O n1(C(C(=O)NC(CNC(CCC(=O)NC)=O)C(C)C)C)c(C)cc(O)cc1=O C1(C(=O)NCCc2n(C)ncc2)CCOCC1NC(C1(CO)CCOC1)=O C1(C(=O)NCC2C(NC(CCC#C)=O)CC2)CCS(=O)(=O)N1 N#Cc1cnc(CN2CCCC(CCNC(=O)CC3CC3(Cl)Cl)C2)c(F)c1 C#Cc1c[nH]nc1C(N1CC(CC=C)(NC(=O)Cc2ccccc2F)C1)=O C1(C(N2CCC(N(C(=O)C(F)=C3CCCC3)CC)C2)=O)CC(C)(C)OC1(C)C C1(C#N)(C(=O)NCCn2ncc(C(=O)NC(c3csnn3)C)c2)CC2CC2C1 Cc1ncnc(C)c1CC(=O)NC1CCCC1NC(C1(C)C=CCC1)=O c1(C(N2CCC(CNC(=O)CCCc3nccs3)C2)=O)c(Cl)ccc(Cl)c1O Cc1cnn(C)c1CC(=O)NCC1CCC(NC(=O)CC2OCCCO2)C1 c1(N2CCC(OC)C(F)C2)cc[nH]c(=NCCCN(C2CCCCC2)C)n1 Cc1ncn(CCNC(C2CC3CC3N2C(c2cnc(Cl)s2)=O)=O)c1C c1(OC)c(C(N2CC3CC2CN(C(=O)CCC(C)(C)C)C3)=O)[nH]c2ccccc12 CN=c1cc(C(N2CCC(CCOC)(NC(=O)C=C(Cl)Cl)C2)=O)cc[nH]1 c1(C(=O)NCC(CN(C(CCC(C)OC)=O)C)O)cccc2nc(C(F)F)sc12 C1(C(=O)OC)CCCN(C2CCN(C(C)=O)CC2)C1=O.c12cc(C)sc1C(=O)N2 N1(C(C2CN(C(C)=O)C2)=O)C(C(=O)NCc2nccs2)CC2CCCCC12 C12(C(=O)NCC(CC)NC(c3sccc3C3CC3)=O)CCC(C)(CO1)C2 Cc1cc(C)c(C(N2CCCCC2CCNC(c2nc(C3CC3)cs2)=O)=O)[nH]1 Cc1cc(Cl)c(C(N2CC(C)(C)CC2CNC(c2nc(C)c(C)s2)=O)=O)cc1C c1(C(=O)NC2CC(NC(=O)C(F)n3cccn3)C2)ccc(C2CCC2)nc1 c1(CN(CC(C)NC(C2C(C)C2)=O)C(=O)COCC(=O)NCCO)ccccc1 c1(OC2C(n3cc(C4(OC)CCOC4)nn3)CC2O)ccc([N+](=O)[O-])cc1O Cc1cc(=NCC(C)(C(C)C)NC(c2ccc(F)c(C)c2)=O)[nH]c(Cl)n1 Cc1nc2cncc(C(N3CCC(C(C)(C)NC(C4C(C)C4(F)F)=O)C3)=O)c2[nH]1 C1(C(=O)NC2CN(C(C(CC=C)C)=O)C2)CC12CCc1ccccc12 c1(C(N2C(CN(C(c3c(C)coc3C)=O)C)COCC2)=O)cccc(Cl)c1Cl N1(C(COCC(=C)C)=O)CCC(C(C)C(=O)NC(c2nc(C)cs2)C)CC1 C(=O)(CC(C)(O)CC)NC(C1CCCCC1)CNC(c1cn(CCOC)nc1)=O N1(CC)CCCCC1C(=O)NCC1CCOC1C(=O)N(C1CCCC1O)C1CC1 C1(C(=O)NC(CNC(=O)CNC(c2ccncc2)=O)C2CC2)CCCOCC1 c1(C(N2C(C(N(CCC(F)(F)F)CC)=O)C(C)CC2)=O)cnc(C)[nH]c1=N CCCC(CC(C)C)C(=O)NCC1CCN(C(c2c(C)cnnc2O)=O)C1 c1(OC)cncc(C=CC(N2CCC(O)(CNC(=O)C3=CCCC3)C2)=O)c1 c1(C(=O)NC2C(OC)CCC2)cccnc1CNC(=O)C(C)OCCN(C)C Cc1cc(C)c(S(N)(=O)=O)cc1C(N1CCCCC1CN(C)Cc1cnn[nH]1)=O N1(C(C(C)=CC2CC2)=O)CC2CCN(C(C3CN(CP(C)(C)=O)C3)=O)C2C1 C1(C(=O)Nc2cc(F)cc(F)c2Br)CCC2(CN(CC(N3CCCCC3)=O)C2)O1 c1(C(=O)NC2CCC(NC(C(C)OCCOC)=O)CC2)ccc2c(n1)CCCC2 C1(O)(CC)CCCN(C(=O)C(CC2CCC2)NC(c2cc(F)ccc2F)=O)C1 C1(C)(C(N2CC3C(CNC(c4cc(C)cc(F)c4)=O)C3C2)=O)CCCCC1(F)F c1(CNC(C2(COC)CCN(C(=O)C(C)CC(C)C)C2)=O)cc(OC)nc(Cl)c1 CC1CN(C(c2ncc(F)cc2F)=O)CCC1NC(=O)CSc1ccc(F)cc1 C#CCC(CC(F)F)C(=O)NC1CCCN(C(c2cc(C)ccc2CC)=O)CC1 N1(C(C)=O)CCCCC1C1CCCN(C(c2cc(C3(C)COC3)no2)=O)C1 c1(C(N2CCC(N3CCCC(CCC)CC3)C2=O)=O)c2c(nn1C)CCCC2 Cc1cc(CC(N2CCC(NC(C3CCCS3)=O)C2)=O)nn1C C1(C(N2CC(NC(Cc3cn(CC)nn3)=O)C2)=O)CC(=O)N(C)C1 C(=O)(C1SCCc2sccc21)N1CC(OCCNC(C2CC(C)(C)O2)=O)C1 c1(NC(C(N2CCCCC(CO)C2)c2oc(C)c(Br)c2)=O)cccc(Cl)c1C c1(SC)cccc(NC(C2CCCN2C(C2(C)CC(F)(F)C2)=O)=O)c1 Cc1ccc(C(=O)N(CC(O)CN(C)C(c2cnccn2)=O)C)c2ccccc12 S(=O)(=O)(c1cc(Cl)cc(Cl)c1)N(C1(C(=O)OCC)CCCC1)CC C(=O)(CCCC(=O)N(C1CC(NC(=O)C=CS(C)=O)C1)C)Nc1c(C)cccc1 N1(C(C2N(S(C)(=O)=O)CCC2)=O)CCC2(CC1)CC2NC(c1cc[n+]([O-])cc1)=O Cc1cc(CC(=O)N(C)CC2COCCN2C(=O)Cn2cnnc2O)cc(C)c1 N1(C(c2c(CNC(C(C)OCOC)=O)n[nH]c2)=O)C(CO)CC2CCCC12 C(=O)(C1CCCc2nncn21)NC(CN(C(C(C#C)(C)C)=O)C)C C1(CNC(C(C)N(CC(F)(F)F)C)=O)CC(NC(=O)CC(=O)N(C)C)CCO1 C(=O)(CCCCCCNC(C1CCC(F)C1)=O)N(C(C)C)CC c1(C(=O)NCC2(OC)CCN(C(=O)COC(C)C)C2)cnc2cc(C)ccn12 N1(C(=O)NC2CCCC23CC3)CCN(CC2NC(=O)OC2)CC1 CCC(CNC(=O)C(C)(c1ccccc1)OC)(CC)NC(c1coc(CO)c1)=O c1(COC)ccc(C(=O)NCC2C3CC2N(C(=O)C2CC2)C3)cc1 Cc1cc(CC(=O)NC2(CN(C(=O)CCC3CNC(=O)N3)C)CC2)cc(F)c1 c1(C(=O)NC(c2cccc(Cl)c2)C(=O)O)cc(I)c(Br)c(F)c1F C(C(CNC(=O)CC(C)CC)C(F)(F)F)NC(c1nc(C#C)sc1)=O C1(C(N(CC(C)NC(C2CCCC2)=O)CC)=O)CCC1CF C=Cn1nccc1C(=O)NC(CNC(=O)Cc1ncc(C)s1)CC(C)C C1(NC(c2ccn(CCOC)n2)=O)CN(C(=O)C(C)(C)CC#N)CCC12CCC2 C=C[Si](C)(C)COC(c1ccc(C(C2CCC(=O)O2)=O)cc1)=O Cc1cc(OCC(=O)NC2(CCCNC(C3(c4cccs4)CC3C)=O)CC2)no1 NC1CCCCC1N=c1[nH]c(N2CCC(F)(F)C(F)C2)nc(=N)[nH]1 C1(C(N2C(CNC(c3cnc(O)s3)=O)CCCCC2)=O)CCn2c(O)nnc2C1 C1(C(=O)NCC2(OC(C)C)CCC2)CN(C(c2ccccc2CO)=O)CC12CC2 N1(C(CSCCNC(C(C)n2ccnc2)=O)=O)CCC(C(C)(C)O)C1 N1(C(C2(F)C(C)C2)=O)CCCC2(CCN(C(=O)C(F)CC3CCCC3)CC2)C1 N1(C(CSCC=C)=O)CC2(C=C(C(=O)NOCCF)CO2)C1 C(=O)(C(C)(C)C(=O)N(C1C2CN(C(c3cc(CCO)oc3C)=O)CC12)C)OCC c1(C(=O)NC2CC(C)(NC(C(CCCC)CC)=O)C2)cnn2cccc(C)c12 c1(C(N(C2CCN(C(C(=O)NCC)=O)C2)C)=O)cnn(C(C)(C)C)c1Cl c1(C(=O)NC(C(=O)NCC(C(C)O)O)(C)C)cccn2cncc12 CC1(C)C=C(C(=O)N2CC(CCNC(c3cc4sccc4s3)=O)C2)C1 c1(C(N2CC(N(C)C(C3CC3(F)F)=O)C(O)C2)=O)cc2cncn2c(O)n1 c1(C(C)Sc2nnc(-c3ccc(Cl)cc3)n2CC(=O)NC(C)(C)C)ccccc1O C1(OC)CN(C(=O)COC(F)(F)F)C(C)(CNC(c2ccoc2C(F)(F)F)=O)C1 NS(=O)(=O)c1cnn(-c2ccnc(C(=O)NC3CCN(C4CNC4)C3=O)c2)c1 c1(C(N(C2CCN(C(C3CCCO3)=O)C2)CC)=O)ccc(F)cc1F Cc1cc(F)c(N)cc1C(N1CCC(CNC(=O)C(F)(F)CC2CC2)C(C)C1)=O c1(C(COC(C2CCN(c3ccccc3)S2(=O)=O)=O)=O)ccccc1[N+](=O)[O-] c1(C(C)=O)cnn(C)c1C(=O)NCC(CO)NC(c1ccns1)=O c1(CC)nn(C)cc1C(=O)NCCC1(O)CN(C(c2cn(C3CC3)nn2)=O)C1 C1(C(N2C(C)(CCC)CC2)=O)CN(C(=O)C2=CCC(C)CC2)CC12CCC2 c1(NCCNC(CC(C)C)=O)ccccc1C(F)(F)F.N12CC3CC3(C1)NC2=O c1(CC(N2C(C(C)(C)NC(c3scc(C)c3)=O)CCC2)=O)ccc2nonc2c1 C1(CCNC(c2ccnc(CO)c2)=O)CSCCN1C(c1ccns1)=O C1(C(=O)NCC(C(C)C)NC(C=CC=CC)=O)CCn2ccnc2C1 Cn1cc(C(=O)NC2C3CCN(C(c4cnsn4)=O)C23)c2cccc(Cl)c12 Cc1cc(C)c(NC(=O)COc2ccccc2)c(O)n1.C12(CC1)C(=O)O2 c1(C(N2CCC(NC(C3ON=C(C)C3)=O)C2C)=O)ccc2occ(C)c2c1 O=C(C1=CCCOCC1)NCC1(CNc2nccc(C(F)(F)F)n2)CCCCC1 c1(C(=O)NCCC2C(CC)CC2)cc2cccc(Cl)c2cn1 c1(CNC(CCC#C)=O)ccc2c(c1)CN(C(c1ccc(N)cc1O)=O)C2 C(=O)(C1=CCC2(COC2)OC1)NCC1CN(C(C=C2CCC(C)C2)=O)CC1O C1(NC(C2CC(=C)C2)=O)CC2CCCC(C1)C2NC(=O)CCP(C)(C)=O Cc1cc(C(N2CC(C3CN(C(C45CCC(CC4F)C5)=O)C3)C2)=O)cc(C)c1C N1(CC)CC(CNC(C2CCCCC2CNC(=O)C(O)c2ccco2)=O)OC1=O C(=O)(C1CCCCc2ccccc21)N1CC(N(C(c2c(SC)scc2)=O)C)C1 N1(C(C(C)CC(N)=O)=O)CCCCC2(CCN(C(c3ccc(F)cc3Cl)=O)C2)C1 C12(NC(c3cc(C)ncc3)=O)CCCC1N(CC(C)CC(C)C)CC2 C1(NC(=O)NC(C2(O)CCCCC2)C2CC2)CCc2nnnn2CC1 C1(NC(c2c(C)nc(C)[nH]2)=O)CN(C(=O)C(C)n2ccnn2)CCC1C C1(C(=O)NC(CC)CNC(c2ccc(-c3ccon3)cc2)=O)CCN(C)C(C)C1 CCCC(C)CC(=O)N1CC(OCCNC(=O)C(C2CCC(=O)N2)C)C1 C(CCC1CCC1)(C(=O)NC1(C)CCCC1C)NC(CCSCCC)=O C(=O)(N1CCC(C(=O)NC2CC(n3ccnn3)C2)O1)C1C(C)(C)CCO1 C(C1=NOC2CCCC12)NC(CN(CC#C)C(c1ccc(C)cc1C)=O)=O C1(C(=O)NC2(c3cn(C4C(=O)NCCCC4)nn3)CCC2)CC2CSCC(C1)C2 N1(C(c2n(C)ncn2)=O)CC2CCCC1C2CNC(C1(C)CC1C(F)(F)F)=O C1(NC(c2cnc(SC)s2)=O)CCN(C(C2CCCCS2(=O)=O)=O)CC1(C)C C(CC(C(C)(C)C)NC(c1[nH]cnc1C#N)=O)N(C(=O)CSCc1cscn1)C CCCCC(C(=O)NCc1ccc(F)nc1F)NC(=O)C(C(C)(C)C)OC C(C(C(=O)NCCc1cnn[nH]1)C(C)C)NC(c1n(CCC)ncc1)=O C1(O)(C(C)NC(C2CC(CC)C2)=O)CCN(C(c2cc(CN(C)C)on2)=O)C1 CC1(C)C(C(=O)NCc2ccc(O)cc2)CCN1C(=O)CSC(F)(F)F C(=O)(CCCC(=O)OC)N1CCC(C)(C(=O)NC(CCC)c2ccco2)C1 C1(C)(C(=O)NCC2CN(C(CN(C(C)=O)C)=O)CC2(C)C)CCCCNC1=O Cc1cccc2[nH]cc(CC(=O)NCC3CCC3NC(=O)Cc3cn(C)nn3)c12 N1(C(c2ccc(OC)nc2C)=O)CCN(C(=O)C=CC2CCCO2)C2(CCC2)C1 CC1CN(C(=O)Cc2cnoc2)C(C)CN1C(=O)CN1CCCC1C c1(C(=O)NCCCCN(C(=O)Cc2cnns2)C)ccc2nc[nH]c2n1 C1(C(=O)Nc2ccc(Br)cc2F)CN(C(c2ccc(Br)cc2F)=O)CC(F)(F)C1 CC(CN=c1[nH]c(=NCCC2CCCC2(F)F)[nH]c2c1CCCCC2)C1CCC1 C1(C(=O)NC)CCCC1N=c1[nH]c(=NCc2cccc(OC)n2)[nH]c2ccsc12 C1(CNC(C(COC)(F)F)=O)C2CCC(C2)N1C(c1ncn(C)c1C)=O N1(C(C2(C=C)CCC2)=O)CC(NC(=O)CC2CCOC2)C(C)(C)C1 c1(C(C)OC(=O)CNC(c2ccccc2)=O)ncccc1C(F)(F)F C1(C(=O)NCCC2CN(C(=O)C=C3CCC3)C2)CCCN(c2ccccn2)C1 C=CCCCCCCCC(=O)NC(CNC(c1cnc(C2CC2)o1)=O)CC=C Cc1cc(-c2cn(C3CCN(C(=O)CCCCCO)C3)nn2)c(F)cc1Cl c1(OC(CC)C)ccc(C(=O)NCCNC(c2ccc(CNC(C)=O)o2)=O)nc1 c1(C(N2CCC(C(C)NC(=O)Cn3ncnn3)C2)=O)ccc(Br)cc1O c1(CC(=O)NCCC2CC(NC(c3nc(CC)sc3)=O)C2)ccc2ncsc2c1 c1(C(N2CCC(NC(c3cn(C)nn3)=O)CC(O)C2)=O)cnc2c(F)cccn12 C1(C(=O)NCCCN(C)C(c2cccc(C(C)(C)C)n2)=O)OC2CCC1C2 C1(OC)(CNC(c2cc(CO)[nH]n2)=O)CCN(C(c2ncc(C)cc2C)=O)CC1 c1(C(N2CCC(C(=O)Nc3c(C)ncn3C)C(O)C2)=O)cc(=O)n2[nH]nnc2n1 C1(NC(c2ccc(Cl)o2)=O)CCC2CCN(C(=O)C3=CCS(=O)(=O)C3)C1C2 Cc1ccc(C(F)(F)F)cc1-c1cn(C2CCCCC2n2cccn2)nn1 c1(C(=O)NC2(COC)CN(C(c3cc(CC)on3)=O)C2)c(O)noc1C C(c1ccncc1)=C(C)C(=O)NC1CC1C1COCC1CNC(=O)Cc1cscn1 c1(C(=O)NC(C(C(C)C)NC(C=CC)=O)C2CCCCC2)cc(S(C)(=O)=O)c(C)o1 c1(OC)ccc(C)cc1C=CC(=O)NC1CC2CN(C(c3ccsc3)=O)CC2C1 CCC(C)CC(N)C(=O)NCc1c(C)nn(C)c1N1CCOCC1 c1(NC(c2ccc(I)c(SCc3ccco3)c2)=O)ccc2c(C(=O)O)c[nH]c2c1 C(c1cc(Cl)sc1Cl)=CC(=O)NCC1C2CN(C(C(C)NC(C)=O)=O)CC21 CC1(C)CC(O)CN(C(C2CCN(C(=O)CN3CCCCC3=O)C2)=O)C1 c1(OC)cccc(NC(C2C(O)CCN2C(c2ccc(OCC3CC3)cc2)=O)=O)c1 Cc1nn(CCC(=O)NC(C)CNC(=O)CC(O)CN(C)C)c(C)c1[N+](=O)[O-] C1(N(C)C(c2ccc[n+]([O-])c2)=O)CC2CCC(C1)N2C(C1CC12CCCC2)=O c1(CNCC(C)(C(C)C)NC(C(C)C)=O)cc(Cl)ccc1[N+](=O)[O-] c1(C(=O)NCC(C(C)C)NC(c2csc(Cl)n2)=O)ccc(-n2cnnn2)cc1 CC(C)CC(C)(CNC(=O)CC1COC(=O)C1)NC(c1ccn(C)c1)=O c1(C(=O)NCC(C)CN(C(=O)C(C)N(C)C)C)cc2n(c1)CCS(=O)(=O)C2 C1(CNC(C2C(C)C2)=O)C2CCC(C2)N1C(=O)CCN1CCCCC1=O C#Cc1ccnc(C(=O)NCC(O)C(=O)NCc2cc(C)cc(F)c2)c1 Cc1ccc2cc(CNC(C)(C)COc3cc(F)c(O)c(F)c3)ccc2n1 c1(C(N2CC(NC(C3C(C)C3)=O)CC23CCC3)=O)ccc(S(C)(=O)=O)cc1N C1(C(N(CCC#C)CC)=O)CCCC(NC(=O)CC2CCC(=O)N2)C1 C(=O)(CCCc1cccs1)NC(C1CC1C(=O)N(C1(c2cnn[nH]2)CC1)CCO)C CC1CS(=O)CCN1C(=O)CNC(=O)CNC(C1CCCC(=O)CC1)=O C1(CNC(CCOCCN(C(=O)Cc2ccnc(O)c2)C)=O)CC2(CCC2)C1 c1(CNC(=O)NC(CCSC)C(=O)N(C)C)ccc(I)c(Cl)c1 C(=O)(CC(C)CC(C)C)N1CC(CC(C)NC(Cc2cc(CC)no2)=O)C1 c1(C(CC)C(=O)NC(C)CCNC(C2CC2F)=O)ccc(OC)cc1 c1(C(N(C(C)CNC(=O)C(C)OCC(F)(F)F)CC)=O)c[nH]c2nccc-2c1C C(CC(C(N)=O)NC(c1cc(CNC(=O)Cn2ccccc2=O)nn1C)=O)OC C(=O)(CCS(=O)(=O)CC(C)C)N1CCC(NC(c2cncc(C#C)c2)=O)C1(C)C c1(CC(=O)NCC(C)CNC(C2CC2c2ccn(C)c2)=O)cnn(C(C)(C)C)c1 C(C(=O)N=c1[nH]onc1C1CCC1)c1c(F)ccc(C(=O)OC)c1 O=C1CC(C(=O)NC2CC(NC(c3coc(C(F)(F)F)n3)=O)C2)CCN1 C12(NC(Cc3ccc(C)s3)=O)CCCC(NC(=O)C=C3CCN(C)CC3)(C1)C2 C#Cc1cccc(C(=O)N(C)CC2CCCCN2C(=O)C=CC(=O)N(C)C)c1F C#Cc1nccnc1NC(C1CCCN1CCNCc1ccc(OC)cc1C)=O C(CN=c1[nH]c(=NCc2ccc3c(c2)OCO3)[nH]c2c1CC(C)CC2)=CC C(N=C(NC(C)CC)N1CCC(Br)=C(C)C1)c1ccc(OCC)nc1 C1(F)(CNC(CNC(C(CC)C)=O)=O)CCC(NC(c2cnn(C)c2)=O)C1 C1(COC)CN(C(C2CC2C2(C)COC2)=O)CCN1C(=O)Cn1nnc(C)n1 N1(CC(=O)N(CC(C)CNC(C2CCCC2C)=O)C)C(=O)CCC1=O Cc1occc(=O)c1OCC(=O)NCC(O)CCNC(C1(C(C)C)CCCO1)=O C(=O)(C(F)C(C)CNC(=O)C(C)NC=O)NC1C(CC=C)COC1 N1(C(Cn2c(C)cnc2)=O)CC(NC(=O)CCc2cn[nH]c2)CC1C c1(CC)ncc(Cl)c(C(=O)NC2(C)CCN(C(=O)Cc3ccn(CC)n3)C2)n1 N#Cc1ccccc1C=CC(N1CC(NC(=O)Cc2ccsn2)C1)=O C(=O)(CCC(=O)C1CC1)N(CC(C)N(C(C=CC)=O)C)C CC(O)CCC(=O)NCC1(CNC(=O)CC2(O)CCCOC2)CCCC1 c1(C(N2CCC2CNC(C2(n3cccn3)CC2)=O)=O)cc2c(nc1O)CCCC2O c1(-c2cn(CC(CCNC(CCOC)=O)(F)F)nn2)ccc(Cl)c(F)c1F CC1CC(C(=O)NCC2(CNC(=O)C(F)=CC3CC3)CCOCC2)CCO1 N1(C(CC(=O)OC)=O)CCCC(F)(CNC(C2(OC)CCOC2)=O)CC1 C1(CNC(C=COCC)=O)CCC2(CCN(C(C3CC3C(N)=O)=O)CC2)CO1 C(CCC(C)CC(=O)NC1C2CC1N(C(c1cncc(C)c1Cl)=O)C2)=C(C)C CCCCC(CNC(c1sc(C)nc1CC(C)C)=O)NC(=O)CCCC(=O)OC Cc1[nH]nc(Cl)c1C(=O)NCC1CC(NC(C2CCCCN2C)=O)C1 C(C(C)(C)CC(=O)NCCc1n[nH]cc1C(=O)N(C)CC1(O)CCC1)N(C)C CC(C)C#CC(=O)NC1(CCNC(=O)C(C)CC2CCCO2)CCC1 c1(C(=O)NCC2C(NC(c3c(OCC)cccn3)=O)CCC2)c(C)cc[nH]c1=N N1(C(C(C=C)(C)O)=O)CCC(C2(NC(=O)CCC(C)CC)CC2)CC1 N1(C(c2c([N+](=O)[O-])ccc(C(=O)OC)c2)=O)CCCC1C1CCCCO1 C12(C(=O)NCC(CC)(CC)NC(=O)C=CC(C)(C)C)CCCN1S(=O)(=O)CC2 c1(C(=O)NCc2ccc(CNCC(C)O)cc2)c([N+](=O)[O-])cnn1CC(F)F C(CCC)(C(=O)N1CCCC1C1CCCN(C(c2n[nH]cc2Cl)=O)C1)=CCC C(=O)(C(C(C)C)C(C)C)N1CC(COC)(NC(=O)C(c2ccccn2)O)C1 CC(CN(C)C(c1csc(O)n1)=O)C(=O)N=c1ccn(C)[nH]1 C(=O)(C(C)(C)CCNC(c1cnn2c1OCC2)=O)NCc1c(CC)c[nH]n1 CCC(C)(C)C(=O)C(=O)N1C(C(=O)NCCC(C2CC2)C2CC2)CCC12CC2 N1(C(C2CC3CC3N2C(C2CCCCC2(F)F)=O)=O)CCC2(CCCO2)C1 c1(C(C)C)c[nH]cc1C(N1CCC(C(F)C(=O)NCC2CC23CC3)C1)=O N1(C(Cn2nnc(C)n2)=O)CCC(C2CC2)C1CNC(=O)CCCN(C)C1CC1 C(C(C)(CC(C)C)NC(C12CSC(C1)C2)=O)NC(C(CC=C)C)=O c1(N2CC(CC)N(C)CC2)ccc(S(=O)(=O)NCC#CC2CC2)cc1Cl C1(C(N2CCC(NC(CC(=C)C)=O)C2C(C)(C)C)=O)COCC2(CCC2)O1 c1(C(=O)NC2CCN(C(C(C)(C)OC)=O)CC2C)c(F)ccc(C#N)c1F C(=O)(C(COC)(CC)CC)NCC(CCNC(C(CC)O)=O)(C)C Cc1cncnc1C(=O)NC1CC(CC(N2CCCC(CC3CC3)C2)=O)C1 CC1C(NC(C2CCC=CCC2)=O)CC2CCC1N2c1nnccc1C#N c1(CNC(N(C(C(CC)C)C)CCO)=O)nnc2ccccn12 N1(C(c2c(C)csn2)=O)CC2CCC2(CNC(=O)C(C)CN(C)C)C1 Cc1ncn(O)c1C(=O)NCC(O)CCNC(c1n[nH]c(C(C)(C)C)n1)=O N1(CCOC(CC)C)CC2(C)CN(C(c3nc4cnccc4s3)=O)CC2(C)C1 CCCCCC(C)CC(=O)NCC(=O)NCC(N1CC(C(N)=O)CC(C)C1)=O c1(C(C)=O)c[nH]c(C(=O)NCC2CC(O)(CNC(C3CC3(Cl)Cl)=O)C2)c1 C(c1cccc(F)c1F)=CC(=O)NCCCOCCNC(=O)C=COC1CCCC1 N1(C(=O)COc2ccccc2C(F)F)C2CCCC1CN(C(=O)C(F)C1CC1)C2 Cc1sc(Br)c(C(=O)NCC(O)CCNC(=O)Cc2cc[nH]n2)c1C Cc1ccn2ncc(C(=O)Nc3ccnn3Cc3cncc(Br)c3)c2n1 Cc1nnc(N2CCCC(CNC(C3CC3(C)C)=O)C2)nc1C C1(CNC(C(CN(C)C)NC(CN(CC)CC)=O)=O)CC(C(N)=O)=NO1 C1(Nc2ncc(C)s2)(NC(C)C(=O)N(C)C)CCN(C)CC1 C1(OC)CCCC(C(=O)NC2(CC(=O)NC3CN(C(=O)CC)C3)CC2)C1 N1(C(CC2(C=C)CC2)=O)CC2CC2(NC(C2CCCCC2C(N)=O)=O)C1 c1(C(=O)NC2(CNC(C34CC(F)(C3)C4)=O)CC2)c[nH]c(=O)c2ccnn12 C1(NC(CCNC(=O)NC)=O)CC(N=c2nc(C3CCCC3)[nH]s2)C12CCC2 CC1CCN(C(=O)C=C2CCCC2)CC1CNC(=O)C(O)CC1CC1 C12(C(=O)NCC(C3CCCC3)NC(c3ccnc(C)n3)=O)CC(C)(C1)OC2C C1(CC)CCN(C(C2CCC2C)=O)C(C(=O)N(C2CCC(=O)N(C)C2)C)C1 Cc1nc(C(=O)NCC(C2CC2)NC(C2CCN2C)=O)co1 N1(C(C2(O)CCOCC2)=O)CCOCC(NC(C2(C(F)F)CCOCC2)=O)C1 C1(C(N(CCC(C)NC(CCCc2c(C)nc(C)s2)=O)C)=O)COCC(C)(C)O1 C(=O)(C(=O)N=S(C)(C)=O)NCC1(NC(Cc2cc(OC)c(F)cc2)=O)CCC1 c1(OC)c(C(=O)NC(CNC(c2ccccc2O)=O)C2CC2)nc(O)nc1O c1(C(=O)NC(C2CCN(C(C3(CO)CCCO3)=O)C2)C)ccnc2nccnc12 c1(C(N2CCC(C3N(C(CC)=O)CCOC3)C2)=O)cccc(-c2cn(C)nn2)c1 C(CC(CC)C(=O)N1CCCC1CNC(=O)C(C)(C)c1ccno1)=CC N1(C(c2ccc(Br)cc2F)C(=O)NC(C(=O)OC)C)C2CCC1CN(C)CC2 c1(C(N2C(C(C)NC(CCCOC)=O)CCCC2)=O)cccc2ccncc12 CC(C)CCCCC(=O)NCC(CC1CC1)C(=O)NC1CCCCCC1CO CC1(C)CN(C(=O)C=Cc2ccccn2)CC1CNC(C1(C)CCC(=O)C1)=O C(=O)(C(C)S(=O)(=O)C(C)C)NCC1(OC)CN(C(c2cnn3c2OCCC3)=O)C1 C12CC(C(O)C1)NC(=O)CCCOC2=O.CCC1C(=O)N1C.C(C)(C)(C)OC Cc1cc(=NCc2cc(C(F)(F)F)cnc2F)[nH]nc1-c1ccccc1 C1(N(C(=O)CCC(N)=O)C)CN(C(c2ccccc2CS(C)(=O)=O)=O)CC1(C)C C=CC1(C(=O)N(C)CC2(C)CCCO2)CCN(C(c2cccc(C)c2C)=O)CC1 N1(C(CN2CCC(C)C2)=O)CCC(C2CC2)(NC(=O)CCC(F)(F)F)C1 N1(C(C(CCC)OC)=O)CCC2(CCc3ccccc3C2=O)CC1 C1(C(N2CCC(n3cc(CNC(c4cncs4)=O)nn3)C2)=O)CCC12CCC2 C=CC(C)(C)CC(=O)N1CCSCC1C(=O)NCC1COCCN1C C1(C)(C(=O)NCC(CNC(C(CC=CC)C)=O)(C)C)CCCC(F)(F)C1 C(C(COC)NC(=O)C(F)C1CC(NC(=O)C(O)C2CCCC2)C1)OC CC1(C)OCc2cc(C(=O)NCCCNC(=O)C3=COCCC3)ccc2O1 n1(CC)cc(Br)cc1C(N1CCC(Cc2cn(-c3ccc(O)nn3)nn2)CC1)=O C(C(CO)(CO)NC(=O)C(C)OCCN(C)C)N(C(c1c(C)snc1)=O)C N1(C(c2cnn(C(C)C)c2F)=O)CCC2(C1)CN(C(c1ccc[nH]1)=O)CC(C)O2 c1(C(=O)NC)ccc(=O)n(CS)n1.c1(CNC(c2nccs2)=O)cccc(C2CC2)c1 c1(CNC(C)=O)ccc2c(c1)CCN(c1nn3cc(-c4ccc(Br)cc4)nc3s1)C2 c1(C(=O)NCC2OCC(C(=O)NCC3CC3(Cl)Cl)C2)cnn2c1OCC2 CC1NC(=O)CCC1NC(c1c(CNC(C2CC=CCC2)=O)nnn1C)=O N1(C(C2(P(C)(C)=O)CC2)=O)CCCC12CCCN(C(C1CCCN1N=O)=O)C2 C1(O)(CNC(C2CN(CC(C)C)C2)=O)CCN(C(c2sccc2CC#N)=O)CC1 CCC(F)(C(=O)OC)C(=O)NCCCCCCNC(=O)C(C)C1CC1 CC1CCCCC1(CNC(=O)C1=CCOC1)NC(c1cnc(C(C)(C)CF)o1)=O c1(SCCC(=O)NCCCN(C(C2C(C)C2)=O)C2CC2)nnnn1C1CC1 Cc1cc(C(N2CC(NC(=O)COCC3CCC3)CCC2C)=O)c(N)c(Cl)n1 CCCC(O)C(=O)NCC(C1CCN(C(c2ncsc2C(C)C)=O)CC1)F O=C(N=c1ccn(C2CN(Cc3cccc(F)n3)C2)[nH]1)c1ccc(Cl)cc1Cl c1(C(=O)NC(CC)(C)CNC(C2CCNC2=O)=O)cccc(F)c1 C(CCCC(C)NC(c1c[nH]nc1C(F)F)=O)NC(c1nc(CC(C)C)sc1)=O C(=O)(CC1=CCCC1)NCC(C)CNC(=O)CN(C)C(N)=O N1(C(c2c(C)cccc2)=O)CCOCC(C)(CNC(c2csc(O)n2)=O)C1 C1(NC(=O)C=CCn2cncn2)C2CCN(C(C3CCC([N+](=O)[O-])CC3)=O)CCC12 Cc1nc(Br)sc1C(=O)NCC1C2CN(C(=O)C=CC(=O)N(C)C)CC12 c1(OC)cc(CN(C2CN(C(=O)CCc3ccoc3)C2)C)cc2c1OCO2 C1(NC(c2c(C)nns2)=O)CCC2CN(c3ncc(F)cn3)CC2C1 N1(C(C(CNC(CCCCCC)=O)(F)C(C)C)=O)CCC2(CNC(=O)O2)C1 Cc1nc(-c2ccccc2)[nH]c1C(=O)NCC1CCCN1C(C1C=CCCC1)=O N1(Cc2ccsc2)CCC2CCN(c3nnnn3C3COC4(COC4)C3)CC12 C1(C(=O)NC(CNC(CN(C)CC)=O)C)COCCN1CC C1(CNC(c2c(C)cc[nH]2)=O)CN(C(C2CCCCN2C)=O)CC1(C)C C1(C(=O)NCC(CCOC)NC(c2cncc(NC(C)=O)n2)=O)NC(=O)OC1C C1(C(N2CCC(N(C(c3cnn(C)c3)=O)CC)CC2)=O)COc2ccccc2C1 CC(C)(CN=c1ccc2ncc[nH]c-2n1)NC(c1ccc(C(=O)NC2CC2)o1)=O N1(C(c2cn(C)nc2C2CCC2)=O)CC2COCC(C1)C(=O)N2 Cn1cc(C(N2CCC3OCC3C2)=O)c(O)nc1=O c1(C(=O)NC2C(C)CN(C(=O)CCC3CCC3)CC2)ccc(P(C)(C)=O)o1 CCCC(CC)CC(=O)N1C2CCC1CC(NC(C1COC(C)(C)O1)=O)C2 C1(CNC(CC2(C=C)CCC2)=O)COC(C(F)(F)F)CN1C(=O)Cc1ccon1 Cc1nc(O)nc(C)c1C(N1CCC(C)C(N(C(=O)C(C)NC=O)C)C1)=O c1(CCC)c(C(=O)NCC2(F)CN(C(=O)C(C)CO)C2)[nH]c(C)c1C(C)=O N1(C(C2C(NC(Cc3c(C)nsc3)=O)COCC2)=O)CC(O)C(O)C1CO c1(N(C2CCC2)C(N2C(C(C3CCC3)=O)CCCC2)=O)c(Cl)ccc2c1OCO2 C#CCCCC(=O)NCCC1(OCC)CN(C(=O)Cc2ccc(CO)cc2)C1 C(CC)(C(=O)N(C1CCN(C(=O)COCCc2ccccc2)C1)CCO)OCC C#CCCCC(=O)NCC(C)(Cn1cccn1)NC(=O)CC1CCOC1=O N1(C(c2nc(C(C)C)nc(O)c2)=O)CC(=O)NC2(CC2)C1 c1(C(=O)NCC(C2CC2)NC(c2c[nH]nc2C(F)(F)F)=O)ccc2nn[nH]c2n1 C(=O)(C(C)(C)S(C)(=O)=O)NC(n1cc(C(N2CC(OC)CC2C)=O)cn1)OCC c1(C(=O)NCc2cc(C(N(C(C)CCO)C)=O)n[nH]2)cncc(CO)c1 c1(C2(NC(=O)NC3(c4noc(C(F)F)n4)CC3)CC2CO)cccc(Cl)c1 n1(CCN2CCC(Cc3ccc(F)cc3)CC2)cnc2c1CCCC2 N1(C(COC(C)=O)=O)CCOCC12COCCN(C(c1cc(CO)c(C)o1)=O)C2 CC1CCC(C(=O)NCc2ocnc2C(N2CC(C3CCCO3)C2)=O)CC1 c1(SC(C(N2CCCC(CNC(C)=O)C2)=O)C)nc(O)c2c(C)c(C)sc2n1 C(c1cc(F)c(F)c(F)c1)=CC(=O)NC(C(C)C)CCNC(C1C=CCC1)=O c1(C(=O)NC2CCC2NC(c2ccc(Oc3ccccc3)o2)=O)cc(Cl)ccn1 C1(NC(C(C)NC(=O)CC(C)(C)C)=O)CC(F)CN(C(C2(CC(F)(F)F)CC2)=O)C1 C1(NC)CCCC1N=c1cc[nH]cc1S(=O)(=O)NC(CCCCOC)C(=O)OC c1(CC(=O)NC2C(CNC(c3ccc(C)nc3N)=O)CC2)nc2ccccc2[nH]1 Nc1ccnc(C(=O)NCC(C2CCCCC2)NC(C2C3CC4C(C3)C24)=O)c1 Cc1nc(Cl)ccc1NC(=O)C(CC(C)C)N(C(=O)C(C)S(N)(=O)=O)C c1(C(N2CC(O)(C(C)NC(CCNC(C)=O)=O)C2)=O)c(C)noc1C(F)(F)Cl C(=O)(CCC(C)(C)[N+](=O)[O-])N1C(CNC(c2cc(F)cc(C)c2N)=O)CC1 Cn1nc(C(=O)NC2CC(CC(=O)NCCNS(C)(=O)=O)C2)cc1C(N)=O Cc1cc(C(=O)NC(C)CC(=O)N(C2CC(C)(C)C2)C)n(C)n1 c1(C(=O)NCCN(CC(C)O)C(=O)COc2ccsc2)cc2ccccc2nn1 c1(COC)n[nH]c(-c2cn(C(C)C(=O)NC(C)C(N)=O)nn2)n1 N1(C(C(CC=C)OC)=O)CCCN(C(c2cccc[n+]2[O-])=O)CC1C c1(OC)cc(-c2ccnn2C)c(OC)cc1CN(c1cccc(Cl)c1C)C Cc1nc(C(C)C)ccc1C(N1CCCCC(NC(c2coc(Br)n2)=O)C1)=O CCC(C)C(O)CC(=O)NCC(C)(CC)C(=O)N(C)Cc1ccc(O)cc1 C(N=c1[nH]c(NC2C(C)C2C)nc2c1CSC2)c1cc(C)c(CO)cc1 c1(C(N2CC(SC)C(NC(=O)C=C(C)C(F)F)C2)=O)cc(C)c2nc(C)cn2c1 C1(NC(c2ccc(C)s2)=O)CCCCN(c2nc(Cl)ncc2F)C1 N1(C(c2ccc(C)s2)=O)CCCCC2(CCN(C(=O)C(O)C(C)C)C2)C1 N1(C(c2ccc(C)cc2C)=O)CC2CN(C(C3COCC3(C)C)=O)CCC12 CC1CN(C(=O)C=Cc2cc[nH]n2)CCC1NC(c1cc(CO)ccn1)=O N1(C(c2ccc(CCC)o2)=O)CC2C(CN(C(=O)CNC(C3CCC3)=O)C)C2C1 N1(C(C2(CCC=C)CCCC2)=O)CCN(CCCNC(=O)C(=O)NC2CC2)CC1 c12cn(C)nc1OC2=O.C(=O)(C(C)NS(=O)(=O)CC)N(CC#N)CC c1(C(N2C(CNC(c3c(C)nc(CO)s3)=O)CCC2)=O)nc2n(c1Cl)CCCC2 C12(CC)CN(C(c3ccc(C)n3C)=O)C(CNC(C3CCC(F)CC3)=O)(C1)C2 C(C)(C(=O)NNC(=O)NCC1CCC1)Sc1n(-c2cccc(OCC)c2)cnn1 C1(NC(C2C(C=C)C2)=O)CN(C(c2cnc(OC)nc2C(F)(F)F)=O)C(C)(C)C1 C1(CN(C(=O)COCC2CCOCC2)CC)CCCN1C(C1C=CCCC1)=O C1(CNC(c2cc(COC)cn2C)=O)CCN(C(=O)C(C)OCC2CC2)C12CC2 c1(C(N2CC(NC(C3(O)COC3)=O)CC(F)C2)=O)c(O)cc(=O)n2c1CCCC2 c1(C(=O)NC2(CNC(C(C=CC)O)=O)CC2)cc(=O)c2cc(Cl)ccc2o1 C1(NCC)CCC(c2nnnn2C(C)(C)CC)(NCCC2CCCOC2)CC1 C(=O)(C(C(C)C)N(C)C)NC1(C(=O)NC(CCSCC)C)CC1 C(=O)(C1c2c[nH]nc2CN1C(C1CCC(=C)CC1)=O)NCC=C N1(C(CN(CCC#C)C)=O)CC2(C(N3CCCCC3CCO)=O)CC1CO2 C1(CCC(=O)NCCC(C(=O)OC)C)CCCCN(C(C2(Cl)CCCCC2)=O)C1 C1(CC)C(NC(=O)C=C=C(C)C)CCCN1C(c1ncn(C)c1C)=O CC1(C)CC(CNC(c2ccon2)=O)CN(C(c2cnn(CCF)c2)=O)C1 C1(CCCC)(C(N2CC(O)(CCNC(c3cnoc3C(C)C)=O)C2)=O)CCCC1 C1(C2CC2)(C(=O)NC2C(C(=O)NC3C(CC)C3)CC2)CC(=O)C1 c1(OCC=C)ccc(C(N2CC(NC(c3oncc3CC)=O)CC2C)=O)cc1 C1(C(=O)NC2(CCCNC(c3ccc(C)s3)=O)CC2)CCCC12CCC2 c1(C(=O)OCC)n[nH]c(=NC2CC(CNC(c3c(OC)ccnc3O)=O)C2)s1 C1(O)(C(C(N2C(C(=O)OC)CC2C)=O)NC(c2c(C)csc2)=O)CCCCC1 CN1CCCC(CC(=O)NC2CC2NC(c2c(Br)cnn2CC(F)F)=O)C1 c1(C(=O)NC(C(C)NC(C2ON=C(CC)C2)=O)CO)cc2ccccc2c(O)n1 CC1CCN(C(=O)C(F)(F)c2ccsc2)CC1CNC(c1c(N)cccc1Cl)=O C12(C(=O)NC3CCC(NC(Cc4c(C)con4)=O)CC3)CC3CC(C(=O)N1)C2C3 c1(N(C)CC2CCN(C(C(C)NC=O)=O)C2)cc(O)nc(C2CC2)n1 N1(C(c2c(C)nncc2)=O)CCC(N(C(=O)Cc2cccc(F)c2Cl)C)C(C)C1 C1(C)(NC(c2cncc(NCC)c2)=O)CCCN(C(=O)COCC2CCOC2)C1 N1(C(C(CC2CN(C(Cc3cn(CC)nn3)=O)C2)F)=O)CC2CCOC(=O)C2C1 c1(NC2(CO)CCCC2)nc(N2CC(C)SC(C)C2)c2ncccc2n1 Cc1ccc(NC2CC2)c(C(=O)NCC(F)CNC(C2CC3C(C2)C3(C)C)=O)c1 C1(C(=O)NC(c2conc2C(C)C)C)(CNC(=O)Cn2cccn2)CCCCC1 N1(C(c2n(C)ccc2)=O)CCN(C(c2scnc2C2CC2)=O)CC(C)(C)C1 C1(C)(CNC(c2ccc(C)s2)=O)CCN(C(C2(Cl)CCCCC2)=O)C1 N1(C(CC2(CC(=O)OC)CC2)=O)CCC(NC(C2CCCC23CC3)=O)C(O)C1 C=CCC(C)(C(F)F)NC(C1CCC(CNC(=O)CCCOC(C)=O)CC1)=O C(=O)(CC(O)CCSC)NC1CN(C(c2cc(OCC)ncc2)=O)C(CSC)C1 c1(C(=O)NCC2(F)CN(C(C(CCC)(C)O)=O)C2)cc2c(s1)CCOC2 C1(C2CC2)(C(N2CCC(NC(C3CCCN(CC)C3)=O)C2)=O)CC=CC1 N1(C(c2cc(C)c(Cl)s2)=O)CCC(CNC(C2CC(N(C)C)C2)=O)C12CC2 N1(C(c2n(COC)ncc2)=O)CCCC1C1CCCN1C(c1c(Cl)n[nH]c1C)=O Cc1oc(Cl)nc1C(N1CCC(O)(CCNC(=O)C(C)Cn2cccn2)C1)=O C(=O)(CC1=NN(C)C(=O)C1)N1CC(C)C(CNC(C2CN(C)CC(C)O2)=O)C1 N1(C(C=C(C)c2ccco2)=O)CC(NC(c2sc(Br)nc2C)=O)CC(C)C1 CC(C)C(CCC(=O)NCCCc1ccccn1)NC(=O)CC1(O)CCCCC1 C1(C(N2CC(NC(C3CCC=CCC3)=O)C2)=O)CC2CCCC(C1)C2 C(=O)(C1=CCSC1)NC(c1n(C)ncc1)C(=O)NCC1(C)CC2CC2C1 c1(NC(C(CCC#C)NC(C2CCCOC2)=O)=O)ccc2nncn2c1 c1(CC(=O)NC2CCN(C(C(CCCC)C)=O)C2)cccc2[nH]ncc12 CC1CCCC=C1C(=O)NCC1CC(F)CN1C(=O)CCc1ccnc(Cl)c1 c1(CC(C)C(=O)N2CCC(CN(C(=O)CC3(C)CC3)C)C2)ccc(F)cc1 C(=O)(C1=NOC2(CCN(S(=O)(=O)c3cc(Br)c(F)cc3F)C2)C1)N(C)CC#N c1(C(=O)NCC(CNC(=O)CCCC(F)F)O)c(Br)ccc2n[nH]cc12 C(N=c1[nH]c(=NCCNS(=O)(=O)C(F)F)[nH]c2c1SCC2)C1CC(OC)C1(C)C N1(C(c2c(CC)nco2)=O)CCOC2(CCCN(C(=O)CCn3ccnn3)C2)C1 c1(C(N(CCCNC(c2[nH]cc(CC)c2)=O)C)=O)oc2ccccc2c1Cl C(=O)(C(F)CCC(C)(C)C)NC(CCCC)C(=O)N1CCC1C(C)O c1(C(=O)NCc2cccc(C)n2)csc(=NCc2cccc(C#N)c2)[nH]1 C1(NC(c2cscc2Cl)=O)COC2(CCN(C(c3cncc(F)c3)=O)C2)C1 CN1CC(NC(=O)CCN(C(C23CC(C#N)(C2)C3)=O)C2CC2)C2(CC2)C1 c1(C(N2CC(O)CC(NC(CNC(CCC)=O)=O)C2)=O)cc2c(n1C)CCOC2 C12(CNC(c3ccc(C(F)(F)F)o3)=O)CC1CN(C(c1ccnc(S)c1)=O)C2 c1(C(=O)OCC)nc(C(N2CCC(CNC(C3CC(C)(C)C3)=O)C2)=O)c(C)s1 C1(C(N2C3CC(CNC(=O)C4CC4)C2CC3)=O)COc2ccccc2C1 N1(C(C2=C(C)OCC2)=O)CCC2(CC1)COC(CNC(C1(C)CCSCC1)=O)C2 CCCCCCN(CCNC(=O)C(C)CC1CCCC1)CC1CCSC1 N1(C(CCc2c(C)ncs2)=O)CCCC12CCN(C(C1CC1C)=O)C2 Cc1cncc(C(=O)NC2C=CC(CC(N3CCCC(C(F)F)C3)=O)C2)c1 C1(N(C(=O)Cc2cnccc2Cl)C)CN(C(=O)CN2CCCC2=O)CC12CC2 CC(CCNC(=O)CCc1nccs1)NC(=O)CC1CC(NC(=O)OC(C)(C)C)C1 Cc1scc(C(=O)NC2(CCC(=O)NC(C)C(O)C(C)C)CCCC2)c1C N1(c2nc(C)cc(CC)n2)CCC2(CCCCN(C(c3ccc(F)s3)=O)C2)C1 C1(CN(C)C(C2(CCO)CC2)=O)CCN(C(c2cscc2-c2ccccc2)=O)C1 C12(NC(c3cc(CCCC)oc3C)=O)CCC1CN(C(c1ncsc1C)=O)C2 C1(CNC(c2cccc(-c3ccoc3)c2)=O)CCN(Cc2nc(O)n[nH]2)CC1 N1(C(C2(C)CCCC2)=O)CCC2(CCCC2C(=O)Nc2nnco2)C1 C1(CC(N2CCC(F)(F)C2)=O)OCC2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CCC12 c1(C(=O)NC2CCCN(C(c3nc(C(C)=O)sc3)=O)C2C)cc2ccncc2s1 N1(C(C2C(C=C)C2)=O)CCCCC1C(C)(C)CNC(=O)CNC(=O)C(CC)CC CC1(NC(C2(C)CCOC2)=O)CCC(NC(c2scnc2C2CC2)=O)CC1 c1(OC)cccc2c(C(=O)NC(C)CN(C(=O)CCc3ccoc3)C)n[nH]c12 Cc1cccnc1CC(=O)N(CCCCNC(C1CC2CC1CO2)=O)C c1(OC)ccc(C2N(CC(C)SC)CC2(C)C)cc1O C1(CNC(COCC)=O)CC(O)(CNC(C2CC2c2ccsc2)=O)C1 CC1CN=C(N2CCN(C(c3nc(Cl)sc3Cl)C(=O)NCC3CC3)CC2)S1 C12(CNC(COCC(C)(C)C)=O)CCC(CC1)N2C(c1snnc1C1CC1)=O Cc1cccc(N(C(=O)C2=NOC(C)C2)Cc2cn(CC(=O)O)nn2)c1C C12(C(=O)NCC(CNC(C(C)CCc3ccccc3F)=O)C)CCCC1CCC2 N1(C(CC(C)NC(COCCSC)=O)=O)CC(C)(C)OCC1C C1(CNC(C=CC=CC)=O)C2CCCC1N(C(=O)CN1C(=O)CCC1=O)C2 CC(C)(C)C(CNC(=O)C=CC=C(Cl)Cl)NC(C1CCOC(C(C)C)C1)=O c1(CCOCCC(=O)NC(C2(O)CN(C(c3cnoc3)=O)C2)C)ccccc1 CC1CN2CCN1CC2C(=O)N(CCCCNC(=O)C1=CC2CCCC12)C C1(C(=O)NCC2CN(C(C3(c4ccnc(O)c4)CC3)=O)C2)(CF)CC(F)(F)C1 N1(C(C(CCCC)NC(c2ccc(CO)cn2)=O)=O)CCC2(COC(=O)N2)C1 c1(C(N(CCC(=O)NC(C(CCC)C)C)C)=O)cc[nH]c2nccc1-2 S(=O)(=O)(c1ccc(NCC2CCOC(C)(C)C2)c(Br)c1)N(C(C)CC(N)=O)C N1(Cc2cn(CC(C(=O)OC)C)nn2)CCC(C(N2CCC(C)(O)C2)=O)CC1 C1(C(=O)NCC(CC)C#N)CCN(C(C2CC(C)(C)CO2)=O)CC1 N1(C(CCCOC(C)C)=O)CCC(C(C)NC(=O)CC2(N(C)C)COC2)CC1 c1(C(=O)NCC(CNC(CC(CC)OC)=O)(C)O)cnn2cccc(C)c12 C(c1cnccc1C)=CC(=O)NCC(CNC(C1(SC)CCC1)=O)CO Cc1cc(N2CCC(CC(F)F)CC2)ncc1S(=O)(=O)NC(CO)C1CCC1 Cc1ccc2nc(C)cc(C(N3CCCC3C(C)NC(=O)CC3CCC3)=O)c2c1 c1(OC)n[nH]c(C(=O)NC2CC(NC(=O)Cc3cncc(C)c3)C(O)C2)c1Cl c1(-c2cccc(SC)c2)cnn2c1CN(Cc1sc3cncn3c1C)CC2 c1(C(=O)NCC(C)N(C(COCC(C)C)=O)C)n[nH]c(=N)[nH]1 N1(C(CN(C)C2CC2)=O)CCC(NC(=O)CC2(C)CC2(Cl)Cl)C1C1CCCC1 C=CC(CCC)CC(=O)NCCOCCN(C)C(c1cc(C)nn1CCC)=O CC1(C)OC(C)(C)C1C(=O)NCC1CCC(NC(c2ccc(O)nc2Cl)=O)CC1 CC1CSCCCN1C(=O)CCCCNC(C1(NC(N)=O)CC1)=O Cc1cc(F)ccc1C(=O)NCC(C(C)(C)C)NC(=O)CC1CNC(=O)N1 c1(C(=O)NCC(CNC(C2CC(CC)OCC2)=O)C)cccc2nonc12 N1(C(CC(C(C)C)O)=O)CCC(C2CCOCC2)(CNC(c2ccoc2Cl)=O)C1 c1(N2CC(F)CC(NC(c3cccc(C(F)(F)F)c3)=O)C2)ncnc2sccc12 N1(C(C2CCC(CNC(CC3CC(C)C3)=O)CC2)=O)CC(C)(CO)CC1(C)C Cc1c(C(=O)NCC2CCCN(C(=O)C=CCBr)C2)cccc1O c1(C(=O)NCCCC2N(C(CC3CCCC(C)C3)=O)CCC2)csc2nnsc12 Cc1nn[nH]c1C(=O)NC1CC(NC(C2(c3ccccc3)CC(C)C2)=O)C1 C#CC1(F)CCN(C(=O)CCOCCCNC(c2csc(CO)n2)=O)CC1 C1(CC)CCN(C(c2cc(CNC(=O)C(C)(C)C3(O)CCC3)[nH]n2)=O)C1C C1(NC(C(C2CCCO2)OC)=O)(Cc2ccccc2F)CCCCC1 CC#CCC(C(=O)Nc1ccc(OCC)cc1)NC(=O)CN1CCOC1=O c1(C(N(CCC(=O)NC(C)CCC2CC2)CC=C)=O)ccoc1CC c1(OC)nc(C(=O)NCC2(NC(C3CCN3C)=O)CC2)sc1C Cn1nc(C2CC2)nc1CC(=O)NCCC1CCN(C(=O)CN(C2CCC2)C)C1 c1(C(N2CC(NC(C(CCCC)O)=O)C3(C2)CC3)=O)nnc(O)c(Br)c1O N1(C(C#CCNC(c2ncnc(C)c2C)=O)=O)CCOC2COCC2C1 Cc1ccc(C(N2CCCC(CN(C(=O)CCc3ccccc3)C)C2)=O)c(C)c1 n1(C(C)C(F)(F)F)nc(-c2cncs2)nc1CCCc1ccsc1 CC(CC(=O)N(C)CCC1CCN(C(C2CCCC2C)=O)CC1)CC(F)(F)F c1(C(=O)NCC2CCCCN2C(=O)CC2CC(F)C2)cn2ccccc2n1 c1(C(=O)NC2(C)CN(C(=O)COC3CCCCCC3)C2)cccc(CC#N)c1 Cc1cccc2c1OC(C(N1CCC(CCNC(C3(O)CC(F)(F)C3)=O)C1)=O)C2 c1(C(=O)OC)cc(OC)cc(C(=O)NC2CN(C(=O)C(N)=O)CCC2F)n1 n1(CC)nc(C)c(C(=O)NCCC2CC(NC(=O)CC3COCCO3)C2)c1C c1(NC(c2nccc(-c3scc(C(N)=O)n3)c2)=O)cc(F)c(O)cc1Cl CC(C(=O)N1CCC(C(=O)NCC2(F)CCC2)CC1)C(F)(F)F c1(C(N2CCC(C(N3C(C(=O)NC)CC3)=O)C2)=O)cnc(C)[nH]c1=N Cc1sc(C(=O)NCCOC2CCN(C(C3CCNC3=O)=O)C2)c(C)c1Br c1(C(=O)NCC(CC=C)NC(=O)CCC2CC2(F)F)cc(Cl)cc(Cl)c1Cl CC1(C)C(NC(=O)CN2CC(=O)NC2=O)CCN1C(=O)C=CC1CCOC1 C=CC1CN(C(C2CN(C(c3sccc3CC)=O)CC2CC)=O)CCO1 c1(CC)ccc2c(CC(=O)NC3C4CN(C(c5csnc5C)=O)CC34)coc2c1 c1(NC(CN(CCOC)C(C2(C#N)CCC2)=O)=O)cccc(O)c1 C1(OC)C=CCN(C(=O)C=CCNC(=O)C(n2cc(C)cn2)C)C1 C1(NC(c2c(C(C)C)ncs2)=O)CCOC(CNC(C2CCCN2C=O)=O)C1 C=Cn1nncc1C(=O)NC(CNC(c1csc(-c2ccccc2)c1)=O)C1CC1 c1(C(=O)NCC(CNC(CC(C(=C)C)O)=O)OC)sccc1S(N)(=O)=O Cc1cc(C(=O)NC(C(N2CCC(OCCF)C2)=O)c2ccco2)cnc1C C1(C(=O)NCCCNC(COCC#C)=O)(C(=O)NCC#C)CCC1 C(=O)(CC(C(F)(F)F)n1cccn1)N(CCC)CCNC(=O)Cc1nc(C)cs1 CCC(C)(C(=O)NC(C)C(CO)NC(=O)C(C)NC=O)OC N1(C(CCCCC=C)=O)CCC(N=[N+]=[N-])(C(=O)NC2CC3CC3C2)C1 C1(C)(C(=O)NCCN(C(Cc2scc(C)n2)=O)CCOCCO)CCOCC1 c1(OC)nc(-c2ccc(C(F)(F)F)cc2O)ccc1C(=O)NC1CCNC1=O C1(OC)CC(CNC(=O)CN2CCCNC2=O)N(C(=O)CCc2ncccn2)C1 C1(CNC(C2C(C)(Br)C2)=O)CC2(CO1)CN(C(c1cc3ccsc3[nH]1)=O)C2 N1(C(C=C2CCC(C)CC2)=O)CCC=C(C(=O)NCCc2cn(C)nn2)C1 CC1CCC(C(=O)NC(C2CC=CCC2)CO)N1C(C1CCC1)=O C=C(C)CC(C(=O)NCC(C)CN(C)C(C1(OC)CCCCC1)=O)OC C=C1CCN(Cc2ccc(OC)cc2)C(C(=O)OC(C)C)C1 Cc1nc2c([nH]1)CC(C(=O)NCC(C)CNC(c1sccc1CN(C)C)=O)CC2 C1(O)(CCNC(CSCC)=O)CCN(C(=O)C=Cc2ccc(F)nc2)CC1 C1(NC(C(C(C)OCC)NC(=O)CCCNC(N)=O)=O)CC2(CCC2)C1OC Cc1sc(=O)n(CCC(=O)N(CCNC(C2CCCC2)=O)CC2CC2)c1C Cc1ccnc2nc(C(N3CCC(O)(CNC(C4CC5CCC5C4)=O)C3)=O)nn12 c1(CC(=O)N(CC(C)NC(C(C)SC(F)(F)F)=O)C)ccccc1OC(F)(F)F N1(C(C2OCCN(C(C)C)C2)=O)C2CCC1C(CNC(c1nncn1C)=O)C2 c1(N(CCCC)C)cc(N2CCOC(C3CC3)C2)nc(C)n1 CCC(C)(CCC(C)C)C(=O)NCCCN(C(=O)Cc1sc(C)cc1C)C c1(NCC(=C)F)ccc(S(=O)(=O)NCCCOC(F)(F)F)cn1 c1(OC)ccccc1CC(=O)NCC1CN(C(c2ccc(CO)nc2)=O)CC1C c1(CC)cnc(-c2ccc(C(C)NCCc3ccco3)cc2)nc1 C1(NC(=O)NCCOc2cccc(OC)c2)CC(C)(C)C12CC2 C(CC(=O)NCC(=O)N(CCCNC(=O)CNC(C)=O)CCO)NC(C)=O C1(C(=O)NC(CC#C)C(=O)NC)CN(C(=O)CCC(C)OCC)CCN1C c1(C(=O)OCCC2CC(C)(C)NC2=O)c(Cl)cc(OC(F)(F)F)cc1Cl C(=O)(C1=Cc2ccccc2C1)NC(CN(C(c1ccoc1C)=O)CC)C c1(OCCC)ccc(Cl)c(F)c1C(=O)N(CCC(C)NC(=O)Cc1nc[nH]n1)C c1(NC2C(F)COCC2)nccc(=NCCc2ccc(C3CC3)cc2)[nH]1 C(C(CN1CCCC1)N=c1cc[nH]c(=NCCCC2CCOC2)[nH]1)OC C1(CCNC(C=CC(C)(C)SCC)=O)(NC(c2cc[nH]c2C)=O)CCCC1 C(C(=O)NC(C)C(=O)NCCN(CCCF)C)(C(C)C)OC C(C1=NOC2CCCC12)NC(c1c(C)cc(CNC(CC(CC)OC)=O)o1)=O c1(CC)cc(C(=O)NC2CCCCC2NC(=O)C(C)C(C)(C)O)ccc1C c1(C(=O)NC(C)(CNC(c2cnco2)=O)Cn2cccn2)ccc2ccsc2c1 c1(C(=O)NC2CN(C(C(C#N)=CC3CC3)=O)C2)ccc2ccccc2c1O CC1(C)CCC(C(=O)NC2CC(O)C2)(NC(C2CCC(=O)O2)=O)C1 C1(C(N(C2(C#C)CC2)C)=O)(CNC(=O)CSC)CCCO1 CCC(C)(CC)C(=O)N1CC2(CCN2C(c2cc(C(=O)OC)on2)=O)C1 C(CO)(CCC(C)C)NC(C1CN(C(C2(CC=C)CCCC2)=O)CC1CCC)=O C1(O)(C(=O)NCC2(F)CCN(C(CC3(C)CC3(Cl)Cl)=O)CC2)CN2CCC1CC2 C1(CC(=O)NCCOCCN(C(=O)CN(C)C2CC2)C)CC(F)(F)C1(F)F c1(C(N2CC(N(C(CC(C)SC)=O)C)C2)=O)cccc(CC(F)(F)F)c1 C1(C(N2CC(CNC(C=C=C(C)C)=O)C(C)(C)C2)=O)Cc2cccnc2C1 C1(OC)CCCC(CNC(=O)C(C2CCCN(C(=O)CC3(C)CCC3)C2)(C)C)C1 C1(NC(C(C)OCCCC)=O)CCCCC1CN(C(=O)C(c1ccccc1)F)C C1(C(N2CCC(n3cc(CN4C(=O)CCCC4)nn3)C2)=O)Cc2nccnc2C1 N1(C(CC(=O)OCC)=O)Cc2n[nH]cc2C1C(=O)N(C(C)C(N)=O)C C1(C)(NC(C2C(C=C)C2)=O)CCN(C(C2CCN(C)C2=O)=O)CC1 C(N=c1ccc(Br)c(S(=O)(=O)NCC2CC23CCOCC3)[nH]1)c1cc(C)n(C)n1 C1(OC)CC(NC(=O)CCc2ncc(F)cn2)CN(C(c2cccc[n+]2[O-])=O)C1 N1(C2(c3cccc(C4(N=[N+]=[N-])CC4)c3)CC2)CCN(Cc2ccccc2Cl)CC1 CCC(CCCC(=O)NC1CCC(NC(C2(COC)CC(=O)C2)=O)CC1)SC N1(C(C2(C)CCCC2)C(=O)Nc2c(C)cc(F)cc2)CCOCC12CCOC2 N1(C(Cn2c(C)cc(C)n2)=O)CCC2CCN(C(=O)CCOCC(F)F)CC12 C(c1ccccc1C)=CC(N1C(CC)C(C(N2CCC(CO)CC2)=O)CC1)=O C(=O)(C1=NOC(C)(C)C1)N1CC2C(CNC(CC(CC)CN(C)C)=O)C2C1 C(C(F)(F)CC(=O)OC(C)(C)C)NC(=O)NC1C(OC)CCC1 Cc1ccc(CC(N2CCCC(C(=O)N(C)CCC3(O)CCCC3)C2)C)cc1 CCN(CC(C)C(=O)OC(C)(C)C)N1CC(=O)NC2(CC2)C1 C1(NC(C(=Cc2ccco2)C)=O)CCCN(C(c2cc(C)n(C3CC3)n2)=O)C1C N1(CC)CCN(CCCNC(=O)CNC(=O)N(C2CCCCC2)C)CC1 C(=O)(C1=CCCCNCC1)NCCC(=O)NCc1cn2ccccc2n1 c1(CC)c[nH]nc1C(=O)NCC(C)NC(C1(n2ccnc2)CCC1)=O c1(C(N2C(C(C)NC(=O)Cc3cccn3C)CCCC2)=O)nccc2occc12 CCS(=O)(=O)c1cccnc1C(=O)C.C(N=c1cc(Br)n(C)[nH]1)(c1nc(N)sc1)C1CC1 c1(NC(c2cc(F)ccc2F)CC)ccc2c(c1)CCNCC2 c1(CC)[nH]c(-c2ccccc2)cc1C(N1CC(C)(NC(c2cnc(C)o2)=O)C1)=O C1(CCNC(C(C)OCC=C)=O)CSCCN1C(c1snc(Cl)c1Cl)=O C1(O)(CC(=O)NCC(C)(C)OCC(=O)N(C2(CC)CC2)C)CCOCC1 N1(C(C2=C(C)CC2)=O)CC2CN(C(=O)C(C)C(F)(F)F)CC2C1 C(=O)(C(O)CC(F)(F)F)NC(CC)C(=O)NC1(CN(C)C)CCCCC1 C1(C(=O)NCCCC(=O)N(CC(CC)C)CC)CC(O)C(F)C1 c1(SCC(=O)NCC2(O)CC(NC(C3(OC)CCC3)=O)C2)cc(C)ccc1C C1(NC(C(CSC)(C)C)=O)CCCCCC1C(=O)NCCn1cc(CO)cn1 c1(CC)cccc(C(=O)NCC(C(=O)NC(C2CCOC2)C)N(C)C)c1 N1(Cc2cnn(C(C)C)c2F)CCC(O)(CO)CC1 CCCC(C(=O)NCC(CC)NC(C12CCC(CC1=O)C2)=O)C(C)C C(=O)(C(CC(C)C)C(C)C)N1CCC(C(=O)NC(c2cnn(C)c2)CC)CC1C C(=O)(CC1=CCCCC1)N1CCN(C(C)CNC(=O)C=C2CCC2)CC1 Cc1cc(C(N2CC(CNC(C3(C)CCN(C)C3)=O)C(C)(C)C2)=O)cc(C)c1F C(C(=O)NCC(C)NC(c1cnc(Cl)c(Cl)c1)=O)(C(F)(F)F)OC(C)=O Cc1ncc(C(=O)NCC2CC(CNC(=O)C3=C(Cl)CC3)CO2)c(=N)[nH]1 C1(NC(C2(COC)CN(C(CSC)=O)C2)=O)CCCC(F)C1 CC(C)C#CC(=O)N1CCC(NC(=O)C=CCCC=C(C)C)C1 CCCCCCCCOCC(=O)NC1COCCC1NC(C1CC(=O)OC1(C)C)=O O=C1NCC(C(N2CCC2CNC(=O)C(=O)NCC(F)(F)F)=O)N1 c1(C(N2C3CCC(C3)C2CNC(C23CCC(F)(CC2)C3)=O)=O)cc(F)ccc1O c1(C(=O)NC2CN(C(C34CC(O)C3C4)=O)CC2O)cc(F)c(F)c(F)c1 c1(CC(N2C(CNC(CN(CCOC)C)=O)CC(OC)C2)=O)ccc(C)nc1Cl C(=O)(C(C)(F)C(=O)N1CCCC(Oc2ccc(C)cc2)C1)OCC n1(CC(F)(F)F)nc2nc1-c1c-2cccc1.c1ccccc1.[nH]1cccc1 Cc1ncc(Cl)cc1C(=O)N(C1CN(C(=O)C(C)(C)c2ccns2)CC1O)C C1(CNC(=O)Cc2cccnc2)CC2CCC(C1)N2C(=O)CN1CCOCC1=O CC(C)(O)C(=O)NC1(C(=O)NCCC2CC(F)(F)C2)CC(CO)C1 C(CC(C)C(C)(C)C)NC(CC(CNC(C(C)OCC=C)=O)C1CCC1)=O c1(SC)cc(C)c(C(=O)NCC2CC(F)(CNC(C3CCCN3N=O)=O)C2)o1 N1(C(CSC)=O)CCN(C(c2c(N)sc(C)c2C)=O)CC1c1cn[nH]c1 N1(C(CCOC)=O)CCN(C(=O)CC(O)C2CCCC2)C(c2cccc(Cl)c2)C1 c1(OC(COC)C)ccc(Cl)cc1S(=O)(=O)NCc1sccc1Cl c1(C(=O)NC(C(=O)NCCC)C)ccc(Oc2ccc(Cl)cc2)cn1 C=CC1(CC(N2CCCC(NC(=O)C(C)CO)CC2)=O)CCCCC1 C12(CN(C)C(=O)NCc3cc(Br)ccn3)CC(CN1Cc1ccccc1)C2 C1(C(=O)NCCCN(C(=O)CC(=O)N(C)C)CCC)CCC(C)(C)CC1 Cc1cn2c(CC(N3CCC(C)(NC(=O)C(C)N4CCC4)CC3)=O)csc2n1 N1(C(C(CC)C)=O)CC2(CCC(CNC(c3cc(Cl)c(Br)[nH]3)=O)O2)C1 c1(CN(CCC)CCNC(=O)CCNC(=O)CC2C(C)C2(F)F)cc(C)nn1C N1(C(C2C(C)CCC2)=O)CCCC1(C)C(N1CCCC1C#N)=O N1(C(C2C(CC)C2)=O)CCC(NC(c2ccc([N+](=O)[O-])cc2Cl)=O)C(F)(F)CC1 C(=O)(C(C#N)C(C)(C)C)N1C(CO)C(C(=O)NCc2cc(C)c(C)nc2)CCC1 C(C1CN(C(=O)C2=CCCOC2)Cc2ccccc21)NC(c1cc[n+]([O-])cc1)=O Cc1c(F)ccc(C(N2CCC3(C2)CN(C(C24CCCCC2C4)=O)C3)=O)c1F C(=O)(C1=CC(O)C(O)C(O)C1)NC(C(Cc1ccc(C(C)C)cc1)N(C)C)=O C1(NC(C(C)OC)=O)(CNC(c2[nH]c(C)nc2C)=O)CCCCC1 c1(-c2nnc(N3C(C)C(C)CC3)n2CCC#N)ccc2c(c1F)CCNC2=O C1(C)(CNC(C(C2CCN(C(c3cc(C)c(C)s3)=O)CC2)C)=O)CCN(C)CC1 c1(N2C(C)(C(=O)Nc3cc(C)cc(Cl)c3)CC2)ncnc2occc12 CCC(CC(=O)NCCCCC(=O)N1CCC(CF)C1)OC c1(CNCC(c2ccccc2)F)nc(Cl)ccc1Cl C(CN=[N+]=[N-])(C(=O)N1CCCC1CSC)NC(CSC)=O N1(C(C2CC(CF)C2)=O)Cc2ccccc2C1.C12CCCC1NC(=O)C2 N1(C(CC)=O)CC2CCC1C1CN(C(C3(C#N)CC4CC4C3)=O)CC21 N1(C(c2cc(C)on2)=O)C2CCC1CN(C(c1ccccc1NS(C)(=O)=O)=O)C2 N1(C(c2nc(OC)nc(O)c2)=O)CC(C)(C)CCC1CNC(c1nocc1C)=O c1(C(=O)NC2(CC)CC2)conc1C(C)NC(=O)CC(C1CC1)C1CC1 CC(=O)CC(C)(C)C(=O)NCC1CCCN1C(c1cnn(CCC(C)C)c1C)=O c1(NC(c2cc(C(CC)C)no2)=O)nc2c(s1)CS(=O)(=O)CC2 c1(C(=O)NCC(C)(C)NC(CC(C)F)=O)nc2ccccc2cc1Cl CC1CCN(C(=O)OC(C)(C)C)CCC1NC(=O)CCCC1CCC1 N1(C(C2CC(C)S(=O)(=O)CC2)=O)CC(N=c2[nH]c3ncc(Cl)cc3o2)C(C)(C)C1 N1(C(C2(OC)CS(=O)(=O)C2)=O)CCC2(CC1)CC(NC(=O)C(O)CN(C)C)CO2 c1(C(N2C(CNC(c3ccnc(S)c3)=O)C=CC2)=O)ccc2c(c1)COCO2 [N-]=[N+]=NC1CC(C(N2CSCC2C(=O)N(CCO)C2CC2)=O)C1 c1(CNC(=O)CC2CC2)ccc(-c2ccncc2)cc1F CC1CN(C(C2(c3ccccc3F)CC2)=O)CC1CCNC(=O)C(C)NC(N)=O C1(CNC(CCNC(N)=O)=O)CN(C(=O)C(O)C(F)F)CCC12CCC2 c1(NC(C(=O)NCCC(C)(C)Cc2ccccc2)=O)c(F)cccc1Cl N1(C(CC2N(C)CCCC2)=O)CC2CC(NC(c3snc(Cl)c3Cl)=O)C1C2 N1(C(c2c(COC)scc2)=O)CCC2(CC(NC(=O)C(Cl)=CCl)CO2)C1 CCC(C(=O)NC(C1CCCN1C(c1cccc(Cl)c1F)=O)C)C(C)C C1(CNC(C2(CCCC)CCC2)=O)CC(C(=O)NCC(C)(O)CSC)=NO1 C1(C(=O)OC)CN(C(c2cc(Br)co2)C(=O)Nc2c(C)cccc2C)CC(=O)N1 C1(CNC(CC(C)(C)C)=O)CC2COCC2N1C(c1cccc(Br)c1)=O N(C(=NCC(C)C)NCCN1CC=CCC1)C1CC(OC)C1(C)C Cc1c(C(=O)N(CCCN(C)C(c2ncoc2-c2ccco2)=O)C)cncc1N C1(CC)CN(C(c2cnc(SC)n2C)C(=O)NCCOC(F)F)CC(C)S1=O n1(CC(=O)OCC)cc(C2CC(NC(=O)C(C)n3ccnn3)C2)nn1 N1(C(C(C2CCC(=O)N2)C)=O)CC2(C1)CN(C(c1ccsc1C(F)F)=O)CCO2 c1(C(N(C)Cc2c(C)ccs2)=O)coc2c1CN(C(=O)C(c1cnn(C)c1)O)C2 c1(C(N2CC(CCNC(=O)Cc3cocn3)OCC2)=O)ccc(F)c2occc12 c1(C(=O)NCC2CN(C(c3cc(C)[nH]n3)=O)C(C)CC2)cc(S(N)(=O)=O)oc1Cl c1(OC)cccc(C(=O)NC(CCSC)C(=O)NCC2(C3CC3)CC2)c1 N1(C(COCC=C)=O)C(C(=O)Nc2cccc(O)c2)CCC1C1CC1 C1(C(=O)NC2C(C)CCN(C(C(CC)(C)CC)=O)C2)Cc2ccccc2O1 N1(C(CC2CC(OCC)C2)=O)CCC(NC(=O)CSc2cccnc2)C1CC C#CC1CCC(C(=O)NCCCC2CCCN2C(c2cc(SC)c(C)o2)=O)CC1 C1(N(C(c2c(F)cccc2F)C)C(=O)C2CC2)Cc2cc(Br)cnc2C1 C(N=c1[nH]c2cccnc2s1)C1CCCC(NC(C2(CC=C)CCC2)=O)C1 N1(C(C2CCCN(C(C3C(C)OCC3)=O)CC2)=O)CCCC2C1CCN2C C(=O)(C(C)C(=O)NCC=CC(N1CC(C)(C)C1C1CC1)=O)OC C1(NC(=O)NCCOC2(C#N)CCC2)CCC2C1C2(F)F C(=O)(CCC(=O)NC(C)CC(C)NC(=O)CCOC1CCOC1)NCCC C(=O)(C(C)(O)CCC)N1CCCC(N(C(Cc2nc(CC)sc2)=O)CCF)C1 C1(C(C)(C)C)CCN(C(=O)CC2CC23CC3)C(CNC(=O)C2=CCCCC2)C1 c1(OC)cc(N2CCCC(N(C)C(C3CC4(C3)CC4F)=O)CC2)ccc1[N+](=O)[O-] c1(C(=O)NC2CN(C(C3(OC)CCC(C)C3)=O)C2)c(C)cc(C)cc1O c1(CCNC(=O)CCC2(NC(c3ccon3)=O)CCCC2)ccc(F)cc1 C1(OCc2cc(N3CCCC(OCCOC)C3)ncn2)C2CCOC2C1(C)C CCCCCCC(=O)NC(C1CCN(C(C2(F)CC2c2ccccc2)=O)C1)(C)C N1(C(C(C(C)O)C)=O)CCC(CNC(=O)Cc2cccnc2Cl)C(C2CC2)C1 CC(C)CC(O)C(=O)NC12CCC(CC1NC(c1ccc(C#N)cc1)=O)C2 C1(C(=O)NC(C(=O)OC)Cc2[nH]cnc2C)OCCCN1C(=O)OC(C)(C)C C=CCCCC(C(=O)N1CCC(CCCO)CC1)NC(c1cc(C)ns1)=O N1(C(C2(F)C(C)C2)=O)CCC2CN(C(=O)CN3CCCC3=O)CCC2C1 C(=O)(C(C)CCC(C)(C)C)NCC(C)NC(=O)Cc1ccc(F)cc1Cl C=CCC(C(=O)NCC)NC(C1CCC1C(F)F)=O.C12C(C1(C)C)CNC2=O c1(OC)cccc(C(=O)NC2(CC(=O)NC3CCC3O)CCC2)n1 Cc1cc(C(=O)NC2CN(C(C3(CO)CC3)=O)CCC2F)c(C)n1C1CCOC1 N(C1CC(C)c2cc(Br)ccc21)C(C1(CC)CCCC1)=O C12(C(=O)NCCC(Cn3cc(C(COC)(C)O)nn3)F)CCCCC(F)(C1)C2 c1(C(N(C(C)CCNC(C2(Br)CC2)=O)C)=O)cc(CN(C)C)on1 C1(C(C)O)C(=O)N1.Cc1ccsc1C(CO)N(C1CCC1)C(=O)OC(C)(C)C C1(CC(=O)NCCCNC(c2ccn(CC)n2)=O)CCCCC1F CC#CCCC(=O)NC1(CN(C(=O)CCOCC(F)(F)C(F)F)C)CC1 N1(C(c2cnc(OCC)nc2)=O)CCC(C)(C)C1CNC(c1cc(OC)n[nH]1)=O Cc1cc(C#N)cnc1C(=O)N(C1CCN(C(=O)Cc2ccnc(O)c2)CC1)C C1(CNC(C2(CC=C)CCC2)=O)CCN(C(=O)C(C)OCCOC)CC1(F)F Cc1ccc(-n2nc(C3CCOCC3)nc2C(N2CCC(F)C2)C)cc1 CCCC(C(=O)NC1CCCCC1CNC(=O)CNC(C)=O)NC(C)=O N1(C(=O)Nc2ccc(C(F)(F)F)cn2)CCN(C(C2C3COCC23)=O)CC1CO CCC(O)C(C)C(=O)NCC1CCN(C(c2cccn2C2CCCC2)=O)C1 N1(C(c2ncn(C(C)C)c2)C(=O)NC2CCCC2)CCC12CCSCC2 C(C(=O)NC1CC(CNC(c2ccc(NC=O)cc2)=O)C1)(C(C)C)SC c1(C(N2CCN(C(c3c(Cl)ncc(C)c3)=O)C(C)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 Cc1ccsc1CC(=O)NC1CC(NC(=O)C=CC2CCOC2)C1 C1(CNC(CCSC)=O)CC2CC1CN2C(=O)Cc1ccc(F)cc1 CCC(Cc1ccc(F)cc1)N=c1ccc2ncc[nH]c-2n1 C(=O)(C1CCCc2ncnn21)N1CCC(N(C(c2ccnc(C(C)C)n2)=O)C)C1 C1(C(=O)NCCOCCN(C)C(c2cc(C(C)(F)F)n[nH]2)=O)CCC=CCCC1 N1(C(C(C)(C)C2CC2)=O)CCC2CCN(C(C34CC(F)(C3)C4)=O)C2C1 CC(O)CC(=O)N1CC(NC(c2cc(C(F)F)[nH]n2)=O)C1 N1(Cc2cn(-c3ccnc(C(=O)O)c3)nn2)CCCN(C2C(C)CC2)CC1 N1(C(C2(CC(C)C)CC2)=O)CC2CC(C1)CN(C(C1CCCC(C)(C)O1)=O)C2 N1(C(C(C)CO)=O)CC2CC1C2CSc1coc(-c2cn(-c3ccccc3)nn2)n1 C1(C(N(CC(C)N(C(C)=O)C)C)=O)CCCCN1C(=O)C(C)=C1CC1 Cc1cccc(C(N2CCCC2C(C)(C)CNC(C2CC23CCOC3)=O)=O)c1F Cc1ncc(Cl)cc1C(=O)NCCCNC(C1CCC1c1ccco1)=O N1(C(c2cnc(C(=O)N(C)C)o2)C(=O)NCCCOC)CC2CCCCCC2C1 N1(C(=O)Nc2c(NC(=O)C3CC3)ccc(C)c2)CCS(=O)C(C)(C)C1 c1(C(N(C2CCN(C(CSCCCC)=O)C2)C)=O)nc2ncc(CCO)cn2n1 CC1(C)CC(C(=O)NCc2c(O)cccc2F)CN(C(C2CC=CCO2)=O)C1 C1(C)(C(N(C)CC2CCN(C(c3c(C)nn(C)c3)=O)CC2)=O)CCCCC1C C(=O)(NNc1cccc(Cl)c1)c1cccc(OCCNC(=O)OCC)c1 CCC(CC)(CCNC(c1ccnn1C)=O)NC(=O)C(c1nc(F)ccc1Cl)C C(=O)(CC1OCCc2sccc21)OCc1nc(CC)on1 C1(C(=O)NC2CC(NC(C3(F)CCOC3)=O)C2)CCN(C2CC2)CC1 C1(C(N2CC3C(C(=O)OC)(C3)C2)=O)C2C(CN1C(c1sccc1OC)=O)C2(C)C c1(OC)nc(C)cc(=NCC(O)CNC(c2cc(CN(C)C)c[nH]2)=O)[nH]1 n1(CCNC(CNC(C(=O)Nc2ccc(N)cc2)=O)=O)cc(Cl)c(O)nc1=O c1(Nc2cnc(-c3ncccn3)s2)ccc(C(=O)NCCOC(C)C)cc1 N1(C(COC(C)C)=O)CCC(C(N2CCC(c3nn[nH]n3)C2)=O)(CF)C1 N1(C(C2COCC(C)O2)=O)CCCCC(C(=O)NCCCc2ccnn2C)C1 CC1(C)CCC(C(N2CCCC2C2(C(=O)NC3CC3)CCC2)=O)CO1 c1(C(=O)NC(CNC(C(N2C(CC)CCC2)=O)=O)C)cc2c(F)cccc2[nH]1 c1(C(N(CCC(C)NC(c2c(C)cc(O)nn2)=O)C)=O)cc2ccccc2s1 Cc1nc2cnn(C)c2cc1C(=O)NC1(CNC(=O)C(O)C(F)(F)F)CC1 C1(C(=O)NC(CSC)(C)CO)CCN(C(c2c(F)cncc2F)=O)CC1O c1(C(N2CC(CCCCNC(c3nnn(C)n3)=O)C2)=O)ccc([N+](=O)[O-])cn1 C1(NC(CN(CCOC)C(c2nc(Cl)cs2)=O)=O)CCC(N=[N+]=[N-])CC1 c1(CN2CC(C(=O)NCCC=C)OCC2)cc(Br)cc(F)c1O CCC(C)CC(=O)NCC1CC(C(N2CC(C)(C)C2C(C)C)=O)C1 C#CC(CCC)NC(c1occc1CNC(=O)C=CCN1CCCC1)=O Cc1ccnnc1C(=O)NC1CC2(C1)CC2C(=O)NCc1cc(=O)cc[nH]1 C1(CNC(c2cccc(CO)n2)=O)CC12CCN(C(=O)CCc1ccsc1)CC2 Cc1cc(F)ncc1-c1cn(C2(C(N3CC(N(C)CCO)C3)=O)CC2)nn1 N1(C(C(C2CN(C(C3C(C)=CCS3)=O)C2)O)=O)CCC(C)(CO)CC1 c1(C(C)OC=O)nnnn1C1CCC1.C(=O)(CN(C(C)(C)C)C)NCCN N1(S(C(CC)C)(=O)=O)CC2CN(C(c3cc(CC(C)C)nn3C)=O)CC2C1 C1(CNC(C=CC=CC)=O)C(C)CCN1C(c1ccc(-n2cncn2)cn1)=O c1(C(=O)OCC=CC)ccnc(C(F)F)c1 c1(C(N2CCC(C3CCCN3C(=O)CC3CC=CC3)C2)=O)coc(Cl)n1 C1(CC=C)(NC(=O)C(O)COC)CCCN(C(=O)Cc2ccc(CC)cc2)C1 c1(NC(=O)NC(c2ncon2)C)cnc(C(F)(F)F)cn1 c1(CC(N2CCC(CN(C(C3C(CC)C3)=O)C)C2)=O)nc(C)sc1C c1(C(N2CC(CCNC(C(CC)C)=O)OCC2)=O)ccc2cccc(CC)c2n1 C12(C(=O)NC(C3CCN(C(CCC(C)OC)=O)CC3)CO)CCCC1C2(F)F N1(C(Cc2c(C)ocn2)=O)C(C(=O)NCCNS(C)(=O)=O)CCC1C1CC1 C(=O)(C#CC1(C)CCCO1)CC.C12CC3CN(CC13)C(=O)C1=CCC(C1)CO2 CC1(C)CCCC(C(=O)NC(C2CCCC2)CNC(=O)C2CC2)CC1 C1(CNC(c2c(C)scn2)=O)(Cn2cc(C3(CO)CC3)nn2)CC12CCC2 N1(C(CC(C)(F)F)=O)CCCC(CO)(NC(c2cc[nH]n2)=O)C1 C1(C(=O)NCc2c(C(N(CC(C)(O)C3CC3)C)=O)n(C)nc2)C2CCC(F)(F)C12 c1(C(N(CCC(C)NC(c2c(C)oc(C)c2C)=O)C)=O)cccc2ncn(C)c12 C(C(=O)NCC(C)OC(F)F)(c1ccoc1)NCC=CC(=O)OCC.C(CCC)O O=C(C1=CC(O)CCC1)NC1CN(C(c2ccc(N3CCC3)nc2)=O)CC1O C1(C(=O)NC2(CNC(C(C)OC(C)(C)C)=O)CC2)CCc2nncn2C1 C(=O)(C(C)C(F)(F)C(F)F)NC1CC(N(C(c2cc(CC)n(C)n2)=O)C)C1 N1(C(CCCOC(CCC)=O)=O)CCCCC1CCNC(=O)C(CC)NC(C)=O n1(CC)cnc(C(=O)NCCCC(C)NC(c2ccoc2Br)=O)c1 C1(CC(=O)NCCC(C)N(C(=O)CC2(CO)CC2)C)CCCCC(=O)N1 N1(C(c2nc(C(C)OC)sc2)=O)CCC(NC(C2CC3(CCC3)CO2)=O)C(O)C1 S(=O)(=O)(CCC(=O)N1CC(CCNC(C(N2CCSCC2)=O)C)C1)NC C(=O)(C1CCCc2scnc21)N1CC2(C(NC(c3c[nH]nc3C3CC3)=O)CC2)C1 C(=O)(C1CCc2c(Cl)cccc21)N(CCNC(C1CCCOC1)=O)CC C1(C2CCN(c3nnccc3C#N)C2)(NC(CCCCC#C)=O)CC1 C12(C(N3CCC(O)(CC)C3)=O)C(NC(=O)Cc3cn(C)nc3C)C3CC1C2C3 N1(C(C(C)(C)SC)=O)CCN(C(c2cc(C)c(C)[nH]2)=O)CC(O)C1 c1(C(=O)NCCC2CCCN(C(C(C=CC)O)=O)C2)cc2cccc(C)c2s1 C=CCC(C(=O)N1CC(CCNC(=O)C#CC(C)(C)C)C(C)C1)C(C)C C(=O)(C1(C)CCc2ccccc21)Nc1cc(NC(C)=O)c(F)cc1 c1(C(=O)NCc2nc(CNC(c3nn(CC)c(C)c3)=O)sc2)cc([N+](=O)[O-])c[nH]1 C(=O)(C(F)(F)c1cncs1)NCC1N(C(CN(C)C(=O)C2CC2)=O)CC1 C1(C(=O)NC(c2sccc2Cl)C)CCC12CCCO2 CC(C)C(C)CN=C(NCC(N1Cc2ccccc2C1)(C)C)NC1CCC1 C(=O)(C(C(C)C)C1CCC1)NC(COCC)C(=O)NC(C)Cc1cncnc1O c1(C(N2CCC(OCCNC(CNC=O)=O)CC2)=O)ncn2ccccc12 c1(C(N2C(CNC(c3c(C)cnc(F)c3)=O)CCC2)=O)cnc2cccc(C)n12 C(c1ccc(S(N)(=O)=O)cc1)=CC(=O)NCCNC(Cc1c(C)n(C)nc1)=O Cc1ccc(C(=O)NCC2CC2CC(=O)NC(c2nc(C)no2)C)o1 CCCCC(CC(=O)N(CC(O)CO)C(C)C)NC(c1cccc2[nH]ccc12)=O c1(NC(C2(F)CCN(Cc3c(OC)cccc3Br)CC2)=O)nc(Br)c(Br)cc1Br C1(CC(N2CCC(O)(CNC(COCCCC(C)C)=O)C2)=O)CCCCC12CC2 CC1Cc2cccc(C(N3CCCC3CN(C(=O)C=CC3(C)COC3)C)=O)c2O1 C1(C#N)(C(N2CCC(OCCNC(c3c(C)ncs3)=O)C2)=O)CC(C)C1 N1(C(C2(NC(C)=O)CCCC2)=O)CC2(CCNC(=O)Cc3cnc[nH]3)CCC1C2 N(C1CCCn2ncnc21)C(=O)NCCNC(c1cnc(O)nc1)=O c1(OC)ccc(F)cc1CN1CCC(C(=O)Nc2cc(O)ccc2C)CC1 C(=O)(C(C)CS(C)(=O)=O)OC.C12(NC(=O)NCC3CC3)CCCN1C2=O N1(CC(=O)NC(CC(C)NC(c2cc(C(=O)OC)sc2)=O)C)CC(=O)NC1=O CC(C)CS(=O)(=O)CCC(=O)N1CCC(C)C(NC(C2CC(C)OC2C)=O)C1C N1(C(CCCCSC)=O)CCN(C(c2cc(C(C)C)[nH]n2)=O)CC(O)C1 N1(C(CC(=C)C)=O)CCC2C(CCN2C(=O)CC2CSc3ccccc3O2)C1 CN=c1nc(C(N2CCC(NC(=O)COCc3cccc(C)c3)C2)=O)cc(C)[nH]1 C1(C)(C(N2CCC(CNC(c3ccc(CCC)s3)=O)C2)=O)CC(C)=NO1 c1(CC2(C(N3CCC(C(C)(C)NC(=O)CP(C)(C)=O)C3)=O)CC2)cccc(F)c1 C1(C(F)(F)F)(C(N(C2C(SCC)CC2)C)=O)CC=CCO1 c1(C(C)NC(C2N(CCC)CCC2)=O)sc(-c2ccc(Cl)cc2)nc1C CCCC(CCC)NC(=O)CCC(C)NC(=O)COc1ccccc1 C1(NC(CSSC)=O)C=CCN(C(c2cn(-c3ccn(C)n3)cn2)=O)C1 N1(C(C2C(CCC)CCC2)=O)CCC(O)(CN(C(=O)C(CO)OC)C)C1 c1(NC2CC3CN(C(c4ccc(OC)c(Cl)n4)=O)CC32)nc(C)nc(O)c1C CC1(C)CCCN(C(C2(CO)CN(C(=O)CCOCC(F)F)C2)=O)CC1 C1(C(=O)NCc2nn(CC)nc2C)CC(C)(C)CCN1C(=O)CCn1ccnc1 S(=O)(=O)(c1ccccc1)N(CC(CN(C)C(=O)NCCC1CC2CCC1C2)O)C c1(OCC(=O)NCCC(C)N(C(=O)CC2CC(=O)NC2=O)C)cncc(Cl)n1 C1(NC(C2C(Cc3ccc(C)cc3)CCC2)=O)CCC(C)N(C(=O)CCF)C1 Cc1nc(CC(C)C)oc1C(=O)N(CCCNC(c1cn(CCCF)nn1)=O)C C(=O)(N=c1nc2cc(Cl)ccn2[nH]1)C1C(C)(C(F)F)C1 N1(C(CCCC=C)=O)CCN(C)CC1C(N1CCN(C)C(CC)C1)=O N1(c2nnc(-c3cc(C)oc3)n2CCCOC(C)C)CCc2ccc(F)cc2C1 c1(CC(=O)N(C(C)CN(C)C(c2n[nH]cc2Br)=O)C)ccc2c(c1)CCO2 N1(C(COCCC(=O)OC)=O)CCC(NC(=O)CC(C)n2cccn2)C12CC2 C#CC1(C(=O)NCC2(C)CCN(C(=O)C(c3cccc(C)n3)(F)F)C2)CCCC1 C(C(O)CC(F)(F)F)Oc1c(C)oc(C(C)(C)C)c1 c1(CC)nc(Cl)c(C)c(=NCC2(NC(=O)C=Cc3ccc(C)c(Cl)c3)COC2)[nH]1 n1(CCC#C)cc(NC(c2n[nH]cc2Br)c2nnnn2CCCSC)cn1 N1(C(COCc2onc(CC)n2)=O)CC(NC(=O)C(C)=CC2CC2)CC1(C)CC Cc1ccc(N(C)CCN(C(=N)N)C(c2ccc(Cl)cc2)c2ccccc2)cc1 C(COC(C)C)(C(=O)NC(c1ccn(C)n1)C)NC(C1C(=C)C1C(C)C)=O N1(C(N)=O)CCC(C(=O)NCC2CCCCN2C(C2CC23CCC3)=O)CC1 N1(C(c2nc(C)oc2)=O)CCOC2(CCN(C(C3(C)CC3C(F)(F)F)=O)CC2)C1 N1(C(CN(CCCCCC)C)=O)CCC(CO)(NC(c2cc(NC)cs2)=O)CC1 Cc1cc(NC(=O)OC(C)(C)C)c(C)cc1NC(N1CC(C#N)C1)=O C1(C(=O)NC2CCN(C(C3(SC)CCC3)=O)C2)(N(C)C)CCC(F)(F)CC1 C1(O)(CC(=O)N(CCOC)C(C)C2CC2)CCN(C(c2coc(OC)n2)=O)CC1 CCCCCC(O)C(=O)NC(CCC)C(=O)N(C)Cc1cncnc1 C(=O)(C(CO)NC(C1COCC1C(N)=O)=O)NC(CN(CCCC)C)C CC1CN2CCCCC2CN1C(=O)Nc1ccc(COC2CCCC2)o1 C1(C(N2CCC(C(C)NC(C3CN(C4CCCCC4)C3)=O)C2)=O)CSCC(=O)N1 N1(C(C=C(C)C)=O)CCC(O)(C(C)NC(=O)CCC2CC2CC2CC2)C1 c1(C(N(C)CC2CCCN2C(=O)CCCn2ccnc2)=O)ncc2[nH]ncc2n1 C(=O)(C(C(C)(C)C)NC(N)=O)NCCC(CCNC(C(C)=CC1CC1)=O)C c1(OC)c(F)ccc(F)c1C(=O)NC(CCNC(=O)COc1ccon1)C(C)C C#CCC(C(=O)NCC1CC1C(=O)OC)NC(=O)CCc1ccncn1 c1(OC)cc(F)cc(C=CC(=O)NC2CN(C(=O)Cc3nnc(C)s3)CC2C)c1 CC1CC(C)(C(=O)NCC(C2CC2)N(C(=O)C=C2CCSCC2)C)CC(C)O1 C(=O)(C(C)C(C)(F)F)NC1C2CN(C(c3n(CC)ccn3)=O)C1C2 CC1=C(C(=O)N2CCC(NC(C3CC4C=CC3C43CC3)=O)C23CC3)SCCO1 C1(NC(CCCC)=O)CS(=O)(=O)N(C)C12CCN(c1ccc(C#N)c(C)n1)CC2 C(=O)(C1CCCn2nccc21)NCC1(OC)CCN(C(C2(F)CCCC2)=O)CC1 C=C(C)CC(C)C(=O)N1CC=C(CNC(=O)COC2CCOC2)CC1 N1(C(CS(=O)(=O)NC(C)(C)C)=O)CCC2(CCC2)C(NC(c2cc(Cl)n[nH]2)=O)C1 c1(OC)ccc2nc(OC3(C)CCCCC3)cc(C)c2c1 c1(C(N(C(C)CN(C)C(C2CCCN2C2CC2)=O)C)=O)cnn2c1OCC2 C1(CNC(C2C(CC)CCC2)=O)(NC(=O)C(=O)NC(C)C)CCC(F)(F)CC1 C(=O)(C1=CCCN(C(=O)OCC(C)(C)C)C1)NC(CNC(C(CC=C)C)=O)CC C1(C(=O)OC)CC(=O)N(C)C1C(=O)NCC1CCN1C(c1nn(CC)cc1Cl)=O CCC(CN(C)C)CC(=O)N1CCCCC(NC(=O)C(C)NC(=O)NC)C1 CC(C)C(O)C(F)(F)C(=O)N1CCN(C2CCCC2NC(=O)COCCF)CC1 c1(CNc2cn(CCNC(C3CCN3C3CCCC3)=O)nn2)ccccc1F CCC1=NOC(C(=O)NCC(O)CC(=O)NCc2cc(CC)no2)C1 N#Cc1ncc(NCC2(F)CC(NC(C3CCCCC3)=O)C2)nc1C#N Cc1ncc(NC(C2(NC(c3cnns3)=O)CCC2)=O)cn1 C1(CC(=O)NC(C)CCCNC(c2cnn(C)c2Cl)=O)CCC2(CC1)CC2 CCCCCCC(C)CC(=O)NC1CCC(CNC(c2[nH]c(O)nc2C)=O)CC1 c1(OC)ccnc(C(N2CC(NC(=O)C=C(C)c3cccs3)C(F)C2)=O)c1F c1(SC)nc(N2CCCC(C(=O)Nc3cccc(Br)c3)C2)ncc1Cl c1(C(=O)NC2CCC(NC(C3CN(CC)C(=O)C3)=O)CC2)ccnc2c1CCO2 Cc1cc(=NC(C)CC2CCC2)[nH]c(N(C)CC23CCCC2OCC3)n1 C(=O)(C=C1SCC(=O)N1C)N(C(C)CNC(C1CCC(C(F)(F)F)O1)=O)C N1(C(C(C2CCCC2)OCC)=O)CCC2(C1)CN(c1ncc(C)c(C)n1)C2 Cc1cc2c[nH]nc2cc1C(=O)NCC(C)N(C)C(C1CCn2cncc2C1)=O c1(CNC(C(CC)N(C(=O)CC2=CCCC2)C)=O)ccc(F)c(O)c1 Cc1nc(Cl)ccc1CC(=O)NCC1CCC1NC(=O)Cc1ccncc1Cl Cc1ccc(CN2CCC2(C)C(=O)NC2CCS(=O)(=O)C2)c(F)c1 [N-]=[N+]=NCCCCCC(=O)NCCn1cc(C(=O)NC2CC23CC3)nn1 N1(C(CC2(C#N)CC2)=O)CCCOC(CNC(c2cnc(C3CC3)o2)=O)C1 Cc1cc(C(=O)N(C)CCN(C)C(C2(C)CCCCC2)=O)c2n[nH]cc2c1 S(=O)(=O)(c1ccc(F)cc1)N1CCCC(NC(=O)NC2C(OCC)CC2)CC1 N1(C(C)C)C(=O)COCC1C(=O)N(CCCCCNC(=O)CCC1CCCO1)C N1(C(C(=O)Nc2ccc(C)nc2)=O)CCCC(c2ccccc2)C1C CC1CCC(NC(c2ccnc(F)c2F)=O)CN1C(C1CN(CC(F)(F)F)C1)=O c1(NC)ccc(C(N2CCC(CNC(=O)CN3CC(C)C3)CC2)=O)cc1F c1(OC)c(C(=O)NCCN(C)C(C2CCC(F)C2)=O)[nH]c2ccccc12 C1(CCC)CN(C(c2ocnc2C)=O)CCN1C(C1CCC1C(F)F)=O C1(CC(=O)Nc2ccc(C(=O)OCC)c(C(=O)O)c2)Cc2cc(F)ccc2O1 CCN=c1[nH]c(C(=O)NCC2C(C)CCCN2C(c2cncn(C)c2=O)=O)cs1 c1(NC(c2n(CC)nnn2)c2ccn(C3CC3)c2)cnc(O)c(C(F)(F)F)c1 C=CCC(C(=O)NC(CCC)C(=O)NCc1cc(COC)no1)C(C)C N1(C(C(CC=C)OC)=O)CC(C2CCCN(C(C3(O)CCOCC3)=O)C2)C1 CC1(C(=O)NC2CC3CCC2N3C(c2cnoc2C2CC2)=O)CC(C2CC2)=NO1 C1(CNC(C(C)O)=O)CCC2(CO1)CC(NC(=O)Cc1sccc1Cl)C2 C1(C(=O)NC(CC)(CNC(c2cc3c(s2)CCC3)=O)CC)Cc2ccccc2O1 N1(CC(=O)N(CCN(C(=O)C(C)Oc2ccccn2)C(C)C)C)C(C)CCC1C C(CNC(=O)C(=O)NCC1(c2ccsc2)CC1)(CSC)OC CN1C(=O)CC(CNC(C2(NC(c3cn(C)cn3)=O)CC(CO)C2)=O)C1=O Cc1cc(NC(c2c(CNC(c3sccc3C#N)=O)nnn2C)=O)cc(F)c1 N1(C(Cc2n(C)ncc2)=O)CCC(C2CC2)C1CNC(=O)CC1CNC(=O)O1 Cc1ccc(Br)c2cc(C(=O)OCc3cnccc3Cl)[nH]c12 N1(C(CC(C)(F)F)=O)CC2(NC(C3CC3(Cl)Cl)=O)CCC1CC2 N1(C(CC(C)C2CC2)=O)CCC(F)C(NC(c2ccc(C(N)=O)s2)=O)C1 CC1CCC(NC(=O)C(=O)NCC2CCCN(CC3CC3)C2)CS1(=O)=O C=CCC(F)(F)C(=O)NC(COC)CC(=O)NC(C)CC(N)=O N1(C(C2C(OC(C)=O)C2)=O)CCC1C(=O)NOCC1(C)CC1 CCCC(C(=O)NCCC1(C(=O)NCC2CCCN2CC)CC1)OCC CC(CC(=O)NC1COCC1C(=O)NCCOCC1CCCC1)n1ccnc1 Cc1cc(NC(=O)CN2CCN(Cc3c(C)cccc3Cl)CC2=O)c(F)c(Br)c1 CC1(C)CCN(C(=O)C=C2CCC2)CC1CNC(c1coc(C2CCCC2)n1)=O N1(C(C(C)Oc2cccc(F)c2)=O)CC2CCOCC2(C(=O)O)C1 C(=O)(C(C)(C(C)C)OC)NC1CCN(C(c2cccc(SCC)c2)=O)C1 c1(C(=O)NCC2CC(NC(C3OCC(C)(C)C3)=O)C2)cncc2cc(Cl)ccc12 C1(C(=O)NC2CC(CCC(=O)NC(C3(O)CCC3)C)C2)CC2CC1CC2O C(=O)(CCCCC(=O)N1CC2CC2(CNC(=O)C(O)C(F)F)C1)OC Cc1cccc(C(=O)C(N2CC3C(NC(c4cn(C(F)F)cn4)=O)C3C2)=O)c1 CC(CC(C)NC(=O)CSc1nc[nH]n1)NC(c1cnc(-c2ccccc2)o1)=O C1(C)(CNC(c2cn(CC=C)nn2)=O)CCN(C(c2ccc(C(C)=O)s2)=O)C1 Cc1nc2cc(-c3nc(NC(C4CCC(=O)NC4)=O)c(C)s3)ccc2s1 C(=O)(CCCCCN(C(=O)CCCOCC1CC1)C)N1CCC(C)C1 Cn1cnc2c1CN(C(=O)C(O)CCCNC(c1ccc(O)cc1F)=O)CC2 N1(C(c2cccc(C)c2)=O)CCC2(CC1)CC2C(N1CCS(=O)CC1C)=O C=CCC(C)(CC=C)NC(c1occc1CNC(=O)C=CC1CCCCC1)=O N1(C(c2c(C)csc2C)=O)CCCC2(CCN(C(=O)CC3CCOC3)C2)C1 c1(C(CNC(=O)C(=O)N(C)Cc2n(CC)ccn2)OC)ccc(F)c(Cl)c1 c1(C(=O)NC2CCC(N(C)C(c3cncc(CO)c3)=O)C2)occ2c1CCCC2 c1(C(N(C2CN(C(C(CC)n3ccnc3)=O)C2)C)=O)ccc(OC(C)CC)cc1 c1(C(N2CCCCC2c2cn[nH]c2)C(=O)NC2CCC2)cccc2ccncc12 N1(C(C(CC)C)=O)CCC2(CCOCC2)C(NC(=O)Cc2nc(C)sc2C)C1 C(N=c1ccc(S(=O)(=O)N2CCC(C)(C(N)=O)C2)c[nH]1)C1(SCC)CC1 C1(CNC(C2(C)C(C)C2)=O)CN(C(C2CC(C)(O)C2)=O)CC1O c1(OC)cc(C)ccc1C(C)NCc1csc([N+](=O)[O-])c1 c1(C(N(CC(C)(F)F)C)=O)cc(CNC(=O)C(C)(C)C2CCOC2)ccn1 C(C1C(C(=O)NC2CN(C(CC(=O)N(C)C(C)C)=O)C2)C1(C)C)=C(C)C C(CC(CNC(=O)CCC=CC(C)C)NC(=O)CC1CC(C(F)F)C1)OC S(=O)(=O)(CCC(=O)N1CCCC1CCNC(=O)CC1CCC1)N(C)C N1(C(C(C(C)C)NC=O)=O)CC2CCC1CN2C(=O)C(c1ccc(Cl)cc1F)O C=C(Br)CC(C)(C)C(=O)NC1CCC(N(C(=O)CCc2cc[nH]n2)C)CC1 Cc1nc(C(=O)N(CC(c2cnn(C(C)(C)C)c2)=O)C2CC2)n[nH]1 C1(CNC(C2(CCOC)CCCC2)=O)CCN(C(=O)CCCCO)CCC1(F)F C(CNC(=O)C(C)(C)O)(CC(=O)N1CCCC1(C)C1CC1)OC C1(CNC(C2CC(=O)NC2)=O)CN(C(=O)COc2ccon2)CCC1(F)F C1(CC(=O)NC(C(=O)NCCc2cnc(C)s2)C)CCC(=O)CC1 N1(C(c2nnn(C)n2)C(=O)NCCC)CCC(Cc2noc(C)n2)CC1 n1(C(C(N2C3CC(NC(CSC)=O)(C3)C2)=O)C)ccc2ccccc2c1=O N1(C(C(C)Oc2cccc(F)c2)=O)CCC2CC1CN2C(=O)C(C)CC1CCC1 N1(C(C2CC(C#C)(O)C2)=O)CCC(C)N(C(=O)CC2CCC(=O)N2)CC1 n1(CC)c(C)nn(CC(=O)NCC(C)N(C(=O)CSc2ccccc2)C)c1=O N1(C(=O)OC(C)(C)C)CC2CCC1C(CN=c1cc[nH]cc1Br)C2 C1(C(=O)NC(C#C)C(C)C)C=CCCN1C(=O)CSC(F)(F)F c1(N(CCC)CC(=O)N)nccc(=NC2COc3ccc(Cl)cc32)[nH]1 CCC(O)CC(=O)N=c1cc(C2CCCCN2C(c2ccc(C3CC3)s2)=O)[nH][nH]1 CC1=CCC(C(=O)NC2CCC2NC(=O)C(C)(C)COC(C)C)CC1 C1(c2cn(CC)nc2)OCCCC1N(C(C1(C)CCOCC1)C(=O)NC1CC1)C C1(C(N2CC3C(NC(c4nnn(CC)c4C)=O)C3C2)=O)CCOCC1(C)C C1(OC)CC2CC(C1)N(C(C1CCCN1C(C1(CF)CC(=O)C1)=O)=O)C2 c1(C(=O)NC(C(=O)NC(CN(C)C)CO)CO)ccc(O)cn1 N1(C(CCc2c(C)ncs2)=O)CC(NC(c2cnn(CC3CCC3)c2)=O)CC(C)C1 CC1CC(=O)NC(C(=O)NCC23CC(NC(C4C5CCCC45)=O)(CO2)C3)C1 CC(C)C(O)C(=O)N1CCC(N(C(=O)Cn2cc(C3CC3)nn2)CCO)C1 C(=O)(C1=CC(C)(C)C1)NC(C(=O)NCCNS(CC)(=O)=O)Cn1cncn1 C(=O)(CCCCCn1cnnn1)NCC(CCNC(C1N(C(N)=O)CCC1)=O)O C1(C(=O)N(CC(F)Cl)C)(NC(C2C=C(C)CS2)=O)CCN(C)C1 C1(NC(CC2CC(=O)NC2=O)=O)CN(C(c2cc(F)cnc2O)=O)CCC1F C1(CNC(CCC(=C)Br)=O)CC(C)CCN1C(c1n[nH]c(CC)c1Cl)=O CC(O)C(C)C(=O)NCC(C)NC(C1(C)CCNC1=O)=O C1(CNC(Cc2c(OC)cccc2F)=O)CC12CCN(C(=O)C(C)CF)CC2 Cc1ccc(F)c(O)c1C(=O)NCC12CC1CN(C(C1CC3CC3C1)=O)C2 c1(C(=O)NCC23N(C(C4CCN(C)CC4)=O)CCC2CC3)cncc2c1CCC2 c1(C(=O)NCC2(CNC(C3CCOC3)=O)CC23CCC3)cnc(O)c(F)c1 c1(C(N(CC(CNC(C2(CC)CCOCC2)=O)O)C)=O)cccc2ncc(C)n12 N1(C(c2n[nH]c(CC)c2C)=O)Cc2occ(C(N3CC(O)CCC3C)=O)c2C1 C12(C(=O)NCC(CC(C)C)(C)C)CC3CC1C2C3(F)F n1(C(CC)CC)nc(C(=O)N(CC(O)CNC(=O)CCNC(=O)CO)C)cc1C Cc1ccccc1OC#CCc1nc(C(c2ccc(Cl)cc2)(C)C2CCC2)no1 C1(N(C(C(C)(C)SC)=O)C)CN(C(c2cccc(OCC(F)F)n2)=O)CC1(C)C N1(C(c2cccc3nc(C)nn32)=O)CCOC2(CCCN(C(=O)CCC#N)C2)C1 c1(CNC(CSCC#C)=O)ccc(C(=O)NCC2N(C(C)=O)CCC2)s1 C=C(C)C(C)(C)C(=O)N(CC(CO)(CO)NC(=O)CNS(=O)(=O)CC)C CC12CCC(CC(=O)NCc3cn(CC4CC(Cc5nncs5)C4)nn3)(CO1)C2 O=C(C#CC1CCCCO1)NC1CCC1CNC(c1ccn(CC(F)(F)F)n1)=O CC1(C)CC(NC(=O)CC2(C)CCN2C(=O)Cc2cc[nH]c2)C(C)(C)O1 Cc1c(C(=O)NC2CCCC2CNC(C2CCC(F)C2)=O)cnn1CC(C)C C12(NC(C3=NOC(C)(C)C3)=O)CN(C(=O)CCC3CC3)CC1CS(=O)(=O)C2 Cc1ncnc2c1CC(C(=O)NCC1CC(C)N(C(=O)CCOC3CC3)C1)CC2 C1(C(N(C(C2CCN(CC(C)C)C2)=O)CC)C)CCN(C(=O)Cc2ccon2)C1 c1(C(=O)NCCCN(C)C(C2CC23CCCOC3)=O)cncc2c1CCCC2 c1(CNC(CCCOC)=O)ccc(CCNC(C2OC3CCC2C3)=O)cc1 CC(C)C(O)(C(=O)NC1CCN(C(=O)C(C2CC2)C2CC2)CC1)C(F)(F)F c1(CN(C(=O)CCc2ccncc2)Cc2ccccc2)ccc(Br)cc1 C1(C(=O)NCC2C(NC(c3cocc3Br)=O)CC2)CCCCO1 CCCC(C(=O)N1CCC(Nc2ccc([N+](=O)[O-])cc2)C1)C(C)C c1(C(=O)NCCC(C(C)C)NC(C2(CC=C)CC2)=O)cc2c(F)c(F)ccc2[nH]1 CCN=C(NCCN1CCCC1)NCc1cc(C)no1.C12CC1C2 C1(C(N(CCC(C)C)NC(C(CC)C)C)=O)CCN(C(c2cncs2)=O)CC1 c1(C(N(CC(=O)N(CC(C)NC(CN(CCOC)C)=O)C)C(C)C)=O)ccsc1 C(=O)(CC1=CCCC1)NCCc1cc(C(N(CC(C)OC)C(C)C)=O)no1 N1(CC)CC(C(=O)NCCC2CCN(C(=O)Cc3cc[nH]n3)CC2)CCC1=O C(CC(O)C(=O)NCC(C(C)C)NC(c1ccc(-c2csc(C)n2)cc1)=O)SC C(=O)(C(C)(C)CCC#N)N(C(C(=O)N(CCCO)CC)C)C1CC1 c1(C(N(C)CC2OCCN(C(CCC#C)=O)C2)=O)cc(F)cc2ccccc12 N1(C(C(c2ccnn2C)C)=O)CCC(NC(c2cc(C3CC3)ns2)=O)C(F)C1 Cc1cc(C)c(C(N2CCN(C(c3cc4cccnc4s3)=O)CC2)=O)c(N)c1 C1(NC(C(C)=CC)=O)CC(OC)CN(C(C2(C(F)(F)F)CCCCC2)=O)C1 C1(CC(=O)NCC2C(CNC(C(Cn3ccc(C)n3)C)=O)C2)CCCCN1C c1(CC)nc(C)c(C(=O)NC(C)CC2CCN(C(C3CC(C(F)F)C3)=O)CC2)o1 N1(C(c2onc(CC)n2)=O)CCC(F)(F)C(CNC(=O)C(CC)N(C)C)C1 C1(C(N(CCCNC(=O)C(C)(C)OC)CC)=O)Cc2cc(Cl)ccc2C(=O)O1 CCCCC(O)CC(=O)N1CCCC(C(N2CCC(C)(CN(C)C)C2)=O)CC1 C1(C(N2C(c3n(C)cnc3)CCC2)=O)(C(=O)O)CC(F)(F)C1 c1(C(=O)NC(COCC)C(=O)NC2CCCC2(F)F)ncncc1Cl N#Cc1nc(Br)cnc1NC(C1CC1NCc1ccc(Br)[nH]1)=O C1(C(=O)OC)CCSC12CN(C(=O)NCC1(C)CCCC(F)(F)C1)C2 n1(CC(N2CC(NC(C3CN(S(C)(=O)=O)C3)=O)C2)=O)cc(C(=O)N(C)C)nn1 c1(CCCC(=O)NCC(CNC(C(CCC)(C)O)=O)CO)csc2ccccc12 c1(CNc2ccc(NC(c3c(C)ccs3)=O)cn2)cc2ncccc2[nH]1 C1(NC(c2c(C)nn[nH]2)=O)(CNC(=O)Cc2ccc(F)cc2)CCCCC1C N1(C(c2c(CC)non2)=O)CC2(C)CC1(C(=O)NC1CCN(CC)C1=O)C2 N1(C(CN(C(=O)OC)C)=O)CC2=C(C1)CN(C(=O)Cc1ncc(Cl)s1)C2 C#CCCN=C(NC1CC(C)(OC)C1(C)C)N(C)Cc1cccc(C(F)(F)F)c1 C(c1ccc(C#N)cc1)=CC(=O)NCC1C(NC(C2(C)CCC2)=O)CCCC1 c1(CN(CC(C)(C)OCCO)C)ccc(C(=O)NC(C2CCC23CCC3)=O)cc1 C=CC1(CNC(C2(COC)CN(C(=O)C(F)CC3CCOC3)C2)=O)CCC1 c1(OC)cccc(C=CC(=O)NCCC(C)(C)NC(C2CC2F)=O)c1OC c1(-n2c(-c3c(Cl)cnc(CC)n3)nc(-c3occc3C)n2)ccc(CC)c(Cl)c1 c1(OC)ncncc1NC(C1CC1C(=O)N(C1COC1)C(c1ccccc1)=O)=O C1(NC(=O)C(F)CC2CN(C(=O)Cn3ccccc3=O)C2)CCn2ccnc2C1 N1(C(=O)NC2CN(CC(F)(F)F)C2)CCC2(C1)c1[nH]cnc1CCN2CC1CC1 c1(C(=O)OCC(=O)N(C2CC2c2ccccc2)C)ccccc1SC(F)(F)F c1(C(N(C)CCc2nccs2)=O)conc1CNC(=O)C(O)C1CCCC1 CCCCC(C)CCC(=O)NC(c1ccccc1)CNC(=O)CS(=O)(=O)CCO C1(NC(C(CC=CC)C)=O)CCC12CCN(C(=O)COc1cccc(F)c1)CC2 N1(C(CCC=CCC=C)=O)CC2CC(NC(=O)C(CC)NC(N)=O)CC1C2 C1(F)(C(=O)NC(C2N(C(c3c(C)nc[nH]3)=O)CCC2)C)CCN(C)CC1 C1(C)(C(N(C(C)CNC(c2cc3n(c2)CCCC3)=O)CC)=O)CC(C(C)C)=NO1 N1(C(C(CC#C)(C)NC(=O)CC2CC(C(=O)OC)C2)=O)CCC(C)C(F)(F)C1 C(C(COC)CC(=O)N1CC2(C)CC1(C(=O)NCCC1CCCCC1O)C2)OC c1(C(=O)NCC(CNC(C2(CC#N)COC2)=O)O)cnn2c1CCC2 C1(C(C)Sc2cccc(F)c2)CCN(c2nnc(SC)s2)CC1.C12CC1NC2=O Cc1cc(F)cc(C)c1C(N1CC(NC(c2ccc3ccsc3c2)=O)C(C)C1)=O c1(C(N2CC(C)(NC(C3C(C)C3)=O)C2)=O)cnc2c(cnn2C)c1 C1(NC(c2cc(Cl)cs2)=O)CCN(C(=O)C=Cc2cncc(O)c2)CCC1CO c1(C(N2CCCC(CN(C(C3CCN(C)C3)=O)C)C2)=O)cc2ccsc2n1C c1(C(=O)NCCC2OCCN(C(c3c(C)oc(CO)c3)=O)C2)ccnc(O)c1F C1(CNC(c2cc(CC)n(C)n2)=O)COCCN(C(C2C(F)(F)C23CC3)=O)C1 c1(C(N2C(CN(C(=O)Cc3ccsn3)C)CCC2)=O)ccc2c(c1)C=CCC2 N1(C(c2nc(C)[nH]n2)=O)C2CCC1CN(C(C1CCCC(F)C1)=O)C2 CN1CCN(C(=O)C(c2cscn2)NC(=O)CN2CCOC2=O)C(CCO)C1 c1(C(=O)NCC2CC(NC(CCc3ncc(C)[nH]3)=O)C2)cc(N)nc(Br)c1 CCC(C)CCCC(=O)CNC(=O)CC1(O)CC1.C12CC(C1)C(=O)NCC2 C1(NC(C2CC(C)(F)C2)=O)CN(C(c2cc(F)cc(F)c2)=O)CC1C1CC1 CC1(C(=O)NCC(C2CCC2)NC(c2cccc(C#N)c2)=O)CC2CCC1O2 c1(C(CF)NC(=O)NC(C(CC)C)CO)cccc2ccccc12 C1(C(=O)NCc2ccoc2C(=O)NC2CC(O)(CO)C2)(OC)CCSC1 C(c1ccccn1)=C(C(=O)NCC(CNC(c1cscc1Cl)=O)OC)C CC(C)CCC(F)C(=O)NC1(C(=O)NCC(c2ccsc2)C)CC(F)C1 CC1=NOC(C)(CNC(C2CC[Si](C)(C)C2)=O)C1 C1(C(=O)NCC2(C3CC3)CC2)COCCN1C(=O)CC1CCC2CC12 C1(C(=O)NCCN(CCCCCC)C(c2sc(C)cc2C)=O)CN(C)CCO1 Cc1ncnc(N2CC3C(CNC(=O)CSCc4ccncc4)C3C2)c1C#N C(CCC)(C(=O)NC1CCCC1NC(=O)CSc1ccc(OC)cc1)=CCC C1(N)(C(N2CCCC(C(=O)NCCC)C2)=O)CC(O)C1(C)C C1(NC(c2n(CC#C)ccc2)=O)C2CC(O)C1N(C(c1cnc(SC)n1C)=O)C2 c1(CC(=O)NC(C)(C)CNC(=O)CC2CC3(CC3)CO2)cnc2ccccc2c1 N1(C(=O)Cc2ccsc2)CCC2CN(C(c3c(Cl)cncc3Cl)=O)CCC2C1 C1(CC)CN(C(=O)Cc2ccco2)CCC1CNC(=O)CC1CC1 N(C1CCCc2cc(CNC(C3C=CCCC3)=O)ccc21)C(c1ccc(C)s1)=O C1(CC(=O)NCCOCCC(C)C)CC2(CC2)CN1C(=O)CC1CCOCC1 C1(n2cc(CNC(c3cnn[nH]3)=O)nn2)CCCN(C(C2(C(F)(F)F)CC2)=O)C1 C1(C(=O)NCc2nc[nH]n2)(COC)CN(C(=O)CC2CCSC2)C1 Cc1nc2cc(C(N3CC4(C3)SCCC4NC(=O)C(C)C3CC3)=O)cnc2[nH]1 C1(C(N2C(C)(C(=O)NCCn3cc(CO)nn3)CCC2)=O)CC2C=CC1CC2 C1(C(N2C(C(N3CC(N=[N+]=[N-])C3)=O)CSCC2)=O)CCC2(CC1)CC2 c1(C(=O)NCC(CN(C(CCc2c(C)nn(C)c2)=O)C)C)[nH]ccc(=O)c1C c1(C(=O)NCCC(C)CCNC(C2C=CCC2)=O)cc2ccc(F)cc2cn1 C1(C(=O)NCC2C(C(=O)NCCSCC=C)CC2)CC(=O)NC(=O)N1 c1(OC)cc(C(=O)NCC(O)CN(C(=O)Cc2cc(C)sc2C)C)cc(F)n1 C(=O)(C1=CC2CCCCCCC12)CC(C)CNC(=O)CNC(c1ccncc1)=O N1(CCNCC(=O)Nc2cnc(C)s2)CCC(C)CC1 c1(SC)c(C(=O)NC2CC(F)CN(C(c3cc4n(n3)CCO4)=O)C2)cccc1F C(C(=O)N1CCC1CF)(c1ccoc1)NC(=O)C=CCO Cc1nnccc1C(=O)NCCC1CCCN1C(=O)C(C)C(=O)OC(C)(C)C c1(OC)ccc(C(=O)NCC2CC(NC(=O)C3=CSCCO3)C2)cc1F C1(CNC(=O)CCOCC2CCCO2)CCCCN1C(C1CCCSC1)=O CC(CC(C)(F)F)C(=O)NC1(c2ccccc2)CCN(C(=O)Cc2nc[nH]n2)C1 C1(CN(C(c2ncsc2NC)=O)CC)CCCCN1C(c1cc(C(C)C)[nH]n1)=O CC(CC(F)(F)F)C(=O)NC1C2CC3C1C3C2C(N1CCCCC1CCCO)=O C(=O)(CS(=O)(=O)CCCc1ccccc1)N(C)CC1CN(C(CCC(=C)Cl)=O)C1 N(C1CN(C(=O)C=CCF)CCc2ccccc21)C(c1nnc(C)s1)=O c1(C(=O)NCC2CCCC2NC(=O)C(F)(F)C(F)F)ccc(O)c(F)c1F C(CCC(C)C)(C(=O)NCC1(N(C)C)CC1)NC(c1nc(C)c(C)s1)=O CN(OC1CCCC1)C(=O)C1CCN1C(C1C=CCCC1)c1ccccc1 Cc1cn(CC(=O)N(C(C)CN(C)C(C2(C)CCC(=O)NC2)=O)C)c(=O)nc1O CC1(C)CN(C(C2C(Cl)(Cl)C23CC3)=O)CC1NC(c1c[nH]c(Br)c1)=O CC(C)(CN(C(c1cn(C2CCCC2O)nn1)=O)C1CC1)CO CC1NC(=O)CCC1CNC(=O)C(CN=[N+]=[N-])NC(c1cncn1C)=O C(=O)(CC(O)CCSC)NC(CCCC)CNC(c1ccc(C)cn1)=O C1(C(=O)NCC(=C)C)CCCCCC1NC(c1cc(C)cc(C)n1)=O Cn1cnc(N2C3CCC2C(C(=O)N(C(c2nccs2)=O)C2CC2)C3)c(Br)c1=O CC1CN(C(=O)C=CC(N)=O)CCC1NC(c1cc(C2CC2)cs1)=O C(=O)(C(O)CC[S+](C)C)N(C1CCC(NC(c2nc(CCC)oc2)=O)CC1)C c1(N(C(CNC(C(C)c2ccsc2)=O)C)C)nc(Cl)c(C#N)s1 N1(C(C2(C(C)=O)CC2)=O)CCC(NC(c2cccc(C(N)=O)c2)=O)C(C)C1 C1(NC(C(CCC=C)NC(=O)Cc2cnn(C)c2)=O)CCn2nnnc2C1 C(=O)(C1CCCc2nnn(C)c21)N(C)CCC1CCCCN1C(=O)C(N)=O C#CCCC(C(=O)NCc1ccco1)NC(c1cc(Cl)ns1)=O Cc1nc(C(=O)NCC(C)(CO)NC(C2CCCCC(=O)N2)=O)ccc1Br CCC(C)(CO)C(=O)NCCC1CN(C(c2cc(C)nc(OC)n2)=O)C1 c1(NC(CCC(=O)N(C)Cc2csc(CO)n2)=O)ccc(F)c(F)c1 C(c1c(Cl)ccc(Cl)c1Cl)=CC(N1CC2CCN(C(C=CSC)=O)CC21)=O c1(CNC(c2ccc(Br)cc2Cl)c2n(CC)nnn2)cccc2c1CCS2(=O)=O C#Cc1cc(C(N2CCN(C(=O)Cc3cccc(F)c3)CC(C)C2)=O)ccc1C O=C1OC(C(=O)NC2CN(C(=O)C=CI)C3(CCOCC3)C2)Cc2ccccc21 c1(SC(C2CCC2)(C)C2CC2)csc2ccc(F)cc12.n12cc(nn1)CN(C)CC2 C1(CNC(=O)Cc2cc[nH]n2)(CO)CCN(C(C2CC(O)C2)=O)CC1 C1(C(=O)NC2(C)CCC(NC(CC=CC)=O)CC2)Cc2cccnc2C1 C(CCSC)(C(=O)NC(C)CNC(=O)CS(C)(=O)=O)OC CC(CC(=O)N1CCC(CF)(NC(=O)CC=CCc2ccccc2)C1)C(C)(C)C c1(N(CCC(N2CCC(N(CC#C)C(C)=O)C2)=O)C)ccccc1O C(=O)(CCCCCC#N)N1CCC1CNC(c1cccc(N2CCC(C)C2)c1)=O c1(C(N2CC(C)C(NC(=O)C(C)(C)CF)C2)=O)cn(C)c(=O)cn1 C1(CNC(C(CC2CC2)NC(C(C)SC(C)C)=O)=O)CC2(CC2)C(=O)O1 c1(NC(CC)CC#N)[nH]c(=NC2CCN(CC3CC3)CC2)nc2scnc12 c1(CC(=O)N(CCNC(c2c(Cl)ccc(CC)c2)=O)C)ccc2c(c1)COC2 c1(OC)ncc(C(=O)NCCCCC(C)NC(=O)C(C)Cn2ccc(C)n2)cn1 N1(C(CCC)=O)CCCC2(CCN(C(=O)C(c3cccc(OC)c3)O)C2)C1 Cc1noc2ncnc(N3CCC(C)C3CNC(=O)CN3CCCS3(=O)=O)c12 C1(CC)(NC(=O)CC2CN(Cc3ccc(O)cn3)CCO2)CCOCC1 N1(C(C#C)=O)CCCC(C)(C(=O)NC2CCC(n3cccc3)CC2)C1 Cn1nc(C(=O)NC2CC(F)CN(C(C3CC3(F)F)=O)C2)c2cc(F)ccc12 Cc1cc(C(=O)NC(CCOCCO)C(=O)N2CCOCC2CCO)cc(C)n1 CN1CC(C(N2CCC(NC(=O)C(C)(C)C(=O)OC(C)(C)C)CC2)=O)CCC1=O C1(N(C(c2ccc(OCC)nc2)=O)C)CCCN(C(c2sncc2CC)=O)CC1 CCN=C(NCC1CN(Cc2ccc(F)cc2)CCO1)NCC1CCCCCC1 n1(CC(C)(C)CO)nc(-c2ccc(Cl)s2)nc1-c1c[nH]ccc1=O Cc1cc(C(=O)N(CC(C)N(C(=O)CCC2CCC(=O)NC2)C)C)n(C2CC2)n1 C12(NC(=O)Cn3ncnn3)CCN(C(c3cc4ccccn4n3)=O)CCC1C2 c1(C(N(CCCN(C(C(C(C)C)NC(C)=O)=O)C)C)=O)ccc(C#N)c(O)c1 C1(NC(=O)C=CCO)CCC(NC(C2CC23CC(O)C3)=O)CC1 CON(CCC(=O)NC1CCCCC1N=[N+]=[N-])C(=O)c1cc(Cl)cs1 c1(OCCC#C)ccc(C(=O)NCC2CC2NC(=O)Cc2noc(C)n2)cc1 C(C)(CCC(=O)NCC(C)(C)OCCNC(=O)C(c1cccc(Cl)c1)C)OCC C(=O)(CCCS(C)(=O)=O)NCC1C2CN(C(C3(COC)CCCCC3)=O)C1C2 c1(OC)ccc(Cl)c(CC(=O)NC(C)(C)CNC(=O)CC(=O)NCC2CC2)c1 C(=O)(CCCS(C)(=O)=O)N1C(C)CN(C(=O)C(C)(O)C2CCC2)CC1 C1(CNC(c2ccc(C(C)=O)[nH]2)=O)CCCC1NC(c1ccnn1CCF)=O CS(=O)(=O)C1(C(=O)NC2CCC(NC(c3cc(C(F)(F)F)ncn3)=O)C2)CC1 C1(C(=O)NC(C)CCc2cn[nH]c2)CC(C)(C)CCN1C(c1csc(Cl)n1)=O C1(OCC)CCN(C(=O)CC2CCN2C(c2cc(C)sc2C)=O)CC1 C=CC1(CC(=O)OC)CN(C(=O)NC(c2ccccn2)C)C1 c1(C(=O)NCC(C)N(C)C(C2OC(C)(C)OC2(C)C)=O)ccc2c(n1)COCC2 C1(N(C)C(c2ccc(C(C)(C)C)[nH]2)=O)CN(C(=O)COCCN(C)C)CC1(C)C O=C(C1=COc2ccccc2O1)NCC1CC(O)CN1C(=O)Cc1ccc(Cl)s1 Cc1ccc2nc(SCC(=O)NC3CCCC3N(C)C)[nH]c2c1.C12(CC1)C(=O)N2 C1(C(=O)OC)CCN(C(C23CCCC2CC(F)(F)CC3)=O)CC12CCC2 c1(C(N2CCN(C(C3CC(CCC)OCC3)=O)CC2C)=O)cc2cccnc2[nH]1 N1(C(CN(C(COC)=O)C)=O)CCC(NC(c2cnc(O)n2C)=O)C1C(C)(C)C c1(C(=O)NCC(CNC(=O)CN(C(=O)C(C)C)C)OC)ncsc1Br c1(C(=O)NCC2CCN2C(c2cc(F)cc(Br)c2)=O)coc2c1CCCC2 C(C(C(=O)N1CC(N2CCCCC2)C1)NC(=O)Cc1nocc1C)OCC c1(C(N2CCCC(N(C(=O)C(F)OC(F)(F)F)CCF)C2)=O)ccc2nsnc2c1 C(=O)(C#CC(C)(C)C)NC(CCOC)C(=O)N1CC(NC(N)=O)C1 C(=O)(C(=O)CC(C)C)NCCCC(=O)NC(CC)Cn1cncn1 n1(CC(C)C2CC2)nc(-c2ccoc2)nc1C1CC1C#N N1(C(c2cc(Cl)ccc2F)=O)CCC2C1CCN2C(=O)C(F)F c1(C(N(CCC)CCNC(C2CC2(C)C)=O)=O)cc(=O)c2ccccc2[nH]1 C(=O)(C(COC)CC(C)C)N(CCC)CCNC(C1(NC(C)=O)CCC1)=O CC1CN(C(=O)CC2(C(F)(F)F)CC2)CC1NC(=O)Cn1cc(Br)cn1 CCCCC(O)CC(=O)N1CC=CC1C(N1CC(C)(C#N)C1)=O C1(NC(c2nc(C(N)=O)sc2)=O)CN(C(=O)CC2CC(=O)C2)CCC1O N1(C(C2CN(S(CC)(=O)=O)C2)=O)CCC2CCCN(C(=O)COCCOC)C2C1 C1(CCC(=O)NCCCN(C(CC2CN(C(C)=O)C2)=O)CCO)CC(C)(C)CO1 c1(COC)cccc(-c2cn(CC3CN(C(c4cnc(O)o4)=O)CCO3)nn2)n1 c1(NC(=O)NC(C)C(c2ccc3c(c2)OCO3)O)cc(C#N)cc(Cl)n1 C1(CNC(C2(F)CCC2)=O)CC2(CCN(c3ncnc4sccc34)C2)CO1 CCCC(C(=O)NC(C)CN(C)C(C)C)NC(c1cc(CC)sn1)=O C1(C)(CCNC(C(CC=C)OC)=O)CCN(C(c2cc(F)c[nH]2)=O)CC1 c1(C(N(C)CC2CCCN2C(c2ncc(N)cc2Cl)=O)=O)cc2c(o1)CCCC2 c1(C(N2C(CCNC(=O)COc3cccnc3)CCC2)=O)nnn2c1CSCC2 c1(CC)cc(-c2nc(CC(C)OC)nn2CC2(C)CCOCC2)n(C)n1 C(CCN(C(=O)COc1ccc(SC)cc1)C)(C(C)C)NC(CC(=O)NC)=O c1(C(=O)NCC2N(C(CN(C3CC3)CC)=O)CCOC2)cc2c(cn1)COCC2 N1(C(c2cn(C)nc2)=O)CCC(C)(CNC(=O)CC2C=CS(=O)(=O)C2)C1 n1(CC)ccnc1C(=O)NCCC1(C(=O)NCCNCCCSC)CCC1 CC1CN(C(c2csc(C(C)(C)C)n2)=O)CC1CNC(=O)CN1CCC(O)CC1 CCC(F)(F)CC(=O)N(C)CC1CCCN(C(c2cccc(C(=O)OC)n2)=O)C1 c1(CNC(CCN(CC#C)C(C2CCOC(C)C2)=O)=O)ccc(F)c(C)c1 CC1C(NC(=O)C(c2ccc(F)cc2)F)CCN1C(=O)C1CC1 C#CCCC(O)C(=O)NCCc1ocnc1CNC(=O)CC(C)(C)OC CC(C)CC(C(=O)NCC1CC(C)CN(C(=O)C(N2CCNC2=O)C)C1)C(C)C N1(C(c2c(Cl)ccc(OC)c2)=O)CCC2(CC1)CC2C(N1CCOC(CO)C1)=O C1(CNC(N(CCn2c(C)ncc2)C)=O)C2CCCCC12 CCCC(C(=O)NC(CO)CCO)NC(=O)CC1(COC)CC1 c1(C(N2CC3C(CNC(C4CC45CCC5)=O)(C3)C2)=O)ccc(F)c2ccncc12 Cc1ccc(CC(N2CCC(NC(=O)C(C)C(C)C)C2C(C)(C)C)=O)cn1 C(=O)(C1Cc2ccc(F)cc21)N1CCC(NC(c2n[nH]c(CC)c2[N+](=O)[O-])=O)C1 N1(C(C(C2CCOCC2)C)=O)CCN(C(c2cc(Cl)ncc2N)=O)CC1C Nc1c(C(=O)NCCN(C(C2CN3CCC2C3)=O)CC2CC2)cc(Cl)cc1F C1(N(C(=O)C=CSc2nc[nH]n2)CC)CCN(C(c2cc(Cl)no2)=O)CC1 Cc1nc(C(=O)N(C2CCCC2)CCNC(=O)C=C2CCC(C)CC2)c(C)s1 C(=O)(CCCC(=O)NCC1CCC1NC(=O)CN1CC=CC1)c1c(N)cccc1 C(=O)(C1=C2CCCN=C2NN1)N1C(C2(NC(CC=C)=O)CC2)CCC1 C1(n2cc(CC=C)nn2)CC2CCC1(NC(C1CC(C)=NO1)=O)C2 N1(C(CNC(CC)=O)=O)CCc2nc(CNC(=O)CCOCC3CCC3)sc2C1 C1(C(N(C)Cc2onc(C(C)OC)n2)=O)CNCc2nccn2C1 c1(N(CC(C)NC(CSc2c(OCC)cccc2)=O)C)ncc2cccnc2n1 C#Cc1cnc(C(N2CCC(O)CC2C(=O)N(C)CCSC)=O)c(C)c1 c1(CC)cnoc1C(=O)NC(C)(C)C(=O)NC(C)CCn1cncn1 c1(C(=O)NC2CCC(CNC(CC3(OC)CC3)=O)C2)cnc2nc(C)[nH]n2c1=O N1(C(c2c(CC)nc[nH]2)=O)CC2CCN(C(=O)CN3CCCCCC3=O)CC2C1 Cc1cc(C(=O)N(C2(C(=O)NC3CCOC3)CC2)C)nc(C)n1 c1(OC)ccc(C(=O)NCCN2CCN(C(=O)C(C(C)O)NC(N)=O)CC2)nn1 CCCCC(F)C(=O)N(CCC(C)(C)NC(c1cncnc1C)=O)C c1(C(=O)NCCN(C(c2cncc(C)c2)=O)C)cc2c[nH]nc2s1 c1(CC)nccnc1C(N1CCN(C2CCN(C(C3CC(=O)N3)=O)CC2)CC1)=O c1(C(=O)NC2C3N(C(C(C=C=C)C)=O)CC(CC3)C2)nn2ccccc2c1Br C=CCC(C)(C)C(=O)NC1CC2(NC(c3ccc(O)nn3)=O)COC1C2 CCCCS(=O)(=O)NCC(=O)N(CCCNC(=O)C=CCO)C(C)C c1(C(N2CCN(C(=O)CSC(F)F)CC2CO)=O)cncc([N+](=O)[O-])c1 N1(C(C2CCCCN2Cc2ccc(-c3ccccc3Cl)o2)=O)CCOCC(O)C1 C(=O)(CCC(C)(C)N(C)C)NC(CCN(C(CCC(=O)NCCC)=O)C)C c1(C(N2CCC(O)(C(C)NC(C=CC(C)C)=O)CC2)=O)cccc2c1C(=O)CC2 c1(C(=O)NC2CC(F)(CNC(C(CC)(C)C(F)F)=O)C2)ccc2c(c1)CCN2C S(=O)(=O)(c1ccc(F)cc1F)NC1CCCN(C)C1 C1(NC(c2cnc(CC)s2)=O)CCC2CN(C(=O)Cc3nonc3C)CCC2C1 N1(C(C(CC)(C)CO)=O)CCC2(C=C(C(=O)N(C)Cc3ccncc3)C2)C1 c1(NC2(CNC(CC3CC(C)(C)OC3)=O)CCCCC2)ccccc1[N+](=O)[O-] Cc1cccc(CCC(=O)N(CCCNC(C2(C)CC=CCC2)=O)C)c1 c1(C(=O)NCC(CNC(C(CCCC)(C)F)=O)C)c[nH]c2ccc(Cl)cc2c1=O n1(CC)c(N(CC2CCCN2C)CC2(c3cccc(Br)c3)CCCC2)nnc1C c1(CC)ccc(C(=O)NC2CCC(C)(CNC(c3[nH]c(C)nc3C)=O)C2)cc1 c1(C(=O)NCCC2(C(N3CC(O)(CC=C)C3)=O)CCC2)ccc(F)c(C)c1 c1(COC)nc(OC)cc(NC(CCNC(=O)C(F)CC2CCCC2)C(C)C)n1 c1(-c2c(OCC(=O)OC(C(C)C)C(=O)N(C)C)cccc2)ccc(F)cc1Cl C1(NC(=O)CC2CC2)CCN(C(=O)COc2ccc(F)cc2Cl)CC1F c1(CCNC(C)C)nc(C)sc1Br.C1(SC)C2CC3C(C2)C13 C1(NC(C(COC)C)=O)CCCN(C(=O)C=Cc2scnc2C)C1C Cc1nc2c(C(=O)NC3CCC(NC(C4CC4(F)Br)=O)CC3)cccc2o1 CC1CCC(C)(C(=O)NCC=C2CCN(C(=O)CCSC3CCCC3)CC2)C1 CCCC(C)(O)C(=O)N1CCN(C(=O)C=Cc2cc[nH]n2)C(C(C)C)C1 C(C)(CCC(=O)NC(C(=O)NCc1cnn(C(C)C)c1)C(C)OC)OCC C(C(C)(C)CC1CN(C(c2cnn(CCO)c2)=O)C1)NC(C(C)OCC1CC1)=O Cc1cc(C(=O)NCC2CN(C(c3cn(C4COC4)nn3)=O)CC2O)ncc1F N1(C(C(C2CCN(C(C3CC3F)=O)CC2)C)=O)CCN(C(C)(C)C)CC1 C1(c2n(CCNC(C3C4COCC34)=O)nnn2)(N2CCCC2)CCCC(F)(F)CC1 C#Cc1ccc(CC(=O)NCC(CC2CC2)C(=O)NC(CO)CCF)cc1 C1(C(=O)NCCOCCC)CCCCN1C(C1(C)CC1(C)C)=O c1(C(N2CCC(CNC(COCCC(C)C)=O)C23CC3)=O)cnc([N+](=O)[O-])n1C CC1CCCCC1CC(=O)N(CCCNC(=O)C(C1CCCCCC1)(C)C)C C=Cc1cnn(C)c1C(=O)NCC1CCN1C(=O)C(C)Oc1cccnc1 c1(C(=O)NCCCOCCNC(CC(=C=C)C)=O)ccc(C2CC2)nc1O CN1CCC(C2(C(=O)N(CCNC(=O)C(C)(C)CC(F)(F)F)C(C)C)CC2)CC1 CCC(C)(CN(C(=O)Cc1cccs1)OC(=O)CC)C(C)O O=C(N=c1cc[nH]cc1Cl)C1CC1NCc1ccc2sccc2c1 C1(CC(=O)N(C2CC(C#N)C2)CC(=O)NCC(C)CO)CCCNC1=O C1(N(C(C(c2ccc(O)cc2)C)=O)C)CCN(C)C1=O c1(OC)ccc(F)c(CN2CCCC2C(=O)NCc2cc(C#N)ccc2Br)c1Br C1(C(N2CC(N3CCC3)C2)=O)CN2CCC1C2.N12CC(O)(C1)C(F)C2=O CS(=O)(=O)c1sccc1C(=O)NC1CCCN(C(C2C3CC4C(C3=O)C24)=O)CC1 C(=O)(N=c1[nH]onc1C1CCC1)NCCCC(C)O C1(CC(N2CCC(CC#C)(C(=O)OCC)C2)=O)CC(=O)c2ccccc2C1 c1(C(=O)NC(C2CCN(C(=O)C(O)C3CCC3)CC2)C)ncc(Cl)cc1F CC1(C)CC(O)CCN(C(c2nc(C3CC3)cs2)C(=O)NCc2cccs2)C1 c1(CN(C(c2coc(C3CCNCC3)n2)=O)CC)cccc(C)c1 N1(C(c2cccc(CC)c2)=O)CCC(N(C)C(c2ocnc2C2CC2)=O)C(C)C1 Cc1c[nH]c(C(=O)N(C(C)CC(=O)NCCC2CCCOC2)C)c1 C1(NC(c2c(C)occ2)=O)CCCCCC1NC(=O)C=C(C1CC1)C1CC1 CC1=C(C(=O)NC2CCCC(NC(C3CC4(C3)CC4F)=O)C2)CCC1 C(=O)(C#CC1(CC)COC1)N1CC(C(=O)NOCCOCCOC)(CC)C1 N1(C(C2(CC)CCCC2)=O)CCC(N(C)C(c2ccnn2C2CCC2)=O)C(C)C1 C1(NC(CNC(CCn2c(C)ncc2)=O)=O)CCOCC1OC(C)(C)C c1(C(=O)NC2CN(C(C3C(=C)CC3)=O)C(C)CC2)ccc(=O)n2c1CCCC2 c1(C(=O)NC(CNC(C(c2c(C)nn(C)c2)O)=O)C2CC2)sc2nccn2c1C c1(SC)ccc(Cl)cc1NC(c1sccc1I)c1nnnn1C(C)C CCC(F)(F)C(C)(C)C(=O)NC1CC(CNC(c2coc(CS(C)(=O)=O)n2)=O)C1 CCC(C)(C)CCCC(=O)NC1CCC(NC(c2n[nH]c(C)c2F)=O)C1 C(CC(F)F)(C(=O)NCC(C)(C)CCC=C)NC(CCOCC#C)=O C(=O)(C(C)(O)C(C)C)NCC(C)CN(C)C(C1(C(F)F)CC(F)(F)C1)=O CCCCC(CNC(C1(F)CC1(Cl)Cl)=O)NC(=O)C(C1CC(F)(F)C1)O C1(C(=O)NCC(C)(C2CC2)NC(=O)CCn2cnnn2)CC2(CCOC2)C1 c1(CC)cnoc1C(=O)NCC(C(=O)NCCNC(=O)NC)C1CCOC1 C1(O)(CN(C(c2cc(CC)[nH]n2)=O)C)CCCN(C(=O)CC(C)C2CCCC2)C1 C1(C)(C(=O)NC(c2ncc(C)cn2)C)CC(O)CN1C(=O)CCc1ncccn1 CCC(CC(=O)NC(Cc1ccccc1)CCNC(c1cnccn1)=O)C1CC1 C#CCC(CC(=O)N(CC(C)CCC)C)NC(=O)CCc1ccccn1 C1(C(C)(C)C)CN(C(c2ncccn2)=O)CCN1C(C1CC(C2CC2)C1)=O C(C(C)(O)CC(=O)NC1CN(c2cc(C(C)C)nc(C)n2)CCC1C)OC C1(C(=O)NC(CC#C)CO)(CNC(=O)COCCN(C)C)CC(C)(C)C1 C1(C(=O)NCC(C)(C2CCC2)NC(C(CCC)O)=O)Cc2nnsc2S1 N1(C(CCCC(C)C)=O)CCC(N=[N+]=[N-])(C(=O)NCc2cncc(F)c2)C1 N1(C(=O)CC(=O)CC2CC3CCC2C3)CCCC(CN2CCC2CO)C1 C1(C(=O)NCC(C)NC(=O)Cc2ccc(F)cc2Cl)C2CCC3(COC(=O)C13)O2 N1(C(Cn2cc(CNC(=O)CCC3CCOC3)nn2)=O)CCCCC1CCCO C(c1ccc(N2CCCC2=O)cc1)=CC(N1CC(O)(C(Cl)(Cl)Cl)C1)=O CC(CCNC(=O)C(O)C(C)(C)C)N=c1[nH]c2ccc(Br)cc2o1 C1(CC(=O)NC(CCNC(C(C(C)C)C#N)=O)(C)C)CCC2CC1C2(C)C c1(C(=O)NC2CC(CCNC(COCCC#C)=O)C2)ccc(S(=O)C(C)C)cc1 Cc1cnc(C(=O)NCC(C2CCC2)NC(C23CCC(C2)C3)=O)cc1Br c1(C(=O)NCC(CC)(CC)NC(C2C(CC)C2)=O)cn2c(n1)CCCC2C C1(CNc2cc(OCC3CCCC3)ccc2)CNCC12CCOCC2 c1(CC(C)C(N2CC3(NC(c4cc(Cl)no4)=O)CCC2C3)=O)ccc(F)cc1F c1(-c2c(C)nn(C)c2)cccc2nc(C(=O)Nc3ccn4ncnc4c3)cn12 C(C1=NOC2(CCC2)C1)NC(C(C1CN(C(c2ccn(C)c2)=O)C1)O)=O CC#CCCCC(=O)N1CCCC(C)C1CNC(C1(c2cccnc2)CCC1)=O C(=O)(CCCC(=O)C1CC1)NC(CNC(CC1(OCC)CCC1)=O)(C)CO C(=O)(C(C)(C)CC(F)F)N1CC(C)C(C)(CNC(c2ccoc2)=O)C1 N1(C(CC)=O)CCC(N(C)C(c2csc(C)n2)=O)CC1 CCC(C)(C)CC(=O)N(C)C(c1ccccc1)c1nnco1 Cc1nn(C(F)F)c(C)c1C(=O)Nc1cnn(-c2ccccn2)c1C N1(C(C(C)(C)C2CCCC2)=O)CCC(CO)C(NC(=O)CC2CC(F)(F)C2)C1 c1(CNC(CCC2N(C(Cc3cc(C)on3)=O)CCCC2)=O)ccc(C)c(O)c1 Cn1cc2c(n1)CCC(C(=O)NCC1CC(F)CN1C(=O)C1CC1)C2 C(CC(COC)N=c1nc(N(C)Cc2cc(Br)cs2)c2c([nH]1)CCC2)OC c1(C(=O)NC(C(C)C)C(C)NC(=O)CNS(=O)(=O)C2CC2)ccc2nonc2c1 C=C1CCN(C(=O)C(C)c2ccco2)C(C(=O)N(CC2=CCCOC2)C)C1 c1(C(=O)NC(CNC(C2C=CCCC2)=O)C2CC2)cc(F)c(Br)c(Cl)c1 CCCC(CC)CC(=O)N1CCOC(CCOC)C1 C1(NC(c2c(CC)nn(C)c2)=O)CCN(C(c2cnnc(C)c2)=O)CCC1CO c1(C(=O)NC(C(C)NC(C=C(CCC)C)=O)(C)C)cc(OC)cc(Cl)c1F c1(COC)nnc2n1CCN(C(=O)C(=O)NC(c1ccccc1Br)CF)C2 Cn1c(C(=O)N(CCN(C(=O)C(O)C(F)F)CC2CC2)C2CC2)cc(Cl)c1Cl C1(OC(CCCC#C)=O)CCCN(C(c2ccc(Cl)cc2)=O)C1=O c1(C(=O)NCCNC(C(C(C)C)C#N)=O)cc2c(Cl)cccc2[nH]1 c1(CC(=O)NC(C(C)C)C(C)NC(=O)CCCOC(C)(C)C)ccc(O)c(F)c1 CCC1=C(C(=O)NCC2CN(C(c3nncn3CC)=O)CCC2C)CCCO1 N1(C(CC(=O)NCC)=O)CCC(O)(CNC(C2CCCS2(=O)=O)=O)C1 C1(CNC(CSC)=O)CN(C(=O)C(c2cscn2)N(C)C)CCC12CCC2 C1(CNC(C=C=C(C)C)=O)CCCC2CN(C(C3CCCN3S(C)(=O)=O)=O)CC12 c1(CC(N2CCCC(C)(NC(=O)CC3CCNC3=O)C2)=O)c(F)cc(F)cc1F c1(CCC(=O)NC2CCN(C(C34CC(OC)C3C4)=O)CC2)c(C)nc(O)nc1C c1(CNC(C2CC3CC3N2C(c2ncc(Cl)cn2)=O)=O)c(F)cc(Cl)cc1F CCCCC(=O)C(=O)N1CCCC(NC(c2oc(CO)cc2C)=O)C1 N1(C(CCc2nc(C)c(C)[nH]2)=O)CC2CCC1C(CNC(=O)C(F)C1CCC1)C2 C1(C2CCN(C(C3CC3Cl)=O)CC2)(NC(CCc2n(C)cnc2)=O)CC1 C1(O)(CNC(c2cc(F)cs2)=O)CCCN(C(=O)C(C2CCCCC2)F)C1 c1(CNc2nccc(-c3c(O)cc(Cl)cc3)c2)cccc2c1OCO2 N1(C(CCCC(CC)NC(CCOCC)=O)=O)CCC12CCC(O)CC2 CC(C)(F)CCC(=O)N1CCC(CNC(=O)CC2(n3cccn3)CC2)C1(C)C C=C(C)C1CCC(C)=CC1CC(=O)NC12CC1CN(C(C1CCCCC1)=O)C2 Cc1cccc(N)c1C(=O)NC(C1CCN(C(=O)Cc2csc(Cl)n2)C1)C C1(CCC)CN(C(=O)C(=Cc2cccs2)C)CC1NC(c1c[nH]cc1CC)=O CC(C)C(C)(O)C(=O)NCCC1CCCCN1C(C1COC(C)(C)O1)=O C1(C(C)NC(c2cnnn2C2CC2)=O)CCN(C(c2sccc2F)=O)CC1 C(C#Cc1cccnc1)NC(C1N(C(C(C(C)C)OCC)=O)CCC1)=O N1(CCc2c(C)ncs2)CCCC2C(NC(=O)Cc3c(C)noc3C)C(C)(C)C12 c1(CC(=O)N(CCC(C)NC(=O)C(C)CC(F)(F)F)C)csc2ccc(Cl)cc12 N1(C(c2cc(C)c(C)nn2)=O)CCCN(C(c2cc(Cl)ccc2Cl)=O)C(C)C1 C(=O)(C1CCCc2ncnn21)N(C)CC1CN(C(=O)C=Cc2cc[nH]n2)CCO1 C1(C(=O)NCCC2(O)CCN(C(C3CC3C(F)F)=O)C2)(OC)CCCCC1 N1(C(CNC(CNC(C(C)(C2CC2)OC)=O)=O)=O)CC(C)OCC1C N1(C(CNS(C)(=O)=O)=O)CCC(O)C(NC(=O)Cn2cccn2)C1 C1(C(N2CCC(=C)C2)=O)C2CC1N(C(=O)CCC1CCOC1)C2 C1(CC)CN(C(c2cc(C)cc(F)c2)=O)CCN1C(=O)Cc1ccsc1C C1(CNC(CCC(C)C)=O)COCCN(C(C23CCN(CC2)C3)=O)C1 C1(CC)CN(C(c2ccn(CC)c(=O)c2)=O)CCC1NC(=O)C1=CCCO1 C12(C(=O)NC(C)CCNC(C3(n4cccn4)CCC3)=O)CCCC(CO1)C2 c1(CCC(=O)NCC2CCC(NC(c3ccsc3)=O)CC2)cnc2n1CCCC2 Cc1cn2cc(C(=O)NCC3(C)CCCN(C(=O)CC4(O)CCOC4)C3)nc2s1 C(C(CC(C)C)NC(=O)C(C)n1cnnn1)NC(c1ccc(CC)s1)=O CC1(NC(C2(C)CCCN2C(=O)C=Cc2ccsc2)=O)CCOC1=O c1(OC)cc(C(N2CC(NC(C3COC(=O)O3)=O)C(C)C2)=O)nc(Br)c1 c1(CC(=O)NCC(CNC(CCC(=O)NCCC)=O)(C)O)cc(F)c(N)cc1F Cc1cc(C(=O)NCCC2CCN(C(=O)C(c3ccccn3)O)C2)ccc1N C(CCCCCC(=O)NCc1cc(O)ccc1F)NC(c1cccc(C)c1N)=O C1(CC)CCCCCCN1C(=O)C(O)CCCNC(=O)CCC(C)c1ccccc1 C1(C)(CNC(C2(N(C)C)CC2)=O)CN(C(=O)C(=O)NCC2CC2)CCO1 CS(=O)(=O)c1cccc(-c2cccnc2NC(c2csc3ccccc23)=O)c1 C1(C(=O)NC(CC)(CNC(=O)CCOCCN(C)C)CC)CC(C(C)C)=NO1 C12(NC(C(C)Cc3ccco3)=O)CCC1CN(C(=O)Cc1ccc(Cl)c(F)c1)C2 c1(C(=O)NC(C(C)NC(CN(C2CC2)CC)=O)C)[nH]ccc1C N1(C(COCc2nnc(C)s2)=O)C2CCC1CC(NC(C1(CO)CCCO1)=O)C2 CC(C(C)(C)C(=O)N1CCC(CCO)C1)NC(=O)COCCF C1(C(=O)NCCC(C(C)C)OC)CN(C(C2CCC(C#N)CC2)=O)CC1C1CC1 C=C1CCC(CNC(=O)C(C2CCCCC2)NC(C2CC2C(=O)OCC)=O)CC1 C1(CNC(C(CC)N(C)C)=O)(OC)CCN(C(C2CCCN2C(C)C)=O)C1 C12(CN(C(=O)CNC(=O)OC(C)C)C1)NC(=O)C(C)OC2.CCC(C)(C)N(C)C CCC(C)C(C)C(=O)N(CC(C)NC(=O)Cc1cc(C)[nH]n1)C N1(C(C(C)NS(CC)(=O)=O)=O)CC2(CCC(CNC(=O)CC3(C(F)F)CC3)O2)C1 C(CC(C)C)(C(=O)NCCOCCCNC(=O)CC(C)(C)C1CC1)OC C#Cc1ccc(C2(NCc3nnnn3C3CC3)CC2)cc1.c1c(Br)cnn1CC c1(CN(C)C(=O)NCCc2nccn2-c2ccccc2)coc(C#N)c1 C12(NC(CC(=O)OC)=O)CCN(C(c3ccc(N4CCCCC4)cc3)=O)CC1C2 C(C(=O)NCC(C1CC1)NC(c1[nH]c(=N)sc1C(F)(F)F)=O)(C(C)(C)C)N(C)C C1(C(N2CC(CCNC(C3CC(N(C)C)CCO3)=O)C2)=O)(SC)CC(F)(F)C1 C1(OC(C)C(N2CCCC2C2CCN(C(c3ccccn3)=O)C2)=O)CCCCC1 C(CC(C)(C)CN=c1[nH]c(=NCc2cocn2)[nH]c2c1SCC2)OC c1(OC)cc(C(=O)NC2CCOCC2C(=O)N(C)Cc2ccncc2F)nn1C CCC(C(=O)N1CC(F)CC1CNC(c1ccc(Br)s1)=O)C(F)(F)F c1(CN(C(=O)CC2CC(CNC(=O)CCc3nccn3C)C2)CC)cncn1C CC1SCCC1NC(c1ccc(-c2ccco2)[nH]1)=O N1(C(CSC(C)=O)=O)CCOCC(NC(c2cccc(I)c2O)=O)C1 C1(NC(c2csc(Cl)n2)=O)CN(C(c2csc(Br)n2)=O)C2CC12 C1(NC(C(C)OCC=C)=O)C2COCC1CN(C(c1cc(C)ccn1)=O)C2 c1(C(=O)OC)cc(C)n(CC(=O)NC2CC2NC(c2cccc(N(C)C)c2)=O)n1 c1(C(N2CCCCC(NC(C(C)CN(C)C)=O)C2)=O)cc(F)c(F)cc1Cl CCCC(C(=O)OC)C(=O)NC1C2CCC1N(C(c1ccc(C(F)(F)F)o1)=O)C2 C(C1CCCN1C(C1CCCSC1)=O)=CC(=O)N(CCC(C)(C)O)C c1(C(=O)NCC2CN(C(=O)C(F)(F)C3CCCCC3)C2)cnn2cnnc2c1 c1(C(N2CCC(C(CO)NC(c3n(CC)nnc3)=O)CC2)=O)cc(C)nc(C)c1 CC(=O)CCCCC(=O)N1CC(C(O)C(N2CCC(N(C)C)CC2)=O)C1 C1(COC)CC2(CCN2C(=O)COC2CCN(C(c3cc(C(C)C)on3)=O)C2)C1 N1(C(C(C)OCC#C)=O)CCC2C1CCN2C(=O)CCc1cccc(Br)c1F C1(NC(c2cc(C)c(C)s2)=O)CCC2(CCCN2C(=O)COCC(F)(F)F)CC1 c1(C(N2CC(C(C)NC(CCC(C)OCC)=O)C2)=O)ccc([N+](=O)[O-])c(O)c1 C(CC(C)(C)OC)(c1n(CCOCC)nnn1)NCC1=CCCOC1 N1(C(CCC=CC)=O)CCC2(NC(=O)CS(=O)(=O)NCC3CCCO3)CC2C1 C1(C(=O)NC2C3CN(C(c4cccc(C(C)=O)c4)=O)CC32)CCC2(CCC2)O1 c1(CC)cccc(F)c1C(=O)NCC(CNC(C1(C(F)F)CCOCC1)=O)OC C12(NC(C3CCC(C)S3)=O)COC(CNC(=O)C=Cc3cnc[nH]3)(C1)C2 c1(C(=O)NCCCC(C)NC(=O)C#CC2CCCCC2)cnc2[nH]c(=N)sc2c1 N1(C(CCC(C)OCC)=O)CCCCCC1C(N1CC(CO)C2(CC2)C1)=O C#Cc1ccc(C(N2CC(NC(C3CCC=CCCC3)=O)CC2C)=O)cc1 c1(C(=O)OC)ccc(S(=O)(=O)N2CC3CN(C(c4snnc4C)=O)CC23)n1C CC1(C)CCCCC1=CC(=O)NC1(CCNC(=O)CCN2CCC(F)C2)CCC1 c1(C(=O)NCC(=C2CN(C(c3n(CC)ncc3Cl)=O)C2)F)cc2occc2[nH]1 Cc1cc(CCC(N2CC(C3(NC(C4COC(=O)N4C)=O)CC3)C2)=O)cc(C)n1 c1(CN(CCCC)C(C2CCCC(C)C2)=O)cccc(O)c1O c1(C(=O)NC(C)C(C)(C)NC(c2cc[n+]([O-])cc2)=O)cccc(C(N)=O)n1 c1(OC)ccnc(OC)c1C(=O)NCCNC(c1cccc(F)c1F)=O C(CCCC(=O)N(C(C)(C(=O)N1CCC1(CO)CO)C1CC1)C)OCC CC(CCNC(=O)CC1CCN(C)CC1)CCNC(C1CC12CCC2)=O Cn1ncc(CNC(=O)CSC(C)(C)C)c1C(=O)NCC1CCC(=O)N1 N1(C(c2nc(C)sc2)=O)CCCCC1C(=O)Nc1ccc(O)cc1 N1(C(C2CC(C)C2)=O)C2CCC1CN(C(=O)CC(O)c1ccccc1)C2 C(CC(N)=O)(C(=O)N1CCC(F)(CF)CC1)NC(CCc1cnc(C)o1)=O C(c1cn(CC2(O)CCN(C(C3CCOC3)=O)C2)nn1)=CC c1(C(c2nnnn2CC2CC2)NCC(CC)(CC)SC)nccc2ccccc12 C1(NC(CCCCC)=O)CC2(C1)CC(NC(C1CCN(C(=O)CC)C1)=O)C2 c1(C(=O)NC2CCC(CNC(C(C)n3cncn3)=O)C2)cc(O)ccc1[N+](=O)[O-] c1(C2(C(C(C)C)N(C)CCOC3CC3)CC2)ccnn1C C1(NC(C2CCCS2)=O)CC1C1CCCN(C(c2cncc(Cl)n2)=O)C1 Cc1nc2cc(C(=O)NCC3C4CN(C(C56CC(C)(C5)C6)=O)CC34)ccc2n1C O=C1CC(C(=O)NC2CC(O)CN(C(C34CC(CO)(C3)C4)=O)C2)=NN1 C(=O)(CC1=NN(C)C(=O)C1)N1C(C(=O)NCC2(CCO)CCC2)CC(OC)C1 C1(C(=O)NCCC2CCC2)COC2(C1)CN(C(=O)C=C1CCOCC1)C2 c1(C(=O)NCC2CC(F)(CNC(C(CCC)O)=O)C2)ccc2n[nH]cc2n1 C12(C(N3CC(C)C(NC(C4CCS(=O)CC4)=O)C3)=O)CC(C)(C1)OC2(C)C c1(C(CNC(=O)CC2CSC2)NC(CC(C)NC(C)=O)=O)ccc(C(C)C)cc1 c1(OC)cc(CN(C=O)Cc2cc(Cl)ccc2Cl)cc(OC)c1OCC(N)=O CCCC(F)C(=O)NC(Cn1cncn1)C(=O)NCC1CCC(C)C1 C1(c2cnn(C)c2)(CNCCC#CC)CCCO1 CON1CCC(C(N2CC(CNC(C3C4CCCC34)=O)C(C(F)(F)F)C2)=O)CC1 C(CC(C)CCCC(C)C)NC(C1=NOCC1)c1n(-c2c(C)cccc2)nnn1 CC1CCC(CNC(c2cncc(O)c2)=O)N(C(=O)COCc2cccnc2)C1 C(=O)(C#CC(C)(C)C)NC1C(C(=O)NC(CC#C)C(=O)OCC)CCCC1 c1(C(=O)NCc2ccc(C)cc2Cl)nccc2c1NCCC2 c1(C(CO)NC(CC2CCN(C(c3n(CC)ncc3)=O)C2)=O)ccc(F)cc1 c1(N)conc1C(N1CCC(OCC(=O)NCC(C)(C)O)C1)=O.CC(=O)C(C)=O C(=O)(C(C)(C)C(C)(F)F)NCC1N(C)CCN(C(c2ccc(O)c(CO)c2)=O)C1 C1(C(=O)NCC2C3CC2N(C(=O)C=C2CCN(C)C2)C3)(OC)CCCCCC1 N1(C(c2n(C=C)ncc2)=O)CCC(C(=O)NC2CC3CCC2O3)C12CC2 C1(C(=O)NCc2c(C(=O)NCC3CSC3)n[nH]c2)CC2CC(=O)C1O2 C(=O)(C#CC1CCCOC1)N1CCN(C(c2ccc(F)cn2)=O)CC1CC1CC1 N#Cc1cscc1C(=O)NCCNC(=O)CC1(O)CCCCC1 O=C(C1CSc2ccccc21)NC1CC2CN(C(C3CCCC34CC4)=O)CC12 n1(CC)nc(C)c2cc(C(N3CCC(NC(=O)C(C)(C4CC4)OC)C3)=O)sc12 Cc1ccc(F)c(O)c1C(=O)NC1CC(NC(=O)CCc2cccnc2C)C1 C1(C(N(C)CC2(CNC(C3CC(O)C3)=O)CC2)=O)CCN(c2ccncc2)C1 N1(CC(=O)NCC2(CNC(c3cnccc3I)=O)CC2)CCCNC1=O c1(C(=O)NC2C(NC(COCC#C)=O)COCC2)cc(OC)c(OC)c(Cl)c1 C1(NC(COC(C)C)=O)CN(C(C2(C#N)CCSCC2)=O)Cc2nccn2C1 C1(C(C(=O)N(CCCCCNC(C2(O)COC2)=O)C)O)CCCCCC1 C1(C(N2CC(C)C(NC(=O)CC(O)C3CCCC3)C2)=O)CCc2ncncc2C1 C1(C(=O)NCC2C(C)(C)C2)CN(C(c2nccnc2Cl)=O)CCC1(F)F N1(CCOCCC)CCCC(CO)C1.C1(=O)CCC(C)N1C1CC1 c1(NCCC2(NC(CC(C)C3CC3)=O)CC2)ccc(C(N)=O)cc1[N+](=O)[O-] c1(CNC(C2C(OC)CN(C(C=CCCC)=O)C2)=O)cncc(C#N)c1 N1(CC(C2CCC2)OC)CCCC1c1ccsc1 C(C(=O)NC1CC1)(C1=NOC2(CCC2)C1)N1C(C(=O)NC)CCC1 C1(CNC(c2c(OC)cc(C)s2)=O)CN(C(c2cnc(C)[nH]2)=O)CCCO1 N(C1CCOc2c(F)cccc21)C(C(C)NC(=O)C1CC1)=O c1(C(=O)NC2C(C)CCN(c3cc(CC)nc(CC)n3)C2)cccc2sccc12 N1(C(=O)C(F)F)CCCCC1C1CCCN(c2nnc(-c3ccccc3)s2)C1 c1(C(=O)NCC2COCCN2C(=O)C(F)CC2CCC2)ccc2c(c1)CCC2 C#CC1CN(C(=O)C(CC)CCOC)CCN1C(=O)C(=O)NOC c1(CNC(N(C)Cc2cc(C3C(C)C3)no2)=O)ccc(C(C)(C)C)nc1 n1(CC(N(CCNC(c2ccc(C#N)cn2)=O)CC)=O)nc2n(c1=O)CCOC2 C1(N(C)C(=O)OC(C)(C)C)(CNC(=O)CCCC(C)(F)F)Cc2ccccc2C1 Cc1ccc(C(=O)NC2CCN(C(=O)C(F)C(C)C)CC2C)c2c1CCCN2 S(=O)(=O)(c1ccc(N2CCC(OCCO)C2)cc1Br)NCC1(C)CCOC1 c1(NCC(=O)N(C2CCN(C(=O)Cc3ncnn3C)C2)CC)ccncc1.C(=O)NC c1(CC(=O)NC2CC2NC(C2C3CC4C(C3=O)C24)=O)ccc(Cl)c([N+](=O)[O-])c1 N1(C(Cn2ncn(C)c2=O)=O)CCC(NC(=O)CCN2CCC2)CC(O)C1 N1(C(c2cc(CC)ncc2)=O)CCOCC(C(=O)NC(C)C2CC2)C1 N1(C(=O)NC2CN3CCC2c2ccccc23)CCc2nccc(CO)c2C1 c1(OC)ccc(F)c(C(=O)NCC2CCCCC2NC(C2CC(OC)C2)=O)c1F C1(CNC(c2cc(C(F)(F)F)no2)=O)CCCCN(C(C2CCCOCC2)=O)C1 Cc1nc(CNC(C2CN(CCC(=O)O)CC2O)=O)ccc1Br c1(CC(=O)NCC(CC(C)C)NC(=O)CN2CCCC2=O)cccc([N+](=O)[O-])c1 N1(C(c2c(C)ncnc2)=O)CCCC(C(=O)NC2(c3ccccc3)CC2)C1C CC(C)CC(C)(O)C(=O)N1CCC(C(=O)NC2(C)CS(=O)(=O)C2)C1 c1(C(=O)NC(CNC(C2CC(SC)C2)=O)C2CC2)ccc(N)c(C)c1Cl N1(C(c2cc(OC)c(OC)cc2)=O)CCCC(NC(C2C=CCC2)=O)CCC1 c1(C(=O)NCC=CCNC(C(CCC)C)=O)cnc(C)nc1COC C(C)(C(=O)NCCCc1nccs1)(C1CCC1)NC(C(C)c1cc[nH]n1)=O Cc1cc(C)c2cc(CNC(Cc3ccc(Br)cc3)C3CC3)[nH]c2c1 C1(CNC(CC2CN(C)C2)=O)CCCCN(C(c2cnn(C)c2)=O)CC1 C1(CNC(c2ccc(Cl)nc2)=O)CCC(F)(CNC(C2(CC(F)F)CC2)=O)C1 CC1CN(C(C2(S(N)(=O)=O)CC2)=O)CC1NC(=O)CC1CCS(=O)(=O)C1 N1(C(CN(C)C2CC2)=O)CC2(NC(=O)Cc3coc(C(F)F)n3)CCC1CC2 C(=O)(C(C)C1CCC1)NCC(=CC(=O)NCC1(COC)CC1)C N1(C(C)=O)CCC(CNC(=O)CCCC(C)C)CC1C.C(CNC)O C1(CNC(C2OCCN(CC)C2)=O)CN(C(=O)C(C)=O)CCN1C C1(N(CCOC)C(c2cnc[nH]2)=O)CCN(C(C2CC(C(F)(F)F)CO2)=O)CC1 c1(CC(=O)NCCOCCn2cc(-c3ccccc3F)nn2)ccc(Cl)c(Cl)c1 C(=O)(C1=COCCO1)NCCc1c(CNC(C2(OC)CCCC2)=O)nco1 C1(C(N2CCN(C(c3cnsn3)=O)C3CCCC23)=O)CCc2cc(F)ccc2O1 C(=O)(C1=CC2(CN(C(c3ccn4ccccc34)=O)C2)OC1)NCC(C=C)O C1(NC(COC)=O)CC(C)CN(Cc2cc(Br)c[nH]2)C1 Cc1cnn(C)c1CC(=O)NC1CCOC(CNC(c2cc(C#N)no2)=O)C1 Cc1nn(CC(=O)NCc2cc(C(=O)NC(C3CCCC3)CO)n(C)n2)c(=O)o1 C1(NC(CCCSC)=O)CC2CCC(C1C)N2C(C1CCN(CC2CC2)CC1)=O C1(N(C(CC(CC)C)=O)C)CN(C(C2(F)CCC2)=O)CC1(C)C N1(C(C2CCC(C(=O)OCC)CC2)=O)CCc2sc(-c3ccnn3C)cc2C1 c1(OC)ccc(Cl)cc1C(=O)NC1CC2CCC1N2C(=O)CCC1CCC(=O)N1 c1(C(N(CCC(C)NC(c2nccc(OC)c2C)=O)C)=O)cc2c(ncn2C)[nH]1 C(=O)(NNc1ccc(CC(C)C)cc1)C1(SC)CCCCC1.c12cn(nn1)CC2 CC1(NC(=O)C(c2ccc(Cl)cc2)O)CCN(C(CC(C)(N)Cn2cccn2)=O)C1 N1(C(C(C2CC2)OC)=O)CCC2(CC1)CC(NC(c1nccc(SC)n1)=O)C2 N1(C(C(CC(C)C)NC(CCCCCC#C)=O)=O)CCC2(CCOC2=O)C1 N1(C(C2CCN(C)C2)=O)CC(NC(C2CN3CCC2CC3)=O)CC2(CC2)C1 C1(N(C(=O)Cn2ccnn2)CCC)CCN(C(c2cnn(CC)n2)=O)C1 C1(NC(c2cc(CC)n(C)n2)=O)CC2CC1N(C(c1sc(OC)nc1Cl)=O)C2 C1(N(C(C=Cc2c(C)ccs2)=O)C)CN(C(c2sccc2C(C)C)=O)CC12CC2 N1(C(c2cc(OC)n(C)n2)=O)CCCC(CC)C1C(=O)NC(c1ccsc1)CO C1(N)CCC2CN(C(=O)CC)CCC2C1.C=CC(C)(CC)C(=O)N Cc1ccc(CCC(=O)NC(C)CCN(C)C(C2(Br)CC2(F)F)=O)cc1 N1(C(c2scc(COC)c2)=O)CCc2[nH]nc(CNC(c3coc(Cl)n3)=O)c2C1 C1(C(=O)NC2CC(CNC(=O)COC(F)(F)F)C23CCC3)COC2COCC2O1 c1(C(=O)OC)nc2ccccc2nc1N(C)Cc1c(F)cccc1F C1(NC(C=CC(C)(C)C)=O)(CNC(C2CC2c2ccco2)=O)CCOC1.C1CO1 Cc1nn2cc(C(=O)Nc3cccc(NC(C4CCCC(=O)N4)=O)c3)nc2s1 CC(=Cn1ccnn1)C(=O)NC1CC2(CCCCN2C(C2CCCOC2C)=O)C1 C12=c3c(scn3)=NC(=NCC3CC(C3)CN1CC)N2.Cc1nccn1-c1ccccn1 C123CCC(CC1)N2C3=O.C(=O)(CC(F)(F)F)NCC(=O)NCC1CCCC12CC2 C1(NC(C(C)NC(C)=O)=O)CC2CC(C1)CN(C(c1cscc1C(N)=O)=O)C2 c1(NC(C)=O)ccccc1COC(c1ncoc1C1C2COCC12)=O c1(C(C)C)ccc(C(=O)NC2CCC(C(N3CCC(CO)C3)=O)CC2)c(Cl)n1 C12(CNC(C(C)(C)C3(O)CCOC3)=O)CC(CN1C(c1coc(CO)c1)=O)C2 C1(C(=O)NCC(C(=O)NC)(C)C)CCCC(NC(=O)CNc2cnn(C)c2)CC1 N1(C(c2cc(OC)n[nH]2)=O)CCC2(NC(=O)CCn3ccnn3)CC2C1 C1(C(=O)Nc2cnn(CC)c2C)(CC)CCCN(C(=O)C=CCO)C1 c1(C(=O)NC2CN(c3snc(CCC)n3)C(C)C2)ccc2c(c1)CC2 c1(N2C(CNC(=O)CCc3ccccc3)CCCC2)ncnc2c(Br)cccc12 CCC(CC)C(C)C(=O)N(C(C)CNC(c1ccn(C(C)(C)C)n1)=O)C C1(N(C(C(C)OCCC=C)=O)C)CCCN(C(=O)CCN2CCCC2=O)C1 C(CC(=O)NCCCCN(CCCNC(C1(NC(N)=O)CC1)=O)C)SC S(=O)(=O)(c1cnn2ccc(=NCCOc3ccccc3)[nH]c12)N1CC(C)(OC)C1 Cc1cc(O)c(Cl)cc1C(=O)NC(CNC(c1c[nH]nc1C)=O)C(C)C(C)C N1(C(=O)NC2C(c3onc(CC)n3)C2)CCNCC1C1CCCC1 CC1(C)CC2(CO1)CN(C(=O)NCC1CCOCC1F)C2 O=C(C#CC1CC1)NCc1ocnc1C(=O)NC1CC=CCC1 Cn1cc(S)cn1.c12c[nH]c(c1)C(=O)NC(C)(C)CNC(=O)CC2.C(C)(C)(C)O C1(N(C)C)CN(C(c2ccc3nsnc3c2)C(=O)NCCCF)C2(CCC2)C1 N1(C(c2cncc(CNC(CCC(C)=O)=O)c2)=O)CC(C)(C)CC1C c1(C(N2CC=CC(NC(C3(c4cccnc4)CC3)=O)C2)=O)cc(CO)nc(Cl)c1 C1(CNC(CCN(C(C)=O)CC)=O)CC2COCC2N1c1cc(=O)n(C)cn1 c1(C(N2C(CCNC(Cc3n(C)ccn3)=O)CCC2)=O)ccn2c(O)nnc2c1 N1(C(c2c(C)nccn2)=O)CC2CC(O)C1C2NC(=O)C(c1cccc(F)c1)C C1(CNC(=O)C2=CCC2)C2Cc3c(Br)cccc3C12 C1(CCC)CN(C(=O)CCCc2cccs2)CCN1C(c1cnc[nH]c1=N)=O c1(C(N(C(C(=O)N2CCC2CN=[N+]=[N-])C2CC2)C)=O)cc2cc[nH]c2cn1 N1(C(C(CC=C)NC(=O)C(F)=CCC)=O)CC2NC(=O)OC2C1 C#Cc1ccc(C(=O)NCC(CC=C)NC(=O)C(O)C(C)(C)C)c(C)c1 c1(OC)cnc2ccc(C(=O)NCCNC(c3coc(Cl)c3)=O)cc2n1 N1(CCNC(=O)C(C2(O)CN(C(C3(c4cccnc4)CC3)=O)C2)F)C(=O)CCC1=O C1(C(=O)NCC(CC(=O)OC)C)CC(O)CCN1C(C1C(C)(C)C1(C)C)=O C(=O)(C1=NNC(=O)CC1)N1CCC(CNC(c2c(CCC)n[nH]c2)=O)(COC)C1 C(=O)(C(C)(Cc1ccccc1)C(C)C)NCCC(=C)CNC(=O)CCCCSC c1(NC(C(C)C)CO)ccc(S(=O)(=O)NC2CCC(CO)C2)cc1C#N C1(CNC(c2c(C)coc2)=O)CC2CCC1N2C(=O)CCC1CCCN1C N1(C(c2cscn2)=O)CC2CCC(C1)N(C(=O)CCOCC1CC1)C2 c1(C(=O)NCCOc2ncccn2)cccc(NC2CS(=O)C2)c1 N1(C(Cc2cnc(C)[nH]2)=O)CCC(NC(C2CCCC2C)=O)C(O)C1 C(CCC1CC1)(C(=O)NCC1(O)CCN(C)C1)NC(COCCCCC)=O N1(c2nc(OCC)c(Br)cn2)CCCC(C2CN(C(=O)CCc3cnc[nH]3)C2)C1 n1(CC)cc(C(=O)NCC2CC2NC(c2cc(C(C)C)oc2C)=O)c(C)n1 C12(C(=O)NCCSCC(=O)NCC(C)(O)CO)C(=O)C3CC1C2C3 CCC(C(=O)N1CC(C2CN(C(=O)C#CC3CCOCC3)C2)C1)C(C)(C)CC C(=O)(C1=NNC(=O)CC1)NC(C1CCCN(C(C2(COC)CC=CC2)=O)C1)C N1(C(CCC=C=C)=O)CCCC2(CCN(C(=O)Cn3cc(S(C)(=O)=O)cn3)C2)C1 Cc1cc(C(=O)NC2(C(N3CC(CSC4CC4)C3)=O)CC(CO)C2)cnc1C c1(C(C(=O)OC)N(C)C(C2CC=CC2)=O)cccnc1 C(=O)(CCCC(F)(F)F)N1CCC(C(C)NC(c2cc(F)c(Br)cc2N)=O)C1 C1(C(=O)NC2CCC(NC(C3C(=C)CC3)=O)CC2)(C(=O)OC)C(C)(C)C1(C)C c1(C(=O)NCC2N(C(C(COC)N(C)C)=O)CC=C2)c(Cl)cc(Cl)cc1Cl C#CCC(C(=O)NCCC(CCC)C1CC1)NC(=O)CCC1(C)N=N1 N1(C(c2ccc(Cn3cc(C(C)O)nn3)cc2)=O)CCOC2(CC3CCC2C3)C1 O(NC(=O)C(CC(N)=O)NC(c1ocnc1CCC)=O)CC=C C1(CC)C(C(=O)NCC(C)(C)C2CCCC2)CCN1C(=O)C=CCN1CCCC1 c1(C(C(=O)NCCC#N)N(CC(F)Cl)C)cn(C)nc1Br C=Cn1ncc(C(=O)NC2(C(=O)NC3(CCF)CC3)CC2C)c1N C(=O)(C1=CC2(CCN(C(c3cc(O)n(C)n3)=O)C2)C1)NC(CC)CO c1(SCCN(C(=O)CSc2ccncc2)C)ccc(Cl)c(Cl)c1 c1(OC)cccc2c(C(=O)NCC(C)(Cc3cccs3)CO)csc12 N1(CC)CCCN(C(C2(F)CCN(C(=O)CCN3CCC3)CC2)=O)CC1 CCCCCC(=O)NCC(N1CCCC1C1CCN(C(=O)CC(=O)NCC)C1)=O C1(C(=O)NCCN(C(c2ccn(C(F)(F)F)n2)=O)C2CC2)OC2CCC1C2 c1(C(N2CCCC(F)(C(=O)NCC3(C)CCCO3)C2)=O)cncc2[nH]ccc12 N1(C(C2CCN(C(OC(F)F)=O)C2)=O)CCC(CC2CC2)CC1 C1(C(N2CCC(O)(C(C)NC(=O)CC3CCS(=O)(=O)C3)C2)=O)C2CC3C(C2=O)C13 C(=O)(CCCC(=O)N(C)CC1CCCN1C(C1CCC=CO1)=O)N(C)C N1(C(C(C)OCCCC)=O)CCCC(NC(=O)CCc2ccn(C)n2)CCC1 N1(c2n(C(C(c3ccc(Cl)cc3)C)C)nnn2)CCc2c(F)cc(Br)cc2C1 CC(C(C)(C)N(C)C)NC(C1CCCN1Cc1ccco1)=O C1(CN(C2CCCCC2)CC=C)CC2(C1)CC(C(F)(F)F)C2 C1(CNC(=O)NCC2CCC(C)CO2)CC12CCOCC2 CCC(C)C(C(=O)NCCCC(C)(C)OC)N(C(=O)C#CC(C)(C)O)C c1(C(=O)NCC2(OC)CN(C(=O)CC3CC=CCC3)C2)cnc2c(C)cccn12 N1(CC(=O)NC2CC(C)N(C(=O)CCCS(N)(=O)=O)C2)CCCC2(CC2)S1(=O)=O C(=O)(C(CC)C(F)(F)F)N1CCC(CC=C)(NC(c2cn(C)nc2COC)=O)C1 CC(C)C(O)C(C)C(=O)NCC(C(=O)N(CCO)CCO)C(C)(C)C C(=O)(C1CCCn2cncc21)NCCC1CCN(C(c2c(C)cnnc2)=O)CC1 N1(C(=O)C=Cc2cccs2)CC2CCC1C1CN(c3ncncc3Br)CC21 C1(c2n(C)nc(C(F)(F)F)c2)CN(C)CCN1C(=O)NCC1CCC12CCCC2 CCCC(CCC)CCCC(=O)NCC(C)CN(C)C(c1ccnc(F)c1N)=O c1(C(N2C(CNC(C(COC)(C)OC)=O)CC2)=O)nc(Br)c2n1CCCC2 c1(C(=O)NC2(C)CCCN(C(c3ccn(C)c(=O)c3)=O)C2)ccc2[nH]ccc2n1 C1(C)(NC(C(OC)OC)=O)CCN(C(c2c(F)cncc2Br)=O)CC1 Cc1nccc(C(=O)NCCC2CCCCN2C(C2CCC(O)C2)=O)n1 CC(CCN(C)C)C(=O)NC1CC(CCNC(=O)C(O)Cc2ccc(F)cc2)C1 C1(C(=O)NC2CCC(CNC(C(C(=O)OC)OC)=O)C2)CC2CCC1C21CC1 c1(CC)cc(C(=O)NC2CC(NC(c3cc(C(C)(C)C)n[nH]3)=O)C2)ncn1 c1(C(N(C(CNC(=O)CS(=O)C(F)(F)F)C2CC2)C)=O)cccc2[nH]nc(O)c12 C(N=c1[nH]c(=NCCc2n[nH]c(=N)o2)[nH]c2c1CCCCC2)C1(CC#N)CC1 C(=O)(C1=CC2C=CC(C1)C2)OCCC1CC(NC(=O)OC(C)(C)C)C1=O C(=O)(C(C)(C(C)C)OC)NCC1C(NC(C(C2CC(C)(C)C2)OC)=O)CCC1 c1(N(CCC(N)=O)C)ncnc2c1ncn2C1CC(O)(CO)C1 C1(C(=O)NC(c2ccns2)C)COCCN(C(c2nc[nH]n2)=O)C1 Cc1c(C(N2C(C(=O)Nc3cnn(C)c3C(C)C)CC2C)=O)cccc1F C1(C(N2CCC(N(C(c3cccc[n+]3[O-])=O)CC)C2)=O)CCC2(CCC2)C1 N1(C(Cc2cc(COC)on2)=O)CC(NC(c2ncccc2C)=O)C2CC12 N1(C(C(C)OCCC(C)C)=O)C2CCC1CN(C(=O)CCC(F)F)CC2 O(C=CC(=O)NCC1CCN(C(C2CCC2C(F)F)=O)C1)CC CC(C(=O)NCCCC(O)C(=O)N1CC(C)(O)C1)C(F)(F)F C(=O)(C(C)S(N)(=O)=O)N1CCN(CC2CN(C(Cn3c(C)ncc3)=O)C2)CC1 CC(C)(C)C(C(=O)N1CC(c2cn(Cc3cnns3)nn2)C1)NC(N)=O CCS(=O)CC(=O)NCCC(C)NC(=O)C(C)N(C)C(=O)OC(C)(C)C c1(CC)ccsc1C(N1CCC(C(C)NC(=O)CN2CC=CC2)C1)=O n1(CC)cnc2nc(=NCCCOCCO)[nH]c(NC3CCN(CC4CC4)CC3)c12 C(=O)(C1CCc2cccc(O)c21)NCC1(CN(C(c2cc(C)nn2C)=O)C)CC1 CCCN=C(NCC(N1CCCCC1)(C)C)N1CCCC(O)(CO)C1 C(Cc1ccccc1)(C(=O)NCCCCCNC(=O)CC(C)c1ccccc1)OC c1(OC)ccc(NC(=O)N(CCC(O)CO)C(C)C)cc1C(F)(F)F C(=O)(CCC(C(C)C)NC(=O)CCP(C)(C)=O)NC(c1nn[nH]n1)CC C1(C(=O)NC(C2N(C(C(C)NC=O)=O)CCCC2)C)CCC2(CC1)CC2 N1(C(C=CC(=O)OCC)=O)CCOCC1CN(C(=O)CCC1CC1(Cl)Cl)C CCC(CC)C(C)C(=O)NC1CCN(C(c2ccc(NC=O)cc2)=O)C12CC2 C123CCCC(CN1CCN2)C3.c1(OC)cc(C)nc(NS(C)(=O)=O)n1 c1(C(C(=O)NCCCN(C(C2CC23CC3)=O)CC)C)ccccc1C S(=O)(=O)(c1cnc(N(CC(O)CC)C)c(Cl)c1)N1CC(COCC)OC(C)(C)C1 CON(CCC(=O)NOCCOC)C(=O)C(C)(O)c1cccnc1 c1(C(N2C(CNC(CCC(CC)OC)=O)CC3(CC3)C2)=O)cc2occc2n1C C1(C(N(CCS(=O)(=O)NC)C2CC2)=O)CCC(n2cc(C(O)C(C)C)nn2)CC1 N1(C(CC(CC)C)=O)CCC2(CC2NC(C2CC23CCSCC3)=O)C1 Cc1c(C(=O)N(C)CC2C3CN(C(=O)C(C)(C)O)CC23)nc(O)c2ccccc12 c1(C(=O)NC2CN(C(c3sc(C)c(O)n3)=O)CC(O)C2)cnc2sccn2c1=O c1(N(CCCC)C(=O)CN2CCCC2=O)c(C)csc1C.C12CCN(C1)C2=O C=CC1CCCCN1C(=O)C(F)CC1CN(C(c2c[nH][nH]c2=N)=O)C1 C1(CC)(NC(=O)Cn2ccnn2)CCCN(C(C2CC2c2ccncc2F)=O)C1 C1(C(=O)NCC2(CNC(c3c(C(C)C)ocn3)=O)CCC2)CCc2c[nH]nc2C1 c1(N2CC3N(C(C4CC4c4ccccc4)=O)C3C2)ncnc2cc(Br)sc12 C1(C)(NC(c2cc(-c3cn(C)nn3)on2)=O)CCN(C(C2CCC(=O)C2)=O)CC1 Cc1cc(C(=O)N(C)CC2CCCN2C(c2ncn(C(C)C)n2)=O)ncc1F N1(C(c2nc(Cl)ccc2F)=O)CC2CCN(C(C3(CO)CC3)=O)CCC2C1 CC(C)C(C(=O)NCCN(C1CCCCC1)C(C1CCCN1C=O)=O)n1cncn1 C(=O)(C(C)C(F)(F)F)NCC(C(C)C)NC(C1(C(C)(F)F)CC1)=O N1(C(c2c(C)cc(F)cn2)=O)CC2CCOC2(CNC(=O)CC2CCOC2)C1 c1(-c2n(CC)ncc2)ccc2ccn(CC(=O)Nc3ccc4[nH]ccc4c3)c2c1 C12CCN(C1)C(=O)C(=O)N2.c1(C(N2CCC2c2cccnc2)C)nncn1C N1(C(c2cnc(C)s2)=O)CC2C(NC(=O)CC(C)CC(C)C)CS(=O)(=O)C2C1 CCC(C)C(O)CC(=O)N1CCCC1(C)C(=O)NCC(C)(C)CC(F)F CC1(C2CCN(C(=O)Nc3cnn(-c4ncc(Br)cn4)c3)CC2)COC(=O)N1 CCC(C(=O)N1CCC(C(C)NC(c2cc(-c3cnccn3)[nH]n2)=O)C1)OC c1(OC)ccc(C(N2CCCC2C(C)(C)NC(=O)CC(C)CF)=O)cc1O Cc1cc(N)cc(C(N2CCCC(NC(c3cnn(C(C)C)c3F)=O)C2)=O)c1F c1(CC(=O)NCC2(C)CC(NC(c3cn(CCC)nc3)=O)C2)c(Cl)cccc1Cl c1(OC)cc(C(=O)N(C(C)CNC(=O)C=C(C)C(F)F)C)cc2cn(C)nc12 C(=O)(C(C)(F)C(F)(F)F)NCC1C(NC(c2sc(CCC)c(CC)c2)=O)C1 c1(CNC(C2CC(C(F)F)C2)=O)ccccc1 c1(OC)cc(NC(c2nc(NC(c3cc(Cl)ccc3Cl)=O)cn2C)=O)cc(O)c1 CCC(C(C)(F)F)NC(C1(C)CCN(C(=O)CC2CC(OC)C2)C1)=O C1(NC(c2ccc(CCCC)cc2)=O)CN(C(=O)C(O)CSC)CC1(C)C Cc1ccnc(C(N2CCCC(C(C)NC(c3ccc(CO)nc3)=O)C2)=O)n1 C(=O)(C1CC(O)c2ccccc21)NC1C(SC)CN(C(=O)COC(F)F)C1 c1(OC)ccc(C(=O)NCCC#N)cc1-n1cc(C(C)CN2CCCC2)nn1 c1(OCC)ccc(CC(=O)OC(CO[Si](C)(C)C)CO)cc1 O=NN1CCCCC1C(N1C2CCC1C(CNC(C1SCCS1)=O)C2)=O CC1CCCN(C(=O)C#CC(C)(C)C)C1CCNC(c1coc(CO)c1)=O N1(C(c2ccc(-c3ccco3)[nH]2)=O)CCN2C(=O)NCCC2C1 C#CCCCCC(=O)NC1CCN(C(c2[nH]ccc2COC)=O)CC1F c1(C(=O)NCC2(C)CCCN2C(=O)C=Cc2ccco2)nc(C2CC2)ncc1Cl C1(C(N(C2CCN(C(c3cccc(CF)c3)=O)CC2)C)=O)CC12CCOC2 C#CC1CN(C(=O)CCCOC(C)C)CCN1C(=O)C=Cc1ncc(C)[nH]1 c1(C(=O)NCC2CN(C(Cc3cc(C)sc3)=O)C2)cc(Cl)cc(Br)c1 CC1=C(C(=O)NCC2CC3(CC(NC(C4(C)CC(O)CN4C)=O)C3)C2)CCCO1 CCC(CC)CCCC(=O)N1CCC1C(N1CCOC(CF)C1)=O NS(=O)(=O)c1scnc1C(N1CCCC1c1cn(Cc2ccncc2)nn1)=O C(=O)(CCCC(C)=O)NCC1N(C(c2c(OC)c[nH]n2)=O)CCC1C N1(C(c2cscc2F)=O)CCOC2CCCCC12 c1(C(N(C2CCN(C(c3ccnc(C)c3N)=O)CC2)C)=O)ccnc2[nH]nnc12 C(=O)(C#CC1(C)COC1)N1CCC(CC=C)(NC(c2cc(C)c(Br)s2)=O)C1 c1(C(=O)OCC)[nH]c(C)c(C(=O)CNCC(c2ccc(Br)cc2)N(C)C)c1C C1(C(=O)Nc2ccc(C(N)=O)nc2)CC2CCC(C1)N2C(=O)CCc1cn[nH]c1 C(N=c1[nH]c2cccc(Br)c2o1)C1C(NC(C2C(=C)CC2)=O)CCCC1 c1(CC(=O)NCC23CC(NC(c4cc(OCC)n[nH]4)=O)(C2)C3)ccc(C)cc1Cl O=c1cc(CNc2cnn(C3CCNC3)c2)nc2ccc(Br)cn12 CC(C)C1=NOC(C(=O)NC(C)C=CC(=O)NCCCc2cncnc2)C1 C1(C(=O)NC(C)(CNC(c2csc(C#N)c2)=O)C2CC2)C2(CCC2)C12CCC2 C1(C(=O)NC(C2(O)CN(C(CC(C)OC)=O)C2)C)COC2COCC12 Cc1ccc(C)c(CC(N2CCN(C(C3CCCN3C)=O)C(CC3CC3)C2)=O)c1 N1(C(C2(COC)C=CCC2)=O)CC2(C1)CN(C(c1ccc(Cl)o1)=O)CC2CO N1(C(CCn2c(C)ncc2)=O)CC2CN(C(c3c(CO)cccc3Cl)=O)C2C1 CC(C)(CCC(=O)NC1CC2CC1N(C(c1csc(Cl)c1)=O)C2)[N+](=O)[O-] O=C1CCC(C(=O)N2CC3(CC(C(=O)NCCC4CCOC4)CO3)C2)=NN1 CC1(C)CCN(C(C2CCS(=O)CC2)=O)C1C(=O)NOCC1CCCO1 C1(NC(C2C(C)C2)=O)CCN(C(C2CCCN(C)C2)=O)CC1C.CCSC N1(C(c2n(CC)cnn2)=O)CC2CCC1C(CNC(c1cnc(O)n1C)=O)C2 CCCCCCC(C)(CC)C(=O)N1CCN(C(=O)Cc2ccon2)C(C)C1 N1(C(c2c(C)nccc2)=O)CCN(C(c2ccnn2C)=O)CC(O)C1 CC1(C)CCC(F)(F)CC1C(N1CCCC1C1(NC(c2cnsn2)=O)CC1)=O c1(OC)ncccc1C(=O)NC(C)CNC(=O)Cc1nc(-c2cccs2)oc1C C(c1ccsc1Br)=CC(=O)NCC1COC(=O)N1 c1(C(N2C3C(CNC(C=CCN(C)CC)=O)C(C3)C2)=O)cc(Cl)cc(Cl)c1N C(=O)(CCC(F)(F)F)NC1CCN(C(c2c(C)cno2)=O)C1C(C)C CC(C1CCCCC1)=CC(=O)NC1CCCC(N(C)C(c2nocc2C)=O)C1 N1(C(c2c(CCNC(c3c(CC)c[nH]c3)=O)n[nH]c2)=O)CCCCC(CO)C1 C1(CNC(c2c(C)nsc2)=O)CCCN(C(C2(CC(C)C)CCC2)=O)C1 c1(SC)ccc(F)cc1COC(C1(C)CCCCCC1)=O C(CC(C)C(=O)NN(C(=O)C=CCOCCOC)CC1(O)CC(CC)C1)=CC c1(C(=O)NCCN(C(C2(c3oncc3C)CC2)=O)CC)ccnc2ccccc12 c1(C(c2ccccc2)NC(=O)Nc2cncc(C(F)(F)F)n2)cc(Cl)sc1Cl c1(C(=O)NC2C(NC(C=C(C)C)=O)COC2)cccc(C#CCO)c1 C=CCCCC(=O)NNC(=O)NCC(c1ccccc1Cl)CO N1(C(c2cn(C)nn2)=O)CCC2CCC(C1)N2C(=O)CSc1nccn1C C1(C(N(C2CCCN(Cc3coc(C4CC4)n3)CC2)C)=O)CC2CC1C1CC21 C1(N(c2cc(-c3ccco3)on2)C(=O)CNC(c2cccs2)=O)CC2CNC1C2 CN1CC(C)(C(N2CCCC(n3cc(C4(CO)CC4)nn3)CC2)=O)CCC1=O c1(C(=O)NC2CCC(CCNC(CCOCC#C)=O)C2)c(F)ccc(F)c1Cl c1(N(C2CNCC2(F)F)C(c2ccn(CCOC)n2)=O)ncnc(C)c1Br CCCC(C)(C)C(=O)N1CCC(C(F)C(=O)NCCC#CCO)C1 C1(C(=O)NC(C(N)=O)C(N)=O)CCc2ccccc2C1O c1(C(=O)NCCOC2CCN(C(C3C(CC)C3)=O)C2)cc(O)cc(Cl)c1Cl c1(C(CN2CC(c3onc(CC)n3)OCC2)=O)ccc2nc[nH]c2n1 N1(C(C(C)(C)N)=O)CCOCC(CN(C)C)C1 C(=O)(C(C)(C)C(=O)N(C)C)N1CCC(NC(c2c(CC)non2)=O)(CF)C1 N1(C(c2cc(OC)n[nH]2)=O)CC(C)CN(C(c2cc(OC)nc(F)c2)=O)C(C)C1 Cn1nnc(CNC(c2ncn(C)n2)=O)c1C(N1CC2(CSC2)C1)=O N1(C(c2c(C)nccn2)=O)CCC2CC2(C(=O)N(CCCCO)C(C)C)CC1 c1(C(N2CCCC3(CNC(CCCC=C)=O)C2C3)=O)cc2ccccc2cn1 c1(C(N2C(NC(C3(COC)CC3)=O)C=CC2)=O)ccc(-c2cn[nH]c2)cc1 Cc1nc(C(=O)N(C)CC2CCCN(C(=O)CC3CCC3C)C2)n(C)n1 C1(NC(c2cc(C)c(Cl)s2)=O)CN(C(=O)Cn2nnnc2C2CC2)CCC1O N1(C(CCC#CC)=O)CCC(C(=O)NCC(c2ccccc2)F)C12CCC2 C1(C(=O)OC)CCCCC1C(=O)N(CCC(C(C)C)NC(C1CC2CC2C1)=O)C CC1CC2(CC(C(=O)NC3CCOC3C(=O)NOC3CCOCC3)C2)C1 N1(C(c2c(C)ncnc2)=O)CC(C(=O)NCCOc2cccnc2)C(F)(F)C1 N(C(=NCc1ccc(OC(F)(F)F)cc1)NC1CCC1)Cc1cnc(C)o1 Cc1cc(C(=O)NC2CC2CNC(c2cc(CC(C)C)[nH]n2)=O)ccc1C1CC1 c1(C(=O)NCC(C)CNC(=O)COCC2(F)CC2)coc(C(F)F)n1 C1(C(=O)NC(CCSC)C)(CNC(c2ccn(COC)n2)=O)CC=CC1 Cc1cc(C(=O)N(C2CCCCCC2)CCNC(C2CN(C)CCO2)=O)ccc1Cl N1(C(C(CSCC)NC(C2CC=CCC2)=O)=O)CCCCN(C)CC1 Cc1oc(C2CC2)nc1C(N1CCC(N(C(=O)C(N)=O)CCO)CC1)=O c1(CC(=O)N(C)CCN(C(=O)CCc2ccn(C)c2)C)ccc(C(=O)N(C)C)cc1 N1(C(C2(COC)CC2)=O)CCOC2(CCCN(C(C3CCCC(C)C3)=O)C2)C1 N1(C(CCOCC#C)=O)CC2CN(C(c3onc(C(=O)OC)c3C)=O)CCC12 c1(CC)ccc(C(=O)N(C)CC2CN(C(C3CCCN(CC)C3)=O)CCO2)nc1 c1(C(=O)NC(C(C)NC(=O)CCc2cncs2)C)c[nH]nc1-c1ccsc1 C(C(CO)(CO)NC(c1c[nH]c(=O)cn1)=O)N(C(C(C=C)C)=O)C O=C(C1=CCCN(C(c2ccoc2)=O)C1)NCCC1CCCCC1O C(=O)(C(F)CC(C)(C)C)N1CCC(CNC(C(=Cc2ncn(C)c2)F)=O)CC1 CS(=O)(=O)C1CCCCC1N=c1cccc(S(=O)(=O)NCCF)[nH]1 C12(CC(N3CC(O)(CNC(c4cccc(Br)n4)=O)C3)=O)CCC(CC1)C2 C=CC(C)(O)C(=O)N(CC(C)C(=O)N(CCCC)C)C C=CCC(C(=O)NC1COCC1O)NC(c1cc(C)sc1C)=O c1(CNC(CC(C2CCCCC2)NC(=O)OC(C)(C)C)=O)cc(CC2CC2)on1 N1(C(c2cn(C(C)(C)C)nc2)=O)CCCC(CNC(C2CCCC2(C)C)=O)C1 Cc1ccnc2ccc(-c3cccs3)cc12 N1(C(C=CC(C)(C)SC)=O)CC2CCN(C(=O)CC3COC(C)(C)CO3)C2C1 c1(CCC(N2CCC(N(C)C(C3(F)CCOC3)=O)C2)=O)cn(C)c2ccccc12 C1(O)(CN(C)C(c2coc(C(F)F)c2)=O)CCN(C(=O)Cc2cn(C)cn2)CC1 Cc1cc(Br)c(C(N2CCCC23CCC3)C(=O)NCCCF)cc1Cl C12(CC(=O)N(C)Cc3ccccc3F)CCC1CN(C(c1ncccc1N)=O)C2 C1(O)(CN(C(C=C(C)C)=O)C)CN(C(C2(F)CCCC2)=O)C1 N1(CC#CC)CCC(C2CCCN(C(C3CCC=CCC3)=O)C2)C1 N1(C(c2c(OC)n[nH]c2)=O)CCC2(CCC2)C(NC(=O)C(C)(CC)OC)C1 N1(C(CC=CC)=O)CCC2CCN(C(c3ccc4c(c3)C(=O)NC4)=O)CC12 CC1(NC(c2ccc(CF)cc2)=O)CCCC1NC(=O)CCCN1CCOCC1 c1(NC(C2CCN(Cc3cncc(OC)c3)C2)=O)ccc(C)c(OC)c1 c1(C(=O)NCC2(CO)CCN(C(C(C)S(N)(=O)=O)=O)CC2)cc(F)cc(F)c1F C(=O)(C(C)C(C)NC(=O)OCC1(CCOC(C)(C)C)CC1)Nc1c(OC)ccs1 c1(C(=O)OC)cc(=NCC2(NC(=O)CC3CCC4(CCC4)O3)CCOCC2)[nH]cn1 c1(CC(C(=O)NCCN(C(=O)CCC2CCOC2)CCC)C)ccc(OC)cc1 S(=O)(=O)(c1ccc(Cl)c([N+](=O)[O-])c1)N1CCC2(N(C(C3CCCS3)=O)CC2)CC1 c1(OC)cccc(C(c2cccc(OC)c2)NC(=O)CC2COC(C)(C)C2)c1 c1(C(=O)OCC)c(NC(C2CCN(C(=O)C(C)CC(N)=O)CC2)=O)sc(C)c1C Cc1cc(C(=O)N(CC(C)O)CCNC(C2CC(C)(C)CO2)=O)ccc1[N+](=O)[O-] O=C(CCCCCC1CC1)NCC1CCCN1C(=O)CCc1cncs1 C1(C(CO)NC(c2cc(C(F)F)no2)=O)CCN(C(C2(CO)CC2(F)F)=O)CC1 c1(NCc2c(F)ccc(N)c2)cc(=NCC(=O)NC2CCCC2)[nH]cn1 N1(C(CNC(=O)OCC)=O)CC(NC(c2ncc(OC)cc2F)=O)CC(O)C1 N1(C(C(=O)NC)CC(C)C)CCOC(C)(C)C1(C)C N1(C(=O)Cc2cnsc2)CCC2(CCO2)CC1 N1(C(C23CCC(OC)C2CC3)=O)CCCC2(CCCN2C(=O)C=CCF)C1 C1(CNC(C2N(N=O)CCC2)=O)CC2CCC1N(C(C1CC(=C3CCC3)C1)=O)C2 C(=O)(C(C)C(C)S(C)(=O)=O)N1C(CN(C(c2c(C)n(C)cc2)=O)C)CCC1 N#Cc1ccc(O)c(CN2CCCC(C(=O)NCc3cnc[nH]3)C2)c1 C1(C(=O)NC2CC(NC(=O)C(c3ccc(F)cc3)=O)C2)CC2CCC1C2 Nc1ccc(S(N)(=O)=O)cc1NC(c1cc(-c2ccccc2)ccn1)=O CCC1=NOC(C(N2CCC(N(C(=O)CC(F)(F)F)CC)C2)=O)C1 C1(NC(CN(c2ccccc2)C)=O)CN(C(c2cc(O)nc(Cl)c2)=O)CC1(C)C c1(CCCC(C)C)nc(CCC2CCCN2C)nn1CCc1cnc[nH]1 c1(C(=O)NC2C(NC(C(C)O)=O)C2)cn(C)nc1-c1cccs1 c1(N(C)C)cccc(C(=O)NC2(CNC(=O)COCCF)CCCC2)n1 Cc1n[nH]c(C)c1CC(=O)NCCC1CCCN(C(C2CCOC(=O)N2)=O)C1 c1(C(=O)NC2CCC(CNC(=O)CCCCCl)CC2)n[nH]c2ccccc12 N1(S(=O)(=O)CC2COC(=O)C2)CCCC(N(c2cc(O)ncn2)CCO)C1 CN=c1nc(C(N2CC(NC(C3C(F)(F)C34CCC4)=O)C(O)C2)=O)cc(C)[nH]1 C1(COC)(NC(=O)CC(C)n2cccn2)CCN(C(=O)C(C)(C)c2cnsc2)C1 C(CC(C(=O)N1CC2CC1C2NC(=O)C=CCO)N(C)C)SC CC(=O)CC(C)(C)CC(=O)N1CC(NC(=O)C=Cc2cn[nH]c2)CC1C C1(NC(=O)CC(C2CC2)C2CC2)CCC(NC(c2cccnc2S)=O)CC1 c1(CCC(=O)N(CC(=O)NC2COCC2O)CC2CC2)nc(O)n[nH]1 Cc1ccc(C(N2CCCCC2CNC(C2(CC3CC3)CCC2)=O)=O)c(O)c1 N#Cc1ccnc(NCc2ccccc2-n2nccn2)n1 N1(C(c2cnc3ncccn23)=O)CCCC2(CCCCN2C(c2ccsc2)=O)C1 C(=O)(C1=NN(C)C(=O)CC1)NC1C(CNC(CCCC(=O)N(C)C)=O)C1 N1(C(C2(C#N)CCOC2)=O)CC(CC(N2CCCC(O)(CO)C2)=O)C2(CC2)C1 C(=O)(C(F)CCC(C)C)NC1C(C(=O)NCCC)CCCC1 N1(C(c2cn(C)c(=O)cn2)=O)CCCC(C2CN(C(=O)C(F)n3ccnc3)C2)C1 c1(C(N(C(C(N2CC3(N(C)CC3)C2)=O)(C)C2CC2)C)=O)cnn2ccc(Cl)c(F)c12 C1(CNC(C=C(COC)C)=O)CN(C(c2ccn(C3CCOCC3)n2)=O)C2CC12 N1(C(=O)N)CC(C(C)(C)C)CC(CN)C1.Cn1cc(-c2csc(C)n2)cn1 C(=O)(C(CCC1CCC1)N1CCC1C(N)=O)N(C1COCCC1O)C(C)C c1(C(C)NC(CN(C(=O)CCc2ccn(C)n2)CCC)=O)ccnc(C)n1 c1(C(N(CC(C)NC(COc2c(C)cccc2)=O)C)=O)cnccc1C#N CCC(C)CCCC(=O)NCCOCCCN(C(=O)Cn1cc(C2CC2)cn1)C CCCCCC(C)(CC)C(=O)NC1CCN(C(=O)C(C)(C)CCC(=O)OC)C1 c1(C(=O)NCC2(C)CCN(C(=O)C(F)C3CCOC3)C2)ncc(C#N)cc1Cl c1(C(NOCC(N2CC(C=C)C2)=O)=O)ccnc(C)c1 c1(Cc2cccc(C(=O)NCC(C)NC(CCC)=O)c2)cccc(C)c1C Cc1cc(C)c(CC(N2CCC(N(C(=O)C(C(C)C)c3ccncc3)C)C2)=O)s1 c1(C(N2CC(NC(C3SC4C=CC3C4)=O)(CO)C2)=O)ccc(CO)cc1 C1(OC)CCn2cc(C(N3CCC4(C3)CN(C(=O)C(=O)NC3CC3)C4)=O)nc2C1 C1(NC(C(=O)NC)=O)CCN(C(=O)CCCC2(C)NC(=O)NC2=O)C12CCCC2 n1(CC(=O)Nc2ncnn3cc(Br)cc23)ccc(=O)c2ccccc12 c1(CC)nc(C)c(C(=O)NCc2ccccc2CN(C)C(C2CC2[N+](=O)[O-])=O)s1 N1(Cc2nn(C)c(=O)n2C)CCC2(NC(C3CC3(C)C)=O)CCCC12 N1(C(C)=O)CC(CC(=O)NOC(CC(F)(F)C(C)C)=O)C(C)C1 C1(O)(CNC(CCN(CC=C)C(c2ccnc(NC)c2)=O)=O)CCC(C)(C)C1 c1(OC)cc(OC)c2c(NC(C3CCC4(CC3)CC4N)=O)ccnc2c1 c1(C(C)NC(c2n(CCCSC)nnn2)CC2CC2)ccccc1Br N1(C(c2c[nH]cc2C(F)(F)F)=O)CC2(CCN(C(C3CC4CCC(C3)S4)=O)C2)C1 c1(C(N(C2CCN(C(C(C(C)C)F)=O)C2)CCO)=O)ccc(Cl)cc1F c1(C(C)C)ccccc1CC(=O)NCC(O)CN(C(=O)Cn1ncccc1=O)C CCC(C)(CCC(C)C)C(=O)N1CC2C(NC(=O)C(=O)C3CC3)C2C1 N1(C(c2c(C)nc(C)o2)=O)CCC2(CC(O)c3ccccc3O2)C1 c1(CC)nc(=N)[nH]cc1C(=O)NC1(CCO)CN(C(=O)CSC)C1 N1(C(c2c(C=O)cccc2)=O)CCc2c(Cl)cccc21 c1(C2C(C(CN3CCC(CC#N)CC3)=O)C2)ccc([N+](=O)[O-])cc1 c1(OC)ccn2ncc(C(=O)NC(CNC(c3sc(C)nc3C)=O)C3CC3)c2c1 C1(Cn2cc(CN(C(c3nc(Cl)cs3)C(=O)NC)C)nn2)CCCCCC1(F)F C1(NC(C2CC(C)C2)=O)CCC(N(C)C(C2CC(=O)C2C)=O)CC1 c1(CC(=O)NC2C(NC(CN(S(CC)(=O)=O)C)=O)CCC2)cccc2ccoc12 C(CCCCC(=O)NC1CC(O)CN(C(c2cccc(O)n2)=O)C1)NC(C)=O S(=O)(=O)(c1ccccc1)NC(C(C)NC(=O)N=c1ncn(C2CCCC2)[nH]1)=O N1(C(C(C)Oc2cccnc2)=O)CCC(NC(=O)C(C2(O)CCCC2)F)C(C)C1 N1(C(Cc2nc(C)c(C)s2)=O)CCC(NC(C2(CO)COC2)=O)C(C)(C)C1 C(=O)(C(C)(O)CC(C)C)N1CC(O)(C(C(N2CCC(OCCC)CC2)=O)F)C1 N1(C(C(C(C)C)n2ccc(C)c2)=O)CCC(C)(NC(=O)CN(C)C(C)C)CC1 N1(C(Cc2c(CC)con2)=O)CCC(CC)CC1C(=O)NCCC(O)C(F)(F)F C1(NC(CCSCC)=O)CN(C(c2cnn(CC)c2Br)=O)CC1(C)C C1(C(=O)NCC(CC)C#N)CCC2CCC1N2C(=O)C=Cc1cnn(C)c1 N1(C(C2(CC=C)CCCC2)=O)C2CCC1C(C)C(NC(C1CCC(F)C1)=O)C2 C1(N(C(CCOC(C)(C)C)=O)C)CCCCC1N(C(=O)C(C)OCCC)C N1(C(c2nc3ccc(OC)cc3cc2)=O)CC(S(=O)(=O)CC(F)(F)F)C1 C(=O)(CCCC(=O)NC1CC1)NCC(CCOC)NC(=O)CC1CC2CC2C1 N1(C(c2c(OC)cnnc2)=O)CC(CNC(C2(C)CCC2)=O)CC(C)C1 C#CCC(C)(C(=O)NCCOCCOC)NC(C1CCC2CC1CO2)=O Cc1cncc(C(=O)N(CCCOCCNC(=O)CC2CC3CCC2O3)C)c1 N1(C(C2(OCC)CCCC2)=O)CCOC2(CCN(C(=O)CC3CC(SC)C3)C2)C1 CCCC(C(=O)OC)NC(=O)NC1CCC(C(=O)OC)C1 N1(C(C2CCCN(CC)C2)=O)CC2CCCC2C1C(=O)N(CCCC(=O)NC)C c1(CNC(C(COC)OC)=O)cccc(F)c1 N1(C(C2(C=C)CCC2)=O)CCC2(CCCCN(C(=O)C(C)(C3CC3)OC)C2)C1 CC(C)(C)CCC(=O)Nc1ccc(F)c(-c2cn(-c3ccc(Cl)nc3)nn2)c1 c1(C(N2CC(C)C(CNC(=O)C3=CCCCCC3)CC2)=O)[nH]cc2c1CCS2(=O)=O CON(CCC(=O)NCC1CCC2(CC2)CO1)C(=O)C1CCS1(=O)=O C1(C(N(C2CC(=C)C2)C)=O)CCCC1CNC(c1n[nH]c(=N)[nH]1)=O N(C(=NCCCC1CCOC1)NC1CCCC1)Cc1c(O)c(F)ccc1 c1(C(N(CCC)CCNC(c2nncn2CC)=O)=O)cc2sc(Cl)cc2[nH]1 N1(c2nnc(C(C)(C)C)o2)CCC(CNC(=O)CC2CC(F)C2)CC1 c1(N(CCCN(C(C2C(CC)OCC2)=O)C)C)nc(O)c2ccccc2n1 c1(N(C)Cc2nccc(C)c2)ccc(S(=O)(=O)N(C)CC2CC2C)cc1Cl C1(C(=O)NCC(C2CC2)OC)CCCC1CNC(c1csc(O)n1)=O CC1(C)CC(NC(C2(Cl)CC2)=O)CN1C(c1cc(Cl)ccc1N)=O O=S(Cc1cccnc1Br)CCCCc1ccccc1 C(=O)(CCC#Cc1ccccc1)NCCCCCCN(C(C=CC=CC)=O)C c1(C(N(C(c2ccccc2)CNC(C(CC)C)=O)C)=O)cc2cccnc2cn1 C1(C)(CNC(C2C(OC)CN(C(=O)CC(=O)N(C)C)C2)=O)CCCC(=O)N1 C(=O)(C(CC(C)(C)C)OC)NCC(C)NC(c1c(CCC)n(C)nc1)=O C1(C(N2C(CN(C(c3c(C)oc(Br)c3)=O)C)CCC2)=O)Cc2nccn2C1 C1(NC(Cn2nc(C)oc2=O)=O)CC(C)CN(C(=O)CCc2nc[nH]n2)C1 Cc1c(C(N2CC(NC(=O)C(C)O)C(C)C2)=O)[nH]c2c1CCCC2 C(C(CO)(CO)NC(c1ccnn1CCF)=O)N(C(c1c(C)c[nH]c1)=O)C C1(NC(=O)Cn2cnc(Br)c2)CCOC2(CCOC2)C1 C1(C(=O)NCC(CNC(C(C=C)O)=O)C(F)(F)F)CC2(C1)CC1(CC1)C2 c1(CC)[nH]c(=N)sc1C(N1CCC(C(C)NC(=O)C(=Cc2ccncc2)C)C1)=O Cc1nc(=O)c2c(C)c(C(=O)NC3COCC3NC(=O)CC(C)F)sc2[nH]1 N1(C(C2(CC)CCCC2O)=O)C2CCC1CC(CNC(C(CC)N(C)C)=O)C2 c1(CC)ccc(C(=O)NC2(CNC(C3CCN(C)C(C)C3)=O)CCOC2)cc1F S(=O)(=O)(c1c[nH]ccc1=NCC(C)(C)OC)NCC(OCC)OCC c1(C(C)CC(=O)N(C)CCN(C(=O)CCc2cc[nH]n2)C)ccc(F)cc1 CCC(C)CCCCC(=O)N1CCCC(NC(=O)COc2cccc(Cl)c2)C1C N1(C(C(C)OCCCC)=O)CCC(OCCN(C(=O)Cc2nnc(O)s2)CC)C1 N1(C(CCCn2cc(C3(C)C(OC)C3)nn2)=O)CCCC1(C)c1cn(C2CCC2)nn1 C1(C(=O)NC(C(C)(C)CO)CO)CCCCCCN1C(=O)CNC=O C1(OC)CC(CNC(C2CN(C3CCOC3)C2)=O)N(C(c2[nH]c(C)nc2C)=O)C1 CCN=c1[nH]cc(C(=O)NCC2CC3CN(C(C4(C)CCCCO4)=O)CC23)s1 n1(CC)nccc1C=CC(=O)N(CC(O)CN(C(=O)C(C)O)C)C C(CC(C)C(F)F)NC(C(CC1CCCC1)NC(C(C)NC(C)=O)=O)=O C1(NC(c2c(OC)noc2C)=O)COC2(CCN(C(=O)CSc3nc[nH]n3)C2)C1 c1(C(=O)NC(C)CCN(C)C(C2CCCC2O)=O)cnc2ncnc(O)c2c1 C(=O)(CCC(C)C)NC1(CNC(=O)C(C2(C)CCCCC2)OC)CC(OC)C1 CCC(CC)C(C)C(=O)N1CCC(NC(=O)CCNC(C)=O)C1 c1(NC(C2N(C(C3(CC=C)CCOC3)=O)C(C)C2)=O)ccc(C)c(Cl)c1 c1(C(N(C(CNC(c2cc(C(C)=O)sc2)=O)C)C)=O)cn(C)c(C)n1 c1(C2C(C(=O)NCCCCC3(NC(C4C(=C)C4)=O)CC3)C2)cccnc1 C1(O)(CCNC(CC=CCC)=O)CCCN(C(c2c[nH]c(=NC)o2)=O)C1 N1(C(C2CN(S(C)(=O)=O)C2)=O)CCCC(C2CN(C(c3ccnnc3)=O)C2)C1 C(=O)(C(C)(O)C(F)(F)F)N1c2nc(-c3csc(C)c3)ccc21.c1(CC2CCNCC2)cnns1 c1(C(=O)NC(CCC)CNC(=O)Cn2nccc2C)c(C)cccc1O c1(C(=O)NC(C(C)NC(c2cccc(CC)n2)=O)(C)C)cc(F)c(O)c(Cl)c1 N1(C(C(CC)C(C)C)=O)CC2CC(NC(C3CCC(N(C)C)CC3)=O)CC1C2 N1(C(CC=CCC)=O)CC(NC(c2c(C(C)C)cnn2C)=O)CC12CCOC2 N1(C(COCCC)=O)CCN(C(=O)Cc2cc(F)cc(Cl)c2)CC1C NS(=O)(=O)c1cc(C(=O)NCC2CCN2C(=O)CC2CCOC2)c(Cl)o1 N1(C(C2(C#C)CCC2)=O)CCN(C(c2cc(F)ccc2Cl)=O)C(CC(F)(F)F)C1 c1(C(=O)NCCC(=C)CNC(C2CC2(Cl)Cl)=O)ccc2c(c1)CCCS2(=O)=O C1(CC(=O)NC2C(CNC(=O)C=CCO)COC2)CC2C=CC1CC2 O=C1OCC2(Br)C(C(N3CC=CC3Cn3cc(-c4cncc(Cl)c4)nn3)=O)C12 c1(C(C(=O)NCCNC(COC)=O)NC(C2CC(=O)C2)=O)ccccc1 C12(C(C)NC(c3coc(CNC(=O)CC(=O)N(C)C)n3)=O)CCC(CO1)C2 N(C1CCc2cccnc21)C(=O)NCCC(=O)O.c1(CN)ccccc1 C1(NC(C(c2cccnc2)C)=O)COCCN(C(=O)CSC(F)F)C1 C1(NC(C(C)(CO)OC)=O)CN(C(c2ccsc2SC)=O)CC2CC12 C12(NC(=O)COC(F)(F)F)COCCC1CN(C(c1cnc3c[nH]nc3c1)=O)C2 c1(C(=O)OC)cc(C(N2CC=CC(NC(=O)C(C)N(C)C)C2)=O)ccc1Cl N1(C(Cn2ccc(C)n2)=O)CC(C(=O)NCCCc2cnn[nH]2)C(C(C)C)C1 Cc1[nH]nc(C(F)(F)F)c1C(N1CCOC(CNC(c2ccc(C#N)s2)=O)C1)=O C(=O)(C1=NOC(C)(C)C1)N1CC(C(C(N2CC(C)=C(C)CC2)=O)O)C1 C=CCCC(C(=O)NCC(O)CN(C)C)NC(=O)C(CO)OC C(=O)(C(C(=O)NCC(N1CC(F)(COCC)C1)=O)C1CC1)NCc1nc[nH]n1 N(C(=NCC1CC(CC(N)=O)CO1)N1CCCC1)CC(C)(C)C c1(C(N(C2CN(C(=O)CC3(O)CCC3)CC23CC3)C)=O)ccc(N)c(Br)n1 c1(CCNC(N)=O)nc(-c2ccccn2)nn1-c1ccccc1F C(CO)(C(C)NC(C1(Cl)CC1)=O)NC(C(C1CC1)SC)=O c1(C(=O)NCC(C)N(C(c2ccnc(C(C)C)n2)=O)C)c(N)cccc1Cl C1(NC(C(C)SCC)=O)CCC(C)(NC(c2cccn(C3CC3)c2=O)=O)CC1 C1(C(N2C(C)(CC(=O)NCCN3C(C)COCC3)CC2)=O)C2CCC(F)(F)C12 c1(C(=O)NC2CC2NC(C2CCS(=O)(=O)N2)=O)ccc(=O)n(CC(F)(F)F)c1 C1(NC(c2cc[nH]n2)=O)CC2CC1N(C(=O)COc1cc(F)ccc1F)C2 C1(C(=O)NCC(N(C(C(C(C)C)C)=O)C)C2CC2)CC(F)(F)CCC1(C)C CC1(C)CCN(C(=O)CCc2nccs2)C(C(N2CCSC3CCC23)=O)C1 Cc1ccc2oc(=NC3CCCC(NC(c4ccnn4CC(C)C)=O)C3)[nH]c2c1 C(=O)(C(C(C)C)n1cnnn1)N1C(C(=O)NCC(COCC)O)C(C)C1 C(=O)(CCCCCCCCC1CC1)N1CCN(C(C2C(=C)CC2)=O)CC1CO C1(NC(C=Cc2cc(OC)ns2)=O)CN(C(=O)C(C)(F)F)CC12CCOCC2 N1(C(c2noc(CC)c2C)=O)CC(F)(F)CC1CCNC(=O)CC1(C)CCCO1 N1(C(CCCC=C)=O)CC=C(CC(=O)NC2CCN(C3CC3)C2=O)CC1 C#CC1CN(C(=O)CCOCCCNC(=O)C(O)CN2CCCC2)C1 N1(C(CC=C)=O)CCC2(CC1)CC2CNC(=O)CC(C)(C)C(=O)OC C1(CC=C)(NC(c2cc(C)ncn2)=O)CCN(C(c2c[nH]nc2CCC)=O)C1 c1(CC(=O)NC(C(C)C)C(C)NC(=O)CCF)ccc2ocnc2c1 Cc1c(CNC(=O)C(C2CCCN(C(=O)C(C)(C)CCF)C2)C)cccc1O N1(C(C=CC=CC)=O)CCC(C(N2CCC(CCCO)C2)=O)CC1 c1(C(=O)NC2CC3(CN(C(c4c(C)nn[nH]4)=O)C3)OC2)ccc2[nH]nc(Cl)c2c1 CC1(O)CCC(CC(=O)NCCCCCNC(=O)Cn2cccc(O)c2=O)CC1 CCC(C)(C)C(=O)C(=O)N1CCC1C(=O)NCC1SCCS1 c1(CC#C)cc(C(N2CCC(CNC(c3cccnc3C(F)F)=O)C2)=O)n(C)n1 N1(C(C(COC)O)=O)CC2(C1)C(NC(c1oc(C)nc1C)=O)CCS2(=O)=O C1(NC(c2c(C)ocn2)=O)CCCCC12CCN(C(=O)C(C)(C)C1CC1)CC2 C(C(C)CN=c1nc(N2CCCC(NC(=O)NC)CC2)cc(C)[nH]1)OCC N1(C(CC(C(N)=O)c2ccc(Cl)cc2Cl)=O)CCC2(CC=CCO2)CC1 N1(C(C=C(C)C(C)C)=O)CCCC(C)(NC(c2cn(CC(=O)N(C)C)nn2)=O)C1 c1(CN(C)C(C2C3CCC2(c2ccc(Br)cc2)C3)=O)ccc(-c2csnn2)cc1 CCC(CC(=O)NC1(CN(C)C(c2nc(Cl)cs2)=O)CC1)OC c1(C(=O)NC(C(CC)C)C(=O)OC)cccc2c1CCC2=O C1(NC(=O)C=Cc2cccc(Cl)c2)CCN(C(c2ccoc2)=O)CCC1CO C1(NC(=O)C=CCNC(c2cnc(Cl)[nH]2)=O)CCN(C2CC2)C1=O CCC(F)(F)CC(=O)NC(C12CCC(CC1)C2)CNC(c1cnoc1C)=O c1(CC(=O)NCCN(C(c2cc(CCCCC)[nH]n2)=O)C)noc2ccccc12 CC(C)(C)C(C(=O)OCC(=O)Nc1cc(Br)ccc1F)C(=O)O C1(COC)CC(CNC(=O)CC2CC(CF)C2)N(C(c2nn(C)cc2C)=O)C1 N1(C(C2C(CNC(=O)CCc3cccnc3)OCC2)=O)CCC2C(C1)C2(F)F C12(C(N3CC(CCNC(c4nc(C(C)C)oc4)=O)C(C)C3)=O)COCC1C2(F)F C12(C(N3C4(CNC(c5c(C)cno5)=O)CCC3CC4)=O)CCC(O)(CC1)CC2 Cn1ncnc1-c1cn(CC2(CNC(C3(Br)CC3(F)F)=O)CC2)nn1 N1(C(C=CC(=O)OCC)=O)CCCN(C(c2cccc(C#N)n2)=O)CC1C C1(C(=O)NC(C2N(C(c3c(CC)nco3)=O)CCC2)C)CC(C2CCCC2)C1 n1(CC)nc(C)cc1C(=O)NCC(=O)NC(C)CC1CCC1 c1(CNC(CN(C)C(C2CCCCC2O)=O)=O)cc2ccccc2[nH]1 CCC(C)CCCC(=O)NC1(C(=O)NCc2cc(C3CC3)no2)CC1 c1(C(=O)NCCC2CCC(NC(C3(C)C(C)C3)=O)C2)ccc(CO)c(Cl)c1 C(CC(C)(C)C)(C(=O)N1CC(C)CC1C(=O)NC12CC(C1)C2)OC c1(CN(C(c2nc(CN(C)C)co2)C(=O)NCC=C)C)ccc(CO)cc1 C1(C(C(=O)N(CCC)CCNC(=O)C=CC(C)(C)SC)OCC)CCCCC1 C12(C(=O)NC(C3(O)CCN(C(=O)C=CCF)CC3)C)CCCC(=O)N1CCC2 C(=O)(C1CCCn2ncnc21)N(C1CCN(C(c2cc(C)c(C)[nH]2)=O)C1)CC C1(C)(CC)C=C(C(=O)NCC=CC(=O)NCCc2ccc(F)nc2)C1 c1(OC)ccc(C=CC(=O)NC(CNC(c2[nH]c(C)nc2C)=O)CO)c(OC)c1 C1(NC(C2CC23CCOCC3)=O)CCSC12CN(C(C1(C(F)(F)F)CCC1)=O)C2 Cc1nn(C)c(C(N2CCC(NC(=O)C(c3ccccc3)NC(N)=O)C2)=O)c1F c1(C(N(CC(C)CNC(=O)Cc2ccn(C)n2)C)=O)ccc2nnn(C)c2c1 c1(C(=O)NC23CC(NC(C4C(C#C)C4)=O)C(OC2)C3)cc(S(N)(=O)=O)ccc1C c1(CNC2CC(C(=O)NCc3cn(C)nn3)C2)ccc(C#N)cc1F C(=O)(C1CCc2cc(F)ccc21)NC(C)CNC(C1C2COCC12)=O C1(NC(CCc2nc(C)c(C)o2)=O)CN(C(C2CCOC2C2CC2)=O)CC1(C)C N1(C(C=Cc2ncc(C)[nH]2)=O)CC(NC(=O)C(C)CF)CC(C)(C)C1 N1(C(c2cc(CC)no2)=O)CC2CC(NC(C3OCC4CCCCC34)=O)C(C2)C1 C(=O)(CC(CNC(NC1=COCC1)=O)CC(C)C)OC C1(C(N2C(CC)C(NC(c3sc(C)cc3Cl)=O)CCC2)=O)CCn2cnnc2C1 C1(NC(C(c2cccc(Br)c2)OC)=O)C2CC1CN(C(C1CC1C#N)=O)C2 c1(C(=O)NCCOC2CN(C(C(C)C3CCCO3)=O)C2)c[nH]c2ncccc12 CC1=C(C(=O)NC2CN(C(c3ccccc3C3CCC3)=O)CC2C)CCCC1 CC(C)CCCC(=O)NCCCC(=O)NCC#CC#CCO c1(C(=O)NCC2(NC(c3c(OC)cnnc3)=O)CCC2)cc2cc(F)ccc2[nH]1 C(=O)(C(C(C)C)n1cc(C)nn1)NCC#CCNC(C(C=CCCC)O)=O c1(SC)ccc(C(=O)NC2CCCC2CNC(=O)COC(C)C)cc1[N+](=O)[O-] c1(NC(=O)C(F)n2cccn2)cccc(NC(C2CC(F)(CO)C2)=O)c1 C1(NC(Cc2ncc(CC)[nH]2)=O)(CNC(=O)Cc2ccccc2)CCCCC1C N1(C(c2ccc(OC)s2)=O)CC2CC(C(=O)NC(C)(CO)C3CC3)C(C2)C1 c1(CNC(c2nccn2C)C)sc(Br)cc1I c1(CC(=O)N(C2CCN(C(C3CCN(C)C3)=O)C2)CC)cn(C)nc1C C=C1CCC(C(=O)NC(C2(O)CN(C(=O)C(C)OC)C2)C)CC1 CCC(CCCC(=O)N1CCCN(C(C)=O)CC1)NC(=O)CCSC c1(C(N2CCN(C(C(C#C)(C)C)=O)CC2C2CCCC2)=O)ncn2ccccc12 C(c1cccnc1)=C(C)C(=O)NC1CC(NC(=O)CC2CCC2C2CC2)C1 C1(C(=O)NC2(CNC(CCOC(C)C)=O)CCCCC2)CCCC2(C1)CC2(F)F C1(NC(=O)NCCCl)CC12CCN(C(c1nnc(C3CC3)s1)=O)CC2 C(=O)(C(C)(F)C(F)(F)F)N1C(CNC(Cn2cc(C3(C)CCCC3)nn2)CO)CC1 C(CCN(C)C)(C(=O)NCc1ncn(C)n1)NC(C1CC(=C)C1)=O C1(C(=O)NCCN(CC)CC)CCCN(C(=O)CCc2ccnn2C)CC1 C1(N(CCOC)C)CC(=O)N(C)C1c1cccc(Cl)c1.c12cc(ncn1)N2 CC1(C)CCCN(C(C2CC3(C2)CC32CC2)=O)C1C(=O)NCc1nc(=O)o[nH]1 Cc1cc(C(=O)NC(C)(CNC(c2ocnc2C2CC2)=O)C2CCC2)cc(C)n1 c1(C(N2C(CNC(CCOCCCOC)=O)CC2)=O)cccc(F)n1 c1(C(N(C2CCN(C(C3CCSCC3)=O)C2)C)=O)cncc(N)c1 n1(CC)ccc(=NC(=O)C2CC(O)CCN2C(=O)C2=CCSC2)[nH]1 Cc1nc(C(C)C)[nH]c(=NCC(C2CC2)NC(=O)CC(C)(O)C2CC2)c1Br c1(C(N2C(CN(C(=O)COc3ccn(C)n3)C)CCC2)=O)cccc[n+]1[O-] C12(CO)CN(N(CC3CCCO3)CC3CC3)CC(CO)(C1)C2 c1(C(CC)C(=O)NCC(C)CN(C)C(c2cn(C)nn2)=O)cccc(Cl)c1 C1(NC(C(C=C)OC)=O)CCCN(C(=O)CC(C)OC)C1 c1(C(=O)NCCC(=O)OC)ccc(-n2cc(C3CC=CCC3)nn2)cc1 c1(CC(N2CCOC(CCNC(=O)C(F)(F)CO)C2)=O)ccc(Cl)cc1F c1(C(N2C(CNC(C(CCN(C)C)O)=O)CC(O)C2)=O)cc2c(s1)CCOC2 c1(COC)nc(Cl)cc(=NCCCC(C)NC(=O)Cc2cnc(C3CC3)[nH]2)[nH]1 C1(NC(c2c(CC)csc2)=O)CCCCC1CNC(c1cnnc(O)c1)=O C1(C)(COC)CC(NC(c2cnc(O)c(C)c2)=O)CN1C(=O)CC1CC(F)(F)C1 C1(C(N2CCCC(CC)(NC(=O)C=Cc3ccoc3)C2)=O)CC12CCCCCC2 CCCCC(C)(F)C(=O)N1CCC(NC(c2cccc(C3CC3)n2)=O)C(C)(C)C1 c1(C(c2n(CCSC)nnn2)NC2CC2C2CCC2)ccc(F)c(C(C)C)c1 C1(C(=O)NC(CC)CO)CCOC1CNC(=O)Cc1csc(C)n1 c1(C(=O)NC2CCN(C(C3CC(CC)C3)=O)CC2)ccc(S(C)(=O)=O)[nH]1 c1(CC)ccc(C(=O)NCCC2CCCN2C(c2ncc(C)cn2)=O)c(Cl)c1 N1(C(c2ccc(OC(F)F)cn2)C(=O)NC(CC)(C)C)CCOC2CN(C)CC12 C1(C(=O)NCc2c(C(N(C)Cc3cocn3)=O)n[nH]c2)CC2CC1CC2O Cc1sc(C(=O)NCC(C)(C)CNC(C2CC3CCC2O3)=O)nc1Br N1(C(C2CCC(C)(C)C2)=O)CCCC(F)(CNC(=O)Cn2cnnc2O)C1 c1(OC(C2(CC=C)CC=CC2)OC)c(C(F)(F)F)cccc1Br C(=O)(C1COc2c(F)cccc21)N1CCC(c2cc(C(F)(F)F)cc(OC)c2)C1 c1(CC)nnc(O)c(C(=O)NC(C)CC(C)NC(C2COCCN2C)=O)c1CC C1(N(C(=O)CC(F)F)C)CCCN(C(c2cscc2C(F)F)=O)C1 C(C(C)(C)C(=O)NCc1ccc(C(N2CCC2C(N)=O)=O)o1)OC C(=O)(CC(C)C(=O)OC)NC1(COC)CN(C(c2ccccc2OC(F)F)=O)C1 C=CCC(C)(C)CN=C(NC1CC1C)NC1CC(c2ccc(F)c(Br)c2)C1 c1(OC)ccc(C=CC(=O)NCC2CCN2C(C2CCCCC23CC3)=O)cc1F c1(CC(N2CC(CNC(C3C(OC)(OC)CC3)=O)C2)=O)coc2cc(Cl)ccc12 C(=O)(CC1CCc2ccccc21)N1CC=C(CCNC(C2CC2F)=O)CC1 c1(C(=O)NC(c2ccccc2)C(C)NC(=O)C=C2CCC2)ccn(C)c(=O)c1 c1(CCC(=O)NCCOC2CCN(C(CCCC#C)=O)CC2)ccc(C)c(C)c1 c1(C(N2CCN(Cc3ccc(OC)cc3Br)C3C2C3)=O)n[nH]c2cccc(F)c12 CCCC(C)(O)C(=O)NC(C)CN(C(=O)COc1ccccc1CC)C C1(NC(c2c(C)cc[nH]2)=O)CCC(n2cc(C3C=CC=CC=C3)nn2)CC1 C1(CCC)CN(C(=O)C=CC(C)CC)CCN1C(c1cn(C)nc1Br)=O c1(CC)ccccc1-n1cc(C(=O)NCCC(C)NC(=O)CCC2CCC2)nn1 N1(C(C2CNC(=O)N2)=O)CC2(CC(NC(=O)C(c3ccccc3)N3CCCC3)C2)C1 C1(NC(CC2CN(C)C2)=O)(CNC(=O)C=CCF)CCOCC1 S(=O)(=O)(c1cccc(C(=O)[O-])c1)NC1CC(C(N2CCC(n3ccnc3)C2)=O)C1 N1(C(c2n(C=C)ncc2)=O)CCCC2(CCN(C(=O)C3=CCCCO3)C2)C1 C1(N(C(C(CSC)C)=O)C)CC2CCC(C1)N2C(c1c(C)noc1C(C)C)=O Cc1ccc(F)c(C(C(=O)O)NC(c2cccc(-c3ccc(Br)cc3)c2)=O)c1 c1(C(=O)NCCC2CCCN(C(C(C)OCC)=O)C2)ccc2c(ccn2C)c1 Cc1ccc(NC(c2cc(F)ncc2NC(c2ccc(Cl)c(I)c2)=O)=O)cc1F C1(NC(Cc2c(C)n(C)nc2)=O)CCN(C(c2cccc(CO)n2)=O)C1(C)C c1(OC(C)C)cccc(CC(=O)NC(C)CCN(C(=O)CC(C)C#N)C)c1 C(=O)(C#CC1CCOCC1)N1C(CNC(c2c(C)ccc(F)c2)=O)C(C)(C)CC1 CC1CN(C(=O)CC2CN(C)C2)CCC1C(=O)NCC1(C)CCN(C)C1 C=CCC(F)(F)C(=O)NCCCN(C(=O)C(c1ccc(F)cc1F)=O)C C1(CNC(C2(CNC(c3n(CC)ccn3)=O)CCCC2)=O)CCC2(CC1)CC2 N12CCC(CC1)N(C(=O)CCn1cncn1)C(=O)C2c1[nH]cnc1C.C1(SC)CC1 C1(OC)CN(C)C(C)(C(N2CCN(CCN(C(=O)C(=O)N(C)C)C)CC2)=O)C1 c1(C(=O)NCC(CC)(C)NC(C2CC2CF)=O)ccc2nccc(C)c2c1 N1(C(C(CC=C)NC(C)=O)=O)CCC(F)CC1C(=O)NCc1[nH]nnc1C Cc1ccc(C(=O)NCC2CCC(C)CN2C(=O)CSCCC(C)C)c(C)c1 C1(CNC(C2(C(N)=O)CC2)=O)CC(C(=O)NCc2cccc(O)n2)=NO1 N1(C(C(C(CC)O)(F)F)=O)CC=C(CC(=O)NC(c2nccs2)C)CC1 CC1CC(=O)NC(C(N2CC(C)(NC(=O)CCOc3ccccc3F)C2)=O)C1 c1(NC(c2nnnn2CC2CCOC2)COC)ccc(OC(C)=O)c(Br)c1 C=CCC(C(=O)N1CCCC1C=CC(N1CC(CO)(OC)C1)=O)NC(C)=O c1(C(=O)NCc2ccc(C(=O)NC3CC(F)(F)C3)cc2)ccc(=O)n(C2CC2)c1 C1(O)(C(N2CC(C3(NC(C4C(C)C4C)=O)CC3)C2)=O)CCCC(C)(C)CC1 C1(C(N2CC3(C(NC(CC(C)n4cccn4)=O)CC3)C2)=O)CC2(C1)CS(=O)(=O)C2 C1(C(=O)NCCC(C)OC)CC2CCN(Cc3ccc(O)c(CO)c3)CC12 C(=O)(CC(=O)N(CC(Cc1ccccc1)NC(C12CCC1CC2)=O)C)NCC#C O=C1Nc2ncc(Br)cc2C12CCC1CC(C(=O)O)(C1)C2 c1(C(=O)NC(CN(C(C(C)CO)=O)C)C)cc2cccnc2[nH]1 C1(C(N2CC(C)(c3cn(Cc4cnoc4)nn3)C2)=O)CCCC1(F)F CC1=CC(CNC(C2(C(C)NC(=O)COC3CCOC3)CC2)=O)SC1 c1(C(N2CCC(N(C(=O)CCc3cnn[nH]3)C)C2)=O)n[nH]c(C2CC2)c1Br Cc1ccccc1-c1ccc(SCCn2cccc2)cn1 C(=O)(C(F)C(F)(F)F)NC(C(=O)N(C1C(C)C1)C)CO CCCCC(C)(F)C(=O)NC1CCOC1C(=O)NCc1ncn(CC)n1 CC(C)C1=CCC(NC(=O)C(C)(C)C(C)NC(=O)CCC2CC2(C)C)CC1 c1(CC)cc(CC(N2CCOCC2CCNC(C2(S(N)(=O)=O)CC2)=O)=O)n(C)n1 c1(C(N2CC(CC(C)NC(CSc3nc(C)[nH]n3)=O)C2)=O)cc(F)cc(F)c1N N1(CC(=O)NCC2CCCC(NC(C3(C(N)=O)CCC3)=O)C2)CCCCS1(=O)=O N1(C(C2N(CC)CC2)=O)CC2CCC(CNC(c3c(C)cnn3C(C)C)=O)C2C1 N1(C(CS(C(C)(C)C)(=O)=O)=O)CCC2(CC1)CCN(C(c1ccc[nH]1)=O)C2 c1(C2(SCC(CC)CNC(C3(NC)CCCSC3)=O)CCC2)ccc(C)cc1 C(=O)(C1=CC2CCCC12)NC1C2CN(C(COc3ccc(C#N)cc3)=O)C1C2 C1(C(=O)NC(C2CCCN2C(=O)CCOCC2CC2)(C)C)C(C2CC2)C1(F)F c12ccc(cc1C(=O)NC1(OCC)CC(c3cn(C)nn3)C1)OC2.OC.OCC c1(C(C)=O)[nH]c2ccccc2c1C(=O)NCCN(C(=O)C1CCc2c[nH]nc21)C CC1CC(NC(c2cn(C3CC3)cn2)=O)CN1C(=O)C(CC1CC1)CC1CC1 C(CC(CNC(=O)CCCc1cccs1)NC(=O)C(C)NS(C)(=O)=O)OC CN1N=CC(CC(N2CCC(OCC(=O)N(C3CCOCC3)C3CC3)C2)=O)C1=O C1(NC(CC)=O)CCC2(CC1)CCN(C(C1CCCN1c1ccncn1)=O)CC2 c1(C(=O)NCC2(COC)CN(C(C3CC(C(F)F)C3)=O)C2)cnn(C)c1C(C)C N1(C(C(C2(O)CN(C(c3c(C)coc3)=O)C2)F)=O)CCCC(N(C)C)C1 c1(-n2cc(C(=O)NC3CCN(CC)C3)nn2)ccc(C)cc1F CCC(CC(C)C)C(=O)N1CCOCC1CN(C)C(C1(OC(C)C)CCC1)=O Cc1nn(C)cc1CC(=O)NCc1ncoc1C1CN(C(c2ccn(C)n2)=O)C1 c1(CC)scnc1C(=O)NCCCN(C)C(C1(c2ccncc2)CC1)=O c1(C(=O)NC2C(OC)CN(C(=O)Cc3cscn3)C2)ccc2nc(O)n(C)c2c1 c1(C(N(CC(CN(C)C(c2ccc(Cl)cc2Cl)=O)O)C)=O)cncc2ccsc12 C(=O)(C(CCc1ccccc1)N1CCOC(CCCC2CC2)C1)NCC(C)C C12(C(=O)NCC(C3CCCCC3)NC(C(CC)SC)=O)CCC(N=[N+]=[N-])C1C2 c1(OC)cc(CN2CC3(CC3)CC2C(=O)NCc2cc(Br)ccc2Cl)cc(Br)c1 c1(N(CCOC)CCNC(=O)C(C)NS(C)(=O)=O)ncnc(Cl)c1C#N C1(NC(CC(=O)NCC#C)=O)CN(C(=O)CNc2ncccn2)CC(F)(F)C1 c1(C(N2CC3(C(NC(c4cc(C)c(F)cc4)=O)CC3)C2)=O)ccc(S(N)(=O)=O)o1 C=CC(C)CC(=O)N(CC(C)NC(=O)C(C)(C)C1CCCC1)C N1(CC(N2CC(CS(C)=O)C2)=O)CCC2(CC1)CC(O)CNC2=O c1(C(=O)NCC2(COC)CN(C(C3CCCO3)=O)C2)ccc(OC(F)(F)F)cn1 C#CC1CC2CCC1N(C(c1coc(CNC(c3ccc(F)c(O)c3)=O)c1)=O)C2 c1(CC)ccc(C(=O)NCC23CC2CN(C(=O)CCC2CC(F)(F)C2)C3)cn1 CC(C)(Cc1ccccc1)C(=O)NCC1CCCCN1C(c1cc(CO)on1)=O Cc1c(C(=O)NC2C=CC(C(=O)Nc3cnn(-c4ccccn4)c3)C2)cnn1C n1(CC)cc(Cl)cc1C(N1CCC(C)(CNC(=O)COCC2CCOCC2)C1)=O C(=O)(CC(C)(C)CNC(=O)CCc1ccncc1)NC(C(C)C)(C)C C1(C(N2CC3(C2)CN(C(C2(CO)CCC2)=O)C3)=O)CCn2nnnc2C1 c1(C(=O)NCC(C2CCOC2)NC(CCCCC#C)=O)ccc2nn[nH]c2c1 N1(C(c2scc(OC)c2OC)=O)CCC(C)N(C(=O)CC2SC(=N)NC2=O)CC1 C(=O)(CCC(=O)N1CC(N2CCCCC2)C1)O.C1(N(C)CC)CCC1C(=O)OC CC(C)CC(C(=O)NCC(F)C1CCC1)NC(C1CN(C2COC2)C1)=O N1(C(C(=O)NCC(F)(F)F)=O)CC2CCC1C(NC(C13CCC(CC1)C3)=O)C2 CC1CN(C)CC(C(N2CC3CC(CNC(c4ccc(N)cc4O)=O)C3C2)=O)O1 c1(-n2ncc(C)c2)ccc(C(=O)NCC2(NC(=O)CN3CC=CC3)CCC2)cc1 C(CCCC(C)(C)C(=O)NNC(=O)C1CCC(F)(F)C1)NC(C1(CC)CCC1)=O CC(CC(=O)N1CCCC1CN(C(=O)CN1CCS(=O)(=O)CC1)C)C(F)F C1(CN(C(C(C)Cn2cccn2)=O)C)COCCN1C(=O)C=Cc1ccc[nH]1 C1(C(=O)NC(CC2CN(C(c3ccc(C)s3)=O)C2)C)CCC(=O)N1C N1(C(c2cc(C)oc2C)=O)CCC(F)(CNC(=O)CNC=O)CC1 c1(NC(C2C(NC(c3c(SC)cccc3)=O)C2)=O)cc(F)ccc1O c1(CCN(CC(C)NC(C2(c3nccs3)CC2)=O)CC)ncccc1O c1(C(=O)NC(C)CNC(c2cc3c(ncn3C)s2)=O)ccc(F)c2cccnc12 C(=O)(C(C)CC(C)(F)F)N1CC(CCC)N(C(=O)C(=O)NCC2CC2)CC1 N1(C(C2C(C)(C)C2(F)F)=O)CCOC(C(=O)NCCOCCC2CC2)CC1 N1(C(c2nnc(CN(C)C)s2)=O)C2CCCC1CNC2 CC(C)(S(C)(=O)=O)c1cn(CCNC(C2(C)CC=CCC2)=O)nn1 c1(C(N(CC(C)NC(CCC#CC)=O)C)=O)c(OC)ccc(Cl)c1F N1(C(C2C=CCC2)=O)CC2(C(N3CC4(C3)CC4(F)F)=O)CCC1CC2 N1(C(C(C=C)(C)CC)=O)CCCN(C(=O)CN(S(C)(=O)=O)C)CCC1 C1(C)(C(=O)NCCCC(C)NC(C2(C(F)(F)F)CC2)=O)Cc2ccccc2C1 CC1CCCCC1OCC(=O)NCCCC(C)(C)NC(=O)Cc1cocn1 c1(CN2C(C(N3CCC(C)(OC)C3)=O)CCCC2)ccc(Br)cc1I C1(NC(C(C(C)O)C)=O)CS(=O)(=O)CC1N=c1ccnc(C2CCCC2)[nH]1 c1(-c2ccc(CNCCS(=O)(=O)NC3CCCCO3)s2)ccc(OC(F)F)nc1 N1(N(C)C)CCC(C(=O)NC(C)(C)COc2ccc(Cl)cc2)CC1 C1(C)(CNC(C(C)Oc2ccccn2)=O)COCCN(C(=O)C(N)=O)C1 C(=O)(CCC(C)CN(C)C)N1CC(CCCCNC(c2cnc(SC)s2)=O)C1 Nc1ccc(S(=O)(=O)N2CCCC2c2nc(C(=O)O)cs2)c(F)c1 C#Cc1cc(C(=O)NC(CC(C)CC)C(=O)Nc2csnc2C)ccc1C C(=O)(CC=C(Cl)Cl)NC1(C)CC(NC(c2[nH]cc(C(C)(C)C)c2)=O)C1 Cc1ccc(C(N2CCCC2CC(=O)Nc2cccnc2F)=O)c(Br)c1 N1(C(C(C)OCC)=O)CC2(CC(CNC(C3(CC4C(OC)C4)CC3)=O)C2)C1 c1(C(=O)NCC2(C)N(C(C(C=C=C)C)=O)CCC2)cc(C)cc2c[nH]nc12 C1(C(=O)NC2CCN(Cc3ccccc3)CC2O)CCn2c(O)nnc2C1 N1(C(c2cc(C(=O)OC)on2)C(=O)NCCC)CCCCC12CCOC2 CC(C)CC(O)C(=O)N(C1CCN(C(C2CC(O)CN2C)=O)CC1)C C1(CC(=O)NOCCF)CCCC(NC(=O)CC2CC(=O)NC2=O)C1 c1(C(=O)NCc2ccc(OC)cc2)ccc2c(C)c[nH]c2c1 c1(C(=O)NC2C(C(C)(C)C)N(C(C3COC(=O)N3)=O)CC2)ccc2snnc2c1 c1(C(=O)NC2CCC(CC(N)=O)C2)cc2ccc(Br)cc2c(=O)o1 C#Cc1ccnc(C(N2CC3(C2)CN(C(=O)CN(c2ccccc2)CC)C3)=O)c1 c1(CNC(C(=O)N(C)C)=O)ccc2c(c1)CCCC2NC(c1cncnc1)=O c1(C(N2CC(C)(C(=O)Nc3cnc(C)c(Cl)c3)C2)=O)c(F)ccc([N+](=O)[O-])c1C C(=O)(C1CCCc2nncn21)NC1(C)CN(C(C(C(C)O)N(C)C)=O)C1 CCN(OC)C(=O)C(C)NC(C1(F)CC=CC1)=O c1(C(=O)NC2(CO)CCN(C(C3COCCO3)=O)CC2)cccc2scnc12 Cc1ncnc(N2CCC(CNC(=O)C3=C(Cl)CC3)C23CC3)c1Br NC(CO)CCC(=O)N1CCCC(c2n[nH]cc2C(N)=O)C1 N1(C(C=CC=CCC)=O)CCC2CN(C(C3(C)CCN(C)C3=O)=O)C2C1 C1(CNC(C2(C=C)CC2)=O)CC2(CO1)CN(C(C1C(C(=O)OC)C1(C)C)=O)C2 C1(CNC(C(CC)NC(C)=O)=O)CN(C(=O)CCCC2CCC2)C2COCC2O1 c1(OC)cccc(C(=O)NCC(CO)NC(C2CC23CC3)=O)c1C N1(C(C(CN(C)C)O)=O)CCN(C(c2[nH]nnc2C2CC2)=O)C2CS(=O)(=O)CC12 c1(OCCNC(C(=O)NC(c2nc(C)on2)C2CC2)=O)cccc2ccccc12 N1(C(C2C(C(=O)OC)C2)=O)CC2CC1C2NC(=O)CCc1ccncc1 CC(C)(C)C1=NOC(C(N2CCC(F)(CNC(C3C4CCC3CC4)=O)C2)=O)C1 C1(C)(C(=O)NCC=CCC(=O)N(C2CC(SC)C2)C)CCOC1C C(C(CC(=O)N1CCC1C)C1CCC1)NC(C1(COC)CCC1)=O N1(C(C(C)NC(C)=O)=O)CCCCC(CNC(c2cc(C(N)=O)co2)=O)C1 c1(C(=O)NC2CN(C(C3CC(SC)C3)=O)CC2C(F)F)ccnn2ccnc12 C1(CC(=O)NC)CN(C(=O)CNC(c2ccsc2)=O)CCN1C(=O)CC(C)C(F)F n1(CCC(=O)NC2(C)CC(NC(CCC(C)OC)=O)C2)ccc(O)nc1=O c1(CC)cc(F)ccc1C(=O)NC1CN(C(=O)Cc2csc(Cl)c2)CC1O C(=O)(C(O)CC(C)(C)C)N1CCN(C(COCc2n(C)ccn2)=O)CC1CO c1(C(C)Nc2ccc3oncc3c2)cc2c(cc1F)NC(=O)CC2 c1(N(C)C)nc(Cl)c(C(=O)NCC2(CNC(=O)CC3CCCS3(=O)=O)CCC2)s1 C(=O)(C(CCCC)N(C)C)NCCC(=C)CNC(=O)CCCc1nc(C(C)C)no1 C1(C(N(C)CC#N)=O)Cc2ccccc2CN1c1ccnc2ccnn12 C1(CC(=O)N(CCC(=O)N(C)Cc2cncnc2)C(C)C)CCCC(C)O1 n1(C2C(OC)CCC2)ccc(=NC(=O)Nc2ccc(CS(=O)(=O)NC(N)=O)cc2)[nH]1 N1(C(C2(CC=C)CCOCC2)=O)CC2CC(NC(C3CC(=O)N(C)C3)=O)C2C1 N1(CC(n2cc(-c3ccc(F)cc3)nn2)C)Cc2ccccc2C1.OC(F)F CC1CN(C(c2sccc2-c2ccc(F)c(F)c2)=O)CCC1CNC(=O)C(N)=O c1(C(N2C3C(NC(C(=O)NCCOC)=O)C(C3)C2)=O)cc(S(N)(=O)=O)n(C)c1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C(=O)NCC(c1ccncc1)C)CCC1CC1 C#CC1(NC(=O)C(C)N(C(=O)COCCN(C)C)C2CC2)CCCCC1 C1(O)(CCCNC(C(C2CCCC2)NC(C)=O)=O)CCOCC1 C(c1ccc(Br)s1)=CC(=O)NC(C)C(C)(C)NC(C1CC1C(F)F)=O C(=O)(C(C)C(C)NC(=O)CN(C(=O)COC)C)N(CCF)CC CC1CC(NC(C2CC3CCCC23)=O)CN1C(c1cccc(C(N)=O)c1)=O Cc1cc(F)c2c(c1)CCN(c1nnc(CC(C)O)n1CC1CCCC1)C2 C1(NC(C(=O)Nc2cccc(C34CC(CC3CO)C4)c2)=O)CC2OCCC2O1 Cc1cc(C(=O)NCC2(Cc3cn(CCN4CCOC4=O)nn3)CC2)cc(C)c1 N1(C(C(COCC)C)=O)CC(F)CC1CNC(=O)COC1CCCCCC1 C(C(C)(O)CNC(C1CCOC1CNC(=O)CSC(C)(C)C)=O)SC C12(NC(Cc3c(Cl)cn(C)n3)=O)COCCC1CN(C(c1cn[nH]c1)=O)C2 C(=O)(C(CC(C)CC)NC(=O)CN(C)C(C)=O)NC(CC#C)C(N)=O Cc1nc2ccc(C(=O)NC(CNC(c3cc4cccnn4n3)=O)CO)cc2o1 C(=O)(C(CNC(C1(Cl)CC1(F)F)=O)CC(C)C)NCc1c(C)n[nH]c1C N1(C(C(C)OCC#C)=O)CCC(NC(c2cnn(CCO)c2C(C)C)=O)C1CC N1(C(CC(C2CC2)NC(C(CC)C#N)=O)=O)CCCC(N=[N+]=[N-])C1 O=S(=O)(c1c(F)cc(Cl)cc1Br)NCCC1=Cc2ccccc2C1 CC(CC(=O)N(CCCNC(C12CC(C)C1C2)=O)CCO)c1ccccc1 N1(C(=O)NC(C(=O)N(C)C)Cc2ccccc2)CCC2(CCOCC2)CC1 C1(C(=O)NC(CC=C)(C)C(F)F)CC(N=[N+]=[N-])CN1C(c1cc[nH]n1)=O C1(CNC(CCC)=O)CC2CCC(C1)N2C(c1ccc(F)c(F)c1)=O c1(OC)c(F)ccc(C(=O)N(CCNC(C2C3CCOCC23)=O)CCOC)c1F N(S(=O)(=O)N1CCCC1C(=O)O)Cc1c(F)ccc(OC)c1F N1(C(C2(NC(C)=O)CCC2)=O)CCC2(CC1)CCN(C(=O)CCC(F)F)CC2C N1(Cc2c(OC)cc(O)cc2)CCC2CN(C(c3scnc3C)=O)CC12 c1(C(N(CC(C)N(C(Cn2c(C)nnn2)=O)C)C)=O)cc2n(n1)C(C)CCC2 C(C(N=[N+]=[N-])C(=O)N(C)CC1CCCN1C(C1(O)CCSCC1)=O)OCC N1(C(c2ccc(CCCC)cc2)=O)CCC(NC(=O)C(C)=CC2CC2)C(O)C1 c1(C(=O)NCCCN(C(=O)Cn2cc(C3CC3)cn2)C)cc(F)c2[nH]nnc2c1 c1(COC)cc(-c2cn(CCCNC(c3cncn3C3CC3)=O)nn2)no1 c1(C(=O)NCC2CN(C(c3nncc(C)c3)=O)CC2C)ccc2ccn(C)c2c1 c1(CN(C(COC(C(C)CN(C)C)=O)=O)C)ccc(F)cc1 c1(C(C(=O)NCC2CCCO2)N(CCC(=O)OC)CC#N)cc(SC)cc(Cl)c1 Cc1cccnc1CC(=O)NCC1(C(=O)N(CCCCO)C)CCCC1 C1(C(=O)NC(CSC)(C)CO)CC(F)(F)CN1C(c1cncc(C#N)c1)=O CCC(CC)C(=O)NCCCCN(C)C(C1C2CCCC12)=O c1(C(=O)NC2CCC(C)N(C(=O)Cn3ncn(C)c3=O)C2)cc2n(c1)CCCC2 C1(NC(C=CCCC)=O)CC(OC)CN(C(C2(c3ccc(Cl)nc3)CCC2)=O)C1 C(=O)(C(C)C(C)n1cccn1)NCCN(C(c1csc(C)c1N)=O)CC c1(OC)ncccc1NCC(=O)NCCOCC(=O)NC(C)C C(=O)(CC(C)CC(C)(C)C)N1CC(C(=O)Nc2cn(CC)nc2)C(O)CC1 CC1CC(C(=O)NCC(F)(F)C(F)F)CCN1C(=O)C(CO)NC(N)=O C1(CNC(C2CCN2C(=O)CC2CCCOC2)=O)(CO)CCOCC1 c1(C(=O)NC(C2N(C(c3n(CC)cnn3)=O)CCCC2)C)cc(C)c(C)c(C)c1 Cc1c(C(=O)NC23CC(n4nnnc4-c4ccccc4)C2C3)ncn1C.C12CCC(F)(C1)SC2 C#Cc1ccc(CC(C)NC(=O)Nc2c(C)ccnc2OCCC)cc1 C(CN=c1[nH]c2cc(Cl)c(S(=O)(=O)NC3C=CCC3)cc2s1)N1CCCC(C)C1 Cc1ncccc1CCC(N1CC2CC2(CNC(C2CCSC2)=O)C1)=O N1(C(c2n(OC)cnc2C)=O)CCCCC(NC(C2(C=C)CCC2)=O)CC1 O=C(C1CCCc2ncnn21)NC1CCN(C(=O)C(F)=CC2CC2)C1C1CC1 CN1CC2(CCN(C(=O)CC3C(NC(c4nocc4Cl)=O)CC3O)CC2)C1 c1(N(C)C(C23CC2CN(S(=O)(=O)Cc2ccccc2)C3)=O)cnc(C#N)cn1 c1(C(=O)NCC#CCNC(c2c(CC(C)C)onc2)=O)ccc(F)c(CSC)c1 CC1(C)COC(CC(=O)NC(C2CCCCC2)CNC(=O)CNc2nccs2)C1 CC(CC(C)(C)C)C(=O)NC(C)CCCNC(=O)C(C(C)(C)C)NC(N)=O N1(C(C2(CC#C)CCC2)=O)CC(NC(C2CC(C#N)C2)=O)C2(CCC2)C1 N1(C(C2CCC(C)C2)=O)CCOC2(CCN(C(=O)C=CCN3CCC3)CC2)C1 c1(OC)c(F)ccc(Br)c1C(=O)OCC1CCCCO1 C(=O)(CS(=O)c1ccc([N+](=O)[O-])cc1)NC1CCN(CC(=O)NC(C)C)C1 c1(C(=O)NCC(CNC(C2(c3cccc(C)c3)CC2)=O)F)nc[nH]c2ncnc1-2 c1(C(N2CCC(CNC(C34CCCC3OCC4)=O)CC2)=O)cc(F)ccc1Cl CCCCCCC(CC)C(=O)NC(C)C(C)NC(c1ccc(C2CC2)nc1O)=O N1(C(c2ccc(CC)s2)=O)CCCC(O)(CN(C)C(C2CCN(C)C2)=O)C1 c1(COC)cc(C(=O)N(C(C(=O)NC2CC3CC3C2)C2CC2)C)ncn1 N1(C(CCCOCCOCC)=O)CC2CCC1CN2C(c1cc(O)nn1C)=O CC1(C(=O)NC2COCCC2NC(C23CCC(CC2)O3)=O)CCS(=O)(=O)CC1 C(=O)(CCCC(=O)NCC(C1CCN(C(=O)CC2C=CCCC2)CC1)O)N(C)C C12(CNC(CNC(CC)=O)=O)CCCC1N(C(c1c(C)nn(C)c1C)=O)CCC2 c1(CC)ccc(C(=O)NCCCC(C)NC(c2ccnn2CCSC)=O)c(Cl)c1 C(CC(C(C)(C)C)NCc1cncc(Br)c1Cl)OC C1(C(=O)NC(CC)C(F)(F)F)CC2CCCC2N1C(=O)C=C1CCCCC1 c1(C(=O)NC(CC)CN(C(=O)CCCNS(C)(=O)=O)C)cc(OC)nc(F)c1 CCC(C)C(O)C(C)C(=O)N1CCCC(CNC(=O)COC(C)(C)O)CC1 C(C)(CCC(F)(F)F)NC.c1(OC)nc(C(=O)NCC2C(=O)N2)co1.C(C)(C)(C)O CC1CN(C(=O)C(c2ccccc2F)N(C)C)CCN1C(=O)OC(C)(C)C C1(NC(C2(NC(C)=O)CCC2)=O)CCC(C(=O)NCC(O)CC(C)C)CC1 N1(CCC(=O)NCCC(CNC(CN(CCC#C)C)=O)O)C(=O)CCC1=O C1(C(N2CCC2CC2CCCCC2)=O)(Cn2cccn2)CCCC1 N1(Oc2ccc(NC(=O)Nc3nc(C(C)C4CC4)on3)cc2)CC(C)OC(C)C1 C1(C)(CC)CC(C(N2CCC(CCOC)(NC(=O)CNC(C)=O)C2)=O)CCO1 c1(NC(=O)NCCC2(CO)CC2)cc(F)cc2c1OCCC2 C(=O)(CCCC(F)(F)C(F)(F)F)N(C)CC1(NC(C2Cc3nccn3C2)=O)CC1 C1(NC(c2coc(Cl)n2)=O)CCC2CN(c3nccc(-n4ccnc4)n3)CC2C1 Cn1c(C(=O)NC2CC3(C2)CN(C(C2CC(=O)NC(=O)N2)=O)C3)cc2sccc12 N1CC2(C1)CN(C(=O)C(C)O)CC(C)(C)O2.CC(C)C(CC=O)C(C)C(C)C N1(C(C(CCC)NC(C)=O)=O)CC(CNC(C2CN3CCN2CC3)=O)C(F)(F)C1 C(=O)(C(C(=O)NC1CC(CNC(c2cc(CO)oc2C)=O)C1)C(C)(C)C)OCC C1(CC(=O)NC(C2CCCCN2C(=O)CC2CCC(C)(C)C2)C)CCCCCC1 C12(NC(C3CS(=O)(=O)C3)=O)CCOCC1CN(C(c1ccc([N+](=O)[O-])cc1)=O)C2 N1(C(C2N(C(C)C)CCC2)=O)CCOCC1CNC(c1ccc(N(C)C)cn1)=O CN1Cc2ccc(C(N3CCC(N(C(=O)CN4CCSCC4)C)C3)=O)cc2C1 N1(C(c2nc(CC)sc2N)=O)CCCC(CNC(=O)C=Cc2ccncn2)CC1 CC1=NS(=O)(=O)NC=C1C(=O)NCC1CN(C(=O)C=Cc2ccc(C(N)=O)o2)C1 CC1CCN(C(=O)CC2CCC(=O)N2)C(CNC(c2cccc(N)n2)=O)C1 CC(C)(C)C(O)C(=O)N1CCCC1CNC(=O)C=Cc1ccc(C(C)(C)C)cc1 CC(C)(C)CCCC(=O)N1CC2CC2(CNC(c2cccnc2OC(F)F)=O)C1 N1(C(=O)CC2CC=CCC2)CCC2CC(C1)CN(C(c1ncccc1F)=O)C2 C1(C(=O)NCC2C(NC(=O)CN3CCCS3(=O)=O)C2)CCC2(CCCO2)CC1 CC1CN(C(=O)C(C2CCCO2)NC(=O)C#CC(C)(C)O)C(C)CO1 c1(C(=O)NCC(C)(CO)NC(C)=O)c(F)ccc(OC(F)F)c1F C12(C(N(C(C)C(=O)NCC)CC)=O)CC(CN(C(=O)CCC3CCCCO3)C1)C2 CC(O)CCCCCC(=O)N1CC2CC(NC(c3cc(F)cc(Cl)c3)=O)CC1C2 N1(Cc2n(C)nnc2)CCC(NC(=O)CC2COC(=O)C2)CC(C)(C)C1 CC1C(=O)NC(C)CN1C(C1CN(C(=O)CN2C(C)CCC2C)CCC1O)=O c1(C(=O)NC2(C)CCN(C(C3(CC#C)CCC3)=O)CC2)c(C)ccc(C)c1O N1(C(N(CC(CC)(F)F)C)=O)CCC(NC(C)(C)C)CC1 N1(C(C2C(OC)CCCC2)=O)CCC(O)(CNC(c2ccccc2)=O)CC1 C#Cc1cc(F)c(C(N2CCOC(CNC(C3(CC)CC3)=O)C2)=O)c(F)c1 C12(OC(=N)O)CCC(C1)CN(C=O)CC(C)CO2.C(CO)OC C1(C(C(=O)NCCC(=O)OCC)N(C)Cc2cc(OC)no2)CCC(F)(F)CC1 C1(N(C2(C)CC3CC3C2)C(c2cn(C)nc2)=O)CCCCC1CNC(C1CCC1)=O CN1CCCC1CCC(N1CC(C(C)(C)O)(CNC(C2CNC(=O)N2)=O)C1)=O C(=O)(C(CC(F)F)NC(C1CC1(F)Cl)=O)NCC1(CO)C(C=C)C1 CCC(CC(F)(F)F)NC(c1ncc(I)cn1)=O N1(C(c2c(OC)cc(C)s2)=O)CC2CN(C(C34CCC(CC3)C(C)O4)=O)CC2C1 N1(C(C=NOC)=O)CCN(CCN(C)C(C2CCS(=O)(=O)C2)=O)CC1 c1(NC(C23CC(Cc4ccc(OCC)cc4)(C2)C3)=O)cc(OC)cc(OC)c1 CON(CCC(=O)NCc1sccc1Cl)C(=O)C(C)C(O)C(C)C N1(C(CC2N(C(CC(C)N(C)C)=O)CC2)=O)CCC(F)(F)C(C)C1 N1(C(c2c(CCC)[nH]cc2)=O)CCCC(C2CC2NC(C2CCCS2)=O)C1 C1(NC(c2c(OC)scc2)=O)CC(NC(C2CCSCC2)=O)C12CCOCC2 c1(C(=O)NC2CC3CCC(C2)N3C(=O)CCOC2CC2)ccc(F)c2occc12 CC1(C)C2CCC(C(=O)N(C3CCN(C(c4sccc4Cl)=O)CC3)CCO)C1C2 C1(F)(C(N2CCC(NC(c3nn(C)c(C4CC4)c3)=O)CC2)=O)C2CCCCC12 c1(C(=O)NCC2C(NC(CCCOCCC)=O)C2)ccnc(NC(C)(C)C)c1 CN1CC(O)CCC1C(N1CC(C(=O)N(CC(F)F)C2CC2)C(C)(C)C1)=O c1(C(=O)NC2CCN(C3CN(C(COCCOC)=O)C3)C2=O)nnc(O)nc1O Cc1c(C(N2CCCC2CC(=O)Nc2cccc(Br)c2O)=O)cccc1O c1(C(N2C(CCCNC(c3c(C)csc3)=O)CCC2)=O)ccc2sc(C)nc2c1 c1(N2CCC(C(N(C)C)=O)C2)nc(=N)[nH]c(=NCCN2CCCC2=O)[nH]1 C1(NC(c2c(C)ccc(C)c2C)=O)CC2(CCC(NC(C3C(C)C3C)=O)CC2)C1 C(=O)(CC1CCc2ccccc21)NCC1(COC)CN(C(=O)C(C)(C)SC)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1C(CC)N(C(C2CN(C)CCO2)=O)CCC1 Cc1nn(CCF)cc1NC(=O)C(C)(C1CC1)N(C)C(C1CC1(C)C)=O N1(C(C(CCOC)N(C)C)=O)CC(CC(=O)NC2CC3CCCC3C2)C2(CC2)C1 C1(C(=O)NC(C)(C)CCCNC(c2ncccc2O)=O)CCc2ncsc2C1 C1(CN(C)C(C2CNC(=O)N2C)=O)CCN(C(C2(C)CCCS2)=O)CC1 N1(C(CSCC)=O)CCC(O)(N(C(=O)COCc2nc[nH]n2)CC)C1 c1(CC(=O)NCC(CC)NC(C(CC#C)(C)CC)=O)ccc(S(C)(=O)=O)cc1 c1(C(=O)OC(C(=O)NCc2ccc(OC(C)C)nn2)=O)cc2c(s1)CCC2 c1(C(N2CCC(C)(CNC(c3ccns3)=O)C2)=O)nc2ccccn2n1 C1(C(N2C(C(C)C)C(C)(C)C2)=O)CCCCCN1C(=O)C(C(C)C)NC=O N1(C(c2cnc(OCC)s2)=O)CCN(C(=O)C(c2cncn2C)O)CC1CCO C1(C(N(CC(=O)NC2CC2)C)=O)COCCN(C(=O)C2=CCOCC2)C1 c1(C(=O)NC2(c3cc(C)on3)CCC2)ccnc(C(=O)NCC#N)c1.C(=O)(C1CC1)N S(=O)(=O)(c1ccc(C(N2CC(CC(C)NC(c3ccsn3)=O)C2)=O)cc1F)NC CC1Oc2ccc(NC(=O)C(N3CCCC4(CCOC4)C3)=O)cc2NC1=O c1(NC(C(CO)NC(CC(C)C2CC2)=O)=O)cccc(N=[N+]=[N-])c1 N1(C(c2n(C)ncc2)=O)CCCC(N(C(=O)CN2CCOC2=O)CCO)C1 Cn1cc(NC(=O)C(Cc2cn[nH]c2)NC(=O)C(C#N)C(C)(C)C)c(O)nc1=O c1(CC(=O)NC2C(C)CCN(C(c3c[nH]c(Br)c3)=O)C2)ccc2nn[nH]c2c1 C1(C)(C(=O)Nc2c(C)nc(F)cc2)CN(C(c2conc2C)=O)C(C)(C)C1 C1(C(=O)NCC2COCC2(C)C)(CNC(CCC2N(C)CCC2)=O)CC12CCC2 N1(CCCC)C(=S)NC(c2ccccc2I)C(C(=O)OCC)=C1C1CCNC1 N1(CN(C)Cc2cccc(CC)c2)C(=O)CN(CC23CCCC2C3)C1=O Cc1ccncc1C=CC(=O)NCC1(C)CN(C(c2cn(C)nc2Cl)=O)CCO1 C(CC1CCC1)(C(=O)NCC1CCC(NC(c2csc(S)c2)=O)C1)OC N1(c2ccnc(C(CC)C)n2)CC2CCCN(C(C3CC34CCOC4)=O)C2C1 c1(CC)csc(C(F)(F)C(=O)NC(C)CCNC(=O)CCn2ccnc2)n1 C1(COC)(CNC(=O)C(N2CCSCC2)C)CN(C(C2(F)CCC2)=O)C1 c1(NC(=O)Cc2csc(Cc3cccc(Br)c3)n2)cccn2ncnc12 Cc1cccn(CC(=O)NC(C)C(C)NC(=O)CC=Cc2ccc(F)cc2)c1=O n1(CCC)c(CN2CC(C(C)NC(C3COC(=O)O3)=O)C2)nnc1C c1(CS(=O)(=O)NC2CCN(C)C2c2ccccc2)cc(Br)ccc1Cl C1(C)(CNC(C(C)NC(C)=O)=O)CN(C(C2(CN(C)C)CC2)=O)CCO1 CC1CN(C(=O)CC2C=CCC2)CCC1NC(C1CC(=O)N(C2CC2)C1)=O CC(C)(F)C(C)(F)CNCc1nnc(C2CC2)n1-c1ccccc1 C1(OC)CCCC(CNC(=O)CCN(CCCO)C(c2ccccc2)=O)C1 c1(OC)cncnc1C(=O)NC1CC(N(C)C(C2CC2C(F)(F)F)=O)C1 C(=O)(C(C)CS(C)(=O)=O)NCCc1c(CNC(C(C)C2CCOC2)=O)nco1 C1(C(N(CCOCCCNC(C(CC)SC)=O)C)=O)CCCNC1=O N1(C(C(C)O)=O)CCCC(C)(NC(=O)COc2ccc(F)cc2Cl)C1 C1(NC(C(C)(C)SC)=O)CC(O)CN(C(c2cnnc(O)c2)=O)C1 c1(C(=O)NCCC2CC(C(N(C3CC(CO)C3)C)=O)C2)cn(CCO)nn1 N1(C(c2c(CC)cc[nH]2)=O)CC2COCC2(C(=O)NCC(C)(F)C(C)(C)F)C1 Cc1ncc(F)c(N(C)CC2CCN(C(c3cnn(C(C)C(C)C)c3C)=O)C2)n1 C(=O)(CS(=O)(=O)C1CCCC1)NC1CCC(NC(CCc2c(C)nccc2)=O)C1 N#Cc1ccc2cc(CNc3c[nH]nc3C(=O)Nc3cccnc3F)[nH]c2c1 CCC(C)(CN(C1CCCC1)C)NC(c1cn(C)nn1)=O C(C)(C)(CN=c1[nH]c(=NCC2CC3(CC(OC)C3)C2)[nH]c2c1CCCCC2)SC c1(C(=O)NCC2(F)CC(NC(c3cccc(O)c3Cl)=O)C2)cnc2ccnn2c1 C(=O)(C1COc2ccc(F)cc21)NC(C(C)(C)C)CCC1CN(C(N)=O)C1 N1(C(C2(CCOCC)CCOC2)=O)CCC2(C1)CN(C(=O)C=CCCC(C)C)C2 Cc1nc(N2CCC(C)(O)C(O)C2)nc2ccc(Br)cc12 C(=O)(C(C)C(=O)N1CCCC1(C)C(=O)NCC(C)NC(=O)OC)NC C123CC1CN(C2)C(=O)NCC3.C1(CC(=O)OC(C)=O)CC2CC2C1 C1(C2CC2)(NC(C(CNC(C2C3CN(C)CC32)=O)CC2CC2)=O)CCOC1 N1(C(C2C(=C)C2)=O)CCCC(CCCC2CCN(C(=O)C3=CCCC3)CC2)C1 CCC(CC)CC(c1nnnn1C1CCC1)NC1COC(CO)C1 CCC(CC(=O)N1CCN(C(=O)Cn2cncn2)C(CC(=O)NC)C1)CC(C)C C(C(=O)NC(COC)C(=O)NCC1(C)CC(C)=NO1)(C(C)C)SCC c1(OCC(=O)NCC2(NC(C(=O)NC(C)C)=O)CCOC2)cc(F)cc(Cl)c1 c1(C(N2CCC(CC(=O)Nc3c(C#N)scc3)CC2)=O)cc(O)c(O)c(O)c1 CCCC(C(=O)NC(C1CCCC1)CNC(=O)C(F)(F)C(F)F)S(N)(=O)=O c1(OC)ncc(C(=O)NC(CNC(c2cccc(N)c2)=O)CO)cn1 c12ccc(cc1)NC(C)C(=O)NCCCNC(=O)C2.C(C)(C)(C)OC(N)=O.S C#CCC(O)C(=O)NC(CC1CCOCC1)C(=O)N(CCC1CC1)CC1CC1 N1(C(C2(C)CN(C(C3(n4cccn4)CC3)=O)C2)=O)CCC2(CC(F)C2)C1 C1(C(N2CC(CC#C)OCC2)=O)CC2(CCN1C(=O)C(O)C1CCCC1)CC2 CCCCCCCC(=O)N1CCC(NC(=O)C(n2cc(Cl)cn2)C)C1CC N(C(=NCCNS(=O)(=O)C(F)F)N1CCC2(CC2)C1)C(C=C)C C1CCc2[nH]c(=NC3CC4CCC(C3)N4C3CC3)nc(N3CCOCC3)c2C1 N1(C(CN(C)C)=O)CCC2(CCCCC2NC(=O)CC2CCNC2=O)C1 C1(NC(COCC=C)=O)CCN(C(=O)Cc2cn[nH]c2)CC1CC c1(C(C(=O)N2CC(CCCCNC(C(C)OC)=O)C2)(C)F)ccc(F)cc1 C1(C(N2CCCC(C)(NC(c3cc(Cl)ncn3)=O)C2)=O)CCn2nccc2C1 N1(C(C(C)=CC)=O)CCCC12CCN(C(c1c(OC)ccnc1O)=O)C2 C1(NC(c2c(C)nnn2C)=O)CCC2CCN(C(C3OCCCC3(C)C)=O)C1C2 c1(C(=O)OC2CN(C(=O)OC(C)(C)C)CC(F)C2)cnc2cc(Cl)ccn12 Cc1sc(S(N)(=O)=O)cc1C(N1CC(N(C(=O)COC2CCC2)C)C(C)(C)C1)=O C(=O)(CCC(=O)NC1CC(CCC(N2CC3CC2CO3)=O)C1)NC CCN=c1[nH]cc(C(=O)NCCN2CCN(C(C3CC3C(=O)OC)=O)CC2)s1 C(=O)(CCC(C)(C)NC(c1n[nH]c(=N)[nH]1)=O)N1CCC(C)(N(C)C)C1 c1(SC)ccc(N2CC(C(=O)NC3CC(NC(=O)C(C)=C4CC4)C3)CC2=O)cc1 c1(C2CC(c3n(CCC4(C)CC4)nnn3)(NCc3cocn3)C2)ccccc1Cl C(C(C)N=c1[nH]c2ccc(Br)cc2s1)NC(c1c(C)cnn1C)=O c1(CN(C)CC2CN(C(=O)Cc3ccc(Br)cc3)C2)c(Cl)ccc([N+](=O)[O-])c1Cl Cc1cc(C(=O)Nc2nccn2Cc2ccc(Br)s2)nc(C)n1 C1(C(N2C(C)C(NC(=O)C=C3CCN(C)CC3)CCC2)=O)Cc2cccnc2C1 c1(C(=O)NC(c2c(C)noc2C)CC(=O)OC)cc(Cl)c(C)cc1OC c1(CNC(C2N(C(Cc3nc(C)on3)=O)C3C(C2)C3)=O)n[nH]c2ccccc12 C1(CC=C)(NC(c2ccc(Cl)o2)=O)CC2CCC(C1)N2C(c1cc[nH]c1CC)=O C(N=C(NCC(C)(C)C)N1CCOC(c2ccc(Cl)s2)C1)c1ccc(C)cn1 C=CCCC(C)NC(=O)C(CO)NC(=O)CC1CC1 N1(C(C(CC=C)(F)F)=O)CC2(C1)SCCC2NC(=O)CN(C(=O)COC)C c1(OCC)oc(C)nc1C(=O)NCCC(C)N(C(=O)Cn1ncn(C)c1=O)C C(CCCC(=O)N1CCC(NC(=O)C(N2CCOCC2)OC)C1)OC c1(OCCOC)cc(-c2cnc(CC)[nH]2)ccc1OCC C12(C(=O)NC3C(CNC(c4ccn(-c5ccncc5)n4)=O)C3)CCCN1CCC2 N1(C(C23CCN(C(c4cccc(Cl)c4)=O)CC2C3)=O)CCOc2ccccc21 c1(C2(NC(c3n(CCCSC)nnn3)C3CCC3)CC2)cccc(C)c1 Cn1c(C(N2CCC2(C)C)=O)ccc1C1COCCN1C(C1SCCCS1)=O N1(C(C2(C#N)CCC2)=O)CCCC(NC(=O)C(c2ccccc2Cl)C2CC2)C1 C1(NC(Cn2c(C)ccn2)=O)CCCC12CN(C(=O)CCC(=O)c1cccs1)C2 C(CC(C)(C)CC(=O)NC(CNC(c1cnn(CC(C)C)c1)=O)CCOC)OC c1(OC(C)C)ncc(C(=O)NC2(C)CC(NC(=O)CN3CCOCC3)C2)cc1Cl C(=O)(C(F)CCC(C)(C)C)NCC1(C(N2CC(F)(F)CC2C)=O)CC(=C)C1 CCC(C)CCCC(=O)N1CC(NC(=O)Cc2cncnc2)CC1(C)C Cn1cc(C2CCCC2C(=O)NCC2(CNC(=O)CCC3CC3CO)CC2)cn1 N(C(=NCC1CCCO1)N1CC2CN(Cc3ccccc3)CC2C1)CC(C)(F)F c1(C(=O)NC(CC=C)CNC(=O)CC(C)C(=O)OC)noc2cc(Br)ccc12 C1(C(=O)NCc2ccc(C(=O)NCC3CC(F)C3)cn2)CC12CCCCC2 c1(C(N2CCC(OCCNC(CC(CCC)C)=O)C2)=O)c([N+](=O)[O-])cnn1C N1(C(c2c(OC)ccs2)=O)CC2CC2(NC(c2ccccc2OC)=O)C1 CC(CCN=c1nc(Oc2ccccc2)cc[nH]1)NC(=O)CC(C)(C)C(F)F C1(C(N2CCC(O)(CCNC(C(=O)NCC)=O)C2)=O)CCCCC12CCC2 N1(C(CC(C)SC)=O)CCC(N(C(=O)C(F)=CC2CC2)Cc2ccccc2)CC1 c1(N2CCC(NC(C3(CO)CC3)=O)C(O)C2)ccn2nccc2n1 Cc1nc(CO)ncc1C(=O)NCC1CCN1C(c1cc(Cl)ccc1Br)=O C1(C)(C(=O)NCC(CNC(C2(C(=O)OC)C(=C)CC2)=O)C)Cc2ccccc2C1 n1(CC(N2CC(C(C)NC(c3c(C)c[nH]c3)=O)C2)=O)c(=O)oc2ccccc12 N1(C(COc2c(CC)cccc2)=O)CCC2(CCN(C(=O)C(C)C(C)CC)C2)C1 C1(C(C)C)(C(=O)NCCOC2(C)CCC2)CCCN1C(=O)C(F)Cl c1(OC)ccc(N(C(c2cncc(OC)c2C)C(=O)NCCC2CC2)C)cc1C c1(C(=O)NC(CCOC)CNC(C2CCC(=O)N2)=O)oc(Br)cc1C C(=O)(C1=C(C(C)(C)C)N(C)C(=O)NC1c1cc(C(=O)OC)ccc1F)OCC CCCCC(CC)CC(=O)N(CCCCN(C(=O)C(c1cn(C)nc1C)C)C)C C(C(F)(F)C(=O)NC1CCN(C2CCN(C(=O)COCCSC)CC2)CC1)OC C(C(=O)Nn1nnc2c1CCCC2)C1N(C(c2c(OC)scc2)=O)CCOC1 c1(OC)nc(N2CC(NC(c3ncccc3OC)=O)CCC2C)cc(C)n1 CC(C(=O)NC1(C)CCN(C(=O)C(F)F)C1)C(F)F c1(CC(=O)NC(C2CN(c3nccc(C#N)n3)C2)C)cccc2ccccc12 c1(NC(C2CC(C)(NC(CCCOCCOC)=O)C2)=O)cc(C)sc1-n1cccc1 N1(C(C(C)(C)NC(=O)C(F)(F)F)=O)CCOCC(NC(C2(CC3CC3)CC2)=O)C1 C(=O)(C(CO)NC(c1sccc1-n1ccnc1)=O)OCC c1(Oc2ccc(COC)cc2)ccc(NC(=O)C(=O)OCCCC#N)cc1F C12(CNC(C3C(C)NC(=O)C3)=O)CC(CO)(CN1C(c1cn(C)[nH]c1=N)=O)C2 Cc1cn2nc(C(=O)NCC3CN(C(C4CC4F)=O)C4(CCC4)C3)cc(C)c2n1 C1(C(C)C)CCN1.C1(C(c2nnnn2C(C)(C)C)(C)OCC)CCN(C)CC1 C=CC(C)(C)CC(=O)NC(Cc1cnn(C)c1O)C(=O)NCc1ccon1 C1(C(=O)NCC2(O)CN(C(C3(c4ncco4)CC3)=O)C2)CC12CCCC2 N1(C(c2c(C)[nH]c(=NCC)s2)=O)CC2CCC(NC(C3SCCCS3)=O)CC2C1 C1(NC(C(C)OC2CC2)=O)CC2(CCN(C(=O)C(CC(F)F)C3CCC3)CC2)C1 C(c1cncc(C)c1)=CC(=O)NC1C(CC)N(C(C2CC(C)C2)=O)CC1 C=C1CC2(C1)CC(C(N1CCC(C(C)NC(=O)C(C)(C)OCC)C1)=O)C2 C(=O)(C1CCOc2ccc(F)cc21)N1C(C)CN(C(=O)COC2CC=CC2)CC1 CC1CC(C(=O)NCC2(NC(C3CC(O)C3)=O)CCCCC2)CC(=O)N1 c1(C(N2C(CNC(C(CCCC)C)=O)C(C)CC2)=O)cc2c(F)ccc(F)c2s1 CC(C)S(=O)c1ccc(C(=O)NCC2CCC2NC(C2CCC(C)CC2)=O)cc1 N1(C(c2ccn(C3CC3(F)F)n2)C(=O)NCCCCCC)Cc2cncnc2C1 N1(C(C(C2CCN(C(c3ccc(OCC)cc3)=O)C2)C)=O)CCC(O)C(F)C1 C1(C(=O)NCC(CC)NC(=O)C=C(C)c2ccsc2)CC2(CCC2OC)C1 C1(OC)CCCCC1C(N1CC(OCCC(=O)NCc2cnccn2)C1)=O N1(CCc2nnc(-c3ccc(OC)c(Br)c3)o2)CCCc2ccccc21 Cc1ncc2n1CCC(C(=O)NCCC(C)NC(=O)CCS(C)=O)C2 C1(NC(CCOCC)=O)CC(NC(C2CCN(CC(C)C)CC2)=O)C12CCC2 c1(C(=O)NCC=C2CCN(C(C3CC(C)(C)C3)=O)CC2)nc(O)nc(O)c1F N1(C(C2(C)CC=CCC2)=O)CC2CCC(C1)N2c1nc(Cl)ncc1C(N)=O CCC(CCC(=O)N1CC(c2ccccc2)(NC(=O)CCCC(C)C)C1)OC C(=O)(CC(C)C(C)(C)NC(=O)C(C1CCC1)OC)NCC1N(C(C)=O)CCC1 N1(CCC)C(=O)CCC1C(=O)NC(CNC(=O)Cc1cn(CC)nn1)C(C)(C)C C1(N(C(=O)C=C(C)C2CC2)CC)CCN(C(c2sccc2OC)=O)C1 CC(C)(N=[N+]=[N-])C(=O)N1CCC1C(=O)NCC1Cc2nccn2C1 C1(CNC(C(=O)N(C)C)=O)CN(C(c2ccc(C#N)cn2)=O)CCC1C(F)(F)F N1(CC(=O)OC)CCCN(CCOCC2(C(F)(F)F)CCNC2)CC1=O C1(OC)COCCC1CC(N1CCCC1(C)CNC(=O)C=C(C)C(C)C)=O N1(C(C=Cc2ccc(=N)[nH]c2)=O)CC2(CCN(C(C3(CF)CC3)=O)C2)C1 c1(N2CC(CNC(c3ccc(F)s3)=O)OCCC2)ncnc2scnc12 N1(C(C2C(CC)C2)=O)CC2OCC(NC(=O)CN3CCC(F)CC3)C2C1 C(C(CC(C)C)C(=O)NCc1cccs1)NC(C(n1c(C)ncc1)C)=O N1(CC)CCCC(CNC(=O)C(c2ccccc2C)NC(=O)OCC(C)(C)C)C1 N1(C(C(c2cnn(C)c2)C)=O)CC2CC1C2C(=O)Nc1cn(C)nc1C(C)C Cc1cc(C(=O)NCC2CCCC(NC(=O)Cc3ccsn3)C2)cnn1 C1(NC(CCSC)=O)C(C)CCN1C(=O)C(c1csc(C)n1)=O.C1(=O)NO1 N1(C(C(C)Oc2ccccc2O)=O)CCC2C(CCN2C(c2cncs2)=O)C1 C1(O)(CCNC(C2CCCS2)=O)CCCN(C(C2SCCCS2)=O)C1 C(=O)(C(F)C(C)CNC(C12CC(CO)(C1)C2)=O)N(C)Cc1c(C)ncs1 C(CC1=CCN(C(=O)CCCC(=O)OC(C)(C)C)CC1)NC(CN1C(C)CC1)=O Cc1[nH]nc(C(=O)NCCCN(C)C(C2COCC2(C)C)=O)c1[N+](=O)[O-] N1(C(C)C)CC(C(=O)NCCC2(NC(C3CC4CCC3O4)=O)CCC2)CC1=O N1(C(C(C)SCCCC)=O)C2CCC(C2)C1CNC(c1cc(C)n(C)c1C)=O c1(C(=O)NCC(C)(C)CNC(C2CC(O)C2)=O)ccc2c(c1)COC(=O)N2 C1(NC(CCc2c(C)c[nH]c2C)=O)CC2CCC(C1)N2C(c1ccncc1)=O C1(C)(CNC(C(Cn2cncn2)NC(c2cc(CC)no2)=O)=O)NC(=O)NC1=O N1(C(CCc2scc(C)n2)=O)CCOCC(NC(C2(F)CCOC2)=O)C1 c1(-c2ccc(OCOC)cc2)ccc2[nH]c(C(=O)NC3(C)CCCCC3)nc2c1 N1(C(C2(C#C)CCC2)=O)CC2CCN(C(c3nc(Br)c[nH]3)=O)CC2C1 N1(C(Cn2cnc(=N)[nH]2)=O)CCC(O)C(NC(C2CCNC2=O)=O)C1 C(=O)(CCC(CF)CF)NCC(c1ccc(C)cc1)NC(=O)CC(C)N(C)C O=C(CS(=O)(=O)C1CC1)NCC(=C1CN(c2ncncc2Cl)C1)F N1(C(c2cc(CSC)c(F)cc2)=O)CCC2CCCN(C(=O)CC(C)(C)C)C2C1 C(=O)(C1=CCCSC1)N1CC(NC(c2c(COC)scc2)=O)C2C1C2 C1(C(=O)NC2CC3(CN(C(C(CC)(C)C)=O)C3)OC2)C2Cc3cc(Cl)ccc3C12 CC(C)CCC(C(=O)NCCF)NC(=O)CC1CSC1 O(NC(=O)CCCC(C)NC(c1c(C)cccc1O)=O)CCOCC=C c1(C(N2CC(NC(=O)Cn3ccnn3)C(O)C2)=O)cc(Cl)cc(I)c1 c1(C(=O)NCC(C)NC(Cc2ccc(CCC)cc2)=O)ncc(C)cc1F N1(C(C2CC(N(C)CC)C2)=O)CCN(C(c2csc([N+](=O)[O-])c2)=O)CC1C c1(C(=O)NC(CNC(C2(OC(C)C)CCC2)=O)C)cn(CC2CCOCC2)nn1 c1(CC)c(C(=O)N(C(C)CNC(C2(C)CCCCO2)=O)C)cccc1F CC1(NC(c2ccn(CC(F)F)n2)=O)CCN(c2ncc(Cl)cn2)C1 c1(CC(=O)NCC2(CCNC(C3CCCC3O)=O)CC2)ccccn1 C=CCC(C(=O)N1CCC(C(N2CCCC(CC)C2)=O)(C(C)C)C1)NC(C)=O O=C(CCCN=c1nccc[nH]1)N1CC2CCCC(C1)N2C(c1ncncc1F)=O N1(CCC(N2CCN(C(C(Br)=C(C)C)=O)C3C2C3)=O)C(=O)NC(C)(C)C1=O c1(C(N2CCN(C(C(=O)NC(CC)C)C)CC2)C)cccc(Cl)c1F C(=O)(C(CC(C)C)NC(N)=O)N1CCC(NC(c2scc(OC)c2OC)=O)C1 c1(C(=O)NC2CCN(C(c3c(N)csn3)=O)C2C2CC2)cnc2nccnc2c1 N1(C(N2C(CC(=O)OCC)COCC2)=O)CCN(C)CC(C)C1 CC1(C)C(NC(=O)COc2ccc(Br)cc2F)C2CCOC12 N1(C(c2c(OC)nsc2)=O)CCC(C2(NC(=O)Cc3cccc(OC)c3)CC2)C1 N1(C(CCC(C)OC)=O)CCC(CNC(c2ccc(C(N)=O)o2)=O)C1(C)C CCCC(C(=O)N1CCC(CNC(=O)C(c2ccc(Cl)c(Cl)c2)O)CC1)C(C)C c1(CC)cscc1C(=O)NC1CC(C)(NC(=O)C(C)OCC2CCCCO2)C1 CC1CC(NC(c2cccnn2)=O)CN1C(=O)CC1CCOCC1 N1(C(C(COCC)NC(c2ccc(Cl)o2)=O)=O)CCOC(CF)C1 C=CC(C)(C)CCN=c1ccnc(N2CCC3CC23)[nH]1 c1(C(N2CCC(CN(C(CC(C)c3ccco3)=O)C)C2)=O)cnn(C)c1F N1(C(C2=CCN(C(c3ccc(C#C)cc3)=O)C2)=O)CC(C)NC(=O)C12CC2 Cc1cccc(C)c1-n1cc(C(C)N(C)C(c2ccc(F)cc2)=O)nn1 CCCCCCCCC(=O)N1CC(n2cc(Cn3cncn3)nn2)(C(=O)OC)C1 C(C(C(=O)NC1CCCC1SC)C(C)(C)C)NC(c1cc(OCC)n[nH]1)=O N#Cc1ccc(NC(C2CCN2Cc2ccc(N3CCCC3=O)cc2)=O)s1 N1(C(C2N(C)CC(O)C2)=O)CCN(C(=O)Cc2cnsc2)C(c2ccccc2)C1 c1(OC)cccc(Cc2nc(-c3n[nH]c(C)c3C)n(Cc3ccccc3)n2)c1 CC1COCCC1n1cc(-c2cc(NC(=O)CC(F)(F)F)ccn2)nn1 c1(C(N2CCN(CCF)CC2)=O)cc2c(s1)CCN(Cc1c(F)cncc1F)C2 N1(C(C=CC(C)(C)SC)=O)CCN(C(=O)C(C)(C)C(N)=O)CC12CCC2 C1(C2CCCN(C(c3ccc(Cl)[nH]3)=O)C2)(NC(CCC=C(C)C)=O)CC1 C(=O)(C1CCc2ccccc21)NCC(C)(O)CNC(=O)CC1CCCSC1 N1(C(CN(C(C)=O)C2CC2)=O)CC2CCCC(NC(C3CCCCC3C)=O)C2C1 Cc1cc(-c2cn(C3CC(NC(C4COCC(C)O4)=O)C3)nn2)ccn1 c1(C(=O)NC(CC(C)NC(c2cc(O)ncn2)=O)C)ncc(Br)cc1Cl C(=O)(C1COc2ccc(Cl)cc21)NCC1CN(C(C2CC(C)(C)OC2)=O)C1 C(=O)(CC(C)C(C)C(C)C)NC1CC(CNC(C2CCC(CCCC)CC2)=O)C1 C(=O)(CC1COc2cc(O)ccc21)N1CC(NC(c2c(C)c(Br)cnc2)=O)C1 C(CC(O)CC(=O)NC1CCCC1NC(C1(C)CCOC1)=O)SC c1(CCC(=O)NC2CNC(C)C2)ccc(C)cc1O.c1(CSCC)ccco1 c1(C(=O)NCC(C)NC(C2(COC)CCCC2)=O)cn2ccn(C)c(=O)c2n1 C(=O)(C1COc2ccccc21)N1CC(NC(c2ccc[nH]2)=O)C2C1CCC2 N1(CCCCNC(C=CCOC)=O)CCCN(C(=O)CC(C)(C)OC)CC1 C1(C(N2CCC(C(C(=O)N(C3(C)CC3)C)F)C2)=O)CC(=O)NC(=O)C1 c1(C(N(CC(CC)NC(C2CSCCS2)=O)C)=O)ncoc1-c1cc(C)no1 c1(C(C(C)C)SC)ccccc1OCC(=O)NC1CC(C)(NC(=O)COC)C1 N1(C(C=COCC)=O)CCC2OCCN(C(c3cccc(N)c3)=O)C2C1 N1(C(c2nccc(CC)c2)=O)CCN(C(c2cc3ncccc3[nH]2)=O)CC1C#N Cc1cncc(C(N2CCC(O)(CNC(C3CCC3C#N)=O)C2)=O)n1 C1(CC)C(C(=O)NCCN(C)CCO)CCN1C(=O)CCC(=O)C1CC1 c1(C(N2CCC3(C(NC(CC=C)=O)C3)CC2)=O)cc2cccc(Cl)c2s1 C(=O)(C1=CCCSC1)NC(CC=C)CNC(C1CCCN1C(C)C)=O C1(NC(C2C(C)CN(C(C3COC(=O)N3C)=O)CC2)=O)CCn2ncnc2C1 C1(NC(C(c2ccccc2)SC)=O)CCSC12CN(C(c1cnccc1C)=O)C2 c1(C(=O)NC(CNC(C(C)NC(C)=O)=O)C(C)(C)C)cc(Cl)ccc1C C#CCC(CC#C)C(=O)NCC1CCC(NC(=O)CC(=O)NCC2CC2)C1 C1(NC(c2cccc(C)c2)=O)CC2CC1CN2C(C1(c2cccc(C)c2)CC1)=O Cn1cc(C(=O)Nc2cccc(NC(=O)CCc3nc(=N)[nH][nH]3)c2)c(C(F)F)n1 CC1CCC(C(c2nnnn2C)NCc2sccc2Br)CC1 C=C1CCC1(C(N1CCC1CNC(=O)Cc1cnn(C(C)(C)C)c1)=O)C(=O)OC C(=O)(CC(CN(C)CC)CC)N1C(CNC(CC2(C(=C)F)CCC2)=O)CC1 C(CC(O)C(F)(F)F)NC(C1(OC)CCN(C(c2cc(SC)oc2)=O)C1)=O C(CNC(c1oncc1C)=O)(CC(C)C)NC(C(C)SCCCC)=O N#Cc1ccc(NCC2(c3ccc(Br)o3)CC2)nc1 C12(C(=O)NCC3OCCN(C)C3)COCC1CN(C(=O)CCS(C)(=O)=O)C2 c1(C(N2CC3CC3(C(=O)Nc3cc(-c4ccccc4)ns3)C2)=O)ccc(F)nc1F C=CC(C)(CCOC)C(=O)NCC1(OC(C)=O)CN(C(=O)CC2CC(N(C)C)C2)C1 CC(C)(C(=O)NCC1(C)CCN(C(=O)C(F)(F)C(F)F)C1)C1=CCS(=O)(=O)CC1 c1(C(N2CC3CC2CN3Cc2ccc(I)cc2)=O)cc(F)c(Cl)nc1Cl S(=O)(=O)(C1CCN(C(=O)C(N2CC(C)(C)C2c2cnn(C)c2)=O)C1)N(C)C C(CCC(C)(C)NC(=O)COCCCN=[N+]=[N-])NC(C(c1ccn(C)c1)C)=O c1(-n2c(C)ccn2)cccc(NC(=O)C(c2cccc(O)c2)N)c1 C(C(CNC(=O)COc1ccc(Cl)cn1)C(F)(F)F)NC(C(CC)OCC)=O Cc1n[nH]c(=NC(C)(C)CCNC(=O)Cc2coc(C(F)F)n2)s1 C=CCN=C(NCC(c1cccc(C#N)c1)O)NCC(C)(C)C1CCCC1 c1(C(=O)NC(CCOC)CNC(=O)C(C)(C)C)ccc2c(c1)NC(=O)C(C)S2 CCC(C(=O)NCCOCCCNC(c1ccc(-c2ccco2)o1)=O)OC c1(CC(C)C(=O)N2CCC(N(CCO)C(c3n[nH]cc3Br)=O)C2)ccccc1F CC(CC(F)F)C(=O)NCC(Cc1ccccc1)N(C(=O)CCNC(N)=O)C N1(C(C(C)N(C(C)=O)C)=O)CC(NC(c2n[nH]c(C3CC3)c2Br)=O)C(C)C1 c1(CN2CC(CC(=O)Nc3n(C)nc(Br)c3)OCC2)cnc(Br)c(F)c1 N1(C(C(=CC2CCCC2)C)=O)CC2CC2(NC(=O)Cc2ccc(Cl)cn2)C1 Cc1[nH]c(=N)ccc1C=CC(=O)N(C1CN(C(C2(O)CCSC2)=O)CC1(C)C)C C1(C2CC2)(NC(c2coc(C3CC3)n2)=O)CCN(C(c2cc([N+](=O)[O-])n[nH]2)=O)C1 c1(C(=O)NC(CNC(c2cc(C)no2)=O)C(C)C)cccn(C)c1=O C(=O)(C(C(C)(C)C)c1ccccc1)N1CC(F)(CN(C)C(c2ccc(Cl)s2)=O)C1 C(c1ccsc1Br)=CC(=O)NC1CC1c1ccc(F)cc1 C1(CCOC)CCN(C(C2C3CN(Cc4ccc(COC)s4)CC23)=O)CC1 C1(CNC(CSCC(=O)OC)=O)CCC(NC(=O)C(c2cccc(F)c2)O)CC1 c1(OCCC)ccccc1CNC(=O)NCc1cnc(Cl)cn1 O=C(NNc1ncnc2cc(Cl)ccc12)c1coc2c(F)cccc12 C1(C(=O)NC2CC(=O)OC2)(CNC(=O)C(=O)NCC(F)F)CCCCC1 Cc1c(Cl)nc[nH]c1=NCC1(O)CCCN(C(=O)C(C)OC(=O)N(C)C)C1 c1(N(C)CC)ccc(C(=O)NC2CCN(C(C3(C)CC=CCO3)=O)C2)cc1 c1(OC(C(=O)NCC(CC)(C)NC(=O)CC2(C)CC2)C)ccccc1Br c1(C(N2CCC(CN(C(CC=C=C)=O)C)C2)=O)ccnc(P(C)(C)=O)c1 N1(C(C(CC)OC)=O)CCC(N(C(=O)C(n2ccc(C3CC3)n2)C)C)CC1 C1(OC)(CNC(c2ccc(CO)nc2)=O)CCN(C(=O)CN2CCCC2=O)C1 c1(C(=O)NCC(c2c(F)cccc2Cl)=O)ccc(F)c(CO)c1 N1(C(C(=O)Cc2cccs2)=O)CCCC12CCN(C(C1CCCN1C1CC1)=O)C2 C1(C(=O)NCc2c(C(=O)NC3CC(CC)C3)[nH]cc2)C(C)(C)C1(C)C n1(CC)cc(C(N2CCC(C)C2CNC(=O)CC2CCC(=O)N2)=O)c(C2CC2)n1 N1(C(C(CC(C)C)=O)=O)CCC(C2CC2)(CNC(C2CC3(C2)CC(F)(F)C3)=O)C1 c1(C(N2C(C)C(NC(c3csc(C4CC4)n3)=O)CC2)=O)cnc2ncccc2c1 C1(CC=C)(NC(c2n[nH]c3c2COC3)=O)CCCN(C(=O)CC2CCCO2)C1 C1(C(F)(F)F)(C(=O)NCC(CC)(C)NC(=O)Cc2sc(O)nc2O)CCCCO1 c1(C(N2CCC(NC(C34CCCN3CCC4)=O)C(O)C2)=O)cncc2sccc12 C#CCC(C)(C)C(=O)NCC1(F)CCC(NC(c2cc(C3CCC3)on2)=O)C1 c1(C(N2CCCC(N(C(C(C)=CC3CC3)=O)CCO)C2)=O)cn(C)c(=O)cn1 N1(C(C(C)=C2CCC2)=O)CCC2(C1)CN(C(=O)C(C)c1ccon1)C2 C(S(=O)(=O)c1ccccc1)c1c(CNC(=O)NC(C)C(F)F)cccc1 CCCC(C)(CCC)C(=O)NCC1(F)CCN(C(C2(C)CC2(F)F)=O)C1 Cc1cccc2oc(N3CCC(C4(NC(C5COCCN5C)=O)CC4)C3)nc12 C#CCC(C)(C(=O)NC1COCC1N(C)C)NC(C1CC2(CC(=O)C2)C1)=O c1(C(=O)NC2C(C)CCN(C(C(CC)N(C)C)=O)C2)c(C)ccc([N+](=O)[O-])c1C N1(C(C2CCN(CC)C2)=O)C2CCC(C2)C1CC(N1CCOCC1C)=O C#CCCCCCC(=O)NC(Cc1cn[nH]c1)C(=O)NC(C)C(C)(C)O Cc1cc(C(c2ccccc2F)NCC2CCCCCC2)ccc1OC(F)(F)F C1(C(N2CC3CCN(C(C4CCCO4)=O)C3C2)=O)CCc2nc(O)nc(O)c2C1 N1(C(C(CSC)(C)C)=O)CC2CS(=O)(=O)CC2(NC(c2cc(C)c[nH]2)=O)C1 CC(C)CC(C)(O)C(=O)N1CC(NC(C2CN3CCN2CC3C)=O)CC2(CC2)C1 C(c1ccc(O)cc1)=CC(N1C2(CNC(C3CC34CCOCC4)=O)CC(C1)C2)=O C(=O)(CC(C)C(F)(F)F)NCC1(C(=O)NCc2c(C)noc2CC)CC(=C)C1 C#Cc1ccc(C(=O)NC(C2CCN(C(c3cncnc3C(C)C)=O)C2)C)o1 Cc1ccc(NC(=O)C2=CCN(C(C3C=CCC3)=O)C2)c(O)n1 CC1CC(NC(=O)NC(Cc2ccccc2Cl)CO)CC(C)S1(=O)=O C1(NC(c2cc(CC)no2)=O)(CF)CCN(C(=O)C(F)OC(F)(F)F)C1 CC1(NC(c2cncc(Cl)n2)=O)CCCN(C(c2c(F)cccc2F)=O)C1 c1(C(N(C2CCCN(C(C(C(CC)C)OC)=O)C2)C)=O)cnc2ccccc2c1 Cc1cccc(C(N2CCC(NC(=O)CC3CC4CCC(C3)C4)C(C)C2)=O)c1F N1(C(CSCC=C)=O)C2CCC1CC(NC(c1cc(Cl)cnc1C)=O)C2 c1(OC)c(Cl)ccnc1NC(N(C(CC(=O)OC(C)(C)C)C1CC1)C)=O C1(N(C(C(CC#C)O)=O)C)CC2CCC(C1)N2C(=O)C(F)C(CC)CC CCCC(C(=O)NC1CCCC1NC(c1nc(C)oc1C)=O)NC(C)=O N1(C(C(C)NC(=O)NC)=O)CCN(C(c2cnc(Cl)s2)=O)C(CC(F)F)C1 Cc1ccc(C(=O)NCC(C)N(C)C(c2cc(-c3ccco3)c[nH]2)=O)s1 c1(CC(N2CC(C)C(NC(c3cncc(Br)c3)=O)C2)=O)ccc2nonc2c1 C1(C(=O)OCC(=O)NCc2nc3c(s2)CCC3)CCCC(O)(C(F)(F)F)C1 c1(C(N2CC(C(=O)NC3CC3F)OCC2)=O)cc2cnccc2[nH]1 N1(C(C(C2CC2)OCC)=O)CCC2(CCN(C(=O)CCc3nc(O)n[nH]3)CC2)C1 C12(CNC(C=C(C)C3CC3)=O)CC(NC(=O)Cc3nc(C)cs3)(C1)C1(CCC1)O2 C1(CCOC)CCN(C(c2ccc(-c3ccc(F)cc3)cn2)=O)CC1 C1(C(=O)NC(c2ccccc2)C(=O)NCC(N2CCCC2)=O)CC=CCC1 c1(NC(c2c(OC)cccc2)=O)cc(NC(=O)C(O)CC(C)C)c(F)cc1F Cc1ccc(OC(C)C(=O)NC2(CNC(c3scnc3C)=O)CCOC2)cc1 CC1CN(C(c2nc(Br)ccc2Br)=O)CCCN1C(=O)C=Cc1ccccc1Br c1(OC)ccc(C(N2CCN(C(=O)C3=CCCOC3)CC2)=O)c(OC)c1Cl c1(C(N(c2ccc(N(S(C)(=O)=O)CCO)cc2)C)=O)ccc(Cl)cc1[N+](=O)[O-] CC1CN(C(=O)C=Cc2ccncn2)CCC1CNC(C1(O)CCOCC1)=O N1(C(CCSC)=O)CCC(NC(c2cc(Cl)c(C)cn2)=O)C(F)C1 O=C1CCC(C(=O)NCc2nocc2C(N2CCC(OCCF)C2)=O)CN1 CC1CN(C(c2cc(C3CC3)[nH]n2)=O)CC2(CCN(C(=O)CCS(N)(=O)=O)C2)O1 C1(NC(C(C=C)(C)CC)=O)CC2CCC1N(C(c1ccc3nccn3c1)=O)C2 Cn1nc(C(=O)NC2CCC3CCN(C(C4CC(O)C4)=O)C2C3)c2c1CCSC2 C1(CNC(CCCNC(CN2CCC(C)C2)=O)=O)CCC(F)(F)C1 c1(C(CNC(CN(C(=O)CC2(C)CC2)CC#C)=O)O)cnc[nH]1 c1(CCCC(N2C(C)(CNC(C3CC4CC4C3)=O)CCC2)=O)cc(F)ccc1F C1(C)(NC(C(CC#C)(C)NC(=O)CC2(C)CCOC2)=O)CCCC(C)(C)C1 N1(C(CSCC)=O)CCC2CN(C(=O)CN(S(=O)(=O)c3ccccc3)C)C2C1 CCCCC(C)C(=O)N(C)CC1CC(C)(C)CCO1.C12CC(OC3CC3)CN1C2=O c1(OC)ccncc1CNC(c1nnnn1C(C)(C)C)C12CC(CO1)C2 N1(C(C(CC)NC(C)=O)=O)CC(C)CCC1C(=O)NCCc1cc(C)ns1 N1(C(c2ccc(C)cc2)=O)CCCC(CCNC(C2(C)CC2C)=O)CC1 C1(N(C(C=CC=CC)=O)C)CC2CCC(C1)N2C(=O)Cc1cc(CC)nn1C c1(C(=O)NC2C(C(=O)NCC(C#C)OC)OCC2)cc(C)c(O)nn1 c1(NC(c2cncc(-c3cc(C)c(C)nc3)n2)=O)cnn2cc(Br)ccc12 c1(C(=O)NCC2C(NC(c3c(OCC)nccc3)=O)C2)ccc(P(C)(C)=O)cn1 c1(CC)c(C(=O)NCCC2COCCN2C(=O)C(CSC)OC)cnn1C CC(CC(F)(F)F)C(=O)N1CC(C)(NC(=O)COC2C#CCCCCC2)C1 c1(C(C)=O)ccccc1NC(=O)C(=O)N(C)Cc1ncco1 C1(NC(CCC(=O)N(C(C)C)C)=O)(CF)CCN(C(c2cc(C(C)C)no2)=O)C1 C(=O)(C(O)CC(N)=O)NCc1c(C(=O)NC(C(=O)NC(C)C)C)scc1 c1(N2CCCC(NC(=O)CCCCCO)C2)ncnc2[nH]cc(I)c12 n1(CCCCC)nc(-c2ccc(N)cc2)nc1Cc1c(Cl)cnn1C C1(CNC(CSC(C)(C)C)=O)CCCC(CNC(=O)C(C)(C)N2CCCC2)C1 C1(CC)CC(C(=O)NCCCOCCCO)CCN1C(C1C2CCC(F)C12)=O N1(C(C(COC)N(C)C)=O)CCCC(N(C(=O)Cc2ncc(C)s2)C)CC1 c1(C(N2CC(OC)(CNC(c3cncnc3)=O)C2)=O)cccc(CO)c1 c1(NC(=O)NCC(=O)NC(CNC(CC)=O)C2CC2)ccccc1.c1(C)ccsc1 Cc1cn2c(=O)c(C(N3CC(C(N4CCC(=O)C(C)C4)=O)C3)=O)cnc2s1 c1(-c2nc(N(C)Cc3cccnn3)sc2)ncccc1F C1(NC(Cc2nc(C)sc2)=O)CC(NC(c2cnoc2C)=O)CC1O N1(C(C2CC(C#N)C2)=O)CCCC(CCNC(=O)Cc2cccnc2)CC1 Cc1coc(C)c1C(=O)N(C1CCN(C(=O)C(C)CF)C1)C C1(C(CNC(C(COCC)C)=O)(C)C)CCN(C(=O)C=CC2CCOC2)CC1 C1(C(=O)NC(C#C)CC(C)C)C(C)OCCN1C(=O)C#CC(C)(C)O N1(C(C2CCC(C)(CC)O2)=O)CCCC(C)(C)C1CNC(C1C(C#N)C1(C)C)=O c1(C(=O)NCC2CCC(C(=O)NCc3cccc(Cl)c3)O2)cc(F)ccc1O C1(C(N(CC(CC)(O)CC)C)=O)CC2(CC(NC(C3CC(C(C)C)=NO3)=O)C2)C1 c1(C(N2CC(Cn3cc(C(C)OCC)nn3)C2)=O)c[nH]n(C)c1=O C(C)(C)(CCCNC(=O)Cn1cnnn1)NC(CN(C(COC)=O)C)=O C(=O)(CCC[N+](=O)[O-])NC1(CC=C)CN(C(C2CCC(=O)N(C(C)C)C2)=O)C1 CN1CCC(N(C2CCN(N(C)C)CC2)C)(CNc2cncn2C)CC1 C1(C)(NC(C(CCN(C)C)O)=O)CCN(c2ncc(F)cn2)CC1 N1(CC)CCCN(C(=O)CC2(CNC(c3cc(C#N)oc3C)=O)CC2)CC1 C(=O)(C1=CCCCC1C)NCCOC(CNC(C(C(=O)OC)C)=O)(C)C c1(OCC)cc(-n2ccnc2)ccc1NC(=O)NCc1nccc(C(F)(F)F)n1 n1(CCC=C)cc(C2(F)CN(C(C3CC(C(=O)OC)C3)=O)C2)nn1 N1(C(C2(C)CC2(Cl)Cl)=O)C2CCC1CC(NC(=O)CCc1ccc[nH]1)C2 C(C)(C(=O)Nn1ccnn1)N(CCC)C(c1ccn(C2CC2)n1)=O c1(C(N(c2cc(OC)ncn2)CC2CNCCO2)=O)c(F)ccc(C)c1Br c1(C(=O)NCC2CN(C(=O)NCc3cnc(CC4CC4)[nH]3)C2)c(Cl)cncc1Cl N1(C(c2cc(C)nc(O)n2)=O)CC(C(=O)NCC2([Si](C)(C)C)CC2)CC12CCC2 C1(F)(Cc2cccs2)COCCN(C(=O)OC(C)(C)C)C1.C1C(O)CSN1C C(=O)(C1=C(C)C(C)(C)OC1=O)N(CCNC(c1cc(C2CC2)cc(F)c1)=O)CC C(c1cc(Cl)ccc1Br)=CC(=O)NC12CC(C1)N(C(C13CCCC1C3)=O)C2 Cc1ccc(C(=O)NC23CC(CNC(=O)CN4C(=O)CNC4=O)(C2)C3)c(N)c1 c1(CC(C(=O)O)NC(=O)CCCCOc2ccc(F)cc2)ccc2c(c1)OCO2 C(=O)(C1=CC2(CN(C(=O)CC3COCC(C)O3)C2)OC1)N1CC(C)OCCC1 c1(C(C)OCC)nc(-c2coc(Cl)n2)n(Cc2cccs2)n1 c1(C(=O)NC(C(C)C)CCNC(=O)Cc2ccon2)cccc2oc(=N)[nH]c12 C1(CNC(C2(CC)CCC2)=O)CN(C(c2csc(=NC)[nH]2)=O)CC(C(F)(F)F)O1 N1(C(c2cccc(NC)n2)=O)CC2(CCOCC2)CC1CNC(=O)CS(C)(=O)=O C(=O)(CCS(=O)(=O)N(C)C)N(CC(CC)NC(=O)Cc1nocc1C)C C1(Cc2nc(COCC)nn2-c2cnc(C)s2)CCCCC1(C)C C1(C(=O)NC2C(CNC(CSCC(N)=O)=O)C2)CC(=O)N(C2CC2)C1 C(=O)(CCCCCC(C)(C)C)N1CC2(CC(CC(N3CC(CN(C)C)C3)=O)C2)C1 c1(CC(O)CN2CCC(O)(c3cccc(Br)c3)C2)ccc(Br)cc1 c1(C(N2CCC(CC=C)(C(=O)NC3CC(C(C)(C)C)C3)C2)=O)cc2occc2[nH]1 c1(CC)nc(C)c(C(=O)NC(CO)C(C)NC(C2CC(c3ccccc3)C2)=O)o1 N1(C(CN(CC#C)C(c2cn(C3CC3)cn2)=O)=O)CC2(C1)CN(CC)C2 C1(C2CC2)(C(N2CC(NC(Cn3c(C(C)C)ncc3)=O)C(O)C2)=O)CC=CC1 c1(C(N(CCCOCCN(C(CCC)=O)C)C)=O)cc(Br)ccc1F C(C)(CC(C)C(F)F)NC(C1N(C(C2CC(O)(CC#C)C2)=O)C(C)C1)=O c1(C(=O)NCC(C2CC2)NC(C(c2ccc(C)cc2)O)=O)c(F)ccc(C)c1F C1(NC(c2ncoc2CC2CCC2)=O)CCC2(CC1)CC2NC(C1CCC1)=O Cc1cc(OC(F)F)ccc1-c1cn(C(C)C(N2COC(C)C2)=O)nn1 N1(Cc2c(F)cc(OC)cc2F)CCCn2nc(C(N3CCOCC3)=O)cc2C1 N1(CCCC(=O)NCCN(C(C2CCSCC2)=O)CC)Cc2ccccc2C1=O N1(C(c2nn(C)c(C#N)c2)=O)CC(C2CN(C(C3CC4(CC4)CO3)=O)C2)C1 c1(OC)ccc(C2CN(CC(=O)NC3CCOC3)CC2N)cc1 c1(C(N2CCC2c2cccnc2)=O)ccc2ccsc2c1 c1(CC)ccc(C(C)CC(=O)N2CC(NC(=O)C(c3ccsc3)N(C)C)C2)cc1 C(CS(=O)(=O)C1CCOCC1)NC(=NCCCOC)NC(c1cccs1)C c1(C(N2CC(NC(c3c(C)[nH]nc3Cl)=O)C(O)C2)=O)c[nH]c2c(F)cccc12 c1(CN(C)C)ccoc1C(=O)N(C(CNC(=O)C(F)n1cccn1)C1CC1)C C(C1=NOC2CN(C(=O)COc3ccccc3)CC12)NC(c1ccnc(C)n1)=O c1(C(=O)NCCCOCCNC(CC=C)=O)nscc1Br c1(C(=O)NC2CCCN(C(CCc3c(C)c[nH]c3C)=O)C2)cc(O)ccc1O C(=O)(C1CCCc2n[nH]cc21)N1CCC(C2(NC(C(=O)N(C)C)=O)CC2)CC1 CCC(COC)C(=O)NC(C)C(CO)NC(=O)CNC(=O)C=Cc1ccccc1 C1(NC(C2(CNC(CNC(=O)OCC=C)=O)CC2)=O)CC12CCCCC2 C1(C(N2C(C(C)NC(c3cnc(O)o3)=O)CCC2)=O)CC2C=CC1C2 C1(C(N2CCN(c3ccccc3)CC2)=O)CC2CCC1N(C(=O)C(F)Cl)C2 c1(C(N2C(C)CC(NC(c3nc(CCC)sc3)=O)C2)=O)cnn2ncccc12 C1(CNC(C2(N(C(c3ccn(C)n3)=O)C3CC3)CCC2)=O)CCNC(=O)C1 C(=O)(C1=C(F)CN(C(C2CCC2C#N)=O)CC1)NC(CC#C)C C(=O)(C(F)(F)C(F)(F)F)NCC1CN(C(Cn2c(C)cnc2)=O)CC1C Cc1cc(C(=O)NC2CCCC2CNC(=O)CC2C=CCCC2)n(C)n1 CC(C)C(O)C(F)(F)C(=O)NCC1CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)CC1C Cc1ccc2nc(C(=O)NC3C4COCC3CN(C(C3COC3)=O)C4)ccc2c1 c1(OC)cn(C)c(C(=O)NCCC(C)NC(=O)C(C)=C2CCCC2)cc1=O C(C(C)(C(=O)N(C)CC1CCCN1C(=O)CN1CCCCC1C)OC)OC N1(CC(COc2cccc(OCC)c2)O)CCSC2(CCCC2)C1 C1(NC(C2C(CCC)CCC2)=O)CCOC(CC)C1 N1(C(C2CN(C)C2)=O)CC(NC(=O)CCc2cc(Cl)cc(Cl)c2)C(F)(F)C1 N1(C(c2n[nH]c(C)c2C)=O)CCC(C2(O)CC(NC(=O)CCS(N)(=O)=O)C2)CC1 CC(c1ccccc1C)=CC(=O)NC(C1CCCN1C(C1CSCC(=O)N1)=O)C CCCCC(C)C(=O)NCCOC1CCN(C(c2nn[nH]c2Cl)=O)C1 N1(C(c2ncccc2Cl)=O)CCC2C1CCCN2C(=O)Cc1cccc(F)c1Cl C#Cc1ccc(C(=O)NCC2CN(C(=O)CCCN(C)C(C)=O)CCN2C)cc1 N1(C(=O)NCc2ccc(C)c(CNC(c3ccco3)=O)c2)CCC(=O)N(C)CC1 CCC(CCC(=O)N1CCC(C(=O)NOCCC(C)C)C12CC2)OC CON(CCC(=O)N(C)Cc1ccc(C)cc1C)C(=O)c1cccn1C C1(C(=O)OC)CCCCN1C(c1ccc(N(C)C)nc1)C(=O)NCC1CCCO1 C1(NC(c2nc(C)sc2C)=O)CC2CC(C1)N(C(=O)CC1CCCCC1(C)C)C2 C(CN=c1[nH]c2c(c(=NC(C)Cc3cnn(C)c3)[nH]1)CCC2)OC(C)C C1(C2(O)CCC2)(CNC(C2C(CNC(C3CC4(CSC4)C3)=O)C2)=O)CC1 N#Cc1ccc(NC(=O)NC(c2ccc(Cl)cc2)CC2CC2)nc1 C1(COC)(CNC(c2cnc(C3CC3)s2)=O)CN(C(=O)C(C)(C)O)C1 CC1CN(C(=O)CSc2ccncc2)CC(C)C1NC(=O)COCc1nccs1 c1(C(=O)NCCCCCNC(c2ccc(C)nc2)=O)ncc(C2CC2)cc1F C1(C)(C(N(C)CCNC(c2ccnnc2O)=O)=O)CCC(O)CC1 C(CCO)(C(=O)NCCC1(NC(=O)CCCOc2ccccc2Cl)CC1)N(C)C c1(OC)cccc2c1CCC2(N)C(=O)NCC(N)CC(C)C C1(CCNC(=O)Cn2ccnn2)(NC(=O)C=Cc2ccsc2)CCOCC1 CN1Cc2c(-c3cnc(C(N4CCC5(CCOC5)C4)=O)nc3)cccc2C1=O CC(C)C(O)C(=O)NCCNC(C1CN(C(C2(S(N)(=O)=O)CC2)=O)C1)=O C1(C(N2CC(F)(CNC(Cc3c(C)con3)=O)C2)=O)Nc2ccccc2C1(C)C C(=O)(C(F)C(CC)CC)N1CC(C(C(=O)NC2(C#C)CCOC2)OC)C1 CC(C)(C(=O)NC1CCC1CNC(c1ccsc1C(F)F)=O)n1cnnn1 CC1CC(NC(=O)CCCn2c(O)nnc2O)CN1C(=O)CCC1CCCOC1 C#CC(C)(C)C(=O)NC(C1CCCN1C(=O)C(C)=CC1CC1)C C#Cc1cccc(C(=O)N(C2CCC(NC(c3cnn(CCC)c3)=O)C2)C)c1Cl CC1C(NC(c2ccco2)=O)CCCN1C(c1ccoc1I)=O c1(C(=O)NCC(CNC(c2c(C)nc(CCC)o2)=O)F)cc(F)c(F)c(F)c1F c1(C(=O)NCCC2CCCCN2C(=O)C(F)C(F)(F)F)ccc2c(n1)CCC2=O c1(C(N2CC(CCNC(=O)C(C)C)(OC)C2)=O)ccc(NC(=O)C(C)(C)C)cc1 c1(CN(C2CCCNC2)CCO)nccc(C2CC2)n1 N1(C(CC(C)OC)=O)CCN(C(=O)CNC(c2nn(C3CC3)cc2Cl)=O)CC1 N1(C(C(C2CCC(=O)N2)C)=O)CC(N=c2[nH]nco2)C2(CCOCC2)C1 N1(C(C(C)OCCOC)=O)CCN(CC(=O)NCC2CCS2(=O)=O)CC1 c1(CCC)nc(=NC(CCN(C(=O)C(C)Cc2cnn(C)c2)C)C(C)C)s[nH]1 N1(C(C=CC2CCN(C(C3(C(C)C)COC3)=O)CC2)=O)CC(=O)N(C)C(C)C1 c1(C(=O)NC2(C)CCN(C(c3cccc(N)c3F)=O)C2)ccc2nc(Cl)nn2c1 c1(N(CCS(C)(=O)=O)C)nc(=N)[nH]c(=NCCN2CC=CC2)[nH]1 c1(CC(=O)NCCC(C)N(C(=O)C(c2cnn(C)c2)C)C)ccc(C(N)=O)cc1 N1(C(c2c(C(=O)OC)ccnc2)=O)CCC2(CCCC2NC(C2(C)COC2)=O)C1 C(=O)(C1=NNC(=O)CC1)N1CCC(NC(C(C)(C)C2CCCC2)=O)CC1C1CC1 CC(C)C1=CCC(C(=O)NNC(C2CCN(C(=O)OC(C)(C)C)CC(O)C2)=O)CC1 CC1CCOCC1C(=O)Nc1cccc(NC(c2cc(C#N)cs2)=O)c1 C1(C(=O)NCC2(C(=O)NCC3CSC3)CC2)CC1C1CCC1 Cc1ccc(C(C)C)cc1NC(c1ccc(OC(F)(F)F)c(-n2cccn2)c1)C N1(C(C(C)N(C)C(=O)OC(C)(C)C)=O)CCN2C(=O)CCCC2C1 c1(C(N2C(CC)CN(C(=O)C(C#N)CC)CC2)=O)csc2ccc(C)cc12 S(=O)(=O)(c1cnc(NCCN(CCS(C)(=O)=O)C)cc1C)N(C(CC)C)C c1(N2CC3CN(Cc4c(C(=O)OC)cccc4)C3C2)nc(C)nc2ccsc12 c1(C(=O)NCC(C)NC(C(c2ccc(Br)cc2)OC)=O)ccc(O)nn1 N1(C(C)C(=O)N(C(C)(C)C)C(C2CC(C)(C(=O)OCC#N)C2)=O)CCCCCC1 N1(C(C(CC)SC)=O)CCC(C)C(N(C(=O)Cc2ccc(C)o2)C)C1 Cc1cc2ncc(C(N3CCC(CNC(c4cnc(S)[nH]4)=O)C3)=O)cc2[nH]1 C(c1ccccc1)=C(CC)C(=O)NCC1CN(C(C2(SC)CC(F)(F)C2)=O)C1 N1(C(C(CC)SC)=O)C2CCCC1CC(NC(C1CC3CCC1O3)=O)C2 c1(C(=O)NC(CC)CNC(=O)CCCSC(C)(C)C)cc(C(F)F)ccn1 c1(C(N2CC3(N(C(C(CCC)C#N)=O)CC3)C2)=O)ccc(OC)c([N+](=O)[O-])c1 C(=O)(CC1CN(C)c2ccccc21)N1CC(C)(NC(CC2CCN(C)C2=O)=O)C1 c1(NC(CC(CC=C)NC(=O)C=CC(C)(C)SC)=O)ccc2nncn2c1 CC1CCC(CNC(=O)Cn2cccn2)N(C(=O)CNC(C2CCCC2)=O)C1 Cn1ccc2c(N(C3CC4CCC(C3)N4)Cc3cc(I)ccc3O)ncnc12 CC1C(C(=O)NC2CC(CO)C2)CCN1C(c1cccc(O)c1)=O N1(C(c2c(CNC(CC(C(C)C)C)=O)noc2)=O)CCc2c(C#N)cccc21 N1(C(C(CCSC)N(C)C)=O)CC2CCN(C(C3CC4C=CC3C43CC3)=O)C2C1 CC1CN(C(=O)COCc2ccnc(C(F)(F)F)c2)CCCN1C(C1CC1F)=O CCCCC(CNC(=O)Cc1ccccc1Cl)NC(c1c(F)cnn1C(C)C)=O c1(OC)ccc(NC(N2CCC(NC(=O)Nc3ccc(I)cc3)C2)=O)cc1 c1(N2CCC3(CCN(C(c4ncccc4Br)=O)C3)C2)ncnc2cccc(F)c12 C(=O)(C(C)NC(C)(C)CC)N(C(CNC(C=CCC)=O)C)C C1(C(C)O)CCCN(C(=O)C(N2CC(O)CC2C2CCC2)=O)C1 Cc1nc(C(=O)NCCCC2CCCN2C(c2ccc(Cl)c(O)c2)=O)cc(O)n1 c1(CCC(=O)NCC(C)N(C(c2cnn(CC)c2C)=O)C)ccc(OC)cc1F CCC(CC)C(C(=O)NCC1CCN(C(=O)C2=NNC(=O)CC2)C1C)OC CC1=C(C(=O)N2CCC2C(=O)NC2(C)CCC(C)(C)CC2)COCC1 C1(NC(C(C)CO)=O)CCC2CN(C(C3CC(n4cnnc4)C3)=O)CC2C1 C1(C(=O)NC(CN(C(CCCCCC#C)=O)C)CC)CCC2(CC1)OCCO2 N1(C(c2occ(C(C)(C)C)n2)C(=O)NC2CCCC2)CCCN(S(N)(=O)=O)CC1 C=CC(O)C(=O)NC1CC(CNC(=O)CNC(=O)OC)C1 C(=O)(CCCC1(NC(=O)CCc2ncnn2C)CCC1)NC(C1CC(C)(C)C1)C C(=O)(C(COC)NC(c1cc(C(C)=O)c[nH]1)=O)N(CC#CC)C C1(NC(C2N(C)CCC2)=O)CCCC12CCN(C(c1cn(C)nc1Cl)=O)CC2 N1(C(CCC(C)N(C)C)=O)CC2CC1CN(C(c1cnn3c1CCC3)=O)C2 C1(CC=C)(C(=O)NCc2ccc(Cl)nc2)CCN(C(c2cn(C)cn2)=O)C1 c1(C(=O)NC2CN(C(C(C)NS(C)(=O)=O)=O)C(C)(C)C2)coc2c(Cl)cccc12 C1(C(=O)NCc2cc(F)ccc2Br)CCC2(CN(C(c3ccc(I)cc3)=O)C2)O1 c1(C(N(C2CCN(C(CN3CC(C)C3)=O)CC2C)C)=O)cn2cccc(F)c2n1 n1(CCC(=O)NC(C)CCNC(C2CSCCS2)=O)cccnc1=O C=C(Cl)CC(C(=O)NCCc1cc(C)no1)NC(c1cc(=N)[nH][nH]1)=O CC1CN(C(C2CCS(=O)CC2)=O)CCN1C(C1(C(F)F)CCCO1)=O C(CC(C(=O)N1CCC(n2ccnn2)C1)NC(c1cc(C)[nH]n1)=O)OC C=CCC(CC(C)C)C(=O)NC1CN(C(=O)CNc2ccccc2)CCC1CO c1(CNC(C2C(O)CCN(Cc3ccc(C)cn3)C2)=O)ccc2c(cnn2C)c1 C1(C)(C(=O)NCC(C(=O)NC(c2cn(C)cn2)C)CC2CC2)CCC(=O)CC1 N1(C(CN(C2CCSC2)C)=O)CCC(C)(CNC(=O)C=C2CCCCC2)C1 c1(CC(C(=O)NC2C(NC(c3n(C)cnc3)=O)C2)O)ccccc1Cl CC1(NC(C2CSC2)=O)CC(NC(c2cc(C(N)=O)co2)=O)C1 C1(C(=O)NCC(=O)NC(C2CCN(C(=O)CCCCO)C2)C)CCC(O)CC1 CC(CN(C)C)CC(=O)NCC(c1ccccc1Cl)NC(=O)CCC1CCC1 CC1(C)CN(C(=O)Cc2ccsn2)CC1CNC(C1CCS1(=O)=O)=O c1(C(=O)NCCC(C)NC(=O)C=C2CCN(C)C2)cc(C(N)=O)co1 N1(C(C(C)(C)OC)=O)CCCCC1C(c1cccc(F)c1)O C1(C(=O)NCCCC(F)(F)F)(COC)C=CCN1C(=O)CSC Cc1nc(C)c(CC(=O)N(CCCNC(c2cn(C(C)(C)C)nn2)=O)C)s1 CC1(C)CC(NC(=O)COCC2CCOC2)CN1C(c1ccon1)=O c1(OC)ccc2c(c1)CCC2C(=O)NC(C)(C(=O)O)C1CCCC1 N1(C(C(C)S(C)(=O)=O)=O)CCN(C(=O)CC2(C3CC3)CC2)CC12CCC2 C1(NC(c2cc(CC)c(C)s2)=O)CN(C(=O)CCC(C)SC)CCC1C(F)(F)F C=CCC(C)(C)CNC(N1CCCCC1Cn1cncn1)=O C1(C(=O)NC(CNC(c2c(C)nncc2)=O)(C)C(C)C)CCC2(CC1)CC2 c12cccc(n1)CN2.C1(CC2C(NC(=O)CCSCCCO)C2)CCCCC1 C1(C(N(CCO)CC)=O)CCOC1CNC(c1cc(C)co1)=O CC(C)(CCC(=O)NC1CCCC(C(=O)NCc2cccc(O)n2)CC1)[N+](=O)[O-] c1(-c2cc(CN(C3C(C)CCC3)C)sc2)ccc2c(c1)NCCC2=O C(=O)(C(C)(C)C(C)NC(C1CC2(C1)CC2(F)F)=O)N(CC(COC)(F)F)C Cc1c[nH]cc(C(=O)N(C2CCCN(C(=O)CCN3CCCCC3)CC2)C)c1=O N1(C(C2CC(O)(CC#C)C2)=O)CCC2CCN(C(c3ccc([N+](=O)[O-])s3)=O)C2C1 Cc1cc(Br)cc(F)c1C(=O)NC(=O)C(Cl)(Cl)Cl C(CCC(C)(C)NC(=O)CCn1cccn1)NC(C1C(C)CCS1)=O C1(CNC(c2cnc(COC)s2)=O)CN(C(=O)CC=C(C)C)CC1(C)C C1(NC(c2n(C)nc(C)c2Cl)=O)CC2CCC(C1C)N2C(=O)CN1CCCCC1 C1(c2c(OC)n(C)nc2)C2=C(C(C)N(C)C2=O)N(C)C(=O)N1C C#Cc1cc(C(=O)NC(C)(CO)C(=O)NCCOCCCO)ccc1C CCCS(=O)(=O)C(C)C(=O)N1CC2(CCCN(C(=O)CC3CCOC3)C2)C1 C1(NC(CC2CC(N(C)C)C2)=O)CC12CC(NC(c1ccnnc1)=O)C2 N1(C(CNC(=O)OCC=C)=O)CC(NC(c2cc(CC)oc2C)=O)CC1C O(NC(=O)C(F)C1CCN(C(c2ccncn2)=O)C1)C(C)C O(NC(=O)C=CCN(C1COC(=O)N1)C(C1(N2CCCC2)CCC1)=O)C(C)(C)C CN1N=C(CC(=O)N2CCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)CC2)CC1=O CCN=c1[nH]c(C(=O)NC(CNC(=O)Cc2cccs2)C(C)C(C)C)cs1 C1(NC(C2N(C)CCOC2)=O)CN(C(c2[nH]nnc2C(F)F)=O)CCC12CCC2 c1(N2CCC(CC)C2)cc(C)c(S(=O)(=O)N2CCC=C(F)C2)cn1 CC(CN(C)C)C(=O)N(C1CC(NC(c2c[nH]c(=N)s2)=O)C1)C C1(CCC=C)(C(=O)NC(C)Cc2nc[nH]n2)CN(C(c2c[nH]nc2OC)=O)C1 C(CO)(CCCCNC(c1cnn(CC)c1)=O)NC(C=CCCC)=O O=C1CN(Cc2ccnc(OCC(F)(F)F)c2)C(=O)N1CCC1CCCO1 c1(C(=O)NCCN(C)C(c2c[nH]nc2C2CCCO2)=O)cccc(F)c1Cl c1(C(=O)NCCNC(=O)C(O)C2CCC2)cc2cccn2cn1 Cc1ccc(C(=O)NCC(C)CNC(=O)C(c2cn(C)nc2C(F)F)=O)cc1Cl C(C(=O)NC1CCCCC1NC(=O)CCCC1CCC1)(C(C)C)OCC(C)C N=C1NC(=O)C(CC(N2CCN(C(c3ccc(-c4ccc(Cl)cc4)s3)=O)CC2)=O)S1 CC(C)(CC(=O)N(C1(c2cccc(Cl)c2)CC1)CCO)n1cc(C2CCCO2)nn1 CCCCCCC(F)C(=O)NC1CC(CNC(=O)C(C)=C(C)CC)CC1O c1(C(=O)NC2CC(C)CN(C(C34CCN(CC3)C4)=O)C2)c(F)ccc2nc[nH]c12 C(=O)(C(C)C(C)(F)F)N(CC(C)NC(CSCC(C)=O)=O)C C(=O)(CCC(C)(F)F)NC(C(N1CC(C)OCC1)=O)C1(O)CCC1 c1(C(C(=O)NC(C)(CNC(=O)C=CC(F)(F)F)C2CC2)F)ccccc1 C1(C#CC(=O)NC(C2CCN(C(c3cc(C(C)(C)C)n[nH]3)=O)C2)(C)C)(CC)CC1 c1(OC)cc(C(=O)NCCC2CN(C(=O)C(C)(F)F)C2)ccc1OCCC(C)C N1(C(c2nccc(CC)c2)=O)CCCCC(NC(=O)CCNc2ccccn2)C1 N1(C(COC)=O)CCCCC(NC(=O)C(Cc2ccccc2)NS(C)(=O)=O)C1 CC1=CCN(C(=O)CCC2(NC(C3CC34CC4)=O)CCC2)CC1 C=CC1(c2cn(CCC(=O)OC)nn2)COCCN1C(=O)CCC1CCOC1=O c1(C(C)C)ccc(C(=O)N(CC(C)NC(=O)Cn2ccccc2=O)C)nc1 C1(NC(C=CCOC)=O)CCC12CCN(C(=O)CC(C)n1ccnc1)CC2 C1(C(N(C2CC(NC(C3CC(C)(CC)C3)=O)C2)C)=O)CC2(CCC2)CO1 N12CCC(CC1)CN(CCC)C2=O.C(C)(C)(C)NC(=O)CC C12(CNC(C(c3ccc(Cl)s3)C)=O)CCC(CC1)N(C(=O)CC1CCC(=O)N1)C2 CN1CCC(c2nnnn2C2CCCCC2)(NC2CC3CCC2O3)C1 c1(-n2c(C(N(CCCNC(c3cnsn3)=O)CC)=O)cnn2)cccc(F)c1 N1(C(c2cnc(SC)nc2)=O)CC2CCC(C1)C2C(=O)Nc1cnc(C#N)cn1 N1(C(C2(CCC)CCC2)=O)CC(OC)CC1CC(=O)N(CCC1CC1)CC c1(OC)ccc(C(F)(F)F)cc1NC(C1CCCN1C(=O)C(F)CC1CC1)=O N1(C(c2c(C)[nH]c(C(C)(C)C)c2)=O)CC2CCC(C1)N2C(C1(C#N)CC1(C)C)=O C12(CCC)CC(C(=O)NCc3ocnc3C(=O)NC3CC(C(C)C)C3)(C1)C2 c1(C(N(C2CN(C(c3coc(CO)c3)=O)CC2O)C)=O)ccc(N2CCCC2)cc1 Cc1nc(C2CC2)oc1C(=O)NC1(C)CCN(C(=O)C(C)CO)C1 Cc1cc(CC(=O)NC2CN(Cc3ccc(Br)c(O)c3)CC2(F)F)cc(C)c1 C(CCCCC)(C(=O)OC)N(C(C1CC(=C)C1)C(=O)NC1CCC1)C c1(C(=O)NCC2CN(C(c3c(C)ncnc3)=O)C(C)CC2)cccc2sncc12 N1(C(C(C)SC)=O)CCN(C(c2c[nH]nc2C)=O)CC1c1ccc(F)cc1 c1(C(=O)NC(C)(C)CNC(=O)Cn2nccn2)cccc(Oc2ccccc2)c1 N1(C(C(CC)SC)=O)CCN(C(=O)Cn2ccc(C3CC3)n2)CC1CCOC C(=O)(C(O)P(C)(C)=O)N1CCCC(CNC(CCC(c2cc(C)sc2C)=O)=O)C1 C(=O)(C(C)CC(C)(C)C)NC(C(=O)NC(CC#CC)CO)CCCC C1(NC(CCC2(C)CN(C(C3CCC(N(C)C)C3)=O)C2)=O)CCC=CCCC1 c1(CC(=O)NCC23OCC(NC(C=CC=CCC)=O)(C2)C3)cc(F)ccc1Cl C1(C(N(C)CC2CCCS2)=O)CN(C(C2C(C#N)C2(C)C)=O)CC12CC2 C1(NC(=O)Nc2cccc(OC)c2)CN(C(=O)C(C)n2cccn2)CC1C#N C1(NC(CCC(=C)Br)=O)CC(F)CN(C(=O)C(C)CN2CCCCC2)C1 N1(CC(=O)NC2CCCC2NC(=O)C2=CCOC2)CCCCCC1=O C1(NC(C(C)(C)C(N)=O)=O)CCC2CC1CN2C(c1cnn2ccccc12)=O C1(NC(C(CC=CC)CC)=O)CC2CCC1CN2C(=O)Cc1cc(F)ccc1O N1(C(c2n(C(C)C)cnc2)=O)CC(NC(=O)Cc2ccnn2C)CC(O)C1 C(C(C(=O)N1CCC(COCC)C1)C(C)C)NC(COCCC)=O C1(CC(=O)OC)CN(C(=O)C(=O)Nc2cccc(C)c2)CC2(CCC2)O1 Cc1cc(N)c(C(=O)NC(CNC(C2CCCC(F)(F)C2)=O)C2CCC2)cc1F N1(C(C=C(CCC)CCC)=O)CC2CC(C)N(C(=O)C(C)SC(C)C)C2C1 C1(CN(C(c2c(C(C)NC(c3cc(C(C)C)no3)=O)noc2)=O)C)CCN(C)C1 Cc1cc(C(=O)NC2CC(CCNC(=O)C(C)OC3CCCC3)C2)cc(C)c1O N1(C(CCCNC(C)=O)=O)CCC2(CC(C(=O)NC(C)CC(F)(F)F)C2)C1 C1(C(=O)NC(C2(C(=O)NCC(C(CC)C)C)CC2)C)CCCCC1(C)C c1(C(=O)NC2(CNC(C3CCC(C)CC3)=O)CCC2)ccc(=O)n(CCF)n1 CC(CCCCNC(=O)C=CCN1CCOCC1)NC(C1(CO)CCOCC1)=O CCCCC(C(=O)NC)NC(=O)CC(=O)NC(c1ccccc1F)C C(C)(CC(C)NC(c1occc1Br)=O)NC(CSCCC(C)C)=O C1(NC(N2CC(CCC)N(CCO)CC2)=O)CCCC2(CCCC2)C1 N1(C(C(C(C)C)c2ccccc2)=O)CC2CN(C(C3COC3)=O)CC2(C)C1 CCC(C)C(C)CNC(C1(SC)CN(C(c2ccc(SC)nn2)=O)C1)=O c1(C(=O)NCC(CC(=O)NCC2(O)CCCC2)OC)cc(O)ccc1C N1(C(c2n(C)ccc2)=O)CCN(C(c2cc(C(F)F)ccc2F)=O)CC(O)C1 C12CCN(CC1F)C(=O)c1cc(n(C)n1)CC(=O)N2.c1(CC)ccc(OC)cc1 C=CCCC(F)(F)C(=O)N1CCN(C(c2nc(=O)n(C)[nH]2)=O)C(CO)C1 N1(C(c2cn(CC)nc2C)=O)CCCC12CCCN(C(c1csnc1Cl)=O)C2 CCCCC(O)C(=O)NCC1CCC1NC(c1csc(Br)c1C)=O N1(C(C2(C(C)C)CC2)=O)CCC(C(C)(O)CNC(=O)CN2CCC(C)C2)CC1 c1(C(c2nnnn2C)NC2CC(OCC)C2)ccccc1OCCN(C)C C(=O)(CCCC(=O)N1CCC(C(=O)N(C)C(c2ccncc2)C)C(C)C1)OCC Cc1cccc(C(=O)NCC(C)(C(C)C)NC(=O)CSC2CCOC2=O)c1F CCCCC(C)CCC(=O)NC(CNC(=O)CC1(NC(C)=O)CC1)CCC CCCCC(O)C(C)C(=O)NCC1CC(C(N2CCC23CCCSC3)=O)=NO1 c1(N2CC(C)SC(C)C2)ccc(S(=O)(=O)NC2(n3cc(C#N)cn3)CC2)cc1Cl Cc1c(C(N2CCN(C(=O)Cc3cc(F)cc(Cl)c3)CC2CF)=O)cncc1Cl CCCCC(C)(F)C(=O)NCCN(C(=O)C(N1CCCCCC1)C)C1CCCC1 C1(CC)CN(C(=NCCc2cn(C)nn2)NCC(=O)NC(C)C)CCO1 Cc1cc(C(=O)NCC2CC2CNC(c2cccc(C(F)F)c2)=O)ccc1Br Cc1ccc(C(=O)NC2CCC2NC(c2nccn2C(C)C)=O)c(Cl)c1 N1(C(c2occ(C)c2)=O)C2CCC1C(C(=O)N(CCC(=O)NC1CC1)C1CC1)C2 C(C(C)CN=c1nc(C2CCCC2)[nH]s1)NC(c1c(CC)nns1)=O N1(C(C2CC(CCC)C2)=O)CCC(NC(c2ncsc2C)=O)C(F)C1 C1(c2ccccc2)(NC(c2cnsn2)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)C1 Cc1nc(O)nc(C)c1C(N1CC(C)(NC(=O)C(C)NC(=O)CC(C)(C)C)C1)=O Cn1nc([N+](=O)[O-])cc1C(=O)NCC1(NC(=O)Cc2ccc(Cl)c(F)c2)CC1 c1(C(=O)NC2CC(F)(CNC(C=CC=CC)=O)C2)ccc2cccnn12 CC(C)CC(C)(CNC(=O)C=Cc1cccc(CO)c1)NC(=O)CCS(C)=O C1(C)(C(N2CC(C)C(N(C)C)C2)=O)CCCN(C(=O)CC2CCCN(C)C2)C1 Cn1ncc(C(=O)NC(Cc2cc[nH]n2)C(=O)NC2CC=CC2)cc1=O C1(O)(CNC(C(C)OCC=C)=O)CCCN(C(c2ccc(CSC)cc2)=O)C1 c1(C(N2C(C(=O)Nc3cncc(OC)c3)CSCC2)=O)cc(O)cc(F)c1 CC(C)CC(C(=O)NCC#CCNC(=O)CCc1ccccc1Br)C(C)C N1(c2cccc(NC(C3CC(C#N)C3)=O)c2)CCC(=O)NC1=O Cc1ccc(C)n1CC(=O)NCC(C1CC1)NC(C1(O)CC(C)(C)C1)=O C1(NC(C(=O)N(C)C)=O)CC(C(=O)Nc2cc(C(F)(F)F)n(C)n2)C12CCC2 C(=O)(C1=CCC(F)(F)CC1)NCCC1CCN(C(CC2(OC)CCC2)=O)C1 Cc1cccc2c1CCOC2C(=O)NCC(C)CN(C(=O)CCCC(C)C)C Cn1nc(C(=O)NC2CCCC(C(=O)OC(C)(C)C)CC2)c(-c2nn[nH]n2)c1C#N C1(C(=O)NCCCN(C(C(C=CC)O)=O)Cc2cccnc2)CCCC12CC2 c1(CC(C(=O)NCC(C)N(C(=O)CC2CCNC2=O)C)(C)C)cc(F)ccc1F O=C(C1Cc2ccccc21)NC1CC2(CCN(C(c3sc(Cl)cc3Cl)=O)C2)C1 C1(O)(CNC(CC(C)C2CC2)=O)CCCN(C(C2(C)CCC(=O)N2)=O)CC1 C(=O)(CCS(=O)(=O)N(C)C)NCC12C(CN(C(C(C(C)C)OCC)=O)C1)C2 C(=O)(CC(C)C(F)(F)F)NCC(CNC(=O)CNS(C)(=O)=O)OC C(=O)(C1CCc2cc(F)ccc21)N1CC(C(=O)NCCS(CC#C)(=O)=O)C1 c1(C(=O)NC2CCC(N(C)C(c3cnccc3Cl)=O)C2)cc(C(F)F)ccc1Cl C1(C(C)(C)C)C(NC(=O)CC2COC(=O)N2)CCN1C(=O)CSC(F)(F)F C1(NC(CCC(=C)Cl)=O)CCCC12CN(C(c1ccc3nsnc3c1)=O)C2 c1(CSC)cc(C(=O)NCCCNC(c2cnccc2C)=O)sc1C C1(OC)CN(C(C2(O)CC2)=O)CC1C(N1CCN(CC(N)=O)CC1)=O C1(CC(=O)N(CC(=O)NC(C)COCC)CCC)CC(O)C1(C)C Cc1ccc(C(N2CC(F)CC2CN(C)C(C2(F)CCOC2)=O)=O)cc1F N1(C(c2ccc(N(C)C)cn2)=O)CCCCC(NC(=O)CCC2CCC2)C1 N1(C(C(C)OCCOCC)=O)C2CCC1CC(N(C(=O)C(N)=O)C)C2 N(C(=NCCN1CCCC1=O)NCC(CO)C(F)(F)F)C(c1ccccc1)C N1(C(CC(C)OC)=O)CCC(C)C1CNC(C1CCN(C(=O)N(C)C)CC1)=O C(=O)(CCC(C)(C)NC(N1CCC(C)(C(=O)NCCF)C1)=O)OC c1(OC(C)(C)C)cc(NC(=O)COC2CC=CC2)ccn1.N12CCCC(C1)C2=O N1(C(c2cc(C)ncn2)=O)CCC2(CCCN(C(=O)CN3CCCC3C)C2)C1 C=CCC(CC=C)C(=O)NC(C1CCN(C(=O)COCC2CCCC2)C1)C N1(C(CCc2cc(C)no2)=O)CCOC2(C1)CN(C(=O)CC(C)c1ccco1)C2 Cc1oc(C#N)cc1C(N1CCC(CCNC(=O)CC2CC=CCN2C)CC1)=O c1(C(=O)NC2COCCN(C(CC3CC(CC)C3)=O)C2)cc(C)cc(C)c1N C#Cc1ccc(C(N2CCC(F)(CNC(=O)CC=C(C)C)CC2)=O)c(F)c1Cl Cc1cc(O)ccc1C(=O)Nc1ccc(C2CCC2)cn1 c1(C(=O)NCC23C(CN(C(C(=O)NCCOC)=O)C2)C3)nn(CC)cc1[N+](=O)[O-] C1(C#N)(NC(C23C(CN(C(c4ccc(C)cn4)=O)C2)C3)=O)CCOCC1 c1(CC)cc[nH]c1C(=O)NCC1(C(=O)N(C23CC(C2)C3)C)CCCO1 c1(SC(c2ccccc2)C)ccccc1C(=O)NCC(C1CCOCC1)(F)F c1(C(=O)NCC2CN(C(C(CC)SC)=O)CC2C)cccc2c1OCC2 N1(C(CCNC(=O)CO)=O)CCC(C(=O)NC2COCOC2)CC1 N(C1CCOc2ccc(Cl)cc21)C(c1c[nH]c2cc(F)c(F)cc12)c1n(C)nnn1 c1(C(N2CC(C)N(c3nc(Cl)ncc3Br)CC2)=O)cnn2ncccc12 c1(C(N2CC3CN(Cc4c(C)c(O)ccc4)CC32)=O)ccc2ccccc2n1 c1(NC(C(N2C(C)CCC(O)C2)c2ccc(OCF)cc2)=O)ccc2c(c1)OCCO2 c1(C(=O)N(C2CC(OC)CN(C(CCC)=O)C2)CC)coc2cc3c(cc12)CCC3 c1(C(=O)NCC(CN(C)C(c2cccnc2)=O)(C)C)cc(=O)cc(Cl)[nH]1 S(=O)(=O)(c1cccc(F)c1)NCC(=O)NC1(CCCNC(CCOC)=O)CC1 CC1=NN(C)C(=O)C1CC(N1CCC(NC(c2nn(C)c(C)c2N)=O)C(C)C1)=O C=CC1CN(C(=O)CCC(CC)NC(=O)CCn2cccc2)CCO1 CC1(NC(=O)C(F)OC(F)(F)F)CCN(C(c2nnsc2N)=O)C1 Cc1cc(C(=O)NC(C)C(CO)NC(C2(n3cnnn3)CC2)=O)co1 C1(C(=O)NCC2CC(NC(C3(C)CC(=C)C3)=O)C2)CC2CC1C1CC21 c1ccc(C(=O)OC)cc1.c12cn(nn1)CC(=O)C1(CCC1)CCNC(=O)N2.CC C(CCN=c1nc2sccc2c(NC(C)CN2CCCC2)[nH]1)(C(C)C)OCC Cc1cccc2c1OC(C(=O)NCC1(NC(c3sc(N(C)C)nc3Cl)=O)CC1)C2 Cc1cc(O)c(CNC2CC(NC(c3cc(=O)cco3)=O)C2)cc1Cl Cc1ccc2c(c1)CCN2C(=O)CCS(=O)(=O)Cc1cccc(C)c1 C=CCCCCCC(=O)NCC1(C(=O)NCC2CC(C)(C)CCO2)CCCCC1 c1(C(N2C(CN(C(=O)C(c3cnn(C)c3)O)C)CCC2)=O)ccn2nccc2n1 Cc1cc(C(N2CC(NC(c3cncc(CO)c3)=O)C(C)(C)C2)=O)nnc1O c1(C(N2CC(OC)C(NC(c3nc(Cl)oc3C)=O)C2)=O)cc([N+](=O)[O-])sn1 N1(C(CCN(CC(F)(F)F)C)=O)CCC(CNC(=O)C2=CSCS2)C1(C)C C(=O)(C1CCc2cccnc21)NC1CCC2(CCN(C(C(C(C)O)(F)F)=O)C2)C1 N1(C(CC2CCN(C(CCCOC(C)(C)C)=O)C2)=O)Cc2n[nH]cc2C1CO N1(CC(=O)N(C(C)C(=O)N(C)Cc2scnc2C)CCC)CCC(=O)CC1 N1(C(c2c(C)c(Cl)cnc2)=O)CCC(NC(=O)CCC(C)C)C(CO)CC1 N#Cc1ccc(Cl)c(C(N2CCCC(CC(=O)Nc3nnc(C4CC4)o3)C2)=O)c1 C(N(O)C(=O)CC(C)CC(F)(F)F)c1cn(C(CCC)CCC)nn1 C(=O)(C1CCc2snnc21)NC(CNC(C(CC(CC)C)C)=O)(C)C CC(C)(O)C(F)(F)CNC(=O)C(N)CCC1CCC1 CN1CC2CCN(C(=O)CC3C4CCCC4N3C(C3(C(N)=O)CC3)=O)CC2C1 Cc1nc(C2CC2)cc(=NCOCCOC(=O)Cc2ccc(C3CC3)cc2)[nH]1 c1(C(=O)NCCCN(C(=O)C(F)(F)C2(O)CCCC2)CC)cncnc1C(C)C C1(NC(c2cnc(C3CC3)s2)=O)COC2CN(C(C3(O)CCSC3)=O)CC12 N1(C(c2ccc(C=C)cc2)=O)CC(C2CN(C(=O)CN3CCC(C)CC3)C2)C1 N1(C(c2ccnc(N(C)C)n2)=O)CC(CNC(C2CCCO2)=O)C2(CCC2)C1 C1(N(C(=O)CSc2cccnc2)C)CCCN(C(C2CCCNC2=O)=O)C1 c1(OC)nc(=NC2CCC3(CC2)CN(C(=O)C(C)=C(C)C)CCO3)nc(OC)[nH]1 N1(C(c2c(C)ncs2)=O)CCC2(CCC2CNC(C2COCCO2)=O)CC1 c1(C(N2CC(NC(C(CC)OC3CCCCC3)=O)C2)=O)cccc(OC(C)C)n1 c1(CCCN2C(C(N(C(C)C)C(C)C)=O)CCC2)ccc(F)cc1 C1(CC(=O)N(C(C)CN(C(=O)C(F)(F)C2(O)CCC2)C)C)CCC2(CCC2)O1 N1(C(CC(=O)NC2CC2)=O)CCC2CCCC12CNC(c1cc(O)cc(=O)o1)=O S(=O)(=O)(c1c[nH]c(C(=O)NCC2(OC)CCN(C(=O)C(C)CF)C2)c1)NC c1(-c2nc(C(C)OCC)nn2CC2CC2)ccnc(CC)c1F C1(N(C)C(C2CC2CF)=O)CN2CCC1CC2.C1(C)COCCO1 C(C(CC(=O)NC1CC(CNC(C2(n3cccn3)CCC2)=O)C1)C(F)F)N(C)C CCC(F)(F)C(C)(C)C(=O)NC1CC1NC(=O)C(C1CCOC1)OC C1(CNC(C(CC)(C)F)=O)CN(C(c2ccnc(Cl)c2N)=O)CCCO1 C1(CNC(c2c(OC)cnc(F)c2)=O)C(C2CC2)CCN1C(=O)CCC1CC1 N12CCC(CC1)C2=O.C1(C2(COCC)CC2)CCCO1.C1C(=O)N1.C1CO1 c1(C(=O)NCCN(C(=O)C(C)(F)CC)CC)cc2ccccc2c(=O)o1 c1(C(=O)NCC(CNC(CCC(C)OCC)=O)O)cc2nc(C)[nH]c2cc1F C(=O)(CCC(C)CN(C)C)NCC1CCCC(CNC(C=CCN(C)CC)=O)C1 N1(C(Cn2c(C)cc(C(F)F)n2)=O)CC2(CCN2C(=O)COC2CCOC2)C1 C(C)(CC(=O)NC1CC1NC(c1cc2cc(Cl)ccn2n1)=O)(C(F)(F)F)N(C)C Cc1cc(C=CC(=O)NCC2(O)CN(C(=O)CCS(C)=O)C2)ccc1Br Cc1cc(F)cnc1C(=O)NCCC1CN(C(C2(C(F)(F)F)CC2)=O)C1 c1(CC)cc(OC)cc(C(=O)NC(C)C(C)NC(C2(O)CCCC2)=O)c1 N1(C(C2CC(OC)C2)=O)CCN(CC2CN(C(=O)C(C)(C)NC(C)=O)C2)CC1 N1(C(COCCOCC#C)=O)CCC(NC(c2n[nH]c3c2CCC3)=O)C12CCC2 C1(NC(CC(CNC(=O)CCC(F)(F)F)OC)=O)CCOC2(CCC2)C1 C(=O)(N=c1cc(C(N)=O)n(C)[nH]1)C1C(CNC(c2ccn(CC)n2)=O)CC1 C1(CNC(CNCCN(C)C)=O)CCOC(CN)C1 C1(CNC(C(C)c2cc[nH]n2)=O)CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1O C1(C(N2C(C)CN(C(C3CC(F)(F)C3)=O)CC2)=O)C(O)C(=O)N(C)C1C c1(CC)nn(C)c(C(=O)NC2CC2CNC(c2cccc(C(C)(C)C)n2)=O)c1Cl C1(C)(CNC(c2c(C)cnnc2)=O)CCCN(C(=O)CC2CS(=O)(=O)C2)C1 CCCC(CCC)C(=O)NCC1CC1CNC(C1(COC)COC1)=O c1(NC)nc2ccc(CN3CCC(O)(C(F)F)CC3)cc2s1 C12CN(C1(C)C)C2=O.C12CC(C1)C(=O)O2.C1(C(C)=O)CCCN1 c1(C(N2C3CC(NC(CC(C)(C)O)=O)CC2CC3)=O)ccc2c(c1)NS(=O)(=O)C2 Cc1nc2ccc(C(N3CC(NC(C4CC=CCO4)=O)CC(C)C3)=O)cc2s1 C1(NC(C2CCCN2C(c2[nH]nnc2C2CC2)=O)=O)CC2CCC1(CO)C2 N1(C(Cn2c(C)nc(C)n2)=O)CCC(CNC(c2nocc2Cl)=O)C(F)(F)C1 c1(OC)ccc(C(N2CCN(C(=O)CC3(C)CCC3)CC2CF)=O)c(Cl)c1OC C(C)(C)(C(=O)NC(C1CCCC1)CNC(c1coc(Br)n1)=O)NC(=O)NCC=C C1(C(=O)NCC2C(CNC(c3nncn3C3CC3)=O)C2)(CO)CCOC1 N1(C(=O)C=CC2CCOC2)CC=C(CCNC(C2(c3cccs3)CC2)=O)CC1 C=CCCCC(=O)N(C)CC1(C)CCCC1NC(=O)C(C)C(F)F C#Cc1c[nH]nc1C(=O)NC1CCC(C)(CNC(=O)CS(=O)(=O)NCC)C1 C=C(C)CC(C(=O)NCC1CC(C)C1)NC(=O)CC#N c1(C(C(C)NC(=O)Nc2cc(C3CCNCC3)no2)OCC)ccccc1F C12(C(N(CCCN(C)C)CCNC(C(C)OCC)=O)=O)CC(C)(C1)OC21CCC1 c1(-c2cn(C3OCCN(C(C(C)(C)C)=O)C3)nn2)ccc2cnccc2c1 N1(C(C2N(C(C)C)CCCC2)=O)CC2CCN(C(C34COCC(C3)C4)=O)CC2C1 N1(C(c2c(C)cnn2C)=O)CCN(C(C2CC(=O)C2C)=O)CC1C N1(C(C2(OC)CCCCCC2)=O)CC2CCN(C(C3CNC(=O)C3)=O)CC2C1 C1(CC(=O)NC(CC=C)C(=O)NC2CCC2)C2CCC(C2)N1C(=O)COC Cc1[nH]c(C#N)cc1NC(=O)C(C)C(C)OC(=O)Nc1ccccc1 Cc1c(Br)csc1C(=O)NC12CC(NC(=O)CC3(C)CC3)(C1)C2 CC12CCC(CNC(=O)Cc3cccc(OCC(F)F)c3)(C1)NC2=O c1(OCc2ccc(COC)cc2)ccc2c(c1)-c1ccccc1C2 C(CC(C(=O)NC1(CCO)CN(C(=O)C(C)OCCN(C)C)C1)NC(C)=O)SC n1(Cc2nc(C(CC)O)nn2-c2ccn(CC)n2)cnc2ccccc2c1=O C(=O)(CC(C)(C)C1CCCCC1)NC1C(CNC(C2N(C(C(C)C)=O)CCC2)=O)C1 c1(C(N2CC(NC(C(C)(C)NC(=O)NCC)=O)C2)=O)ccc2cnccc2n1 C1(C(N(CC#CC)C)=O)CCCC(NC(c2cccc(C)c2F)=O)CC1 c1(C(=O)NCC(CNC(=O)CCCc2cccc(Cl)n2)F)ccc(O)c(F)c1F CC1CN(C(c2cc(Cl)no2)=O)CC1NC(c1cn(CC2CCOCC2)nn1)=O c1(C(N2CCN(C(C=C(C)C)=O)C3(C2)CCC3)=O)cc(S(C)(=O)=O)ccc1Cl C(=O)(C1COc2ccccc21)NCC1CN(C(c2cc(C)on2)=O)CC1(F)CO CC(C)(C)CCCC(=O)N(CCC(=O)NCCCCCF)C1CC1 c1(NCC(=O)NC(C)(C)C)ccc(-c2ccc(C(F)(F)F)s2)cn1 C1(C(=O)NCC(C)OC)CC(O)CN1C(=O)C(O)CCNC(=O)OC(C)(C)C C1(CNC(NOCc2ccc(OC)cc2)=O)N(C(c2cnns2)=O)CCC1(C)C CCC(C)C(O)CNC(=O)NCc1c(Cl)cnn1C C#CC1(NC(=O)CC(C(F)(F)F)NC(=O)C(c2ccccc2)C)CC2CCCC12 c1(C(N2CC3C(NC(C4CC(c5nnc[nH]5)C4)=O)(C3)C2)=O)ccc(Cl)c(F)c1F c1(CNC(C(CC)N(C(=O)C(O)C2CC2)C)=O)cc(C)ccc1F CCC(Cc1ccccc1)C(=O)NCCC1(NC(=O)C=CS(C)=O)CC1 c1(OC)cccc(NC(C2CC(F)CN2C(=O)C=Cc2ccsc2)=O)c1Br CCCCC(O)C(C)C(=O)NC1CC(C(N2CC(N3CCCC3)C2)=O)C1 c1(SC)ccc(CNC(C23CCCC2(C(N)=O)C3)=O)cc1Cl c1(C(N(CCCCN(C)C(C2CCC2C(N)=O)=O)C)=O)ccc(F)c(CO)c1 CC(=NOCC#N)C(=O)N(CC(C)C(=O)NC(C)CC1CCC1)C CC(C)CC(CNC(C1CCN(C(N)=O)CC1)=O)NC(=O)Cc1cccnc1Cl C(=O)(C(CC1CCC1)NC(c1cn(CC)cn1)=O)NC1(CCCC)CC1 CCS(=O)CC(=O)NC(C)C=CC(=O)NCC(C1CC1)N(C)C N1(C(C2N(CC)CCC2)=O)CC(C)(C)CC1CC(=O)NCC1(CCOC)CC1 C1(O)(C(=O)NC2C(CNC(c3c(C)ccc(C)n3)=O)CCC2)CN2CCC1CC2 CCCCCCC(C)CC(=O)N(C)CCN(C)C(c1c[nH]nc1S(N)(=O)=O)=O C(=O)(C1SCc2cccnc21)NC1CCC(NC(c2c(N)ccc(CC)c2)=O)C1 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CC(N(C(=O)CC(C)(C)COC)CC)C1 C1(C(=O)NC(C2CCN(C(c3conc3C3CCCC3)=O)C2)(C)C)C2COCC12 c1(CC)c(C(N2CCC(CO)C(NC(=O)C(C)(C)C#N)C2)=O)oc2ccccc12 CCC(F)(F)CC(=O)NCC(F)CNC(C1CCC(=O)N1c1ccccc1)=O C1(NC(C2C(=C)CC2)=O)CCCC(NC(c2cc[nH]c2C)=O)CC1 CC(C)CC(C)CN=C(NCC(=O)N(C)C)NC1CCS(=O)(=O)C1 c1(OCC)ccccc1C1(C(N2CC(NC(C3CCSC3)=O)C(O)C2)=O)CC1 C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC(O)(C(CNC(CCCOCC)=O)(C)C)C1 c1(C(=O)NC(C)(C)CCNC(=O)CSCCC#N)ccc2nsnc2c1 C1(CNC(CC2N(C)CC=CC2)=O)CN(C(C2(CN(C)C)CC2)=O)CCC1(C)C c1(C(=O)N(CCNC(C23CSCC2C3(F)F)=O)C2CC2)ccc([N+](=O)[O-])s1 Cc1c(Cl)ccnc1C(N1CCOCC1CCNC(=O)C(F)C1CCC1)=O c1(CCC)nnc(S)n1CC(=O)NCCC1CCN(C(c2cncc(O)c2)=O)C1 N1(C(C=CC2(C)COC2)=O)CCCC12CCN(C(=O)Cn1nccn1)C2 C1(C(=O)NCc2c(CCNC(C3C=CCC3)=O)ocn2)Cc2nnsc2S1 N1(C(C2(C(O)C(F)(F)F)CCC2)C)CCN(Cc2cc(C#N)cn2C)C(C)C1 Cc1nc(C(=O)N(CCNC(C2CCC2n2ccnc2)=O)C2CC2)c(C)n1C1CC1 S(=O)(=O)(c1cc(OC)ccc1Cl)N1C(CC)CN(C(=O)CSc2nc[nH]n2)CC1 C=C(Cl)C(C)(C)C(=O)NCC(F)CNC(=O)C(c1ccc(F)cc1)(C)O Cc1nc2c(C(=O)NC(C)C(C)(C)NC(=O)C(C3CCCCC3)F)ccnc2[nH]1 Cn1ccc(C=CC(N2CC(CC(F)C(=O)NCC(C)(O)CO)C2)=O)c1 n1(CCC(=O)O)nc(C)nc1C.C1CC(C)(C)N1CC=CON1CCSCC1.CC C(=O)(C#CC1CCCC1)N1CC(NC(C(C2CCOCC2)OCC)=O)(COC)C1 c1(C(=O)NCC2C3CN(C(CC(C)CF)=O)C2C3)ccc2nonc2c1 Cc1cc(C)n(C(C)C(=O)NCCN(C(=O)Cn2cncn2)C2CC2)n1 Cc1nc(CC(=O)NC2CCN(C(=O)Cn3nnnc3C3CC3)C2)sc1C CN(CCC(=O)Nc1ccc(F)cc1F)N(C)CCn1ccnc1 C(=O)(C1=CC2CCC=CCCC12)OC.c1(CC)cc2c(c(F)c1)NC2=O C1(CNC(C2(CC#C)CC2)=O)CCCCN1C(c1cnc(C(C)=O)s1)=O CC1(C)CN(C(C2CC(O)CN2C(C2(C#N)CCOC2)=O)=O)CCC1CO c1(C(C)C)cc(C(=O)NC2CCCCC2NC(C2CNC(=O)C2)=O)c(C(C)C)[nH]1 NS(=O)(=O)CCC(=O)NC1CN(C(c2cccc(N3CCOC3=O)c2)=O)C2CC12 N1(c2nc(N3CCOC(C)(C)C3)cc(C)n2)CC(=O)N2CCCCC2C1 C1(NC(c2ccnc3[nH]ncc23)=O)C2CCN(C(c3ncccc3Cl)=O)CCC12 c1(CC)ocnc1C(=O)NCCN(CCOCCO)C(C1CCC1C(F)(F)F)=O N1(C(C(=Cc2cccs2)C)=O)CC(CNC(C2CCNC(=O)C2)=O)CC(C)C1 Cc1ccc(F)cc1NC(C1C2CCC(C2)C1NC(c1cc(F)cn1C)=O)=O c1(C(=O)NCC2C3CCCC2N(C(=O)C2=CCSC2)C3)cc2cc(Cl)ccn2n1 C1(NC(CC(CC)C)=O)CC2CCC1N2C(c1ccc(Br)cc1N)=O c1(C(N2CC(OCC(=O)NC(C=C)C)C2)=O)ccncc1CC CC1(C(=O)NCC2CC(NC(c3ccc(C4CCC4)nc3)=O)C2)CCCCO1 C#CC1CC2(CC2)CN1C(C1CC(C)CN1C(C1CCC(C)(C)C1)=O)=O c1(SCC(N2CCC(CNC(CCC(=O)NC)=O)C2)=O)ccc(Cl)cc1Cl N1(C(=O)CO)CCCC2(CCN(C(C3(Cc4ccccn4)CC3)=O)CC2)C1 N1(C(c2cnc(C(=O)OC)s2)=O)CCCN(C(=O)C=CC2CCCC2)C(CO)C1 c1(C(=O)NC2CC(NC(C(CC)C#N)=O)C2)cc2c(ccn2C)s1 CCCC(C)(CC)C(=O)NC1CC(C)CN(C(c2ccc(C(=O)OC)c(O)c2)=O)C1 C12(CNC(c3cc(C)nn3C3CCC3)=O)CCC1CCN2C(=O)CCNC(N)=O c1(C(NOCCCC)=O)[nH]ccc1C(=O)NCC1C(C(=O)OC)CCC1 Cc1ccc(F)c(C(=O)NC(C2(O)CCCCC2)C(N2CC3CC(C)C3C2)=O)n1 N1(C(C2C(C(C)C)CCO2)=O)CCC(C)(CC(=O)NC2C3CCC2CC3)C1 CCCS(=O)(=O)CC(=O)NCC(C1CCCC1)NC(C1CCC(CC)NC1=O)=O c1(CCC(=O)N(CCCNC(C2CNC(=O)N2)=O)CC)cc(F)cc(F)c1 c1(C(=O)NC(CCNC(C2C(C)CC2C)=O)(C)C)cncc2sccc12 N1(C(c2c(CC)nco2)=O)C(C(N2CC3(CCCCC3)C2)=O)C2CC(O)C1C2 CC1CS(=O)(=O)CCCN1C(=O)C(C1C2CC3CC(C2)CC1C3)N c1(C(N2CC(CCOC)C(C)C2)C(=O)NCC(=C)C)ccc(CC(C)C)cc1 N1(C(C(C)(C)CO)=O)CCC(n2cccn2)(CNC(=O)C=Cc2cncs2)CC1 CSC=CC(=O)NCC1(O)CN(C(=O)C=CCN2CCC2)C1 C(C)(CO)(C(=O)NCC1CC1CNC(c1cc(-c2csc(C)n2)c[nH]1)=O)OC c1(N2CC3CC(NC(C=C(C)C(C)C)=O)C3C2)ccc(C#N)cc1[N+](=O)[O-] Nc1c(C(=O)NC2CC3CC(NC(C4CCNC4=O)=O)C2C3)sc2nccnc12 C(=O)(C(C)CC(C)(C)C)NCC1CCN(C(Cc2[nH]n(CC(C)C)c(=O)c2)=O)C1 c1(C(=O)NC(CNC(CN(C(COC)=O)C)=O)C(C)C)ccc(C)c([N+](=O)[O-])c1 C(=O)(C1CCCc2nc[nH]c21)N1CCCN(C(c2ccc(O)nn2)=O)CC1CO CC1CC(NC(N2CCN(CC(=O)N(C)CCNc3cccs3)CC2)=O)CCO1 c1(COC)ncsc1C(=O)NC(C)CCCNC(c1[nH]cnc1C)=O C=Cc1cncc(C(=O)NC2(C(=O)NC3CC=CC3)CC2(C)C)c1 N1(C(=O)OC)CCCC(n2cc(NC(=O)Nc3cnc(C)n3C(F)F)cn2)C1 c1(OC)cc(C(=O)NC2CC(F)(CNC(=O)C(C)n3cccn3)C2)ccc1C N1(C(C(C)OC(C)(C)C)=O)CCC(C2(NC(C3CN(CP(C)(C)=O)C3)=O)CC2)C1 C#CC1CN(C(C23CCCCC2C3(F)F)=O)CCN1C(c1nc(CC)oc1C)=O CC1C(NC(C2CCS(=O)CC2)=O)CCCN1C(C1CC2C=CC1C2)=O CCCC(C(=O)N1CC(CS(C)=O)C1)NC(c1cnn(C)c1Cl)=O C1(CC)CCc2sc(C(N3CCCN(C(=O)CCCOC)CC3CO)=O)cc2C1 C(CNC(=O)CCCN1C(=O)CNC1=O)(C(C)C(C)C)NC(c1cnc(C)o1)=O C(=O)(C1Cc2ccccc21)NC(CC)(CNC(c1cccc(O)n1)=O)CC c1ccc2oc(O)nc2c1.C(=O)(C1=CCCN(CO)C1)C(=O)NCc1ccco1 c1(C(=O)NCCN(CC(C)O)C(=O)C=CC2CC2)cn(C)nc1C1CCOC1 c1(C(N2CC(O)(C(C(=O)NCc3onc(C)n3)F)C2)=O)ncnc(C)c1C N1(CC)CCCC1CCCNC(=O)Cc1cnn(CCOCCCN=[N+]=[N-])c1 C1(N(C(=O)CC(=O)OC(C)(C)C)C)CCCN(CCCNC(=O)C2=CCCS2)C1 CCC(C)CC(C)C(=O)NCC#CC(=O)NCc1nnn(C)n1 C(=O)(C1CCCc2ncnn21)N1CC(N(C(C2=C(C)OCCC2)=O)C)C2(C1)CC2 CCCCS(=O)(=O)NC(C)C(=O)NC1(c2ccccc2)CN(C(=O)C(C)(C)F)C1 c1(C(=O)OC)cccc([N+](=O)[O-])c1OCC12CC1CN(C(=O)CNC(=O)OC)C2 N1(C(C2CC(C(=O)OC)C2)=O)CCC2CN(C(c3c(O)nnc(C)c3C)=O)CC12 N1(C(C2CCC(NC(=O)OC)C2)=O)CCC(C)(NC(=O)Cc2n[nH]c(C)n2)CC1 c1(C(N(C2CC(OCC)C2)C)=O)cnc(CNC(c2cc(O)cs2)=O)nc1 C(C(C)(C)CO)(c1ccccc1)NC(C(Cc1cccs1)NC(C)=O)=O C1(NC(C2CN(C(=O)NCC)C2)=O)CC2(C1)CC(C(=O)NC1(C)CCCC1C)C2 C(=O)(CCCC(C)CC)NC(CCC#C)C(=O)N1CCCCC(C)C1 c1(C(=O)NC(CC2CN(C(C(C(CC)CC)C)=O)C2)C)[nH]c2ccccc2c1Cl C12(C(=O)NCCN(C(=O)CCC(=O)c3ccccc3)C)CCC(C(F)F)(CC1)C2 N1(C(CC2N(C)C(=O)CC2)=O)CCN2CCOCC2(C(=O)O)C1 C1(NC(C=C(COC)C)=O)CCN(C(=O)CC(N2CCCCC2=O)C)CC1O C(CC)(CCCO)NC(CC1(NC(CCOCCC)=O)CCC1)=O N1(C(C(n2cc(C(C)(C)OC)nn2)C)=O)CC(=O)CC(C)C1 Cc1cccc2c(C(=O)NCCC(O)CNC(C3CC(O)CN3C)=O)n[nH]c12 C12(CNC(C3C(OCC)C3)=O)CCC(CN(C(c3cccn4cncc34)=O)C1)C2 NS(=O)(=O)c1cc(Br)ccc1NCCCCC(F)(F)F C1(C(N(CCCN(C(C2C(C#C)C2)=O)C)C)=O)COc2ccc(OCC)cc2C1 N1(C(CC(=C=C)C)=O)CC(NC(C2CN(C3CCOC3)C2)=O)CC12CCCCC2 c1(OC)cc(C(=O)NCC2CCCC2CC(N2CC(CO)C(O)C2)=O)ncn1 O=C1CCc2cc(Cl)c(S(=O)(=O)N3CCC(c4ccsc4)C3)cc21 CC1(C(N2CCC(C(CO)NC(=O)CC3CC3)CC2)=O)CCNC(=O)C1 N1(CC)N=C(C(=O)N2CCN(C(C3CC3c3cccs3)=O)CC2)CCC1=O N1(C(c2c(C)con2)=O)CCC2(C1)CN(C(c1cnccn1)=O)CCO2 C(C)(N=c1nc2c(cnn2C)c(NC2CCN3CCCC3C2)[nH]1)c1cnc(C)s1 N1(C(c2ccc(C#N)[nH]2)=O)CCC2(CC(NC(=O)Cc3cccnc3O)CO2)C1 c1(C(=O)NC2CC(C)CN(C(C34CCC(CC3)C4)=O)C2)cnc2c(ccn2C)c1 c1(CC)nccnc1C(N1CCC2CC12C(=O)Nc1cn(C)nc1O)=O Cc1noc(C)c1CC(=O)NC(C)(C)CNC(=O)C(C)NC(N)=O C(CC(C)C)(C(=O)N1CC(C)(O)CO1)C(C=C(CC)C)=O.NC c1(SC)cc(C(N2CCC(CO)C(NC(C3(C#N)CCCC3)=O)C2)=O)ccc1F C(=O)(C(C)(C)CS(C)(=O)=O)NCC1CCC(NC(c2cc(C)c(=O)n(C)c2)=O)C1 C1(F)(CN2C(C(=O)NC3N(C(C)=O)CCC3)CC2)CCN(C(=O)C#CC(C)C)C1 c1(CC)ncc(C(N2CC(O)CC2CC(=O)NCCC(=O)NC(C)CC)=O)cn1 c1(C(N2C(C)CC(CC(=O)N(CCCC(=O)OC)C)C2)=O)cnc(O)c(C)c1 N1(C(c2ccc(C(C)C)o2)=O)CC2CN(C(=O)CC3CCCN3C)CC2(C)C1 C1(NC(c2cccc(COC)c2)=O)CS(=O)(=O)CC1NC(c1cnn(CC)c1)=O C1(CC(=O)NCCN(CC(=O)N(C2CCC2O)C)CC)CCC(O)C1 C(C(C(=O)OC)CN(CC)CC)OCC(n1cc(CCC2CC2)nn1)CO n1(C(C)C)ccc(=NC(=O)c2cc(CNC(C3(F)CC=CC3)=O)on2)[nH]1 c1(CCNC(C2CC(C)(SC)C2)=O)ccc(CNC(C2CCCC2O)=O)cc1 c1(C(=O)NC)[nH]c(NC(=O)CSc2ccc(C(=O)NC3CC3)s2)c(C)c1C(C)=O c1(C(N2CCCCC(CNC(C(C)OCC)=O)C2)=O)nc2ccccc2nc1C C1(NC(C2(C)C(C)C2)=O)CN(C(=O)Cc2ccnc(Br)c2)C(C)(C)C1 N1(CC(N2CC(CN(C)C(C3C4COCC34)=O)C2)=O)CCc2ccccc2C1 Cc1cc(Cl)c(F)cc1NC(=O)CN1CCOCC1.C12CC1OC2=O C1(O)(C(=O)NCCCN(C(C)C)Cc2ccn(C(CC)CC)n2)CCOCC1 c12cc(C)c(cn1)S(=O)(=O)N1CCC(C1)N2C(=O)OC.C1(OC2CC2)CCOC1C C1(C(=O)NC2(C(=O)OC)CSC2)CCN(S(=O)(=O)C(F)(F)F)CC1 S(C1CCc2c(Br)cccc21)c1ccc(Br)c(CN2CCOCC2)c1 Cc1ccn2cc(C(=O)NC3(CCNC(C4(C)CC4Br)=O)CC3)nc2c1 C1(NC(c2cc(CNC(=O)CCc3cn[nH]c3)on2)=O)CCN2CCC1C2 S(=O)(=O)(c1ccc(-c2cccc3ccnn23)cc1)N1CC(C)C(CO)CC1 N1(C(C2(OCC)CCC2)=O)CC2CC2(NC(c2ccc(CN3CCCC3)o2)=O)C1 CCC(C(=O)NC1CC(C(=O)N(Cc2ccccc2)OC)C1)NC(N)=O O=C1Cc2cc(C(=O)NC3CC4CN(C(C5CC5C(C)O)=O)CC34)ccc2N1 N1(C(c2c(CC)cccc2)=O)CCCCC(NC(=O)C(C)NC(C)=O)CC1 c1(NC(C23C(CN(C(c4ncn(C)c4)=O)C2)CC3)=O)cccc(F)c1C#N c1(OC)ccc(C)c(C(=O)NCC(CO)NC(C2COCC2(C)C)=O)n1 Cc1cnccc1CN(C(=O)C(Cn1ccnn1)NC(=O)CN1CCNC1=O)C C1(OC)CCC(C)(C(N2CC(O)(C(C)NC(=O)C(=O)N(C)C)C2)=O)CC1 N1(C(c2cccc(I)c2)C(=O)NCCC(=O)OCC)CCOCC2(CCC2)C1 c1(C(N2CCC(NC(C(C(C)C)C3(C)CC3)=O)C2C)=O)ccnc2cc[nH]c12 N1(C(C=CC(=O)OCC)=O)CCN(C(c2ncc(F)cc2F)=O)C(C#N)C1 N1(C(CC)=O)CCCN(C(C2CN(CC(F)(F)F)C2)=O)CC1C(C)C n1(C(C)C)ncc(C(=O)NCCCN(CCO)C(c2coc(Cl)c2)=O)n1 n1(Cc2ccc(C)cc2)cc(Br)c(=NC(=O)Nc2cc(F)c(I)c(F)c2)[nH]1 C(=O)(C#CC1CCCCC1)N1C(C)CCN(C(=O)Cn2nc(Cl)ccc2=O)CC1 c1(C2(C(=O)Nc3cnnn3C(F)F)CCC2)ccc(Cl)cc1.C12(CC1)C(=O)NC2 C1(NC(C(c2ccccc2F)C)=O)CCC(C)N(C(C2C3C4CCC(C4)C23)=O)C1 N1(C(c2cc(C(C)C)on2)=O)CC(C)CN(C(=O)CCCC(N)=O)CC1C c1(CNC(=O)NCC(c2cccc(Br)c2)(C)C)nc2c([nH]1)CCCC2 N1(C(C(C)CC(F)F)=O)CC2CC(C1)CN(C(=O)C=Cc1cccc(CO)c1)C2 c1(C(N(C2CCN(C(=O)COc3ccsc3)C2)CC)=O)nocc1Cl CC1(C)CC(CC(N2CC(c3ccccc3)(NC(=O)Cc3csnn3)C2)=O)CO1 C1(C(=O)NCCNC(C)=O)CCC=CC1NC(=O)COC1CCCOC1 n1(CC)ncc2cc(C(N3CC4CCC3CN4C(c3csc(Cl)c3)=O)=O)cnc12 N1(C(c2c(OC)nccc2)=O)C2CCC1C(C)C(NC(=O)CC(C)(O)C1CC1)C2 N1(C(CC2C(C)C2)=O)CCc2sc(CNC(c3nncs3)=O)nc2C1 N1(C(c2cnc(CC)[nH]2)=O)CC2CCC(C1)C(NC(C1CCCC(=O)C1)=O)C2 C(Cc1ccccc1)(C(=O)NNC(=O)OC)NCC1C(C(=O)OCC)OCC1 C(=O)(CCCCCC(C)O)N1C(CNC(CCc2cc(C)no2)=O)CC(F)(F)C1 CC1CN(C(c2cccnc2SC(F)F)=O)CCC1CNC(c1csnc1Cl)=O Cc1cc(C)c(CC(N2CC(O)CC2CNC(c2coc(C(F)(F)F)c2)=O)=O)s1 c1(OC(C)C)ncccc1C(=O)NCC(CO)NC(=O)C(C)CC1CCCC1 C(CC(C)C(=O)NC(CC1CC1)CC(=O)N1CCCC1CC(N)=O)OC N1(C(CCOCCOC)=O)CC2(CCCC(CNC(c3n[nH]c(C)c3O)=O)O2)C1 C1(N(C(C2C(C#C)C2)=O)CCOC)CCN(C(C2(C3CC3)CCC2)=O)CC1 N1(C(C(CCNC(=O)C=Cc2ccco2)OC)=O)CCN(C)CC1C N1(C(Cc2c(C)cccc2)=O)CC2CCN(C(C3CCOCC3(C)C)=O)CC12 c1(OC)cccc(I)c1C(N1CC2(CC(C(=O)NCC3CCC(F)C3)C2)C1)=O N1(CC(=O)N(CCC(C)NC(=O)C=C2CCC2)C)CCCC(C(F)(F)F)C1=O c1(C(N(C(C=C)CO)Cc2ccccc2)=O)cccc(-c2cncn2C)c1 C1(Cn2cc(CCNC(C)=O)nn2)CCCN(C(=O)Cc2ncc(Br)s2)C1 c1(CC(=O)NCC(C)(C2CC2)NC(=O)C=C2CCCC2)c(F)cncc1Cl C1(NC(c2c(C)scn2)=O)CCCCC1NC(=O)CCCOC(C)C c1(C(=O)NCC(C(C)C)NC(C(CSC)O)=O)cccc(N=S(C)(C)=O)c1 N1(C2CN(C(C3(C)CCC3)=O)C2)CCN(C(c2cncc(Cl)n2)=O)CC1 N1(CCC)CC2CCC(C1)N2Cc1ccc(O)cc1 C1(C(CNC(C=C(C)C(C)(C)C)=O)C)CCN(C(C2(CF)COC2)=O)CC1 CC(C)CC(O)C(=O)N1CCC(NC(=O)Cc2ncn3c2CCC3)C12CC2 C(=O)(C1=NOC(C)C1)NCCC1N(C(CC(CC)C)=O)CCCC1 C1(NC(C2N(CC)CCC2)=O)CCOCC1NC(=O)CCC(F)F Cc1cc(CN(C(=O)C=CC(C)NC(C2CCNC2=O)=O)C)no1 c1(C(=O)NC2(COC)CN(C(=O)CC3CCC4CC34)C2)nnn(C2CC2)c1C N1(C(C23C(CN(C(C(C)CBr)=O)C2)CC3)=O)CCc2sccc2C1 c1(C(N2CCC(CCNC(c3cncc(C(C)=O)c3)=O)C2)=O)ccc(N)cc1F CCCCC(C)C(=O)N1CCC(C(CO)NC(=O)CCC2CCCC2)CC1 CCC(C)CCC(=O)NC1CN(C(=O)Cc2cc(C(C)C)no2)CC1O C=CCCCC(C(=O)N1CC(C)(F)C1)NC(c1n[nH]cc1C#C)=O C1(NC(C2CCCCCC2)=O)C2CCCCN(C(=O)CC3CCSCC3)C12 c1(OC)cc(C)c2cc(C(=O)NC3(CF)CCN(C(C4CCOC4)=O)C3)[nH]c2c1 CCCCCCCCC(=O)N1CCC(O)C(N(C(=O)CSS(C)(=O)=O)C)C1 C1(NC(c2cscn2)=O)COC2C(NC(c3cccnc3OC(F)F)=O)COC12 c1(C(CNC(=O)Nc2ccc(F)cc2)Nc2csc(C(F)F)c2)ccccc1Cl C1(CN(C(c2scnc2C(F)F)=O)C2CC2)COCCN(C(C2CC(F)C2)=O)C1 CC1CC(CNC(=O)CC(C)(C)c2ccccc2)CCN1C(c1nccn1C)=O C(=O)(CC=C(Cl)Cl)NCC(C(=O)N(C1CCSC1)C)NC(N)=O N1(C(C2=C(C)CC2)=O)CC2(CC(NC(c3cccn3C(C)C)=O)CO2)C1 N1(C(C(C)SC)=O)CC2CCN(C(C3CCCC(=O)C3)=O)CC12 C1(C(=O)NCCCCCN(C(C(CC)F)=O)C)CC(OC)C(OC)C1 CC1(C)CCCOC1C(=O)NCC1CCC(NC(c2cnc(O)c(F)c2)=O)C1 N1(C(CC=CC)=O)CCCCC1CCN(C)C(c1cncnc1C1CC1)=O Cc1c[nH]c2cc(C(N3CC(C)(CNC(=O)CN4CCOCC4)C3)=O)ccc12 C(=O)(CCN=C(NCC(C)(C)C)NCCOC1CCCCC12OCCO2)NC C(=O)(CC(C)C(F)(F)F)NC1CC(C)(NC(C2CC(OC)C(OC)C2)=O)C1 c1(C(=O)NCC2CCCN(C(CC3CCC(C)C3)=O)C2)cc(O)cc(C#N)c1 N1(C(C2CC(C)(CC)OCC2)=O)CCC2CCN(C(c3coc(C)n3)=O)C2C1 c1(C(=O)NC(c2ccccc2)CNC(C2C(C)C2)=O)ccc(F)c2[nH]ccc12 N1(C(C(C(C)NC(=O)COC2CCC2)C)=O)CC2(CNC(=O)C2)C1 N1(C(c2cc(C)c(C3CC3)cc2)=O)CC(O)C2(CCOCC2)C1 C1(C)(CNC(c2ncc(OCC)nc2)=O)COCCN(C(C2SCCCS2)=O)C1 c1(C(=O)NCC2(F)CCCN(C(CCC=C)=O)C2)nccn2nc(C)cc12 C(=O)(C(C)CC(F)F)N(CC(=O)NCc1cnc(COC)[nH]1)C c1(C(=O)NC(CC(C)C)CNC(=O)CC(C)(C)C2CC2)cc2c[nH]nc2s1 n1(CCOC)nnnc1C(CCC1CCCC1)NC(COC)C1(C)CC1 CC(=O)CCCC(=O)N1CCC(C)C(NC(c2c(Cl)cnn2C)=O)C1 N1(C(c2ccn(CCC)n2)=O)CC2CN(C(C3OCCCC3(C)C)=O)CCC12 c1(C(N2CC3C(CNC(C4CC4(F)F)=O)C3C2)=O)nnc(O)c2c1CCCC2 c1(OCCC(=O)NCC2(C(=O)NC3CC(SC)C3)CCC2)ccccc1Cl c1(CC)ccc(C(=O)NCC2(NC(=O)CCc3ccc(Br)cn3)CC2)cc1 c1(C(N2CCC(n3c(C(=O)OCC)ncn3)C2)=O)cccc(C(F)(F)F)c1C c1(CC(=O)NCC2N(c3c(C(=O)OC)cncc3)CCC2)cn2cc(C)sc2n1 c1(C(=O)NC2CC(C)N(C(=O)Cc3cc[nH]c(=N)c3)C2)cnc2ccnn2c1O c1(C2(C)C(C(=O)NCC(C)CNC(=O)C(F)C3CCOC3)C2)ccccc1 N1(C(c2c(OC)csc2)=O)CCC(C)(C)C1C(=O)NCC1(C)CC(O)C1 c1(COC)nc(=N)[nH]cc1C(=O)N(CCCN(C(=O)CCCCCSC)C)C C1(C(=O)NC(C(CC)C)CO)CC12CCN(C(=O)C(c1cccc(O)c1)C)CC2 c1(C(C)C(=O)NC23CC(NC(=O)Cn4ccnn4)(C2)C3)ccc(F)c(F)c1 CC1CN(C(=O)C(=O)Nc2cnn(C)c2C(F)(F)F)CC1(C)Cn1ccnc1 Nc1cc(C(N2CC3CC2(C(=O)NC2(C4(O)CCC4)CC2)C3)=O)cc(F)c1 N1(C(C(C2CCCN(C(=O)C(CN(C)C)N(C)C)C2)C)=O)CC(CO)CC1(C)C c1(-n2c(C3(C)C(C)OCC3)nc(C3CSC3)n2)ccccc1S(C)(=O)=O c1(C(=O)NCC2(OC)CN(C(=O)COC(C)C)C2)csc2c1CCCC2 N1(C(CCOCC(C)C)=O)CCCC(CNC(=O)C(C)SCC2CC2)CC1 C(=O)(CCCCCF)NC1CCN(CCNC(C2N(C)C(=O)CC2)=O)CC1 CC1CN(C(=O)CCC2(C#N)CCC2)CC(C)CN1C(c1cnc(N(C)C)o1)=O C1(C(=O)NC2CCN(C(c3c(C)nc(CO)s3)=O)C2(C)C)Cc2ccccc2C1 C1(CC(=O)NC(C)CN(C)C(C2CCC(F)CC2)=O)CC2(CCCC2)CO1 N1(C(CCCCCC=C)=O)CC2CC(C)N(C(=O)C(C)Cn3ccc(C)n3)C2C1 C(=O)(C(CO)C(F)(F)F)N1C(Cn2cc(CCCCC)nn2)C=CC1 CC1(C)C(C(N2CCCC(NC(c3coc(Br)c3)=O)C2)=O)C1(C)C N1(C(CC)C)CCC2(CC1)CC2(C)C(=O)NCC1CCc2nccn2C1 c1(C(=O)NC2CCC(C(=O)NCC(C)(C)C)C2)cc2cccnn2n1 C(=O)(CCC(C)NC(=O)CN(C)CCOC)N(CCC#C)C N(C1CCc2ccc(O)cc21)CCC(C)(C)NC(=O)OC(C)(C)C C1(C(=O)Nc2ccccc2CO)CC12CCN(C(C1CC1(F)F)=O)C2 c1(C(c2nnnn2-c2cccc(OC)c2)NCC(CC)OC)sc(C)nc1C C1(C(=O)NCCSCC2CC2)CNCC12CCCCCC2 C(CO)(CCCCNC(=O)OC(C)(C)C)NC(C(CCSC(CC)=O)OC)=O CC1(F)CN(C(c2ccc3c(c2)CCCN3)=O)CCN(C(C23CC(C2)C3)=O)C1 n1(CC(N2CC3CC3(C(N3CC(O)C(O)C3)=O)C2)=O)cc2ccccc2n1 C1(C(N2CCC(C)(CC(=O)NCc3ncccc3NC)C2)=O)(CC)CCOCC1 c1(C(=O)OCc2c[nH]c(=N)o2)ccc(COC(F)F)cc1 C1(CC(=O)N(C)CC2CN(C(=O)CC3C=CCCC3)C2)CCCNC(=O)C1 c1(COCC)cn(CC2CCCN2C(=O)CCCc2cncs2)nn1 C(=O)(C(C)CS(C)(=O)=O)NCC1CCN(C(C2ON=C(C(C)C)C2)=O)CC1C C1(NC(C23CC(C(=O)OC)(C2)C3)=O)COC2(CCN(C(c3cc(F)cn3C)=O)C2)C1 N1(C(C=CCOC)=O)CCC(C=C)(C(=O)Nc2cccc(C)c2C)C1 CC1CCc2n[nH]cc2C1C(=O)NC(C)CC1CN(C(C2(C(N)=O)CC2)=O)C1 C(CC(O)CO)NC(=O)NC(C)C(F)F.C1CN1 C1(C(=O)NCCCn2cc(-c3cnc(C)s3)nn2)CCC2CCCCC2C1 Cc1cc(C(=O)N(C2CN(C(C3CC3C3CCCO3)=O)C2)C)sc1C N(C(=NCC=CCC)N1CCN2C(=O)OCCC2C1)C(C=C)C CC(C)(C(=O)NCCCCCCNC(c1cnc(C2CCCO2)s1)=O)C(F)F N1(C(CCc2cc(C)n(C)n2)=O)CCC(NC(C2CC(O)C2)=O)C1(C)C C1(CNC(C2C(NC(CCNC(=O)OCC)=O)CCO2)=O)CC1C1CCCC1 C1(C(=O)NCc2cccc(NC(Cc3n(C)ncc3Cl)=O)c2)CCC(C)(C)OC1 c1(NCC(CC)(C)OC)ccc(S(=O)(=O)N2CCCC3(CCC3)C2C)cc1Br N1(C(CCC(=O)NC)=O)CCC(C(N2CCC(C)(CN(C)C)C2)=O)C(O)C1 c1(OCCC(=O)NCC(C2CC2)NC(CSCCC)=O)ccc([N+](=O)[O-])cc1 C1(CNC(C(CSC)OC)=O)CCCCN(C(C2(C)CCC3CC3C2)=O)C1 N1(CCNC(=O)Cn2ccc(C3CC3)n2)CCCN(C(C2CC23CCCC3)=O)CC1 N1(CC(=O)N(c2ccc(C#N)cc2)CCS(N)(=O)=O)CCc2ccc(Cl)nc2C1 C(CC(=O)NCCN(C(C1(C)CC1F)=O)C1CC1)OCCC C(=O)(C1CCCc2nn(C)cc21)NC(C)C(F)(F)F C1(O)(C(CNC(c2n(CC)nnc2)=O)C)CCN(C(=O)CCC2CC(F)(F)C2)C1 N1(C(Cc2c(C)ccs2)=O)CCC(NC(=O)CCc2nccn2C)C12CCCC2 CCC(CC(=O)N1CC=CC(C(N2CCC(CC3CC3)CC2)=O)C1)C(C)(C)C N1(C(C2(COC)CC2)=O)CC2CC(NC(c3ccc(O)nc3Cl)=O)C2C1 CCC(COC)(c1nnnn1CCCOC)Nc1csc(Cl)n1 C(=O)(CCCCC(F)F)N1CC(COC)(NC(C2CC=C(C)CC2)=O)C1 c1(C(=O)NCC2C(NC(c3coc(Cl)n3)=O)COC2)ncc2cc(Cl)ccn12 O=C(CC1OCCc2ccsc21)NC1c2ccc(Br)cc2OCC1Cl C1(CNC(c2n[nH]c(C)c2Cl)=O)CN(C(C2CCN(C)CC2)=O)CC1(F)CO N1(C(C2CC(C)(C(=O)OC)C2)=O)CCN(C(c2cccc(=O)o2)=O)C(C)C1C C1(N(C)C(c2occc2-c2cnn(C)c2)=O)CCN(C(c2ccnc(S)c2)=O)CC1 Cn1c(Cl)nc2nc(Cl)nc(N3CCC(C(F)(F)F)C(C(N)=O)C3)c12 CC1(C)COCC(NC(=O)CCC2CC(NC(=O)C(F)C(F)(F)F)C2)C1 C12(CNC(=O)CCN3CCC3)CC1CN(C(=O)C(Cc1cccc(Cl)c1)=NO)C2 N1(C(Cc2c(CC)con2)=O)CCC(CC)(NC(=O)CC2CCC(F)(F)C2)CC1 C1(NC(c2cncc(C(F)F)c2)=O)C2CCC1N(C(c1cc(C3CC3)ns1)=O)C2 c1(C(=O)NC(c2cc(OC)ns2)C)ccc(S(=N)(=O)N(C)C)cc1 c1(C(N2CC(CNC(c3ccc(F)c(F)c3)=O)C2)=O)ccc2c(c1)COCO2 O=C(C1=Cc2ccccc2C1)NC1COCC1NC(=O)Cc1ncc(Cl)s1 N1(CC(=O)NCCN(C)C(c2csc3cncn23)=O)CCC(=O)NC1=O C#Cc1ccc(C)c(NC(C2CCCN(C(=O)CC3CCC(=O)N3)CC2)=O)c1 N1(C(=O)NCc2cn(C3CCN(CCCl)CC3)nn2)CCCC(CCF)C1 CC(C)CN=C(NCC12CCC(CC1)O2)N1CC2CC(C1)c1cccc(=O)n1C2 C1(CCNC(C2(C)CCCC2)=O)CCCN(C(C2(CF)CC(F)(F)C2)=O)C1 c1(C(=O)NCC2(O)CN(C(C3COCCO3)=O)C2)cnn2cnnc2c1 Cc1nc(O)nc(C)c1CC(=O)NC1CCCC1NC(C1CC12CCCCC2)=O CC1CCCN(C(c2ccnn2CCF)=O)C1CNC(=O)CSS(C)(=O)=O c1(N2CCC(OCCF)C2)nc(N2CCC3(CCSC3)C2)c2ccsc2n1 N1(C(C(N2CC(C)(NC(C(N3CCNC3=O)C)=O)C2)=O)C)CCc2ccccc21 C1(C(=O)NC(CNC(c2ccnc3cc[nH]c23)=O)CO)C2Cc3ccccc3C12 C1(CN(c2ccc(C(N)=O)[nH]2)C)CN(C(C2CCCN(C(N)=O)C2)=O)CCO1 c1(CNC(CCCOCC=C)=O)cccc(NC(C2OCCC2(C)C)=O)c1 C1(CNC(=O)CCCC2CCC2)CCC2(CO1)CC(NC(=O)CC1C=CCC1)C2 C12COCCN1C2=O.C1(CC)CC(NC(=O)CCC(=O)NC2CC2)C(O)C1 c1(C(C)(C)C#N)cc(C(N2CCOCC2)=O)cc(CO)c1 Cn1ncc(I)c1C(N1CCOCC1Cc1cn(C2(C)CC2)nn1)=O c1(N(CC(C)NC(c2nccnc2N)=O)C)nc2cccnc2s1 N1(Cc2ccc(OC)nc2)CCC2(CC1)CC2C(=O)Nc1ccns1 N1(C(c2cc(C)cc(N)c2)=O)CC2CN(C(=O)CCC3CCN(C)CC3)CC2C1 C=C(F)C1(CC(N2CC(O)CC2CNC(c2ccnc(C)n2)=O)=O)CCOCC1 CC(C)(C)C(CO)C(=O)N1CCCC(NC(=O)Cc2nc([N+](=O)[O-])n[nH]2)CC1 N1(C(C2C(C)C2)=O)CCC(C)(NC(c2cc(C(F)(F)F)ncn2)=O)C1 c1(CC(=O)NCC2CN(C(Cn3cnc(=N)[nH]3)=O)CC2O)c[nH]c2cccnc12 N1(C(CC2ON=C(CC)C2)=O)CCC(CNC(c2cnc(O)o2)=O)C1(C)C c1(C(N2CCC(NC(C(C)CC3CCCCC3)=O)C2)=O)ncccc1OCCF N1(C(C(C)C2CC2)=O)CCOCC(F)(CNC(=O)CCCCC(N)=O)C1 CC1OCCC1COC(c1ocnc1CNC(=O)OC(C)(C)C)=O Cc1ncoc1CNC(=O)C(O)CNC(=O)CCCC1CCC1 CCC(C(=O)NCCC(=O)N(CC)CC)NC(=O)C(C)CO N1(C(CNC(=O)C=Cc2cccnc2)=O)CCC2CCCCC12 C1(CCC)C(=O)NCCN1C(=O)CC1CCC(NC(C2CCCC(=O)C2)=O)CC1 S(=O)(=O)(c1cc(Cl)ccc1Cl)N1C2CC(N3CCN(CCC#N)CC3)C(C2)C1 N1(C(CCCN(C)CC2COC2)=O)CCCC(C(=O)Nc2ccccc2)C1 C1(C(N2CC(OCC#C)C2)=O)CCN(C(c2ocnc2CC#C)=O)CCO1 N1(C(CCC(C)OCC)=O)CCC(C)(C(=O)NC(C(O)CO)C2CC2)CC1 c1(C(N(CCCCNC(C23CCCCC2C3)=O)C)=O)c(O)cc(F)cc1F N1(C(c2c(CC)cccc2)=O)CC2CC(N(C)C(c3ccc(OC)s3)=O)C1C2 C(=O)(CCS(N)(=O)=O)NCC1(F)CN(C(COCCC)=O)C1 c1(C(=O)NCC2CCC(C(N3C(CC)C(C)CC3)=O)O2)ncc(F)cc1F N1(C(C23CCC(OC)(CC2)C3)=O)CCN(C(=O)CN2CCOCC2=O)CCC1C CSC1=C(C(=O)N2CCC(CNC(=O)C(F)F)C(C)C2)CCCC1 N1(C(C=CC(=O)OC)=O)CC2(COC(CNC(c3cnn4ccn(C)c34)=O)C2)C1 c1(NC(c2cccc(C)c2F)c2n(CCC)nnn2)cc([N+](=O)[O-])c(C)cc1C c1(C(=O)NCCCN(CCCNC(C(C)SC)=O)C)cnc(C(C)C)nc1 c1(C(N(CC(CN(C(=O)C(F)n2ccnc2)C)O)C)=O)cc2cc(Cl)ccc2[nH]1 C1(C(N2CCCN(C(c3ccc(N)c(Br)n3)=O)CC2)=O)CCc2ncnn2C1 N1(c2n(CC(=C)C)c(C(F)F)nn2)CC=C(C2(C(=O)OCC)CCC2)CC1 C(=O)(CCCS(=O)(=O)NCc1cc(C(=O)Nc2ccccc2C(C)C)no1)OC c1(C(N(C)CC2CN(c3nc(OC)c(Br)cn3)C2)=O)cc(Cl)c(F)cc1F C(=O)(CCCCCC(=O)NCC1CCN(C(C2CCC2C)=O)CC1)OCC C1(NC(CC=CCC)=O)CC2CCC1CN(C(c1cc3c(ncn3C)s1)=O)C2 N1(CC)CC(CNC(C2CCCC(CNC(C3CCCCC3C)=O)C2)=O)OC1=O c1(C(N(C2CN(C(=O)CC3CC(CF)C3)C2)C)=O)cnc(O)o1 C=CCC(CC(C)C)C(=O)N1CCCC(N(c2cc3nncn3c(C)n2)C)C1 C1(C(N(C2CCN(C(c3cc(C)n(C(F)F)n3)=O)C2)CCC)=O)CC(F)CN1C C(=O)(C(C)(C1CCC1)NC(=O)CN1CCSCC1)NCC(C)(O)C1(C)CC1 CC(C)C(O)C(=O)NCC1CC1C(=O)NCc1cnccn1 n1(CC)cccc1C(=O)NCC1CC1CC(=O)NCC(C)(C)CC1CC1 C1(CNC(Cn2nc(C)oc2=O)=O)OCCCC1(C)C c1(CC)onc(C(=O)N(C)CC2CCCN2C(c2ncc(Cl)s2)=O)c1C c1(NC2C(C(F)(F)F)C2)[nH]c(=NCC(F)C2CC2)nc2sccc12 C1(C)(C(=O)NCC(C)(C)SC)CC(O)CN1C(=O)C(C)CC1CC1 N1(C(c2c(C)occ2)=O)CC(NC(=O)C(C)(O)C(C)C)CC(F)C1 C1(c2nnnn2C)(NCc2cccc(C(=O)OC)c2)CCN(C)CC1C CCC(C)C(O)C(=O)N1CCC(CNC(c2ccc(Cl)cc2OC)=O)C1(C)C N1(C(CC2CC(CC)C2)=O)CCC(CNC(c2cc(N)cnc2C)=O)CC1C c1(C(=O)NC2CCCC(NC(c3cccnc3S)=O)C2)ccc2oc(S)nc2c1 N1(C(C(C)NC(=O)C2CC2)=O)CCC(C(=O)NCC2(C#N)CCCCC2)C(C)(C)C1 C12(C(N(C(c3ccccn3)CC)C)=O)CC(CO1)N(C(=O)OC(C)(C)C)C2 Cn1nc(C(=O)NCC2(NC(C3CCCN3C=O)=O)CCC2)cc1-c1cccs1 C1(C(N2C(CC(=O)NCCc3ccncc3F)CCC2)=O)CC2(CCC2O)C1 Cc1csc(C(C)C(=O)NC2CC(NC(=O)C(C)NS(C)(=O)=O)C2)n1 c1(C(=O)NC2CN(C(CCC(=C)Cl)=O)C(CO)C2)cc(F)c(F)cc1Br C(C(N=[N+]=[N-])C(=O)N(C(CNC(c1ccc([N+](=O)[O-])[nH]1)=O)C1CC1)C)OCC c1(C(N2C(C)CN(C(=O)C#CC3CCC3)C(C)C2)=O)ccnc2cc(Cl)ccc12 N1(Cc2nc(N(CCCC(C)O)c3ncccn3)sc2)CCS(=O)(=O)C2CCCC12 C1(N(C)C)CN(C(N2CC(OCC(C)(F)F)C2)=O)c2ccccc2O1 N1(C(c2ccn(C(F)F)n2)=O)CC2CCC(C1)N2C(c1c[nH]cc1Br)=O c1(C(N2CCN(C(c3cncc(OC)c3)=O)CC2)=O)ccc2ncsc2c1 c1(NC(c2cc(-c3ccncc3)[nH]n2)=O)ccc2c(c1)nnn2O N1(C(C(=O)NCc2cccc(Cl)c2)c2cnc[nH]2)Cc2ncsc2C1 C1(O)(C(C(=O)N(C(C)C(=O)NCCCn2cnnc2C)CCC)C)CCCCC1 C(=O)(C(O)C1=CCCCC1)NCc1ccc(CN(C(CCC(C)C)=O)C)cc1 N1(C(c2c(CCC)[nH]cc2)=O)CC(C)(C)CC1CNC(C1CCCC(F)(F)C1)=O O(NC(=O)N(CCCOC)C(C)C)C(C=C)C C1(C(N(CCNC(c2cc(Cl)ncc2O)=O)CC2CC2)=O)CCC2(CCC2)C1 C1(CNC(C(F)=CCC)=O)CC(NC(C2CN(CC(F)(F)F)C2)=O)C12CCC2 C1(C(=O)NC)CCN(c2cc(NCC3CCN(C(N)=O)C3)ncn2)CC1 N1(C(C23CCN(C(C4(NC(C)=O)CC4)=O)C2CCC3)=O)CCC(O)CC(C)(C)C1 Cc1c(C(=O)NC(C)CNC(=O)C(N2CCCCC2=O)C)c(Cl)nn1C C1(C(=O)NCC2(C(=O)NCC3CCC3(F)F)CC(=C)C2)CCCOCC1 C(=O)(CCCC(C)(C)NC(=O)C(C)OC(C)=O)NC(CC)CCCO c1(OC)nc(C(=O)NCC(C2CCCCC2)NC(=O)CC(C)(C)O)cc(O)n1 N1(C(CN)=O)CCC2(CC2C(=O)Nc2cccc(CF)c2)C1 N1(C(C2N(C(CC3CNC(=O)O3)=O)CC(O)C2)=O)CC2CCC(O)C2C1 Cc1cccc(C(=O)NCCNC(=O)Cc2cccnc2O)c1 c1(C(N2CC3C(CNC(c4cocn4)=O)C3C2)=O)ccc(F)cc1OC(F)F C(=O)(CC(C)C(F)F)N1CC(NC(CCN(CC)CC)=O)C(C)C1 C1(NC(C2(C)CCCCO2)=O)CCOC2(CCN(C(=O)CSC(=N)N)CC2)C1 c1(OC)ccc(C(=O)OC)cc1C(c1ccccc1)NC(=O)C(F)(F)F C1(CCNC(c2nccc(CC)c2)=O)C(C)CCCN1C(=O)C=CBr Cc1ccc2c(=O)c(C(=O)NC3CC(NC(=O)C#CC4CCCO4)C3)c[nH]c2c1 N#Cc1cc(C(=O)NC2CC2NC(=O)Cn2nc(-c3cccs3)oc2=O)no1 Cc1cncc(C(=O)NC2CCCC2NC(=O)C(O)CCN(C)C)c1C C1(c2ccccc2)(NC(C(C)NC(C2CCCC2=O)c2nn[nH]n2)=O)CC1(C)C N1(C(C(COC)C)=O)CCC(C)(C)C1CC(=O)Nc1ccc(Cl)c(OC)c1 c1(C(N2CC(NC(CCCCC(=O)NC)=O)C3C2C3)=O)ccc2c(c1)C(=O)OC2 C1(NC(=O)CN2CCOCC2)CC2(C1)CN(C(c1ccc(Cl)c(Cl)n1)=O)C2 C1(C(N(CCNC(c2ccc(NC(C)C)cc2)=O)C)=O)COC(C)(C)CO1 C1(C2CCCN(C(C3(N4CCCC4)CCC3)=O)C2)(NC(c2c(C)nsc2C)=O)CC1 c1(CC(=O)NCC2(NC(C3C(C=C)C3)=O)CCCC2)ccccc1SC c1(C(=O)NC2C(CNC(C(C)(C)c3cc[nH]n3)=O)CCC2)cccc2ccnn12 C#CC1CN(C(=O)CNS(C)(=O)=O)CCN1C(c1ccc(F)cc1F)=O N1(C(c2cc(OC)cc(F)c2)=O)CCC2(C1)CN(S(=O)(=O)CCCCCl)C2 N1(C(C2CC(F)(F)C2)=O)CCCN(C(=O)Cc2cnc(C3CC3)[nH]2)C(CO)C1 C(C(Cc1ccccc1)CC(C)C)NC(CN1CC(C(=O)OC)C(F)C1)=O Cc1cnccc1C=CC(=O)NCC(c1cccnc1)NC(C1CCC1C)=O C1(NC(C(C)(C)c2cnsc2)=O)CC2CCC(C1F)N2C(c1cnsn1)=O C(=O)(CCCN(C)N=O)N1C(C2(NC(C(COC)(C)C)=O)CC2)CCC1 C1(NC(c2cnc(Cl)s2)=O)CCOCC1NC(C1CC12CC2)=O c1(OC)ccc(CC(N2CC(NC(=O)CN3C(=O)CNC3=O)C3CC23)=O)cc1Cl N1(C(CCCN(C)N=O)=O)CCN(C(c2c[nH]c(=N)s2)=O)C2CCCCC12 CC(C)(O)C(F)C(=O)NCC(C)(C)OCCNC(=O)CN1CCOCC1 C(=O)(C(C)(C)C(F)F)NCCN(C(=O)CC1CCCN(C(C)=O)C1)CC C1(C(=O)NCC2C(C(C)C)C2)CCC(C)N1C(c1cccnn1)=O c1(NCC(=O)NC(CNC(Cc2c(C)occ2)=O)CO)cccc(C#N)c1 c1(C(=O)NCC(CC)NC(=O)COC2CC=CC2)c(N)cc(C)cc1F c1(C(=O)NCC2(NC(CCC)=O)CCCCC2C)cc(O)cc(C#N)c1 C(=O)(CCCCCC(C)C)N1CCCC(N(C(CCCC)=O)CCO)C1 C1(NC(Cc2c(OC)cncc2)=O)CC2(CCN(C(=O)C(C)c3ccco3)C2)C1 CC(C(=O)NCCNC(c1ccc(C(F)(F)F)c(O)n1)=O)C(F)(F)C(F)F C12(NC(C(CCSC)O)=O)CCC(C1)N(C(c1ccsc1SC)=O)C2 N1(C(C2C(=C)CC2)=O)Cc2nccn2CC(NC(c2cccnc2OCC)=O)C1 C(=O)(CCC(F)(F)C(F)F)N(C1CCCCCC1)CCNC(CSCCOC)=O c1(C(N2CCCCC(CNC(=O)CC3(O)CCC3)C2)=O)noc2cc(F)ccc12 C#Cc1cccc(C(C(=O)NC(c2ccccc2)C)N(C)CCSC)n1 C1(NC(CCSC)=O)C2CC3C1C3C2C(N1CC(F)(F)C1C1CC1)=O C(=O)(C(C)C(O)C(C)C)N1CC(C2N(C(c3c(C)cn(C)n3)=O)CCC2)(O)C1 CCC(C(=O)NC(C)C(CO)NC(c1ccnc(C(C)(C)C)n1)=O)C(C)(C)CC C12(NC(CSC)=O)CCCN(C(C3CN(SC(F)(F)F)C3)=O)CC1C2 Cc1ncc(CNC(=O)C(=O)NC(C2CCCCC2)C(C)C)s1 N1(C(c2nc(C)sc2C)=O)CC2CC(NC(=O)C(c3cccc(F)c3)C)C1C2 C1(c2n(C)ncc2)CN(C(=O)C(F)(F)c2cnccn2)CC1NC(=O)CC1CC1 CN1CCC(CCNC(C2CC=CCN2C(c2ccn(C)c2)=O)=O)CC1 CC1CN(C(c2ccc(-c3nn[nH]n3)cn2)=O)Cc2ccccc21 c1(C(=O)NCC(C)(C)NC(C(CC)n2cccn2)=O)ccc2snnc2c1 C1(N(C(=O)OC(C)(C)C)CC)CCC(C(F)(F)F)N(C(c2nc3sccc3s2)=O)C1 C#CCCCC(=O)N1CCC(CO)(NC(c2ccc(C3CCOC3)cc2)=O)C1 c1(OC)cccc(C)c1NC(=O)CC1COCCN1Cc1cncc(C)c1 C(=O)(C1Cc2ccc(Cl)cc21)N(CC(CN(C)Cc1ccc(S(C)=O)cc1)O)C C(=O)(CCC(C)(C)F)N1C(CNC(C2C(OC)CCC2)=O)C(C)CC1 C1(CS(C)(=O)=O)CN(C(=O)CCCNC(N)=O)CCN1C(C1CC(=C(F)F)C1)=O N1(C(c2cnc(OCC)s2)=O)CCN(C(=O)CCc2ccon2)C(C2CC2)C1 N1(C(c2c(C)ccn2C)=O)CCC(NC(=O)C(C)P(C)(C)=O)C(F)(F)CC1 N1(C(c2ccc(=O)n(C)c2)C(=O)NC)CCC2CCC(O)CC2C1 c1(C(=O)NC(C(CO)NC(C(CO)N(C)C)=O)C)nn(CC(F)(F)F)cc1Cl c1(C(=O)NC(C(C)C)CCN(C)C(C2CCC(F)C2)=O)ccc2nc(O)[nH]c2c1 C(=O)(CCCC(=O)N1C(C(=O)NC2(C)CC(N(C)C)C2)CC1C)OCC c1(N(C)Cc2nccs2)nc(=NC2CC=CCCC2)[nH]c2ccsc12 c1(CNC(=O)C=CCC2(NC(=O)CCCCO)CCC2)cc(CO)on1 C1(C(=O)NC(CC=C)CNC(c2nc(C)no2)=O)CCc2nnc(O)cc2C1 N1(C(CCCCCCSC)=O)CCC2CCC(C1)N2C(c1cccn(C)c1=O)=O c1(C(N2C(CN(C(C(COCC)C)=O)C)CCC2)=O)cnnc(C)c1C C1(NC(C(CC=C)C)=O)C2CC3C(C2)C13C(=O)N(C)Cc1cc(C)on1 N1(C(CC(c2c(OC)cccc2)C)=O)C2CCC1C(NC(c1cnc(C)s1)=O)C2 C1(CNC(c2cnc(C)o2)=O)CCCCC1N1CCN(C(=O)C(F)C(C)C)CC1 C(=O)(C(CCO)NC(=O)C1CC1)NC(C)CNC(C1(C(C)(C)C)CCCC1)=O.OC C1(C(=O)NC(C2CN(C(c3coc(Cl)n3)=O)CCO2)C)CCCCS1(=O)=O Cc1ncc(C(=O)NC2CC(C)N(C(c3cnn(C)c3C)=O)C2)cc1N C(CCN=c1ccnc(C(C)NC2CCCCCC2)[nH]1)OC(CNC(=O)OC)=O C(=O)(C=CS(F)(F)(F)(F)F)N1CC(C)(CNC(=O)Cc2ccc(F)cc2F)C1 C(=O)(C1=CC2CCCCCC12)NCC12N(c3nc(C)cc(OC)n3)CC(C1)C2 C(=O)(CS(C)(=O)=O)NCC(C1CCN(C(C2CCCN(CC(F)F)C2)=O)CC1)C c1(C(N2CCC(C(=O)NC(CO)C(C)O)(CC)CC2)=O)cc2ccccn2c1 c1(NC(=O)NCC(CC)OC)cccc(OCCN(C)C)c1 Cn1[nH]c(-c2nc(CCO)nn2-c2cccc(Cl)c2)nc1=O c1(C(N2CC(CC(C(=O)NC3CC4CCCCC34)F)C2)=O)cc2cccn2cn1 C=CCC(C)(CC)C(=O)NCCC1(O)CN(C(c2ccc(=N)[nH]n2)=O)C1 c1(C(=O)NCCNC(=O)C=CI)cnn(CC2CC2)c1 C(N=c1[nH]c(=NCC=CBr)c2sccc2[nH]1)c1[nH]cc(Br)c1 C1(NC(C=CC(C)NC(=O)C(Cl)Cl)=O)CCCC(C)(C)C1 c1(COCC(=O)N(CC(C)N(C(C=C(C)I)=O)C)C)ccccc1C CC1(C(N2CC(NC(c3ccsn3)=O)C2)=O)CCCCC1(F)F CON(CCC(=O)NCC1CCC(O)C1)C(=O)c1cccn1C1CC1 c1(OC)ccc(F)cc1C(=O)NCC1(O)CCN(C(=O)C2=C(Cl)CCC2)C1 c1(OC)ccc(C(=O)NC(CNC(=O)CN2CCNC(=O)C2)C2CCC2)nc1Cl c1(C(=O)NCCC2CCCCN2C(C2COCCO2)=O)cc(Cl)c(Cl)c(Cl)c1 N1(C(C2(OC)CC2)=O)CCC(NC(c2ccc(C)cc2OC)=O)C(F)C1 N1(C(COCC(C)C)=O)CCCC(CNC(=O)Cc2cncnc2O)CC1 Cc1coc(C(N2CCCC2CNC(C2CCOC2(C)C)=O)=O)c1C N1(C(c2c(SC)cn(C)n2)=O)CCC(F)(F)C(CNC(c2ncsc2C)=O)C1 S(=O)(=O)(CCCN=c1ccnc(NC2CCCC2OCC)[nH]1)N(CC)CC CC1OCCC12CN(c1nccc(=NCc3ccc(C(F)F)cc3F)[nH]1)CCO2 C12(NC(c3ccc(C(C)C)s3)=O)CCCCCC1N(C(C1CCCCS1)=O)CC2 c1(C(=O)NC2C3CN(C(CC4ON=C(CC)C4)=O)C2CC3)nccn2nccc12 CC1CN(C(=O)CSc2cccc[n+]2[O-])CC1CNC(c1ncnn1C)=O O=C(CS(=O)(=O)C1CCCC1)NCC(CNC(c1cccc2ncnn12)=O)CO C1(C(N2CC3CC3C2)=O)CC(O)CN1C(c1cc(Cl)c(Cl)s1)=O c1(CC)c(C(N2CCC2CNC(C2C(Cl)(Cl)C23CC3)=O)=O)cnn1CC c1(CNC(C2CC2C(=O)Nc2ccon2)=O)ccccc1-n1cccc1 CC1CC(NC(=O)Cc2ccccc2)CCN1C(=O)Cc1ccsc1 N1(C(CSc2ccc(OC)cc2)=O)CCC2(CCN(C(c3cn[nH]c3)=O)C2)C1 C1(C(C)C)CN(C(=O)CC(CC2CC2)NC(=O)CC2COCC2O)CCO1 c1(C(=O)NC2CCC(CCC)C2)cccc(CNC(=O)CS(C)(=O)=O)c1 C1(CC)CN(C(=O)C(C)OC)CCN1C(C1CC(N(C)C)C1)=O C1(C)(CNC(CC2(CSC)CC2)=O)CCN(C(=O)CCCc2n[nH]c(=N)s2)C1 c1(CNC(C(C(C)C)O)=O)ccc2c(c1)CCN(C(C1CCCN1C(C)C)=O)C2 C1(C(=O)NCCCC2CCN(C(c3nc(C)n(C)n3)=O)CC2)CCC12CCCO2 N1(C(c2c(C)ncn(C)c2=O)=O)CC2COCC(C1)C2NC(=O)Cc1cccs1 C1(O)(C(C)NC(C(C)NC(=O)NC)=O)CN(C(=O)CC2CCCO2)C1 c1(C(N2CCCC(CN(C(C(CC3CC3)OC)=O)C)C2)=O)cc(C)ccc1C C1(C(N2C(C)CC(NC(C3CC(=C)C3)=O)C2)=O)CCC(C)=C(C)C1 C1(CC(=O)NCCCC(C)CO)CCN(C(c2ncc(F)cc2N)=O)C1(C)C CC1(CNC(=O)NC2(CC(=O)NCCNc3cc[nH]c3)CCC2)CCCS1 N1(C(c2ccc(C#N)nc2)C(=O)Nc2ccccc2)CC2OC(=O)OC2C1 c1c(C)nc(C)n1C.CCCC(=O)N1CCC1CS(N)(=O)=O c1(C(=O)NC2CC(C)N(Cc3nc(=O)n(C)[nH]3)CC2)ccc2oc(O)nc2c1 CC1=CC(C(=O)NC(C(=O)N(C)Cc2ncnn2C)C2CCCO2)SC1 N1(C(C2(CC=C)CC2)=O)CCN(C(=O)CCOC2CCCCC2)C(C2CC2)C1 C1(NC(c2cccc(N3CCCC3=O)c2)=O)(CO)CCN(C(c2ccoc2)=O)C1 C(CCCCCC(=O)NCc1cc(C2CC2)on1)NC(c1nn(CC)nc1C)=O c1(C(N2CC(CNC(CSCCOC)=O)C3C2C3)=O)ccc(C)cc1C C#CC1CCC(CNC(c2csc(CNC(C3CCC4CC3CO4)=O)c2)=O)CC1 Cc1nc(C(N2CC(c3ccccc3)CC2C)C(=O)NC2CCC2)sc1C Cc1ccc(-n2cc(C3CCCN(C(c4ncccn4)=O)C3)nn2)cc1 N1(C(C)=O)CCCC1C(=O)NCC(C)N(C(=O)Cc1nonc1C)C1CC1 N12CCOC(C)(C1)NC(=O)CC2.C1(COC(=O)NC(C)C)CCCN1C(C)C C1(C(=O)NCC(C2(O)CN(C(C(C)(C)OC)=O)C2)(C)C)CCCC(C(=O)OC)C1 c1(CC)ccccc1SCC(=O)NCC(C1CCOC1)NC(c1n[nH]c(C)n1)=O C1(C(=O)NC(C(=O)N(C)CC)C)CCN(C(=O)C(C)=CC(C)(C)C)C1 O=C(C1=CCCS1)NC(CNC(c1cncc(F)c1)=O)C1CC1 N1(C(C(C)NC(C2CCCC2)=O)=O)CC=CCC2(CCCC2)C1 c1(CNC(C2CC2NC(c2ccc(Br)s2)=O)=O)cnc(O)nc1O c1(C(N2CCC(CCNC(C=CCC)=O)C2)=O)cc(Br)c(O)nc1C C1(C(=O)NCCOCCC#C)C(CC)CCN1C(=O)C(C1CCOCC1)F C1(CNC(c2nccc(C#C)c2)=O)CN(C(c2conc2C)=O)CC(C)(C)C1 c1(CNC(CNC(COCC)=O)=O)nnc2nc(C)cc(C)n12 C(c1cnccc1C)=CC(=O)NC1CC(CNC(c2nc(COC)[nH]n2)=O)C1 C1(C(N(C)CC2(CNC(COCC(=C)C)=O)CC2)=O)CC1(F)F N1(C(c2cncc(C(=O)OC)c2)=O)CCC2CN(C(=O)CN3CCC3C)CC2C1 C1(NCC(=O)NCC#C)(CO)COC1 c1(C2(NC(=O)CSc3ccccc3)CC2)ccc(OC(F)F)cc1 c1(C(=O)NC(C)CN(C)C(c2cncn2C)=O)ccc2c(c1F)CCC2 C(C(C)(C)CC(=O)NC(CC1CC1)CO)NC(c1n(CC)ccn1)=O c1(C(N2C(C)CC(NC(C3(C(F)F)CCCC3)=O)C2)=O)ccc(Cl)c(F)c1 c1(NCCNC(c2n(C)nnn2)CC2CCC2)cccc(Cl)c1 c1(NC(C(C(C)NC(c2cc3n(n2)CCO3)=O)(C)C)=O)ccc(O)c(=O)cc1 S(=O)(=O)(c1ccc(NCC2COCCO2)c(Br)c1)NC(C)(C)CCCO N1(C(CC2(C)CC2)=O)CC23CCCC2(C1)CN(C(C1CCCC(=O)N1)=O)C3 C=CCC(CC(C)C)C(=O)NC1(CNC(=O)C(C)CCc2cccc(F)c2)CC1 CCC(CC(=O)NC1CCN(C(=O)Cn2ncn(C)c2=O)CC1F)C(F)F c1(-c2cc(CC(=O)NCc3ccccc3F)ncc2)cc(F)c(F)c(F)c1F N1(C(CN(C(C)=O)C)=O)CC2CCC(CNC(=O)Cc3cn(C)cn3)C2C1 N1(C(Cn2c(C)ncc2[N+](=O)[O-])=O)CCCC2C1CCN2C(=O)Cc1cnsc1 C1(CNC(C=CC(C)(C)SC)=O)CN(C(=O)C(C(C)C)n2cnc(C)c2)CCO1 C1(OC)CN(C(=O)CNC2COCCN2C)CC1NC(=O)OC(C)(C)C Cc1cc(C(=O)NCC(O)CNC(=O)C(C)(F)F)cc(F)c1C C(N=c1[nH]cnc2ccsc12)C1CCC(NC(c2sccc2F)=O)C1 N1(C(CCCC(=O)NCC)=O)CC(CNC(=O)C(O)C(C)CC)C2CCCCC12 C1(C(N2CCC(NC(CN(CC)Cc3ccc(Cl)cc3)=O)C2)=O)C2CCN1CC2 c1(C(=O)NC2CC(NC(CC(=C)C)=O)C23CCC3)ccc(C)c2ncccc12 Cc1cn(CC(=O)NC(C)CCN(C)C(c2cn[nH]c2)=O)c2ccccc12 CC1CN(C(c2ccc(CC3CCC3)o2)=O)CCC1NC(=O)CCc1cnoc1 C1(C(=O)NC(C2CN(C(c3n[nH]c(C(C)(C)C)n3)=O)C2)C)CC=CCC1 c1(NC(C2CC(=C)CN2CCc2c(O)n[nH]c2C)=O)ccc(F)nc1F O=C(C1=C(Cl)CCC1)NCC1CCCCN(C(=O)COC2CC(F)(F)C2)C1 c1(-c2c(C)cccc2C)cc(=NC(=O)CC(C)c2ccc(F)cc2)[nH][nH]1 c1(C(=O)NCCCNC(CSc2n(C)nnn2)=O)cncc(OCC(F)(F)F)c1 C1(NC(c2ccc(CC)cn2)=O)CC(F)CN(C(=O)CCOCC2CCCO2)C1 C1(CNC(Cc2cc(C)ns2)=O)CC2(CO1)CN(C(=O)C=C(Cl)Cl)C2 C1(CN(C)C(c2ccc(O)nc2)=O)CCN(C(C2CCOC2C(F)(F)F)=O)CC1 C1(CNC(CCc2ccc(C)o2)=O)CN(C)CCN1C(c1cncc(Cl)c1Cl)=O Cc1ccc(F)c(C(=O)NC2CCC2NC(C2(CO)CC23CCC3)=O)c1 c1(NC(c2n(CC(=C)C)nnn2)c2cscc2C)cc2n(n1)CCCCO2 c1(C(N2C(C)C(NC(=O)CC3CCOC3)CC2)=O)ccc2c(c1)CC2 N1(C(c2c(C(C)C)cccc2)=O)CCC2(CC1)CC2NC(C1(C)CC=CCO1)=O c1(-n2c(C3N(C)C(=O)CCC3)nc(C3CC3)n2)nnc2n1CCNC2=O c1(C(N(CCCN(C(CCOCCC)=O)C)C)=O)ccc2c(c1)CC(C)(C)O2 c1(C(=O)NCC#CCNC(C2CC3CCC2O3)=O)cc2cc(O)ccc2[nH]1 C(C1c2ccccc2CC1C)NCc1cc(OC)c(F)cc1F C12(C(N3CC=C(C)CC3)=O)CCC(CN(C(c3cnn(C(F)F)c3)=O)C1)C2 N1(C(C2(C)C(C)C2)=O)C2CCC1C(NC(=O)COCCF)C2 CC#CCC(CO)NC(C1CCC(C2CC2)N1C(c1cnn(C(F)F)c1)=O)=O c1(CNCCCCC(C)(C)C)ccnc(S(C)(=O)=O)c1 CCC(C)(CCC(C)C)C(=O)NC1CCN(C(=O)CCc2nc(O)n[nH]2)CC1O C1(C2CCN(C(C3CC3[N+](=O)[O-])=O)C2)(NC(=O)C=CC2CCCCCC2)CC1 N1(C(C(CC)C)=O)CCN(C(c2ncn(C(C)(C)C)n2)=O)CC12CC2 Cc1ccc(C(=O)NCCN(C(=O)CC(C)O)C(C)C)c(F)c1C C1(c2cn(CCCC(=O)NCCN3CCC(CSC)C3)nn2)(OC)CCCCC1 c1(C(=O)NCC(CC(C)C)NC(=O)C2=NOC(C)C2C)ccc(S(N)(=O)=O)cn1 C1(NC(=O)CC2CCCOC2)CCOC12CCN(C(=O)C=CC1CC1)CC2 N1(c2sc(C#N)c(Cl)n2)Cc2ccccc2C(CNC(c2cnccc2Cl)=O)C1 Cc1cc(C(=O)NCC2C(O)C(O)CN2C(C2CCS(=O)(=O)N2C)=O)cc(F)c1 N1(C(C2CC(C)(NC(C3C(CCC)C3)=O)C2)=O)CCC2CC1C(=O)O2 C1(C(=O)NC(C2OCCN(C(c3ncc(OC)cn3)=O)C2)C)CNC(=O)CC1C CC1CN(C(c2cn(C)nn2)=O)CC1CC(=O)NCCc1cccs1 c1(NC(CCOCCOC)=O)cccc(NC(C2(C)CCC(C)C2)=O)c1 Nc1cc(Cl)nnc1C(N1CCC(O)(CNC(c2c[nH]c(C(F)(F)F)c2)=O)C1)=O C(=O)(C(C)(C)C(=O)N(C)C)NCCNC(C(C1CC(F)(F)C1)OCC)=O c1(C(N2C(Cc3cn(C(C(C)O)C)nn3)CCC2)=O)ccc(Cl)c(Cl)c1 c1(OC)cc(C(=O)NC2(C(N3CC(O)(CNC(C)=O)C3)=O)CC2)cc(F)c1 Cc1ccc2c(c1)CC(C(N1CCC(NC(C3CCN(C)C3)=O)C1)=O)S2 CC1CN(C(C2CCCC2)=O)CCC1CNC(=O)C(C)(C)C1CC1 c1(C(C)NC(Cn2c(C)ncc2)=O)ccc(CNC(=O)C(O)C2CCCC2)cc1 N1(C(C2CC(C)OC2)=O)Cc2nccn2CC(NC(C23CCCC(C2)OC3)=O)C1 c1(NC(CCC)=O)ccc(OC2CCN(C(c3ccc(C(N)=O)o3)=O)C2)nc1 CCC(C)CC(=O)C(=O)NCC1CN(C(=O)CCS(N)(=O)=O)CCC1C C(=O)(C(F)C(C)(C)O)NC(C)(C)CCCNC(c1csc(C(F)(F)F)n1)=O n1(CCC)ccc(C(N2CC(C(N)=O)(CNC(=O)CC(O)C3CCCC3)C2)=O)n1 C(CC1=CCN(C(=O)CC2=CCCCC2)CC1)NC(C1CC2(CC(=C)C2)C1)=O c1(NC(=O)Cn2cnc(C(=O)O)n2)cccc(-n2cc(CO)nn2)c1 c1(NC(C)CC(C)(C)OC)nc2ccccc2nc1NC(C)CCC1CCCC1 N1(C(C(C2(C)CC2)NC(=O)CC(C2CC2)C2CC2)=O)CC(=O)NC(C)C1 Cc1c(NC(c2c(-c3ccc(CCCO)cc3)cnn2C)=O)cc(F)cc1Br c1(C(N(CCCCNC(C(CC)c2cccnc2)=O)C)=O)ncnc(O)c1Cl C1(C(N(CC(=O)N(CCC(=O)NC)C)CC)=O)CC(=O)N(OC)C1 c1(CN(C(C(=O)OCC)CC)C2CC2)c(Br)cc(OC)c(F)c1F N1(C(C2(C#C)CC2)=O)CC(NC(=O)CCCN(C)C(C)=O)C(C)C1 N1(C(c2c(CC)cno2)=O)CCOC(CCNC(c2cscn2)=O)C1 CC1(C)CN(C(=O)CC2(Cc3ccccc3)CC2)CC1NC(C1(C)CC1Br)=O C(=O)(C1=CC2(CCOC2)C1)NC1CCC(C(N2CC(N(OC)C)C2)=O)CC1 CCCCCC(=O)NC1CCCC(NC(=O)C(C)C#N)C1 CC(Cc1cnn(C)c1)C(=O)NC1(CCCNC(=O)COC2CC2)CCCC1 N1(c2ncnc(C(=O)OCC)c2OC)CCC=C(C(=O)NC2CNCCC2)C1 c1(CC(N2CCC(NC(CC3CCN(C)CC3)=O)(CF)C2)=O)ccc(Cl)c(Cl)c1 C(CC(C)(C)C(=O)NC1CCN(C(c2nccn2C)=O)CC1CO)OC O=C(C1=CC2CCC(C1)C2)NCC(=O)NCC(N1C2C=CCC1CCC2)=O C(=O)(C(C)(C)CCCNC(c1cnc(C)n1C)=O)NC(CC)C(O)C(C)C N1(C(c2ccc(Cc3ccccc3)s2)C(=O)NCC)CCN(C2(C)CCC2)CC1 N1(C(C2C(C)=C2)=O)CCC(NC(=O)C=C2CCSCC2)C12CCCC2 c1(CCNC(=NCC=C)NCCC2(C)CC2(F)Cl)ccc2c(c1)OCCO2 c1(C(N(CC(O)CNC(c2ccccn2)=O)C)=O)sccc1S(C)(=O)=O c12ccc(cc1)[nH]2.C1(CC=C)CCCC1(c1nnnn1CCCF)OCCOC C(=O)(C1=C(C)OCCS1)N1CCC2C(NC(c3nn(CC)nc3C)=O)C2C1 N1(C(c2cc(CSCC)on2)=O)CCC2(CCN(C(c3cccc(C)c3)=O)C2)C1 NS(=O)(=O)c1ccc(NCCOCCF)cc1Br C1(OCC(=O)NC(C(=O)NCc2ccoc2)C2CCCO2)CC=CC1 c1(CNC2(c3nnnn3CC)C(CCC)COCC2)cccc(F)c1OC(F)F C1(C(C)C)CN(C(c2cnc[nH]2)=O)CCCN1C(c1cc(S(N)(=O)=O)c[nH]1)=O Cc1ccc2cc(C(N3CCN(C(=O)Cc4cncnc4)C(C)C3)=O)ccc2n1 c1(C(=O)NC(C)CNC(C2CC2[N+](=O)[O-])=O)ccc(N)c(Br)n1 C1(O)(CN(C)C(C2(CF)COC2)=O)CCCN(C(C2CCCCN2C)=O)C1 C(=O)(CC(C)C(F)(F)F)NC(CCC)CCCN(C(=O)Cc1cnc[nH]1)CC CCC(C)CC(C)C(=O)NC1(CC(=O)NCC2(SC)CCC2)CCC1 c1(C(=O)NC(C=CC(=O)NC2C(OC)C(O)C2)(C)C)nc(=N)cc[nH]1 c1(OC)cc(F)c(F)cc1NC(=O)C(c1ccc(C)cc1)C C(CC(=O)N1CCCCC1CCNC(=O)C=C(C)c1cccs1)(C(F)(F)F)OC C1(CNC(C2CC=CCO2)=O)CN(C(c2sccc2F)=O)C2CCCCC12 Cc1cccc2c1CN(C(C1CC3(CCC3)CN1C(=O)COC1CC1)=O)C2 c1(C(=O)NCCC2(C)CCN(C(C(C)(C)N(C)C)=O)C2)c(F)ccc2occc12 C12(NC(CCCC#C)=O)CCCC1N(C(=O)C(c1ccn(C)c1)C)CCC2 O=C1COC(C(=O)NCC(C2CCCC2)NC(C2CCSC2)=O)C1 N1(C(C(CC)SC)=O)CCN(C(c2[nH]nc(C(F)(F)F)c2C)=O)CC1C1CCC1 c1(C(N(C2CCN(C(C3C(C)C3C)=O)C2)C)=O)cccc(Cl)c1O CCC(Cc1ccccc1C)C(=O)N(C)Cc1cc(C#N)cs1 Cc1cc(C(N2CC(C3(NC(=O)COCCOCCO)CC3)C2)=O)cc(Cl)n1 c1(NC(CNC(c2cccc(OC)c2)C(=O)O)=O)cn(C)c2ccccc12 c1(OC)cccc(Cl)c1C(=O)NCCCCNC(C1CCCC(C#N)C1)=O C1(CNC(CC2CN(C)C2)=O)CN(C(c2cncc([N+](=O)[O-])c2)=O)C2(CCC2)C1 C1(CC(=O)N(CCCNC(c2csc(CC(F)F)n2)=O)C(C)C)CCCS1(=O)=O CN=C(NCC1CCOC1)NCC(CC1CCC1)CO c1(CCC)nsc(N)c1C(=O)NCC(C1CC1)NC(c1cn(CCC(C)C)nn1)=O CCC(C)C(C(=O)NCC(CO)NC(C1(C)CC=CCC1)=O)NC(C)=O C(C)(CCC(=O)N(C1CCN(C(C2CC2F)=O)CC1)CCO)OCC C(c1ccc(C(=O)OC)cc1)=C(C(=O)NC(c1ccccc1F)CC)C c1(C(=O)NC(CCN(C(C=CC=CC)=O)C)C)ccc2ccn(CC(F)F)c2c1 c1(NC(C(C2CC2)NC(C2(CCC=C)CC2)=O)=O)cc(F)ccc1OC CP(C)(=O)c1ccccc1C(=O)NCCCOCCNC(c1c[nH]c(=O)cn1)=O C1(CNC(C2CCC(CNC(C(C)SCC)=O)O2)=O)CCCCC1(C)C C1(CNC(C2CC2Br)=O)CCCCN1C(=O)CCc1cccc(O)n1 c1(-c2cc(C(N3C4CN(C)CC3CC4)=O)sc2)cccc2c1cnn2C C1(CC)(CC)CC(N=c2nc3c(cnn3C(C)C)c(NCCS(=O)(=O)NC)[nH]2)C1 C#Cc1ccccc1C(=O)NCC1CCCN1Cc1ccnn1-c1ccccc1 C1(NC(c2scnc2C(F)F)=O)C=CCN(C(C2CC=CCC2)=O)C1 C1(F)(CNC(CCC2(C)CC2)=O)CCN(C(=O)CSc2cn[nH]c2)C1 C1(CC)(CNC(=O)C(CO)NC(=O)C(C)c2ccco2)CCCC1 C(CNC(C1(C(F)F)CC1)=O)(C(C)(C)C)NC(c1c(CC)[nH]cc1)=O c1(C(N(C2CCN(C(COCCCC)=O)CC2)C)=O)cc(CC)cc(F)c1 N1(C(=O)NC2(C(C)(C)C)CCNC2)CCOc2ccc(Cl)cc2C1 CC1(C(=O)NCc2ccnc(F)c2)CCN(C(c2ccccc2S)=O)C1 C=CC1(C(=O)NC2CC3(CCC3)C2O)CCN(C(=O)CCOCC(C)C)C1 c1(C(=O)NCc2cc(C(N3CCC(C)(CC)C3)=O)ncc2)cccc(C)c1F C(CN=C(NCC(C)Cc1cccc(C)c1)NCC1CCCC1OC)SC N#CCCCCC(=O)NCC12CC1CN(C(c1ccc(C(F)(F)F)c(F)c1)=O)C2 C1(NC(NNC(C23CN(C(C)=O)C(C2)C3)=O)=O)CCC(F)(F)CC1 c1(C(=O)NCC2OCC(CNC(c3nnn(C)n3)=O)C2)cc2ncccc2[nH]1 C(=O)(CCCC(C)(F)F)N(C1CCCN(C(CCCc2nc(C)sc2)=O)C1)C N1(C(C(F)=CC)=O)CC(C)(CNC(=O)CC2CCCC2(F)F)CC1(C)C c1(N(S(C)(=O)=O)C)cccc(C(=O)Nc2ccccc2C(N2CC(O)C2)=O)c1 N1(C(c2cc(C(=O)OC)cn2C)C(=O)NC2COC2)CC2CC=CCC2C1 N1(C(C(c2cccc(F)c2)C)=O)CC(NC(c2cnn[nH]2)=O)CC12CCOCC2 C(=O)(C(C)(F)CC1CCCC1)N(CCCNC(c1sccc1F)=O)C C1(C(=O)NC2CC(=O)OC2)C2CCC(C2)N1C(c1ccnc(C(F)F)c1)=O C(=O)(C(CCOC1(CC#C)CCC1)NC(=O)Cc1ncoc1C)NCCO Cn1cc([N+](=O)[O-])c(C(=O)NCC(C)(C)CCNC(C2CCC(=O)N2)=O)n1 C1(NC(CSCC(C)C)=O)CN(C(C2CCC(=O)N2CCN(C)C)=O)CC1C C1(NC(C(C=C=C)C)=O)CCC2(CC1)CC(NC(c1ccc(COC)s1)=O)C2 c1(C(=O)NCC2C3CN(C(C4(C=C)CC4)=O)CC32)c(OC)cccc1OC C1(NC(=O)CS(=O)(=O)C2CC2)CCC2(CCN(C(c3csnn3)=O)C2)C1 C#CC1(C(=O)NCc2ncccc2Cl)CCN(C(=O)C(c2ccc(C)o2)C)CC1 CCCC(C)C(=O)NC12CC1CN(C(C1CC(O)(CCC(C)(C)C)C1)=O)C2 c1(C(=O)NC2CC(C)(C)N(C(C3CCN3C3CCC3)=O)C2)ccc(F)c(O)c1F c1(C(=O)NCC(C)N(C(c2n(CC)ncc2)=O)C)ccc(C)c(O)n1 C#Cc1cnn(CC(N2CC(CNC(C3C4CC5C(C4)C35)=O)(OC)C2)=O)c1 c1(NC(c2ccnc(Br)c2F)c2n(CC)nnn2)ccc2c(ccn2C)c1 CC1(C(=O)NC2CCCCC2NC(C2(C3CCC3)CC2)=O)CC(C#N)C1 C1(NC(CNC(C2C(C)C2)=O)=O)CN(C(=O)C=CC(=O)OC(C)(C)C)CC1(C)C CC1CN(C(c2ccc(O)nc2)=O)CC(CCNC(=O)CC2CCC=CCC2)O1 c1(C(=O)OC)ccnc(N2CCC(OCCNC(=O)CC3CCOC(CN)C3)C2)n1 CCC(C)C1C(=O)N1.c1(CSC)nc(CCNC(=O)CN(C)C(=O)OC)n[nH]1 c1(OC)cc(CCC(=O)NC2CCC(CNC(C34CSCC3C4)=O)C2)on1 Cc1ccc(CNC(=O)C(C2CCN(C(c3csc(C)c3C)=O)C2)C)cc1C S(=O)(=O)(c1cnc2ccccc2n1)NC(C(=O)N(C)C)Cc1ccccc1 CCC(C(=O)NCC(C)NC(c1nc2cccnc2s1)=O)C(C)(F)F C1(NC(c2cc(C)c(O)nc2)=O)CC2(CCN(C(C3(CO)CCCO3)=O)CC2)C1 N1(C(CCCN(C)C)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)C(CC2CC2)C1 C1(CNC(C(C=CC)O)=O)COCC2(CCN(C(=O)Cc3coc(C)n3)CC2)O1 CCC(C)CC(C)C(=O)NC1C=CCN(C(=O)Cc2cscc2C(=O)OC)C1 C(=O)(C(C)C(O)C(C)C)NC1C(NC(c2c(OC)oc(C)n2)=O)CCC1 N#Cc1ccc(C(N2CCN(C(=O)CCN3CCCC3)CC2)=O)c(F)c1F N1(C(C2(NC(C3CCC(C)O3)=O)CC2(C)C)=O)CC2CCC1C(O)C2O N1(C(c2c(C)cccn2)=O)CCCC(C2CN(C(c3cn4c(n3)SCC4)=O)C2)C1 c1(CC(=O)NC2(C)CCN(C(CCCC=C)=O)C2)cn2c(C)cncc2n1 C1(CNC(C(CCC)OCC)=O)CC2COCC2N1C(=O)C(O)CCSC c1(C(=O)NCCC2(NC(C(C(C)C)C#N)=O)CC2)cc2c(cc1F)OCC(=O)N2 C(CC(C)(C)CC(=O)NC1CCN(C(c2nc(O)[nH]c(=O)n2)=O)CC1C)OC N1(C(c2c(C)cn(C)c2)=O)CCN(C)CC1C(=O)NCCCC1(O)CCC1 C1(NC(COC2(C)CCCC2)=O)CCOC(CNC(=O)CC2(O)CCCOC2)C1 Cc1c(C(=O)NC(CNC(c2coc(C(F)F)n2)=O)CO)[nH]c2ccccc12 c1(CNC(N)=O)cccc(C(C(=O)C(=O)NC2(C3CCCO3)CCCC2)=O)c1 O=C1CCC(CC(N2CCC(N(C(=O)C(=O)Nc3ncc[nH]3)CCO)C2)=O)N1 C1(NC(CN(C)C2CC2)=O)CCC(CN(C(=O)CCc2cccnc2)C)CC1 c1(C(N2CCN(c3ccc(Cl)cc3)CC2)=O)ccn2ccsc12 c1(COC)cc(C(c2nnnn2C)NCC2CCOC2(C)C)ccc1Br C1(C)(C(=O)NCC(CN(C(C2CCN(C)C2=O)=O)CC)(C)C)CNC(=O)C1 c1(OC)nccc(Br)c1C(=O)NC1CCC(N(C(=O)CS(C)(=O)=O)C)C1 c1(CCN(CCC(=O)NC(C(=O)NCCC)C)C)ccccc1 Cc1cccnc1C(=O)NC1CC(NC(=O)Cc2sc(C3CCC3)nc2C)C1 O=C(C1CCSc2ccccc21)NC1CCC(N2CCCS2(=O)=O)CC1 C=CCCCCCCCC(=O)NCCC1(CNC(C2OCCC2C(C)C)=O)CC1 C1(CNC(C(CCC)F)=O)CC(C(=O)NC(CCO)C(F)F)=NO1 c1(C(N2CCC(C(C(=O)NC3(CSC)CC3)C)C2)=O)ccccc1C#N N1(C(C(c2cccnc2)C)=O)CCCC(N(C(=O)CC2C=CS(=O)(=O)C2)C)CC1 C(C(=O)N1CC2COCC2O1)C1N(C(CCC(C)(F)F)=O)CCC1 c1(CN(C(C2C(C)C2(F)F)=O)C)nn(C)cc1Br Cc1c(CN2CC(C(N3CC(F)C(F)C3)=O)C(O)C2)sc2ccccc12 CC1CCC(C)C1NC(=O)C(c1cccnc1)NC(=O)COC1CCCC1 N1(C(C(C)Cc2ccccc2)=O)CCC2CN(C(=O)C3=CCCS3)C2C1 N1(C(C=CC(C)NC(c2cnc(Cl)n2C)=O)=O)CC(CO)C1(C)C c1(C(=O)NC23CCN(C(c4n(CC)ccn4)=O)CC2C3)cc(C)c(F)cc1F C1(C(N(C)CC2C(NC(CCCC#C)=O)CCC2)=O)COC2COCC2O1 N1(C(Cn2nnc(=N)[nH]2)=O)CC2(CCC2NC(C2CC=CCC2)=O)C1 C1(C(=O)N(C(C2CCCCCC2)CO)CCO)CCCCN1C(C1CCCCC1)=O c1(NC(COC(C(=O)OC(C)C(=O)C2CCOC2)C)=O)c(F)cc(F)cc1Cl C(=O)(C1OCCn2ccnc21)N1CCC(C)(NC(Cc2ccc(C)s2)=O)CC1 C12(C(=O)NCC(C3CC3)NC(c3c(N(C)C)cccc3)=O)CCC(CC1)OC2 C(C(=O)N(C)OCC1CC1)(c1ccnn1C)NC(C(C=CC)O)=O N1(C(c2c(C)ccnn2)=O)CCCC(C2CCN(C(=O)C3=CC(C)(C)C3)C2)C1 C1(CNC(C=CCCC)=O)CCCC2(CN(C(=O)CC3CCCCN3C)C2)O1 c1(CNC(CCOC2CN(C(C(C=C)O)=O)C2)=O)ccc(CC)cc1 C1(NC(C(C2CCCO2)OC)=O)CCN(C(=O)COCc2cccc(C)c2)CC1 c1(OC)cnc(C(=O)NC(CNC(c2ccc(Cl)c(C)c2)=O)C(C)C)c(OC)n1 c1(C(=O)NCC(CCNC(=O)C(C2(O)CCCC2)F)OC)cc(S(N)(=O)=O)cs1 c1(CN2CCC(NC(Cc3nnc(C)o3)=O)C(F)C2)cccc2c1OCCO2 O=C(CCCN1CCCC1)NCC1CC1CNC(c1sccc1C1CC1)=O C1(NC(C(C(C)C)O)=O)CCN(C(=O)CC2CC=CCN2C)C1(C)C C1(CNC(C(COCC)NC(=O)C(C2CCOCC2)=O)=O)CCC(F)(F)C1 N1(CCC(=O)NC2(C(F)(F)F)CCS(=O)(=O)CC2)C(=O)C2CC=CCC2C1=O c1(C(N(c2ccc(OC3CC3)cc2)CC(=O)O)=O)cccc(C(F)(F)F)c1 c1(CNC2CCC(C(=O)Nc3n(CC)nnn3)OC2)ccc(I)c(O)c1 C1(NC(C(CCC2CCC2)NC(c2cnns2)=O)=O)CCCC2(CCC2)C1 n1(CC(N2C(CN(C)C)C(c3ccccc3)C2)=O)cc(S(N)(=O)=O)cn1 C1(C)(CCNC(CSCCN(C)C)=O)CCN(C(c2nocc2Cl)=O)CC1 c1(C(N2CCC(CC=C)(NC(c3cc(Cl)ns3)=O)C2)=O)cc2n(n1)CCC2 C1(C(N2C(C(C)O)CC2)=O)CC(=O)CN1C(=O)C1=C(Cl)CC1 C1(NC(CCCOCC=C)=O)CCN(C(=O)Cn2nc(C)nc2C)CCC1(F)F c1(C(N2CCOCC2)CNCc2ccc(C(=O)OCC)o2)ccccc1 N1(C(COC2(C)CCOCC2)=O)CC(F)(F)CC1(C)CNC(C1CCNC1=O)=O c1(CC(=O)OC)ccc(OC)c(S(=O)(=O)N2CC3C(CC(=O)OC)C3C2)c1 Cc1nc2cc(C(N3CC=CC(NC(C4CC(=O)N4)=O)C3)=O)cnc2[nH]1 N1(CC)CCC2(CCCN(CC3CCC(COC)CO3)C2)C1 CCC(CNC(=O)C(c1ccc(-c2ccccc2)nc1)(C)C)C(=O)O c1(C(N2C(CCNC(Cn3c(C)cnc3)=O)CCC2)=O)ccc2ccccc2n1 N1(C(C=CCCC=C(C)C)=O)CCCC(O)(CNC(=O)C(N2CCCCC2)C)C1 Cc1cc(F)c(C(N2CCOCC2CNC(=O)CCc2scnc2C)=O)cc1F Cc1nc(C=CC(N2CCCCC(N(C(=O)C(C)c3cccs3)C)C2)=O)[nH]c1C CC1C(C)N(C(=O)C=Cc2nccs2)CCN1C(c1ccc(Cl)cc1)=O N1(C(CC(C(F)F)NC(CCC2(C#N)CCC2)=O)=O)CCC2(CC1)CC2C#N c1(C(=O)NC2CN(C(c3c(C)ncs3)=O)C2)cc2c(nc1O)CCCC2O CC1(C)CC(NC(c2ccc(N3CCCC3)cc2)=O)CN1C(C1C=CCC1)=O C1(CNC(CNC(C(c2cccnc2)C)=O)=O)CCCN(C)C1=O C(=O)(C(CO)C(C)(C)C)NC(C(=O)N(CC(CCC=C)O)C)CCC N1(C(C2CC(OCC)C2)=O)CC2(C1)CN(C(c1ccc(N)cc1C)=O)C2 N1(C(C2N(C)C(=O)OC2)=O)CCC2(CC(NC(=O)Cc3csnn3)C2)C1 CCC(C(=O)N1CC2(C1)CN(C(c1cnccc1C)=O)C2)C(C)C C1(C(=O)Nc2c(CC)nc(Br)s2)Cc2ccccc2O1 c1(C(=O)NC(CNC(c2c(CC)c[nH]n2)=O)C(C)(C)C)ccc2ncnn2c1 C1(CNC(C(CC)NC(N)=O)=O)CCN(C(c2cc(C)ccc2N)=O)C(C)C1 C1(C(N2CCC3CCN(C(C4CCOC4)=O)C3C2)=O)CCC2(CC1)CC2(F)F Cc1cc(C(N2CC(NC(=O)CN3CCOCC3)CC(F)C2)=O)nc(C(F)F)n1 C1(CNC(C2(SC)CCC2)=O)CN(C(=O)C=CCF)CC12CC2 CCC(CCC(=O)NCC1C(C(N2CCC(C(C)C)C2)=O)C1(C)C)OC CCN=C(NCC(F)=C)NCC1CCC2CC12.C1(=C(F)CF)CCOCC1 c1(C(=O)NC2CCCCN(C(C3CN(C)C(=O)C3)=O)C2)nccn2nccc12 N1(C(C)=O)CCCCC1C(=O)NCC(C(C)(C)C)NC(=O)Cn1c(C)csc1=O N1(C(C=CC(C)OC)=O)CCCCC1C(=O)NC1(C)CC(C(=O)N(C)C)C1 N1(C(C(C=C)O)=O)CC(C(=O)N(CC(=O)NC(C)C)C)C(CC)C1 c1(OC)cncc(C=CC(N2CCC(Oc3ccc(F)cc3F)C2)=O)c1 C12(CNC(CSCC)=O)CCCCC1N(C(c1cnc(C(C)(C)C)s1)=O)CC2 C(=O)(C1=C(Cl)CCCC1)N1C(C(C)NC(c2ncc(C)cc2C)=O)CCC1 C(C(=O)NC1CCC2(CC2)C1)(C(C)(C)C)NC(C(C=C)CC)=O N1(S(CC)(=O)=O)CCCC1C(=O)NC(C)CCNC(=O)CCc1ncc[nH]1 N(C(=NCCc1ccc(Cl)cc1Cl)NCC(=O)NC1CC1)CC1N(CC)CCC1 C(=O)(CC(CC)SC)NCc1cn(CC(=O)NCC)nn1 O=C1CC(CNC(C2(O)CCCC2)CCO)C12CCC2 C(=O)(C(CC)C(=O)N1CC2(NC(=O)CCc3cc(C)[nH]n3)CCC1C2)OCC N1(C(=O)OCC(C)C)CCC2(CC1)CC2CNC(C1CC=CCC1)=O c1(CC(=O)N(CC(C)NC(CCCNC(=O)OC)=O)C)ccc(OC)c(F)c1 N1(C(c2scc(OCC)c2)=O)CCCN(C(c2oc(OC)nc2C)=O)CC1 C=CCC(C(=O)NCCC(=O)NC(N)=O)NC(=O)CN1CCCCCC1 N1(C(c2ccc(NCCCC)cc2)=O)CCN(Cc2ccc(C)cc2Cl)CC1C C1(NC(C(CC=CC)NC(=O)CCOC)=O)C2CCCC1CC2 c1(C(=O)NC2CN(C(C3CCN(C(CC)=O)C3)=O)C2)ccc(C(C)(C)C)cc1N N(C1CCc2cc(Cl)ccc21)C(C)=O.n1(CCSC)nnnc1C1C2(CCC2)N1 c1(C(=O)NCC(CC)NC(c2c[nH]cc(F)c2=O)=O)ccc(Br)c(C)c1F C1(NC(c2ccc(COC)cc2)=O)CCCCCN(C(c2ccc(F)s2)=O)C1 c1(C(=O)NCC(CCCC)NC(=O)C(C)(C)C2CC2)ccnc2[nH]cnc12 CC(C)(C)C(S(=O)(=O)N1CCC(CC2(O)CCC2)CC1)c1ccccc1 N1(C(c2c(C)cns2)=O)CCCC(C)(NC(=O)C=CC(N2CCOCC2)=O)C1 C1(C(=O)NCC2C(C(=O)NC(CSC)(C)CO)CCCC2)CCCC(C#N)C1 N(C)(S(=O)(=O)N(C)C)CC(=O)NCC1(C)N(C(C=CCCC(C)C)=O)CCC1 Cc1c(C(N2CCSCC2CCNC(C2(C)CC2)=O)=O)nnn1-c1ccn(C)n1 c1(C(N2C(CNC(C(C(=O)OC)C)=O)COCC2)=O)cn2nc(C)sc2n1 CCCC(CNC(C1CCC(O)CC1)=O)C(=O)N(CC=Cc1ccccc1)CC CC(C)CS(=O)(=O)CC(=O)NC1CCCCCN(C(=O)Cc2ccoc2)C1 CNS(=O)(=O)N1CCC(C(N2CC3CC2C3NC(=O)C(C)c2cccs2)=O)CC1 C1(NC(CC2(C(=O)OC)CC2)=O)CC(C2CCN(C(C3CN(S(N)(=O)=O)C3)=O)C2)C1 N1(C(=O)Cc2cnccn2)CC2CCCC(C1)N2C(=O)Cc1cccnc1O C1(C(=O)NC(CC)C)CCCCN(C(=O)CCCC(C)C)C1 N1(C(C(F)OC)=O)CCC(c2ccccc2)(NC(=O)CCN(C)CCO)C1 c12ncccc1NC2=O.c1(C(=O)OC)csc(CO)c1.C12CC(C1)NC2=O C1(C(N2CCCCC(NC(C=COCC)=O)C2)=O)Cc2cc(C)ccc2S1(=O)=O C1(C(N(CCCC)CCOC)=O)CC2CC2N1C(c1cccc(=O)o1)=O N1(C(C(CC(CC)C)C)=O)C2CCCC1CN(C(=O)CN1CCS(=O)(=O)CC1)C2 N1(C(=O)CSC(F)(F)F)CC(C2CN(C(c3cccc(F)c3Br)=O)C2)C1 C(=O)(CC(C)CF)N(C(CNC(CCNC(=O)OCC)=O)C1CC1)CCO C1(C(=O)NCc2cc(C(C)C)on2)CCCCN(C(C2(C(F)(F)F)CC2)=O)C1 C12(NC(c3nc(OCC)oc3)=O)CCCCC1N(C(=O)CCC1CCC1)CC2 C1(CC(=O)NCC(CNC(c2c(C(F)(F)F)cn(C)n2)=O)O)CCCS(=O)(=O)C1 c1(C(=O)NCC2CCC(NC(C3(OC)CS(=O)(=O)C3)=O)C2)cc2c(s1)CCCC2 N1(CCNC(C(C)Sc2ccccn2)=O)CCCN(C(=O)Cc2cncs2)CC1 CC12C3C4C1C1C2C3C41C(N1CCC(NC(C2CCCN2C2CCCC2)=O)C1)=O N1(C(CN(C2CC2)CC)=O)CCCC(C2CCCN2C(=O)Cn2[nH]cnc2=N)C1 c1(C(CO)N(CCC(N)=O)CC)cccc(S(C)(=O)=O)c1 Cc1cc(C(=O)NCc2nc(C(=O)N(CC(C)C)C)c(C)o2)cc(O)c1 N1(C(C(CC)n2cccn2)=O)CC2(CC(CNC(C3CCC(C)(C)OC3)=O)C2)C1 c1(C(N(C2CN(c3ccn4nccc4n3)C2)C)=O)cc(Cl)c(Cl)c(Cl)c1 C1(C(=O)NC(C)CO)CC(C)(C)CN1C(=O)CCc1cnn(C)c1 c1(SCC)ccccc1C(N1CC(C(C)NC(=O)CSCC2CCCO2)C1)=O C(=O)(C1=CS(=O)(=O)CCC1)NCC1(NC(C(C)OC)=O)CCCCCC1 C1(C(=O)NC2CC(CCNC(CCCOC)=O)C2)CCC(C)(C)C1 C12(C(=O)NCCCN(C(c3c(C)nco3)=O)C)CCCC1C2(F)F C=CCC(CC)C(=O)N1CC(C=C)(CC(=O)NC2CN(C)CC2(C)C)C1 c1(C(N2C(CC)CN(C(C3CC3C(F)F)=O)CC2)=O)ccc2c(c1)CCN2C CCCC(CNC(=O)CCNC(N)=O)C(=O)N1CCCCC1 C1(NC(C2CC(CC)N(C(=O)C=CC(=O)N(C)C)CC2)=O)CCc2ncnn2C1 N#CC1CN(C(=O)CCC2CCCN2C(=O)CCCCN=[N+]=[N-])CCO1 c1(C(=O)NCCCNC(C2(CO)CC2)=O)ccc(-n2ccnc2)cn1 N1(C(C(C)N(C)C)=O)CCC2(CCC2)C(NC(=O)Cc2cc(Cl)n(C)n2)C1 C1(C)(C(=O)NCC2CCC(NC(c3c(C)ncnc3)=O)CC2)CC2CCC1C2 N1(C(C(=O)NCCOC)=O)CC(NC(=O)C=Cc2ccc(C3CC3C)o2)CC(O)C1 c1(C(N2CC(CNC(CCOCCC)=O)OCCC2)=O)cc2c(C)cccc2o1 O=C(C1=C2CCN=C2NC=C1)NCC1CCCSCC1 C1(C(N2CCC3CC3C2)C(=O)NC2CCOC2)CCC2COCCC2C1 CC1CCC(NC(=O)C=Cc2cn[nH]c2)CN1C(C1CCCCC12CC2)=O c1(NCc2ncc(OC)o2)ccc(OC(=O)NCC(C)N=[N+]=[N-])cc1 Cc1ccc(-n2cccc2)c(C(=O)N(C)Cc2cn(Cc3ccccn3)nn2)c1 c1(C(=O)NCCN(C(c2cn(C)c(=O)n2C)=O)CC)c(C)nc2ccnn2c1C N1(C(C2=CCC(C)CC2)=O)CC2CC(C)N(C(=O)CC3CC(=O)NC(=O)C3)C2C1 c1(C(=O)NCC2CCN(C(=O)CN3CSCC3=O)C2)cccc(-n2cnnn2)c1 C1(CC(=O)NC2(CCNC(C(C)(O)C3CCC3)=O)CC2)CCCS1(=O)=O C1(CC(=O)NC2CCC(NC(c3c(NC)cncc3)=O)C2)CCC(C)(C)CO1 c1(C(=O)NCCC(C)(C)NC(Cc2cnc(C)o2)=O)sc(=N)[nH]c1C Cc1cc(N)c(C(=O)NCC(F)CNC(=O)Cc2cc(C(C)C)no2)c(F)c1 c1(C(=O)NC2CCC(N(C(=O)C=CCO)C)C2)ncc(F)cc1F N1(CCN(C(CCC(=O)N(C)C)=O)C)CC(NC(c2ccccc2)=O)CCC1=O N1(C(CN(C2CC2)CC)=O)CCC2(NC(c3cccc[n+]3[O-])=O)CCCCC12 N1(C(C2(CCOC)CCC2)=O)CC2CCC1C(NC(=O)C(F)(F)C(F)(F)F)C2 C1(C(C(=O)CCN(C(C(C)CN(C)C)=O)CC(C)C2CC2)O)COC(C)(C)O1 C1(NC(N2CCC2c2cccc(F)c2)=O)(CO)CC(O)C12CCC2 C1(C(=O)NC2CCC(NC(Cn3ccc(C)n3)=O)C2)CC(F)C(=O)N1 N1(C(C=C(C)C2CC2)=O)CCCC(C)(C(N2CCNC(=O)C2CCO)=O)C1 Cc1ccc(Br)c(CC(=O)NCC2COCCN2C(=O)C=CS(C)=O)c1 C(CC(C(=O)NOC1CCC(O)C1O)NC(=O)C(C)CC(N)=O)SC C1(NC(CC2(CSC)CC2)=O)CC(CC(=O)NCCN2CCCCC2=O)C1(C)C Cc1csc(C(=O)NC2CC2NC(C2CCCCCC2)=O)c1Br c1(CCC)cc(C(=O)N(CC(C)(C)NC(C2CCN2CC)=O)C)ccn1 N1(C(C2CCCC2C)C(=O)Nc2ccc(OCC)cc2)CCN(C)CC1C#N CC(C)C(CCN(C)C(C1(C)CC(F)C1)=O)NC(=O)CCOCC1CC1 c1(C(N2CCC(NC(=O)CC3CCCC3)C2)=O)c(F)cccc1Br c1(SC)cc(C(=O)NC(C)CC2CN(C(C3(F)CCOC3)=O)C2)ccc1[N+](=O)[O-] C1(C(N(CCCNC(C2(n3nccn3)CC2)=O)C)=O)CCC(NC(N)=O)CC1 CCC(C)(C)C(O)C(=O)N1CC2(C1)CN(C(C1CCS(=O)(=O)C1(C)C)=O)C2 C1(NC(C(COC)(C)O)=O)CCN(C(c2ccc(C3CC3)c(Cl)c2)=O)CC1(C)C N1(C(C(CC)COC)=O)CCCC12CCN(C(c1ccc3c(c1)CCC3)=O)CC2 C1(C(=O)NC2CCC2CNC(C23CC4CC2C3C4)=O)CC2(CCC2)CO1 CC(C)(O)C(F)C(=O)N1CCC(CO)(NC(c2ccnc(C(F)(F)F)c2)=O)C1 S(=O)(=O)(CC(=O)NC1(C(=O)N(C)CC2CC(F)C2)CCCC1)NC C(=O)(C(C(C)C)C(C)C)NCCOCC(=O)NC(c1nc[nH]n1)CC c1(CC)cc(Cl)ccc1C(=O)NC1CC2CCC1N2C(c1ccccc1C)=O c1(OC)cccc(-n2cc(CNC(N3CC(N4CCOCC4)C(C)C3)=O)nn2)c1 c1(-c2cn(CC3CN(C(C(C)=CC(c4ccccn4)=O)=O)C3)nn2)c(Br)c(C)nn1C C1(NC(c2c(C)ccc(C)n2)=O)CC2CCC(C1C)N2C(=O)CCc1cnoc1 N1(C(c2c[nH]c(=NC)s2)=O)CCC(NC(=O)C(C)S(N)(=O)=O)C(F)C1 C1(C(=O)NC(C(=O)OCCCC)C)CN(Cc2cnc(Cl)cc2OC)CCC1O C(c1ccc(C(N)=O)cc1)=CC(N1CC=CC(NC(c2cnn(C)n2)=O)C1)=O N1(C(C(CC#C)NC(c2cnn(CCC)c2)=O)=O)CC(CO)C(C)(C)C1 N1(C(C2CN(CCOC)C(=O)C2)=O)CCC2(CCCN2C(C2C3CCCC23)=O)C1 C(CC1CCOCC1)(C(=O)N(CC(C)SC)C)NC(CCC1CC(OC)C1)=O C(C(CNC(=O)COC(C)(C)C)S(C)(=O)=O)NC(c1nc(C(C)C)sc1)=O C(=O)(CC(C)(C)C(F)(F)F)NC1C(C)CCN(C(c2c(Cl)cn(CCC)n2)=O)C1 c1(CN2CCC(CNC(=O)NCCC(C)OC)CC2)ccc(Cl)c(F)c1 N1(C(c2ccc(C(C)C)o2)=O)CCC(NC(=O)CC=CC(C)(C)C)C(C(C)C)C1 CC(CCCNC(c1ccc(Br)o1)=O)NC(C1CC1c1ccccc1)=O c1(C(=O)NC(C)CCCCNC(=O)C=C(Cl)Cl)ccc2cc[nH]c2c1F N1(C(c2cccc(N(C)C)c2)=O)CCC(C2CCN(C(=O)CC34CC(C3)C4)C2)C1 N1(C(C2C(C)OCC2)=O)CCN(C(c2cnoc2)=O)CC12CCC2 C1(NC(c2nn(C)c(C(F)(F)F)c2)=O)C2CC3CN(C(C4CCCS4)=O)C1C3C2 c1(SCC(N2CCN(C(c3ncccn3)=O)C3C2C3)=O)c[nH]c2cc(F)ccc12 N1(C(C2CC=C(C)CC2)=O)CCC2(CCN(C(=O)CCCC(C)(C)C)C2)C1 c1(C(N(CC(CC)NC(=O)C(C)n2cnnn2)C)=O)cn(CC)nc1C C(=O)(CCCC(C)=O)N1C(CN(C(C(CC2CC2)OC)=O)C2CC2)CCC1 c1(NC(CCOCCOCCOCCN=[N+]=[N-])=O)ccc2cccnc2c1N c1(C(=O)NCC(=O)NCCNC(c2c(C(C)=O)ccs2)=O)ccccc1Cl c1(C(=O)NC2C(C(=O)NCc3ccc(C)c(C)c3)C2)ccc2c(Cl)ccnc2c1 c1(NCCC2(C(=O)OC)CCCCC2)ccc2c(n1)CCCC2 c1(NC(C2C(NC(C3C(C(=O)OC)C3)=O)CCCC2)=O)ccc(N(C)C)c(F)c1 C1(C(NOCCCOCC)=O)CC(NC(=O)CCC2(C#N)CCC2)C(O)C1 c1(C(=O)NC2CCN(C3CC3)CC2)coc2ccc(Cl)cc12 S(=O)(=O)(CC(=O)N1CC(NC(=O)C(CN(C)C)N(C)C)C(C)C1)NC C#CC1(O)CC(C(N2CCC(CNC(=O)CSCCOC)C2)=O)C1 C1(OC)CCCC1C(N1CCC1C(=O)NC(C)C(C)n1cccn1)=O c1(OC)ccc(C(=O)NCC2(O)CCCC2C)c2ccccc12 N1(C(C(N2CCCCC2)C)=O)CCC(CNC(C2(C)CC(F)(F)C2)=O)C12CCC2 c1(SC)cccc(NC2CCC3CC2CN3C(=O)CCC[N+](=O)[O-])c1[N+](=O)[O-] C(CCCC(=O)N1CC(C)(NC(=O)C(C)OCC(C)C)C1)OCC c1(C(C)NC(c2cnc(Cl)s2)c2nnnn2Cc2ccccc2)cn2ccnc2s1 C1(N(C(=O)CCC2CC2)C)CCCCC1NC(C1(c2ccccc2)CC1)=O CCCC(CCC)CC(=O)NC12CCC(C1)N(C(c1ccn(C)c(=O)c1)=O)C2 C1(C(=O)NCC2CCCC2)CC2CCCCC2N1C(C1CC(O)C1)=O C(C1=CCCN(C(=O)C(C(C)C)C2CCC2)C1)NC(C1N(CC)CCC1)=O CC1OCC2(CCN(C(C3(Br)CC3)=O)CC2)C1NC(=O)CC1(O)CCC1 N1(C(c2cn(CC=C)nn2)=O)CCC2(CCN(C(c3ccnc(CO)c3)=O)C2)C1 C1(C(=O)NC(C#C)C(C)OC)CCOCC1NC(C1(CC#C)CCCO1)=O C1(C)(CNC(COC2(C)CN(C(C3C(C(=O)OC)CC3)=O)C2)=O)CSC(C)=N1 C(=O)(CC(C)(C)CN(C(=O)CC1CCCSC1)C1CC1)N1CC(SC)C1 C#CCCCCC(=O)N1CCCN(CCCCNC(=O)Cc2cnsc2)CC1 C12(C(=O)NC(C#C)(CC)CC)CCCC1CN(C(=O)C(C)SC(C)C)C2 N1(C(C)OC2(C(=O)OC)CCOC2)CCN(C(=O)C(=O)NC(C)C)CC1 Cc1nc(C(N2CCOCC(F)(CNC(=O)C=C3CCC3)C2)=O)c2ccccn12 Cc1cc(C(=O)N(C2CCN(C(c3cn[nH]c3)=O)CC2)C)nc(O)n1 N1(C(c2cc(COC)no2)=O)CCC2CCC12C(=O)NC(C)(C)C N1(C(C2CCC(=O)C2)=O)CCCCC1C1CCCN(C(=O)CCc2ncc[nH]2)C1 c1(C(N2CCC(O)(C(CNC(C(C#C)(C)C)=O)C)C2)=O)cc(C(N)=O)ccc1F N1(C(C(=O)NCC(=O)NC2CC2)=O)CCN(C(=O)CO)CC1CCO N1(C(CN(C)CCO)=O)C(CNC(=O)C=Cc2cscn2)CC2COCC12 Cc1c(NC(C(C)(C)C)=O)nc(Br)n1C.C12CC(=O)N(C1)Cc1nc2no1 CCC(C(=O)NC1COCCN(C(c2conc2C2CCC2)=O)C1)C(C)(F)F Cc1cc(=NC(C)c2ccncc2C)[nH]c(N2CC3CC2CS3=O)n1 C(C(CCOC)NC(=O)CCSC(=O)NC1CCCCC1)NC(COC)=O.C(C)(=O)C N1(C(c2cccc(C#C)c2)=O)CCCN(C(c2cc[nH]c2C)=O)CC1C C1(C(=O)NC2(C)CN(C(=O)CCCN3C(=O)CNC3=O)C2)CC2CC1CC2(F)F C(=O)(C1=CCCC1C)N1CC(F)(CNC(C2(COC)CC=CCC2)=O)C1 C1(C)(NC(CCC2CCN(C(CCc3cc(C)[nH]n3)=O)C2)=O)CCN(C)C1 C(=O)(C1Cc2ccccc21)NCC(CC(C)C)C(=O)N1CCCCCCC1C Cc1cc(F)cnc1C(=O)NC(C)CNC(=O)CCC1(C)CCC(=O)N1 C1(O)(C(C)C(=O)NC(C)(CNC(=O)C(C)(C)n2cnnn2)CO)CCOCC1 C(CCCCCCCO)=CC(=O)NCCCN(c1nnc(-c2ccccc2)s1)C N1(C(C(=O)NCCOC)=O)CC2CC(NC(C3(COC)CCCC3)=O)C1C2 C1(CNC(C(CC)Sc2nc(=N)[nH][nH]2)=O)CN(C(=O)CCCC(C)C)CCC1O N1(C(COc2c(C)occc2=O)=O)CCN(C(=O)COC2CCCC2)CC(O)C1 c1(C(N(CCCCNC(c2n(CC)ncc2)=O)C)=O)cccc2c1COC2 N1(C(c2n[nH]c(C)c2O)=O)CCCC(F)(C(=O)NCC(C)(O)CN(C)C)C1 C1(NC(c2n(CC)ccc2)=O)CCC(C)N(C(=O)CCCC#N)C1 Cc1nc2ccc(CN3CCC(C(=O)N(C)C(c4nccs4)C)CC3)cc2o1 c1(C(=O)NCC(C)(Cn2cccn2)NC(CCC=CC)=O)[nH]cc2c1CCC2 C(C(=O)NNc1ccc(Br)c(Cl)c1)(C1CCCCCC1)NCSCC N#Cc1ccc(F)c(CN2CC(O)(CNC(c3nc(Cl)sc3Cl)=O)C2)c1 C1(C(=O)NC(C(C23CCC(CC2)C3)NC(CC)CC(=O)OC)=O)CCCCC1(F)F c1(C(=O)NCC2(NC(C(F)=CC)=O)CC2)ccc(OC)c(C(C)C)c1 c1(CC(N2CCC(N(C(c3c(C)ocn3)=O)C)C(C)C2)=O)cn2ccccc2n1 C(=O)(C(CCN(C)C)NC(c1c[nH]nc1C)=O)N1CC(O)(COC)C1 C1(C)(C(=O)NC2C(NC(C(COC)COC)=O)C2)CCCCCC1 CS(=O)(=O)CC(=O)N(CCNC(=O)CN1CCCC1)CCc1cccc(Cl)c1 C=CC(CC)CC(=O)NC1CCCC1C(N1CCOC(CCF)C1)=O c1(OCC)nn(C)cc1NC(C1(O)CCN(Cc2ccccc2OC)C1)=O c1(NC(C2N(Cc3c(C)c(Br)ccc3)CC(O)C2)=O)cc(Br)ccc1[N+](=O)[O-] Cc1nn[nH]c1C(=O)NC1CCCC1NC(=O)Cc1nocc1C(C)C N(C1CN(C(=O)CO)Cc2ccccc21)C(c1cn(C)nc1-c1ccccc1)=O C1(OC)CN(C(C2OCCC2C(C)C)=O)CC1NC(c1cnccn1)=O c1(CN(C)Cc2ccccc2F)ccc(CN2CCCC2=O)cc1 C(C1c2ccsc2CCN1C(c1ccc2cccnn12)=O)NC(CCC(N)=O)=O N1(C(C(C)NC(C)=O)=O)CCC=C(CNC(C2CCC(=O)N(C)C2)=O)C1 C1(C(=O)NCC(=O)NC(CCNC(C(C)c2cncs2)=O)(C)C)CCS(=O)(=O)C1 N1(C(C(C)OC)=O)CCC=C(C(=O)NC2CC(N(C)C)C2(C)C)C1 c1(CC)cc(N)c(C(=O)NCCNC(=O)C(F)(F)Sc2cnn(C)c2)c(F)c1 C(=O)(CCC(=O)NC)NCC1(C(C)(C)O)CN(C(C2C(OCC)C2C)=O)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C)C=CC(N1CCC(F)(F)CC1)=O c1(C(=O)NC2CN(C(C(C)(C)O)=O)CC2N=[N+]=[N-])cccc2c1OCCCO2 C1(C(N2CCC(NC(=O)CCCNC(=O)C3CC3)C(O)C2)=O)Cc2cccnc2C1 C(=O)(C(C#N)C(C)(C)C)NC1C(NC(c2cc(CC)on2)=O)COC1 C(C(C)(C)C(=O)N1CCCC(OCC)C1)N(C(C1C(CCC)C1)=O)C C1(CC(=O)N(C)CCNC(c2ccn(-c3cccnc3)n2)=O)CCC1C1CC1 C1(NC)CCOCC1.C1(SCC)CN(C=O)C1.C1(=O)NCCN1 c1(C(=O)NCC2(OC)CN(C(c3cc(=O)n(C)o3)=O)C2)cc(C(F)F)ccc1F c1(C(=O)NC2C(NC(C(C)(C)SCC)=O)C2)cc(OC)c2ccccc2n1 Cc1sc(-n2cnnn2)c(C(N2CCC(C)(CNC(=O)C=CCF)C2)=O)c1C CC(C)C(C)CC(=O)N1CCC(NC(c2cccnc2Sc2ccccc2)=O)C1 c1(C(N2C(C)CCC(CNC(c3ncc(F)cn3)=O)C2)=O)cccc2c1CCN2 C1(COC)CN(C(=O)C(O)CN2CCCC2)CCN1C(=O)C(F)CC(C)C CC(C)C(C(=O)NCCN(C)C(C1CCCN1Cc1ccsc1)=O)n1cncn1 N1(C(C2(CC=C)CC2)=O)CCCCC(C(=O)NCC(C)(C)C(=O)OCC)C1 C1(C)(CNC(COCCOC)=O)CC(F)(F)CN1C(c1cc2ncccc2o1)=O N1(C(C(C)(C)C)=O)CCCC(C2CCCN(Cc3cc4cc(F)ccc4[nH]3)C2)C1 c1(C(=O)NC(C(C)NC(=O)CSC(F)F)C)onc2ccccc12 c1(C(=O)NC(C)CNC(=O)CC2C(C)(C)C2(C)C)c[nH]nc1[N+](=O)[O-] c1(CNCC(=O)N(CC(C)(C)C)C)cnc(-c2ccccc2)o1 c1(CC2(NC(CCC=C)=O)CCCC2)c(F)cc(C#N)cc1Br C(CC(N)=O)(C(=O)NCC12CCC(CC1)CC2)NC(C(n1ccc(C)n1)C)=O Cc1ccccc1C1CC1C(=O)NC1(CCNC(c2cnncc2O)=O)CCC1 c1(-c2n(C(CC)C)nc(-c3ccc(Cl)cn3)n2)ccc2c(C)nn(C)c2n1 CC(C)C(C(C)C)C(N)C(=O)NCC(N1CCOCC1C)(C)C C1(C(=O)N(CC(C)NC(=O)CC2(C)OCCO2)C)(OC)CCCSC1 c1(C(=O)NC(CCCNC(c2cn(C)nn2)=O)(C)C)ccc(C#CC2CC2)cc1 C1(CNC(c2c(C)snn2)=O)CN(C(c2cc(Cl)ncc2N)=O)C2COCC2O1 N1(C(c2cc(COC)oc2C)=O)CC2CC(NC(=O)Cc3cccnc3)C(C2)C1 C(=O)(C(C)(O)C(C)(C)C)N(CCC(C)NC(c1c(C)c(Cl)cnc1)=O)C c1(C(N(C2CCN(C(=O)Cc3cnccc3Cl)CC2)CC)=O)c(C)cccc1O C(=O)(CC1=CCOCC1)NC1CN(C(c2c(C)nn(C(C)C)c2C)=O)CC1(C)C N#Cc1ccc(OCC2CN(C(CC(=O)CN3CC4CC4C3)=O)C3C2C3)cc1 c1(C(=O)NC(C)CCO)coc(CNC(C2(O)CCSC2)=O)c1 C1(NC(C(CSC)O)=O)CC2COCC(C1)N2C(C1C2(CC2)C12CC2)=O c1(OC)cc(C(=O)NCCCN(C(=O)CC2CCC(C)O2)CCO)ccc1C c1(C)ocnc1CONC(=O)c1cn[nH]c1.C1(C)C=CCOC1 C1(C(=O)NCCOC2(CNC(C=CC)=O)CCOCC2)CCc2nnnn2CC1 c1(NC(C(c2cccs2)NC(C(C)=CC(C)(C)C)=O)=O)ccc(Cl)nc1 CN1CCC(CCC(=O)NC2(CNC(=O)C=Cc3cn[nH]c3)CCCC2)CC1 C1(CNC(C2(CC)CC2(F)F)=O)CC(NC(=O)CCc2cn(C)cn2)C(O)C1 N1(C(C(C)OC2CCCC2)=O)CC2CC1CCN2C(=O)C(=O)N(C)C C1(CNC(c2scc(C(C)=O)c2)=O)CN(C(=O)C(=O)Nc2ncc[nH]2)CC1(C)C c1(C(N2CC(NC(c3ncc(C)nc3)=O)C(F)C2)=O)c(Cl)ccc(Cl)c1F N1(C(C(C)=CC2CC2)=O)CCC(C(=O)NOC2CCOC2)CC1 C1(C(N2C(C)CC(CNC(CCc3onc(C)n3)=O)C2)=O)CC2(CC2)CN1C C1(C(=O)NC(C)CNC(=O)COc2ccc(Cl)nc2)CC(C2CC2)=NO1 N1(C(c2cc(CC(C)C)[nH]n2)=O)CC2CC(C1)N2C(=O)Cn1ccnn1 C1(NC(c2n[nH]c(CC)c2C)=O)CC2CC1N(C(c1cnn(C)c1C1CC1)=O)C2 C1(C(=O)NCCC2CCCN(C(C3(CC)CCCCO3)=O)C2)CCCC(=O)CC1 c1(C(=O)NC2C(OC)CN(C(C34CC(COC)(OC3)C4)=O)C2)cc(F)ccc1O c1(C(N2C3C(NC(CCC=C)=O)CC(C3)C2)=O)cnc2ccnn2c1 C(C1CCCCC1)=CC(=O)NCC12CC1CN(C(C1(CO)CC(F)(F)C1)=O)C2 N1(C(c2c(CC)noc2C)=O)CCC2(CCC(NC(c3cc(Cl)n(C)n3)=O)C2)C1 N1(C(c2nc(C)n(C)c2)=O)CC2CCC(C(=O)NCC3CCCC(C)(C)C3)(C2)C1 Cc1cc(C(=O)N(CCC(C)N2CCCC2)C)c2cccc(O)c2n1 C(=O)(C(C)(C)CNC(c1cc(C)on1)=O)NCC(C(C)C)OC C(=O)(C#CC1CCOCC1)N1CCC(F)(C(N2CCOCC(C)C2)=O)C1 C(C)(C(C(=O)NCC1(C)CC1)C(C)C)NC(c1c(OC)n(C)nc1)=O C1(N(C(C2CN(C)C2)=O)CC2CC2)CCN(C(=O)C=Cc2ccc[nH]2)CC1 C1(=O)C(C(C)C)N(C)C2(F)CN1C2.C(=O)(C(CC1CCC1)OC(C)=O)NC C1(NC(C(C)(C)n2cnnn2)=O)CCOCC1NC(c1cnn(C(C)(C)C)c1Cl)=O c1(C(N(C2CN(C(c3c(C)oc(Br)c3)=O)C2)C)=O)ccc2[nH]ccc2c1F C(CC(C)C)(C(=O)Oc1ccc(CN2CCCCC2C(=O)NCCF)cc1)OC C1(CCNC(COCCOCCOC)=O)(C(=O)NCC2C=CCCC2)CCOC1 S1(=O)(=O)c2ccc(c(F)c2)NC2CC(C2)CN1.C1(OC)CCOC1C(C)C N1(C(C=CCCC(C)C)=O)CC2(C1)CN(C(c1ocnc1C1CC1)=O)CC2CO c1(CNC(=O)NCC=C(C)C)c(NC2(O)CCCNC2)sc2c1CCC(C)C2 Cc1noc(C)c1-n1nc(C(C)C)nc1CC(O)Cc1ccccc1Br C1(C(N2CCCC(CNC(C3(C)CS(=O)(=O)C3)=O)C2)=O)CCc2nccn2CC1 Nc1ccc(C(=O)NC2(CNC(C3CCCOCC3)=O)CCC2)c2cnccc12 C1(C(=O)NC(CNC(c2ccc(SC(C)C)cc2)=O)CO)SC2C=CC1CC2 C1(C(=O)NC(C)CCCCNC(c2cnn(C)c2C(F)F)=O)COC2(CCC2)C1 C#CC1C(C(=O)NC2CN(C(=O)Cc3c[nH]nc3O)CC2C(F)F)C1(C)C c1(C(=O)NC2(C)CC(NC(CC3C(C)(C)C(O)C3)=O)C2)c[nH]c2cccc(F)c12 C1(CC)(CNC(=O)CC(C)F)CCN(C(c2cn(C)nc2-c2cccs2)=O)CC1 c1(C(N2CC(CN(C(CC(CC)C)=O)C)C2)=O)cnc(Cl)cc1Cl C=C(CNC(=O)C(c1cncn1C)N(C)C)CCNC(c1c[nH]cc1Br)=O c1(CCC)nc(C(=O)NCC(C)(C)CNC(=O)Cc2nc[nH]n2)co1 c1(C(C(=O)NC23CC(C(F)(F)F)(C2)C3)F)ccc(SC(F)(F)F)cc1 C1(C(=O)NCCC2CCN(C(C(C)(C)CC3CC3)=O)CC2)CC2C(C1)C2(F)F CC1CN(CCCNC(=O)C(c2cc(F)ccc2Br)C)CC(C)O1 C#CC1(NC(=O)C(CNC(c2cnc(O)o2)=O)CC=C)CCCCC1 C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)NCC1(F)CC(NC(C(C)N(C)C)=O)C1 c1(CN2CCC(NC(c3ccc(F)cc3I)=O)C(O)C2)csc2ccc(Cl)cc12 C1(NC(CN2CC(C)(OC)C2)=O)CN(C(=O)CC(O)C2CCCC2)C2(CCC2)C1 c1(C(=O)NCCC(=C)CNC(=O)CC2CC3CCC2C3)c(S)n[nH]c1C Cc1c(C(N2CC(C)(C)CC2CNC(C2CC2(Cl)Cl)=O)=O)cncc1N C(=O)(C(O)CSC)NCC(CNC(CCN(CCCCC)C(C)C)=O)F CCCCC(C)C(=O)N1CCCC1(C(=O)N(C)Cc1cnc(C)s1)CC C12CCCCC1C(=O)N2C.C1(CN(C(=O)C(F)F)C)CCC(=O)N1 c1(C(N(C(C(C)SC)C)C)=O)cc(C)n(C2CCCOC2)c1C C(=O)(C(F)C(=O)N1CC(OC)C(NC(c2ccc(O)nc2)=O)C1)OCC Cc1nnc2n1CCN(C(=O)C(CC1CCC1)NC(C1CC3CCC1CC3)=O)C2 N1(CCN(CCC)CC)CCC2(CCCN(C)C2)C1 N1(C(CC(COC)NC(=O)C2=NOCC2)=O)CC2(CC2)CC1C c1(C(=O)OC)nn(C)c2c1C(OC(c1cc(C(F)(F)F)n(C)n1)=O)CCCC2 Cc1cc(C(N2CCC2CNC(c2ccc(C(C)F)cc2)=O)=O)c2nccn2c1 C1(C(=O)NCC2CN(C(=O)CCn3ccccc3=O)CCO2)CCC2(CC1)N=N2 CCC(C)C(C(=O)NCC(C)C(C)(C)C)NC(=O)OC(C)(C)C c1(OC(C)C(N2CC3CC2CN3C(=O)C2=CCSC2)=O)ccc2c(c1)CCC2 n1(CC)cnc2nc(=NCC#CC3CC3)[nH]c(NCC3CC4(CC4)CO3)c12 C(C(CC(C)C)C(=O)NCCCC1C=NNC1=O)NC(CCC(C)=O)=O C=CCCC(O)CNC(=O)CCC1(NC(C2C3CCCC23)=O)CCC1 C1(NC(=O)Cc2ccoc2)CC(O)CN(C(c2cnn(CCO)c2)=O)C1 C=C1CC2(C1)CC(C(=O)NC(C)CN(C(=O)CS(=O)(=O)CC1CCCO1)C)C2 c1(OC)ccc(CNC2CC2C(N2CCC(C)(O)C2)=O)c(Cl)c1OC c1(C(=O)NC2CC(OCC)C2OC2CC2)sc(C(C)Nc2ccccc2)nc1C C1(C(N2CCC(OC)C2)=O)CC(NC(=O)Cn2nccc2C)C12CCC2 c1(N(C)C)ccnc(C(=O)NC2CCN(C(c3ccc(C(N)=O)[nH]3)=O)C2)c1 c1(C(N(CC(CN(C)C(c2nc(Cl)cs2)=O)O)C)=O)cccc2c1OCCC2 C(C(C)(C)CCNC(C1CC(n2cnnc2)C1)=O)NC(c1c(C)[nH]cc1)=O c1(CNC(CN2C(C)CCC2)=O)ccc2c(c1)CN(C(=O)C#CC1(C)COC1)C2 CC1CN(C(C2(Cc3ccc(O)cc3)CC2)=O)CCCN1C(C1CC1(Cl)Cl)=O C1(CCCNC(C2C(NC(=O)CCc3ccc[nH]3)CC2)=O)CCOC1=O C1(C(=O)NCC2(O)CCN(C(C34CCC(C3)C4)=O)C2)(CC)CCNC1=O Cc1nc(C(=O)N(CC(O)CNC(=O)CCn2cccn2)C)c(Br)s1 C1(NC(=O)COCc2cccc(O)c2)CCN(C(=O)CC2CC2)CCC1(F)F c1(C(CCC)C)nc(-c2cscc2F)n(-c2ccc(Br)cc2)n1 C1(NCC2CC(OC)C2)CC2(CCN(C(c3ccc(Cl)nn3)=O)CC2)C1 C12(C(=O)NCC#CCNC(c3cc(N)cc(F)c3)=O)C3CC(CC13)C2(F)F C=CCC(C)C(=O)NCc1ncc(C(=O)N(C(C)C(C)C)C2CC2)cn1 N1(C(C=C(C)C2CC2)=O)CCCC2(NC(=O)Cc3ccsc3Cl)CCCC12 c1(C(C)C)ccnc(C(c2nnnn2C(C)C)NC(c2cccc(Cl)c2)C)n1 CC1CN(C(=O)C=Cc2cn(C)cn2)CC(C)C1Nc1nc(Cl)ncc1Br N#Cc1ccc(C(=O)N(c2nc(C(F)(F)F)cc(Cl)n2)C2CCNC2)c([N+](=O)[O-])c1 c1(CN(C)C)ccccc1NC(C1CCCCN1S(=O)(=O)CCCCl)=O c1(CCC(=O)NCC2C(CNC(C(C)(C)CO)=O)C2)ccc2ccccc2c1 CC1c2c[nH]nc2CCC1C(N1CCOC(CN(C(=O)CSC(F)(F)F)C)C1)=O c1(C(=O)NCCC2CCN(C(C3(CC)CC3)=O)C2)ccnc2c(C(N)=O)cnn12 Cc1noc(C)c1C(N1CC(CNC(c2ccoc2C2CC2)=O)C(O)C1)=O N1(C(C(C(=O)OCC)F)=O)CCC2(CC1)CC(NC(=O)CC(C)(C)CC)CCO2 N1(C(CC2C(C)CCC2)=O)CC(C)OC2(CCN(C(=O)Cc3nncs3)C2)C1 c1(SCCCC)cccc(C(N2CC3CC3(NC(C3CCN(C)CC3)=O)C2)=O)c1 C1(CNC(N2C(C(C(=O)OC)(C)C)CCC2)=O)CC=C(C)CC1 C#CCC(C(=O)N(C1CCCS1)CC)NC(c1ccn(C2CC2)n1)=O C12(NC(CC=C=C)=O)CCCCC1N(C(=O)Cc1cnccn1)CC2 C1(C(C)C)(C(=O)NCCC2CC2C)CCN(C(c2n[nH]c(=N)[nH]2)=O)C1 c1(OC)cc(C=CC(=O)N(C)CC2CCCN2C(c2csc(C(N)=O)n2)=O)sn1 Cc1ccc(C(=O)NC2CC(NC(C3(C)CC4CC4C3)=O)C2)cc1OC(F)F c1(C(=O)NC2C(CNC)CCC2)cc(I)ccc1N N1(C(c2ccc(C3CC3)c(Cl)c2)=O)CC2CCCOC2C1 N1(C(c2n[nH]cc2I)=O)CC2COC(C1)C2O N1(c2ccc(C)nn2)N=C2C3(CC(C(=O)NC4CC4)(C1)C3)C2=O Cc1cc(F)c(C(=O)NC2CC3CN(C(=O)CSC4CC4)CC3C2)cc1Br c1(NC(C(n2ccc3ccccc3c2=O)C)=O)cc(Br)cc([N+](=O)[O-])c1 c1(OC)nc(C)ccc1C(N1CCC(CO)(NC(C2C(C)(C)C2(F)F)=O)CC1)=O C1(c2onc(C(C=C)(C)N)n2)CCN(C(=O)CC(=C)C)CC1 c1(OC)ccc(NC(=O)C(CC(C)=O)NC(=O)CCOCC(F)(F)F)cc1C C1(F)(CNC(=O)CSCC(F)(F)F)CCC(NC(C2CCC2)=O)C1 C#CCCCCCCC(=O)N1CCC(C)C(CNC(c2cnn(C)c(=O)c2)=O)C1 CCCC(CC1CCCCC1)C(=O)NCC(O)CNC(c1cnc(C(F)F)s1)=O c1(C(=O)NCCCN(C)C(C2CC2c2cnnn2C)=O)cnc(C2CC2)nc1 C1(N(CC(C)C)CCO)CCN(C(=O)C(C)C2CCOC2)CC1 C(=O)(CC(C)(C)C1CC1)N1CCC(CNC(C=NOC)=O)C1 CC(C)(C)CC(F)C(=O)N1CCCC(CC(=O)NCCC(O)CCO)CC1 C(=O)(C#CC1CCCCC1)N1CCCC(NC(CSC)=O)C(F)C1 c1(C(=O)NCC(C2CC2)NC(=O)C(O)C2CCC2)n[nH]c2c1COCC2 c1(-c2ccc(OC)nc2)ccc2[nH]c(C(=O)NCc3ccccc3CO)cc2n1 c1(C(=O)NC2CN(C(CN(C3CC3)CC)=O)C2)ccnc(SCC(F)(F)F)c1 CCC(CC)CC(=O)NC12CCN(C(=O)Cn3nc(C)cc3C)CC1C2 C(=O)(C1COc2ccccc21)NCCCN(C(=O)C(C)(C)Cc1cnn[nH]1)CC C(C(=O)C(C)(C)C)OC1C(C(=O)Oc2c(C(=O)OCC)csc2)CC1 C(CC(CNC(=O)CC1CC(OC)C1)NC(c1cc(C(=O)OC)co1)=O)OC c1(C(C)NC(CC2N(C(c3cnc(OC)s3)=O)CC2)=O)ccnc(F)c1 CC(CCCN=c1ccc(C(F)(F)F)n[nH]1)NC(c1cccc2c1OCC2)=O c1(C(N2CCCCC(NC(CC(CC)O)=O)C2)=O)cnc2ccccc2c1C N1(C(C(C)OCC2CC2)=O)CCOCCC1C(=O)NCC=CC1CC1 c1(CCC)cc(C(=O)NC(CNC(=O)CC2CCCCC2)CC)no1 CC1=C(C(=O)N2CCN(C)C(C(=O)NC(CO)C(=O)N(C)C)C2)CCO1 c1(N2C(=O)CC(C(=O)NC3(CNC(C(C)(C)OC)=O)CC3)C2)ccc(Cl)c(F)c1 C1(CNC(c2c(COC)cccc2)=O)CC2CCC1N2C(c1cc(CO)on1)=O c1(C(=O)NCCN(C(CNC(=O)OCC)=O)C2CC2)cnc(C(C)OC)s1 N1(C(C2CN(C)C2)=O)CC2CC2(NC(=O)CCCC2CCCO2)C1 C1(NC(CC2CCCC(C)C2)=O)C2CC3C1C3C2C(=O)NCC(C)(C)F N(C(=NCCc1cnccn1)NCC1CC(F)(F)C1)CC(c1ccc(C)cc1)O c1(C(=O)NCC(CC(C)C)NC(C2(C(N)=O)CC2)=O)coc2cc(F)ccc12 N1(C(C(C)(C)OC)=O)CCC(C)(CC(=O)N(C)CC2CCC(C)CC2)C1 n1(CC(=O)NC(C2CN(C(=O)COc3ccc(Cl)nc3)C2)C)cccnc1=O C1(O)(CCNC(C2CC(NS(C)(=O)=O)C2)=O)CCCN(C(c2cc[nH]n2)=O)C1 C1(C(=O)NCCC2CC(NC(=O)CCOC3CCOCC3)C2)CC2(C1)CC2(F)F c1(C(N2CC(C)(C)OCC2CCO)=O)ccc2c(c1)CCOC2 c1(C(=O)NC(CC=C)CNC(=O)CCC2CC2(C)C)c(CO)noc1C Cc1nsc(C)c1C(N1CC(C(C)NC(C2CCCCN2C)=O)C1)=O N1(C(CC(=O)OCC)=O)CC(NC(=O)C(C)N(C)C)C(C)C1 c1(N2CC(C(C)NC(=O)CCC(F)(F)F)C2)cc(C(F)(F)F)ncc1[N+](=O)[O-] C#CC12C3C4C1C1C2C3C41C(=O)NCC(C)(C1CC1)NC(C1CCS(=O)(=O)N1)=O C(C)(C(CC(=O)N1CCCCC1C)NC(=O)CCC(=O)C1CC1)OC C1(C(N(CC(C)NC(CCC(C)SC)=O)C)=O)Cc2ccccc2N1 C1(C(N(C2CC3(CC3)C2)C)=O)CC2CCCC2N1C(c1cccc[n+]1[O-])=O n1(CC)cccc1C(=O)N(CCNC(C1CCCN1C1CCCCC1)=O)C1CC1 C1(NC(=O)CCc2cncnc2)CC(F)CN1C(=O)NC1CC(F)(F)CO1 C1(O)(CNC(CCC(C)OCC)=O)CCCN(C(=O)COCCCN(C)C)C1 C1(CC)CN(C(=O)CC2CC2CC)CC1C(=O)NCC1CCCOC1 c1(C(N2CCC(C)C2CNC(=O)CCc2cocn2)=O)cc2n(n1)CCO2 c1(C(=O)NCC(C)N(C(C2CCN(C)C2)=O)CC)cccc2occ(Br)c12 CC1CCC=C1C(=O)NCC1CCC1C(=O)N(C1CC1)CC1(O)CCOC1 N1(C(C(CC=C)CC)=O)CCCN(C(=O)CSCc2ccncc2)CC1C(C)C N1(C(CC(CCC)O)=O)CCCC2(CCN(C(C3(C)CC3C)=O)CC2)C1 N1(C(CC(=C)C)=O)CC2C(CNC(c3ccc(-n4ccnc4)cc3)=O)C2C1 c1(OC)c([N+](=O)[O-])ccc(CNC(=O)CCNC(C2CCOCC2)=O)c1O CC(C)=C=CC(=O)NC12CC(CNC(C3CC3(F)Cl)=O)(C1)C2 c1(C(=O)NCCCN(C(C(C)CN2CCOCC2)=O)C)cc(F)cc(Cl)c1 c1(OC)ccc(F)c(C(c2nnnn2CC(F)F)Nc2cnoc2)c1F C1(C(N(CC(C)NC(c2ccccc2Br)=O)C)=O)Cc2nncn2C1 C1(CNC(=O)CCCCNC(=O)CCN2CCOC2=O)Cc2ccccc2C1 c1(C(C)F)cccc(NC(=O)CCC2(C)CCN2C(=O)C(c2ccccc2)F)c1 c1(C(C)C)[nH]ccc1C(=O)NCC(C)N(C(=O)CN(C)C(C)C)C c1(C(N(C2CCN(C(=O)C=C(C)C3CC3)C2)CC#C)=O)cc(OC)ns1 N1(C(CCC(CC)OC)=O)CCOC2CCN(C(c3ccc(F)c(F)c3)=O)CC12 Cc1ncsc1CC(=O)NC1(C(F)F)CC(NC(C2CCC(C)C2)=O)C1 Cc1cc(CN2CCOC(CC(=O)NC3CNC(=O)C3)C2)ccn1 N1(C2CCCN(C(C(C(C)C)n3cnnn3)=O)C2)CCN(C2CCC2)CC1=O C(CN=C(NCC(C(F)(F)F)n1cccn1)N1CC(O)C(C)(C)C1)OCCOC C1(C(=O)NCC23OCC(NC(C(C)OC)=O)(C2)C3)CC2CCCC2C1 CC1(C(N2CCC2CNC(=O)CCC(=O)c2ccncc2)=O)CCCCO1 C(=O)(C(C(C)(C)C)C1CCC1)NCCC(C)NC(=O)CC1CC(=O)NC(=O)C1 C1(CS(C)(=O)=O)CN(C(C2(CCO)CC2)=O)CCN1C(=O)Cc1ccco1 N1(C(c2cc(SC)oc2)=O)CC2CC(NC(=O)CN3CCCCS3(=O)=O)CC2C1 c1(C(=O)NCC2C(CNC(=O)CCCn3ccnn3)C2)ccccc1OC1CC1 Cc1cccnc1CCC(=O)NCC(C)NC(c1ccccc1CC#N)=O N1(C(CC(CNC(C(C)c2cccs2)=O)(C)C)=O)CCN(C)CC(O)C1 c1(C(=O)NCC2(CNC(CCS(C)=O)=O)CCCC2)c(N)cccc1F C(CC(=O)NCC1CCN(C(c2c[nH]nc2C2CC2)=O)C1)(C(C)C)OCC CCCCC(C)C(=O)NCC(CC(=O)NCC(F)(F)C(F)F)OC CC(C)CC(CNC(C1CCS(=O)(=O)N1)=O)NC(=O)CSc1nncs1 C(=O)(C1=CC2CCCCCC12)NC1C=CCN(C(c2c(C)[nH]c(=NCC)s2)=O)C1 n1(CCNC(C(C2CCN(C(C=CC(CC)C)=O)C2)F)=O)cnccc1=O CC(N=c1nc(N2Cc3ncsc3C2)c2cccc(F)c2[nH]1)c1cnn(C)c1 C1(NC(C=Cc2cc(OC)ns2)=O)CC(N=c2[nH]c(SC)nc(Cl)c2C)C1 C1(CNC(CN(CCC)C)=O)CC2COCC2N1C(c1cc(CC)ccc1O)=O N#Cc1cc(OCC2CCC3(CC2)CSC3)cc(Br)c1 N1(C(C(CC)F)=O)CC(CO)C2(C1)CN(C(C1CCc3nnn(C)c3C1)=O)C2 C1(C(N2C3C(CNC(C4(C)CC4)=O)C(C3)C2)=O)CC(c2cccc(Cl)c2F)=NO1 N1(C(COC2CN(C(C3C(C)OCC3)=O)C2)=O)CCOC(C(C)(C)C)C1 c1(OC)ccc(COCC(=O)NC23CC(NC(=O)COCC4CC4C)(C2)C3)cc1 c1(C(=O)NCCC(=O)NC(C)C)cnc(CNC(C2(C)CCCC2O)=O)nc1 C(c1cc(F)cc(F)c1)=CC(N1CCC(NC(C(CC)NC(N)=O)=O)C1(C)C)=O Cc1cc(C(=O)NC2(C)CCN(C(=O)C(F)C3CC3)C2)c2cccc(C)c2n1 C(C)(CCCCC(=O)OC)NCC(=O)NCCCCC CC1(NC(=O)CCc2ccc[nH]2)CN(C(=O)CSCc2cscn2)C1 c1(OC)cc(C(N2CCC(C)C2C(=O)NCCCOCCCO)=O)ncn1 C#CCC(C)C(=O)N1CCCC(CN(C(=O)CN(C)C(c2ccsc2)=O)C)C1 N1(CC(N2C(C(N(C3CCN(C)C3=O)C)=O)CC=CC2)=O)C(=O)CCCC1=O c1(C(=O)NCC(C2CC2)NC(C2C(CCC)C2)=O)ccc2c(O)nc(S)nc2c1 C1(C(=O)NC2CC(CO)C2)COC2CN(C(=O)CC3CCOC3)CC12 c1(C(=O)NC(C2CN(C(=O)CCc3cn[nH]c3)C2)C)cc(C(F)(F)F)cs1 N1(C(C(C(C)C)NC(N)=O)=O)CCOCC(C(N2CCCC(CN=[N+]=[N-])C2)=O)C1 C1(CNC(C=CCN(C)CC)=O)CCCC1C(=O)NC(c1ccn(C)n1)(C)C C1(C(=O)NC(CC)C2CC2)CC2CCN(C(=O)NC3CCCC3)CC12.C(CO)N c1(C(N2CC3C(NC(CCC(CC)CC)=O)(C3)C2)=O)ccc(F)c(S(N)(=O)=O)c1 C1(C(N(CCNC(C(CC)n2nccc2C)=O)CCOC)=O)COC(C)(C)CO1 O=C1CN(C(=O)CCS(=O)(=O)N2CC2)C2CCN(C(=O)C#CC3CC3)CC2N1 C#CCC(C)C(=O)N1CC2(NC(c3sc(OC)nc3Cl)=O)CC1C2 C(=O)(CCC(=O)N(C)C)N(C)CC1N(C(C2N(C(C)=O)CSC2)=O)CCC1 N1(C(C(C)CN(C)C)=O)CCCC1(C)CNC(C1(n2cnnn2)CC1)=O N1(C(COCCCOC)=O)CCCC1(C)CNC(=O)C=Cc1csc(C)n1 c1(C(N(C(C)C(=O)NCC2(CO)CCC2)C)=O)cc(Cl)c[nH]1 Cn1cc(S(N)(=O)=O)c(C(N2CC(NC(C3(CC4CCC4)CC3)=O)C2)=O)n1 c1(C(C)NC(=O)CCN(C(=O)CCc2cccnc2)CCO)ccn(C)n1 N1(C(Cn2c(=O)cc(C)nc2)=O)CC(CNC(C2CC(=O)N2)=O)OC(C)(C)C1 C1(C(C)C)(C(=O)NC(C2CN(C(=O)CCNC(=O)C=CCl)C2)C)CCCO1 c1(OC)ccc(C(=O)NCC(F)CNC(=O)CCc2ncc[nH]2)cc1C1CC1 C(=O)(C1Cc2c(Cl)cccc21)NC(CNC(c1ccc(CC#N)cc1)=O)C1CC1 C#Cc1cncc(NC(C2CCC(C)N(C(=O)C(=O)NC)C2)=O)c1 N1(C(C(C)NC(c2c(C)onc2)=O)=O)CCC(C)N(C(C2SCCS2)=O)CC1 N1(C(C2(CCC)CC(=O)C2)=O)C2CCC(C(=O)NC3CC4(CCC4)C3O)C1CC2 c1(C(=O)NCC2C(NC(=O)CCC3CCCO3)C2)ccn(-c2cccs2)n1 c1(C(=O)NC(CCCNC(C2C(CSC)C2)=O)C)ccc(C(F)(F)F)nc1O N1(C(c2cccc(NC)n2)=O)CCC2CN(C(c3cncnc3)=O)CCC12 c1(C(=O)NC2C(NC(=O)C3=CCOCC3)CC2)csc2ccccc12 CCC(CCCC(=O)N(CCSC)CC)NC(C1(C(C)(C)O)CC1)=O C1(C(=O)NCC(CNC(C(Cc2ccsc2)NC=O)=O)O)CC2CC1C1CC21 C1(=CC(N2CC(C)N(C(=O)CS(C)(=O)=O)CC2)=O)CCCCCC1(F)F N1(C(c2cncc(SCC)n2)=O)CCCCCC1CNC(C1CCSCC1)=O c1(C(N2CC(C)C(NC(C3CC(C)(C)C3)=O)C2)=O)ccc([N+](=O)[O-])cc1N c1(C(C(=O)N(CC(C)NC(c2cncnc2)=O)C)C)c(F)cccc1F C1(NC(c2c(OC)nsc2)=O)CCC2(CC1)CN(C(c1ncoc1C(C)C)=O)C2 C1(NC(CC=CCCCCC)=O)CC(O)CN(C(=O)Cc2cnccc2C)C1 N1(C(C(C)Cn2cccn2)=O)CC(C2(NC(C3CCCC(O)C3)=O)CC2)C1 c1(CNCc2onc(CC(=O)NC)n2)nn(C2CCC2)cc1Br C1(Nc2c(C)noc2C(=O)O)CC2CCC(C1)O2 C(C)(C(C)CC)(c1n(CCNC(c2cnccn2)(C)C)nnn1)OCC C1(NC(C(CC(=C)Cl)NC(c2ccc(C)[nH]2)=O)=O)CC2CCC(C1)N2C CCC(C(=O)NCC1(CNC(c2ccccc2NC(N)=O)=O)CCCC1)C(C)O CCC(CC(F)F)C(=O)N1CC2(CCC2)CC1CNC(c1cnc(S)nc1)=O C1(NC(C(c2ccccc2)OCC)=O)CC2C(NC(C3(CO)CC3)=O)C2C1 C1(C(=O)NCC2CC(CC)C2)CCC2CCC1N2C(c1cc(O)ccc1C)=O c1(CC)[nH]ccc1C(=O)NCCNC(=O)C(=O)NCCn1ncc(C(=O)NC)c1 c1(C(=O)NCCC2CCCN(C(C(C3CC3)OCC)=O)C2)cncc(N)c1C c1(C(=O)NC2CCC23CN(C(c2ccc(F)cc2O)=O)C3)ncnc2ccsc12 n1(CC(N2C(CCNC(C(F)=CC)=O)CCCC2)=O)cc(Br)c(O)nc1=O C12(C(N(C)CC3CCCN3C)=O)CCC(CC1)N(C(=O)C(C1(O)CCCC1)F)C2 C1(C(C)NC(C2CC3(CC3)CO2)=O)CCN(C(C2CC23CCOC3)=O)CC1 C(c1ccc(Br)cc1F)=CC(N1CC2C(NC(=O)COCC(F)(F)F)C2C1)=O Cc1cccn2ncc(C(=O)N(C3CN(C(=O)C(O)CN4CCCC4)C3)C)c12 C1(C)(CN(C)C(C2CCCOCC2)=O)CCCC1NC(=O)Cc1ccsc1 C(=O)(C1=NOC2COCC12)N1C2CC(CNC(=O)Cc3ccc(CO)cc3)(C2)C1 Cc1cc(CC(N2CC(O)(CNC(=O)CCOc3ccccc3)C2)=O)ccc1O N1(C(CCC(=O)NC)=O)CCC(NC(=O)CSC(F)(F)F)C(O)C1 c1(C(=O)NCCCN(C(=O)CCc2ccccn2)C)cc(O)nc2cnccc12 CC(C)(C)CC(O)CNC(=O)NC1(C2OCCOC2(C)C)CCC1 c1(N2CC(NC(c3cnn(C(C)C)n3)=O)C(C)(C)C2)ncc(Br)cc1[N+](=O)[O-] CCC(O)C(C)C(=O)N1CC(CNC(=O)C(F)(F)CC2CC2)C(C)C1 C1(C)(C(N2CC(CCNC(C#CC3(CC)CC3)=O)OCC2)=O)CC(C(C)C)=NO1 C(=O)(C(F)C(=O)N1CCCCC1CCNC(c1cnc(S)n1C)=O)OCC CC(C)(C(=O)N1CC(NC(C2(c3ccc(Cl)cc3F)CC2)=O)C(O)C1)C(N)=O C1(CNC(CCC2(NC(COC3(C)CCCC3)=O)CCC2)=O)NC(=O)CC1(C)C N1(C(C2(CCOC)CCCC2)=O)CCCC2(NC(c3nn(C)cc3Cl)=O)CC2C1 N1(Cc2nnc(C)o2)CCC(C(C)NC(=O)CNC(c2cccc(F)c2)=O)CC1 N1(C(C(C)OC2CCCC2)=O)CC(NC(c2csc(Cl)c2Cl)=O)C(C)(C)C1 CCS(=O)c1ccccc1NC(c1cc[nH]c1C1CCCC1)=O C1(C(N(C(CNC(=O)OC)=O)C)C)CCN(C(=O)CNC(c2ccco2)=O)CC1 S(=O)(=O)(c1ccc2[nH]c(=NC3COC(C)(C)C3)ccc2c1)NCCCC(C)O c1(C(=O)NC2CC(NC(=O)CC3CCC34CCC4)C2)c(Cl)ccc(Cl)c1O N1(C(CC2CCCN(C(c3cnc(Cl)s3)=O)C2)=O)CCCCCC1CO c1(NCCC(=O)NC(CC)CNC(C2CCC3(CC3)C2)=O)oc(C)nc1C#N C1(CNC(COCCCN=[N+]=[N-])=O)CC(C(=O)NCCS(C)(=O)=O)=NO1 N1(C(CN(C(c2cc(CC)[nH]n2)=O)C)=O)CCN(C(c2cc(C)[nH]c2C)=O)CC1 Cc1cccc(Br)c1C(N1CCC1CNC(C1CCCC12CC2)=O)=O N1(C(CC(C=C)C)=O)CCN(C)CC1CNC(=O)CN(C(=O)C(C)C)C C1(NC(c2nc(C)[nH]c2C(F)(F)F)=O)CN(C(c2cncnc2C)=O)CC12CC2 C1(C(N2CCC(C(C)(C)NC(c3ccnc(C)n3)=O)C2)=O)CC2COCC2C1 N1(c2ccnc(C(CC)C)n2)CCC2(CCN(C(=O)CCc3cncn3C)C2)C1 N1(C(c2cccc[n+]2[O-])=O)CCCC2(CCN(CC=C(Cl)Cl)C2)C1 C(C(C(F)(F)F)N1CCN(C(=O)OC(C)(C)C)CC1)NC(C1(CC)CCOC1)=O C(=O)(C(C)(C)C(=O)NC(c1ccccc1)C(=O)NCC1CCC(=O)NC1)N(C)C N1(C(C2CC(CNC(c3cccc(C)c3O)=O)OC2)=O)CCOC(C)(C)C1C Cc1cc(C)c(NC(C2CCCCC2NC(c2ccc(F)c(Br)c2)=O)=O)cc1Br c1(C(N2CCC(C)(OC)C2)=O)cnn2cccc(-c3cc(C)cnc3F)c12 C1(NC(C(COCC)NC(C2CCC(=O)N2)=O)=O)CC(CO)C12CCC2 C12(C(=O)NCC3N(S(CC)(=O)=O)CCC3)CC1CN(C(=O)CCOC)C2 Cc1nc2cc(NC(C3CCC(NC(c4n[nH]c(C)c4C)=O)CC3)=O)cnc2[nH]1 CCS(=O)(=O)CC(=O)NCCCCC1CCN(C(c2cccc(C)c2Cl)=O)CC1 C1(NC(Cc2cn(C)nc2)=O)C=CCCC1C(N1CCC1C(N)=O)=O c1(C(=O)NC(CNC(c2c(C)nn[nH]2)=O)C)ccc(CN2C(=O)CCC2=O)cc1 CC1=NN(C)C(=O)C1CC(=O)NC1CC(F)(CNC(C2CCC(C)(O)CC2)=O)C1 c1(NC(CN2CCN(C(C(C)C3CC3)=O)CC2)=O)cc(F)cc(F)c1 C1(C(N(C)C)=O)CCC(C(=O)NCC2COCCN2C(c2ccc(C#N)o2)=O)CC1 c1(CSC)cc(C(N2CCCC(NC(c3ccc(CF)cc3)=O)C2)=O)sc1C Cc1nc(=N)[nH]c(=NCC2(c3ccc(Cl)cc3)CC2)[nH]1 CCC(CC(=O)N1CCCC(O)(c2cn(C3(C(=O)NC)CC3)nn2)CC1)C(C)C c1(C(=O)NC(CCCNC(C2(CCC=C)CCCC2)=O)C)cccc(O)n1 C1(NC(c2c(C)nc(CO)s2)=O)CCCCN(C(C2CC(C)(C)O2)=O)C1 c1(CN2C(CNC(=O)NC(CCSC)C(=O)N(C)C)CCC2)ccc(O)c(O)c1 CC1C(C(=O)Nc2nnccc2C(F)(F)F)CCN1C CCC(C(=O)N1CCC(N(CCO)C(c2cnn(CCOC)c2)=O)C1)C(F)(F)F N1(C(C2(OCC)CC2)=O)CCC2(CCCN(C(C3COCCC3(F)F)=O)C2)C1 N1(C(C(C(C)C)NC(C)=O)=O)CCC(C2(NC(=O)C#CC(C)(C)C)CC2)C1 C(=O)(C(O)CC(F)(F)F)N1C(C(=O)NCC2CCN(CC)CC2)(C(C)C)CCC1 c1(C(=O)NCC2(COC)N(C(C(C=C=C)C)=O)CCC2)cc2cncc(C)c2s1 C=CCC(CNC(c1cncn1C1CC1)=O)C(=O)N(C1CC(CO)C1)C C1(NC(c2scc3c2OCCO3)=O)COC2(C1)CN(C(=O)C(O)C(F)(F)F)C2 N1(C(C(C)c2cc[nH]n2)=O)CCCC2C1CCCN2C(=O)CC1CSCCO1 c1(N2CC(COC)OCC2)ccc(S(=O)(=O)N(CCN2CCCC2)CC)c(Br)c1 Cc1cc(CNC2CC(C(=O)NCCC(C)(C)C)C2)c(C)cc1Br N1(C(C(=O)NC(CC)(C)C)CC(C)C)C2CCC1c1ccccc12 C(C)(CNC(=O)CNC(N1CCCC1)=O)(CC(C)C)NC(c1c(C)n(C)cn1)=O C(CC(C(=O)N1CCC(C)(CC(=O)N(C)Cc2cscn2)C1)OC)OC N1(C(C2CCN(C(CC(C)n3ccnc3)=O)C2)=O)CCC(N(C)C)CC1 CN1CCC(O)(C2(C(=O)NCC(C3CCC3)NC(C3(C4CC4)CC3)=O)CC2)CC1 C1(NC(CCC#C)=O)CCCCC12CCN(C(C13CCC(CC1)C(C)(C)O3)=O)C2 c1(C(N2C(C(=O)OC)CC=CC2)C(=O)NC2CC2)ccc(Br)c(F)c1 c1(C(=O)NCC(C)CN(C)C(c2ccc(C(C)(F)F)nc2)=O)n[nH]cc1[N+](=O)[O-] CC1CN2CCN1C(C(N1CCC(CCNC(C3(C)CC(C#N)C3)=O)C1)=O)C2 C12(C(=O)NCCCCN(C(CS(C(C)C)(=O)=O)=O)C)CC3CC(C1)CC(C)(C3)C2 c1(C(N2CCCC(CNC(CC(C)F)=O)(CO)C2)=O)n[nH]c2c1CCCC2 Cc1ccc(C(=O)NC2CN(C(=O)CCSC3CCCC3)CC2C)c2c1CCC2 c1(OC)c(C(=O)Nc2cccc(C3CC3)c2)cccc1F C(=O)(CCS(N)(=O)=O)NCCNC(c1cc(CC)c(C)s1)=O N1(C(CC=CCC)=O)CC(C)(C)CCC1CNC(C1CCCC(F)(F)C1)=O C(C(=O)N1CCC(NC(C2(C)CCC(OC)CC2)=O)C(F)C1)(C(C)(C)C)OCC CC1CC(C(=O)N(CC(N2CCC(c3ncco3)C2)=O)C2CC2)=NO1 c1(C(N2CC3CC(CNC(C4CC4F)=O)C3C2)=O)nncc2ccccc12 C1(CC)CCN(C(=O)CCC2CCN(C(=O)CCc3ncccn3)CC2)CC1 N1(C(C(C)OCC(C)C)=O)CCCCC1c1cn(CC2CCCCCC2)nn1 N1(C(C(C(C)OC)NC(=O)C=CC2CCC2)=O)CCCC(CO)CC1 C1(CNC(=O)C#CC2CC2)CN(c2ncnc3sccc23)CCC12CCC2 c1(C(N2C(CN(C(CNC(c3c(C)occ3)=O)=O)CC)CC2)=O)cc(F)ccc1O N12CC(CC1(C)C)C(=O)NCC=CC2=O.C1(C(COC)C)CCCC1 C1(NC(c2c(C)nns2)=O)(CNC(=O)Cc2ccco2)CCOCC1 n1(C(CNC)=O)ccc2ccccc12.C12C3C4CC5C1C3C45CNC2=O c1(OC)ccc(C(=O)NC2CC(C)N(C(=O)CC3CSCCS3)C2)c(F)c1N N1(C(=O)C2=CC(O)CCC2)CCC2(C1)CN(C(C1(C3CC3)CC1)=O)CCO2 c1(OC)cc(C(=O)NC(CNC(=O)C(O)C(C)(C)C)CO)c(F)cc1N C12(C(=O)NC(CCCNC(c3ncc(OC)cn3)=O)C)CCCC1CCC2 C(C(C)(C(=O)NC1CC1NC(=O)Cc1nc(C)sc1C)OC)OC c1(C(CNC(CSCC=C)=O)NC(c2nocc2Cl)=O)ccc(N(C)C)cc1 C1(C(=O)OCC)CCCN(C(=O)CN2CCOC2=O)C1 CCCCC(CC)CC(=O)NCCC(C)(C)C(=O)NC1CC(OC)C1 CC1CCOCCN1C(c1[nH]ccc1CNC(=O)CCCC1CC1C)=O S(=O)(=O)(c1ccc(NCCCN2C(=O)CCC2=O)c(F)c1)NCC(CC(C)C)O c1(NC(c2cccn(CC(=O)NCCOCC)c2=O)=O)ccc2[nH]ccc2n1 C1(NC(c2cccc(F)c2)=O)CC2CN(C(=O)CCn3cccnc3=O)CC2C1 C(=O)(C1=CC2C=CC1C2)NC(C(C)C)C(=O)NCCC1CCCC1(C)C C1(C(=O)Nc2ccc(CCCC)cc2)CN(c2ncncc2OC)CC(F)(F)C1 C1(COC)CN(C(C2CC(C(N)=O)C2)=O)CCN1C(=O)C(O)CN1CCCC1 C(CCCCC(=O)NC1CN(C(c2cc(C(F)F)on2)=O)CCC1C)OC C1(CNC(C2C(=C)C2)=O)CCN(C(=O)C(c2ccc(F)cc2)C)CC1 C1(C)(C(=O)NC2CCC(C(=O)NCc3c(C)scc3)CC2)CC2C=CC1C2 C1(NC(N(CCCOCC)CC)=O)CCCN(c2ccc(C#N)cc2)C1=O C=CC1(C(=O)N(C2CCSC2)C)CCN(C(=O)Cc2n[nH]c(C)n2)CC1 c1(C(=O)OC)cc(Br)cc(Br)c1NC(C1CC2CC2N1C(C1CCCC1C)=O)=O C1(NC(C=Cc2cc(C)no2)=O)CCN(C(=O)C(C)(C)CC(C)C)CC(C)(C)C1 C1(O)(CCNC(C2CC2C(F)F)=O)CCCN(C(c2cccc(F)c2Cl)=O)C1 C1(O)(CN(C)C(c2cncc(C3CC3)c2)=O)CCCN(C(=O)Cc2cc[nH]c2)C1 S(=O)(=O)(c1ccc(NCC2CC2)c(Cl)c1)NC(C)CN(C)C.c1(C2CC2)nnnn1CS N1(C(c2ccn(CCCC)n2)=O)CCCOC(CNC(=O)CC2CC2)C1 Cc1cc(NC(=O)C#CCNC(=O)C(C2CCOCC2)O)cs1 c1(C(=O)NCC2CCN2C(C2C3COCC23)=O)cccc2sncc12 N1(C(c2csc3c(O)ccnc23)=O)CCOc2ccc(CN3CCOCC3)cc21 N1(C(CCSC)C(=O)NC(C)C)CCC2(CC1)CNC(=O)N2 c1(CC)cc(F)ccc1C(=O)NCCC(C)NC(=O)Cc1cc(Cl)cnc1C CC(CC(C)NC(=O)Cn1nccn1)NC(C1CCC2CC12)=O C1(C(N2C(C)CCC(NC(c3cnn(C(F)F)c3)=O)C2)=O)Cc2ccncc2C1 c1(C(=O)NCC(N)=O)ccc(NC(=O)Nc2ccccc2)cc1 C(=O)(CC(O)CC(C)(C)C)N(CCC(c1cccs1)NC(C(COC)C)=O)C N#CC1(C(=O)NC2CCC(CNC(C3(C4CCC4)CC3)=O)CC2)CCOCC1 n1(CC(=O)NCC2CN(C(C=CCCC)=O)CC2(F)CO)cc2ccccc2n1 c1(C(=O)NCC2CC(NC(C3COCC(C)O3)=O)C2)coc2c(Cl)cccc12 CC#CCC(C(=O)NCC(C(=O)OC)OC)NC(C1CN2CCC1C2)=O C(=O)(CC(C)C(F)(F)F)NCC1(C)CCN(C(c2cc(C)nnc2)=O)CC1 N1(C(C(CC2CCC2)OC)=O)CCN(C)CC1C(=O)NCCN1CCC(C)C1 C1(C(=O)NC(C)(CNC(c2cc3sccc3[nH]2)=O)CO)CCCC12CCOCC2 c1(CCNC(C2(n3cc(CN4CCCC4)nn3)CC2)=O)cnc(CC2CC2)s1 N1(C(CC(CC)C)=O)CC2CCN(Cc3cccc(Cl)c3OC)C2C1 c1(NCC2(CNC(COCCOC)=O)CC23CCC3)ncc(Br)cc1C#N C1(N(C(=O)C(CC2CC2)OC)CC=C)CCN(C(C2CCC2C(F)F)=O)CC1 c1(C(=O)NC(C2CCN(C(COCCC=C)=O)C2)(C)C)cccc2c1COC2 CCCCCCCCCC(=O)NCC(CC)NC(=O)C(C)(F)C(F)(F)F C1(C(=O)NC(CCC(C)(C)c2ccccc2)=O)Cc2cccnc2C1 c1(NC(C)=O)cc(CC(=O)NCC(O)CO)ccc1O.C12CCN(C1)C(=O)C2 Cc1cc(C(=O)N(CCCN(C)C(C2CCCCC2O)=O)C)c(O)nc1C N1(C(C=CCC)=O)CCCC(C(C)(O)CNC(c2cccc(COC)c2)=O)C1 C1(NC(CN(c2ccncc2)C)=O)CN(C(=O)Cn2ncccc2=O)CC1F c1(NCC(C)OCC=C)cc(Br)ccc1S(=O)(=O)NCc1cc(Br)cs1 C1(NC(C2(C)CCCC2)=O)CN(C(c2ccnn2C2CCC2)=O)C2CCCCC12 C(=O)(CC(C(F)F)n1ccnc1)NCC1(NC(c2c(C)n(C)cc2)=O)CCCC1 C1(NC(C(CC=C)NC(C)=O)=O)CN(C(=O)Cn2ccnc2C)C(CC)(CC)C1 c1(N(C)C)cc(F)c(Br)cc1-n1nc(C2CCC(F)(F)CC2)nc1-c1cnsc1 C(C(CC(C)C)c1nn[nH]n1)N(C(C(CC)F)=O)C(=O)Cc1ccccc1 CC(C)(CCCNC(c1sccc1Cl)=O)NC(C1CC(O)C(F)C1)=O c1(C(=O)NC(CNC(C2(C)CC2)=O)C2CCC2)cc2c(C#N)c(F)ccc2[nH]1 C(CO)(CCCCNC(C1CC2(C1)CC(C)C2)=O)NC(c1c(C)cc(SC)o1)=O C1(C(N2CCC(NC(CCCC)=O)CC2)=O)CN2CCN1CC2C N1(C(C(C)CC2CC2)=O)CC(CN=c2[nH]nc(Nc3ccccc3)o2)C2(COC2)C1 C1(C(=O)NC(C2CCCCC2)C#C)CN(C)CCN1C(=O)CCC=C(C)C C1(NC(c2cc(C)ns2)=O)CC(C)CN(C(c2n[nH]c(C3CC3)c2Cl)=O)C1 N1(C(CC2C(C)OCC2)=O)CCC2(CC1)CCN(C(C1CCN1C)=O)CC2 N1(CCCCCNC(C2CC(C)OC2)=O)CCN(C(=O)CSC(F)F)CC1 CC(C)(C)CC(O)C(=O)NC1CCC(NC(c2csc(C(F)F)c2)=O)CC1 c1(C(N(C(CNC(CC(CC)CN(C)C)=O)C2CC2)C)=O)cc(C)c(C)nc1C C(=O)(C(C(C)(C)C)NS(C)(=O)=O)NCCC1OCCN(C(C=CCOC)=O)C1 c1(CCC)sc(C(=O)N(C2CCC(NC(c3cccc(N)c3)=O)C2)C)cc1CC CCC(C)CCC(=O)NC1(C2CN(C(c3sc(C(F)(F)F)cc3C)=O)C2)CC1 CC(F)(F)C(F)C(=O)NCCCC(O)C(=O)NC1CC(C)(C)C1 c1(OC)cccnc1CCCNC(C1CC(COC(C)(C)C)CN1C(=O)OC)=O C1(NC(C2(F)CN(C(C3C(C(C)C)OCC3)=O)C2)=O)C2CCC(F)(F)C12 c1(C(=O)NCCC2N(C(C3C(C)C3)=O)CCSC2)nn(C)c2ccc(Br)cc12 N1(C(c2[nH]nnc2-c2ccccc2)=O)CCCCC1C1CCCN1CC(Cl)=CCl Cc1cc(C(N2CCCCC(NC(C34CCC3CC4)=O)C2)=O)c2ccccc2n1 C(CCCC(=O)N1CCCC(NC(C2(CCOC)SCCCS2)=O)C1)SC C1(C(N2C(CNC(CC(C)n3cccn3)=O)CC2)=O)C2CCC1(C)C2(C)C C12(CNC(c3c(C)nc[nH]3)=O)CCCC1CN(C(C1CC13CCC3)=O)C2 CC1CC(C(=O)NCCCn2ccnc2)N(C(c2ccccc2O)=O)C1 C1(O)(C(C)NC(CS(CC)=O)=O)CCN(C(C2(n3ccnc3)CCCC2)=O)CC1 C1(C(=O)OC)CN(C(=O)C(=O)Nc2ccccc2Br)CC1(C)COCC(F)F C1(C(=O)NCC(c2cccc(O)n2)O)CC2CC2N1C(C1CC2CCC1O2)=O c1(C(=O)NCC(C(C)C)(C)NC(C2COCCOC2)=O)cccc2sncc12 N1(C(c2cn(CC)nc2C)=O)CCN(C(c2cnn(C(C)(C)C)c2)=O)C(C)C1C C1(C#N)(C(=O)NCC(C)NC(c2c(C)ccc(C(F)(F)F)c2)=O)CC12CCCC2 c1(C(=O)NC2C=CCN(C(c3nc(COC)[nH]n3)=O)C2)c(C)oc(C)c1C CC1CC(NC(=O)CC2(C#N)CC2)CN(C(=O)C(c2cncn2C)O)C1 N1(C(c2c(C)occ2)=O)CC2COCC2(C(=O)N(C2CC2C2CC2)C)C1 CCC(CC(=O)N1CCCC1C(C)NC(c1conc1COC)=O)SC C1(N(C(=O)CSc2n[nH]c(O)n2)CC)CCCN(C(=O)C(C)n2ccnn2)CC1 c1(C(=O)NC2CCN(C(=O)Cn3cc(Cl)cn3)C2)ncc2[nH]ncc2n1 Cc1cccc(Cl)c1C(N1CC(O)(C2CCCN2C(=O)C2=CSCS2)C1)=O N1(C(C=C(C)C(F)F)=O)CCS(=O)(=O)C(CCNC(c2cc(C)c[nH]2)=O)C1 C(c1ccc(=N)[nH]c1)=CC(N1CC(C(C)NC(=O)CC2CC(=O)NC2=O)C1)=O N1(C(Cc2c(O)ccc(C)c2)=O)CC2(CCN(C(C3CC4CC3C4)=O)C2)C1 Cc1ccccc1C=CC(N1CC2CCC2(CCNC(c2cncnc2)=O)C1)=O C1(C(=O)Nc2cn[nH]c2)CN(C(C2CC2c2ccc(F)cc2)=O)CCS1 C1(C(=O)Nc2nc(C)c(C(=O)NC(C)CF)s2)CCc2[nH]c3ccccc3c2C1 CC(C)C(CCC(=O)NCC1CC12CCC2)NC(c1ccnn1C1CC1)=O N1(C(Cc2n(C)cnc2)=O)CCC(c2ccccc2)(CNC(=O)C2=CCC2)CC1 c1(C(N2CCC(N3CC(C(C(=O)OC)O)C3)C2)=O)cccc(F)c1F c1(N(CC(=O)Nc2ccc(CC)cc2)C(C)C)cnc2ccccc2c1 CC(C(=O)N(CC(O)CNC(c1ccc[n+]([O-])c1)=O)C)P(C)(C)=O C1(NC(c2ccc(C(C)(F)F)cn2)=O)CCSC12CN(C(c1scnc1Cl)=O)C2 N1(C(CNS(NC)(=O)=O)=O)CCC(c2ccccc2)C(c2ccccc2)C1 C1(N=[N+]=[N-])(C(=O)NC2C(OC)C(O)C2)CCN(C(c2nc(Cl)oc2C)=O)C1 CCCCC(F)C(=O)N1CC(C2CN(C(=O)C(O)C3CC3)CCO2)C1 C(C(C)(C)C(=O)N1CCCC(CCC(=O)NCCCc2ccsc2)C1)N(C)C CCCCC(CC(=O)NCC=C(C)C)NC(c1[nH]nnc1CC)=O C1(CNC(C(C)=C(C)C)=O)CN(C(=O)C(c2ccn(C)n2)C)CC(C)(C)O1 C1(C(N2CCC(N(C(c3c(C)occ3)=O)C3CC3)C2)=O)CCC(OC2CCC2)CC1 C12(CCC(C)(C)C1)C(=O)N2.C1(=O)CC(=O)O1.C(C)(C)(C)CCSC(C)C C1(CNC(c2ccc(OC(F)F)nc2)=O)CN(C(c2n[nH]cc2I)=O)CCO1 CC(O)C(C(=O)NCC1C2CN(C(C3(N(C)C)CCOCC3)=O)CC12)N(C)C C=C1CC2(C1)CC(C(=O)NC(C1CCN(C(C34CC(CO3)C4)=O)C1)C)C2 Cc1[nH]cc(C(N2CCC3(CC2)CC3CNC(c2cnccn2)=O)=O)c(=O)c1Cl N1(C(C(C)C2CC2)=O)CCN(C(=O)CSc2nncs2)C(C2CCCC2)C1 C(C(CO)(CO)NC(c1cncc(C)n1)=O)N(C(C(C)(C)OCC)=O)C N1(C(CCn2ncc(C)c2)=O)CCC(NC(C2(F)CCCC2)=O)C(C(N)=O)C1 C1(C)(CC)CCC(C(=O)NCC2(CNC(=O)C=Cc3ccncn3)CCC2)O1 c1(C(=O)OC)c(F)cc(NCc2cc(Br)c(O)nc2C)cc1Br n1(C(CC)(C)C)nnnc1C(c1cc(-c2ccco2)on1)NCC1CCC1(F)F c1(C(=O)NCCC(C)N(C(CCOC(C)C)=O)C)ccc(F)c(S(N)(=O)=O)c1 C(C(=O)NOCCO)(C(C)C)NC(C(CNC(C)=O)C)=O c1(CC(=O)NCC2(O)CN(C(=O)CO)C2)csc(N2CCCC2=O)n1 CC1C(NC(=O)C=Cc2cscn2)CC2CCC1N2C(c1ccc(N)cc1)=O N1(C(C(CCN(C)C)NC(c2sccc2C2CC2)=O)=O)CCN(C)C(CO)C1 CC1(CNC(C2(Cc3cccs3)CCCCC2)=O)CCCN1C(C1CCCC1)=O N1(C(c2n(CC)ncc2)=O)CCC=CC1C(=O)N(C)Cc1ncc(C)o1 c1(OC)cc(C(=O)NCC2CC3CN(C(C4(N(C)C)CCC4)=O)CC23)cc(Cl)c1 c1(CC(=O)N(CC(C)NC(=O)CCc2cccc(Cl)c2)C)c[nH]c2ncccc12 CC(C)(CC(F)F)C(=O)NCC1C(Cn2cc(CNS(C)(=O)=O)nn2)C1(F)F c1(C(C(=O)NCCCc2cn(C)cn2)OC)ccc(C#N)cc1F c1(C(N2CC3C(NC(c4n(CC)cc(Br)c4)=O)(C3)C2)=O)cncc(C)c1C CCCCCCC(C)C(=O)NCC(CNC(=O)CCNC(=O)OC)CO c1(CCCSCC)nc(-c2cccc(N)n2)nn1-c1cccc(C)n1 CCCCC(F)(F)C(=O)NCC1(C(=O)N=c2ccn(C)[nH]2)CCCC1 Cc1cc(CNC(C2CC(C)(NC(=O)CC3CC4(CC4)CO3)C2)=O)cc(C)c1 C1(NC(c2cn(C)nn2)=O)CCC(CNC(=O)CCn2cccnc2=O)CC1 C1(C(N2CCC2CNC(=O)C(C(C)C)NS(C)(=O)=O)=O)(OC)CCCCC1 CC(C)CC(O)C(=O)N1CCC(F)(C(=O)N(CC(O)CO)C)C1 C1(CCC(=O)N(CC#C)C)CCCN(C(C2(CC(=O)OC)CC2)=O)C1 c1(C(N2C(CO)CC(NC(C3C(CCC)C3)=O)C2)=O)c(OC)ncnc1OC c1(C(=O)NC(CC)(CC)CCNC(C2CCCSC2)=O)csc2ncnc(O)c12 C(=O)(C1=C(C#N)CCC1)NC(CC=CC)C(=O)Nc1cn(CC)nc1C c1(C(=O)NCC2C(NC(c3c(C(N)=O)nccn3)=O)CCC2)n[nH]c2c1CCC2 C(C(C)C(C)C(=O)NC(C)(C)CNC(c1ccc(CN(C)C)[nH]1)=O)OC Cc1nc(C(=O)NCCCCCN(C)C(=O)C2CC2)ccc1C(=O)N(C)C Cc1cc(N2CCOC(c3ccc(F)cc3)C2)nc(NCC2CCCS2(=O)=O)n1 N1(C(CC(c2c(F)cccc2F)C)=O)CCC(C)C(NC(c2csnc2Cl)=O)C1 C1(O)(C(=O)NCC2(CC(=O)N(CC(C)C)CCN(C)C)CC2)CCCCC1 c1(C(=O)NC2(CC=C)CCN(C(=O)C(O)CN3CCCC3)C2)ccc(C)nc1C N1(C(c2c(C)n[nH]c2)=O)CCC2(CCN(C(=O)CC3CCCCC3(F)F)C2)C1 c1(NC2CCN(C(C(CC)N(C)C)=O)C(C)C2)ncnc2sc(CC)cc12 C1(C(C)(C)O)(CNC(COCCOC)=O)CN(C(=O)CCCF)C1 C1(C(N2CC(C(C(=O)NCCCNC(=O)OC)O)C2)=O)CCCC(=O)CC1 N1(C(CCOCCC)=O)CC2CCC(C(=O)NCC(=O)NOC)(C2)C1 N1(C(c2c(OC)c(Cl)ccc2)=O)CC(NC(c2cn(C)cn2)=O)CC(C)(C)C1 N1(C(C(C)=C(CC)C)=O)CCN(C(=O)C(CC)c2cccnc2)CC(C)C1 c1(C(=O)NC(CC=C)CNC(c2csc(C(F)F)n2)=O)cc(C)c(F)cc1Cl Cc1ccc(C(=O)N(C2CCCC(NC(=O)C(C)(C)c3cc[nH]n3)C2)C)cc1O c1(CC)nc2c(C(=O)NC(CO)C(C)NC(=O)CCn3cncn3)ccnc2[nH]1 N1(C(c2c(OC)nccc2)=O)CCCC(C)(CNC(C2CCS(=O)(=O)N2C)=O)C1 C1(NC(CCc2cnn(C)n2)=O)CCC2CCN(C(c3ccncc3)=O)C12 N1(C(c2cnn(C(C)C)n2)=O)CCCCC(CCC(=O)NCCC(C)(C)CO)C1 C=CCCCC(C(=O)NC(C)CCOCC)NC(c1nocc1C)=O N1(C(C(c2cn(C)nn2)NC(=O)C#CC(C)(C)C)=O)CCC2C(C1)C2(F)F CCC(C(=O)N)N(C)CCO.C(C(=O)C1CC1)(CCOCCCO)NC1CC1 N1(C(C=C(CC)C)=O)CC(OC)CC(C)C1.C12(CC=CC1)C(=O)NC2 C1(N=c2[nH]c(Cl)c(C#N)s2)(CC)CCN(C(C2CC3CCC2C3)=O)CC1 N1(C(c2c(C)nns2)=O)Cc2ccccc2CC1CNC(C1(C)CC(F)C1)=O C1(F)(CNC(C2C(CC(C)C)C2)=O)CN(C(c2ncn(-c3ccccc3)n2)=O)C1 C1(NC(c2cc(CNC(C3C(C)CC3)=O)on2)=O)CC(O)C(F)C1 c1(C(=O)NC(C)CCN(C)C(C2(F)CC2C)=O)csc2ccccc12 N1(C(c2c(C)nsc2)=O)CCC2CC1CN2C(c1cc(C2CC2)on1)=O CCCCC(C(=O)NCCC(C)(C)CC)NC(c1nn(C)cc1C)=O C(CO)(C(C)NC(=O)CN1CC2CC2C1)NC(COCCC(C)C)=O c1(C(=O)NCCCCc2scc(C)n2)ccc(C(F)(F)Br)nc1 C(=O)(C(F)(F)C(O)C(C)C)NC(CC1CN(C(Cc2c(C)cc(Cl)nc2)=O)C1)C Cc1c(F)ccc2[nH]c(C(=O)NCC(C)CNC(C3CCCO3)=O)cc12 c1(C(=O)NC(CN(C(C2C(CCC)CCC2)=O)C)C)nc2ccccc2[nH]1 Cc1c(C(=O)NCC(C)(C2CC2)NC(C2CC23CC3)=O)c[nH]c1C#N N1(C(Cc2c(C)scc2)=O)CCN(C)CC1C(=O)NCC(C)N(C)C C(C(CC(C)C)C(=O)NC(C)(CNC(=O)CC1(NC(C)=O)CC1)CC(C)C)OC c1(OC)c(C(c2nnnn2C(C)C)NC2CC(CF)C2)c(C)nn1C C1(C2(NC(C(c3cnn(C)c3)C)=O)CC2)CCCN1C(=O)C(F)=CC1CC1 C1(NC(C)=O)C(C)CN(C(=O)CCCNC(c2nc(=N)cc[nH]2)=O)CC1C N1(C(C(C)OCC(C)C)=O)CCC(F)C(NC(c2nocc2C(C)(C)C)=O)C1 N1(CC2(C)ON=C(C)C2)CCCC(C(N2CCCC(CC3CC3)C2)=O)CC1 C1(CC(=O)NCC2CC(CNC(C3(F)C(C)C3)=O)C2)CCCCN1C C12(NC(CNS(CC)(=O)=O)=O)CCCC1N(c1nccnc1F)CC2 C(=O)(N=S1(=O)CCC(C)(CNC(=O)OC(C)(C)C)CC1)C1(C)CN(C)C(=O)CC1 N1CC(S(N)(=O)=O)C1.C#CCC(C=O)C1CC1CC(C)(C)C1(O)CCC1 N1(C(C2CC=C(C)CC2)=O)CCC2C1CCCN2C(c1ccc(Br)o1)=O C1(C(=O)NCC(CNC(C(c2cccc(OC)c2)O)=O)C)CN2CCN1CC2C N1(C(CC2CN(C)C2)=O)CCC2(C1)CN(C(=O)C(O)C1CC1)CCO2 CC(O)C(F)(F)C(=O)N1CCC(C(C)(C)CNC(c2cnccn2)=O)CC1 CCC(C)(CC)C(=O)NC1CN(C(=O)CCCNS(C)(=O)=O)C(C)(C)C1 N1(C(CCCC)=O)CCc2ccccc2C1CNC(C1(C(F)(F)F)CC1)=O c1(NC(CC)CCCO)nc(C)cc(=NC2CCn3ncnc3C2)[nH]1 Cc1nc(NC(C2CCC(C)N(C(=O)OC(C)(C)C)C2C)=O)nc(Cl)c1C C1(C(=O)OCC)(C(=O)NCC(C)C2CCC2)CC(C)=C(C)C1 C1(CNC(=O)C=C2CCOCC2)CN(C(C2(C(F)F)CC2)=O)CC12CCOCC2 c1(OC)cc(C(=O)N(CC(C)CNC(=O)C=C(C)C2CC2)C)ccc1C#N C1(O)(CNC(C(C2CCCO2)NC(Cc2ccn(CC)n2)=O)=O)CC(C)(C)C1 c1(OC)cnc(C(=O)NCC23CC2CN(C(=O)COCC2CCOC2)C3)cn1 N1(C(C2(CC#C)CCC2)=O)CCN(C(=O)Cn2nnc(=N)[nH]2)CC12CCC2 c1(NC(c2cc(C)c(Cl)cc2F)=O)cc(O)c2c(=O)n(C)c(=O)n(C)c2n1 c1(C(=O)NCC(C)(CC(C)C)NC(C2C(C=C)C2)=O)cnn2c(C)cc(C)nc12 C1(NC(C2CC(OC)C2)=O)CC2CC1N(C(=O)CC(C)c1cnn(C)c1)C2 C=CC(C)(C)CC(=O)N1CC(NC(=O)Cn2cc(C)c(C(F)(F)F)n2)C2CC12 c1(OC)c(C)cc(C(=O)NC(=O)C(Cl)=CCl)cc1C.C(CCN(C)C)N1CC1 c1(C(=O)NCC2(O)CCCN(C(c3coc(O)n3)=O)C2)noc2c1CCCC2 C12(NC(C=CCNC(C(C)(O)C3CC3)=O)=O)CCN(CC1)C2 CC(C)(C)C(CN=c1nc(O)c2ccccc2[nH]1)NC(C1CC2C=CC1C2)=O C(C)(CC(C)(C)O)NC(C(C1N(C(CN(CC)CC)=O)CCC1)(C)C)=O C(=O)(C1=CC2(CCN(C(=O)Cc3ccnc(O)c3)C2)C1)NC1C(O)CCN(C)C1 c1(CCCNC(=O)NC2(OCC(C)(C)C)CC2)cccnc1 N1(C(C(CC)(C)CN(C)C)=O)CC2CN(CCOCCCN=[N+]=[N-])CC2C1 CC1C(NC(=O)Cc2cnsc2)CCCN1C(c1cnc2n1CCC2)=O C1(CCNC(c2c(C(C)(C)C)n[nH]c2)=O)CN(c2ncc(F)cn2)CCS1(=O)=O C1(C(=O)NC2CCC(NC(CC3CCN(C)CC3)=O)C2)CCCCC12CC2 N1(C(C(CCC)N(C)C)=O)C2CCC1CC(CNC(C1(C)CCCC1C)=O)C2 Cc1scc(CNC(=O)C(C)CNC(=O)CC2CCC(=O)N2C)c1C C(=O)(CCCC(=O)NCC(CO)NC(=O)C(c1ccccc1F)O)OC(C)(C)C C12(NC(C(C)O)=O)CCCC1N(C(=O)C(C)S)CC2 c1(C(=O)NCCC(CNC(=O)C(C)S(C)(=O)=O)OC)cc(F)ccc1CO CC1CCN(C(=O)Cn2ncn(C)c2=O)CC1NC(c1cnc[nH]c1=N)=O N1(C(C2(CC)CC2)=O)CCC(NC(=O)COC2CCCOC2)C(F)C1 C1(C(N(CC(C)NC(c2ccc(Cl)c(N)c2)=O)C)=O)CCc2nc[nH]c2C1 N1(C(CC2(C=C)CCC2)=O)CC(NC(C2CCC2C(=O)NC)=O)C(COC)C1 CC1CCCN(C(c2ccco2)=O)C1CNC(=O)CCN1C(=O)CCC1=O c1(C2C(NCc3c(C)cccc3)C2)cccc2c(-c3cc(F)cc(C#N)c3)cccc12 CC1(C)CCCCC1C(=O)NCC1CCN1C(c1c[nH]ccc1=O)=O C1(C#N)(C(=O)NC(CCNC(C(c2c(C)nn(C)c2)C)=O)C)CCOCC1 CC(C)(C)CCCCNC(=O)CC1(NC(=O)CSc2nc[nH]n2)CC1 c1(C(=O)NC2C(C(=O)NCCC3CC(OC)C3)CC2)ccc2ccoc2c1 c1(NC(CCOCCN(C(C(CC)COC)=O)C)=O)cccn2nccc12 N1(C(c2ccc(OCC=C)c(OC)c2)=O)CCCN(C(=O)CC(F)F)CC1C c1(NC(CCNC(C2C(CC)OCC2)=O)C)nc2c(cc1C#N)CCOC2 O=C1CCC(CC(N2CCCCC2CNC(C2(c3nccs3)CC2)=O)=O)CN1 Cn1ncc(C(=O)NC2CCCC2CNC(=O)CC2CCC(=O)NC2)c1C1CC1 C(=O)(C(=O)C(C)(C)C)CCN1CCC(C(=O)NC2(OC)CC(O)(C(F)(F)F)C2)CC1 CC(C)CC(CCO)NC(C1CCN(C(c2ccoc2)=O)C1)=O C1(C(=O)OC)Cc2c[nH]nc2CN1C(=O)C(O)CC(O)CO C(CC(C)(C)C(=O)NCCCN1CCC(NC(C2C(F)(F)C23CCC3)=O)C1)OC CC1=C(C(=O)N2CC3CN(C(c4cccnc4)=O)CC(C2)O3)S(=O)(=O)CCO1 c1(C(=O)NC(C(C)C)CCN(C)C(C2CC(CF)C2)=O)cc2ccsc2n1C N1(C(c2cc(CNC(C3C(C)CCC3)=O)on2)=O)CC(CO)C(O)C1 C1(C(=O)NC(CCCC)CNC(C2CC(OC)C2)=O)CCCCS1(=O)=O C1(NC(c2ccccc2C(F)F)=O)CN(C(=O)C(O)CC2CC2)CCC1O Cn1ccc(C(C)(C)C(=O)NC2CC(NC(=O)C=CCSc3ccncc3)C2)n1 C(c1cncc(F)c1)=CC(=O)NCC(CNC(C(CC)(F)F)=O)C C1(C(=O)NCC2CC(NC(C3(C)CC3)=O)C2)COc2ccc(Cl)cc2C1 c1(CNc2ccc(C)c(OC3CCOC3)c2)ccc2c(c1)NC(C)C2 c1(OC)cc(N(C)C)ccc1CN1CCOCC1CC(=O)NCCCCCN(C)C c1(OC)ccccc1N(C)C(C1(O)CCN(C(=O)Cc2ccccc2)C1)=O c1(C(c2nnnn2C2CC2)Nc2cn(COC)nc2)cnc(C)nc1 c1(C(=O)NC2(CO)CCN(C(C3CCOCC3)=O)C2)cnn2c(=O)cc[nH]c12 Nc1cc(Cl)ncc1C(N1CC(CNC(=O)CCn2cc(Cl)cn2)C2(CC2)C1)=O C(CC(=O)NCc1cncc(C#N)c1)(C(F)F)NC(C1(C)N(C)CCC1)=O c1(CCC(N2C(C)CC(CNC(C=C(C)C)=O)C2)=O)ccc2ccn(C)c2c1 C(=O)(CC(C)CN(C)C)NCC1(CNC(C(CO)NC(C(C)C)=O)=O)CCC1 C1(NC(C2CCCN(C(C)=O)C2)=O)CC2CCC(C1)N2C(C1CC(C#N)C1)=O c1(C(=O)NC2CN(C(C(c3n(C)ncc3)O)=O)CC2O)cc2ccccc2s1 CS(=O)(=O)c1ccc(C(N2CC3CC4CC3C2C4)C(=O)NC2CCOC2)s1 Cc1ccn(CC(N2CCC(CNC(c3c[nH]nc3-c3cnn(C)c3)=O)C2)=O)n1 Cc1cc(N2CCN(CCNC(=O)C(c3ccccc3)C)CC2)c(F)cc1[N+](=O)[O-] c1(C(=O)NCCCN(CCO)C(C2CCC(O)C2)=O)nnn2c1CCCCC2 c1(C(N2C3(CNC(C(C)C)=O)CCCC(C2)C3)=O)cnc2ncc(Cl)cn12 C(=O)(CC(C(C)(C)C)NC(C1CC1C(N)=O)=O)NCc1c(C)nc(C)o1 C1(NC(c2n(CCC)nc(C)c2)=O)CCN(C(=O)CC2(CO)CCC2)CC1(C)C C1(NC(c2c(OC(C)C)ccc(Cl)n2)=O)CC2CN(C(=O)C(C)(F)F)CC2C1 n1(C(CC)C)ccc(=NC(=O)C(CCNC(C2CCC(F)CC2)=O)OC)[nH]1 c1(OCC)ncc(C(N2CC3(CC(NC(C4OCC4(C)C)=O)C3)C2)=O)cc1Cl c1(OC)ccc(Br)c(NC(N2CCC(c3ccccc3)C2C)=O)n1 c1(C(=O)NC2CCC(Nc3ncc(OCC)cn3)CC2)c[nH]c2ccc(O)cc12 CC(O)CC(C)CN=c1[nH]c(=NCCC2(n3cc(Br)cn3)CC2)[nH]c2cc[nH]c12 N1(C(C(=O)NCCCC(C)OCC)=O)CCCCCC1c1ccco1 c1(C(N2CCN(C(C(CC)n3cccn3)=O)CC2)=O)c(F)cc(Cl)cc1Cl C1(O)(C(=O)NC2C(NC(C(Cn3ccc(C)n3)C)=O)COC2)CCC(C)(C)CC1 C1(NC(c2ccc(C(C)=O)o2)=O)C2CC(NC(=O)CCc3ccc(F)nc3)CC12 Cc1ccc(-n2cc(CCCCNC(c3cncc(F)c3Cl)=O)nn2)c(F)c1 c1(C(=O)NCCC2CCN(C(C3(COC)C=CCC3)=O)C2)cnc(Cl)cc1N CC1(C)CC(CNC(C2CCC2)=O)CN1C(c1csc(-c2cccc(Cl)c2)n1)=O C1(C(N2CC(CO)C3(CCC3)C2)=O)CC(c2ccccc2[N+](=O)[O-])=NO1 N1(C(C(=O)NC2CCN(C(C(=O)OC)C(C)C)CC2)=O)CCn2nc(C)cc2C1 c1(OC)cc(OC)c(C(=O)N(C)CCNC(C2CC(C(C)=O)C2(C)C)=O)cc1Cl C1(NC(C(C(C)C)OCC)=O)CC(O)CN(C(C23CCOC(C)(C2)C3)=O)C1 C12(C(N3CCN(C(C=CC(c4cn(C)nc4)=O)=O)CC3)=O)CC3CC(CC1C3)C2 C#CC1CN(C(=O)C(C)C=C)CCN1C(=O)COC1CCCC1 N1(C(C(CC)N(C)C)=O)CC2CC1CN(C(=O)CCN(C)C(=O)OC1CCCC1)C2 N1(C(C(C)OCC=C)=O)CCC2(CCCN2C(=O)CC23CCC(CC2)C3(C)C)C1 C(CC(=O)NCC(C)(O)CCO)(C(F)F)NC(C1CC=C(C)CC1)=O C1(C(N(C2CCN(C(=O)Cc3cc[nH]n3)CC2)CCOC)=O)CCS(=O)(=O)CC1 C(=O)(C1CCCn2ccnc21)N1CC=CC(NC(c2nn(C)c(Cl)c2Cl)=O)C1 N1(C(CCSCCC)=O)CC(CNC(=O)CCC2(C#N)CCC2)CC1C C1(C(=O)OC)CC2(CCC2)CN1C(c1cnn(CC(F)F)c1)C(=O)NCCCF O=[N+]([O-])c1cccc(Oc2ccc(-c3noc(CCc4ncccn4)n3)cc2)c1 C1(O)(C(=O)NC(C)CNC(C2CC2(F)F)=O)CCCC(C)(C)CC1 c1(C(N2C(C)(C)C(NC(=O)C(F)CC3CCC3)CC2)=O)ccc(P(C)(C)=O)cn1 c1(NCC(CC(C)(C)C)OC)ccc(S(=O)(=O)NC2COCC2F)cc1C#N C(=O)(C(C)(C)CCC#N)NCC1CC(NC(c2c(C)nc(C3CCCO3)s2)=O)C1 C1(C)(C(=O)NCC(C)NC(=O)CNc2ccccn2)CCNC1=O N1(C(C2CN(S(CC)(=O)=O)C2)=O)CCn2c(CNC(C3(F)CC3C)=O)nnc2C1 C1(NC(c2cn(CC)nc2)=O)CN(C(C2CCO2)=O)CCC1(C)C N1(C(=O)COCC2CC2)CCN(C(=O)CCc2cscn2)C(CCO)C1 C1(C(N(C)CC2CCCN(C(c3cn(C)nc3Cl)=O)C2)=O)CCCS(=O)(=O)C1 CCCCCC(F)C(=O)NCCn1cnc(C(=O)NC2CCC(F)CC2)c1 N1(C(C2(C3N(C(c4n(CC)nc(C)c4)=O)CCC3)CC2)=O)CCCSCC1C n1(CC)cnc2c(N3CC(CN(C)C(C4CCC(=O)N4)=O)C3)nc(Cl)nc12 N1(C(c2c(C)nc(C)s2)=O)CC2CCC1C(NC(c1c[nH]nc1C(F)F)=O)C2 c1(C(N2C(C)C(C)S(=O)(=O)CC2)=O)ccc2c(c1)C(C)(C)S(=O)(=O)N2C N1(C(C2(COC)CC2)=O)CCC2(CCN(C(C3CC4CC3CC4(F)F)=O)C2)C1 C(=O)(CCC(F)(F)F)NCCC(C)NC(=O)CCOCCN(C)C1CC1.C(C)(C)(C)NC N1(C(C2N(Cc3nccc(OC)c3)CC(F)(F)C2)=O)CCc2nc(Br)sc2C1 C(CCC(C)C)(C(=O)Nc1cnccc1CO)NC(C(CC#C)O)=O C1(C(=O)NCc2c(C)noc2)CCCN1NC(=O)C1COCC1(C)C N1(C(C(COC)COC)=O)CCC(NC(c2cc(N(C)C)ccc2F)=O)C(F)C1 CON1CCC(C(N2CCCCC2CC(N2CC(CC(F)F)C2)=O)=O)CC1 N1(C(c2cc(C)oc2C)=O)CC2(CO)CC1(C(N1CCCC(C)(F)C1)=O)C2 C12(C(N3CCCC(C(C)NC(c4nocc4Cl)=O)C3)=O)CCC(CC1)CC2 C1(CN(C(C(CSC)OC)=O)C)CCCN(C(c2cccc(C(=O)OC)n2)=O)C1 CC(C(=O)NC1CN(C(=O)CCCCN2CCCCC2)C1)C(C)(C)C c1(C(=O)NC2C(NC(=O)CCF)CCOC2)ccc(Br)c(O)c1 c1(NC(CSCC(=O)NCCNC(C(=C(C)C2CC2)F)=O)=O)ccc(C#N)cc1 CC1CCN(C(C2CNC(=O)N2C)=O)C(C)C1NC(=O)Cc1ccoc1 C1(NC(C2CC(C)OC2)=O)(CNC(=O)OC(C)(C)C)CCCCC1C c1(NC(=O)OC)cccc(NC(=O)CC(Cc2ccccc2)c2ccccc2)c1 N1(C(C2(CC=C)CCCC2)=O)CCC(O)C(NC(c2cnn(C)c2CC)=O)C1 c1(C(N2CCC(NC(C=C(C)C3CC3)=O)C(F)C2)=O)c(F)ccc(O)c1O n1(CCC)ccc(C(=O)NC(C)(C)CC=CC(=O)N(C)CC2COCCO2)n1 Cc1cocc1C(=O)NC1(C(=O)NCC2CC3(CC3)C2)CC(CO)C1 C1(C)(NC(C(C(C)O)NC(C=CC(CC)C)=O)=O)CCC(C)(C)CC1 C=CCC(CC=C)C(=O)N1CCC2C(NC(=O)C(CC)OC3CCCC3)CC12 CC(C)CC(C)(CNC(C1CC2CC1CC2O)=O)NC(=O)Cn1ncn(C)c1=O c1(CC)ccc(C(=O)NCCC2CC(F)(F)CN2C(=O)C=CCOC)c(F)c1 N1(C(c2cc(CC)[nH]n2)=O)CC(C)(C)CC1CNC(=O)C(C)CSC(F)(F)F C(CCCCC(=O)NCC1CC(NC(c2ccc(C)nc2OC)=O)C1)=CC c1(C(=O)NCC2N(C(C3CNC(=O)N3)=O)CCC2)ccc(O)cc1F c1(OCCOC)ccc(F)cc1C=CC(=O)NCC(c1cc(Br)ccc1Br)O C=CCC(C(=O)NCCOCCNC(C1CN(C(C)C)C1)=O)C(C)C.C1CCCC1 C1(C(=O)NCC(C2(O)CCN(C(c3c(C)nsc3C)=O)C2)C)(OC)CCCSC1 C1(C(N2CCC(N(C(=O)C=CC3CCOC3)C)CC2)=O)(CC)CCCCC1 N1(C(C=NOC)=O)CC2CCCCC2(NC(C2CC(=O)NC(CC(C)C)C2)=O)C1 N1(C(C)=O)CC2N(C(=O)Nc3nn4cc(C)nc4s3)CCC2(C)C1 S(=O)(=O)(c1ccc(C#N)c(NC2(c3cccs3)CC2)c1)NCCC(CCC)O CC(CCCc1ccccc1)C(=O)NC1COCC1NC(C1CCCCC1)=O S(=O)(=O)(c1cccc(NC(C2(n3ccc(I)n3)CNC2)=O)c1)Nc1cc(C)on1 c1(Cc2n(CC)c(NCP(C)(C)=O)nn2)cc(F)cnc1Br Cc1ccc(CCCC(N2CC(NC(c3c(C)coc3C)=O)C(O)C2)=O)cc1C c1(C(N(CC(C)NC(=O)CN(C)C(C)=O)CC)=O)csc(-c2cn[nH]c2)n1 c1(OCC(N2CCC(CCOC)CC2)=O)ccc2[nH]ccc2n1 CCCC(CC)C(=O)N1CC(CC(=O)NCC2SCCS2)CC1(C)C CCCCC(O)CC(=O)NC1CC(CNC(C2CC2c2ccc(C)cc2)=O)C1 C1(C(=O)NCCOCCNC(C(C)OCC(C)C)=O)CCCC1P(C)(C)=O C=C(Cl)CCC(=O)N1CCCC1CCCNC(c1cc(C(C)(C)C)n(C)n1)=O C(=O)(C1=C(F)CN(C(C2C=C(C)CS2)=O)CC1)NC(CCC)(C)CC C(CCCCC(=O)NCCCCC(=O)N1CCC(c2ccco2)C1)SC N1(C(C(CC)SC)=O)CC2(CNC(c3coc(C(F)F)n3)=O)CC2(C(F)(F)F)C1 Cc1c(F)cc(C(N2CCCC(c3nccs3)C2)=O)c(F)c1N C(CC(Cl)=CC(=O)N(CCCNC(c1cocn1)=O)CCO)N(C)C N1(C(CCNC(=O)OC)=O)CCCC(C2CC2NC(=O)C(C)c2cccs2)C1 C1(C(N2CCC(CC)C2)=O)CCN(C(=O)Cc2ccoc2C)C12CC2 c1(C(N2CC(C)(NC(C3CC3(C)C)=O)C2)=O)ccc(Cl)c(S(N)(=O)=O)c1 c1(OC)ccc(C(c2nnnn2C2CCC2)Nc2cccc(F)c2)cn1 c1(CN2C(C(=O)NC(C)C(=O)OC(C)(C)C)CC(F)C2)sc2ncccc2c1Cl S(=O)(=O)(c1cccnc1N1CCCC(F)C1)N(CC1(C)CCCC1)CC1CC1 C(=O)(CC(C=C)CCC)NC(C(=O)NCC(C#C)CC1CC1)Cn1cncn1 c1(CC(=O)NCc2nc(C(=O)Nc3ccns3)co2)ccc(O)cc1 CCCC(C)(CC)C(=O)NC1CCCN(C(c2noc3ncccc23)=O)CC1 N1(C(c2ccc(C)c(C(C)(C)C)c2)=O)CCCC12CCN(C(C1CC1C(N)=O)=O)C2 c1(C(=O)OCC)cnc(=NCC(C)NC(=O)COCC2CCCO2)[nH]c1 Cc1cc(C(N2CC3CC2C3C(=O)Nc2cc(Cl)nc(Cl)c2)=O)cnc1F CC1CN(Cc2cccs2)CCN1C(c1ccc(C(F)(F)F)nc1Cl)=O C1(NC(CCC(=O)NCC)=O)CCN(C(=O)CC2CCOC2)CCC1CO n1(CC)cc(S(=O)(=O)N2CC(SC(C)C)C2)cn1.N12CCC(C)(C1)C2=O C1(NC(N2CC(n3ncc(C(=O)OCC)n3)C2)=O)CCC2(CCC2)OC1 CCCC(C)(CC)C(=O)NC1CCCCC1NC(=O)Cc1cc(C)cs1 N1(C(c2c(OC)n(C)nc2C)=O)CCCC2(CCN(C(=O)C(C)(O)C3CC3)C2)C1 c1(C(=O)OC)cc2c(cc1NCCC1CCN(CC(F)(F)F)CC1)OCO2 N1(C(c2c(CC)nc(C)[nH]2)=O)CC2CC(O)C1C2NC(C1CCCS1)=O C1(NC(CC(=C=C)C)=O)CC2COCC(C1)N2C(=O)C(C)OC1CCOC1 c1(C(C)C)ncc(-c2cn(C3CCCC3NC(=O)CNC3CC3)nn2)o1 N1(C(C2OCCN(C)C2)=O)CCC2(CCC2NC(C2CCC(F)(F)CC2)=O)CC1 N1(CC(N2CCC(C3CCCCO3)C2)=O)CCC(F)CC1 N1(C(c2ccc(CC)cc2N)=O)CCC2(CC1)CC2NC(=O)C(C)(C1CC1)OC C1(C(=O)NCCC2OCCCN(C(CNC=O)=O)C2)CCC2(CCOCC2)O1 c1(-n2cc(CN)nn2)cc(C(=O)NCc2ccc(NC)cc2F)cc(F)c1 CC1(O)CCCN(C(C2CCC(CNC(c3cc(F)ncc3Br)=O)CC2)=O)C1 N1(C(c2ccc(OC)s2)=O)CCC(NC(=O)CCSc2ccccn2)C(C)C1 CC1CCN(C(C23CCC(C)(CO2)C3)=O)CC1CNC(=O)Cc1cccc(F)c1 C1(C(=O)NC(CCC)CO)CN(C(C2CN(C(C)=O)C2)=O)CC(C)(C)C1 c1(C(N2CCC(NC(CC(C)(C)O)=O)C23CC3)=O)cc(F)c(C#N)c(F)c1 c1(C(=O)NCC2CCN2C(=O)COC(F)F)cc2oc(Br)cc2[nH]1 O=C1CC(C(=O)N2CCCCC(CNC(=O)C(C)(C)N3CCCCC3)C2)=NN1 c1(C(=O)Nc2ccc(-c3cccn(C)c3=O)s2)n[nH]c2c(F)cccc12 c1(C(N(C(C)CNC(=O)CCCc2cnccn2)C)=O)ccc(C2CC2)cn1 c1(C(N2C(CNC(c3cccc(N)n3)=O)CC2)=O)n[nH]c2ccccc12 C(N=c1[nH]cnc(Cl)c1C(=O)OC)C1CCC(NC(c2nc(CC)sc2)=O)C1 c1(CC)cc(C(=O)NC(CNC(c2c(OC)cccc2Br)=O)CC)cc(O)n1 c1(C(C(=O)NCC=C)N(C2CCC(C)C2)C)ccc(C)c(I)c1 C(=O)(C1CCCn2cnnc21)NC1(CNC(C2(N=[N+]=[N-])CC2)=O)CCC1 CON1CCC(C(N2CC(C)(C)CC2C(=O)NC2(CCF)CCC2)=O)CC1 C1(CNC(C(CC)(C)C)=O)(NC(=O)CCC(=O)c2cnn(C)c2)CC2CCC1C2 C(=O)(CCC(C)(C)C#N)N1CCN(C(c2cc(CC)c(O)cc2)=O)CC1 c1(C(c2n(CC(=C)C)nnn2)NCC2C=CCC2)ccc(-c2scnc2C)cc1 c1(C(N2CC(N)C(O)C2)C(=O)NC(c2ccccc2)C)ccc(F)cc1Cl c1(CNC(C2CCCS2)=O)cncc(C(=O)NOCc2nc[nH]n2)c1 C(CC1CC1)(CC(=O)N(C)CCc1cnn(C)c1)NC(C1(C(=O)NC)CC1)=O N1(C(CCOCCOCC)=O)CCC2CN(C(=O)CN=S(C)(C)=O)CCC2C1 C#CCC(O)C(=O)C(CCO)=O.c1(CNC2CC2)cccnc1.C12(CCC1)C(=O)N2 c1(C(N2CC(NC(c3cc(OC)no3)=O)C(OC)C2)=O)ccc2c(c1)NCC2 Cc1cc(NC(=O)CC2CCCN(C(c3cncn3C3CC3)=O)C2)cc(C)c1F O=C1CC(C(=O)NCC(C2CCCC2)O)N(C(C2(CCCCO)CC2)=O)C1 C1(CC(=O)NCc2ccc(C(=O)NC(CSC)(C)C)o2)CCC(C)CO1 C(C)(C)(CC(F)C(=O)N1CCSC(C)C1C)NC(C(CC=C)CC)=O N1(C(=O)OC(C)(C)C)CC2(CCC2)CC1CNC(C1CCC(N=[N+]=[N-])C1)=O c1(COCC(=O)NC(C2C(=O)NC2)=O)ccc(N2CCOCC2)c2cccnc12 C(=O)(CCCN=[N+]=[N-])N1CCCC(CN(C)C(c2nc(Cl)cs2)=O)C1 C[Si](C)(C)c1ccc(-c2csc(NC(=O)CC3CCCC3)c2)cc1 C(=O)(C1=COCCO1)N(C1CCCCC1)CCNC(c1cc(C(C)C)n(C)n1)=O c1(NCCOCC(=C)C)cc(C)c(S(=O)(=O)NC2CCCC(F)(F)C2)cn1 c1(C(=O)NCC2N(C(c3ncn(C(C)C)n3)=O)CC(F)C2)ccc2nccn2c1 N1(C(=O)COCc2ccccc2)CCC2CN(CC3CC3)CC12 CCCC(CCCNC(=O)CC1CCCC(C)(C)C1)NC(c1c[nH]nc1SC)=O Cc1ccc(C=CC(=O)N(C2CCC(NC(=O)Cc3ccoc3)C2)C)o1 Cn1cc2cc(C(=O)NC3CC(O)CN(C(=O)C4=NOCC4)C3)ccc2n1 C(c1cnc(O)nc1O)=CC(N1C(C)C(NC(c2nn[nH]c2Cl)=O)CC1)=O Cn1c(I)cc2c(N3CC(C(=O)Nc4cncc(C(F)(F)F)c4)C3)ncnc12 CCCCC(=O)C(=O)NCC(O)C(=O)NC(C(C)C)c1nc[nH]n1 Cc1cc(=O)n(C)nc1C(=O)NC1(CN(C(=O)C(CCO)N(C)C)C)CC1 N1(C(C(C)NC(=O)CC(C)(C)C)=O)CCC2(C1)CN(C(=O)C(=O)NC1CC1)C2 Cc1cc(C(C)C(=O)NC23CC(NC(=O)CC4CSCCS4)(C2)C3)cc(C)c1 C1(C(=O)NC2CCN(CC)C2)CC=CCC1C(=O)NCC1=C(C)CCC1 C(C(=O)NOC(C)C)(C1CCCC1)NC(c1cc(CC)sn1)=O C1(CC(=O)N(C2CC(COC)C2)C)CCC(NC(C2(C)CSC2)=O)C1 c1(C(=O)NC(CC(C)C)CNC(=O)C(=O)NCC2CC2)ccc(F)c(F)c1 c1(CNC(C(CC#C)NC(=O)Cc2cnc(C)s2)=O)ccc(F)c(C)c1 CC1CCC2(CC1)NC(=O)N(Cc1nnc3ccccc3n1)C2=O C12CCC3(CCN(CC3)C1=O)O2.CC(CNC(=O)OC(C)(C)C)S(C)(=O)=O C1(C(=O)OC)(COC)CCCCN1C(=O)Cn1cc(-c2ccc(Cl)nc2)nn1 C1(CC(=O)NC2CC3(CC(C)(C)C3)C2)C(=O)Nc2ccccc2S1(=O)=O CC(C)CC(C)CC(=O)N1CCC1CNC(c1cc(=N)[nH]cc1Br)=O C1(NC(C(N2C(C)CCC2C)C)=O)CC2CCC(C1C)N2C(c1ccnn1C)=O N1(C(C(C)NC(=O)CCC2CCCCN2C)=O)Cc2ccccc2C1 Cc1cccnc1C(=O)N(C1CC1)CC1CCCN1C(C1CC12CC2)=O C1(C(=O)NCCC(C)NC(=O)Cc2cnsc2)CCC(=O)N(CC(F)(F)F)C1 N1(C(c2c(C)n[nH]c2)=O)CC(NC(=O)COCCN(C)C)CC1(C)C N1(C(c2cc(CC)no2)=O)CC2CCC1(CNC(C1CCCC(C)CC1)=O)CC2 C(=O)(C(CC(=O)OC)NC(C)=O)N1CC(CC=C)(NC(=O)CCCCF)C1 C1(NC(CC#N)=O)CC2(C1)CC(NC(C1(c3cncnc3)CCCC1)=O)C2 C(CN=c1[nH]nc(-c2ccon2)s1)N(C(=O)C=Cc1cncc(F)c1)C1CCC1 N1(C(C2(CC=C)CC2)=O)CCCC(C2CN(C(=O)CC3=NNC(=O)C3)C2)C1 C(=O)(C(CC1CCOC1)NC(c1ccc(OCC2CC2)s1)=O)OCC C1(NC(=O)CC2CC(F)(F)C2)Cc2ccccc2C1NC(=O)Cc1cscn1 N1(C(C(C2CCC2)OC)=O)CC(CO)(NC(c2cc(C(F)(F)F)cs2)=O)C1 N1(C(C(C(C)C)SC)=O)CCC2(CCN(C(c3cc[n+]([O-])cc3)=O)C2)C1 CN1CC(C)(NC(C2(F)CCN(C(=O)CC3(O)CCCCC3)CC2)=O)CCC1=O c1(CNC(C2(CNC(C3C(CC)CCC3)=O)CCC2)=O)cc(C)c(C)o1 c1(OC)ncc(C(=O)NC(c2ccc(F)cc2)CC(=O)Nc2sncc2C#N)cn1 c1(CC(=O)NC(CNC(c2cccc(-n3cncn3)n2)=O)CO)cncc(O)c1 c1(C(N2CCCC(CNC(C(C)n3ccnn3)=O)C2)=O)ccc(F)cc1F c1(C(N(CCCNC(C(CC)C(C)C)=O)C2CC2)=O)cc(F)c(OC)c(Cl)c1 C1(C(=O)NC2(C)CCN(C(c3n(CC)nnc3)=O)C2)Cc2nccnc2C1 N1(CCC(=O)NC(CC(C)NC(CSCC=C)=O)C)C(=O)C2CC=CCC2C1=O C=Cn1nncc1C(=O)NC1(C)CC(NC(=O)CSC(F)F)C1 N#CC1(C(N2CCCC(NC(=O)CSCc3cccs3)C2)=O)CCCCC1 C(=O)(C1=CCC(C)(C)CC1)NC(C)C(C)(C)C(=O)N(C)CC1CCCOC1 CC1CN(c2ccc(C(N3CCC(O)(Cc4ccc(Cl)cc4)C3)=O)cc2)CCN1 N1(C(C(C2CC=CCC2)NC(c2nocc2Cl)=O)=O)CCCC(F)(F)C1 c1(CN2CCN(C(c3n(C)cc(Br)n3)=O)C3C2C3)ccc(C#N)c(F)c1 N1(C(CSCC#C)=O)CCCCC1CCC(C)(C)NC(c1ccnn1C(F)F)=O C#CCCCC(=O)N(CC(Cc1ccccc1)NC(c1ccc(OC)cc1)=O)C C12(OC)CNCC(C(N3CC(Cn4cncn4)C3)=O)(C1)C2 c1(OC)cc(F)c(Br)cc1S(=O)(=O)Nc1ccc(C2CNC(=O)C2)cc1 C(=O)(C(CN(C)C)NC(=O)C(F)n1ccnc1)N(CCC(C)O)C C1(NCC2C(C(C)C)C2)CCCC1Cc1ccccc1 C1(C(=O)NC2CC(NC(C(CC)CC(C)C)=O)C2)CCC2(CC1)NC(=O)NC2=O N1(C(CCCC2C(C)C2)=O)CCC(CC(=O)NC(C)CC(=O)N(C)C)C1(C)C C(=O)(C1=NOC2(CCC2)C1)NC1CC2CC(NC(C3C(CC)C3)=O)CC21 c1(SC2CCCCC2C)cccc(OC)c1.C=C(C)CO c1(NC(N(CC(=O)NCC(C)C(=O)O)CC)=O)cc(C)ccc1C Cc1noc2ncc(C(=O)NC(C)CNC(C3(F)CCOC3)=O)cc12 C(=O)(C(CC(N)=O)NC(=O)Cn1cc(CSCCSc2ccccc2)nn1)OC C12(C(=O)NC(CN(C(=O)Cc3c(C)n[nH]c3C)CC)C)CCCC1(C(N)=O)C2 c1(C(=O)NCCC(=C)CNC(c2c(C)nn(C)c2Cl)=O)cc(C)ccc1CC C1(C(N(CCNC(CC(=C)C)=O)CCOCCO)=O)CC2C=CC1C2 Cc1cnc(F)cc1C(=O)NC1CCN(CCNC(C2CC2C)=O)CC1 C(=O)(C(F)C(=O)NCC1(C(=O)NC2(C)CC(O)C2)CC(C)(C)C1)OCC c1(C(=O)NC2C(C)CN(C(c3cc[nH]c3)=O)C2)c(F)c(F)c(Br)c(F)c1F C1(C(c2n(CC(=C)C)nnn2)NCCn2cncc2CC)CCCCCCC1 c1(-c2cc(C(=O)NC3C(NC(c4cc(C)sc4)=O)CC3)n[nH]2)ccc(C)c(C)c1 N1(C(C2CN(c3ccc(OC)c(C)c3)C(=O)C2)=O)CCC(OC)CC12CC2 N1(C(C2N(CC)CCOC2)=O)CCC(F)(CNC(c2cn(C)cn2)=O)CC1 C1(NC(CCOCCC)=O)CN(C(=O)CCN2C(C)CCCC2C)C2CCCC12 CC1(CNC(=O)CC2CCC(O)C2)CCCN(C(C2CCC2)=O)C1 c1(SC)ccc(C)c(C(=O)NCC(C(C)C)NC(=O)CC#N)c1 C(=O)(CCC(C)OC)N(CC(C(N1CC(C)(CC=C)C1)=O)C)C C=C(C)CN=C(NCCN1CCC(C)(C)C1)NCC1(c2ccc(Br)cc2)CCC1 N1(CC)CC(C(=O)NCC#CCNC(=O)CN(c2cnccn2)C)NC1=O N1(CCC(=O)NCC2C(NC(=O)CCCc3cc[nH]n3)C2)C(=O)CCC1=O C1(C#N)(NC(c2c(C(=O)OC(C)C(=O)N3CCCC3)nco2)=O)CCOC1 C1(C(=O)NC2CCC(OC)C2)CCCN(C(C2(CC3CC3)CC2)=O)CC1 C1N=C2C=C(N=CN2)NC12CCC2.c1(CCSC)ocnc1C C1(OCC(=O)NCCSCC(F)(F)F)CCNCCC1c1ccccc1 N1(C(C2C=CCN(C(C3CCCOC3)=O)C2)=O)CCCC12CCCCC2 C(CCCN=c1[nH]c(=NCCC(C)SC)c2sccc2[nH]1)c1ccc(OC)cc1 c1(C2(O)CN(Cc3cnn(CC4CCOC4)c3)C2)ccc(F)cc1F c1(NC(N2CCCC(C(C)NC(=O)CCc3cncs3)C2)=O)cc2c(s1)CCC2 c1(NC(CC(C)N2CCCC2=O)=O)c(F)cc(Cl)cc1F S1(=O)(=O)CCN1Cc1ccccc1.c1(COCC(=O)OCC)nc[nH]n1 C(=O)(CC(C(F)F)NC(C1C(C)C1C)=O)NCC(C(=O)NC)(C)C N1(C(C(C=CC)O)=O)CC(C)(C)CC1CNC(C1(O)CCCCC1)=O N1(C(C(C)=CCC)=O)CCOC(C(=O)NCCn2ccnc2C)CC1 CC1CC2CCC(C(N3CCN(C(C4C=CC=CC=C4)=O)CC3C)=O)CN2C1 CCC(C#N)C(=O)N1CC(F)CC1C(=O)Nc1cnn(C(C)C)c1 Cc1c(C(=O)NC(CNC(=O)CC2C=CCCC2)CO)cccc1Br N1(C(CC2C(C)CCO2)=O)CC2N(C(c3ccn4ccnc4n3)=O)CCC2(C)C1 CC(CC#N)C(=O)NCCN(C(=O)CCn1cncn1)C c1(C2CCC2)ccc(Cl)cc1.C(=O)(CCCNC(=O)ON)N(CCCOCC)C(C)(C)C c1(C(=O)O)ccc(C(N2CCC(F)(F)C2)=O)c(Cn2cc(-c3ccoc3)cn2)c1 C1(C(=O)NC(C#C)C)CN(C)CCN1C(c1ccc(OC)nc1)=O C1(NC(c2c(C(C)C)n(C(C)C)nc2)=O)CCCN(C(=O)OC(C)(C)C)C1C C12(CCNC(c3ccc(C(C)(C)C)[nH]3)=O)CCC1CN(C(=O)CCCC(N)=O)C2 Cc1nc(C(C)C)ccc1C(=O)NC1C2CC1N(C(c1c[nH]nc1Br)=O)C2 CC1(C)CC(CC(=O)NCC2CC(O)C2(C)C)N(C(=O)CN2CC3CC3C2)C1 C1(OCC)CC(F)(F)C12CCCC2.C12CCCCN1C2=O c1(OC)cc(C(=O)NC2CC(CNC(=O)C(=O)N(C)C)C2)ccc1C C1(NC(C(C(CC)(C)C)O)=O)CC2CCC(C1C)N2C(=O)Cc1cc(C)nn1C N1(C(C=Cc2ccc(C)o2)=O)CCCC(C)(CNC(C2CCCC23CCC3)=O)C1 CC(C)C(C(=O)NC(C)(C)C(C)NC(C1(COC(C)C)CC1)=O)NC(N)=O CN1CCC(C)(NC(=O)Oc2ccc(OC(C)(C)C)nc2)C1 Cn1cnnc1CCC(=O)NCCc1ocnc1CNC(c1ccc(CO)s1)=O CC(C)C(CNC(=O)CCc1cnccn1)C(=O)NC(CN1CCCC1)CO S(=O)(=O)(c1cccnc1NC1(CO)CCCC1)NCCC12C(C)(C)C(CC1)CC2 C12(C(=O)NCCN(C(C)C)C(c3ccnnc3S)=O)CC(C1)C(C(F)(F)F)O2 C1(CC(=O)NCC2(CNC(CCNC(N)=O)=O)CCC2)CNC(=O)O1 c1(CNC(C(C)OCC#C)=O)nc2c(s1)CN(C(c1[nH]cnc1C)=O)CC2 Cc1cc(NC(c2nnnn2CCCF)CCC2CCCC2)cc(Cl)c1 Cc1cc(Cl)c(C(=O)NC2CCN(C(=O)C=Cc3ccncc3)CC2CO)cn1 Nc1cc(C(=O)NC2CCCC2NC(c2cncc(C(F)(F)F)c2)=O)cc(Cl)n1 c1(C(N2C(C)CCC(NC(C(c3ccc(Cl)s3)C)=O)C2)=O)n[nH]c2c1CCOC2 CC(CN(C(=O)CCOCCOC1(C)CC1)C)C(=O)NOCCOC N1(C(c2c(C)cco2)=O)CC2(C1)CN(C(C1CC1C1CC1C)=O)CCO2 c1(C(N2CCCN(C(C3C(=C)CC3)=O)CC2)=O)cc2c(cc1Cl)NC(=O)CO2 Cc1ccc(Br)c(N2CCN(C(=O)C(=O)NC3CC34CCOCC4)CC2)c1 c1(CN2C(C(=O)Nc3ccc(Cl)c(Br)c3)CSCC2)cc(Cl)c(Cl)cc1O N1(C(c2ccc[n+]([O-])c2)=O)CC2CCC(C1CO)N2C(=O)CC1CCCO1 C1(C(=O)NCC2(C(C)(C)O)CN(C(C3(F)CCCC3)=O)C2)CC12CCSCC2 C1(N(C(CN(C)C2CC2)=O)C)CCC2CN(C(=O)C(=O)N=S(C)(C)=O)CC12 C#CCC(CC#C)C(=O)NC(CN(C)C(c1cccc(OC)n1)=O)CC c1(C(N2CCN(C(C3(CO)CCC3)=O)CC2)=O)ccc2oc3ccccc3c2c1 C1(C(N2CC(CN(C)C(c3cnnc(O)c3)=O)C2)=O)(CC)CCCCC1 C1(NC(CN(C)C(=O)C2CC2)=O)CCCN(C(C2CC3(CC(=O)C3)C2)=O)CC1 C(=O)(C1=CCC(NC(=O)C(C)(C)N2CCCC2)C1)N(CCCC(=O)OC)C c1(C(N(CC(CC)NC(c2ccco2)=O)CC)=O)ccc(F)c(CC2CC2)c1 c1(NC)cncc(C(=O)NC2CCCCC2NC(C2(F)CCOCC2)=O)n1 C(=O)(C1=CCCCC1P(C)(C)=O)NC(C1N(C(CCCNC(C)=O)=O)CCC1)C C1(NC(c2nn(CC)c(O)c2)=O)CN(C(=O)C=CCN2CCOCC2)CCC1C N1(C(CNC(CCC)=O)=O)CC(NC(=O)C(CO)c2ccccc2)CC(F)C1 C1(C)(NC(C(C)=CC)=O)CCCN(C(c2ccccc2-c2cnn(C)c2)=O)C1 Cc1cc(Cl)c(Cl)cc1C(N1C2CNCC1C2)=O.C.CCS c1(CC)ccc(OC(C2CCN(CCN(C)C)CC2O)=O)c(CC2CC2)c1 C1(C)(C(N2CC(C)C(NC(C3(C(F)(F)F)CCCC3)=O)C2)=O)CC2(CCC2)C1 C1(C(=O)NCC2CN(C(c3c(CC)oc(C)c3)=O)C(C)C2)CCC2(CCC2)O1 CC(C)CCC(C(=O)NC1CN(C(=O)C2CC2)C1)NC(=O)CC(O)CN(C)C C1(NC(c2n(C)ncc2Cl)=O)CN(C(C2CC2c2ccnn2C)=O)C2(CCC2)C1 C1(NC(C2(C)N(C(C(C=C)CC)=O)CC=C2)=O)CC(C)N(C)CC1C c1(CCC(=O)NC2(CNC(c3c(CCC)nco3)=O)CCC2)cccc(Cl)c1 C(=O)(CC1=CCCCC1)NC1C(NC(c2cccc(C(C)C)c2)=O)CCC1 N1(C(C(CC(=C)C)NC(c2cccc(F)c2F)=O)=O)CCn2ncnc2C1 CCC(CCC(=O)NCCC1CCCCO1)NC(=O)C1CC1 C(CC(=O)N(C1CC(C(N)=O)C1)C)N(C(c1cc[nH]c1)=O)CC C#CC1(C(N2CCC(CCN(C)C)C2)=O)CN(C(c2ccc(O)nn2)=O)C1 Cc1onc(Cl)c1C(N1CCN(CCCNC(=O)CC2(C)CC2)CC1)=O Brc1[nH]nc2ncc(-c3nc(CCCc4ccccc4)nn3C3CCSC3)cc12 N1(C(C(C(CC)CC)OC)=O)CCCC2(C1)CN(C(C1CCC3(CC3)C1)=O)C2 N1(C(C=C(CC)CC)=O)CC2(CCN2C(=O)COCP(C)(C)=O)C1 Cc1ccc2c(n1)CN(C(=O)CCC(CC)NC(C1C(C#N)C1(C)C)=O)C2 CCC(C(=O)N1CCCC1C(C)NC(=O)Cn1nccc1C)n1nccc1C C1(CCC(N2CC(O)(CN(C(CCCOC)=O)C)C2)=O)C(=O)NN=C1C C1(CC)CN(C(c2cc(C)c[nH]2)=O)CCN1Cc1ccc(C)cc1 N1(C(C(C)CN(C)C)=O)CCN(C(C2CCC(=O)NC2)=O)C(CCO)C1 N1(C(C2CC(C)(NC(C(C)N=[N+]=[N-])=O)C2)=O)CCC12CCCSC2 N1(C(=O)Nc2ccc(SC)cc2)CCCC(C)(C(=O)NC(C)CO)C1 N1(C(C)=O)CCCC1C(=O)NCC1(NC(=O)C(C)C2CCCO2)CCC1 c1(CCC(=O)NC(CCCCNC(CSCCC(C)C)=O)C)ccc(Cl)c(Cl)c1 C1(=O)C(O)C(O)C(=O)NCC23CC(CO2)N(C3)C1=O.C(C)(C)(C)OOC c1(Nc2scc(C)n2)ccc(C(=O)NC(CNC(=O)CC2(C)CC2)C2CC2)cc1 c1(CCCC=C)cn(C2CC3(C(=O)NCCOCC4CCCO4)CC23)nn1 c1(C(N2CCC(Oc3ccc(CC)cn3)C2)=O)cccc(C(C)C)c1F N1(C(c2c(C)c[nH]n2)=O)CC2CC(NC(=O)CN3CCCC3C)CC1C2 N1(C(C2CN(C(CC3CCC(C)(C)O3)=O)CC2(F)F)=O)CC2COCC2(C)C1 c1(OC)cc(C(=O)NC2CCCC(CNC(=O)CCOC(C)=O)C2)cc(F)c1 Cc1cc2ccc(C(N3CC(C4CN(C(=O)CN(S(C)(=O)=O)C)C4)C3)=O)cn2c1 C1(C)(C(=O)OC2CC(=C)C2)CC(OC(C)(C)C)C1 C#CCCCCCC(=O)N(CCNC(c1cccc(Cl)c1C)=O)C1CC1 N1(C(CC(C(F)(F)F)OC)=O)CCCC(C2CCN(C(C3(Cl)CC3)=O)CC2)C1 Cc1[nH]c(=NCc2ccc(O)nc2)sc1C(=O)Nc1ccnc(Cl)c1Cl C#Cc1ccc(F)c(C(=O)NCCOC2CN(C(C3(C)CCCC3(F)F)=O)C2)c1 CC(C(=O)N(CCCCNC(=O)C(F)n1cccn1)C)C(C)(C)O C1(F)(C(=O)NC2C(OCC)CCC2)CC2CC1(c1ccccc1)C2 C#Cc1ccc(C(N2CCC(CCNC(=O)C(C)(C)OC)C2)=O)cc1 CN1CCN(C(=O)C(=O)C2CCCC2)CC1NC(=O)C(F)(F)F.C1CCO1 C1(C(=O)OC)CN(C(C(=O)NCCCSC)c2cccs2)CC(C)(C)O1 C1(CN(C(C=C(CC)CC)=O)C)CN(C(c2csc(C(F)F)c2)=O)CCO1 Cn1ccc(CNC(=O)C(CC2CC2)NC(=O)CCc2ccn(C)n2)n1 c1(C(N2CC3N(C(COC)=O)C3C2)=O)cc2c(C)snc2s1 Cc1nc(CO)sc1C(=O)NC1CCC1NC(=O)C=Cc1cscn1 C1(NC(C2(C(=O)OCC)CC2)=O)CN(C(c2ccc(C)nn2)=O)CC1C1CC1 C1(C(N(CCCOCCN(C(CCNC(C)=O)=O)C)C)=O)C2COCC12 C(=O)(C1=CNC2=NCCCC2=C1)N1CC=CC(NC(=O)CCN2CCCCC2)C1 c1(C(N2CC(O)(CNC(CCCOC)=O)C2)=O)cc(N)cc(C)c1F Cn1ncc2ccc(CC(N3CCCC(CCC4CCCNC4)C3)=O)cc12 CCCCCCCCNC(=O)CC(CNC(C1CCC(C)(C)OC1)=O)C1CCC1 n1(CC(=O)N(C(C)CNC(C2CCN2C)=O)C)ccc(O)nc1=O c1(C(=O)OC)ccc(C=CC(N2CCC2CNC(=O)COCc2nccn2C)=O)o1 c1(CC)cccc(C(=O)NC2CCN(C(=O)Cc3cc(C)no3)C2CC)n1 c1(SCc2cn(CC)nc2)c2c(nn1CC)CCC2 Cc1cccc(C)c1C(N1CCC(CF)(NC(=O)CNS(C)(=O)=O)C1)=O n1(CC(=O)NC(CC(C)NC(=O)CC(O)CN(C)C)C)ccccc1=O CCCC(CC)CCC(=O)NC1CC(CO)N(C(=O)C(C)OCC(C)C)C1 n1(CC)cc(CC(=O)NCCc2n[nH]cc2C(=O)N(C)Cc2csnc2C)nn1 C(CN=c1ccc(C(=O)NCC2CN(C(C3CCCC3OC)=O)C2)c[nH]1)OC C1(NC(CCS(C)=O)=O)CCC2(CC1)CC(NC(C1(C(F)F)CC1)=O)C2 C(CNC(=O)Cn1cnc(=N)[nH]1)(C(=O)N1CC(SC)C1)OC C12(NC(c3ccnc(F)c3F)=O)CCCCCC1N(C(=O)Cn1ccnn1)CC2 C1(NC(C2(C)CC(=C)C2)=O)CC2(C1)CC(NC(=O)C(C)C1CCCO1)C2 C(=O)(CCS(N)(=O)=O)N1C(CC)C(C(=O)NCC2CSCCO2)CC1 C12(CNC(c3c(Cl)ccc(CC)c3)=O)CN(C(c3cnc(S)[nH]3)=O)CC1CCO2 C1(NC(C2N(C(=O)C=Cc3ccncc3)CCN(C)C2)=O)CCn2nccc2C1 Cn1c(O)nc2ccc(C(=O)NC(CNC(C3CC34CC(O)C4)=O)CO)cc12 C1(C(=O)NCC2(C)N(C(CCn3c(C)cc(C)n3)=O)CCC2)CC(C)CC(C)C1 Cc1ccc(-c2ccccc2)cc1C(=O)NCC(C)NC(=O)C(C)(C)C(C)O C1(C(N2CC(F)(CNC(c3ccc(F)c(F)c3)=O)C2)=O)C(F)(F)C12CCC2 C(=O)(C(F)(F)C(F)(F)F)N1CC(CN(C(=O)C=Cc2cc(F)cc(F)c2)C)C1 c1(C(N2C(C(C)NC(C3(c4ncco4)CCC3)=O)CCC2)=O)ccc(Cl)cc1O CN=c1[nH]cc(C(=O)NCCNC(=O)Cc2cccc(C(F)(F)F)c2)s1 CCCCC(O)C(=O)N1CC(F)(C(=O)NC(c2ccccc2F)C)C1 c1(C(=O)NCC(CN(C(C(C(C)C)n2ncc(N)n2)=O)C)C)cccc(=O)n1O c1(C(=O)NCC2C(NC(CCc3ccc(C)s3)=O)C2)ccc2oc(C)nc2c1 c1(NCCCC(CC)O)ccc(S(=O)(=O)NC2(C3CCCC3)CC2)cn1 C1(C(=O)NC2C(C)(CN(C(CCCC=C)=O)C)CCC2)CN2CCN1C(C)C2 C1(C)(C(=O)NCCCN(C(C)C)C(C2CCC3CC23)=O)CCOCC1 C1(C)(c2cccc(C(=O)NCCN(C(C(C)CF)=O)C)c2)NC(=O)NC1=O c1(C(N2C(CC(=O)NC3CNC(=O)N3)CCC2)=O)coc(-c2ccccc2)n1 c1(C(=O)OC)cncn1CC(=O)N(C)CC1CCCN1C(=O)C(C)OC N1(C(Cc2cn(CC)nc2)=O)CC2(CC2)CC1CNC(C1(CCOC)CCC1)=O C(=O)(CS(=O)(=O)CCO)NCC1C2CN(C(c3ccn(C)c3)=O)CC21 CC(C(=O)NC(C1CCN(C(C2(C#N)CCCCC2)=O)CC1)(C)C)C1=CCCC1 C=CCCC(C)(C)C(=O)NCC(C)N(C)C(c1ccc(-n2cncn2)cc1)=O CCC(CC(F)F)C(=O)N(C1CCN(C(=O)CCSCC(N)=O)C1)C C(=O)(CCCCC(=O)OC)NCCN(CC(C)O)C(C1(COC)CC12CCC2)=O C1(CCNC(c2ccnc(CNC(C3CCC4(CC4)C3)=O)c2)=O)CCCC2CC12 c1(CC)ccc(C(=O)NC2(C(=O)NCCC(=O)NO)CC2(C)C)cn1 c1(OCC)ccc(CNC(C2CCS(=O)(=O)CC2)(C)C)c(F)c1F N1(C(CCC2(CCC#C)N=N2)=O)CCCCC(CCCC)C1.C(=O)(C(C)(C)CO)N C(=O)(C1CCOc2ccc(Br)cc21)NC1CC(C)(NC(CCC#C)=O)C1 Cc1cnc(C(=O)NCC2CCCC(CNC(C3CC(C(F)(F)F)C3)=O)C2)cn1 c1(OCC#C)ccc(CNC2CC2C(=O)Nc2cnc(Cl)c(C)c2)cc1OC N1(C(c2cc(SC)oc2C)=O)CCCC(C)C1CNc1ncncc1I c1(NC(CNC(c2ccc(C)nn2)=O)C(C)C)cc2nnc(C)n2cn1 C(=O)(CC(C)CC(=O)N1CCC(C)C1CNC(C1CC2(CCCCC2)C1)=O)OC c12cc3cc(OC)c(OC)c(c3[nH]1)NC2=O.CCCCCCNS(=O)(=O)CC c1(C(=O)NC(C2CCN(C(=O)Cn3cccc3)CC2)C)c[nH]c2nccc-2c1 c1(C(N2CC(NC(=O)CCc3ncc[nH]3)C(F)CC2)=O)n[nH]c2ccccc12 c1(OC)ccc(CNc2cn(CCC3CCCO3)nn2)c(Br)n1 C1(COC)CC(CNC(c2cc(C(F)F)cs2)=O)N(C(c2cnc(O)n2C)=O)C1 C12(NC(CCc3ccc(C)o3)=O)CC1CN(C(=O)CC1CCOC1=O)C2 c1(CC(C(=O)NC(C)CNC(=O)CC2(O)CCC2)F)ccc([N+](=O)[O-])cc1 c1(C(=O)NCC(c2ccccn2)C)cccnc1CNC(=O)C(C)(C)CF C(CC(C)C)(C(=O)N1CC2CC1CN2C(C)C)NC(CC1CC(=C)C1)=O C1(CCNC(C(C)NC(CC)=O)=O)CC(OC)CN1C(c1nccnc1C)=O c1(C(=O)NC2CCC(CCNC(c3ccc(C)nn3)=O)C2)nn(C)cc1[N+](=O)[O-] N1(C(C)=O)CCN(C(=O)CC2(NC(=O)C(F)F)CCC2)C(C)C1 C(=O)(C1=CC2(CCOCC2)C1)NC1C(CNC(c2cn(CC)nc2)=O)CCCC1 c1(C2C(C(N(CCCN(C)C(c3csnn3)=O)C)=O)C2)ccn(C)n1 c1(C(=O)NC2C(CNC(C=CS(C)=O)=O)CC2)nnc2ccccc2n1 C1(NC(C(CSC)(C)NC(c2ccnc(O)c2F)=O)=O)CCC2CCCC1O2 C=CCC(C(=O)N(CC(=O)NOCC1CCCC1)CCOC)OC Cc1ccc(C)c(C(=O)NCC2CC(NC(C3(C)CCCS3)=O)C2)c1N C(=O)(C(C)(C)CS(C)(=O)=O)N(C1CN(C(=O)C(CO)NC(N)=O)C1)C c1(C(=O)NC2C(NC(c3ncn(C(C)(C)C)c3)=O)CCC2)ccc(Cl)c(Cl)c1O Cc1sc2nc(CN=c3[nH]c(NCCN(C)CCO)nc(=N)[nH]3)nc(O)c2c1C C(CC(C)(C)C)(C(=O)NCCCC1(NC(C2(O)CCCCC2)=O)CC1)OC Cc1ccc(C(=O)NCCCN(C(=O)Cn2cc(C3CCOC3)cn2)C)s1 C1(OC)CC(C(=O)NCc2ccc(O)cc2)N(C(c2ccc(F)cc2)=O)C1 c1(C(=O)NCC(CNC(=O)CCc2cnc[nH]2)CO)cccc2cncn12 c1(OCCC(=O)NC(C(CO)NC(CC(C)(C)O)=O)C)cc(F)cc(F)c1 C(CCC(=O)NCC(C(C)C)NC(C1(C(=O)N(C)C(C)C)CC1)=O)=CC c1(C(=O)NCC2(C)CCN(C(CCOCC)=O)C2)cc(C)cnc1C C1(C(=O)NC2CC2)CCCCN(C(C2CCCN(Cc3cc[nH]n3)C2)=O)C1 CC(C)CCCC(=O)NCC1CC1NC(=O)C(CC(F)F)C1CCC1 c1(C(=O)OC)cnc(C(=O)N(CC(C)NC(=O)CC2CCC(C)C2)C)cn1 CON(CCC(=O)NCCCN1CC=CC1)C(=O)C1CCN(C)C1 N1(C(CC2C(C)CCCC2)=O)CCC2(NC(C3CCCC(=O)N3)=O)CCCC12 c1(C(=O)NCC2C(C(=O)NCc3nc(CC)sc3)CCC2)ccc(C#N)s1 C1(NC(=O)CCC2CC2(Cl)Cl)Cc2ccccc2N(C(c2ccc(Cl)nc2)=O)C1 C(=O)(CCCC(=O)N1CC2(CO)CC1(C(N1CCC1C(=O)NC)=O)C2)OCC N1(CCN(C2CCCC(CC(F)(F)F)C2)CC(=O)OC)CCN(C)CC1CO N1(C(C2(CCNC(COC)=O)CC2)=O)CCCC2CN(C(C)=O)CC12 N1(C(C2N(C)CC2)=O)CCCN(C(C2CC(=C3CC3)C2)=O)C(c2ccccc2)C1 N(C1CN(C(C2CC(C)C2)=O)Cc2ccccc21)C(c1ncccc1C(C)=O)=O Cc1cc(N2CC(CCO)OC(C)(C)C2)nc(=NC(C)CC(C)(C)C)[nH]1 c1(C(=O)NC(CC(C)NC(C(C)(C)OCC)=O)C)cc(N)c(C)c(N)c1 C1(NC(CC=C(C)C)=O)C=CCC(C(=O)NCC2(F)CCOCC2)C1 N1(C(c2c(C)nns2)=O)CCC(C)C(CC(=O)N(C2CC(O)C2)C)C1 N1(C(C(C)=O)Cc2cc(C)ccn2)CCC(N2CCOC2=O)CC1 C1(CNC(CC=C)=O)CN(C(=O)CCC(C)N(C)C)CC1(C)C c1(OC)cc(C(=O)NCCNC(=O)C#CC(C)(C)C(C)(C)C)c([N+](=O)[O-])cc1OC c1(C(=O)NC2CN(c3nccc(C(C)C)n3)CC2O)ccc([N+](=O)[O-])nc1 N1(C(C(c2cccnc2)OC)=O)C2CCC1C(NC(=O)C=CC(C)C)C2 C12(NCC3CCN(C(C)=O)C3)CCC(n3cc(C(=O)NC4CN(C)C4)nn3)(CC1)C2 CC1(CNCC(O)CNC(=O)CCN)CCC1 c1(-n2cc(C3N(C(C4CCCC=C4Br)=O)CCOC3)nn2)ccc(F)c([N+](=O)[O-])c1 c1(C(N2CC(NC(=O)C#CC3(C)CC3)CC(OC)C2)=O)cc(N)c(F)cc1F C12(C(N(CCCO)C(C)C)=O)CCC(NS(=O)(=O)c3cccnc3)(CC1)CC2 CCC(C(=O)NCCN(CC(C)O)C(c1n[nH]cc1C(=O)OC1CC1)=O)OC C#Cc1ccc(C#N)c(NC(=O)NC(c2cnnn2C)CC)c1 CN=c1nc(N2CCc3c(nnn3C)C2)[nH]c(=NC2CCN(CC(F)F)C2)[nH]1 C1(N(C)C(C2CC(CNC(C3(CCCF)CC3)=O)C2)=O)CCCC1C#N c1(C(N2C(C(=O)NCCOCCCC)CCC2)=O)noc(C)c1C c12cnccc1SC2=O.N1(CC=C(C)C)CCC(C2CC(N)C2)C1 C=CCCCCCCC(=O)NCC(CC(=O)NC(C)CCOC)C1CCC1 C1(C(N2CCC(SC)CC2)=O)C2CC(O)C(C2)N1C(=O)C(C)C1(O)CCC1 CC(CCNC(=O)CCCSC(C)(C)C)N=c1[nH]c(C2CC2)nc(=N)[nH]1 Cc1ccc(NCC(=O)NC(C)CC(C)NC(c2cnn(C)c2)=O)c(C)c1 CC(O)C(C)(C)C(=O)N1CC=CC(NC(=O)CCC2CCCCO2)C1 Cc1c(N(C)Cc2cn(C(C)C(N3CCCOCC3)=O)nn2)cnn1C(C)(C)C C1(CC(=O)NCc2ncn(CC)n2)CC(NC(=O)C(C)C)C1(C)C C#CC(C)(C)C(=O)NCC1CCCN1C(c1n[nH]cc1-c1ccccc1)=O C=C=CC(C)C(=O)NC1(C(=O)NCC23CC(F)(C2)C3)CC1(C)C c1(OC(C)C)ccc(C(=O)NCC2CC(NC(=O)C(O)CC3CCCC3)C2)nn1 c1(C(N2CCC(C)(NC(C3CNC(=O)C3)=O)C2)=O)cc(Br)cc2c1CCN2 c1(N2CC(C)=C(C)CC2)nc(N(CC2=CCCOC2)C)c2c(n1)CCC(C)C2 C(C(C(C)C)N(C)C)NC(CCOCCOCC)=O.C(=O)(CCCOC(=O)O)N N1(C(c2cc(C)cc(C(N)=O)c2)=O)CC2CCC(CNC(c3cccs3)=O)C2C1 N1(C(CNC(C(N2CCOCC2)C)=O)C(F)F)CCN(C(c2ccccc2)=O)CC1 C1(CNC(C2C(C(N)=O)C2)=O)CN(C(=O)C=Cc2ccsc2Br)CCO1 C1(NC(=O)NCCN(CC2(n3cncn3)CC2)CC)CCCCC1n1cccn1 c1(COC)ccc(Cc2cc(Nc3ccc(-c4nn[nH]n4)c(C)c3)ncn2)c(F)c1 Cc1coc(C2CC2)c1C(N1CC=CC(NC(=O)CCCSC(C)(C)C)C1)=O N1(C(c2ccc(CC)o2)=O)CC23CCCC2(C1)CN(C(c1cc(C#N)no1)=O)C3 C(CCCCCNC(=O)CCOC1CC1)N(C)C(C1CC2C=CC1C2)=O C(=O)(CCC(C)(C)OC)N1CC(O)(CCNC(c2c(OC)nsc2)=O)C1 C1(C(=O)NC(C)C(O)C(F)F)(CNC(C(CO)OC)=O)CC2(CC2)C1 c1(NC(C(c2ccc(F)cc2)(C)O)=O)cnc2n[nH]c(Br)c2c1 c1(OC)nccc(C(=O)NCc2cc(C(=O)NC(C)C(C)n3cncn3)n(C)n2)n1 c1(CC)cc(C(=O)NCC(c2ccc(N)cc2)O)n(-c2ccccc2)n1 c1(SC)ccc(OCC(=O)N(CCCCCNC(c2cc(C(N)=O)c[nH]2)=O)C)cc1 N1(C(c2c(OC)csc2)=O)CCCC(C(=O)NCc2cn(C3CC3)nn2)C1 Cc1cc(OCCC(N2CCCC(NC(=O)C#CC(=O)O)C2)=O)cc(C)c1 Cc1ccc(C(N2CCCCCC2CNC(=O)C(F)CC2CC2)=O)cc1F CCC(C)C(O)C(=O)N(C)CC1CCN(C(c2ccc(-n3ccnn3)cc2)=O)C1 N1(C(c2n(C)cnc2)=O)CC2(CCC2NC(C2CC23CC(C)(C)C3)=O)C1 C1(NC(C2CC(CC)C2)=O)CCC(O)CN(C(=O)CC=Cc2ccccc2)C1 C1(NC(COCCC#C)=O)(CNC(C2(C(N)=O)CC2)=O)CC2CCC1CC2 C(=O)(C1CCc2nccn21)NCC1(O)CCCN(C(CNC(N)=O)=O)CC1 C1(C(N(C2CCN(C(C3(C)CCCCO3)=O)CC2)CC)=O)CCn2nncc2C1 C(=O)(C1CCCn2c(C)cnc21)NC(CNC(c1cccc(SCCC)c1)=O)C c1(C(=O)NCC(C2CCC2)NC(c2c(C)c[nH]n2)=O)cc2ncccc2[nH]1 CCCC(C)CC(=O)NCCCCC(CO)NC(=O)Cc1cncnc1 c1(OC)cc(C(N2CCC(C)(NC(=O)COCC3CC3)CC2)=O)cc(F)c1 Cc1c(Cl)cnn1CC(=O)NCC1CCCC1NC(c1ccccc1C(C)O)=O C1(CNC(C(C)(C)N(C)C)=O)CC2CCC(C1)N2C(C12CCC1C2)=O c1(C(=O)NCC(C2CC2)NC(c2n(C)c(Cl)c(Cl)c2)=O)c(F)ccc(Cl)c1N C1(C)(C(=O)NC2CC(N(C(=O)CCC3CCCC3)C)C2)CCOCC1 CCC(C)(CCC(C)C)C(=O)NC1CC1NC(=O)C(C)(C)c1cnco1 n1(C(C(C)C)Cc2ccccc2)nc(-c2nc[nH]n2)nc1-c1cc(Br)cn1C CS(=O)(=O)C(CNC(c1ccc(C#N)cn1)=O)CNC(C12CCCN1CCC2)=O c1(C(N(C)CC2(CNC(C(CCC)C(C)C)=O)CC2)=O)cnc2c(ccn2C)c1 c1(OC)cc(N(C)CC2CCCN2C(C2CC2(C)C(C)C)=O)nc(OC)n1 C(=O)(C(F)C(F)(F)F)NC(CCSCC)C(=O)NC1CCCC1C1CC1 Cc1cc(CC(=O)N(CCCNC(=O)C(C)c2ncco2)C)n[nH]1 c1(C(=O)NCC=CCNC(C(N=S(C)(C)=O)=O)=O)c(Br)ccc2n[nH]cc12 C1(Cn2cc(C(COC)(C)O)nn2)CN(C(c2sc(C)nc2Br)=O)CCO1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC(C)CNC(c1ccc(C(C)(C)C)cc1)=O c1(COC)nc2cc(-c3ccnc(OCCOC(C)C)c3)ccc2o1 C(=O)(C#CC1(C)CCCO1)N1CC(O)(CNC(CN(C)C(c2cccs2)=O)=O)C1 Cn1cc(C(=O)NC2CN(C(=O)CC3CCOC3)C(C)(C)C2)c2cc(F)ccc12 C1(C)(COC)C=CCN1C(=O)C(C)(C1CCC1)NC(c1cccc(CC#N)c1)=O c1(CN(c2ccnc(C3(N)CCC3)n2)CC2CC2)ccc(F)c(F)c1 C(=O)(C1=NOC(C)C1C)NCC(C(C)C)NC(c1c(OC)ccnc1O)=O Cc1csc2cc(C(=O)NC3CC4CN(C(c5ccnnc5O)=O)CC4C3)[nH]c12 CCC(COC)C(=O)NC(CC1CC1)CC(=O)N(CC(C)OC)C N1(C(C23COC(CF)(C2)C3)=O)CCC2(CC1)CC2NCC1CC12CCOCC2 CC1CC(NC(C2CCOC2=O)=O)CCN1C(c1ccc(CN=[N+]=[N-])cc1)=O N1(C(C(CSC)C)=O)CC(O)CC1CC(=O)NC1(CC2CC2)CC1 C12(C(=O)NCCS(C)(=O)=O)CC(CCO1)N(C(C1CCCC(=O)N1)=O)C2 N1(C(c2cc(CCC)[nH]n2)=O)CCC2CCN(C(=O)CSC(F)F)C2C1 C(=O)(C(C)C(C)(C)C)NCC1(O)CCN(C(c2c(SC)snn2)=O)C1 C12CCCCN1C(=O)C(C)S2.C(C(F)(F)F)OCC(C)N(CCCC)C c1(C(=O)NCC(C(C)O)C)cccc(CNC(=O)CC(=O)NC(C)(C)C)c1 C1(C(=O)NC(C2OCCN(C(Cn3c(C)nnn3)=O)C2)C)CC2CC2CC1C C(CC(N)=O)(C(=O)NCCN1CCC(O)CC1)NC(c1c(CC)nc(C)o1)=O CC1CCN(C(c2occc2CNC(c2ccc[n+]([O-])c2)=O)=O)C1CO C1(NC(C(=O)NCC)=O)CCOC2(CCN(C(=O)C#CC3(C)CC3)CC2)C1 C1(NC(c2c(C(C)(F)F)cccc2)=O)CCN(C(c2ccc(O)nc2)=O)CC1F C12(C(=O)NC3CN(C(Cn4c(C)ncc4)=O)CC3C)CCC(N(C)C)(CC1)CC2 C(=O)(C(C)C(C)C)NC(C(CO)NC(C1CC(OC)(OC)C1)=O)C C(=O)(C(C)C1=CCCC1)N1C2CC(CNC(c3c(N)ccc(C)c3)=O)C1CC2 CC1=C(C(=O)N2CCN(C3CCN(C(C4CCOC(C)(C)C4)=O)C3)CC2)CCC1 c1(C2(CC(=O)NCCN(C)C(C34COCC3C4)=O)CC2)ccccc1 C1(NC(CNc2cccc(C(N)=O)c2)=O)C2Cc3ccccc3C12 N1(C(=O)OC)CC(C)(OCC2CC(C(F)(F)F)(OCC(=O)OC(C)(C)C)C2)C1 N1(C(C(C)OC2CCOC2)=O)CC2(CCC2)CC1C(=O)NC1(N2CCOCC2)CC1 CCC1=NOC(C(=O)NCC(C(C)C)NC(=O)CCc2cnc(O)[nH]2)C1 N1(C(c2n(CC)ccn2)=O)CCC2CCC(C1)N2C(c1coc(C#N)c1)=O CC1CN(C(c2ncccc2N)=O)CC1C(N1CCC(CF)C1)=O N1(C(C2(OCC)COC2)=O)CC(C(=O)NOC2CCC2)C(C2CC2)C1 O=C(CC1=CCCCC1)NC1(c2ccccc2)CCCNCC1 C12(C(=O)NCCN(C(=O)Cn3nnc(=N)[nH]3)CCOC)CC1COC2(C)C C1(C(=O)NCCCNC(COCCC=C)=O)(C(=O)OC(C)(C)C)CC2CCC1C2 C1(NC(Cc2ccc(C)s2)=O)COC2(C1)CN(C(=O)CCCc1n[nH]c(=N)s1)C2 CC(F)(F)CCC(=O)NC1CCC(NC(C2CCOC2c2nccn2C)=O)CC1 C(=O)(C1CCCc2nc(C)[nH]c21)N1CCCC(CN(C(COCCC)=O)C)CC1 C(=O)(C1Cc2cccc(Cl)c21)NCCCNC(Cc1ccn(C(C)C)n1)=O N1(C(CN(C(=O)C(O)Cn2cncn2)CC#C)=O)CCc2nocc2C1 c1(C(=O)NC2(C)CN(C(C3CC(Cl)(Cl)C3)=O)C2)cnc(S(C)(=O)=O)s1 CC(C)(C)CC(O)CC(=O)N1CCCC(C)(NC(=O)CCOCC(F)(F)F)C1 c1(C(N2CCCC(CNC(c3[nH]c(CC)c(Cl)n3)=O)C2)=O)cc(C)c(F)c(C)c1 C1(C(=O)NC2C3(CN(C(C45CC(C)(C4)C5)=O)C3)CC2)CC(c2ccccc2)=NO1 Cc1cc(C(=O)N(CC(C)(C)CNC(C2CC(N3CCCC3)C2)=O)C)ncc1N C12CCN(CC1)C2.c1(NC(=O)NCC2(c3cc[nH]n3)CC2)ccnc(C(F)F)c1 C1(CC(N2CC(C)C2)=O)CN(C(=O)Nc2cncc(F)c2)CCO1 N1(C(Cc2c(C)non2)=O)CCCC2CN(C(=O)CC3CSCCO3)CCC12 CC(C)C(O)C(C)(C)C(=O)N1CCC(NC(C2CCC(N(C)C)CC2)=O)C(O)C1 c1(C(=O)OC)c2cccc1NC(=O)CNC(=O)O2.c1(OC)cc(Br)cnc1C CC(C)C(C)(CNC(=O)C(C)NS(C)(=O)=O)NC(=O)CSc1nnc(S)s1 C(=O)(NN1Cc2ccc(Br)cc2C1=O)c1c(C(F)(F)F)ccc(C#C)c1 c1(CN=C(NCC(CC)(C)C)NC2CC2C)cccc(C)c1O CC(Cc1cccnc1)N=c1[nH]c(=NCC2CCCCN2C)c2ncccc2[nH]1 C(=O)(CCCCCCCS(C)(=O)=O)N1C(CN(C(=O)C=CC2CCC2)C)CCC1 C1(C(=O)OC)CC(c2ccccc2)CN(C(=O)NC2CC2c2cnn(C)c2C)C1 C(CCNC(C1CC1c1ccccc1F)=O)(C(C)C)NC(C(COC)C)=O c1(CC)cc(C(=O)N(C)CCNC(C2CC3C=CC2C3)=O)cc(C)c1 C1(C(=O)NC2CCC(CNC(c3ccnc(CO)c3)=O)CC2)SC2C=CC1CC2 CC1C(NC(=O)CSC(F)(F)F)C(C)CCN1C(=O)CC1CC1(Cl)Cl C(=O)(CCCCCN(C(=O)C(c1ccccc1)F)C)NCc1n(CCC)ncn1 CC(C)(C)C(O)C(=O)NC1COCC1CNC(c1cnn(C2CCC2)c1)=O N1(C(C(C)NC(N)=O)=O)CC2(C1)CN(C(=O)CC(O)C1CCCC1)CC2CO Cn1c(NC(N2CCN(S(C)(=O)=O)CC2)=O)nc2cccc(Cl)c12 N1(C(C(C)c2cccs2)=O)CCN(C(c2nccn2C)=O)CC1c1cccnc1 c1(C(=O)NCCC2C(C)CN(C(c3ccc(O)nc3)=O)C2)c(F)cncc1Cl C1(CN(C(c2cnc(C(C)O)s2)C(=O)NCC=C)CCC#C)CCS(=O)(=O)C1 C(CCCCCCCO)=CC(=O)NCC1CN(C(c2cc(NC)nc(Cl)c2)=O)C1 c1(OCC)ccnc(NCCC2CCCCN2C(c2cc(C(C)C)oc2C)=O)n1 CC(C)(C(=O)NC1CC1NC(=O)CC1CCC(C2CC2)O1)n1cc(Br)cn1 N1(C(C(C)NC(CC)(C)C)=O)CCC(O)(C(C)NC(=O)CCCn2ccnn2)C1 C1(NC(=O)OC(C)(C)C)CC2CCC(C1)N2.C12CC(O)C1CC(=O)N2 C1(CCC(=O)NCc2ccncn2)CC(C)(C)CO1.C1(N(C(=O)C)C)CC(O)(C)C1 Cc1cccc(C)c1S(=O)(=O)N(C1CS(=O)(=O)CC1O)C N1(C(c2ccc(CCCCC)o2)=O)CCCCCC(NC(=O)COCCSC)C1 c1(C(=O)NC2CC(CC(=O)NCC3(C)CCCCC3)C2)cnc(O)c(Br)c1 Cn1cc(NC(C2CC(NC(c3cc(Cl)cn3C)=O)C2(C)C)=O)c(C#N)n1 C(=O)(C1=NOC(C)(C)C1)NCCOCC(N1C(C)CCCC1C)=O Cn1c(C(N2CC3CC3(NC(c3cccc(C(F)F)c3)=O)C2)=O)cnc1[N+](=O)[O-] c1(COC)cccnc1C(N1CCC(C(C)C(=O)NCCC2CC2)CC1)=O C(=O)(C1(C)CCn2ccnc21)NCC(C)(C1CC1)NC(=O)Cn1cc(CO)nn1 c1(C(=O)NCC(CNC(CCCCC)=O)OC)ccc2cnc(C)cc2c1 C1(NC(CSCC(C)C)=O)C=CCN(C(c2coc(Cn3cccn3)c2)=O)C1 c1(C(N2C3CC(NC(C4CC4F)=O)(C3)C2)=O)ccc(-c2ccncc2)c(F)c1 N1(C(C(C)OCCOC)=O)CCN(C(c2cnn(C(C)(C)C)c2N)=O)C(C)C1 N1(C(Cc2c(C)ocn2)=O)CC2CCC(C1)N2C(=O)CCN1CCCS1(=O)=O c1(C(=O)NCCCCN(CCCNC(C(C2CC2)OCC)=O)C)ccc(C)nn1 C1(C(=O)NC(CC=CC)C(=O)N2CCCC2CNC(N)=O)CCOCC1(C)C N1(c2snc(CCOC)n2)CC2(C1)SCCC2NC(=O)C1=CCOCC1 Cc1ccc2cc(C(N3CCN(C(=O)CC(O)C(C)C)CC3CF)=O)cnc2c1 N1(C(Cc2n[nH]c(=NC)s2)=O)C2CCC1CC(N(C(=O)Cc1cnsc1)C)C2 c1(C(N2C(CNC(C3(C)CCCO3)=O)CC2)=O)cn(CC#N)c2ccccc12 C1(CNC(C2(CC(C)C)CCC2)=O)C2CN(C(=O)C(C)(C)c3cnsc3)CC12 c1(N2C(C(=O)NC3(C4C(=O)NCC4)CC3)CCC2)ncc([N+](=O)[O-])cc1Br c1(C(N2C(CNC(C(CSC)O)=O)CCC2)=O)cc(N)c(F)c(F)c1F N1(C(C2(C3CCCO3)CCC2)=O)CCCC1C(=O)NCC.C12COCC1CN2 CCN=C(NC1C2CN(C(C3CCC3)=O)CC12)N1CCC(C)(F)C1.C(C)(C)(C)N C(=O)(C(F)(F)C(O)c1ccccc1)NCC1N(C(C(C)C)=O)CC(O)C1 CN1CCOC(C(=O)NC2CCN(CCNC(C34CCC(CC3)O4)=O)CC2)C1=O N1(C(C2CC(OC)C2)C(=O)NCCSC)CCc2ccc(O)cc2C1 c1(CC)cc(C(N2CC(CNC(C3SCCS3)=O)(COC)C2)=O)ns1 n1(CC)nc(C(C)C)cc1C(=O)NC1CCN(C2CNC2)C1=O CCC(C)CC(=O)NC(C)(C(=O)NCC1CC[Si](C)(C)C1)C1CCC1 C1(C(N(C(CO)CO)C)=O)CCCN(C(=O)C(c2ccccc2)O)CC1 C1(NC(C2N(CC)CC2)=O)CN(C(=O)CCCc2nnc(C)n2C)CC1C(F)F N1(C(C(CCC)NC(N)=O)=O)CC2CC(C1)N(C(c1cc(C)nc(Cl)c1)=O)C2 N1(C(CNc2cc(C#C)nn2C)=O)CCOCC(C)(C)C1 CCC(C)CCCCC(=O)N1CC2(CCCN(C(=O)CC(C)(O)COC)C2)C1 CCC(O)C(C)C(=O)NCC1(C)CCN(C(=O)CCc2cc(Br)cs2)C1 c1(CC(=O)NCC2N(C(c3n(CC)ccc3)=O)CCOC2)cc(O)nnc1O N1(C(C2(CC)CCN(C(C(CCC)N(C)C)=O)C2)=O)CCN2CC(O)CC2C1 C(CC(C)C(=O)NC(c1nocc1C(=O)NCCC(C)O)C)=CCC CCC(CNC(=O)COC1CCN(C(=O)CCCCNC(N)=O)C1)CC(C)C CCCCCCC(C)CC(=O)NCc1csc(CNC(=O)C=CSC)n1 c1(C(N2C(CN(C)C(C34COCC3C4)=O)CCC2)=O)cc(=N)[nH]c(Cl)n1 C(=O)(C(C)(C)C(c1nnnn1CCCF)NC1CCCC1CF)OC c1(OC)cc(C)c2cc(C(=O)N(CCNC(C3CCS3(=O)=O)=O)C(C)C)oc2c1 C1(NC(C(C)C#N)=O)CC2CCC1(C(=O)NC1CCC(C(C)O)CC1)C2 N1(C(C(CC=CC)C)=O)CCCC(N(C(=O)CNC(=O)CCC)C)CC1 c1(OC)c(C(=O)NC(C)CC2CCN(C(=O)CC(C)C)CC2)cccc1C CC(C)C(C#N)C(=O)NC(Cc1cnn(C)c1O)C(N1CCOCC(O)C1)=O CC1OCCN(C2CCN(C3CCNCC3)C2=O)C1(C)C C1(C(=O)NCCNC(C(C)OCC2CC2)=O)(Cc2cnn[nH]2)CCOCC1 N1(C(C2ON=C(C)C2c2ccccc2)=O)CCCC(NC(=O)C(C)C)CC1 C(=O)(N1CCC(C(=O)NC2(C)CCSC2)O1)C1(CC)CC1 n1(CC)c(C(=O)NCC2CCCN(C(c3ccncc3Cl)=O)C2)cnc1O c1(C(=O)NC2(CF)CCN(C(=O)C3CC3)C2)ccc2c(c1)CCOC2 N1(C(CC(C(C)C)C)=O)CCC2(CC1)CCN(C(c1cc(Cl)c([N+](=O)[O-])[nH]1)=O)C2 c1(CNC2(SCC)CCC2)nncn1C CCCCC(C)C(=O)NC1CC(C)(CNC(C2(C)CS(=O)(=O)C2)=O)C1 N1(CCOc2ccc(CCC(=O)NCCC=CC=C)o2)CCCC(C)(OC)C1 N1(C(C(C)C2CCOC2)=O)CC2CCCC1C2CNC(=O)CN(C)C(=O)C1CC1 C(C)(C(C(C)C)NC(c1ncoc1CC)=O)NC(c1c(CC)con1)=O O=C(N1CC(c2cn(C3CCCC3)nn2)CO1)c1cc(-n2ccnc2)[nH]n1 CC(C)CC(S(=O)(=O)Oc1cncc(NS(C)(=O)=O)c1)c1ccc(F)cc1 CC(C)C(C(=O)NC1(CNC(C23CCCC2(C(N)=O)C3)=O)CC1)NC(N)=O C12(C(N(C(CNC(C(c3c(C)cccc3)C)=O)C)C)=O)COC(CCO1)C2 CC1CC(NC(=O)C=Cc2ncc[nH]2)CN(C(=O)CC(C)(C)C)C1 C(C)(C)(CCCCNC(=O)C(C)=CC1CC1)NC(c1nc(CCC)sc1)=O C1(C(=O)NC2(CNC(CCC(C)N(C)C)=O)CC2)CCCCCS1(=O)=O C1(F)(CNC(=O)C=Cc2cnccn2)CCCN(C(=O)C(O)C(F)(F)F)CC1 N1(C(c2c(C)nsc2)=O)CCC(CCC(=O)NCCOC2CCC2)CC1 C(c1cnn(C)c1C)=CC(=O)NC1C(NC(c2ccc(COC)cc2)=O)CC1 c1(CNc2ccc(N(CCCO)CC)cc2)cccc(OC(F)(F)F)c1Cl C(=O)(C(CNC(=O)C(F)C(C)(C)O)C(C)C)NCC1(CCC=C)CC1 C1(CNC(Cc2c(SC)cccc2)=O)CC2(CO1)CN(C(C1CCCOC1)=O)C2 N1(C(CNC(c2ccc(C(=O)NC)nc2)=O)=O)CCN(C(=O)C(C)O)CC(C)(F)C1 C(CCC(C)(C)C(=O)NCCc1nc(C)no1)NC(c1ncn(CC)n1)=O c1(CNC(CN(CCCCCC)C)=O)cc(O)nc(CNC(=O)C(C)C(C)C)n1 c1(OCC)nc(C(=O)N(C(C)CCNC(C2CCCCS2)=O)C)ns1 c1(C(=O)NCC(CNC(CCSCCC)=O)C)cncc2[nH]ccc12 C#CC1(NC(C2(CNC(C3CC(C)CCO3)=O)CCC2)=O)CCC(C)CC1 C1(CNC(c2csnn2)=O)CC(O)CN1C(=O)C1=CCCS1 C1(c2nc(C3ON=C(C(C)(C)C)C3)on2)CCc2nnnn2CC1 c1(C(=O)NCCC2(NC(C(COC)C)=O)CCC2)c(Br)cnn1C c1(C(N2CCC(CN(C)C(C3CC3(Cl)Cl)=O)C2)=O)ncncc1N Cc1cc(F)ncc1NC(=O)N(CCC(N)=O)CCO.C1CN1 C1(CC(=O)NC(CCC=C)C)N(C(c2cc(CC)ncn2)=O)CCC1(C)C c1(C(N2CCCC(N(CCC)CCO)C2)=O)c(C)sc(C)c1C CC12C3C4C1C1C2C3C41C(=O)NC1CCC(NC(c2cc[nH]c2)=O)C1 N1(C(CNC(=O)OC)=O)CC(F)CC1CNC(=O)CCC1CCCOC1 C1(NC(C(C)N(C(CC2C(C)C(=O)CC2)=O)C)=O)CC(=O)N(C)C1=O Cc1sc(S(N)(=O)=O)cc1C(=O)NC1CCCCC1NC(=O)C(C)c1cc[nH]n1 C(CCCC(=O)N1CCC(C)CC1CNC(c1cc(Cl)cn1C)=O)(OC)OC N1(C(C#CC(=O)N(C)C)=O)CC2(CCN(C(=O)CCCCC3CC3)C2)C1 Cc1cc(=NCC2CCN2C2CCCCC2)[nH]c(=NCC2(CC3CC3)CC2)[nH]1 c1(C(=O)NC2CCC(NC(c3cnc(C)s3)=O)C2)ccc(N2N=CCC2=O)cc1 Cc1cc(F)cc(C(N2CCCC(CNC(C3(O)CC3)=O)C2)=O)c1N O=C(CC(O)c1cnc[nH]1)N1CCCC1c1cn(CCc2ccccn2)nn1 CC1OCCCC1C(=O)NCCN(C(=O)C=C(Cl)Cl)C1CC1 c1(C(N(C)CCN(C)C(C2(C3CCC3)CCC2)=O)=O)nnn2c1CSCC2 C1(CC)CN(C(C2(S(C)(=O)=O)CCC2)=O)CCC1NC(=O)CSc1cnn(C)c1 CC(C)C.C1(C)(CNC(=O)CNS(C)(=O)=O)C(=O)N1 c1(NC(c2c(NCc3scc(C)n3)cnc(F)c2)=O)ccc2ccccc2n1 CC1(CCO)CCN(C(=O)CC2CCN(C(=O)Cc3cscn3)CC2)CC1 C1(CNC(c2n(CC(=C)C)nnn2)c2sccc2Br)CCC2(CC2)C1 C1(CC)CCOCCN1C(=O)CCCC1(NC(c2ccc(C#N)cn2)=O)CCC1 C(C(CNC(C1(C)CC1(Cl)Cl)=O)S(C)(=O)=O)NC(c1c(CC)n(C)nn1)=O N1(C(C(F)=C(C)C)=O)CCN(C(=O)CCc2ccc(F)cc2F)C(C2CC2)C1 c1(OCC)ccnc2sc(C(=O)NCC34CCCC(CO)(CO3)C4)cc12 c1(NC(CC)CO)ccc(NC(=O)C(=O)N(C(c2cccnc2)C(C)C)C)cc1 C12(C(=O)NCCC(C)NC(CCSC)=O)CC3CC(C1)C(F)(F)C(C3)C2 c1(OC)ccc2cccc(NC(=O)NCC(c3ccccc3C)C)c2c1 C1(CNC(CCCOCC)=O)CN(C(=O)C(c2ccccc2F)F)CCC1(C)C CC(C(=O)N1CCC(OCCNC(=O)C(c2cccnc2)C)CC1)C(F)F C(=O)(N=c1ccn(C2CN(C(C3(Nc4c(CC)noc4)CCOC3)=O)C2)[nH]1)OC Cc1cccc(C(C(=O)NCC(F)F)N(C)CC2COCCO2)c1F C1(C(=O)NCC(C)(Cn2cccn2)NC(c2ccccc2)=O)CN2CCN1CC2 C(=O)(CC(CC(C)C)NC(=O)CSC(F)(F)F)NC(CC=C)(C)C(F)F N1(C(c2snc(OC)c2Br)=O)CCC2CN(C(=O)CO)C2C1 N1(C(CC=CC=C)=O)CC2CCOCC2(NC(=O)COCc2cccc(Cl)c2)C1 CCC(CCC(=O)NC(C)(C)CN1CCN(C(=O)Cc2cc(C)ns2)CC1)OC c1(C(N2CC(CC=C)(NC(=O)CCCc3cccs3)C2)=O)c(C)ncn1O N1(C(C(CSC)C)=O)CCOC2(CCN(C(=O)CCC3CCC(=O)N3)C2)C1 C(=O)(N1OC2CCC1CC2)C1N(C(C(C=C)CC)=O)CCCC1CC c1(CC(N2CCC(N(C(C=CCCCCC)=O)C)C2)=O)ccc(Br)c(F)c1 C(CCC1CCC1)(C(=O)N(C1CCC1C)C)NC(COC)=O C(=O)(CC(CN(C)C)CC)N(C1CN(C(C(CC)=CCCC)=O)C1)C C1(CN(C)C(C2CC2[N+](=O)[O-])=O)C2CN(C(=O)Cc3nccn3C)CC12 c1(C(N2CC(F)(C(=O)NCC3CC(C(=O)OC)C3)C2)=O)c(C)cccc1Br N1(C(c2c(CC)con2)=O)CC(CCNC(c2c(C)noc2C)=O)C(C)C1 N1(C(c2cn(C)nc2)=O)CCOCC1CCNC(=O)CC1CCCCC1O c1(C(=O)NC(C(=O)NCCCC(=C)Cl)CCc2nn[nH]n2)cc(C)n(C)c1C C1(C(C(=O)NC2C(NC(=O)CCCN3CCCC3)C2)O)CCCCCCC1 Cc1cc(=NCC2CC2(C)C)[nH]c(N2CCOC(c3cccc(OC)c3)C2)n1 c1(C(N2CC(CC(C)NC(c3c(CC)c[nH]c3)=O)C2)=O)cnn(C)c1Cl N1(C(C(COC)C)=O)CC2CCCC(C(N3CCC(C)C(CO)C3)=O)C2C1 C1(CC(C)=O)CCCCN1CCc1cccc(I)c1 c1(C(N(C)CC2CCCN(C(C3C(=C)C3)=O)C2)=O)sc(C#N)cc1Cl C(=O)(CC(N)C(C)(C)C)N1CCC(C(=O)OCC)(NC)CC1 C(=O)(C1Cc2ccccc21)NC12CCC(C(N3C(CN=[N+]=[N-])CCC3)=O)(CC1)C2 C1(NC(=O)Cc2csc(Cl)c2)CCCC2CN(C(=O)C(Cl)=CCl)CC12 N1(C(CCC(=O)NCC)=O)CC(C)CN(C(c2conc2C2CCC2)=O)CC1C c1(CNC(C2(C)CN(Cc3ccc(OC(C)=O)cc3)C2)=O)cc(F)c(F)c(F)c1 Cc1nc(=N)[nH]cc1C(=O)NCCC(C)CCNC(=O)CC1(CO)CC1 C1(NCc2n(C)c(Cl)cn2)CC12CCC(C(=O)OC(C)(C)C)CC2 CCCCC(CNC(=O)CCc1ncccc1C)NC(C1CC2(CC2)CO1)=O C(=O)(C(C)(C)C(=O)NC(C)CNC(c1sccc1C)=O)OC c1(C(N2CC3N(C(CC#N)=O)C(CC3)C2)=O)noc2cc(F)ccc12 C(=O)(CCCS(C)(=O)=O)NC(C)CCNC(c1cn(C2CCC2O)nn1)=O c1(C(=O)NCC(CN(C(C2CC3CCC(C2)C3)=O)CC)(C)C)c(F)cccc1F C1(CNC(CCN(CC(F)(F)F)C)=O)CCC(F)(CNC(=O)Cn2ccnn2)C1 c1(C(N(C)CC2(O)CCN(C(c3nccc(C)n3)=O)C2)=O)ccc2[nH]ccc2n1 N(C(=NCCCCl)NCCN1CC2(COC2)C1)CC(C)C(F)F.N1CCCC1 C1(NC(CC(C)=CC(=O)NCC2(C)CSC(C)=N2)=O)CC(C)(C)CN1C C1(C(N2CCC(CC=C)(NC(=O)C(c3ccncc3)C)C2)=O)CC12CCSCC2 CC1=C(C)CC(C(=O)NC(C2CCN(C(C3CC4(CC4)CO3)=O)CC2)(C)C)CC1 Cc1cc(C(N2CC=CC(C(=O)NC(C3CCCC3O)C)C2)=O)c(C)nn1 c1(C(N(C2CCN(C(C3CC(F)(CO)C3)=O)C2)CC)=O)ccc2nc(O)[nH]c2c1 C1(CC(=O)NCC23CC(NC(C45CCC(CC4)C5)=O)(C2)C3)CCC(F)(F)CC1 N1(C(C(C)C2CC2)=O)CCC2C(CCN2C(=O)CO)C1.S(C)(=O)(=O)NCCC1CC1 N1(C(C2CC(C)OCC2)=O)CCCC(CNC(=O)C=Cc2cncs2)CC1 c1(CSCC(=O)NCCN(C(=O)CCCn2ccnn2)CC(C)O)nccn1C C1(CNC(C(F)=CCC)=O)CN(C(=O)CCOC2COC2)CCC1C(F)(F)F CC1CN(c2nc(C(C)(C)C)ns2)CCC1Nc1cc(Cl)n(C)n1 c1(C(=O)NC(C(C)NC(c2ccc(OCC=C)cc2)=O)C)ccc(C)nc1OC C(=O)(CC(Cc1cccs1)CC1(C=C)CCC1)NCc1cc(C(=O)OCC)n[nH]1 N1(C(c2ncn(CC)c2)=O)CCC2C(C(=O)Nc3cn(C)nc3O)C2C1 N1(C(C2CCCOCC2)C(=O)NCCCC(=O)OCC)CC2CCC(O)C2C1 c1(C(N2CC3C(CNC(c4cc(CC)no4)=O)C3C2)=O)cc2c[nH]nc2s1 c1(C(=O)NC23CC(CNC(C4N(C)CCC4)=O)(C2)C3)sc2sccc2c1Cl C1(C(N(C2CCN(C(=O)CC3CC3(C)C)C2)CC)=O)CC(F)(F)C1 CON1CCC(C(=O)NCCCCC2CN(C(C3(C)CC3(F)Cl)=O)C2)CC1 Cc1sc(O)nc1C(=O)NC(C)CC(C)NC(=O)CCn1cc(Cl)cn1 N1(OC)CCC2CC(C(=O)NCCC3CCCC(C)C3)C2C1.c12ncc(s1)CS2 CCC(C)C(C(=O)N1CC(OC(=O)CC)C1)NC(=O)C(O)C(F)(F)F Cc1ccc2c(c1)C(C(=O)NC(C)CCCNC(=O)COc1ccccc1)C2 Cc1cc(C)nc(CCNC(=O)CC2CCN(C(C3SCCS3)=O)C2)n1 Cc1cc(C)n(CCC(N2CCOC(CCNC(c3cnc[nH]3)=O)C2)=O)n1 c1(C(=O)NC23C(CN(C(CN(CC)CC)=O)C2)C3)cc(Br)c2ncccc2c1 N1(C(CC=C)=O)CC(C(=O)N(C2CCCCC2)C)C2(CCC2)C1 n1(CCC(N2C(C(N3CC(C(=O)OC)C3)=O)CC2)=O)nc(C)cc1C C(=O)(CC(C(F)(F)F)n1ccnc1)NCCCN(C(=O)Cc1cnoc1)C(C)C c1(CC)cc(C(N2CCC(O)C(N(C)C(C3C(C)(C)C3(F)F)=O)C2)=O)ccc1O C1(C(=O)NCCC(C(=O)NC2(C)CCCC2O)OC)CC2CC1CC2O c1(OC)c(C(=O)NCC2CCCC2NC(C23CC(C2)C3)=O)c(C)nn1C c1(OC)c(F)ccc(F)c1C(=O)N(C)CC1(O)CCN(C(C2CC2C)=O)C1 C12(C(=O)NC3C4CN(C(C(C)Cc5ccncc5)=O)C3C4)CC3CC1C2C3O N1(C(c2c(CC)ccs2)C(=O)NC2CCOC2)CCC(c2ccccc2)C(O)C1 C1(CNC(CC2CN(C)C2)=O)CN(C(c2cccc(O)n2)=O)CC1O Cc1cc(C(N2CCN(C)CC2C(=O)NC(C)CS(C)(=O)=O)=O)cc(O)n1 N1(C(C2CCN(C(c3c(CC)cno3)=O)CC2)=O)CCCC(C)(N(C)C)C1 c1(C(=O)NC(CN(C(C(C)CNC(=O)OC(C)(C)C)=O)C)C)cc(=O)n(C)cn1 N1(C(CCCN(C)C)=O)CC2(CC(CC(N3CC(C)(CN(C)C)C3)=O)C2)C1 CCC(CC(C)C)C(=O)N(CC(C)(C)CNC(=O)CC1CCCCC1O)C C(=O)(CC(C)CNC(C1CCS(=O)CC1)=O)N(C1CSC1)CC#C N1(C(CN(CCOC)CC)=O)CC(NC(=O)C(C2CC2)OCC)C(C(F)F)C1 C1(CNC(C2(C)CSC2)=O)CCN(C(C2CC=CCC2)=O)CC1C1CC1 N1(C(C(C)NC(CC)=O)=O)CCC(COC)(NC(=O)CC(C)(C)C2CC2)CC1 CCC(CN(C)C)C(=O)N1CCC(C(=O)NCC(=O)NCC)C1C CC1SCCCC1C(=O)O.C12(CCOCC1)C(NC(N1C3CCC1CC3)=O)C2 C1(NC(c2cccc(N(C)C)n2)=O)CCCN(C(C2(Br)CC2)=O)CC1 C(c1ccc(F)cc1)=CCC(=O)NC(C1CCN(C(CNC(CC)=O)=O)CC1)C c1(C(N2CCC(NC(C(C)Oc3cccc(F)c3)=O)C2)=O)csc2ccncc12 c1(NCC(=O)NCC2(NC(C34CC(C)C3C4)=O)CCC2)ccc(F)cc1 Cc1ccc(CCNC(CO)CC(F)F)cc1C c1(C(C(=O)NCCN(C(=O)C(C)CSc2ccccc2)CC)O)cccc(N)c1 C1(CNC(CC(=O)OC(C)(C)C)=O)CCCN(C(C2(C)CC2Br)=O)C1 C(=O)(C1=CS(=O)(=O)CCC1)NC1C(C)(C)CCN(C(CC2CC(C)C2)=O)C1 C=C(Cl)CC(C(=O)NCC(=O)NCCO)NC(c1ncnc(C)c1C)=O c1(COC)ccc(NC(C)=O)o1.C12(CCC1)C(=O)N(C)CCCN(C)C2=O Cc1nc(C(=O)NC2CCCC2NC(C2CC(=O)NC(=O)N2)=O)ccc1[N+](=O)[O-] C(C(C)(C)CN(C(=O)C(CN(C)C)NC(=O)CN1CCCC1=O)C)OC Cc1n[nH]c2cc(C(=O)NC3CCCCC3NC(C3(C)CCCS3)=O)ncc12 S(=O)(=O)(c1ccccn1)N1CCN(C(c2cccc(SC)c2)=O)C(C(F)(F)F)C1 C1(C(N(C)CCO)=O)CC=CC(n2cc(C(C)(C)NC3CCC3)nn2)C1 CC(C)(O)C(C(=O)NCc1n[nH]cc1C1CC1)NC(=O)CC1CCOC1=O C1(C(N2CC(CCNC(=O)C3CC3)OCC2)=O)CC2(CCCCC2)S1(=O)=O C1(NC(C(C)=C2CC2)=O)CS(=O)(=O)CC1NC(=O)CCc1ccc(C(N)=O)cc1 c1(C(=O)NC2CN(C(C3CC4OC3C3CC43)=O)C2)c[nH]c2c(Br)cccc12 N1(C(C(CC=C)NC(C)=O)=O)CC(O)CCC1C(=O)NCC1CN(C)CCN1C c1(C(C(N2CC(CCNC(c3c(OC)ccnc3)=O)C2)=O)C)ccc(F)cc1F C1(C(N2CCC2(CO)CO)=O)CCC(O)CN1C(c1cc[nH]c1)=O CN1CCC=C(CNCc2scc(OC)c2OC(F)F)C1 c1(OC)nccc(C(N2CCCC(c3ncc(-c4ccccc4)[nH]3)C2)=O)c1Br C(=O)(CCCC(C)C)NC1C(CNC(c2c(CC)n(C)nn2)=O)CCC1 C1(C(=O)NCc2nnc(CC)s2)CC(C)CN(C(C2OC3CCC2C3)=O)C1 c1(C(N2CC(C(=O)Nc3cccc(F)c3Cl)NCC2)=O)c(F)cc(Br)cc1Br C(CC(C)C(=O)NCCOC1(CNC(=O)Cc2cccs2)CCOCC1)=CCC c1(C(C)(C)C)ccc(C(C)(C)NC(c2ccc(CN=[N+]=[N-])cc2)=O)cc1 C(=O)(C1(C)CCCc2ccccc21)N1CC(CCNC(C(=O)OC)=O)C1 c1(C(=O)NCC2C(NC(c3c(CC)nccn3)=O)CCCC2)c(C)ncnc1O C1(O)(C(C)NC(=O)C=CC(C)(C)SC)CCN(C(c2c(C)n[nH]c2C)=O)C1 C1(C(N(C(C(C)C)C)C)=O)CSCCN1C(=O)Cn1ccccc1=O C12(NC(=O)Cc3csc(-c4ccccc4)n3)CCN(C(c3ccoc3)=O)CC1C2 C12(NC(C3CC4(C3)CC3(CCC3)C4)=O)CCCCCC1N(C(C1COC1)=O)CC2 C1(=CCC)CCN(C(C2CN(CCN)C2)=O)CC1 c1(C(N2CC(C)C(CNC(c3ncncc3F)=O)CC2)=O)ccc(Cl)c(Cl)c1N c1(C(=O)NC(C2CN(C(c3cnn[nH]3)=O)C2)C)cc(Cl)c(Br)[nH]1 C(=O)(C1=CS(=O)(=O)CCC1)NCC1N(C(C2CCOC2)=O)CCC(C)C1 C1(NC(C2(C(N)=O)CC2)=O)COCC1C(=O)NCC1(C2CC2)CC1 Cc1ncc(C(=O)NC23CCC2CN(C(c2cnn(C)c2F)=O)C3)c(C(C)C)n1 CCC(=O)CCC(=O)N(C(C)C(=O)NCc1ccc(F)nc1C)CC O=C(CCCc1nccs1)NCCCN(CCO)C(c1cnc(C2CC2)o1)=O C1=CC(=O)Nc2ccc1cc2.C(C(C)(C)CC1CC1)NC(C(C)OCCOC)=O CCCCC(O)C(=O)N1CC(CNC(C2(C)CC3CC3C2)=O)(OCC)C1 C(=O)(C(C)(C)CC(=O)N1CC(C(=O)NC(C)CCC(F)(F)F)CC1(C)C)OC c1(C(=O)NCC=C(C(=O)N(C(CC)C)C)C)cncc(CO)c1 CC1CC(CCNC(=O)NC(c2cccc(Br)c2)c2ccccn2)CC(C)(C)C1 C1(C(=O)NCCC2CN(C(c3c(CC)nc[nH]3)=O)C2)CC(C(C)(C)C)=NO1 CC1CN(C(C2Cc3cscc3C2)=O)CCC1N=c1ccnc(Cl)[nH]1 C(C1COC(C)(C)O1)=CC(=O)NC1CN(C(c2c(C)cco2)=O)CC1C c1(C(=O)NCC(CCNC(Cc2cn(C)nn2)=O)O)cccc2nc(O)[nH]c12 CN=c1nc(N(C)CCOC)[nH]c(=NCCC2CC(C)OC(C)C2)[nH]1 c1(CCC(=O)NC2C(NC(c3c(SC)ccs3)=O)CC2)nc(O)c2cnn(C)c2n1 c1(-n2cc(CNC(C3CCCC(=O)O3)=O)nn2)ccc(Cl)cc1Br C1(NCc2c(C)oc(-c3ccccc3)n2)CCCOC12CCNCC2 N1(C(c2ccc(OC)cc2)C(=O)NC(CC)(C)C)CC(C)OC(C)(C(F)F)C1 CC(CNC(c1nnc(O)nc1O)=O)C(F)C(=O)N1CCC1(CO)CO C(=O)(CC1CS(=O)(=O)c2ccccc21)N1C(C)CCN(C(C(C)=C2CC2)=O)CC1 C(=O)(C(O)CCC(C)C)NC(C(=O)NCC(=C)C)CCC1CC1 N1(C(CCS(C)(=O)=O)=O)CCC2(COC(CNC(c3c(Cl)ccnc3F)=O)C2)C1 c1(OCC(N2C(C)CC(NC(=O)C(C)(C)C(F)F)C2)=O)nn(C)cc1[N+](=O)[O-] CC1(C)C=C(C(=O)NC2CCN(CCNC(=O)CC3CC(C)(C)C(=O)N3)CC2)C1 N1(C(C2C(CC)CCN2C(C)=O)=O)CC(NC(=O)CN(C)C)C2CCCC12 N1(C(c2c(OC)cncc2)=O)CC2(C1)CN(C(=O)C(C)(C)N1CCOCC1)C2 CCCCC(C(=O)NC(CCO)C(F)(F)F)NC(c1ncn2c1CCC2)=O c1(C(=O)NCC2CN(C(C(CC=C)C)=O)C(C)(C)C2)oc2cc(Cl)ccc2c1C c1(C(=O)NC(CNC(CCC)=O)CC(C)C)ccn2c(Br)cnc2c1 c1(-c2scc(NC(C3(Br)CC3)=O)n2)cc(F)c(CO)c(F)c1 c1(C(C(N2CC(NC(C=CCCC)=O)C(OC)C2)=O)(C)C)c[nH]c2ccccc12 N1(C(c2cnc(C)nc2)=O)CCC2(C1)CN(C(=O)CC(C)(C)CN(C)C)CCO2 c1(C(=O)NCCC(C(N2CCc3nc[nH]c3C2)=O)OC)ncn2ccccc12 C(=O)(C(C)(C)CCS(C)(=O)=O)N1CC2C(CNC(C(C)c3ccsc3)=O)C2C1 c1(C(=O)NC(C2CCN(C(C(C(C)C)(C)O)=O)CC2)C)cnc2cccnc2c1 CC1(CNCc2nnc(-c3ccc(Br)o3)o2)CC(O)C1 c1(C(N2CCCC(O)(CCNC(C(C)(F)F)=O)C2)=O)cnc(=NCCF)[nH]c1 CN1C(=O)OCC1C(N1CCCC1C(C)(C)C(=O)NCC1(C#N)CC1)=O S(=O)(=O)(c1ccc(N2CCC(c3ccc(Br)cc3)C2)c(Br)c1)N(CCOC)C N12CC(F)(F)CC1C2=O.c1(NC2CCN(C(C)=O)CC2)nnc(C)c(C)n1 C(=O)(C(C1CN(C(=O)CC2CC2(C)C)C1)OC)N(C(C)COC(C)=O)CC c1(NC(CC)CNS(C)(=O)=O)ccc(S(=O)(=O)CC)cc1 CC1C(NC(c2ccccc2CCN(C)C)=O)CCCN1Cc1cccnc1 c1(C(=O)NCC(C(C)C)(C)NC(C2CCC(=O)N2C)=O)csc2cccc(F)c12 CC(C)C(CNC(=O)C=Cc1ccc[nH]1)C(=O)NCCc1cncn1C N1(C(C2CCC(CC)O2)=O)CCN(C(c2cc(C)nnc2O)=O)CC1COC N1(C(C2C(C)SCCC2)=O)Cc2ccc(CNC(c3ccc(O)nc3)=O)cc2C1 C1(C(=O)NCC(C)(C2CCC2)NC(CN(C)C(=O)C2CC2)=O)CC(F)CN1C Cn1nc(C2CCCOC2)cc1C(=O)CN1CC(C)(C)C1 C1(O)(CN(C)C(c2n[nH]cc2Cl)=O)CN(C(=O)C(C)(O)C2CC2)C1 c1(SCCC(=O)NC2CCN(C(=O)C(F)CC3CCCC3)C2)ccccc1Cl N1(C(C2CN(CCC)C(=O)C2)=O)CCCC(C)C1CNC(=O)CCC(C)(C)F C(=O)(CC(C)C(=O)OC)NCC(C(=O)NC(CCC)C1CCC1)N(C)C CC(C)C(C(=O)N1CCCC1)NC(=O)CC(C)O C1(F)(CNC(C(C=C)OC)=O)CCCN(C(=O)C(C2CCOC2)OC)CC1 C1(C(N(C2CCC(NC(CCCCN(C)C)=O)CC2)C)=O)CC12CCCOC2 CC(C)(C)C(CNC(C1COCCN1C(C1CC(F)(CF)C1)=O)=O)CO C=C(C)CC(=O)N(CCNC(=O)C(c1cc(Br)cs1)N(C)C)CCOC N1(C(c2cccnc2)C(=O)OCC)CCC(O)C(O)C1 n1(C(C)C)cc(C(=O)NCC(C)CN(C(=O)CC2(CSC)CC2)C)ccc1=O c1(NC)nc(C(F)(F)F)ccc1C(N1CC(c2cc[nH]n2)C(C)(C)C1)=O CC1CN(C(C2(CF)CN(C(c3cc[nH]c3)=O)C2)=O)CCC1CO c1(C(C)N(C(=O)C(C2CC=CCC2)NC(=O)C(=O)NCC2CC2)C)cnn(C)c1 c1(OC(=O)NNC(=O)NC(COC(C)C)C)cc(Cl)cc(Cl)c1 C(=O)(CC(C)(F)F)N(C1(CCO)CCCC1)C(C(C)C)C Cc1nc(O)sc1C(N1CCC(C(C)C(=O)NC2CC(CO)N(C)C2)C1)=O Cc1nc(C)c(C(=O)NCC(O)CN(C(=O)C=Cc2cn(C)cn2)C)[nH]1 C1(C2CN(C(=O)Cn3cccc(C)c3=O)C2)(NC(CCn2c(C)ncc2)=O)CC1 C=CC(C(=O)NC1CC(CC(=O)NCC(CO)OC)C1)OC C12(CNC(C3=CC(C)(CC)C3)=O)CCCC1N(C(c1csc(C(C)C)n1)=O)CC2 C1(C(=O)NCC2C(CC)CCN2C(c2cscn2)=O)CCC(O)CN1C C1(CC)CCOC1C(=O)NC1CC(C)(NC(=O)CCc2ccoc2)C1 N1(C(C2CCN(C)C2)=O)CCC2C(C1)CN2C(c1ccc(-c2ccco2)o1)=O c1(OC)ccc(C(C)NC(=O)CSCC2CCCO2)cc1Cl c1(C(N2CCC(C(=O)NC(CC#C)CC)C2C)=O)cccc(C#N)c1 c1(N(C)CC2CCCN(C(c3cnc(C)[nH]3)=O)C2)ncnc(C)c1C#N N1(C(c2nc(C(C)NC(C(CC)C#N)=O)oc2)=O)CC2(CCC(C)OC2)C1 C1(NC(C2C(C)(C)C2)=O)CC(CNC(=O)C=Cc2cncnc2O)C12CCC2 N1(C(C(C)=C(CC)C)=O)CCN(C(=O)CP(C)(C)=O)CC1c1ccnn1C N1(C(c2cc(CC)nn2C)=O)CCC2(CCCN2C(C2CCCN2C)=O)C1 C12(CC(OCC)CC)CC(CO1)N(C(=O)C(C1(O)CN(C(=O)OC(C)(C)C)C1)F)C2 S(=O)(=O)(c1cccc(=NCC(C)SC)[nH]1)NC1CCC(CC)CC1 Cc1cc(Br)cnc1C(N1CCC(C)(NC(=O)CN2CCOCC2)CC1)=O N1(C(C2CCCOCC2)=O)CC23CCCCC2(C1)CN(C(C1CCCOC1)=O)C3 CCC(O)C(F)(F)C(=O)NCC(C1CCCN1C(c1occc1Br)=O)(C)C C(CCC(=O)N1CCC(CC(N2CCC(c3ncco3)C2)=O)C1)OC(C)(C)C C1(NC(CCOCCC)=O)CCCC1CNC(=O)Cc1cnns1 CCC(Cc1ccccc1)CC(=O)NCCNC(=O)C(C)(C)n1cccn1 N1(C(CC2CC(=O)C2)=O)CCCC(CO)(CNC(C23CCC(C2)C3)=O)C1 C1(NC(C2(CC)CC2)=O)CC2CCC1CN2C(C1CCCN1C1CC1)=O O=C1CCC(n2ccnc2-c2cccc(-c3cccc(Cl)c3)n2)CN1 CCN=c1[nH]c(C)c(C(N2CC(CNC(C3CCN3C)=O)CCC2C)=O)s1 C1(CCNC(C2CC3(CCCC3)C2)=O)CC(F)(F)CN1C(c1ccncc1)=O C1(C(=O)NC(CC)(CNC(c2cccnc2N)=O)CC)CN2CCC1CC2 N#CC1CCN(C(=O)Cc2csc(Cc3ccc(F)cc3)n2)CC1 N1(C(C2CC(=O)CC23CCC3)=O)CC(C2CCN(C(C3CC34CCC4)=O)CC2)C1 N1(C(CSCCCC)=O)CC(NC(=O)CC(CC)C2CCC2)C2(CCOCC2)C1 c1(OC)ncc(C(=O)NCC2(F)CC(NC(c3csc(Cl)c3)=O)C2)s1 CC1(C)COC(C(=O)NC2CC2NC(=O)CCOCCN(C)C)CO1 c1(CC)cc(C(=O)NC2CCN(CC(CC)CC)C2)no1 Cn1ccc2cccc(C(N3CCC(CF)(NC(c4cnccc4Cl)=O)C3)=O)c12 C=CC1(CC(=O)NC(CNC(C2CC2C2CC2)=O)CO)CCOCC1 c1(C(=O)NCC(C)(C2CCC2)NC(C(C=C=C)C)=O)ccc(OC)nc1Cl CCCCCCCCN(CC(=O)NC1CN2CCC1(CO)C2)Cc1ccccc1 c1(N2CCN(C(c3c(OC)csc3)=O)C3(C2)CC3)ncnc2cc(F)ccc12 N1(C(c2cc(CC)oc2)=O)CCCCC1CN(C(=O)CNS(N)(=O)=O)CC C=CC(C)(O)CC(=O)NC1CC2(C1)CN(C(=O)C(C)Oc1ccc(SC)cc1)C2 c1(SCC2(CNC(NC(c3ccccc3)C)=NC)CC2)ccc2c(c1)OCCCO2 c1(C(=O)NCc2cc(C(N3CC(CCC)OCC3)=O)sc2)cc(C#N)oc1C C1(NC(C2CC2[N+](=O)[O-])=O)CCC(CNC(C2(O)CC2)=O)CC1 CC1(C(=O)NCC2CN(C(c3ccoc3Br)=O)CC2O)COC(=O)OC1 N1(C(C=CCNC(=O)CCn2ccnc2)=O)CCn2nccc21 c1(NC(c2c(NC(C3CCC(=O)N3)=O)cccc2F)=O)ncnc2[nH]c(Br)nc12 CCCCS(=O)c1ccc(-c2csc(=NCCNS(=O)(=O)C(C)C)[nH]2)cc1 Cc1ccc(N2CCN(C(C)C(=O)Nc3ccc(F)cc3Br)C(C)C2)cc1C N1(C(CN(CCC)C)=O)CCN(C(c2ccnn2CC(C)C)=O)CC1CF C1(C(=O)NC2C3(CC(NC(c4c(OCC)cccc4)=O)C3)C2)CC(=O)NC(C)C1 C(=O)(C1=COCCC1)NCC(C1CCN(C(C(CCOC)C)=O)CC1)(C)O Cc1nc(Cl)ncc1NC(C1C=CCN1C(C1CCCS1)=O)=O c1(OC)cc(OC)c2c(c1)N(C(=O)NCCCC1CC1)CCC2 Cn1cccc1C(=O)NCC(C1CC1)NC(C1CCCN1Cc1nnn(C)n1)=O CC(C)C(C)CC(=O)N1CCC(C(C)NC(=O)Cc2cc(O)nnc2O)CC1 C=CCC(C)C(=O)NC1CN(C(=O)C(CC=C)NC(c2ccccc2)=O)CC1F c1(C(=O)NCC2CCCCN2C(=O)Cc2cocn2)cnc2cc(Br)ccc2c1 N1(C(c2nccc(C(=O)OC)c2)=O)CCC(C)(C(N2CCC(COC)C2)=O)CC1 Cc1cnc(C(C)NC(C2CCCC2CNC(c2csnc2Cl)=O)=O)nc1 CCC(C)(C)CCCC(=O)NCC1CC(O)CN1C(c1cncc2ccsc12)=O n1(C)nc(C)c(C(=O)NC2(CCCOC)CC2)c1C.C12CC1CC2=O.C1CC1 C(=O)(C(O)CC(N)=O)N1C(C(=O)NCC(CSC)(C)C)CSCC1 C(=O)(C(O)C(C)CC)NCCn1ncc(C(N(CCCCCC=C)C)=O)c1 c1(C(CC)NC(C=CCNC(CCC(C)SC)=O)=O)ccc2c(c1)OCCO2 c1(C(N2CCCC(N(C(C(CC)OCC)=O)C)C2)=O)cc2c(cc1N)CCC2 C1(C(=O)NCC2(F)CN(C(CNC(C(C)(C)C)=O)=O)C2)CCc2ncccc2C1 N1(C(CCC(=O)NCC)=O)CC2(CCC2)CC1C(N1CCC1CC(=O)NC)=O C1(C(=O)N(C)CC2(NC(c3ccncc3C)=O)CC2)(COC)CCOCC1 Cc1nccnc1CCNC(=O)C(C)(C1CC1)N(C(=O)C=CC(F)F)C C=CCCCC(C)(C)C(=O)NCCC1(NC(=O)C(C)n2cnnn2)CC1 N1(C(C2(CC#C)CCCCO2)=O)CCC(C)(CNC(=O)CC2(CSC)CC2)CC1 N1(C(C2(COC)CC2)=O)CCOC(CCCNC(=O)Cc2ccon2)C1 C#Cc1cccc(CC(N2CCC(C(=O)NCCC(C)N3CCC3)C23CC3)=O)c1 N1(c2nccc(C)n2)CCN(C(C23CC(CN2C2CC2)C3)=O)CC1C N1(C(C(c2ccccc2)SC)=O)CCCC(CO)(NC(c2occ(C)c2C)=O)C1 c1(OC)ccnc(C(N2CC(CO)(NC(c3ccc(SC)cc3)=O)C2)=O)c1 N1(C(=O)Cc2csnn2)CCC2CC12C(=O)NC1CC1c1ccsc1 c1(NC(C)=O)ccc(C(N2CCC(O)(C(C)NC(C3COCCO3)=O)C2)=O)cc1 N1(C(c2ccc(C)cc2N)=O)CCCC2CN(C(=O)COC3CC3)CCC12 C1(n2c(C(c3cn(C)nn3)(C3CC3)Nc3nc(C)c(C)[nH]3)nnn2)CCC(F)(F)CC1 C1(C(=O)NCCOCCC(=O)NC2(C)CC(O)C2)CC2CCC1CC2 C1(C#N)(C(=O)NCC(CNC(c2coc(C(=O)OC)c2)=O)OC)CCC(=O)CC1 C1(NC(CCOCC(C)C)=O)CCCC(C(=O)N(C2CCC2)C2CCC2)C1 C1(C(=O)NCCCN(C(=O)Cn2cccn2)CCO)CCCCC1n1cccc1 CC1=C(C(=O)NC(CC2CC2)CC(=O)N(C2CCCNC2=O)C)CC1 CC(C)(C(=O)NCC1CC(F)(CNC(=O)C=Cc2ccc(O)cc2)C1)C(F)F N1(C(CSC)=O)CCC2(CC2C(=O)NCC(CSC)OC)C1 C=C(C)C(C)(O)C(=O)NCCCCC(C)NC(c1cccnc1OCCO)=O C12(C(N(C(CNC(c3nc(C(C)C)sc3)=O)C)C)=O)CCC(=O)N1CCS2 CON=CC(=O)NCC1(CC(=O)N(CCCF)C)CC1 c1(C2C(C(N3CC(NC(CCCC=C)=O)C(C)C3)=O)C2)ccc(C)c(C)c1 C1(C(N2CCCC(NC(C=CCOC)=O)C2)=O)CC(=O)c2cc(Cl)ccc2O1 C1(NC(CC(n2c(CC)ncc2)C)=O)COCCC1NC(=O)C(=O)NC(C)C C(=O)(CS(=O)(=O)CC(=O)OC)NCC(C)(C1CC1)NC(C(CCOC)OC)=O C(CCCC(=O)N1CCOC(C(=O)NC2CCN(C3CC3)CC2)C1)(OC)OC CC1=C(COC(c2c(Cl)cnc(F)c2Cl)=O)C(C)(C)CCC1 CC1(C(=O)NCc2ccccn2)CC12CCN(C(=O)COc1ccccc1)CC2 c1(CNC(CN2CCN(C(C3(SC)CC3)=O)CC2)=O)cc(C)cc(F)c1 CC(C)S(=O)(=O)CC(=O)NC1CC2CN(C(C3(N4CCCC4)CCC3)=O)CC2C1 C=CCC(CC)C(=O)N1CCC(CNC(C2CC3(CCO2)CC3)=O)C(O)C1 c1(C(=O)NCc2cn(C3C(OCC)COC3)nn2)ccnc(-c2nccs2)n1 C(=O)(C1=NNC(=O)CC1)NCC(=C)CCNC(=O)CCCOCCOCC C=C(C)CCCC(=O)NC(C)CC(C)NC(c1ccc(-n2ccnc2O)cc1)=O CC1CC(C)(C(=O)NC(C)(C)CN2CCN(C(=O)C(C)(C)CC#N)CC2)CCO1 N1(C(C(C)OC(C)=O)=O)CCCC(C(N2CCCN(CCO)CC2)=O)C1C CC(C)(C)C(CC(=O)NCC(F)CNC(c1cnn2cccc(Cl)c12)=O)C(F)F C(=O)(C(CO)C(C)(C)C)NCC1N(C(CN2CCC(C)CC2)=O)CC(O)C1 C1(NC(C2(CC)CC2)=O)(CNC(=O)C(C)NC(=O)NC)CCCC1 C(C(=O)N1CC2CC2C1C(=O)NCC(C)CC1CCCC1)(C(C)C)OC c1(C(=O)NCC2(O)CN(C(c3cccc(N)n3)=O)C2)c(F)ccc(Br)c1F N1(C(CSCCC(C)C)=O)Cc2occ(NC(=O)Cc3cnsc3)c2C1 CC1(C)CCCOC1C(=O)NC1CCCN(C(c2cc(N)cc(F)c2)=O)CC1 c1(C(=O)CN2CCCCCC2)cccc2c1OCC(C(=O)O)C2 C(=O)(C(C)C(C)(F)F)NC(C(C)NC(C(C(C)C)O)=O)CO C1(C(=O)OC)COC(CCC(=O)N(C2CC2)Cc2ccc(Cl)s2)C1 C=CC1OCCC1NC(c1cc(CNC(C2(C#N)CCOC2)=O)on1)=O c1(C(N2CC3C(CNC(c4c(C)cccc4)=O)(C3)C2)=O)cncc(O)c1Cl C1(CNC(C2(OC)CCSCC2)=O)CCC(C)CN1C(=O)COCC1(F)CC1 c1(C(N2CCC(C3N(C(C(C#N)=CC4CC4)=O)CCC3)C2)=O)ccc(CO)cn1 N1(C(CCSCC)=O)CC(NC(c2ccc(C)c(OC)c2)=O)CC1(C)COC c1(C(=O)NC2CN(C(C(CC)CCOC)=O)CC2C)ccc(S(C)(=O)=O)cc1N c1(C(=O)NCC(CN(C(C2(CC#C)CCC2)=O)C)C)ccn(CCO)c(=O)c1 c1(C(N2C3C(CNC(c4cnc(O)s4)=O)C(C3)C2)=O)cc(Cl)ccc1Cl N1(C(CCCOC)=O)CCN(C(c2cc(C)sc2C)=O)C(c2ccncc2)C1 Cn1ccc(C=CC(=O)NC2CC2NC(c2ccc(Cl)o2)=O)c1 CC(N=c1ccnc(N2CCC(CC#N)C(F)(F)CC2)[nH]1)c1nccc(=N)[nH]1 c1(C(C(=O)NC(C)CCN(C(=O)Cc2cncn2C2CC2)C)C)ccccc1F N1(C(C(CCC)F)=O)CC2CCCC(CNC(c3cn(C)nc3C(F)F)=O)C2C1 N1(C(C2OCCC(NC(c3c(CC)con3)=O)C2)=O)Cc2cccc(C#N)c2C1 O(N1CCC(CC(=O)NC(CNC(=O)C=CC(=O)OCC)CO)CC1)CC C1(C(N(CCNC(C(C(C)C)NC(=O)OC(C)C)=O)C)=O)CC2CCC1CC2 c1(C(=O)NCC(CNC(c2ccnc(CC)n2)=O)C)cccc(C)c1C(F)(F)F CN1CC=C(CC(=O)NC(CNC(c2ccc([N+](=O)[O-])[nH]2)=O)C2CC2)CC1 CCC(CCCC(=O)NCC(C)CC1CC1)NC(c1sccc1C)=O CC1CC(C)CN(CCN2CCN(C(C(=O)Nc3ccsc3)c3ccco3)CC2)C1 N1(C(C(C=C)(C)C)=O)CCC(C(F)(F)F)C(NC(=O)C(c2cncn2C)O)C1 C1(CNC(CC2(COC)CC2)=O)CCCCN1C(=O)C(C)CN(C(=O)COC)C Cc1nnc2n1CCC(C(N1CCC(NC(C3CCC(=O)N3)=O)CC1)=O)C2 C1(C)(CNC(c2ccc(OC)s2)=O)CC(OC)CN1C(=O)Cc1[nH]cnc1C C1(C(=O)NC2C(C)(C)C2C(=O)NCC(C)(F)CO)CCC2(CC2)C1 C1(C(=O)NC(C(C)NC(c2ccc[nH]2)=O)CO)CC(C)(C)C(C)(C)C1 C(N1CCCC(n2ccnn2)CC1)=Cc1nnc(C(N)=O)n1-c1ccccc1 Cc1cc(=NC2CCCC2C#N)[nH]c(=NCc2cccc(S(=O)(=O)C(F)F)c2)[nH]1 N1(C(CN(c2ncccn2)C)=O)CCC2CC1CN(C(C1COCC(C)(C)O1)=O)C2 C(=O)(C(C(C)O)NC(=O)CC1CC(C)C1)NCC(COC)OC c1(CNC2CCN(C(c3ccnc(F)c3F)=O)CC2F)cnc2[nH]ccc2c1 c1(CC(=O)NCC(CNC(C(CN(C)C)(C)C)=O)F)ccc2cccnc2c1 C1(COC)(CNC(C2CC(N)C23CCC3)=O)CCN(C)CC1 C1(Cn2c(N3CCC(C(=O)NCCC(C)C)CC3)nnn2)CCCS(=O)(=O)C1 c1(CC(=O)NCC(N(C(CC=C(C)C)=O)C)C2CC2)coc2ccc(C)cc12 N1(C(c2c(C(C)C)occ2)=O)CC(NC(c2cncc(N)n2)=O)C(C)C1 C1(NC(C(C)OCCC=C)=O)CC2C1CCN2C(c1ccnc(S)c1)=O C(=O)(C(=O)CCC(C)C)N1C(C2(NC(C(CC(C)C)NC(C)=O)=O)CC2)CCC1 N1(C(c2c(OC)csc2)=O)CC(NC(=O)C2=CCN(C)C2)CC1(C)C C1(C(=O)NCC2(CN(C)C(C3CC3(Cl)Cl)=O)CC2)OCC2CCCC1C2 Cc1cc(C(=O)NC(C(N2CCCCC2CF)=O)c2ccco2)nnc1O C1(OC)(CNC(=O)C=C(C)c2ccsc2)CCN(C(C2(C#N)CC2(C)C)=O)C1 C(=O)(C1=CCS(=O)(=O)C1)N(CC(CNC(C(CC)(C)C#N)=O)(C)C)C c1(-c2cc(C(=O)NCC=CCNC(C(=O)NCC(F)(F)F)=O)on2)cccc(Cl)c1 N1(C(CNS(CC)(=O)=O)=O)CCCC(O)(CNC(=O)CCc2ccn(C)c2)CC1 c1(C(=O)NCC(C)(C)NC(c2n(C)ccn2)=O)cc(Br)cn1C C(=O)(C1CCc2nccn21)NC(C)(CO)C(=O)NCCC1(O)CCCCC1 C1(CNC(=O)CC2CC=CC2)CN(C(c2ccn3cccc3c2)=O)C2(CCC2)C1 N1(C(CC2(COC)CC2)=O)CC(NC(c2c(C3CC3)cnn2C)=O)C(SC)C1 N1(C(c2cc(CC)sn2)=O)CCC(C)C(C(=O)NCc2ncccc2OCC)C1 c1(COCC)cc(CC(=O)N(CC(C)(C)CNC(=O)CSC(C)C)C)no1 c1(C(=O)NCC2N(C(C(C)SC(C)C)=O)C3C(C2)C3)ccnn2ccnc12 C(=O)(CCCCCN(C)C(C)C)N1CC2C(c3cn(CCCN(C)C)nn3)(C2)C1 C(C)(CCC(=O)c1cccs1)N(CCN(CC=C)C)CCN(C)C C1(CCC)(C(=O)NC2CC2NC(c2ccccc2OC(F)F)=O)CCNC1=O c1(CC(C(=O)NCC(CNC(=O)COCC2CC2)F)O)cc(Cl)sc1Cl c1(C(CC(=O)NCC(CNC(CCN(C(C)=O)C)=O)F)C)c(C)n[nH]c1C Cc1nccn1CCCC(=O)NCC(C)CN(C(=O)CCN1CCCCC1)C C1(NC(C(C(CC)C)O)=O)CCSC12CN(C(c1cnc(N)c(N)c1)=O)C2 C(=O)(CCCCCNC(=O)Cc1cc(F)ccc1F)N1CCC(O)(C(C)C)C1 CCC(CC(=O)N1CC2CCOC2(CNC(=O)CSC)C1)C(C)(C)C c1(C(=O)NCC2C(NC(COC(CC)C)=O)CC2)cccc(N)c1Br C1(NC(c2cncc(C)c2)=O)CCC(C)N(C(c2cc(CO)oc2C)=O)C1 Cc1coc(C(c2nnnn2CSc2ccccc2)NC2(C)CC2(C)C)c1 C=CCC(CC=C)C(=O)N1CCC(NC(=O)CCCCOC)C(CO)C1 CC1CN(C(C2(C#N)CCCOC2)=O)CCN1C(C1CNC(=O)C1)=O C(=O)(CS(=O)(=O)CCC)N1CCN(C(C(C=C=C)C)=O)C(C(F)F)C1 CN1CCCC2CN(C(C3CC4(C3)CC3(CNC3)C4)=O)CCC12 c1(C(N2CC(C(C)NC(=O)Cc3cccs3)C2)=O)ccc([N+](=O)[O-])c(O)c1 N1(C(C(C)N=[N+]=[N-])=O)C2CCCC1CN(C(c1ccnc(CO)c1)=O)C2 c1(C(=O)NCCC(=C)CNC(c2cnoc2CC)=O)c(Br)c(C)nn1C c1(NCC2(C)N=C(C)SC2)ccc(S(=O)(=O)NCc2c[nH]nc2C(C)C)cc1Br N1(Cc2c(C)occ2C(=O)O)CCCC(N2CCCC2=O)CC1 Cc1[nH]cc(C(N2CCCC(C)(CNC(c3ccc[nH]3)=O)C2)=O)c(=O)c1Cl O(NC(=O)C(C)(C)CCNC(c1c[nH]c(=NC)s1)=O)CC(=C)Cl CCC(C(=O)NC(CNC(c1ncccn1)=O)C(C)C)C(C)C C1(C(N2CCC(NC(=O)C3=CCCCC3)CC2)=O)CC12CCc1ccccc12 C12(NC(c3cn(C)nc3)=O)CCCN(C(c3cnc4n3CCS4)=O)C1C2 c1(OC)ccc(C=CC(c2nnnn2CCC2CC2)NCC2CC2)cc1 CCC(O)C(C)(C)C(=O)NC1CC(CCNC(=O)C(C)(C)c2ccccn2)C1 CC1CN(C(=O)C=Cc2cnccn2)CC(CCNC(c2cc(Cl)c[nH]2)=O)O1 Cc1cc([N+](=O)[O-])cc(C(N2CC(CNC(=O)CN3CCOCC3)CC2C)=O)n1 CC1(C(=O)NCC2(CNC(=O)CC3CCC(C)(C)C3)CCCC2)CS(=O)(=O)C1 C1(C(=O)Nc2c(O)ncnc2O)C2CC(F)C(C2)N1C(c1ccco1)=O c1(C(=O)O)c(N(C)C)cccc1C(F)F.n1(C(C)C)cc(C2CC2OCC)cn1 Cc1cc(C(F)(F)F)nn1CC(=O)NCCCNC(c1c(Cl)cnn1C(C)C)=O c1(C(=O)NCC2N(C(C(CC)(C)OC)=O)CCCC2)c(F)ccc(F)c1Br C(N=c1nc(N2CC=CC2)c2ncn(C)c2[nH]1)c1snc(C(C)C)n1 c1(CC(N2CC(CN(C(C(C)CN(C)C)=O)C)C2)=O)cccc(C(F)F)c1 CC1(CNC(c2cccn2C2CCCC2)=O)CCN(C(c2ccoc2)=O)C1 n1(CC(=O)NC2(C)CCN(C(C3C(C)=C3)=O)C2)ccc2cc(F)ccc12 c1(C(=O)NCCCCCN(C)C(C2(C)CCCCO2)=O)cccc2nsnc12 N1(C(C2C3(CCN(C(C(CCCC)CC)=O)CC3)C2)=O)CCc2c(cnn2C)C1 C1(NC(CCCC(=C)C)=O)CC2CN(C(=O)CC3CCC(O)C3)CC2C1 C1(NC(C2C(NC(=O)C(F)F)CC2)=O)(CO)CCOCC1 c1(NC(Cc2c(-c3ccc(C4(C)CCCC4)cc3)csc2)=O)ccc(F)cc1Br C1(NC(C2CCN(c3ccc(Cl)nn3)CC2)=O)CN(C(=O)C=CCO)CC12CC2 N1(CC(=O)NCC2(C)CC(NC(c3n(C)ccc3)=O)C2)CC(=O)NC1=O N1(C(C=C(CCC)C)=O)CC(NC(C2CCC(C)O2)=O)CC1CO C(=O)(C1CCCc2nn[nH]c21)N1CC2C(NC(C#CC3(C)CC3)=O)(CC2)C1 O=C(C=NN1CCCCC1)N1CC2CC(F)(F)C2C1 CC1=C(C(=O)NCC2CCN(C(c3cn(C)nc3C(C)C)=O)CC2O)CCO1 c1(NC(CSCC(N2C(CC(C)=O)CCC2)=O)=O)cccc2ccccc12 C(CS(=O)(=O)CC(=O)NCC(C)(C(C)C)NC(c1cc(C)c(F)c(C)c1)=O)OC CCC(C)(C(=O)N1CC2CN(C(=O)C=C3CCN(C)C3)CC2C1)C(F)F c1(C(=O)NCc2cscn2)ccc2c(c1)S(=O)(=O)C=C2 CC1OCCCC1C(=O)NCc1ccc(CNC(c2sccc2CO)=O)cc1 C(C(C)(C)CNC(C1(n2cccn2)CCCC1)=O)N(C(=O)C(O)C1CCC1)CC CCC(CNC(=O)CC1CC2(C1)CN(C(C1CC1C(=O)OC)=O)C2)C(C)(F)F CC(C)CCC(=O)C(=O)NC(CCN(C)C)C(=O)NC(C)(C)CCCF C12(NC(C3CC(OCC)C3)=O)CCCC1CN(C(c1cccc(F)c1Cl)=O)C2 C1(C(=O)NCC(C(CC)C)C)CN(C(C2(C)C=CCCC2)=O)CC(C)(C)C1 c1(CN(CCNC(=O)NC2(OC)CCCCC2)CC)ccc(O)cc1C c1(C(=O)OC)cc(C(=O)NCCC2CCC(F)(F)C2)cc(C(C)C)c1 C(CC1NC(=O)c2ccccc21)OC(c1c(F)ccc(Br)c1Cl)=O Cc1ccnc(C(C)(C)C(=O)NCCCN(C(=O)CC(=O)NCC(F)(F)F)C)c1 C1(CC(C)C)CN(C(C2(C)CCN(C(=O)CN3CCCC3C)C2)=O)CCO1 C12(NCC3N(C(c4c(CC)n[nH]c4)=O)CC(OC)C3)CCC(C(=O)NC)(CC1)C2 N1(C(C=C)=O)CCC(C(=O)NCC2CC(F)(F)C2)C(O)C1 N1(C(c2cn(CCC)nc2)=O)CCCCC2(CCN(C(=O)CSC(F)F)C2)C1 CC1(C(=O)NCCCOCCNC(c2csc(C3CC3)n2)=O)CCCC1 Cc1cncc(C(N2CCC(C(F)F)(CNC(c3snc(O)c3Cl)=O)C2)=O)c1 c1(-c2cc(C(N(C3CC(C(N)=O)C3)C)=O)n[nH]2)ccccc1F C1(CNC(C2(CC)COC2)=O)CN(C)CCN1C(C1CC2(CC2)CO1)=O C=CCCC(C(=O)NCCN(CC)CC)NC(=O)Cc1ccccc1CC C12(NC(C(C)CF)=O)CCCC(CN(C(=O)CN3CCCOC3=O)C1)C2 N1(C(C(C)(C)NC(=O)OC)=O)CCCC(F)(C(=O)NCCCN(C)C)C1 Cc1cnnc(O)c1C(N1CCC(C)(CNC(=O)CC2(C)CCOCC2)C1)=O CCCC(CC)C(=O)NCC(O)CCNC(c1cnc(CC(C)(C)C)s1)=O CCC(C)(O)C(=O)NCC(C)C(=O)NCCC12CC(CCO1)C2 N1(C(C2N(C)CCC2)=O)CCC(C(=O)NCCCOCC(F)F)C1(C)C N1(C(C2(CC)CCN(C(C(CC)C(F)(F)F)=O)CC2)=O)CCN2C(=O)CCC2C1 C(=O)(C1=NOC2(CCC2)C1)NC(C(C)C)C(=O)NC(C1CCCC1)C CCC(CC)C(F)C(=O)NC1CCCC1CNC(=O)CCc1ncc[nH]1 C(C)(C)(CCCC(=O)N1CC=CC1C(=O)N(C)C)NC(CC(=O)OCC)=O c1(CCN(CC=C)Cc2nn[nH]n2)csc(C(C)(C)C)n1 Cc1ccc(CC(=O)NC(Cc2ccccc2)CCNC(C2CC2(Cl)Cl)=O)cn1 O=C(N=c1ccc(C2CCOCC2)n[nH]1)N1CCC2CC2C1 c1(C(=O)NCC2N(C(C(C(C)C)NC(N)=O)=O)CC2)cccc(Br)c1N N1(C(c2nncc(CCC)c2)=O)CCC(CO)(NC(c2coc(CO)c2)=O)CC1 CON1CC(C(=O)NC2CCCC2C(=O)NCCC(C)(C)N(C)C)CC1=O c1(C(N2CC3(C(C(=O)NCc4cncc(Cl)n4)C3)C2)=O)cc2ccccn2n1 C(C(=O)NCCOCCN(C(=O)Cc1nccs1)C)(C(C)C)SCC CC#CC1CCN(C(=O)C(Cn2cncn2)NC(c2cnn(C(C)C)c2)=O)CC1 c1(C(=O)NCCCC2(NC(C3CC=CC3)=O)CC2)cnn(CCO)c1 c1(C(N2C(C)(CNC(C3(C)CCCO3)=O)CCC2)=O)cc(O)c2ccsc2c1 CC1(CNC(C23CCCC2C3)=O)CCCN(C(c2ncnc(O)c2F)=O)C1 C1(C(=O)NC2CCCN(C(c3ccc(CC)o3)=O)C2)CC(=O)NC(=O)N1 C1(C(=O)NCC(C)(C)NC(C2CCC(CC)O2)=O)CC(C)(C)C(C)(C)C1 C12(C(=O)NC3CN(C(C(C(C)C)SC)=O)C(C)CC3)CC3CC(C1)CC(F)(C3)C2 C1(OC)CC(NC(=O)CCC=Cc2ccccc2)CN(C(=O)C(C)C#N)C1 C(=O)(C(C)S(=O)(=O)C1CCOCC1)NCC(CNC(=O)Cc1cncs1)OC C1(CN(C(C2CC(SC)C2)=O)C)(CNC(C)=O)CC1(F)F C12(NC(CCCC(=C)C)=O)CCCC1N(C(=O)CN1CCCNC1=O)CCC2 C1(C(C)C)CCCC1C(=O)NCc1cc(C(=O)NCc2ncc(CO)[nH]2)co1 N1(C(C(CCC=C)(C)C)=O)CCC2(CCC2)C(NC(C2CCOCC2(C)C)=O)C1 N1(CCNC(CCCC)=O)CCC(NC(c2cnn(CC3CCOC3)c2)=O)CC1 N1(C(C2(n3cnnn3)CC2)=O)CCC2CCCC12C(N1C2CSCC1C2)=O Cc1nn(CCO)c(C)c1C(=O)NCC1COCC(C)O1 N1(C(c2ccc(CC)o2)=O)CCCN(CCCCNC(C2CC(=O)N2)=O)CC1 N1(c2nc(C)cc(C(=O)OC)n2)CC2CCC1CN2C(=O)CCN1CCC(F)C1 CN1CCCC(CC(=O)NC2CCC2CNC(=O)CC2(CSC)CC2)C1 CC1(NC(c2cc(O)ncn2)=O)CCCN(C(=O)C=Cc2ccccc2)C1 c1(C(=O)NCC(C)N(C(=O)CCCN2CCCC2)C)cccc2c1ncn2C CC1(C)CCC(C(=O)NCCN(C(=O)C(O)Cc2ccccc2)CC2CC2)CC1 c1(C(=O)NC2(C)CN(C(C=C(C)Cl)=O)C2)cc(Cl)cc(F)c1N N1(C(c2n(C(C)C)ccn2)=O)CCC2(CCCCC2NC(=O)C(C)CF)C1 CCC(C(=O)N1CC2CC1CN(C(C1(SC)CCC1)=O)C2)C(C)(F)F c1(C(=O)NCCN(CCOC)C(c2cc(Cl)c[nH]2)=O)ccc(CF)cc1 C(=O)(C(C)C(C)C(C)(C)C)NCCN(C(=O)C(C)(C)OC)CC S(=O)(=O)(c1c[nH]ccc1=NCc1ccc(C(=O)NCCO)cc1)N1C(C)CSC1 CC(C)C(C(=O)N1CCC2CC2(C(N2CC3(C2)CC(C)(O)C3)=O)CC1)C(C)C C1(C)(CC)C=C(C(=O)NCCCCC(CO)NC(=O)Cc2c(C)nn(C)c2C)C1 N1(CCc2cn(CC)nc2)CCOC(C)(CNC(C2(C)CCNC2=O)=O)C1 c1(C(=O)NC(C)CCCNC(C2(C3CC3)CCCO2)=O)cnc2nccn2c1 C1(NC(c2ccc(CNC(C)=O)s2)=O)CCC(C)N(C(=O)C(O)C(F)(F)F)C1 c1(C(=O)NC)cccc(S(=O)(=O)NCC23COCCC2C3(F)F)c1 n1(C(C(=O)OC)C)cc(CNC(C2CC2C(C)(F)F)=O)nn1 CP(C)(=O)c1ccnc(-c2noc(-c3ocnc3NS(C)(=O)=O)n2)c1 N1(C(c2cc(C)c(O)nn2)=O)CCN(C(=O)C=Cc2cnc[nH]2)CC(C)C1 C(=O)(N=c1[nH]oc2ccc(Cl)cc12)NC1CN(C)C(C(F)(F)F)CC1 C(CN=c1cc(C)c(S(=O)(=O)N2CCC(S(C)(=O)=O)CC2)c[nH]1)OCCOCC C#CC1(C(=O)NCCOC(C)(C)CC)CCN(C(C2CC(CCOC)C2)=O)C1 c1(OC)cc(C(=O)NCC2CC(NC(=O)COCCC(C)C)CC2O)ccn1 C(=O)(C(O)CC(N)=O)NC(CNC(C=C(CCC)CCC)=O)(C)Cn1cccn1 CCC(CC)C(F)C(=O)N1CC(O)(CN(C(=O)CC2CCC(C)C2)CC)C1 O=C(CS(=O)(=O)Cc1cccs1)NCC12CC1CN(C(C1C3(CC3)C13CC3)=O)C2 C1(CN(C(CSCC#C)=O)C)CN(C(C2CC2c2ccccc2Cl)=O)CCO1 N1(C(C2N(C)CC2)=O)CCC(O)(CNC(=O)CC2CSC2)CC1 c1(C(=O)OCC2CC(OCC)C2)cc(F)ccc1SC C1(C#N)(C(=O)NCCCN(C(C2(C)CC2C)=O)CC)CCOCC1 C1(NC(COCCOCC#C)=O)COCCN(C(=O)CCc2cnc(C)o2)C1 Cc1ccc(-c2cc(C(=O)NC(CNC(c3occc3C)=O)CO)no2)c(C)c1 c1(C(=O)NC2C(C(=O)Nc3c(C(=O)OC)n[nH]c3)C2)cc(C)c2cc[nH]c2c1 n1(CC)c(C(N2CC(CNC(=O)COCc3nc(C)no3)CC2C)=O)cnc1O C(C1CN(C(C2C=C2C)=O)Cc2ccccc21)NC(c1scc(OC)c1)=O CC1CCOC1C(=O)NCCC1(CNC(c2cc(-c3ccccn3)ns2)=O)CC1 C1(C(C)C)CN(C(=O)Cc2ccnn2C)CC1C(=O)NCC(F)CO C1(OC)CCCN(C(=O)CC(C)NC(C2(CO)COC2)=O)CC1 C1(F)(CNC(c2c(C)nc(C(C)C)o2)=O)CCCN(C(c2ccc(Cl)cn2)=O)C1 C1(CC)COC(C)(C)CN1C(C1CC2CCC(C1)N2C(=O)CC(C)(C)C)=O N1(C(C2(CC)CNC(=O)C2)=O)CCN(C(=O)Cn2ncn(C)c2=O)C(CCO)C1 C=CCCCCCC(=O)NC(C)C(CO)NC(C1(COC)CC(F)(F)C1)=O c1(C(N(CCOC)CCNC(=O)C(c2ccccc2)O)=O)cncc(OC)c1 c1(C2CC2)cc[nH]c1C(=O)NC1(C(=O)NCC(CO)C2CCC2)CCC1 C1(C(N(CCC(N2CC(O)(CC)C2)=O)CC2CC2)=O)CC12CCOC2 C(=O)(C1CC(NCC(=O)NCc2ccccc2F)c2ccccc21)OCC CC(C)C(Cc1ccccc1)C(=O)N1CCC(NC(c2cccc(Cl)c2)=O)C1 C1(CNC(CCOCC#C)=O)CN(C(=O)CC(C)(C)C)CCC12CCOC2 N(C(=NCCc1ncccc1C)NCC1C=CCC1)C(C=C)C CCC(C(=O)NCC1(C)CN(C(c2ccnn2CCF)=O)CC1C)C(C)(F)F c1(C(=O)NCC(CNC(C(CC)=CC)=O)OC)ccc2cccnc2c1O c1(N(C(C(C)OC)=O)C)ncccc1Oc1ccc(Br)cc1 c1(OCC(=O)NCCN2CCN(C(=O)C(Cl)(Cl)Cl)CC2)ccc(F)cc1F N1(C(C23C(CN(C(=O)C=Cc4nccs4)C2)C3)=O)CCC(F)(CO)CC1 c1(CN2CCCC(CNC(c3cc(CC)n(C)n3)=O)C2)cccc2c1OCO2 C1(CNC(C=C(COC)C)=O)(OC)CCN(C(C2(Cl)CC23CCC3)=O)C1 Cc1oc(Cl)nc1C(=O)NCCNC(=O)CCCN(C(N)=O)Cc1ccc(Cl)cc1 Cc1cccc2nc(CNC(C3CCCN(CCCC4CCCO4)CC3)=O)cn12 N1(C(C)=O)CCCCC(F)(F)C1.N12CCCC(C1)C(C)CC2=O CCCCC(CCCC)C(=O)N1CCC(C(C)(C)NC(=O)C=CS(C)=O)C1 C1(NC(C(COC)C)=O)CN(C(=O)C(C(C)(C)C)NC(C)=O)CC2(CCC2)C1 C1(C(N2CCC(=CCNC(COC3(C)CCC3)=O)CC2)=O)CCCC1P(C)(C)=O C(=O)(C1=NNC(=O)CC1)N1CCC(C)C(NC(C2(c3ccno3)CCC2)=O)C1 N1(C(CCc2n(C)ccn2)=O)Cc2[nH]nc(C(N3CCOC4CC34)=O)c2C1 C(=O)(CC(CN(C)C)CC)N(C(CC(=O)NC1CC(CC)C1)C)C CON(CCC(=O)N(C1CS(=O)(=O)C1(C)C)C)C(=O)CC1CC(=O)NC1=O C(CNC(=O)CSCc1ccccc1Cl)(CC(C)C)NC(C1C(C)(CC)C1)=O N1(C(c2c(C(C)C)n[nH]c2)=O)CCCCC(CNC(=O)CSc2ccccn2)C1 C(c1c(F)cccc1F)=CC(N1CC(O)CC(NC(c2ccc(=O)oc2)=O)C1)=O C(=O)(C1SCc2cccnc21)NC12C(CN(C(C(C)=CC)=O)C1)COCC2 Nc1ccc(Br)c(C(=O)NCC2CCC(NC(=O)C(O)C3CC3)CC2)c1 C1(c2ccccc2)CCN(CCCc2nc[nH]n2)CCO1 C1(N(C)C(C2(S(C)(=O)=O)CC2)=O)CN(C(=O)C(c2cccn2C)=O)CC1(C)C C(=O)(C#CC(C)(C)O)NCC1CCN(C(C(C=CCCC)O)=O)C1 c1(SC2(C(=O)NCC(C3CN(C(c4cc[nH]c4)=O)C3)C)CCC2)ccccc1 c1(C(=O)NCc2cccc(CNC(C=CS(C)=O)=O)c2)ccc2n[nH]cc2c1F CC1CN(C(C2C3CC2N(C(=O)Cc2csnn2)C3)=O)CCO1 C(=O)(C(O)CC(C)(C)C)N(CC(C)NC(c1cnccc1C#N)=O)C N1(C(c2n(C(C)C)ncc2Cl)=O)CC(NC(c2ccc(Cl)c(F)c2)=O)CC(F)C1 c1(N(C)C)ccc(F)c(C(=O)N(C2CCCC(NC(=O)C=CC3CCC3)C2)C)c1 c1(N2C(C)CC(NC(c3ccc(CN(C)C)o3)=O)CC2)ncn(C)c(=O)c1Br CC1CC(NC(C2(NC(C3CC(F)(F)C3)=O)CSC2)=O)CCS1 C(C)(CCN=c1ccc([N+](=O)[O-])c[nH]1)NC(c1c(OC)n(C)nc1C)=O C(=O)(CCC(C)(C)OC)NCCC(C(C)C)NC(CCC(=O)NCC)=O N1(S(CC2(C)OCC(C)(C)OC2)(=O)=O)CCC(=C(Br)Br)CC1 CC1(CNC(C2(C)CC2(F)F)=O)CN(C(C2CCC(F)(F)CC2)=O)CCO1 Cc1ccc(C(=O)NCC2CCCCN(C(c3c(C)noc3C)=O)C2)c(Cl)c1C CC(C)C(CCNC(=O)COC(F)(F)F)NC(C1(c2cccnc2)CCC1)=O C1(CNC(C(COC(C)C)(C)C)=O)CCN(C(=O)CCc2nncn2C)CC1O C1(C(=O)NCCOCCCNC(c2cncc(OC)n2)=O)CCC(=C(F)F)CC1 c1(C(=O)N=c2cc(Cl)cn[nH]2)ccc2c(-c3ccc(CO)cc3F)cccc2n1 Cc1cc2c(C(=O)NCC3CC(NC(c4cc[nH]c4C4CC4)=O)C3)nccn2n1 c1(OC)ncc(C(=O)NC(C)C(C(C)C)NC(=O)Cc2ccoc2)c(C)n1 N1(C(c2ncn(C)n2)=O)CCC(O)(CCNC(c2cncc(F)n2)=O)C1 N1(C(C(=O)NCCCOC)C)CCC(F)(F)C(CNC(=O)CCC(C)C)C1 C(=O)(C1=CS(=O)CCC1)N1CCCC(C)C1CNC(=O)Cn1cnc(C(N)=O)n1 c1ccc(F)c(C#N)c1.c1(CNC(C2(C)CC2C(=O)OC)=O)ccc(F)cc1 C1(NC(c2cc(SC)oc2)=O)CN(C(=O)CC2CCCC23CC3)CC1(C)C Cc1nc(CC(C)C)oc1C(N1CC=CC1CNC(=O)CC(C)C1CCCC1)=O CCC(C(=O)N(C)CC1CCCN(C(=O)C(C)SC)C1)C(C)(F)F c1(C(=O)NC2CN(C(C=C(C)Cl)=O)CC2C2CC2)cn2cccc(C)c2n1 c1(C(N2C(CCNC(C3CC(=O)NC3)=O)CSCC2)=O)cc[nH]c2nccc1-2 N#Cc1cccc(C(=O)NC2CN(C(=O)CC3CCCCC3)CCC2(F)F)c1Cl C(CN(C)C)(C(=O)NCC1(O)CCCC1)NC(C(C)OCC#C)=O C1(C(=O)NCCc2cn(C)nn2)CC2(CCC2)CN1C(C1CC(CF)C1)=O C=CC(C)(CCOC)C(=O)N1CCCCC(NC(=O)C(CC)CO)C1 Cc1nn(C)c2sc(C(N3CCC(CNC(C4CC5CCC45)=O)C3)=O)cc12 N1(C(c2c(CC)ocn2)=O)CC2CC(C(N3CCC3C3CCCC3)=O)(C2)C1 C(c1cccc(Cl)c1)=C(C)C(=O)NC1(CO)CN(C(C2(C#N)CC=CC2)=O)C1 c1(C(N2CC(CNC(C3CC(=C)C3)=O)C3(C2)CC3)=O)ccc2c(Cl)nccc2c1 C1(C(=O)NC2CC(C)(NC(c3c(N)cn(C)n3)=O)C2)CC(=O)NC1(C)C Cc1cn2nnc(C(N3CCN(C(C4CC4F)=O)C(C)C3)=O)c2c(O)n1 c1(C(=O)NCCCN(C(=O)CCC2CCCN2C)CCC)ccc(C)nc1OC N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CC(NC(=O)Cc2cncs2)CC(F)C1 c1(NC)ccc(C(N2CCN(C(=O)C#CC(=O)N(C)C)CC2C(F)F)=O)c(Cl)c1 c1(N(C2CCS(=O)(=O)C2)C(C2(C)CCCS2)=O)ccccc1C=O N1(C(c2cnc(C(C)C)[nH]2)=O)CCC(CCCNC(c2ccc(Cl)cn2)=O)CC1 c1(C(=O)NC2CN(C(c3ccc(C(C)=O)[nH]3)=O)C(C)C2)ccc(C2CC2)cc1C c1(C(C(=O)OCC2C(C(=O)O)C2)(F)F)ncccc1F C=CCC(C(=O)NCC1(F)CC(NC(=O)C(c2ccccc2)=O)C1)NC(C)=O C=CCC(C)(C)C(=O)NCC1CCCCN(C(=O)C(C)CC(N)=O)C1 n1(CC)cnc2[nH]c(=NC(C)c3cnn[nH]3)nc(N3CCC(F)(CO)CC3)c12 C1(OC)CC(OC)CN(C(C2CCC(Cl)C2)=O)C1 N1(C(c2cc(C)nc(C)c2)=O)CC(NC(c2[nH]cc3c2CCC3)=O)CCC(O)C1 C1(C)(CNC(C(CN(C(CC2CC(=C)C2)=O)C)C)=O)CCCC(=O)N1 c1(CC)nocc1CN(C(=O)C(c1cccs1)NC(=O)CC(=O)N(C)C)C N1(C(c2cc(OC)c(C)cc2)=O)CC2CCCC(NC(C3CCSCC3)=O)C2C1 C(=O)(CCOCC1CCC1)NCCCN(C(C1CC1C(=O)OC)=O)CC c1(C(N2CC=CC(NC(C3C(C)(C)CC3)=O)C2)=O)ccc(C#N)c(O)c1 c1(C(=O)NC(C2CCCN(C(c3scnc3Cl)=O)C2)C)cc([N+](=O)[O-])nn1C c1(N2CC(CC=C)(NC(C3CCOC3CC)=O)C2)ncnc2ccc(O)cc12 N1(C(c2n[nH]c(C)c2C)C(=O)NC2(C)CC2)CC2CS(=O)(=O)CC2(C)C1 N1(C(C(CC)O)=O)CC(C)(C)OC2(C1)CN(C(=O)C(C)NC(=O)OC(C)(C)C)C2 C12(N(C(c3c(C)nc(CO)s3)=O)C)CCN(C(=O)COC3CC(F)(F)C3)CC1C2 c1(C(N2CCOCC2CCC)C(=O)NCC=C)ccc(C)c(C)c1 c1(C(=O)NC2CCN(C(c3nc(C)oc3C)=O)CC2)cnc2ccccn12 N1(C(C(C)OCCCC)=O)CC2(C)CN(C(c3cc(CCC)on3)=O)CC2(C)C1 c1(C(=O)NCC(CC)(CC)NC(=O)C(C(C)C)C(C)C)ccn2cc(C)nc2c1 c1(C(N(CCCNC(C2(c3cccs3)CCCC2)=O)CC)=O)cnc(N)cn1 N1(Cc2n(C(C)C)ccn2)CCOC(C)(Cc2nc(N3CCCCCC3)no2)C1 Cc1ccc2c(C(=O)NC3CCC3CNC(c3cc(C)c(C)o3)=O)c[nH]c2c1 Cc1cnn(C(C)C)c1C(=O)NCC1CCCC(CNC(C2C=CCC2)=O)C1 C1(O)(CNC(C2(CC=C)CC2)=O)CC(C(=O)NCC(CO)N(C)C)C1 C1(CC)CN(C(=O)CC2CCCC(=O)C2)CC1CNC(=O)CNC(=O)CC(C)C c1(C(N2CCCC(NC(C)=O)C2)C(=O)NC2CCC2)ccc(CO)cc1F c1(C(N(C2CCN(C(=O)C(C)CC3CCCC3)C2)CC)=O)c[nH]nc1Cl N1(C(C2C(C(=O)OC)C2)=O)CC(C2CN(C(=O)C=Cc3ccc(OC)cn3)C2)C1 C(C)(C(=O)N(CC(=O)N(C12CC(C1)C2)C)C1CC1)[SH](CCCC)C1CC1 Cc1cc(C(=O)C(N2CC(F)(F)CC2CNC(c2n[nH]c(O)n2)=O)=O)ccc1F C1(NC(Cc2cc(C)sc2)=O)C2CC(O)C1N(C(=O)CCCNC(N)=O)C2 c1(C(N(C)CCN2CCN(C(C3CC4CCC34)=O)CC2)=O)ccn2cnnc2c1 C(C(=O)NCc1csnc1OC)(C(C)(C)C)NC(c1cccc(OC)c1)=O C=CC1OCCCC1C(N1CC(C(F)(F)F)CC1CNC(=O)CSC1CC1)=O c1(C(=O)NC2C(NC(COCCC)=O)C2)ccc([N+](=O)[O-])cc1[N+](=O)[O-] N1(C(C(CC(C)C)C)=O)CC=C(C(=O)NC2CCCCCCC2C)CC1 c1(C(N2CCCCC2CCO)=O)cc2cc(-c3ccsc3CO)cnc2[nH]1 C1(O)(CC(=O)NC2CCN(C(CCCOCCOCC)=O)C2)COC(C)(C)C1 N1(C(COCC(=C)C)=O)CCC(CN(C(=O)C(C)n2cccc2)C)CC1 C1(NC(CN(CCC=C)C(C2C=C(C)CS2)=O)=O)CCCC1CCO c1(SC)cc(=NC(=O)C2CC23CC(NC(C24CC(CO)(C2)C4)=O)C3)[nH]n1C c1(C(N2CCC(CNC(CSCC(C)C)=O)C2)=O)c(Cl)nsc1Cl C=C(CNC(=O)CC1CCN(C(=O)COCC2CCCC2)C1)c1ccccc1 c1(OC)ccc(F)c(C(N2CCC(N(C)C(c3ccc(F)c(C)c3)=O)C2)=O)c1F c1(C2CN(C(C3C(CNC(=O)COC(F)F)CCO3)=O)C2)ccncc1 c1(C(=O)NC2(CC)CC2)nc2n(c1Cl)CCN(C(=O)Cc1ccc(Cl)cn1)C2 c1(CN2CC3N(C(c4cc(Br)c[nH]4)=O)C3C2)cccc(Cl)c1Cl C1(C(N2CCC(O)(C(F)F)C2)=O)CC(F)(F)CN1C(c1cc[nH]n1)=O c1(C(N(CCCNC(=O)C(CCC2CC2)SC)CC)=O)ccc(C#N)c(OC)c1 C(=O)(C1=CCCCO1)N(CC(C)O)CCNC(=O)C(C)(C)C1(C)CC1(F)F C(C(O)CC(=O)N1C(c2cncc(Cl)c2)CCC1(C)C)N(C)C C1(F)(C(=O)NC2CN(C(CC)=O)C2)CCCN(C(c2nccn2CC)=O)C1 CCCCCCC(C)C(=O)NC(CCC(C)C)C(=O)NCC(C)(C)C(C)(F)F Cc1ccc(C(N2CCC3(NC(c4ccc(C(F)F)cn4)=O)CC3C2)=O)c(O)c1 c1(C(=O)NCCOCCNC(Cc2cc(C)cc(C)c2)=O)n[nH]c2c1NCCC2 CC1(C)C(C(=O)NC2(CNC(=O)C=CC3CCCC3)CCC2)C1c1ccccc1 C1(C2(O)CCN(C(c3ccc4ncnn4c3)=O)CC2)(NC(C2C(=C)C2)=O)CC1 C1(C(N(C(C)CNC(c2[nH]nnc2C2CC2)=O)CC)=O)C2CC3CC(C2)CC1C3 CCS(=O)(=O)c1cccc(C(=O)NC2CCCCC2NC(=O)C(CO)N(C)C)c1 c1(OC)cn(CC(=O)N(C)CCN(C(=O)CCC(=O)N(C)C)C)c(C)cc1=O c1(C(N2CC(N3C(=O)CC(NC(C(C=C=C)C)=O)C3)C2)=O)c(F)ccc(Cl)c1F C12(CNC(CCCC)=O)CCCCC1CN(C(c1coc(CC)n1)=O)C2 C1(C(N(C)CC2CCC(NC(C(CSC)O)=O)CC2)=O)CCCC(C)CC1 C1(N(S(C)(=O)=O)C)CCN(C(=NCC2CCSCC2)NC2CC2c2ccccc2)C1 CC1(C(N2CC(NC(C3CCN(CC(F)(F)F)CC3)=O)C(O)C2)=O)CC(F)(F)C1 c1(C(N(CCCCNC(CN(CC)CC)=O)C)=O)n[nH]c2c1CCOC2 N1(C(CC(CC)OC)=O)CCCC2(NC(c3cc(C)n(C)c3)=O)CC2C1 C(=O)(C(C(=O)NCCCCCNC(=O)CC1CCC(C)(O)CC1)C(C)C)OCC c1(C(C)C)nnc(CC(N2CC(NC(=O)CCSc3nccn3C)C2)=O)o1 C1(NC(Cn2ncc(C)c2)=O)CCN(C(C23CC(C2)C(C)O3)=O)CC1F c1(OC(F)F)ccc(CCCCNC2CCN(C3CC3)CC2)cc1 N1(C(c2cc(C)ccn2)C(=O)NCC(=C)C)CCc2cc(OC)cc(OC)c2C1 C1(F)(C(N2C(CNC(Cc3nc(C)sc3Cl)=O)CC2)=O)CCCN(C)C1 N1(CCC)CCCC1C(=O)NCC(CO)NC(c1cnn(C2CCC2)c1)=O CCCC(CCCO)C(=O)N1CCC(NC(=O)CNS(=O)(=O)N(C)C)CC1C C1(COC(c2cc(OCC)n[nH]2)=O)CCOC(C2CCNCC2)C1 CC1CC(CNC(c2cn(C(F)F)cn2)=O)CN1C(=O)Cc1cccnc1 c1(OC(C)C(=O)Nc2cccc(-n3ccnn3)c2)ccc(F)cc1Br c1(C(=O)NC2CC(CNC(=O)C(c3ccc(F)cc3)O)C2)cccc2c1CCO2 c1(OC)cccc(CNC(c2cnn(C)c2)C2CCCC2)c1O CCCC(C)(CC)C(=O)NCC1CCCN1C(=O)CC1(CSC)CC1 C1(O)(CCNC(=O)C(c2ccc(Cl)cc2)O)CCN(C(=O)CC2CC=CC2)CC1 CCC(C)C(O)C(=O)N1CCN(CCNC(c2cc(O)ccc2F)=O)CC1 CC1(C)CC(NC(c2cncc(-n3cccc3)c2)=O)CN(C(c2cncs2)=O)C1 C(CN=C(NCC1(O)CCC1(C)C)N(C)Cc1cnn(C)c1C)N(CC)CC c1(C(=O)NC2CN(C(Cc3ccc(OC)cc3)=O)C3C2C3)cncc([N+](=O)[O-])c1 n1(CCC(=O)NCC(C2CC2)NC(=O)Cn2nnc(=O)[nH]2)cnc2ccccc12 N1(C(c2n(CC)ncn2)=O)CC2CC1CN(C(=O)C=CC1CCCO1)C2 C(=O)(C(C(C)NC(c1cncn1C)=O)C(C)C)Nc1c(C)cc(Cl)nc1 Cc1nc2ncnn2c(NC(C)CN(C)C(c2cccnc2O)=O)c1C C1(CNC(=O)CN2CCC2)CCCN(C(C2C(F)(F)C23CCC3)=O)CC1 c1(CC)ccc(O)c(C(N2CCC(N(C(=O)C(C)P(C)(C)=O)C(=O)OC)C2)=O)c1 N1(C(c2scc(-c3ccc(CC(=O)NC)s3)c2Br)=O)CCC(C)CC(C)C1 C1(CCOC)CN(C(=O)C(C)(C)SC)CCN1C(C1CC1c1ccc(C)cc1)=O n1(CC(=O)N(C2CCN(C(C3CC(=C)C3)=O)C2)CC#C)ccc(O)nc1=O N1(C(C(c2ccccc2O)OC)=O)CCN(C(c2ccnn2C(F)F)=O)CC1 c1(C(N2C(COC)CN(C(C3(O)COC3)=O)CC2)=O)n[nH]c2c1CN(C)CC2 c1(NC(=O)NCC(=O)NCC2(O)CN(C(C3C(CC)C3)=O)C2)c(F)cccc1F C1(C(=O)Nc2c(C)cc(NC(=O)CCn3ccnn3)cc2)CN(C)C(=O)CCO1 C#Cc1cnn(CC(=O)NC2(CCCC(=O)NCC(C)(C)N3CCC3)CCC2)c1 c1(CC(C)C(=O)NCC2CC(NC(c3cc(Cl)no3)=O)C2)ccc(Cl)cc1 CC(=Cn1ccnn1)C(=O)NC1CCC2CN(C(c3csc(O)n3)=O)CC2C1 C1(CNC(c2ccc(C#C)o2)=O)CC2(CC2)CN1C(=O)Cc1ccc(Cl)c(Cl)c1 C1(NC(c2c(C)ccs2)=O)CCC(C)(C)CC1CNC(C1COC1)=O C1(OC)CC(NC(C2CCS(=O)CC2)=O)CN(C(c2ccncc2C(F)F)=O)C1 C(C)(C)(C(=O)NCc1cc(C(N2CC(CC3CC3)C2)=O)n[nH]1)OC(C)=O C(CC(N)CC(C)(C)C)N(C(C1CCCCC1)C)C c1(OC)n[nH]c(=NC(=O)c2ncc(Cc3ccccc3)nc2C)cc1CO C=CC(C)(C)CC(=O)NC1CC(C)CN(C(c2nn(C)c(C3CC3)c2C)=O)C1 Cc1ccn2cc(C(N3CCC(N(C(=O)CC4CC4C4CC4)C)C3)=O)nc2c1C c1(C(=O)NCCN2CCN(C(CC3ON=C(C)C3)=O)CC2)c([N+](=O)[O-])cnn1C C=CC1(NC(=O)C(C)(C2CCC2)NC(c2ccon2)=O)CCCC1 C1(NC(C2CC23CCCCC3)=O)CC2CCC1N2C(=O)CCCc1ccncc1 c1(C(N2CCCC(OC)C2)=O)cc([N+](=O)[O-])sn1.C1(=O)CC(=O)N1C1CC1 C1(CC(=O)N(C)CC2CCN(C(c3ccc(C)o3)=O)C2)(CN(C)C)CCCCC1 CC1CN(C(C2CC2C2CN(C(=O)CC3CCCC(=O)C3)C2)=O)C12CCOCC2 n1(CC(=O)N(CCC(C)NC(=O)C=CC(=O)N(C)C)C)nnnc1C1CC1 C1(C(=O)OC(C)(C)C)(CC)CCCCN1C(C1C(C)C1(C)C)=O N1(C(CC(C)(F)F)=O)CCCC2(C1)CN(C(c1c(Cl)cnn1C1CC1)=O)CCO2 C1(CNC(c2c(CC)nccc2)=O)CCN(C(=O)CCOC(C)C)CC1C C1(C(=O)NCC(C)CNC(C2CC(=C3CCC3)C2)=O)OCC1(C)C C1(NC(=O)C=Cc2ccco2)CCN(c2ccc([N+](=O)[O-])cc2)CCC1CO c1(NC(C2CC(C(=O)NCCN(C(=O)OC)C)C2)=O)nc(C)ccc1F N1(C(COCC=C)=O)CCOCC(NC(=O)C=C(CC)CC)C1 N1(C(C(CCC)OC)=O)CC2(CCC2)CC1C(N1CC(OCC)CCC1C)=O C1(F)(CNC(C2CCS(=O)CC2)=O)CC2CCC(C1)N2C(C1CC2CCC1O2)=O CC1(C)CC(NC(=O)Cc2c(F)cccc2F)CN1C(=O)CCC1CC1(F)F C(=O)(C(CC)C(F)(F)F)NC1CCCN(C(c2c(CC)n(CC(C)C)nc2)=O)C1 C(=O)(C1=CCC(C)CC1)N1C(C(=O)NCCC2(COC)CCC2)CC(C)C1 C(=O)(NNc1cc(Br)ncn1)c1cc(C#C)c(C)nc1 C1(C(=O)NC2CC(C)CN(C(=O)C=Cc3cnc[nH]3)C2)CC2(CO1)CC(F)(F)C2 Cc1ccnc(C(N2CC(N(C)C(c3ncoc3C3CC3)=O)C2)=O)n1 S(=O)(=O)(c1cc(C(=O)N=c2cccn[nH]2)n(C)c1)Nc1ccc(OC)cc1 CC1CN(C(=O)C(O)Cc2cnc[nH]2)CC1CNc1cc(O)ncn1 C1(NC(c2c(OC)c(C)cs2)=O)CCN(C(C2CC3(CC3)CO2)=O)CC1(C)C N1(C(C(C)(C)n2cnnn2)=O)CC2(CCCC2NC(=O)CN2CCNC(=O)C2)C1 C1(C(N)=O)CC(=O)N(CNC(=O)CCOCCC2CC(NC(=O)C(=O)NOC)C2)C1 C(=O)(C(F)C(C)CNC(c1cc(O)ncn1)=O)N(CC(C)(C)O)CC C(=O)(C1=CCC(C)CC1)N1C(CNC(c2c(C)c(O)ccc2)=O)CC1 C1(C(C)C)CN(C(C2CC(O)C2)=O)CCC1NC(=O)CC1CCSCC1 C1(C(N2CCC(O)(c3cn(-c4cccc(Br)c4)nn3)CC2)=O)CC12CCCCC2 c1(C(=O)NCC2N(C(c3cnc(CC)[nH]3)=O)CC2)cnn2ccc(Cl)c(F)c12 CC(=O)CCN=C(NCC1CC1C(F)F)N1CCC(n2cncn2)C1 C(=O)(C(CC(N)=O)NC(=O)C(C)OC)NCC1(CCC)CCC1 C(=O)(C(C)(C)CC(F)(F)F)NCC1(CNC(C=C(C)C)=O)CCC1 c1(CC)nn[nH]c1C(=O)NC(C1CCCN1C(=O)C(C)SC)(C)C CC1CCN(C(=O)Cn2cc(C3CC3)cn2)C1c1cn(CC2CCC2)nn1 N1(C(c2ccc(CO)o2)=O)CCCC2CN(Cc3cccc(O)c3)CCC12 CC1=C(C)CC(C(=O)NC2(CNC(c3c(Cl)c(C)nn3C)=O)CCCC2)CC1 c1(C(=O)NCCOCCN(C)C)csc(C(=O)Nc2ccc(Br)o2)n1 C1(C)(CCC(=O)NCC(C)(C2CCC2)NC(=O)CCCn2ccnn2)CC1(F)F C(C)(C(CC(=O)NCC1(C(=O)N(C)C)CC1)NC(=O)CN=[N+]=[N-])OC c12cnccc1C(=O)N2.N1(CC)CCCC(c2cn(CCNC)nn2)C1 C1(C(N2CC(C)C(O)C2)=O)CC2(CC2)CN1C(c1sccc1Cl)=O N1(C(c2n(C(CC)C)ncc2)=O)CCCCC1CNC(c1cc[nH]c1C)=O C=CCCC(CC(C)C)C(=O)N1CC(CN(C)C(c2cocn2)=O)C2(CC2)C1 N1(C(C(C)OCCCCCC)=O)CCC(C)(C)C(CNC(=O)CCC=C(C)C)C1 C(C)(N=c1[nH]c2c(c(=NC3CCCn4ncnc43)[nH]1)SCC2)c1cc(C)oc1C N1(C(C=CC)=O)CCC2(NC(=O)CCOc3ccc(F)c(F)c3)CC2C1 C12(C(=O)NC(C)C(CO)NC(C3CC4CC4C3)=O)CC3CC(F)(C1)CC(F)(C3)C2 C1(CC(N2C(C(C)O)COCC2)=O)CN(C(=O)Cc2cnoc2)C(C)(C)C1 CC(C)CC(CNC(c1cc(CS(C)(=O)=O)on1)=O)NC(c1cscn1)=O N1(C(=O)C=CCO)CC2CCC1C1CN(C(C3(CF)COC3)=O)CC21 C1(NC(c2nccc3[nH]ccc23)=O)COC2(C1)CN(C(C1CCCS1(=O)=O)=O)C2 c1(CC(=O)NC(C)C(CO)NC(C2(C(F)(F)F)CC2)=O)cccc2c1CCC2 N1(C(C(C)NC(=O)OC)=O)CC(N(C)C(c2cc(C(N)=O)co2)=O)C2(CC2)C1 Cc1cc(C(N2CC(CCNC(C3(C#N)CC34CCC4)=O)C2)=O)nc(C)c1 N1(Cc2cnc(-c3c(OCC)cccc3)nc2)CC2CC(C(=O)OC)C1C2 CC(CCC(=O)NCCCCC1CN(C(c2cccc(COC)c2)=O)C1)S(C)(=O)=O CCCCC(=O)C(=O)NC(C)(C(=O)NCCCn1ccnc1C)C1CCC1 N1(C(C(C)C2CCOC2)C(=O)NCc2ccco2)CCCOCC12CCCC2 C1(NC(c2ccc(CSC)o2)=O)CC2CCC1CN2C(C1COCCO1)=O C=CCCC(C)(C)C(=O)NC(CNC(=O)CCc1cnco1)Cc1ccccc1 c1(OC)ncnc(OC)c1C(N1CC(N(C)C(c2coc3c2CSC3)=O)C1)=O O=C1CCC(C(=O)NCCOC2CCN(C(c3cc(C4(O)COC4)on3)=O)C2)C1 C(=O)(C(F)C(=O)NC(Cn1cccn1)C(=O)NCC1CCOCC1)OCC N1(C(C(N2C(CC)CCC2)=O)=O)CCCCC(CNC(=O)CCn2ccnn2)C1 N1(C(C)(C)C)CC(NC(=O)N(CC(O)CN2CCCC2)C(=O)C2CC2)CC1=O CC(C(C)(O)Cc1ccccc1)NC(=O)C(=O)NCc1ccncc1Cl N1(c2nc(Cl)ncc2Br)CCCC2(CC=CCC2)C1.c1(C=O)coc2ccc(Cl)cc12 c1(C(N(CCN(C(Cn2ccc(C)n2)=O)C)C)=O)cc2ncccc2o1 Cc1[nH]nc2c1CC(C(=O)NCC(F)(F)Cn1cc(-c3cc[nH]n3)nn1)CC2 C1(C(=O)OC)CCCCC1C(=O)NC(c1nn[nH]n1)C1CC1 C#Cc1ccc(C(=O)NCc2ccc(CO)cc2)o1.C1(C(=O)N)CC(OC)C(OC)C1 CN1C(=O)CN(C(C2(C)CCN(C(C3CC3[N+](=O)[O-])=O)CC2)=O)CC1=O Fc1ccc2nc[nH]c2c1CNc1nc(C2CCOC2)cs1 N1(c2c(C#N)ccc(Cl)n2)CCC2CCN(C(=O)CCc3cscn3)CC2C1 N1(C(CC2(C=C)CN(C(C3(CCCC)CCC3)=O)C2)=O)CCOC2COCC12 CN1CCN(C(C2(F)CC2)=O)CC1CNC(C1CC(F)CN1C)=O C(=O)(C(O)CC(F)(F)F)NCc1ccc(C(=O)NC2C(CC)COC2)cn1 C1(CNC(C(C)SCC)=O)CN(C(=O)Cc2cccc(NC(C)=O)c2)CC1O c1(SC)ccc(C(=O)NC(C)CCCNC(=O)C(F)(F)CN(C)C)c(Cl)c1 c1(CNC(CCSC)=O)n[nH]c2c1CN(C(c1cc(F)cc(C)c1C)=O)CC2 CCC(CC(=O)NCCCCCN(C)C(c1cc(C)n(C2CC2)n1)=O)C1CC1 C1(C(=O)NC(CC)CNC(=O)C(C)CF)CCc2ncnc(C)c2C1 c1(C(=O)OCCOCCN(C)Cc2nc(COC)[nH]n2)nc(C(C)C)cc(C)n1 c1(OC)ccc(C(=O)NC2CC(C)(NC(=O)C(C)CS(C)=O)C2)c(F)c1 c1(NC(C2N(C(c3[nH]cc(COC)c3)=O)CCCC2)=O)ncc(C)cc1Cl c1(OC)cc(C(N2CCOCCC2C(F)F)C(=O)NC2CC2)cc(OC)c1OC CC(C)C(C)CC(=O)N1CCN(C(c2ccc(N)c(N)c2)=O)C(CCO)C1 CC(F)(F)C(F)C(=O)NCC1(C)CN(C(c2cn(C3CCC3)nn2)=O)CCO1 CNS(=O)(=O)N1CCC(C(=O)NCCOCCN(C(=O)C(C)N2CCC2)C)CC1 C1(C#N)(C(=O)NCC(C)NC(c2cnn3ccsc23)=O)CCCOC1 C1(NC(c2sc(C)c(C)c2C)=O)COC2(CCN(C(=O)CN(C)C3CC3)C2)C1 N1(C(c2c(C)cc(C)[nH]2)=O)CC2CCC1CN2C(C1CC1c1cccs1)=O c1(OC)ccc2nc(C(=O)NC34CCC(CC3)N(C(=O)CC(C)CF)C4)cn2n1 C=C(C)c1cccc(NC(=O)C#CCNC(c2cc(CC)nn2C)=O)c1 C12(C(=O)NC3CCC(NC(c4ccc(C#N)s4)=O)CC3)CCCCN1CCC2 c1(C(N(C2CC(NC(=O)CC3CC34CC4)C2)C)=O)scnc1C1CCCC1 N1(C2CN(C(=O)COC(F)(F)F)C2)CCCN(C(c2cc(Cl)ns2)=O)CC1 C1(C(=O)O)CC2(CCC2)CN1C(C1CC12CC2(F)F)=O c1(NC(CC2ON=C(CC)C2)=O)ccc(NC(C2CNC(=O)N2)=O)c(C)c1 N1(C(=O)NCCC2CCOC2C2CC2)CCCNS1(=O)=O N1(C(COC(C)=O)=O)CC2(CC2)CC1C(=O)Nc1sccc1C#N C(=O)(CC1=CCCC1)NCC(CNC(C1CC(C(F)(F)F)C1)=O)OC c1(C(=O)NC(CC=C)CNC(c2cnc(C(C)OC)s2)=O)ncnc(OC)c1F C1(CNC(C(C(C)C)SCC)=O)C2CCC(C2)N1C(=O)COc1cccc(C)c1 N(C(=NCCCC(C)(C)O)NC1CC(C)(CC)C1)C(C=C)C CCCCCCC(CC)C(=O)N1CCCCC(C(=O)NCC2CC3C=CC2C3)C1 C1(C(=O)NC(C2(C(N3CCC3CN=[N+]=[N-])=O)CC2)C)CC2(CCC2)CO1 C1(CNC(C(c2ccccc2)OC)=O)CC2(CC(C(=O)O)C2)C1 NC12CCN(CC1)NC(=O)C(=O)NC2.C1(O)(CO)CCOCC1.c1(C)ccccc1 Cc1nn(CC(=O)N(CCCNC(=O)COC(C)(C)C)CCO)c(C)c1[N+](=O)[O-] C1(O)(CNC(C2(OC)CC2)=O)CCN(C(=O)CCc2cccnc2Br)C1 C(C)(C)(CCC(=O)N1CCOCC(NC(C2CC2(F)F)=O)C1)N(C)C CCCC(C(=O)N1CC2CCC1C(CNC(=O)CCCc1ncco1)C2)C(C)C N1(C(C2C(C(=O)OC)CC2)=O)CC(C(=O)NCCCn2nccn2)C(C2CC2)C1 c1(NC(C2(C)CN(Cc3ccc(F)c(Br)c3)C2)=O)ncc([N+](=O)[O-])cc1Br c1(CC)nnc2c(C(=O)NC(CNC(c3cc(Cl)cnn3)=O)CC)cccn12 C1(NC(C(C)=C2CCCC2)=O)COCC1NC(=O)Cc1cc(C)[nH]n1 C1(O)(CC(=O)NC2(CO)CN(C(C3CCC3c3ccccc3)=O)C2)CCCOC1 C1(C(=O)NCC(CC(=O)NCCOCCOCC)C)CC(=O)NC(=O)C1 CC(C)(C)C1=NOC(C(N2CC3COCC3(NC(=O)CSCC(F)(F)F)C2)=O)C1 c1(CNC(C(=O)NC(=O)NC(CC)C)C)ccc2c(c1)CCCN2C(C)=O N1(C(C(C)N(CC)CC)=O)CCC2(CC2NC(c2ccn(C)c(=O)c2)=O)C1 c1(C(=O)NC2(CNC(CCNC(=O)NC)=O)CCCC2)cnc(CSC)nc1O n1(CCC)cccc1C(=O)NC1CCC(CCNC(=O)Cc2n[nH]c(C)n2)C1 c1(C(=O)NCCC2N(C(C(C)CF)=O)CCC2)cccc2c1CCCC2 c1(C(N(C(CNC(CCSC)=O)C)C)=O)ccc2c(c1)N(C)CC2 N1(C(C2(C)CC2)=O)CCN(C(C2CCN(C(c3cccc(CO)c3)=O)CC2)=O)CC1 C=CCCCC(=O)NC(CCF)C(=O)NCCC1CCCN1C C1(OCC)CCN(C(=O)C(C)N(C(=O)CCCC2CC2)C)CC1 C(=O)(CC(C1CC1)NC(=O)CNC(C)=O)NCC(=O)NCCOC NC1CC(F)(Cc2c(CNC(=O)C(=O)NCc3cccnc3)c[nH]n2)C1 c1(N2CCC(C(C)(C)OC)CC2)cc(NCC2(O)CCCCCC2)nc(C)n1 CC(=O)CCCC(C)C(=O)N1CC(C2CN(C(=O)CC3CCCSC3)CCO2)C1 c1(C(N)=O)cc(OCC(=O)NC2CN(C(=O)C=C(Cl)Cl)CC2CO)cc(F)c1 C(C)(C(C(=O)N1CCOC(C)(CC)C1)C(C)C)NC(c1c(C)nc(CC)o1)=O CC1CCCCN1CCC(=O)NCCC1CC(NC(=O)C(C)N2CCC2)C1 N1(C(CCCCC=C)=O)CC(C)CN(C(=O)CC2(COC)CC2)C(C)C1 C#CC(CNC(c1ncoc1CNC(=O)C(C1(O)CCCC1)F)=O)CC(C)(C)C Cc1ccc(NC2COCCN(CC(=O)NNC(=O)Nc3nccs3)C2)c(Cl)c1 CCC(C(=O)N1CCC(C)(CNC(=O)CCCN2CCCCC2)C1)C(C)C CCC(CC)CCC(=O)N1CCCOC(CNC(C2CCCCS2(=O)=O)=O)C1 C1(NC(Cc2cc(C)no2)=O)CC2(C1)CC(NC(=O)C(C)(C)Cc1cnn[nH]1)C2 CN1C(=O)CCC1CC(=O)NCC1(NC(=O)C(C)Sc2ncccn2)CC1 C(=O)(CC(C)(CN(C)C)C(F)(F)F)NCC(N1CCCCCC1)C Cc1nsc(C(=O)NCC2CCC2C(=O)NCc2ccc(O)nn2)c1N Cc1nc(C)c(CC(N2CC(CNC(=O)CCc3cccc(O)c3)CC2C)=O)s1 C1(NC(c2c(CC)nns2)=O)CN(C(=O)CNS(=O)(=O)C2CC2)CC2(CCC2)C1 c1(C(N2CCC3CN(C(C(N(C)C)C4CC4)=O)CC32)=O)ccc(S(N)(=O)=O)cn1 N1(C(COC(C)=O)=O)CC2CCC1C(OC(=O)CCn1c(C)ccc1C)C2 c1(CCC)ccc(C(C)C(=O)Oc2ccc(C(=O)OC)cc2)cc1 Cc1ccccc1-c1nc(-c2cncs2)nn1CCCCO C(=O)(C(C)(C)C(C)(F)F)NC1CN(C(c2ccc(-c3ccc(C)o3)s2)=O)C1 c1(CCC(=O)NC2C3(CC(NC(Cc4nc(C)[nH]n4)=O)C3)C2)nnc(O)nc1O c1(CCC)ccc(Oc2ccc(C(=O)NC(C3CCCC(C)C3)CC)cc2)cc1 N1(C(CCc2cc(C)ncc2)=O)CCC2(CCC(C(N3CCC3)=O)CC2)CC1 c1(OC)ccc(C(N2C(C(=O)NCC(c3ccccc3)C)CC3CC23)=O)c(Cl)c1 C1(C(C)NC(=O)Cc2cnsc2)CCCN(C(=O)CCC2CCCCCC2)C1 C(=O)(C(O)C(C)(C)C)NCC(CNC(CSCC#C)=O)C c1(OC)cc(CC(=O)NCCCCC(C)NC(c2cncs2)=O)ccc1F N1(C(c2occ(C)c2)=O)CC2CCC1C1CN(C(=O)Cc3cncnc3)CC21 N1(C(CCC)=O)CCC2(C1)CN(C(C1CC3CCC1CC3)=O)CC(C)O2 CC(C)CCC(O)C(=O)N1CC(C(=O)NCc2nncn2C)CC(C)C1 Nc1c(C(=O)NC2CC2NC(C2CC3(CCCC3)CO2)=O)sc2ncccc12 C1(C(N2C(CN(C(C(=O)NC(C)C)=O)C3CC3)CCC2)=O)CCCCCC1 C1C(C(C)C)CC(=O)O1.C(CCC(=O)OC(C)(C)C)NC(=O)N.C(C)(C)(CC)OC C1(CNC(Cc2c(C)noc2)=O)CCC(C)CN1C(c1ccn(C)n1)=O c1(C2CCN(Cc3ccc(C)c(O)c3)CC2)ccc(C)c2ccccc12 C1(NC(=O)CC2C=CCCN2C(C2CC(OCCF)C2)=O)CCc2nn[nH]c2C1 N1(C(c2ncc(OC)cn2)C(=O)NC(CC)C)CCC(F)(F)C(C#N)C1 Cc1ncc(Br)c(N2CCC(NC(c3cc(N4CCCC4)ccn3)=O)CC2)n1 Cc1csc(C(=O)N(C)CC=CC(=O)NC(c2ccn(C)n2)(C)C)c1C N1(C(c2cnn(CC)c2C)=O)CC2(CCC2)CC1C(N1CC2CC2C1)=O C=CC1(C(=O)NCC(CO)NC(c2cnc(C(F)(F)F)cn2)=O)CCOCC1 Cc1c(-c2nn[nH]n2)cnc2c1N(C(=O)COC1CC1)CCO2 N(C(=NCCc1cccs1)NCCN1CC(C)OC(C)C1)C(COC)CC(C)C Cn1ncc(C(N2CCN(C(=O)CN3CCCC3=O)CC2)=O)c1OC(C)(C)C CC1C(NC(=O)CN2CCCCC2)C(C)CCN1C(C12CC=CC(C1)OC2)=O C1(NC(C(=O)N(CCCCC)C)=O)CCC(C#N)CC1 CN1CCCCC1C(=O)NC1CC(C(=O)NC2C3CCC2CC3)C1 C1(CC=C)(NC(=O)CSCCc2ccccc2)CCN(C(=O)C(CSC)OC)C1 C1(CNC(C2CCCC2)=O)CC12CCN(C(c1cc3c(s1)CCC3)=O)CC2 c1(C(=O)NCC(C)(C)NC(C(C2CC2)SC)=O)c(F)ccc(F)c1F C(=O)(C1CCCc2c(Br)cccc21)OC1CC(C)(C)C1 N1(C(C(C=C)OC)=O)CCC(CC)CC1C(N1CCCCCC1C)=O N1(C(C(C)=CC2CC2)=O)CC(C)(C)OCC1CNC(c1cncc(F)c1C)=O c1(CNC(C2CC(NC(C3=C(C)CC3)=O)C2(C)C)=O)ccc(C)cc1C N1(c2nc(O)n(C)c(=O)c2)C2CCCC1CN(C(C1(CN(C)C)CC1)=O)CC2 C12(NC(C(C)C3CC3)=O)CCCCC1CN(C(=O)Cc1cncc(Br)c1)C2 C1(CCC)CN(C(C2CCC(O)C2)=O)CCN1C(=O)C=NOC C12(C(=O)NCC(CNC(C(C)C(C)O)=O)CO)CC3CC(CC(C3)C1)C2 C1(C(=O)NCc2c(COC)nccn2)CNC(=O)CN1C(=O)CC=C(C)C N(C(=NCCS(=O)c1ccccc1F)NC1CCC1)C1CCN(C(C)=O)CC1 C1(NC(C(C)N(C(=O)CC(C)N(C)C)CCC)=O)CC2(CCCCO2)C1 Cc1nsc(C(N2CCCC2C=CC(=O)N(C(C)CN(C)C)C)=O)c1N c1(C(N2CCC(C)(NC(c3ccc(OC)nc3)=O)CC2)=O)cc(Cl)c(F)cc1O C1(NC(COCCCN(C)C)=O)CCC(O)CN(C(c2cnn[nH]2)=O)C1 c1(CC)ncc(C(=O)NCC2CC(O)CN2C(c2cccs2)=O)c(C)n1 CC1(C)CCCOC1CNC(c1[nH]ccc1CNC(c1ccnnc1O)=O)=O C(C1=NOC2CN(C(C3CC=CCC3)=O)CC12)NC(C1CN2CCCN1CC2)=O C(=O)(CC(C)C(F)(F)F)NC1(CNC(C23C(C(=O)OC)(CCC2)C3)=O)CC1 c1(C(N2CC(C(C)(C)O)(CNC(=O)CNC=O)C2)=O)cc(F)ccc1Cl c1(C(N2CCC(C(C)NC(Cc3c(C)non3)=O)C2)=O)cc(S(N)(=O)=O)c(C)s1 CC1(C(=O)NCC2(CC(N3CCOC(C(N)=O)C3)=O)CC2)CCC(O)CC1 C1(NC(c2c(C)nc[nH]2)=O)CC2COCC(C1)C2NC(=O)CC(C)C(C)C c1(C(N2CCC3CN(C(C4CN5CCC4CC5)=O)C3C2)=O)ccn2ccccc12 N1(C(COC(C)C)=O)CCC=C(C(=O)NC(C)CCN2CCCC2)C1 C(=O)(CC1CS(=O)(=O)c2cc(Cl)ccc21)N1C2(CC(=O)N1)CCCCC2 C1(NC(C(C)=CC)=O)CN(C(=O)Cc2ccoc2)CC2(CCOCC2)C1 C1(F)(C(=O)NC2C(C(=O)NCCC3(COC)CC3)COC2)CC=CCC1 c1(OC)ccc2c(c1)C(C(=O)O)CCN2C(C1CC12CCC(=O)CC2)=O N1(C(C(C2CC(F)(F)C2)OCC)=O)CCCC(NC(=O)C(C)NC(=O)NC)CC1 N1(C(c2c(NCC)cccn2)=O)CCC(NC(=O)Cc2cncnc2)C(O)C1 C(O)(C(F)(F)F)C1CC(NC(=O)NC2CCOC2)C1 N1(C(C2C(=C)C2)=O)C2CCC1C(NC(c1cccc(-n3nc(C)cc3C)c1)=O)C2 c1(C(=O)NC2CN(C(C(C)N(C(C)=O)C)=O)CC(F)C2)nc2ncccn2n1 c1(NC(C2C=CCN2Cc2c(O)cccc2Cl)=O)ccc2[nH]c(=O)ccc2c1 CC1(CNC(C2CCSC2)=O)COCCN(C(=O)CCc2ncc[nH]2)C1 C(=O)(C(C)C(=O)OC)N1CC(C(C(=O)N(CC(O)COC)CC)O)C1 N1(CC)CC(NC(C2(CNC(=O)Cn3nnnc3C)CCCO2)=O)C(C)C1 C1(C(=O)NCC2COCCN(C(C(C)=C(C)C)=O)C2)CCc2cnc(C)n2C1 C(=O)(C(C)CC(C)(C)C)N1CCC(C)C1CNC(=O)C(c1ccc(Cl)s1)C C#CCC(C(=O)NC(c1nc(C)oc1C)C)NC(C1CCC(C)O1)=O Cc1cc(C(=O)NC2CCCC2C(N2CCOCC(O)C2)=O)cnc1F N1(C(C2CCC(=C)CC2)=O)CC2CCCC2C1C(=O)NC1CCOC1C N1(C(C)=O)CC2CCC1CN2C(c1csc(C2CC2)n1)C(=O)NCCC#N C(=O)(C1=CCCSC1)N(CC(C)N(C(=O)CC1CC=CC1)C)C Cc1ccnnc1CN1CCC(c2noc(CC(F)(F)F)n2)CC1 c1(OC)ccc(C(=O)NCC2(NC(c3ncncc3F)=O)CCC2)c(O)c1 c1(C(N2C(CNC(Cc3ncc(C)s3)=O)CC(C)(C)C2)=O)scc2c1OCCO2 N1(C(C(C)N(CC(F)(F)F)C)=O)CCCC1CN(C(=O)CC1CCCC1O)C N1(C(CC(=C)C)=O)CCN(C(C2CCN(C(c3ccnnc3S)=O)CC2)=O)CC1 C(=O)(C1c2ccccc2C(=O)N1C)NC1CCN(C(C(C(C)C)NC2CC2)=O)CC1 c1(C(N(CCOCCN(C(CN(CC(C)C)C)=O)C)C)=O)ccn(C(C)(C)C)c1 c1(C(=O)NC2CN(C(C(CCC)OC)=O)CC2C)ccc(C(C)C)nc1F C1(CNC(C2(OC)CCCC2)=O)CC2(CCN(C(C3C=C3C)=O)CC2)CO1 c1(COC)ccc(NC(c2nc(-c3ccc(F)nc3)cs2)=O)cc1 C(c1ccc(Br)c(Cl)c1)=CC(=O)NC1(C)CN(C(CC(COC)C)=O)C1 C1(O)(CNC(C2(C=C)CC2)=O)CCN(C(=O)C(F)(F)COC)CC1 CCCCCC(O)C(=O)N1CCC(N2CCN(c3cc(O)ncn3)CC2)C1 C(C(C)NC(C1(CCF)CCOCC1)=O)(C(C)C)NC(c1cc(C)sc1)=O c1(C(N(CC(C)(C)C)CC(F)(F)F)=O)ccc(N)c2cnccc12 N1(C(c2ccc(O)c(Cl)c2)=O)CC2CCN(C(=O)Cc3ncccn3)C2C1 C1(C(N2CCCC(CNC(Cc3c(SC)cccc3)=O)C2)=O)CC(F)(F)C1(C)C c1(Cn2c(C(N(C3CCCCC3)CCC#N)=O)nnn2)cnc(C2CCC2)[nH]1 CCCC(CC)CCC(=O)N(CCNC(c1ccc2c(c1)C(C)CO2)=O)C1CC1 c1(CN2CCCC(C)C2C(=O)O)ccc2nccnc2n1 c1(C(N2CCN(C(C3(C(F)F)CC3)=O)CC2CF)=O)ccc(CO)cc1F O=C1CSc2ccc(C(=O)NC3CCC(NC(C4CCNC4=O)=O)CC3)cc2N1 N1(C(=O)CC2CC3(CCC3)C2)CCCN(C(c2c(O)cccc2Cl)=O)CC1 N1(C(c2c(F)ccc(C)c2)=O)CCS(=O)(=O)C(CCNC(C2CC2C(F)F)=O)C1 C1(CNC(c2nn(C)c(C3CC3)c2)=O)CCCN(C(c2ccc(Cl)nn2)=O)CC1 c1(CC=CCC(=O)NC2C(CNC(C3(CC=C)CC3)=O)C2)ccccc1Cl Cc1nc(C2CC2)[nH]c1C(=O)NCC(C)NC(=O)C(C)SC(F)(F)F Cc1cc(=O)oc(C)c1C(=O)OC(Cc1ccccc1)C(N)=O c1(OC)ccc(C)cc1C(=O)N(CCC(C)NC(=O)C(CCO)N(C)C)C N1(C(C(C)n2cccn2)=O)CC2CCN(C(=O)CCN3CCCCC3)CC12 CC1(C)COc2c(C(=O)NCCOCCCNC(c3n[nH]c(=N)[nH]3)=O)cccc21 Cc1cc(C(C)C)nc(=NCC(C)N(C)C(C2CC23CCc2ccccc23)=O)[nH]1 N1(C(C(CCC)C)=O)CCN(C(=O)C(CCO)N(C)C)C(CS(C)(=O)=O)C1 Cc1noc2ncc(C(=O)NC3CCC4CC3CN4c3cncc(Cl)n3)cc12 c1(C(=O)NCC(CC)NC(c2cscc2F)=O)ccnc(Cl)c1OC c1(C(N(CC(C)CO)C)=O)sccc1CNC(=O)C=CC1CC1 C#Cc1ccc(C(N2CC(F)(F)CC2C)C(=O)NCCC2CC2)cn1 C1(C(=O)NC)COC2(CCN(C(=O)NC(c3noc(C4CC4)n3)(C)C)CC2)C1 C1(COC)(CNC(=O)COCC2CCCOC2)CN(C(C2CC(F)C2)=O)C1 Cc1nc(C(=O)NC2(CF)CCN(C(c3cccc(O)n3)=O)C2)ccc1Br c1(C(N(C(CNC(c2cc(C)cc(Cl)c2N)=O)C)C)=O)ccc2nnc(S)n2c1 c1(C(=O)NC2CCN(C(C=C(CCC)CCC)=O)CC2)ccccc1S(C)=O Cc1ccc(-n2ccc(C(N3CCSCC3CCNC(=O)C(C)(C)F)=O)n2)cc1 C1(CNC(CN(C2CC(C#N)C2)C(c2cc(C3CC3)on2)=O)=O)CCC(F)(F)C1 C1(CCC)CCCCN1C(=O)CC1(CNC(c2ccccc2COC)=O)CC1 c1(C(N2CCC(C(F)(F)F)C2)=O)n[nH]c2c1CN(C(c1sccc1F)=O)C2 N1(C(C(=O)NCC(CC)(c2ccccc2)c2cccs2)=O)CCC(CO)C1 C1(CO)(CNCC2(Br)CC2(F)F)CCCO1 CC1(C)C(NC(=O)C(F)(F)c2ccccc2)CCN1C(c1ccc[nH]1)=O N1(C(C(C2CCCCC2)C)=O)CCC(C)(C)C(C(=O)NCc2nncn2C)C1 c1(C(=O)NCC(C)N(C(=O)Cc2csc(Cl)c2)C)cncn1C C12(C(=O)NCC(CCOC)NC(C3CC4CC3CC4O)=O)C3CC(CC13)C2(F)F N1(C(C(C)OC)=O)CCCC2(CCCN(c3ncc4c(n3)CCC4)C2)C1 Cc1c(C(=O)NC2CCC(C)N(C(=O)COCC3CCC3)C2)cccc1Cl C1(CNC(C2CC(C)OCC2)=O)CN(C(=O)Cc2cccc(C#N)c2)CCN1C C12(CNC(C3ON=C(CC)C3)=O)CCC(C1)N(C(=O)Cc1c(F)cccc1Cl)C2 C1(NC(c2cnc(C(C)O)s2)=O)CC2(C1)CN(C(=O)CC(C)C(C)C)C2 C1(CNC(=O)C2=CCSC2)CCCCN(C(c2coc(C3CCCC3)n2)=O)CC1 Cc1c(C(N2CCC(C3CCCN3)C2)=O)nn(C)c1N.C(c1cnn(C)c1C)=C c1(CC)c(C(=O)NCC2CCN(C(=O)CC(C)(C3CCC3)N(C)C)C2)nnn1C C1(C(=O)NCCC(COC)C)CN(C(=O)CN2CCCCC2C)CC1C c1(-n2cc(CN3CCCC(F)(C(=O)OC)C3)nn2)cccc2c1OC(C)(C)C2 N1(C(c2cn(CC)nc2)=O)CCC(C(=O)NC2C3CCCC23)(CF)C1 C12(C(=O)OCC)CCC(n3cc(CCO)nn3)(CC1)C2.C12CC1C1CC1C(=O)N2 Cc1c(C(N2CC(C(C)NC(=O)Cc3ccc(C(N)=O)cc3)C2)=O)cncc1F C1(C)(CCC(=O)N(CC(O)CNC(C2CCCC2)=O)C)CC1(F)F N1(C(C2C(CC)CCC2)=O)CCC=C(C(=O)N(C2CCN(C)C2)C)C1 N1(C(CCOCCNC(c2nc(C)c(C#N)cc2)=O)=O)C2CCC1CC1(C2)N=N1 Cc1cc(C)c(C(N2CC(NC(c3ccoc3CC(N)=O)=O)C(O)C2)=O)c(C)c1 CN1CCOCC1CNCC1CCCOCC1 c1(C2(C(=O)NCC(CC)NC(=O)CSC3CCOC3=O)CC2)ccc(F)cc1F C12(C(=O)NC3CC(C)(NC(c4c(OC)cccc4)=O)C3)CCC(C1)C(C)(C)O2 N1(C(Cc2scc(C)n2)=O)CCC(C(F)(F)F)C(NC(c2csc(=N)[nH]2)=O)C1 Cc1ccc(C=CC(=O)NCCCC(C)NC(=O)C(C)(C)c2cccnc2)s1 C(=O)(C(C(C)NC(=O)OC(C)(C)C)C(C)C)OCc1c(OC)ccc(Cl)c1 Cc1cc(=NC(=O)NCC2CCCOC2C(C)(C)C)[nH]n1C(c1ccccc1)C C1(Oc2c(C)cccc2)CCN(N2CCC3(CCC3)CC2)CC1 C=C(C)C(C)(C)C(=O)NC1CCC1NC(=O)CC1(c2ccccc2)CC1 CC1(C(=O)Nc2ccc(N3N=CCC3=O)cc2)CCN(C(c2cnsn2)=O)C1 N1(C(C(CC)C#N)=O)CC(C)(C)C(NC(=O)C(C)n2cccn2)C(C)(C)C1 c12ccc(cc1)CC(=O)N2CC.C1(SCC)CCN(C(=O)CCC2OCCO2)C1 C1(CC)CN(C(=O)NCCC2CCC(C(=O)OC)CC2)CCC1C(=O)NC CC(C)(O)CC(=O)NC1CC(O)(CNC(c2cn(CCCF)nn2)=O)C1 N1(C(Cc2c(C)ncs2)=O)CCC2CCCC12CNC(=O)CCCS(N)(=O)=O N1(C(C(CC)(C)C)=O)CC2(CCCN2C(c2cccc(OC(F)(F)F)c2O)=O)C1 C1(C(=O)NCC(C2CC2)OC)(NC(C2CC(SC)C2)=O)CCSC1 c1(C(=O)NC(CNC(C(CC)NC(N)=O)=O)CO)cc2cc([N+](=O)[O-])ccc2o1 c1(C(=O)NC2CN(C(c3n(CC)ncn3)=O)CC(O)C2)cccc2ccn(C)c12 c1(C(=O)NCCCCC(CO)NC(C2(OC)CCC2)=O)ccc2c(c1)CCCS2 C1(=CC(=O)NCC2C(NC(C3N(CC)CCC3)=O)CCCC2)CCC(C)(C)CC1 C1(NC(c2c(C)noc2)=O)CCC(CNC(c2cncn2C)=O)CC1 c1(C(C)C)nc(CN(C(c2sccc2Br)C(=O)NC2COC2)C)cs1 C(CN(C(=O)Cc1csnn1)C1CC1)(CC(F)(F)F)NC(=O)COc1cccnc1 C#Cc1ccnc(C(=O)N(C2CN(C(=O)CCC(C)CN(C)C)C2)C)c1 C12(CNC(CCSCCC)=O)CCCC(CN(C(=O)C(O)CSC)C1)C2 c1(C(CNC(=O)Cc2cccs2)NC(=O)CCc2nncs2)cccc(Cl)c1 C1(NC(CCc2cccc(-n3cc(CCCOC)nn3)c2)=O)CC2OCCCC12 C1(C(=O)NC2(CCNC(c3cc(C)ns3)=O)CCC2)CCCC2(CC2)C1 C12(CNC(c3c(C)nn[nH]3)=O)CCC(CN(C(c3cc(=O)n(C)cn3)=O)C1)C2 C1(N2CCN(C(C3C(C)CC4CC4C3)=O)CC2)CCC2CNCCC2C1 c1(C(N(CCCNC(C2C(CCC)CCC2)=O)CCO)=O)cc(C)c(Cl)cc1F S(=O)(=O)(c1ccc(O)cc1)N1CCC(C(=O)Nc2c(C)nccn2)C(O)C1 Cn1cc(C(F)(F)F)c(Cc2ncccn2)n1.c1(CNC(=O)NC)ccccc1 N1(C(CC2(CC)CCC2)=O)CC(NC(c2cnn(C(C)C)c2C)=O)CC2(CC2)C1 C1(C(=O)NCC2(Cn3cc(Cn4cccn4)nn3)CC2)CC2(CCC2O)C1 C#Cc1ccc(C(N2C3CCC(C3)C2C(N2CC3CC2CN3C)=O)=O)c(Cl)c1 N=c1[nH]cc(CCC(=O)NCC(O)CNC(=O)CC2COCCO2)[nH]1 N1(C(c2scc(COC)c2)=O)CCCC(NC(=O)CCC2CCOC2)C1C C1(O)(CNC(=O)C(c2ccccc2)O)CCCN(C(=O)CCc2nccs2)CC1 C12(C(NOCC(CC)C)=O)CC(C)(CN1C(=O)CN(C)C(N)=O)C2 C(=O)(C1=CC2(CCOCC2)C1)NC1CC2(N(C(C(CC)SC)=O)CCCC2)C1 c1(OC)ccc(CC(N2CCC(=CC(=O)NCCCCSC)CC2)=O)cc1 c1(C(=O)NC(C(C)NC(C2(CC=C)CCCC2)=O)C)cc(C)ccc1[N+](=O)[O-] C1(CC)(NC(=O)CC#N)CN(C(=O)C(F)CC2CCOC2)C1 c1(C(C(=O)N(CC(COC)C)C)NC(=O)C(C)NC(N)=O)ccnn1C c1(C(=O)NC(CNC(c2c(OC)c[nH]n2)=O)C2CC2)ccc2nc[nH]c2c1 C1(C)(C(=O)OC)CC(Nc2sc(Br)cc2F)CN1C(=O)C1CC1 c1(C(=O)NC(CN(C(c2c(C)coc2C(C)C)=O)C)C)c(Cl)ccc2c1OCO2 C1(NC(c2n(C(C)C)cnc2)=O)CN(C(C2CC(O)C2)=O)CC1c1cnn(C)c1 Nc1c(C(N2CCC(F)(CNC(=O)C(F)=CC3CC3)C2)=O)cnc2ccnn12 c1(N2CCCC(C(=O)Nc3cccc(C)c3Br)C2)[nH]cnc2nc(Br)cc1-2 C1(OCC#C)CCN(C(c2c[nH]nc2CCNC(=O)C(COC)OC)=O)C1 Cc1ccnc2c(C(N3CCC4(C(N5CC6CC6C5)=O)CC4C3)=O)cccc12 C1(NC(C2(COC)CCCO2)=O)CC2CC(C1)N(C(=O)Cc1ccccc1F)C2 C1(O)(C(C(=O)NCc2c(C)nn[nH]2)NC(=O)CC2CC3(CC3)C2)CCCCC1 C1(NC(c2ccoc2Cl)=O)CCCC(C(N2CCCC(CO)C2)=O)C1 C1(NC(C2CC23CC3)=O)CCC12CN(C(=O)C=CCCc1ccccc1)C2 C=C1CCCN(C(=O)C(CC)NC(C2CCCN2C(C)=O)=O)C1 N1(C(C=NOC)=O)CC(NC(c2cnn(CC(F)(F)F)n2)=O)C(C2CC2)C1 CC(CC(=O)NC1C=CC(C(=O)NC2COC(C(F)F)C2)C1)C(F)F C1(NC(CCC(N)=O)=O)CCOC12CCN(C(C1CCNC(=O)C1)=O)CC2 c1(C(=O)NC2CC(C)N(C(c3ccc(Cl)c(Cl)c3N)=O)C2)cccc2cncn12 c1(C(N2CCC(CCN(C(C=C(C)C)=O)C)CC2)=O)cccn2ncnc12 c1(C(N(C2CC(NC(C3CCC(=C)CC3)=O)C2)C)=O)cccc2c1CNC2=O c1(NC(c2nc(C(F)(F)F)cc(C)n2)=O)cc(F)cc(F)c1F C1(CCOC)CC(c2nnnn2C)(Nc2cnn(CC(F)F)c2C)CCO1 N1(C(c2cc(C)on2)=O)CC(NC(=O)COCCc2ccccc2)CCC(O)C1 c1(CC)[nH]nc(C(=O)NCC2CCN2C(=O)Cn2ncnc2C(C)=O)c1[N+](=O)[O-] CS(C)(=O)=Nc1cnn(CC(N2CC3(CCC3)C2c2ccco2)=O)c1 N1(C(c2nc(CC)[nH]n2)=O)CCC2CCC(C1)N2C(=O)Cc1cncc(F)c1 S(=O)(=O)(c1cc(C)cnc1NCC(C)CC1CC1)NCC=CCCC CCC(CNC(C1CC1C)=O)(CC)C(=O)N1CC(COC)C1 C(C)(C)(CC(=O)N1CCCC(CN(C)C(C2C3CCCC23)=O)C1)SC N1(C(C(C=C)CC)=O)C(C(N2CCC2C2CCC2)=O)CC2CCCC12 c1(C(=O)NCC23CC2CN(C(=O)CCN2CCOCC2=O)C3)cc2c(s1)CCC2 C1(NC(Cc2c(C)ncs2)=O)C2CN(C(=O)C(C(C)C)n3cnnc3)CC12 C1(C2CCOCC2)(COC(C(C)OCCC(C)C)=O)CC1 N1(C(c2ccc(CC)[nH]2)=O)CC2CCC1CN2C(C1CCCC1F)=O C1(CNC(CCN(C(C)C)C(c2cccc(CO)n2)=O)=O)CC12CCOC2 C1(C(=O)O)(NC(=O)OC(C)(C)C)CSC1.N12CCC1C2 N1(C(CN(CC=C)CC=C)=O)CCC(C(N)=O)CC1 S(=O)(=O)(c1ccc2c(c1)CC(=O)N2C)NCC(N1CC2COCC2C1)C CCCC(O)CC(=O)N1CC=CC(NC(c2cccc(SC)c2Cl)=O)C1 C1(NC(c2c(C)nns2)=O)CC2CN(C(=O)CCC(C)(C)F)CC2C1 C(=O)(C1=NOC2(CCC2)C1)N1C(CC(=O)N(CCN(C)C)CCO)CC(O)C1 CCCCCC(F)C(=O)N1CCC(C(=O)NCCc2ccc(C)s2)(CO)C1 C(c1ccc(Cl)cc1F)=CC(=O)NCC12CC(NC(C(CCCC)O)=O)(C1)C2 c1(C(=O)NC2CC(CCNC(=O)CC3CCC(O)C3)C2)ccc2nnn(O)c2c1 CCCC(C(=O)NCc1cc(OC)ns1)NC(=O)CC(C)F CC(C)CC(C)C(=O)NCC1C(C)CCN1C(c1ccc(-n2cncn2)nc1)=O c1(C(=O)N(CC2N(C(C=CC=CCC)=O)CCC(C)C2)CC)cc(F)c(C)cc1N C(=O)(CN=c1cc[nH]cc1)N1CC(C)OC(C(N2CCCC(C)C2)=O)C1 C1(NC(CN(C)C)=O)CCS(=O)(=O)C2(C1)CC(CNC(=O)C(C1CC1)N(C)C)C2 N1(C(C(CC)C#N)=O)CCC(C2CC2)(CNC(c2ccc(OC)s2)=O)C1 N1(C(C=CCN(CC#C)C)=O)CC2(CC2)CC1CNC(=O)CCC1CC1C c1(NCc2c(C)noc2)ncccc1S(=O)(=O)NC1CCC(C(C)C)CC1 C(C(=O)NCCN(C(c1cncc(C(=O)OC)c1)=O)CC)(C(C)C)OCC N1(C(C2CCN(C)CC2)=O)CC(NC(=O)CSc2cnn(C)c2)CC(F)C1 C1(NC(c2c(C(C)C)cco2)=O)CCCN(C(=O)CCc2nncn2C)CC1 N1(C(C(CC#C)(C)NC(c2n[nH]c(C)c2Cl)=O)=O)C2CCC1CC1(CC1)C2 C1(CNC(C(C2CCC(=O)N2)C)=O)CCN(C(C2CCSCC2)=O)C12CC2 C(=O)(CCCC(=O)NCC(C)(C)NC(c1sc(C)c(Br)c1C)=O)OC CCC(C)(O)C(=O)NCC1CC(O)CN1C(=O)C(c1ccccc1)OC C1(C(=O)NC2CN(C(=O)OC(C)(C)C)C2)CCN(C(C2CC2(F)Cl)=O)CC1 n12cc(nn1)CC(=O)N(N1CCCC1C(=O)O)CC2C.CC(C)C(O)c1cccs1 C(=O)(C(C)CC(C)(F)F)NCCC1N(C(C(C)SCCCC)=O)CCC1 c1(OC)cccc(O)c1C(=O)NCC1CCN(C(=O)Cc2cccnc2)C(C)C1 c1(N2CCC(CC(N3CCCC(C(=O)OC)CC3)=O)C2)nc(Cl)nc2[nH]cnc12 N1(C(CCOCCN(C)C)=O)C2CCC1C(CNC(=O)CCN1CCCC1=O)C2 CC1CCN(CCSc2ccn(C)c(=O)c2)CC1C(F)(F)F Cc1onc(-c2ccccc2)c1C(N1CCC(CNC(c2ccnnc2)=O)C1)=O C(=O)(CC(C)CC(C)(C)C)N(C(C)CNC(c1cnc(C2CC2)nc1O)=O)C C(=O)(CCCC(C)(C)CC)N1C(CNC(C(CC)OC)=O)(COC)CCC1 C1(CNC(c2c(CC)[nH]cc2)=O)CC2CCC1N(C(=O)CC(C)C1CCCO1)C2 CC1CN(C(C2(C)CCCO2)=O)CC2(CCN(C(=O)Cc3cccc(N)c3)C2)O1 C1(NC(C2(C)CC(F)(F)C2)=O)CC2CC(C1)N(C(=O)Cc1ccc(F)c(Cl)c1)C2 C12(C(N3CCC(N(C(c4cn(CC)nc4)=O)C)C3)=O)CC(C)(C1)OC2(C)C C1(C(=O)NC23CC(OCC)(C2)C3)(CNC(=O)CC2CC2C(F)(F)F)CCCCC1 c1(C(=O)OCc2cc(C(F)F)n[nH]2)sc(C(F)(F)F)cc1Br c1(OC)cc(O)ccc1-c1ccc(C2CCN(C(=O)CC(C)(C)O)C2)cc1 CC1CN(C(=O)CN2CCCNC2=O)CC(C)N1C(C1CC12CCOCC2)=O N1(C(c2c(C)occ2)=O)CCN(C(=O)CCCCNC(N)=O)C(C)C1 C1(=CC(=O)NCC2COCCN2C(C2COCCO2)=O)CN2CCC1CC2 C1(NC(CS(N)(=O)=O)=O)CN(C(C2CC2(F)F)=O)C2(CCC2)C1 C(C1=CCN(CC(c2ccc(F)cc2)O)CC1)NC(c1c(C)nns1)=O c1(C(=O)NC2CC(Nc3ncc(C#N)cn3)C23CCC3)ccc2nc(O)[nH]c2c1 CCC(CC(F)F)C(=O)NCCOCCNC(c1cc(Br)c(C)s1)=O N1(C(c2[nH]nnc2C)C(=O)NCCCSCC)CC2(CCCC2)C1C(C)C O=C(C1CCCc2cncn21)N1CCC2OCCN(C(c3cocn3)=O)C2C1 C12(C(=O)NC(CNC(C(=Cc3ccccc3)OC)=O)CO)CCC(CC1)C2(C)C C(CCC(O)C(=O)NCc1ccc(C#N)cc1)NC(CC=CC(C)(C)C)=O C(=O)(C#CC1CCCC(NC(=O)OC(C)(C)C)C1)OCCC(CSC)O N1(C(C(CC)C)=O)CC(CNC(=O)CCN2CCN(CC)CC2)OC2(CCC2)C1 CC1(C)CCC(CC(=O)NCC2(C)CCC(NC(c3ccnnc3O)=O)C2)CC1 C12(NC(c3cn(CC)nn3)=O)CCC(C1)N(C(c1[nH]nnc1C)=O)C2 CCCCC(F)(F)C(=O)NCC(CC(C)C)C(=O)N1CC(=O)NC(=O)C1C C(=O)(CCCS(C)(=O)=O)NC1C(CNC(CCCN(C)C)=O)CCCC1 c1(CC(=O)NCCC(C)CCNC(c2cscn2)=O)cccc2ccoc12 Cc1cc2scc(CC(=O)NC3CC(CNC(C4CCC(C)(C)OC4)=O)C3)c2s1 c1(CN2CCCC2)cc(Cl)cc(I)c1.CC12CCCN1C(=O)N2 c1(OC)cc(CNC2CCC(C(=O)NCC(C)(F)F)CC2)cc(F)c1F Cc1nc(O)c(C(=O)NCC2CC2NC(=O)C(C)OC2CCCC2)cc1Br N1(C(C2CC=CCC2C)C)CCCCC12CCN(Cc1ccccc1)CC2 CCCCCCC(C)C(=O)NOCC(=O)NCCCc1nncn1C c1(CNC(C2C3CN(C(c4ncn(C)n4)=O)C2C3)=O)ccc(C(F)(F)F)c(F)c1 c1(C(=O)NC2CC(NC(c3c(CC)ncs3)=O)C2)n[nH]c2c1CC(C)(C)C2 c1(CC)ccc(C(=O)NCC(CCOC)NC(C2(c3ccnn3C)CC2)=O)[nH]1 C1(OC)CCC2(C(=O)N(C3CCN(C(c4ccc(C(N)=O)o4)=O)C3)C)CC12 CC1CN(C)CCCN1C(=O)CCC1CCCN(C(=O)Cc2ccc(O)cn2)C1 CC(C)(CS(C)(=O)=O)C(=O)NCC1CCCCN(C(=O)CN2CC3CC3C2)CC1 c1(C(N2CCC(O)(C(=O)Nc3c(C)ccnc3Br)C2)=O)c(O)ccc(F)c1F C(=O)(C(S(C)(=O)=O)C1CC1)N1CCC(COC(c2c(OCC)scc2)=O)CC1 c1(C(C(=O)N2CC(N(C(=O)CCN3CCOC3=O)C)C2)O)cccc(Cl)c1 Cc1ccc(C(=O)NC(CC(F)F)c2ccccc2)cc1-n1cnnn1 C(=O)(C#CC(C)(C)O)NC1CCCC(N(C(=O)Cn2cc(C(F)(F)F)cn2)C)C1 C1(CNC(C2C(C)C2)=O)CC2CCC(C1)N2C(C1(C)CC1(F)Cl)=O N1(C(COC(C)(C)C)=O)CC2CC(C1)N(C(c1cc(C#N)c(N)cn1)=O)C2 c1(C(=O)NC2(CNC(c3ccnc4[nH]nnc34)=O)CC2)cc2cc[nH]c(=O)c2s1 c1(C(=O)NCC(CC)NC(c2cc(O)nc(Cl)c2)=O)cc2c(C)cccc2[nH]1 N1(C(CC2C(C)CCO2)=O)CCOC(CN(C)C(C2CC3(CCC3)C2)=O)C1 c1(C(=O)OC(C)(C)C)nccnc1C(=O)OCC(N1CC(c2ccccc2)C1)=O N1(C(c2noc(CC)c2C)=O)CCCC(O)(CNC(=O)Cc2ccnc(O)c2)C1 C1(OC)CC(F)CN(C(c2cc(CNC(=O)C=CC(F)F)nn2C)=O)C1 C12(C(=O)NCC3(O)CCN(C(C(C)C(C)(F)F)=O)CC3)CCCCC1NC(=O)C2 N1(C(c2nc(CC)sc2)=O)CCC2CCN(C(=O)C(C)CCCC(C)C)C2C1 N1(C(c2cncc(COC)c2)=O)CC2CCC1CC2NC(=O)C(C)S(N)(=O)=O N1(C(c2cnc(SC)nc2O)=O)CC2CCC(C1)N2c1nnc(C#N)s1 N1(C(c2cccc(OC)c2N)=O)CCN(C(=O)C(C)C(C)(F)F)CC(CO)C1 c1(C(N2CC(O)(CNC(c3c(OC)nccc3)=O)C2)=O)cc(F)cc(N)c1F c1(C(N2CCCC3(NC(C(CCC)C)=O)C(C2)C3)=O)cc(F)c(F)c(O)c1F CC1COCC(CC(=O)NCC2(F)CN(C(c3cn(C(F)F)cn3)=O)C2)O1 Cc1nnc2c(C(N3CC=CC(NC(c4cc(Br)n(C)n4)=O)C3)=O)cccn12 C#CCC(O)C(=O)N1CC(C2CN(C(=O)CCCCc3cccc(O)c3)CCO2)C1 C1(C2CCS(=O)(=O)CC2)(NC(C=Cc2n(CC)ncc2)=O)CC1 CC1(C)CC(CNC(C2CCCC(=O)N2)=O)CN(C(=O)CCc2csc(=N)[nH]2)C1 N1(C(C(C#C)(C)C)=O)CCCC(CNC(=O)C(C)Cc2ccc(Cl)cc2)CC1 CCCCCCC(C)C(=O)NCCC1(C(=O)N(CC(O)CO)C)CC1 c1(CC(CC(=O)OC)NCCCC2CCCCN2)ccc(F)c(Cl)c1 CC1=C(C(=O)N2CCCCC2CCCNC(c2csc(O)n2)=O)CC1 C1(NC(CCc2cnc(C)s2)=O)CCCCN(C(c2ccc(CF)cc2)=O)C1 N1(C(C2C(CNC(c3occ4c3CCC4)=O)CCO2)=O)CCCC(F)CC1 C(=O)(C(C)(C)C(C)(F)F)NCC(C(=O)NCCc1ncn(CC)c1)(C)C c1(C(N2CC(C)C(NCc3ccc(-n4cccc4)cc3)C2)=O)cc2c(s1)CSC2 C1(C(N2CCCC2c2cn(-c3ccc(Br)c(Cl)c3)nn2)=O)CCc2nnc(O)n2C1 O=C(CCN=C(NCCSc1ccc(F)cc1)NC1CCCC1)OCC1CC1 Cc1cc(C(=O)NC2CCCC2CNC(C2(C)CCCCC2)=O)cc(N)c1O C(=O)(C(CC)C(=O)N1CCC1CNC(c1cn(CC)nc1C)=O)OCC c1(C(N(C2CCCN(C(C3(OC)CCCCC3)=O)C2)CC)=O)cn(C)c(O)n1 C1(C(=O)Nc2c(OC)ccc(S(C)=O)c2)CCc2cc(Br)ccc2NC1=O C1(n2ncc(C(=O)NC(CNC(C(=O)NCC)=O)CC)c2)CCS(=O)(=O)C1 C1(N(C(=O)NC(c2cccs2)C)CCF)CCOC1 C1(CC=C)(C(=O)N(C)CC2CC2(C)C)CCN(C(=O)CCC=C(C)C)C1 C(C)(C)(C(=O)NCc1cc(C(=O)NCC2=CCCC2)no1)OC CC(C)CC(C(=O)NCC(C)OC(F)F)ONC(=O)CCc1cscn1 C1(C)(C(N2CCCC(CN(C(CC3(OCC)CCC3)=O)C)C2)=O)CCN(C)C1=O C#Cc1ccccc1CC(N1CCC(CO)C(NC(C2(CO)CCOC2)=O)C1)=O CC1=NS(=O)(=O)NC=C1C(=O)NCC1(C(N)=O)CN(C(C2CCCSC2)=O)C1 Cc1ncc(C(=O)NC2CC2NC(=O)C(C(C)C)C2CCC2)c(C)n1 C(N=c1[nH]c(=NCCOc2nncs2)c2sccc2[nH]1)C1C(C)(C)OCCO1 C#Cc1cncc(C(=O)N(CCCN(C)C)CCNC(c2ccnc(S)c2)=O)c1 C1(NC(C(n2cc(Cl)cn2)C)=O)CC2(C1)CC(NC(=O)CC1SC(=N)NC1=O)C2 c1(CN2C3CCN(C3)C2=O)ncccc1OC(F)F.CC(C)CCOC(C)(C)C CC(C)(C)CCC(=O)NC(CNC(c1ccc(-c2ccc(Cl)s2)cn1)=O)C1CC1 Cc1ccc2c(c1)C(CNC(=O)C(CN(C)C)N(C)C)CC2 c1(C=O)ccccc1-c1nc[nH]n1.c1(C(C)OC)noc(CN(C)CCl)n1 O=C1CCC(CC(=O)NC2(CF)CCC2)N1.C12(CC1)CC(=O)N2 C=Cc1cnn(C)c1C(=O)NCC12CC(CO1)N(C(C1CCOC(=O)CC1)=O)C2 N(C(=NCCC1CC2C=CC1C2)NCC12CCCC1C2(F)F)CCOCC c1(C(=O)NCC2CN(C(c3cn(C)c(=O)cn3)=O)CC2O)occ2c1CCCC2 c1(OC(C)C)nccc(C(=O)NC2CCC2NC(=O)C(C)N2CCCC2)c1F C1(NC(Cc2c(OC)ccc(F)c2)=O)CCN(C(=O)CSC)CC12CCC2 C1(CNC(COCCSC)=O)COCCN(C(c2cc(OC)nc(F)c2)=O)C1 C1(C(N2CCC(C(C)NC(c3csnn3)=O)C2)=O)Cc2cncn2C(=O)N1 CCC(C)(C)C(O)C(=O)N1CCCC(CN2CCN(C(=O)CC3(C)CC3)CC2)C1 N1(C(C(C)SCCCC)=O)CCCCC12CN(C(=O)Cn1cncc1C)C2 c1(CC(=O)NCCCN(C(C)C)Cc2cncn2C2CC2)ccc(Cl)c(F)c1 C1(C(=O)NCCC2(NC(CCCOCCOC)=O)CC2)CC2CC1CC2O c1(NC(C2(C#C)CN(C(=O)C(Cl)Cl)C2)=O)cc(C#N)ccc1O c1(C(=O)NCC(CNC(c2c(Br)n[nH]c2C)=O)OC)cnc(N)c(N)c1 CCC(F)C(=O)NCC(C)CN(C(=O)CCSCc1ccccc1)C C(=O)(CC(C)(C)C(=O)NCC1CCN1C(C1CC2(CCC2)C1)=O)OC c1(CNC(C(CCC)OCC)=O)nnc2n1CCN(C(C1CC1F)=O)C2 c1(CC)cccc(C(=O)NCC(C)=CC(=O)NC(c2cnc(C)s2)C)n1 c1(CN(c2ccc(Br)cc2)CCCC)ccc(Cl)c(C)c1OC C(C1=NOC2(CCN(C(=O)OC(C)(C)C)C2)C1)Sc1cnc(C(C)=O)s1 c1(C(N(C2CCN(C(=O)C(CC)=CC)CC2)CC#C)=O)cc(C)c(Cl)cn1 C12CC13CCN(C3)CC(=O)N2.c1(N)ncc(Cl)cc1Cl.c1(OC)ccccc1O C1(C)(CNC(CN(C(=O)CCc2conc2C)CCC)=O)CC2CCC1C2 N1(C(=O)CN2CC=CC2)CCN(C(=O)CC2CCC2)C2(CC2)C1 CC1(C)CCC(C)(C(N2CCC(CNC(=O)C(c3cccnc3)O)C2)=O)CC1 c1(N2C3CC(CNC(CC(C)c4ccccc4)=O)C2CC3)cc(O)nc(=O)n1C c1(N2CC(NC(c3cccc(C(C)=O)n3)=O)C(C)C2)nnc(C)c(C)n1 C1(CNC(c2scc(C)c2Br)=O)CN(C(c2[nH]cnc2C)=O)CCCO1 N(C1CS(=O)(=O)Cc2ccccc21)C(c1c(C)c(N)cc(O)c1)=O N1(C(C(C)OCCC=C)=O)CCC(NC(C2CC2F)=O)C(OC)C1 Cc1cc2ncn(CC(O)COc3ccc(Cl)cc3Cl)c2cc1C C(C(O)C(=O)N(C)CCc1noc(C)n1)NC(C=C(C)C(F)F)=O C1(O)(CNC(C(Cc2c(C)noc2C)C)=O)CCN(C(=O)C(F)=CCCF)CC1 CC(CN(C)C)CCC(=O)NC(C(=O)NOCC1CCC1)c1cccnc1 c1(C(=O)NC2(CNC(c3cc(Cl)ncc3O)=O)CCOC2)cc2c(s1)CCCC2 C1(C(=O)NC2(C)CC=CC2)CN(C(=O)Cc2cccnc2O)CCO1 N1(C(c2cccc(I)c2)C(=O)NCCCC)CC=C(c2cc(C)cc(C)c2)CC1 n1(CC(N2CCCC(CNC(c3cccc(OC)c3)=O)C2)=O)ccc(C)cc1=O N1(C(C2CCC(CC)CC2)C(=O)NC2CCOCC2)CC2CCC(C(=O)OC)C2C1 N1(CC)CCCC(C(=O)NCC(CCOC)NC(=O)C(c2ccccc2)OC)C1 C(=O)(CN=c1cc(C)nc(N2CCC(CNc3ccccc3)CC2)[nH]1)NCC C1(NC(c2n[nH]c(C)c2C)=O)CN(C(=O)C(O)CC(C)(C)C)C2CCCCC12 C=C1CC2CCCC(C1)N2C(=O)C(C1CCN(C(=O)C(CC)OC)CC1)C Cc1ncnc(C)c1C(=O)NCC1(C)CCCC1NC(c1ccc(F)s1)=O CC(C)CC(C(=O)N(CC(C)(C)N(C)C)C)NC(=O)C(=O)C(C)C C(CCCCC(=O)N1CCC(C(CC)CC)C1)NC(CCSCCC)=O CC1CCN(C(c2cc(Br)sn2)=O)CC1NC(c1ccccc1C(N)=O)=O C(C(CC(C)C)C(=O)NCC#N)n1cc(-c2n(C3CCN(C)CC3)ncc2)nn1 O=C(C1Cc2c(Cl)cccc21)NCC1CC2(CC2)CN1C(=O)CCn1ccnn1 C1(NC(C2CCN(C(CC)=O)C2)=O)CC2(C1)CN(C(c1csc(Cl)c1)=O)C2 N1(C(CC2(C=C)CC2)=O)CCC(CCOC)(NC(=O)CCc2cc(C)no2)CC1 CC1CCCCC1(C)C(N1CCCC(CN=c2[nH]nc(-c3ccon3)s2)C1)=O c1(C(=O)NCC2C(NC(C3C(C(=O)OC)CC3)=O)C2)ccc(F)cc1Cl c1(C(=O)NCC(CNC(C(C)(C2CC2)NC(C)=O)=O)F)cc(F)cc(Cl)c1 c1(CN2CC3C(OCC)C3C2)cccc(SC(C)(C)C)c1C(F)(F)F Cc1cc(N(C2CC3(CNC3)C2)C(C2CCC(OC(F)F)CC2)=O)ccc1Cl C1(C#N)(C(=O)NCC(C)NC(c2nn(C)cc2CN)=O)CCc2ccccc2C1 c1(C(=O)NC2C(CNC(COCC(=O)OC)=O)CC2)sc(C)nc1CC(C)C C(=O)(CCCCCCCBr)N1C(CC)CN(C(=O)C(C)S)CC1 C1(C(=O)NC2CC(C)(NC(=O)COCCCOC)C2)(OC)CCCC(C)C1 c1(C(=O)NCC2CC(NC(C=Cc3ncc(C)[nH]3)=O)C2)cnn2ccn(C)c12 C(CCCC(C)(C)C(=O)NNC(=O)C1(CF)CC1)NC(C=CC1N(C)CCC1)=O C1(NC(CN2C(C)CC2)=O)CCC(NC(=O)Cn2nnc(C(C)(C)C)n2)C1 N#Cc1c[nH]ccc1=NC(CNC(C1CC(c2ccccc2)C1)=O)CO C12(C(=O)NCCC(C)CO)COCC1CN(Cc1cnc(-c3ccccc3)s1)C2 Cc1cc(C(=O)N(CC(C)CNC(=O)CC(C)c2ccco2)C)c(C)o1 C1(N(c2cnns2)C(C23CC(C(F)(F)F)(C2)C3)=O)CC2CC1CN2 Cc1oc(C(F)(F)F)nc1C(=O)NC(C)(C)CCN(C(=O)CCC1CCOC1)C C(CC(C(=O)NC(C)(CC)C(=O)OC)OC)NC(C1(C#C)CC1)=O CC(CCC(C)(C)C)C(=O)N1CC(CNC(C2CC(=O)C2(C)C)=O)C1 Cc1noc(C)c1C(C)C(=O)N(C)CCNC(c1cc(Cl)nn1C)=O Cc1cc(C(N2CCN(C(C3CC(C)(C)CCO3)=O)CC2CCO)=O)nc(C)n1 Cc1ncnc(C)c1CC(=O)N(C)CCOCCCN(C)C(C1CCOCC1)=O N1(C(CN(CCC#C)C)=O)CCCC1(C(=O)NCCC(COC)OC)CC C1(C(=O)NCCC2CC(C(=O)NC(C)CC3CCCC3)C2)(CO)CCOC1 c1(C(N2C(CNC(=O)OC)CC2)=O)ccc2c(c1)COCC2 C(S(=O)(=O)c1ccccc1)c1ccc(C(=O)OC)o1.C12CN(CC1C(=O)O)C2=O N1(C(c2ccc(OC)s2)=O)CCCCCC(NC(c2cc(OC)nc(F)c2)=O)C1 C(C)(C(=O)N(C)CC1C2CN(C(c3cc(C)ccc3Cl)=O)CC12)(C(C)C)OC c1(C(=O)NCCNC(CNC(=O)OC)=O)cc(=O)c2ccccc2[nH]1 Cn1cc(CC(C(=O)O)NC(c2cnn(Cc3ccccc3)n2)=O)cn1 C(=O)(CCC(O)C(C)(C)C)N1C(CN(C(CN2CCC(C)CC2)=O)C)CCCC1 c1(NC(C(=O)N(C(C)Cc2cccc(F)c2)C)=O)cc(F)c(F)cc1F CC1CC(CNC(c2ccccc2O)=O)CN1c1ncncc1I C1(C(=O)NC2CN(C(C(C)(C)F)=O)CC2O)C2CC(F)(F)CC12 C(CCC)(C(O)C(=O)NCC1(S(C)=O)CC1)NC(CCCCCC)=O c1(C(=O)NC(C(C)NC(c2ccccc2[N+](=O)[O-])=O)C)cc2ccnc(Cl)c2[nH]1 c1(C(=O)NCC(C)NC(C2CC(O)(CC#C)C2)=O)cc(OC)c(OC)c(N)c1.OCC C1(C(C)NC(C(Cc2ccco2)CO)=O)CCN(C(=O)C(C)C)CC1 C=CCC(C)C(=O)N1CCC(N(C(=O)CCCn2cccn2)CC2CC2)CC1 C1(C(=O)NCCc2c(CNC(C34CC(C)(C3)C4)=O)nco2)CCN(C2CC2)C1=O CCC(C(=O)NC1CCC(NC(=O)C(C)=C2CCCC2)C1)NC(N)=O C1(CNC(=O)CSC(F)(F)F)CCCN1C(C12CC(c3ccccc3)C1C2)=O C1(CC)CCC(NC(=O)CN(C2COCC2O)C(=O)CN2CC(C)(C)C2)CC1 Cc1nc(C(N2CCCC23CCN(C(=O)CC2C=CCC2)C3)=O)c2ccccn12 C1(CNC(CCN(C(=O)C(CSC)OC)CC#C)=O)CCNC(=O)C1 N1(C(CC(CC)O)=O)CCC(O)C(C(=O)Nc2ccc(O)cc2C(N)=O)C1 N1(C(C(OC)OC)=O)CCC2(CCC(NC(=O)Cc3ccc(F)c(Cl)c3)C2)CC1 C=C(C)C1OCCCC1C(N1CCCC1C(C)NC(c1[nH]nc(OC)c1Cl)=O)=O c1(CN2CC(CC(=O)Nc3cnc(OCC)nc3)C2)cccc(S(C)(=O)=O)c1 c1(N2CCC(C(=O)NC)CC2)ncnc(NCCNCc2ncc(C)cn2)c1C c1(OC)ccc(OC)c(S(=O)(=O)NC2CCN(C3CCOC3)CC2)c1 Cc1cc(O)n2ncc(C(=O)NC3CC(CNC(C4CCN(C)CC4)=O)C3)c2n1 O=C(C(O)C1=CCCCC1)NC1CC(C(N2CCCC2CF)=O)C12CCC2 C1(CNC(=O)C=Cc2cn[nH]c2)COC(C(F)(F)F)CN1C(=O)Cc1ccns1 CC1(C)CCN(CCNC(C2CC(n3cc(CCN4CCSCC4)nn3)C2)=O)C1 CCCCCC(C1CC1)NC(C1CCC1NC(C1(C)C=CCCC1)=O)=O Cc1c(Br)ccc2c1CCN(C(c1c(C)oc3ncnc(O)c13)=O)C2 c1(C(=O)NC2(C)CCN(C(=O)COCCN(C)C)CC2)cc2cccn2c(O)n1 c1(CC(N2CCCC(c3nn[nH]n3)C2)=O)cc(F)ccc1F c1(C(N2C3C(N(C(=O)CCCCCF)C)CC(C3)C2)=O)ccc2ccncc2c1 C(=O)(C(C(C)Cc1ccccc1)N(CC(C)CCC)CC=C)NC N1(C(c2c(OC)cnnc2)=O)CCOCC(C(=O)NC2CCCC(CO)C2)C1 C(=O)(C(C)(CC)CO)Nc1[nH]nc(-c2ccc(OCC)cc2)n1 c1(C(N2CCC(COC)CC2)=O)nc2ccccn2c1-c1cc(F)c(O)c(F)c1 Cc1cnc(C(=O)NC2CCCN(C(c3cc4c(s3)CCCC4)=O)C2)cc1C#N C=C=CC(C)C(=O)NC(CNC(=O)CCOc1ccccc1OC)C1CC1 CC1CC(CNC(=O)C(C2CCCCC2)NC(=O)Cc2cnnn2C)=NO1 C12(C(N3CCN(C4CCN(C(C5C(C)C5)=O)C4)CC3)=O)CC3CC(C(=O)N1)C2C3 N1(C(C2(C)CCC2)=O)CCC(Oc2ccccc2NCCS(C)(=O)=O)CC1 N=c1ccc(C(=O)NC23CC2CN(C(C2(CCF)CCOCC2)=O)C3)n[nH]1 C(CC(CC)C(=O)NCC1CC(F)(CNC(c2n[nH]cc2Cl)=O)C1)=CC C1(NC(CC(=C)C)=O)CCCCC12CCN(C(c1ccc3c(c1)CCC3)=O)C2 c1(C(=O)NCCCC(C)NC(C2C3CCCOC23)=O)ccc2cccc(Cl)c2n1 C1(CNC(c2cnn(CCCC)c2C)=O)(CO)CCN(C(C2CC2(Cl)Cl)=O)CC1 N1(C(c2c(C)coc2)=O)CC2CCC2(N(C(=O)CCc2cc(C)sc2C)CC)C1 N1(C(c2cc(C)n(C)c2)=O)CCC2CN(Cc3cccc4occc34)CC12 C(=O)(CCN=C(NCC(c1ncc(C)s1)(C)C)NC1CN(C2CC2)CC1C)NC N1(C(c2cc(OCC)n[nH]2)=O)CCN(C(C2CCC2CO)=O)CC(C)C1 C1(C(=O)Nc2cnn(CCO)c2)(CC)CCCN(C(=O)C(C2CC2)OC)C1 N1(C(C2CCC(CNC(=O)CN3CCCC3=O)O2)=O)CCCC(O)(C2CC2)C1 CC1C(C(=O)NC2COCC(C)(C)C2)CCCN1C(=O)Cn1cncn1 c1(C(=O)NCC2(OC)CC2)cccc(CCNC(=O)OC(C)(C)C)c1 C(C(COC)C(=O)NC1CCN(C(C2CC(n3cccn3)C2)=O)C1C(C)C)OC C(=O)(C1=CC2(CCN(C(=O)C(CO)C(C)(C)C)C2)C1)NCCC(COC)(C)C C(C(C)C(=O)NCC(C)(C)CC1CN(C(c2conc2C2(C)COC2)=O)C1)OC CCCCCC(O)CC(=O)NCC(C)(CO)NC(c1cc(C#N)cs1)=O c1(CC(=O)NC2C(NC(C(C3CCC3)OCC)=O)COC2)cccc2sccc12 Cc1conc1C(N1CC(O)(C(F)C(=O)NC(CO)C2CC2)C1)=O CC1(C)NC(=O)CC1C(N1CCCC(CC(=O)NCCCn2cnnc2)C1)=O C1(C(=O)NC(C)CC(=O)NCCc2nncs2)CCCC(C)(C)C1 Cc1ccc(C(C)NC(=O)CC2CN(C(=O)C3=NOCC3)CC2C)cc1 FC1(F)CCC(n2nc(Cc3ccccc3)nc2-c2ccc(Br)cc2)C1 C1(C(=O)NCC(CNC(=O)CCOCC(F)F)F)CC2(CCCC2)CO1 CC1(C)CCCN(C(c2cc(Cl)c[nH]2)=O)C1CNC(c1cccnc1N)=O N1(C(C#C)=O)CCC(C(=O)Nc2nc(Cl)ccc2I)C(O)C1 C1(NC(c2ccc(C)cc2)=O)CC(C)CN(C(=O)CN(C)C)C1.C(C(=O)O)SCC N1(C(C2(NC(C(CC)C(C)C)=O)CSC2)=O)CCCCCCCC1 C1(CCNC(CCN(C)CC)=O)CCCN1C(C1CCC(C(N)=O)O1)=O N1(C(CC(=C)I)=O)CC(CNC(=O)CC(C)OC)C(C)C1 C=CC(CC(=O)N(C)CCN(C)C(c1c(C)coc1C1CC1)=O)c1ccccc1 c1(OC)cc(C)c(CNC2CC(c3ccnc(C)c3)(C(=O)O)C2)c(C)c1 c1(C(N2CCC(OC)(CNC(c3cn[nH]c3)=O)C2)=O)cc2ccncc2s1 Cc1oc(C)c(C(N2CCC(NC(=O)CSCc3ccccn3)C2)=O)c1C n1(CC)cc(C(=O)NCC(C)(CO)NC(C23CC(F)(C2)C3)=O)c(C(F)(F)F)n1 CC#CCCCC(=O)N(CCCNC(C1COCCN1C(C)=O)=O)C1CC1 CCC(CC(=O)NCCCCNC(c1cccc(CS(N)(=O)=O)c1)=O)SC c1(COC)nc(NCc2nccn2C)cc(=NC2CC(n3cncn3)C2)[nH]1 C1C2=CCN(CC2)N2CCN1CC2.c1(CC)ncc(N)cn1.C(C)(C)(C)OC=O C(=O)(C1=CNC2=NCCC2=C1)N1C(C2CCN(C(=O)Cn3cnnc3O)C2)CCC1 CC1CC(C(=O)N(C)CCNC(C2(c3ccno3)CCC2)=O)CC(C)C1 Cc1[nH]nc(C(=O)NCC2C3CC2N(C(C2CC2C2CCC2)=O)C3)c1Cl c1(NC(C2(F)CCN(Cc3c(OCC)cccc3Cl)C2)=O)ncnc2occc12 C(=O)(C(O)CCC(F)(F)F)N1CC2(CC(NC(=O)Cn3cnnn3)C2)C1 C1(NC(c2c(N)ccc(CCC)c2)=O)CC(NC(=O)COCC)C12CCOCC2 Cc1cccc(Br)c1C(=O)Nc1ccc(Cn2cc(CC(O)C(C)C)nn2)cc1 CC1c2cc(Br)cc(F)c2CCN1C(C1CCN(C2COC2)C1)=O c1(C(=O)NCCC(=C)CNC(c2cnc(OC)nc2)=O)cnc2c(c1)CCC2 CC(=O)CCCCC(=O)NC1CCCC1CNC(=O)Cn1cc(C)ccc1=O C1(C(=O)NCCOCCCNC(CCCC=C)=O)CS(=O)(=O)CC12CCC2 c1(C(c2nnnn2C(C)C)NC(CC)C(C)C)cccc(O)c1 c1(OCCOC)ccc(C(N2CC(CCCCNC(=O)CS(C)(=O)=O)C2)=O)cn1 Cc1c(C(N2CCC(NC(=O)C(C)C3CCCC3)C2(C)C)=O)cnc2nncn12 C1(NC(C2(C)N(C)CCC2)=O)CC2CC1N(C(=O)Cc1cc(C3CC3)on1)C2 c1(OC)ccc2c(c1)C(C(=O)NCc1cscc1C)CCC2 CC(CCC(=O)NCc1ccc(CNC(C2(C#N)CCC2)=O)cc1)N(C)C C=CC1(C(=O)NCC(C)(C2CC2)NC(=O)C#CC(=O)N(C)C)CCCCC1 c1(C(C)C)ccccc1NC(CN(c1cccnc1)CC(C)C#N)=O CCCC(CNC(c1ncncc1C)=O)C(=O)NC1CC(Cl)(Cl)C1 c1(COC(C2(C(=O)O)CC(F)C2)=O)ccc(Br)cc1[N+](=O)[O-] C1(NC(=O)OC(C)(C)C)CN(N2CCC(O)(C(F)(F)F)CC2)CCO1 Cc1n[nH]c(C)c1C(c1nnnn1C(C)C)Nc1cccc(Cn2ccnc2)c1 N(C(=NCCSC)NC(C1(F)CC1)C)CCSC c1(NCCc2ccc(OC)cc2)cc(S(=O)(=O)N(CC(C)C)CC)ccc1C#N C=CC1(C(=O)NCC2(O)CCC(C)(C)C2)CCN(C(C2CCC=CCC2)=O)C1 C1(CNC(C(C)n2cncn2)=O)C(C)CCN1C(C1COC(C)(C)C1)=O C(=O)(CCS(N)(=O)=O)NC(CCNC(c1nc(C(C)OC)sc1)=O)(C)C c1(C(=O)NC2C(NC(c3cc4cccnn4n3)=O)C2)c[nH]c2ccc(Br)cc12 Cc1sc(O)nc1C(=O)NCC1(F)CCN(C(C2CCN(C)C2=O)=O)C1 C1(NC(C2CN(C)C(=O)N2)=O)CCCC(NC(=O)CCN2CCNC(=O)C2)CC1 C(=O)(C1=COCCC1)N1CCC(O)(CN(C(C(C(C)C)n2cnnn2)=O)C)C1 C1(NC(c2cc(OC)c(O)cc2)=O)CN(C(c2cc(C)n(C)n2)=O)CC(C)(C)C1 N1(C(C(C)Cc2cnco2)=O)CCC2(CC1)CC2NC(C1CCCN1N=O)=O N1(C(C(CC)=CC)=O)CCC(C)C(NC(c2ncc(N(C)C)cn2)=O)C1 CCCC(O)C(CO)NC(C1CC2CCC1N2C(=O)CCCC1CC1)=O c1(C(=O)NC(CC)CN(C)C(C2CSCCS2)=O)cncc(N)n1 c1(C(N2CCC(=CCNC(C3C(CCC)C3)=O)CC2)=O)c(Cl)cc(Cl)nc1N c1(C(N(CCCCNC(=O)C(O)c2ccco2)C)=O)ccccc1Br C1(C(=O)OC)CCCC(n2cc(C3CCN3C(c3cnn(C)c3C)=O)nn2)C1 c1(C(=O)OC)cccc(NNC(=O)NC2CCn3c(C)cnc3C2)c1C C1(CNC(C=Cc2scc(C)n2)=O)CCN(C(C2CC23CCC3)=O)C12CCC2 c1(SCC(=O)OC(C)(C)C)nc(C)cc(NC(C2ON=C(C)C2)=O)c1C#N Cc1ccn(CC(C)C(=O)NC2CCC(NC(c3ccn(C)n3)=O)C2)n1 C1(C(=O)NCC(CC)NC(c2c[nH]nc2C2CCCO2)=O)CCC(=O)N1 CC1CN(C(=O)NC2C3CCC4C(C3)CC24)CC(C)N1C C(=O)(C#CC1CCCCC1)NCC(C(N1CCC(C(C)C#N)CC1)=O)(C)C N1(C(CN(C(=O)OCC)C)=O)CCCC2(CNC(c3oncc3C)=O)CC12 C1(C2CCCC2)(C(N(CC(C)NC(=O)C(O)CC2CC2)C)=O)CCNC1=O N(C1CN(C(c2cnnn2C2CC2)=O)Cc2ccccc21)C(CC(C)(F)F)=O C12(C(=O)NCCN(C(C(C)SC)=O)C)COC(C1)C2 N1(C(=O)OC(C)(C)C)CC2(CC(NCCCc3cc(F)cc(F)c3)C2)C1 C1(NC(CCC=C)=O)CN(C(c2cc(C#N)ccc2Cl)=O)CC1S(C)(=O)=O C(=O)(C(CC1CCOCC1)NC(=O)C(C)N1CC(C)C1)N(C1CCOCC1)CC C1(O)(CC(=O)N(CCCNC(=O)CC=CC(C)(C)C)C(C)C)COC(C)(C)C1 C1(CNC(c2c(C)nn(CC)c2Cl)=O)CN(C(=O)C2=CCCC2)CC2(CCC2)O1 c1(CC)cc(C(=O)NC(CO)C(C)NC(c2sccc2SC)=O)ncn1 N1(C(CC(=O)OCC)=O)CCN(C(=O)C(C(C)(C)C)NC(N)=O)C2CCC12 N1(C(C(CC)=CCCC)=O)CC(C(=O)NC(C2(CO)CC2)C)CC12CCC2 C1(NC(C(C)OC)=O)C2CCC1CN(C(c1ccc3c(c1)OCO3)=O)C2 c1(CC)c(C(=O)N(C)CCN(C(C2C3CCCOC23)=O)C(C)C)nnn1C N1(C2(C(=O)NC(C3CN(C(=O)C=CCN(C)C)C3)C)CCC2)CCOCC1 C1(C(N2C(C)CC(CNC(=O)Cn3cc(Cl)cn3)C2)=O)CCCC(=O)N1C N#CC1CN(Cc2ccc(I)cc2F)CCN1C(C1CC=CCC1)=O n1(CC(=O)N(CCCNC(COCC(=C)C)=O)C(C)C)cnc(C(N)=O)n1 C1(C)(CN(C(=O)CC=C(Cl)Cl)C)CCCC1NC(=O)C(O)CCn1cncn1 N1(C(CC2N(C(COCCCOC)=O)CC(O)C2)=O)Cc2ccnn2CC1C N1(CC)CCC(C(N2CC3C(C(=O)NC4CC(CCC(N)=O)C4)C3C2)=O)CC1 C1(NC(CCSCC)=O)CC12CCN(C(=O)CC1(n3ccnc3)CC1)CC2 Cc1cc(=NC2CCCN(C3CC3)C2)[nH]c(N2CCOC(C)(C(C)C)C2)n1 CC(C(=O)NCc1ccsc1C(=O)NC1(C)CCCOC1)S(C)(=O)=O N1(C(C(CC=C)CC)=O)CC(C(=O)ON(CC(=O)OC)C)CC(C)(C)C1 c1(C(N2CC(C)C(NC(=O)C(F)=CC3CC3)CC2)=O)ccc2nnn(C)c2n1 N1(C(c2ccnc(OC)c2F)=O)CC2CN(C(=O)CCCSC(C)(C)C)CC2C1 N1(C(c2cccnc2)=O)CCC(F)(F)C(C(N2CC3CC(C2)O3)=O)C1 N1(C(C2C(C(=O)OC)C=C2)=O)CCC(CNC(=O)COC2CCC2)CC1 c1(CCN=C(NC(c2cccs2)C)NCCS(C)(=O)=O)cccc2ccccc12 C(=O)(C#CC1CCCO1)N1CC2C(CNC(c3cc(Br)cs3)=O)C2C1 C#CC1CCCN(C(c2cc(Cl)c(Br)cc2F)C(=O)NCc2cccs2)CC1 c1(C(N2CCCC(c3cn(CCN(S(C)(=O)=O)C)nn3)C2)=O)occ2c1CCC2 N1(C(C(F)=CCOC)=O)CCCCC(NC(=O)CCc2ccc(OC)cc2)C1 n1(CCOC)cc(C(=O)NCC2CC(NC(C3CCOC3CC)=O)C2)ccc1=O c1(C(=O)NC(CN(C(CNS(CC)(=O)=O)=O)C)C)ccc2c(c1)NC(=O)CCC2 c1(OC)cc(C(N2CC(CNC(=O)C(C)C(F)F)C(C)(C)C2)=O)cc(Cl)c1 C1(CC)CN(C(c2ccn(COC)n2)=O)CC1C(N1CCCC(CO)C1)=O c1(CN(C(=O)C=CCC(C)(C)NC(C2CN(C3CCC3)C2)=O)C)cccc(F)c1 c1(NC(c2ccc(OCCNCCc3nn[nH]n3)cc2)=O)cccc(F)c1F N(C)(S(=O)(=O)N1CCCCC1C1CCCN(C(=O)C(C)C)C1)C(C)C1CC1 C1(NC(c2cccc(CC)n2)=O)CC2CC1CN(C(C1CC1c1cnn(C)c1)=O)C2 Cc1n[nH]c(C)c1C(C)C(=O)NC(C)CC(C)NC(=O)CCCCF c1(C(=O)NCCCN(C)C(C2COC2)=O)ccc2[nH]c3ccccc3c2c1 N(C(=NCCC(=O)N1CCCC(C)C1)NCCOC)CC(CC)NC1CCOCC1 c1(C(=O)NCC2CC(Nc3n(C)cc(Br)n3)C2)cc2ncccc2[nH]1 c1(C(=O)NC(CC(C)NC(c2cc(C)sc2C)=O)C)cc([N+](=O)[O-])c(O)cc1N C1(C(=O)NC2C3CCN(C(C(c4cccc(C)c4)=O)=O)C32)CCCC(C)(C)O1 c1(C(=O)NC2(CF)CN(C(c3c(C)scn3)=O)C2)noc(C2CC2)c1C c1(C(=O)NC2CN(C(CCCCN(C)C)=O)C3C2C3)cc(O)nc2ccccc12 C(C1=CCN(C(C23CC(F)C2C3)=O)CC1)NC(C1CC(C)OCC1)=O c1(OC)cnc(F)cc1C(=O)NCCC1CCN(C(=O)C(C)(C)C(C)O)C1 C1(C)(C(=O)NCC(C2CCC2)NC(c2c(CCC)[nH]cc2)=O)CCCCNC1=O c1(NC(C)=O)ccc2c(c1)CCC2NS(=O)(=O)CCOC(F)F c1(CC)cc(Cl)ccc1C(N1CCC(CO)(NC(c2nccc(Cl)c2O)=O)C1)=O N1(C(c2cc(N)c(F)cn2)=O)CC2(C1)SCCC2NC(c1cnc2n1CCS2)=O C1(C(=O)NC(CNC(C(C)=C(CC)C)=O)C(C)(C)C)CC2(C1)CC21CC1 C1(NC(C2CCSC2)=O)CC2(CCCCN2C(=O)CSc2cccs2)C1 C1(NC(COC(CNC(C(C(=O)OC)OC)=O)(C)C)=O)(CO)CCC(F)(F)CC1 Cc1ccc(C)c(NC(=O)CC2CCCN(C(C3CC3c3ccoc3)=O)CC2)c1 C1(NC(CC2(C(=C)F)CCC2)=O)C2CC1N(C(c1ccccc1C)=O)C2C C1(C#N)(CC(=O)NC(CNC(CC(C)c2ccco2)=O)C(C)(C)C)CCCCC1 c1(C(=O)NCC2(F)CC(NC(CC3(C)OCCO3)=O)C2)cnc2sccc2c1 Cc1nc(O)nc(O)c1NC(N1CCN(CC#Cc2cccnc2)CC1)=O N1(C(CCc2ccc(C)o2)=O)CCC2CC(NC(C3(C(F)F)CC3)=O)CCC2C1 N1(C(C2N(CC)CC2)=O)CCC(C)(CNC(c2c[nH]c(C#N)c2)=O)C1 C(=O)(C1=NNC(=O)CC1)N(C1CN(C(c2ccc(=O)n(C)c2)=O)C1)C [N-]=[N+]=NC(CCC(N)=O)C(=O)N1CCCC(CC2CC3(CCC(CO)O3)C2)C1 C(CCC(O)C(=O)OCC)NC1(c2n(CC=C)nnn2)CCC1CC n1(CC#C)cc(NC(=O)C(C)NC(=O)C(C)OCC2CC2)cn1 C1(C(=O)NCc2c(C)csc2)CN(C(C2CCC(=O)N(C)C2)=O)C(C)(C)C1 CC1CC=CCC1C(N1CCC(CCNC(C2CN(C3CCOCC3)C2)=O)C1)=O C12(C(N3CCCC(COCC)C3)=O)C(NC(=O)CCP(C)(C)=O)C3CC1C2C3 C1(NC(C(COCC)NC(c2cc(C(N)=O)co2)=O)=O)CCC(=O)NC1C c1(C(N2CCC(C)(CCNC(C3N(CC)CC3)=O)CC2)=O)cc(F)c(C)cc1N c1(C(N2CCCC(NC(c3cc(C(F)(F)F)cs3)=O)C2)=O)c(F)ccc(F)c1F C1(C(N(CC(CC)NC(=O)CC2(n3ccnc3)CC2)C)=O)CC=C(C)CC1 Cc1nc(O)[nH]c1C(=O)NC(CNC(=O)CN(c1cnccn1)C)CO C#CCC(C)(C(=O)NCC1CCCN(C)C1=O)NC(c1coc(CCC)n1)=O N1(C(C2(OCC)CC2)=O)CC(CNC(c2ccncc2C)=O)C(C)(C)C1 C1(OCC)CCCN(C(c2c(I)cnn2C)C(=O)NC2COC2)C1 C1(CCCC)C2=CC=NSC(CC)(C(C)NC(=O)CSCC1)CNC2=O c1(C(=O)NCC(CC)(C)NC(C2CCC2C#N)=O)cc2cccnc2[nH]1 c1(C(=O)NCCOC2CCN(C(COC)=O)C2)cc(C)c(F)cc1F c1(SCCC(c2cc(OC)ncc2)=O)cc2c(Br)c(C(=O)O)cc(C)c2[nH]1 Cc1nsc(C(=O)NCCCNC(=O)C(N2CCC(C)C2)=O)c1Nc1ncc[nH]1 N1(C(C(C=C)(C)CCOC)=O)CC2(C=C(C(=O)NCC3COCC(C)O3)CO2)C1 N1(C(c2c(C)c(Cl)c(Cl)s2)=O)CCCC2(CC(NC(c3ccncn3)=O)C2)C1 C(=O)(C(=O)N=S(C)(C)=O)N1C(CNC(c2nn(C)c(=O)cc2)=O)CCCC1 CN1CC(C(=O)NCC2(C)CCCN2C(c2cc(Br)no2)=O)NC1=O c1(C(=O)NCCC2ON=C(C)C2)[nH]c2ccc(F)cc2c1Cl c1(CC)ccc(C(N2CC3CC2CCN3C(C2CC2C(F)(F)F)=O)=O)cc1C#N Cc1c[nH]c2ccc(-c3cc(C(=O)NC4CC5CCC4C5)ccn3)cc12 c1(C(=O)NC(CN2CCCC(C)C2)C)cc2cn[nH]c2cc1O c1(C(=O)NC2C(NC(C3(C)COC3)=O)COCC2)cccn(C2CCC2)c1=O c1(CN2CC(C)(CC(=O)NCCC3CCOCC3)C2)ccc(I)c(O)c1 N1(C(C=COCC)=O)CCCN(C(=O)CC2CN(C)C2)C(c2ccccc2)C1 c1(C(C(=O)NC(c2ccccc2)C)N(CC#CC)C2CC2)ccccc1Cl C1(F)(NC(c2cccc(OC(C)(C)C)c2)=O)CCCN(C(C2C(OC)C2)=O)C1 C(=O)(CCC1=NNC(=O)CC1)N1C(CNC(CCC(C)OC)=O)C(O)C(O)C1 CCC(CC)C(=O)NCC(C1CCN(C(=O)C(C)Sc2ccccc2)CC1)F C1(CNC(C2(C#C)CCC2)=O)CCCCN(C(=O)C(C)C(F)(F)F)C1 c1(C(=O)NCC2CC2)ccc(C(N2CCC(N(C)C(C3CC3C#N)=O)C2)=O)cc1 C1(NC(C2=CCCCC2C)=O)COC2(CCN(C(C3CC(F)C3)=O)CC2)C1 c1(CCC(=O)NC(C(CO)NC(CN(C)CC)=O)C)nc2ccccc2o1 C(=O)(CCCCC(=O)NC)N1C(CCN(C(CCCC#CC)=O)C)CCCC1 c1(C(N2CCC(OC)(OC)CC2)C(=O)NCC(F)F)ccc2nsnc2c1 c1(C2(OC)CN(C(=O)Cc3c(Cl)cnn3C)C2)ccc(Br)cc1 c1(SCC(N2CCC(N(C(C(C)NS(CCC)(=O)=O)=O)C)C2)=O)ccccc1O Cc1cc(Br)ccc1CN(C(=O)C(=O)NC(C)CN1CCOCC1)C C(CCC(=O)N=S(C)(=O)C1CC2(CNC2)C1)Oc1ccc(C)cc1 CN=c1nc(N2CC3CC2C2CC32)[nH]c(=NCC(C)(C)S(C)(=O)=O)[nH]1 c1(C(=O)NCC(C)NC(c2c(C)con2)=O)cnn(C(C)C)c1Br C1(NC(Cc2ncc(C)o2)=O)CC(F)CN(C(c2ccc(-c3cc[nH]n3)s2)=O)C1 Cc1[nH]ccc1C(N1CCC(CCNC(=O)CC(C)F)C1)=O C1(C)(NC(C=CCNC(c2c(CC)nc(C)o2)=O)=O)CCC(C)=C(C)C1 C(CC(C(=O)N1CCOC(CC(N)=O)C1)NC(=O)COC1CC1)=CC N1(C(CN(C(CC(=C)Br)=O)C)=O)CCN(C(=O)CCc2ccn(C)n2)CC1 Cc1csc(=NCC(=O)NC2(CNC(C3CC4COCC4C3)=O)CCOC2)[nH]1 C1(C(N2C(CNC(C3CNC(=O)O3)=O)CC(C)(C)C2)=O)CN2CCCN1CC2 CCC(CNC(=O)CCN(C)CC)NC(=O)C(C)c1cccs1 Cc1cnc(C(N2CCCCC2CCNC(=O)CCOC2CCOC2)=O)cn1 C1(CNC(C2CC(OC)C2)=O)CCCCN(C(C2(C)CCCC2C)=O)C1 C1(C(=O)NC2C(C)CN(C)CC2)C(C2CC2)CCN1C(c1ccccc1)=O N1(C(Cc2c(C)nccc2)=O)CC2CC1CN2C(c1n[nH]c(C)c1F)=O c1(N2CC3CN(CC)CC3C2)ccc(S(=O)(=O)NC2(c3ccsc3)CC2)cn1 c1(C(C(=O)N(C)CCN(C(=O)CSn2cncn2)C)n2cccc2)ccccc1 N1(C(C(CC)C2COC2)=O)CCCN(C(c2cnc(Br)s2)=O)CC1C C1(NC(c2ccccc2-n2cncn2)=O)CCN(C(C2(CF)CC2)=O)CC1CO CCC(CC)CN=C(NCc1ccc(F)cc1)N1CC2C(C1)C2(C)C c1(NC(C(CC=C)C)=O)ccc(C(=O)NC2(C)CC2)cc1C c1(C(N2C(CNC(=O)CCC3CCCO3)CC2)=O)sccc1Cl C1(C(=O)NCCCCN(C)C(C2(N3CCOC3=O)CC2)=O)(OC(C)C)CCOC1 N1(C(C(CN(C)C)N(C)C)=O)C(CC(=O)N(C2CC3CC3C2)C)C2CCCC12 C(=O)(C(CCS(C)=O)N(C)C)NC1C(NC(C(C)=C(C)C)=O)CCOC1 C1(CCC(=O)NCCn2ncc(C)c2)CCN(C(=O)C(C)NCCCCO)CC1 C1(C(=O)NC2C=CCN(C(C3C(OC)CCC3)=O)C2)CCC(C)C(C)C1 C1(C(=O)Nc2cc[nH]n2)CCCN(C(C2C3CN(C(=O)CC4(O)CC4)CC23)=O)C1 c1(C(=O)NC2CC(CCNC(CN(C)CC)=O)C2)noc2c1CC(C)(C)CC2 C(=O)(CCCCCNC(=O)C1CC1)NCCC1OCC(C)(C)C1 C1(NC(C2CCCN(C)C2)=O)CN(C(=O)CSc2ncccn2)CC(F)(F)C1 CC(C)C(O)C(=O)N(C1(NC(=O)CCc2ccn(C)c2)CC1)C c1(CC(N2CCC(N(C(=O)CSC(F)F)CC)C2)=O)cc(C)nn1C c1(C(C(C)OC(c2sccc2-c2ccc(F)cc2)=O)=O)ccc2c(c1)OCO2 CCC(C)C(O)C(=O)NC1CC2CC1N(C(=O)CSc1ccccc1F)C2 c1(C(N(CC(CC)NC(=O)COC2CC=CC2)CC)=O)cccnc1 N1(C(CSCC=C)=O)CCC(C(=O)NCCC(=O)NCC(C)C)C1 C(=O)(C1=CCCCO1)N1CC2C(C(=O)NCCNC(C34COCC3C4)=O)(C2)C1 C1(C(C)C)CN(C(c2cccn2C)=O)CCCN1C(c1cc(C2CCC2)n[nH]1)=O C1(C)(CCC(=O)NC2CC(CC)C2)CCCN1C(=O)C(C)C(=O)OC c1(C(=O)NC2(CNC(c3n(CC=C)ccc3)=O)CCOC2)cc(F)cc(Cl)c1N c1(CC)ccc(Cl)c(C(N2CCN(C(C3CCCC3(C)C)=O)CC2C2CC2)=O)c1 C(S(C)(=O)=NC(=O)CCc1nc2ccccc2[nH]1)NC(=O)OC(C)(C)C C(=O)(C(C)CCNC(=O)CC(CC1CC1)NC(=O)C(=Cc1cn[nH]c1)C)OC N1(C(c2c(CC)cco2)=O)CCC2CC(C(=O)NCC3CCCO3)C2C1 c1(C(N(C2C3CN(C(CC(CC)C(F)F)=O)CC32)C)=O)ccc2oc(O)nc2c1 Cc1ccc(F)c(CNC(C2CCN(C(c3c(C)n[nH]c3C)=O)CC2O)=O)c1 C1(N(C(C(C)NC(CC)(C)C)=O)C)CCN(C(C2(c3ccc(C)s3)CC2)=O)C1 N1(C(C)C)CC2CC1CN2C(=O)C(Cn1cccn1)NC(=O)C(C)N1CCCC1 Cc1[nH]c(C2CCN(CCC(C)N(C)C)CC2)cc1C(N1CCC12CCC2)=O C(CN=c1[nH]c2c(c(=NC3CC=C(C)CC3)[nH]1)CCCC2)OC(CC)(C)C c1(C(=O)NCCCOCCNC(c2c(C)n[nH]c2C)=O)coc2cccc(O)c12 C1(NC(C2(c3ccc(N(C)C)cc3)CC2)=O)CC2CC1N(C(=O)C(O)CF)C2 Cc1cc(C(N2CCCC2C(=O)NCCC(=O)N(C)C2CC2)=O)cc(O)n1 c1(C(N2C(CNC(CN(C)CC)=O)CC2)=O)cnc(N2CCOCC2)s1 c1(C(=O)NCCN(C(C=CC)=O)C(C)C)cnn(C)c1C(C)C c1(C(C(C)NC(=O)CC(C)C2CC2)NC(=O)C(C)(C)C)cccc([N+](=O)[O-])c1 C1(NC(CCSCC)=O)CCN(C(c2cn(C(C)C)nc2C)=O)CCC1CO C#Cc1cccc(C(C(=O)NCSc2ccccc2OC)Nc2cnn(CC)c2)n1 n1(CCOC)nnc2c(N3CCCC(NC(=O)CC(=O)OC)C3)ncnc12 N1(C(C(C#C)(C)C)=O)CCCCC2(CCN(C(=O)C(C)(C)CS(N)(=O)=O)C2)C1 C(C(=O)N1CC(N(C)C(c2snc(O)c2Cl)=O)C1)(C(C)C)NC(C)=O CCCCCCC(CC)C(=O)NCC1CCCN1C(c1ccc(C)[nH]1)=O c1(N(C)Cc2scc(C)n2)nc(NC2CCC(=O)NC2)c2ccsc2n1 N1(C(=O)C=CCN2CCCC2)C2CCC(C(N3CCCC3CF)=O)C1CC2 N1(C(C(C)=C(C)C)=O)CC=C(CCNC(C2CC2c2ccccc2)=O)CC1 N1(C(C(=O)NCC)=O)CC(C)(C)c2ncc(-c3cc(C)cnc3OC)cc21 C1(OCC)CC(C(N2CCCC(O)C2)=O)N(C(C2(c3ccccc3)CC2)=O)C1 C1(C(=O)NCCCNC(c2ccnc(OC)c2Br)=O)CCCCN(C)C1=O C=CCN=c1[nH]c(C(=O)NCC2CCCCC2NC(=O)CCC(C)(F)F)cs1 c1(C(N2CC(CC(C)NC(C(C)NC(=O)C(C)(C)C)=O)C2)=O)cnc(N)c(O)c1 CCCS(=O)(=O)CC(=O)N1CC(C(C)NC(c2cnn(C)c2C)=O)C1 N1(C(Cc2nc(C)oc2)=O)CCCC1(C)CNC(c1ccn(C2CC2(F)F)n1)=O C(C)(C)(CC(=O)N1CC(CNC(=O)CCn2cncn2)C(O)C1)OC Cc1nc2ccc(C(=O)NCCC(C)N(C(=O)CN(C)C3CC3)C)cc2[nH]1 C1(C)(C(=O)NCC2C(NC(C3CCC(C)CC3)=O)CCCC2)CCOC(C)C1 C(C(=O)N=c1cc2ccccn2[nH]1)(C1CN(C(=O)CC2(N(C)C)CCC2)C1)OC c1(C(N2CCC(NCC3CC3)C2)=O)cccc(S(=O)(=O)N(CCC#N)C2CC2)c1 C1(N(C)CC2(CC(=O)N(CCOc3ccccc3)CC)CC2)CC(=O)C12CCC2 N1(C(CCSCCCC)=O)CC(CC(=O)NC(c2cccnc2)C)CC1(C)C C(=O)(CS(=O)(=O)C1CC1)NC1C(CNC(C(CC(C)C)OC)=O)C1 N1(C(C2=CC(C)(C)C2)=O)CC2CCC(C1)C(NC(C1(C)CCC3CC3C1)=O)C2 C1(C(=O)NC(c2ccncc2)CC)CC2CC2N1Cc1ccc(SC)cc1 CC(=O)CCC(=O)NC(c1nocc1C(=O)N(C1CCC2CC12)C)C N1(C(c2c(C)nco2)=O)CC2(CO)CC1(C(=O)NC(c1ccc(F)cc1)C)C2 c1(OC)cc(F)cc(C=CC(=O)N(c2cc(F)cc(C#N)c2)C2CC2)c1 Cc1nn2ncccc2c1C(N1CCC2CC2(NC(c2ccsn2)=O)CC1)=O N1(Cc2c(C#C)cccc2)CC2(CCC(C(=O)NCc3cnccc3C)O2)C1 CON(CCC(=O)N1CC(C)CC(C)C1)C(=O)c1c(C)nn(C)c1C CC(C)CC(F)C(=O)NC(C)CNC(c1ccccc1-n1ccnn1)=O C(CC(C(=O)NOCc1ccccc1)NC(=O)CC1CCOCC1)OC c1(C(=O)NCC(C2CCOC2)NC(CCOCC)=O)cc2cc(Cl)c(Cl)cc2[nH]1 C(=O)(N=c1cc(C(C)C)o[nH]1)N(CCCCc1ccccc1)C.CO c1(C(N2C(c3ccccc3)CC(C)C2)=O)nn(C)c(=O)c2ccccc12 c1(SC)ncc(Cl)c(C(=O)NCC2(F)CCN(C(c3cccnc3Cl)=O)CC2)n1 C1(=O)n2[nH]c(=NC(=O)C(C)S)c3c2CN(C3)C(=O)N1.C1(CC)CCC(C)CC1 C1(C(=O)NCC(F)CO)CCCC12CCN(C(c1ccc(O)c(I)c1)=O)C2 C1(C(N2CCC(C(C#C)C)CC2)=O)CN(C(=O)CC2(COC)CC2)CCC1(C)C C(=O)(C(C)(C)CCC#N)N1CC(CCNC(C=Cc2ccc(SC)s2)=O)OCC1 C1(CC)CN(C(=O)CC2(O)CCCC2)CCC1NC(=O)CCN1CCN(C)CC1 c1(C(N2C3CN(Cc4cccc(O)n4)CC23)=O)c(Cl)cccc1I C1(C(=O)NCc2nccc(C(N(C3C(C)C3)C)=O)c2)CC2(CC(=O)C2)C1 CC1CCN(C(c2cnc(C#N)s2)=O)CC1CNC(=O)Cc1ccnc(F)c1F C1(NC(c2cc(OC)nc(F)c2)=O)(CNC(=O)C(N)=O)CC2CCC1CC2 Cc1ccc(C(N2CCCC2CNC(c2ccnn2CC(F)F)=O)=O)cc1N c1(NC(C=C)COC)[nH]c(=NCCC(C)(C)OC)nc2c1ncn2CC S(=O)(=O)(c1ccc(NCC2CN(C3CC3)C2)c(Br)c1)NCCN(S(C)(=O)=O)C c1(CC)occ(C)c1C(=O)NC1CCCCC1CNC(c1scnc1C(F)F)=O N1(C(c2cn(C)nn2)=O)CCCC(Cc2cn(CC(N3CCSCC3)=O)nn2)C1 C1(NC(CN(C)CC)=O)CN(C(c2ncc(C)cc2C)=O)CC(C)(C)C1 N1(CC(N2CCC(N(C(C(C)Cc3ccccc3)=O)CCO)C2)=O)C(C)CCC1C c1(CNC(C(C)O)=O)nc(CNC(c2ccnc(NS(C)(=O)=O)c2)=O)cc(O)n1 N1(C(COCCC)=O)CC2CC(NC(=O)Cc3cc(Cl)ccc3Cl)CC1C2 c1(OC)ccc(S(C)(=O)=O)cc1C(=O)NC1CCN(C(=O)CCCCl)CC(O)C1 c1(NC(CC)CNC(C2CCN(C)C2)=O)nc(C)cc(C)c1C(=O)OC C1(CC)C(NC(=O)CCc2cccnc2)CCN1C(c1coc(Cl)c1)=O N1(C(CC(=O)NC2CC2)=O)CCC(O)(C(F)(F)CNC(c2ccc(=O)oc2)=O)C1 Cc1cnn(C)c1C(=O)NCC(C1CCCCC1)NC(=O)CC12COC(C)(C1)C2 c1(COC)cccc(C(=O)NC2CC(CNC(C3(C)C=CCCC3)=O)C2)n1 c1(CCC(=O)NCCNC(C=C)=O)ncc(-c2ccccc2)o1 N1(C(C(F)=C(C)C)=O)CC(NC(=O)CC2CCCOC2)C(N=[N+]=[N-])C1 Cc1c(NS(=O)(=O)CC2CC3C(C2)C3(F)F)cccc1N=[N+]=[N-] C(=O)(CCCCC(C)(C)C)N1CC(C2(NC(Cc3n(C)ccn3)=O)CC2)C1 N1(C(=O)Nc2ccc(Oc3cccc(C#N)c3)cc2)CC2C3C=CC(O3)C2C1 c1(C(=O)NC2C(CNC(C(C)OCCCCCC)=O)CC2)nc(Cl)c(CC)[nH]1 N1(C(Cc2cccc(SCC)c2)=O)CCN(C(=O)CC2CC(=O)C2)CC1CCO c1(C(N2C(CCNC(c3ccc(CCC)[nH]3)=O)CCC2)=O)cccc(F)c1CC C1(CC(=O)N(C2CCN(C(C(CC)SC)=O)C2)CC)CC2(CCC2)C1 c1(CNC(C2CC(F)C2)=O)nc2c(s1)CCN(C(=O)CCCF)C2 CC1(C)CC(C(=O)NCC2CN(CCN)C2)CN1C(c1cc(C(F)F)no1)=O c1(CC2(C(N3CC(NC(C4CCCO4)=O)C3)=O)CC2)ccccc1 c1(N2CCCC(CCNC(=O)C=CC3CC3)C2)ccc([N+](=O)[O-])cn1 C(=O)(C(C(C)(C)O)NC(=O)C(=Cc1ccco1)C)N1CCC(CSC)C1 c1(C(=O)NC2(C)CCN(C(c3cnc(C(F)(F)F)o3)=O)C2)cccc2cncn12 N1(Cc2n(C)ncc2-c2cnsc2)C(C2(O)CC2)CC2CCCC12 C#CCC(CC(F)F)C(=O)NCCC1COCCN1C(=O)CCOC Cc1csc2c(CN3CC4CCC(CN=c5ccnc(CO)[nH]5)(C4)C3)cccc12 c1(C(=O)NCC2C3CN(C(c4c(C)cccc4)=O)CC32)cccc2c1OCC2C c1(C(N2CCC(N(C(c3ccn(C(C)C)n3)=O)CC)C2)=O)cnn(C)c1Cl c1(C(N2CCCC(C(N3C(CCC)COCC3)=O)C2)=O)ccc(F)cc1Br N1(C(COCCOCC#C)=O)CCCC(F)(C(=O)NCc2ccc(NC)nc2)C1 c1(C(=O)Nc2sc(C)c(C3CCCOC3)n2)ccc2cncn2c1C CCCC(C)CC(=O)N1CC(C)(CCC(=O)NC(CCO)C(F)(F)F)C1 C1(NC(c2c(SC)cccn2)=O)CC2(C1)CC(CNC(=O)Cc1coc(C)n1)C2 C(=O)(CC(C(F)(F)F)OC)N1CC2(CN(C(C3CCC(CCC)CC3)=O)C2)C1 C#CCC(C(=O)N(CCCOC(C)C)C)NC(c1cc[nH]n1)=O C1(NC(CCN(C(=O)CC(C)F)CC#C)=O)CC(=O)N(CCC)C1 Cc1cc(C)c(C(=O)NCC2CCOC2C(=O)NCC(O)C(C)C)s1 C(=O)(C(O)(CNC(=O)CS(C)(=O)=O)C(F)(F)F)OC(CC=C)CNC(C)=O c1(C(=O)NCC(C2CCC2)NC(=O)CCn2cncn2)c(Cl)nsc1Cl Cc1c(C(=O)NC2CCCC2(C)CNC(=O)C(C)O)[nH]c2c(Cl)cccc12 C1(C(N2C(CCNC(C3(C)CCOC3)=O)CCC2)=O)CC2C=CC1C21CC1 C1(NC(C(CC#C)C)=O)CC2CCC1N(C(c1c(C)cc(C)nc1O)=O)C2 c1(C(C)C)cc(C(N2CCOC(CNC(C3(N(C)C)CC3)=O)C2)=O)cc(Br)c1 N1(C(C(C)N(C(c2ccc(C#N)o2)=O)CC)=O)CC(C)CCCC1C n1(CC(=O)NC(C)CCNC(c2cccc(Br)c2)=O)ncc(O)nc1=O c1(C(N2CC(OCCNC(c3c[nH]cc3Br)=O)C2)=O)cccc2c1CCCC2 C(CC1=CCN(C(=O)C(C)n2cnnn2)CC1)NC(C(c1cccc(F)c1)C)=O C(CNC(c1cn(C)c(=O)n1C)=O)(CC(F)(F)F)NC(Cc1ncc(CC)[nH]1)=O C(C1(O)CCc2ccccc21)NC(=NCCC)N(C)CC(C)OC CCC(F)(F)CC(=O)NCCOC1CCN(C(C23CC(C(C)(C)C)(C2)C3)=O)C1 C(=O)(C(F)(F)C(F)(F)F)N(C)CC1(O)CN(C(c2sccc2F)=O)C1 CC12CCC(O)C(C1)N(C(C1CC(C(F)(F)F)CN1)=O)C2 c1(C(N2C(C)(C)CC(NC(=O)CCc3nncs3)C2)=O)ccc2c(c1)OCC2 C1(CNC(c2n(C=C)nnc2)=O)CCN(C(=O)C(CSC)OC)CC1C1CC1 N1(C(COCC#C)=O)CC(NC(=O)C(C)(O)CCC)CC2(CCC2)C1 c1(C(N2C(C(N3CCCC(O)C3)=O)CCCC2)=O)cc(F)c(F)c(O)c1F c1(C(N2CCCC(C(=O)NCc3ncccc3Cl)C2)=O)cn2cc(F)ccc2n1 CCCCCCCCC(=O)N(CC(C)CNC(c1cnn(C(C)C)c1C)=O)C c1(C(C)=O)nc(C(=O)NC(C)CC2CN(C(c3ccc(Cl)o3)=O)C2)cs1 c1(NCC(=O)N(C2CCN(C(c3cn(C)nc3O)=O)C2)CC)ccc(F)cc1 C1(NC(c2cnc(C)o2)=O)CN(C(c2cnsc2)=O)CCC1C C(=O)(CS(C)(=O)=O)OCCCN(C(CC)C)C c1(OC)cc(C(=O)NC23CC(C(N4CCOC(C#N)C4)=O)(C2)C3)ccc1Br C1(CC)CN(C(=O)C(C2(O)CN(C(C3(Cl)CC3(F)F)=O)C2)F)CCN1C c1(NCCCCSC)nc(N2CCC(CC#N)C2)nc2scnc12 C1(C(=O)NCc2nc(CNC(=O)Cn3cnnc3)sc2)CCS(=O)(=O)N1 N1(C(CCCC(=O)NCC)=O)CC(NC(C23CCC2CC3)=O)CC12CCOCC2 C1(C(=O)NCC(CNC(CCc2ccc(C)s2)=O)CO)CCC2(CC1)CC2 N1(C(C(C2CC2)SC)=O)CCCC(C(=O)NOCC2CCC2)C1 c1(N2CCCC(C(C)NC(C(C)CF)=O)C2)ncnc2scnc12 CC(C)(CCNC(=O)C=CC1CCCC1)C(=O)NC(C(C)(C)O)C1CC1 C1(C(N2CCCC(CC(C)C)C2)=O)CN(C(C23CCC(C2)OC3C)=O)CCN1C c1(CNC2=NCC(C)C(CCC)N2)ccc(S(=O)(=O)N)c(F)c1.C(C)(C)OC N1(C(C=CC)=O)CCC(C)(C(N2CCC2C=C)=O)CC1 c1(C(N(CCC(=O)NCC2CCC(CC)CC2)C)=O)cc2n(n1)CCC2 N1(C(C2(OC)CC2)=O)CC2CCCC1C2CNC(c1cc(C2CC2)nnc1O)=O CCCS(=O)(=O)C(C)C(=O)N1CC(NC(=O)Cc2ccc(C)cc2)CC(F)C1 CC1(C)CCN(C(=O)CCC2CC2)C(C(=O)NCc2nccc(O)n2)C1 N1(C(CNC(C(C)OCC)=O)=O)CCN(C(=O)Cc2cn[nH]c2)CC1 CCCC(C)C(C)NC(=O)CC(C)(C)NC(c1ccncc1F)=O N1(C(c2cncc(NC)c2)=O)CCC2(NC(c3cnc(C)cn3)=O)CC2C1 C(=O)(C(C)(O)CC(F)(F)F)N1CCC(CNC(C(C)(C)N(S(C)(=O)=O)C)=O)CC1 C(=O)(CC(C)C(F)F)N(C1CCN(C(=O)CCc2c(N)cnn2C)CC1)CC#C c1(CC)nnc2n1CCCC2C(=O)N1CCC(NC(=O)COC)C1 c1(CC(=O)NC2CCN(C(C(C)CC3CCCCC3)=O)C2)ccc(O)cn1 NS(=O)(=O)CC(=O)NCc1cn(CCNC(C2CCOC2C(F)(F)F)=O)nn1 N1(C(CN(C2CC2CC(C)(C)C)C)=O)CCCC(C)(NC(=O)CN(C)C)C1 C1(NC(=O)Cn2cccc2)CCCC2CN(C(=O)Cn3cc([N+](=O)[O-])cn3)CC12 C(=O)(C1=CCCOCC1)N(CC(CC)NC(=O)C1=CCN(C)C1)C C1(NC(c2n(CC)c(O)nc2)=O)CN(C(=O)CCC=C(C)C)CCC1C(F)(F)F N1(C(C2C(=C)C2)=O)CCOCC(CNC(c2cc(-c3ccc(F)cc3)no2)=O)C1 Cc1cccc(CNC(C2C3CC2N(C(=O)C=Cc2cccc(O)c2)C3)=O)c1F C1(C(N2CC(CCNC(CCC)=O)OCC2)=O)CCc2nc(C)[nH]c2C1 c1(C(=O)NCC(CNC(CC2(OC)CCC2)=O)OC)cnc(-c2ccsc2)s1 C(C(=O)N(C1CCN(C(=O)CCNc2cccnc2)C1)CC)(C(C)C)OCC C1(C2(O)CCN(N(CC(F)(F)F)CC(C)C(=O)OC)CC2)(C(=O)NC)CC1 c1(N(C(CC(c2cccc(C)c2)C)=O)C)cccc2c1CCCC2 CCCCCC(=O)NCC1C(C)CCN1C(=O)CC12CC(c3ccccc3)(C1)C2 C1(CNC(CSCC=C)=O)CN(C(=O)C#CC2CCCCO2)C2(CCOCC2)C1 c1(OC)ccc(N)c(C(=O)NC2CCN(C(c3cc(Cl)cs3)=O)C2C)c1 c1(CC)ccc(C(=O)NCC2CC(O)CN2C(=O)CCC(F)F)cc1F C12(CCNC(c3cc(C(OC(F)(F)F)=O)no3)=O)CC(CNC(=O)C(F)OC)(CO1)C2 c1(C(c2nnnn2-c2ccccc2C)NCC(CSC)OC)cc(Br)c(C)s1 c1(NC(C(c2ccco2)NC(c2c(C)occ2)=O)=O)cccc(C(F)F)c1 C1(OC(C)C(=O)NC2CC2CNC(=O)CC(C)(C)C)CCOCC1 C1(COC)CN(C(c2cc(C)nn2C)C(=O)NCCCSC)C1(C)C CC1(C)CC2(CC(C(=O)Nc3ccc4c(c3)CCO4)C2)C1.N12CC(C)(C1)NC2=O c1(C(N2C(CC(C)(C)C)CN(C(C3CC3F)=O)CC2)=O)ccc2c(n1)OCCO2 c1(CC)ncncc1C(=O)NCC1CN(C(=O)Cn2nccn2)C2CC12 O=NN1CCCC1C(N1CCC(Cn2cc(CC(c3ccccc3)O)nn2)C1)=O C(=O)(C#Cc1ccc(Br)cc1)NC1Cc2c(nc(C)s2)CC1 N1(C(c2ccc(C(N)=O)cn2)=O)CCC2(CC1)CCN(C(=O)CCOC1CC1)C2 N1(C(CS(CCOC)(=O)=O)=O)CCOC2CN(C(=O)Cc3nonc3C)CC12 CCCCC(C)C(=O)NC(C(=O)NCC(C)(C)OC)C1CC1 C1(C)(NC(c2ccn(CC)n2)=O)CCN(C(C2CCC(C(=O)OC)C2)=O)C1 CC1(C)CC(NC(=O)CSc2nncs2)CN(C(C2C3CCCOC23)=O)C1 c1(NCC(c2ccc(N)s2)=O)ccsc1CNS(C)(=O)=O.C1(CO)CCC1 C1(CCOC)(C(N2CC(C(F)F)CC2CO)=O)CCN(C(=O)OC(C)(C)C)C1 C(=O)(C1=CCCC(C)(C)C1)NC(C)CC(=O)NCC1N(C(N)=O)CCCC1 Cc1ccc(C(N2CCN(C(=O)CCCCN(C)C)CC2C)=O)c(N)n1 C1(OCCCN(C)CC)CC2(C1)CC2C(=O)NOC(CO)C(=O)OC C(=O)(C(COC)OC)C1C(CC(=O)NC2CC(OCC)C2)C1.C1(C)CO1 c1(OC)c(Cl)cc([N+](=O)[O-])c(Cl)c1C(=O)NCc1cc(C(C)C)on1 CCC(C)(F)C(=O)NCC1CCCN1C(=O)CN(c1ccccc1)C C(=O)(CCCC(F)(F)C(F)(F)F)N1C(C)(C)C(NC(c2nc(Cl)cs2)=O)CC1 C1(NC(CSCCCC)=O)CN(C(c2ccc(C(=O)CF)cc2)=O)CC1SC C1(C)(C(N(CCC)CCNC(=O)CSCCSc2ccccc2)=O)CC2CC2C1 C1(C(=O)NC(CC(=O)Nc2cn(CC(=O)OCC)nc2)(C)C)CCCCC(=O)N1 c1(OC)c(C(N2CCC(NC(=O)C(CC(F)F)C3CCC3)C2)=O)cccc1F C(=O)(CCCC(CC)NC(=O)CC(C)F)N(CCOCC=C)C c1(C(=O)NC2C(NC(C(CCSC)O)=O)CCC2)ccnc2[nH]ncc12 C1(NC(CCSCC)=O)CCCC1C(c1nnnn1C)(C)OC Cc1nc2cc(C(=O)NC3CN(C(=O)C(C)S(N)(=O)=O)CC3N=[N+]=[N-])cnc2[nH]1 N1(CCC(=O)NCCC(CCC)C)C(=O)SC(=Cc2ccc(OC)cc2)C1=O c1(C(N2CCC(C)=C(Br)C2)C(=O)NC2CC(C(=O)OC)C2)cc(Cl)cc(Cl)c1Br C1(NC(C2CC(=C)C2)=O)Cc2ccccc2N(C(=O)C(C)C(CC)CC)C1 CC1CC2(CCN(c3ncnc4[nH]ccc34)CC2)CN1C(c1nc(=O)n(C)[nH]1)=O Cc1ccnnc1C(=O)NCC(C(C)(C)C)NC(c1ccc(F)o1)=O C1(CN)CN(Cc2c(O)cncc2Cl)CC12CC2 Cc1ccc(C(CNC(=O)C(F)=CC2CC2)NC(C2CCCN(C)C2)=O)cc1 C(=O)(C(C)(COC)CC)NCC1CCCN(C(c2cnn(CCOC)c2C)=O)C1 C1(C(C)C)CN(C(=O)CC2CC3C=CC2CC3)CCCN1C(=O)C1=COCCO1 C1(CNC(C(CNC(=O)Cc2ccc(C)cc2)OC)=O)CC2CCCC2C1 CC1(NC(=O)CCCC#N)CCN(C(c2cc(CS(C)(=O)=O)on2)=O)CC1 c1(C(=O)NCC(CC)N(C)C(c2cc(C3(C)CC3)n[nH]2)=O)cc(C)cnc1OC c1(C(=O)NCCC2OCCN(C(c3c(C)cc(CO)o3)=O)C2)cncn(C)c1=O C1(C(=O)NC(CCN(C(=O)C(F)C(C)(F)F)C)(C)C)CCC2(CCCC2)C1 Cc1cc(CN(C(=O)C(=O)NC2CN(C3CCC(C)CC3)C2)C)n(C)n1 N1(C(C2N(CCC)C(=O)CC2)=O)CC2(c3cn(CC=CCOC)nn3)CCC1CC2 C(=O)(C1=NN2CCCN=C2N1)N1CC(NC(C(CC)F)=O)C(F)CC1 n1(CC)ncn(NC(=O)C(F)(CNC(=O)CN(C)C(=O)OC)C(C)C)c1=O N(C(=NCC(C)(C)C(C)C)NC1CCCC(OC(F)F)C1)C(CC)C c1(OCC)cnc(C(N2CC(O)(C(F)C(=O)N(C(C)CN(C)C(C)=O)C)C2)=O)cn1 c1(C(c2n(CCOCC)nnn2)Nc2cnn(CCSC)c2)ccc(Cl)c(F)c1 CC(C(CO)NC(C1(SC2CC2)CC1)=O)NC(=O)C(=O)N(C)Cc1ccccc1 c1(C(=O)NCC2(C(C)(C)O)CN(C(c3cc(C)ns3)=O)C2)ccncc1C1CC1 c1(C(=O)NC(CNC(C(CC(C)C)F)=O)(C)CC(C)C)cc2cc(O)ccc2[nH]1 N1(C(CC(=C=C)C)=O)CC2C=CC1C(C(=O)NC13CC(c4ccccc4)C1C3)C2 C(CCCCC(=O)N1CCCCCC1CO)NC(=O)C=Cc1cnccn1 C(=O)(C(CC(C)C)C(N)=O)NCc1ccc(C(C)NC(COC)=O)cc1 C#CCCCCCC(=O)NC1CCCC(CC(=O)N(CC(F)F)CCO)C1 C(=O)(C1=CC(C)(C)C1)NCC1(NC(CC(CC)c2ccccc2)=O)CCCC1 CC#CCCC(=O)NCCCN(C(=O)Cc1ccccc1Cl)Cc1ccccc1 Cc1cc(N)c(C(=O)NC(CNC(c2cc3sccc3s2)=O)C2CCC2)cc1F c1(NC(=O)NCC(=O)NC2CCS(=O)(=O)C2)ccc(F)c(Cl)c1 N1(C(c2cc(C(C)C)nn2C)=O)CCCC(C(=O)Nc2cccnc2)CC1 CC1CN(C(=O)COc2ccc(Cl)nc2)CCN1C(=O)CCN1CCCC1 C(=O)(C1=CCCCC1)NC1(CC(=O)NCC(C(N)=O)O)CC1 c1(C(N(C)CC2CCN(C(=O)C=CCOCC(F)(F)F)C2)=O)cc[nH]c(=N)n1 c1(CNC(=O)NC2(CC)CCCCCCC2)nc2ccc(Br)cc2s1 N1(C(c2ccc(C)[nH]2)=O)CCC2CC12C(=O)NC(c1ccns1)C Cc1cscc1C(N1CCC1(C)CC(=O)NC1(C(C)C)CCC1)=O c1(C(=O)NC2CC(NC(C=CC)=O)C2)ccc2c(c1)c(I)nn2C Cc1cc(C(=O)NC2CCC(CNC(c3cnc(C(C)C)s3)=O)C2)nc(C)n1 N12CCCC(C1)C(=O)OC2(COC)C.C(=O)(C(C)CF)NCc1ccccc1 c1(C(=O)NC2CN(C(c3c(C#C)c[nH]n3)=O)C(C)C2)cc2ccc(Br)cn2c1 c1(CC)oncc1C(=O)NCC1CCN1C(=O)Cc1nc(-c2ccccc2)no1 C#Cc1cc(C(=O)NC2CCC(NC(C3(C(F)F)CCCO3)=O)C2)cc(F)c1 N1(C(C2(COC)C=CCC2)=O)CC2CCC1CN2C(=O)COCc1ccccc1 CC1COC2(C1)CN(C(c1sccc1CNC(=O)C(C)S(N)(=O)=O)=O)C2 c1(CSCC)ccccc1C(=O)NCC1(O)CN(C(=O)CC(C)N(C)C)C1 c1(NC(N2CC(C)(N(C(=O)CC(=O)OC(C)(C)C)C)C2)=O)cc(Cl)n(C)n1 C12(C(N3CCN(C(C(CC#C)C)=O)C(CC)C3)=O)C3CCC(CC13)C2(F)F N1(C(C(CC)C)=O)CCCC(C2CN(C(C)C(=O)Nc3ccc(Cl)c(F)c3)C2)C1 Cc1cc(C(=O)N(C2CCCC(NC(=O)C=CCCC(C)C)C2)C)cc(Br)c1 c1(CN(CCC(=O)OC)C(=O)NC(CSC)CO)ccccc1 c1(C(=O)NCC2CN(C(CC3CCC(C)(C)CO3)=O)C2)onc2c1CCCC2 CCCC(C#N)C(=O)NC(Cc1ccco1)C(=O)NC(c1ccnc(F)c1)C c1(CC)ccccc1C(CNC(=O)C(F)CC)NC(c1sncc1C)=O S(=O)(=O)(c1ccccc1S(=O)(=O)N(C)C)NC(C)Cc1cccc2c1CNC2 Cc1cc(NCC2(C)CCN(C(C3(C)CCN(C)CC3)=O)C2)n2nc(C)nc2n1 C1(CC)CN(C(=O)C=C2CCN(C)CC2)CCN1CCSC N1(C(C(C)(C)CF)=O)Cc2ccnn2CC(NC(C23CCCC(CCC2)C3)=O)C1 C(=O)(C(CNC(c1cccnc1S)=O)CC1CCCC1)NCC1CC(C)C1 C1(NC(C=CC2(C)CCOCC2)=O)C2CCCN(C(=O)CC3(C)CC3)C2C1(C)C C1(N(C(CSC)=O)C)CN(C(=O)Cc2ccc(-n3cnnc3)cc2)CC1F C1(C(=O)NCCc2c(OC)ccc(F)c2)COC2(CCC2)CO1 C(=O)(C1CCCc2nn[nH]c21)N1CC2(C(NC(C=C(C)Cl)=O)CCC2)C1 C1(CNC(COCC(C)(C)C)=O)COC(CNC(c2cn(CCO)nn2)=O)C1 CC(C)(C)CC(O)C(=O)N1CC(CNC(=O)Cc2ccsn2)C(F)(F)C1 Cc1cnc(C#N)c(-c2cc(C(=O)NCC3(O)CCC3)ccn2)c1 C1(C(=O)NCCCNC(Cc2n[nH]c(=NC)s2)=O)CCN2CCOCC12 c1(C(=O)NCC2C3CN(C(C4(C#N)CCCC4)=O)C2C3)cc2c(F)cccc2s1 C1(CC)CCC(C(=O)N(C)CCN2CCN(C(=O)C(C)N3CCC3)CC2)CC1 C(C)(C)(CC=CC(=O)NC(C)C(F)(F)F)NC(C1C(OC)CC1)=O Cc1ncc(Cl)c(C(N2CC(O)(CN(C(=O)C(O)C(C)N(C)C)C)C2)=O)n1 C1(NC(c2cscn2)=O)CCCCC12CCCN(c1ccc([N+](=O)[O-])cc1Br)C2 CCC(C(=O)NC1(CNC(c2ccc(OC)c(Cl)c2)=O)CCCCC1)C(F)(F)F c1(C(C(=O)NCCCN(C(=O)COCCF)CC)(C)F)ccc(F)cc1 C(=O)(CC(C)(C)C#N)NC1CC(NC(C2C(C(=O)NCC#C)C2)=O)C(O)C1 C#CCC(O)C(=O)NC(C)(CNC(c1ccc(CSCCC(N)=O)cc1)=O)CC N1(C(C=NOC)=O)CCC(NC(=O)C=Cc2sccc2Br)C(F)C1 C1(CC)COCC1(c1nnnn1C1CCC(C(=O)OC)C1)NCCn1cnnc1 CCCC(CC)C(=O)NC(CC)CC(=O)NC1CCC(OC)C1 S(=O)(=O)(CCNC(c1nnnn1CC1CC1)(CC)C1CCCC1)NC(C)(C)C c1(C(=O)NC2(CNC(c3cnsn3)=O)CCC2)ccc(-n2cnnc2)cc1 c1(C(=O)NC2CC(NC(=O)C(F)CC3CCCC3)C(O)C2)ccc([N+](=O)[O-])s1 CCCC(C(=O)N1CCC2C(C(N3CCC(NC(=O)NC)C3)=O)C2C1)C(C)C c1(CC)ncc(C(=O)NCCN(C(C2(CC)CCC2)=O)C2CC2)s1 CCC(C)(CC)C(=O)N1CCC(O)(C(C)NC(=O)CSCCC(C)C)C1 Cc1ccc2c(c1)CC(N(C)C(=O)C1CC1)C2.C1CCCC2(CNC2)O1 C(=O)(C(=O)C(C)(C)C)NC(C1CN(C(=O)CSCC2CCCCO2)CCO1)C Cn1ncc2c1CC(C(N1CCC(F)(CNC(=O)CCCCCF)C1)=O)CC2 C(=O)(C(C)CC(C)(C)C)NC(CN(C(c1cccc(OCC=C(C)C)c1)=O)C)C N1(C(Cc2[nH]c(=N)sc2)=O)CCC2(CC1)OCCCC2NC(=O)COC(F)(F)F C(c1nccs1)=CC(=O)N(C1CC(NC(=O)C(C)(C)N2CCCC2)C1)C c1(C(=O)NC2CC(C)N(C(c3cn(C)[nH]c3=N)=O)CC2)c[nH]c2ccccc12 CC1(C)C(C(=O)NC2CC3CC(NC(c4ccc(C#N)cn4)=O)C2C3)CC1(F)F N#Cc1ccc(C(N2CCC(O)(CNC(=O)CCc3ncc[nH]3)CC2)=O)c(O)c1 C1(CC)CN(C(C2CCC(C(C)C)N2C(c2ccncc2OC)=O)=O)CCN1C C1(C(N(CC(C)CNC(C2CCN2)=O)C)=O)CCCN(C(=O)N(C)C)C1 c1(C(N2CC(O)CC(NC(c3cc(F)cc(F)c3)=O)C2)=O)ccc2ncsc2c1 C1(CC=C)(NC(=O)CC(C)(C)O)CCN(C(C2CCC2(F)F)=O)CC1 C(=O)(C(C)(F)C(F)(F)F)N1CCC(C)(CNC(c2ncc(C)cc2C)=O)C1 C1(C(N2CC(CCn3cc(CN(C(C)C)C)nn3)C2)=O)CC(F)(F)C1C C1(CC)CCN(C(C)=O)C1C(=O)NCCNC(c1cncs1)=O N=c1nc2c(c[nH]1)CC(C(N1CCN(C(C3CC(=O)CO3)=O)CC(O)C1)=O)CC2 N1(C(C2C(=C)C2C(=O)OC)=O)CCC2(CC1)CC2CNC(=O)C=CCCC C1(NC(C(CC2CN(C(CC=CC)=O)C2)F)=O)CC(C)(OC)C1(C)C c1(C(=O)NC2C(C)CN(C(C3(C)CC3(C)C)=O)C2)cnc2ccc(Cl)cn2c1=O N1(C(C2C(C)C2)=O)CC(C)(C)OCC1CNC(c1ccn(CCF)n1)=O c1(NCC2C=CC(NC(=O)CNC(=O)C(O)c3ccco3)C2)ncccc1O C12(NC(Cc3cc(CC)nn3C)=O)CC3CCC(C1C2)N3C(=O)C(=O)NCC#N c1(C(=O)N(CCCNC(C2(Cl)CC23CCC3)=O)C2CC2)cc2c(s1)CCOC2 CCC(C)CCC(=O)N1CCOCC(NC(=O)CCNC(=O)CC(C)C)C1 N1(C(C2(CCC=C)CC2)=O)CC(CNC(=O)C=CC2CCCN2C)OC(C)(C)C1 C12(C(N(CCOCC#C)C)=O)CC(C)(CN1C(C1CC1CCC)=O)C2 CC(C)(CC(F)F)C(=O)NCCSCc1cn(Cc2ccccn2)nn1 Cc1cc(CNCC(c2cnn(C)c2)N2CCCC2)ncn1 C1(CNC(=O)COC2CN(C(=O)CC3CC(CO)C3)C2)CCCS1 CCCCCCC(=O)NCCC1(NC(C2CCN(OC)CC2)=O)CCCC1 C1(NC(CC2C(C)(C)OCC2)=O)CC12CCN(C(c1cccc(O)n1)=O)CC2 N1(C(CC2(C(=C)F)CCC2)=O)CC2(CCC2NC(c2cncc(C=C)c2)=O)C1 C=CCC(C(=O)N1CCN(CCCNC(C2(F)CC=CC2)=O)CC1)C(C)C N1(C(CNC(CC)=O)=O)CCN(C(=O)CC(C)C)CC1 C12(C(N3CCN(C4CCN(CC)C4)CC3)=O)CCC(F)C1CC2 C1(C(=O)NCCN(C(=O)CCCCC#N)C)CC2CCCCN2C1 N12CCCN(CC1)C(=O)CC(=O)N1CC(O)CC1C2=O.C(C)(C)(C)OC(C)=O CCC(CCc1ccccc1)C(=O)NC(C)CN(C(=O)C(C)CCO)C c1(C(=O)NC2(CNC(C(C3CCC3)OC)=O)CC2)ccnc(C(C)(C)O)c1 N1(C(CCSCCCC)=O)CC2CC(NC(=O)Cc3c(C)nn(C)c3C)CC2C1 N(C1CCCc2n[nH]cc21)C(C1CCC(=O)N(C)C1)=O.C#CCC1C(=O)N1 C1(N(C)C(c2cncc(Cl)c2)=O)CC(N=c2[nH]nc(C(C)(C)C)o2)C12CCC2 c1(C2(C(=O)NC(CN(C(=O)CCn3ccnc3)CC)C)CCC2)ccc(Cl)nc1 C1(NC(=O)Cn2ccnn2)CC2CC(NC(C3CC3[N+](=O)[O-])=O)C1C2 O=C(N=c1[nH]onc1C1CC1)C1CCN(Cc2cnc(C3CC3)s2)CC1O Cc1nc(O)nc(O)c1CC(N1CCN(C(=O)COC2CCC2)C(CF)C1)=O c1(OC)c(-c2ccc(C(=O)N(C)C3CC3)c(C)c2F)cc(C)cc1C c1(OC)cc(F)c(C(N2CCC(NC(=O)C(F)=C3CCCC3)C2)=O)c(F)c1 C=CCC(C(=O)NC(CC(=O)NCCC(C)C=C)C1CC1)NC(C)=O C1(C)(C(N2CC(NC(COCCCCC)=O)C(CCC)C2)=O)CCC12CCC2 c1(NC(C2C(NC(C(C(=O)OCC)C)=O)C2)=O)nccc(Br)c1Cl C#Cc1ccc(C(=O)N(CC)CC2CCCCN2C(=O)C(C)S(N)(=O)=O)nc1 C1(SC)CCC(c2nc(-c3cccc(OC(C)C)n3)nn2C2CCC2)CC1 c1(N2CCC(CC(=O)Nc3cc(OCC)ncc3)C2)nc(C)nc2c1CCC2 c1(CN2CC3CN(C(=O)COc4ccc(Cl)cc4)CC32)cc2ccc(Br)cc2s1 c1(C(N2C(C)(CNC(C=CS(C)=O)=O)CCC2)=O)nccn2ccnc12 CC1(C)CC(CNC(C2CCCC2O)=O)N(C(=O)C2=C(Cl)CC2)C1 N1(C(C(C)CF)=O)CC(NC(c2ccc(F)c(Cl)c2)=O)CC1(C)C CC(C(=O)NC1(CNC(=O)CC=CC(C)(C)C)CCC(F)(F)CC1)C(F)(F)C(F)F C(=O)(CCCCCNC(N)=O)N1CCC(NC(COC(CC)CC)=O)(COC)C1 C(=O)(C(O)CC(C)(C)C)N(CC(C)O)CCNC(c1n(CC)cnn1)=O c1(CC)nc(NC2CN(C(=O)C(C)(O)C3CC3)CC2C)ncc1C CC1(CCNC(=O)C=CC2CCCC2)CCN(C(=O)CS(N)(=O)=O)C1 N1(C(c2n(CC)nnc2)=O)CC(CNC(C2(SC)CC2)=O)CC12CCC2 N1(CC(N2C(CNC(c3c[nH]c(=NC)o3)=O)CCCC2)=O)CCC(=O)NC1=O C#CCC(C)(C)C(=O)NCC(C1CCC1)NC(=O)C(F)n1cccn1 c1(C(=O)NCCC2CC(NC(C(C)C(F)F)=O)C2)ccc2ccsc2c1 C1(C(=O)Nc2nc(C(F)(F)F)cs2)CCC(NC(=O)NC23CNCC2C3)CC1 c1(C(=O)NC(c2cncs2)C)cnn(CCNC(C2CSC2)=O)c1 S(=O)(=O)(CCCC1CC1)NC(=O)C(CN1CCCC1)c1ccccc1 C1(NC(C(C)c2cccs2)=O)CCC(F)(CNC(C2CC(=C3CC3)C2)=O)C1 C(=O)(C(CC(C)C)NC(C)=O)N(CCCNC(=O)CC1(C)OCCO1)CC c1(N(C2CN(C(c3ccc(Cl)c(Br)c3)=O)C2)C)ncc2ccccc2n1 c1(C(=O)NCC(CC=C)NC(=O)C#CC2CCOC2)cnn2cccc(C)c12 N1(C(CCC2CC(C)C2)=O)CCCC1C(C)(C)NC(=O)Cc1ncsc1Cl N1(C(CC2CCN(C(=O)NCCOC)CC2)=O)CC2COCC2(CO)C1 N1(C(c2cnsn2)=O)CCN(C(C2C(Cl)(Cl)C23CC3)=O)C(C2CCC2)C1 S(=O)(=O)(c1cccc(C(F)(F)F)c1)N1C(C(=O)Nc2c(C)nsc2)C=CC1 C(=O)(CC(O)CC(C)(C)C)N1CCC(CN(C(C2C(CC)C2)=O)C)CC1 c1(OC)cccnc1C(=O)NC(C)C(C)(C)NC(=O)CP(C)(C)=O c1(NC(C(Cc2cccs2)NC(=O)OC(C)(C)C)=O)ccncc1N1CCCC1 O(N=C1CCCCCC1)CC(=O)N(CC(CN(C(c1csc(C)c1C)=O)C)O)C C1(CN(C(CSCCC(C)C)=O)C)CCN(C(C2CN(S(C)(=O)=O)C2)=O)C1 C12(NC(CCC(=O)OCC)=O)CCC(CN(C(=O)C(F)C(C)(C)O)C1)C2 Cc1ncc(C(N2CCN(C(=O)C=Cc3ccc(Cl)cc3)C(C)C2)=O)cc1C#N Cc1ccc(O)cc1CNC(C1N(C(c2ccc(Cl)cn2)=O)CCC1(C)C)=O CC(CC(=O)NC1CCC1NC(c1cncnc1)=O)C(F)F C1(C(=O)NC2C(NC(CCC(=C)Cl)=O)COC2)CCc2nc(C)sc2C1 N1(C(COCCC=C)=O)CC(C)CN(C(c2ccoc2)=O)C(C)C1 CC1(NC(=O)CCc2ncco2)CCN(C(=O)Cc2ccc(C(F)(F)F)cc2)C1 c1(C(N2CCCC(C(C)NC(c3cnc[nH]c3=N)=O)C2)=O)ccc2scnc2c1 C1(NC(C2(F)CCCC2)=O)CC2CCC(C1)N2C(=O)CCCn1ccccc1=O c1(C(N(C(CNC(c2cc(C)c(Cl)s2)=O)C)C)=O)cncc2sccc12 C1(NC(C2(COCC)CC2)=O)CCC(C)(C)N(C(=O)CC(C)n2ccnc2)C1 C1(C(=O)O)CCN(N2CCC(c3ccccc3)(C(=O)O)CC2)CC1 N1(C(CN(CC)CC)=O)CC2(CNC(=O)Cc3ccc(Cl)cc3)CCC1C2 N1(C(C2C(CC)C2)=O)CCCC2CCN(C(=O)CSCc3cscn3)CC12 CCCC(CNC(=O)CCCNC(N)=O)C(=O)N1CC(N(C)C)C(C)C1 N1(C(CC2C(C)CCO2)=O)C(C(=O)NC2C=CCC2)CC2CC12 C1(C(=O)Nc2c(N)sc(-c3ccccc3)n2)CC2CN(C(c3cccs3)=O)CC12 c1(C(=O)NCC(CCOC)NC(c2sc(=N)[nH]c2C)=O)cc(C)ccc1F c1(C(=O)NCCNC(COCCCOC)=O)ccncc1O CC(C)(C)CCC(=O)N1CC2CC1C2CNC(C1NC(=O)OC1(C)C)=O c1(C(N2C(CCNC(C(C=C)(C)O)=O)CCCC2)=O)cn2ccnc2cn1 C=CC(C)(C)CC(=O)N1CC(CC)(NC(C2C3CCC(=O)C23)=O)C1 CC1(C)CCN(C(c2ccsc2Cl)=O)C1CC(=O)NCC(C)(O)C1(C)CC1 C1(C(=O)NCC(C)(C2CC2)NC(c2coc3c2COC3)=O)CC(S(C)(=O)=O)C1 C(CC(C)(O)C(=O)NC1CCOC(C(N2CC(C)(C)CC2C)=O)C1)N(C)C C1(C(=O)NCC(C2CCC2)OC)OCCC1CNC(=O)CN1CSCC1=O c1(C(=O)NCC2N(C(C(C=C)O)=O)CC(C)(C)C2)cc2cc(OC)ccc2cn1 CN1C(=O)CCC1C(=O)NC(C)(CNC(c1[nH]ccc1C1CC1)=O)C1CCC1 c1(C(=O)NCC2CN(C(CCC)=O)C3(C2)CCC3)cnc2c(C#N)cnn2c1 Cc1cn2c(C(=O)NC3CCCN(C(=O)CS(=O)(=O)C4CC4)C3C)c(C)nc2s1 C12(NC(C(CC3CCC3)OC)=O)CCCCCC1N(C(c1csc(Cl)n1)=O)CC2 C1(C(=O)NCCCn2c(C)nnc2)CCOCCN1C(=O)C1=CCSC1 N1(C(C2=CC(C)(C)C2)=O)CCCC2(CCN(c3nc4cc(F)c(F)cc4s3)C2)C1 C1(CC(=O)NC2CCN(CCC)C2)COCCN1C(=O)CCc1cccc(C)c1 c1(CC)ccc(C(=O)NCC2(C)CCCN2C(=O)CC(C)(C)F)nc1 N1(C(C(C=C)CC)=O)CCC(C2CC2)C1C(N1CC(C)(C)C1C(=O)OC)=O N1(C(C2N(C)CCOC2)=O)CC(NC(c2ccc(-n3cncn3)cc2)=O)C2CC2C1 C=C1CCN(C(=O)CC(F)(F)F)C(C(NC[Si](C)(C)C)=O)C1 C#Cc1ccc(C(N2CCC(CO)(CNC(=O)C#CC(C)C)C2)=O)cc1F S(=O)(=O)(c1ccc(NCC(O)CC(N)=O)c(Cl)c1)NC1(C)CCCOC1 c1(C(N2CCC(CN(C(=O)CCC(=O)N(C)C)C)C2)=O)[nH]c2ccccc2c1Cl C1(NC(C(CC)C(C)O)=O)CCC2CN(C(C3CC3(F)F)=O)CCC2C1 C(N=c1nc2ncn(C)c2c(NCCCC(F)(F)F)[nH]1)c1c(C)cc(C)cc1C CCCCC(O)C(=O)N1CCC(NC(c2n[nH]cc2I)=O)CC1 n1(CC(N2C(CNC(C(C(C)C)n3cncn3)=O)CCC2)=O)nc(O)ccc1=O C1(NC(c2ccc(CNC(C)=O)s2)=O)CC2(C1)CN(C(C1CCOC1)=O)C2 C1(CCC)(CC2CC2)CCCN1C(=O)CC1CCN(CCc2ccccc2C)C1 CC(CCC(=O)NC1CCCC(NC(=O)CCCCN2CCOCC2)C1)N(C)C C(=O)(C#CC1CCCO1)N1C(C)(CNC(c2cc(C)sc2)=O)CCC1 C=CCC(C(=O)NCC1CC(NC(c2cc3c(s2)CCCC3)=O)CCO1)C(C)C C1(CNC(Cc2c(C)ccc(F)c2)=O)CC2CCC1N(C(C1CC(C)(C)O1)=O)C2 C(=O)(C(C)C(C)(C)C)NC1(C(=O)NC(c2ccn(C)n2)CC)CCC1 C12(CNC(=O)CCc3ccc(Cl)s3)CCCC1N(C(=O)CCCC1CC1)CCC2 c1(CN2CC(NC(c3cccc(C(N)=O)c3)=O)C(O)C2)c(Cl)ccc(F)c1F C1(c2onc(C(C3CC4CNCC34)C)n2)CC12CCN(C(=O)OC(C)(C)C)C2 Cc1nc(Cl)nc(N2CC3(COC(CNC(C4CCCCC4)=O)C3)C2)c1F c1(-n2cc(C3CN(C(=O)CCn4cccn4)C3)nn2)ccc(F)cc1 N1(C(C(C)OC)=O)CCC2(CCC(CNC(c3cccc(Cl)c3C)=O)CC2)CC1 C(=O)(CCC(C)NC(=O)C=C(CC)CC)N(CCCC=C)C C1(N(C(=O)C=CCF)C)CN(C(C2CC2C#N)=O)CC1O Cc1cccc2c1N(C(=O)CCCCN1CCCC1)CCN2 Cc1cc(Cl)c(C(=O)NCC2CC2CNC(=O)CC2CC(F)(F)C2)cc1C c1(CCC(=O)N(C2CCN(C(=O)CNS(N)(=O)=O)C2)CC)ccc(F)nc1 c1(C(=O)NCC(=O)NCC=C)ncc2n1CCNC2 c1(OCC)cccc(CCC(=O)NC(CNC(C2C3CC4C(C3)C24)=O)C(C)C)c1 N1(C(c2cc(OC)ncn2)=O)CC(C2CCCN(C(=O)C(O)CCC(C)C)C2)C1 c1(C(=O)NC2(CNC(=O)CC3CCC3)CCOCC2)cnc2cc(O)ccc2c1 CCCC(C)N(CCC(=O)NCC1(N(C)C)CCC1)NC(=O)CC1CCC1 C=CC1(C(=O)Nc2cscc2C)CCN(C(C2CNC(=O)CC2C)=O)C1 N1(C(C2CCN2C(c2nccs2)=O)=O)CC2CCC(C1)O2 N1(C(c2ccc(C(C)=O)s2)=O)CCCCC1C1(NC(c2ccccc2Cl)=O)CC1 c1(C(N2CCN(C(=O)C=CCF)CC2CO)=O)cc(F)c(CO)c(F)c1 c1(C(N2C3CC(CC(NC(CC#N)=O)C3)C2)=O)cc2ccc(Cl)cc2s1 N1(C(C(C=CCCC)O)=O)C(C)CC2CN(C(c3nn(C)cc3Cl)=O)CC12 c1(C(=O)NCC(CNC(=O)C(C)N(C)C(C)=O)OC)ccc(S(C)(=O)=O)[nH]1 c1(C(=O)NCC(CC)NC(c2c(Cl)cnn2C2CCCC2)=O)cn(C)nc1O C1(OC)CN(C(C2(C)CCCC2)=O)CC1C(=O)NCC(C)CC1CCC1 c1(C(N2CCC3C(C2)CN3C(=O)C(O)CN2CCCC2)=O)cccc2c1NCC2 c1(NC(CC2C(CNC(COCC)=O)C2)=O)cncc(Br)c1C C1(C(=O)NCCN(C(c2c[nH]nc2C2CCOC2)=O)CC)(CO)CC=CC1 C1(NC(CCC(=O)NCCC)=O)CC2CC1N(C(c1csc(=NC)[nH]1)=O)C2 CS(=O)(=O)C1(C(=O)NC(CNC(c2cccc[n+]2[O-])=O)C2CCC2)CCOCC1 c1(C(=O)NC2CCCC(NC(C3(C)CC3(F)Cl)=O)C2)ccc2ccccc2c1O C1(CC)CNCCC1NC(c1ccc(C)cc1)CO c1(N(C)Cc2ccc(C)o2)nc(N2CC(=O)NC(C(C)C)C2)c2ncccc2n1 CC(C)C(O)C(=O)N1CC(F)CC1CNC(C1C2CCC1CC2)=O N1(C(CCC(=O)NC(c2c(C)c(Br)ccc2)C2CC2)=O)CCSc2ccccc21 C(c1ccccc1Cl)=CC(=O)NCC1N(C(c2cc(C(C)=O)c(C)o2)=O)CCC1 c1(C(N2CCN(C(CC=C=C)=O)CC(CO)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(C(N2CCC(N(C(c3c(O)cc(C)nn3)=O)C)C2)=O)cccc2c1CCC2 Cc1ncc(F)c(N2CCOCC2CN(C)C(C2CCC(C)C(C)C2)=O)n1 c1(C(N2CCC(N(C(=O)C3=NOCC3)CCC)C2)=O)ccc2cnoc2c1 N1(C(C(C)=CC)=O)CC2ON=C(CNC(=O)CSS(C)(=O)=O)C2C1 c1(CC(c2n(CC)c(N3CCCC(C)C3)nn2)C)ccc(F)c(F)c1 C(C(O)C(=O)NC1(CO)CN(C(=O)C(F)CC2CCOC2)C1)=CC c1(OCC)sccc1C(=O)N(C)CCNC(=O)C(C)CSC(F)(F)F N1(C(C(=O)NCC(c2cccc(F)c2)N(C)C)=O)CC2CS(=O)(=O)CC2(C)C1 N1(C(COCCC#C)=O)CCC(C(=O)NOCC(O)CO)(C(=O)OC)C1 N1(C(C=CC=CC)=O)CCC(NC(c2cn(C(F)F)c(C)n2)=O)C(O)C1 N1(CC)C(=O)CCC1CC(N1CCC(O)(CN(C(=O)CC2(C)CCOC2)C)C1)=O Cn1cc(Cl)cc1C(=O)NC(CNC(c1cccnc1O)=O)C1CCC1 N#Cc1cc(Br)ccc1C(N1CC(NC(=O)COc2ccc(Cl)nc2)C1)=O Cc1ccc(C(N2CCC(C(C)NC(C3(C(C)C)CCCO3)=O)CC2)=O)c(C)c1 C1(C(=O)NC(C)C#N)CC2(CCN(C(c3ccnc4cc[nH]c34)=O)C2)C1 c1(NC(c2noc(C)n2)CC)cc(C)c([N+](=O)[O-])cc1Br c1(C(=O)NC(CC(=O)NC(CO)CCF)CC2CC2)cnn2c1CCC2 C(=O)(C1=CC2CCCC12)NC(C1CCN(C(C(COC)C)=O)C1)C CCC(C#N)C(=O)NCC1CCCCN1C(=O)Cc1cccnc1 c1(C(N2CC(C(=O)NCC3CCOC3C)(CC)C2)=O)c(C)nsc1C c1(N2CCN(C(C(n3cc(C4(O)CSC4)nn3)C)=O)CC2)cncc2nnnn12 C(=O)(CCN=C(NCc1sccc1C)NCC1CCCC1N1CCOCC1)NC CCCCCCCCC(=O)N1CC(CNC(=O)COCCC)C2(CC2)C1 c1(OC)cc(F)ccc1NC(C1C=CC(NC(c2cn(C)nn2)=O)C1)=O C12(NC(C(CC)CC)=O)CN(C(c3c(C)ccc(C)c3C)=O)CC1CS(=O)(=O)C2 N1(C(c2ccc(C)cc2O)=O)CCCC2(CCN(C(c3c[nH]c(Br)c3)=O)C2)C1 CC1(C)C=C(C(=O)N2CC(F)(F)CC2CCNC(=O)C(F)OC(F)(F)F)C1 C1(C(N(CC)Cc2cnn(C)c2)=O)COC2(C1)CN(C(C1CC3(CC3)C1)=O)C2 C12(C(=O)NC(CCC=C)CO)CC(CN(C(c3nc(COC)oc3C)=O)C1)C2 N1(C(CS(N)(=O)=O)=O)CCCC2CCN(C(=O)COCCF)CC12 c1(C(C(=O)NCC)N(C)C(c2cccc(Cl)c2)C)ccc(CC)nc1 C1(CNC(CCCC(C)=O)=O)C2CCCC1N(C(C1CC1C)=O)C2 C=C(C(=O)N1CCN(C2CCN(Cc3cc(C#N)ccn3)CC2)CC1)C(F)(F)F c1(C(N(C2CCC(n3cc(-c4ccccn4)nn3)CC2)C)=O)ccc(C#N)cc1 N1(C(C(CC)N(C)C)=O)CCC2(CC1)CC(NC(c1cc(Br)n[nH]1)=O)CO2 c1(N(CCOC)Cc2cccc(C)c2)cc(=NC(C)CC2CCC2)[nH]c(Cl)n1 c1(CC(=O)N(CC(=O)NC(C#C)CC2CCC2)C2CC2)ccnn1C C#CCCCC(C)C(=O)NC1CCC12CN(C(c1cnc(Cl)s1)=O)C2 C12(CNC(c3c(C)nco3)=O)CCCC1N(C(=O)C(C)C(C)C)CCC2 C1(NC(c2nc(C)[nH]n2)=O)CN(C(=O)C(C)Sc2ccccn2)CCC1C c1(C(=O)NC(C2CCCN2C(c2ccn(CC(F)(F)F)n2)=O)(C)C)ccc(Cl)o1 Cc1cc(C(=O)NC(CO)C(C)NC(=O)Cc2cc(Cl)n(C)n2)c(C)s1 CC1(C)NC(=O)CC1C(N1CCC(C(=O)NCC2(O)CCOC2(C)C)CC1)=O c1(C(=O)NC2(C)CC(NC(C(CC)(C)COC)=O)C2)cn2c(n1)CC(C)CC2 c1(C(CC)NC(C2CCC2CNC(=O)CCNC(=O)CO)=O)ccn(C)n1 c1(N2CCC(CC=C)C2)nc(N2CCC(N(C)C)(CO)CC2)nc2ccccc12 c1(-c2ccc(SC)cc2)c(C(=O)NC(C2CCC2)C2CC2)nn2c1CCCC2 CCCC(C(O)C(=O)N1CC(N(C)CCOC)C1)NC(=O)CC(=O)OCC Cc1cc(C(=O)NC(CNC(c2coc(C3CC3)n2)=O)C2CCC2)nn1C(F)F C1(C2CCCN(c3nc4cccc(Br)c4o3)C2)(NC(C2=NOC(C)C2)=O)CC1 C=CC1(CC(=O)NC2CCC(C(C)C)CC2)CN(C(=O)CN2CCC(OC)C2)C1 C=CC(C)(CC)C(=O)NC(CNC(C1CC(O)CN1C(N)=O)=O)CC(C)C N1(C(c2c(C)cc(OC)c(C)c2)=O)CCCC2c3ncn(C)c3CCC12 N1(C(CN(CC)CC)=O)CCC2C(NC(c3cc4scnc4[nH]3)=O)CC12 c1(C(N(CCNC(C(C2CCOC2)OCC)=O)CC)=O)cccc2c1C(=O)CC2 c1(C(CC)NCc2ccnn2C)cc(O)ccc1F C1(NC(C2CCC(NC)CC2)=O)C2CCC(C2)C1C(N1CC2CCC2C1)=O C(=O)(C(F)(F)c1cnn(C)c1)N(CCC(C)NC(=O)C(C)CN1CCOCC1)C CC(O)(CNC(=O)Cc1cc(C2CC2)on1)CNC(=O)Cn1nccn1 C1(Cc2cn(CCOC(C)=O)nn2)CCCN(C(=O)CC2CCCOCC2)C1 c1(OCC)ccc(NC(C2CC(=O)N(c3ccccc3C)C2)=O)cc1S(N)(=O)=O N1(C(CC=CCNC(C(C)NC(N)=O)=O)=O)CCc2nc[nH]c2C1 c1sc2c(c1C=C)CCC2.n1(CC(=C)C)nnc2c1CCCC2 C(CCSC)(C(=O)NCCCN1CCCC1C)NC(CC(C)c1ccco1)=O.C1CC1 c1(C(=O)NCC2CCCCN2C(C2CCC(F)CC2)=O)cnn2c1OCCCC2 c1(C(=O)NC2CC(C)N(C(=O)Cc3csc(=N)[nH]3)C2)cc(C2CC2)cc(F)c1 CCC(CC(C)C)C(=O)NC1CCCC1(C)CN(C)C(c1nc(C)ncc1Cl)=O c1(CN(C2CC(c3c(C)con3)C2)C=O)cc(Cl)cc(Br)c1OCCO c1(CC(CNC(NC(CC)C)=S)C)ccccc1Cl C1(NC(C2(C)CCCN2C(c2ncccn2)=O)=O)CCn2ncnc2C1 C(=O)(CC(C)CC(F)(F)F)NC1CC2CC(NC(c3c(C)csc3)=O)CC21 c1(C(N2C(CNC(CCOC)=O)CCCC2)=O)ccc(C#N)cc1Br C1(CNC(c2c(Cl)cc(C)s2)=O)CN(C(c2ccc(C(N)=O)s2)=O)CCC1(C)C c1(OCC)ccc(C(C)NC(C2(F)CN(C(c3cnn(C)c3Cl)=O)C2)=O)cc1 C1(NC(CCCOC(C)(C)C)=O)C2CC3C1C3C2C(N1CCC(O)(C(F)F)C1)=O c1(C(N(CC(C)NC(c2ccc(-c3ccon3)cc2)=O)C)=O)cnn2c1OCC2 C(CN=c1[nH]c(=NC(C)CCn2ccnc2)[nH]c2c1CC(C)CC2)N(CC)CC C1(C(=O)NC2CC(N(C(CCCCC=CC)=O)C)C2)C2CCCCCCC12 C(=O)(CC(C)(C)CC(=O)NCCCCc1cn(-c2cnnn2C)nn1)OC N1(C(C(CSC)O)=O)C2CCC1CC(F)(CNC(=O)C=Cc1cnn(C)c1)C2 C(C(CC)CC)N(C(C(c1cnn(C)c1)NC(CCC)=O)=O)C(C)C n1(CCN(C)C(C2CSCCN2)=O)cc(COCC(F)(F)F)nn1 O=C(O)CCCCCCCOC(=O)CC1SC2=NCCN2C1=O C(C1CCCCC1)=C(C(=O)N(CC(C)N(C(CC(C)C)=O)C)C)F C1(c2n(CC(=C)C)nnn2)(NC(C2CCOCC2)CC)CCS(=O)(=O)CC1 C1(CC)CCCC(NC(C2CC(F)(F)CN2C(c2cnc(OC)s2)=O)=O)CC1 CCCCC(C(=O)N(C(C)CNC(=O)CC1(O)CCC1)C)ON=C(C)C C(=O)(CC(F)(F)F)N(C1CC1)CC1N(C(C(Cc2ccsc2)NC=O)=O)CCC1 c1(C(=O)NC2C(CNC(C(C(C)(C)C)N(C)C)=O)C2)csc(=NC2CC2)[nH]1 CC(CNC(=O)Cc1cncnc1O)C(F)C(=O)NCCCC(N)=O C1(CC(N2CC(C(C)OC)C2)=O)CCCCN1C(=O)C=C1CCC(C)CC1 N1(C(C2OCCN(C)C2)=O)CC2CC(C1)C2NC(=O)C(O)CC1CCOCC1 Cc1cnc2nccc(C(N3CC4CC4(CNC(C4CC4(Cl)Cl)=O)C3)=O)c2c1 C1(OC(C)C(=O)OCC2CCC2)CCCCC1.C1(C(N2CCC2)=O)CC(O)CN1 CC1(C)CCOC(C(=O)NCCCOCCNC(=O)CSc2cccs2)C1 N1(C(c2c(SC)cccc2)=O)CCN(C(C2(C3(O)CCC3)CC2)=O)CC(C)C1 C(C)(C)(CCC(=O)NC1CCCC(NC(c2ccc(C#N)[nH]2)=O)C1)OC n1(CC2(C)CCC2)cc(CC2CCN(C(=O)CN3CCSCC3)C2)nn1 N1(C(=O)NC(c2cccc(C)n2)CC)CCOC2CNCC12 C1(CNC(C(C)OCCCC)=O)CCCC12CCN(C(C1(C#N)CCC1)=O)CC2 N1(C(CC(CCC)(C)O)=O)CCN(C(C2CCC(=O)NC2)=O)CC12CCC2 C(CC(C(=O)NCC(C1CC(C)(C)C1)O)NC(=O)CC1(C#N)CC1)=CC c1(CSC(CC)C)nc(C(C)OC)n(-c2ccc(F)cc2)n1 C1(CC(=O)NCCCN(C)C(c2ccc(CO)s2)=O)CCCS1(=O)=O Cc1nc(C)c(Cn2c(N3CCC(OCc4ccccn4)C3)nnc2C(C)C)[nH]1 C1(C(=O)OCC)OCCNCC1N(C(c1ccc(C)nc1C)=O)C(C)C c1(N2C(C(=O)NCCC(=O)NCCCCC#C)C=CC2)ncc2c(ccn2C)n1 CC1(NC(=O)Cc2cnsc2)CCN(C(c2nc(-c3cccs3)no2)=O)C1 c1(CN2CCN(C(CCOC)=O)C(CC#N)C2)cn(C)c2cc(F)ccc12 c1(CCC)n[nH]cc1C(=O)N(CC(O)CNC(c1ccsc1)=O)C N1(c2cc(C)nc(N3CCCC(C)(F)C3)n2)CCC(N)C(C)(C)C1 O=S(=O)(c1cc(Br)c(Br)s1)N1CC2CCC(C1)N(Cc1ccc(Cl)c(Cl)c1)C2 N(C(=NCCc1ccccc1)Nc1ccc(OC)c(OC)c1)C(C#C)C1CCC1 c1(OC)cccc(N(C(=O)C(C2CN(C(=O)CNc3ccccn3)C2)OC)C)c1 C1(C)(NC(C(n2cc(Cl)cn2)C)=O)CCCN(C(=O)C(N2CCC(C)CC2)=O)C1 N1(C(C2C(C#C)C2)=O)CCC2(CC1)CCN(C(C1CCc3ccnn3C1)=O)CC2 CC1(C)CC(NC(=O)C(F)C(F)(F)F)CCN(C(C2(C(F)F)CCCCC2)=O)C1 CC(C)C(C(=O)NC1CN(C(C2(OC(N)=O)CC2)=O)CC1C(F)F)NS(C)(=O)=O Cc1ncc(-c2cn(CC3(O)CCC3)nn2)cn1 CC1CN(C(C2(C3CCCO3)CCC2)=O)CC1n1cc(-c2ccncc2F)nn1 C1(CCNC(c2conc2C(F)(F)F)=O)CCCCN1C(C1CCCC12CC2)=O c1(C(N2CCCC(N(C(COCCOC)=O)C)CC2)=O)cc2ccc(Cl)nc2s1 Cc1ccn(C)c(=O)c1NC(=O)C(F)CC1CN(C(=O)CCc2nc[nH]n2)C1 CCC(O)C(C)C(=O)NC1(C(=O)NCCC(C)(C)CO)CC(F)(F)C1 c1(C(N2C(C(N3CCC(CSC)C3)=O)C=CCC2)=O)ccccc1C#N C(=O)(CC(C)C)NC(CCN(C(C1CC(C(=O)OCC)C1)=O)C)C CCC(CC1CC1)C(=O)N1CCC(N(C(=O)CC#N)CC2CC2)CC1 C(=O)(CCCCC(=O)N1CC2CC1(C(=O)NC1CC1C1CC1C)C2)OC c1(N(CCNC(C(C)SC)=O)CCOCCO)ncc(C)c(C)n1 c1(CC)ccnc(CNC(=O)C(CO)NC(C2CC23CC3)=O)c1 C1(NC(CN(CC(C)C)C(c2ccc(C)o2)=O)=O)CNC(=O)C1(C)C N(C(=NCc1ccccc1Cn1cccn1)NC(C)C)C(C#C)C(C)C Cn1ccc2cccc(C(N3CCC(CN=c4nn[nH]n4C)C3(C)C)=O)c12 C1(CNC(NNc2cn(C)nc2)=O)C2Cc3cc(Cl)ccc3C12 C1(NC(c2c(CNC(C(C)(C3(C)CC3)OC)=O)cco2)=O)Cc2cscc2C1 C1(NC(Cc2cc(OC)c(C)cc2)=O)CN(C(=O)C(O)CN(C)C)CCC1(C)C C1(C(=O)NC(CN(C(c2cnc3sccn23)=O)CC)C)CCc2c[nH]nc2C1 CCC(C)CC(=O)C(=O)N1CCC(C(=O)N(c2cccc(F)c2)C)C(C)(C)C1 c1(OC)cc(F)c(C(=O)NCC2CN(C(c3cc(C)c(F)c(C)c3)=O)C2)c(Cl)c1 c1(NCC(C=C)C)ncccc1S(=O)(=O)NCc1cccn(C)c1=O c1(C(=O)NC2CC(NC(c3n(C)ncc3[N+](=O)[O-])=O)C2)cnc2c(c1)ncn2C N1(C(C(C2CCN(C(C(CC)C)=O)CC2)C)=O)Cc2n[nH]cc2C1CO N1(C(CCC(C)NC(c2ccc(C#N)o2)=O)=O)CCC2CCC(C1)S2 CCCCC(O)CC(=O)N1CCC(C)N(C(c2nc(C)ncc2Cl)=O)CC1 CCCCCCC(=O)NCc1cc(C(=O)NCc2ncc(C)s2)co1 C#Cc1cnc(C(=O)NC(CCNC(=O)C(C2CCCCC2)O)C(C)C)c(C)c1 N(C)(C(=NCCC#N)NCCCOC1CCC1)CCN(CCCC)C c1(C(N(C(c2ccncc2)C)C)=O)cnc(CNC(=O)CC2CCOC2C)nc1 C(=O)(CCCCCC(C)O)NCC(C(C)C)NC(C(C)(C)SC)=O CC1(C)CCC(N=c2[nH]c(=NCCC34CCCC3C4)c3cc(F)cc(F)c3[nH]2)C1 c1(C(=O)NCC2(CNC(C34CCC(CO3)C4)=O)CCCC2)ccn2nnnc2c1 C1(C(=O)NCC2(F)CCN(C(C3(CF)CCC3)=O)C2)OCC2CCCC1C2 C=CC(C)(C)C(=O)NCC1CCCN(C(=O)CC23CCCC2C3)C1 Cc1c(O)ccc(C(=O)NC2CCCC(NC(=O)C(O)C3CCCC3)C2)c1C C(C(CNC(c1cc2occc2s1)=O)C(F)(F)F)NC(c1nc(C)nn1C)=O c1(SC)nc(N2CCC(C(=O)Nc3cc(C)no3)C(O)C2)ncc1Br C1(O)(C(=O)NC2CC(OCC(=O)NCC3OCC(C)C3)C2)CCOC1(C)C C1(NC(COC2CC(NC(C(=Cc3ncn(C)c3)F)=O)C2)=O)CC2CCC(C1)S2 N1(C(CC2CC(=O)NCCC2)=O)C2CCC1CN(C(C1COCCO1)=O)CC2 N1(C(C)C)CC(N=c2[nH]c3c(c(=NCCCn4cccn4)[nH]2)COCC3)C1 c1(NC)c(C(N2CC(CNC(=O)CC3CC3(C)C)C(O)C2)=O)sc2nccnc12 c1(C(=O)NCC2(O)CC(CNC(C3(O)CC(CF)C3)=O)C2)ccn2nccc2n1 C1(NC(C(CC=C)CC)=O)CCC2(CC1)CN(C(C1CCN(C)CC1)=O)CCO2 c1(CC(=O)NC(CN(C(=O)CN2CCOCC2)CC)C)cccc(COC)c1 N1(C(C2N(CC)CC2)=O)CCCC1CNC(=O)CCc1cn(C)nn1 c1(OC)cc(Cl)c(Cl)cc1C(N1CC(NC(=O)C(F)(F)C(C)O)CC(C)C1)=O c1(-c2cn(CCCN(C(C3(C)CC3)=O)C3CC3)nn2)ccc2c(c1)OCO2 C1(NC(c2c(C(C)(C)C)con2)=O)CC2CN(C(=O)C3=CCOC3)CC2C1 N1(C(C(C)C(C)(F)F)=O)CC(CNC(C2(O)CCC2)=O)CC12CCOCC2 C(=O)(C(CNC(C1CC1Cl)=O)C(C)(C)C)N(CCC)C N1(C(CSCCC)=O)CCN(C(=O)CC(C)COC)C(c2ccnn2C)C1 c1(C(N(C(CCNC(C=CC(=O)OCC)=O)C)C)=O)nnn(C)c1CC c1(C(=O)NC2CC(C)(NC(=O)C=CCF)C2)ccnc(CO)c1 C1(NC(CCOC)=O)Cc2ccccc2C1NC(c1ccc(N(C)C)cc1C)=O CC(C)(C)CCC(=O)N1CCCC(NC(c2cnc(C(C)(C)C)s2)=O)C1 Cc1nonc1CNC(=O)C(CC1CCC1)NC(=O)C(C1CC1)C1CC1 C1(OC)CN(C(C2CCS(=O)(=O)N2)=O)CC1NC(c1cncc(Cl)c1)=O CC(C)C(C)(CNC(=O)CSc1ccoc1)NC(=O)COC1CCCC1 C1(C)(C(NOCC2CC(=C)C2)=O)CCCN(C(c2ncccc2C)=O)C1 Cc1ccn2c(C(N3CCC(NC(=O)CCC4CCC(=O)N4)C3C)=O)cnc2c1 c1(CC(N2CC(NC(c3cc(F)c[nH]3)=O)C3C2C3)=O)cccc2ccccc12 Cn1c(-c2cccc(NC(C3OCCC4CNCCC34)=O)c2)nc2ccccc12 c1(C(N(C2CN(C(C3CCN(CCF)CC3)=O)C2)C)=O)ccnnc1O C(N=c1[nH]c(N(C)Cc2ncnn2C)nc2ccccc12)c1c(C)cco1 C1(C)(C(N2CCC(CCNC(C(C)SCC)=O)C2)=O)CCCN(C)C1 Cc1cc(F)c(C(N2CCC(F)(C(=O)Nc3cnccc3C(N)=O)C2)=O)cc1Br c1(C(N2CCC(C)(CCNC(C3CC3C#N)=O)C2)=O)cccc(C(F)F)c1Cl C1(CCC(=O)N(CC(C)N(C(C)=O)C)C)(NC(c2csnc2C)=O)CCCC1 C1(C(=O)NCCOC2CN(C(C(C)=C3CC3)=O)C2)NC(=O)CC1C c1(C(=O)NC(C)CCNC(C2CCOC2)=O)cncnc1C1CC1 C=C1CC2CC(C1)CC(c1nnnn1CC1CC1)(NC1(CCO)CCC1)C2 Cc1cc(C(=O)NCC2(CO)CC23CCC3)c(O)nn1.N12CCCC(C1)C2=O CC#CCCCC(=O)N1CCCC1CN(C(C12CC(C)C1C2)=O)CC N1(C(CSC)=O)CC2(NC(=O)CC(C(F)F)c3ccc(F)cc3)CCC1C2 c1(C(N2CCCN(C(=O)CSC3CCS(=O)(=O)C3)CC2)=O)cn2c(n1)CCC2 N1(C(C(C(C)CNC(c2cnn(C)c2C#N)=O)F)=O)CCOCC(C)(F)C1 N1(C(C(C2CCN(C(c3ccccn3)=O)C2)C)=O)CC2CCCC2C1 c1(C(=O)NC2CN(C(=O)CC3CC(F)C3)CC2O)ccc2nc(C3CC3)oc2c1 C1(NC(=O)C=Cc2cccs2)CCCC12CN(C(c1occc1F)=O)C2 CON1CCC(NC(=O)C(Cc2cn[nH]c2)NC(C2CC3(CC3)CO2)=O)CC1 C#Cc1ccc(C(N2CCC(C(=O)NCCCCC3CC3C)C2C)=O)cc1C C(C(CC(F)(F)F)NC(=O)C(C1CC1)C1CC1)NC(C(C1CCC1)OC)=O c1(NCCNC(C(=O)OCC)CF)c(Br)c(Cl)cc(Cl)c1[N+](=O)[O-] N1(C(Cc2cccc(SC)c2)=O)CCCN(C(c2cnc3n2CCC3)=O)CC1C N1(C(C2(C#C)CC2)=O)CCC2(C1)CN(C(=O)CCN1CCC(F)C1)C2 c1(C(N2C(C)CC(CNC(C3C(C)CCCC3)=O)C2)=O)ccc2ccccc2n1 N1(C(C2CCN(CC)C2)=O)CCC(C(=O)NCC2CC(C)=NO2)CC1C c1(C(=O)NC(CN(C(=O)C(C)(O)c2ccccc2)CC)C)nnn(CC)c1C C(=O)(CCCN=[N+]=[N-])N1CCCC(CN(C(=O)CC(O)C2CCCC2)CC)C1 c1(C(=O)NC2C(C)CCN(C(CCCOC)=O)C2)cc2c(s1)COCC2 N1(C(C2(C)COC(=O)OC2)=O)CCC(C)(C)C(NC(=O)CCc2cn[nH]c2)C1 c1(C(=O)NCCCN(C(C(C2CCC2)OC)=O)CCO)cccc2nn(C)cc12 C1(CCC)CCCC1C(=O)N(CCN(C)C(c1cnoc1CC)=O)C(C)C CC1CCC(CCNC(=O)C(CC2CC2)NC(=O)C(C)O)CC1 C1(COCC)CCN(C(=NCCC(C)C)NCC23CCC(CC2)OC3)C1 c1(CC)c(C(N2CC3CC2(C(=O)NC(C)COCC2CC2)C3)=O)cnn1C C(=O)(CC(C)(C)CNC(c1cc(CO)on1)=O)NC(C)Cc1ccco1 S(=O)(=O)(c1ccc(NCC2CC23CC3)c(Cl)c1)NC(C)C(C)(C)CO c1(-c2ccc(NC(c3nccc(C(C)=O)c3)=O)cc2)c(C)nc(C)nc1O C=C(C)CC(C(=O)NC1CCC1NC(c1ccnn1CCN(C)C)=O)OC n1(CC(=O)NCC(C(C)C)NC(=O)CC(C)n2cccn2)ccc(=O)n(C)c1=O C12(C(N(CC#CC)C)=O)CCC(NC(C3CNC(=O)CC3C)=O)(CC1)C2 c1(C(N2C(CN(C(C=C(COC)C)=O)C3CC3)CCC2)=O)ccc(OCF)nc1 c1(-c2c(C(=O)OC)scn2)c(C(=O)NC(=O)C2=CC=NC(=O)C2)cc(Cl)cc1Cl C1(C(=O)NCC(CC)(CC)CC)CC2CC1CN(C(C1(C)CC1C)=O)C2 C1(NC(CC(C=C)C)=O)CC2CCC1N2C(c1cnn(CC2CCCC2)c1)=O C(=O)(C(C)(COC)CC)NC1CCN(C(c2cn(CCC=C)nn2)=O)CC1 c1(OCCC(=O)NCC(CCCC)NC(=O)CSC(C)C)ccc(C)cc1C C(=O)(C1=NOC(C)(C)C1)NC1(CC=C)CCN(C(C2(F)CCC2)=O)C1 C#CCCCC(C)C(=O)N1CC(C(C)(C)O)(CNC(c2cn3ccsc3n2)=O)C1 C1(C(=O)N(CCNC(=O)CCCC2CCOCC2)C2CC2)(OC)CCC(C)C1 C(N=c1nc[nH]cc1C#N)C1OCCN(C(CC2C(OCC)COCC2)=O)C1 N1(C(c2c(C)c[nH]n2)=O)CCCC2C(NC(C3COCCN3C=O)=O)C(C)(C)C12 C=CCCC(C)C(C(=O)NC1CCCC1)N1CCC(C(=O)OC)CC1(C)C N1(C(C=C(CCC)C)=O)CC(C(=O)N(C(C)C(C)SC)C)CC(C)C1 C(=O)(CC(C)(C)C1CC1)NCC(CCOC)NC(c1ncn(C)c1C)=O N1(C(=O)OCCC)CCN(C(=O)NC2CC(C)(C)OC2=O)C(C2CC2)C1 Oc1cc(-c2nc(-c3ccc(Oc4ccccc4)nc3)nn2C2CC2)cnn1 C=Cn1nccc1C(=O)NC(CNC(C1(c2cccnc2)CC1)=O)CC N1(C(CC(C)N(C)C)=O)CCC(NC(c2cscc2C(N)=O)=O)CC1 n1(C(C)C)ncc(C(=O)NCCC2(NC(=O)CC3CCOC3C)CCC2)n1 CC#CCC(C(=O)NC1CC(=O)N(O)C1)NC(=O)COc1cc(C)on1 C(=O)(C(C)(C)S(C)(=O)=O)NC(CN(C(C=CC=CC)=O)C)C CCCCC(CC)CC(=O)N1C2CCCC1CN(C(=O)C=C(C)c1cccs1)C2 Cc1nc2sc(C(=O)Nc3ccc4nnc(C(C)C)n4c3)cn2c1Br C1(C(=O)NCC2C(C)CN(C(=O)C=CCF)C2)CC2(C1)CC(O)C2 CC(C(=O)NCCCC1(NC(C2SCCS2)=O)CC1)C(C)c1ccc(F)cc1 C(=O)(C(F)(F)C(F)(F)F)N(CCCNC(=O)Cn1ccc([N+](=O)[O-])n1)CC C1(C(N(C)CCNC(=O)Cc2cocn2)=O)CCCCC1F N1(CC)CC(C(=O)N(CC(C)NC(c2cc(F)ccc2Cl)=O)CC)CCC1=O c1(NC(=O)CC2CCN(C(=O)C(O)Cc3ccc(O)cc3)C2)cnc(Br)c(Br)n1 C(CCCC(=O)NCC1CCCN1C(=O)Cc1n[nH]c(=N)s1)SC Cc1cc(CCC(=O)NCC2COC(CNC(=O)C(=Cc3c[nH]cn3)F)C2)on1 c1(OC)cc(C(=O)NCC2CN(C(=O)C(C)SC)CC2(F)F)nc(C)c1 Cc1cc(C)n(CCNC(=O)C=Cc2cn[nH]c2)n1 C1(C(N(C)CC2(C(=O)NCC3(F)CCC3)CC2)=O)CCCCC1(C)C Cc1ccc2[nH]c(C(=O)N(CCN3CCCC3)C(c3ccccc3Cl)=O)cc2c1 N1(C(C(CC)N(CC)CC)=O)CCC(F)(F)C(CNC(=O)C=CC(C)C)C1 c1(NC(COC2CC(NC(C3CC(SC)C3)=O)C2)=O)cc2ccccc2nn1 O=CN1CCCC1C(N1CCCC1CCNC(=O)C(F)(F)c1ccncc1)=O N1(C(C2(O)CCN(S(=O)(=O)CC3CCC3)CC2)=O)CCC(C2(O)CC2)CC1 N1(C(c2ccc(S(=O)(=O)NCCCOC)cc2)=O)CCC2C(=O)NC(=O)C2C1 C1(N(C(c2scc(OC)c2)=O)C)CCN(C(C2(O)CC(C)(C)C2)=O)CC1C C(CCC(C)C(=O)N1CCC(N(C)C(c2cc(OC)ns2)=O)CC1)OC N1(C(C(CC)(C)C(F)F)=O)CC2(C1)CN(C(c1c[nH]c(=NC)o1)=O)CCO2 C1(CN(C(Cc2cnc(C)o2)=O)C)CCCN(C(C2(C(C)C)CCC2)=O)C1 c1(N2CCCC(C(=O)NCC(C3CCCO3)O)C2)ncnc2ccccc12 Cc1oc(SC(F)F)cc1C(=O)NC1CCCC(CNC(C2(O)CCOCC2)=O)C1 C1(C(=O)NCC(C)(C)CCNC(=O)CNS(C)(=O)=O)Cc2nccn2C1 CC(C)CC(O)C(=O)NCc1ccccc1CN(C(=O)CCc1cnn(C)n1)C C1(CC)CN(C(c2cc(CNC(=O)CC(C)OC)ccn2)=O)CCS1 N1(C2CCN(C(C=CCN(CC)CC)=O)C2)CCN(C(=O)C#CC2CC2)CC1 C(=O)(C(CNC(=O)CSC1CC1)CC1CCCC1)NCC(CC)(C)OC n1(CCOC)ncc(C(N2CCCC2CNC(c2ncccc2SC)=O)=O)c1C c1(C(=O)NC(C2CCCN2C(c2cnn3c2CCC3)=O)C)cc(=O)cc(Cl)[nH]1 C1(C)(NC(C2(COC)CN(C(=O)C(Cl)Cl)C2)=O)CN2CCC1CC2 c1(OC)cc(OC)nc(N2CC3C(CNC(c4conc4C)=O)C3C2)n1 c1(C(N(CC(C)N(C(=O)COc2ccsn2)C)C)=O)ccc2c(c1)N(C)C(=O)C2 N1(C(C(C=C)CC)=O)CC2CC(NC(=O)CC(C)F)CC(C2)C1 C1(CCCCNC(CNC(CC)=O)=O)CCCN(C(=O)CC2(CO)CCCC2)C1 C1(C(N2CCC(C)N(C(=O)CN3CC4CC4C3)CC2)=O)CCCN(S(N)(=O)=O)C1 CCC(C)(C)C(=O)C(=O)N1CC(NC(=O)C(C)Cn2ccnc2)CC1C c1(NC(CCN(C(c2ccc(CC)[nH]2)=O)C)C(C)C)ncnc(Cl)c1[N+](=O)[O-] C(c1ccc(Cl)cc1)=C(C(N1CC(OCCNC(C2C(OCC)C2C)=O)C1)=O)C C(=O)(C(F)(F)CO)NCC1(CCNC(Cn2cc(C(N)=O)nc2)=O)CC1 C(C(C(C)C)NC(C1CCCN1c1ccncn1)=O)NC(C=C(C)C)=O CC1(C)CN(C(=O)C(c2ccccc2)F)CC1C(=O)NCC1(CO)CC=CC1 N1(C(CN(C(=O)CC#N)CCC)=O)CCC(NC(C)=O)C1 CCCC(CCC)CC(=O)NC(C(=O)NCC(CC)(CC)CC)C1CC1 c1(C(N(C)CC2(CNC(=O)C(C)(C)c3cc[nH]n3)CC2)=O)nnc(S)n1C Cc1c(C(=O)NC2CCC(NC(=O)C(F)(F)C3CC3)C2)ccc2c1CCC2 c1(CC)ccc(C(=O)NC2(C(N3CCC(C)(O)C3)=O)CC2(C)C)cc1 c1(CN(C)C)ccc(C(=O)NC(C)(C)CN(C)C(C2C3CCCC23)=O)cn1 CC1CCC(C(=O)NCC23CCCC2CCC3)CN1C(=O)C(F)C(F)(F)F C1(CNC(C2CCC2)=O)CCCN1C(c1cnn(CC(F)(F)F)n1)=O N1(C(C(C)(C)CC#N)=O)CCC2CC(NC(c3cccc(F)c3F)=O)CCC2C1 c1(C(=O)NC2CCCN(C(CC3C(C)CCCC3)=O)C2)nc2cccnc2s1 N1(C(C(C2CCC2)OCC)=O)CCC2CN(C(c3cn(C)cc3C)=O)CC2C1 c1(C(=O)NC2CN(C(CC(C)(C)C)=O)C2)cc(S(N)(=O)=O)c[nH]1 C1(C(N2CCC(C)(C(N)=O)C2)=O)CCCCCN1C(=O)CCCn1ccnc1 N1(C(C(N2CC3C(CN(C)C(=O)OC(C)(C)C)C3C2)=O)=O)CCC2C(C1)C2(F)F n1(C(C)C)cc(C(=O)O)c(C(F)F)c1.N12CCC(F)(C1)C2=O.N12CC(C1)C2=O CC1(NC(c2cocn2)=O)CCCN(C(c2ccnc(OC3CC3)c2)=O)C1 c1(C(=O)NC(CCCC)CNC(c2csc(C(N)=O)n2)=O)sc2nccn2c1C C(=O)(CCS(C)(=O)=O)N1C(C)(C(=O)NCCC2COCC2O)CCC1 N1(C(CC2(CC)CN(C3(c4ccnc(Cl)c4)CC3)C2)=O)CC2(CNC(=O)OC2)C1 C(C(=O)N(C)O)NC(C(C1CCN(C(=O)C(n2ccnc2C)C)C1)C)=O N1(C(CC(CC2CC2)NC(CCCC(=O)OC)=O)=O)CCc2c(C)cccc21 c1(C(=O)NCC(CN(C)C(c2cnn(C)n2)=O)O)cc(F)ccc1Br c1(C(N2CCC(NC(C3CC(OCC)C3)=O)(CF)C2)=O)cc2c(Cl)ccnc2s1 N1(C(COCC(=C)C)=O)CC(C)CN(C(c2cc3ccccc3s2)=O)C(C)C1 N1(C(C(=O)NC2(CC=C)CN(C(=O)C(C)C3CCC3)C2)C)CCC(O)CC1 C1(=O)NNc2ccc(c(Br)c2)CN1.CC1(C)C(Cc2ccccc2)C1(C)C Cc1nc(O)[nH]c1C(=O)N(C)CCOCCNC(c1csc(-c2cn[nH]c2)c1)=O C(=O)(CC(F)(F)C(F)(F)F)NCCC12CN(C(CNC(N)=O)=O)C(CC1)C2 N1(C(c2nc(C)n(C)c2)=O)CC(NC(c2cnc3[nH]cncc2-3)=O)C(N=[N+]=[N-])C1 C1(CC#C)CN(C(=O)CCCNC(=O)CN2CCN(C)CC2)CCO1 n1(CC(=O)NCCN2CCN(C3CCN(CC)C3=O)CC2)ccc2ccccc12 C1(CC#C)CN(C(=O)C(C)CNC(=O)CCc2ccn(C)n2)CCO1 C(CC(C)(C)C(=O)NCC1(CF)CCC1)NC(c1ncc(NC)nc1)=O C1(C(N2CC(O)(C(CNC(C(C)N3CCC3)=O)(C)C)C2)=O)CC2C=CC1O2 CC1(C)CC(C(=O)NOCC(F)F)(CNC(C2CC2Cl)=O)C1 C1(C(=O)NC2C(C(C)C)N(C(c3cc(Cl)cc(Cl)c3)=O)CC2)CC2C(C1)C2(F)F N1(C(c2ccc(C#N)nc2O)=O)CCCC12CCN(C(=O)CCc1cccs1)C2 C1(CNC(CNC(=O)NC)=O)COC(C)(C)CN1C(=O)C(O)CC1CC1 C1(CCNC(Cc2c(Cl)cn(C)n2)=O)C2CC3CC(C2)CC1C3 c1(C(=O)NCC(CN(C(C2C(OC)CCC2)=O)C)C)ccc2cnccc2c1 Cc1nnc(O)c(C(N2CCC(C(F)CNC(=O)CCF)CC2)=O)c1C c1(OC)ccc([N+](=O)[O-])c(CN2CCC(O)C(C(=O)NCC(F)CO)C2)c1 C(=O)(CCCCNC(C1(N(C)C(c2cc(OC)ns2)=O)CCCC1)=O)NCC N1(C(CNC(C)=O)=O)CCN(C(c2cn(CCO)nc2C)=O)CC2(CC2)C1 C1(C(=O)NC2CCCN(C(C=CC=CC)=O)C2CC)CC=C(C(C)C)CC1 C1(CC)CN(C(c2nc(O)c(C)s2)=O)CCC1NC(=O)C(F)OC(F)(F)F C1(NC(C(=CC2CCCC2)C)=O)CCCC(NC(c2c[nH]c(=N)o2)=O)C1 C1(C(N2CC3C(CNC(C=CC(=O)N(C)C)=O)C3C2)=O)CNC(=O)CC1(C)C N1(C(c2n[nH]c(CC)c2Cl)=O)CCCC(C)(CNC(=O)CN2CCC(C)C2)C1 CCCC(C)C(C)c1noc(C2CCCC2)n1.C(=O)(CCC(N)=O)N C(=O)(CCCCCCCCCO)N1CC(C(C)NC(CC)=O)OCC1 C(CC(F)F)(C(=O)NCCC1NC(=O)NC1=O)N(C)C(c1cc(C2CC2)on1)=O C1(F)(C(=O)NCCC2(C)OCCO2)CCN(C(c2ccccc2I)=O)C1 c1(N(C(CC)=O)C(c2ccc(O)cc2)=O)cc(F)ccc1-c1cccc(OC)c1 C1(C(=O)Nc2c(C#N)nc(C)o2)CC2CCC1N(C(C1C3C=CSC13)=O)C2 S(=O)(=O)(c1ccc(C(N2CC(NC(=O)CNS(N)(=O)=O)C2)=O)cc1)NCC(C)C C=C(C)CCCC(=O)N1CCCC(C(N2CCC2CC(=O)NC)=O)C1CC N1(C(c2[nH]cc(C)c2)=O)CCOCC1CC(=O)NOCCc1ccccc1 C1(NC(c2cn(C)nc2)=O)CCN(C(C2CCC2c2ccc(F)cc2)=O)CC1 N1(C(C(C)SC)=O)CCCC(CCNC(c2ncsc2C2CC2)=O)C1 CCCC(C#N)C(=O)N1CCC(CNC(c2ccon2)=O)CC1C Cc1noc(N)c1C(N1CC(=C(F)CNC(=O)COCC2CCCO2)C1)=O N1(C(CCCCC(=O)OC)=O)CCN(C(=O)C2=NOC(C)C2C)C2COCC12 C(=O)(C1=CCN(C(=O)C=CC2CCCC2)CC1)N(C(CO)CO)CC C1(CC(C)C)C(=O)N1.C1(C)(NCC=C(C)C)CCN(C(=O)CNS(N)(=O)=O)C1 C1(NC(c2n(CC)nnc2)=O)CN(C(=O)CSCc2cscn2)CC1C1CC1 C1(c2cccc(Cl)c2)(Cn2cc(CCC(CC)O)nn2)CCOCC1 C1(NC(C=CCCC)=O)CCCN(C(=O)C(C2(OC)CCCCC2)(F)F)CCC1 C1(NC(Cc2cn(C)nc2)=O)CCCCN(C(c2cnc(Cl)c(N)c2)=O)CC1 c1(OC)ccc(S(=O)(=O)NC2CC2C(=O)Nc2ccn3cnnc3c2)cn1 C1(C(=O)NCC)CC12CCN(C(c1cncc(OC(C)C)c1)=O)C2 c1(CC)nc(C)c(C(N2CC(O)CC2C(=O)N(C)CCc2ncccn2)=O)o1 C1(NC(CCC#C)=O)CCCCC1NC(c1c(C)nsc1NC1CC1)=O N1(C(C2ON=C(C)C2)=O)CCC(C)CC1Cc1ccccc1.c1(=O)c(=O)n1CCCCO C1(C(=O)OC)CCN(Cc2cn(CCN(C)C(c3ccsc3C)=O)nn2)CC1 C=C(C(=O)N(C1CCNCC12CC2)CCNc1ccccc1OC)C(F)(F)F N1(C(CC(CC)C2CC2)=O)CC(CNC(C2CCCC2)=O)C(C)(C)C1 Cc1cccc(C(N2CCOCC2)C(=O)NCc2ccccc2OCC(=O)O)c1 CCC(C)(COC)C(=O)N(C)CCNC(=O)Cc1ccc(Sc2ccccc2)cc1 N1(C(C2(C=C)CCC2)=O)CC(CNC(=O)C(C(C)(C)C)NC(N)=O)CC(C)(C)C1 N1(C(Cn2ncc(C)c2)=O)CCc2ccccc2C1CNC(C12CC(CO1)C2)=O c1(OC)ncc(C(=O)NC2CCCC2NC(=O)C(C)NC(N)=O)nc1C C(CCN(C(=O)CSc1nc[nH]n1)C)(C(C)(C)C)NC(CC(CC)OC)=O C12(NC(c3cc(OCC)n[nH]3)=O)CCC(CNC(=O)Cc3nc[nH]n3)(CC1)OC2 CC1CCC(=CC(=O)NCC2(C(=O)NCC3CCOCC3)CC=CC2)CC1 C(=O)(CC=C(Cl)Cl)NC(C(=O)NCc1c(CC)nn[nH]1)Cn1cncn1 N1(C(C(C)(C)NC(=O)OC)=O)CCCC2(C1)CN(C(C1CC1C1CC1)=O)CCO2 C1(C(=O)NCC2(F)CCN(C(C(N(C)C)C3CC3)=O)CC2)CCCC12OCCO2 N1(C(c2cccc(CC)n2)=O)CC(C(N2CCOCC2CC(N)=O)=O)C(F)(F)C1 CCCC(CC)CCC(=O)NC1CC(NC(=O)C(C)NC(C)(C)C)C1 C1(C(=O)NCCCCCNC(C2(SC)CC(O)C2)=O)C(Cl)(Cl)C12CC2 N1(C(CCc2c(C)nn(C)c2)=O)CCC(NC(=O)CC2C=CS(=O)(=O)C2)C1(C)C c12ccccc1[nH]c(=O)c(=O)[nH]2.NC1CCCC1C(=O)N(c1ccccc1)C C1(CCC(=O)N(CC(C)O)CCNC(CC2CN(C(C)=O)C2)=O)CCCC(=O)N1 c1(C(=O)NC2C=CC(C)(C)CC2)ccccc1S(=O)(=O)C(F)F CC#CCCC(=O)NC1(C)CCN(C(c2c(C)nsc2NC(=O)OC)=O)C1 N1(C(c2ncn(C)c2)=O)CCC2CCN(c3ccnc(-c4nccs4)n3)CC2C1 CC1(CNC(=O)Nc2ncc(C(F)(F)F)cc2I)CCCC(=O)N1 c1(CC(=O)NCC2ON=C(C)C2)noc(C)c1C#N C(CCCCCCCCCCO)N(C(=O)C(N1CCC1(C)CCN)=O)C c1(-c2c(C)c(F)ccc2)cc(C(=O)Nc2ccc(OC)nc2)cc2cc[nH]c12 C1(CC=C)(OC)CN(C(c2nnn(C)c2)=O)CCO1.C(=O)O N1(C(c2ccc(Cl)s2)=O)CCOC2(CCN(c3nccn4nnnc34)CC2)C1 N1(C(CSCCN(CC)CC)=O)CCCC(NC(C2(C)OCCO2)=O)C1 C(c1ccccc1OC)=CC(=O)NC1(CC=C)CCN(C(=O)C(C)(C)CCC)C1 c1(C(=O)NCC(CN(C(=O)CCN2CCNC(=O)C2)C)O)cccc2nn[nH]c12 C1(NC(C(C)=C(C)C)=O)CCCC(NC(=O)C(F)C(C)C)C1 CCCCC(O)C(C)C(=O)NC1CCCCN(C(=O)CSc2cn[nH]c2)C1 CC(C)(C(=O)NC1COCC1NC(C1(c2cccs2)CCCC1)=O)n1ccnn1 Cc1cc(C(N2CCCC2C2CCN(C(C3(C(C)(F)F)CCC3)=O)C2)=O)no1 c1(NCC(C)NC(=O)CNC(C2CC(F)C2)=O)cccc(NCC(F)(F)F)c1 CCC(C)C(O)CC(=O)NCCC(C(N1CCCC(F)CC1)=O)OC N1(C(C(=O)NCCOC)=O)CC(NC(=O)COCC2CCCCO2)CCC1C N1(C(C2CC(OC)C2)=O)CC(C)(C)C(NC(C2C=CCCC2)=O)C(C)(C)C1 N1(C(C=C(CC)C)=O)CCC(COC)(NC(=O)CN(c2ccncc2)C)C1 C1(C(=O)NC2CCC2NC(C2CC(CCO)C2)=O)(CC)CCCC1O c1(C(=O)NC(CN(C(=O)CCCc2cccs2)CC)C)c(C)noc1C1CC1 C12(CNC(c3[nH]ccc(=N)n3)=O)CCCCC1CN(C(=O)C=Cc1ccco1)C2 c1(C(=O)NC(C(C)C)CNC(=O)Cn2cc(Cl)cn2)ccc(Cl)c(C#N)n1 N1(CC)C(=O)COC(C(=O)NC2CC2CNC(=O)C=CBr)C1c1nccn1C Cc1nc(C(N2CCC3(CC3C(=O)NCCCSCCO)C2)=O)ccc1C#N Cc1cc(C(=O)NC2CCN(C(=O)C=Cc3cn(C)nn3)C(C)C2)cnc1O CC1CN(C(=O)C(Br)Br)CC1c1cn(Cc2ccc(F)cc2)nn1 c1(CCC)nc(C)c(C(=O)NC(CNC(C2CC(=O)N(C)C2)=O)CO)o1 c1(N(CC(F)(F)Cl)C)nc(N2CCC3(C)C(F)(F)C3(C)C2)c2ncccc2n1 O=C(C1CCc2snnc21)N1CC2CC1C2NC(c1ccc2c(c1)CCO2)=O N1(C(C(c2ccc(C)o2)C)=O)CCCCC1CCN(C(=O)CCCN(C)C)C N1(C(C(C)CS(C)(=O)=O)=O)CCC(C2(NC(C3(C)CC3Br)=O)CC2)CC1 C(=O)(C(CO)C(F)(F)F)NC(C(=O)N(C)Cc1ncccn1)C(C)(C)C N1(C(c2cc(C)c(C)[nH]2)=O)CC23CCCC2(C1)CN(C(=O)C(CO)C(C)C)C3 C1(C(=O)NC(c2ccc(OC(C)C)cc2)CC#N)CCCCC(C)(C)C1 Cc1cc(C(N2CC(NC(C3CC4(CC4)C3)=O)C(n3cccn3)C2)=O)ccc1F CC1CC(=O)Nc2cccc(C(N3CCC4(CCCCCC4)C3)=O)c2N1 n1(CC)cc(C(=O)NCCCN(C)C(c2ccsc2C#N)=O)c(C2CC2)n1 Cc1ncc(Cl)cc1CC(=O)NC(CNC(=O)CC(C)N(C)C)CC(C)C N#Cc1cc(C(N2CC3(CNC(=O)CCF)CC2CCO3)=O)cc(O)c1 CCC(C(=O)NCC1CCC1NC(=O)CCN(C)C(C)=O)n1cncn1 C1(NC(c2csc(Cl)c2)=O)(CO)CCN(C(=O)CCOc2ccc(F)cc2)CC1 c1(OC)cc(F)ccc1N1CCN(CCN2CC3CCC2C3)CC1 c1(C(N(C2CCC(NC(=O)CCOCCOC)CC2)C)=O)cccn2cnnc12 N1(C(c2c(CC)cccc2)=O)CCN(C(=O)C(CC)OC)CC1C C1(CCC(N)=O)CCCCN1N1CCOC(c2ccc(F)c(Cl)c2)C1 N1(C(C(C)NC=O)=O)CCN(C(=O)CCn2cncn2)CC1Cc1ccccc1 C1(C(N2CC(C)(C)C(CNC(C3COC3)=O)C2)=O)CC2CCCC(C1)C2 C1(N(C(c2n(CC)cnn2)=O)C)CCN(C(c2cnc(Cl)s2)=O)CC1 c1(CC)ccccc1OCCC(=O)N(C)CC1CCCN(C(=O)C(C)(C)CF)C1 c1(OC)ccc(NC(=O)CCCCCN(C(=O)C(C)OC)C)c(C)c1 c1(C(=O)NCC(CC)NC(=O)C(O)CN(C)C)cccc(N)c1C Cc1cc(OCc2ccccc2Cl)c(NC(=O)Cc2ccc(OC)cc2)cc1F C1(C(=O)NC(C(C)C)CNC(=O)C(C)n2ccnc2)CCS(=O)(=O)C(C)C1 c1(OC)ccc(F)c2[nH]c(C(=O)NC3CC3NC(C3(C#N)CC4CC4C3)=O)cc12 N1(C(C2N(C)CCC2)=O)CC2(CC(NC(C3(c4cccnc4)CCC3)=O)CO2)C1 c1(C(N2C(CNC(C3ON=C(C)C3)=O)CC(O)C2)=O)cnn2c(C)ccnc12 C1(OC)(CNC(=O)CC2COCCN2C)CCN(C(c2cnncc2C)=O)CC1 c1(C(N2CC(NC(C3(C)CCCCO3)=O)C(O)C2)=O)cn2c(n1)CCCC2 C1(C(N(CCC)CCN(C)C)=O)CCC2CCC1N2C(=O)C=CC(F)(F)F n1(CCOC)cc(C)c(CN2CCOCC2c2nc(C(C)(C)C)n[nH]2)n1 N1(C(=O)CC2CC3(CCC3)C2)CC2=C(C1)CN(C(c1snnc1C1CC1)=O)C2 c1(CC(=O)OC)ccc(NC2CN(c3ccnc(COC(C)(C)C)n3)C2)cc1 N1(C(CC2C(C)(C)C2)=O)CCN(C(=O)CSCC(N2CCCC2)=O)CC(O)C1 CC(C)(C#N)C(=O)NCC(O)CC(=O)NCc1cccc(Cl)n1 CCCC(F)C(=O)NCC(C)(CNC(=O)C(C)=C1CCC1)OC N1(C(c2cc(C)cc(Cl)n2)=O)CCC2(CCCCN(C(=O)Cn3cnnc3)C2)C1 C#CCCN=C(NCc1ccc(OC)nc1C)NCc1ccccc1CSC Cc1ccc(F)cc1C(=O)NC(C)C(C(C)C)NC(C1(c2ccnn2C)CC1)=O N1(C(C(C2(OC)CC2)OCC)=O)CCC(O)C(NC(=O)C(C)(C)C2CCOC2)C1 N1(CCN(C(C(C)N(C(COCCC=C)=O)CCC)=O)OCC)CCCC1C CC1(C)CC(CNC(=O)CCc2cccc(Cl)c2)CN1C(=O)Cn1nnc(=O)[nH]1 CC1OC2(CNC(=O)C(C)C3CCOC3)CC1(NC(c1cnc(Br)s1)=O)C2 c1(-c2nc(CCC(CCC)NC(c3ccccc3)=O)on2)nc(C)c(C)[nH]c1=O c1(C(=O)OC)cccc(C)c1S(=O)(=O)NC1CC1C(N1CC2CCC(C1)O2)=O Cc1ccc(C(=O)NCCC2(C)CCN(C(C3CC4(CCO3)CC4)=O)C2)c(C)c1 O=C(CCCCNC(C1C2CCCOC12)=O)NCc1cccc(CO)n1 C1(CNC(c2nc(CCC)sc2)=O)CN(C(c2sncc2C)=O)CC1C C12(C(=O)NC3(C)CCOCC3)CC(CN(C(=O)CC=Cc3ccccc3)C1)C2 C(=O)(CCCCCF)NCCNC(C1CCCN(C(C(CCC)C)=O)C1)=O C1(COC)(NC(=O)CC(C)SC)CCCN(C(c2cnc(C3CCC3)s2)=O)C1 C(=O)(C1=CC(O)C(NC(=O)C#CC2(CC)COC2)C1)N1C(C=C)CC1 c1(-c2c(C(=O)NCC3(CCNC(C(C)=CC)=O)CC3)c[nH]c2)ccc(F)cc1 c1(C(CC(=O)NCCCCCN(C(=O)C#CC2CC2)C)O)cccc(F)c1.C(=O)CN C1(C(N(CC(C)CNC(=O)C(C)C2CCCC2)C)=O)CN(CP(C)(C)=O)C1 C1(C)(C(=O)NCC(CNC(C2(SC)CCC2)=O)C)CCCOC1 CCC(C)CC(=O)N1CC(O)CC1Cc1cn(CC2CC(F)(F)CO2)nn1 CCC(CC)C(C(=O)N(CCNC(C1CCCSC1)=O)C(C)C)OC c1(NC(C=C)CSC)ncccc1S(=O)(=O)NCCS(N)(=O)=O C(N=c1nc(CS(C)(=O)=O)[nH]s1)C1CCCN(C(C)=O)C1 Cc1cc(Cl)c(C(=O)NCCCOCCN(C(=O)CC2OCCC2C)C)s1 c1(N(C(CCNC(c2occ(C)n2)C)=O)C)ccccc1Br CCC(C)(C)CCCC(=O)NCC1CCCN1C(C1C2Cc3ccccc3C12)=O C1(C(=O)NC(C)Cn2ccnc2)CNC(=O)CN1C(=O)CN1CCSCC1 C=CCCCCCC(=O)N1CC(CNC(=O)CC2CCN(C)CC2)CC1(C)C N1(C(C(COC)(C)C)=O)CCC(NC(c2ccc(S(C)(=O)=O)s2)=O)C(CO)CC1 C1(C(N(CC(C)NC(C2(CF)CC2)=O)C)=O)CC2(CCCC2)CO1 c1(C(=O)NCC(CNC(Cn2c(=N)nc[nH]2)=O)F)ccc(F)c2[nH]ccc12 C(=O)(C#CC1CCOC1)NC1CN(C(C(c2cccc(C)c2)(C)C)=O)CC12CC2 CC(C)CCC(C(=O)NC1CNC(=O)C12CC2)NC(=O)CCC1CCCC1 Cc1cn2cccc(C(N3CC(F)CC3CNC(C3CC3C3CC3)=O)=O)c2n1 C#CC1C(C(=O)NCCN(C(=O)CC2CCN(C(C)=O)CC2)C)C1(C)C c1(C(N2CCN(C(C(CSC)O)=O)CC2)=O)cnc(N2CCCCC2)c(Cl)c1 CC1(C)CC(C(=O)NC2(C)CCOC2=O)N(C(C2CCC2(F)F)=O)C1 C1(C)(N(C(=O)C(N)Cc2cccnn2)C)CC2(CCC2)C1 CC1CN(C(C2CCC23CCC3)=O)CCCN1C(c1c(O)cccc1F)=O C1(NC(COCCCC(C)C)=O)CCN(C(=O)Cc2ccnn2C)C(C2CC2)C1 c1(CC(N2CCCC(N(C(Cc3c(C)nsc3)=O)C)C2)=O)cnn2c1CCCC2 C12(NC(c3nc(COC)sc3)=O)CCCC1CN(C(c1nnn3c1CCC3)=O)C2 CON1CCC(C(=O)N(C(C)CN(C)C(c2c[nH]c(=N)nc2C)=O)C)CC1 C(c1cncc(O)c1)=CC(=O)NCC(C)N(C)C(C1CC12CC(F)(F)C2)=O Cn1c(COCC(=O)NCc2ccccc2CNC(C2(F)CC2)=O)nnc1S c1(C(=O)NC2(COC)CCN(C(=O)C3=NNC(=O)C3)C2)csc2cccnc12 c1(CNC(C2N(C(c3c(C)scn3)=O)CCOC2)=O)ccc(Br)c(F)c1 C1(C)(CNC(CC(C)SC)=O)CCCC1NC(c1ccc(CCN(C)C)cc1)=O c1(C(N2C3CN(C(C(F)=C(C)C)=O)C(C3)C2)=O)cc(C(F)(F)F)ccc1Cl c1(C(N2CCN(C(COCCC)=O)C(C)CC2)=O)cccc2c1C(C#N)C2 C(=O)(C(CNC(=O)C=Cc1nccs1)C(C)(C)C)NCC(C(CC)C)C c1(CC)nc(C(=O)NCCCN(C(=O)CC2CCC(C(F)(F)F)O2)CC)cs1 c1(C(=O)NCCNC(C2CCCN3CCCCC23)=O)cn2ccc(CO)cc2n1 Cc1nc(C(F)(F)F)c(C(=O)NCC(C(C)(C)C)NC(c2scc(C)c2C)=O)o1 C(C)(C)(C(=O)NCC)OC1(CN(C)C(C2CC(O)(Cc3ccccc3)C2)=O)CC1 C1(NC(c2c(C)nccc2)=O)CCOC2(CCN(C(=O)CNC(C)(C)C)CC2)C1 c1(C(=O)NCC2(CCNC(CN(C)C(N)=O)=O)CC2)cccn(O)c1=O C1(C(=O)NC2(C)CN(C(C(C(C)(C)C)NC(C)=O)=O)C2)CCn2c(O)nnc2C1 c1(CN)cc(CC(=O)NCC2(c3ccccc3)COCCO2)ccn1 N1(C(=O)C(F)(F)C2(O)CCCC2)CCN(c2ccccn2)C(=O)C1 c1(C(N(CC(C)NC(CS(=O)(=O)NC)=O)C)=O)cnc2nccn2c1 Cc1cccc2c1CCN(c1ccc(S(=O)(=O)NCC(C)CCO)cc1F)C2 N1(C(C2N(C(c3cc(C)nn3C)=O)CCSC2)=O)CCOCC(C)(F)C1 C(=O)(C1=CCC(C)CC1)NC(CCCNC(c1c(CC)cccn1)=O)CO c1(CC)ccc(-c2ccc(C(=O)N(C(C)CC)CC3(C)CC(F)(F)C3)o2)cc1 c1(C(=O)NCC=CCNC(C(CC)(C)F)=O)cc2n(n1)CC(C)NC2=O C1(CCNC(CN(C(=O)Cc2cncc(F)c2)CCOC)=O)CCN(C)C1=O c1(C(=O)NCC2N(C(c3c(OC)nn(C)c3)=O)CCCC2)cccc2c[nH]nc12 c1(CC)cccc(C(N2CCC(NC(c3ccc(Br)o3)=O)CC2)=O)c1O c1(SC)cncc(Oc2ccccc2NC(=O)Nc2ccc(C(=O)OC)cn2)c1 Cc1cnc(N2CCC(C)S(=O)CC2)c(S(=O)(=O)NCCc2cnco2)c1 c1(C(=O)NC2CCC=CCCC2)sc2ccccc2c1Cc1nc[nH]n1 c1(OC(=O)NCC)cccc(-c2nc(C(CC)NC(C)(C)C)n(C(C)C(C)C)n2)c1 C=CCCCCC(=O)NCC1C(C)CCN1C(=O)C(c1cccc(C)n1)(F)F Cc1cc(NC(C2C3CC2N(C(=O)Cc2cccc(Cl)n2)C3)=O)cnc1Cl C1(CC(=O)NC)SC(=Nc2ccc(C)cc2)N(CC(CO)C(C)C)C1=O c1(OC)cc(C(N2CC3CC3(CNCc3ccc(C(=O)O)s3)C2)=O)ccc1Br c1(C(N2CCOCC(NC(C(C)(C)SC)=O)C2)=O)cc2c(F)cccc2s1 CCCCCS(=O)(=O)CC(=O)NCCC1CC(NC(=O)Cc2cn[nH]c2)C1 C(CC(C)(C)CC(=O)N1CCC(C)(NC(=O)Cc2c[nH]nc2O)CC1)OC C(=O)(C1=C(Cl)CCC1)NC1C(NC(CNC(c2c(OCC)cccc2)=O)=O)C1 Cc1cncc(C=CC(=O)NC2CCC2NC(c2cccc(C(F)(F)F)n2)=O)c1 C#CC1CCN(C(=O)Nc2cnn(CC(C)(C)O)c2C)C1 C(=O)(CCC(=O)N(C)C)NC(C)CCNC(C1CC(CF)C1)=O c1(C(N2CCOC(C(N3CCN(CCF)CC3)=O)C2)=O)ccc(F)c(C(F)(F)F)c1 N1(C(C=Cc2cnc(OC)nc2)=O)CCN(C(c2cc(O)no2)=O)CC1C#N C1(c2nnnn2C(C)(C)C)(NCCCC(C)(C)C)CCCCCCCCCCC1 N1(C(CC2C(C)CCO2)=O)CCC(NC(=O)C(F)(F)c2ccccc2)CC1C c1(C(=O)NC2CC(CC(=O)NC(C)CN(C)C)C2)c(OC(F)F)cccc1F N1(C(COCCC)=O)CCC(C(F)C(=O)NCCCc2ccccn2)C1 C1(C(C)NC2CCSCC2)(CNC(=O)OC(C)(C)C)CCC(C)(C)CC1 N1(C(c2ccc(OCC(C)C)cc2)C(=O)NC(C(=O)OC)C)CCOCC1CF Cc1ccc(NC(=O)C(N2CC(NC(=O)C(C#N)C3CC3)C(C)C2)=O)cc1C C1(OC)CCC2(C(N3CCCC(C(=O)Nc4nc(C)cs4)C3)=O)CCC12 c1(OCCS(C)(=O)=O)cccc(NCC2(O)CCCSC2)c1 c1(C(N2CCCC(C(C)NC(c3c(C)nc(C)s3)=O)C2)=O)ccn2cncc2c1 c1(C(=O)NCC(C)NC(CC2CC(C(C)C)OCC2)=O)cncc2ccccc12 N1(C(C)C)CCCCC1C(=O)N(C)CC1CCCN1C(=O)CCC(C)O C1(CC=C)(NC(C2CCCC2C(C)C)=O)CCN(C(=O)CC=CC(C)(C)C)C1 C1(C(N2CCCCC(CNC(=O)CCOC3CC3)C2)=O)CC2(C1)CS(=O)(=O)C2 c1(C2(C(C3C(n4cc(C(C)(C)CO)nn4)CCCC3)=O)CC2)ccc(F)cc1Cl c1(C(N2CCC(CNC(c3scc(OC)c3)=O)C2)=O)sc(F)cc1Cl C=C(C)C1OCCC1CNC(=O)CCC(CC)NC(C1(C#N)CC1)=O c1(C(C(=O)NC(C)(C)C)N(C2CCCCC2)C(C)C)sc(Cl)cc1Br N1(C(Cc2cn(C(C)C)nc2)=O)CCC(CNC(=O)C(F)(F)C(C)O)C12CC2 c1(C(c2nnnn2CCSC)NCCC2(OC)CCC2)cc2cc(Br)ccc2o1 CC(C)(F)CCC(=O)NC(C1CCCCC1)CNC(=O)CC=C(Cl)Cl c1(C(N(CCN(C(=O)CCC2OCCO2)C(C)C)C)=O)sccc1SC(F)F C12(NC(C(C3CCOC3)OC)=O)CCOC(CNC(c3cncnc3)=O)(C1)C2 c1(C(=O)NCC2(CNC(C(C)OCCOC)=O)CCC2)cccc(O)n1 C1(C(=O)NC2CC(CNC(C=C3CCN(C)C3)=O)C2)CCC2(CCCCC2)C1 O(P(C)(=O)CNC(=O)CCN(C(=O)C(CN(C)C)CC)CCCO)CC c1(C(=O)NCC2C(NC(c3cc(F)ccc3F)=O)CCC2)csc2c1CCCC2 c1(C(=O)NCC(CNC(CC(C)C)=O)(C)O)ccc(S(C)(=O)=O)c([N+](=O)[O-])c1 c1(CNC(c2c(I)cnn2C)c2n(CC)nnn2)csc(C)c1C N1(C(Cc2cc(C)sc2)=O)CCN(C(c2ncc(F)cc2C)=O)CC1CF c1(C(C)C)cccc(C(=O)NCCC2CC(NC(c3nc(=O)n(C)[nH]3)=O)C2)c1F C12(C(N3CCN(CCCNC(c4cc(C)sc4)=O)CC3)=O)CCC(F)C1CC2 N1(C(CCn2cnc(=N)[nH]2)=O)C(C(N2CC(OCCO)C2)=O)CCC12CC2 N1(C(CC(CNC(c2ccn(C(F)F)n2)=O)OC)=O)CCOC2COCC2C1 Cc1nc(N(CC(C)C#N)C)cc(NC2CCN(CC3CC3)CC2)n1 C1(CCCC)CN(C(c2ncc(Cl)cc2F)=O)CCN1C(=O)C(C)CC1CC1 C1(C(N(CCN(C)C(c2cccc(C3(C)CC3)c2)=O)C)=O)CC2CCC1C2 n1(CC(=O)NCC(C)(C2CC2)NC(c2cnc(C(C)O)s2)=O)ncn(C)c1=O C=C(C)CC(C)C(=O)NCC1(F)CCC(CNC(c2cnnc(C)c2)=O)CC1 N1(C(c2c(F)ccc(C)n2)=O)CC2CCN(C(=O)C=Cc3cncc(O)c3)C2C1 C(=O)(C(C(=O)NCC(C)N(C)C(C12CC(C)(CO1)C2)=O)C(C)C)OCC CC(C)CC(=O)C(=O)N1CCC(C(N2CCC3(CC(CO)C3)C2)=O)O1 CC1CCCN(C(=O)CCn2cnnn2)C1CNC(C1(C(F)(F)F)CCCC1)=O CC1(C)CCC(CO)N(C(C2(NC(C3CCSC3)=O)CCOCC2)=O)C1 c1(OC)cc(C(N2CCC3(CCC3)C2)=O)ncc1C1=COCCC1 C1(OC)CCN(C(c2conc2CNC(=O)CSCCOC)=O)CC1C C1(C(=O)OC)CN(CC(C2CCCCC2)O)C2(CCCCC2)C1 C1(C(N(C2(CC)CC2)C)=O)CN(C(c2scc(C)c2C)=O)C(C)(C)C1 c1(C=O)cnn2c1CCCC2.C1(C(C)NCC2CCCCO2)CCN(CCl)CC1 N1(c2ccnc(N3CC(C)(F)C3)n2)CCCC2CCCCC12 C12(NC(CC(C)(C)C3CC3)=O)CCCCCC1N(C(=O)C=Cc1cc[nH]c1)CC2 CCC(CCC(=O)N(CC(=O)NCc1cc(C)on1)CC1CC1)OC c1(C(=O)NCC(CNC(C(CC)NC(C)=O)=O)C)ccc(C)nn1 CCCC(CCCO)C(=O)NC1CCN(C(=O)C(n2cc(C)cn2)C)C(C)C1 C1(C(N(CCC(C)NC(=O)CCC(=O)N(C)C)C)=O)COc2ccccc2C1 C(=O)(CC(O)C(C)CC)N(CCNC(C(CC)C(C)C)=O)CCOC N1(C(c2c(OC)ccs2)=O)CCC2(CCN(C(=O)CNC(=O)C(F)(F)F)C2)C1 n1(CCNCC(CC(=O)N(C)C)=O)c(Cc2ccccc2)nc2ccccc12 C1(NC(c2c(C)cc(Br)o2)=O)CCN(C(=O)Cc2cnc[nH]2)CCC1CO C1(C(=O)NCC(C)NC(c2cnc(C(C)(F)F)s2)=O)CC(=O)N(C)C1 N1(CC(=O)NCC(CCC)NC(=O)CC2C(=O)NN=C2C)CCCNC1=O C1(CN(C(C2CN(CC)C2)=O)CC)CCN(C(=O)C(O)CC2CCOCC2)CC1 C1(NC(c2cc(C)oc2)=O)CCCN(C(c2cccc(C)c2Cl)=O)C1C Cc1ccc(C(=O)NCC2(NC(=O)CC34CCCC3C4)CCOC2)cc1O C12(C(N(C3CCCN(C(C4CCCCS4(=O)=O)=O)CC3)C)=O)CC(C)(CCO1)C2 c1(OC)ccccc1C(C)C(=O)NCC1(C)CC(NC(c2cn(C)cn2)=O)C1 C1(C(N(CC#CC)C(C)(C)C)=O)CC(NC(=O)OC(C)(C)C)C(O)C1C1CC1 c1(C(=O)NCC2CCCC(NC(=O)CCc3cnc[nH]3)C2)cc2ccccc2[nH]1 CN1CC=C(CC(=O)N2CCC3CCN(C(=O)CC4CCOCC4)C3C2)CC1 C1(NC(=O)CCc2cccs2)CC2CCC1N(c1ncncc1Cl)C2 N1(C(c2c(CCC)occ2)=O)CCCCC(CNC(c2ocnc2C2CC2)=O)C1 N1(c2[nH]c(=NCC3(CC)CCCCC3C)ncn2)CC2(CCCCCC2)C1 C1(OCC(=O)NCc2cc(N(C)C)sc2)CCN(C(=O)CCC2(C#N)CCC2)C1 c1(C(=O)NCCCCCC)cc(C2=CCCC2)cn(C)c1=O CC1CCN(C(=O)C(C)(C)n2cc(Cl)cn2)CC1NC(C1CN2CCN1CC2)=O C(=O)(CC(C)(C)CCOC)N(C1CCCC1)CCNC(CC(C=C)(C)O)=O C(=O)(C(C)C(C)C)N(C(C)C(=O)NC1(C)CC(O)C1)CC C1(C(=O)NCCOCCC=C)CN(C(c2nccs2)=O)CC12CC2 C(=O)(N=c1[nH][nH]c(C)c1Br)C1C(C(=O)Nc2cc(SC)cc(C(F)(F)F)c2)C1 C1(OC)CC(F)CN(C(c2ncoc2CNC(=O)CCc2nc[nH]n2)=O)C1 c1(OC)cc(Br)c(C(N2CC3CC3(CNCc3cc(C)ccc3F)C2)=O)cc1O O=C1CCC(C(=O)N2CCCC2CNC(c2nccn3nccc23)=O)=NN1 N1(C(C(CC)NC(C)=O)=O)CC2(CCN(C(c3nc(C(C)NC)no3)=O)CC2)C1 C(=O)(CCCCN(C)C)NCC(C)(C1CC1)NC(c1nc(OCC)sn1)=O N1(C(C=Cc2cn(C)nn2)=O)CCC2(CCN(C(C3CC(O)C(F)C3)=O)CC2)C1 c1(CNC(CCN(C(C2(CC)CCC2)=O)C)=O)cccc(Cl)n1 c1(CC(C)C(=O)NCCCCCCNC(C2CC2CF)=O)ccc(Cl)c(Cl)c1 C1(C(N2CCC(O)(C(C)C)C2)=O)CC2(CCN1C(c1ccnn1C)=O)CC2 C(C(C)(C)CC(=O)N1CCC(C)(C(N)=O)C1)NC(C(CSC)C)=O c1(OCCC)c(OC)cc(C(=O)NCC(C)N(C(=O)CC(O)C(C)C)C)cc1Cl C(=O)(C(C)(C)c1ccn(C)n1)NCCCN(CC)CC1CCOCC1 n1(CC(=O)NCC(CNC(CCc2cc(C)n(C)n2)=O)F)cccc(N)c1=O c1(C(N2CCC(NC(C(CC)(C)C)=O)C2C(C)C)=O)nccc(Cl)c1Cl C(=O)(C1=C(F)CN(C(=O)C#CC2CCCCC2)CC1)N1CCC(COC)C1 N1(C(c2ccno2)=O)CCCC2(CCCCN2C(c2cc(F)ccc2F)=O)C1 N1(C(c2c(SCC)nccn2)=O)CC(NC(c2sc(F)cc2Cl)=O)C(C)(C)C1 C1(F)(CNC(C2(C=C)CCC2)=O)CCN(C(C2COCCN2C)=O)C1 C1(NC(c2nn(C)c(Cl)c2)=O)CN(C(=O)CN2CCC(CO)CC2)C2CCCC12 C1(NC(CC2C(C)CCO2)=O)COC2(CCN(C(=O)C=CC3CCC3)CC2)C1 c1(NC(c2nn(C)cc2SC)c2n(CC(=C)C)nnn2)cccc(C(=O)OCC)c1 Cc1ccc(N)c(C(=O)NC2(CN(C)C(c3csc(F)c3)=O)CC2)c1 c1(C(=O)NCCCCC(C)NC(C2CC2(C)C(F)(F)F)=O)ccc2c(c1)OCC2 N1(C(CCCSC)=O)CCC(CO)CC1CO c1(OC)ccc(CC(=O)NCC2CCN(C(C3CN(C(N)=O)C3)=O)C2)cc1F N1(C(c2c(SC)ccs2)=O)CCN(C(=O)C(C2CCCCC2)O)C(C)C1 C1(C(N2C(CNC(c3ccc(C#N)cc3)=O)CC2)=O)CCn2cncc2C1 c1(C(=O)OC)ccc(C(=O)N(C)CC2CN(C(c3ccccn3)=O)C2)cc1C C1(N(C(=O)C(F)Cc2ccccc2)CC)CCCN(C(=O)C(Cl)=CCl)C1 C1(C(=O)NC(CNC(c2ccn(C(C)C)n2)=O)C2CCC2)CN2CCN1CC2C Cc1cccc(CN(C(C)CN2CCOCC2)CC2CCC2)c1 C#Cc1ccc(C(=O)NC2CC(C)(NC(=O)C(CC)OCC)C2)o1 Cc1ccc(-c2ccsc2C(=O)NC2CC3(C2)CC3NC(=O)C(C)C)cc1 c1(C(N2C(CN(C(COCC)=O)CC)CCC2)=O)ccc([N+](=O)[O-])c(N)n1 C(=O)(C(C)C(C)CC)N1CCC(C(CNC(C(COCC)(C)C)=O)(C)C)CC1 n1(CCN2C3C(C(=O)OC)CC(CC3)C2)ccc2cc(Cl)ccc12 N=S1(=O)CCC(NC(C2CC3CC(=O)CC(C2)N3)=O)c2cc(F)ccc21 c1(C(=O)NCC=CCNC(c2cnsc2)=O)cccc2[nH]ncc12 N1(C(c2c(SCC)ccc(Cl)c2)=O)CC2CC(NC(=O)CSC3CC3)CC2C1 Cc1cn(C)cc1C(N1CC(O)CC1CNC(C1CCCCN1C)=O)=O N1(C(CCC(=O)OC)=O)CCCC(CCNC(c2cc(C(C)(F)F)n[nH]2)=O)CC1 c1(NC(c2c(C)ccnn2)=O)cnc2cnccn12 CC1(CO)CN(C(C2C=CC(NC(C3(c4ccccc4)CC3)=O)C2)=O)CCC1O c1(N2CC(C(C)NC(=O)C(C)(C)C(F)F)OCC2)nc(Cl)ncc1[N+](=O)[O-] C1(CNCc2ncn(C)c2)(NC(=O)OC(C)(C)C)CCOCC1 C12(NC(C(CCC#C)O)=O)CCCC1CN(C(c1cc(CC)c(C)s1)=O)C2 N1(C(C(C)SC(C)C)=O)CCCC12CCN(C(=O)CSC1CCOC1=O)CC2 C1(C)(OC)CCCN(C(C2CC(O)CN2C(=O)CCC(=O)N(C)C)=O)C1 C1(C(=O)NCCCC(=O)NCCNS(C)(=O)=O)(CC)CCCCC1 c1(C(N2CCC(C)(Cn3ccnn3)C2)C(=O)NC)nccc(OC)c1OC C1(NC(C2C(OC)C2)=O)CN2CC1C2.c12cccc(c1)NC2=O.C1CC1.C(C)(C)O CC1CN(C(c2ncccc2Br)=O)CCC1N(C(=O)CCC(F)F)C C1(NC(C2C=CCC2)=O)COC2CN(C(c3ccc(-c4ccccn4)o3)=O)CC12 N1(C(c2c(OC)ccs2)=O)CCCC(C)(NC(c2ccn(C(F)F)n2)=O)C1 C1(NC(c2ccc(C)s2)=O)COC2(C1)CN(C(C1CC(C)OC1C)=O)C2 c1(CC(=O)NCC(C)(CO)NC(c2ccc(COC)[nH]2)=O)ccnc(C(N)=O)c1 C1(CC(=O)NC(CCC)(C)CC)CCCN(C(=O)Nc2c(C)noc2C)C1 C(CCC(C)C(=O)NC(CNC(c1ccnc(OC(F)(F)F)c1)=O)C(C)C)OC Cc1cccc2c1OC(C(N1CC3C(NC(C4(O)CCCCCC4)=O)C3C1)=O)C2 c1(CCOC(=O)CN2CCc3ccccc32)ncnc2sc(Cl)nc12 CC1(C(=O)NCC#CCNC(C2(c3cccc(Cl)n3)CC2)=O)CC2(CCC2)C1 C1(CNC(CC(C)NC(=O)CN=[N+]=[N-])=O)C(C)(C)C1(C)C c1(C(=O)NCC(CNC(=O)C(O)CCc2ccccc2)OC)cnccc1Cl C(=O)(CCC(=O)NN(C)C)N1C(C(C)C)CN(CCO)CC1 C=CC(C)(CC)C(=O)N1CCC(C(=O)Nc2cnc(O)c(C)c2)O1 CC(CC(=O)NCCC1CC(F)(F)CN1C(=O)C(C)n1ccnn1)P(C)(C)=O N#Cc1ccc(C(N2CC(NC(C3CC(C(F)F)C3)=O)CC23CCC3)=O)cc1Cl N1(CC)CCCC1C(=O)NCC1CC(NC(c2scnc2C(F)(F)F)=O)C1 N1(C(c2c(C)snn2)=O)CCC2(CCCN2C(C2CCN(CC(F)(F)F)C2)=O)C1 N1(c2nnc(CCOC)n2CC2CCOC2)CCC(S(=O)(=O)CC)CC1 C12(C(=O)NCCN(C(CC(CC)C)=O)CC)CCC(C(=O)OC)(CO1)C2 c1(N(C)C)nnc(C2CC2)n1CC.N1(CCOCCOC)CCCC1 C(=O)(CS(F)(F)(F)(F)F)NC1C(C)N(C(=O)COc2cccnc2)CC1 C1(C(N(CCNC(C23CCCC2(C(N)=O)C3)=O)CC)=O)Cc2ccc(F)cc2O1 C#CCCCCC(=O)NCC1COCC1NC(C1(F)CCN(C)CC1)=O C1(CN(C(CC)C(=O)N2CCCC2C(N)=O)c2ccccc2)(OC)CCOCC1 c1(CC(C)C(=O)N(C)CC2CCCN2C(=O)CCc2cc[nH]n2)ccccc1F C1(NCc2c(N(C)C)cccc2)CCN(C(c2cc(F)nc(F)c2)=O)CC1F CC1CCC(NC(c2c(F)cncc2Cl)=O)CN1C(c1ccnn1C)=O CC1CN(C(c2cccc(F)c2N)=O)CCN1C(C1CCOC(C)(C)C1)=O Cc1ccc(=NCCC(=O)NCC2(F)CCC(CNC(=O)COC(F)F)C2)[nH]c1 Brc1cc2n(c1)CCN(Cc1cc3ncccc3[nH]1)C2 N1(CCC(=O)N(C2CCC(NC(=O)CC3OCCCO3)CC2)C)CCOCC1=O C#Cc1cnc(C(N2CC(OC)CC2C(=O)NC(CO)CC(F)(F)F)=O)c(C)c1 N#Cc1c(F)ccc(C(N2CCN(C(=O)CCC(CF)CF)CC2)=O)c1F N1(C(CCn2cnc(=N)[nH]2)=O)CCOC(CCNC(c2cccnc2)=O)C1 c1(-c2c(OCC)nccc2SC)ccc2nc(C(=O)N=c3cc(C)o[nH]3)cn2c1 c1(SCC)ccccc1-n1cc(CN2CCC(CC#N)(COC(C)C)C2)nn1 c1(OCC)cnc(C(=O)NCC23CC(NC(=O)CCSCC(C)C)(C2)C3)c(Cl)c1 N1(CC)CC(C(=O)NCCN(CCOC)C(C2CCCCN2C(C)=O)=O)NC1=O c1(C(=O)NCC2CCN2C(c2cnns2)=O)cc(Cl)ccc1Cl C1(NCn2ncc(C(=O)OCC)c2)CCC(Cc2ccccc2)CC1 S(=O)(=O)(c1cccc(C(=O)NCC2CC2NC(=O)CC#N)c1)N(C)C1CC1 C1(C(=O)NCC(O)CNC(=O)CCCCF)(NC(C(CC)C)=O)CCCCC1 c1(C(=O)NCC2(C)N(C(C3C(C)C3)=O)CCC2)cc(O)c2cc(F)cc(F)c2n1 Cc1c(C(N2CCN(CCCNC(=O)C(C)C)CC2)=O)cccc1C1CC1 C1(CC)CCOCCN1C(=O)C(CNC(=O)CCOCC(F)F)N(C)C N1(C(C(=O)NCCC(=O)OCC)C2CC2C)CCCC2(C1)OCC1CC21 C1(CNC(C2CC2(F)F)=O)CN(C(c2nc(Cl)cs2)=O)CC12CC2 N1(CC)CCN(C(=O)CC2C3CCCC3N2C(=O)CCc2ccn(C)c2)CC1C N1(CCOC)CCC(C(=O)N(CC2CC(F)CN2CCOC)CC)CC1 C1(C(N2CC(OCCF)C2)=O)CC(O)CN1C(C12COCC1C2)=O C1(C(=O)NCC(C)CN(C)C)COC2(C1)CN(C(=O)CCc1ccsc1)C2 C(C(C)CC(=O)NC1C2CC1N(C(=O)C(C(C)C)Sc1ccccc1)C2)OC c1(C(N(CCC(=O)N(CC)Cc2cn(C)nn2)CCO)=O)n[nH]c2ccccc12 N1(C(C(F)OC)=O)CC(NC(c2cc(N)ccc2O)=O)CC12CCOCC2 C1(CNC(C23CC(OC)C2C3)=O)CCN(C(=O)C=Cc2cccnc2C)CC1O CC1CN(C(c2cnns2)=O)CCC1CNC(=O)C(C)(C)CCF C=CC(C)(C)CC(=O)N1CCC(NC(=O)C(c2cccc(C)c2)C)C12CC2 N1(C(Cc2nc(C)oc2)=O)CCCC(NC(=O)C(C)C(C)(F)F)C1C c1(NC(C2CN(Cc3cc(O)cc(Cl)c3)CCO2)=O)cccc2ncc(Br)cc12 c1cc2[nH]c(=NCC3CCCN3CCCO)[nH]c(=NC3CCCC3)c2[nH]1 C(C(C)(C)CC(=O)N1CCOC(C)C1C)NC(C1C(C)OC(=O)N1)=O C1(C#C)(C(=O)NC(C#C)CC2CCCC2)CN(C(c2[nH]ccc2CC)=O)C1 N1(C(c2nc(CC)oc2)=O)CCCC(CC(=O)N(C(C)CO)CC2CCC2)CC1 Fc1cc(N(Cl)Cl)cc(CN(c2ccccc2)CCCCN2CCCCC2)c1 N1(C(CC(CC)OC)=O)CC(CNC(c2scnc2C2CC2)=O)C2(CC2)C1 CC1CC(CCNC(c2ccn(C(C(=O)OC(C)(C)C)(C)C)n2)=O)CCO1 C1(NC(C(C(C)C)F)=O)CCC(C)N(C(=O)C(C)OCc2ccncc2)C1 C1(NC(CCCNC)C(=O)OC)COc2ccccc2C1 c1(C(=O)OC)cccc(C(=O)NCC#CCNC(=O)CC2CCCC(O)C2)n1 N1(C(CC=CC)=O)CCN(C(c2cccc(CSC)c2)=O)C(C(C)C)C1 N(C(=NCC(C)(O)C1CC1)NCC1CC(=O)N(CC2CC2)C1)CC1C(CC)CCO1 N1(C(c2ncn(C)c2)=O)CC2CCC(CNC(C3(C4(C)CC4)CC3)=O)(C2)C1 C(=O)(CC(O)C(C)CC)NC(C(=O)NCc1cnc(CC)s1)C1CC1 C12(CNC(c3ncsc3Br)=O)CC1CN(C(=O)CC1(C(F)F)CC1)C2 Cn1cc(C(=O)NCC2CC(F)CN2C(=O)C(=O)NCCC(N)=O)n(C)c1=O C=C(C)CC(C(=O)NCC1(O)CCCCCC1)NC(c1cc(C(C)=O)[nH]n1)=O CC1(C)CC(NC(C2(O)CC(F)(F)C2)=O)CN1C(=O)C1=CCSC1 c1(C(N2CCC(CNC(c3c(NCC)scn3)=O)C2)=O)cc(C)c(F)cn1 c1(C(N(C2CCCN(C(c3cn(C)cn3)=O)C2)CC)=O)ccc2c(c1)N(C)CC2 Cc1cnc2nc(C(N3CCC4(CCCN4C(=O)CC=C(Cl)Cl)C3)=O)nn2c1 N1(C(CC2(CC)CCOCC2)=O)CCN(C(C2CC(=O)N(OC)C2)=O)C(CO)C1 c1(C(=O)NC(CNC(c2cnc(C(C)C)[nH]2)=O)C2CCC2)ccc2[nH]ccc2n1 N1(C(C(CC)OCC)=O)CCN(C(=O)Cc2c(F)cccc2F)C(CCO)C1 C(=O)(C(F)C(=O)NCCC1(OC)CN(C(c2sc(C)nc2CC(C)C)=O)C1)OC c1(C(=O)NCC2(NC(C3CC4CC4C3)=O)CCCCC2)cnc2ncccc2c1 Cc1ccc(C(N)=O)cc1C(=O)NC1CCN(Cc2c(C)nn(C)c2Cl)CC1 c1(C(=O)NC(C2CN(C(=O)CC3(C4CC4)CC3)CCO2)C)cccc(CO)c1 C1(NC(C(C)NS(C)(=O)=O)=O)CC2CN(C(c3cccc(C(C)(F)F)c3)=O)CC12 C1(N(C(CC=CC)=O)C)C2CN(C(=O)C(CC)Sc3ccccc3)CC12 N1(C(C2(CC)CNC(=O)C2)=O)CCCC(CC(=O)N(C2CC2C)C)CC1 C1(CC(N2CCC(NC(C(C(C)C)NS(N)(=O)=O)=O)CC2)=O)CCC(=O)NC1=O C1(N(c2c(OC)nc(Br)cn2)C(c2coc(C)n2)=O)CC2(CCNCC2)C1 N1(C(C(CC)OCC)=O)CCN(C(=O)C(C)(C)CCOC)CC1c1cccnc1 c1(C(C)=O)ncnc2c1ncn2C1CC1.c1(C(=O)NCC(O)CN)coc(C2CC2)n1 c1(C(CCC(c2nnnn2CC)C2CC2)NCC(CO)C2CC2)ccc(Cl)cn1 C1(CNC(Cc2n(C)ccn2)=O)N(C(=O)CC(C)(C)C#N)CCC1(C)C c1(C(N2CCC(C(C)NC(=O)CCn3ccnn3)C2)=O)ncn2cccnc12 C1(C2CCN(C(=O)CCC3OCCO3)C2)(NC(C2CCn3ncnc3C2)=O)CC1 Cc1cc2cc(C(N3CCCC(CN(C(=O)C(C)CO)C)C3)=O)ccc2cn1 C=C(C)CC(C)C(=O)N1CC(OCCNC(c2c(C)cccc2Br)=O)C1 c1(C(C(=O)N(CCC)CCNC(c2nocc2C)=O)C)ccc(F)c(Cl)c1 N1(C(C2N(C)CCN(C(C(CC)(C)C)=O)C2)=O)CCC(F)(F)C(F)C1 N1(CCCNC(C(CC)N(C)C)=O)CCN(C(C2(SC)CC2)=O)CC1 c1(C(C)=O)cnc2sc(C(N3CC(F)(CF)C3)=O)c(C)c2c1 c1(C(N2CC(CC=C)(C(=O)NC(C)C(C)CCC)C2)=O)cc2ccccc2o1 CC(CC(=O)NC1COC(c2cccnc2)C1)c1ccco1 c1(C(C(N2CC(NC(c3ncn(CC)c3)=O)(CO)C2)=O)C)cccc(Cl)c1 C(=O)(CCCCc1ccc(OC)cc1)N(CC(CC)NC(=O)C(C)(C)C1CC1)C C(=O)(CCCCC(C)=O)NCC1(C(=O)NCC(C(C)C)OC)CC=CC1 C1N=C2NC=NC(=C2C)NCC12CCC2.C(CS(=O)CC)SCC N1(C(c2c(CC)nco2)=O)C2CCC1C(CNC(c1cc(OC)ccc1N)=O)C2 Cc1cc2ccc(C(N3CCC4(CCC(NC(=O)C5=CC(C)C5)C4)C3)=O)cn2c1 Cc1cc(C)c2nc(N3CCCCC(CNC(C4(C)CCC(=O)N4)=O)C3)sc2c1 C1(CC(=O)N(C2CCN(c3ncc(C(C)(C)O)cn3)C2)CC)CCCNC(=O)C1 c1(CCC(N2CCCN(C(COC(C)(C)C)=O)CC2)=O)cccc2ccccc12 N1(C(C2CC(=O)NCC2)=O)CC2CC1CN2C(c1cc(C2CCOCC2)n[nH]1)=O CC1CN(C(=O)C(C)(C)CF)CC1NC(C1CCN(CCS(N)(=O)=O)CC1)=O c1(C(=O)NC(CNC(=O)Cc2cccc(CO)c2)CO)ncc(C2CC2)cc1F c1(C(N2CC(C(C)NC(=O)C(O)C3CC3)C2)=O)ccn2ccccc12 C(=O)(C(O)CC(F)F)N(C1CCCN(C(C2CCC(C)(C)CC2)=O)CC1)C C1(C(=O)NC2C(OCC)CCC2)CCCCCN1C(c1ccsc1)=O N1(CCC)CCCC(C(=O)NC(CNC(=O)CCc2cnc(C)o2)C(C)C)C1 CCC(C)C(C(N)=O)NC(c1csc(CNC(=O)CCc2ncnn2C)c1)=O Cc1cc(Br)cc(C(=O)NC2CC(NCc3c(Cl)cccc3I)C2)c1O C(=O)(C1=CC2CCCC12)N(CCNC(c1n(CC=C)ccc1)=O)C(C)C C1(C(=O)NCC(C)NC(C2(C3CCOCC3)CC2)=O)COC2(CCC2)CO1 Cc1cnc(C(=O)NC(C)(C)C(=O)N(CC(C)O)C)cn1 c1(C(=O)NC2CN(C(c3c(CC)ncnc3)=O)CC2C)c(F)ccc2c1OCC2 c1(C(N2C(C(=O)NC3(CC#C)CC=CCC3)CCC2C)=O)cn(C)c(=O)cn1 C1(CNC(CC(=C)Br)=O)CCC(F)(CNC(=O)C(F)CC2CC2)C1 C(N=c1[nH]c(=NCC2(CO)CC23CCC3)c2sccc2[nH]1)C1C(CCC)C1 c1(OC)cc(C(=O)NC2CCCCC2CNC(C2(CO)CCCC2)=O)ccc1C C1(C)(CNC(c2nc(CCC)sc2)=O)CCN(c2nc(C(F)(F)F)ns2)C1 c1(CC)c(C(=O)N(CC(C)NC(=O)C(C)n2cccc2)C)cccc1C c1(OC)cc(O)c(C(=O)Nc2cc(C(C)C)cc(C(C)C)c2)cc1OC N1(C(CCCCC=CC)=O)CC(C(=O)NC(C)CN(C)C)CC(C)(C)C1 N1(CCCC(=O)N(C2CCN(C(C3CC3(C)C)=O)CC2)C)C(=O)NC(C)(C)C1=O N1(C(C2=C(C)OCC2)=O)CC2(C(=O)N=c3ccn(C4CCC4)[nH]3)CCC1CC2 N1(CCC)C(=O)NC2(CCN(Cc3nnc(-c4sccc4Br)o3)CC2)C1=O c1(C(=O)NCCC2OCCN(C(C(CSC)O)=O)C2)ccc(O)cc1C N1(C(C(C=C=C)C)=O)CCN(C(c2ocnc2C2CC2)=O)CC1C(F)F N1(C(c2nncc(OC)c2)=O)CCN(C(c2ccoc2C2CC2)=O)C(C)C1 C(=O)(C(C(C)C)C1CCN(c2cc(NC(C)(C)C)ncn2)CC1)NC(=O)OCC Cc1nn(C)c(C)c1CNC(=O)C(CO)NC(c1ccc(F)s1)=O c1(C(=O)NCC2(CNC(=O)CCOCC(F)F)CC2(F)F)cnc(O)c(F)c1 CC1(C)CC(=O)C(N(C2CC2)Cc2cn(C(C)(C)C)c(=O)nc2O)C(C)(C)C1 c1(CC(=O)NC2C(NC(c3ccc(CC)cn3)=O)CCC2)cn2cc(C)sc2n1 N1(C(CN2CC(=O)NC2=O)=O)CCOC2CN(C(C3CCCCS3)=O)CC12 CC1(C)CN(C(C2(C(F)(F)F)CCC2)=O)CC1CNC(=O)CN1CCOCC1 c1(C(=O)NCC(C2CC2)NC(C2(COC)CCOC2)=O)ncnc2cc[nH]c12 c1(N(C2CCCN(C(c3cc(C4(C)CC4)n[nH]3)=O)C2)C)nc2cccc(Br)c2o1 c1(C(N2CC(CCNC(C3(NC(C)=O)CCC3)=O)C(C)C2)=O)cc(C#N)[nH]c1C c1(OC)ccc(F)c(C(=O)NCC2(C)CC(NC(c3cc(CO)c[nH]3)=O)C2)c1F C(=O)(C(C(C)C)c1ccc(Cl)cc1)NC(CN(C(c1cc(C)sn1)=O)CC)C CC(C(=O)NC1CCCCCCC1NC(C1CCC1)=O)S(=O)(=O)C1CCOCC1 C1(CC)CN(C(=O)C=Cc2cn[nH]c2)CCC1NC(c1cccc(Cl)n1)=O Cc1ccnc(F)c1-c1csc(NC(c2cc(Cl)n(C)n2)=O)n1 c1(OC)ccc2c(c1)CC(C(=O)NCC1C3CC1N(C(=O)CNC=O)C3)CC2 N1(C(C2CN(C(C3(CC(=O)OC)CC3)=O)CC2C)=O)CC(C)(C)OCC1C C1(CC)CCN(C(C23CCC(CC2NC(c2cccc(F)c2C)=O)C3)=O)CCO1 Cc1nc2ccc(C(=O)NC(C)(C)CCNC(C3(C)CCNC3=O)=O)cc2n1C Cc1ccc(C(N2CC(CNC(=O)CC(C(F)F)n3ccnc3)C2)=O)c(O)c1C N1(C(c2onc(CC)n2)=O)CCC(NC(C2(C)CCCOC2)=O)C(CO)CC1 N1(C(CC2C(C)(C)CCCC2)=O)CCc2ccc(Br)cc2C1C(F)(F)F Cc1cc(C(N2CC(CO)(NC(=O)CNc3cccc(F)n3)C2)=O)cc(Cl)c1 N1(CC)CCC(C(C(F)(F)F)N(C)C)CC1.c12ccc(s1)c(=O)[nH]2 C1(CC)CCN(C(C2CCN(CC)C2)=O)C1C(=O)NOCC1CCOC1 c1(CC)occc1C(=O)NCC1CCN(C(N)=O)C1.C12(CC1)CCCC(=O)N2 C1(O)(C(N2CCN(C(c3c(C(C)C)ncnc3)=O)CC2C)=O)CN2CCC1CC2 c1(SCC(=O)NC(CNC(CC(C)C)=O)CO)cccc(F)c1 S(=O)(=O)(c1ccc(Br)cc1)N1C(CCC(SC(C(=O)NC)CC(C)SC)=O)CCC1 c1(OC)c(C)cc(C(N2CCC(CNC(=O)CCCCBr)C(F)(F)C2)=O)cc1C S(=O)(=O)(c1cc(Br)c(F)cc1F)N1CCC(CC(=O)NCc2ncc(C)nc2)C1 CCC(C(C)CN(C)C)NC(C1CCN1C(=O)CC(Cl)Cl)=O C=CC1(C(N2CC(C)(C)C2C2CC2)=O)CCN(C(C2CC2(F)Cl)=O)CC1 CC1(C(=O)NC2CCCC2CF)CCCN1C(c1ccc(O)cn1)=O C1(F)(CNC(CCC(=O)N(C)C)=O)CCN(C(=O)Cc2ccccc2)CC1 CC(C)C(O)CCN=c1[nH]c(=NCc2ncoc2C(C)(C)C)c2sccc2[nH]1 C1(N(C(C2C(=C)C2)=O)C)CCCCN(C(=O)Cc2cncn2C2CC2)C1 c1(C(=O)NC(C)CCCNC(=O)Cc2cn(C)nn2)cc2c(O)ncnc2cn1 N1(C(Cn2c(C)nnn2)=O)CC2CC1CN(C(=O)CCOCCOCCCO)C2 CC(C=CS(C)(=O)=O)N=c1[nH]c(N2CCCCC(CO)C2)nc2c1CCC2 C1(C(N(C)CC2CC(=C)C2)=O)(NC(=O)CN2CCCCCC2)CCCC1C CC1CN(C(C2CCC(C3CC3)N2C(=O)CC2CCC(C)(C)C2)=O)CCS1=O Cc1cccc(C(CN)C(=O)NCC(c2cccc(O)c2)O)c1 N1(C(C(C2CCCCC2)OC)=O)CC(O)CC1CNC(C1(CCF)CCC1)=O C1(NC(N2CCN(C(c3cccc(=S)n3O)=O)CC2)=O)CCn2ncnc2C1 c1(C(=O)NCC2(CNC(C3CC4C=CC3O4)=O)CC2(F)F)cc2n(n1)CCCO2 Cc1cc(C(=O)N(CCCNC(C2CC2c2cnn(C(C)C)c2)=O)C(C)C)n[nH]1 N#Cc1ccccc1CN1CCOC2CC12.N12CCCC1CCC2=O N1(C(C2(SCC)CC2)=O)C2CCC1CC(CNC(=O)C(CC)CC(F)F)C2 C1(NC(c2c(C)c(Cl)ccn2)=O)COC2CN(C(=O)CCCc3ncco3)CC12 c1(C(=O)NCC2(C)OCCN(C(C(CCC)C)=O)C2)cc([N+](=O)[O-])oc1C c1(C(N2C(C(C)NC(C3(COC)CCCO3)=O)CCC2)=O)csc2nccn12 Cc1ccc2cc(C(=O)N(CCNC(=O)C(N3CCOC3=O)C)C(C)C)cn2c1 C(=O)(CC(C)(C)C(C)(F)F)NC1CCN(C(C2ON=C(C(C)(C)C)C2)=O)CC1 CC(C(C)(C)C)=CC(=O)N(C1(C(=O)N(C(C)C(C)C)C)CC1)C Cn1nc(C(=O)NC2CC(CNC(C3CCCC3O)=O)C2)cc1C1(Cl)CC1 c1(N2CCC3(CN(C)C3)C2)nc(=NCP(C)(C)=O)[nH]c2c1CCCC2 C(CC(=O)NC1CCC1O)(C1CC1)NC(C(=O)NC(C)C)=O CC(C)(C)CC(=O)NCC1(C(C)(C)C)CCN(C(=O)COC(C)(C)C)C1 N#Cc1ccc(Br)cc1CNC(=O)CN1CCN(Cc2c[nH]ccc2=N)CC1=O C1(O)(C(C)NC(C2CC2C(F)F)=O)CCN(C(=O)CC2(C)CCOCC2)C1 N1(C(C)=O)CCN(C(=O)CCOC(CC2(OCC)CC2)=O)CC(O)C1 O=C(CCCCC1CC1)NCC(O)CCNC(c1sccc1-c1ccccc1)=O C(CC(C(C)(C)C)NC(c1ccc(F)cc1Cl)=O)N(C(C1CCN(CC)C1)=O)C N1(C(c2c(CC)nccc2)=O)CC2(CO)CC1(C(=O)NCC1C=CCC1)C2 C1(NC(CSCC=C)=O)CC(F)CN(C(c2ccc(O)c(CO)c2)=O)C1 Cc1ccc(Cl)cc1C(=O)NC(C1CCCN1C(c1cc(C(C)(C)C)no1)=O)C c1(C(C(=O)NCCC(Cn2cc(C3(C)CCCO3)nn2)F)O)ccc(F)c(Br)c1 N1(C(C(CC)O)=O)CC(c2ccccc2)CC1C(=O)Nc1ccc(F)cn1 C12(C(N3CCC(C(C)C)(C(N4CC(n5cnnn5)C4)=O)C3)=O)CCCC1C2(F)F CCC(C)(C(=O)NC(C1(O)CN(C(c2cc(CN(C)C)on2)=O)C1)C)OC CC1CN(C(C2CCCN2C=O)=O)CCN(C(=O)C(O)Cc2ccccn2)C1 Cc1cc2[nH]c(C(N3CCN(C(c4ccsc4Cl)=O)CC3C)=O)cc2o1 c1(C(N2CC(C(N3C(CCOC)CCCC3)=O)C2)=O)cccc2ncc(Br)cc12 Cc1scc(C(=O)NCCC2(O)CN(C(c3ccncc3O)=O)C2)c1C c1(C(N(CCCO)C(C)C)=O)cccc(CNC(C2CCCC(O)C2)=O)n1 CCCCCCC(C)(C)C(=O)N1CCCC(CO)(NC(=O)C(O)CC(C)C)C1 CCC(CC(=O)NCC#CCNC(=O)C=CC1CCCN1C)C1CCC1 N1(C(c2ncc(N)nc2)=O)CCc2ccccc2C(NC(=O)CC2(CO)CC2)C1 c1(C(N2CC(CNC(CCCC=C)=O)OCC2)=O)cc(C(C)C)cnc1O N1(C(CCc2ccc(C)o2)=O)CCC(C)(C)C(NC(C2(C)CCCCC2)=O)C1 C12(NC(Cc3nc(COC)sc3)=O)CCN(C(C3(C#N)CC=CC3)=O)CC1C2 c1(OC)ccc(SCCC(=O)N2CCC2COC(C2(C)CCNC2=O)=O)cc1OC c1(CNC(=NCCC)NCCN2CCOCC2)cccc2c1OCCCO2 C1(Cn2cc(-c3cc(C(C)=O)nn3C)nn2)CC(F)(F)CN1C(=O)C(C)CO O=C(C1=C(Cl)CCCC1)NC(c1ccccc1)CNC(C1CC1C1CC1)=O N1(CCC#C)CCN(C(=O)C(C2CCCN(C(=O)CCC(C)N(C)C)C2)C)CC1 N1(C(CCOCCOCC)=O)CCC(C(=O)NC(CO)(CO)CO)C(C)C1 c1(OC)cccc(OC)c1C(=O)NC1CC(NC(C2CSCN2C)=O)C1 c1(CC(=O)N(CCC(=O)NC2CCOCC2)CCC)ccc(SC)cc1 c1(C(N2CCOCC(NC(C=CC(C)C)=O)C2)=O)ccc2c(c1)CCC(=O)N2 c1(NCCNC(=NCC)NC(C)CCn2ccccc2=O)ccc(C)cc1C C(=O)(C(C)CCC(C)(C)C)NCC1(CNC(CC(CC)C(C)C)=O)CCCCC1 N1(C(c2c(C(F)(F)F)nc(C)n2O)=O)CC(NC(=O)C(C)C)CCC(O)C1 Cc1ncccc1C=CC(=O)NCC1(F)CN(C(=O)C(C)(C)O)C1 N1(C(c2ccccc2)=O)CCS(=O)(=O)CC1.n12c(nnc1O)C1CCN(CC1)CC2 C1(CC(N2CCC(CC)C2)=O)CCN(C(=O)C(C)n2cccc2)CC1 N1(C(C(C(CC)CC)OC)=O)CCOC2CN(C(=O)CCP(C)(C)=O)CC12 N1(C(C2CC3CCC2N3C(=O)CSC(F)(F)F)=O)CC2CCC1C(O)C2O CC1CN(C(c2cc3sccc3[nH]2)=O)C(C)CN1C(c1ccc([N+](=O)[O-])o1)=O C1(C(=O)NCCC(C)(C)CNC(C2CC3(CCC3)CO2)=O)CCCCC12CCC2 c1(-c2ccc(C(C(=O)NCC=C)N(c3ccccn3)CCOC)o2)ccccc1Cl c1(C(=O)NC(C(=O)NCC2(CO)C(C)(C)C2)Cc2cn[nH]c2)nc(=N)cc[nH]1 C1(C(=O)NCc2cccc(C(N3CCC(CC4CC4)C3)=O)n2)CC2CCCC2C1 N1(C(c2scc(C)c2)=O)CC(NC(c2csc(C(C)(C)C)n2)=O)C2(CCC2)C1 c1(C(=O)NC2CC23CC(NC(=O)C(F)Cc2ccccc2)C3)cc2c(s1)CCC2 C12(C(N3CCCC(CCNC(C(C)CF)=O)C3)=O)CC3CC(CC(C3)C1)C2 c1(C(=O)NCC2N(C(C3CCCN(C)C3)=O)CCCC2)ccc2c(c1)nnn2C c1(C(=O)NC2C(N(C(CCc3cc(C)no3)=O)C)CCCC2)cncc(Cl)c1C C1(C)(C(N(CCC)CCC)=O)CCN(C(=O)C(C)(O)COC)C1 C1(C(=O)NCC(CNC(=O)C(c2ccn(C)n2)C)OC)CCNC1=O N1(C(C(c2ccco2)NC(CCOC)=O)=O)CCCN(C)CCC1 C1(C(=O)NCC23OCC(NC(C(C)(C)OC)=O)(C2)C3)COc2cc(F)ccc2C1 c1(C(=O)NC2C(CNC(C3C(CC)C3)=O)C2)ccccc1NS(=O)(=O)CC N1(C(c2c(C)nn(CCO)c2)=O)CCC2(C1)CN(C(=O)Cc1cnsc1)C2 c1(C(N(CC(=O)NC(CC#C)CO)CCOC)=O)ccccc1F Cc1cc(C)c(C(=O)NCC(C)(C)CC(=O)N(C)CCn2cnnc2)cn1 c1cc(F)ccc1Br.c1(OCC)cccc(CNC(=O)Cc2ccccc2Cl)c1 C1(C2(C)OCCO2)CCN(c2nnc(-c3cc(Br)n[nH]3)n2CC2CCCO2)CC1 S1(=O)(=O)c2ccc3c(c2)CCN3C(=O)c2ncn3c2CN1CC3.C(C)(=O)NC N1(C(C#CC(=O)N(C)C)=O)CCC(C2CCN(C(C3CC4(C3)CC(F)C4)=O)C2)C1 c1(C(N(CCCNC(=O)Cc2cnn(C3CCC3)c2)CC)=O)[nH]c(C)nc1C c1(C(=O)NC2C(NC(c3nc(CCC)oc3)=O)C2)cncc(-n2cnnn2)c1 C1(C(=O)NC(C(C)(C)C)CNC(C2CC2(F)F)=O)CC2C(C1)C2(F)F N1(C(c2c(SC)cccc2)=O)CC2(CNC(C3(C)CCOC3C)=O)CC(F)(C1)C2 C(=O)(CCCCCC(C)O)N(C1CCN(C(=O)Cc2ccc(F)c(F)c2)C1)CC C(=O)(CCC(CC)OC)NCC(CN(C(C1CC(C)=NO1)=O)CC)(C)C C(C)(C(C)C)=CC(=O)N(CC(C)C)CC.C(C(C)O)N N1(C(C2N(C(C3N(C)CC(C)(C)C3)=O)CC=C2)=O)CC(C2CCCCC2)C1 Cc1sc(Cl)c(C(=O)N(C)CC2CCN(C(c3ccc(C(N)=O)cc3)=O)C2)c1C C1(NC(CCCc2nc(C)sc2)=O)CC(C)N(c2nnc(C(C)C)o2)C1 c1(OC)cc(=O)n(C)cc1C(=O)NC(CO)CCCCNC(C1COCCO1)=O C1(OC(C)=O)CCC(CN=C(NC2CC2)NC2CC(OC(C)(C)C)C2)CC1 c1(C(N2CC(CNC(CCC)=O)N(C)CC2)=O)cc2c(C)cccn2n1 C1(COC)(NC(=O)CCOC(C)C)CCN(C(=O)C=Cc2cnc[nH]2)C1 C1(NC(c2cnc(C)s2)=O)CC2C1CCN2C(=O)CN1CCN(C2CC2)C1=O C(=O)(C(C)CC(C)C)N1CCC(N(C(=O)COCCCOC)CCCC)CC1 c1(C(=O)NC23CCC(C2)N(C(=O)C2=CCCSC2)C3)c[nH]c2c(Cl)cccc12 C1(NC(c2cn(C(C)C)nc2Br)=O)CCN(C(=O)Cc2ccco2)CC1C C1(COC(C(c2ccc(C(C)(C)C)cc2)(C)C)=O)CC2CC1C1CC21 C1(CNC(C=CC2N(C(C(OC)OC)=O)CCC2)=O)CCC2(CCC2)O1 CCCCC(CC)CCC(=O)NCCOCCNC(=O)CSCc1cccnc1 S(=O)(=O)(c1cnn(CCF)c1)NC(c1ccc(NCc2ccccc2)cc1)=O c1(C(C(N2CC(O)(CNC(C3CCCO3)=O)C2)=O)O)cccc2c1OCC2 CCC(COC)C(=O)N(CC(C)(C)C(=O)NCc1nc(C)cs1)C C1(C)(CCNC(C(CCC)N(C)C)=O)CCCN(C(=O)C(CC)OC2CCCC2)C1 C(C(C)C(=O)NCC(C1CCC1)NC(=O)C(C)(C)c1cnsc1)SC c1(NC2(c3n(CC)nnn3)CCOC(CC(C)C)C2)ccc2ncccc2c1 C1(C(=O)NC2CCN(C(C)(C)C)C2=O)CNc2cccc(Br)c2O1 c1(C(=O)NC(C)(CNC(c2cnc(Cl)s2)=O)C2CCC2)ccnc2cc[nH]c12 C(=O)(C(F)C(C)(F)F)N1CC(N(C(=O)CC2C=CCC2)C)C1 c1(C(C(N2CCC(C(C)NC(C3(OC)CC3)=O)C2)=O)(C)C)ccccc1F C#CC(CNC(C1(OC)CCN(C(c2cccc[n+]2[O-])=O)C1)=O)CC(C)(C)C Cc1ccc(Cl)c(O)c1C(=O)NCCC1(O)CN(C(C2CC23CC3)=O)C1 N1(CC)CC(C(=O)N(C(C)CNC(c2c(C)cc[nH]c2=N)=O)C)c2ccccc21 c1(CC(=O)NCC(C2CC2)NC(c2ncoc2C2CCOCC2)=O)ccccc1 N1(C(C2C(C)CCC2)=O)CCC(OCCNC(=O)Cc2cncs2)CC1 C1(C(C)(C)C)CCC(C(=O)NCC2CCC(NC(c3cccc(F)n3)=O)C2)CC1 c1(C(=O)NCC2(C)OCCN(C(CC(=C)C)=O)C2)ccn2ncc(Br)c2c1 N1(C(C2CN(C)C(=O)N2)=O)CC(NC(c2ccc(CS(C)(=O)=O)o2)=O)C2(CC2)C1 C1(CCCNC(=O)CCc2ncc[nH]2)CN(C(=O)CCC2CC2(Cl)Cl)CCO1 Nc1ccc(-c2cn(CCOCCN(C(=O)C3=CCOC3)C3CC3)nn2)cc1 S(=O)(=O)(c1ccc2c(c1)CCCC2)N1CCC(O)(CNC(C2(CC)CC2)=O)CC1 N1(C(c2cc(OC)n[nH]2)=O)CCN(C(c2ccsn2)=O)C(c2ccccn2)C1 C(=O)(CCCCC(C)CC)NCC1(C(=O)NCc2c(CC)nns2)CC=CC1 C1(C(N(CCCn2cnnc2)C)=O)CCC2CCC1N2C(=O)OC(C)(C)C C1(C(C)C)(C(=O)NC(CO)C2(O)CC2)CCN(C(=O)C(c2cnn(C)c2)C)C1 Cc1c(Cl)cnn1CC(=O)NC1CCOCC1NC(=O)CC1CC2CC2C1 Cc1ncsc1CC(=O)NCC(C)CN(C(=O)CN(C)CCO)C C1(OCCCCC)CN(C(=NCC(C)(C)C2CCC2)NCC2CC23CC3)C1 N1(C(c2c(OCC)nccc2)=O)CC2CC(C)N(C(=O)CCOC3CC3)C2C1 C1(C2CC2)(CNC(c2cc(C)ncc2C)=O)CCN(C(C2(C)CCSCC2)=O)C1 N1(C(C(C)C)=O)CCCCC2(CCN(C(c3cccc(C4CC4)n3)=O)C2)C1 CC1(C)CC(NC(=O)CC2(CNC(C3C(C)(C)C3(F)F)=O)CC2)CO1 C1(NC(C(C)OC2CCCC2)=O)CN(C(c2cc(Br)co2)=O)CC1CO C(=O)(C1CCCc2n[nH]cc21)N1CCC(NC(C2N(C)C(=O)CC2)=O)C(F)C1 C(=O)(C1CCCc2ncnn21)NC1C=CC(NC(=O)CN2CCC(CO)CC2)C1 N1(C(c2c(C)nc(CNC(CC(CC)C(C)C)=O)o2)=O)CCC2(CNC(=O)O2)C1 C(=O)(CN=c1cc[nH]cc1)NCC1CCCC(C(=O)NCc2c(C)noc2C)C1 c1(C(N2CC(NC(CCSCCCC)=O)C3C2C3)=O)cc([N+](=O)[O-])ccc1SC C1(CNC(C(C#C)(C)C)=O)CC2CCC(C1)N2C(c1scnc1C(F)(F)F)=O n1(CC)cc(C(=O)NC2(C)CN(C(=O)C=Cc3cnc[nH]3)C2)c(C(F)(F)F)n1 C1(CC(=O)NC2CCCC(C(C)C)C2)CC2(C1)CN(C(=O)Nc1ccccc1)C2 C1(C)(C(=O)NCCCCNC(c2c(C)nn(C)n2)=O)CCCCCC1 C1(CNC(c2cc(C)on2)=O)(NC(c2cncc(Cl)n2)=O)CCCCC1C C(CCCCCNC(C1CC1(F)Cl)=O)NC(C1(CC=C)CC1)=O Cc1cc(-c2cn(C3(C(N4CCC(CC5CCOC5)C4)=O)CC3)nn2)cc(C)c1 N1(C(C2(C)CCCO2)=O)CCC(C2CCN(C(c3c(F)ccnc3F)=O)CC2)C1 CC(C(C)C(=O)NCC1(C)CCOCC1)NC(c1ccn(C)c1)=O C1(NC(C(F)OC)=O)CCN(C(=O)CCCS(N)(=O)=O)CCC1CO c1(C(=O)NC(C)CNC(c2ccsn2)=O)c(Cl)cccc1[N+](=O)[O-] N1(C(c2cc(CC)c(C)s2)=O)CC(NC(=O)CN2CCNC(=O)C2)CCC1C C1(NC(CCC(=C)Cl)=O)CCSC12CN(C(c1nc(C)c(C)[nH]1)=O)C2 CS(=O)(=O)c1cc(C(N2CCCC23CN(C(c2csc(Br)c2)=O)C3)=O)ccc1F N1(C(c2cn(CCCOC)nc2)=O)CC2CCN(C(=O)CCC(CF)CF)CC12 c1(C(=O)OCc2ccc(C(=O)OC)c(OC(F)F)c2)cccc(F)c1C#N CN1CCC(C(=O)NC(C2CCOC2)CNC(=O)CCSCC(N)=O)(C(F)F)C1 C(=O)(C1=CS(=O)(=O)CCC1)NC1C(NC(c2n(C)ccn2)=O)C1 N1(C(CC(C)F)=O)CCC(F)(CNC(C2CC(=O)N(C(C)(C)C)C2)=O)C1 CCCC(C(=O)NCCCC(C)NC(c1ccc(OC)o1)=O)OCC c1(C(N2CCC(OC)(CNC(=O)CC(C)N(C)C)C2)=O)n[nH]c2c1CCOC2 c1(CNC(C2CC(NC(C(c3ccccc3)OC)=O)C2)=O)ccc(O)cc1 C1(CNC(c2cc(C)nc(C)c2)=O)CC2CCC1N(C(=O)COc1ccsc1)C2 C1(C(C)NC(=O)CSc2n[nH]c(O)n2)CCCN(C(C2CS(=O)C2)=O)C1 N1(C(c2n(CC)nnc2)=O)CCC(NC(c2ccsc2C)=O)CC1C N1(C(CCN(C(=O)C(C)S(=O)(=O)CC)CC)=O)CCCC(CNS(=O)(=O)CC)C1C N1(C(CSCCC)=O)CCCC2(CCN(C(C3CC4(CCO4)C3)=O)CC2)C1 C1(C(N(CCNC(c2c(C)ccc(OC)c2)=O)C)=O)CCCC12OCCO2 C1(C(=O)NCC(C(CC)C)CO)CC(N=[N+]=[N-])CN1C(=O)CC(C)CC c1(OC)cc(NC2CC3(C2)CC(NC(=O)CCCCCO)C3)nc(OC)n1 C1(C(=O)NCC2(N(C)C)CC2)CSCN1C(c1ccns1)=O Cc1cn2c(n1)CCC(C(=O)NC(C)CCNC(c1ccc3n[nH]cc3n1)=O)C2 c1(NCc2c(NCc3cc(OC)c(F)cc3F)ccs2)ncnc2[nH]c(C)cc12 Cc1cnsc1C(N1CC(O)(CCNC(=O)Cc2ccccn2)C1)=O C(=O)(C1=CCC(NC(=O)CCc2cn(C)cn2)C1)NC(CCCC)CC c1(C(N(CC(C)NC(c2n[nH]c(C3CC3)c2Cl)=O)C)=O)cc2c(nc1O)CCC2 CC(CC(=O)N1CC2(CC(NC(=O)CN3CCSCC3)CO2)C1)P(C)(C)=O N1(C(CCN(C)C)=O)CCN(C(=O)C(C)(C)CF)C2(CC2)C1 Cc1c(C(N2CC3C(CNC(=O)Cc4ccon4)C3C2)=O)[nH]c2cc(Cl)ccc12 c1(C(N2CCC(N(C(c3csnn3)=O)CC)C2)=O)nnn(C)c1C c1(C(=O)NCCC(C)N(C(C(C=C=C)C)=O)C)ccc(C)c(OCC)c1 N1(C(c2ccnnc2)=O)CC2COCC2(C(=O)NCC(c2cccc(O)c2)O)C1 n1(CC(C(=O)NCCNC(CCCc2cc(C)no2)=O)C)nnc2ccccc12 C1(C(N(CCNC(=O)Cc2cc[nH]n2)C2CC2)=O)C2Cc3ccccc3C12 C1(C(N2CCC(CNC(CSC(C)C)=O)C2)=O)CC2CSCC(C1)C2(F)F CCC(CC)(CCNC(=O)CC1(OC(C)C)CC1)NC(c1ccc(C)cn1)=O C1(C(=O)NCCCC(C)NC(=O)C(C2CCCCC2)C)(OCC)CCCCCC1 C1(C#N)(C(N2CCC(C(C)NC(C=C(CCC)CCC)=O)C2)=O)CC2CC2C1 N1(C(CS(CC)=O)=O)CC2CC(O)C1C2NC(c1cc(C)c(Br)o1)=O c1(C(C)NC(c2nn(CC)c(Br)c2Cl)=O)nnc2ccccn12 c1(C(=O)NC2C(NC(C(C(C)(C)O)F)=O)CC2)cc2c(cc1O)OCO2 N1(C(CC(C)(C)N(C(=O)CSCC(N)=O)C)=O)CCC(C2CC2)CC1 C1(C(N(CCNC(C(Cn2ccc(C)n2)C)=O)C)=O)CCc2cnnn2C1 c1(C(=O)NCC(C)NC(c2cc(C3CCC3)on2)=O)cnc2c(c1)nc(O)n2C N1(C(C2CC2c2cccc(Br)c2)=O)CC2CCN(c3ncccn3)C2C1 N1(C(c2cc(C)ns2)=O)CC2CCN(C(=O)CC(C)F)C2C1 CCCC(CC)CCC(=O)NC1(C)CC(NC(c2ccc(C(C)C)c(Cl)c2)=O)C1 C1(C)(C(=O)NCC=C(C(N2CC(O)(C(=O)OC)C2)=O)C)CCC(C)C1 N1(C(C2CCN(C(c3cc(SC)oc3)=O)CC2)=O)CC(F)(F)CC1CN(C)C CN=c1nc(C(=O)NC2CC2Nc2ncc(C(=O)OC)cc2C#N)cc(C)[nH]1 Cc1ccc(C(N2CCCC2C(N2CCC(C)CC2)=O)=O)c([N+](=O)[O-])c1 c1(CNC2CC3(CC(NC(Cc4nc(C)sc4C)=O)C3)C2)c(Cl)cc(F)cc1Cl c1(C(C(=O)NCCOC)N(C2CCCCC2C)CC)nc(Cl)ccc1Br C(=O)(C#CC1CCCCO1)N(C1CCCN(C(CC(COC)C)=O)C1)CCO c1(C(=O)NC(CSC)(C)C(=O)N2CC3CC3(CO)C2)cc(O)ccc1F C1(NC(=O)NC(c2cccc(OC)n2)c2ccccc2)CC2(CCOCC2)C1 Cc1ccc(C(N2CCC(=CCNC(c3c(C)nc(C)n3O)=O)CC2)=O)nc1C N1(C(C2C(n3cc(-c4n(C)ncc4)nn3)CCCC2)=O)CCS(=O)(=O)C(C)(C)C1 c1(CC(=O)NCC2(OC)CN(C(C3CCCCC3F)=O)C2)ccc(Br)cc1C C(=O)(CC(C)C(F)(F)F)NCCC1(NC(C2N(CC)CCCC2)=O)CCC1 C=CCN=C(NCCSc1ccc(-c2ccco2)cc1)N1CCN(CC)CC1 N1(C(C2C(C)(C)OCC2)=O)CC2OCCN(C(=O)Cc3cnns3)C2C1 C=CCCCC(C(=O)N(C1CC(O)C1)C)NC(=O)CC1=NCCCC1 C1(N(C(c2n(C(C)C)ncc2)=O)C)CCCCN(C(C23CCC2C3)=O)C1 c1(C(N2C3(CNC(COC)=O)CCC2CC3)=O)cc2c(Br)cccc2s1 C(CCS(=O)(=O)c1ccc(Cl)cc1)C(=O)NCc1cnc(C(C)C)[nH]1 c1(OC)cc(N)c(F)cc1C(=O)NC1(CNC(c2cncnc2C)=O)CCC1 C1(C(N(CC(C)NC)C(c2c(SCC)cccc2)=O)=O)CCc2n[nH]cc2C1 CC(N=c1[nH]c(=N)[nH]c(=NCCCn2cncn2)[nH]1)c1cccc(F)c1F N1(C(CC)=O)CC(CNC(C2C=CCC2)=O)C(F)(F)C1 Cn1c(C(N2CCC(O)(Cn3cc(C4CCC4)nn3)C2)=O)cnc1S Cc1ccc(O)c(C(N2CC(O)CC2(C)C(=O)NOCC(N)=O)=O)c1 CC1CCCC1(C)NC(c1conc1C(C)NC(C1(CN(C)C)CC1)=O)=O c1(OCC=C)c(C(=O)NCC2C=CCN2C(C2CC3COCC3C2)=O)cccc1C N1(C(c2c(C)cnnc2)=O)CCC(O)(CCNC(C2(C#N)CC(C)C2)=O)CC1 c1(-n2cc(CNC(c3c(CO)cccc3Br)=O)nn2)ccc(Br)cc1C(F)(F)F N1(C(C=CSC)=O)CC2(NC(C3CCS(=O)(=O)C3)=O)CCC1CC2 C(=O)(CCC(O)C(C)(C)C)NCCCCC(C)NC(c1c[nH]nc1C(C)(C)C)=O c1(C(N2CCC(NC(C(CC(C)C)NC(C)=O)=O)C2)=O)csc2cc(C)ccc12 CC1(O)CCC(C(=O)NC2CC(NC(C3CC(C)(O)C3)=O)C2)CC1 C1(C(N2C(CC(=O)N(C)CC3(C4CC4)CCC3)COCC2)=O)CCOC(=O)CC1 N1(CCOC(C2CCN(C(c3cccc(F)c3)=O)CC2)=O)C(=O)CCCC1=O CC(C)C(CCN(C(=O)C(F)CC1CC1)C)NC(c1csc(Br)n1)=O CS(=O)(=O)C1CCCCN(C(=O)Nc2cc(F)c(F)c(F)c2)C1 N#CC1(NC(c2ncccc2C(F)(F)F)=O)CCN(Cc2sccc2Cl)C1 C1(C(N2C(C)CC2CO)=O)CN(C(C2CCCCC2O)=O)CCN1C c1(C(=O)NC2C(CNC(C(C=C)(F)F)=O)CCC2)ccc(N(C)C)c([N+](=O)[O-])c1 c1(C(N2CCC(NC(C(CC)OC)=O)C(C)C2)=O)c(N)cc(Cl)cc1F c1(C(C)C)cc(=NCC2CC(C)N(C(c3ccn(C)n3)=O)C2)[nH]cn1 c1(C(=O)NCC2C(NC(C(C)c3ccsc3)=O)C2)cnc2sccc2c1 C(=O)(C(F)(F)C(O)C(C)C)N1CC(O)(CCNC(C(CC=C)CC)=O)C1 c1(C2C(NC(CC(c3ccc(F)cc3)N)=O)CCC2)cccc(Cl)n1 O=C(CCCc1ncco1)NC1CC(F)(CNC(=O)CC2(c3ccon3)CC2)C1 C1(NC(CN(S(C)(=O)=O)C)=O)CN(C(c2cc(C3CC3)no2)=O)CC1S(C)(=O)=O CC(C)C(CO)C(=O)N1CCCC1(C)CNC(C1CSCCS1)=O N1(C(C(C)(C)C2CC2)=O)CCOC2(C1)CN(C(=O)CC1(N3CCCC3)COC1)C2 CC(CCn1cncn1)N=c1[nH]c(=NC2CCN(C)CC2)c2cc(Cl)ccc2[nH]1 N1(C(C2CC(F)(CC)C2)=O)CC(O)CC1CNC(=O)C(F)=C(C)C1CC1 c1(C(=O)NCC2CC3CN(C(C=C(C)C(C)C)=O)CC32)cc2ccsc2c(O)n1 c1(CC)c(C(=O)NC(C2CCCN(C(c3cn(C)[nH]c3=N)=O)C2)C)csc1C O=C(CC1CCOc2ccccc21)NC1CN(C(=O)C#CC2CC2)CC12CC2 C(=O)(CCCCC(=O)N1CCC2CCCC12C(=O)NC(c1ccn(C)n1)C)OC Cc1nnc(C(N2CCCC2c2cccs2)C(=O)NCC(F)F)n1C c1(NC2C(F)COC2)nccc(=NCc2cncn2Cc2ccccc2)[nH]1 N1(C(C2(C)CC(C)C2)=O)CC2CC1C2CNC(c1cnc(C(C)(C)C)s1)=O Cc1[nH]c2ccc(Cl)cc2c1C(=O)NCC1COCCN(C(C23CCC2C3)=O)C1 CCC(COC)C(=O)NCC(C)CC(=O)N1CCCC1C(=O)N(C)C c1(CCC(N2CC(NC(C3(NC(=O)OC)CCCC3)=O)C2)=O)nnc(O)nc1O C(=O)(C#CC12CC3CC(CC(C3)C1)C2)NC1C(NC(C2N(C)CC(O)C2)=O)CC1 C1(CNC(C(C)OCC#C)=O)CC12CCN(C(=O)C(C1CCOCC1)O)CC2 CC#CCCCCNC(=O)CCC(C)NC(c1cc(OC)nn1C)=O Cc1cccc2c1CC(C(=O)NC1CC1NC(=O)Cc1ccc(F)cc1F)O2 C1(SCC(=O)N(CC)CC2CCCN2C(c2ccccc2)=O)CCC(F)(F)C1 c1(OC)cc(C)ccc1C(N1CCCC(O)(CNC(c2cc(OC)n[nH]2)=O)C1)=O C1(CN(C(CCc2onc(CC)n2)=O)C)CCN(C(C2CC(C)C2)=O)CC1 C(=O)(N1CCC(C(=O)NCC2CC(C(C)(C)C)C2)O1)c1cn(CC=C)nc1 c1(C(N2CCN(CCNC(CC(=O)OCC)=O)CC2)=O)ccc2nc(O)oc2c1 C1(C(=O)Nc2c(C)ncnc2)CCCCN(C(=O)CCCC2CC2C)C1 C1(CNC(C(C=CCCC)O)=O)C2CCC(C2)N1C(C1(N(C)C)CCCCC1)=O CC1(C)CC(C(N2CCCC2CCNC(C2CC2Cc2ccccc2)=O)=O)C1 c1(C(N(C2C(C)CCN(C(CCCOC(C)C)=O)C2)C)=O)cnn2ccccc12 C1(C(N(C(CNC(CNC(C)=O)=O)C2CC2)C)=O)C=C(C)CS1 c1(C(=O)NC2C(C(C)C)CN(C(=O)CC3CC3)CC2)nccc2ncccc12 c1(C(=O)OC)cc(C)nc(N(CCCN(C)C(C2CCCN(C)C2)=O)C)n1 N1(C(C)C)CCCC(NC(C2OCCC2NC(=O)Cn2ncn(C)c2=O)=O)C1 N1(C(C=C(C)C(=O)O)=O)CCOC2(COCCN(C(=O)C(C)n3cnnn3)C2)C1 c1(SC)cc(C(N2CCC(NC(c3cc(=O)n(C)cn3)=O)C(F)C2)=O)ccc1F c1(OC)cc(C)c(C(=O)NC2CCCCN(C(=O)CCC3CC3)C2)cc1Br Cc1nc(CC(=O)NCC(C)(C2CC2)NC(c2n[nH]cc2Cl)=O)n[nH]1 C1(C(=O)NCC2CCN2C(=O)CC=CC(C)(C)C)(COC)CCCCO1 Cc1n[nH]c(C)c1CC(=O)NC1CCC(NC(=O)CCN2CCCCC2C)C1 c1(NC(C2CCN(Cc3ncc[nH]3)CC2O)=O)cccc(Cl)c1[N+](=O)[O-] N1(CC(C)CC2CCC2)CCC(O)C2(CCOCC2)C1 C1(OC)(OC)CCC1CNC(=O)NCCn1nccc1C C1(F)(CNC(c2c(CC=C)cccc2)=O)CCCN(C(=O)C(C)(O)CC)C1 C(=O)(C1CCCn2cc(C)nc21)C1OCC(=O)N(CCOC)C1c1ccccc1 N1(C(CCOC(C)=O)=O)CCC2CCN(C(=O)CCc3nncn3C)CC12 C1(C(N2CC3(C2)SCCC3NC(C2(F)CCCC2)=O)=O)Cc2ccccc2N1 Cc1nn(CC(=O)NC(C)(CNC(C2(CCF)CCC2)=O)CO)cc1Br C1(C(C(=O)NCCOCCNC(C2(c3ccno3)CCC2)=O)O)CCCCC1 Cc1nc(C)n(CC2CN(C(=O)CCC3CCC(=O)C3)CCO2)n1 c1(C(C(=O)NCC(C)N(C)C(c2cn[nH]c2)=O)O)ccccc1 C(c1cccnc1C)=CC(=O)NCCCN(C(=O)CCC1CCCN(C)C1)CC N1(c2c(C#N)ccnn2)CC2C3CCC(C2C1)N(C(=O)C=Cc1ccc(Cl)s1)C3 N1(C(COCCOCCOC)=O)CC(NC(c2snc(Cl)c2Cl)=O)C(O)C1 C1(NC(C(COC)N(C)C)=O)CN(C(=O)CN2CCC(CO)CC2)CC2(CC2)C1 c1(CC(=O)NC(C(C)NC(CCC#C)=O)C)ccc(Br)cc1C#N C1(C(N(CC(C)N(C)C(c2ccnc(C(N)=O)c2)=O)C)=O)CCc2cncn2C1 Cc1ccc(C2CC2)cc1NC(=O)C(=O)N(CC(C)(O)C(F)(F)F)C N1(C(c2c(C)noc2)=O)CCC(F)(F)C(CNC(C2Cc3nnc(C)n3C2)=O)C1 c1(C(=O)NCC(C)(C2CC2)NC(=O)CSc2n[nH]c(O)n2)nc(Cl)cs1 CC1CN(C(c2cscc2C2CC2)=O)CCC1NC(c1cc2n(c1)CCC2)=O c1(OCC)c(C(=O)NCC(C)CNC(c2cnc(OC)c(C)c2)=O)cccc1F C1(C(=O)NC2(COC)CN(C(c3ccc(CC)cn3)=O)C2)CCCCC1C1CC1 CN1CCN(C(C2(C#N)CC(=O)C2)=O)CC1C(N1CC2CC2C2CC12)=O c1(-c2nc(C3(CC)CCOC3)on2)cccc(S(=O)(=O)CC(F)(F)F)c1 N1(C(c2cnc3[nH]ccc3n2)=O)CCC2CCC(C1)N2C(C1CC12CCC2)=O CN1CCCC(C)(C(=O)NCC2CC(CNC(c3cc(Cl)cs3)=O)C2)C1 C1(=O)CCC(=O)NCCCN2CCC3C(C32)N1.c1(C(=O)OC)csc(C(C)C)n1 C1(Cn2cc(C(C)OCC)nn2)N(C(C2(C(F)F)CC2)=O)CC1(C)C CCCCC(C)CCC(=O)N1CC(NC(=O)Cc2nc(C3CC3)cs2)CC(F)C1 N1(C(c2c(F)ccc(C#C)c2)=O)CCCC2(C1)CN(C(c1cc(C)c[nH]1)=O)C2 N1(C(C(CC)OC)=O)C(C)CN(C(=O)Cc2ncn(C)c2C)CC1C N1(C(C2N(C)C(=O)CC2)=O)CC2=C(C1)CN(C(=O)C(c1cccc(Br)c1)O)C2 C12(NC(C3C(C)(C)C3)=O)CCCC1N(C(c1cnc3ccnn3c1N)=O)CCC2 c1(C(=O)NC2C(CNC(CN(C(COC)=O)C)=O)CC2)cccc2nncn12 Cc1cc(Cl)cc(C)c1C(=O)NCCCCCNC(c1cccc(F)c1O)=O c1(OCC)ccc(CNC2C(CO)C2(C)C)cc1OC(=O)CC C1(C(=O)NCC(C)N(C)C(c2cc(Cl)cnn2)=O)CCCOC1c1ccccc1 CC1CN(C(C2CCCN(C)C2)=O)CC(C(=O)NC23CC(C2)C3)O1 C(=O)(CCC(=O)NCC1CCCC1NC(c1ccc(C2COC2)cc1)=O)NC Cc1cc(F)ccc1C(N1CCN(C(=O)C(C)SC(F)(F)F)CC1C1CCC1)=O C(CC)(C(=O)NC(CNC(C1(NC(N)=O)CC1)=O)C(C)C)OCC c1(NC(c2c(OC)nc(C)cc2)=O)sc2c(c1C(=O)Nc1cccnc1)CCC2 N1(C(c2ccc(N(C)C)nc2)=O)CCC(C)(C(=O)Nc2ccc(CO)cc2)CC1 C(=O)(C=C1SCC(=O)N1C)N1C2CC(NC(COC)=O)C1CC2 CC(C(C)C(=O)Nc1cncc(CO)c1)NC(c1ccncc1N)=O CC1C=C(C(=O)NCC2CN(C(c3ccc(O)nc3)=O)CC23CC3)CC1 c1(C(=O)NCC2(F)CCC(NC(c3cc(C)sc3)=O)C2)ccc(Cl)nc1O c1(C(=O)NC(CC2CN(C(C(CC=CCC)C)=O)C2)C)cc(=O)c(OC)cn1C c1(CCC(=O)N(C(CCN(C(CC2(C(=O)OC)CC2)=O)CC)C)C)cccc(F)c1 C1(NC(c2cnc(C)nc2C2CC2)=O)CC2CCC(C1)N2Cc1cnsn1 C(=O)(C(O)C1=CCCCC1)N1CC(NC(c2ccc(C#C)cn2)=O)C(O)C1 CC1(C)CC(C(=O)NCc2ccnc(CO)c2)CN1C(C1C=CC=CC=C1)=O c1(C(=O)NCC(CNC(CC(C)NC(N)=O)=O)(C)O)[nH]nc([N+](=O)[O-])c1Cl C1(COCCC(=O)ONCCCCC)CC12C1CC3CC(C1)CC2C3 C(=O)(C(C)(F)C(C)(C)F)NCCn1ncc(C(N(CCCC(C)(F)F)C)=O)c1 CCCCC(O)C(C)C(=O)N1C2CCCC1CN(C(c1nn(C)cc1C)=O)C2 c1(CN2C(C(=O)NC)CCC2C)nccc2c1[nH]c1ccccc21 c1(CC)ccc(N)c(C(=O)NC(C)CN(C(c2ccc(OC)nc2)=O)CC)c1 C(=O)(C1=CCCOCC1)N1C(C)CC(NC(C2CC3(C2)CC3(F)F)=O)C1 C1(C)(C(=O)NC2CC(NC(CCCc3ccc(SC)cc3)=O)C2)CCN(C)C1=O C(CCN=C(NCC(c1ccc(OC(F)F)cc1)C)N1CCSC(C)(C)C1)OCC C1(C(C)C)C(C(=O)NCCC2CCCC3CC23)CCN1C(c1cccc(O)n1)=O C1(COC)CCN(N2C3CCC2CC(c2nccn2C)C3)C1 N1(C(c2ccoc2C2CC2)C(=O)NCCC)CCOC(C2CCCC2)C1 C1(C(N(CCN(C)C(c2oc(C3CC3)nc2C(F)F)=O)C)=O)CC(=O)NC1(C)C CC1CCCCC1CC(=O)NC1CC(CNC(c2c[nH]nc2C(F)F)=O)C1 c1(C(=O)NC2CCN(C(c3c(OC)c[nH]n3)=O)C2)cc(C(F)(F)F)ncc1OC C1(C(=O)NCCC2(CNC(=O)CC3CC3C(F)(F)F)CC2)CCCC1F c1(CC2CCN(S(C)(=O)=O)C2)cn(CC(=O)Nc2ccn(C)n2)nn1 Cc1cnc(F)c(C(N2CCCC(CO)(NC(C3CCC(C)(C)OC3)=O)C2)=O)c1 Cc1cc(C(C)C)ccc1C(=O)NC1CCN(C(=O)CCn2cccn2)C1 CCCCCCCCN(C)C(C1(NC(=O)CC2(O)CCCCC2)CC(O)C1)=O C1(C(=O)Nc2cc(O)ncn2)CN(C(=O)CC2CCC3(CC2)CC3)CC12CC2 C1(C(N2C(COC)CC2)=O)CNC(=O)CN1C(c1cc(C)oc1C)=O C#CCC(CC(=O)NCCS(N)(=O)=O)NC(c1cncc(Cl)c1)=O c1(-c2ccc(CN(C(=O)NC(C)C)C)nc2)cc(Sc2ccccc2)ccc1F c1(Cc2cn(Cc3c(OCC)ccc(Br)c3)nn2)cc2c(cnn2C)nc1O N1(C(C(=O)NC(C)C)=O)CCC(C(C)C(N2CCC(CC(N)=O)C2)=O)C1 c1(C(N2CC(NC(C)=O)C(CC3CC3)C2)=O)cnc(O)c(F)c1 n1(CC)ncc2c(C(=O)NC(c3ccc(C(C)C)cc3)C)cc(C3CC3)nc12 C(CCC(N)C(=O)N1CCC(c2ncc(Br)cn2)CC1)OC N1(c2cc(OCC)ncn2)CC(C2CCN(C(c3cnc(Cl)cc3C)=O)CC2)C1 C1(C(=O)NCC(CCNC(c2cnc(CC(C)C)s2)=O)O)OCC2CCCC12 N(C1CCCn2ccnc21)C(C1C(C=CC)CN(C(=O)CC(C)COC)C1)=O C1(CCN(C(=O)CC2CC3(CCC3)C2)C)CCN(C(c2cscn2)=O)CC1 C12(NC(c3cnc(CC)[nH]3)=O)CC1CN(C(=O)CCc1ccccc1Br)C2 c1(C(=O)NCC2CC(C)N(C(c3ccco3)=O)C2)cnc2ccc(C#N)cn12 Cc1ccccc1C(=O)NCC1(NC(C2(C(=O)N(C)C(C)C)CC2)=O)CCCC1 CC1CC(CO)CN1C(=O)CCCCN(C(=O)Cc1ccccc1O)C Cc1nc(CC(=O)NCc2csc(CNC(c3cc(C(N)=O)cs3)=O)n2)n[nH]1 c1(C(N2CC3C(NC(c4ncc(C)cc4C)=O)(C3)C2)=O)coc2c1CCCC2 N1(C(C(=O)NCc2ccc(C3C(C)C3)o2)=O)CC2(CC(C(=O)OC)C2)C1 c1(SC)cncc(C(=O)NCCN(C(=O)C(C2CCOCC2)F)C2CC2)c1 C(C1CN(C(=O)CC2CCCC(C)(C)C2)CC1C(=O)NCC(C)N(C)C)=CC C(C(CNC(c1cnn(C(C)C)c1C)=O)C(F)(F)F)NC(CC1(C=C)CC1)=O C#CCC(CC(=O)NC1CN(C(C2CCCC2O)=O)CC1C)c1ccccc1 N1(C(Cc2nc(COC)sc2)=O)CCC(NC(C2CC(=O)NC2(C)C)=O)C(C)C1 C(=O)(CCCCCN(C)C)NCC(CNC(c1cncc(OC)n1)=O)F c1(C(=O)NCCCCCN(C(COCC(=C)C)=O)C)cncc(SC2CC2)c1 c12nnnn1CCC(=O)NC(C1CC1)C2C.N1(C(=O)N(C)C)CCC1CCF CC(C)CC(C(=O)NCC1CC(NC(=O)C=C2CCCC2)C1)n1ccnc1 N1(C(C2N(CC)CCOC2)=O)CCN(C(c2cc(C)c(O)nn2)=O)C2CCC12 c1(OC)nccnc1C(N1CCOC(CC(=O)NCCCN2CCC(O)C2)C1)=O C1(C(=O)NCC(c2nncn2C)C)CCCCN1C(=O)CCC(N)=O C1(CNC(=O)C2=C(Cl)CC2)CCCC2(CN(C(c3c[nH]c4ncccc34)=O)C2)O1 C1(C(=O)NCC(CN(C(C2(CC)COC2)=O)C)C)CC(c2ccccc2C)=NO1 C1(NC(Cc2c(C)noc2Cl)=O)CN(C(=O)CC2NC(=O)CNC2=O)C(C)(C)C1 N1(CC(=O)N(C2CCCN(C(c3cc(C)nnc3)=O)C2)C)CCCNS1(=O)=O c1(C(=O)NC23CC(NC(c4nn(C)c(C(C)(C)C)c4)=O)(C2)C3)ccc(N)c(N)n1 C1(CNC(C2(OC)CCSC2)=O)(NC(=O)C(C)c2ccsc2)CC2CCC1CC2 C1(C)(C(=O)NCCN(C)C(c2cocc2C(N)=O)=O)COC(=O)N1 c1(C(N2C(C)CC(NC(=O)C(C)(C)CF)C2)=O)ccc(Br)c(Cl)c1 C(=O)(CCCCC(=O)N(CC(O)CNC(=O)Cc1cccc(OC)c1Cl)C)OC C1(C(=O)NCCC(C)NC(Cc2c(F)ccc(C)c2)=O)CC2(CCOCC2)CO1 Cc1sc(Br)nc1C(N1CC(F)C(F)C1)C(=O)NC1CCCC1 C1(C)(CC)CC(NC(=O)COCC(F)(F)F)CN1C(c1cccc(F)c1OC)=O CCC(C)C(=O)C(=O)N1CC(N(C)C(C2CC(C3CC3)=NO2)=O)C2(CC2)C1 N1(C(CCC(CC)OC)=O)CCCN(C(c2ccnc(OC)c2Br)=O)C(C)C1 C#Cc1ccc(C(=O)NC2(CNC(=O)C(c3cc(C)cc(F)c3)C)CCC2)nc1 N1(C(Cn2nnc(C)n2)=O)CCCC(NC(=O)CCOCCN(C)C)C(F)C1 c1(OC)cncc(-c2ccc(CN3CCC(NC(=O)C(C)S)CC3)cn2)c1 Cc1nc(Cl)ccc1CC(N1CCN(C(=O)Cc2ccco2)C(COC)C1)=O C1(CCC(=O)N(CCOC)CCNC(C2CC(C)(C)C2)=O)CCCN(C)C1 c1(C(N2C(CNC(C(C)NS(C)(=O)=O)=O)COCC2)=O)cc2ccnc(Cl)c2[nH]1 Cc1ccc(C(=O)NCCC2CCCCN2C(C2CCCOCC2)=O)c(O)c1 c1(C(N2C(C(=O)NCC(C)CC3CCC3)C3CCC2C3)=O)ccc2cncn2c1 c1(CCC(=O)C(=O)N(CCC(=O)OC(C)C)CCO)ccc(Br)cc1 c1(CC)cc([N+](=O)[O-])ccc1C(=O)NC1CN(C(=O)CN(S(C)(=O)=O)C)C2CC12 C(=O)(CCCCCCN=[N+]=[N-])NC1C(OC)CN(C(c2cc(C)[nH]n2)=O)C1 Cc1cc(C(N2CC(NC(=O)Cn3cc(C4CC4)cn3)CC2(C)C)=O)c(C)n1C C1(NC(c2c(SC)nccn2)=O)CN(C(C2CC3CC2C2CC32)=O)CC1(C)C c1(C(=O)NC(CNC(C=CC(=O)OCC)=O)C)c(Cl)cc(C(F)(F)F)cc1Cl CN1CCN(C(=O)C(CCF)NC(=O)C=C2CCCCC2)CC1=O C(=O)(CCCC(F)(F)F)N(C(C)CCNC(=O)Cc1ccccn1)C C(=O)(CC1=CCCC1)NC1CN(C(CCN(CCC(C)(C)C)C)=O)C1 CC(CNC(N1CCC(C(N)=O)C1)=O)S(N)(=O)=O C1(CNC(C(c2c(C)noc2C)(C)C)=O)CN(C(=O)CN(C)C2CC2)CC1(C)C c1(-c2cnc(NCc3ccc(C)c(C(=O)O)c3)s2)ccc(F)c(C(F)(F)F)c1F Cc1ccnc(C(=O)NC23CCC(NC(=O)Cn4ccnc4C)(CC2)C3)c1F N1(C(COCCCC)=O)CCCC2(C1)C(NC(=O)C(C)=CC1CC1)CCN2C C1(NC(c2c(C(C)NC(C(C)NC(=O)C3CC3)=O)noc2)=O)CC2CCC(C1)O2 C(=O)(C1=CCCOC1)NC1CCC(CCNC(CN(C)S(N)(=O)=O)=O)C1 c1(C(N2CCC(CCNC(C(C)Cc3ccco3)=O)C2)=O)cnccc1Br C#Cc1ccc(CNc2cc(NC3CN(CCC(=O)C4CC4)C3)ncn2)cc1 N1(C(c2n(C)cc(Br)c2)=O)CCC(NC(c2ccnn2C(F)F)=O)C(F)C1 C#CCC(CC(F)F)C(=O)N1CCC(CC(C)NC(=O)C=CC2CC2)CC1 C1(CC(=O)NC(c2cncnc2)C)CCCN1C(=O)C=CC1CCOC1 c1(C(N2CC(F)(C(=O)Nc3ncn(C)c3)C2)=O)cnccc1Nc1ncc(F)cn1 C1(NC(CN(C(=O)C=CC(=O)OC(C)(C)C)C)=O)COCC1C1CC1 C1(C(NOC(CC)C)=O)CCC(O)CN1C(c1cc(C#N)cs1)=O c1(CCC)onc(C)c1C(N1CCN(C(C2CC3(C2)CC3F)=O)CC1)=O c1(CCC(N2CC(N(C(=O)CCCF)C)C(C)(C)C2)=O)nc2cccnc2[nH]1 CC1CN(C(c2csc(C3CCCO3)n2)=O)CC(C)N(C(=O)C2=NNC(=O)C2)C1 c1(C(=O)NC(CNC(Cn2ncc(CC)c2)=O)CCOC)cc(F)ccc1F c1(CC(=O)NC(CCCC)CNC(=O)CCCCOCC)ccc(OC)c(F)c1 C1(CC(C)NC(C(F)=C(C)C)=O)CCN(C(C2(CO)CC2(F)F)=O)CC1 c1(NC(CCCOC)C)ccc(NC(=O)C(O)Cc2ccccc2)cc1F C(=O)(C(C)Cn1cccn1)NCCCN(C(=O)C(C)(C)c1ccccc1)CC N1(C(c2oc(CC)c(C)c2)=O)CC2(CCN2C(C2CC=CCC2C)=O)C1 N1(C2CCN(C(Cc3c(C)noc3)=O)C2)CCN(C(C2CC(F)C2)=O)CC1 c1(C(N(CC(C)(C)NC(CCCCOCCC=C)=O)C)=O)cc2c(s1)CCC2 c1(C(N2CCC(CNC(C(C3CC3)OCC)=O)C2)=O)cc(N2CCCC2)ccn1 C#Cc1cccc(C(=O)N(C(C)CNC(=O)Cn2cc(Cl)cn2)CC)c1F [N-]=[N+]=Nc1ccccc1C(=O)NCC12CC(CO1)N(C(=O)CNC(=O)C1CC1)C2 C1(COC)CNC(C(=O)NC2CCC(C)C2)C1 Cc1scc(C(=O)NCCC2(CNC(=O)CCc3cnn(C)c3C)CC2)c1C Cc1c(NC2(C(N)=O)CCN(C(=O)COC3CCC(C)CC3)CC2)ncnc1Cl CCC(C)C(CC(=O)NCC(C)(C)OCCO)c1ccccc1 c1(C(=O)NC2CN(C(=O)CCn3cnnn3)C3CC23)cccc(Cl)c1Cl c1(C2(NC(C3C(NCC(C)O)C3)=O)CCC2)c(F)cccc1F Cn1cnn(CCC(=O)NC2COCC2n2cc(CC(O)C3CC3)nn2)c1=O c1(C(=O)OC)sc(C)cc1NC(C1(Sc2ccccc2)CC(C(=O)O)C1)=O N12CCC1(C)CC(=O)NCCCCOCC2=O.N(C)(C(C)=O)CC N1(C(CC=CCC)=O)CCC2(CCCC2NC(=O)C(F)(F)COC)CC1 N1(C(C(c2ccccc2)NCC)=O)CCCC(N(C(=O)CCN(C)CC)CC)C1 N1(C(COCC#C)=O)CCCC(COC)(NC(c2ccc(-c3cc[nH]n3)s2)=O)C1 C1(CCOC)(NC(=O)CCn2ccc(C)n2)CCN(C(C2CC23CC(O)C3)=O)C1 c1(C(=O)NCC2C(CNC(COCC=C)=O)C2)cc(Br)c2[nH]cnc2c1 C1(NC(CC(CC)C)=O)CC2CN(C(c3c(C)noc3C3CC3)=O)CC2C1 c1(C(=O)NCC2N(C(CSCCOC)=O)CCCC2C)cc(C)cc(C)c1N N1(C(CC2CCC(=O)CC2)=O)CCC(C(N2CCCCC2CF)=O)C12CC2 C(c1ccc(Cl)s1)=CC(=O)NCC1(COC)CN(C(=O)C(C)(C)c2ccsc2)C1 CC(C)CC(C(=O)NC1CC1c1ccccc1)ONC(=O)C=Cc1cnccn1 N1(C(C(CC)OC)=O)CC(NC(c2cc(OC)nn2C)=O)CC12CCC2 S(=O)(=O)(c1ccc(C(=O)O)cc1F)N1CCC(CS(N)(=O)=O)CC1 C1(NC(c2ccc(CO)s2)=O)CC(CNC(C2(O)CCSCC2)=O)C(O)C1 c1(CC(=O)NC(CNC(C(C)SCC)=O)(C)CO)csc2ccccc12 CC1CN(C(=O)CCC2CCC2)CCCN1C(=O)CCC1CCC(=O)C1 CC1CCC(NC(=O)CCc2cccc(O)n2)CN1C(=O)C1=CCCOC1 Cc1cc(CNC(=O)CC2CN(Cc3ccc(Cl)cc3F)CCO2)cc(C)c1F c1(N2CCC(C(=O)NC(C(C)C)C)CC2)nccc2cccnc12 c1(-c2ccc(C)o2)nc(C)c(C(=O)NCC2CCC(NC(=O)C(C)N(C)C)C2)s1 c1(C(=O)NCCN(C(CNS(CC)(=O)=O)=O)C(C)C)csc(S)n1 C12(C(=O)NCCN(C(CC(C)(F)F)=O)CCOC)CCOC1CCOC2 c1(CNC(C2CCCN(C3C(C)CN(C)CC3)CC2)=O)nnc2c(=O)[nH]ccn12 N(C1c2ccccc2CC1NC(=O)CC(=O)NC1CC1)C(C(C)OCC#C)=O c1(N(C)Cc2c(C)ncs2)nc2cc[nH]c2c(=NCC2CC(=O)NC(C)C2)[nH]1 CCC(C)CCC(=O)NCC1(NC(C2COCC2(C)C)=O)CCC1 C(CCCC(=O)N1CC2CC2(CNC(c2cnn(CC(F)(F)F)n2)=O)C1)OCC C1(CC)CCCC(N=c2[nH]c(=NCC(C)(C)c3cccnc3)c3[nH]ccc3[nH]2)C1 N1(C(CCC=CC)=O)CCN(C(=O)C(C)C2CCCO2)CC1CCO c1(C(=O)NC2C=CCN(C(C(CC)(F)F)=O)C2)ccnc2c1CCC2 c1(NC(N(C)CCNC(c2ccccc2Cl)=O)=O)ccc(=O)n(CCl)c1.C(C(F)(F)F)N CC1=C(C(=O)NCC(CO)NC(c2cc(C)cnc2C)=O)CCC(C)(C)C1 N1(C(CC2CCC(C)CC2)=O)CCC2(C1)CN(C(=O)CNc1nccs1)CCO2 Cc1conc1C(=O)NC1(CCNC(c2scnc2C(C)C)=O)CC1 c1(NCCNC(COCC)=O)cc(=NC2CCCN(CC)C2)[nH]c(COC)n1 CC1CN(C(c2snc(O)c2Cl)=O)CCC1NC(=O)CN1CC(=O)N(C)C1=O C#CC1(C(=O)NCCCC2(NC(c3cccn3C)=O)CC2)CCCC1 N1(C(CC(C)(C)C#N)=O)CCCCCCC1C(=O)NCCC1=CCOCC1 C1(C(=O)NC(CCCCNC(CCC#CC)=O)CO)Cc2ccccc2C1(C)C C1(OCC)CC2(C1)CC2C(=O)N(C)CC1CCN(C(C2(OC)CCOC2)=O)C1 c1(C(N(CCCNC(C2OCC(C)C2)=O)C2CC2)=O)ccnc(S)c1 c1(C(=O)Nc2scc(CN3CC(C)OCC3)n2)nccc2c1NCCC2 C1(C(=O)OC)CC2CCC(C1)N2C(c1cc(-c2csc(C)n2)cn1C)=O N1(C(C(Cn2ccnn2)NC(C=Cc2cc(C)no2)=O)=O)CCC(F)C(F)C1 C1(NC(=O)CCCc2nccs2)CC12CCC(NC(c1cnc[nH]1)=O)CC2 C1(C(N2CC(NC(C(C(=O)OC)C)=O)(CO)C2)=O)CCCN1S(=N)(=O)N(C)C C1(COC)CN(C(=O)CC2CC=CCC2)CCN1C(=O)C(C)=C1CCC1 CC(=O)CCCC(C)C(=O)N(C)CC1CCCCN1C(=O)CC1CCC(=O)N1 C=CCCCC(=O)NC(C)(CNC(=O)C(F)(F)CO)CC N1(C(c2c(C(=O)OCC)c[nH]c2)=O)CCC(C)C(CNC(c2cnnn2C)=O)C1 N1(C(CC2(C)N(C(C3N(C)C(=O)CC3)=O)CC2)=O)CCC(N=[N+]=[N-])C1 C1(C(c2cncc(OCC(F)F)c2)C(=O)O)CC(=O)C12CCC2 N1(C(C2(C)C(C)(C)C2)=O)CCC(C(=O)Nc2cncc(-n3cccn3)n2)CC1 C1(NCc2ccc(C(=O)OCC)[nH]2)CCN(Cc2ccc(Cl)nc2)CC1O C1(CN(C(=O)C=CCC(C)(C)NC(C2(C)CCCS2)=O)C)CCCC2CC12 C(C(C)C)(C(F)(F)F)NC(CC(CC)NC(=O)CNC(=O)C(C)(C)C)=O C(=O)(C(N=[N+]=[N-])C(C)C)NC(CC=C)CC(=O)N(C1CC2CC2C1)C Cc1coc(C2CC2)c1C(N1CCOC(CNC(=O)C(C#N)C2CC2)C1)=O CC(c1ccccc1)=CC(N1CC=CC(C(=O)NC(CO)CCF)C1)=O C(=O)(C1=CCC(C)CC1)NC1C(C=C)CN(C(=O)Cc2sccc2Br)C1 c1(C(=O)NCCN(C(C(c2c(C)cccc2)C)=O)C)noc2c1CC(C)CC2 C(=O)(C1=CS(=O)CCC1)N1CC2C(NC(c3c(C)cns3)=O)C2C1 Cc1cc(C(=O)NC2CCCN(C(=O)Cc3cocn3)CC2)c2c(c1)CCC2 N1(C(C(COC(C)C)NC(CSCC#C)=O)=O)CCCC2(CC2)C1 N1(C(C2C(C)(C)CCN2C(=O)CC2=CCCC2)=O)CC2(CCOCC2)C1 CC=C=CCCN=c1[nH]c(=NCCCCN(C)C2CC2)[nH]c2c1CCC2 N1(C(c2cc(CC)nn2C)=O)CCOC2CN(C(c3cnc(C(C)O)s3)=O)CC12 N1(C(c2c(C)nc(CC)s2)=O)CCC2CCC12CNC(=O)CNC(=O)NC c1(C(C(=O)NCCCC)N(C)C(c2ccc(Cl)cn2)C)ccccc1CO n1(C(N2CCC(CNC(=O)CSC3CC3)C2)=O)c(=O)oc2ccccc12 S(=O)(=O)(c1cccnc1N1CC2CSCC2C1)NC(CCCCCC)C Cc1cc(F)c(F)cc1NC(c1nnnn1C1CC1)C1CCOC1 CCCC(C)C(CC)(c1nnnn1-c1ccccc1)NCCN1CCCC1=O N1(C(CCC=CC)=O)CCN(C(C2CC2c2ccn(C)c2)=O)C(CC)C1 N1(C(C(F)OC)=O)CCc2ccccc2C1CNC(c1cncc(Cl)c1Cl)=O CC(O)CC(C)(C)CNC(=O)C(C1CC1)NC(c1cc(Cl)n[nH]1)=O C1(C(=O)OC)CN(C(=O)NC(c2c(Cl)cccc2Cl)C)CC(F)(F)C1 C1(N(C(c2ccccn2)=O)CC)CCCN(C(c2cn(CCOC)nc2C)=O)C1 Cc1cccc(CNCc2ccc(-c3c(O)cccc3F)cn2)c1Br C(=O)(CCCC(C)(C)NC(c1cn2c(n1)CCC2)=O)NC(C(C)C)CC(=O)O C(=O)(CCCCC(N)=O)N1CCC(N2CCN(C(C3CC(CC)C3)=O)CC2)C1 CN1CCCN(C(=O)CCCNC(=O)CC2C=CCC2)CC1=O CCC(C)(C)CC(=O)N(CCCNC(=O)Cc1cnn(C)c1)C1CC1 C(CNC(=O)CSC(F)(F)F)(CC(=O)N(C1CCOC1)CCO)OC N1(C(C(c2ccccn2)C)=O)CCC(Oc2ccccc2)C1 C1(CNC(c2c(OC)nsc2)=O)(NC(=O)Cc2cc(C)[nH]n2)CCC(C)(C)CC1 C(=O)(CC(C)(C)C(C)(F)F)N(CCCCCC)CCNC(=O)CC1OCCC1C CC(C(C)(O)C(=O)N1CCC(C)(NC(c2cnc(Cl)s2)=O)CC1)c1ccccc1 c1(C(=O)NC2(CNC(c3cc(CCOC)on3)=O)CC2)n[nH]c2ccc(O)cc12 N1(C(CC=CCC)=O)CC(CN(C(=O)C(CC)CCOC)C)C2(CC2)C1 n1(CCC)ncc(C(=O)NC2CCC2NC(c2ccc(=N)[nH]n2)=O)c1C C1(CNC(CCOC)=O)(OC)CCN(C(c2cccc(C3CC3(F)F)c2)=O)C1 C1(NC(c2c(C)coc2)=O)CC(C)CN(C(=O)CCc2cccc(Cl)c2)C1 C1(CC)CN(C(C2CC3COCC3C(=C(C#N)O)O2)=O)CCN1C(C)=O c1(NC(C2CCCN(CC(=C)C)C2)C)ccc2c(c1)CCCS2(=O)=O c1(C(=O)NC2C(NC(=O)CC3(O)CCC3)CCC2)cccc(N2CCOCC2)c1 c1(C(=O)NCC(CC)NC(=O)C=CCCC(C)C)ccc(N(C)C)cc1 C1(NC(C(C(C)C)c2ccccc2)=O)CCCCN(C(=O)C=Cc2ncco2)C1 CC(C(=O)N1CCC=C(CNC(C23CCC(C2)C3)=O)C1)S(N)(=O)=O C1(CNC(C=Cc2ncn(C)c2)=O)CCC2(CCN(C(c3cnc[nH]3)=O)CC2)O1 N1(C(C(CCC)(C)C)=O)CC2CCC(C1)C(NC(=O)C(C)Cc1ccccc1)C2 C1(NC(CC(C(C)(F)F)(C)C)=O)CCCC12CCN(C(C1(C)COC1)=O)CC2 CC(C)(C)C(=O)CCC(=O)N1CC=CC(C(=O)NCC2(C)CC(F)(F)C2)C1 N1(C(c2c(OC)cc(C)s2)=O)CCC2CCN(C(=O)CCCC(C)C)C2C1 C1(NC(C2(CC=C)CCOC2)=O)C=CCN(C(=O)CC2(N3CCCC3)CC2)C1 c1(-c2nc(C(=O)NCc3cccc(C4CCC4)c3)sc2)c(C(=O)O)cccc1F C12(NC(=O)Cc3c(F)cncc3Cl)CCCC1CN(C(c1cc[nH]n1)=O)C2 c1(C(=O)OC)cc(C)n(C(C)C(=O)NC(C)CCNC(=O)CN2CCC2C)n1 C1(C(=O)N)C2CCC3C(C2)CC13.C(C1=CCN(N(CCC)C)CC1)SCC=O.O=C N1(C(c2c(CC)con2)=O)CCC2(CC2NC(c2cn3ccsc3n2)=O)C1 C(=O)(C(CC)C(=O)N(C)CCN(C(=O)CCCc1ccc(C)s1)C)OCC c1(C(N2C(CNC(CC3(C=C)CC3)=O)CCCC2)=O)ccc(F)c2ncccc12 N1(c2c(C(=O)OC)nccn2)CCCC2(NC(=O)Cc3sccc3C)CC2C1 c1(OCC)cc(CC(N2CC3C(NC(C4CN(S(C)(=O)=O)C4)=O)C3C2)=O)ccn1 CCCC(C(=O)N1CCC(C(=O)NCCOCCC(=O)NC)(OC)C1)OC CC(CS(C)(=O)=O)N(C1CC1)Cc1ccccc1OCC(F)(F)F N1(C(C(CNC(c2cn(CC=C)nn2)=O)CC2CC2)=O)CC(O)CC1(C)CO c1(OC)oc(C)nc1C(=O)N(C1CCCN(C(=O)COC2(C)CCC2)C1)CCO N1(C(C=CSC)=O)CCCC12CCN(C(c1ccc(C(F)(F)F)cc1C#N)=O)C2 N1CC(CC(=O)NC2(c3nn[nH]n3)CC2)C2(CC2)C1.c1(CC)cc(C=O)ncn1 C1(NC(C(C2CC(F)(F)C2)OC)=O)CCN(C(=O)C(C)(C)C(F)F)CC1C C1(C(N(CC(C)NC(C23CC2CNC3=O)=O)CC)=O)CCC2(CCC2)C1 N1(C(C(C=C)O)=O)CC2(CCN(C(C3CCCN(Cc4cccnc4)C3)=O)C2)C1 Cc1ccc(OCC(O)CSC2CSC2)cc1 C1(CNC(C=Cc2ncn(C)c2)=O)CC2CC1CN2C(C1(CO)CC1)=O C(=O)(C1=CS(=O)CCC1)N(C)CC1CN(C(C2CC3CCC2C3)=O)C1 C1(C(=O)NC2CCC(CC(=O)NC(C#C)(C)C3CCOC3)C2)CC2(CCC2=O)C1 O=C(C1=Cc2ccccc2C1O)NCCCNC(c1ccoc1C1CC1)=O c1(OCC(N2CC(CNC(CCC#CC)=O)C3C2C3)=O)c(F)cccc1F C(=O)(C1=CCCCC1C)N1C(C(=O)NCCC(=O)OC)CCC1C(C)C c1(CCC(=O)NCCCCNC(C2C(CC)OCC2)=O)cccc(C#N)c1 c1(CNC2(c3n(CCC)nnn3)CCCC2OC)cccc(Cl)c1Br C(CCCCC(=O)NC12COC(CNC(=O)CCOCC3CCCO3)(C1)C2)OC C1(N(C(c2cc(CC)ncn2)=O)C)CC2CC1N(C(c1ccc(Cl)cc1)=O)C2 C1(CCNC(CN(C(=O)C(O)CN(C)C)C(C)C)=O)CCC(C)(C)C1 Cc1c(C(=O)N(C)CC2CCN(C(C3C(F)(F)C34CC4)=O)C2)nn(C)c1Br C1(CCC(=O)NCC(COCC(C)C)O)CCN(C(=O)CC2(O)CCC2)C1 C1(C(N2CCN(C(CS(N)(=O)=O)=O)C(CCO)C2)=O)CCOC2(CCCC2)C1 N#Cc1cn[nH]c1C(=O)NCCOC1CN(C(=O)CCCc2ccccn2)C1 C(=O)(CCC(C)(F)F)N1CCC(C(NOCCC#C)=O)C1C(C)C c1(C(=O)OCC)[nH]cc(CNC(C23CC(c4ccccc4)C2C3)=O)c1C N1(C(C(C2CN(C(C3N(C)SCC3)=O)C2)O)=O)CCC(CO)C1(C)C Cn1ncc(Cl)c1CC(=O)NC1CCCC(NC(=O)CC(=O)OC(C)(C)C)C1 c1(C(N(C)CC2CCN(C(c3cnc(O)c(F)c3)=O)C2)=O)cc2scc(Cl)c2[nH]1 C1(NC(c2nc(C(C)C)oc2)=O)CCC2CN(C(=O)C=Cc3cnc[nH]3)CC2C1 c1(C(N(CC(C)N(C(c2c(CC)nns2)=O)C)C)=O)cc(OC)cc(OC)c1 c1(C(N2CC(CCC=C)(NC(=O)CSC)C2)=O)ccc(OC(CC)CC)cc1 Cc1nc2c([nH]1)CN(C(=O)C(C)(CO)NC(=O)CCCn1ccnc1)CC2 CC12CNC(C(N3CCC(Oc4ccc(Cl)c(Cl)c4)C3)=O)(CO1)C2 C1(C(=O)NCC2C(CC(=O)NCCC(C)F)C2)CCOC1C Cc1ccc(C(C)(F)F)cc1C(=O)N(CCCNC(c1cnc(C(C)O)s1)=O)C C1(NC(c2ncnc(OC)c2F)=O)CC1C1CCCN(C(C)=O)C1 c1(C2(C(N3CC(NC(c4cccc(-n5cccc5)n4)=O)C3)=O)CC2)ccc(F)cc1 N1(C(c2c(CC)c[nH]c2)=O)CC2CC(NC(c3ccc(S(N)(=O)=O)s3)=O)C(C2)C1 CC(C)C(C(=O)NCC1CCN1C(c1cncn1C)=O)n1ncc(N)n1 C1(C(=O)NCC(CN(C(c2ccc(C)o2)=O)C)O)CC12CCC(=O)CC2 C1(NC(c2ccc(CC)[nH]2)=O)CCCCCC1C(=O)N(C1C2CCCC12)C c12cc(nn1C)CNC2=O.C1(c2ccccc2)(CC(=O)N(C)C)CCCC1 C(=O)(C(O)CC[S+](C)C)N(CCN(C(c1ccncc1OC)=O)CC)CC Cc1ccnc(C(N2CC(N(C(=O)CN3CC4CC4C3)C)C(C)(C)C2)=O)c1N C1(NC(c2c(Cl)cc(C)c(F)c2)=O)C2CC3CN(C(C4CCCCC4)=O)C1C3C2 C1(NC(C(CC)N(C)C)=O)C2CC3C1C3C2C(=O)NCCCC1(O)CCC1 c1(CC)ocnc1C(=O)N(C(C)CC(=O)NCC(CC1CC1)CO)C CCCCCCC(C)C(=O)N1CCC(C2CC2)(CNC(=O)CCC(C)(C)O)C1 C1(OC)CCCC(CC(=O)NCCCCCN(C)C(C2CC2c2cncs2)=O)C1 c1(C(C(=O)NC2(C)CN(C(=O)COCC3CCCO3)C2)OC)ccc(Cl)cc1 c1(C(=O)NC2CN(C(c3ccc(CC)s3)=O)CC2C)cccc(S(N)(=O)=O)c1 c1(CNC2OCC(NC(=O)OC(C)(C)C)C2O)c(C(F)(F)F)cccc1F c1(C(C(=O)NC(CC)C)N(C)CCc2cnn(C)c2)ccc(C(C)(F)F)cc1 C1(NC(c2c(C)nc(CO)o2)=O)CN(C(=O)COC2CCCCCC2)C(C)(C)C1 c1(C(c2ccc(Cl)cc2O)=O)c(O)cc(O)cc1O.c12ccc(cn1)c(=O)[nH]2 C(CN=c1nc(N2CCOC(c3cn[nH]c3)C2)c2c([nH]1)CCOC2)OCCC c1(C(=O)NC23CC(CNC(C4CC5C=CC4C5)=O)(C2)C3)cc2ccccc2o1 N1(C(C2CC(C)(F)C2)=O)CCC(CO)C(NC(=O)CC2OCCCO2)C1 C(N=c1nc2sccc2c(N2CCC3(CCCC3)C2)[nH]1)C1C(C)(C)CCO1 C(=O)(C(F)C(=O)NC1(C(N2CCC(O)(CN(C)C)C2)=O)CC(O)C1)OCC CCC(C)(C(=O)NC1CC(NC(c2ccc3cnoc3c2)=O)C1)C(F)F N1(C(C(c2ccc(Br)s2)OC)=O)CCN(C(=O)CC(F)F)CC1C C1(CCC)(NC(=O)CN2C(=O)CNC2=O)CCCN(C(=O)CS(N)(=O)=O)C1 C1(CNC(C=C(C)C(C)C)=O)CN(C(=O)Cn2nnc([N+](=O)[O-])n2)CC(C)(C)O1 N1(C(c2c(CC)cno2)=O)CCCC12CCN(C(C1CCCN1C(C)=O)=O)C2 CCCC(C(O)C(=O)NC1CC2(C1)CC21CCC1)NC(c1cncc(CO)c1)=O CCCCC(CC)CC(CC)(c1nnnn1C1(C)CC1)NCCN(CC)CC O=C(CCCCCCC(=O)N1CCC1)OCC(C1CC1(Cl)Cl)=O C1(CNC(C2(C)CC(=C)C2)=O)CC(C(C)C)CCN1C(=O)C=Cc1cncn1C N1(CC)CCCC(C(=O)NC2C3CCN(C(=O)C(c4cccc(OC)c4)=O)C23)C1 Cc1cc([N+](=O)[O-])ccc1OC=C(C#N)C(=O)N1CC(COC2CCCC2)C1 C1(CNC(c2c(CC)nc[nH]2)=O)CCN(C(c2ncnn2C(C)C)=O)CC1 C(CC(O)C(=O)N1CC(CC(F)F)C1)NC(c1n(CCC)ncc1)=O CN1N=C(C(=O)N2CCOC(C(=O)NC3CC3c3cnn(C)c3)CC2)CCC1=O Cc1c[nH]cc1C(=O)NC(C)CNC(c1ccn(C(C)(C)C)n1)=O c1(C(=O)NC2(CCC(=O)Nc3ccccc3CO)CCCC2)cccc(CO)n1 c1(C(N2CCN(c3cc(C)cc(Cl)n3)CC2)=O)cc(C)c(C)n(C)c1=O N1(C(C2(C)CC2(F)F)=O)CC2CN(C(c3cncs3)=O)CC2C1 C(=O)(C(C)CCCC(C)C)NC1CCN(C(C2(CC)CCCCO2)=O)CC1(C)C N1(C(c2cn(C)nc2)=O)CC(CNC(c2cnn[nH]2)=O)C2(CCOCC2)C1 N1(C(C2(OC)CCSC2)=O)CCC(C2(O)CC(NC(C3CCO3)=O)C2)CC1 c1(OC)ncc(C(=O)NC2C=CC(CNC(c3sccc3SC)=O)C2)cn1 CCCC(C(=O)N1CC(O)(C2CCCN2C(=O)C=Cc2ccco2)C1)NC(C)=O C1(C(=O)NCC2(C)CCCN(CC(=O)NC(N)=O)C2)CCC2(CCC2)CC1.O C(=O)(C(F)C(C)C)NCC1(O)CN(C(C(c2ccccc2)SCC)=O)C1 Cc1cc(C)c(CC(N2CCCC(CNC(=O)COC3COC3)CC2)=O)c(C)c1 Cc1nc2ccccc2c(C)c1C(=O)NCC(O)CNC(c1cc(O)cs1)=O C1(NC(C2CC(SC)C2)=O)CCN(C(=O)C(C)(C)S(C)(=O)=O)CC(C)(C)C1 c1(NC(N(CC#CC)C)=O)c(C)nc2ccc(Br)cn12 Cc1nc(C(N2CCOC(CCNC(C3CCN(C)C3=O)=O)C2)=O)cc(O)n1 c1(C(N2C(CNC(C3CCn4cnnc4C3)=O)CCC2)=O)ccc2scnc2c1 c1(COC)ccc2[nH]cc(CSc3cc(C)nn3C)c2c1 C1(NCC(C2CCC(N)C2)=O)CCCC2(C1)CC(O)C2 C1(C(C(=O)OC)(C)C)CCN(C(=O)CSCC(c2nn[nH]n2)c2cccs2)CC1 C(=O)(CCCCCC(C)O)NC(C1N(C(c2nc(CC)oc2C)=O)CCC1)(C)C c1(C(=O)OCC)cc(C(C(=O)NCCCSc2nccs2)N(C(C)C(C)C)C)on1 c1(C(=O)OC)cccc(NC(C2COCCN2C(=O)C#CC(=O)O)=O)n1 c1(CC(=O)OCC)cc(NC(C2CC3(CC3)CN2C(=O)CCOC)=O)ccc1Cl N1(C(c2c(C)cco2)=O)CCC2(CC1)CN(C(=O)CCC(=O)N(C)C)CCO2 c1(CN2CCC(NC(c3cc(Br)cnc3Br)=O)C2)c[nH]c2ccc(F)cc12 S(=O)(=O)(c1cccnc1NCc1cnoc1)N1CCCC(COCC)C1 n1(C(CC)(C)C)nnnc1C(c1cnc(C)s1)NCc1nc(Cl)cs1 c1(C(=O)NC(C2(O)CN(C(Cc3c(C)nsc3)=O)C2)C)ccc2sccc2c1 CC1CCc2sc(C(=O)NCC(C)(C)OCCNC(C3(C)CC(F)C3)=O)cc2C1 C1(C(=O)NCC(C)NC(=O)CCc2nncs2)COCCN1CC1CCC1 C1(C(=O)NC(C)CCN(C)C(C2(CC#N)COC2)=O)CCC(=O)N(C2CC2)C1 N1(C(CC2C(C)(C)C2)=O)CCC(CCCCNC(=O)CNS(N)(=O)=O)CC1 CCCCC(C(=O)N1CCCC(F)(C(=O)NC2CC(=O)N(C(C)C)C2)C1)N(C)C N1(C(c2cc(CC)nnc2C)=O)CCCN(C(C2CCC2C(C)(C)C)=O)C(C)C1 S(=O)(=O)(c1ccccc1F)N1CC2CN(C(c3c(C)nc(F)cc3)=O)CC2C1 C(=O)(C(CC(C)C)N1CCCCC1=O)NC1CN(C(CN(C)CC)=O)C1 CC(CCC(=O)NOCC1(F)CCC1)NC(=O)Cn1[nH]cnc1=N N1(C(c2c(CCC)nns2)=O)CC(NC(=O)C(C)CO)CC2(CCOCC2)C1 C(=O)(C(CO)C(F)(F)F)N1C(C(=O)NC2CC(O)C(O)C2)CCC(C)C1 c1(C(N2C(C)(C(=O)NC(C)CN(C)C)C=CC2)=O)cc(C#N)ccc1N C1(C)(C(N2CCC(OC)(CNC(=O)CCS(C)(=O)=O)C2)=O)CCCCCCC1 c1(CC(C(=O)OCC)NC(c2ncnc(C(F)F)c2Br)=O)ccc(F)c(Cl)c1 c1(OC)ccc(C(N2CCC2(C)C(N2CCOC3(CC3)C2)=O)=O)c(C(F)F)c1 C=CCC(C)(C)CN=c1nc2sccc2c(NCCCNC(C)=O)[nH]1 c1(C(C)NC(=O)CC2CC(CNc3cc(CO)c(C)o3)C2)cnn2ccccc12 C1(CCOC)(NC(=O)CC=C(C)C)CCN(C(C2CC2Cl)=O)CC1 C1(CNC(=O)Cc2ccc(Cl)cn2)CC2CCC(C1)N2C(=O)C(O)c1ccsc1 c1(C(=O)NCC(CC(C)C)NC(C(CCC)C)=O)c[nH]c2ccc(F)cc2c1=O c1(C(N2C(C(=O)Nc3ccc(O)c(F)c3)CCC2)=O)cccc2c(Br)cccc12 N1(C(C2CC3(CC(=O)N3)C2)=O)CC2CC(NC(c3csc([N+](=O)[O-])c3)=O)CC2C1 C1(CNC(c2n(C)c(S)nc2)=O)CC12CCN(C(=O)C(O)C(F)F)CC2 c1(C(=O)NCCCN(CCO)C(C2CCC(F)(F)CO2)=O)c(F)cc(F)cc1F n1(CC(=O)NC2CN(C(C3CC(C)(C)C3)=O)C3C2C3)cc(Cl)c(O)nc1=O c1(C(=O)NC(C2N(C(c3ccc(C#C)o3)=O)CCC2)C)cnn2c1CC(C)CC2 S(=O)(=O)(c1cc(Cl)ccc1Cl)NC(CC(=O)NC(C(=O)OC)CSC)C c1(OC)cc(Br)ccc1CN1CCOC(CNC(c2cc(F)ccc2O)=O)C1 O=CN1CCOCC1C(N1CC2CC1C2NC(=O)CCCOc1ccccc1)=O C#Cc1cc(C(N2CC(NC(=O)C(C)SC(C)C)CC(F)C2)=O)cc(Br)c1 CCCCS(=O)(=O)CC(=O)NCCN(CC(C)O)C(c1cnc(C(C)C)nc1)=O n1(CC(c2ccc(Br)cc2I)=O)ccc(=O)c([N+](=O)[O-])c1 C1(C)(NC(c2c(C)cc(C)[nH]2)=O)CCN(C(=O)C(F)CC2CCC2)CC1 Cc1c(C(N2CC(NC(=O)COCc3nccn3C)CC(F)C2)=O)cccc1F C1(OC)CS(=O)(=O)CC1C(=O)C(c1cccc(C(F)(F)F)c1Cl)C#N N1(C(C(C)C2CCOC2)=O)CCC2(NC(c3cccc(C4CC4)c3)=O)CCCC12 c1(C(N(C(CCNC(c2cn(C(C)C)nc2)=O)C)C)=O)ccc(F)cc1O N1(C(c2n(C)c(S)nc2)=O)CC2CC(N=c3ccnc(CO)[nH]3)C2C1 NS(=O)(=O)c1ccc(CCC(N2CCCC2CC(c2cccc(F)c2)O)=O)cc1 c1(C(=O)NCCCN(C(C2(Br)CC2(C)C)=O)CC)ccc2c(O)n[nH]c2c1 C1(Cc2nc(C)[nH]n2)CCCCN(C(N2CCC(C)C2)=O)C1 C1(NC(c2ncc(F)cc2F)=O)CC2CN(C(=O)Cc3cnsc3)CCN2C1=O C1(C(C)C)CCC(NC(=O)C(C2CCCO2)C2CC2)CC1 c1(C(=O)NC2CCN(C(c3cccc(OCC)c3)=O)C2)cnc(O)c2ccsc12 c1(NC(COc2ccc(OC)cc2)C=O)nc(OC(C)C)cc(C)n1.OC c1(OC)ccc(C(=O)NC(C)(C)CN(C(=O)CCS(=O)(=O)N(C)C)C)c(C)c1 Cc1ncccc1C=CC(=O)NC(C)(CNC(C1CCOC1)=O)CO C(=O)(C(O)C(F)(F)F)N1CCC(NC(C2CC(F)(F)C2(F)F)=O)C1 C12(CC(=O)NC34C(CN(C)C3)C4)CCC1CN(C(c1cscc1Cl)=O)C2 C12(C(N(CCN(C)C(c3cscc3Br)=O)C)=O)CC(F)C1C2 C(CC(F)F)(C(=O)NC1CCCC1N(C)C)N(C)C(C1CC2CCC2C1)=O c1(C(=O)NC2(C)CCN(C(c3c(CC)nn[nH]3)=O)C2)cnc2c(F)cccc2c1 C1(CC)CN(C(=O)CCSC)CC1NC(=O)C(C(C)C)c1cnn(C)c1 C1(C2CC2)(CNC(=O)C=C(Cl)Cl)CCN(C(=O)CCN2CCCS2(=O)=O)C1 c1(C(=O)OC)cc(Br)c(F)cc1N(C1CCNCC12CC2)C(=O)C(OC)OC C1CC2CCC(C1)N2C(=O)CC(C)C(C)C.c1(SC)cccnc1C(=O)NCC1CC1 c12nnnn1CCNC(C)CCNC2.C(C)(C)(C)OCCCC.C(C)(=O)OC C1(C(=O)NCCCN(C(=O)CC2CCC(=O)N2)C)CCc2nccn2C1 c1(C(=O)NCC(CC=C)NC(=O)CCCC(=O)N(C)C)cc(F)c(C)cc1F CON(CC1CC1)C(=O)C(CCOCCO)NC(=O)CC1CC(C)=NO1 C=CCCC(C)(C)C(=O)NCC(CC(=O)N1CC(CO)(CO)C1)OC c1(OC)cc(C)cc(C(=O)NCC2(NC(=O)C(O)C(C)C)CCCC2)c1O S(=O)(=O)(c1ccc2c(c1)OCC2)NC(c1csc(-c2ccccc2Cl)n1)=O C(=O)(C1Cc2ccccc21)NCC(CN(C(C(n1cc(C)nc1)(C)C)=O)C)C N1(C(C(C(CC)C)N(C)C)=O)CC2(NC(c3sccc3F)=O)CCCC2(F)C1 N1(C(COCCSC)=O)CC(C(C)NC(C2CC2(C)C)=O)C1 C#CCC(C)(CC)C(=O)NCC(CNC(=O)C=CC(=O)OC(C)(C)C)CO CC1C(NC(=O)C2=CCCO2)CC2CCC1N2c1nnco1 Cc1ccc(C(=O)NC23CCC2CN(C(C2CCCN2C(C)C)=O)C3)c(O)c1 CC1(C)OCCC1(O)C(=O)NCC1CCN(C(C2(O)CCCCCC2)=O)CC1 C1(C(N2CC(C(C(=O)NCC3(CCC=C)CC3)O)C2)=O)CC(=O)C1(C)C C1(CNC(CCC2(C)CN(C(=O)CCC(=O)C3CC3)C2)=O)CCC2(CCC2)C1 CCCC(C)CC(=O)NCC(C(=O)NCCN1CCCCCC1)N(C)C C(=O)(C1=CC2(CCOC2)C1)NCCC1(CNC(C2CCCC(C)CC2)=O)CC1 CCCC(C)(CC)C(=O)N1CC2CCCC2(C(N(C)CP(C)(C)=O)=O)C1 c1(N2CCCC(NC(C(C)Cc3ccccc3)=O)C2)ncnc2c1ccn2C C1(C)(C(=O)NC(C)COCc2ccccc2)CC=CCO1 C1(CC(C)NC(c2cncc(OC)c2C)=O)CC2CCC(C1)N2C(=O)C(F)F C1(CNC(c2cnc(C)[nH]2)=O)CN(C(=O)Cn2cc(C(=O)C3CC3)nn2)CCCO1 C1(CNC(=O)CCOC2CCC2)CCCC2CN(C(=O)CC3OCCO3)CC12 C1(NC(C(C=C)C)=O)CCOC(C(=O)NCC2(C)CCCC2O)C1 C12(CNC(C(CC)n3ccnc3)=O)CCC(C1)N(C(C1(C(C)(F)F)CCC1)=O)C2 O=C(C1COc2ccc(F)cc21)NCC1(NC(c2ccco2)=O)CCOC1 S(=O)(=O)(c1cccnc1N1CC2CCC(NS(C)(=O)=O)(C2)C1)N1C(C)SCCC1 C1(C(C)C)CN(C(c2cn(C)cn2)=O)CCC1NC(c1sccc1CN(C)C)=O C1(C(C(=O)NC(C)(C)C)OCCN(CCOCCOCC)C)CCCC1(C)C C(C)(CCC#N)(c1nnnn1C1CCC(C(N)=O)C1)NCc1cn(CCC)nc1 N1(C(c2c(C)cccn2)=O)CCC2(CCCC2C(N2C3CCC2CC(O)C3)=O)C1 n1(CC(=O)NC2C(NC(C3(OC)CCOC3)=O)CC2)c(-c2cccs2)nnc1S C1(c2nnnn2CCCF)(NCCc2ccc(OC)c(F)c2)CCCC(C#N)C1 c1(C(=O)NC2CC(C)N(C(c3cc4ccccn4c3)=O)C2)nc2c(s1)CCCC2 c1(CCC)cc(C(N2CCCC2CCNC(C23CCC2C3)=O)=O)ccn1 N1(CC)CCCN(C(C2(NC(=O)CCC3CCCC3)CC2(C)C)=O)CC1=O c1(C(=O)NC2CC(NC(c3cccc(C(N)=O)c3)=O)C2)cccc2nc(O)[nH]c12 Cc1nc2c(o1)CCN(C(C1CC1NC(c1ccc(I)c(F)c1F)=O)=O)C2 C(CCCCC(=O)NCC(C)(CO)NC(c1ccc(C(F)(F)F)c(N)c1)=O)OC N1(C(CCc2cc(C)on2)=O)CCC(C2CCCN(C(C3CC=CCC3)=O)C2)C1 C1(CNC(c2c(CC)nn(C)c2Cl)=O)COCC2(CCN(C(=O)CC(C)C)C2)O1 c1(C(N2CC(CC#N)C(C)C2)C(=O)NCCOC)cc(OC)c(C)c(OC)c1 Cc1noc(Cl)c1CC(=O)NCC(C)CNC(=O)C(c1ccccc1)OC(F)F Cc1cc(C(=O)NC(C)CC(C)NC(=O)C(C)(F)F)cn(C)c1=O N1(C(C2C(C)CCC2)=O)CCC(C2(NC(c3cccc(Cl)c3O)=O)CC2)CC1 C1(CN(C(=O)C(F)CC2CCOCC2)C)CCN(C(=O)C=CC2CCCC2)C1 c1(CC(C)C)cccc(C(N2CC(NC(=O)C(C)OC(=O)N(C)C)C2)=O)c1 C1(NC(C(C(C)O)C)=O)Cc2ccccc2C1NC(c1csc(=N)[nH]1)=O C1(N(C(c2ncoc2Br)=O)CC)CCN(C(c2cc(Cl)cnn2)=O)CC1 CCCS(=O)(=O)CC(=O)N1CCCN(C(=O)CN2CCC(C)(O)C2)CCC1 C1(CC(=O)NCC2COC(CNC(=O)C(F)(F)C3CCCC3)C2)CC2(CC2)CO1 CN1C(=O)CCC1CC(=O)NC(c1ccccc1)CNC(=O)CCCN(C)C N1(c2nc(C)cc(OC)n2)CC2(CCCC2NC(=O)CCC2CCC(=O)N2)C1 C1(NC2CCC2)CN(S(=O)(=O)CC23CC(C(F)(F)F)(CO2)C3)C2CC12 C(C(=O)NCC(C)(C)CCNC(=O)Cc1cccs1)(C(C)(C)C)N(C)C c1(C(N(CC(CC)NC(C2CCCN2C)=O)CC)=O)cc2ccsc2n1C O=C1CCCCC(C(=O)NC2(CO)CCN(C(=O)Cn3ncnn3)C2)N1 C1(NC(C(CN(C)C)O)=O)CCN(C(c2cc(O)nc(O)n2)=O)C12CC2 c1(N2CCC(N3CCN(C(C(CC)C)=O)CC3)CC2)nc(OC)c(F)c(C)n1 C1(NC(Cc2nc(C)[nH]n2)=O)CCN(C)C12CCCN(C(C1CNC(=O)N1)=O)C2 c1(CC)c[nH]c(C(N2CCCC2C(C)NC(=O)Cc2cnoc2)=O)c1 CCS(=O)(=O)CC(C)NCC(=O)OC(C)(C)C CC1CC(O)CN1C(=O)C=CCN(C(=O)CC1(C#N)CC1)C C12(CNC(=NCCOC)NCC(C)OC(F)F)COCCN1C(=O)OC2 Cc1cc(C(=O)NCC(C)(F)CNC(c2cnn(C)c(=O)c2)=O)c(C)c(C)c1 N1(C(C(C=C)(C)C)=O)CCC2(CC1)CN(C(c1onc(CC)c1C)=O)CC2CO C12(CC(=O)NCCC3CN(C(C(C4CCOC4)OCC)=O)C3)COCC(C1)C2 N1(C(C(CC)(F)F)=O)CC(C(=O)NCC(c2nccs2)C)CCC1(C)C N1(CC(=O)N(C2CCC(NC(C(C(C)C)OC)=O)CC2)C)C(=O)C(C)C(C)C1=O C1(c2cn(CC(=O)O)nn2)CN(C(c2conc2CN2CCCC2)=O)CCO1 c1(C(N2CC(CC)C(NC(c3cc(C)c[nH]3)=O)CC2)=O)c(C)ccc2nonc12 N1(C(c2cn(CCC=C)nn2)=O)CCC(C)C1CNC(c1cn(C)cn1)=O N1(C(c2cnc(C)n2-c2ccccc2)=O)CCC2(CC(NC(=O)C(C)CF)C2)C1 CCC(CC)CCCC(=O)NCC#CC(=O)NC(C)C(N)=O CC1CC(NC(=O)C2=CCSC2)CN1C(=O)CC1COC(=O)C1 C(CC(C(=O)NC(C)C(C)(C)CO)NC(=O)Cn1nc(C)cc1C)=CC O=C(O)CC1CN(CC(=O)Nc2nccn2Cc2ccccc2)c2ccc(Br)cc21 C1(C(N2CC(C(C)NC(C(=O)NCC)=O)OCC2)=O)CN2CCN1CC2C C1(CNC(Cc2cccc(SC)c2)=O)CC(C)(C)CN1c1cnc(C#N)cn1 N1(C(CCC=C)=O)CCN(C(=O)CCCc2ccc(OC)cc2)CC1CCC C12CCN(C1C1CC1)C(=O)c1cn2nn1.CC(C)C(=O)NCCC1CCCC1 N1(CCNC(=O)CCC2OCCO2)CCN(C(c2cscn2)=O)CC12CCC2 C(=O)(C(O)C(F)(F)F)NC1(C(N2CCC(C(C)(C)C)CC2)=O)CC1 C(CC(C)C(=O)N1CCN(C(=O)CN(C)C(C2(C)C=CCCC2)=O)CC1)OC C1(C(N(CC(C)(C)O)C)=O)CC12CC(NC(=O)C(N)=O)C2 CS(=O)CCC(=O)N1CCC(CCC(C)(C)NC(=O)CCc2ccncc2)CC1 C12(C(N3CC=C(C)C3)=O)C(NC(c3cccc(C#N)c3)=O)C3CC1C2C3 C1(CNC(C(CC)N(CC)CC)=O)(OCC)CCN(C(C2CC=CCC2)=O)CC1 C12(CNC(c3c(CC)ncnc3)=O)CCC(C1)N(C(=O)C(C(C)C)NC(N)=O)C2 C12(C(=O)Nc3cc(CC)cc(F)c3)CCN(C(C3(C)CNC(=O)N3)=O)CCC1C2 C(=O)(C(CO)C(C)C)N1C(Cn2cc(CCC(C)=O)nn2)CC1 CS(=O)C1CCC(NC(=O)NC2(c3ccnc(Cl)c3)CCC2)C1 C(=O)(C(F)C(C)C(F)(F)F)NC12CC(CNC(C3(C=C)CCCCC3)=O)(C1)C2 C1(C(=O)NC2C3CCN(C(C4CC(=C)C4)=O)C3C2)Cc2nn(C)cc2C(=O)N1 [N-]=[N+]=NC1(C(N2CCCC2CF)=O)CCN(C(c2cnn(CCF)n2)=O)C1 N1(C(CC(C)(C2CCC2)N(C)C)=O)CC2CCN(C(c3cc(F)c[nH]3)=O)CC12 C#CCC(C(N)=O)NC(=O)C(C1CCC1)NC(c1cc(F)c[nH]1)=O c1(CC)ccc(C(=O)NCC(F)CNC(C2CC2c2cccc(F)c2)=O)cc1N c1(OC)ccc(-c2nnc(C(=O)Nc3ccccc3)o2)cc1.N12CCCC1C2=O N1(C(C2N(CC)CCCC2)=O)CCCN(C(=O)CSCCC(C)C)C(C2CC2)C1 N1(C(C(C)NC(=O)OC)=O)CCOC2(CCN(C(=O)C(C3CC3)SC)CC2)C1 C1(CNC(=O)Cc2csc(Cl)n2)CN(C(=O)Cc2cncs2)CC2(CCC2)O1 N1(C(COCCC=C)=O)CCCCCC1C(=O)NCc1ccc(F)cc1F C(CC(C)C)(C(=O)OC)ONC(=O)C1CC1.c1(OC)nnc(C2CCC2)s1 c1(C(N(C2CN(C(C3(F)C(C)C3)=O)CC23CC3)C)=O)cccc2nc(O)oc12 C(C(=O)N1CCCO1)NC(=O)CCC1(NC(=O)CC2CC3C=CC2C3)CCC1 C1(C(=O)NC2(C#C)CCOC2)CCC(O)CN1C(c1cncs1)=O C1(NC(CCN(CCC)C)=O)CC12CCN(C(=O)C(F)(F)C(F)(F)F)CC2 C1(NC(c2ccc(C)cc2)=O)CC(C)CN(Cc2cccc(C)c2O)C1 c1(C(C(=O)N(CCN(C(=O)CC(C)F)C(C)C)C)(C)C)ccc(F)c(Cl)c1 C(=O)(CS(=O)(=O)C1CCCC1)N(C)CC1CCCCN1C(c1nc(=O)n(C)[nH]1)=O N1(C(=O)CC2CCOCC2)CC2(CCCN2c2nccc(-c3ccccc3)n2)C1 CC1(C)COCCC1C(N1CC(F)(CNC(C23COCC(C2)OC3)=O)C1)=O c1(C(=O)NCCCOCCCNC(CC2C(OCC)CC2)=O)cc(C2CC2)no1 C1(C(N(CC(C)(C)O)CC)=O)CCC2CCC1N2C(C1CC2(CC2)CO1)=O c1(OC)ccc(C(=O)NCCOCCOCCNC(C2(C)CC3CC3C2)=O)cc1C CN1CCC(C)(CNC(=O)C(Cc2cn[nH]c2)NC(=O)CC2CC2(C)C)C1 C(=O)(C(O)CC(F)(F)F)NCC(C(=O)NC1(C(COC)O)CC1)N(C)C CC(C)CC(CC(=O)N1CCOC(C2CC2)C1)NC(=O)C#CC(C)C CCCCCC(C)NC(=O)CN(C(=O)CC1CCN(C)CC1)CC N1(C(C(C)Oc2ccc(Br)nc2)=O)CCC(C(=O)O)CC12CCCC2 N1(C(c2c(C)nn[nH]2)=O)CCC(NC(c2cn3cccnc3n2)=O)C(CO)CC1 N1(C(c2cnc(NC)s2)=O)CCC2CN(C(=O)C=C(C)CN3CCOCC3)C2C1 c1(NC(N2CC(c3cc(C(F)(F)F)n[nH]3)C2)=O)sncc1Br C(C(C(=O)N(CC(F)(F)CC)C)C(C)(C)C)NC(C(CCC)NC(C)=O)=O C1(C(=O)NCC2N(C(C3(OC)CCOCC3)=O)CC2)CCC2(CC1)CC2 C1(C(N2CC(C(=O)N(C)CCN(C)C(C)=O)(CC)C2)=O)CCCC(=O)C1 c1(C(=O)NC(CNC(c2cc(OCC)no2)=O)(C)CO)ccc2nsnc2c1 N1(C(CC2(C)CCN(C(CCCCNC(C)=O)=O)C2)=O)CCCCC(CO)C1 N1(C(Cc2c(C)nccc2)=O)CC2(COC(CNC(c3ccn(C)n3)=O)C2)C1 c1(C(=O)NCCn2nnc(-c3ccccc3)n2)ccc(=O)n2c1CCC2 N1(C(CN(C2CCCC2)C(=O)C2CC2)=O)CCC(F)(F)C(F)C1.C1CO1 c1(C(=O)NC2COCCN(C(C(C)n3cnnn3)=O)C2)cccc2nccn12 CC(C)C(C#N)C(=O)N(CCC(C)NC(c1cn(C(F)(F)CO)nn1)=O)C c1(-c2ccc(C(=O)CCSC)o2)ccc(-c2nccn2CC(C)N2CC2)cc1F N1(C(C(C)=CC)=O)C2CCC1CC(NC(C1CCC1C(F)(F)F)=O)C2 C(=O)(CCCCCSC)NC(CC=C)CNC(=O)CC1CCCC(F)(F)C1 C(=O)(C(C(C)(C)C)NC(=O)CC(C)(C)C)N(CC(C)O)CC N1(C(=O)NCC(c2ccc(Br)cc2)C)CCOC(C(F)(F)F)C1 N1(C(CCCC(=O)OCC)=O)CC=C(C(C)(C)C(=O)N2CCC(CSC)C2)C1 C1(NC(c2cc(CCOC)on2)=O)C2CCC1N(C(=O)CC(C)CF)C2 c1(OC)ccc(C)c(C(=O)NC2(C)CCN(C(=O)C(F)C(C)(F)F)C2)c1 CC1CN(C(C2(O)CCCCC2)=O)CC(C)C1NC(=O)CNC(c1cccs1)=O c1(CN2CCC3(C(C(=O)NC(CC(=O)OC)C)C3)C2)cccc2[nH]ccc12 C1(CNC(CC=C)=O)CCCCCN1C(=O)C(O)Cc1cn(C)cn1 c1(CC)cc(Cl)ccc1C(=O)NC1CC(NC(=O)Cc2cn(C(C)C)nn2)C1 c1(OC)ccc(C(N2CCC(NC(c3cncn(C)c3=O)=O)C2(C)C)=O)cc1C c1(NCC(c2cn(C)nc2)O)ccc(Br)c(S(=O)(=O)NC2CCCC(CO)C2)n1 c1(OCC)ccc2cc(C(N3CC(O)(CNC(=O)C(C)C(C)(F)F)C3)=O)[nH]c2c1 N1(C(c2ccc(C)o2)=O)CCC2C1CCCN2C(c1cncnc1C)=O CCC(CCC(=O)N1CCC(CO)C(O)C1)NC(=O)CCc1cccnc1 CN1CCC(C)(C(N2CCC(C)(C(=O)NCC3C=CCCC3)C2)=O)C1 C(=O)(C1=CS(=O)CCC1)N1CCC(N(C(C(OC)C2CC2)=O)CC2CCCO2)CC1 c1(CC(C(=O)NC(C)CNC(c2ccc(Br)s2)=O)C)cccc(Cl)c1 c1(C(N2CCCN(C(C=C(CCC)C)=O)C(CO)C2)=O)cc(S(N)(=O)=O)c(C)o1 S(=O)(=O)(c1ccc([N+](=O)[O-])cc1C(F)(F)F)N(C1CCCCC1)C(C)C CN=S(C)(=O)c1ccc(C(=O)NCCCCNC(=O)CCCNC(=O)OC)cc1 C(=O)(C1=CCOCC1)NCc1ccc(C(=O)NCC2C(C)(C)CCC2)nc1 CCC(C(=O)NC12CCOC(CNC(c3cc(C)ccc3OC)=O)(C1)C2)C(C)O c1(CC=C)ccccc1C(=O)NC(C(=O)NCCCOCCCC)c1cccs1 C1(C(=O)NCC2C=CC(NC(c3c(C)coc3)=O)C2)OC(C)(C)OC1(C)C CN=c1nc(N2CCCC(C(=O)N(C)C)C2)[nH]c(=NC(C)CCn2cncn2)[nH]1 C12(NC(c3n(CC)c(O)nc3)=O)CCCC1N(C(=O)C=CCN1CCCC1)CC2 C(=O)(CS(=O)(=O)C1CCCC1)N(CCCCN(C(=O)CCCCNC(N)=O)C)C C(C(C(=O)NC(CO)C(C)C)NC(=O)CCCC1CC1)SCC C(CC(CC)C(=O)NC1CC(C)(C(=O)NCc2ncccc2C)C1)=CC N1(C(c2n(C)nnc2)=O)CCC(C)(CNC(=O)CNC(c2ccoc2)=O)C1 Cc1ccncc1-c1c[nH]nc1C(=O)Nc1cncc(F)c1 CC1CCC(NC(c2cccc(N)c2)=O)CN1C(=O)C1=CCCCC1 Cc1nc(CC(=O)NC2(CNC(c3ccc(C(N)=O)[nH]3)=O)CC2)cs1 c1(CCNC(c2n(CCCC)nnn2)c2cnc(C)s2)ccc(SC)cc1 C=CC(C)(O)CC(=O)NC(Cc1cn(-c2ccc(CC)cc2)nn1)C(=O)OCC N1(C(Cc2ccc(CC)cc2)=O)CCC(C)CC1CNC(C1C=CCCC1)=O CC(C)CC(F)(F)C(=O)NC(C)CNC(c1cccc(-c2ccccc2)c1)=O C(=O)(C(C(C)(C)C)OC)N1CCC(CCC(C)(C)NC(CS(CC)=O)=O)CC1 C1(C(=O)NC(C)CNC(=O)C(C)(C)C(N)=O)CCC(S(N)(=O)=O)CC1 CC1(CNC(=O)CC2CC(F)(F)C2)CCCN(C(=O)CCC2CC3CCC2C3)C1 c1(C(N2CCCC(C3N(C(C=CC(C)C)=O)CCCC3)C2)=O)ncc(N)cc1Cl C1(C)(C(N2C(C(N(CC(O)CO)C)=O)CCC2)=O)CC(F)(F)C1 CCCC(CCC)=CC(N1CCOC(CN(C)C(C2CCCN2C2CC2)=O)C1)=O Cc1cn2c(-c3nnc(N(C)CCC4CC4)n3C(C)CCCC(C)C)c(C)nc2s1 N1(C(C2C3CN(C(C4C(CC)CCO4)=O)C2C3)=O)CC(=O)NCC1C(N)=O C(=O)(C(F)CCC(C)(C)C)NC1(CF)CN(C(CCC(C)OC)=O)C1 c1(OC)cc2c(cc1C(=O)NC(C)CCNC(c1cnsn1)=O)CCC2 c1(SC)ccsc1C(=O)NCC1CCCN1C(=O)C(C)CO Cc1c(Cl)cnc(NC2CC3CCC2N(C(=O)CC2COCCO2)C3)c1C#N N1(C(COC)=O)CCCC2CCN(C(C3(OC(C)C)CCSCC3)=O)CC12 c1(SCCC(=O)N(C2CCN(C(=O)C(C#N)CC)C2)CC)ccc(C)cc1 C(C(=O)NCCCF)(C1=CCCCC1)N1C(C)C(C)N(C)CC1 CCC(CC(=O)N1CCC1(C)CC(N1CCCCC1CF)=O)CC(C)C c1(NC(C(=O)NC(CNC(C(C)=CC)=O)C(C)C)=O)ccc(Cl)c(F)c1 Cc1c(C(=O)NCC2CC2CC(=O)NCc2cn(C)nn2)noc1C1CC1 N1(C(C2CCC(=C)CC2)=O)CC(NC(c2cc(CCC)nc(O)c2)=O)C2(CC2)C1 CCC1(C(=O)NC2CC(NC(=O)CN3CCC3C)C2)CCCc2ccccc21 c1(SC)cc(C(=O)NC23COC(CNC(C4(C#N)CC4(C)C)=O)(C2)C3)ccn1 C1(C(=O)NC)(CNC(C(CC)SC2CCCC2)=O)CCCN1C(c1cnc(C)[nH]1)=O C1(C(=O)NCC#CCNC(C(CC(C)C)C)=O)CN(CP(C)(C)=O)C1 CC1=C(F)CN(C(C2C3CCC(C3)N2C(=O)CCc2ncccn2)=O)CC1 C(CNC(C1CC1C(F)F)=O)(CC(F)(F)F)NC(c1c(=N)[nH]cnc1)=O CC(=O)CCCC(=O)NCC1CN(Cc2nc(CC(C)C)no2)CCCO1 C1(c2cn(CC(=O)NCc3nc(Cl)ccc3Cl)nn2)CCCS(=O)(=O)C1 C1(C(N2CC(C#C)OCC2)=O)CC2CN(C(=O)CCCN(C)C)CC2C1 CC1(C)CC(NC(c2c(O)cccc2F)=O)CN(C(C2(N(C)C)CC2)=O)C1 C1(CC(=O)NC2CC(NC(=O)Cc3cc[nH]n3)C(O)C2)CCC=CCC1 C12(OC)CCC(C(=O)NCC3CCC3NC(c3oc(C4CC4)nc3C)=O)(CC1)C2 N1(C(C(=O)NCc2ccc(Br)s2)=O)CC(CO)OC2(CCC2)C1 N1(C(Cn2ncc(CNC(=O)COC)c2)=O)CC(CC)C2(CCC2)C1 c1(C(=O)NCCC2CC(NC(c3c(C)ncnc3)=O)C2)csc2cncn12 C1(NC(C2CCC(C)C2)=O)(CF)CCN(C(=O)Cn2ccccc2=O)C1 N1(C(C2C(C)(C)C(=O)C2)=O)CC(C(=O)NCCc2ccco2)CCC1(C)C c1(C(N(CC(CC)NC(=O)Cc2ccc(Cl)cc2Cl)C)=O)ccc(F)c(C)c1 Cc1cc(C(=O)NCC2CCN2C(=O)C=Cc2ccsc2)cc([N+](=O)[O-])c1O Cc1cccc2[nH]cc(CCC(=O)NCC3CC(F)(F)CN3C(C3CCC3)=O)c12 C(CCCCCC(=O)NCCc1nccs1)NC(c1ccc(C#N)[nH]1)=O c1(NCC(CNC(=O)OC(C)(C)C)OC)ccc2c(c1)C(=O)CCCC2 N1(C(C2CCN(C)C2)=O)CCCC12CCCN(C(=O)Cn1cnc([N+](=O)[O-])n1)C2 C1(CNC(C=C=C(C)C)=O)CC(F)(F)CN1C(=O)C(=O)NCC1CC1 C1(N(C(=O)C(COC)N(C)C)CCCC)CCN(C(=O)CC2CCCO2)CC1 C=C(C)C(CC(=O)NC1CCCN(C(=O)C(O)C2CCC2)C1)OCC N1(C(CCc2c(C)n[nH]c2C)=O)CC(NC(=O)COc2cnn(C)c2)CCC1C C1(NC(Cc2c(C)nc(SCC)s2)=O)COCCN(C(=O)CC2CCC(=O)O2)C1 C1(c2nc(C3CC3)no2)(COC)C=CCN1C(c1cc(OC)ncn1)=O Cc1cc(Cl)nc(Cl)c1NC(C1CCN(C(=O)C(CO)c2ccccc2)CC1)=O CCC(CCC(=O)NCCC(C)(C)C(=O)NC1CN(C)CC1(F)F)OC c1(C(N2CCCC3CCCC23)C(=O)NCC=C)ccc2c(c1)COC2(C)C N1(C2CN(C(Cn3cc(C(N(c4ccccc4)CC)=O)nn3)=O)C2)CCCS1(=O)=O N1(C(c2c(C)cccc2)=O)CCC(O)CC1C(N1CCNCC(C)C1)=O Cc1cc2c(CC(=O)NCC(C)NC(c3snnc3C3CC3)=O)csc2s1 N1(C(C2(C)CCCS2)=O)CC2(C1)CN(C(C1(O)CCC1)=O)CC2CO C1(CNC(CCCCNC(=O)CCOC2CCC2)=O)CC2CCCC2C1 C=Cn1nncc1C(=O)NC(C)CCN(C)C(c1ccc(OC(F)(F)F)cc1)=O C1(N(C(CC(CC)C)=O)C)CN(C(=O)CCc2cc(C)cs2)CCC1O C1(C)(C(=O)NCC(=C)C)CCCN(Cc2c(C)n[nH]c2C)C1 CCCC(C)C(=O)NCC(O)C(=O)NC1(CO)CC(C)C1 N1(C(c2c(C)cn(C)n2)=O)CCCOC(CNC(c2cc(Cl)c[nH]2)=O)C1 c1(C(=O)NCC(C(C)(C)C)NC(CCN(C(C)=O)C)=O)cn2c(n1)C(C)CCC2 CC1(C)CCC(CNC(c2cc(Cl)c(Cl)[nH]2)=O)N(C(c2ccc(F)cc2F)=O)C1 c1(CC(=O)NC2C3CCN(C(C=C(C)C(F)F)=O)C32)cnn2c1OCCC2 C(CCCCC(=O)NCC(C)C)n1cc(-c2c(C)n(C)nc2)nn1 N1(C(C2ON=C(CC)C2)=O)CCCCC(C(=O)NCC2(CCOC)CCC2)C1 C=CC1(C(N2CC(C(C)(C)O)(CNC(=O)CCn3ccc(C)n3)C2)=O)CCC1 N1(C(c2ccnnc2O)=O)CC2(CCN(C(=O)Cn3ccc(C4CC4)n3)CC2)C1 C1(C(N(C)CC2COCCN2C(=O)CC2CCC(=O)N2)=O)CCc2n[nH]cc2C1 N1(C(C2C3C(NC(C=C(CCC)C)=O)C4C(C3)C42)=O)CCc2cccc(C)c21 C1(CNC(=O)COC2CCCC2)CC2CCC1N2C(C1CCS1(=O)=O)=O c1(C(=O)NCC2C3CN(C(c4ccc(=N)[nH]c4)=O)CC32)ccc2nc(O)[nH]c2n1 C1(C(=O)NCCCCNC(C2CCC=CCC2)=O)CCc2nccn2CC1 c1(C(=O)NCCC2(C(N(C)CC3(C)CCCC3)=O)CCC2)sccc1C#N N1(C(N(c2ccc(Cl)cc2Cl)C)=O)CCCC12CCCN(CCO)C2=O C1(C(=O)NCC2(F)CC(NC(Cc3c(C)ccs3)=O)C2)CCc2nncn2C1 C1(CCOC)CN(C(=O)CC(F)F)CCN1C(=O)CCCCCSC N1(C(CN(C(=O)C(C)n2cccc2)C(C)=O)=O)CCN(C(c2cccs2)=O)CC1 C1(CCCC)CCCC1(c1nnnn1C1COC1)NC1(CC2CCC2)CC1 N1(C(c2ccc(CN(C)C)o2)=O)CC2CCN(C(=O)CCOCC(F)(F)F)C2C1 c1(OC)ccc(C(=O)NC(C)(C)CNC(C2(C(N)=O)CCC2)=O)nc1OC N1(C(CSCC(C)C)=O)CCCC(C2(NC(=O)C(C(C)C)n3cncn3)CC2)C1 N1(C(C(=O)NCC)COC(=O)NC(C)(C)C)CCN(C2CCNC2=O)CC1 Cc1nc(C)c(CC(=O)OC(C)(C)C)[nH]1.C12CCCN1C(=O)C(C)CNC2=O C(CCCCC(=O)N1CCOC(C)C1)N(C(C=CC(C)(C)SC)=O)C C1(C2C(=O)NC(C)CN2CCOC(C)(C)C)CCC(C)(C)CC1.C1(SC)CCC1 c1(C(N(CCN(C(=O)CN2OC(C)(C)CC2=O)C)C)=O)cncc(Cl)c1Cl c1(NC(C(C)Oc2ccccc2F)=O)nc2cc(F)c(F)cc2[nH]1 N1(C(C(CC)Br)=O)CCC2(CC1)OC(CNC(C)C(=O)OCCCl)c1ccccc12 N1(C(C2CCCC(C)C2)=O)CCCC(C)(C)C1CNCC1C2CC3C(C2)C13 O=S(=O)(c1c(F)cccc1F)NC1COC2(CCCCC2)C1 c1(C(=O)NC2(CNC(CCC(C)OC)=O)CCC2)c[nH]c2nc(F)ccc12 S(=O)(=O)(c1cnn(CCF)c1)NC(C1OCC(C)C1)(C)C N1(C(CCOCCOC)=O)CC(CNC(C2CNC(=O)O2)=O)N2CCC1C2 C(N=c1[nH]c(C(=O)NCCOCC)cs1)c1ccc(C#C)s1 C(CC(=O)NC(C)Cc1cn[nH]c1)(C1CC1)NC(CC1CC(C)C1)=O N1(c2nc(N3CCN(CC)CC3)c3c(n2)CCS3)CCc2c(C)cccc2C1 C1(C(=O)NCCSCC(=O)NC23CC(C2)C3)CCCC(CO)CC1 c1(C(=O)NC2CC(NC(c3cc(-c4nc(C)sc4)sc3)=O)C2)ncccc1Cl c1(CC(C)=O)cccnc1C(F)(F)F.c12ccc(s1)C(=O)OC2 CC1CN(C(=O)CC2CCCN2C(C23COCC2C3)=O)CC1CO c1(C(=O)NC2(CN(C)C(C3CC(O)C(F)C3)=O)CC2)cc(Br)cnc1N C=C=CC(C)C(=O)NCC(=O)NC1C(=O)NCC1O CCCCC(CNC(C1OCC1(C)C)=O)NC(c1ncccc1OC(F)F)=O C1(O)(CC(=O)NC)CCCN(CC(c2cc(F)ccc2OC)O)C1 Cc1c(C(N2CC(CO)(NC(=O)Cc3ccc(F)cc3)C2)=O)sc2nccn12 Cc1ccc(F)c(OCC(=O)N(C2CCCN(C(C3CCCCO3)=O)CC2)C)c1 c1(NC(C2CCC(NC(c3ccc(CC=C)cc3)=O)C2)=O)cc(Cl)ccc1Cl c1(C(=O)NC2(C(N3CCC(CC)CC3)=O)CC2(C)C)ncc(C)cc1F Cc1ncc(NC(=O)C(C)CNC(=O)C(C)(C)n2ccnn2)cc1C#N c1(OC)ccc2[nH]c(C(=O)NC3CC3NC(C3(C)CCS(=O)(=O)CC3)=O)cc2n1 C(C(=O)NNc1ncnc2c1oc1ccccc21)c1cc(OC)c(C)cc1 N1(C(c2ccc(C(C)C)nc2)=O)CC(NC(=O)C(C)S(C)(=O)=O)CC(F)C1 N1(C(C2CC(OCC)C2)C)CCC(NC(=O)C(N2CCOCC2)=O)CC1 c1(CNC(C(c2ccoc2)NC(C=CCN(CC)CC)=O)=O)cc(C)co1 C1(NC(=O)NCC(C2CCOCC2)F)CN2CCC1C2 Cc1c(C(=O)NC2CC(NC(=O)C(=C3CCCCC3)F)C2)ccn1C(C)C N1(C(c2c(C(C)C)con2)=O)CCN(C(=O)CCCSC(C)(C)C)CC12CC2 c1(C(C)C(=O)NCCC2CSCCN2C(C2CC(F)C2)=O)ccc(F)cc1F n1(CC2(CC)CC2)ccc(=NC(=O)CCOC2CC2)[nH]1.C1CNC(=O)N1 N1(C(Cc2n(C)ccn2)=O)CCC(CO)(NC(=O)CSc2nnnn2C)CC1 N1(C(C(N2CCSCC2)C)=O)CC(NC(=O)Cc2nc(=N)[nH][nH]2)CC12CCOC2 CCC(N=c1[nH]c(=NC2CCCC2OC)[nH]c2c1CCCCC2)c1ccn(C)n1 c1(CC)ncoc1CNC(C1CC(F)(CNC(=O)CC(C)F)C1)=O C12(CNC(CC)=O)CCC(CN(C(C3CC(=O)N(CCF)C3)=O)C1)C2 CC1CCN(C(c2cc[nH]c2)=O)CC1CNC(=O)CCC(C)(C)F c1(OCC(=O)NC2CCC(CCNC(c3ccc(F)o3)=O)C2)cccnc1 N1(CCCCCOC)C(=O)CN(C(c2cccc(C(C)(C)C)c2)C)C1=O C1(F)(CNC(C2CC3CCC2O3)=O)CCN(C(=O)CCCc2cncs2)C1 C1(CC=C)(NC(C2CC2C(C)C)=O)CCCN(C(c2ccnn2CC(C)C)=O)C1 c1(CC)onc(C(N2CCC2CC(=O)Nc2nc(C)co2)=O)c1C c1(OC(C)C(=O)NCC2CCCC2NC(C2CNC(=O)N2)=O)ccc(F)cc1Cl C1(C(N)=O)CCCN(CCC(=O)NCC2CC(F)(CNC(C3CC34CC4)=O)C2)C1 C(CC(C(C)C)NC(=O)CSCCC(F)(F)F)N(C(C(F)OC)=O)C CC(C(=O)NCCCNC(=O)CNc1ccc(C(F)(F)F)cn1)C(F)F C(C(=O)NC1CN(C(C2(C)CCCO2)=O)C1)(C(C)C)NC(=O)OC C(C(=O)NCC#CCNC(c1ccnnc1O)=O)(C(C)C)c1cnc(C)s1 C(C)(C)(C(=O)NCc1ccccc1)OCC.C1C(CC)CC2C(CC(=O)N1)C2 FC1(F)CC2CC1CC2(c1nnnn1CC(F)F)NCC12CCC(CC1)OC2 C1(O)(CC(=O)NCC(C)CNC(=O)CC2CCCC(=O)C2)CCCN(C)C1 C1(CCOC)CCN(c2ccnc(NCC(C)(C)OCCO)n2)CC1 N(C(=NCC1CCC1)NCc1cncs1)C(C)Cc1ccnn1C C12(C(N3CCC(C)(NC(C(CSC)O)=O)C3)=O)CCC(N=[N+]=[N-])C1C2 c1(-c2n(CC=C)nc(-c3ccccc3C(F)F)n2)c[nH]c2cc(C)ccc2c1=O C1(C(N2CC(C(C)NC(=O)Cn3nnc(C4CC4)n3)C2)=O)CCCN(C2CC2)C1 C1(CNC(CN(CCC)C(c2sc(F)cc2C)=O)=O)(CO)CC(C)(C)C1 c1(OC)ccc(Cl)c(CN2CC3CC(CN)C3C2)c1F CCCCCC(=O)NCC(c1ccccc1)NC(c1onc(C)c1C(F)(F)F)=O C1(NC(CN(S(CC)(=O)=O)C)=O)(COC)CN(C(=O)CCC2CCCOC2)C1 C=CC1CCCN(C(c2cnn(CCNC(c3cnccc3N(C)C)=O)c2)=O)C1 N1(C(C(CCC)C#N)=O)CCC(C)(C)C(CNC(=O)CC2(CSC)CC2)C1 N1(C(c2nnc(C)s2)C(=O)NCCC#N)CCOC2(CCCCC2)C1 N1(C(C(CC2CC2)OC)=O)CCCC(CNC(=O)COC2CC2)CC1 C1(NC(=O)C(F)=C2CCCC2)CCN(C(=O)Cc2ccccc2F)CC(O)C1 Cc1cc(C)c(C#N)c(NCCC2CCC(NC(=O)CCc3nc[nH]n3)C2)n1 N1(C(c2n(C=C)ncc2)=O)CCN(C(=O)COc2ccccc2Cl)C(CF)C1 C(C(O)CC(=O)NCc1ncccc1O)NC(=O)CCC1CC1(F)F C1(O)(CNC(CN(CC)CC)=O)CCN(C(C2(C#N)CCC2)=O)C1 C1(C(N(OC)CC2CC2(C)C)=O)CC2C=CC1N(C(=O)COCCCN(C)C)C2 C1(NC(N(C)C)=O)CCCN(N2CCN(C3CCCCC3)CC2)C1 C(=O)(C#CC1CCCCO1)N(CC(CNC(C1CC(C#C)(O)C1)=O)C)C c1(C(=O)NC2COCCC2NC(=O)C(C2CCCCC2)O)cnc2n1CCS2 c1(CC)oc(C)cc1C(=O)NC(C)C(C)NC(c1ccoc1Br)=O N1(CC(=O)NCCN(C(=O)C(C)Sc2ccccn2)CC)C(=O)CN(C)C1=O N1(C(N(c2ccc(Cl)cc2)C)=O)CCC(Nc2nc[nH]n2)CC1.C12(CC1)SC2 C1(NC(C(c2ccc(F)cc2)OC)=O)CCCC1(C)CNC(C1(Br)CC1)=O Cc1ccc(N2CCCC(CCNC(c3cc(CO)c(C)o3)=O)C2)c([N+](=O)[O-])c1 N1(C(C(C(C)C)NC(=O)OC)=O)CCCC(CCNC(c2cn[nH]c2)=O)CC1 S(=O)(=O)(c1ccc(Br)cc1NCC1(CSC)CCOC1)NCCC1(SC)CC1 N1(C(CCC(=C)Cl)=O)CC2(CC(C(=O)NC(C)(C)CC3CC3)CO2)C1 C(=O)(C1OCCc2c(O)cccc21)NC1C(NC(c2cccs2)=O)CC1 NS(=O)(=O)CC(=O)NCC1CC(F)(CNC(=O)CSC(F)(F)F)C1 C(=O)(CCCCC#Cc1ccccc1)N1C(C)CC(NC(=O)CC2CC=CC2)C1 C1(NC(C(C)C2CC2)=O)CC2CCCC(C1)N2C(=O)CS(=O)(=O)NC1CC1 c1(C(N(C2CN(C(=O)C3=COCCO3)CC23CC3)C)=O)cc(Cl)c(Cl)cc1O Cn1c(C(=O)NCCC(C)(C)CNC(=O)CCC2CC2(Cl)Cl)cnc1S c1(C(C(=O)NCC(=C)C)N(C2CC=CCC2)C)nc(-c2ccccc2)cs1 N1(C(C=CCNC(C23CCCC2C3)=O)=O)CC2COCC2(CO)C1 N1(C(c2n(C)nnc2)=O)CCN(C2CCN(C(=O)CNC(C3CCC3)=O)C2)CC1 c1(C(=O)NCC(CC=C)NC(=O)COC(F)F)cc(F)ccc1NN1CCOCC1 c1(C(C)F)ccc(C(=O)N(C)CCN(C)C(c2ncoc2Br)=O)cc1 C(=O)(CCC(C)NC(C12CC1CN(C(C1(O)CCCCC1)=O)C2)=O)OC C1(C(=O)NCCCCCC2CC2)(NC(C)=O)CCCC1C c1(N(C)C)cccc(C(O)CNC2CCC(C(=O)NC3CC3)CC2)c1 c1(C(=O)NCCCN(C)C(C23CC(F)C2C3)=O)cc(F)cc2ccncc12 c1(-c2n(CCOC)nc(COC)n2)nccc(OC(C)C)c1Br N1(C(CCC=C)=O)CC2CC1CN2C(C1CCCC(F)(F)C1)=O C1(C(=O)OC(C(CC)C)C)CC2C=CC1NC2 c1(C(C)C)cncc(C(=O)NC2CN(C(C3(O)CCSCC3)=O)CC2F)c1 N1(C(C2CN(CC)C(=O)CC2)=O)CC(CO)C2(C1)CN(C(=O)Cn1cccc1)C2 c1(N2CCC(COCC)C2)nnc(CC)n1NC(C)C(C)C C12(C(=O)NCc3n(C)nc(C(F)(F)F)c3)CCC(CC1n1cc(CO)nn1)C2 C(=O)(C(C)(O)C1CCC1)N(C)CCn1cc(C(C)(C)O)nn1 Cc1cc(C(=O)NC2CN(C(C3COCCOC3)=O)CC2C)ccn1 c1(N2CC3C(CN(CCC(=O)NCC)CC)C3C2)nc(C(C)C)nc(C)c1CC C1(NC(=O)CCCF)CCCCC12CCN(C(=O)Cc1cc(F)cc(F)c1)C2 c1(C2C(C(N(C(C)CCCO)C)=O)C2)cccc(F)c1 C(Cc1ccccc1)(C(=O)NOC(C)(C)C)NC(C(CC1CCC1)OC)=O c1(C(N2CC(N(C(Cc3cc(C)no3)=O)C)C2)=O)coc2c1CS(=O)(=O)C2 c1(OC(C(=O)NCC2CCN(C(CCCCC)=O)C2)C)ccccc1C#N Cc1cnc(NCc2c(Cl)cccc2Cl)c(S(=O)(=O)NC2CC3CCC2O3)c1 CCC(C)(F)C(=O)NCC(c1cccc(OC)c1)NC(c1nccnc1C)=O c1(C(C)C)nccc(C(=O)NCC=CCNC(C2CC(C(F)(F)F)CO2)=O)n1 C#CC(CCC)NC(=O)C(C)(C)NC(c1cc(COC)[nH]n1)=O CN=S(C)(=O)c1ccc(C(=O)NCCNC(c2ccc(O)c(C)c2)=O)cc1 Cc1c(F)ccc(Cl)c1C(N1CC2CCC2(CNC(c2ccc(C#N)s2)=O)C1)=O c1(C(=O)NC(CC(C)NC(C(C)(C)OCC)=O)C)n[nH]c2c1CCCC2 C1(NC(C2CC(=C)C2)=O)CCN(C(=O)C(C)Cc2ccc(O)cc2)CC1O Cc1cc(C(=O)NC(C)C(C)NC(c2cc(Cl)n[nH]2)=O)c(F)cc1N n1(CCOC)cc(C(=O)NC(C)CC(C)NC(c2cc(C)ns2)=O)c(C)n1 c1(NC(C(N2CCC(N)(CC)CC2)=O)=O)cc(F)cc([N+](=O)[O-])c1 c1(C(=O)NC2CC(NC(C(CCC)C)=O)C2)c(Br)ccc(F)c1OC C1(NC(c2n(C)c(S)nn2)=O)CCC2CC1CN2C(c1n[nH]cc1F)=O N1(C(c2cccc(NC(C)=O)n2)=O)Cc2cc(Cl)ccc2CC1c1ccccc1 c1(CC)c(C(=O)N(C2CCC(NC(=O)CC3(OC)CC3)CC2)C)csc1C C1(NC(CCC(=O)NCC)=O)CCN(C(=O)C(F)C(C)(C)O)C12CC2 C12(CC(=O)NC3CC3CNC(=O)COc3cccnc3)CCCC1C2 c1(NC)cncc(C(=O)NC(C(N2CCC(C(C)C#N)CC2)=O)C2CC2)c1 Cc1ccccc1OCCCC(=O)NC1CC1NC(C1(C(F)F)CCC1)=O c1(C(=O)O)ccc(F)c(CN2CCC3(CC3C(N3CCC(F)C(O)C3)=O)C2)c1 c1(C(N2CC3C(CNC(c4n[nH]c(C)c4O)=O)C3C2)=O)ccc(F)c2occc12 Cc1nc(C)c(CNC(=O)CC2COCCN2C(=O)C(O)CN(C)C)[nH]1 N1(C(c2cncc(CSC)c2)=O)CC2(C1)CN(C(=O)C(CSC)OC)CC2CO CCCCCC(C)C(=O)N(c1ccc(F)cc1Cl)C1C2CCC1CNC2 c1(C(N(CCC=C)CCOC)=O)cn2ccc(-c3cc4sccc4s3)cc2n1 N1(C(CC(C)F)=O)CCN(C(c2cc(F)ccc2Br)=O)C(CO)C1 Cc1csc2c(=NCCNC(c3c(C)nn4ccccc34)=O)[nH]cnc12 N1(C(COCCCCC)=O)CC(NC(=O)CC2CC23CC3)C(n2ccnn2)C1 C1(CNC(c2c(CC)c[nH]n2)=O)CC2(C1)CN(C(C1CCCC(OC)C1)=O)C2 Nc1ncc(-c2cn(CC3CCN3C(=O)C(C3CC3)C3CC3)nn2)cc1C(=O)O c1(C(=O)NC(C(=O)NCC(C)(C)OC)CO)ccsc1C#N C12(NC(C3C(CC)C3)=O)CCC(CC1)N(C(c1cn(C)nc1C(F)F)=O)C2 N1(C(C2(CC#C)CCCC2)=O)CCCC(CNC(C2COCCC2C)=O)C1 c1(NC(C2N(C(CCN(C)C3CC3)=O)CCSC2)=O)cccc([N+](=O)[O-])c1 C=C(C)CC(C(=O)NCCC1(C)CCOCC1)NC(C1CCCO1)=O C(=O)(C1CCCc2nn[nH]c21)NC(C1(O)CCN(c2nccc(SC)n2)C1)C CCCCCC(O)CC(=O)N1CCC(NC(C2CCC(CC)CC2)=O)C(O)C1 c1(C(N(C2CN(C(c3c(C)nc(CCC)o3)=O)C2)C)=O)cnc2ccccc2c1 C1(OC(=O)NCc2nnn(C)c2C(=O)OC2CCC2)CCCN(C(C)(C)C)CC1 CCS(=O)CC(=O)N1CCC(C2CCCN2C(c2ccoc2Br)=O)CC1 C1(CC=C)(C(=O)NCC=CCNC(=O)C(C)NC(C2CCC2)=O)CC=CC1 c1(C(=O)NCC2C(NC(Cc3c(C)noc3C)=O)CCC2)c(F)cccc1[N+](=O)[O-] C(CC(C)(C)C)(C(=O)NCCNC(=O)C(C)Cn1ccc(C)n1)OC c1(CN2CCC(CC(=O)NCc3ncc(C)nc3)C2)cc(F)cc([N+](=O)[O-])c1 C1(CC)OCCC1C(=O)NC1CCOC1C(=O)NCC1(C(N)=O)CCC1 CC(C)(C)C(CNC(c1c[nH]c(=N)s1)=O)NC(c1cn(C2CCOCC2)nn1)=O C1(C(=O)NC2CCN(CC)C2)CC2(CCN(C(C34CC(CO)(C3)C4)=O)C2)C1 c1(CO)ccnc(OC2CCC(NCC3CC3)C2)n1 C=C=C(C)CC(=O)N(CCC(=O)Nc1cccc(C(C)F)c1)CC=C C1(C#N)(C(=O)NCC2(COC)N(C(CCOCC#C)=O)CCC2)CCCCCC1 CC1(C)C(CNC(c2cnc(=N)[nH]c2)=O)CCN1C(c1coc(Br)n1)=O CC1CCc2nc(CNC(=O)C(=O)NCC(c3ccccn3)C)sc2C1 N1(C(Cc2cccc(OCC)c2)=O)CCOCC(F)(CNC(=O)C(C)C(C)C)C1 c1(CNC(Cc2c(C)noc2)=O)ccnc(C(=O)N(C)CCOCC2CC2)c1 C1(CNC(c2c(C)cns2)=O)CN(C(=O)Cc2cnns2)CC1O c1(C(=O)NC(C)C(CO)NC(C2(C)CCCO2)=O)ccnc2ccncc12 Cc1ccc2c(c1)C=C(C(=O)NCC(C)N(C)C(c1ccnnc1S)=O)CO2 N1(C(c2cnc(-c3ccccc3)nc2)=O)CC2(CC(C3CC3)=NO2)C1 c1(C(=O)Nc2ncc(-c3ccc(COC)cc3)s2)c(C)cccc1C C(CC(=O)N(C)CC1CCN(C(c2cnco2)=O)C1)(C(C)C)OCC c1(C(=O)NC(c2cn(C(c3ccccc3OC)CC)nn2)C)nccnc1N c1(CC)ccc(C(N2CCC2CNC(=O)CCc2cc(C)nn2C)=O)c(C)n1 C1(NC(C2(OC)CCC2)=O)COC2(CCCN(C(c3cc(F)ccc3C)=O)C2)C1 N(C(=NCCCN1CCCCC1)NCc1ccccc1)Cc1cnn(CC)n1 N1(C(=O)NCC2(C=C)CCC2)CC(c2ccc(C)cc2)OCC1C C1(CNC(C2CCC(F)(F)CC2)=O)CC2CCC1N2C(c1cnccn1)=O CC1=CCN(C(=O)C(Cc2ccco2)NC(=O)C(C)N2CCC2)C1 n1(CC(=O)Nc2ncc(COCCO)s2)c2ccccc2c(=O)c2ccccc12 C1(CC(=O)OC)CCN(C(=O)C=C(C)C2CC2)C(C(=O)NOC2(CC)CCC2)C1 N1(C(C(CCCC)NC(=O)CN2CCCC2C)=O)CC2CCC(C1)C(=O)O2 CC1(C)CCC(C(=O)N(CCCNC(C2CCCS2)=O)CCO)OC1 C1(C(N2CCCC(CCOC)C2)=O)C2CC(CC2F)N1C(=O)C(C)S c1(OC)cc(N2CC=CC(NC(c3cnc(F)c(C)c3)=O)C2)nc(OC)n1 CC1CC(NC(=O)CN(C)C(c2ccsc2)=O)CN1C(c1ncoc1C1CC1)=O C(=O)(CC(CNC(c1ccc(Cl)cn1)=O)C1CCC1)N(C1(CO)CCCC1)C N1(C(Cc2c(C)nn(C)c2Cl)=O)CCC2(COC(CNC(=O)C=CC(C)C)C2)C1 C1(NC(c2ccc([N+](=O)[O-])s2)=O)CC12CCN(C(=O)CC1CSCCS1)CC2 C1(C(=O)NC2C(CN(C)C)CCC2)CCC2(CC2)N1C(c1c(C#N)cnn1C)=O Cc1nccnc1C(N1CC(OC2CCN(C(C3CN(C)C(=O)N3)=O)CC2)C1)=O C(CC(=O)NN1CCCC1C(=O)Nn1cnnc1C)c1cccc(C)c1CO CN1CCN(C(=O)CC=C(Cl)Cl)CC1C(=O)NC1(CO)CCOCC1 C(C(C(=O)NCC(O)(C1CC1)C1CC1)C(C)(C)C)NC(C(C(C)C)SC)=O C1(O)(CNC(c2ccc(C3CC3(F)F)cc2)=O)CCN(C(C2CCCC2)=O)CC1 c1(C(=O)NCC=CCC(N2CCC(CC(=O)NC)C2)=O)cn(C)ccc1=O c1(OC)cccc2c1C(CNC(=O)NCC(C)(C)C(O)C(C)C)CC2 O=C(CCCC(F)(F)CO)NCC(=O)OCCN(CC(F)F)C1CC1 c1(COC(C2C=C(C)SC2)=O)ccc(OC2CC2)cc1 C=C(C)CCCC(=O)N1CCC(CCNC(c2ccc(N)c(Cl)c2)=O)CC1C C=CC1(C(=O)NCc2cc[nH]c2C(N2CCC23CN(C)C3)=O)CCOCC1 c1(CNC(CN(C(c2c(OC)ccs2)=O)C2CC2)=O)cc(O)ccc1F Cc1nn2c(c1C(=O)NC1CCCC1NC(C1(CC(F)F)CC1)=O)CCCC2 c1(N(C)C)nc(NC(C2CC2NC(=O)CC(F)(F)F)=O)cc(O)n1 c1(OC)cccc(Br)c1C(N1CCN(C(c2ccc(Br)cc2O)=O)C(CO)C1)=O CCC(CNC(C1CCCCC1OC)=O)(CC)C(=O)Nc1cnn(C(C)C)c1 c1(CC(C)C)ccc(C(N2CC(NC(=O)CC3CCCCCC3)C2)=O)cc1 CC(C)CC(CNC(c1nncn1C(C)C)=O)NC(c1scnc1C(F)(F)F)=O c1(NCCOCC(=C)C)cc(Br)ccc1S(=O)(=O)NCC=C(C)C c1(C(N2C(C)CC(NC(C(C)(C)SC)=O)C2)=O)cc2ncccc2cc1Cl c1(C(c2nnnn2CCC2CC2)NC(c2ccsc2OC)CC)cccc(C)c1 C=C(C)CCC(=O)NCC1(OC)CN(C(c2cnc(C(C)(C)C)nc2)=O)C1 c1(CN(C)CC)cn(C2(C(=O)NC(c3cccnc3)(C)C3CC3)CC2)nn1 Cc1cc(NCCOCCN(C(=O)C(=O)Nc2ncc[nH]2)C)cnc1O C1(CNC(=O)NCCCC#CC)CC12CC(CO)C2 C(CC(C)C)(C(=O)NC1CCC(NC(=O)Cc2cccc(O)c2)CC1)OC C(=O)(CCC(=O)c1ccccc1Br)NCC(C)NC(c1cccnc1)=O c1(CC)ccc(C(C)(C)C(=O)NCC2(NC(c3ccc(CO)s3)=O)CC2)cc1 c1(C(=O)NCC2C(CNC(c3cc(C)nn3C3CCC3)=O)C2)cccc(O)c1Cl C1(NC(CCC2(NC(C3CCCC(=O)C3)=O)CCC2)=O)CC2CC1C(O)C2O C(=O)(C1CCCc2ccccc21)NCC1CC(NC(C(CN(CC)CC)F)=O)C1 C1(CNC(C2C(OCC)C2C)=O)CCCN1C(c1c[nH]cc1CC)=O c1(C(=O)NC(CNC(CC2(OC)CC2)=O)(C)CO)ccc2c(c1)CCCC2=O n1(CC(=O)NC2CCCC(NC(C3(F)CC3)=O)CC2)cnc2sccc2c1=O C1(NC(C(C)SCCCC)=O)(CNC(c2ccc(F)cn2)=O)CC(F)(F)C1 N1(C(c2cc(C(CC)CC)no2)=O)CC2CC(C1)C2NC(c1cnsc1)=O C1(C#N)(NC(C(C)NC(=O)OCC2CCCC2)=O)CCN(C(C)(C)C)CC1 C1(CNC(C=C(C)c2cccs2)=O)CN(C(=O)CC2COCCN2C)CC1(C)C C1(CN(C(C2CCCCC2)C)C)CCc2cc(F)ccc2O1 C1(CCN=C(NCC(c2ccnc(C)n2)F)NC(C)C)COc2ccccc2O1 C12(CCC(=O)NC(CC)CNC(=O)C=Cc3nccs3)CCC(CC1)C2 c1(C(N(CCNC(CC2CC(CC)OCC2)=O)C)=O)cc(C#N)c2n1CCCC2 CCCCC(CNC(=O)Cn1ncn(C)c1=O)NC(c1scnc1C1CC1)=O C1(C(C)C(=O)NCC2(C(N)=O)CC2)CCN(C(c2cnn(CCF)c2)=O)C1 N1(C(CCC=CC)=O)CCC(CO)C(NC(=O)CCc2cccc(C)c2)C1 N1(C(C2C3CN(C(C4C(CCOC)C4)=O)CC32)=O)CCCC(C(N)=O)CC1 C1(CC=C)(C(=O)N(CC(C)CNC(=O)C(CC)=Cc2cn[nH]c2)C)CCOC1 C=C(C)C(CC(=O)NCC(C)(C(C)C)NC(=O)Cc1ccc(Cl)cc1)OCC C(c1nc(C)cs1)=CC(=O)N(C(CN(C(CNC(=O)OC)=O)C)C)C C(=O)(C(C)(C=C)CCOC)N1CCOCC(NC(C2(C#C)CCCC2)=O)C1 CCC(CC)C(C)C(=O)NC1CCN(c2ncnc(C(C)(C)C)n2)CC1C C1(C)(NC(C2CC(n3cc(C(C)N(CCF)C(C)C)nn3)C2)=O)COCCO1 C1(CN(C(Cc2cc(C)ns2)=O)C)CCCCN1C(=O)C(C)CC1CCCCC1 c1(NC(=O)CCc2ccc3c(c2)OCO3)cc(OC(F)(F)F)nc2ccccc12 Cn1ncc(C(F)(F)F)c1C(=O)NCC1CCC1NC(=O)CNc1nccs1 c12cc3sc(cc3s1)C(=O)NC2.c1(-n2cc(C(CC)O)nn2)cccc(CO)c1 CCC(C#N)C(=O)NCCN(C)C(c1coc(-c2ccsc2)c1)=O CC1CCN(C(C2CC(Cl)(Cl)C2)=O)CCN1C(C1CC(C)(C)CO1)=O c1(C(N2CCC(CCNC(CC(C=C)(C)O)=O)CC2)=O)ccc2ncc(C)n2c1 C(=O)(C1=CC(C)(C)C1)NCC(C)N(C)C(c1cnoc1-c1cnn(C)c1)=O C1(CC(=O)NCC(C(C)C)NC(c2c[nH]cc(Cl)c2=O)=O)NC(=O)CNC1=O C1(NC(C23C(C)OC(C)(C2)C3)=O)CCCC2CN(C(C3CCC(C)(C)C3)=O)CC12 c1(NC(C2C(C(=O)OC)C2)=O)ccc(F)c(C(=O)Nc2ccc(Br)cc2O)c1 C(C(C)(CC)C(C)O)NC(c1c(CCNC(c2cn(CC)nn2)=O)n[nH]c1)=O c1(CNC(CCC2N(C(Cc3ccc(C)nc3)=O)CCC2)=O)cnc(F)cc1C c1(C(=O)NC(C2OCCN(C(c3c(CC)ccs3)=O)C2)C)cc(F)cc(C)c1N C1(N(C)CC)CCC(C(=O)NCC2CCN2C(=O)C=CC(=O)NC2CC2)CC1 CC1CN(C(c2ccc(Cl)nc2O)=O)CCCN1C(=O)CCc1cc[nH]n1 c1(C(=O)NC2(CNC(=O)Cc3nnc(O)s3)CCC2)cc2c(F)ccc(F)c2s1 N1(C(c2nccc(C)c2)=O)C(CNC(=O)Cc2cnc(C)[nH]2)CC2CCCC12 C1(CNC(CCC(C)(C)F)=O)CCN(C(c2csc(C(F)F)n2)=O)CC1(F)F c1(C(=O)NC(CC=C)C(=O)NCC2(F)CC(CO)C2)cc(C)c(F)cn1 C1(C(=O)NCC(COC)C(C)C)CCN(C(=O)C(C)(C)CC#N)O1 c1(C(=O)OC)ncc(OC(=O)NCc2ccc(N3CCCCC3)c(F)c2)cc1Cl C(=O)(C(C)C(F)(F)C(F)F)N1CC(SC)C(NC(=O)CC(C)CN(C)C)C1 CC(O)CCCCCC(=O)NCC1CN(C(=O)C=CCO)CC1C(F)(F)F C1(NC(Cc2ccc(C)s2)=O)CCCN(CC(=O)N(C)C)C1=O N1(C(c2cc(C)no2)=O)CCOCC1CNC(c1ccc(-c2ccccc2)nc1)=O c1(C(N(C)CCNC(C2CC3CCCN(C2)C3)=O)=O)ccc(Br)c([N+](=O)[O-])c1 c1(C(=O)NC2CC(F)(CNC(c3cc(F)cc(Cl)c3)=O)C2)ccc(Cl)cc1F N1(C(C2(CC(=O)OC)CC2)=O)CCC(NC(=O)CC2CCCNC(=O)C2)C(O)C1 C(C(C)(F)C(C)(C)F)NC(C(C)(CO)NC(CC1CC(N(C)C)C1)=O)=O c1(CC(N2CC(OCCNC(CC3CCN(C)C3)=O)C2)=O)sc(O)nc1O c1(C(=O)NCC2CCC(NC(c3nc(C)n(C)c3)=O)C2)nccc2ccn(C)c12 S(=O)(=O)(c1c[nH]ccc1=NC1Cc2cscc2C1)N(CCCF)C CCC(CC)C(=O)NCC(=O)NC(C)C(C)(C)NC(=O)Cc1sccc1Cl c1(C(N2C(CC)CCC(C)C2)=O)cc2cccc(Br)c2n1C CC1CC(C(=O)NC2CN(C(c3cncc(C(N)=O)c3)=O)C2)CCO1 c1(C(=O)OC(C(C)NC)C)cnn2ccc(OC)cc12 CC1(NC(C2CC(O)CCN2C(=O)CC2CCOCC2)=O)CCCC1(F)F C12(CNC(C(C)OCC=C)=O)CCC1CN(C(=O)CCCC1CCOCC1)C2 C1(NC(CCOC(C)C)=O)C2CC1CN(C(c1n[nH]cc1[N+](=O)[O-])=O)C2 C1(NC(C2(C(=O)NC)CC2)=O)CCC(O)CN(C(c2cccc(=S)n2O)=O)C1 Cc1ccc(C=CC(N2CC(NC(=O)CC3CCCCN3C)C3(CC3)C2)=O)cc1 c1(OC(C)C)ccc(F)cc1NC(C1CC12CN(Cc1c[nH]ccc1=N)C2)=O n1(CC)nc(C(=O)NC(C)CNC(=O)C(F)(F)c2ccc(Cl)s2)ccc1=O C=CCCC(CC(C)C)C(=O)NC1(CF)CCN(C(=O)CCCCC(CC)CC)C1 C(=O)(CCCCC#N)N(CCCN(C(=O)CCN1CCCCC1)C)C C[Si](C)(C)C1(CNC(=O)C(F)C2CC(NC(C34CSCC3C4)=O)C2)CC1 c1(OC)cc(C(=O)NC2CCC2CNC(=O)C(C)(C)OC)cc(Cl)c1OC(C)C N1(C(=O)C(c2ccccc2F)O)CCC2(CO)CN(C(C34CC(C3)C4)=O)CC2C1 C=C(C)C1CN(C(C2C3CCC(C3)N2C(c2cccnn2)=O)=O)CCO1 CC(C)CC(C)C(=O)N1CCCCC1CNC(=O)CCSc1ccccc1 C1(NC(c2c[nH]nc2F)=O)CC2CC(C1)N(C(=O)C1=COCC1)C2 N1(C(CC(COC)C)=O)CC(NC(=O)CCCS(C)(=O)=O)CC2(CCOCC2)C1 C1(N(C(C(c2cncnc2)C)=O)CCO)CCN(C(c2cc(F)cs2)=O)C1 N1(C(C(CC)(C)C)=O)CC(C2CC2C(N2CCC(N(C)CC)CC2)=O)C1 C1(C2CC2)(CNC(=O)Cc2ccno2)CCN(C(=O)CC2CSCCS2)C1 N1(C(CC2CC(OC)C2)=O)CC(c2cn(CCCC(=O)O)nn2)(NS(C)(=O)=O)C1 n1(CC)cncc1CNC(=O)C(N)Cc1nc[nH]c1Br C(=O)(C1=C(C)S(=O)(=O)CC1)NC1CCC2CCN(C(c3cc(OC)ncc3)=O)C21 N1(C(CCCC(=O)NC(C)C)=O)CC(NC(c2cncc(F)c2)=O)C2(CCC2)C1 C(N=c1[nH]c(C2CC2)nc(C)c1C)C1(OC)CCC(C)C1 c1(C(=O)NCCN(C(C2C(CC)OCCC2)=O)C)c(S(C)(=O)=O)cnn1C C1(C(=O)NC(CC=C)CC)CCC2(CC2)N1C(=O)CC1CC(CC)C1 c1(OCC(N2CCC(NC(C(C(C)C)N(C)C)=O)C2)=O)ccc(S(N)(=O)=O)cc1 C1(C(N(CC(C)CNC(C2CCC(C3CC3)O2)=O)C)=O)CCCCN1C(N)=O N1(C(C(=O)Nc2ccc(OC)cc2C)CC2CCCC2)CC=CCC12CCCC2 c1(C(c2n(CC(=C)C)nnn2)NCCCC(C)O)cnc(OC)nc1 C12(C(=O)NC(CN(C(CN(CCC#C)C)=O)C)CC)CCC(C)(C1)OC2 Cc1ccnc(C(=O)NC(C2CCCC2)CNC(=O)CC2CC2(C)C)c1 C1(C(N2C(CNC(CCS(C)(=O)=O)=O)CC2)=O)CC12C1CC3CC(C1)CC2C3 Nc1cnc(C(N2CC(CNC(=O)C=CC3CC3)C3CC23)=O)cn1 c1(CC(C(=O)NCC2(F)CN(C(CC(=C=C)C)=O)C2)C)ccc([N+](=O)[O-])cc1 N1(C(C(CSC)O)=O)CC(NC(C2CN(c3ncccn3)C2)=O)C(C)C1 Cc1[nH]nc2c(C(=O)NC3CN(C(=O)COC4CCC4)CC3C3CC3)cccc12 C12(CNC(c3cc(OCC)no3)=O)CC1CN(C(c1ccc(C)cn1)=O)C2 C1(=CCNC(=O)CC2CC3CCC2O3)CCN(C(=O)Cc2cnccn2)CC1 C(=O)(CCCC(C)(C)NC(C1CC1(F)Cl)=O)N(CC(=O)NC(C)(C)C)C Cn1cc(CC(N2CCC(NC(C3CCC3)=O)C2)=O)c2ccccc12 c1(C(=O)NCC2CCCC(NC(CC=C)=O)C2)cccc2c1CCN2 c1(-c2c(OC)ncnc2)ccc(N=c2nc[nH]n3cc(Br)cc23)cc1F C1(CNC(CC(CC)(C)C)=O)CN(C(=O)CCNC(C2CCC2)=O)CC(C)(C)O1 C1(N(C(c2coc(CO)c2)=O)CC)CCCN(C(=O)Cc2cccc(C)c2)CC1 c1(NC(C2N(C(c3cc(C)sc3C)=O)CC(=O)NC2)=O)ccc(C#N)cc1O N1(C(C(CC)OC)=O)CCOCC(C)(CNC(=O)C=CC2CCCC2)C1 C1(N(CCCC)C(C2CCCN2C)=O)CCN(C(=O)C(F)=C(C)C)CC1 c1(C(=O)NC2C(N(C)C(c3ccoc3)=O)CCCC2)ccc(F)c2c1CCC2 c1(CC)nnc(C)cc1C(=O)NC(CNC(C1(F)CCS(=O)(=O)C1)=O)C1CCC1 C1(NC(C=C(C)C(F)F)=O)COC2(CCN(C(c3cc(CO)ccc3C)=O)C2)C1 C1(NC(CCc2onc(C)n2)=O)C2CC3C1C3C2C(N1CCC(C2CC2)C1)=O C12(COC)CN(C(C3C(C)OC(C)C3C)=O)C(CO)(C1)C2 C1(N2CCN(C(C(=O)NC(CC)(C)C)CCN(C)C)CC2)CC(C)(OC)C1(C)C C(=O)(CCCC(=O)NOC(C)(C)C)N(CC(CNC(C(CC)C(C)C)=O)(C)C)C c1(SCC(=O)NC2CCCN(C(C3C(C#N)C3)=O)CC2)nnc2ccccn12 Nc1cnc(C(N2CCCC2C(N2CCC(C(F)(F)F)C2)=O)=O)cn1 N1(C(c2c(C)nc(C)s2)=O)CCN(C(c2cc(C)c(N)cn2)=O)C2COCC12 CC1CN(C(c2ccc(Cn3cc(CNC(=O)C(C)O)nn3)cc2)=O)C(C)C1C c1(C(N2C(C)CC(NC(=O)Cc3cnn(C)c3)CC2)=O)csc2c(O)ccnc12 C1(NC(CC2(CNC(c3cc(C)cc(F)c3)=O)CC2)=O)CC(C)N(C)CC1C N1(C(c2c(NC)cnnc2)=O)CC(CNC(=O)C(C)NS(C)(=O)=O)C2(CCC2)C1 Cc1nc(NC(C2CCCN(C(c3cccc(O)c3)=O)CC2)=O)cnc1Cl c1(C(=O)NC2C(CC(N3CC(C#CC)C3)=O)C(O)C2)ccn(C)c(=O)c1 N1(C(C23CC(C)(C2)C3)=O)CC2(CCN(C(C34CCCC(C)(C3)OC4)=O)C2)C1 c1(C(=O)OC)ccc(NNC(=O)C(=O)OCC(N)=O)nc1 N1(C(c2n(C(C)C)cnc2)=O)CCC(CCN(C(=O)CCC2CC2)C)CC1 C1(CNC(C2(C#C)CC2)=O)C(C)CCCN1C(=O)CC1(O)CCCCC1 N1(C(=O)C(F)C2CCCC2)CC(C2CCN(C(C3CCC(C)(C)O3)=O)CC2)C1 c1(OCCC(=O)NCC(CC=C)NC(c2ccncc2C)=O)ccccc1O C(=O)(CCCCCO)NCC(C)N(C(=O)C(O)CCc1ccccc1)C c1(C(N2CCN(C(C3=NNC(=O)C3)=O)CC2CCO)=O)cc2n(n1)CCNC2=O C1(CN(C(=O)C(C)C2CCC2)CC)CCN(C(c2cc(Cl)n[nH]2)=O)CC1 c1(C(N(CCCCNC(C2CC2(C)C)=O)C)=O)cc2c(F)ccc(Br)c2[nH]1 C(=O)(CC(CC)CCCC)N(C1C(N(C(CCC=CCC=C)=O)C)CCCC1)C C12(C(N(CCC(C)NC(C3CCOC3C)=O)C)=O)CCN(CC1)S(=O)(=O)C2 N1(C(CCc2n[nH]c(=N)s2)=O)CCC2C(C1)CN2C(c1c[nH]c2ccccc12)=O N1(C(C2(OCC)CC2)=O)CCC(NC(c2cc(O)ncc2Br)=O)C(CO)C1 n1(CC)nc(C(=O)NC(C)C(C)NC(c2[nH]ccc2C)=O)c(=O)c2ccccc12 N1(C(C(CC)(CNC(C2CC2Cl)=O)CC)=O)CCOCC2(CCC2)C1 C(c1nc(C)cs1)=CC(=O)N(C1CCN(C(C2OCCC2C(C)C)=O)C1)CCC Cc1ccc(C(=O)NCC23CCC(CC2)CN3C(C2(C)CCOC2)=O)c(F)c1F N1(Cc2cnc(N(C)C)nc2)CCC(C(=O)Nc2ncc(C(F)(F)F)cn2)C(O)C1 c1(C(N2CCC(CCOC)(NC(C(C=C)C)=O)C2)=O)cc(F)cc(F)c1 C1(C(N(C(CCCC)C)C)=O)CC2(CC(NC(C3(CCF)CCC3)=O)C2)C1 C1(NC(C(C(=O)OCC)=O)c2ccccc2)CC2CCCCN2C1=O c1(C(N2CCN(C)CC2CNC(C2CC3(C2)CC3F)=O)=O)cnc2n1CCOC2 c1(CC)ccc(C(=O)NCC(C2CC2)NC(c2ccc(C(F)(F)F)nn2)=O)cc1 CCCCC(CNCC(F)(F)C(C)C)CC c1(CC)ccccc1C(=O)NC(C)C(C)NC(=O)C(CC)Oc1ccccc1C N1(C(CCCC(=O)N(C)C)=O)CC2(NC(=O)CC3CC(C)(C)C3)CCC1CC2 c1(C(N(CCCNC(=O)C=CI)CC)=O)cccc(O)c1C CC1CN(C(=O)CC2CC3CCC2O3)CC1CNC(c1cncc(O)c1)=O c1(C(N(CC(CN(C(COCCSC)=O)C)O)C)=O)[nH]nc2c(=O)n(C)cnc12 C1(CCNC(C2(COC)COC2)=O)CCC(NC(=O)CC=C(C)C)C1 C1(CCO)(NC(C(C)O)=O)CN(C(=O)CCCNC(N)=O)C1 C#Cc1cc(C(N2CCCOC(CNC(=O)CC3(COC)CC3)C2)=O)ccc1Cl C1(C(=O)NC(CNC(c2c(C)ncn2O)=O)C)C2CCC1(C)C2(C)C Cc1cnc(C(=O)N(C)CC2CN(C(=O)C(F)CC3CC3)CCO2)cn1 CC1=C(C(=O)N2CCCC2CCNC(c2ccc(C)s2)=O)CCO1 CCC(C)(C)CC(=O)NCC1(F)CC(NC(c2cc3scnc3[nH]2)=O)C1 c1(SC)cc(C(N2CC3CC3(CNC(c3ccc(CO)o3)=O)C2)=O)c(C)o1 O=C(CC1=CCN(C(=O)Cn2cccc2)CC1)NC1CCC2(CCC2)C1 C#Cc1cccc(CC(=O)N(CC(C)(C)NC(=O)CC2CC(F)C2)C)c1 Cc1n[nH]c(C)c1CC(C)C(=O)NCCCC(C)NC(=O)C=CC(C)(C)C Cc1cc(C)c(C(=O)NCC2CC(O)CN2C(=O)Cn2ccnn2)c(O)n1 c1(C(=O)NCC(CC)OC)ccc2n[nH]cc2c1.C1(=O)C(CC)N1CC C=CCCN=C(N)NCC.N1(CCc2ccnc(N3CCCC3)c2)CCC(C)CC1 Cc1nscc1-c1noc(CNC(=O)C(COCc2ccccc2)N(C)C)n1 c1(C(=O)NC2CN(C(C3CC3c3cncnc3)=O)C2)ccc(Cl)cc1F c1(C(=O)NC(C)(C)CNC(C2CC2(C)Br)=O)ccc(O)nc1 N#Cc1ncc(C(=O)NC(CNC(c2cc(-c3cnccn3)[nH]n2)=O)CO)s1 Cc1cc(C)c(C(N2CC(O)CC2CNC(c2nn(C)cc2Cl)=O)=O)cn1 CC(CCCCO)NC(=O)CCN(C(=O)C(C)n1cncn1)C N12CCC(C(C)C1)NCC2=O.c1(OC)cc(C=Cc2ccccc2)sn1 N1(C(CC=C)=O)CC(OC)CC1C(=O)Nc1sc(C)nc1-c1ccc(OC)cc1 C=C(C)CC(C)C(=O)NCCC1(O)CCCN(C(c2ncn(C)n2)=O)C1 c1(C(=O)OC)cccc(CN2CCSCC2C(=O)Nc2cncnc2O)n1 c1(CC(=O)NC23CC(NC(=O)CCc4cc(Cl)no4)(C2)C3)ccc(F)cc1F Cc1ccc(N(C)C(c2occc2CNC(=O)C(C2CCCCC2)C)=O)cc1C C(C(C)(O)CCCO)c1cn(C2CCN(CC)C2=O)nn1 c1(C(N(CCNC(C(C(C)C)NC(=O)OC)=O)C)=O)ccc2c(c1)COC2(C)C C1(C(N(c2cn[nH]c2)C)=O)C2CN(C(=O)CCCn3ccnn3)CC12 CN1CC(NC(C2CN(C(=O)CCc3ccccc3)CCN2C)=O)CCC1=O C(=O)(CS(=O)(=O)C(C)C)N1C(C(=O)NC(CCOC)COC)CCOCC1 N1(C(C2C(C)(C)CCO2)=O)CCC2(CC1)CC(NC(C1(F)CCC1)=O)CO2 C1(NC(C(C)=C2CC2)=O)CN(C(=O)CCCc2ccc(O)cc2)CC1C C1(NC(c2nn[nH]c2C(F)(F)F)=O)CCCC(NC(c2nsnc2O)=O)C1 C1(NC(C(C)N2CCC2CN(C(=O)CCn2cncn2)C2CC2)=O)CCCCC1 C1(C)(CNC(C(F)(F)C2(OC)CCC2)=O)CCCN(C(=O)CN(C)C(C)C)C1 C(=O)(C(O)CCS(C)=O)N1CCCN(C(c2c(C)ncs2)=O)CC1.C1C(=O)N1CCC(C)C c1(C(=O)NC(C(C)C)CNC(=O)C=Cc2ccco2)ccc(S(N)(=O)=O)c(F)c1 C(CCO)(C(F)(F)F)NC(C(C1CCCN(C(C23CC(F)(C2)C3)=O)C1)(C)C)=O N1(C(c2ccc(SC)o2)=O)CCOCC(F)(CNC(C2CCCOCC2)=O)C1 N1(S(CCC)(=O)=O)CCCC(C(=O)N(C)CCN(C(=O)C(C)OCC)C(C)C)C1 C(=O)(C(CC)(CC)C(C)C)N1CCC(CNC(C2(CCC=C)CC2)=O)CC1 c1(CCOC(CN2CCC(OC(C)(C)C)CC2=O)=O)cc(F)c(Cl)cc1Cl CCC(CCCC(=O)N1CC(CCO)C1)NC(c1csc(C)n1)=O N1(C(CN2C(C)CC2)=O)CCC2(CCCN(C(C3CC(O)C3)=O)C2)C1 C1(CC=C)(NC(=O)CNc2ncccn2)CCCN(C(C2(C#N)CC2(C)C)=O)C1 C1(c2cn(CCN(CC)CC)nn2)CCCCN1C(c1ccc(O)nn1)=O N1(C(C(C)NC(C)=O)=O)CC2(CCOCC2)CC1CNC(c1c(C)ncn1O)=O N1(C(Cn2c(C)ccc2C)=O)CCC=C(C(=O)N2CCCC(CC(C)C)C2)C1 c1(OC)ccc(CC(CNC(=O)C(N)Cc2cccc(Br)c2)CO)cc1Br CCCCS(=O)(=O)CC(=O)NCCN(C(c1csc(CSCOC)c1)=O)CC1CC1 C(=O)(C(C)C(O)C(C)C)NCC1C2N(C(C(c3cccc(C)c3)=O)=O)C(CC2)C1 C=CC(C)(O)CC(=O)NCC1(NC(=O)CCc2csc(C)n2)CCCCC1C C1(C)(C(=O)NC2CN(C(C(C)Cc3ccc(F)cc3)=O)C2)COCC1(F)F C1(C(=O)NC2CCCC2C(N)=O)(CC)CCN(C(=O)CC23CCCC2C3)CC1 N#CC1(CNC(=O)C(O)CCCNC(=O)CC2CCCSC2)CCCCC1 N1(C(C(CC)OC)=O)CC(NC(c2ccc(NC=O)cc2)=O)C2(CC2)C1 c1(C(C)NC(=O)COc2ccon2)ccc(CNC(=O)C(C)CC2CCC2)cc1 c1(C(C)C(=O)OCC(c2ccncc2)=O)cc(F)cc(F)c1 C(=O)(C1CCCc2nc[nH]c21)N1CCCCC(CNC(=O)CC2CS(=O)(=O)C2)C1 c1(C(N(C2CCCC(NC(=O)CCCCC#N)C2)C)=O)ccc2nccn2n1 N1(C(CCNC(N)=O)=O)CCC2CC1CN2C(=O)C=Cc1ccc(Br)cc1 C1(CN(CCCC)C)CCN(C(c2ccc(F)cc2)C(=O)NC2(C)CC2)CC1 c1(C(=O)NC2CC(NC(c3c(C)cn(C)n3)=O)C2)ccc2c(c1)CCC(C)N2 Cc1sc(O)nc1C(=O)N(CC(=O)NCC1CCC(=O)NC1)C(C)C C1(NC(c2cn(C=C)nc2)c2nnnn2CC(=C)C)CCCCN(C)C1=O c1(C(N2C(CNC(CN(CCC)C)=O)CC(O)C2)=O)cc2c(s1)CCS(=O)(=O)C2 CCC(CNC(=S)NCC(Br)=C(C)C)C(C)C c1(CC(=O)NCc2cn(CC3CNC(=O)O3)nn2)n[nH]cc1C(=O)OC(C)(C)C N#Cc1cn[nH]c1C(=O)NC1CCC1NC(c1ccc(C(F)F)s1)=O c1(NC2CC(F)(CNC(C3CCCCC3)=O)C2)ncc2cccnc2n1 C#CCC(C)(C(=O)N1Cc2c[nH]nc2C1)NC(=O)Cc1ccoc1 c1(CC(C2(C)CCOC2)NC(CC)(C)c2nn[nH]n2)ccc(F)cc1 c1(C2C(C(=O)NCCN(C(=O)CC3(C)CCCO3)CC)C2)ccc(Cl)cc1F c1(C(N2CCCC(CNC(C(C3CC3)OC)=O)CC2)=O)ccc2[nH]ccc2c1 N1(C(C2C(CC)CCO2)=O)CC(C(=O)Nc2cnc(C)nc2C)C(C)(C)C1 CC(C)(C)C(C(=O)NOC1CCCCC1)NC(=O)CCCCC(N)=O C1(N(C(c2ccc(OC(C)C)nn2)=O)C)CCCN(C(=O)C(C)(C)C2CC2)CC1 C1(NC(CC(C)C(F)F)=O)CN(C(C2CCS(=O)CC2)=O)C2(CCCC2)C1 c1(C(=O)NC(C2CCCC2)CC)cc(C(F)F)[nH]n1 C1(C(=O)NCc2c(C(=O)NC(CC#C)C(=O)NC)scc2)CC2(CCC2=O)C1 Cc1cnc(C)c(NC(C2CCN(C(=O)C(C)OCC(C)C)C23CC3)=O)c1 N(C1CC2(CN(C(=O)C(O)CSC)C2)n2ccnc21)C(C1(C=C)CCOCC1)=O S(=O)(=O)(c1ccc(Cl)nc1)NC1CN(C(c2c(C)ccc(Br)c2)=O)CC1(F)F Cc1nnc(C(C(=O)Nc2ccccc2)N(C2(C)N(C(C)C)CC2)C)s1 C1(SCC)CC(C(=O)NCc2c(OCCO)cccc2Br)CC(=O)N1 CC(CS(C)(=O)=O)C(=O)NCC(O)CCNC(c1ccc2nccn2c1)=O CCN=c1cc(C(=O)NC(COC)CNC(=O)C(C)CC2CCC2)cc[nH]1 C(=O)(C1=NOC(C)C1C)NCC(C)CNC(C1Cc2ccccc2C1)=O C12(NC(Cc3cc(C)[nH]n3)=O)CC1CN(C(C1CCS(=O)(=O)C1)=O)C2 Cc1cc(C(=O)N(CC(C)NC(=O)CC(C)(C)C2CC2)C)c(F)c(Br)c1 N1(C(CC(=C=C)C)=O)CCC(NC(c2cccc(P(C)(C)=O)c2)=O)C2(CCC2)C1 c1(C(=O)NC2CC3(CN(C(C(CC=C)CC)=O)C3)C2)cc2cc(Cl)cc(C)c2[nH]1 C1(CNC(C(CC#C)O)=O)CN(C(=O)Cc2ccccc2C)CCC12CCC2 C1(C(=O)NCC2C(OCC)CC2)CCCCCCN1C(c1cnnc(C)c1C)=O Cc1ncc(C=CC(=O)NC2CC2CNC(c2cnc(N(C)C)o2)=O)s1 C12(CCNC(=O)CC(O)C3CCC3)CCC(C1)N(C(=O)Cc1cncs1)C2 c1(C(=O)NC(C(C)(C)NC(C(C)=C2CC2)=O)C)ccc(N)c(OCCO)c1 C12(C(N3CC(C(C)NC(C(C)=CC)=O)C3)=O)CCCC(CO1)C2 CC(C)CC(C(=O)N1CCN(C(c2ncccc2O)=O)CC1)N1CCCC1=O O(N1CCC(NC(=O)CCN(C(c2ccc(C)cc2)=O)C2CC2)CC1)CC c1(C(=O)NCC2(F)CCCN(C(C3(CCF)CCC3)=O)C2)cc(F)c(Cl)cc1Cl Cc1cc(Br)c([N+](=O)[O-])cc1C(N1CC(NC(c2[nH]ccc2C)=O)C(F)C1)=O c1(CNC(CC(C)NC(CC2(C(=O)OC)CC2)=O)C)nccc(-n2cccn2)n1 Cc1cc(NC(=O)C2=CCN(C(C3CC4CC4C3)=O)CC2)cc(C)c1O c1(CC(=O)N(CC(C)NC(=O)CCNC(C)=O)CC)cc(SCCCC)c[nH]1 c1(C(N(C2CC(NC(c3cc(C)ncc3)=O)C2)C)=O)ccc(F)cc1Cl CC1(C)CC(CCNC(C2CCOC2CNC(C2(C)CCC(=O)C2)=O)=O)CO1 C(CCC(=O)NC1(C(=O)O)CC=CC1)NC(C(C)=C(CC)C)=O c1(OC)ccc(Br)c(CN2CCC3(CC3C(=O)NCC(O)CO)C2)c1 c1(C(N2CCC(NC(C3CCN(C(C)=O)C3)=O)C23CC3)=O)ccnc2[nH]nnc12 C#Cc1ccc(F)cc1C(N1CCC(NC(c2cnc(F)c(F)c2)=O)C1)=O N1(C(c2c(OC)cc(Br)cc2)=O)CC2CCN(C(c3cc4ncccn4n3)=O)C2C1 C(=O)(C(C)(C)CCCO)NC(C)CNC(c1c(C)nc(C2CC2)o1)=O C1(CNC(CC(C(C)C)O)=O)CC2CCC(C1)N2C(C1CC(C)(C)C1)=O c1(C(c2nnnn2C2COC2)NCC(C)F)cc(Br)oc1Br c1(CNC(C2CCC(CC(=O)OC)CC2)=O)cc(OC)c(OC)c(OC)c1 C1(CN(CCCC2OCCO2)CC)CC(O)C1(C)C Cc1[nH]c(=N)ccc1CN1CCC2(COC2)C1 N1(C(CN2CC(C)(C)C2)=O)CC2CC2(CNC(C2(n3ccnc3)CCCC2)=O)C1 c1(C(=O)NC2(CC(=O)NC3(C)CN(C(C)=O)C3)CCC2)cccc(F)c1 C1(C(=O)NC(C(C)NC(=O)CC2OCCCO2)C)C2CCC1(c1ccco1)C2 N1(C(CNC(C(CC)C)=O)=O)C(CC(=O)N(CCN=[N+]=[N-])C)C2CCCC12 C1(NC(C(C)NC(C)=O)=O)(CNC(c2ocnc2C)=O)CCOC1 C#CCCC(C(=O)NCC1CC12CCC2)NC(=O)C(CC)NC(N)=O N1(C(c2ccsc2Cl)=O)CCC2CCN(C(C3CCn4ccnc4C3)=O)CC2C1 c1(C(N(CCCNC(=O)C=CSC)CC)=O)ccc(OC)c2cn[nH]c12 c1(C(C(=O)NCCC(C)NC(=O)C2=CCCC2)O)ccccc1I c1(C(N(CCNC(c2n(CC)ccn2)=O)C)=O)ccc2c(c1)SCCN2 CC1CC1C1CC1NC(=O)C(Cc1cnn(C)c1O)NC(=O)Cn1nccn1 c1(C(N2CCCC(NC(C3CCCC(=O)C3)=O)CC2)=O)ccc2nc(Cl)nn2c1 C1(C(=O)NC2(C)CC(NC(CC(CC)CC)=O)C2)CCc2nc(CC)ncc2C1 C=CCC(C)(C)CC(=O)NC(C1CCN(C(=O)C(C)Cc2cnco2)C1)(C)C C1(C(=O)OC)CCN(C(C2CCOC(C)C2)C(=O)NCCC2CC2)CC1C C12(C(=O)NC3CN(C(c4csc(Br)c4)=O)C3)CCCCC1CC(F)(F)C2 N1(C(Cc2nnc(C)o2)=O)CCC(NC(=O)CC2(CO)CCCCC2)CC1C c1(CNC2CCC(NC(c3n(CC)nc(C)c3)=O)C2)c[nH]c2ncc(Br)nc12 N1(C(c2n(CC)ccn2)=O)CC2CC(NC(C34CCC(CO)(CC3)C4)=O)CC2C1 C1(NC(C(F)=CCC)=O)CCCCC12CCCN(C(c1cnc(N)c(N)c1)=O)C2 CC(C)CC(O)CC(=O)NC(C1CCCN(C(=O)C=Cc2nccs2)C1)C N1(CCNC(C2CC(=O)N(c3ccccc3)C2)=O)CCC(CO)(CCl)CC1 C1(C(N(C)CC2N(C(c3n(CC)nnc3)=O)CCOC2)=O)CCCCC12CCC2 C12(NC(=O)NC3CC34CCOCC4)CC(CO)(C1)OC21CCNCC1 C1(C(=O)NC(C#C)C2CC2)CCCCCCN1C(C1CC2CCC(C1)O2)=O N1(C(C2(c3ccc(C)nc3)CC2)=O)CC(N(C)C(c2n[nH]cc2C)=O)C2(CC2)C1 CCC(CC)(CO)C(=O)NC(C)CCNC(=O)C(C)Sc1ccc(Cl)cc1 N1(C(C2CN(C)C(=O)CC2)=O)CC(C(=O)N(C2CCOC2)C2CC2)C2(CCC2)C1 C1(C)(NC(C(Cn2cncn2)NC(CCSCCCC)=O)=O)CCOC1=O C1(C(C)NC(c2ccc(Cl)c(F)c2)=O)CCC2(CC2)CN1C(=O)OC(C)(C)C c1(C(=O)NCCOCCN(C(c2cc(CC)on2)=O)C)cnn(C)c1Br CCC(CC)(CCNC(c1cnn(C(C)C)c1)=O)NC(=O)CC1COC(C)(C)C1 CCC(C)(CNC(C1CC2(C1)CC21CC1)=O)C(=O)NC1CCN(C(N)=O)C1 c1(C(N)=O)cc(NC(=O)C(=O)N2CC(n3cccc3)C2)cc(C(N)=O)c1 N1(C(Cn2c(C)ccn2)=O)CCCC(CNC(C2(C)CSC2)=O)CC1 CCCC(C(=O)OC)C(=O)N(CCC(=O)NCC1=CCCN(C)C1)OC c1(C(=O)NCCC(=O)NCC(n2cccn2)C)nc(=N)cc[nH]1 C1(F)(CNC(C(N(C)C)C2CC2)=O)COCCN(C(c2cc(Cl)nnc2O)=O)C1 C1(CNC(c2nc(CC)sc2)=O)CC(COC)CN1C(c1cn(C)nn1)=O c1(CN(C(CN(CC)CC)=O)CC)ccoc1C c1(C(=O)NCCCCCNC(C(CC)C(=O)OC)=O)cc2cccnc2nc1C C1(NC(C2CC(=C)C2)=O)CCN(C(c2cc(C(=O)OC)ccc2Cl)=O)CC1(C)C CC1=CCN(C(C2CC(N(C(=O)Cc3cc(C)nn3C)C)C2)=O)CC1 c1(OC)cncnc1N1CCSCC1C(=O)NC(c1cccc(F)c1)C C#CCC(C)(C)C(=O)N(C)CC1(CNC(c2cccc(C)c2N)=O)CC1 C1(NC(C=CC=CC)=O)C2CC3CN(C(c4cccc(C#N)c4Br)=O)C1C3C2 Cc1cnnc(O)c1C(N1CCCC(N(C(=O)C(N2CCN(C)CC2)C)C)C1)=O N1(C(CC(C)C)=O)CCCCC1C(=O)NCC(C)(O)CNC(C1CC(C#N)C1)=O c1(CNc2nc(-c3c(F)ncc(OCC)c3)sc2)ccc(C)c(C#N)c1 CC1CCC(N(C)C(=O)Nc2cc(CC(C)(C)C)nn2C(C)(C)C)CC1 c1(C(=O)NC2CCC(N(C(=O)C(=O)NCC3CC3)C)C2)n[nH]c2c1COCC2 N1(C(C2(CC)CCOC2)=O)C2CCC1C(C(=O)NCc1csc(Cl)n1)C2 C(C1CN(C(=O)C(C)OCC2CC2)CC1C(=O)N(C)CCC1CCC1)=CC c1(CC)cc(C(N2CCC3C(NC(c4nnc(O)nc4O)=O)C23)=O)ccc1Br Cc1cc(C(N2CCC(N(C)C(C3CCS(=O)(=O)N3C)=O)C2)=O)c(O)c(C)c1 N1(C(N2CCC(OCC(=O)NCC)C2)=O)CCCCC1CCO N1(C(CCCCCOC)=O)CCC(NC(c2cnc(C(C)C)s2)=O)C12CCC2 CCCCC(O)CNC(c1c(CNC(C2CC2OC(C)(C)C)=O)nnn1C)=O C12(C(=O)OCC(C)C3CC3)CCCN1S(=O)(=O)CC2 N1(C(=O)NC2CC(C(=O)OC)(C(=O)OC)C2)CCOC(c2cnn[nH]2)C1 Cc1ncccc1CCNC(C1C=CCN1C(=O)CCl)=O C1(NC(CC#C)=O)CN(C(c2cccc(F)c2Cl)=O)CC1(F)F N1(C(CS(=O)(=O)NCC)=O)CC2CC(C1)C2NC(=O)Cc1cccc(OC)c1F C1(C(C)C)(C(=O)NCCCc2cc(O)n[nH]2)CCCN1C(C1CCCCO1)=O Cc1ccnc(O)c1C(=O)NCCN(C(=O)Cc1cn[nH]c1)C N1(C(CC2(N(C)C)COC2)=O)CCN(C(C2(C)CC2(F)F)=O)CC12CC2 N1(C(CC2CC(C)C2)=O)CCCC(C)(NC(=O)CCOc2cccnc2)C1 C(C1c2ccsc2CCN1C(C1CC2(CSC2)C1)=O)NC(C1CCN(C)CC1)=O c1(CCC(=O)NC2CC2CNC(C2(CCF)CC2)=O)ccccc1F Cc1cc(Cl)ccc1C(=O)NC1CC(CNC(c2cncnc2C(C)C)=O)C1 CC(C)(O)C(F)C(=O)NC1CCC(CNC(=O)CC2CC(N(C)C)C2)CC1 c1(C(=O)NC(C)CN(C)C(C2CC3(CCOC3)C2)=O)cc2ccc(Cl)c(F)c2o1 CC1CN(C(=O)C(F)OC(F)(F)F)CC1n1cc(CC2(O)COC2)nn1 N1(C(c2c(C)n[nH]c2)=O)CCC2(CC1)CC(CNC(=O)C1=CCCC1C)C2 c1(NCc2ccc(OC)nc2)nc(N2CC3CC3(CO)C2)nc2ncn(C)c12 CCC(CC(=O)NCC(c1ccccc1)CNC(=O)CCF)OC COn1cnc(C)c1C(=O)NCC(O)CNC(=O)C(C)NC(c1cnoc1C)=O C1(C(=O)NC(C)CNC(=O)CC23CC(C2)C3)CCOC2(CCCC2)C1 C1(NC(CC=CC=C)=O)CC(CNC(C2CN(C(N)=O)C2)=O)C1(C)C c1(OC)ccccc1CC(C)=CC(=O)NC(C)C(C(C)C)NC(C1COC1)=O C=CCC(CC(=O)NCCOCC(C)(C)O)NC(=O)Cc1cccc(O)c1 c1(NCc2c(Cl)cc(N3CCOCC3)cc2)cnc2c(Cl)ccnn12 c1(NC(c2cccc(C)c2N)C2CC2)[nH]c(=NCCSC(F)F)nc2ncn(C)c12 C(C)(CCC(=O)NCC1CCCCN1C(c1cc(C2CC2)ncn1)=O)OC N1(C(=O)OC(C)(C)C)CCCC2(CNCc3ccnc(O)c3)CCCCC12 C1(OC)CCC2(C(N3CC(CNC(=O)Cc4ccnc(OC)c4)C(C)C3)=O)CC12 N1(C(C(CC)(F)F)=O)CC2CCCCC2(CNC(=O)CCCOC(C)C)C1 N1(C(c2c(SC)cccn2)=O)CC2ON=C(CNC(C3(C4CC4)CC3)=O)C2C1 N1(C(C2CCC(NCc3c(C)n[nH]c3)CC2)=O)CCC2(CCOC2)C1 Cc1c(CC(=O)NCC2(C(=O)NCC(O)C(C)O)CC=CC2)cnn1C C1(CNC(CCCCC#C)=O)CC12CCN(C(=O)C(=Cc1cccnc1)C)CC2 c1(C(c2n(CCCSC)nnn2)NCCCC(C)CO)cccc2[nH]ncc12 C1(C2CCOCC2)(NC(CN(C(=O)C#CC(C)(C)C)C)=O)CC1 N1(C(C2N(CC)CCCC2)=O)CC=C(CCNC(c2c[nH]nc2C(C)C)=O)CC1 CCC(C)C(C(=O)NCC12CC(C)(CCO1)C2)N(C(=O)CC1(COC)CC1)C c1(C(=O)NC(C(N2CC(CC)(OC)C2)=O)Cc2cn[nH]c2)ccc(C2CC2)cc1 C#CC1CN(N2CCC(C)(C(C)C)CCCC2)CC1O Cc1nc(N)cnc1C(=O)NC1(C)CCC(NC(=O)CC2CCCCC2)CC1 CC(O)CC(CNC(=O)CNC1(c2nn[nH]n2)CCC1)c1ccccc1 N1(C(C2N(CC)CCOC2)=O)CCCC2(CCN(C(c3csnc3Cl)=O)C2)C1 C1(C(=O)Nc2c(OC)nccc2)CCN(C(=O)CC(C)O)O1 N1(C(C2(OC)CC(C)C2)=O)CCOC2(CCN(C(c3cc(C)nc(C)c3)=O)C2)C1 c1(C(=O)NC2C(NC(=O)CC(C(F)F)N3CCOCC3)C2)ccc2occc2c1 N1(C(C)=O)CCOC(C(N2CCCC2C2(NC(C3CC(Cl)(Cl)C3)=O)CC2)=O)C1 C(=O)(C1=CC2CC=CCC12)C(C1(C(=O)NCCCOCCOCC)CCC1)=O c1(C(=O)NCC(C)(C2CC2)NC(CC(C)C2CCCC2)=O)[nH]nc2c1CCC2(C)C C1(CNC(C(CNC(=O)CCOCC(F)F)OC)=O)(COC)CC2CC2C1 c1(C(N2C(CNC(=O)C3=CCCCO3)CC(OC)C2)=O)cc(C)c(Cl)cc1F n1(CCCC)nnnc1C(COc1ccccc1)NCC1(COC)CCC1 c1(C(=O)NCC(CNC(C2CCCN2C=O)=O)OC)ccc(C)c(C)c1O N1CC(C(N2CC(C(CCC)O)C2)=O)CC(C)(C)C1.C1C(O)CCS1.SC.CC Cc1cc(F)c(N)cc1C(=O)NC(C)CCCNC(c1occ2c1CCOC2)=O N1(C(CCC(CC)C)=O)C2CCC1CC(C(=O)NC1CCN3CCC1C3)C2 N1(C(C(C)=O)=O)CC2(CCC(CNC(=O)C(Cl)(Cl)Cl)O2)C1 C12CCC(CC1)NC2=O.C1(NC(CC2CC(=C)C2)=O)CC(CO)(CO)C1 C1(O)(CCNC(CCC=CC(C)C)=O)CCN(C(C23CCCC2C3(F)F)=O)CC1 C1(NC(=O)NC(C)C(c2ccc(Br)cc2)O)CC2CCC(C1)N2C c1(C(N(CC(O)CNC(C2(N=[N+]=[N-])CC2)=O)C)=O)nn(CC(F)F)cc1[N+](=O)[O-] c1(CC)conc1C(=O)N(CC(CC)NC(=O)CN(C)C(N)=O)C C1(NC(=O)CC2(NC(=O)NCCCl)CCCC2)CCCC2(C1)N=N2 c1(C(=O)NCC2C(CNC(c3cnc(OC)s3)=O)C2)cn(C)nc1Br c1(CC(C)C)ccc(C(C(=O)NC2CCCCC2)N(C)CC2(C)CCCO2)cn1 c1(C(N2CCC(OCCNC(C(C)C#N)=O)CC2)=O)cccc(F)c1F N1(C(Cc2ccc(C(C)=O)s2)=O)CC(NC(=O)Cc2cn(C)nn2)C(C)(C)C1 N1(S(c2n(C)ccn2)(=O)=O)CCc2sccc2C1c1cccs1 N1(C(c2cccnc2F)=O)CC2CCC(C1)C2NCc1ccc(Cl)c(F)c1 C1(CNC(=NCCC(C)=O)NCC2CC3(CC3)CO2)CCCN1S(=O)(=O)N(C)C c1(NC2C(CC)CN(C(=O)C3=CC(C)(C)C3)CC2)ncc(C#N)cc1F CS(=O)(=O)c1coc(C(=O)NC2CCCC2NC(C2CCC(N=[N+]=[N-])CC2)=O)c1 CCC(CC)CC(F)C(=O)NCCOCC(N1CCC1COC)=O C(=O)(CC(C(F)(F)F)NC(=O)C1=NOC(C)(C)C1)NC(C(=O)NC)(C)C C1(CC(=O)NCC(CO)NC(C(C)=C2CC2)=O)CCN(C)C1=O S(=O)(=O)(CCC(=O)N1CCCC1C(C)(C)NC(=O)Cc1ccn(C(C)C)n1)NC C#Cc1cc(C(N2CCCCC(CNC(c3sccc3OC)=O)C2)=O)cc(F)c1 c1(C(n2cc(C3CCCN3C(=O)Cn3cccn3)nn2)C)cccc(C(N)=O)c1 C(=O)(C(C(C)C)C(C)C)NC(c1cnn(C)c1)C(=O)NC(c1c(C)ncs1)C CCCC(C)C(=O)N1CCCCC1CCNC(=O)Cc1cnn(CC)c1 C1(NC(=O)CCOCC(F)(F)F)CC2(C1)CC2NC(=O)COc1ccccc1 C(=O)(C1=CCc2ccccc21)N1CCC(C(C)(C)NC(C(CCCC)F)=O)C1 n1(CC)c(C(=O)NC(C)(C)CN(C(=O)Cc2cnc(C)[nH]2)C)nc2ccccc12 c1(OC)cc(C(=O)N(C2CCN(C(=O)Cc3nc(C)no3)C2)C)cc(O)c1O C(=O)(CCCS(N)(=O)=O)N1C(C2(NC(CCOCC(C)C)=O)CC2)CCC1 C1(COC)(NC(=O)CSC2CCCC2O)CCN(C(C2(c3cc[nH]n3)CC2)=O)C1 c1(C(COC(C2(C(C)NC(=O)N(C)C)CC2)=O)(C)C)ccc(Br)nc1 c1(C(N2CC3CN(Cc4nc(C)oc4)CC3C2)=O)cccc2cccnc12 c1(CC(=O)NCC2(C)N(C(c3c(COC)cco3)=O)CCC2)ccc(O)c(F)c1 c1(C(=O)NC(c2cccnc2)C(=O)NC(CC(C)O)C)cnc(O)c(F)c1 C=CCCCC(=O)N1CCCC1C(C)NC(=O)CCC1CCCN1C N12CCC(c3ccccc3)C(C1)NS(=O)(=O)CC2=O.CC1CCC(C(=O)O)CC1 c1(OC)ccc(Br)c(F)c1CN1C(C(=O)NC(C#N)C(N)=O)CCC1C C#CC1(C(=O)NC2(C(=O)O)CCCC2C)CCCCC1 C(=O)(C1=CCC(NC(c2cc(C)n(C)n2)=O)C1)NCc1c(C)cccn1 N1(C(C(N2C(CCCNC(c3c(C)cno3)=O)CCC2)=O)C)CCC(O)CC1 CC1(CNC(c2cnc[nH]2)=O)CCCN1C(=O)CC12COCC(C1)C2 C1(CNC(=O)C(=O)N2CC(Cc3cccnc3)C2)CCCCC1O C1(C)(CNC(C(=O)N(C)C)=O)CCCN(C(c2ccc(N)c(O)c2)=O)C1 N1(C(C(c2ccc(C)s2)C)=O)C2CCCC1CN(C(c1ccnn1C)=O)CC2 c1(CC)nn(C)cc1C(=O)N(C1CCC(NC(=O)C(C)OC2CCOC2)C1)C S(=O)(=O)(c1cnc(NC(C2CCOC2)C)c(Cl)c1)N(CCCCO)CC CCC(C)(C)C(O)C(=O)N1CCC(CNC(c2ccc(SC(F)(F)F)s2)=O)CC1 c1(OCCOC(C)C)ccc(F)cc1C1CCCN1CCCC(=O)OC c1(OCC)cccc(NC(=O)C(C2CCOC2)N(CC(=O)OC(C)(C)C)C)c1 C(=O)(C(C)CN(C)C(c1c[nH][nH]c1=N)=O)N(C(C)C(=O)NC)CC C1(F)(C(=O)NCCOCCNC(C(C)N(C)C)=O)CC12CCCCC2 C1(COC)(CNC(C2CC2(C)C)=O)CCN(C(=O)CN2CC3CC3C2)CC1 C1(C(=O)NOCC2CCCCC2)(CC=C)CCCN1C(c1cnncc1C)=O CC(C)CCCCCCC(=O)NC1CN(C(=O)C(C)NS(C)(=O)=O)C(C)(C)C1 N1(C(C2(OCC)CCCC2)=O)CC2(CCC2NC(=O)C=CCO)C1 c1(N(CCOCC=C)C)nc(=NCc2csc(O)n2)[nH]c2c1CCCCC2 C1(CCCC)CN(C(=O)CNS(=O)(=O)N(C)C)CCN1C(=O)C#CC1CC1 C1(NC(C(C2CN(C(C)=O)C2)OC)=O)CCCC1C(=O)O CC(CC(=O)N(C)CC1CCN(C(C2(CN(C)C)CC2)=O)C1)P(C)(C)=O.C(=O)N c1(NC(c2n(-c3c(C)cccc3C)nnn2)C)ccc2ncoc2c1 C1(C(=O)NCC2CC(NC(=O)CC(C)N3CCCC3=O)C2)(OC)CCOCC1 C(c1c(C)noc1C)=CC(=O)NCC1N(C(c2c(C)cc(C)o2)=O)CC(O)C1 N1(C(C(C)N(C(C)=O)C)=O)CC(O)(C2CCN(C(=O)C(O)C(F)F)CC2)C1 c1(CC)sc(=N)[nH]c1C(=O)NCC(C)CNC(=O)CCc1nccs1 N1(CCS(CC)(=O)=O)CCCC(NC(=O)C2=NOC(C(C)(C)C)C2)C1C c1(C(N2CC(CC)N(C(=O)C=CCO)CC2)=O)cnc2c(c1)CCOC2 c1(-c2cccc(C)n2)ccc2cc(C(=O)NC3CCNC3=O)oc2c1 C(=O)(C(C)CCC(C)(C)C)NC1(CNC(C(COCC)C)=O)CCOCC1 CC#CCC(C(=O)NCC1CNC(=O)CO1)NC(c1sc(C)nc1C)=O c1(C(=O)NC2CC(NC(C(CCOC)OC)=O)C2)cc2nc(=O)ccn2[nH]1 N1(C(C2CCC(CNC(C(OCC)OCC)=O)CC2)=O)CCOC(C)(C)C1C C1(CNC(C(CCSC)O)=O)CCC2(CN(C(=O)C(=O)Nc3ccccc3)C2)O1 c1(CN(C2CCC3CC2CN3)Cc2ccc(F)cc2)ncnc2c1oc1ccccc21 N1(C(C(c2ccco2)NC(CC2C(C)=NNC2=O)=O)=O)Cc2cncnc2C1 c1(-c2nc(CC(CC)C)nn2Cc2ccccc2N(C)C)cnn2c1CCCC2 C1(C)(CNC(C=CCOC)=O)CC(C(=O)N(C)C(C2CC2)C2CC2)C1 c1(OC)nc(Br)cnc1NC(c1cc(-c2c(F)cccc2F)cnc1OC)=O CC(C)C(Cc1ccccc1)C(=O)Nc1ccnn1-c1cccnc1 C12(C(=O)NCC(CC(C)C)OC)CCCC1CN(C(=O)C(Cl)Cl)C2 c1(C(C)C)cc(=NCCCCC(C)NC(C2CC3(CC3)C2)=O)[nH]cn1 C(=O)(CN=S(C)(=O)c1ccc(Cl)cc1)N1CCCC(NC(C(C)CO)=O)C1 c1(C(=O)NC2C(NC(C3(C=C)CCC3)=O)C2)ccc(OC)cc1OCCC c1(CC)[nH]c(C(=O)N(C)CC2CCN(C(c3ccnc(O)c3)=O)C2)nc1Cl C1(NC(CN(C(C)=O)C)=O)CC2CC1N(C(c1cccc(-c3nc[nH]n3)c1)=O)C2 N1(C(c2c(CC)noc2)=O)CCC2CN(C(=O)CC3SC(=N)NC3=O)CC2C1 c1(SCCC(=O)NC(C)CCN(C(=O)C(C)c2cc[nH]n2)C)ccc(Cl)cc1 c1(C(N2C3CC(C(=O)Nc4c(C)cccc4Br)C(C3)C2)=O)ccc2[nH]ccc2n1 CC1(C(=O)NCc2ccccc2SCC(N)=O)CCCN(C(c2cnn[nH]2)=O)C1 CCC(F)(F)CC(=O)NCC1(C(=O)NC2CCC(COC)C2)CC12CCC2 CCC(C(N)=O)NC(=O)CC1CCN(C(=O)CC2CCSCC2)C1 Cc1[nH]nc2ncc(C(=O)NCC3(NC(=O)C(C)CN(C)C)CCOC3)cc12 C(c1ccc2[nH]ccc2c1)=CC(N1C(c2n(CCOC)ccn2)C(C)(C)C1)=O c1(-c2cc(O)c(F)cc2)n[nH]c(=NCCCF)s1 C1(C(C)NC(c2cc(C)ns2)=O)CN(C(=O)Cc2cnccc2C)CCO1 c1(CN2CC(C)(CC(=O)Nc3cnccc3CO)C2)c(Cl)cc(Br)cc1Cl C1(N(C(CCc2onc(CCC)n2)=O)C)CN(C(=O)CC(C)(C)OC)CCC1C Cc1ccc(C(=O)NC2CC(=O)N(c3ccc(Cl)cc3Cl)C2)c(N)c1Cl C12(NC(c3cc(C)nc(Cl)c3)=O)CCCC1N(C(c1occc1C)=O)CC2 CCC1=NOC(CC(=O)NC2(CCNC(=O)C(c3ccccc3)C)CCCC2)C1 C1(C)(NC(C)=O)CCN(C(=O)CN(C(=O)CC2C(C)(C)C2(C)C)C2CC2)C1 CC1CC(CNC(=O)CCCC2CC2)CCN1C(C1CCC2(CCC2)C1)=O C1(C)(NC(=O)NC(c2cccc(C)c2)C(=O)O)CCCN(Cc2ccccn2)C1 Cc1cc(C(=O)NC(CNC(c2cnc(C(C)C)s2)=O)C(C)C)no1 c1(N2CCN(C(C)CO)CC2)nc(=NCCC2=CCCCCC2)[nH]c2c1CCC2 S(=O)(=O)(c1cnc2c(Br)csc2c1)NCCS(N)(=O)=O N1(C(c2c(OC)cc(F)c(F)c2)C(=O)NC2CCC2)CC2CS(=O)(=O)CC2(C)C1 c1(C(N2CCC(CCN(CCC(C)C)C)CC2)=O)cc2sccc2[nH]1 C(C(C)(CC(=O)NCC(C1CCC1)NC(=O)C(C)(C)O)C(F)(F)F)N(C)C n1(CC)nncc1CNC(=O)NC(C)C1CC1 C(CC(=O)NC1CCS(=O)(=O)C1)(C(F)F)NC(C(CC=C)NC(C)=O)=O c1(CC(=O)NC2(CN(C(=O)COCC3CCCCO3)C)CC2)ccc(Cl)s1 c1(CC(=O)NC(C)CC(C)n2cncn2)ccc(Oc2ccccc2)cc1 c1(C(N2CC(OC)CC(NC(CSCC)=O)C2)=O)cc(F)c(F)cc1Cl C12(NC(c3cncs3)=O)CCCC1N(C(c1nnc3ccccn13)=O)CC2 c1(C(C2CC2)OCC)nc(CC2(c3cccs3)CC2)n(-c2cnc(C)s2)n1 Cc1ccccc1COC(C)C(=O)NC1CC(NC(c2cnnn2C)=O)C1 c1(C(=O)NCC(CNC(c2c(C)snn2)=O)C)c(C(F)(F)F)ncn1O c1(OC)cc(OC)c(C(=O)N(CC(O)CN(C(=O)C(C)NC(N)=O)C)C)c(N)c1 C(C(C)(C)CCNC(=O)CC12CCCC1C2)NC(CCCn1ncc(C)c1)=O c1(CONC(=O)NCC2CC2(Cl)Cl)cccc(Cl)c1 N1(C(C(=O)N(CC(=C)C)CC)C)CCC(C(=O)NCCC2CC(C)(C)CO2)CC1 C1(C(N2CCC(CN(C(C(C)=CC)=O)C)C2)=O)CC12CCOc1ccc(Cl)cc12 c1(N2CC3C(C(=O)Nc4cc(OC)cc(Br)n4)(C3)C2)ncnc2[nH]cc(C)c12 N1(C(C2C(=C)C2)=O)CCCCC1C(=O)N(C1CN(C(C)=O)C1)C C1(NC(c2c(C)nn(C)c2)=O)CN(c2cc(C(N)=O)nc(Cl)n2)C2CCCCC12 c1(C(=O)NC(CC=C)CNC(c2cc(C3CCOCC3)on2)=O)cncc(C)n1 CS(=N)(=O)C1CN(C(C2(NC(C3CC4(CCC4O)C3)=O)CCSC2)=O)C1 c1(OC)ccc(C(c2nnnn2CC(F)F)NC2CC3CC3C2)cc1F N1(Cc2ccc(CC(C)C)cc2)CC2(CCN2C(=O)Cc2ccccc2Cl)C1 c1(OC)ccccc1C(C)C(=O)NCc1ccc(CNC(C2CC(C)C2)=O)cc1 c1(CC(=O)NCCCCCCN(C(COC(C)C)=O)C)ccc(Cl)c(Cl)c1 N1(C(CCSCC)=O)CCCC(C(=O)NCC(O)C(C)C)C1 C(=O)(C(C)(O)C(F)(F)F)N1C(CNC(CC(C=C)(C)C)=O)CN(C)CC1 C1(C)(CC(=O)NC(C2CCCC2)CNC(C(C)CF)=O)CCS(=O)(=O)N1 C1(CN(C(CCNC(CC(C)C)=O)=O)C)CCCCN1C(C1CN(C(C)C)C1)=O c1(CNC(CCOCC#C)=O)ccc2c(c1)CN(C(c1sc(CO)nc1C)=O)C2 CCCCCC(O)C(=O)NCC1CCN(C(c2sccc2Br)=O)C1 C1(C(N2C(CN(C(=O)Cc3cnc(C4CC4)[nH]3)C)CCC2)=O)CCCCNC1=O c1(C(N2C3CC(NC(C4CCC(C(=O)OC)CC4)=O)(C3)C2)=O)cn(C)c(=O)cc1C c1(C(C)(C)C(=O)NCC2CCN2C(=O)CC2(O)CCOC2)cccnc1F c1(NC(Cc2ncc(C)[nH]2)=O)ccc2c(c1)nnn2C C1(NC(c2ccc(N(C)C)c(F)c2)=O)CN(C(C2CCOC2)=O)C2(CCCC2)C1 C(C(=O)NC1CN(Cc2cccc(-c3ccccn3)n2)CC1F)(C(C)C)OCC C(CO)(C(O)C1CCC1)NC(=O)C(=O)N1CCC1C1CCC1 c1(C(N2CC(N(C)C(C34CCC(F)(CC3)C4)=O)C2)=O)cc2c(nc1O)CCSC2 C1(C(N(CCCN=[N+]=[N-])C)=O)CC(O)CN1C(C1CCC(=O)N1)=O N1(C(C)=O)CCC(C)(NC(C(C2CCCOC2)OCC)=O)CC1.C1(=O)CCCN1 N1(c2nccc(SC)c2)CCOCC(C(N2CC(=O)NC(=O)C2)=O)C1 N1(C(c2c(C)cnnc2O)=O)CCN(C(=O)CSC2CCOC2=O)CC(C)(F)C1 C1(C(=O)NC(CC=C)(C)C)CCCCC1CNC(=O)CC1CC(=O)NC1=O C1(NC(=O)CC2CCOCC2)CN(C(c2ccc3occc3c2)=O)CC12CCC2 c1(C(=O)NCC2N(C)CCN(C(c3cc(O)no3)=O)C2)n[nH]c2c1CCSC2 Cc1ncnc(C)c1C(=O)NCC1(C)CCCN1C(C1C=CC=CC=C1)=O C1(C(=O)NC(COCC)C(=O)Nc2cc(C)sc2C)CCOC(CC)C1 c1(C(N(CC(C)N(C(C(C)C2CCCC2)=O)C)C)=O)ccc(C(F)(F)F)c(F)c1 N1(C(CC(CN(C)C)O)=O)CCC(CNC(=O)CCCCN(C)C)C12CCC2 CC1(C)OCCC1CNC(=O)C(C1(O)CCC1)NC(C1CCC(F)(F)C1)=O C(=O)(CC(C)C(F)(F)F)N1CC(C)OC(C(=O)NCc2conc2C2CC2)C1 c1(C(=O)NC2CC3(CC(NC(C(CCC)O)=O)C3)C2)ccc(Cl)c(C)c1F C1(CC(=O)N(CCNC(=O)CC2CCCC2O)CC2CC2)CCCC(O)C1 C(=O)(C(Cc1cn[nH]c1)NC(C1(CC=C)CC=CC1)=O)NCC(C=C)O c1(C(=O)OCC)ccc(NC(=O)C(=O)NC2CCNC2=O)cc1S(N)(=O)=O c1(C(=O)NCC(O)CNC(C2CC3CC3C2)=O)csc(CCc2ccccc2)n1 Cc1c(C(N2CCC2Cn2cc(C3CC(F)(F)C3)nn2)=O)cncc1Br c1(N2CCCC(NC(C(COC)(C)C)=O)C2C)nc2ccc(Br)cc2s1 Cc1cnc(C(N2CCC(CN(C)C(C3CC4CC4C3)=O)C2)=O)cc1C c1(CNC(C(C)CC2CC2)=O)ccccc1CNC(c1c(Br)nnn1C)=O C1(NC(CCCC(=C)C)=O)CN(C(c2ccc(F)c(C)c2Cl)=O)CCC12CCC2 c12cc(OC)cc(c1)N2.c1(C(=O)Nc2ccc(CC)cc2)ccnc(OC)c1F c1(C(N2CC=CC(NC(CC3CC(=C)C3)=O)C2)=O)ccc2c(c1)S(=O)(=O)NC=N2 c1(NC(C)C(C2CCCCC2)NC(C2CCOC2)=O)ncccc1[N+](=O)[O-] N1(C(C2C(CCOC)C2)=O)CCC2CC1CN2C(c1cccc(C(N)=O)n1)=O C1(NC(C(F)=CCC)=O)CC(O)CN(C(c2scc(C)c2OC)=O)C1 N1(C(c2cnc3n2C(C)CCC3)=O)CCC2(CCOCC2)C(NC(=O)CCF)C1 N1(C(c2n(CC=C)ccn2)=O)CCN(C(C2CCCOC2C)=O)C(C)C1 C=CC(C)(CC)C(=O)NCCCOCCC(=O)NCc1cc(O)ccc1F Cc1ccc2c(c1)CCC(C(=O)NCCCC(C)NC(=O)Cc1ncc(C)s1)O2 c1(OC)cccc(F)c1CN1C(C(=O)Nc2cccnc2C#N)CC2CC12 C1(CC(=O)NCCCNC(c2c(C)oc(C(C)(C)C)c2)=O)CC2(CCOCC2)CO1 C(N=c1cc(NCC2CC2CO)nc(CC)[nH]1)CCC(=O)NC(CC=C)=O c1(C(N2CCC(OC)(CNC(=O)C(C)O)CC2)=O)cc(F)c(Br)c(F)c1 C1(NC(C(C)(C)C2CCC2)=O)CC(CNC(c2cocc2Br)=O)CC1O C12(C(=O)NC3CCCC(C#C)C3)CCC(CC1)N(C(C1CC(SC)C1)=O)C2 C1(C(=O)OC)CCN(C(=O)C2CCC2CNC(=O)CC2(O)CCCOC2)O1 c1(C(C)C)[nH]ccc1C(N1CC(F)(CNC(=O)C(c2ccccc2)C2CC2)C1)=O Cc1ccc(=N)[nH]c1C(=O)NC1CCC1CNC(=O)CC1CC(C)(C)C1 N1(C(C2(C)ON=C(C)C2)=O)CC2CC(NC(=O)CCN(C)CCO)CC2C1 c1(OC)ccnc(C(=O)NC2CC(F)(CNC(C3(C(C)C)CC3)=O)C2)c1F CC1CC(=O)NC1C(N1CC(O)(CNC(=O)COc2ccccc2O)C1)=O N1(C(=O)CC(F)(F)F)CC2(C1)CN(C(C1(O)CCOC1)=O)CC2CO c1(C(=O)NC2CCCC(NC(c3ccc(NC)cc3)=O)C2)c(C)ncnc1O CC1(C)CC(C(=O)NOCCC(=O)NC2CCNC2=O)N(CCO)C1 c1(C(=O)OCC)cc(CCCNC(N2CCC(Cn3cncn3)C2)=O)on1 S(=O)(=O)(c1cc(F)ccc1C(N1CCN(C=O)CC1)=O)N1C(C)CC(C(=O)O)C1 C1(CC(N2CC(COC)(CNC(C3CCCO3)=O)C2)=O)CCC2(CCC2)CO1 N1(Cc2cc(OC)cc(OC)c2)CC2(CCN(C(=O)C=CC(C)C)CC2)C1 c12c(F)cc(cc1Cl)CN(C1CCOC1)C2=O.c1(N(C)C)nc(C(=O)O)cs1 C1(NC(CCN2CCN(CC)CC2)=O)CC2CCC1N(C(=O)C(C)SC)C2 N1(C(c2c(NC)nccc2)=O)CCCC2CN(C(C3(C)CCOCC3)=O)CC12 Cc1cc(NC(c2c(C(F)F)cccc2Cl)=O)cc(C)c1 C#Cc1cn(C)nc1C(=O)NCC(C)C(=O)NCCCCCCC N1(C(c2c(C)scn2)=O)CC2(C1)CN(C(c1c(C)noc1C1CC1)=O)CCO2 N1(C(c2n(CC)cnn2)=O)CCC(COC(C23CC(OC)(C2)C3)=O)CC1 c1(CCC(N2CC(F)(CNC(C(C)OCC(C)C)=O)C2)=O)cccc(O)c1 C1(C(N)=O)(CNC(C2CCC2C(N)=O)=O)CN(C(C2CCC(=O)N2)=O)C1 c1(C(N2CC3C(NC(C4CN(CCC)C(=O)C4)=O)C3C2)=O)cc(C)c(C)c(F)c1 N1(C(C2CC(C)CC(C)C2)=O)CCC(C)(C)C(NC(=O)CCN2CCCCC2)C1 C1(NC(c2c(C)cc(C(F)F)o2)=O)CN(C(C2(C)CC2)=O)CCC12CCC2 c1(NC)cnc(C(=O)NC2CCC2NC(c2cc(C(C)C)sn2)=O)cn1 C(CN=c1[nH]c(=NCC2CCCC(F)(F)CC2)[nH]c2c1SCC2)c1[nH]c(=N)sc1 CC(C(=O)N1CCOC(CCCNC(C2(c3nccs3)CC2)=O)C1)S(N)(=O)=O N1(C(c2ccc(C#N)c(Cl)c2)=O)CCC2(CCC2)C(NC(C2CC=CCO2)=O)C1 N1(C(CSC(C)C)=O)CC2(CNC(=O)CCc3cccnc3F)CCC1C2 Cc1cc2cc(C(=O)NCC3CN(c4nc(Cl)ncc4F)CCO3)oc2cc1C c1(C(=O)NCC(CO)NC(CC2(C)CCCCC2)=O)cccc(F)c1N C(c1c(F)cccc1F)=CC(N1CCC(CNCC(=O)Nc2ccccc2)C1)=O c1(C(N(CC(CNC(C2(C)CCN(C)C2=O)=O)O)C)=O)cnc2sccn2c1=O c1(C(=O)NCCN(C(=O)CC(C)C2CCCCC2)CC)ccc2c(n1)CCCC2 C1(NC(c2c(OC)n[nH]c2)=O)C(C)CN(C(c2[nH]c(O)nc2C)=O)CC1C c1(N2CC(CCCCNC(C3(C)ON=C(C)C3)=O)C2)cc(C)c(C#N)c(C)n1 Cc1cc(C(=O)NC2COCC2n2cc(C(C3CCOCC3)C)nn2)ncc1Br C=C1CCC(C(=O)NC(CCNC(C2CNC(=O)C2)=O)C(C)C)CC1 C1(C#N)(C(=O)NC(C2CCN(C(c3ccc(CCC)[nH]3)=O)C2)(C)C)CC12CCC2 c1(NCCCCC(C)NC(C2CN(C)CC(C)O2)=O)ncc2c(ncn2C)n1 CC(C)CCCCCC(=O)N1CCOC(C(C)NC(=O)C(C)n2cncn2)C1 C1(C(=O)OC)CCN(C(=O)C=CC2CCN(C(=O)Cn3ccc(C)c3)CC2)O1 C(=O)(C(CN(C)C)NC(C1COCC1C(N)=O)=O)NCC(CC1CC1)OC N1(C(C)=O)CCCC1CN(CC1(Oc2ccccc2)CC1)Cc1ncc(C)s1 C1(CC#C)(C(=O)NCC(O)CN(C(=O)Cc2cncn2C)C)CCCCC1 C12(CC(=O)NCC(C)Cc3cn[nH]c3)CCC1CN(C(c1ncccc1F)=O)C2 C1(CC)(NC(c2coc(Cl)c2)=O)CCCN(C(C2CC(c3ccccc3)O2)=O)C1 N1(C2CN(C(C3(C)CC3C(F)(F)F)=O)C2)CCN(C(c2ncc[nH]c2=O)=O)CC1 CCC(CC)CC(C(=O)NCC(F)F)N1CCOCC1c1ccc(C)o1 N1(C(C=C(C)C(F)F)=O)CCCCC(NC(=O)CC2OCCCC2(C)C)C1 N1(C(c2[nH]cc(C(C)=O)c2)=O)CCC2C1CCCN2C(C1CCC(CO)CC1)=O c1(NC(CCNC(C2(C=C)CCC2)=O)=O)cnc2[nH]ncc2c1 N1(C(CCC(C)C)=O)CCC2CN(C(C3(C(F)F)CCOCC3)=O)CCC12 C1(F)(CNC(CCC(C)OCC)=O)CCC(CNC(=O)Cc2cnn(C)c2)CC1 c1(C(=O)NC(CCNC(CCC=CC)=O)(C)C)nc(S(N)(=O)=O)c2ccccn12 CC(C)(C)CCCCCC(=O)N1CCC1CNC(c1c(O)ncc2c1CCC2)=O C1(C)(CC(=O)N(CC(C)NC(=O)C=CSC)CC)CCS(=O)(=O)N1 CN1CCCC(F)(C(=O)NCCC2(O)CCCN(C(=O)Cc3cnccn3)C2)C1 C=C=CCCC(=O)N(CCNC(C1CCCC1C)=O)CC Cc1ccc(=N)[nH]c1C(=O)NC1(CNC(=O)CC2CCCN2C(C)C)CC1 N1(CCC)CC(C(N2CCC(NC(c3cnn(C)c3)=O)CC2)=O)CC1=O Cc1cccc(C(=O)N(CCC(=O)N(C2CC2)C(C)C2CC2)C)c1N O=C1CC(C(N2CCCOC(CCNC(=O)C=CC=C(Cl)Cl)C2)=O)CC(=O)N1 c1(N2CCC(C(CC)C)CC2)ccc(Br)c(S(=O)(=O)NC(C2(OC)CCC2)C)n1 c1(C(N2C3C(NC(CCC(=O)NC)=O)C(CC3O)C2)=O)cn2c(C)cccc2n1 c1(N2CCC(C(=O)NC3CCOCC3)C2)ccc(NCC2CCNC2)cc1 S(=O)(=O)(c1ccccc1C#N)Nc1c(C(C)OC)cc(F)cc1 N1(C(CCCC#CC)=O)C2CCC1CC(N(C)C(C13CCC(OC)C1C3)=O)C2 CCC1CN(c2cc(N3CCN(CCO)CC3)ncn2)Cc2ccccc21 N1(C(CSc2ccc(OC)cc2)=O)CC2(C1)CN(C)CCO2 N1(C(C=CC)=O)CCC2(CC1)CC2C(=O)N(C1CC1)CC O=C1CC(C2CCN(C(c3cnc4ccc(-c5nn[nH]n5)cn34)=O)CC2)CN1 CC(C)CC(C)(O)C(=O)N1CCN(C)C(C(=O)NOCc2ccccc2F)C1 N1(C(CC(C)OC)=O)CCC(C)(C)C(NC(c2ccc(C)cc2Cl)=O)C1 N1(C(c2c(OC)nccn2)=O)C2CCC(C2)C1CC(=O)NC1CC1c1ccsc1 N1(C(C(CC#C)NC(=O)CNC(=O)OC)=O)CCC(O)CC12CC2 CC1CCCC=C1C(=O)NC(C)(C)CCNC(c1conc1C1CCCO1)=O C1(CNC(CCCN(C(C)C)C)=O)CCN(C(c2cc(C3CC3)ns2)=O)CC1C Cc1ccc(C(=O)NC(CNC(=O)CC2CCC(=O)C2C)C2CC2)cc1O C1(N(c2scc(CN3CCOCC3)n2)C)CCCCC1C1CC1.CO c1(CN(CC(CC)Oc2ccccc2F)C=O)cnc(F)c(Cl)c1 C(=O)(C(C(C)NC(c1cncc(OC)n1)=O)C(C)C)NC(CCCC)(C)C C(CC(C(=O)N1CC(O)(C#N)C1)NC(=O)C(c1ccccc1)C)SC CC(O)C(C(=O)NCc1ccoc1C(=O)NC1(c2cccs2)CC1)N(C)C c1(OC)cc(C(=O)NCCC2(C)CCCC2)cc2cccnc12 c1(OC)ccc(C(N2CCCC2(C)C(=O)NCC(F)F)=O)c(Br)n1 c1(CC)c(C(=O)NCC(C2(O)CCN(C(=O)CN(C)C(N)=O)C2)C)csc1C C(C(=O)NC(C)C(CO)NC(=O)C(O)CC1CCCCC1)(C(C)C)OC C(C)(CCC(=O)NCCCNC(=O)Cc1ccc(CC)s1)OCC C(=O)(CC(F)(F)F)NCC(N1C(CNC(=O)C=Cc2ncc[nH]2)CC1)=O C1(NC(CC(CNC(C(CC)NC(N)=O)=O)OC)=O)CCC(C2CC2)C1 N1(CC(N2CCC(CCC)C2)=O)CCCC(N(C(=O)CSC(F)F)CCO)C1 c1(C(C)C)c(Cl)ncnc1NNC(=O)C1(c2ccc(Cl)cc2Cl)CC1 C#CCC(C)(C)NC(=O)CC1CCCC1NC(=O)C(CC)N(CC)CC CC(CC(=O)NCC1CC(O)(CNC(c2cnc3c[nH]nc3c2)=O)C1)P(C)(C)=O N1(C(C2CC(C)(NC(=O)CCN(C)C)C2)=O)CCC2CCC(C2)C1 c1(C(=O)NCC2C=CC(NC(CN(C(=O)OCC)C)=O)C2)nnn(C)c1C1CC1 CC1OC2(C(N3CC(F)(CNC(=O)CCCC4CC4)C3)=O)CC1C2 c12ccc(c(C(F)(F)F)c1)CC2.CN(C)CCN(CCNC(=O)C1CC1)C CN(C1CCCc2c1cnn2C)C(=O)NC(CC(F)F)C(=O)O c1(C(=O)OCCCc2c(C)cccc2)c(C)ccc2ncccc12 Cc1cc(C(N2CCCC2CNC(C23CCCC2OCC3)=O)=O)cc(C)c1Br N1(C(c2c(CC)nns2)=O)CCCC(C(C)NC(c2c(C)noc2C2CC2)=O)C1 CCCCC(C)C(=O)NC1(C)CCN(C(C2CC3(CC3)C2)=O)CC1 c1(C(=O)NC(CN(C(c2c(CC)nco2)=O)C)CC)cnn(C)c(=O)c1 c1(C(N(C2CCCN(C(c3cn(CC)nc3C)=O)C2)C)=O)cc(Cl)c(O)cc1C c1(CC(=O)NCC(CNC(=O)CC2CC3CCC2O3)OC)ccc(F)c(Cl)c1 C(=O)(CC(F)(F)F)NC(CCNC(C(C1CCC(=O)N1C)C)=O)(C)C c1(C(=O)NCC2(O)CN(C(C3C(C=C)CC3)=O)C2)cnn2ccccc12 c1(CC(C)C(=O)NC2C=CCN(C(=O)C(C)CCO)C2)ccc(Cl)cc1 n1(CC)cnc2nc(N3CCCC(CC#N)C3)nc(NCc3cc(C)on3)c12 C(=O)(C1=CC2(CCN(C(=O)C#CC(C)(C)O)C2)C1)N1CC(C)(C)OCC1(C)C c1(C(=O)NCC(CNC(c2c(OC)nccc2)=O)O)cnc(C)c(N)c1 C1(NC(C(CC=C)NC(c2cc(C)[nH]n2)=O)=O)CCCC(O)CC1 c1(C(=O)NC(c2ncc(Br)cn2)CC)ccc2c(C)cc(Cl)nc2c1 C1(C#N)(C(N2CCC(O)(CN(C(CCOC(C)C)=O)C)C2)=O)CC2CC2C1 Cn1ncc(C(N2CCCCC2C(=O)NCC2CCCSC2)=O)c1C#N C1(NC(=O)COC(F)F)CCCCCN(C(=O)C(O)CC(F)(F)F)C1 N1(c2cc(OCC)ncn2)CCC(O)(C2(NC(=O)COC)CC2)CC1 O=C(C1=C(Cl)CCC1)N1CC(NC(C2(C(N3CCOCC3)=O)CC2)=O)CC1CO c1(C(N2CCN(C(C3CC(=O)C3)=O)C2)=O)ccc2ccnn2c1 C1(NC(C(c2cc(C)oc2C)C)=O)CN(C(c2cnns2)=O)CC12CCOCC2 c1(C(N2CCC(NC(C3C(OCC)C3)=O)C2(C)C)=O)cccn2ccnc12 N1(C(CN(S(CC)(=O)=O)C)=O)CC(NC(c2cnn(CCO)c2)=O)C(C2CC2)C1 c1(C(N(C2C3CN(C(=O)CCc4nc(O)n[nH]4)CC23)C)=O)ccc2ncnn2c1 N1(C(C=CC=CC)=O)CCC(C(C)C(N2CCC(c3ncco3)C2)=O)C1 N1(C(C(C)OC2COC2)=O)CC2(CCC2)CC1CNC(=O)CCCCNC(N)=O C1(CC(=O)N(C)CC2(CC(C)C)CC2)CC(O)CN1C(=O)C(c1cnn(C)c1)C N1(C(CCNC(C(=C)F)=O)=O)CCN(C)C(=O)C1C c1(NC(=O)OC(C)(C)C)nccc(NC(c2cnn(-c3cccnc3)c2)=O)c1Br Cc1ccc2c(C(=O)NC(CNC(=O)C(C)c3ccsc3)CO)csc2c1 C1(NC(=O)Cn2ncnn2)COCCN(C(=O)Cc2ccncn2)C1 c1(CC)ncc(C(N2CC(CNC(=O)CC(C)C)C(C)(C)C2)=O)c(C)n1 C1(F)(CNC(CCc2n(C)cnc2)=O)CCC(CNC(=O)CC2(C)CCCC2)C1 C=C=CC(C)C(=O)N(C1CCN(C(=O)Cc2cc(CNC)on2)C1)CCO.SCC C(=O)(CC(CCN)C(F)(F)F)NCCC(CCC(C)C)C C(=O)(C1=CCCC1(C)C)N1CCC(C(C)(C)NC(COc2cc(C)on2)=O)CC1 CCCC(O)C(=O)N(C)CCN1CCN(C(=O)CN(C)CCC)CC1 C(=O)(C(C)(C)C(F)F)NCCCN(C(C1C(C=C)OCC1)=O)C(C)C C1(OC)(CNC(c2nnsc2C)=O)CCN(C(c2cnn(C(C)(C)C)c2C)=O)C1 C(=O)(C(C)(C)C(F)F)NC(C)C(C)C(=O)N(C)Cc1ccco1 C(C(=O)NCC(=O)N(C1CCCC(C)C1)C1CC1)(C(C)C)NC(=O)OC C1(NC(CCN(S(C)(=O)=O)C)=O)CCC(N(C(=O)CC2CC(C)(C)CO2)C)CC1 C=C(Cl)CCC(=O)N1CCOCC1.C1(C(N(C2CC2)C)=O)CN(C=O)CCO1 C1(NC(CCN(C(C2C(C)CC2)=O)CCO)=O)CCN2CCCC12 CC1CCn2c(C(N3CCCC(NC(=O)CC(C)C4CCCC4)C3)=O)cnc2C1 C(C(CC)N=c1[nH]c(=NC)[nH]c(=NCc2cc(C)nc(C)n2)[nH]1)N(CC)CCNCC CC1CCCN(C(C2CC2CNC(C2(N(C)C)CCC2)=O)=O)C1.C1C(=O)N1 CC1CN(C(=O)C(C)(C)c2cnsc2)CC1NC(c1cnco1)=O C1(OC)COCCN(C(c2cccc(F)c2Cl)=O)C1.C12C3CN(CC13)C(=O)N2 C1(C(=O)NCCc2nc(C)oc2C)CC(C)(C)CN1C(=O)C(C)Cn1ccnc1 N1(C(CN(C)C)=O)CC(CNC(c2nsc3ccccc23)=O)OC(C)(C)C1 c1(CC(C(=O)NC2C(NC(c3cncc(C)c3)=O)CCC2)C)ccc(F)cc1F n1(CC)ncc2cc(C(=O)NCC(C)NC(c3cnsn3)=O)cnc12 C1(CCNC(C2(COC)CCCC2)=O)CC2CCC(C1)N2C(=O)C(C)C(C)(C)C c1(OS(CC2C(C)CCC(C)O2)(=O)=O)cc2c(cc1[N+](=O)[O-])OCCO2 C(=O)(C(F)(F)CC(C)C)NCCC1(C)CCN(C(C(CCOC)C)=O)C1 c1(C(=O)NC2C(NC(=O)C=Cc3cccs3)C2)cc([N+](=O)[O-])ccc1OC(F)F c1(CCCC(=O)NC2(C)CCN(C(=O)CC3COCCOC3)C2)ccc(F)c(F)c1 c1(N2C(CNC(C3C(C)OC(C)C3)=O)CCCC2)ncnc2sccc12 CCC(C)(CN=c1cccc(S(=O)(=O)NCc2cc(C)sc2C)[nH]1)C(N)=O C(O)(C(F)(F)F)C1(C(N(CCCNC(C2CC23CCC3)=O)C2CC2)=O)CC1 c1(C(=O)NC(CN(C(=O)CCCc2nc(C)cs2)CC)C)ncn(C)c1C Cc1cc(C)c(C(=O)NCCC(C)(C)NC(=O)CC2CC2(C)C)c(C)c1Br c1(CN2CC(CC(=O)NCC3(NC(C)=O)CCC3)C2)cc(O)ccc1C CC1CN(C(c2csc([N+](=O)[O-])c2)=O)CCC1NC(=O)CSc1n[nH]c(O)n1 C#Cc1ccc(F)cc1C(N1CCCC(C)(NC(=O)C=CC2CCCN2C)C1)=O N1(C(Cc2cc(COC)on2)=O)CC(CNC(=O)C(CC)CCOC)C(F)(F)C1 c1(C(N2CC(CNC(C3CC(CF)C3)=O)C2)=O)ccnnc1 c1(C(=O)NC2CN(C(CP(C)(C)=O)=O)C2)ccc(Br)c(F)c1N c1(OC)c(C(=O)NC2C3CC2N(C(c2ccnc(C)c2)=O)C3)oc2ccccc12 C1(C(=O)NC2CC(NC(=O)Cc3cc(C)no3)C2)(CC)CCOC1 C1(NC(CCCC(=O)N(C)C)=O)C2CC(O)C1N(C(=O)C(O)c1ccsc1)C2 c1(C(=O)NC2(C)CN(C(c3cnc(C)s3)=O)C2)cc[nH]c(=N)c1Cl O=C1NCc2c1ccnc2C(N1CCCC(c2nnno2)C1)=O N1(C(Cc2scc(C)c2)=O)CCC(F)(C(=O)NC(c2ncn(C)n2)C)CC1 c1(C(N(CC(CN(C(c2cnc(C(C)C)s2)=O)C)O)C)=O)ccc(F)nc1 c1(CCN(C(=O)C(C2CC2)NC(c2ccsc2Cl)=O)C)ccncc1 C1(NC(c2cn(CCCOC)nc2)=O)CCCN(C(c2nc(C)oc2C)=O)CC1 C1(C(=O)NCC(CCNC(CCC(=C)C)=O)(C)C)CC2CCC(C1)N2C(C)C N1(CC2C(C(=O)NC3CC(CNC(C=CC(C)C)=O)C3)C2)CCOCC1 N1(C(c2ccc[nH]2)=O)CCC(NC(C23CCC(CO2)C3)=O)C(CO)C1 C(CCCC(CO)NC(=O)Cc1coc(C)n1)NC(C1CN(CCC)C(=O)C1)=O C1(NC(CN(C)C)=O)CN(C(C2CNC(=O)N2)=O)CC1F CC1CCN(C(C2(F)CCOCC2)=O)C1CNC(c1cccc(NC(N)=O)c1)=O N1(C(Cc2ccc(C)nc2)=O)CCCC(O)(CNC(=O)C2=CCCCC2)CC1 C=CC(C)(O)CC(=O)N(CC(C)(C)CNC(C1CCC(C)O1)=O)CC N1(CC(=O)NC(=O)NC2CC2)CCC2(NC(C3(F)CCOCC3)=O)CCCC12 C(C(CC(C)C)NC(c1[nH]nnc1C)=O)NC(c1cnc(C)s1)=O C(CC(C)(C)C(=O)N1CC(NC(C2CC(=O)N2)=O)C(n2ccnn2)C1)OC n1(C(C)(C)C)cnc(C(N2CC(CF)(NC(c3csnc3Cl)=O)C2)=O)c1 C1(C(=O)NC(C)CNC(=O)CNC(=O)OC(C)(C)C)(CN(C)C)CCCO1 Cc1nc(C)n(CC(=O)N(CC(O)CNC(c2nnc(S)n2C)=O)C)n1 CC(C)CC(CC(=O)NCC1CCC(C)(C)O1)NC(c1cc[nH]c1C1CC1)=O N1(C(Cn2c(N)cc(C)n2)=O)CCN(C(C2CC2F)=O)C(C(C)C)C1 C1(NC(CCCN(C(C)=O)C)=O)CC(C)N(C(=O)CN(C(=O)C(C)C)C)C1 C(C#Cc1cccc(Cl)c1)NC(=O)Nc1ncsc1Br c1(N2C3C(C(=O)NCc4ccc(SC)cc4)C(C3)C2)ncc2sccc2n1 C(=O)(C(F)(CNC(c1snc(C)c1N)=O)C(C)C)N(CC(C1CCC1)OC)C C1(C)(NC(C2CCC(C(C)=O)O2)=O)CCCN(C(C2(c3oncc3C)CC2)=O)C1 c1(C(=O)NC2CN(c3snc(SC)n3)C(C)CC2)cc2c(cnn2C)nc1O CC1CN(C(c2c[nH]nc2C2CCCO2)=O)CC1CNC(C1CCCO1)=O C(=O)(C(CC(C)C)C(C)C)N1CC(CNC(c2cncc(SC)c2)=O)C(C)(C)CC1 NC(=O)CCCC(=O)NC1CC(CNC(=O)CSCc2ncc[nH]2)C1 C(c1ccccc1F)=CC(=O)NC12CC(CNC(C(CC)SC)=O)(C1)C2 C1(C(N(C2CCC(NC(c3cc(C(F)F)cs3)=O)CC2)C)=O)CCCCN1N=O c1(C(=O)NC2(SC)CN(C(=O)CN3CCC(O)CC3)C2)cc[nH]c2nccc1-2 N1(C(C(=O)NC(CC)C)CC2CCCCC2)CC2(C(=O)OC)CC1CO2 c1(C(=O)NCCCCN(C(c2nccc(OC)c2)=O)C)ccc(Cl)cc1OC c1(OC)ccc(C(F)F)cc1C(=O)NC1CN(C(=O)C(C)(F)F)C2CC12 N1(C(C(C=CC)O)=O)CCC(CNC(c2c(C)cccc2OC)=O)C(F)(F)CC1 C1(NC(=O)CCc2nc(Cc3ccccc3)no2)CCOCC12CCCC2 Cc1csc2c(C(N3CCC4(CC3)CC4CNC(C3CC3C)=O)=O)ncnc12 c1(CNC(C2OCCN(Cc3c(C)ccc(Br)c3)C2)=O)cnc2ccccc2c1 C1(CNC(=O)NC(c2ccnc(Cl)c2F)C)CCCC12CCC2 c1(CN2C(C(C)C)CNCC2)cc(Cl)ncc1Br C(=O)(CCCCCCNC(=O)C1=CCCCCC1)NC(CCC)C1CC1 c1(C(N2CC3C(NC(CS(CC)=O)=O)(C3)C2)=O)c(C)nn(C)c1Br c12ccccc1C(NC(=O)C(C(C)O)NC(N)=O)CNC2=O.c1(CC)cnc[nH]1 C1(N(C)C)CCOC(C(N2CCC(N3CCCOCC3)CC2)=O)C1 Cc1[nH]nc(C(N2CCC(CCNC(=O)C(C)Sc3ccccc3)C2)=O)c1C CCC(C)C(O)C(=O)NCCCCCCN(C(=O)CC1CNC(=O)C1)C c1(OC)cccc(F)c1C(=O)NC1CN(CCn2cccn2)CCC1C N1(C(c2c(Br)cn(C)n2)=O)CCCC(C(N2CC3CC2CN3)=O)CC1 C1(C(=O)NCC2(CN(C(C(C)OCCC=C)=O)C)CC2)COc2ccccc2C1 C1(C(=O)NC2CCN(C(c3cnn(C)c3C#N)=O)C2)(OC)CCCCCCC1 c1(OC)ccc(C(c2ccccc2)(C2CC2)NCC2CC(F)(F)C2)cc1 c1(C(=O)NC2(C)CN(C(c3cccc(F)c3)=O)C2)ccc(N)c(F)c1Br N1(C(C2(C=C)CC2)=O)CC2C(N(C)C(c3cnc(C(F)(F)F)s3)=O)C2C1 CC1(CC(=O)N(CCNC(C2CCCN2C2CC2)=O)CCOCCO)OCCO1 C(c1cn(C)nn1)=CC(=O)NC(C1CN(C(=O)CC2CN(C)C2)CCO1)C Cc1cc(C(=O)N(C(C)CN(C(=O)C(C)Oc2ccccn2)C)C)cs1 Cc1ccc(Br)cc1CNC(C1COCCN1C(c1ncc(Cl)cn1)=O)=O c1(C(=O)NCC2(C)CC2)cc(CC(c2ccccc2)=O)nn1C.C12CC1NC2=O c1(C(=O)NC(CN(C(C(CSC)C)=O)C)C)cccc(C2(C)CCO2)c1 N1(C(C(C)OC(C)=O)=O)CCC2CN(C(c3cc(C)no3)=O)CC12 CCC(CC)(C(=O)OC(C)(C)C)C(=O)NC1CCCC1CNC(=O)C=CC(C)(C)C C1(C)(C(=O)OC)CC(OC)CN1C(=O)CCCC1CNC1 CC(C)CCC(=O)C(=O)NC1CC2CCC1(C(N1CC(O)C(N=[N+]=[N-])C1)=O)C2 C1(COC)(NC(=O)C=CC(F)(F)F)CCN(C(C2CCN2S(C)(=O)=O)=O)C1 C1(C(=O)NCCCNC(C(C)(C2CC2)OC)=O)Cc2cc(Cl)ccc2O1 C=CCCCCCC(=O)N1CC(C)(C(=O)Nc2cc(C)c(O)c(C)c2)C1 N1(C(CC(=C)C)=O)CC(C)N(C(c2c(F)ccc(F)c2OC)=O)CC1C N1(C(C2CC23CCCC3)=O)CC2CCCCCC12 N1(C(c2c(C3C(C)C3)noc2)=O)CCC(C2CC2)(NC(=O)COCC(F)F)C1 C1(C(N(CCS(N)(=O)=O)C)=O)CCN(C(c2cc(C(N)=O)[nH]n2)=O)C(C)(C)C1 c1(OC)ccc(C)nc1C(=O)NC1CCC12CN(C(c1ccc(F)cc1N)=O)C2 CCCC(C(=O)NC)NC(=O)C(c1cccs1)NC(c1cccn1C)=O C(=O)(CC(C)C(F)(F)F)NC1CCCC(C(N2CCC(C)(COC)C2)=O)C1 C(C)(C)(CCNCC(O)C(=O)N1CCOCC1)OC c1(C(N2CCCC2CCCNC(C2(C3CC3)CCC2)=O)=O)ccn(C(F)(F)F)n1 N1(C(C=CCCC)=O)CC(NC(=O)CCC2CCC(=O)C2)C(n2cccn2)C1 CC(C)(C)C#CC(=O)NC1CCC(NC(c2cc3occc3[nH]2)=O)C1 c1(C(=O)OC)cnc(F)cc1C(C)(C)NCCc1cocn1 Cc1nc2ccccc2n1CCC(=O)NCCCNC(=O)C(c1cnn(C)c1)O CC(C)C1=NOC(C)(C(=O)NCC23CC2CN(C(=O)C(c2ccccc2)=O)C3)C1 c1(C(N2CC(C(C)C)N(C(N)=O)CC2)=O)cccc2nc[nH]c12 c1(OC)ccc(S(=O)(=O)CCN2CCC(c3ncco3)CC2)cc1 C1(C#N)(C(=O)NCCNC(C(C)(C2CC2)OC)C(=O)O)CC12CCOCC2 c1(C(=O)NC2C(C)CCN(C(C(CCOC)C)=O)C2)cncc2c1CCNC2=O N1(C(C(COC)N(C)C)=O)CC2CC1CN2C(c1ccnc(C(F)(F)F)c1N)=O C(CCC1CC1)(C(=O)NOC(C)(C)C)NC(c1n(C)c(C#N)cc1)=O C(C(C)C(=O)NC1CC1CNC(c1ccc(COC)o1)=O)OCC c1(C(N2CCC(O)(CNC(C3(C)CC(C)(C)C3)=O)C2)=O)ccn(CCO)c(=O)c1 c1(C(=O)NC(CCN(C(c2c(C)c[nH]n2)=O)C)C)cc2ccc(Cl)cc2s1 N1(C(COC(CC)(C)C)=O)CCC(F)(C(=O)N(CC(c2ccsc2)O)C2CC2)C1 c1(OC)cc(=O)oc2c(C)cc(C)cc12.C12Cc3nnsc3S1(=O)=NC2=O N1(c2cc(NCc3[nH]nnc3C)nc(C)n2)CCC2(CCC2)S(=O)(=O)CC1 C1(NC(C=CC)=O)CCOC12CCN(C(=O)C(C(C)C)c1cnc(C)s1)CC2 Cn1ccc(S(=O)(=O)N2CCN(C(c3cc(Cl)c(Cl)cn3)=O)CC2C#N)n1 C=CCC(F)(F)C(=O)NC1CCN(C(=O)C(CC)N2CCCC2=O)CC1 c1(C(c2nnnn2CCCF)NC(c2csc(C3CCC3)n2)C)nc(C)cn1C c1(C(=O)NCCC2C(C)CN(C(=O)CCNC(N)=O)C2)cccc(F)c1C#N S(=O)(=O)(c1ccc(NCCCN2CCOC(C)C2)c(Cl)c1)NC(CCC=C)C c1(C(N2C(C)CC(NC(c3cc(C4(C)CC4)on3)=O)C2)=O)cccc2nccn12 C12(CNC(=O)CC3CCSC3)CCC(NC(c3ccnnc3O)=O)(CO1)C2 c1(C(N(C2CC(NC(c3cocc3Br)=O)C2)C)=O)ccncc1Cl C1(OCCn2cc(C(N(C)CCO)CC)nn2)CCCN(C(=O)C(O)C2CC2)C1 c1(C(C)C)nn(C)cc1C(N1CC=CC1CNC(c1cncnc1)=O)=O c1(C(=O)NC(CCCC)CNC(C2(C(=O)N(C)C)CC2)=O)cc(C)ccc1Cl Cc1cc(=O)oc(C)c1C(N1CCC(N(C)C(c2cnn(CC3CC3)c2)=O)C1)=O CC(C)(C)C(CNC(c1ccoc1)=O)C(=O)NCCSCCSC(F)F CC(=O)CCN=C(NCc1cc2c(s1)CCCC2)N1CCC(n2cc(C)cn2)C1 C1(C(=O)NCC2C(C)CCN2C(c2cnc(Cl)s2)=O)CCC2(CC1)CC2 C#Cc1ccc(CCCC(=O)NC2CCCN(C)CC2)cc1 N1(C(c2cccc(NC(C)=O)c2)=O)CC(NC(C2CCOC2)=O)CC(F)C1 c1(C(N2C3CN(C(=O)C(F)(F)Cl)CC32)=O)c(F)ccc([N+](=O)[O-])c1F N#Cc1ccc(CNCC(S(C)(=O)=O)c2ccccc2)s1 Cc1nc(C(F)(F)F)c(CNC2CCOCC2c2ccc(F)cc2)s1 c1(C(=O)NCC2(F)CCN(C(C3(F)CCCCC3)=O)C2)ccc2c(c1)CCC2 CCN=c1[nH]c(C)c(C(=O)N(C2CCCN(C(=O)C(C3CC3)OCC)CC2)C)s1 C1(CC=C)(C(=O)NCC(CC2CC2)OC)CCCN1C(c1cc(CC)n(C)n1)=O N1(C(c2n(C)ccc2)=O)CC(NC(=O)CNC(=O)NC2CC2)CC(C)(C)C1 N1(C(c2c(CC)n(C)nc2)=O)C2CCC1C(C(=O)Nc1cnc(OC)c(C)c1)C2 C(=O)(CC(C1CC1)NC(C)=O)NC(C(=O)NCCC=CCCC)C N1(C(CC(=O)OCC)=O)CCC(C)(NC(=O)C(C(C)C)OC)C1 CCC(F)C(=O)N(C1CN(C(=O)C(C)N(CC(F)(F)F)C)C1)C c1(OC(c2c(CC)nn(C)c2)=O)ccc(OC(F)(F)F)cc1C CCCCCCCC(=O)N1CCC(F)(C(=O)Nc2ccc(I)cc2C#N)C1 c1(C(N2CCCC(NC(c3nccc(C)c3)=O)CC2)=O)cc2nc(C)ccc2o1 C1(c2nnnn2Cc2ccccc2)(NCC(=O)OC(C)C)CC2CC1CC2 N1(C(c2ncn(C(C)C)c2)=O)CCC12CN(C(=O)C=Cc1ccncn1)C2 C(CC(C)C(=O)NCC(C1CC1)N(C)C(c1ccc(C(N)=O)nc1)=O)=CC C1(CNC(COCCOCC)=O)CC2CCC(C1)N2C(=O)CCc1ccc(C)s1 c1(C(=O)NC(C2CCN(C(=O)Cc3ccco3)C2)(C)C)ccc(O)cc1 C1(CCC)CCCC1C(=O)NCCCN(C(=O)CCN1CCCC1=O)C N1(C(C23C(C)OC(CO)(C2)C3)=O)CC(NC(C2CCOC2)=O)Cc2ccccc21 C(=O)(C(C)C(C)S(C)(=O)=O)NC(C)CN(C(=O)CCSc1nnnn1C)C CC1CCn2cc(C(N3CCC(C4CCCN4C(C4CCOC4)=O)C3)=O)nc2C1 C(=O)(C1CCc2cccnc21)NCC(CN(C(CCC(=O)OCC)=O)C)(C)C C(=O)(CCC(F)(F)C(F)F)N1CC(NC(COC(C)C)=O)C2C1CCC2 CC(C)CCC(O)C(=O)NC1(CO)CCN(C(C2(F)CCN(C)CC2)=O)CC1 N1(C(CCC#C)=O)CC(CNC(=O)CSc2nc3ccccc3[nH]2)N2CCC1C2 C1(CNC(c2cnc(C(C)=O)s2)=O)CCCN(C(=O)C(Cl)=CCl)C1 C(=O)(C(c1ccoc1)NC(=O)C=CCOC)N(CC#CC)C CC1CC2(CCC2)CN1CCCOc1cccc(C(=O)O)c1 C(=O)(CCCCn1ccnn1)NC(C)CNC(C1(c2ccccc2)CCOC1)=O Cc1c(NC(=O)NC(C)C(C)C)cccc1C(c1nccc(O)n1)C1CC1 c1(NC(=O)Cn2cncn2)nccc(=NC2CC3(CCC(NCCCF)CC3)C2)[nH]1 N1(C(c2cnc(C)[nH]2)=O)CCCN(C(c2cc(-c3ccoc3)[nH]n2)=O)CC1C c1(N(CCCC)C)ccc(NC(c2csc(Br)n2)c2nnnn2C(C)C)cc1 CC(O)C(F)(F)C(=O)N(C)CC1CCCN1C(c1cnoc1-c1cccs1)=O C1(C(=O)NC(C)C(CO)NC(C2(C)CCCCCC2)=O)CC12CCCCC2 C1(NC(C2(C)CCOC2)=O)CCCCC1CC(=O)NCCN1CCOCC1 Cc1cc(N2CCC(N(C)C(c3cc(C(F)(F)F)cc(Br)c3)=O)C2)nc(C)n1 C(=O)(C#CC1CCOCC1)N1CC(CCCNC(CSCC(C)C)=O)OCC1 c1(C(=O)NC2CC(C)N(C(=O)C(=O)NC(C)(C)C)CC2)cnc2c(c1)CCCO2 c1(C(N2CCN(C(Cc3onc(C)n3)=O)CC2CO)=O)c[nH]c2cc(Cl)ccc12 Cc1nccc(C(=O)NCC(C2CC2)NC(C2CC2Cc2ccccc2)=O)n1 C(=O)(C(C)(C(C)C)N(C)C)NC1C(OC)CN(C(C2(CSC)CCCCC2)=O)C1 CC1(C)CN(C(C2CCN(C(=O)C(C)(C)n3cccn3)CC2O)=O)CC(=O)N1 C(=O)(CCC(=O)NN(C)C)NCC1CCN(C(c2c(C)cc(O)c(Cl)c2)=O)CC1 CN1CC(C(=O)NC2CCCC2NC(=O)C(F)CC2CCOCC2)CCC1=O C1(N(C)CCNC(c2ccccc2NCc2ccccc2)=O)CCCCC1(C)O CCCC(C(=O)N(C1CN(C(=O)CC2=NNC(=O)C2)C1)C)S(N)(=O)=O C(=O)(C(C)(F)C(=O)N(CCCCCC(=O)NCC1=NOC(C)C1)C)OC S(=O)(=O)(c1cccc(=NC(C)c2cccn2C(F)F)[nH]1)NCCCNC(=O)NC n1(CCC(=O)NC2CC(C)(NC(C(CC=C)NC(C)=O)=O)C2)cnc([N+](=O)[O-])c1 C=CCCCC(C)(C)C(=O)NC1CCC(F)(CNC(c2cnco2)=O)C1 C1(CNC(c2c(C)cnnc2)=O)CN(C(=O)CC2CC2(C)C)CC2(CCC2)O1 C(C1CN(c2ccc([N+](=O)[O-])cc2)Cc2ccccc21)NC(C1(C)CC1(F)Cl)=O N1(C(CNS(N)(=O)=O)=O)C2CCC1C(F)C(NC(c1cn3ccsc3n1)=O)C2 Cc1ccccc1C(N1CCCCC1c1n[nH]cc1C(=O)NC1CCOC1C)=O N1(CC)CCCC(C(=O)NC(C2CN(C(C3CCCN3C=O)=O)CCO2)C)C1 C1(C(=O)NC2CCCN(CCc3cccc(Cl)c3Cl)CC2)CCCCC1C1CC1 c1(C(=O)NC(c2c(SC)cccc2)CO)ccc(S(N)(=O)=O)cc1[N+](=O)[O-] c1(C(N2CC(CNC(C(CCC)C)=O)C(F)(F)C2)=O)c(C)nc2sc(C)nn12 C(C(CCO)CC(C)C)NC(CC(C)OC)c1nnnn1C1(C)CC1 c1(C(N(C)CC2(CNC(=O)CC3CCOC3)CC2)=O)c(F)ccc(F)c1Cl Cc1c(Br)ccc(C(=O)NC2C=CC(C(=O)NCc3ccc(Cl)c(Cl)c3)C2)c1F N1(C(C2CCC(OC)CC2)=O)CC(C2CC2)(C(N2CCC(OCC3CC3)C2)=O)C1 C1(CN(C(C(=O)N(C)C)=O)C)CCCN(C(c2ccc(C3(O)COC3)cc2)=O)C1 N1(C(c2on(C)c(=O)c2)=O)CCC2(CCCC2NC(=O)C2=CCCCC2)C1 N1(C(C2OCCN(CC)C2)=O)CCN(C(=O)CCCN2CCOCC2)CC1C c1(C(N2C(C3(NC(c4c(CC)csc4)=O)CC3)CCC2)=O)c[nH]c2nccc-2c1 c1(OC)ccc(F)c(C(N2CC(NC(c3cccc(Cl)c3O)=O)C(O)C2)=O)c1 C1(C(=O)NCCC2N(C(CC3C(=O)NC(=N)S3)=O)CCC2)CCOCC12CCC2 c1(C(N(CC(C)NC(CSCCCC)=O)CC)=O)cnc(OC)cn1 N1(C(C2N(C(C(C)NC(CC)(C)C)=O)CCCC2)=O)CCC2CC1C(=O)N2C N1(C(c2c(C)onc2)=O)CCC2(CC1)CN(C(C1(N3CCCC3)CCC1)=O)C2 C(=O)(N1CCCO1)C1(NC(CC2(C)CCOC2)=O)CCC1 C1(CNC(Cn2cc(C(=O)OC)nc2)=O)C(C)CCCN1C(C1(F)CCCC1)=O C1(O)(CNC(C2C3CCCC23)=O)CCN(C(c2ccc(C(F)F)cc2)=O)CC1 Cc1ccc(F)cc1C(F)(F)C(=O)N(CCCNC(c1cc(Cl)n(C)n1)=O)C C(=O)(C1=CCCOCC1)N1CC(C2CC2)(C(N(C(C#C)C2CCC2)C)=O)C1 c1(OC)cc(C(=O)N(C2CCN(C(=O)Cc3csc(Cl)c3)C2)C)nn1C c1(C(N(CCOCCCNC(CNC(CCC)=O)=O)C)=O)cc(C)c[nH]1 C1(NC(C(C)OCCOCC)=O)CCCN(C(c2ccnc(S)c2)=O)C1C c1(C(N(CCNC(C2COCCC2C)=O)CC)=O)nn(C)cc1S(C)(=O)=O Cc1cc(C2CC2)ccc1C(N1CC2CC1C2NC(=O)CSc1ccccn1)=O CCC(C)(COC)C(=O)NCc1ccc(C(=O)NC2(C)CC2)o1 C(=O)(C(COC)CC(C)C)N1C(CC(=O)NC(CC)C(C)CN(C)C)CC1 C12(NC(c3n(CC)ccc3)=O)CC1CN(C(C1(C)CCSCC1)=O)C2 N1(C(C2CC(CC)C2)=O)CCCC1CNC(=O)Cn1cnc(C(N)=O)n1 c1(CC)nnsc1C(=O)NCC1CC(F)(CNC(=O)C(C#N)C2CC2)C1 c1(-c2cn(CCNC)nn2)ccc(C)c(Oc2ccc(NC(=O)N(C)C)cc2)c1 C1(CCO)(NC(c2nnnn2Cc2cccs2)C2CCCC2)CCOCC1 N1(C(c2n(CC=C)ccc2)=O)CC(NC(=O)C(C)C(C)(F)F)CC12CCOCC2 CC1CCC(C(=O)NC(C)Cc2cnccn2)N(C(=O)CCCC#N)C1 CC1CCN(C(=O)C(C)(C)C#N)CC1NC(c1ncc(Cl)cc1F)=O C=CCC(CC)C(=O)N(CCCCC(=O)NC1CCCCNC1=O)C c1(C(=O)OC)ccc(C(=O)NCC(C)CNC(c2cn(C)nc2Cl)=O)c(C#N)c1 c1(NC(c2cccc(-c3nc(C4CC4)no3)c2)=O)ccc(I)cc1I c1(C(N2CCN(C(Cc3cn(C)nc3)=O)CC2C2CC2)=O)cnn2c(Cl)cccc12 C1(C(N(C2CC(O)C2)C)=O)CC1C1CN(C(c2ccnn2C)=O)C1 N1(C(c2cnn(CCC)c2Cl)=O)CC2CCN(C(=O)CCOC(C)C)CC12 C1(NC(N)=O)CCCC(C(=O)NC(C)CCNC(=O)COc2ccc(Cl)cc2)C1 C1(C(=O)OC)CCC1(C)C(N1CC(C)(NC(C)=O)C1)=O N1(C(c2cc(COC)no2)=O)CCCC2CN(C(=O)CC3=CCCC3)CCCC12 c1(OC)ccc(CCC(=O)OCc2cc(Br)ccc2OC(C)C)cc1O N1(C(C(C(C)C)SC)=O)C(C(=O)NOCc2cccc(C)n2)CCC12CC2 N1(C(C23CC(C)C2C3)=O)CC2(CCCN(C(=O)CCC(N)=O)C2)C1 C(=O)(C#CC1(C)CC1)N(CC(CC)NC(=O)C(c1cccc(Cl)c1)O)C c1(OC)cccc(C2=NOC(C(=O)N(CCCn3cc(C(C)O)nn3)C)C2)c1 C(=O)(C(C)C(F)F)NCCC1(NC(Cc2cnc(C)s2)=O)CC1 N1(C(C=CC=CCC)=O)CCC(CNC(c2cc(N(C)C)ccc2F)=O)C(C)C1 C1(CNC(=O)NC(CCCC)CO)CC2CCCCC12 c1(C(N2CCC(N(C(C3CC(C)(C)O3)=O)CC)CC2)=O)ccc2c(c1)NC(=O)C2 N(C(=NCCC1CCC1)NC1CCC1C(N)=O)C1C(N)CCCCC1 C#Cc1cccc(C(=O)NC23CC2CN(C(C2CC4(CCC4)C2)=O)C3)c1Cl C(C(C)C(C)C(=O)N1CCC(OCCNC(c2cccnc2)=O)CC1)OC CC(C)(C)CCC(=O)N1CCOC(CCCNC(=O)C=Cc2cocn2)C1 C#CCC(C)C(=O)NCC1(CNC(=O)C(O)C2CC2)CC1(F)F C(=O)(N=c1cc(C)n(CCN(C)C)[nH]1)Nc1cc(SC)nn1C c1(SC)nc(N2CCCC2C(=O)NCC2CC(n3ccnn3)C2)cc(Cl)n1 C1(NC(COCC#C)=O)CCN(C(c2ccc(CO)cc2)=O)CC1CCC Cc1nn(C(C)C)c(C)c1C(N1CC(NC(=O)C(C)(C)O)CC(F)C1)=O N1(C(CSCCC)=O)CCC(CNC(C2(c3ccccc3)CC2(C)C)=O)CC1 N1(Cc2cn(CCS(C)(=O)=O)nc2)Cc2cc(Br)cnc2C1.C12CC1C(=O)N2 c1(CNC(c2occc2CNC(C2(Cl)CC2(F)F)=O)=O)ncc(Cl)cn1 N1(C(c2cn(CC)nn2)=O)CCC2CC1CN2C(=O)Cc1cccc2c1OCO2 Cc1c(C(=O)NC(C)CC2CN(C(C3C4CCCC34)=O)C2)oc2c(Cl)cccc12 N1(CCCNS(CC)(=O)=O)CCC(NC(C2(C#N)CC2(C)C)=O)C(C)C1 c1(C(C)(C)C)conc1C(=O)NCC=CCNC(=O)C(C)(O)C1CCOC1 C(=O)(C(O)CCS(C)=O)N1CC2C(CNC(c3c(OC)ncnc3OC)=O)C2C1 O=C(C#CC1CCCCC1)NCC1N(C(C2CCCOC2)=O)CCCC1(C)C Nc1c(C(=O)NCCNC(C2CC(N3CCCC3)C2)=O)nnn1-c1ccccc1 CC(CCNC(=O)CCN(CCCO)C(=O)CN1CCOC1=O)CCO C(=O)(CS(=O)(=O)C1CC1)NCCC1CCN(C(CCc2c(C)n[nH]c2C)=O)C1 C(C)(CCC(F)(F)F)NC(C(CSC)(C)NC(C1CC12CCCCC2)=O)=O c1(OC)nc(C)ncc1C(=O)NCCCCC(C)NC(c1cccc(CO)c1)=O C=CC1(CO)CCN(C(=O)CCC2CCCN2C(=O)CCOCCOC)CC1 N1(C(CCC(C)SC)=O)CCC(NC(C2(F)CCCCC2)=O)C12CCC2 C(CC(C(C)C)NC(=O)CC1(CSC)CC1)NC(C(CC)SC)=O C1(NC(CCc2ccn(C)n2)=O)CC2CC(NC(=O)C3=CCCOC3)C2C1 C1(NC(C=CC=CC)=O)CN(C(=O)CC2(OC(C)=O)CCCCC2)C2(CCC2)C1 C1(CNC(C2C(NC(CC3C(C)=NNC3=O)=O)CC2)=O)CCC(C)(C)CC1 c1(OC)cc(NC(C2(NC(C3COCCO3)=O)CCN(C)C2)=O)ccc1O c1(C(=O)NCCCC2N(C(CCC=C(C)C)=O)CCC2)ccnc(C2CCC2)c1 CC(O)(C(=O)N1CCCC1CC(N1CCCCC(F)(F)C1)=O)C(F)(F)F C1(C(=O)NC2CC(F)(CNC(C=CC)=O)C2)CCn2c(C)nnc2C1 C(C(C(=O)NCc1cc(C)co1)C(C)(C)C)NC(C(COC(C)=O)C)=O c1(C(N(CCCNC(c2cn(C(F)F)cn2)=O)C(C)C)=O)nc(=O)n(C)[nH]1 C1(NC(c2ccc(N3CCCC3)cc2)=O)COCCN(C(=O)C=CBr)C1 N1(C(c2cnc(SC)nc2)=O)CC(NCc2ccc(Br)nc2)C2(CC2)C1 c1(NC2(CNC(C(C)C(C)(F)F)=O)COC2)nc2ncc(Cl)cc2o1 C#CC1CCN(C(C2(CF)CCN(C(C3CC3(Cl)Cl)=O)C2)=O)C1 c1(CCC=CC(=O)NCC2CN(C(C3CN(C4CCOC4)C3)=O)C2)ccccc1 N1(C(c2c(CC)n[nH]c2)=O)CC(CC(N2CCC3CC23C)=O)C2(CC2)C1 c1(C2C(C(N(C3CC(NC(=O)C=CC4CC4)C3)C)=O)CC2)nc(S)n[nH]1 Cn1nc2c(c1C(N1CCC(CNC(c3ccsn3)=O)C1)=O)CS(=O)(=O)CC2 CCC(C)CCCC(=O)NCCC1CSCCN1C(c1cc(SC)n(C)n1)=O c1(CC(=O)NC(CCNC(C=Cc2cncc(C)c2)=O)C)cccc2cn[nH]c12 C(=O)(CCC(=O)NN(C)C)N1CC(C)N(C(c2cc3c(ncn3C)[nH]2)=O)CC1 C1(C)(C(=O)OC)CCCN(c2nn(Cc3ccc(Cl)cc3)cc2I)C1 CC(CCC(=O)NCc1cc(O)ns1)NC(=O)CC(C)(C)O CC(C)(CS(N)(=O)=O)NC(=O)NC1CC(C)(NC(=O)Nc2ccccc2)C1 C1(C(N(CC=CC(=O)OC)CC)=O)CCCC1NC(=O)NC c1(C(=O)NCCOC2CN(C(C(C)C3CCCO3)=O)C2)cccc2sccc12 c1(CC(C(=O)OC)NC(c2c(Cl)csc2Cl)=O)ccc(Br)cn1 c1(OCC)cc(C(F)(F)F)ccc1OC1(CNC(c2cn(CC)nn2)=O)CC1 C(CCC(=O)NCc1ccoc1C)(C(C)C)NC(CCC#C)=O c1(CC)nc(Cl)nc(N2CCC(C)(NC(=O)CSC)C2)c1Cl N1(C(C(=O)Nc2ccc3c(c2)COC3=O)=O)CCc2cc(Br)cc(Cl)c2C1 CC1(CNC(=O)C=CCn2cncn2)CCCN1C(C12CC(O)C1C2)=O N1(C(C2CCC(SCC)CC2)=O)C2CCC1C1CC1(NC(=O)Cc1cnns1)C2 N1(c2n(CC)ncc2)CCCC(NC(=O)NCC2(F)CCOC2)C1=O c1(C(=O)NC2C(C)N(C(c3cn(C4CC4)cn3)=O)CC2)ccc2c(c1)CC2 C1(C(c2n(C(C)C)nnn2)NCc2ccccc2C(F)(F)F)(CO)CCOCC1 C=CCC(CC(C)C)C(=O)NC1CN(C(C2(CF)CCC2)=O)CC2(CCC2)C1 C1(CC(=O)N(C2CSC2)C)CCCC12CN(C(=O)CCc1cccnc1)C2 c1(COCC)cc(N2CCC(C(=O)Nc3cccc(C(C)C#N)c3)C2)ncn1 C1(C(=O)NC2CCCN(C(C3(C(C)C)CNC(=O)C3)=O)C2)CCC(C#N)CC1 c1(C(N2CC(Nc3ncccn3)C3CCCC3C2)=O)cc(F)cc2ccoc12 C1(NC(c2ccnn2C(F)F)=O)CCCCN(C(=O)C=Cc2ccncc2)C1 N1(C(c2cccc(C#N)c2)=O)CCC(NC(C23CC(CO2)C3)=O)C(CO)CC1 C(C)(C(C)NC(=O)NCC1(O)COC1)(C1CC1)OC n1(CCC)nnnc1C(c1sccc1C(=O)OC)NCC1(CO)CC1(C)C C(=O)(C(F)(CC)C(=O)OC)NC(CC1CN(C(c2ccc(NCC)cc2)=O)C1)C C(=O)(C(CCOCCO)NC(c1ccc(O)nn1)=O)Nc1ccc(C2C(C)C2)o1 N1(C(CC(=O)N(C)C)=O)CCCC2C1CCN2C(=O)CSCC1CCCO1 c1(CC(=O)NCCN(C(c2ccn(CC)c2C)=O)C2CC2)c[nH]c2ccccc12 C1(C(=O)N(CCCNC(C2(C)CCCS2)=O)C)(OC)CCCOC1 c1(C(=O)NCC(N2CCC(CN(C(=O)CNC=O)C)CC2)=O)ccc(O)c(N)n1 c1(C(=O)NCCN(CCC)C(C2CCC(=O)N2)=O)cc(C)n(-c2ccon2)c1C c1(C(C)C)ccc(NC(=O)C(N2CCN(CCN)CC2)C)cc1 N#Cc1ccc(N(CCC#N)C(c2ccc(N3CCCC3=O)o2)=O)cc1 C(=O)(C1CC(O)c2ccccc21)NCC1C(CNC(c2cn[nH]c2)=O)C1 N1(C(C2CC(CC)OCC2)=O)CCN(C(c2ccc(Cl)c(O)c2)=O)C2(CC2)C1 CCC(CC)C(=O)N1CC2CC2(CNC(=O)CCC(=O)NC)C1 N1(C(C(=O)NC2CCC2)C2CCSC2)CC2(CC2)CC1c1ccccc1 C(=O)(C(C)(C)CC(C)(C)C)NC1C(CNC(c2nn(C)c(=O)cc2)=O)CCCC1 C1(CC)CC(C(F)(F)F)CCN1C(=O)Cc1ccc(C)cc1Cl C1(NC(CSCCCC)=O)COC2(CCN(C(c3cc4nc[nH]c4cn3)=O)C2)C1 C(C(=O)N1CC2C(NC(=O)CCn3ccc(C)n3)C2C1)(C(C)C)NC(C)=O C#CCCC(=O)NCCCN1CCC(C(=O)NCc2cc(OC)ns2)C1 C(=O)(CS(=O)(=O)N1CCOCC1)NC(CNC(=O)Cn1ncnn1)C1CCC1 C1(CNC(C)=O)CCCN(C2CCN(CC(=O)O)C2=O)C1 C(=O)(C(C)CC(C)C(C)=O)NC(C(=O)N(C)Cc1scc(C)c1)CCF N1(C(C(CC)COC)=O)CCN(C(=O)CCc2ccc(Br)cn2)CC1C C12(CNC(c3ccc(CSC)o3)=O)CC1CN(C(C1CCCO1)=O)C2 CC#CCC(C(=O)NC(C)CCc1cn[nH]c1)NC(c1cnco1)=O c1(C(=O)NC(CN(C(c2nn(C)cc2Cl)=O)CC)C)csc2cc(Cl)ccc12 C(=O)(CC(C)(C)CC(=O)N(C)CC1CCCN1C(c1cccc(=O)o1)=O)OCC C(=O)(C(CC(C)C)N(C(=O)C(C)C(=O)OC)C)NC(c1cn(CC)nc1)C CC1(C)C(CNC(C2(F)CCCC2)=O)CCN1C(c1ncccc1O)=O N1(C(Cn2ncc(C#C)c2)=O)CC(CC(=O)NCCC(C)(C)C)C2(CC2)C1 C1(NC(Cc2c(C)cccn2)=O)CCN(C(=O)CNS(C)(=O)=O)C12CCC2 C(N=C(NC(C)C)N1C(C2CC2)CC2CCCCC12)c1c(OC)cc(C#N)cc1 C1(CC(=O)Nc2ccc(OC3CCCNC3)cc2)CC2CC(N)C2C1 C1(C(N(CCCCCC)C)=O)CCN(C(C2CCCN(CCOC(C)=O)C2)=O)CC1 CC(CC(=O)NCC1CN(C(c2ccccc2)=O)CC12CCC2)C(C)(C)C C1(CNC(CC(CC)C)=O)CN(C(C2CCCC(O)C2)=O)CCC12CCOCC2 C(C(C)(C)CNC(=O)CC1CCOC1=O)N(C(=O)CCc1cnn(C)c1)C C=CC1(C(=O)NCC2Cc3nccn3C2)CCN(C(C2CCC(N(C)C)C2)=O)C1 c1(CCC(=O)OCCC(C)N(C)C)ccccc1 CC1CCCN1C(c1cn(CCNC(C2CC2C2CC2)=O)nn1)=O C(=O)(CCC(C)(C)N(C)C)N1CC(O)(C(C(=O)N(CCCC(C)(F)F)C)F)C1 C(=O)(C(CO)C(C)(C)C)N1CCC(C(=O)NCCc2onc(C)n2)C12CC2 C(C(F)C(=O)NCC1(O)CCSC1)C1CN(C(c2cnsc2)=O)C1 N1(C(=O)Cn2ncnn2)CCCCC1c1cn(CCN2CCNC2=O)nn1 C=Cn1nccc1C(N1CC2CC2(NC(c2cnc(C(C)(C)C)s2)=O)C1)=O CC(C(=O)N(C(C)CN(C)C(c1c[nH]ccc1=N)=O)C)C(=O)N1CCOCC1 N1(C(C2C(CCC)C2)=O)CC2(CCN2C(=O)COc2cc(F)ccc2F)C1 c1(C(=O)NCCN(C(=O)CCc2cnn(C)n2)CCOC)cc(C)c(C)o1 c1(C(=O)NCC2(C(N)=O)CN(C(C(C)OCC#C)=O)C2)cccn(C2CC2)c1=O C1(C(N2CC(C)C(NC(=O)CCn3ccccc3=O)C2)=O)CC(C)(C)OC1=O Cc1cnn(C(C)C(=O)NC2CC(C(C)NC(c3occc3C)=O)C2)c1 c1(CN(C)C(c2n[nH]cc2CNC(c2ncn(C)n2)=O)=O)nccn1C C1(C(C)NC(c2cc(C(F)F)[nH]n2)=O)CCCCN1C(=O)CC(F)F c1(CCN(CC)CC)nc(-c2ccco2)nn1-c1ccc(OC(F)F)cc1 C(C)(CCC(=O)NC12CC(C1)N(C(c1cc(-c3ccccc3F)no1)=O)C2)SC CC1CS(=O)CCN1C(=O)CC1CCCN1C(=O)CN1CCCCC1C N1(C(C2CC(C)(C)CN(C(=O)CC34CCCC3C4)C2)=O)CCC12CCCOCC2 c1(C(N(C2CCCC(NC(=O)CO)C2)C)=O)cccc(Cl)c1 C1(N(C(c2cc(CC)ncc2)=O)C)CN(C(C2CCCN2C)=O)CCC1C C(=O)(C1CCCc2nc[nH]c21)N1CC2(CC(NC(COCCC=C)=O)C2)C1 N1(C(c2cc(C#N)on2)=O)CCCC(NC(c2ccc(N3CCC3)nc2)=O)CC1 C1(CNC(c2ccc(C#C)o2)=O)CN(C(c2cc(C)sc2C)=O)CCC1C N1(C(C2(CCOC)CC2)=O)C2CCC1CN(C(=O)CCC1CC1)CC2 N1(C(C2CC(C#C)(O)C2)=O)CCC2CC(CNC(=O)C3=COCCO3)CCC2C1 N1(C(C2N(C(c3nc(COC)oc3)=O)C3C(F)CC2C3)=O)CCCC12CCCC2O N1(C(COCC(C)C)=O)C(CNC(=O)C=CC=C(Cl)Cl)CC2CC12 c1(C(N2CC(O)(C(C(=O)NC(C(=O)NC)C3CC3)F)C2)=O)ccc(C#N)o1 O(NC(=O)CNC(=O)C(CC1CC1)NC(=O)CC1(COC)CC1)CCOC C1(C(N(C2CC(NC3CCCN3C(=O)C(=O)N(C)C)C2)C)=O)CCCCCC1 c1(C(=O)NCC(=C)CCNC(=O)CC2CC(F)C2)cnc(O)n(C)c1=O C1(C(C(=O)NCC(C)C)(C)C)CCCCN1C(=O)COC(=O)Nc1ccccc1 c1(OCC)c(OC)cc(C(=O)NC(CNC(C23CC(C2)C3)=O)CC)cc1Cl C1(CNC(c2coc(C(F)F)n2)=O)CC2CCCC(C1)N2C(=O)C(F)C1CCC1 N1(C(C2N(C(N)=O)CC(O)C2)=O)CCC2(C1)CN(C(c1cc(CO)ccn1)=O)C2 C1(N(C)C(C2CC(OCC)CCO2)=O)CCN(C(c2cn(C)c(C)n2)=O)CC1 N1(C(c2c(NC)nccc2)=O)CC2(CCC2)CC1C(=O)NC1CC(F)(F)C1 C#CC12CCC(C(=O)N(CC(C)NC(C3CCC(COC)CC3)=O)C)(CC1)CC2 CC1OCCC1C(N1CCC1CN(C(=O)CCC1CCC(=O)C1)C1CC1)=O N1(C(CC2C(C)C2)=O)CC2CCC(C1)C(NC(C1CCOCC1(C)C)=O)C2 C#Cc1cccc(C(=O)N(C)CCOCCN(C)C(C23CC(CO2)C3)=O)c1F N1(C(c2ccc(-c3ccc(OC)cc3)o2)=O)CC(C(=O)O)CCC1C N1(CC)CCN(CC(N2CC(NC(=O)C(F)=CC3CC3)C2)=O)CC1 C1(C(N(CC(C)N(C(C)=O)C)C)=O)(NC(c2cc(O)ncn2)=O)CCN(C)C1 C1(N(C(=O)NC2CC(C(C(=O)OCC)F)C2)C)CCc2cc(Br)ccc2C1 c1(C(=O)NCC(CC=C)NC(c2ccc(CO)s2)=O)ccc(O)c(F)c1F C(C)(C)(C(=O)N(CCCCCNC(C1(C(F)F)CCCC1)=O)C)NC(=O)OC c1(SCC(=O)NCCN(C(=O)NC)CC)ccc(S(=O)(=O)N2CCOCC2)cc1 C(=O)(CCC(=O)NN(C)C)NC(C(=O)N(CCC1CN(C)C1)C)CCC1CCC1 c1(C(=O)NCCOCCCN(C)C(c2ccc(F)cc2)=O)ncncc1Cl c1(NCC2(NC(C(C=C)O)=O)CCCCC2C)ccnc2ncnn12 c1(C(=O)NC2CSC2)cn2cccc(Br)c2n1.C12CCC(CC1)C(=O)NC2 CCC(CC)(CC)C(=O)NC1CCC(CNC(c2cc3n(n2)CCCC3)=O)CC1 S(=O)(=O)(c1cn(C)cn1)NCC(N1C(CNC(C(C(C)C)NC=O)=O)CC1)=O c1(C(=O)NC(CNC(C(C)(CO)OC)=O)CC(C)C)ccc(F)c(Cl)c1 CCC(COC)C(=O)NCCCN(CCCCNC(C1CC1CC)=O)C CC1CN(C(C2CC23CCC3)=O)CC1NC(c1cnccc1N1CCOCC1)=O c1(OC(C(=O)NC(C)CC2CN(C(c3ncc[nH]3)=O)C2)C)ccccc1Cl c1(C(=O)NCc2cn(C3CC(CC(=O)OC)OCC3)nn2)cc2sc(C)cc2s1 C1(CN(C2CNCCOC2)Cc2n(C)ccn2)CC2(CC(=O)C2)C1 CCCCCCCCC(=O)O.N1(Cc2n(CC)ccn2)CCN(C2=NCCS2)CC1 N1(C(c2c(C)nc(COC)s2)=O)CC(NC(c2cnc(Cl)n2C)=O)CC(C)C1 N1(C(C(CCC)(C)O)=O)CCC2(CC1)CN(C(c1ccc(OC)nc1C)=O)C2 N1(C(COCCC=C)=O)CCN(C(C2CC2C(F)(F)F)=O)CC1C1CC1 C(=O)(C(C)(C)CCCF)N1CC(OCC)(CNC(=O)C(c2cccc(F)c2)F)C1 C(=O)(C(C)CS(C)=O)N(CCNC(c1n[nH]c(C)c1Br)=O)C(C)C c1(C(=O)NCC2OCCN(C(C3(COC)CCOC3)=O)C2)cc(O)cc(Cl)c1 N1(C(CCCN(C(=O)COC(C)(C)C)C)=O)C2COCC1C2 N1(C(CC(C)O)=O)CCCC12CCCN(C(c1ccc(-c3cccs3)[nH]1)=O)C2 N1(C(=O)Cc2cscn2)CCCC(F)(C(=O)NC(CC2CC2)CC2CC2)C1 C1(CNC(c2c(C)nc(O)s2)=O)CC2CCC(C1)N2C(C1CCN(C)C1=O)=O C1(C(=O)NC(c2ccn(C)c2)C(=O)O)CC2CN(C(=O)OC(C)(C)C)CC1O2 Cn1nc(C(=O)NC(C2CCCCC2)C(=O)NCC2CCC(=O)NC2)cc1C#N c1(C(N(C(CCNC(CCC#CC)=O)C)C)=O)cnc2ccc(C)cn2c1=O c1(C(=O)NC(C)Cn2cc(C3(C)CCCO3)nn2)c(F)cccc1Br C1(C(N2CC(CCNC(=O)Cn3nccn3)C2)=O)CC2CSCC(C1)C2 c1(C(=O)NC(C2CN(C(C3CCC3c3nc[nH]n3)=O)C2)C)ncn(C(C)(C)C)n1 Cn1cnc2c(C(N3CC=C(CNC(=O)C(C)(F)C(C)(C)F)CC3)=O)cccc12 Cc1cc(C(=O)NC2CN(C(C3CCCC3(C)C)=O)CC2O)cc(C)c1Cl C(C)(CC(=O)NCc1ocnc1C(=O)N(CC(C)C)CCO)OC C(C1CCCCC1)=CC(=O)NC1CCCCC1NC(=O)CC1CCCC1 CC1CC(=O)NCC1C(=O)NCCCOCCC(=O)NCC1CCCCO1 N(C1CCCc2ccoc21)C(C(CC(C)(C)NC(CCC1(C)N=N1)=O)F)=O C1(NC(c2csc(C(F)(F)F)n2)=O)CCC(CC(N2CCCCC2CO)=O)CC1 N1(C(C(CCCOC)C)=O)CCC(F)(F)C(CNC(=O)CCCn2ccnn2)C1 c1(C(=O)NCC2N(C(c3n(C)ncc3)=O)CCCCC2)cccc2cncn12 CC1CN(C(C2(C(=O)NC3CC3)CC2)=O)CCC1N(C(=O)CP(C)(C)=O)C C1(Cn2cc(CCSC)nn2)C(C2CC2)CCN1C(c1cnc(O)o1)=O CCC(CO)C(=O)N1CC(O)(CCNC(=O)C(n2nnnc2C(C)(C)C)C)C1 c1(OC)ccccc1C(c1ccccc1)NC(=O)CNC(C1CCN(O)C1=O)=O N1(C(C2CCN(CC(C)C)C2)=O)CCC(F)C(NC(=O)CCCN(C)C(C)C)C1 CCCCCCCN(C1CCCCC1)C(c1cc(C)on1)=O c1(OCC(C)OC)cc(Cl)c(Cl)cc1C(c1nnnn1CCCSC)NC1CC1 c1(OC)cc(C(=O)NCCN2CCCOCC2)ccn1 CC(N=C1NS(=O)(=O)c2ccccc21)C(=O)N(CCO)Cc1cccc(Br)c1 c1(C(=O)NC2C(NC(C(C)OCC)=O)COCC2)cc(Br)cc(C)c1F CCN=c1ccc(C(=O)NCCC2CN(C(c3csc(CO)n3)=O)C2)c[nH]1 CS(=O)(=O)c1ccc(CNC(C(=O)C(F)(F)F)c2ccccc2)s1 c1(C(N2CCN(C(C(C)(C)SC)=O)CC2CCO)=O)ccc2n[nH]cc2n1 N1(C(C(C)NC(=O)CC(F)(F)F)=O)CCC(NC(=O)CCc2cncs2)CC1C Cc1[nH]cc(C(N2CCC(F)C(NC(=O)Cc3c[nH]ccc3=O)C2)=O)c(=O)c1Cl C(N=c1[nH]c(=N)[nH]c(=NCc2cc(-c3ccccc3)on2)[nH]1)C1CCN(CC)C1 c1(C(N2CCC3CN(C(c4cc(SC)oc4)=O)C3C2)=O)cc2ccc(F)cc2[nH]1 C1(C#N)(C(N(CCCNC(c2c[nH]nc2C2CCOC2)=O)CC)=O)CCCOC1 CC1CC(O)CN(C(=O)C(C2CCCN(C(=O)CCn3cnnn3)C2)(C)C)C1 C12(C(NOCC=C(C)C)=O)CC(CO1)N(C(c1ccc(CF)cc1)=O)C2 C1(C(C(=O)NCCN(C(C(C(C)C)SCC)=O)CC2CC2)O)CCS(=O)(=O)CC1 C1(CCO)(NC(c2n(CCCCCC)nnn2)c2ccncc2)CCOCC1 CC1(C)C(NC(=O)C(=O)NCC(F)(F)F)CC1CNC(=O)CNC(=O)COC CCCCC(CC)CC(=O)NCC1(F)CCN(C(c2c(C(C)C)n[nH]c2C)=O)C1 N1(C(C2CCN(C(COC)=O)C2C)=O)CCC2(CC1)CSC2 c1(CN(C)C)cc(C(=O)N(CCCNC(=O)C(C)(F)c2ccccc2)C)ccn1 N1(C(C2(SC)CN(C(C3Cc4nccn4C3)=O)C2)=O)CCOCC(O)C1 C=CCC(CC(C)C)C(=O)NC(C)(C(=O)NCC1(CC)CCCCO1)C1CCC1 N1(C(C(CC)N2CCCC2=O)=O)CCC(C)(NC(c2cc(C3CC3)ncn2)=O)C1 C(=O)(CCCCC(=O)N(C)CC1(O)CCN(C(C2CC(O)CN2C)=O)CC1)NC C=C(C)CC(C(=O)N1CC2CC1CC2O)NC(c1ccsc1Cl)=O C1(NC(COCCC#C)=O)C(C)CN(C(c2cnc3ncccn23)=O)CC1C C(=O)(CC(C(F)(F)F)NC(C1(C)CC(C)(C)C1)=O)NCc1n(C(C)C)ccn1 c1(C(N2CC=C(CNC(C(C)SCCCC)=O)CC2)=O)ccc2sc(O)nc2c1 N1(C(c2c(CC)cns2)=O)CCCC(NC(=O)CCN(C)CC)C1C C(=O)(C(C)(C(C)C)NC(C)=O)NC(CNC(c1cc(CC)oc1C)=O)C1CC1 N1(C(C(CC)C#N)=O)CCN(C(c2cccc3oncc23)=O)C2COCC12 O=C1CCC(C(=O)NCCc2n[nH]cc2C(=O)NCC2(O)CCOC2)N1 C1(NC(C2CCS(=O)(=O)CC2)=O)CC2(C1)CC(CNC(C1CC3CCC1O3)=O)C2 C12(C(N(C3CN(C(Cc4c(C)ccs4)=O)CC3F)C)=O)CC3CC1(CO)CC3C2 c1(C(=O)NC(C(N2CCCC(OC)C2)=O)(C)C2CCC2)cc(=O)n(C)cn1 CC(C)C(CCN(C(=O)C(C)(O)c1ccccn1)C)NC(C1(C)CC(C)(C)C1)=O C1(NC(c2c(C)coc2)=O)CCC(C)(C)CC1CNC(c1ccnn1CCF)=O CCC(CN(C)C)C(=O)N(CC(=O)NC(c1ccn(C)n1)C)C S(=O)(=O)(c1cccc2c(C)ccnc12)NC1c2ccc(OC)cc2OCC1 c1(C(N(C)Cc2nc[nH]n2)=O)cc(CNC(=O)CSc2ccon2)[nH]n1 c1(N2CC=CC(NC(c3c(OC)cc(Cl)cc3)=O)C2)nc(C)nc(C)c1F C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(C(C)NC(c2ccc(Cl)c(F)c2F)=O)C1 c1(OC)cc(CC(=O)Nc2cccc(CF)c2)c(Br)cn1 C1(C(=O)OCC(=O)CCC2CCCCO2)CCC(O)C1O Cc1ccnnc1N(C(c1ccccc1Cl)CNC(=O)COCC1CC1)C(C)C C1(C(=O)NCCN(CCCC)C)OCCC1NC(C1CCC1C)=O C1(C(=O)Nc2cn(C3CN(CCOCCOC)C3)nc2)CC(S(C)(=O)=O)C1 CC1CC(NC(=O)C=Cc2cc[nH]n2)CCN1C(c1cc(Cl)ccc1F)=O C1(C(N2CC(CN(C)C(c3csc(-c4cnc[nH]4)n3)=O)C2)=O)CCCC1C1CC1 CC1Oc2c(C(=O)N=c3ccn(-c4ccnc(C)c4Cl)[nH]3)cccc2C1C N1(C(CCC(C)(C)C)=O)CC(NC(=O)CC2CC(F)(F)C2)C2(CCC2)C1 C(=O)(C(C)(C)CCC#N)N1CCCC(CCNC(C2(CC)CC2(F)F)=O)C1 C(=O)(CCCCCNC(c1cocc1C)=O)N(CC)CC1CCCO1 c1(NC(CC2OCCN(C(C3C(C)C3)=O)C2)=O)nnc2n1CCCCC2 N1(C(C=CC=CC)=O)CC2CCC(C1)N(C(c1cn(C)nc1Cl)=O)C2 N1(C(C=CC=CC)=O)CCN2CCN(C(c3ccc(F)cc3Cl)=O)CC2C1 c1(C(N(C2CC(C#N)C2)CC(=O)NCc2snc(C)n2)=O)cnc2ccccn12 C12(C(=O)NCC(C)(CO)NC(c3n(C)nc(O)c3)=O)CC3CC(C(=O)N1)C2C3 N1(C(CC2CCC(NC(C(CC)(C)CC)=O)C2)=O)CCC2(CCN(C)C2)C1 C(=O)(C1CCCn2cncc21)N1CCCC(O)(CCNC(C2(C=C)CCC2)=O)C1 Cc1nn(C2CC2)cc1-c1nc(-c2coc(C(C)(C)C)n2)no1 N1(C(C(N2CCNC2=O)C)=O)CCN(C(=O)C(C)(F)F)C(c2cccc(Cl)c2)C1 c1(C(=O)OCC)coc(CNCC(C2CCCO2)O)n1 C1(CNC(c2c(C(C)(C)C)n[nH]c2)=O)(CO)CCN(C(=O)CC2OCCO2)CC1 N1(C(CC(C)(C)O)=O)CCc2c(C(N3CCNC(=O)C3)=O)cccc2C1 C12(NC(=O)C=Cc3cccc(O)c3)CCCC1CN(C(C1CCOCC1)=O)C2 c1(OCC)ccc(C(=O)NC2CCCC(NCC(F)CO)C2)c2ccccc12 C1(CNC(CCCCC)=O)CCN(C(C2COC(=O)N2C)=O)CC1C C1(NC(C(c2cncnc2)C)=O)CCC(NC(=O)Cc2cccc(CO)c2)CC1 CN1CC(NC(C2CC(N(C)C(c3ccc(C4CC4)o3)=O)C2)=O)CC1(C)C N1(C(c2ccc(C)s2)=O)CCOCC1CN(C)C(C1CCN1C)=O C1(C(N2CCC(C3CC3)(CNC(C=CC)=O)C2)=O)CCc2nc(C)cn2C1 c1(C(=O)NCC2C(C)(C)CCN(C(=O)CC#N)C2)ccc2c(O)nnc(O)c2c1 N#Cc1c[nH]ccc1=NCC1(O)CCCN(C(C2CCc3ccccc3O2)=O)C1 O=C(C#CC1CC1)NCC1(CNC(C2C=CC2C(=O)OC)=O)CC1(F)F C1(C(=O)NCC(C(C)(C)C)NC(Cn2c(C(C)C)ncc2)=O)CCCC2(CC2)C1 C(S(=O)c1ccccc1)c1c(C(=O)OC)occ1 C(=O)(C(=O)N=c1[nH]n(C(C)C)cc1C)NC(CC)CNC(C1CCC1)=O N1(c2ccnc(NCC3(CF)CCC3)n2)CCC2(CCC3(CC2)OCCO3)C1 CC1CC(NC2CCCCCC2c2ccc(Cl)cc2)CC(C)(C)C1 c1(C(N(CCNC(c2cc[nH]c2C2CC2)=O)C2CC2)=O)cc(F)cnc1O N1(C(C(C)C2CCC2)=O)CCC12CN(C(=O)CNC(=O)CN(C)C)C2 C1(CNC(c2cc(CO)[nH]n2)=O)COCCN(C(=O)CC2CCCCC23CC3)C1 C12(C(C)C)COC(CNC(c3cccnc3C(N)=O)=O)(C1)C2.C12CC1CNC2=O N1(C(C(C=C)(F)F)=O)CCCC2(C1)CN(C(=O)CCc1cncnc1)CCO2 c1(CN2CC3C(C(=O)Nc4c(C)cccc4Br)C3C2)cc2ccccc2o1 C#CC1(O)CN(C(C2CC=CCC2NC(=O)CC2CCCC3CC23)=O)C1 CC1(C)C(NC(c2cc(CO)[nH]n2)=O)CC1CC(=O)NCCn1cccnc1=O c1(NC(c2ccsc2Cl)=O)ccc(C2(Nc3ncncc3F)CCC2)cc1 C1(CNC(CCN(CC(C(C)C)C)C)=O)CN(C(C2CCCCC2)=O)CC1C.C1CC1 C1(C(=O)NCc2n(C)ccc2)CC2OCCC2N(C(c2ccc(C=O)s2)=O)C1 CCC(CC1CCCCC1)C(=O)N(CCCNC(c1c(C)nsc1N)=O)C C1(CNC(C(c2ccnn2C)C)=O)CC(F)CN1C(C1CC1(C)C(F)(F)F)=O CC(C)(C(=O)NCc1c[nH]nc1C(=O)NCCC1CCCC2CC12)C(F)F C1(CN(C)C(=O)NC23COC(CC(=O)OC)(C2)C3)CCCN(CC2CC2)C1 C1(CNC(c2c(C)cco2)=O)CN(C(=O)C(O)CC(F)F)C2(CCC2)C1 Cc1cccc(F)c1C(=O)NCC(C1(O)CCN(C(c2coc(CO)c2)=O)C1)C C1(C2(O)CCOC2)(C(=O)OCC(c2ncc(Br)cc2F)=O)CC1 c1(CC)cc(C(=O)N(CCC(=O)NC2C3COCC23)CCO)n(C)n1 c1(N(C)C)ccc(N(CCCc2ccco2)C)cn1 N1(C(CC)=O)CC2COCC(C1)N2C(c1[nH]cnc1-c1cn[nH]c1)=O c1(C(N(CCOCCN(C(CSCCC)=O)C)C)=O)cc(C(C)=O)cn1C C1(NC(CC2CCN(C(CN3C(C)CCC3)=O)C2)=O)CC2CC3C(C2)C13 N1(C(C2OCCN(C)C2)=O)C2CCC1CC(O)(CNC(=O)Cc1ccsn1)C2 N1(C(c2nc(C)oc2)=O)CCSCC1C(=O)Nc1ccc(-c2ccsc2)nc1 N1(C(c2nccc(C)c2)=O)CCCC(C(=O)NCc2cc(C)ns2)CC1 C(=O)(CC(C)C(C)(C)CC)NCCC1CN(C(C=CCCC=C(C)C)=O)C1 Cc1ncc(C(N2CCC(O)(CN(C(=O)C(CO)N(C)C)C)C2)=O)cn1 N1(C(C(COC)OC)=O)CC(NC(c2nocc2C2CC2)=O)C(C)(C)C1 Cc1cccc2cc(C(=O)NCC3CCCCN3C(C3CC4(CC4)CO3)=O)[nH]c12 c1(C(=O)NCC(CC)NC(c2ccnc(C)c2)=O)cn2cc(C)ccc2n1 c1(OCC(=O)NCC2N(C(C3N(CCOC)CCC3)=O)CC2)ccc(Cl)cc1 c1(NC(N2C(COC)CCOCC2)=O)cccc(C#Cc2ccccn2)c1 n1(CCOCC)nnnc1C(c1cc(OC)ns1)NC1CC(CC(N)=O)C1 c1(C(=O)NC2(CCCNC(C(C)SCCCC)=O)CC2)nc2cc(F)ccc2s1 c1(C(N(CCC)CCNC(=O)CCC(C)C)=O)ncnc2c1c(Br)cn2C Cn1ncc([N+](=O)[O-])c1NCCC1CCN(C(c2cc(Cl)nc(Cl)c2)=O)C1 c1(OC2(C(=O)NC(CC)CNC(c3ccc(F)s3)=O)CC2)ccccc1F C1(NC(C2C(C)CCO2)=O)CCN(C(=O)C=CC(=O)N(C)C)CCC1CO N1(C(CC2(C)CCC2)=O)CC(F)CC1CC(=O)NC1C=CCCCC1 N1(C(C(C)N(C(c2ccc(CN(C)C)[nH]2)=O)C2CC2)=O)CCC(CCCO)CC1 N1(C(C2CNC(=O)N2)=O)CC2(CCN(C(c3cnccc3Br)=O)C2)C1 C1(C(=O)Nc2ccc(COC)cc2)(CC)CCCN(C(=O)COCCF)C1 CC1CCC(NC(c2cscc2Cl)=O)CN1C(C1NC(=O)OC1C)=O N1(C(C(C)Oc2ccccc2Cl)=O)C2CCC1CN(C(C1CC1(C)C(F)F)=O)C2 N1(C(C2CCN(CC)CC2)=O)CC2(CCCC2)C1C(N1CCC([N+](=O)[O-])CC1)=O n1(CCC)nc(C)cc1C(=O)NC1CCCCC1CNC(c1ncsc1CC)=O C=C1CCC(CNC(=O)CCOCCNC(c2cnn(C(C)C)n2)=O)CC1 c1(C(=O)NCC(CNC(c2c(CC)con2)=O)F)ccc(C(C)C#N)cc1 N#Cc1cncc(CNC(=O)CCC2CCCN2C(C2CCC(O)C2)=O)c1 c1(C(=O)NCC2CCN2C(C23CC4CC(CC2C4)C3)=O)ccc2c(c1)COCO2 C1(CCNC(c2cc(C)[nH]n2)=O)CCN(C(C2C=CC=CC=C2)=O)CC1 C1(C(N(C)CC2(O)CCN(C(c3cc(Cl)cnn3)=O)C2)=O)CC2COCC(C1)C2 N1(C(=O)Nc2ccc(C(=O)OC)c(C)c2C)CC2CCCCCCC12 C1(C(=O)NC(C2CCCCO2)CC)CCCCC1NC(=O)C=C(C)c1ccco1 C1(CNC(C2C(CNC(C=CCC)=O)CCC2)=O)CC(=O)N(CC)C1 N1(C(C(C)OCC2CC2)=O)CC2CN(C(c3cc4sccc4s3)=O)CC2C1 N1(C(C(C2CC2)OC)=O)CC2CCCC(C1)N2C(=O)C(C)c1ncco1 Cc1ccc(C#N)cc1C(=O)NC1CCCC1NC(=O)C(C(C)C)NC=O N1(S(=O)(=O)c2cn[nH]c2)CCC2CN(c3ncnn4cc(Br)cc34)CC2C1 c1(C(=O)OC)ccc(C(CO)NC(=O)Nc2ccc(-c3ccoc3)cc2)cc1 C1(C(=O)NC2C(C)CN(C(=O)C(C)O)C2)CNC(=O)CC1(C)C C1(NC(=O)CCC2CCOC2)CCN(C(C2CC3C=CC2C3)=O)CC12CCC2 c1(OCCOC)ccc(CNC2CCCC(C(=O)OC)CC2)cc1-c1nn[nH]n1 N1(C(CN(c2c3c(nn2C)CCC3)C)=O)CC(NCCOC(F)(F)F)CC(C)(C)C1 c1(C(N(C(C(=O)NCCCC(=C)Cl)C)CC)=O)ncncc1C Cc1ccc(F)cc1C(F)(F)C(=O)NC(CNC(c1c(Cl)cnn1C)=O)C(C)C C(=O)(C(C)(C)C(=O)NCC1CC(C(=O)Nc2ccccc2C(C)C)CO1)OCC N1(C(C(C)c2ncco2)=O)CCCC(F)(CNC(c2cc(O)ncn2)=O)C1 CC(CC(=O)N1CCC2(CC(C(N3CCC4(C=CCO4)C3)=O)C2)C1)CC(C)(C)C c1(CNC2CC3N(C(c4c(CC)cno4)=O)C(CC3)C2)c(F)cccc1[N+](=O)[O-] C1(C(=O)NCC(C(C)C)(C)NC(=O)C(Cl)=CCl)CC12CCOc1ccc(F)cc12 N1(C(C(CC)OC)=O)CC(NC(c2c[nH]c(Br)c2)=O)CC12CCCCCC2 CCS(=O)CC(=O)NCC1(COC(c2cncc(OC(C)C)c2)=O)CCOCC1 c1(C(=O)NCC2CCC(C)N(C(c3ccc(O)cc3)=O)C2)cccc(N=[N+]=[N-])c1 C(=O)(C(F)C(C)C(F)(F)F)NCCC(C)(C)NC(c1ccnc(OC)c1F)=O c1(NC(C)=O)ccc(C(N2CC3CCC3(CNC(c3cnn[nH]3)=O)C2)=O)cc1F CCC(C)(C#N)C(=O)N(C(C)(C)CC(=O)NCC1CC(=O)N(CC)C1)C C1(C)(CNCC(C)C)CS(=O)(=O)CCO1 C12(C(=O)NC(CCN(C(CNC(=O)OC)=O)C)C(C)C)CCC(C1)C2(C)C N1(C(C(C)(F)F)=O)CCC2(CCCC2NC(=O)CC2CC=CCC2)CC1 CC(CCNC(=O)Cc1cnccc1Cl)CCNC(=O)COc1ccc(F)cn1 c1(CN(CCC)CCNC(C2CC2(F)F)=O)nnn(CCO)n1 CC1CN(c2nncs2)CCN1C(c1coc(Br)n1)=O CC(C)CC(C)CNC(c1ccccc1C(C)(C)CNC(=O)OC(C)(C)C)=O c1(NC(NCC(CN(C(=O)OC(C)(C)C)CC)C)=S)ccccc1 c1(CC)nonc1C(=O)NC1CCC(CNC(=O)C(CC)Oc2ccccc2)C1 N1(C(c2ccn(C)c(=O)c2)=O)CC2CC(C1)C(CO)C2NC(C1CCCCC1)=O c1(C(=O)NCC2CCN(C(C(CC)OCC)=O)C2)cccc[n+]1[O-] C1(c2n(CC=C)nnn2)(NCCOC2CC2(F)F)CCC2CCCC2C1 Cc1nc2cncc(C(=O)NCCCCNC(=O)C(C)OCC3CCCO3)c2[nH]1 c1(CC(=O)NCC(N2CCOC(CNC(C3CCCC3)=O)C2)=O)ccccc1Br C1(CNC(c2c(C#C)c[nH]n2)=O)CN(C)CCN1C(=O)Cn1ccc(C(F)F)n1 c1(C(C(C)C)NC(=O)NC(c2ccc(C)cc2C)(C)C)nc2c(s1)CCCC2 Cc1nn(C)c(C)c1C(C)C(=O)NCC1CN(C(=O)CCn2ccnn2)CCO1 CC(C)CC(O)C(=O)N1CCN(C(=O)COC2CCCCC2C)C(CCO)C1 N1(C(CCOCC)=O)CC2CC(C1)C2N=c1cc(C)c(C#N)c(C)[nH]1 c1(CNC(C2CCN(Cc3ncc[nH]3)CC2)=O)ccnc(Cl)c1F CC(CC(=O)NC(C)CC(=O)N(C)CC1CC1(C)C)n1ccnc1 C12(C(=O)NC(C(=O)OC)C(C)C)CCC(CN(C(C3CNC(=O)N3)=O)C1)C2 N1(C(C2(CC#C)CCOC2)=O)CC(NC(c2cn(C)cc2C)=O)C(O)C1 N1(C(c2ccc(SCC)cc2)=O)CC(CNC(c2[nH]cnc2CC)=O)C2(CC2)C1 c1(C(=O)NC(CNC(C2(CC)CCOC2)=O)CC)sc2ccc(C#N)cc2c1C c1(-n2cc(C3CCN(C(CCN=[N+]=[N-])=O)C3)nn2)c(Cl)cccc1Cl N1(C(C(C(C)C)F)=O)CCC2CCCC(C1)N2C(c1ccc(CN=[N+]=[N-])o1)=O Cc1c(C(=O)NCC2CC2CNC(C2(CF)CC2(F)F)=O)cnn1C c1(C(N2C3C(C(N4CCC(F)C4)=O)C(C3)C2)=O)cc2ccccc2cc1O N1(C(C(C2CCOCC2)OC)=O)CCCC(NC(c2cnnc(O)c2)=O)C1 CCC(O)C(F)(F)C(=O)NCC12CC(CO1)N(C(c1ncc(Cl)cc1Cl)=O)C2 Cc1cn2c(n1)CCC(C(N1CC(NC(c3c(C)ncnc3O)=O)CC1C)=O)C2 C1(CCC)(NC(C(C)OCC#C)=O)CCCN(C(=O)COCC2CC2)C1 N1(C(c2ccc(C(C)(C)C)o2)=O)C2CCC1CC(NC(C1CCOC(=O)N1)=O)C2 c1(C(N2C(COC)CN(C(=O)C3=CCC3)CC2)=O)ccc(Br)c(Cl)c1F C1(NC(C(C)=CC=C)=O)CCCC(C(N2CCS(=N)(=O)CC2)=O)CC1 N1(C(CSCCOC)=O)CC2(CCCC2)C1C(=O)NCCN1CCOC(C)C1 N1(C(COCCCCCC)=O)CCC2(CC1)CC2NC(=O)C(C)CC(F)(F)F CC(CCS(C)(=O)=O)NC(=O)C(O)CC1CC(F)(F)C1 c1(CCN)cc(C)ccc1OC.C1(CC)(c2nnnn2C)CC1CC C1(CNC(C=CCC)=O)CN(C(=O)CC2CCC(C)(O)CC2)CCN1C C(=O)(CCCC(C)(C)C#N)N(C1CN(C(C2(F)CCOC2)=O)CC12CC2)C C1(C)(C(=O)NCC2(C(C)NC(c3cc(O)n(C)n3)=O)CC2)CCCC1(F)F c1(C(=O)NCC(C)(CC)NC(CC(CC)C2CC2)=O)cnc(OC)cc1C(F)F Cc1ccc(NC(=O)C(=O)NC2CN(C3CC3)CC2C)cc1S(C)(=O)=O C1(NC(C(=Cc2ccco2)C)=O)CCCC(CNC(C2C(C)C2C)=O)C1 C1(NC(C2C(CC)CCO2)=O)CC2CC1CN(C(C1CCC(C)CC1)=O)C2 CC1CCN(C(=O)Cn2cc(C#N)cn2)CC1CNC(c1csc([N+](=O)[O-])c1)=O C1(C(C)(C)NC(C(C)N2CCCC2)=O)CCCN1C(C1CCN1C)=O C(C(C)CC(C)C)N1CC(CC=C)(NC(C2CCCN2C2CC2)=O)C1 C1(NC(NCC2(C(C)C)CC2)=NCCC2CC2)CCC12CCCCC2 N1(C(c2c(C)non2)=O)CCC(C)(C)C1C(=O)N(CC(O)C(F)(F)F)C c1(CC(N2CCCC(NC(Cc3c(C)nsc3)=O)C2)=O)cccc(F)c1F N1(C(c2ccc(Cn3cc(Cl)cn3)cc2)=O)C2CCC1c1ccccc12 C(C(C)(C)C#CC(=O)N1CCC(C)CC1C)NC(c1n[nH]c(CC)c1C)=O C(=O)(C(=O)C(F)(F)F)NC1(CN(C(=O)CC(O)C2CC2)C)CC1 c1(CC(=O)O)cccc(NC(c2cn(C3CC3)nn2)=O)c1 c1(C(N(C2CCN(C(c3c(C)noc3C)=O)CC2)CC#C)=O)cncc(CC)c1 CCC1=NOC(C(=O)NC(C(=O)NCC2(C3CCC3)CC2)c2ccoc2)C1 n1(CCC)ccc(CNC(c2ccnn2C)c2nnnn2C(C)C)c1 Cc1cc2c[nH]nc2cc1C(N1CCCN(C(C2(C)CC=CCO2)=O)CC1C)=O N1(C(C2(C)C(C)OC(C)(C)O2)=O)CC23CCCCC2(C1)CN(C(=O)CCCF)C3 CC(C)CC(F)C(=O)N(C1CN(C(C2CN(C(N)=O)C2)=O)CCC1O)C C1(C(N2CC(c3c(CNC(CC(C)SC)=O)nco3)C2)=O)Cc2ccccc2N1 c1(C(=O)NC(CC)CNC(=O)CC2CC(CF)C2)cc2scc(C)c2[nH]1 N1(C(c2cc(C(=O)O)cc(Cl)c2)=O)CCC(CNC(=O)CC(F)(F)F)C(F)(F)C1 N1(Cc2c(OC)c(=O)cco2)CCC2OCCNC2C1 C1(NC(C=CCC)=O)CCN(C(=O)CC(c2ccc(CC)cc2)C)C(C)C1 c1(CC)nc2sc(C)cn2c1C(=O)NCC1C=CCN1C(=O)C#CC1CCCO1 c1(Cn2cc(CCC(CC)O)nn2)ccc(C(=O)N(C)CC2CCCOC2)nc1 C=CC(CCC)CC(=O)NCCC1(O)CCN(C(=O)Cn2cc(C)cn2)C1 C1(C(N2CC3C(CNC(c4n(C(C)C)ccn4)=O)C3C2)=O)CC(=O)C12CCCC2 N1(C(C2C(CC)C2)=O)CCC(O)C(N(C)C(c2ccc[n+]([O-])c2)=O)C1 N1(C(c2c(C)nc(CC)o2)=O)CC2CCC1CC2NC(=O)C(C(C)C)NC(N)=O C1(C(=O)NC(C)C(C)(C)CO)N(C(=O)CC2(O)CCOCC2)CCC1(C)C C(c1cncc(O)c1)=CC(=O)NCCN(C(CN1CCC(C)C1)=O)CC1CC1 CC(CC(N)=O)C(=O)NC1CC(C)CN(C(=O)Cc2csc(Cl)c2)C1 c1(C(=O)NC(CCN(C(CCc2ncc(C)[nH]2)=O)C)C(C)C)cn2ccnc2s1 N1(C(CCC(CCC)CC)=O)CC=C(C(C)(C)C(=O)NCc2cccc(O)c2)C1 c1(C(=O)NC2C3(CC(NC(=O)CCc4cccs4)C3)C2)ncn2c1CCC2 O(NC(=O)CC1CCC(NC(C2CCSCC2)=O)C1)CCCCC C(=O)(C1=C(C#N)CCC1)NCC1C(NC(c2c(C)n(C)nn2)=O)C1 CCCCCCC(C)CC(=O)NCC1(F)CCCN(c2nnnn2CC)C1 CC#CCCC(=O)NC1(CF)CCN(C(=O)C(C)OCCN(C)C)C1 CC1CC(=O)NCC1C(N1CCC(CO)(CNC(c2ccc(F)s2)=O)CC1)=O C(=O)(CCCCCC(C)(C)C)NCCC1CCCN(C(C(CC)OC)=O)C1 CC(C)C(C)(C)C(=O)N1CCC(CNC(=O)C(c2ccc(Cl)cc2)C)C1 C(=O)(CC(C)(C(F)F)N(C)C)NCC(C)CN(C(=O)CC(C)(C)C)C c1(C(=O)NC2CCOCC2NC(C2CSC2)=O)cc(F)c(Cl)cc1Cl C1(CNC(C2C(NC(CCSC)=O)CCO2)=O)CCC(=O)NC1 N1(C(C(c2ccc(C)s2)C)=O)CC(CNC(=O)C(C2CC2)C2CC2)CC12CCC2 N1(C(c2c(C(C)C)cco2)=O)CCC2(C1)CN(C(C1CC(F)(F)C1(C)C)=O)C2 Cc1nn(CCC(=O)NC2CN(C(=O)Cc3ccco3)CC2F)c(C)c1C N1(C(C(C)n2ccnn2)=O)CC(C2CC2)(C(=O)NCCCS(C)=O)C1 c1(C(=O)NC(C(=O)N(CCC#C)CCO)CCN(C)C)cccc2[nH]ncc12 c1(C(N(C(CC)CC(=O)NC(c2cccnc2)CC)C)=O)cc([N+](=O)[O-])c[nH]1 C(C)(C)(CCCC(=O)NC1CC(CF)C1)NC(C(N1CC(C)C1)C)=O C#CCCCCCC(=O)NCC(C1CCC1)NC(c1cccc(C(N)=O)c1F)=O c1(C(C)C)n[nH]c2ccc(NC(N3CCC(NC(=O)OC(C)(C)C)CC3)=O)cc12 C1(C(=O)NC(C(N2CCC(C)C2)=O)(C)C)CC2OC1C1CC21 C#CCCCCCCC(=O)N1CCC(C=C)(C(=O)NC(C)Cc2cnc[nH]2)CC1 C(c1cc(Br)cs1)=CC(=O)NC(C(C)NC(C1CC1(C)C)=O)CO CC1OC2(C(=O)NCC3CCN3C(=O)CSC3CCCCO3)CC1C2 C1(N(C(c2c(C)nsc2C)=O)C)CCCN(C(=O)Cc2cccnc2)CC1 C1(CNC(c2cn(C)nc2C(F)F)=O)CCN(C(=O)CCc2ncc[nH]2)C12CC2 c1(C(N2CC(O)CC(NC(=O)COC(F)(F)F)C2)=O)ccc2c(c1)CCOC2 N1(C(C2CCN(CCC#C)CC2)=O)CCCC(NC(=O)C=NOC)C(F)C1 N1(C(C=C(CC)C)=O)CCC(C)(NC(=O)Cn2cncn2)C1 N1(C(C2CC(C#N)C2)=O)CC2CCCN(C(c3ncc[nH]c3=O)=O)C2C1 C1(C)(C(=O)NC2CC(CCC(=O)C(C)=O)C2)CCCS1.CC(C)(O)CNC CCC(CC(=O)NCC(c1ccccc1)NC(c1nc(O)c(C)s1)=O)CC(C)C c1(OCC)cc(F)ccc1CNC(c1c[nH]nc1-c1cnccn1)=O N1(C(c2cnc(C)nc2)=O)C2CCC1CC(NC(C1CC3(CC3)C1)=O)C2 c1(-n2c(C(C(CC)C)OC)nc(-c3cncnc3)n2)ccc(Br)c(C)c1 c1(C(N(CC(C)CNC(=O)CN(C)C)CC2CC2)=O)cnc(OC(C)C)cn1 C1(C(C)=O)CC(C)CN(C(c2cn(C)c(-c3ccccn3)n2)=O)C1 CCN=c1[nH]cc(C(=O)NCCCCC(C)NC(=O)C(n2cc(C)cn2)C)s1 CCCCC(CNC(c1cnsn1)=O)NC(=O)CC1CCOC1 N1(C(CN(C(CCCCSC)=O)C2CCC2)=O)CCN(C)C(C(C)C)C1 N1(C(C2C(C)=C2)=O)CCC(C)C1CNC(=O)C(CN(C)C)c1ccccc1 C=CCC(C(=O)NC(c1cccc(Cl)c1)CNC(C1(CC)COC1)=O)NC(C)=O C(=O)(C1=CCCN(C(c2ccccc2Cl)=O)C1)N(CCCC(F)(F)F)C c1(CN(C(C2CCC(N)C2)C)Cc2ccccc2Cl)ccc(F)cc1 C1(NCc2ccc(C(=O)OC(C)C)[nH]2)CN(C)CC1C(F)(F)F N1(C(c2c(C)cccc2O)=O)CC2CN(C(=O)CC34CCCC3C4)CC2C1 N1(C(C)=O)CCN(OCC(C2CCCN(C(=O)CO)C2)C)CC1 c1(C(=O)NC2C3CCN(C(C(C)N(C(C)=O)C)=O)C3C2)cc(F)c(C)cc1Cl CC(CCCOCc1ccccc1)NC(CCCC1CC1)c1nnnn1CCF N1(C(C=C(C)Cl)=O)CCC(NC(c2ccnnc2S)=O)C1C(C)C N1(C(c2cc(CC(C)C)[nH]n2)=O)CCC(CNC(C2CN(C(C)C)C2)=O)C1(C)C N1(C(C2CC(SC)C2)=O)CC(C)CCC1CNC(c1cc(Br)c(C)o1)=O C#CCC(C(=O)N1CC(C(N2CC(OC(C)C)C2)=O)C(CCC)C1)C1CC1 CCCCCCCCC(C)CC(=O)NCC1CC(NC(=O)CCC(C)CC)CC1O C1(CC(N2CCC(CC(N)=O)C2)=O)CC(F)CN1C(C1CC1C(F)(F)F)=O C(C)(CO)(C(=O)NC(CNC(=O)CN1CCCNC1=O)C(C)C)OC C=CCC(C)(CC=C)NC(=O)CCC1CCCN(C(=O)CCC(C)OCC)C1 c12ccnc(c1)C(C)(C)CO2.c1(N(C2CCCO2)C(C)=O)cc(O)n(C)n1 c1(CN(CC(C)NC(=O)C(=O)NC2CCSC2C)C)cccnc1 c1(CNC(=O)Cc2ccsn2)nc(CNC(=O)CN2CCCCC2=O)cc(O)n1 N1(CC(=O)N(c2nnnn2CC(=O)OC)CC(C)NCC)C(=O)CCC1=O C1(C(N2CC(NC(C3C4(CC(C)(C)C4)C3)=O)C2)=O)CS(=O)(=O)CC12CC2 C(=O)(C#CC1CCCO1)N(C)CC1(O)CCN(C(c2ccc(COC)o2)=O)C1 C1(=O)CC(O)CN1.c1(CC(=O)OCC)occc1C(N1CCCCC1)=O CP(C)(=O)CC(=O)NC1COCCC1NC(c1ccnn1C1CC1)=O N1(C(C2C(C)C2)=O)CCC(NC(=O)CCCN(C)C)C12CCC2 C(=O)(CCC(F)F)NC(CC=C)CNC(=O)C(C)Sc1nncn1C Cc1ccc(F)c(C(=O)NCCCN(C(=O)C(C)(C)F)C)c1 N1(C(c2csc(Cl)c2)=O)CCC(NC(C23CC(CO2)C3)=O)C12CCC2 C1(NC(c2c(C)scn2)=O)CN(C(C2CCC2C)=O)CC12CCS(=O)(=O)CC2 C12(C(=O)NCc3cncc(F)c3)CCC(CC1)N(C(C1CC(O)CN1)=O)C2 n1(CC(=O)NC(C2CC(C(=O)N(C)CC3CCCO3)C2)C)cnc(C#N)n1 N1(C(c2cc(OC)nc(C)c2)=O)CCC(NC(c2cc(C)oc2C)=O)C(C)(C)C1 c1(-n2cc(CC(=O)N(C3CCSC3)C(C)C)nn2)cccc(C=O)c1.CO C1(N(C(c2cc(C3CC3)ccn2)=O)CC)CCCN(C(=O)CCC2OCCO2)C1 c1(OC)ccc(SCC(=O)NC2C3CCN(C(=O)C=CC(C)(C)C)C23)cc1 c1(C(=O)NC2C(C)CN(C(=O)Cc3cccnc3)CC2)ccc2c(c1)CCCS2 c1(C(=O)NCC2OCCN(C(C(C)=C(C)C)=O)C2)cc(C)cc(C)c1C Cc1cc(C(=O)NC(CNC(c2ccc(-c3ncc[nH]3)nc2)=O)CO)ncc1F O=C(C1=CCCCO1)NCC1CN(C(c2cn(CCC3CC3)nn2)=O)CCCO1 c1(C(=O)NCC(CC)NC(C2(C(C)C)CCC2)=O)cccc(-n2cc(C)cn2)c1 n1(CC(=O)NC(C2(O)COC2)C)cc(SCCCO)nn1 N12CC(C3CC3)(C1)OC1CCN(C1)C(=O)C(C)C2=O.C(C(N)=O)O.CCS c1(C(=O)NCc2nc(C)on2)ccc2[nH]nc(-c3cccc4cc[nH]c34)c2c1 C1(NC(C(C)n2cncn2)=O)CCN(C(=O)COCc2ccccc2)C1C Cc1[nH]nc(C(=O)NCC23CCCC2N(C(c2cn[nH]c2)=O)CC3)c1[N+](=O)[O-] c1(C(C(=O)NC2CCOC2)N(C)Cc2cn[nH]c2)cn(C)nn1 Cc1nc(=NC2CCC3CN(C(c4cc(CN(C)C)c[nH]4)=O)CC23)s[nH]1 C12(NC(c3cc4ccccc4o3)=O)CCCCC1CN(C(=O)CN1CCCC1)C2 c1(NCCN(C(=O)CC2CCOC(C(C)C)C2)CC)cc2oc(C)c(C)c2[nH]1 C(=O)(CCS(C)(=O)=O)N1CCC(C(=O)NC(CC=C)CC)(CC)C1 Cc1cc(-c2cnc(NCc3ccc(C#N)cn3)c(C)c2)c(C)cc1CO CCCN=C(NCC1(S(C)(=O)=O)CC1)N1CCC(CC2CCCC2)C1 C1(C(=O)NCc2cc(Br)ncc2F)C2CCC1CN(Cc1ccc(CO)o1)C2 N1(C(c2cc(CC)on2)=O)CCCC2CCN(C(C3(c4cccs4)CC3)=O)CC12 C1(CC(=O)NC(CC)CNC(=O)CCc2ccccc2C)CN2CCN1CC2 Cc1cccc(CC(=O)Cc2ccccc2CN2CC(O)CC2C)c1 C1(C(=O)NC2(CC)CCOCC2)C2CCN(C(=O)C=CC(C)C)CCC12 c1(C(N2C(C)(C(=O)Nc3cnc(Cl)cc3I)CCC2)=O)cc(Br)cc2cc[nH]c12 N1(C(C(C)C#N)=O)CCCCC1CNC(C1CC(OC(F)F)C1)=O N1(C(c2c(CC)noc2)=O)CCCCC1C(C)NC(c1nocc1C1CC1)=O N1(C(C(=O)N(C)C)C)CCC(C(O)C(=O)N(CC(c2ccccc2)O)C)CC1 c1(C(N(C(C)=O)C)C)c(C)nn(CCC(=O)OC)c1C.c1(C)nccs1 N1(C(N(CCCNC(C2CCN2Cc2ccccc2)=O)CC)=O)CCC(C)CC1 c1(SCC(=O)NCC2C(NC(C(C)OC)=O)CCC2)ccsc1[N+](=O)[O-] c1(C(N2CCC(CCNC(c3cc(C)nn3C)=O)CC2)=O)ccc2cnnn2c1 c1(OC)ccc(C)c(C(=O)N(CCNC(=O)CCc2cnccn2)CC2CC2)n1 c1(C(N2C3CC(CN(C(c4cscc4C(F)F)=O)C3)C2)=O)ccc2n[nH]cc2n1 N1(C(CC(CC)C(C)(C)C)=O)CC(N=c2[nH]c3ncc(Cl)cc3s2)CC1C C1(NC(=O)CC2C=CCC2)CN(C(=O)C2=NOCC2)CCC12CCOCC2 C(=O)(C(F)(F)C(O)C(C)C)NCCC(C(C)C)NC(c1cc(O)ccc1N)=O C1(NC(c2c(OC)scc2)=O)CCC2CCN(C(c3cccc(=S)n3O)=O)C1C2 C1(C)(CNC(C2(CC=C)CCCC2)=O)CCN(C(c2c[nH]nc2C)=O)C1 C(=O)(C(O)CCN(C)C)N(C(C)CNC(C1CCCC1C)=O)C c1(C(=O)NCC(CNC(c2cc(CCC)on2)=O)O)cccc2c1CCOC2 C(C1c2ccsc2CCN1C(=O)C=CCO)NC(C(CN(C)C)(C)C)=O c1(OC)ccc(C(=O)NC(C)CN(C(=O)CC(C)C2CC2)C)cc1O C1(C(=O)NCCC2(OCC)CCC2)C(C)CCN1C(c1ccc(O)nn1)=O c1(C(=O)NC2CN(C(c3cncc(N)n3)=O)CC2CO)cccc2c1CCCC2 c1(C(N(CCN(C(=O)C#CC2CCCC2)C)C)=O)n[nH]c2c1CCCC2 c1(C(=O)NC23CC(NC(c4ccc(SC)cc4)=O)(C2)C3)ccc(C(F)F)nc1O Cc1nc2cc(N(C3CC4CNC3C4)C(C3CCCN(C)C3)=O)ccc2o1 N1(C(CC(C)F)=O)CCCC(C2CN(C(c3conc3C(C)(C)C)=O)C2)C1 c1(C(C(=O)NCC2(OC)CN(C(C3(F)CC=CC3)=O)C2)C)ccccc1C CCCC(CNC(c1cnncc1OC)=O)C(=O)N1CC=C(CO)CC1 CC#CCCC(=O)N1CCC(N(C(=O)CCc2nc(-c3cccs3)no2)C)C1 CC(C)(C(=O)N1CCCCO1)C1CCN(C(c2cccc(=O)o2)=O)C1 n1(CC(=O)Nc2c(C)cc(I)cc2)ccc(=NC(=O)c2cncc(Cl)c2)nc1O n1(CC)nc(C)c(C(=O)NCC2(NC(=O)C(C)C#N)CC2)c1C N1(C(=O)Nc2cncc(C)c2)CCCS(=O)(=O)CC1c1cnn(C)c1 C12(CNC(C=CCOC)=O)CC(CN1c1cc(Cl)ncn1)C2 C=C(C)CC(C(=O)NCc1cccc(O)n1)NC(c1ccc(N)cn1)=O c1(C(=O)OC)sc(C(=O)NC2CC2)nc1C.C12(CC1(C)C)CCNC(=O)N2 c1(C(N2CCC(NC(Cc3scc(C)c3)=O)C(C)C2)=O)n[nH]c2ccc(Cl)cc12 CC(C)(C(=O)NC(CC(=O)NC1CNC(=O)C1)C(F)F)C(N)=O Cc1nc(CNC(=O)C(C)n2ccnn2)oc1C(=O)NOCC1CCCO1 c1(C(=O)NCCC(C)CCNC(C2CC3CCC3C2)=O)cc(F)c(N)cc1F c1(C(=O)NCCC(CNC(C(C(CC)O)C)=O)(C)C)c[nH]c2nccc-2c1 Cc1sc(O)nc1C(=O)N(C1CN(C(C2CCC(O)(c3ccccc3)C2)=O)C1)C c1(OC)ccc(CCCC(=O)NCc2ccccc2C2CCC2)c(Br)c1 N1(C(c2sc(C)c(O)n2)=O)CC2(C1)C(NC(=O)CSc1nncs1)CCS2(=O)=O c1(OCC)ccc(C)cc1C(=O)NCC(C)CNC(=O)Cc1ncccc1C N1(C(CCC#N)=O)C2CCC(C2)C1CNC(=O)CSC1CC1 CC(C)CC(C(=O)NC1C2CN(C(C3CCCN3C(C)C)=O)CC12)N(C)C c1(NC(=O)OC)cccc(C(=O)NC2(CO)CC(NC(=O)C=C(C)C(C)C)C2)c1 c1(NC(=O)NC2C(C(=O)Nc3ccc(C)cc3)CCC2)cccc(F)c1I N1(C(C(CC)(C)CNC(c2cn(C)c(=O)cn2)=O)=O)CCC(C)C(F)(F)C1 c1(NC(c2cc(-c3cccc(-c4ccc(F)cc4)c3)on2)=O)cc(Br)cnc1O N1(C(COCC=C)=O)CC(CO)(CNC(=O)COCc2cccnc2)C1 C1(C(N(C)CC2CCCN2C(=O)CCCC(C)(C)C)=O)CC2(CCOCC2)CO1 c1(C(N2CC(C)C(NC(c3cccc(CS(C)=O)c3)=O)C2)=O)cccc(O)c1F CCC(CC)C(C)N=c1cc(Cl)nc(-c2ccc(F)cc2)[nH]1 Cc1cc(S(=O)(=O)NC(C2CCOCC2)CCO)n(C(C)C)n1 c1(CC(=O)N(C)CCNC(C2(c3cccs3)CC2)=O)ccc([N+](=O)[O-])cc1F CC(C(=O)NCCCN(C(=O)CC1CCCN1C)Cc1ccccc1)C(F)(F)F N1(CC)N=C(C(=O)NCC2CC2NC(C2(C)CCC(C)(C)CC2)=O)CCC1=O C(=O)(CCCCCCNC(c1cn[nH]c1)=O)N1C(COCC#C)CCCC1 C1(C(=O)NCCOCCCO)CCN(C(C2CCCO2)=O)C12CCC2 c1(C(=O)NCCN(C(c2cc(CC)c(CC)o2)=O)C)cc(C)c(F)cc1Br C(=O)(CC(O)CC(C)(C)C)N1CCCC(C(N2C(C#C)CCC2)=O)C1CC Cc1cc(C(N2CCC(CNC(=O)C3=CCCC3)CC2)=O)c2n[nH]cc2c1 c1(C(=O)NCC2(C)N(C(CCCC#C)=O)CCC2)cc2c(s1)CCC2=O c1(CC(=O)NCC(CNC(c2c(CC)csc2)=O)(C)C)c[nH]c2cnc(Cl)cc12 Cc1nc2ccc(C(=O)NCC3CC(NC(=O)C(Cl)=CCl)C3(C)C)cc2nc1C CC(C)CC(O)C(=O)NC1C=CCC(C(=O)N(CC(c2nn[nH]n2)C)C)C1 N1(C(c2nc(C(C)C)oc2)=O)CCC2CN(C(c3cc(O)cc(Cl)c3)=O)CCC12 C1(NC(C2(CC)CCC2)=O)(CF)CCN(C(=O)C(C)COC(C)=O)C1 C1(C)(C(=O)NCC(C)CN(C(=O)CC2CC2C)C)CC1(Cl)Cl C1(C(=O)NC2(C(C)O)CC2)CC2C=CC1N(C(c1c[nH]c(C#N)c1)=O)C2 c1(NC(C(C)C)c2ncc[nH]2)ccc(N2CCCC2)cc1C(F)(F)F c1(NC(COC2CN(C(C(CSC)O)=O)C2)=O)ccc(CNC(N)=O)cc1 C1(N(C(c2c(C)nc(-c3ccccc3)s2)=O)C)CCN(C(=O)C(C)O)CC12CC2 O=C(C1=CCCSC1)NC1CC2CC(NC(C3CC=CC(O)C3)=O)C2C1 c1(C(N)=O)ccsc1NC(C1CCN(Cc2ccc[nH]2)C1)=O CCCC(C(=O)NC1CC(F)(CNC(=O)C(C)n2ccnc2)C1)OC Cc1cccnc1CCC(=O)NC(C)(CNC(=O)CC(=O)OC(C)(C)C)C1CC1 c1(OC)cc(C(N2CCC(NC(=O)CCc3nc[nH]n3)C2)=O)c(N)c(Br)c1 N1(C(CC(=C=C)C)=O)CCC2(CC1)CC(CNC(=O)C(C1CCOC1)OC)C2 N1(C(=O)CCC(F)F)CC23CCCCC2(C1)CN(C(=O)CCC1CCCO1)C3 O=NN1CCCCC1C(N1CC2CCC2(CNC(=O)CCC2CCC2)C1)=O CC(=O)CCCCC(=O)N1CCCC1CNC(=O)CCOC1CCCCC1 c1(C(=O)NC2CCN(C(c3c(C)cc[nH]3)=O)C2(C)C)ccc2c(n1)CCC2 C(=O)(C1=C(Cl)CCOC1)N1CC(C)C(C)(CNC(c2c(F)cccc2Cl)=O)C1 c1(NC(C2(C(C)NC(C(CC)OC)=O)CC2)=O)cccc(F)c1OC C(=O)(C(CC)CC(F)F)NC(CC)CN(C(=O)Cn1ncc(O)nc1=O)C c1(C(=O)NC2CC(C(=O)NC3CCOCC3)C2)cc(F)c(Cl)cc1Cl c1(C(=O)NC2CCN(C(C(C)(CO)OC)=O)C2)oc2c(C)ccc(C)c2c1C C#CC(CNC(=O)CC(CC)NC(C1(C(N)=O)CC1)=O)C(C)C N#Cc1ccccc1C1(CNC(C2C(C(=O)O)C2(F)F)=O)CCC1 CC(N=c1[nH]c(N2CCS(=O)(=O)CC2)nc2c1CCC2)C1CCCCC1 CC1(C)CCN(C(=O)Cc2ccsc2)CC1NC(=O)C1=CCS(=O)(=O)C1 N1(CCOCCOC)CC(n2cc(C)nn2)C(C)C1.c1(C(C)N)ccccc1.CCO O=c1c2cc(Br)sc2nc(Cl)n1C1CCN(CCc2ccncc2)CC1 C1(NC(C(C(C)NC(=O)CCN2CCCC2=O)C)=O)CCC(C#N)CC1 C1(CC)(C)CCCN(C(=O)CC2CC2C(F)(F)F)C1.C(C1CCCN1C)=CC(=O)N C(=O)(CC(C(F)F)NC(C1(C)CC2C=CC1C2)=O)NCc1cn(CC=C)nn1 c1(C(N(C)CC2C3CN(C(C(CC)(C)F)=O)CC32)=O)cnc2ccccc2n1 N1(C(c2nc(CC)sc2N)=O)CC(NC(C2C=CCC2)=O)CC2(CCOCC2)C1 N1(C(C(C)OCC)=O)CCN(CC2CN(C(=O)C(c3cccc(C)c3)C)C2)CC1 N1(C(CCC(=O)NC)=O)CC2CCC1CN2C(=O)Cc1cc(C)sc1C C=CC1(C(N(CCN(C)C)Cn2nc(C)cc2C)=O)CCN(C(C)=O)C1 C1(NC(c2ccoc2)=O)CC2CCC1CC2NC(C1Cc2nnsc2S1)=O N1(C(CC(=O)N(C)C)=O)CC2COCCC2(NC(c2cccc3scnc23)=O)C1 Cc1c(F)ccc(C(N2CC3(CC3)CC2CNC(=O)C(O)CC(C)(C)C)=O)c1C c1(CC(=O)NC(CNC(c2nncc(OC)c2)=O)C2CCC2)ccc(C)c(F)c1 c1(CC(N2CC3(C(NC(CCC=C)=O)CC3)C2)=O)c[nH]c2cccc(C)c12 S(=O)(=O)(c1cc(Br)ccc1Br)N1CC(CC)N(c2ncnc3c(Br)csc23)CC1 C12(NC(CN(CCOC)C)=O)CCCC1N(C(c1cc(C)c(Cl)cc1F)=O)CC2 C1(N(C)C(c2csc(Br)c2)=O)CCCN(C(C23CC(O)C2C3)=O)C1 c1(NC(C2N(Cc3ccnc(OC)c3F)CC(F)(F)C2)=O)c(Cl)cc(Br)cc1Br C1(C(=O)NCCc2n(C)nnc2)CN(C(=O)COc2ccccc2)CC(C)(C)C1 N1(c2ncc(SC)cn2)CC(NC(C2CC3(CCC3)C2)=O)CC(F)(F)C1 c1(OC(N(C2CCCC2C)C)=O)cnn(C(C)(C)C(=O)OC(C)(C)C)c1 CCC(C(=O)NNC(=O)NCCC(C)SC)c1ccc(C)cc1 C=CCC(C(=O)NCC(C)(C)NC(=O)CC1CC(C(F)F)C1)C(C)C C1(C(C)C(=O)NC2(CN(C3CCCC3)C(=O)COc3ccsn3)CC2)CCC(=O)N1 c1(-c2cc(CC)c(O)cc2)cc(S(=O)(=O)NCCN2CCOCC2C)ccc1OC C1(C(=O)NCC(CC)NC(c2cnc(=N)[nH]c2)=O)CC2CCC1C2 C1(CNC(c2c(C#N)ccnc2)=O)CC12CCN(C(=O)NCCCCl)CC2 C1(NC(c2c(C)cc[nH]2)=O)C2CC1CN(C(c1cc(-c3ccncc3)on1)=O)C2 CC1(C)COCC(C(=O)NCCN(c2ccccc2)C(c2c[nH]ccc2=O)=O)O1 c1(CC)nc(C)c(CC(=O)NCC(CNC(=O)C(C)=C(C)C)CO)c(C)n1 O=C(C1CCCc2nn[nH]c21)NC1CCN(C(c2ccoc2Cl)=O)CC(O)C1 O=C1NCC(C(=O)NC2(CC(=O)NCC3CCC4CC34)CCC2)O1 C1(CSC)CCN(C(c2ccnn2C)=O)CC1.c12cn(nn1)CCN1CCSC21 CC1CCN(C(C23CCCN(CCC2)C3)=O)CCN1C(=O)CCC(C)N(C)C C(=O)(C(C(C)C)Sc1ccccc1)NC(C(CO)NC(c1cc(C)ns1)=O)C c1(-c2c(OC)ccnc2)nc2c(s1)CC(C(=O)Nc1ncc(Cl)cc1I)CC2 CCC(CC(=O)NC(C)CC1CN(C(=O)C(c2ccccc2)N(C)C)C1)C(C)C c1(C(=O)NC(C2CCCC2)CNC(c2nc(OCC)sn2)=O)cc(=O)c(C)c[nH]1 N1(CC2CC(C(C)C)OCC2)CC2CN(C(=O)CCCC3CC3)CC2C1 C(=O)(C1=CC2CCCCC12)NCC(N(C(CCC=C(C)C)=O)C)C1CC1 CC1CC(CNC(c2ccns2)=O)CN1C(=O)OC(C)(C)C c1(C(N2CCCC(CO)C2)=O)cc2c(-c3ccoc3)cncc2s1 C(=O)(CN=S(C)(C)=O)NCC1(NC(CCC(C)N(C)C)=O)CCCC1 N1(C(C(N)=O)=O)CCCC(c2cn(CC(=O)O)nn2)(CO)C1.C12CCCC1C2 C(=O)(C(F)(F)CC(C)C)N1CC(N(C(CCC(=O)NCCC)=O)C)C(O)C1 C1(NC2CC(NC(CSCC)=O)C2)CCCCC1N=c1ncnc2[nH][nH]c(C)c1-2 C(C)(C)(CCCCC(=O)N1CCCC(NC(=O)CN2CCNC(=O)C2)CC1)OC C1(C(N)=O)CN(C(C2C3CC4C(C3)C24)=O)CCC1NC(C1SCCCS1)=O c1(SC)ccnc(N2CCC(C(C)(C)CNC(c3ccc(F)s3)=O)CC2)n1 CC(C)C(F)(CNC(=O)C=CCF)C(=O)NCC1(CO)CCN(C)C1 c1(NC(c2c(C)cnn2C)c2n(CCOC)nnn2)cc(C)cc(O)c1 C12(NC(CC=C)=O)CCCCC1CN(C(c1cccc(NC(C)=O)n1)=O)C2 CCC(C)(COC)C(=O)NC1CC2(C1)CC(CNC(C1CC(OC)C1)=O)C2 N1(C(=O)NCCn2cnc(C#N)n2)CCc2nocc2C1 C(=O)(C(C)CC(C)(C)C)NCC1(C)CCCN(Cc2cc(C)sc2)C1 C1(n2c(-c3ccc(CCC)s3)nc(C(C)O)n2)CCCS(=O)(=O)C1 C1(C(=O)NC(CNC(c2ccc(C(F)F)o2)=O)CO)CC(F)(F)CS1 C(=O)(C1CCN(C)c2ccccc21)c1nnc(C2C(C)CN(C)C2)o1 C(=O)(CC(C(F)(F)F)n1cccn1)N(CCC(C)NC(=O)C1=C(C)CCC1)C CC(C)(C)C(CNC(C1CCC(C(N)=O)C1)=O)C(=O)NCC1(CO)CC1 c1(-c2nc(CCC(C)C)nn2Cc2ccccc2)ccc(S(=O)(=O)C(C)C)cc1 Cn1nc(C(=O)NC2(CO)CCN(C(C3CCCS(=O)(=O)C3)=O)C2)ccc1=O C(=O)(C(C)C1=CCCC1)NCCN1CCN(C(c2ccc(C)nc2)=O)CC1 n1(C2CN(C(C3(CC)CC3)=O)C2)cc(CNC(c2ccnn2C)=O)nn1 Clc1ccccc1C(c1nnnn1Cc1ccccc1)NCC1CC2CCC1C2 C(=O)(C(F)C(C)C)NCCC1(C(N2C(C#C)CC2)=O)CCCC1 c1(C(=O)NC2CC(C)(NC(C3CCS(=O)(=O)N3)=O)C2)c(C(F)(F)F)cccc1O Cc1nsc(CNC(c2nnnn2C)(C)Cn2ccnc2C)n1 N1(C(c2cc(CNC(C3(O)CC3)=O)ccn2)=O)CCC2CCC(O)C1C2 CCCC(O)(CCC)CC(=O)N1CCN(C(=O)CC(O)C2CCCC2)CC1CO Cc1ccc(C)c(CC(=O)NC2C=CCN(C(c3nc(C)n(C)c3C)=O)C2)c1 Cc1c(Cl)cnn1CC(=O)NCC(CNC(=O)CC1CCCOC1)CO N1(C(c2cc(C(C)(C)C)no2)=O)CCN(C(C2CC2c2cn[nH]c2)=O)CC1CO C1(C(=O)OCCC(C)(C)C)(COC)C=CCC1 c1(CC)nc(N(C)CC2CCCN2C(c2nc(C)oc2C)=O)cc(C)n1 c1(C(N(C2CCCN(C(C(CN(C)C)(C)C)=O)C2)C)=O)nc[nH]c2ncnc1-2 O(NC(=O)CC(C)C(C)(C)NC(N)=O)CC(=O)NC1C(C)C1C c1(C(=O)NCC(CN(C(c2c(COC)cc[nH]2)=O)C)O)ccc(CO)cn1 C1(C(=O)NCC(C2CCOC2)NC(C(C)c2ccsc2)=O)CC(=O)NC1(C)C C1(C(=O)NC(CCOC)CNC(C2CC2C)=O)C(C)(C)C1(C)C N1(C(CC=CCC)=O)CC(NC(c2oc(C3CC3)nc2C)=O)CC1(C)C C1(CNC(c2cc(C)c(O)nc2)=O)CN(C(=O)Cc2ccon2)C2(CCC2)C1 N1(C(C(C)C2CCCC2)C(=O)NCSC)CCCN(c2cccc(CO)c2)CC1 c1(C(N2CC(NC(C3C(C)(C)CC3)=O)C2)=O)cc(C(F)F)ccc1F CC(O)C(F)(F)C(=O)NCC12CC(NC(c3cccc(N)c3F)=O)(C1)C2 c1(C(N2C3CCC2CN(C(C2(N(C)C)CCCC2)=O)C3)=O)cccc2c1CCO2 C1(NC(=O)Nc2c(NC(=O)NCC)ccs2)CCCC1(C)CSC C1(NC(C(C(CC)O)C)=O)CC2(CCCCN2C(=O)CN(CC(C)(C)C)C)C1 C1(CN(C)C(C2(NC(=O)C(F)F)CC(CO)C2)=O)CCCC2CC12 C1(CC(=O)NCC2(F)CN(C(=O)COC3CC3)C2)CC=CCC1 C1(C(=O)NCC(C)CC2CC2)(NC(=O)CCc2nccn2C)CCC(C)(C)C1 C=CCC(C)C(=O)NCCCCCN1CCN(C(=O)C(=O)C=CCCC)CC1 Cc1c(SC2(C(N3CC(NC(=O)CN(C)C)C(C)C3)=O)CC2)oc2ccccc12 c1(N(C)C)ccc(C(=O)NCC2(C)CCN(C(C3CCOCC3)=O)C2)nn1 C1(CNC(CC(C)c2ccco2)=O)CC(NC(=O)C=CC(C)(C)C)CCO1 c1(OC)cncnc1NC(=O)C(O)CCCl c1(NC(=O)OC)cccc(C(=O)NC2CN(C(C3CCCC3O)=O)C2)c1 C1(NC(C2CCN(C(=O)NC)CC2)=O)CCSC12CN(C(=O)C(C)C#N)C2 C12(CNC(c3cc(CF)on3)=O)CC1CN(C(=O)COc1ccccc1F)C2 C1(C)(C(=O)NCC2N(C)CCN(C(=O)Cc3ccsn3)C2)CCC(F)(F)CC1 C1(CC(=O)NCC(=O)NCC(=O)NCCC2CC(C)C2)C=CCCC1 C1(C(N(C(CC)C2CC2)C)=O)CCC(O)CN1C(C1CC=CC(O)C1)=O c1(C(N(CCN(C(=O)CN2CC3C=CC2C3)C)C)=O)noc2c1CC(C)(C)CC2 N1(C(C2(F)CCN(C(C(C(CC)O)(C)C)=O)C2)=O)CCc2nc(O)[nH]c2C1 c1(C(C(=O)NC(CNC(c2nccc(C)c2)=O)CC(C)C)C)ccc(F)cc1F N1(C(c2n(CCN(C)C)ncc2)=O)CCOC(CNC(C23CC(C2)C3)=O)C1 CC1=C(C(=O)N2CC3CC(NC(c4c(Cl)ccc(F)c4F)=O)CC3C2)CCCC1 C1(F)(C(=O)OC)COCCN(C(=O)NCc2cc(CSN)cn2C)C1.C(C)(C)C C1(CNC(C(CC)=CC)=O)CCN(C(=O)CC2CC2C(F)(F)F)CC1O C1(C(=O)NCc2cc(C(=O)NCC(C)(CO)OC)on2)CCCC(=O)CC1 C#Cc1cnc(C(=O)NCC(C)CN(C)C(c2c(OC)cccc2F)=O)c(C)c1 C#Cc1cn(C)nc1C(=O)N(C(C)CN(C)C(c1scnc1COC)=O)C C(=O)(C1CCCc2c[nH]nc21)NC1(CNC(CSSC)=O)CCOCC1 Cc1c(C(N2CCCC2C(C)(C)C(=O)N(C)Cc2ccncn2)=O)cccc1O CC1OC2(C)CC1(C(=O)NCC1CC(CNC(=O)CS(N)(=O)=O)CO1)C2 c1(C(N2C(C(=O)NCc3n(CC)ncn3)(C(C)C)CCC2)=O)ccc([N+](=O)[O-])[nH]1 CC1(C(=O)NCCN(C2CCCCC2)C(C2CC(C(F)F)C2)=O)CCC2CC2C1 C1(NC(C2CC=CCC2)=O)CC2CCC1N(C(C1CC1c1ccncc1F)=O)C2 c1(C(=O)NC2C3CN(Cc4c(C)nc(C)o4)CC32)c(F)ccc(F)c1Cl C1(NC(CCC(=O)NC)=O)CC2CC1N(C(c1cccc(Br)c1Cl)=O)C2 Cc1cc(C)c(CNC(=O)C(C)(C)C2CCCN2C(=O)C(=O)C2CCCC2)cn1 c1(CC(C(=O)NC(c2ccsc2Br)C(=O)OC)OC)ccc(F)cc1 N1(CC2ON=C(C(C)C)C2)CCN(S(C)(=O)=O)CCC1C C(C(C)(C)C#CC(=O)NC1C(=O)OCC1(C)C)NC(CCCCC#C)=O N1(C(c2c(C)noc2C)=O)CC2CCCCC2(NC(=O)CCCCN(C)C)C1 C1(NC(c2c(CC)cncc2)=O)COC2(CCN(C(=O)C(C)(C)CF)CC2)C1 C1(CCOC)CN(C(c2scc(C)c2C(F)(F)F)=O)CCCO1 C1(NC(=O)CCC2CCC2)CCN(C(C2CC2F)=O)C12CCC2 C1(C(N2CC(C)C(NC(C3(S(C)(=O)=O)CCCC3)=O)C2)=O)CCCC2CCCN12 Cc1ncc(C(=O)NCC2(C(C)(C)C)CCN(C(=O)CCF)C2)c(C)n1 N1(C(c2cc(CC)[nH]n2)=O)CC2CN(C(=O)CC3C=NN(C)C3=O)CC2C1 C1(n2cnnn2)(CC(=O)NC2C(CNC(=O)CC3CCC3)COC2)CCOCC1 c1(OC)ccc(Cl)c(C(=O)NCCN(C(=O)Cc2cncn2C2CC2)C)c1 C1(NC(CCC(=O)NC)=O)CCN(C(c2ocnc2C(C)C)=O)CC1C S(=O)(=O)(c1csc(C(=O)NC(C2CCCN2C(=O)C(C)=C2CC2)C)c1)NC CC(C)C(O)CC(=O)N(C1CCCN(C(=O)C(C)CN2CCOCC2)C1)CCF N1(C(CN(CC)CC)=O)CCCN(C(=O)COC2CCOCC2)CC1CO N1(C(CSCCC)=O)CCC(NC(=O)C=Cc2cnc[nH]2)CC1c1ccccc1 c1(C(N2CCC(CC=C)(NC(=O)C(F)OC(F)(F)F)C2)=O)c(N)ccc(C)c1F c1(OC)c(C(=O)NCC(C)(C(C)C)NC(c2cn(C)cn2)=O)oc2ccccc12 Cc1ncc(C#N)cc1NC(=O)CC(C)N(C)C(c1ncc2ccccn12)=O N1(C(C(c2n(C)cnc2)O)=O)CC2CCOC2(CNC(c2ccco2)=O)C1 CCCC(CNC(c1coc(COC)n1)=O)NC(=O)C(C)(O)C1CCC1 C#CCC(C(=O)NCCCCC1CCCN(C(C2C3CCC2CC3)=O)C1)C1CC1 C1(C)CCN(C(C2CCCN2N(C)NC(C2(c3cccs3)CC2)=O)=O)C1.C1CC1 Cc1cnc(NCC2CCCC(CNC(c3cnn(C(C)C)c3C)=O)C2)nc1 C(=O)(C(F)(F)CO)NC(c1cccc(NS(C)(=O)=O)c1)C.C12CN(C1)C2=O CC(C)S(=O)(=O)C(C)C(=O)NCCC1CN(C(c2ccn(C)c2)=O)CCCO1 CC1OCC2(CCN(C(=O)C3=CCNCC3)CC2)O1 c12c(cccc1C)C(=O)N1CCCCC1CCNC2=O.C1(NC(C)=O)CC1(F)F N1(C(C(F)OC)=O)CC(CNC(=O)Cn2nccn2)C(O)C1 C(=O)(CC(CNC=O)CC(C)C)N(C1CCN(C(c2ccc(N)cn2)=O)C1)CC CCCC(C)(O)CC(=O)N1CCN(C(C2(S(C)(=O)=O)CC(O)C2)=O)CC12CC2 CCCC(CCCNC(=O)Cc1ccon1)NC(=O)C(C)(C)c1ccns1 c1(OC)ccc(Cl)c(C(=O)NC(CCNC(c2ccnc(S)c2)=O)C(C)C)c1N FC1(F)CC12CCCN(Cc1cnc(C3CCC3)o1)C2 C1(CC(=O)NCc2cn(CC)nc2)CC2(CC2)CN1C(C1CC2(CCC2O)C1)=O c1(C(=O)NCCOCCN(C)C(C2CC2(C)C)=O)cccc(-n2cnnn2)c1 Cc1ccc(C(=O)NCCCc2ncco2)c(-n2cc(C(C)O)nn2)c1 C#CCC(C(=O)NCC(C)(C)C(N)=O)NC(C1CN(CC)CCO1)=O CC1(C)CN(C(C2(O)CCCCC2)=O)CC(CNC(=O)Cc2cccs2)O1 c1(N2CC(=C(CNC(CC)=O)F)C2)nc(Cl)nc(C2CC2)c1C#N C12(C(=O)NCC(CC)(CC)NC(=O)C#CC3CCC3)CCC(CC1)CO2 c1(C(N2CCN(C(C(=O)OCC)C)CC2)C(=O)NC(C)C)cc(F)c(Cl)cc1Cl C1(C(=O)NCC2(NC(c3c(Cl)cc(C#N)s3)=O)CCC2)CCOC2(CCC2)C1 c1(C(=O)NCCN(C(C(CC)C2CCOCC2)=O)C)nn(C)cc1Cl N1(C(N2CCCC2=O)=O)CCOCC(C(=O)NCCC(=O)NC2CCCCC2)C1 c1(N2CCC(CN(C)C)C2)nnc(-c2ccco2)n1CCc1cncc(F)c1 c1(C(N2C(CCNC(C(C(C)(C)O)F)=O)CCC2)=O)nnc2ccccn12 c1(C(C(=O)NC2(CO)CN(C(C(C)OCC#C)=O)C2)O)ccccc1Cl CN1CC(C)(C)CC1C(=O)N(C1CCCN(C(=O)CCCN2CCCCC2)C1)C Cc1c(C(=O)O)c[nH]c1CSc1ccnc(NC2CC2)c1 c1(CC(=O)NCC(C)CN(C)C(c2cnc(C(C)O)s2)=O)cnn2ccccc12 C1(C)(NC(C2N(C(CCCOCC)=O)CC2)=O)CCC(C)(C)C1 c1(NC(CCC)CCC)nc(C)cc(=NC2CC3C(C2)C3(F)F)[nH]1 c1(C(=O)NC2(C)CCN(C(CN(C)C3CC3)=O)C2)cc2c(Cl)cncc2s1 Cc1cc(C(F)(F)F)nc(NCC2COCCN2C(=O)Cn2ccnc2C)n1 c1(C(C)NC(N2CCN(C(=O)Cc3ccn(C)c3)CC2)=O)cccc(C#N)c1 C1(C(=O)NC(C#C)CC)(CC)CN(C(c2nccn2C)=O)C1 C=CCC(C)(C)CNC(C12CCC1C2)=O C(=O)(C1CCCn2cnnc21)NC1C(C)CN(C(=O)C(F)=CC2CC2)CC1 Cc1cccc2c(CC(=O)NCCCN(C)C(C3C4CNC(=O)C34)=O)c[nH]c12 C(=O)(C(O)CCN(C)C)NC1CC(C(=O)NC(C)Cc2nncn2C)C1 Cc1ccc(-c2noc(C(N3CCC(CNC(=O)CNC4CCC4)C3)C)n2)cc1 Cc1cc(C2CC2)ccc1C(=O)N(C)CCOCCN(c1ccccc1)C c1(-c2ccc(CCOC)cc2)n[nH]c2c1CN(C(=O)C1=CCCC1)C2 n1(CCNC(N2CCC(CCCF)CC2)=O)cnc2c1CCCC2 N1(C(C2(C3CCN3C(=O)OC(C)(C)C)CCC2)=O)CCCCC1CNC(C)=O n1(CCOC(C)C)cc(C2(OCCO)CC2)nn1 C1(CNC(c2n[nH]cc2Cl)=O)(CO)CCCN(C(=O)C(=CC2CCCCC2)F)C1 C1(NC(CC(CC)SC)=O)CN(C(=O)COC2CC2)CC12CCOCC2 C12(C(N3CCCC(C)C3)=O)COCC1CN(C(c1ccc(Cl)cc1F)=O)C2 c1(C(N2CC(CNC(=O)CC3CCOC3)C(O)C2)=O)ncc(Br)cc1F N1(C(c2n[nH]c(CC)c2Cl)=O)CCC2CCN(C(=O)C(O)CC(C)(C)C)CC2C1 Cc1nc2c([nH]1)C(C(=O)NCCCCN(C(=O)CCc1ccc(C)o1)C)CCC2 N1(C(C2C3C=CC(CC3)C2C(F)F)=O)Cc2cc(Br)ccc2CC1C(=O)O C(=O)(C1=C(Cl)CCC1)NCC1C(NC(CC=C=C)=O)CC1 C1(CC(N2CCCC(CCNC(=O)COC3CCOC3)C2)=O)CCCOCC1 C(CCCCC(=O)NOCC(N1CCN(C(C)(C)C)CC1)=O)OC C(CCC(O)C(=O)NCC1CNC(=O)C1)NC(CC=CC=C)=O N1(C(c2occ(C)c2)=O)CC(CNC(=O)CC2OCCCO2)CC(C)C1 c1(C(=O)OC)ccc2c(c1)CN(C(c1sc(C)cc1Br)=O)CCO2 c1(CC(=O)NCC(CO)NC(CS(CC)(=O)=O)=O)cn2cccc(C)c2n1 C1(C(=O)NCCCCC2CN(C(c3nn[nH]c3Cl)=O)C2)(OCC)CCCC1 CC1(C)CCC(CC(N2CC(O)(CNC(C3CCCC(F)C3)=O)C2)=O)C1 C1(F)(CNC(=O)Cc2cc(Cl)ccc2Cl)COCCN(C(C2CNC(=O)C2)=O)C1 C1(C(=O)OC)CCN(C(C2CC3CC3C2)C(=O)NCCCCCNC(C)=O)C1C N1(C(CS(N)(=O)=O)=O)CC2CS(=O)(=O)CC2(NC(=O)CCN2CCCC2=O)C1 C1(C(C)C(c2ccccc2)=O)CCCCN1C(C1CCCN1C(N)=O)=O n1(CC)nc(C(=O)N(CC(C)N(C(=O)CC(C)=C(C)C)C)C)c(Br)n1 c1(C(=O)NC23C(CN(C(c4c(C)occ4)=O)C2)CCC3)cc2ccsc2c(O)n1 c1(C(=O)NC(C2CCN(C(CS(=O)(=O)NC)=O)C2)C)csc(S(C)(=O)=O)c1 c1(NC(CN(C(=O)COCC2CC2)CC)=O)cnccc1CN(C)C C(=O)(CCC(F)(F)CN=[N+]=[N-])N1CCC(O)(C(C)NC(CC(C)C2CC2)=O)CC1 CCCC(C(=O)NCCCCF)NC(=O)CN(C)C C(CC(=O)NCc1cccnc1C)(CC(C)C)NC(C(CC=CC)CC)=O c1(CNC(C2C(S(C)(=O)=O)(Cc3ccccc3)C2)=O)cc2cn[nH]c2cn1 n1(C(C)CC(=O)N2CCC(N(C)C(c3cnn(C)c3)=O)C2)cnc2ccccc12 CCC(C)C(O)C(=O)NC(C1CCN(C(=O)C(O)Cc2cnc[nH]2)CC1)C N1(C(C=CCC)=O)CCCC(C(=O)N(C)Cc2ncn(C)n2)C1C C(=O)(C(F)(F)C(F)F)NC1CCCC(NC(C(C)OCCC=C)=O)C1 c1(C(N2C(C)CC(NC(=O)CC(F)(F)F)C2)=O)ccc2c(O)nccc2n1 C1(NC(CN(C(C2(CCCC)CCC2)=O)C2CC2)=O)CSCC1C N1(C(C=CC=CC)=O)CCC(CO)CC1.C1(=O)CC(C)CN1C c1(C(N2C(C(=O)Nc3cnc(Cl)nc3)CC3CC32)=O)noc2c1CCCC2 C1(C)(C(=O)NC2C(CNC(CCCNC(C)=O)=O)CC2)CC(C2CC2)=NO1 CC1C(NC(C2CC3CCC2C3)=O)CCN1C(=O)C1CC1 c1(C(N(C(C)C)CCNC(=O)C(O)C2CC2)=O)cc2sc(Cl)cc2[nH]1 C1(NC(C(CC)NC(N)=O)=O)CCC2CCN(C(c3ncccn3)=O)C1C2 c1(C(N2C(C)(C)C(NC(=O)COCCO)CC2)=O)cc(F)cc2ccncc12 c1(C(=O)NC(C)(C)CCNC(C2CCCCN2S(C)(=O)=O)=O)ccc(C#N)cc1 C1(CNC(CC2CC(=C)C2)=O)(CO)CCN(C(=O)C(C)(Cl)Cl)C1 C(CCCCNC(=O)CCC1CCOCC1)N(C(C)C)C(C1CCC(C)O1)=O C12(NC(COCC)=O)CCCC1CN(C(c1cc(-n3cccn3)ccn1)=O)C2 N1(C(C2CC23CC3)=O)CCCC(CC(=O)NCc2ccncc2Cl)C1 c1(C(=O)NCC(CN(C(=O)C2=CCCOCC2)C)O)nc2cc(O)ccc2[nH]1 Cc1ncc(C(=O)N(CCC(=O)NCC23CCCC2C3)CC2CC2)c(=N)[nH]1 C1(NC(=O)C(C2CCOCC2)=O)CCCCCN(C(C2CC(C3CC3)=NO2)=O)C1 C=CCCCCCCCC(=O)NC1CN(C(C23CCCCN2CCC3)=O)CC1C C1(O)(C(C)NC(C=CC=CC)=O)CN(C(C2CC2C(F)(F)F)=O)C1 C(=O)(CCCC(=O)NC(C1CCN(C(c2ccncc2F)=O)C1)(C)C)OCC C1(CC(=O)N(CC(=O)NC2CC2OC(C)(C)C)CC#C)CCOC1C C12(NC(CC(CCCC)O)=O)CC3CCC(C1C2)N3C(c1ccc(=N)[nH]c1)=O c1(C(C)(C)C(=O)N2CCC(CNC(C3(CO)CCCO3)=O)C2)ccc(Cl)cc1F C1(CCOc2cccnc2)CCCC1(C)C.C12CC(C1)NC(=O)N2CC c1(CC(COC)C(=O)NC2CSCCN2CCOC)ccc(F)cc1F CC1(C(N2CCCC(CNC(c3ccc[nH]3)=O)C2)=O)CC2CCC(C1)S2 CC1Oc2ccccc2OC1C(=O)NCC1(CNC(c2cnc(O)s2)=O)CCC1 CCCCC(C)(CO)NC(C1(N(C)C(c2ccc(O)c(F)c2)=O)CC1)=O c1(C(N2CCCC(C)(CNC(CC)=O)C2)=O)cc(F)c2nc(C)cn2c1 c1(C(N2C(CC(=O)NC(c3ccc(F)cc3)C)CCC2)=O)ccc(O)c(F)c1F c1(NC(c2ccc(-c3c(O)ccc(C)c3)cc2)C)ncnc2n[nH]cc12 c1(NCC(CNC(CCC(C)SC)=O)C)ncnc(O)c1Br CC(C)CCC(O)C(=O)N1CCC(C(C)NC(=O)C(F)C2CCC2)CC1 C(=O)(CS(=O)CCC(F)(F)F)NCCCN(CCCNC(C1(SC)CCC1)=O)C N1(C(c2scc(COC)c2)=O)CC(NC(C2(c3cccs3)CC2)=O)CCC1C C(=O)(CCCC(F)(F)F)NC(C)CCCCNC(=O)CN(C1CCSC1)C N1(C(CCC2N(C(CN=[N+]=[N-])=O)CCCC2)=O)CCOC2(CC2)C1 C(=O)(CCC(C)(C)C#N)NC(CC(=C)C)C(=O)NCCC1(C)CC1 O=C1CC2C(NC(C3(NC(=O)COCCN(C)C)CC(O)C3)=O)CC2O1 C(=O)(C1=NNC(=O)C1)NC1C(CC)N(C(c2cc(Cl)cc(Br)c2)=O)CC1 C(=O)(CCCC(=O)NC1CCC1NC(c1scc(C)c1C)=O)N(CC)CC C1(C(N(CCN(C(=O)CN(C)C)C(C)C)C)=O)CC12CCC(C)(C)CC2 C=C1CCN(C(C2C3CCC(C3)C2C)=O)C(C(N2CC(F)(C(=O)OC)C2)=O)C1 N1(C(c2n(C)cnc2)=O)CCN(C(C2(CF)COC2)=O)CC1c1cccc(F)c1 c1(C(=O)NCCN(C(=O)CCCOC(C)(C)C)CC)cnn(C(C)C)c1C c1(C(N2CCC(NC(c3c(C)onc3O)=O)CC2C)=O)ccc2c(c1)CCN2C N1(C(C(C2(C)CC2)NC(CCn2ccc(C)n2)=O)=O)CCC2CN(C)CC12 C1(OC)CC2(C1)CC(C(=O)NC1CN(C(=O)C(C)SC)CC1c1cnn(C)c1)C2 c1(CCC(=O)N(CC(CC)NC(c2cc(C)c[nH]2)=O)C)ccc(Cl)cc1 C1(Cl)(C(=O)NC2CC(OC)CN(C(C)=O)C2)CC12CCOCC2 c1(C(C)C)cccc(NC(c2cncnc2)c2nnnn2CC2CCCO2)c1 N1(C(c2occ(C)c2)=O)C2CCC1C(CO)N(C(c1cccc(N)c1)=O)C2 c1(CNC(C2CCN(C(c3cccs3)=O)CC2O)=O)cc(F)cc(Br)c1 CCCC(CCCNC(C1CCOC1)=O)NC(c1cncs1)=O C(=O)(C1=C(CC)OCCS1)NC12C(CN(C(C3(CC#C)CCCO3)=O)C1)CC2 c1(C(C)C)nnc(C=CC(N2CC3CC3(NC(=O)CC3CCC(O)C3)C2)=O)o1 C12(NC(=O)CCCC3CC3)CCCCCC1N(C(=O)Cc1sccc1Cl)CC2 CN1CC=C(CC(=O)N2CCC(NC(=O)CN(C)S(N)(=O)=O)C(C)(C)C2)CC1 c1(C(=O)NCC(C)CNC(c2cnc(C3CC3)s2)=O)ccc(Br)c(F)c1 N1(C(C(C=C)OC)=O)C2CCC(C2)C1C(N1CC=CC1COC)=O c1(C(=O)NC(C)C=CC(=O)NCCC(C)(C)F)ccc(Cl)cn1 Cc1cc2cc(C(N3CC(C)CCC3NC(=O)OC(C)(C)C)=O)[nH]c2cc1Cl c1(C(N(C(CN(C(C(C)NC(CC)=O)=O)C)C)C)=O)c[nH]cc(F)c1=O c1(C(=O)NCCCC(=O)NC2CN(C(CC)=O)CC2C)ccc2c(c1)CCC2 CS(=O)(=O)C1CN(C(=O)Cn2nccn2)CC1NC(C1CCc2nncn2C1)=O C1(C2(O)CN(C(=O)CCC3CCCC3)C2)(CNC(=O)CN2CCCS2(=O)=O)CC1 C1(CNC(C(=O)N(CCCCO)CC)=O)CCN(C)C1 c1(CC)ncc(C(N2CCC(N3CCCC3)C2)C(=O)NCCOC)cn1 c1(NC(C2C(NC(C(C)O)=O)CC2)=O)ccc2c(c1)CCC2 C(CC(=O)N=S(C)(=O)C1CCCCC1)C1CCCC(C)C1 c1(N2CC(NC(CCN(CC)CC)=O)CC(C)(C)C2)c(C#N)cccc1[N+](=O)[O-] N1(C(C(CC#C)C2CC2)=O)CCN(C(=O)Cn2ncnn2)CC1C1CCCC1 O=C1CN(C(c2cc[nH]c2)=O)C(C(=O)NOCc2ccccc2)CN1 CC(C)C(C)(CNC(C1(C)CC=CCC1)=O)NC(=O)COC1(C)CCOCC1 Cc1cc(C(=O)N(CC(C)CNC(C2(O)CCSC2)=O)C)ncc1C(F)F C12(CNC(C3COC(CNC(c4coc(C5CC5)n4)=O)C3)=O)CCCC1C2 C12(CNC(=O)NCCS(CC)=O)OCCCC1C2(F)F Nc1ccc(C(=O)NCC2(CNC(c3cc4scnc4[nH]3)=O)CCCC2)cc1F C1(C2CC2)(CNC(c2c(SC)cnn2C)=O)CCN(C(c2nc(Cl)sc2C)=O)C1 c1(OCCCC)ccc(C=CC(=O)NC2CC2NC(c2cccc[n+]2[O-])=O)cc1 N1(C(C=CC(=O)N(C)C)=O)CCC2CN(C(C34CC(F)(C3)C4)=O)CCC2C1 c1(CC(=O)NCC(CC)NC(=O)CC(C)(C)CCOC)c[nH]c2cc(Cl)ccc12 C(CCCCC(=O)NC1CC2(C1)CC(NC(=O)CNC(N)=O)C2)NC(C)=O CCCC(C)CC(=O)NCCCCCN1CCN(C(C2CCC(C)C2)=O)CC1 C1(CNC(C(F)=C(C)C)=O)CC2(CC2)CN1C(=O)Cc1cnc(C)[nH]1 C12(CNC(c3cccc(CC)c3)=O)CN(C(C3CC4CCC3O4)=O)CC1CCO2 C(CC1=CCN(C)CC1)C(=O)NC(c1ccc(CC(F)(F)F)cc1)C CN1C(=O)CCC1C(N1CCC(F)(C(N2CCC(CF)(CO)C2)=O)C1)=O C(=O)(CCC1=NNC(=O)CC1)N1CCC(C2CC2)(NC(c2cnc(OC)s2)=O)C1 c1(C(=O)NCC(CCOC)NC(C2(COC)CC=CC2)=O)sc2cncn2c1C CC1CN(C(=O)C(C)(C)C2CCC2)CC1NC(C1CCCN1c1ncccn1)=O N1(C(c2cncc(CC)c2)=O)Cc2ccc(CNC(=O)CCCC(N)=O)cc2C1 N1(C(CCC(=C)C)=O)CCC2(NC(=O)C3=NOC(C(C)(C)C)C3)CCCC12 N1(C(CN(C(=O)OC)C)=O)CCC(O)C(NC(c2sncc2C)=O)C1 Cc1ccn(C(C)CC(=O)NCC2CCN2C(=O)CCc2cn(C)cn2)n1 c1(CN(C(c2ccccc2)CO)C)cccc(S(N)(=O)=O)c1.N12CCCC(C1)C2 C1(C(=O)NC2CCCCCC2)C(C2CC2)CCN1C(C1(N(C)C)CCC1)=O Cc1cc(=NC2CC2N(c2ccccc2)C)[nH]c(N2CC3CCC(C2)C3O)n1 C1(CCC)CN(C(=O)C(C)(C)COCC)CCN1C(=O)C(CC)c1ccccc1 C1(NC(C2C(C)(C)C2)=O)C2CC3C(C2)C13C(=O)N1CC(O)CO1 N1(C(C(C)SCCCC)=O)Cc2nccn2CC(NC(c2cnsn2)=O)C1 c1(C(=O)NC2(CNC(C(C(C)O)(F)F)=O)CCCCC2)ccc2oc(O)nc2n1 CCCC(C)(CC)C(=O)NC1CCC2CCN(C(c3cc(C)nc(O)n3)=O)C12 C1(C)(CCNC(Cc2ccc(C)s2)=O)CCN(C(=O)C2=CCOC2)C1 c1(C(N2CCC(O)(C(C)NC(=O)Cn3ccnn3)C2)=O)ccc(N)cc1O C1(CC)CCN(C(=O)C(C)=CC(C)(C)C)C(C(=O)Nc2cccc(CO)c2C)C1 N1(C(c2c(C)onc2-c2ccccc2F)=O)CC2(CCN2C(C2CC2(F)F)=O)C1 CN1CC(C)(C(=O)NC2CC(CNC(C3C=CCCC3)=O)C2)CCC1=O n1(CC(N2CCN(C(C(CCC)C#N)=O)CC2C)=O)ccc2ccc(F)cc12 C1(O)(CNC(=O)CCC2CC2CC2CCCCC23CC3)CCCN(CC2CC2)C1 N1(C(c2ccc(SC)o2)=O)CC(C(=O)NCC2(SC3CC3)CCC2)C(F)(F)C1 CCC(CC)(CO)C(=O)NC12CC1CN(C(=O)CCc1cccc(F)c1F)C2 N1(C(C(C)OC(C)(C)C)=O)CC2(CNC(C3CC3F)=O)CC1CO2 CCCCC(CO)NC(=O)NCCC(N1CCOCC1)=O c1(C(N2CCOCC(NC(c3ncn(C(C)C)n3)=O)C2)=O)ccc(S(N)(=O)=O)s1 C12(NC(COCCC)=O)CC3CCC(C1C2)N3C(C1CCc2nnnn2C1)=O c1(C(=O)NC2(CC=C)CCNC2)cc2nc(O)[nH]c2cc1N C1(C(=O)NCCCCN(C)C(c2csnc2C2CC2)=O)CC2CC1CO2 c1(C(N2C(C)CN(C(C3CCCCN3N=O)=O)CC2)=O)ccc(S(N)(=O)=O)s1 C(=O)(N=c1[nH][nH]c2c1CN(Cc1cc(Br)cc(Br)c1F)C2)c1cc(C)[nH]c1 C1(CNC(c2cn(CC)nn2)=O)CN(C(c2csc3nnsc23)=O)C2CCN1C2 C(=O)(CCCCCF)NCCC1CC(C(=O)NCC2ON=C(CC)C2)C1 c1(OC)cc(CNC(=O)NCC2C=CCOC2)sn1 C(=O)(C(F)(F)C(F)F)N(CC)CC1CCN(C(=O)CC2CCCS2(=O)=O)C1 C(C(O)CC(=O)N1CCOC(CNC(=O)CCCC2CCCC2)C1)N(C)C c1(C(=O)NCC(CC(C)C)NC(CC(=C)Br)=O)ccc2cc[nH]c2c1F c1(CCC(N2CCOCC(CNC(c3cnn[nH]3)=O)C2)=O)nc2cnccc2[nH]1 N1(C(CCC(C)O)=O)CC2CN(C(=O)CN3CCOCC3)CC2C1 C1(Oc2cc(C)cc(C#N)c2)CCC2CN(C(=O)OC(C)(C)C)CC12O C1(C(=O)NCC(CC)Oc2ccccc2F)CCN(C(=O)CN(C)C)CC1 C1(NC(CCn2ccc(C)n2)=O)CCCCN(C(c2cnn(C)c2F)=O)C1 C(C(C)CC(=O)NCC(c1ccc(C(F)(F)F)cc1)O)OC C1(N(C(CSCC#C)=O)CC)CCCN(C(c2nn(C)cc2C(F)(F)F)=O)C1 c1(OC)ccc(C=CC(N2CCN(C(=O)CCCSC)CC2C(C)C)=O)cc1F Cc1cc(C(=O)Nc2ccc(Br)cc2I)cc2c1CCC2 c1(C(=O)NC2CCN(C(CCOCC#C)=O)C(C)C2)cc([N+](=O)[O-])ccc1SC N1(C(c2[nH]cc(C)c2C)=O)CCC(O)(CNC(c2c(C(C)C)n[nH]c2C)=O)CC1 c1(C(=O)NCC2(F)CN(C(Cc3c(F)ccc(C)c3)=O)C2)cc([N+](=O)[O-])cn1C N1(C(C2C(C#C)C2(C)C)=O)CCCC2(C1)CN(C(c1coc(CO)c1)=O)C2 c1(CNC(C2CCCSS2)=O)cccc(CNC(C2CCCC3CC23)=O)c1 C1(CC=C)(NC(=O)CCC(C)SC)CCN(C(=O)CCCc2sccc2C)CC1 C1(C(C)C)CN(C(=O)CCCC(N)=O)CCC1NC(c1cn(C)nn1)=O N1(C(CN(C(COC)=O)C)=O)CC(O)(CN(C(=O)CC2CC2C)C)C1 C12(NC(C3(c4cccc(OC)n4)CC3)=O)CC(CNC(=O)C(C)(C)O)(C1)OC2C C1(C(N2CCC(NC(C(C)c3ncco3)=O)(CO)C2)=O)(C(F)F)CCN(C)CC1 N1(C(Cc2cn(C)nc2)=O)CCCC(C2CCN(C(C3CCCO3)=O)CC2)CC1 C1(NC(c2c(O)cccc2F)=O)CN(C(=O)C=CC2CCCO2)CC12CCC2 C(CC(=O)NC1CC1NC(=O)CC1CCSCC1)(C(F)(F)F)OC c1(NC2c3cccc(OCC)c3CC2)ncc(C)cc1[N+](=O)[O-] c1(C(=O)NCC2C(NC(c3c(C)c(Cl)ccn3)=O)C2)ccc2ccnc(Cl)c2n1 C1(O)(C(CCNC(c2nc(OCC)sn2)=O)C)CCN(C(=O)C(C)OCC2CC2)C1 N1(CCNC(C=C(C)C(C)(C)C)=O)CCCN(C(C2CCCCN2C)=O)CC1 N1(C(c2cccc(NC(C)=O)c2)=O)CCN(C(=O)C(F)C2CCC2)C(CCO)C1 c1(C(=O)OC)cccc2sc(C(=O)NCC(C)(C)NC(C3C4CCCC34)=O)cc12 c1(CN(c2c(C(N)=O)cccc2Cc2ccccn2)C)cc(Br)ccc1O c1(C(N2CC(NC(C3(F)C(C)C3)=O)C(O)CC2)=O)cc2c(ncn2C)s1 c1(CCC(=O)NCCCCNC(CCC=C)=O)cccc2cn[nH]c12 c1(C(=O)NCC(C(C)(C)C)NC(CC2(COC)CC2)=O)ccc2nc(C)sc2c1 S(=O)(=O)(c1cnc(NCC(=O)NC2CCC2)c(Cl)c1)N1C(CC)CCOCC1 c1(OC)n[nH]c(C(=O)NCC2(CCNC(C3(C)CCC(=O)N3)=O)CC2)c1Cl N1(C(c2c(C)cc[nH]2)=O)CCn2ncc(CN(C(=O)C(C)CS(C)(=O)=O)C)c2C1 C=CCCC(C(=O)NC1CCS(=O)CC1)NC(=O)CNC(C1CC1C)=O c1(C(N(C(CN(C(CCCCOC)=O)C)C)C)=O)nccc2ccn(C)c12 C1(CNC(C2Cc3nncn3C2)=O)CC12CCN(C(=O)Cn1nccn1)CC2 CC1(C)CN(C(=O)CC2(O)CCOCC2)CC(C)(C)C1NC(C1CC1C(N)=O)=O CCC(F)(F)C(C)(C)C(=O)NCCN(CC(C)O)C(c1ncoc1C1CC1)=O C(=O)(N=c1cc(C)n(CCO)[nH]1)C1C(CC)CCN1C(=O)CC1(C#N)CC1 c1(OCCC(=O)NC2CN(C(C(CC)COC)=O)C2)ccc(Br)c(C)c1 C1(CC)CN(C(C2C(C)(C)OC2(C)C)=O)CCN1C(C1CC1C(C)(F)F)=O Clc1cc(Cl)ccc1-n1ncnc1-c1ncc(CC(C2CC2)C2CC2)s1.N C(=O)(C1CCCc2ncnn21)N1CCC2(CCN(C(=O)CC3CC=CC3)C2)C1 c1(CCC=C)ccccc1NC(c1cc(COC)no1)c1nnnn1C(C)(C)C c1(C(N2CCCC(C)(NC(c3n[nH]cc3F)=O)C2)=O)ccc(S(C)(=O)=O)cc1 C(CC(F)F)(C(=O)NOC(CO)C(C)C)N(C(c1nc(C)sc1)=O)C C1(NC(C(CSC)(C)C)=O)CCN(C(=O)C(C(C)(C)C)NC(C)=O)C(C)C1 N1(CC)Cc2ccccc2C(NC(=O)Nc2c(Cl)nc3sccn23)C1 Cc1ccncc1C(=O)Nc1nc(C(=O)O)c(C(C)C)s1 N1(C(C2(OC)CC2)=O)CC2CCC1CN2C(c1ccc(SC(F)F)o1)=O C(=O)(CC(C(F)(F)F)NC(=O)CNC(C)=O)Nc1cn(CCOC)nc1 C1(F)(CNC(Cc2cn(CC)nn2)=O)CCC(CNC(c2cnn[nH]2)=O)CC1 CCC(C(=O)N1CCC(NC(c2cc(C3CCOCC3)no2)=O)CC1)C(C)C C(C(C(=O)N1CC(CNC(=O)CCC2CC2C)C1)OC)OC C1(CC)CN(C(=O)CSC)CCN1C(C12CCC(NC(C)=O)C1C2)=O N1(CC)N=C(C(=O)N(C)CCC2CCCCN2C(=O)C=CS(C)=O)CCC1=O N1(C(C(C=C)(F)F)=O)CC2CCN(C(c3cccc(CC(C)C)c3)=O)CC2C1 C=CCCC(CC)(c1nnnn1C1CCCCC1)NC1(C)CC1(C)C C=CCCCC(C(=O)N1CC2CC(O)CC2C1)NC(c1ccoc1)=O C(CC(C)CC)(C(=O)NC1(C#C)CCOC1)NC(c1n(CC#C)ccc1)=O c1(CN2CC(C)N(C3CC3)CC2)nc2ccc(Br)cn2c1N c1(C(N(C)CC2CCCN2C(C2CCC(F)CC2)=O)=O)c(O)ccc(F)c1F C1(CN(C(=O)COc2cccnc2)CC)CCN(C(C2(C)CCC(C)C2)=O)CC1 C1(CNC(CSCC=C)=O)CCC(C(=O)NCC2CC23CCC3)CC1 N1(C(c2cccc(OCC)c2)=O)CCC(C(F)(F)F)C(C(=O)O)C1 C(c1ccc2c(c1)CCO2)=CC(=O)NCC1CCN(C(=O)CCN2CCCC2)C1 CC(F)(F)CC(=O)NCC12CC1CN(C(C1(CF)CC1)=O)C2 c1(OCC)ccc(Cl)c(C(=O)NCCCCNC(c2ccn(C(C)(C)C)n2)=O)n1 Cc1noc(Cl)c1CC(N1CCC1CNC(=O)CCN1CCCCC1)=O C(=O)(C(C)(C)CNC(C1CC(C)N1C(c1n[nH]c(=N)[nH]1)=O)=O)NCC C(=O)(C1CCCc2ccnn21)N1C(CCNC(CN=S(C)(C)=O)=O)CC(F)(F)C1 Cc1cc(Br)cc(F)c1C(=O)NCCN1CCN(Cc2ccc(O)cc2)CC1 Cc1cc(C(=O)NC(CO)C(C)NC(=O)C(C)(C)Cc2cnn[nH]2)cn(C)c1=O N1(C(C)=O)CC(C)(NC(=O)C=CC(C)NC(=O)CN(C2(Cl)CC2(F)F)C)C1 Cc1[nH]nc2ncc(C(N3CCC4C(C3)CN4C(=O)CCCOC(C)C)=O)cc12 C(C(=O)NCCC(O)CNC(c1csc(C(F)F)c1)=O)(C(C)C)NC(COC)=O n1(CC)nncc1C(=O)N(C1(C(=O)N(C)Cc2cc[nH]n2)CC1)C C1(C(N(C2CN(C(C(COC)OC)=O)C2)C)=O)Cc2ccccc2N1 Nc1c(C(=O)NCC2(O)CN(C(C3CC4CCC3O4)=O)C2)cccc1Br N1(C(c2cnsc2)=O)CCCC2(CCN(C(c3cc(F)cc(Cl)c3)=O)C2)C1 c1(C(=O)NC2(CNC(CC(CC)OC)=O)CC2)cc(C)n(C(C)C)c1C C1(C(=O)NC(C2(O)CCCCC2)C)CC(O)CN1C(=O)CCC1(C)CC1 C1(C(=O)NC(CC)CNC(=O)CN(C)C2CC2)CCc2cnnn2C1 c1(C(=O)NC(CCCC)CNC(=O)C(C)COC)cc(C(N)=O)cc(F)c1 c1(C(=O)NC2CCCC(CNC(CCC#CC)=O)C2)ccc(Br)c(F)c1C C1(NC(CCCC(=O)NCCC)=O)CN(C(=O)C(C)N2CC(C)C2)CC2(CC2)C1 c1(N2CC3C(NC(c4scc(C)c4Cl)=O)C3C2)ncc2cc(Br)ccc2n1 CC1COC2(CCCC2)CN1C(c1c(Cl)ncn1C)C(=O)NCCC1CC1 N1(c2cn(C)nc2)CCN(C(=O)C(=O)Nc2cc(C(N)=O)ccc2CN)CC1=O CN1CC(NC(=O)CCC2CCN(C(c3cnn(C)c3)=O)CC2)C(=O)N1 c1(-n2c(C(CCOCC)NCCc3cc(C)ccn3)nnn2)c(C)cccc1C C[Si](C)(C)C#Cc1ccc(CNS(=O)(=O)CCCC(=O)O)cc1 c1(C(N2CC(CC(C(=O)NCC(C)N(CC)CC)F)C2)=O)cnn(C)c1C C1(CNC(c2ncccc2Br)=O)CCCCCN1C(=O)C=CC1CCCO1 C1(CNC(C2CCCC2(F)F)=O)CCCN(C(=O)Cn2cc(CO)nn2)C1 C(CN=c1[nH]cc(C(F)(F)F)s1)c1c(C(C)OC)cc(F)cc1 CC1CN(C(c2ccccn2)=O)CC(C)CN1c1cccc(F)c1C#N C1(NC(CCc2cnc(C)s2)=O)CCN(C(=O)Cc2ccon2)CC1C(C)C N1(C(c2cn(CCC)nc2)=O)CCC(CC(C)NC(c2ccc(=N)[nH]c2)=O)CC1 CCCC(CC(C)C)C(=O)NCC1(C(=O)NC2(C)CC2)CC2(CC2)C1 Cc1ccc(N(c2ncc(C(F)F)cc2I)C(C)C)c(C)c1 N1(C(C2C(COC)C2)=O)CCCC1(C)CNC(=O)CP(C)(C)=O N1(CC(C)C)C(=S)NC(c2nn(C)cc2Br)C2=C1C(c1ccccc1Br)NC2=O c1(OCC)ccc(C2(C(=O)N(CC(C)(C)CNC(=O)C(CC)SC)C)CC2)cc1 N(C1C(=O)Nc2c(Cl)cccc21)c1nccc(=NCc2nnc(C(C)C)n2C)[nH]1 c1(C(N2C3(CNC(C(C(C)C)NC(C)=O)=O)CC(C2)C3)=O)cn(C)c(=O)cn1 C(C)(C(CC(=O)NC1(c2cc[nH]n2)CC1)NC(c1cc(=O)cc(C)[nH]1)=O)OC c1(C(=O)NC2CN(C(Cc3c(C)nc(C)s3)=O)C3C2C3)ccc2nc(O)[nH]c2n1 N#Cc1ccnc(N2CCC(NC(=O)C=CC3CCCO3)C2)n1 CCC(CC)C(C)C(=O)NCC=CC(N1CCC(C(=O)NC)C1)=O c1(C(N2CC(CNC(C3(F)CCCC=C3F)=O)C2)=O)ccc(F)cc1Cl C1(C(=O)NCCCc2nc[nH]n2)CCN(C(c2cccnc2S)=O)C12CC2 C(=O)(C(C)(C)N(C)C)NCCOCCCCC.C1(=O)C(F)CC2CN1C2 c1(C(C)=O)cn(CC(N2CCCC2CCNC(=O)CSc2nccn2C)=O)nn1 CC(C)C(C(=O)NC1CC(N(C(=O)CCc2ccccn2)C)C1)N(C)C Cc1ccc(C=CC(=O)NC2CCCCC2NC(C2CCNC2=O)=O)s1 CC(C)(C#N)CCCC(=O)N1CCC(CNC(=O)C2=NNC(=O)C2)C12CC2 C1(C(N2CC(CO)(CC3CCC3)C2)=O)(SC)CN(C(=O)CCN(C)C)C1 C(=O)(CC1=CCCCC1)NCc1cccc(NC(C2(OC)CCCOC2)=O)c1 C1(NC(c2cncc(Cl)c2)=O)CCC12CN(C(c1cncc(C3CC3)c1)=O)C2 C(CC(C(=O)N(C)CCc1ccccn1)NC(C1CCC1C#N)=O)OC CC(C)C1=NOC(C(=O)NCCC(O)C(=O)NC2CCCC2(C)CO)C1 CC1(NC(C2(C)CC2(F)F)=O)CCCC(F)(F)C1O C1(NC(c2c(F)ccc(C)c2)=O)CN(C(c2cn(C)nc2Cl)=O)CC1S(C)(=O)=O C=CC1(C(N2CCC(C)CC2CNC(=O)CNc2ccccn2)=O)CCOCC1 c1(OCC)ccc(C(=O)NCC2CCCCN2Cc2noc(C3CCC3)n2)cn1 c1(C(N2CC(C(C)C)N(C)CC2)C(=O)NCC2CC2)cc(Br)cc(Cl)c1F C(=O)(C(O)CC(F)(F)F)NCCc1c(CNC(COC(CC)CC)=O)nco1 c1(CCNC(C23CC(C2)C3)=O)ccc(-n2cc(CON3CC=CC3)nn2)cc1 c1(C(=O)NCCC2N(C(CC=CCC)=O)CCC2)ccc2c(c1)C(C)(C)CO2 C(=O)(CCCCCBr)NC1CC(C(=O)Nc2cc(CC)no2)C1 C#Cc1ccccc1CC(=O)NC1(CCOC)CCN(C(=O)C(C)C2CC2)CC1 C1(C(N2C(C)CC(NC(c3occc3Br)=O)C2)=O)CCc2c[nH]nc2C1 N1(C(CSC)=O)CCN(C2CCCN(C(c3csc(C(F)(F)F)n3)=O)C2)CC1 Cn1cnc2cnc(N(C3CCCC3)C(c3ocnc3C(F)F)=O)nc12.C1CN1 C=CC1CN2CC1NC(=O)CCCC2=O.C(=O)(COC(C)C)NCC(=C)F c1(C(N2CC(OC)C(NC(=O)CC3CS(=O)(=O)C3)C2)=O)c(N)cccc1Cl N1(C(COC(C)C)=O)CCC2CCC(NC(c3cc(C(N)=O)cn3C)=O)C1C2 c1(C(=O)NC2CCC(NC(=O)CCCC3CCOCC3)C2)ccccc1Br c1(CC)cc(NC(=O)CCC2CC(NC(=O)C(O)C3CCC3)C2)cc(C)c1 C1(CC(=O)NC2CC(CNC(c3cccc(C(C)C)n3)=O)C2)CCC2(CC1)CC2 C12(C)CCN1C2=O.C1(OC(=O)NN(C(C)C)C)CCN(C(c2ccco2)=O)C1 C1(CC(=O)NCC2CCC(C)CN2C(C2CCCC2)=O)(OC)CCC(C)(C)CC1 C1(C(C)C(=O)NC2COCC2F)CCCN(C(=O)CCc2cncnc2)C1 C1(NC(C(c2cn(CC)nc2)=O)=O)CCCCC1CNC(=O)C(C)C c1(C(C)C)cc(C(=O)NC2CCOCC2CC2CCN2C(=O)CO)c(C(C)C)o1 N1(c2ccc(-n3c(C)cc(C)n3)cn2)Cc2cncnc2C1.C(CCN)NC(=O)CN Cc1cnn(CC(=O)NOCC(=O)NCCCC2CCCCC2)c1 Cc1c(C(N2CC(CC(=O)NC(c3cccnc3)C)CC2(C)C)=O)[nH]ccc1=O c1(N2CCC(c3ccc(C)cc3)CC2)ncnc2c1ncn2CCC1(CSC)CC1 Cc1ccc(CC(=O)NCCCCNC(c2ccc(=O)n(C)c2)=O)cc1Cl N1(C(COC(CC)C)=O)CCCN(C(=O)C=Cc2ccsc2C(F)(F)F)C(C)C1 c1(C(=O)NCC2CC(NC(CC3(C)CCCO3)=O)C2)cccc(CO)n1 N1(C(c2c(C(C)C)n[nH]c2)=O)CC2CCN(C(=O)CC3CCC(F)(F)CC3)C2C1 Clc1nc(N2CC3CNCC2C3)c2[nH]c(Br)cc2n1 C1(C(=O)O)CC2(CCSCC2)CN1C(=O)Cc1csc(-c2ccco2)n1 C(CCCCC(=O)N1CCC(C)(CC(=O)N(C)CC2(CO)CC2)C1)N(C)C C1(COC)CN(C(c2cc(C(F)F)ccc2Cl)=O)CCN1C(=O)CC(C)(C)O Cc1cc(C(C)(C)C(=O)NC2CC2NC(c2cccnc2C2CC2)=O)ccc1F c1(C(=O)NC2CCCN(C(c3cncc(C)n3)=O)C2)sc(Br)c(C)c1C CC1(C)CCC(CNC(=O)CCc2ccsc2)N(C(c2ccc(Cl)o2)=O)C1 C1(F)(CNC(c2cc(C)[nH]n2)=O)CCCN(C(=O)C=C2CCOCC2)C1 c1(CC(N2CC(CNC(c3c(C)[nH]nc3Br)=O)C2)=O)ccc(F)c(Cl)c1 C1(NC(C=Cc2c(C)ccs2)=O)CCN(C(C2(C#N)CC=CC2)=O)CC1O c1(OC)ncc(-c2noc(CC3CCCN3C3CCOCC3)n2)c(=N)[nH]1 c1(C(=O)NC2C(OC)CN(C(=O)CC(O)C(C)C)C2)nc2ccccc2s1 N1(C(Cc2ccc(OC)cc2C)=O)CCCN(C(=O)C(OC)OC)CC1C(C)C CCC(C)(C)C(O)C(=O)N1CCC(N(CCO)C(=O)OCC(C)(C)C)C1 c1(N2CC(c3c(CNC(C(C)(C)NC(C)=O)=O)nco3)C2)nc(C)nc2n[nH]cc12 C(=O)(CC(O)C(C)C)NC(CCC(=O)N1CC(O)(CC(C)C)C1)C c1(NC(=O)Nc2cc(OC)c(OC(C)C)cc2)ccc2c(c1)CN(C)C2=O c1(NC)ccc(C(=O)NC(C)(CO)C(=O)NCCC(Cl)Cl)cc1 CC(CN1CCOCC1)C(=O)NCC1(F)CC(NC(C2(c3cc[nH]n3)CC2)=O)C1 N1(C(C(CC=C)C)=O)C2CCCC1CN(C(C1(F)CCOCC1)=O)C2 CS(=O)(=O)CCCC(=O)NC1CN(C(=O)CCN2CCC(F)C2)CC12CC2 CC1(c2nn[nH]n2)CCN(C(c2cnc(OCF)cn2)=O)C1 c1(C(=O)NC2C(NC(CCCCC)=O)COC2)cc([N+](=O)[O-])c(C)c([N+](=O)[O-])c1 O=C1CCCC2(CCCN(C(=O)C(N3CCCC3c3cc(F)cc(F)c3)=O)C2)N1 c1(CC(N2CCC(N(C(=O)Nc3cccnc3O)CC)C2)CC)ccc(F)cc1 c1(N2CCC3(CC(NC(c4ccc[nH]4)=O)C3)C2)c(F)cc([N+](=O)[O-])cc1F c1(C(=O)NCC2(C)COC2)nc(N2CCC(C(C)OCC)C2)cc(C)n1 c1(C(=O)NCC2CN(C(C=CC=CC)=O)CC2(C)C)cc2c(nn1)CCCO2 Cn1nnc2cc(C(N3CC(NC(=O)COCC4CC4)C4(CC4)C3)=O)sc12 Cn1ccc(C(=O)NCC(CNC(c2ncccc2C(F)F)=O)CO)cc1=O N1(C(Cc2c(CC)cccc2)=O)CCN(C(c2ccc(C)cc2)=O)C(CCO)C1 c1(C(=O)NCC(CC(C)C)NC(=O)C(Cl)=CCl)ccc2nnc(O)n2c1 CCC1=NOC(CNC(C2CC(N(C)C(C3CCCO3)=O)C2)=O)C1 C(C(C)(C(=O)N1CC=CC(O)C1)NC(c1ncsc1C)=O)SC CCCCCC(F)C(=O)NC(C1(O)CCCCC1)CNC(C1C=CCC1)=O c1(C(=O)NCCC2CN(C(CCC(=O)NC)=O)CC2C)cnc2c(c1)COCC2 C1(NC(C2CC2(F)F)=O)CCCCN(C(=O)Cc2csc(Cl)n2)C1 N1(C(=O)NCC2(CCO)CC2)CC2CCCCN2c2ccccc21 C(C(=O)N1CCCc2ccnn21)(C1CC1)NC(=O)C=CCF CC1(C)CCC(N=c2cccc(S(=O)(=O)NCCC3CCCCC3O)[nH]2)C1 C1(NC(C2(CF)CCC2)=O)CCOC12CCN(C(C1(C(F)F)CCCO1)=O)CC2 N1(C(COC(CC)CC)=O)CCN(C(c2cccc3ccnn23)=O)C2COCC12 C1(C#C)(C(=O)NC(C#C)C2CCC2)CCN(C(C2CC(C)(C)CO2)=O)C1 n1(CC(=O)N(CC(CN(C(c2cc(OC)nn2C)=O)C)O)C)cnc([N+](=O)[O-])c1 c1(C(N(c2ncc(OC)cn2)C2CC(N)C2)=O)ccc(F)c(C)n1 C1(CC(=O)NCC(CC(C)C)NC(CNC(CC)=O)=O)CCC(F)(F)CO1 c1(N2C3C(NC(c4ccn(C(F)F)n4)=O)(CCC3)CC2)nc(Cl)nc2[nH]cnc12 c1(C(=O)NC(CNC(c2scc(OC)c2)=O)C(C)C)ccc2c(c1)CN(C)CC2 N1(C(C(C2CC2)NC(C2CC(O)C(F)C2)=O)=O)Cc2cncnc2C1 C1(NC(Cc2cccc(OC)c2)=O)CCN(C(C2OCCO2)=O)C(C)C1 C1(CCNC(CCOC(C)C)=O)CSCCN1C(=O)Cc1coc(C(F)F)n1 c1(CC)nc(Cl)cc(=NC2CC(CNC(C3C4CC5CC(C4)CC3C5)=O)C2)[nH]1 N1(C(C(CC)OC)=O)CCC2(CCN(C(c3cc4cccc(Cl)c4s3)=O)C2)C1 c1(C(=O)NCCCC(C)NC(Cc2c(C)cccn2)=O)cc(O)cnc1N C1(CNC(c2ccc(C)s2)=O)CCC2CN(C(C3(C)CCCO3)=O)CC12 c1(C(N2C3C(NC(C(COC)(C)OC)=O)C(C3)C2)=O)cnc2c(C)cccc2c1 C#CC1(O)CCCN(C(=O)C(F)(CNC(C2(SC)CC2)=O)C(C)C)C1 C=CCC(CC=C)n1cc(C(C)(C)NC(C2CCOC2C)=O)nn1 c1(-c2cc(C)c(OC)c(C)c2)ccc2c(C(N3CCC(F)(F)C3)=O)n[nH]c2c1 Cc1cc(C(F)(F)F)c(N(CCCNC(C2(F)CCCC2)=O)C)nc1C CS(=O)C=CC(=O)NCC(CO)NC(=O)CCC(=O)c1ccc(OC(F)F)cc1 c1(CC(N2CCCC(N(C(=O)C(F)C(F)(F)F)CC)CC2)=O)ccc2c(c1)CCO2 N#CC1(C(=O)NCCCCNC(C2CCOCC2)=O)CCCCCC1 C(=O)(C(CCC1CCC1)NC(c1nonc1N)=O)N(C)Cc1ccsc1 Cc1sc2ncc(C(=O)NC3CCCCC3n3cccn3)n2c1C Cc1cc(C)n(C(C)C(=O)NC(C)C(C)(C)NC(c2cc(CC(C)C)[nH]n2)=O)n1 O=C(CCOCCOc1ccccc1)N=c1nc(-c2ccccc2Cl)[nH]s1 N1(C(CSCCCC)=O)CCN(C(C2(C)CC(C)=NO2)=O)CC1C c1(C(N2CCCC(NC(c3c(C)ncc(N)c3)=O)C2)=O)cc(S(N)(=O)=O)co1 C#CC1(NC(=O)CC2CCCC2NC(=O)C(C)(C)Cl)CCC(C)(C)C1 c1(C(C)C)cnc(O)c(C(=O)NC(C)(CNC(=O)CCC=CBr)C2CC2)c1 N1(C(c2n(CC=C)ccc2)=O)CC2(CC(NC(c3cnn(CCC)c3C)=O)C2)C1 c1(C(N2CCCN(C(c3cc(C)ns3)=O)CC2C)=O)cc2cc(O)ccc2[nH]1 c1(NC(C(CO)NC(c2cc(C)cc(O)n2)=O)=O)cccc(C#N)c1C N1(C(c2c(C(C)C)ncs2)=O)CC(NC(C2CC(C)(C)C2)=O)C(C2CC2)C1 Cc1ccc(C(=O)NCC(C2(O)CCN(C(=O)Cc3nncn3C)C2)C)nc1O C1(C)(C(N2CC=CC(NC(c3cc(C)oc3)=O)C2)=O)CCCCC1(F)F c1(C(N2C(C)(C(N(C3CCN(C)C3)CC)=O)CC2)=O)ccc(CO)cn1 c1(C(=O)NC(CCCC)CNC(C2(C#N)CC2)=O)cnc(F)c(Cl)c1 C1(CNC(Cc2cccc(C)c2)=O)CCCC2(CN(C(C3CC34CC4)=O)C2)O1 c1(OC)ccc(Br)c(F)c1CN1CCn2ncnc2C1 c1(OC)cccc(-c2ncc(C(N3CC(C(=O)N(C)C)C3)=O)s2)c1 N1(C(C)C)CCCN(C(C2CCC(NC(=O)C(C#N)C3CC3)CC2)=O)CC1 C1(NC(=O)CC2CCOC2)CC2CCC1N2C(c1c(Cl)nsc1Cl)=O CCCCCC(F)C(=O)N1CC(OC)C(C(=O)NCCCc2cccs2)C1 C1(NC(c2nnc(C)s2)=O)CC(CNC(=O)Cc2cc[nH]c2)C12CCC2 N1(C(c2c(CC)onc2)=O)CCN(C(C)CNC(=O)C(C)(COC)OC)CC1 CC(CC(=O)N1CCC(C(C)(C)NC(=O)Cn2cccc2)C1)C(F)F Cc1ccncc1N(C(=O)C(C)CNC(=O)COC1CCCC1)C c1(C(C(=O)NC(CNC(C(c2cncnc2)C)=O)C2CC2)(C)C)ccccc1F c1(CCCC(=O)NCCN(C(Cc2c(C)cco2)=O)C(C)C)ccc(F)c(F)c1 N1(C(c2c(F)cc(O)cc2F)=O)CC2(C1)CN(C(=O)C(O)C1CCC1)CC2CO CCCN=C(NCc1cccc(OC)c1OC)NC1C(F)(F)C12CC2 c1(OCCC)cc(C)ccc1CNCc1ccn(C)c1C1CCC1 c1(C(N(CC(CNC(C(F)OC)=O)C)C)=O)ccc(C(N)=O)c(Cl)c1 N1(C(C2(NC(c3ncn(C)n3)=O)C(C)CCC2)=O)CC=C(CO)CC1 C(=O)(CC(F)(F)CC(=O)N1CCCC(NC(c2cccc(CO)c2)=O)C1C)OC C1(O)(CNC(c2c(CC)cco2)=O)CCCN(C(c2ccncc2C(F)F)=O)C1 c1(C(N(C)CC2N(c3nnc(C)s3)CCC2)=O)nn(C)c(Cl)c1Cl c1(N(C(CCC(=O)N(C)C)=O)CC(=O)N(C)C)ccc(C(F)(F)F)cc1Cl c1(OCC)ccc(SCC(=O)NCC23CC2CN(C(=O)C(C)(C)C#N)C3)cc1 CC1CCC(C(=O)NCc2cccc(C#N)n2)N(C(c2cc(C(F)F)[nH]n2)=O)C1 c1(CC(=O)N(C2CN(C(c3cc(C(CC)C)no3)=O)C2)C)ccc2nsnc2c1 C1(C)(NC(c2ncn(C)n2)=O)CCN(C(c2cc(C(F)(F)F)ccc2Cl)=O)CC1 N1(C(C(CC(C)C)NC(C2N(CC)CCOC2)=O)=O)CC2C3CCC(C3)C2C1 CC=C=CCCN=C(NCc1csc(C(F)(F)F)c1)NCC(C)C N1(C(C2CCNCC2)=O)CCOC2(C1)C1CC3CC(C1)CC2C3 C1(NC(c2ccc(CSC)o2)=O)C2CC(NC(c3c(C)noc3C)=O)CC12 C1(N(C(CC2(OC)CC2)=O)C)CCCC2CN(C(=O)C=CC(C)(C)SC)CC12 CCC(F)(F)CC(=O)NC(C)(CNC(=O)C(C)OCC1CC1)C(C)C C(CC(=O)NCC1(CO)CCN(C(C2(C)CC=CCC2)=O)CC1)(C(F)(F)F)OC O=C1CC(C(=O)N2CCC(C(F)C(=O)NCc3ccc(O)cc3)C2)=NN1 c1(C(=O)NCC2(C)CCCN(C(C3(C#N)CC=CC3)=O)C2)nnn2ccccc12 C=CCCCCCC(=O)NCCCCC1(NC(=O)C(F)CCC)CC1 c1(OC)cc(OC)c2cc(NC(C3COC(CN)C3)=O)[nH]c2n1 C1(C(=O)NCC=C(C)C)COCCC1NC(c1ccon1)=O N1(C(CC2ON=C(CC)C2)=O)CC(NC(c2c(CC)cccc2F)=O)CC(C)C1 O=C1CC2CC1CC2C(=O)NC(C1(O)CCCCC1)C(=O)N1CCC1C1CCC1 FCCCN=C(NCc1ccc(Cl)cc1)NCc1ccc(OCC2CC2)cc1 C1(C(N(CCCN(C(C2CN(CC)C(=O)C2)=O)C)C)=O)CCN(C)C(C)C1 C(=O)(C(C)C(C)NC(C1CCO1)=O)NCc1nc(CC)[nH]n1 c1(NC(=O)NCCCN(C(C)=O)CC2CC(OC3CC3)C2)ccccc1 c1(CC#N)cccc(C(=O)NCC2CCC2NC(=O)C=CCO)c1 C(CCCC(CO)NC(=O)CC1CCC(C)(C)CC1)NC(Cn1ccc(C)n1)=O N1(C(C(=Cc2cccnc2)C)=O)CC2CC3CC2C1C3NC(C1CCC1(F)F)=O c1(-c2cc(CNC(c3c(NC)cnnc3)=O)ncc2)cnc(F)cc1C C1(C(N(CCN(C(C2CC(C(F)(F)F)(OC)C2)=O)C)C)=O)COC2(CCC2)C1 c1(C(=O)NCC2CN(C(c3cnn(CC)n3)=O)C2)ccc(OC(F)(F)F)nc1 c1(C(=O)NC23CC(C(N(C)CC45CCC(CC4)C5)=O)(C2)C3)cc2cc[nH]c2cn1 c1(CCSc2n(C(F)(F)F)c(CC3CC3)nn2)nc2c(Cl)ccnc2[nH]1 C(=O)(C(CC(C)C)NC(C)=O)NC(CNC(Cc1cn(CC)nc1)=O)(C)C(C)C CC1CN(C(c2cccc(C(N3CC4(CCOCC4)C3)=O)c2)=O)C(C)(C)CO1 c1(C(=O)OCC)c[nH]c(=NCC2(C)CCN(C(=O)C(C(C)C)N(C)C)C2)s1 Nc1ncc(C(=O)NC2CCN(C(=O)Cc3csnn3)C2)cc1CO N1(C(C(C)(C)OCC)=O)CCC(NC(=O)CCCOc2ccccc2C)C(C)C1 C1(CCN(C(=O)C(C2CC2)N(C)C)C)CCN(C(=O)CCC2(C)N=N2)CC1 c1(OCC)cc(C)ccc1OCCC(=O)Nc1ccc(CC)cc1 C(=O)(C(O)C(F)(F)F)N1C(CNC(C2CCC(CCC)CC2)=O)CC(COC)C1 C(N=c1[nH]nc(CO)s1)C1CN(C(C2(F)CCCCC2)=O)C1 Cc1cc(C(N2CCC(CC(=O)NC(C3CCCC3)C)C2)=O)cc(C)c1F N1(c2nccc(OC(C)C)n2)CCCN(C(c2cc3ncccn3n2)=O)C(C)C1 C(C)(N=c1ccnc(NCc2csc(-c3ccccc3)n2)[nH]1)c1c(CC)nns1 c1(CC(=O)NC(C(C(C)C)Nc2cnccc2Cl)C)ccc2ccccc2c1 c1(CC(C(=O)NC(C)(C)CNC(=O)CC(C)F)OC)ccc(F)cc1 N1(C(c2c(OC)csc2)=O)CC2CC(NC(=O)C(C)N3CCC3)CC2C1 c1(CC(=O)NCCN(CCOC)C(C23CC(C)(C2)C3)=O)ccccc1F C1(C)(NC(Cc2cccc(C)c2)=O)CCN(C(=O)COCc2ncnn2C)CC1 c1(CC(=O)NC(C2CCOCC2)C(=O)OC)nc(C)sc1Cl Nc1cc(C(=O)NC2C3CN(C(=O)OC)CC23)ccc1F.C12CC(C1)OC(=O)C2 C1(NC(C23OCC(COC)(C2)C3)=O)COC2(C1)CN(C(=O)C(C)CC1CCC1)C2 CCC(CC)C(CNC(c1c(OC)cccc1N(C)C)=O)NS(C)(=O)=O S(=O)(=O)(c1cnnc(C)c1C)NC1(C(=O)OC)C(C)C1C n1(CC)nc(C(=O)NCCC2CCCN(C(c3ccncc3)=O)C2)c(Br)n1 N1(C(c2oc(CC)c(C)c2)=O)CC(CC(=O)N(C(C)CCSC)C)C2(CC2)C1 c1(NC(c2nc(C)n(C)c2C)c2n(CC)nnn2)nc2cnccc2[nH]1 N1(C(CSc2c(C)n[nH]c2C)=O)C2CCC1CN(C(=O)C(C)C(C)C)CC2 N1(c2ncc(C)cn2)CCC(O)C(c2nc(C(=O)N)no2)C1.C(C1CC1)CCO C1(NC(Cc2cccc(C)c2)=O)CC(O)CN(C(c2cnccc2C)=O)C1 C(=O)(C1=CCCCC1C)N(C1CC(C(=O)NC(C(=O)NC)(C)C)C1)C N1(C(C2(C)N(C(c3cccc(C)c3C)=O)CCC2)=O)CCC(O)C(C)(C)C1 C1(COC)(NC(=O)Cc2cn(C)nn2)CCN(C(=O)CC(C)(C)O)C1 c1(C(N(C(C)CCNC(=O)CN2CCC2C)C)=O)cn(C)nn1 c1(CN(C(=O)CCC2(C)CC2)C)cccc(CNC(=O)C(C)(C)c2cnco2)c1 c1(CCC)cn(CC2(CN(C(c3cocn3)=O)CC)CC2)nn1 C(=O)(C(C)(O)CC(C)C)NC(CNC(c1cc(C)c(O)cc1)=O)C c1(C(=O)NCC(C)NC(c2c(SC)csc2)=O)cccc2ccc(C)nc12 Nc1ccc(C(N2CCC(NC(C3CC4CC3C4)=O)CC2)=O)cc1Cl n1(CCC)nnnc1C(CCOCC)NC(CC)C(=O)OCc1sccc1C CC1CC2(CC(NC(C3(NC(C4CCCCN4C)=O)CC(F)C3)=O)C2)C1 c1(C(N2C(C)C(NC(C3CC3F)=O)CCC2)=O)cccn2c(CO)nnc12 Cc1nn(C)c(C)c1C(=O)NC1CC(C)CN(C(c2cccn(C)c2=O)=O)C1 C1(CNC(CCCN(C)C)=O)CCCCN1C(=O)COCCC1CCCC1 C1(F)(C(N(OCC)C(C)C)=O)CCCN(C(=O)CN(C)C2CC2)C1 c1(C(=O)NCC2CC(OC)CN2C(c2cc(C)cc(F)c2)=O)c(C)cncc1F c1(N2CC(CCSC)OCC2)cc(C)c(S(=O)(=O)NCC(F)CO)cn1 c1(C(S(=O)(=O)c2ccc(Cl)nc2)=O)ccc2nc(-c3ccc(I)cc3)sc2c1 Cc1nc(F)ccc1-c1cn(CC(F)CCNC(C2(CO)CC2C(F)(F)F)=O)nn1 c1(C(C(=O)NCC=C)N2CCC2c2ccc([N+](=O)[O-])cc2)ccc(C)c(F)c1F c1(C(=O)NC2C(CNC(CCSCCCC)=O)CC2)cnccc1N(C)C C(C(CNC(c1occc1-c1ccccc1)=O)CO)NC(=O)CCn1cnnn1 C(=O)(CCC(F)(F)F)NC(C1CCCN1C(c1ccc(C2CC2)cc1)=O)C C(=O)(CCCCCC#N)NCC(C(C)(C)C)NC(c1c(C)nn(CCC)c1C)=O Cc1cc(Br)sc1NC(=O)OC(C)(C)C.C1(=O)NNC(=O)C12CC2 c1(CC)conc1C(N1CC(C(C(=O)NC(CC)CO)OC)C1)=O c1(C(N(C2CC(NC(=O)Cc3ccoc3)C2)C)=O)cnc(O)cc1C(F)(F)F CON=CC(=O)NCC(C)(Cn1cccn1)NC(c1ccsc1Br)=O C1(CC(=O)NCC(CN(C(=O)CN2CCC(C)(C)C2)C)(C)C)CC2CCC1C2 C(=O)(C(C)(F)C(F)(F)F)NCCCc1cn(-c2scc(C(=O)OCC)n2)nn1 c1(C(=O)NC2C(CC)N(C(C3CCCC3)=O)CC2)ccc2c(n1)OCC(=O)N2 c1(N2CC(CNC(C(CC#C)(C)C)=O)N(C)CC2)nc(C)nc2c(C)csc12 c1(C(N(CCCCCNC(=O)CCOCC(F)(F)F)C)=O)cccc(OC)c1 CC1(CNC(=O)C=Cc2cccnc2)CCCC1NC(=O)CCc1cccnc1 c1(CCC(=O)NCCC2CCN(C(=O)C3=CCSC3)C2)ccc(Cl)cc1F c1(C(N2CCCC2CCNC(C23COCC2C3)=O)=O)cnn2c1S(=O)(=O)NCC2 C(=O)(N=c1cc(C)o[nH]1)C1(C)CCCN(C(C2CCC(CCCC)CC2)=O)C1 CCC(C)C(C)(O)CNC(=O)CCN(C(c1c[nH]c(C)c1)=O)CC1CC1 c1(C(=O)NCCOCCNC(C2C(C(=O)OC)C2)=O)noc(C2(C)CC2(F)F)n1 C1(CCNC(CC(=C)C)=O)C(C)CCCN1C(=O)COCC(=C)C c1(CN2CCC3(C(C(N4CCC(NCC#C)CC4)=O)C3)C2)c(F)cc(Cl)cc1F N1(C(c2cc(C(C)=O)sc2)=O)C2CCC1CN(C(c1cc3n(n1)CCCC3)=O)C2 C(=O)(CCC1(C)N=N1)N(CC(=O)NC(C1CCCC1)CC)CC1CC1 C(=O)(C1=NN(CC)C(=O)CC1)N1CC(O)(CN(C(C(CC)F)=O)C)C1 c1(C(=O)NC2(CF)CCN(C(c3n(CC=C)ccc3)=O)C2)cn(C)ccc1=O Cc1cccc(C(=O)NC(c2cn(C)nn2)C(N2CCOC(C3CC3)CC2)=O)c1C C1(C(N2CC(C)C(NC(c3ccc(CC#N)cc3)=O)C2)=O)CCC2C(C1)C2(F)F Cc1cccn2ncc(C(=O)NC3CC(NC(=O)CC4CC5CC5C4)C3)c12 Cc1sc(C)c(C(N2CC(NC(c3ncn4c3CCC4)=O)CC(F)C2)=O)c1C#N c1(CC)cc(=NC(=O)NC(c2nnc3n2CCOC3)C)cc[nH]1 N1(C(c2ccc(F)cn2)C(=O)NCCCC)CCCCC12CCC2 N1(C(CC2(N(C)C)COC2)=O)C2CCC1CN(C(C1CCS(=O)(=O)N1)=O)C2 Cc1ncccc1CC(=O)NC1CN(C(c2cn(C)nc2C)=O)CC1C(F)(F)F c1(C(N(C(C)C(=O)NC(C2(CO)CC2)C)CC)=O)ncccc1F C1(C)(C(N(CCN(C(C)C)C(c2cnnn2C)=O)C)=O)CCCN(C)C1 C1(OC)CC(NC(C23CCCN2CCC3)=O)CN(C(c2cncc(N)c2C)=O)C1 c1(C(C)C)ccc(C(N2CCC(OCCNC(C3(C)CCCO3)=O)C2)=O)c(F)c1 Cc1ccc(C(N2CC(NC(=O)COCC3CCC3)CC(F)C2)=O)c(F)c1F C(CC(C)C)(C(=O)NC1(CC(N)=O)CCC1)ONC(C1CC=C(C)CC1)=O Cc1cnc(N(C)CC2CCCCC2)c(S(=O)(=O)NCc2ccc(C)c(F)c2)c1 N1(C(COC(C)(C)C(F)(F)F)=O)CC(F)(F)CC1CNC(C1CC1(C)C)=O N1(C(C2C(CCC)CN(C(=O)CC3(C)OCCO3)C2)=O)CCC2(CCCC2)CC1 N1(C(C(C)N(C(c2c(C)oc(Cl)n2)=O)C)=O)CC(CO)CC(C)C1 c1(NC2(CC=C)CN(C(=O)C(C)C(C)O)C2)ncnc2c1ccn2C(C)C C1(C(=O)NC2CC(NC(=O)CCCc3cnn[nH]3)C2)OC2CCC1CC2 C(=O)(CCCCCC#N)NC(C(C)NC(CCC(=C)Br)=O)(C)C Cc1ccc(Br)c(CNCC2(CF)CCN(C(=O)OC(C)(C)C)C2)c1 c1(C(C(N2C(C(=O)NCC(C)C)CCC2)=O)C)ccc(N(C)C)cc1 c1(CC(=O)NCC2(NC(C3C(C#C)C3)=O)CCOCC2)cccc2nonc12 C(C(CC)(CC)C(=O)NC1CC(O)C(O)C1)NC(c1ncc(CC)cn1)=O c1(C(N2CC(C)C(CNC(=O)CCc3ccncn3)C2)=O)c(F)ccnc1F C1(NC(C(C)O)=O)CN(C(c2cc(Cl)cc(Cl)c2O)=O)CC2(CCOCC2)C1 C(=O)(CC(C)C(C)(C)NC(c1cnn(C)c1)=O)NCC(C)S(N)(=O)=O c1(C(=O)OC)ccnc(N2CCC(c3ccccc3)CC2)c1I C(C(C)C(F)C(=O)NC1(CCOC)CCCC1)NC(COCCCOC)=O c1(C(N2CCC(N(C(COCCC#C)=O)CCC)C2)=O)ccc(C)cc1 C1(CNC(CN(CC)CC)=O)C(C2CC2)CCN1C(c1ncn2c1CCCC2)=O c1(OC(C)C(N2CCC(NC(=O)CCc3cc(Cl)cs3)C2)=O)ccccn1 N1(C(C2CCN(C)C2=O)=O)CCC(O)C(NC(C2(CC3CCC3)CC2)=O)C1 C(=O)(C(C(=O)OC(C)(C)C)C(C)C)NCCCCCCN(C(C(C=C)(C)O)=O)C O=C1CCC(CNC(=O)CN(C2CCC2)C(c2ccn(C3CC3)n2)=O)N1 N1(C(C(C)OC)=O)CCCC12CCN(C(c1c(C3CCCC3)noc1C)=O)C2 N1(C(c2c(C(=O)NCc3c(CC)cccc3)cccc2)=O)CC2(C)CC1(C)CO2 C1(C(N(CCCNC(c2ccc(C3CCC3)nc2)=O)CC)=O)CC2CCCC2C1 C1(C(C(=O)N(CCC(N)=O)CC)(C)C)CCCN(C(=O)CC(C)C)C1 c1(C(=O)NCC2C(NC(C(C)Cc3ccco3)=O)C2)cccc2c1CNC2=O Cc1cccc2cc(C(N3CCC4(NC(c5ncccc5O)=O)CC4C3)=O)oc12 c1(NCC2C(NC(C(CC)OC)=O)CCC(C)(C)C2)cccc(F)c1[N+](=O)[O-] Cc1cc(C(=O)NCC(CC(C)C)NC(c2sncc2C)=O)c(Cl)cn1 c1(C(=O)NC(CNC(C2(SC)CCC2)=O)C2CC2)cc(C)nn1CC(F)(F)F N1(C(=O)CC2CCCN(C(=O)Nc3ccccc3)C2)CCc2cc(O)ccc2C1 C1(C(N(C)CC2CCN(C(c3cccc(C)c3Cl)=O)C2)=O)CC2(CCCCO2)C1 N1(C(c2cc(C)on2)=O)CC(N(C)C(c2ccc(NC(N)=O)cc2)=O)C(O)C1 C12(C(=O)NC3(CNC(C(C)N(C)C)=O)CCCCC3)CCC(N=[N+]=[N-])C1C2 c1(OC)cc(C(=O)NCC2CC3CC3N2C(c2ccnn2CCF)=O)cc(F)n1 C(=O)(CCCC(F)(F)CO)NC(CCCCNC(C=CC(C)(C)C)=O)CO O=C1CC(C(=O)NC(c2cccnc2)C(=O)NCCCC(F)(F)F)CCN1 CCS(=O)CC(=O)NCCc1ocnc1CNC(=O)C=CS(C)=O C1(C(=O)Sc2ccc(-n3cc(C(C)(C)OC)nn3)cc2)CCOC2(CCCC2)C1 c1(C(N2CC(F)(CNC(C3C(C)(C)CC3)=O)C2)=O)ncn2cc(Br)sc12 c1(C(=O)NC(C(C)NC(C(COCC)(C)C)=O)C)ccc(OC)c(F)c1 C(=O)(CC(C1CC1)C1CC1)N1CC(CC(C)NC(C2C(CCC)C2)=O)C1 c1(C(=O)NC(C)(C)CCNC(=O)CC2C=CCCC2)cnc2c(c1)NCC2 C1(O)(CCNC(C2(Cl)C(C)(C)C2)=O)CCCN(C(=O)Cc2ccsc2)C1 N1(C(=O)CC2(N3CCCC3)CC2)CCOCC(NC(C2(O)CCSCC2)=O)C1 n1(CC(=O)NC(C2(O)CCN(C(C3(O)CCC3)=O)C2)C)cnc2c1CCCC2 C1(CCC=C)(C(=O)NCC=CC=C)CN(C(=O)C(C2CCCCC2)O)C1 N1(C(C(CSC)O)=O)CCN(C(=O)CCCN2CCN(CCOCC)CC2)CC1 C(=O)(CCCS(C)(=O)=O)N1C(CNC(C2N(C(C)C)CCCC2)=O)CC1 C1(CNC(C2C3COCC23)=O)CCCCN1C(C1(F)CCCC1)=O N1(C(C2C(CCOC)C2)=O)CC(CNC(c2cc(Cl)c(C)cn2)=O)C2(CC2)C1 C1(CCNC(c2c(C)[nH]cc2)=O)CC(F)(F)CN1C(=O)CNc1cccc(F)c1 C1(N(C=O)O)CCCCC1Cc1c(CC)nsc1.C1CCCC(F)C1 N#Cc1ncc(NC2CC3CCC2N(C(=O)C(F)(F)C2CCCC2)C3)nc1C#N C1(NC(c2cn(CC)nc2)=O)CC2CCC(C1)N2C(=O)CCN(C1CC1)CC C#Cc1ccc(CC(=O)N(CCNC(c2nn(C)nc2Br)=O)C(C)C)c(F)c1 C(=O)(C(C(C)CC)N(C(=O)CN1CC2CC2C1)C)NCCC#C Cn1nnc2c1CCN(C(c1cc(CO)on1)=O)C2.C12(CCC1)CCNC2=O Cc1nn(Cc2ccccc2Cl)c(=O)n1C1CCCC1 CC1CN2CCN1C(C(N1C3CCC1C(CNC(=O)C(=O)NC1CC1)C3)=O)C2 N1(C(=O)COC2C=CCC2)CC2CCCC(C1)N2C1CCc2c(Cl)cccc21 CCC(C)CCC(O)CC(=O)N1CCC(NC(=O)C=CC2CCC2)C(CO)CC1 c1(C(=O)NCC2CN(C(C3CCC(=O)N3)=O)CC2(F)F)cc2nc[nH]c2cc1F C1(C(N2C(C(=O)NC(C)(C)C)CC(OC)C2)=O)CC12CCSCC2 C(CCN=C(NCC1CCC1)NC1CCS(=O)(=O)C1)OCC c1(CC)nccnc1C(=O)NCCCOCCCNC(=O)C=Cc1ccncn1 c1(C(=O)NC2CCCN(C(CC3C(=O)NC(=O)N3)=O)C2)cn2ccnc2cn1 Cc1cc(-c2ncc[nH]2)ccc1NC(c1cnc(C2CCOCC2)o1)=O c1(SCC(=O)NCC2(NC(C=CC(CC)=CC)=O)CC2)ccccc1[N+](=O)[O-] C1(C(C)NC(C2CCCO2)=O)CCCN1C(=O)C=C1CCSCC1 C(=O)(CC(C)C(F)F)N1C(CN(C(c2nn(CC)c(C)c2)=O)C)CCC1 C1(CC(=O)N(CCCCNC(=O)C(C)(C)c2ccsc2)C)CN2CCC1CC2 C1(CC(=O)N(CCCNC(CC=CC)=O)C)CCCCN1C N1(C(CCOC(C)=O)=O)CC=C(C(=O)NC(C)C(F)F)C1 C1(OC)CN(C(=O)CCCC#N)CC1NC(=O)CC1CCOC1 C1(C(C)NC(=O)Cc2cnc[nH]2)CCN(C(C2(C3CCCCO3)CC2)=O)C1 C=C(F)C1(CC(=O)NC2(C(=O)NCCCN3CCCC3=O)CC2C)CCC1 c1(C(=O)NC2CC(NC(CCCCCCC)=O)C2)cnc2c(C)cnn2c1 N1(C(C(=O)NC)C(C2CCC2)OC)CCOC2(CCN(C)CC2)C1 C1(CC(C)(C)C)CN(C(=O)C(=O)NCC2CCCN2c2ccccc2)CCO1 c1(C(=O)NCCCCNC(C(n2ncc(C)c2)C)=O)cn(C)nc1Br N1(C(CC2CNC(=O)O2)=O)CCN(c2cc(C3CC3)no2)CC1 C=C(C)C1OCCC1C(=O)NC1CN(C(=O)C(=Cc2ccccn2)C)CCC1F C(=O)(C(O)CC1CCCCC1)N(C1CCCC1)CCCNC(C(C1CC1)SC)=O N1(C(C#CC(C)(C)O)=O)CCC2(C1)CN(C(C1CC13CCCC3)=O)C2 Fc1ccc(NC2(c3nnnn3C3CCC3)COC2)c(F)c1Cl N1(C(c2c(CC)nns2)=O)CCC(C)C1CNC(=O)CC1CSCCS1 C(=O)(C(=O)C(C)(C)C)NC(C1CCN(C(C2OCCOC2(C)C)=O)CC1)C CCCC1C(N2CC=CC(C(=O)OC(C)(C)C)C2)C(=O)N1.N(C)CC CC1C(C)N(C(=O)CCOc2cccnc2)CCN1C(c1cc2n(n1)CCC2)=O C1(C(C)NC(COC(CC)(C)C)=O)CCN(C(c2ccn(C(C)C)n2)=O)C1 CC1=NN(C)C(=O)C1CC(=O)NCCC1CC(NC(C2CCSCC2)=O)C1 C1(CNC(c2c(C(=O)NC(c3ccccc3)C)cccc2)=O)CCC2(CC2)CO1 c1(C(C(=O)NCC(CC)NC(C=CC=CCCCCC)=O)F)ccc(F)cc1F C1(C(=O)NC2CC(Cn3cc(CCS(N)(=O)=O)nn3)C2)CC2(CCO1)CC2 c1(CCC)cc(C(=O)NC2(CO)CN(C(c3nn(C)cc3SC)=O)C2)c(C)o1 CC1CCCC1(C(=O)NOCCC#N)NC(c1cccc(SCCCO)c1)=O CC(C)CC(O)C(=O)N1CC(NC(c2ccc(F)c(F)c2)=O)C(C(F)(F)F)C1 C(C(CC(=O)NCCCCCF)NC(=O)COCC1CCC1)OC C1(CNC(COCCCC#C)=O)CCCCC1NC(=O)CCC1CCC1 C1(NC(C)C(C)n2ccnc2)CCN(CC(c2ccc(F)cc2)N(C)C)CC1 C1(CCCC)C(=O)NCCN1CC(C1CCC2(CC1)CC2)=O C(=O)(C(C)CC(=O)NC1CC2CC(NC(c3cc(Cl)cs3)=O)CC12)OC C1(NC(=O)CCc2cnoc2)CCSC12CN(C(C1C3CCCCCC13)=O)C2 c1(C(=O)NC(CC)(CNC(C2(S(C)(=O)=O)CC2)=O)CC)coc2cc(C)ccc12 c1(CC(=O)NC(C(C)NC(C(C)=CC)=O)(C)C)csc2cc(Cl)ccc12 c1(C(=O)NCC(C)NC(=O)COCC(F)F)cccnc1Sc1ccccc1 N1(c2nc(C)nc(Cl)c2)CCC2(CCCC2NC(C2CCOC2)=O)CC1 C1(C(N2CC(N3C(=O)CC(NC(c4ccc(C)o4)=O)C3)C2)=O)CC12CC(C)(C)C2 C1(OCC)CN(C(C2CCC(NC(=O)CC3CCCO3)C2)=O)CC12CC2 c1(C(=O)OCC)cc(CN2CCC(CO)(COC)CC2)ccc1O.c1ccccc1 c1(C(=O)NC2(CN(C)C(C3CC3C(F)F)=O)CC2)cnc2nccn2c1 N1(C(Cn2ncc(C#C)c2)=O)CC(C(N2CC3C(C2)C3(F)F)=O)C(F)(F)C1 N1(C(C2C=C(C)CS2)=O)CC2CCC2(CNC(=O)CC2(C)CCCCC2)C1 C1(OC)(CNC(c2nccn2C(C)C)=O)CN(C(c2sccc2OC(F)F)=O)C1 Cc1c[nH]cc(C(=O)NCC(C)(CNC(=O)C(C)(O)CCN(C)C)OC)c1=O C1(C(=O)NCC2(CN(C(=O)C=C3CCCC3)C)CC2)CCc2nncn2C1 c1(NCCOC)cc(C(N2CCC(C(C)NC(=O)Cc3ccsc3)C2)=O)ccn1 C1(CNC(C2(COCC)CCC2)=O)(CNC(c2cncc(Cl)c2)=O)CC12CCC2 N1(C(C)C(N2CCC(N)CC2)=O)CCCCC1C1=NCCN1C O=C(C1=NOCC1)N1CCCCC1CNC(C1(n2cc(Cl)cn2)CC1)=O c1(C(C)NC(c2c(CNC(c3c(CC)c[nH]c3)=O)cc[nH]2)=O)cccc(O)c1 c1(CN2CCCC(C(=O)Nc3ccc(O)cc3F)C2)cnc2ccccc2n1 CC1=C(C(=O)NCC2(F)CCC(CNC(C3CC(C4CCC4)C3)=O)C2)SCCO1 Cn1nc(C(=O)NC2CCC2NC(C2(c3ccccc3)CCCO2)=O)ccc1=O N1(C(C2C(C)OCC2)=O)CC2CC3CC2C1C3NC(c1nccn2nccc12)=O C12(C(=O)NCC(CC)NC(c3cnc(C(C)OC)s3)=O)CCC(CC1)CC2 Cc1noc(CC(=O)NC(C(=O)NCCN(C2CCCC2)C)c2cccs2)n1 Cc1n[nH]c(C)c1CC(=O)NC(C1CCCCC1)CNC(C1CC2CC1C2)=O Cc1cccnc1C=CC(N1CC(CNC(=O)Cc2ccccc2)C(O)C1)=O c1(OC)cc(Cl)c(S(=O)(=O)N2CCOC(C)C2(C)C)cc1Cl C1(CC(=O)N(C(CSC)C)C)C2CCCC2N1C(=O)CCP(C)(C)=O C1(c2ccccc2)(CNC(CCCOC)=O)CCN(C(c2cnco2)=O)C1 C(=O)(CCCCCCCCCO)NC(C)(CNC(c1cc(CO)[nH]n1)=O)CO N1(C(CCN(CCOCCOC)C)=O)CC=CC(C(=O)NCC2(N(C)C)CC2)C1 N1(C(c2nccc(OC)c2OC)=O)CCC(O)(C2CCN(C(=O)C3CC3)CC2)C1 N1(C(c2scc(OC)c2)=O)CCC(CF)(NC(=O)CC(C)c2ccco2)C1 N1(C(c2ccc(C)[nH]2)=O)CC2CCC1C(NC(C1(C)CCCCC1)=O)C2 c1(CC)ccc(C(=O)NCCCCC(C)NC(c2cccs2)=O)cc1OC CC(CC(F)(F)F)C(=O)N1CCC2CC12C(=O)N(C1CC(O)C1)C C1(C(C)=O)C(C(=O)N(CC(=O)NCc2nncs2)C2CC2)C1(C)C c1(C(=O)NCC2N(C(C3(OC)CCCC3)=O)CCC2)occ(C)c1C c1(CC(N2C(CNC(=O)CCC3CCC(=O)N3)CCC2)=O)cccc2ccoc12 CCC(C)C(C)N=c1nc2sccc2c(NCc2c(F)cccc2Cl)[nH]1 Cc1ccc(C=CC(=O)NC(C2CCCC2)CNC(c2ccc(Cl)o2)=O)cc1 c1(C(=O)NC(CN(C(C(C)CN(C)C)=O)C)C)cc2c(Cl)c(F)ccc2[nH]1 C(C1(C)CCOCC1)=CC(=O)N(CCCN(C(C1(COC)COC1)=O)C)C c1(CC)ccc2c(c1)CN(C(c1ncsc1C)C(=O)NC1CCCCC1)CC2 C1(NC(c2c(C)nncc2)=O)CCSC12CN(C(c1cc(CO)[nH]n1)=O)C2 N(C(=NCC1CCOC1)N(C)Cc1ccco1)CC(COC)(C)OC N1(C(C(CC(C)C)O)=O)CC2CC(NC(c3c[nH]nc3F)=O)CC(C2)C1 C(=O)(NNC(=O)C(N)=O)OCc1cn(Cc2cccc(OC)c2)nn1 C#Cc1cccc(CC(N2CCC3(NC(c4cc[nH]c(=NC)c4)=O)CC3C2)=O)c1 C(C(F)(C(=O)NCC(C)(C1CC1)OC)C(C)C)NC(c1c(CC)cncc1)=O C(=O)(CCCCC(=O)N1CC(NC(c2c(COC)cnn2C)=O)C(C)C1)NC C(C(CC(C)C)C(=O)NCCC(O)CNC(c1ccc(O)nc1C)=O)OC Cn1cc(C(C(=O)NC2C=CCC2)NC(c2cscn2)=O)nn1 c1(N(CCC(C)(C)C)C)nccc(=NCCCCc2ccc(Cl)s2)[nH]1 c1(C(N2CC(N(C)C(c3c(F)ccc(O)c3F)=O)C2)=O)cc2c(cn1)COCC2 c1(C(N2C(C(=O)Nc3c(C(=O)OC)cnn3C)CC2)=O)ccc(COC)c(F)c1 C1(C(N2CC(CNC(c3n(CCOC)ncc3)=O)(COC)C2)=O)C(C#N)C1(C)C O=S(=O)(CCN=c1[nH]c2ccccc2c2ccccc12)Nc1cc(F)cc(F)c1 C(=O)(C#CC1(C)COC1)N1CCOCC(NC(C2(OCC)CCN(C)C2)=O)C1 C#Cc1ccc(C(N2CC(NC(c3ccc(F)c(C)n3)=O)C(C)C2)=O)cc1 C1(O)(CN(C(C(=O)NC(C)C)=O)C)CCN(C(c2cnc(N(C)C)o2)=O)C1 C1(C(=O)NC(C(C)C)CO)C(O)CCN1c1ccncn1 c1(C(N(CC(CNC(CCCCOC)=O)C)C)=O)c(N)ccc(F)c1C CCC1(C)COC(=O)CCNC1=O.C1(CSC)CCCC12CC2 Cc1cnc2c(C(=O)NC3CC(NCc4ccc(C#N)nc4)C3)cnn2c1 C(CCN(C)C(C1(CC(F)F)CC1)=O)(C(C)C)NC(CCC=CC(C)C)=O C1(C(N2CCC(NC(CC(C(C)C)O)=O)(CF)C2)=O)CC2(C1)CC1(CCC1)C2 C1(O)(C(=O)NC2CCC(c3cn(C(C)(C)C)nn3)C2)CN2CCC1CC2 c1cc(C)n(C)n1.C1(C)(C)CCNC(=S)N1.CS c1(OCC)cn(C)c(C(=O)NCC2CCN2C(c2[nH]c(C)c(C)c2C)=O)cc1=O CC#CCCC(=O)N(CC(C)CNC(=O)C(c1ccc(Br)cc1)CC)C S(=O)(=O)(c1ccc(N2CC(F)C(F)C2)nc1)N(C)Cc1cccc(F)c1F C(CC(=O)NCCCC(C)(C)OC)(C(C)(C)C)NC(C=CC)=O CC1(C)CC1(C)C(=O)NC1CCCC1NC(=O)CN1CCSCC1 c1(C(=O)NCC2CC(CNC(C3COC3)=O)OC2)cn2cccnc2n1 N1(CC)CCN(CC(=O)NCCCCNC(C2CCCC(=O)O2)=O)CC1 c1(C(C2CC2Cc2ccc(Br)o2)=O)ccccn1.N C1(S(C)(=O)=O)(C(=O)NCC(CCNC(CCC=CCC=C)=O)O)CCOCC1 C(=O)(C1CCCc2scnc21)N1CCC(O)(CCNC(CSCCC(C)C)=O)C1 c1(OCCC(C)C)ccccc1C(N1CCCC(n2cccn2)C1)=O Cc1c(C(=O)NC2CC(OCC(=O)NCC3CN4CCC3C4)C2)cccc1F c1(C(=O)NC2CC(CNC(c3c(C)[nH]cc3)=O)C2)csc(S(N)(=O)=O)c1 c1(OC)ncc(C(=O)NC2CCCN(C(=O)CCc3cc(C)[nH]n3)C2C)nc1C C1(NC(COCCC(C)C)=O)CN(C(=O)Cc2cn(C)nc2C(F)F)CC12CC2 C(C)(C(=O)N(C)C(c1ncccn1)C)(N(C(C(C)C1CC1)=O)C)C1CC1 N1(C(C2(C)C(C)OCC2)=O)Cc2[nH]nc(C(=O)NCCOC3CC3)c2C1 N12CCC(C(CO)C1)C2=O.c1(C(C)OCC)ccn(-c2ccccc2)n1 C1(N(C(CN(C(C(C)OCC=C)=O)C(C)C)=O)C)CCOC(C)C1 c1(NC(C2N(c3ncc(CC)cn3)CCOC2)=O)cnccc1[N+](=O)[O-] c1(NC(COC)C2CC2)ncc(C)cc1S(=O)(=O)NCc1ccc2c(c1)OCO2 N1(C(C(C)=CC2CC2)=O)CCN(C(c2ccn(C)n2)=O)C2CCCCC12 C1(C(=O)NC(c2ccccn2)C)(NC(c2cc[nH]n2)=O)CC1(C)C C1(O)(C(=O)NCCN(C(C(C2CCC2)OC)=O)C2CCCC2)CCOC1(C)C N1(C(c2n(CC)ccn2)=O)CCOC2CCN(C(c3cc(C#N)c[nH]3)=O)CC12 c1(CNC2CCC(NC(C3CCC(=O)NC3)=O)C2)cc(Br)cc(Cl)c1F C1(NC(c2c(C)n(C(C)C)cc2)=O)CN(C(=O)C2=NOC(C)C2)CC12CCC2 Cn1cc(C(C(=O)OC(C)(C)C)N(C2CCOCC2)CF)c2ccccc12 c1(C(=O)NC2C(CNC(C(C)OC3CCCC3)=O)CCCC2)ccc(N)c(N)n1 C(=O)(CCCCc1cccc(O)c1)N(CC(C)NC(=O)CC1CCC12CCC2)C n1(CCC(=O)NC(CC)CNC(C2CCNC(=O)C2)=O)ncc2ccccc12 N1(C(COCC)=O)CCC(C(=O)N(CC(C)C)CCO)CC1 Cn1ccn2ncc(C(N3CC(NC(=O)CSc4cccs4)CC3(C)C)=O)c12 C(CCCCC(=O)Nc1csc(C)c1)NC(C(C1CCOC1)OC)=O c1(C(N(C2CN(C(c3cc(CCCCC)[nH]n3)=O)C2)C)=O)n[nH]c2c1COCC2 c1(C(=O)NC(CNC(CC(=O)OCC)=O)CO)sc(S(N)(=O)=O)c(C)c1Cl c1(C(=O)NC2CC(CNC(C=Cc3n(CC)ncc3)=O)C2)cc2c(s1)CCSC2 c1(CC(=O)NC2CCN(C(c3ncc(C)cn3)=O)CC2O)c(C)cc(C)nc1O C1(NC(c2nn(C)nc2C(F)(F)F)=O)CC2CCC(C1F)N2C(=O)C(Cl)=CCl C(=O)(CCC(C)(C)C#N)NC(C(=O)NCC(CC=C)(F)F)COCC C1(C(=O)NCC23CC(NC(Cn4ncc(C)c4)=O)(C2)C3)CCC2CCC1O2 C1(OCC=C)CCN(C(=O)C(=O)NC2CCCCN2C)CC1.C(C(F)(F)F)O N1(C(C(C=CC)O)=O)CCC(CN2CCC2c2cn(-c3cccc(Cl)c3)nn2)CC1 Cc1cc(OCC(N2CCOC(C(C)NC(c3ccc[nH]3)=O)C2)=O)ccc1Br Nc1c(C(=O)NCC(O)CNC(=O)C=Cc2cscn2)sc2ncccc12 Cc1cc(C2CC2)ccc1C(=O)N(CCNC(C1CC1Cl)=O)C(C)C c1(C(N2CCCC(NC(C(C(C)O)NC(C)=O)=O)CC2)=O)cc(C#N)cc(C)n1 Cn1cc(C(=O)NCCCNC(=O)CC2(N(C)C)COC2)ccc1=O N1(C(C2N(C=O)CCC2)=O)CCCC2CN(C(=O)C(F)(F)c3cscn3)CC12 C(=O)(C(F)CC(C)(C)NC(=O)CN1CCNC(=O)C1)NCc1cn(C(C)C)nc1 C(=O)(CCNC(c1ccco1)=O)N(C1CCC1)CCN(C)C CC(C)C(O)C(=O)NC(C)(C)CNC(c1ccnc(OCCO)c1)=O c1(C(=O)NC2CC3(C2)CC(NC(CCNC(C)=O)=O)C3)ccc(S(C)(=O)=O)cc1C n1(CC)c(NC(=O)C(=O)NCc2ccc(N=[N+]=[N-])cc2)nc2ccccc12 C1(NC(C(C)(C)c2cnsc2)=O)CCN(C(=O)C=C(Cl)Cl)C1c1ccccc1 C1(CC)CN(C(c2csnc2Br)=O)CCC1NC(c1cn(C)ccc1=O)=O c1(OCC)cccc(NC(C2(C(=O)Nc3ccc(OC4CC4)cc3)CC2)=O)c1 CC1CC(NC(c2cc(-c3ccco3)c[nH]2)=O)CN(C(c2nc(Cl)cs2)=O)C1 C1(C(=O)NC(CCC)C2CC2)(CC)CCCN1C(=O)C=CCF CC(C(=O)N(C)C)C(C)(C)C.C12C=CCN(C1)c1ccc(cn1)C(=O)N2 CC1COc2ccc(C(N3CCCC3c3nncn3C)=O)cc21 c1(N(C(C(C2CCCN(C(=O)CCC(=O)C3CC3)C2)C)=O)C)cccc(F)c1 C(C(=O)NCc1c[nH]nc1C(=O)NC1CC(C)CCC1O)(C(C)(C)C)SC Cc1cnccc1C(C)C(=O)NC1CC2(C1)CC2NC(c1cc(CO)n(C)n1)=O C12(C(N3CCC(NC(C(C(=C)C)(C)C)=O)C(C)C3)=O)CCCC1CC(=O)CC2 Cn1c(CNCC2(C(=O)Nc3cccc(C(F)(F)F)c3)CC2)cc2ccccc12 C1(NC(=O)Cc2ccc(F)nc2)CC2CCC1N2C(=O)CC1CCOC1 C=CC1(C(=O)N(CC)OCC)CCN(C(c2cncnc2)=O)C1 c1(C(C)C)c[nH]nc1C(=O)NC1CCC(N(C(=O)CC(=O)N(C)C)C)C1 CC1C(CCC(=O)NCCCN(C(c2cc(Cl)c[nH]2)=O)C2CC2)CC(C)N1C C#CCC(C)(CC)C(=O)NC1CN(C(=O)CCCCC)CC1CO N1(C(C(C)(C)OCC)=O)CC(CNC(=O)C(F)(F)C(C)(C)O)OC2(CCC2)C1 c1(OCC)ccnc(NC(C2CCN(C(=O)CCOC3CCOCC3)C2)C)n1 C1(NC(C(CSC)(C)C)=O)CC2CCC(C1)N2C(=O)Cc1cncnc1O c1(CC(=O)NC(CC)(C)CNC(=O)C2=CCOCC2)coc2ccccc12 CC(C)(CC#N)C(=O)Nc1cccc(NC(C2CC3CCC2C3)=O)c1 c1(OCCC)ccc(NC(=O)Nc2ccc(-n3cncn3)cc2)c(C)n1 C(=O)(C#CC(=O)NC1CCOC(CNC(=O)CNC(=O)CC(F)(F)F)C1)N(C)C c1(C(N2CCN(C(C(C)OC)=O)CC2)=O)ccc2nc(O)n(C)c2c1 C(=O)(CCC(=O)NC(CC1CCC1)C(=O)N(CC(C)CC)C)NCC N1(CCC)CCCC1C(=O)NC(C)(C)C(=O)NC1CCCC1CN(C)C C1(C)(NC(c2cn(CCC)nn2)c2nnnn2Cc2ccccc2)CCC(C)C1 CCCC(CCC)CC(=O)N1CC(C)(NC(=O)C=C2CCC(C)CC2)C1 c1(C(=O)NCCC2(NC(C3C(CC)OCC3)=O)CCC2)ccc2oc(C)nc2c1 c1(C(=O)NCC2N(C(C3CC(=C)C3)=O)CC(OC)C2)nccc(Br)c1C C1(CNC(COC(C)=O)=O)CC(NC(=O)CCc2nnc(C(F)F)o2)C1(C)C N1(C(c2cncc(C3CC3)c2)C(=O)NC)CCc2[nH]nc(C(F)(F)F)c2C1 Cc1c(C(=O)NC2CC(C(=O)NCCC(F)(F)F)CC2O)ccn1C C1(CNC(C(C)(C)C2CCC2)=O)CN(C(=O)CCCn2cccn2)C2(CCC2)C1 C1(OCC)CC2(C1)CC2C(=O)NC(CN(C)C(c1ccnn1C)=O)CC CC1CN(C(c2ccnn2C)=O)C(C)CN1C(C1COCC1C(N)=O)=O c1(C(=O)NCC(C)N(C)C(C2CCCSC2)=O)conc1C1CCC1 S(=O)(=O)(c1ccccc1)NC(C)C(=O)NC1CCCN(CCCc2ccsc2)C1 c1(OCC)ccc(C)cc1NC(=O)C=CCC1(NC(C2(C)OCCO2)=O)CCC1 Nc1cc(C(=O)NCCC2(O)CN(C(C3CC3CF)=O)C2)ccc1F N1(C(C=C(C)c2cnn(C)c2)=O)CC(C)(C)OCC1CNC(c1cc(O)cs1)=O CC(O)C(C(=O)NCC=CCNC(=O)C(c1ccccc1Cl)C)N(C)C c1(C(N2CCC(C)(C(=O)Nc3nccc(C)c3Br)C2)=O)cc(C)c(CO)c(C)c1 CC(C)(C)C(O)C(=O)NCC1COCCN1C(=O)Cn1cc(F)ccc1=O C(C(C(=O)NOCCCC1CC1)C(C)(C)C)NC(C1OCCN(C)C1)=O c1(C(=O)NC2CCN(C(c3cccc(C(F)F)c3)=O)CC2)ccc(F)c(F)c1F C1(C(N(CCCN(C)C(C2(F)CCOC2)=O)C)=O)CCc2ncsc2C1 Cn1cc(Br)c(OCC(=O)NCCCNC(C2CCCC2O)=O)n1 CCC(CC(=O)N1CCCC1CNC(=O)Cc1ccc(Cl)cn1)c1ccccc1 N1(C(C2(C)CC(F)C2)=O)CC(C(=O)NCCCS(N)(=O)=O)C2(CC2)C1 c1(C(=O)NCC2(O)CN(C(C=C(C)C)=O)C2)cc2c(Br)cccc2c(=O)o1 N1(C(c2ccc(C)nc2)=O)CCCN(C(c2cnc(N(C)C)nc2)=O)CC1 c1(CC(N2CCC(C(N(OCC)C)=O)C2)=O)ccc(C#N)cc1 c1(OC)cccc2ncnc(N3CCC(CNC(c4ncccn4)=O)C34CC4)c12 c1(C(=O)NC(CNC(=O)Cc2nnc(O)s2)CO)cc(=O)cc[nH]1 C1(NC(CCSCCC)=O)CCC2(CCN(C(=O)CC(C)C)C2)C1 C1(C(N(CCCCNC(C2CCCCN2C)=O)C)=O)CC12CC(F)(F)C2 C1(OC(CC(C)C)=O)CCCCCC1.C1CC(=O)NCCN1CCO c1(C(N2CCC(C)(CNC(C(C)C3CCC3)=O)C2)=O)ccc2oncc2c1 C(CC)(CC)(CCNC(=O)C(C)(C)CC)NC(c1cccc(CC)n1)=O N1(Cc2ccc(OC)c(I)c2)CC(C(=O)NCC2CCOC2)CC(F)(F)C1 c1(NC(=O)OC)cccc(C(=O)N(C2CCC2NC(=O)C(C)C)C(C)(C)C)c1 CCCC(CCCO)C(=O)N1CCC(C)(NC(c2cccc(S(C)=O)c2)=O)C1 C(=O)(C(C(=O)N(C)CCNC(=O)Cc1cncn1C1CC1)OC)OC c1(C(N2CCCC(N(C(CC(COC)(C)C)=O)C)C2)=O)coc(S(N)(=O)=O)c1 C1(NC(C(C)CC2CCCC2)=O)C=CCC(C(=O)NCC(C)(O)CCO)C1 C(c1cnn(C)c1)=CC(=O)NC(C1(O)CN(C(=O)Cc2csc(NC=O)n2)C1)C C(=O)(CC(C)CC(C)(C)C)N1CCN(C(c2nncc(OC)c2)=O)C(C(F)F)C1 c1(OC)ccc(C(=O)NCC#CCNC(=O)CCCOc2cccc(Br)c2)nn1 c1(C(N(C2CC(NC(=O)C(O)C3CC3)C2)C)=O)cccc2c(Cl)c(Cl)sc12 C#CCC(C)(C(=O)NC1CCCC1C(N)=O)NC(C1COCCN1CC)=O c1(CNC(C(C)(C)NC(c2n(CC)ncc2)=O)=O)cccc(Cl)c1 CCCC(C)(CC)NC(=O)C(c1cnn(C)c1)NC(=O)Cn1nccn1 N#Cc1c(F)ccc(F)c1NC(C1CC(CC2CC2)C1)=O c1(C(N2CC(NC(COCCC(C)C)=O)C3(C2)CC3)=O)cn2cccc(Cl)c2n1 c1(C(N2C(CNC(C=CCC)=O)CC(C)(C)C2)=O)ccc2c(C)noc2n1 c1(NC(C(=O)NC(CC=C)=O)=O)ccc(OC(c2ccc(F)cc2)C)cc1 c1(C(C)C)nc(C(=O)NCCC2CCN(C(=O)Cc3cscn3)C2)co1 N1(C(c2c(F)ccc(F)c2Cl)=O)CC2CCCN(C(C3COC3)=O)C2C1 C1(CC)C(C(=O)NC(C)CS(C)(=O)=O)CCCN1C(c1ccc(CO)o1)=O C1(NC(c2cnc(CC)[nH]2)=O)CC2CN(C(=O)Cc3csc(Cl)c3)CC12 N1(C(c2noc(C)c2-c2nn[nH]n2)=O)CCC(c2ccccc2)CC1C(F)(F)F c1(C(N2CC(COC)OCC2)C(=O)NCC2CCCO2)cc2occc2s1 C1CCc2ccccc2C1.c1(OC)cc(NC(=O)CC2CCCN2C=O)ccc1F CCCC(CCC)=CC(=O)NCCC1(O)CN(C(=O)Cc2cnns2)C1 C12(CNC(Cn3ncn(C)c3=O)=O)CC(C1)C(NC(=O)CC1(O)CCC1)CO2 c1(C(N(CC(CNC(C2(CC=C)CCCC2)=O)C)C)=O)ccc(P(C)(C)=O)s1 c1(C(=O)Nc2ccnc(OC)n2)cc(C)c2sccc2c1 Cc1cccn(CC(N2CCOCC(NC(=O)C=Cc3cn(C)cn3)C2)=O)c1=O Cc1nc(C2CC2)nc(O)c1C(=O)NCC(C(C)C)NC(C1(C)CCCCC1)=O C1(C)(NC(C(C)SCC)=O)CC(C(N2CCC2C2CCCC2)=O)C1 C(=O)(C(C)P(C)(C)=O)OCC1(CC)CCOCC1 c1(CNC(=O)Nc2cccc(C3(OC)CC3)c2)c2c(nn1C)CCC2 Cc1cc(C(=O)NC2CCN(C(C3CC3c3ccsc3)=O)CC2O)cc(C)c1 C(=O)(CC(C)(C)C#N)N(CCC(=O)NCC12CCCCC1C2)C(C)C Cc1ccc(F)cc1Cn1nccc1-c1cccc(-c2ccco2)n1 CC1CCCCC1NC(=O)COC(=O)Cc1ccccc1 N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCC2CN(C(C3(C4CC4)CC3)=O)CCC12 Cc1ccc(F)c(C(=O)NCCOCC(=O)NCc2cc(=O)cc[nH]2)n1 N1(C(C2CC(C)C2)=O)CCC(OCC(N2CC(NC(=O)C(C)C)C2)=O)CC1 C=C(Cl)CCC(=O)NC1CC(N(C(=O)CC(C)C2CC2)C)C1 n1(CC(COC)O)cc(C#CCNC(=O)CC(C)(C)C#N)nn1 CCC(CC)(CO)C(=O)NCC(CO)NC(=O)Cn1nc(C)cc1C(F)F n1(CCC)cc(C(=O)NCC(F)CNC(c2cncc(C(C)C)c2)=O)c(C)n1 Cc1ccc(C(N2CC(NC(c3nc(Cl)sc3C)=O)C(C)C2)=O)cc1F O=C(C#CC1CCOC1)NC1CCC2CN(C(c3ccc(O)cn3)=O)CC12 C(=O)(C1CCCn2nccc21)N(C(CC)CNC(=O)C(C)Cc1cnc[nH]1)C N1(C(c2c(CNC(C=C(CC)CC)=O)cnn2C)=O)C2C=CC(C2)C1CO C1(C(=O)O)CCC2CCN(C(c3cc4ncccc4s3)C3CC3)C12 C(=O)(C(C#N)C(C)(C)C)N1CCC(C)(CC(=O)NC(c2nc(C)on2)C)C1 Cc1ccc(I)c(C(=O)NC2CCCN(C(c3ccnc(F)c3F)=O)C2)c1 c1(C(=O)NC(CC)CNC(=O)C(C)(C)C2CCCCO2)cccn2cnnc12 c1(C(N2C(C(C)NC(C(C)OCCCC)=O)CCC2)=O)ncncc1Br CC1(CNC(c2cnn(CC(F)F)c2)=O)COCCN(C(=O)C=CC(F)(F)F)C1 C1(NC(C2C(C)C2)=O)CC12CCN(C(=O)C1CC1)C2 N1(C(C=C(CC)C)=O)CC2CCN(C(=O)C=CCOC)CC2C1 Cn1ncc2c(C(N3CCC4CCN(C(C5CCN5C)=O)CC34)=O)cccc12 NC12CCCC1CN(C(=O)C(N)CCOCc1ccccc1)C2 Cc1cc(Br)c(C(N2CC(CNC(C3(C(F)F)CC3)=O)CC2C)=O)s1 C1(CC(=O)NCC(C=C)(C)C)CC(O)CN1C(c1coc(C(N)=O)c1)=O N1(C(c2cc(CC)no2)=O)CC=CCC1C(=O)NC(CC)C(C)(F)F c1(C(=O)NC(CC(C)C)(C)CNC(=O)C(C)P(C)(C)=O)ccc2c(c1)CCCC2 c1(-c2cn(CCC3CC(NC(c4c(C)nccc4)=O)C3)nn2)ccc(Cl)cc1Cl CC(CCCCNC(C1CC1(C)C(F)F)=O)NC(=O)C=CCOCC(F)(F)F C1(C(=O)NCC2CCC(CN(C(c3c(C)nns3)=O)C)CC2)CCC(C)NC1=O c1(C(N2C(CO)CC(NC(C(CC=CC)C)=O)C2)=O)ccn2c(C)cnc2c1 C1(CNC(C(CC)N(CC)CC)=O)(CNC(c2ccc(N)cn2)=O)CCCCC1 Cc1nn(C)c(Cl)c1C(N1CC2C(CNC(=O)CC3CCC(C4CC4)O3)C2C1)=O C1(CNC(C(C=C)(F)F)=O)CN(C(=O)Cc2n[nH]cc2Br)CCC1(F)F C1(NC(CC(C)(C)OC)=O)COC2CN(C(C3(C)CC4CC4C3)=O)CC12 CON(CCC(=O)N(C)CC1CCCO1)C(=O)C1(C)CCC(=O)NC1 C1(NC(Cc2c(OC)ccc(C)c2)=O)CCC2CN(C3CCCNC3=O)CC2C1 CC(C)CCCOCC(=O)NCCC(C)NC(c1ncoc1C(F)(F)F)=O Cc1cc(=NC2CCCC(NC(=O)CCc3cccnc3)C2)c(C#N)c[nH]1 C1(NC(CC=C=C)=O)CCN(C(=O)CCOc2cc(Cl)ccc2Cl)C(C)C1 C1(NC(c2cnc(C)o2)=O)CC(C)N(C(c2cnc(C3CCOCC3)nc2)=O)C1 C12(C(=O)NCC3N(C(C4C5CC6C(C5)C46)=O)CCCC3)CCCCCC1OCC2 C(=O)(C(N=[N+]=[N-])C(C)C)NC12CC(C(=O)NCCc3c(C)ccnc3)(C1)C2 N1(C(C(C(C)C)C)=O)C2CC=C(C(=O)NCc3cc(O)cc(F)c3)C1CC2 C#Cc1cnc(C(N2CCC(CC)C2CNC(=O)C(C)NC=O)=O)c(C)c1 c1(CNC(N2CCOC(Cn3cnnn3)C2)=O)cc2cc(Br)ccc2o1 C(=O)(CS(=O)(=O)CC(C)C)N1CCN(C(C(C)OCOC)=O)C(CC2CC2)C1 Cc1c(C(=O)NC2(C#N)CCN(Cc3ccc(F)c(F)c3)C2)ccc(F)c1F C(=O)(CCCS(N)(=O)=O)NC1(C)CCN(C(c2ccc(C(=O)NC)c(F)c2)=O)C1 c1(C(N2CCC(C(C)NC(C3C(C(C)C)OCC3)=O)C2)=O)cc2n(n1)CCOC2 N1(C(C(CO)N(C)C)=O)CCC(F)(F)C(CNC(=O)Cn2cc([N+](=O)[O-])cn2)C1 C(C(CC1CC1)C(=O)NCC1(F)CCOCC1)NC(C1(OC(C)=O)CC1)=O C1(C(=O)NCCCCN(C(CCOCC(C)C)=O)C)CCCC1c1cnn(C)c1 C(=O)(C(CC(C)(C)C)NC(c1cn(C(C)C)cn1)=O)NC1(C(C)O)CC1 N1(C(C(C(CC)C)=O)=O)CCN(C(=O)C2=CCCOCC2)CC(C)C1 c1(C(=O)NC2C3CN(C(CC(C)(F)F)=O)CC2C3)cnc2ccc(Cl)cn2c1=O CC1CC(NC(=O)CCN(C(C2CCOC2)=O)C2CC2)CO1.N(C)C C1(NC(CCC(=O)NC)=O)CN(C(=O)CCc2scnc2C)C(C)(C)C1 C(=O)(C(C(C)C)C(C)C)NC(CCNC(c1c(-c2cc(C)no2)ocn1)=O)C c1(N(C)C)nc(O)c2c(ncn2C)n1.N1CC(C(=O)NC2CCC2)CC1=O C(=O)(C(C)(C)CCCNC(=O)CCOCC1CC1)NC(C)Cn1cccn1 c1(CC(=O)NCC2CCCN2C(c2c(Cl)ccnc2F)=O)ncc(F)cc1F c1(C(=O)NC2CC3(CC(CNC(C(C(C)C)F)=O)C3)C2)nccc2ncccc12 c1(C(N2CC(CNC(C3C(CCC)CCC3)=O)(OC)C2)=O)c(C)cc(=O)oc1C CCC(CC(=O)NCCNC(=O)Cc1csc(CSC)n1)C(F)F C1(C(=O)NC(CNC(CS(=O)(=O)NCC)=O)CC)CCn2c(C)cnc2C1 c1(OC)ccc2[nH]cc(CC(=O)NCC(O)CNC(c3cccs3)=O)c2c1 C1(NC(c2cc(C)cc(Cl)c2)=O)CC2CC1CN(C(C1CC(C)CCO1)=O)C2 N1(C(C2C(C)C2C)=O)CCCC1(C)C(=O)N(C1CCC(F)(F)C1)C N1(C(C(=O)N(CC(CNC(C=C(C)C(C)C)=O)O)C)C)CCN(C)CC1 C(=O)(C(CCc1ccc(Cl)cc1)C(C)(C)C)c1nnc(C2C3(CC(COC)C3)C2)o1 c1(CC)ccccc1N(C(N1CCN(C2CCC(C(=O)O)C2)CC1)=O)CC Cn1ncc2c1CCC(C(=O)NC1(C)CCCN(C(C3(C4CCC4)CC3)=O)C1)C2 N(S(=O)(=O)N(C)C)CC(=O)NC(CC)CNC(C1CC1CCOC)=O C(C)(CC(=O)NCC12CC(NC(=O)CCCc3nccs3)(C1)C2)SC Cc1ncc2n1CC(C(N1CCC(N3CCN(C(=O)C(C)CF)CC3)C1)=O)CC2 c1(OC)cnc(F)c(C(=O)NC2(CCNC(c3[nH]nc(OC)c3Cl)=O)CCC2)c1 C1(C(=O)NC(C2CCCCC2)CO)CN(C(=O)C(O)CC2CCCC2)CCO1 Cc1cccc(C2CCN(N3C(COC(C)(C)C)C(N(C)C)C3)CC2)c1C.C(=O)O c1(C(=O)NCCNC(C2(C)CC(=C)C2)=O)c[nH]c2c(C)cc(F)cc2c1=O Cc1nn(C)c(C)c1NC(=O)C(C)N(C)CC1CCCN1C(=O)C(C)C(C)C C1(CC)CN(C(=O)CC2CC2CNC(C2COC(=O)N2C)=O)CCS1 c1(CC(=O)OCC)nc(C)c(N(CCCN(C)C)Cc2ccccc2)cc1C C12(NC(CC=CC)=O)CC(NC(c3cc(-c4ccccc4)sn3)=O)(C1)C2 c1(NC(=O)NCC)ccc(C)c(F)c1.C1(=O)C(CC2CCCC2)COC2CN1C2 c1(OCCOC(Cn2nc(C)c(Cl)c2)=O)nc2cc(Cl)ccc2s1 C1(C(=O)NCCCNC(C)=O)CCC(OC2CCC2)CC1.C1CNO1 c1(OC)ccccc1Cn1cc(C2CCCN2C(=O)C(Br)Br)nn1 c1(C(=O)NCC2CCN(C(C3CCCCC3)=O)CC2)ccc2c(c1)CCNC2=O C(C(CNC(=O)CN(C(=O)CN1CCCC1C)C1CC1)C(C)C)OC c1(OC)nc(C(=O)NC(C)CCNC(C2CC2C(c2ccccc2)=O)=O)ns1 Cc1cc(Br)cc(C(=O)N(CC(C)CNC(=O)CC2CCC23CCC3)C)c1C Cc1c(NC(=O)C(=O)NC2(C)CCC2)cnn1-c1ccc(Cl)cc1 C12(C(=O)NCC3C(C)CCN3C(=O)CN3CCC3C)CCC(F)(CC1)CC2 C(C)(CC(C)N=c1nc(C2CC2)[nH]s1)NC(c1c(CC)c[nH]n1)=O c1(-c2cn(CC(C3CN(C(=O)COC4CC4)C3)F)nn2)ccc(F)nc1 CCC(CC)(CC)C(=O)N(CCCC(=O)NC(c1ccco1)CO)C C(C)(C)(CCCC(=O)N1CCC(N(C)C)CC1)NC(c1c(C)cc(CC)o1)=O c1(NC(c2cc(OC)ns2)C)cc(N2CCOCC2)nc(C)n1 N1(C(c2c(C)nsc2)=O)CCC(C2CCN(C(c3cc(N)ccc3Cl)=O)CC2)C1 c1(C(=O)NCC2CN(C(C(C)(C(C)C)NC(C)=O)=O)CC2C)cc(C)nc(C)c1O C(=O)(C(C)C(O)C(C)C)NC(c1ccc(CNC(C2(C(=O)NC)CC2)=O)cc1)C C(=O)(C(C(C)(C)C)OC)NCC(=C)CCNC(C1(N2CCCC2)CCC1)=O c1(C(N)=O)cncc(NC(C2(C)CC(NC(c3cccnc3O)=O)C2)=O)c1 N1(C(=O)NC(Cc2ccc(F)cc2)C2CC2)CCSc2ccc(C(=O)O)cc21 C1(NC(=O)CNC(C2CCCCC2)=O)CC(O)CN(C(c2ccccc2Cl)=O)C1 N1(C(C2C(C(=O)OC)CC2)=O)C2CCCC1CN(C(=O)C(C)(C)C(C)(F)F)CC2 N1(CC)CCC1C(=O)N(C1CCCC1)CCNC(=O)C(C)NC(c1ccco1)=O C(C(=O)NC1C2CC3C1C3C2C(=O)NC1CC(CN(C)C)C1)(C(C)(C)C)SC Cc1nscc1CC(=O)NCCOCC(=O)NCCCC1CCCC1 C1(C(N2CCC(OCCNC(CCCC)=O)C2)=O)CCC(=O)CC1(C)C N1(CC)CCC2OCCN(C(=O)Nc3cc(Cl)cc(C)c3C)C2C1 c1(C(=O)NCC=CCNC(C(C)OCC)=O)c(C)cc(OC)cc1F c1(C(N2CC(n3cc(C(C)OCC)nn3)C2)=O)ccc(C(=O)N(C)C)cc1 N1(C(C(COCC)C)=O)CCC2(C)CN(C(=O)C=CC(C)C)CC12 c1(C(N2C(C)(C)C(CNC(=O)CC3CC=CCC3)CC2)=O)ccc2cnoc2c1 c1(CSC)cc(C(=O)NCCC2CN(C(=O)C=CC(C)C)CCCO2)ccc1F N1(C(c2c(C)nn(C)c2)=O)CC2CC(N=c3nc(-c4ccccc4)[nH]s3)C2C1 Cc1cnc[nH]c1=NCC1CCCC(NC(=O)CN(C)CCO)C1 C12CCN(C(C)C1)C2=O.C1(NC(CC=CC=C)=O)CC2CC3C(C2)C13 CN1CCCC1(C)C(N1CCCC1C(C)(C)CNC(c1ncc(Br)cn1)=O)=O C12(CNC(CNC(=O)OC)=O)CCC1CN(C(=O)CCCN1CCCCC1)C2 c1(OC)cccc2ccc(C(N3CCC3CF)=O)nc12 Cc1cccc(CC(=O)NCC(O)CCNC(=O)CN(C2CCCC2O)C)c1 c1(CNC(=O)CC2CC3CNC2C3)ccc2c(c1)CCC2 c1(C(C)C(=O)NCC2CCCN(c3cc(O)ncn3)CC2)cccc([N+](=O)[O-])c1 C1(NC(c2c(COC)noc2)=O)CCN(CCNC(C2CC(C)(C)C2)=O)CC1 CCC(CNC(c1sc(C)cc1Cl)=O)N=c1[nH]c2ccc(OC)nc2s1 N1(C(CC=CC=C)=O)CCOC2(CCN(C(C3CCCC4CCCN34)=O)C2)C1 n1(CCC)ccc(C(=O)NC2CCC(NC(c3cc(Br)no3)=O)C2)n1 CC(C)CC(C)CC(=O)NC1CCCC1C(=O)NCC(O)CC1CCCC1 N1(C(C2(O)CCCC(C)CC2)=O)CC2(CCC(NC(C3CSCCS3)=O)CC2)C1 c1(C(CNC(=O)NCC(=O)Nc2cccc(C)c2)C)ccc(F)c(Br)c1 c1(CN2C(C(=O)NCCOCCOC)CCC2C)cc(Br)cc(F)c1F N(C1CCOc2cc(Cl)ccc21)C(CCCOC)C(=O)OC C1(CN(C)C(C2C(CC)C2)=O)CCCN1C(=O)C=CCOCCOC Cc1nc2ccc(C(=O)NCCOC3CCN(C(=O)CCCF)C3)cc2[nH]1 c1(C(=O)NC2CN(C(C3(CCN4CCCCC4)CC3)=O)C2)cccc(F)c1 c1(C(N2C(C(=O)NC3CC(C)OC3=O)CCC2)=O)cc2ccccc2o1 C1(C(=O)NCC2C(NC(C(C=C)(C)C)=O)COC2)CCOCC1(C)C CC#CCCCC(=O)NC(C1CCN(C(c2ccccc2C2(C)CC2)=O)CC1)C c1(C(=O)Nc2n(C(CC)C)ncc2)coc2cccc(F)c12 CC(C)(C)CC(O)C(=O)NCC1CC(F)CN1C(c1ccc(OC(F)F)cn1)=O c1(C(N(CC(C)NC(=O)C(C)OC2CCCCC2)C)=O)ncc(Cl)cc1Cl c1(CN(C(C2C(OC)(OC)CC2)=O)C2CC2)ccc2c(c1)CC2 c1(SCCC(=O)NC2CC2NC(=O)Cn2cccn2)nc2ccccc2s1 C1(C(=O)O)(OC)CCN(C(C)C(N)=O)CC1.n12cnc(C)c1CNC(=O)C2 N12CCOC(C1)OCCC2=O.C(C)(C(=O)N1CC(N(C)C)C1)OCCOC Cn1cnnc1SCC(=O)NCC1(C(C)(C)O)CN(C(C2(n3cncn3)CC2)=O)C1 N1(C(C=C2CCC(C)C2)=O)C2CCC1CN(C(=O)CNS(=O)(=O)C1CC1)C2 C(C(=O)N(C)Cc1ccccc1)(C(=O)O)NC(C1CCC1)C c1(-c2occ(C(=O)NC3CCCN(C(C4(F)CC4)=O)C3)n2)ccc([N+](=O)[O-])cc1 c1(C(N2C3CCC(NC(CCCSC)=O)C(C3)C2)=O)nc2cncnc2[nH]c1=O N1(C(c2cccc(OCC)c2)=O)CCN(C(C2(F)CC2)=O)C2CCCCC12 N1(C(C2(C)CCOC2)=O)C(C(N2CCC(O)C(C)(O)C2)=O)C2CC(O)C1C2 C1(CC(=O)NCC=CCNC(c2nccs2)=O)CCC(O)CC1 N1(C(c2nccc(C)c2)=O)CC(C(N2CCCC2C(F)(F)F)=O)CC(F)(F)C1 N1(CCCNC(=O)CSC(F)(F)F)CCN(C(C23CCCCC2C3)=O)CC1 C(=O)(C(C)CC(F)F)NC1C(OC)CN(C(=O)CCc2ccncn2)C1 N1(C(=O)Cn2cnnc2)CCCC(N=c2[nH]nc(C3CC3)o2)CC1 c1(C(=O)NCCCNC(c2c(CC)onc2)=O)ccc(=O)n(-c2cnn(C)c2)c1 N1(Cc2ccc(OC)cc2Br)CCN(C(C2CCCCC2)=O)C2(CC2)C1 C1(C(N2CC(N3C(=O)CC(NC(C(C)C4CC4)=O)C3)C2)=O)CN(C)CCN(C)C1 C1(C)(NCCC(=O)N(CCC(=O)OC)CCCOC)CCCC1(C)C c1(NC2CCOC2=O)ccc(OCC(N2CC(CNCC)C2)=O)cc1 c1(OCC)ccccc1C=CC(=O)NC1CC2CC1N(C(C13CC(C)C1C3)=O)C2 c1(C(=O)NCC(CC)NC(=O)C(F)C2CCC2)cc(COC)[nH]n1 C=C1CC2CCC(C1)N2C(=O)C(CNC(c1oc(C)cc1C)=O)CCC c1(C(C(=O)NC2CCOCC2)N(CC)CC2CCC2)cccc(C2CC2)c1F N1(C(COCCOCC)=O)CCC(C2CN(C(C3CCOC3(C)CC)=O)C2)CC1 CCCCS(=O)(=O)CC(=O)NCC1CC2CCC(C1)N2C(=O)C=CC1CCCO1 Cc1ccc(CN2CC(C)(NC(C3CCCN3C)=O)C2)cn1.c1(C)ccco1 c1(C(=O)NCCCCN(C)C)ccc2c(n1)CCC(C)(C)C2 C#CC(C(C)(C)C)NC(=O)C(COCC)NC(=O)CC1CCC(C)(C)C1 C1(C(=O)NCC2CCCC2OC)(NC(CSCC)=O)CCC(C)(C)CC1 N1(C(c2cc(C)c(C)o2)=O)CCC(NC(c2cnc(Cl)c(N)c2)=O)C(CO)C1 C(=O)(CS(=O)(=O)Cc1cccs1)N1CCC(CC=C)(NC(c2cnn(C)n2)=O)C1 C(=O)(CC(C)C(F)(F)F)NC1CCCN(C(c2n(C=C)ncc2)=O)CC1 c1(NC(C2CC(CC(=O)N(C(C#C)C3CCC3)C)C2)=O)ccc([N+](=O)[O-])o1 CC1=C(C(=O)N2CCN(C(c3ccc(N)cc3F)=O)CC2C(C)C)SCCO1 c1(CN2C(CC(=O)OCC)C(=O)NCC2)ccc(F)cc1C#N c1(C(C)NC(=O)C(CN(C)C)NC(=O)COCCCN(C)C)ncn(C)n1 c1(CC(=O)NCC(C2CC2)NC(CCc2cc(C)on2)=O)ccc2nsnc2c1 C12(NC(C(CO)OC)=O)CCC(n3cc(-c4cccc(F)c4)nn3)(CC1)C2 c1(C(N2CC(C3(NC(c4ccc(C)cn4)=O)CC3)C2)=O)cc(Cl)cc2c1OCC2 c1(C(N(C2CCN(C(C3CC(F)C3)=O)C2)CC)=O)cccc(C(N)=O)c1 Cc1c(C(=O)NCCCCCCNC(=O)C(C)(C)CF)cc(C(F)(F)F)cc1N N1(C(c2ccc(OC)cc2F)=O)CCCC2(CCCN2C(c2cc(C)ns2)=O)C1 CCC(C)CC(C)C(=O)NCC1CC2(CO1)CN(C(=O)COC1CCCOC1)C2 N1(C(C(c2ccccc2)C)=O)CCC2(CC1)CN(C(=O)CC(C)F)CC2CO N1(C(C)=O)CCCC2C(NC(C34CC(C#N)(C3)C4)=O)C(C)(C)C12.C(CN=[N+]=[N-])C1CC1 c1(C(=O)NCC2CCN(C(c3cc(C)[nH]n3)=O)C2)cc2c(C)c(Cl)ccc2[nH]1 C1(C(=O)NCCC(C(=O)OC)C)CCCCCN1C(=O)CC1C=NN(C)C1=O N1(C(C(CN(C)C)NC(C2CCCOC2)=O)=O)CC2CCCC(O)C2C1 C(=O)(N=c1cc(C)n(C2CCC2)[nH]1)c1c(C)cccn1.c12occc1CNC2=O C1(C(N2CCC(C)(NC(=O)CCn3cncn3)C2)=O)CC(C2CCC2)C1 N1(C(C(c2ccc(Cl)cc2)C)=O)CC2CC2(CNC(=O)Cn2ncnn2)C1 Cc1ccc(O)c(C(=O)NC2CC(NC(c3cnc(C(N)=O)s3)=O)C2)c1 N1(C(C2CC(CCC)OCC2)=O)CC2(CC(CNC(=O)Cc3ccoc3C)C2)C1 CCC(CCN=C(NCCF)NCC1CCCC(N2CCCC2)C1)SC c1(C(N(C2CC(NC(C3N(CC)CCOC3)=O)C2)C)=O)ccnc2c1ccn2C C(=O)(CP(=O)(C(C)C)C(C)C)NC1C(C)(Cc2cccc(C)n2)CCC1 CCC(CO)(C(=O)NCC1COCCN(C(c2cc(CCO)on2)=O)C1)OC C(=O)(C1CCCc2nn[nH]c21)N1CC(CCNC(C(C(CC)C)OC)=O)(OC)C1 N1(C(=O)NCC2CCN(CCCC)CC2)CCn2cccc2C1C(=O)OC c1(CC(=O)NC(C)C=CC(=O)N(C)Cc2ccccn2)cnnn1C c1(C(=O)NC2CC(NC(C3CC(=O)NC3)=O)C2)cccc(-c2ccc(O)nn2)c1 C(=O)(C(O)CN1CCOCC1)NC1CN(C(C2C(C)C2C)=O)C1 C1(S(C)(=O)=O)(C(C2CCC(N(C)C(c3ccccc3)=O)CC2)=O)CNC1 c1(C(=O)NC(C)CCN(C)C(c2cc(CO)[nH]n2)=O)cc(C2CC2)ccc1Cl c1(CNC2(c3n(Cc4nnn(C)n4)nnn3)CCC2C(F)F)ccc(Cl)c(Br)c1 c1(C(=O)NCc2c(C(N(C(CSC)C)C)=O)occ2)cc(N)cc(F)c1 C1(C2CCN(C(C3CN(C)CC3C)=O)CC2)(NC(CCC(=C)Cl)=O)CCC1 C1(C(=O)NCCOCCCN(C(c2cnc(C)[nH]2)=O)C)CC2(CCC2)CO1 C(=O)(C(CNC(=O)CC(C)SC)CCC)NC1(C=C)CCC1 C(=O)(CC(C)(C)C=C)N1CCC(CC=C)(C(=O)N(CCCC(=O)NC)C)C1 N1(C(C(C)OCCOCC)=O)CCCCC(N(C(=O)C2=COCC2)C)C1 C(=O)(C(C)S(N)(=O)=O)NC(C1CCN(C(C2CC(N3CCCC3)C2)=O)CC1)C Cc1ccc(S(=O)(=O)CCC(=O)N2CCC(C)(NC(=O)Cc3cncs3)C2)cc1 c1(OC)cc(Cl)ccc1C(N1CCCCC(NC(=O)CC(=O)OC(C)(C)C)C1)=O C1(NC(CC(C)c2ccco2)=O)(CO)CCCN(c2ccc(C#N)nc2)C1 c1(NC(C2N(CC(C=C=C)C)CSC2)=O)cc(F)ccc1O CCC(C(=O)NC(C(=O)NC(C)CC(F)(F)F)c1cccs1)C(C)(C)CC CCC(C)(C)C(C)CC(=O)NCC(c1cccc(Cl)c1)NC(c1ccsc1C)=O C(=O)(CS(=O)(=O)C1CCCC1)NCC(CNC(C(c1n(C)ccc1)=O)=O)(C)O c1(C(C)NC(=O)C(=O)NC2CC(n3ccnn3)C2)ccc(Br)cc1 C12(CNC(C(c3cccc(O)c3)C)=O)CC(CN1C(=O)Cc1ccc(O)nc1)C2 N1(C(C2CC23CCC3)C(=O)NCC=C)CCCC(O)(C2CC2)C1 C1(C(N2CC(F)(CNC(c3c(C)cncc3)=O)C2)=O)CCc2ccccc2C1 C12(NC(CN(C3CCC3)C)=O)CCCN(C(c3cc(F)c(N)cc3F)=O)CC1C2 c1(OCC)nc(C)ccc1C(N1CCC12CN(C(c1ccsc1C#N)=O)C2)=O C1(C)(NC(C2(COCC)CC2)=O)CCCN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 c1(C(C)C)cc(C(=O)Nc2nc(C(=O)NCc3cnccn3)cs2)n[nH]1 c1(-c2scc(C(N3CCCC(OCC4CCOCC4)C3)C)n2)cccc(C#N)c1 c1(C(=O)OC)cc(C(=O)NCC2(NC(c3ccoc3Cl)=O)CCC2)[nH]n1 n1(CC(N2CCC(CCNC(C(CC)NC(C)=O)=O)C2)=O)c(C)cc(O)cc1=O C1(C(=O)NCC=C2CCN(C(=O)CCc3ccsc3Cl)CC2)CC2C=CC1CC2 C1(NC(N2CC(C(=O)OC(C)(C)C)C(F)CC2)=O)CCCC2(CCOC2)O1 c1(C(=O)NCC2(CN(C(C=C(C)C)=O)C)CC2)c(C(C)C)n[nH]c1C C1(CC(=O)NC2C(C)(C(F)F)C2)CCCCC1NC(=O)C(O)CN(C)C N1(C(CN(C)CC)=O)CC2CCCC2(NC(c2cc(SC)c(C)o2)=O)C1 c1(NC(=O)NC2C3(CC3)C23CC3)cc(Cl)nc(C2CCOCC2)n1 c1(C2C(C(=O)NCc3ccc(C(F)F)nc3)C2)ccc(F)cc1Cl CC1(NC(=O)CNc2ccccc2)CCN(C(C23CSC(C2)C3)=O)CC1 n1(CCN(CCCC)C)c(N2CCC3CC3C2)nnc1-c1ccccc1 c1(OC)ccccc1OCC(=O)NC1CC(NC(C2CC(SC)C2)=O)C1 C1(NC(=O)Cn2ncnn2)CC(F)CN(C(C2CCOC2c2ccncc2)=O)C1 c1(C(N(CCCOCCN(C(=O)C(C)(C)CC2CC2)C)C)=O)cc(Cl)nnc1O CC1(C(=O)NCC(O)CNC(C2(c3c(Cl)cccc3Cl)CC2)=O)CCCC1(F)F N1(CC)CCCC(C(=O)NC2CC(NC(=O)Cc3ccc(C)cc3)C2)C1 Cc1c(Cl)cnn1CC(=O)NC1CC(F)(CNC(=O)CCOC2CCCCC2)C1 c1(CNC(=NC)NCC(O)(COC)COC)c(N2CCCC2)ncnc1Cl c1(C(N(C2CCC(NC(=O)CCC(C)(C)C)CC2)C)=O)ccc2nccn2c1 N1(C(CS(CCC)(=O)=O)=O)CC2CN(C(C34CC3CNC4=O)=O)CC(C1)O2 c1(C(=O)NCCCC(C)NC(=O)Cc2cc(Cl)cs2)nc[nH]c2nccc1-2 c1(OC)cc(C(N2CCOC(C(C)NC(c3cc[nH]c3)=O)C2)=O)cc(F)n1 C12(C(N(C3CCCCC3)CCNC(C=CS(C)=O)=O)=O)CCC(CF)(CC1)CC2 CC(C)(CNC(C1CCC12CCC2)=O)CCNC(=O)COc1ccccc1 N1(C(C(CC)n2cncn2)=O)C(C(=O)NCCn2cnnc2C)CCC1C1CC1 C1(C(C)=O)CC(C(=O)NCCCCn2cc(-c3cnn(C)c3)nn2)C1(C)C c1(OC)ccnc(C(=O)NC2CCCC(NC(=O)C=C3CCC3)C2)c1N C1(C(N2CCC(C)(CNC(c3ccoc3)=O)C2)=O)CC2(C1)OCCO2 N1(C(CCOCC#C)=O)CCN(C(c2cc(C)nn2CC)=O)CC1CC(F)(F)F C1(N(C(CCOCCOCC)=O)C)CN(C(c2ccnnc2)=O)CC1F C1(C(=O)OC)CCN(C(=O)C(CNC(C2(C(N)=O)CC2)=O)CC2CC2)C1C c1(C(=O)NC23C(CN(C(c4n(CC)nnc4C)=O)C2)C3)c(F)c(N)cc(Cl)c1F C1(C(N2C(C)CCSCC2)=O)C2CC(O)C(C2)N1C(=O)CCCF c1(CSC(C)C(=O)NCCN(C(c2ccc[nH]2)=O)C2CC2)ccccn1 C(=O)(C1=CC2(CCOC2)C1)NCC=CCC(=O)NCc1n[nH]c2c1CCC2 C1(CNC(c2scc(C)c2Cl)=O)CC2(CCC2)CN1C(c1ccn(CC#N)n1)=O c1(CC(=O)N(C(CN(C)C(C2CCCO2)=O)(C)C)C2CC2)cc2cc(Cl)ccc2[nH]1 C1(C2CCCNC2)(NC(C(C)(O)c2cccnc2)=O)CC1 Cc1cc(C#N)cc(C(=O)NCC(O)CNC(c2nc(C(F)(F)F)cs2)=O)n1 N1(C(c2csc(Cl)c2)=O)CCN(C(C23CC(CC(F)(F)F)(C2)C3)=O)CC1 c1(C(=O)NCCNC(c2cc(C(N)=O)[nH]c2)=O)ncnc2cc[nH]c12 O=C1CC(CC(=O)NC2(C(F)(F)F)CC3(CCC3)C2)c2ccccc2N1 N1(C(C(C=C)OC)=O)CC2CN(C(=O)C=CSC)CCC12 C=CCC(Cc1ccccc1)C(=O)NCC(C)CN(C)C(c1cccc(C)n1)=O N1(C(c2[nH]c3nc(C)sc3c2)=O)CCN(C(c2cnc(O)n2C)=O)C2(CCC2)C1 C1(NC(c2c(Cl)csc2Cl)=O)CCCN(C(c2cnoc2)=O)CC1 C1(NC(=O)COC(F)(F)F)CN(C(=O)CC2CCCCC2O)CC1CC1CC1 c1(C(=O)NC(C)(CNC(C2(C(=O)CCl)CC2)=O)C2CC2)nc(=O)o[nH]1 C1(NC(CSCCNC(C(C)C2(O)CCC2)=O)=O)CCCC(O)C1O CC1OCCC1(C)NC(C1OCCC1CNC(=O)CC1CC2CCC1C2)=O CCC(CCC(=O)Nc1cccc(Cl)c1)NC(c1cc(C#N)cs1)=O C=CC(C)C(C)C(=O)NCC1(O)CCN(C(c2cn(C)nc2Br)=O)CC1 CC(C(F)F)=CC(N1CC(CNC(=O)CNC(C2CC2C)=O)C1)=O N1(c2n(CC3(F)CCC3)nnn2)CCOCC2(C1)CC2(F)F N1(C(c2ccn(C)c(=O)c2)=O)CCc2sc(C(N3CCCC(O)C3C)=O)cc2C1 CCC(CCOC)C(=O)N1CCCCC1CNC(=O)CC1CC=CCC1 c1(CC(=O)NCC(=O)Nc2cccc(C(F)(F)F)n2)cc(F)ccc1F c1(CN(C(C2C(C(=O)NCC#C)C2)=O)CC)ccc(Br)c(Cl)c1 CC(C)C(C)(O)C(=O)NCC1CCN(C(C2CCC(=O)N2C)=O)CC1O C1(C)(OC)CCN(c2ncnc(N3CCC(C(C)(C)C)C3)c2C)CC1 CCC(C)(C(=O)N1CCC(C2CCCN2C(c2cncnc2C)=O)C1)OC C(=O)(C1CCc2nccn21)NCC1CN(C(c2ccc(=NC)[nH]c2)=O)CC12CC2 C(=O)(CCCCCC(C)C)NC1C(OC)CN(C)C1.C(=O)C(C(C)OC)N c1(NC(CC)CC(F)(F)F)[nH]c(=NC2CCCN(C)CC2)nc2c1ncn2CC CCC(C)(C)C(C)CC(=O)N(CC1CCCCC1)CC1CC(=O)N(C(C)(C)C)C1 C1(NC(c2ncncc2Cl)=O)(CO)CCCN(C(c2ccc(F)o2)=O)C1 c1(OCCOC)ccc(C(=O)NC2(C)CC(NC(=O)CC3C=CCC3)C2)cn1 N1(C(c2c(CC)[nH]nc2Cl)=O)CCCC(C)(NC(c2cccc(C(F)F)c2)=O)C1 N1(C(C)=O)CC2CC2(C(=O)N(CCCCN(C)C(C2CCN2C)=O)C)C1 CC1(C)CC(NC(C2CCCO2)=O)CN(C(=O)Cc2csc3nccn23)C1 C(C(C(C)C(C)C)NC(c1cnn(C(F)F)c1)=O)NC(c1ccc(C(C)=O)[nH]1)=O N1(C(C(C)(F)F)=O)C2CCC(C2)C1C(=O)NOC1CCCC1 N1(C(C(C(C)NC(c2cc(O)n(C)n2)=O)(C)C)=O)CCc2n[nH]cc2C1 N1(C(c2cc(C(C)C)on2)=O)CC(NC(=O)CNc2ccccc2Cl)CC(F)C1 CCC(CN(C)C)CC(=O)NCC1(F)CC(CNC(C2C3CC4C(C3=O)C24)=O)C1 c1(C(N2C(CNC(c3c(C)ccnc3)=O)COCC2)=O)cnc2ncccc2c1 N1(C(C(C)C(C)O)=O)CCCC(O)(CN(C(=O)CCn2ccnc2)C)C1 c1(NC(C2CC2C(=O)NC(c2ccc(Cl)cc2)CO)=O)cnn2cccnc12 C1(C2CC2)(CNC(C(CC)F)=O)CCN(C(=O)CC(=O)NC)C1 N1(C(C2C(C)(C(F)F)C2)=O)CCCCCC1CNC(=O)Cc1ccccc1 c1(OCC)ccc(CC(N2CCC(CNC(=O)C(C(C)C)SC)(OC)C2)=O)cn1 CC1Cc2cccc(-c3cccn3Cc3ccco3)c2C(=O)O1 C(=O)(C(C(C)(C)C)OC)N1CCC(CC)C1CNC(c1cc(C)oc1C)=O c12ccc(O)c(c1)C2.C1(OC(C)(C)C)CCNC1C(=O)ON c1(C(N(C2CN(C(c3nc(C)nn3C)=O)CC2O)C)=O)nn(C)c2ccccc12 N1(C(c2[nH]c(C)c(C(C)=O)c2C)=O)CC2(CCCC2NC(=O)CCCN(C)C)C1 N1(C(C2C(CCC)CN(C(=O)CCc3cccs3)C2)=O)CCCC(CCO)CC1 Cc1c[nH]cc1C(=O)NCC=CCNC(C1COC(C)C1)=O Cc1c(N(C(=O)C(O)CNC(C2(F)CCOC2)=O)C)cccc1F C1(NC(C2(O)CC(C)(C)C2)=O)CCCCCN(C(=O)CN2CCP(C)(=O)CC2)C1 N1(C(C=C(C)Cl)=O)CC2CCN(C(c3nsc4ccccc34)=O)C2C1 c1(C(=O)Nc2cc(Br)ccc2I)cc2ccc(-c3cc(O)c(F)c(F)c3)nc2[nH]1 C1(CN(C(CC#N)c2ccccc2)C2CC2)CC(O)CN1C(=O)OC(C)(C)C C1(C(N2CC(NC(C(C)(C)CF)=O)C2)=O)CCn2c(cnc2-c2ccccc2)C1 c1(C(N2C(CN(C)C(C3C(C(F)F)C3(C)C)=O)CCCC2)=O)cc(=O)n(C)cn1 Cc1cccnc1-n1cc(C2C(C)CCN2C(C2(CC(C)C)CCC2)=O)nn1 CC(CC=Cc1ccccc1)C(=O)NCCN(C)C(c1nsnc1O)=O c1(SC(C)C(=O)N(C)CCN(C)C(c2ccns2)=O)nnnn1C1CC1 C12(CCC(=O)NCC(CO)NC(c3c(C)ncs3)=O)CCC(CC1)C2 c1(-c2c(OC)c(F)ccc2F)ccc2ccnc(NC(=O)C3=C(C)OCC3)c2c1 C1(CC(=O)NC2CC2C2CCC2)CCN(C(C2(F)CCOC2)=O)CC1 c1(C(=O)NCC2CC(CC(=O)OC)C2)cc(SC(c2cccs2)=O)nn1C c1(C(C)C)nc(C(C2CC2)C2CC2)no1.C1(C(=O)OC(C)(C)C)N(C=O)CC12CC2 c1(C(=O)NC2CC3(CN(C(C(C)NS(C)(=O)=O)=O)C3)C2)cc2c(nn1)CCOC2 N1(C(C2OCCN(CC)C2)=O)CC2CC1CN2C(=O)CC=C(C)C Cc1nc2ccnn2c(NCc2ccccc2Oc2ccc(F)cc2)c1C CC1(CNC(c2occc2-c2ccccc2)=O)CCN(C(C2(F)CC2(C)C)=O)C1 N1(C(c2cc(C)[nH]c2C)=O)CC2CCCC1CN(C(C1CCCCC1)=O)C2 C(C(C)(O)CNC(=O)C(C)C1CC1)NC(C(C)OCCN(C)C)=O O=S(=O)(c1ccc(NCCOC2CC2)cc1Cl)NC1CCn2ccnc2C1 c1(C(C)NC(c2ccc(-c3cc[nH]c3)cc2)=O)nnc2ccccn12 Cc1nc[nH]c1CC(=O)NCC(O)CN(C)C(c1cc(CCCO)on1)=O C(CC(C)C(F)(F)F)NC(C(CCOC)NC(c1ncc(CC)cn1)=O)=O c1(C(=O)NCCCCCNC(c2c(C)cnnc2)=O)cncc2cnccc12 C1(CC=C)(NC(c2nocc2Cl)=O)CCN(C(=O)C(C)=CCO)C1 C12COc3cc(nn3C1)C(=O)N2C.c1(C(=O)OC(C)(C)C)cccc(S(C)=O)c1 C(CN=C(NCC1(OC)CCC(C)(C)C1)NC1CCN(c2ccccc2)C1)OCC C1(CC(=O)NC(CNC(C2CC(CCC)C2)=O)(C)CC)(OCCC)CCCCC1 CC(C)CC(CNC(=O)CC1(O)CCCCC1)C(=O)NCC1CC1C C1(C(N2C(C)CC(NC(c3cnns3)=O)C2)=O)Cc2ccccc2CO1 c1(C(=O)NC2CCC(NC(c3cn(C)nc3)=O)CC2)ccc2cccnc2c1O C1(C2N(C(Cc3c(C)con3)=O)CCC2)CCN(C(C2(C)CCCCO2)=O)CC1 C1(n2cc(C(CC)(C)O)nn2)CCCCC1CNC(=O)CCC1CCC(=O)C1 N1(C(COC2(C)CCC2)=O)CC(C)(C)OCC1CNC(=O)CN1CC(=O)NC1=O c1(C(=O)NC2CC3(C(NC(C(CCC)OC)=O)C3)C2)cc2c(Cl)ccnc2s1 CN1CCCN(C)C1=NCC12CC(CN1)C2.c1(C)ccccc1 N1(C(c2c(C)n(C)cc2)=O)CCN(C(C2CCCSC2)=O)C(C)C1 c1(OC)cccc(C(CF)NC(=O)CSCCNC(=O)NC)c1 N(C(=NCCCCCCC(C)C)NC1CCCCC1)C1CC(OCC(=O)OC)C1 Cc1scnc1C(=O)NC1CCC(CCNC(=O)Cc2cc(Cl)cs2)C1 Cc1nc2c(C#N)cnn2c(C)c1CCC(=O)NCCCN(CC(C)(C)O)C1CC1 C12(CC(N3CC(N4CCN(C(CN5CC(C)C5)=O)CC4)C3)=O)CCCN1CCC2 c1(NC(CC2CN(C(c3n(CC)ccc3)=O)CC2C)=O)ccc2occc2c1 c1(OCC(=O)N(CC(C)NC(c2c(C(C)C)cco2)=O)CCO)ccc(Cl)c(F)c1 C1(CNC(C(C=C)(F)F)=O)CN(C(=O)CC2CCCC3(CC3)C2)CCCO1 C#Cc1ccc(C(=O)NCC(O)CN(C(=O)CCc2nnc(S)n2C)C)o1 N1(C(c2c(CC)cno2)=O)CC(NC(c2cc(F)n(C)n2)=O)CC1(CC)CC C(C(=O)NC1CC(CNC(c2ccc(C)cc2)=O)CC1O)(C(C)C)OC c1(C(N(C2CCN(C(C3C(c4ccc(C)cc4)C3)=O)C2)C)=O)nc(C)ccc1F CC(C)CC(C)C(C(=O)NC(C)C)N1CCCCC1CN1CCOCC1 CCC(C(c1nn[nH]n1)N(c1ccc(C(N)=O)cc1)C)C(C)C c1(C(=O)NC(C(C)C)CNC(C23CC=CC(C2)OC3)=O)cc2nccn2c(O)n1 c1(OCCOC)ccc(C(=O)NCC(C2CCCC2)NC(C2CC2(F)F)=O)cc1 Cc1nncn1NC(=O)C1CCCN1C(=O)CC1(C)CC1 CC1CN(C(c2nccs2)=O)CCC1NC(=O)C(F)=C1CCCC1 c1(C(N2C(C(=O)NC3CN(C(N(C)C)=O)C3)CC2)=O)ncccn1 C#CCC(C)(C(=O)NCC1CCCO1)NC(c1nnn(C)c1CC)=O c1(C(N(C2CCN(C(c3c(CC)non3)=O)C2)C)=O)cc(F)cc2c1CCC2 Cc1ccc(F)c(S(=O)(=O)N2CCc3[nH]nc(C(N4CCCC4CO)=O)c3C2)c1 CC1CCc2nc(C(N3CCC3CNC(=O)CN3CCCC3C)=O)cn2C1 c1(C(=O)NCCN(C(=O)C=Cc2cnn(-c3ccccc3)c2)C)nc(=N)cc[nH]1 C(=O)(C1=CCC2CCC1N2C(C1CCCSC1)=O)NCCC1=CCN(C)CC1 CC(C(=O)NCC1CN(C(C2(F)CC3(CCC3)C2)=O)CCCO1)S(N)(=O)=O CC1=CCN(C(c2cccnc2CNC(=O)CSc2cn[nH]c2)=O)CC1 N1(C(C(C)NC(N)=O)=O)CCN(CC(C)NC(c2ccc(CO)o2)=O)CC1 C1(CNC(c2cccc(C)c2)=O)CC(C)(C)CCC1NC(c1nc(C)c(C)s1)=O CC1(C)C(CNC(=O)C=CC2CCCO2)CCN1C(c1csc2nnsc12)=O c1(C(=O)NC(C)CN(C)C(C2(F)C3CCCC23)=O)ccc(Cl)c2ccccc12 S(=O)(=O)(c1ccc(O)c(-c2nn[nH]n2)c1)N1C(C)CC(O)C1 N1(C(CCSCCSC)=O)CCN(CCN(C(=O)Cc2ccn(C(F)F)n2)C)CC1 CC(C)CCC(=O)NCC(=O)NCC(C)(O)CNC(=O)C=Cc1cocn1 c1(C(=O)NCC(CC)NC(=O)CN2CCCCC2)cn(C2COC2)nn1 N1(C(C(C=CC)O)=O)CC(C)C(C)(CNC(c2cnn(-c3ccccc3)n2)=O)C1 C(=O)(C1SCCc2ccccc21)NC(C)(C)CCNC(C1CC2(CC2)CO1)=O N1(C(CC(C)(C)O)=O)CC(NCc2c(O)cccc2O)CC(F)C1 Cc1sc(N)c(C(N2CC(NC(=O)C(F)CC3CCC3)C3(CC3)C2)=O)c1C C1(C(=O)NCc2c(CCNC(C(CC)(C)O)=O)ocn2)Cc2ccc(F)cc2O1 c1(NC2(c3n(CCC)nnn3)CC(CS(N)(=O)=O)C2)cc(OC)cc(OC)c1 C1(CNC(c2cc(C)oc2C)=O)CC(C)CN(C(C2CCCCCN2C)=O)C1 c1(OC(C(=O)NCCN(C(C(F)=CCC)=O)CC)C)ccc(F)cc1 n1(CC)ncc(C(=O)NC2CCCCC2CN(C(c2sc(F)cc2Cl)=O)CC)c1C C12(COC)CC(CNC(c3ccc(F)c(F)c3)=O)(CN1C(C1CCC(F)C1)=O)C2 n1(CC(=O)N(CC(C)NC(C2CC2(C)C(F)F)=O)C)cnnc1O Cc1cc(O)cc(C)c1C(=O)NCC(CNC(=O)C(C)(C)c1nncn1C)CO c1(C(N(C)CC2N(C(C3C(C)CCO3)=O)CCCC2)=O)cn(C)c(=O)n1C c1(C(=O)NCC2CN(C(Cc3n[nH]c(=NC)s3)=O)C3C2C3)cnc2cc[nH]c2c1 CCC(CC)CC(=O)N1CCC(=CCNC(c2cnc(C)o2)=O)CC1 N1(C(CCSCCC)=O)CC(CCNC(c2cc(C)c[nH]2)=O)OC(C)C1 C=C1CCC(C(=O)NC2(c3cccc(F)c3)CCN(C(C3COC3)=O)C2)CC1 C1(NC(C2(COC)CC(=C)C2)=O)CC(C(=O)NCCc2cc(C)no2)=CC1O Cc1ncccc1CCC(=O)NC(C)CN(C)C(C1CCC(O)C1)=O c1(C(N(C(CNC(C(CC(=C)C)C)=O)C)C)=O)cnc(O)n(C)c1=O c1(NC(c2n(C(C)C)cnn2)C)nc2ccccc2nc1N1CC2CC1C2 CCCCCCC(C)C(=O)N(CCC(N1CCC2C(C(N)=O)C2C1)=O)C1CC1 Cc1cnc(C(=O)NCCC(C)(C)C(=O)NC2CCCCCC2)cc1C Cc1ncnc2c1CC(C(=O)NC(C1CN(C(C3CCS(=O)(=O)N3)=O)C1)C)CC2 C1(NC(c2ccc(CCC)[nH]2)=O)CN(CC(O)CC(F)(F)F)CC(C)(C)C1 c1(OCCC)ccc(Nc2ccc(C(=O)NCC(C)O)cn2)cc1CO C(=O)(CCCCCS(N)(=O)=O)N1CCN(C(c2[nH]n(C)c(=O)n2)=O)C(C(F)F)C1 Cc1ccc(C=CC(N2CCCCC2CCCNC(=O)C(C)(O)C2CC2)=O)cn1 CC(C)(C)C(CO)C(=O)NC1CC=C(C(N2CCC3(CCC3)CC2)=O)C1 C(=O)(CCCC(=O)N1CCCCC1C1CCCN(C(C2(C(C)=O)CC2)=O)C1)NC N1(C(C2(NC(C(=CC3CCCC3)C)=O)CCOCC2)=O)CC(C)C(O)C(C)C1 c1(CNC2CCC(C(=O)Nc3c(OC)nc(C)nc3)C2)c(F)ccc2occc12 c1(C(N(CCC(C)NC(c2cn(CCCF)nn2)=O)C)=O)cnccc1Cl C1(N(c2nc(C)cc(C)n2)C(C(C)NC(C=C)=O)=O)CCNCCC1C c1(C(=O)NCCN(C(c2c(CC)c[nH]c2)=O)CC)cc2c(C(F)F)nn(C)c2s1 c1(OC)ccc(CC(N2CC3(CCN3C(c3ccc(O)c(F)c3)=O)C2)=O)cc1C C(=O)(CC(CC)CC)N(CC1CCN(C(COCC(=C)C)=O)CC1)CC C1(CNC(Cn2nc(C(=O)OCC)c(C)n2)=O)COC2(CCCCC2)O1 CC(C)C(C)C(=O)NC(C1CCN(C(=O)CNC(C2CCOCC2)=O)C1)(C)C c1(C(=O)NCCC2COCCN2C(c2ns[nH]c2=O)=O)csc2cccnc12 O=C1OC2CCC1CN(C(c1ccc3occc3c1)C(=O)NC1COC1)C2 C1(C(=O)NCCCCN(C)C(C2CC(O)(C(F)(F)F)C2)=O)CCC2(CCC2)C1 c1(C(=O)NC2C(C)CN(C(=O)CN3CC(=O)NC3=O)C2)cc([N+](=O)[O-])cnc1N C1(C(=O)NC2CC(C#C)C2)CSCCN1C(C1CC(C2CC2)C1)=O Cc1ccc(CNC(=O)CN(C(C)C)Cc2cnsn2)cc1C c1(NC(C2CN(C(c3c(F)ccnc3Cl)=O)CCN2)=O)cnc(F)c(Br)c1 c1(C(=O)NCC(C)N(C)C(C2C3CC4C(C3=O)C24)=O)ccc2c(c1)CC(=O)N2 Cc1ccc(C(=O)NCC2CCCCC2NC(=O)C2=CCSC2)cc1N C(=O)(C#CC1(C(F)(F)F)CC1)NC(C)CCCCNC(=O)C=Cc1ccn(C)c1 CC(CN=c1[nH]c(N2CCC(CC(F)F)C2)nc2c1CSC2)c1cccc(Cl)c1 C1(COC)(CNCc2ccc(CN(C)C)cc2)CC(F)(F)C1 c1(NC(N2CCC(C(C)C(=O)Nc3cccc(O)n3)CC2)=O)cccc(Cl)c1Cl N1(C(COCCNC(C(NOC)=O)=O)=O)CC2(CC(CO)CO2)C1 CC1CC(C(N)=O)CN(C(=O)CCCc2cc(F)ccc2F)C1 c1(CC)ccccc1C(=O)NCCOCC(=O)NC(C(=O)NC)C1CC1 Cc1cc(C(=O)NCC(C)(O)CNC(C2C(C)C2C)=O)c(N)c(Cl)c1 CC(c1ccccc1)=CC(N1CCC(O)C(N(C)C(C2CCC(C)(C)C2)=O)C1)=O CCCCCC(O)CC(=O)N1CCCN(C(=O)COc2ccc(Cl)cc2)CC1C Fc1cc(CNCC2CCCC3(CC3)C2)cc2ccccc12 Oc1cc(C(F)(F)F)ccc1NCCN1CCS(=O)(=O)CC1 c1(CC)ccc(-c2nc(CC=C(Cl)Cl)n(-c3cccnc3C)n2)cc1 C12(CC)CN(C1)C(C)c1nnnn1CCOC(=O)C2.N1CCOCC1.C1(C)N=N1 Cc1cc(C(N)=O)cc(C(=O)NC2CCOCC2NC(=O)CC2CCOC2=O)c1 CCCC(CCNC(=O)C#CCNC(C1CC1CC(C)(C)C)=O)C1CC1 C1(OC)CC(CNC(=O)CCOc2cccnc2)N(C(=O)C=C2CCC(C)C2)C1 N1(C(=O)NCCCNC)CCc2cc(OC)c(OC)cc2C1C C1(F)(CNC(c2nn(C)c(Cl)c2)=O)CCCN(C(=O)C2=CCCCO2)CC1 Cc1ccc(C(F)C(N2CCC(NC(=O)CC3CCOC3)CC2)=O)cc1 C(CC(C(=O)Nc1ccc(C2CC2)nc1)NC(=O)COCC(F)F)=CC C=CC1OCCC1NC(N1CCC(C)(c2cccc(Br)c2)C1)=O c1(-n2c(C(=O)NCC=CCNC(=O)COC3CCOC3)cnn2)ccccc1Cl C1(NC(C=CC(N)=O)=O)CCCOC12CCN(C(c1cc(F)cnc1Cl)=O)CC2 c1(C(N(C)CC2CCN(C(=O)OC(C)(C)C)C2)=O)ccccc1S(=O)(=O)C(F)F c1(C(=O)NC2CCCC(NC(Cn3ncc(C)c3)=O)C2)cc2sc(Cl)cc2s1 C1(NC(c2cc(Br)co2)=O)CN(C(C2(CCO)CC2)=O)CC1C(F)(F)F C1(C(=O)OC)CC(COC(=O)CCNc2ccc(Cl)cc2)C1(C)C C(=O)(C(C)C(O)CC(C)C)NCC1(F)CN(C(c2ccc(C)nc2)=O)C1 CCCCCC(CC)C(=O)NC1CN(C(c2ccnn2CC)=O)CC2CC12 c1(C(N(CCNC(C(C)C2CCOC2)=O)C)=O)cc(Cl)cc(Cl)c1N C1(C(N2CC(C(C)NC(CC(=O)OCC)=O)OCC2)=O)(CF)CC2(CCC2)C1 C1(NC(C=CC(=O)NC2CC2)=O)CN(C(=O)CC2COCCO2)CCC12CCC2 C1(C(=O)NC)Cc2ccccc2CN1C(C1Cc2ccc(C(=O)O)cc2C1(C)C)=O C1(N(Cc2nc(C)[nH]n2)Cc2ccccc2)CN(CC2CCCCS2)CC12CC2 Cc1ccc(C)c(C(=O)NC2CN(C(C3C(C)(C)OC3(C)C)=O)CC2F)c1C N1(C(CCC(=C)Br)=O)CC2CCC2(CCNC(=O)Cn2nccc2C)C1 c1(C(=O)NC2(CC)CCCN(C(C3(SCC)CC3)=O)C2)ccc2[nH]ccc2c1 c1(CCC(N2C(C(C)NC(C(C)=C(C)C)=O)CCC2)=O)c(C)n[nH]c1C C1(CNC(C2N(C(Cc3cc(C)no3)=O)CC2)=O)CC2(CCC2)C1 c1(OC)ccnc(C(N2CCC(C)(CO)C2)=O)c1.N12CC=CC1C2=O c1(C(=O)NC(CNC(C(CN(CC)CC)F)=O)C(C)C)cc(F)c(F)c(F)c1 N(C(=NCCCF)NCC1(C)C=CCCC1)C1CCC(SC)C1 C(=O)(CC(C(F)(F)F)n1cccn1)NCC=CCNC(c1c(C)cccn1)=O N1(CC)N=C(C(=O)N2CCOCC(CNC(=O)CC(C)P(C)(C)=O)C2)CCC1=O c1(C(=O)NCC(C2CC2)NC(C(C=C)OC)=O)ccc2cnnn2c1 c1(CCCC(=O)N(C)CC2OCCN(C(CCC(=C)C)=O)C2)ccc(C)c(C)c1 C(C(C)(C(=O)NCC1CCCCC1)NC(=O)C=C(C1CC1)C1CC1)SC N1(C(C(CC)(C)O)=O)CCC2(CCOCC2)C(CNC(c2ncccc2Cl)=O)C1 C1(C(N2CCC(CCNC(c3nc(N(C)C)oc3)=O)C2)=O)CCC2(CCC2)CC1 c1(N(C(C)CCNC(C2CCCN2C)=O)C)c(C#N)cnc2ccccc12 n1(CC(=O)N(C2CN(C(=O)CCc3cncc(Br)c3)C2)C)cccnc1=O N1(CC)CCCCC1C(=O)N(CC(=O)N(C)Cc1ccoc1)C1CC1 N1(C(c2c(C)cn(C(C)C)c2)=O)CC2CN(C(=O)CCC=CC(C)C)CC2C1 c1(OC)csc(C(=O)NCC(C)CN(C(=O)C(C)(C)c2ccccc2)C)c1OC C1(CCCNC(CCSC(C)(C)C)=O)CCCN1C(c1ccc[nH]1)=O N1(C(C(CC)C)=O)CCN(C(c2sc(Br)c(C)c2C)=O)CC1CC C=C(C)CCCC(=O)N1CCCC(CCC)(NC(c2cncc(OC)c2)=O)C1 CCC(CC)C(=O)N1CC2CC2C1C(=O)NCCC(C)N1CCCC1 CCN=C(NCCc1snnc1C)NCCC1(C)CC1(F)F CC1CN(C(=O)CCNc2ccccc2)CC1NC(C1CC12CCOC2)=O C1(C(=O)OCc2c(OC(C)(C)C)nccc2)CC2(CCOCC2)CO1 CC(CCCCNC(C1CC1C#N)=O)NC(=O)CC1(C)CC(F)(F)C1 c1(OCC(=O)NCC(CCNC(C=C2CCN(C)C2)=O)O)c(F)cccc1F c1(OCC)ccc(F)cc1C(N1CCN(C(=O)C=Cc2ncc[nH]2)C(CF)C1)=O CSC=CC(=O)NCC1(NC(c2scnc2C(C)C)=O)CCC1 c1(OC)cnc(Cl)c(CC(N2CCC(CN(C)C)C2)=O)c1.C12CC1C(=O)N2 c1(CC)nn(C)cc1N.c1(CN2C(=O)C(=O)N3C(CC3)C2)ccccc1F C(=O)(CCN(OC)C(=O)C1CCCC(C#N)C1)NC(C#C)(C)C1CCC1 C1(C)(c2nc(C(C)C)on2)CCN(Cc2cnn(CC3CCOC3)c2)C1 c1(C(CNC(=O)NC(CCC)c2cccs2)(C)O)cccc(Cl)c1 c1(CCNC(C(C2CCN(C(C3CS(=O)(=O)C3)=O)C2)C)=O)cnn(C)c1 C1(NC(CC2CCCN(C(Cn3c(C)ncc3)=O)C2)=O)COC2(CCC2)C1 C=C(C)CC(=O)NCCCOCCN(C)C(c1csc(CCCCC)n1)=O C1(NC(Cc2nc(C)sc2)=O)CC2CC(C1)N(C(c1cnn(C(C)C)c1C)=O)C2 N1(C(c2c(C(C)C)occ2)=O)CCC(CCCNC(c2cn(C)nc2O)=O)CC1 N1(C(=O)CSCC2CCCCO2)CCC2(CC1)CCN(C(C1CC(F)C1)=O)CC2 C1(NC(c2cncc(OC)c2)=O)CC(O)CN(C(=O)Cc2ncccc2C)C1 c1(OC)ccnc(O)c1C(=O)NCC1(NC(C2CCNC2=O)=O)CCOC1 c1(C(=O)NC2CC2NC(C2C=CCS2)=O)ccc(F)c(Cl)c1F c1(N2CCC(SC)CC2)nc(=NCCN(C)C)[nH]c2ccsc12 N#CC1CCN(C(C2COCC2NC(=O)Cc2cc[nH]n2)=O)C1 C12(NC(c3cnco3)=O)CCCC(NC(C3CC4(CC4)C3)=O)(C1)C2 c1(OC)cc(S(=O)(=O)N2CCCC(CNS(=O)(=O)c3ccncc3)C2)ccc1Br C(C)(C)(CC(F)C(=O)N(C)CC1(C)CCC1)NC(C(N1CC(C)C1)C)=O n1(CC=C)cccc1C(=O)NCC=CCNC(=O)C(C)Cc1ccco1 CN1CC=C(CC(=O)N2CCC(O)C2C(N2CC(F)(CF)C2)=O)CC1 c1(CC)c(C)nn2ccc(C(=O)OCC3CCC(OC)CC3)nc12 c1(C(N2CCN(C(c3nccc(C)c3)=O)C(C#N)C2)=O)c(F)ccc2[nH]ccc12 C1(n2cnc(C(=O)OC)n2)CCCN(N2CCC3CCCCCC3C2)C1 N1(C(c2n(C)nnc2)=O)CCOC(CCNC(C2CCC(OC(F)F)CC2)=O)C1 c1(-c2nc(CC3(OC)CCOCC3)n(C)n2)cccc(S(C)(=O)=O)c1 c1(CNC(C2SCCN(C(c3ccc(OC)s3)=O)C2)=O)cccc(O)c1F C1(NC(c2c(CC)cc[nH]2)=O)CC2CN(C(c3cnc(CC4CC4)s3)=O)CC2C1 N(S(=O)(=O)N1CCC(n2c(=O)oc3ccccc23)C1)(CCCC)CC N1(C(c2ncncc2-c2cnn(CCN3CCC3)c2)=O)CCc2cccc(Cl)c2C1 C1(C(C)(C)C)C(NC(=O)C(=O)NC(C)C)CCN1C(c1ccc(NC(N)=O)cn1)=O N1(C(C=C(C)C)=O)CC2CCN(C(c3ccc(C)c(CO)c3)=O)C2C1C C1(NC(CC(C(=O)OC)C)=O)CCC2(CC1)CC(NC(=O)Cc1csc(C)n1)C2 c1(C(=O)NC(C(=O)NC(C2CCOC2)C#C)c2cccs2)coc(C)c1 C1(NC(C(c2cccnc2)OC)=O)CCC(CNC(=O)CC=C(C)C)CC1 C(=O)(C(C)(C)CCC#N)NCC1CCC(C(N(C)CC2CC(=C)C2)=O)O1 N1(C(CNC(C)=O)=O)CCC(CCNC(c2ocnc2C)=O)CC1C N1(C(Cc2nc(C(C)C)sc2)=O)CCC2(CC1)CC2NC(c1cc(C#N)c[nH]1)=O N1(C(=O)CC(F)(F)Cl)CCN(C(C2CC(O)C2)=O)CC12CC2 C1(C(N2C(C)C(NC(c3ccc(F)c(O)c3)=O)CC2)=O)CC(C)(C)SC(C)(C)C1 CN1N=CC(CC(=O)NC2COCC2C(=O)NCC2CCC3(CC3)C2)C1=O c1(CC)nccn1C(C)CC(=O)NCCCCCN(C(=O)C(CC)N(C)C)CC C(CC(C)(C)C(=O)N1CCOCC(NC(C2CC2C(N)=O)=O)C1)SC c1(OC)cc(C(=O)NCC2C3CN(C(=O)COC(C)=O)CC23)cc2c1OCCO2 Cc1csc(CCNC(=O)C(CC2CC2)NC(c2cc(Cl)c[nH]2)=O)n1 N1(C(c2ccc(C(C)C)s2)=O)CCC(NC(c2ccc(Cl)o2)=O)C(C)C1 O(C=C(C#N)C(=O)N1CC(CN(C(=O)Cc2ccc(Cl)c(F)c2)C)C1)CC N1(C(c2cc(C)sc2)=O)CCC2(CCC2NC(c2cn3cc(C)sc3n2)=O)CC1 C(=O)(C(C)(CO)NC(=O)Cc1cccs1)N(C)Cc1nc(C)[nH]n1 C(=O)(C(C)(C)CC(C)(C)C)NCC(CNC(CCC(=O)NC)=O)F C(=O)(C1=CCCSC1)NCCN(CC(C)O)C(c1n(CC#C)ccc1)=O CC(C)C(CNC(=O)C(C)n1cncn1)NC(c1cnn(CCF)c1)=O CC1CCN(C(=O)CCc2ccc(F)nc2)CCN1C(C1(C2CCCO2)CC1)=O C(=O)(CCC(=O)NC(C)(C)CCNC(=O)C(C)(C)N1CCCCC1)NCCC CCCCC(F)C(=O)N1CCCC1(C)CCC(=O)NCC(=O)NC1CCC1 N1(C(C2CC(C(C)C)OCC2)=O)CC2(C1)CN(C(C1CC1c1ccccc1)=O)C2 N1(C(CC2(CNC(c3c(C)snc3)=O)CC2)=O)CC=C(C(C)(C)C)CC1 C1(N(C(=O)COCC(F)F)C)CCC(NC(C2CCN(CC(F)F)CC2)=O)CC1 C1(F)(CNC(C(C)SC)=O)CCCN(C(=O)CCNC(=O)Cc2ccncc2)C1 c1(SC)cccc(=Nc2cccc(S(=O)(=O)NC3CCc4cc(F)ccc43)c2)[nH]1 N1(C(C(C(=O)OC)C)=O)CCC2(CCC(NC(=O)CC(C)(C)SC)C2)CC1 N1(C(C(C)OCCOC)=O)CC2CC1CN2C(c1sc(Cl)c(Cl)c1OC)=O N1(C(CCCSC)=O)CCN(C(C2(c3cccc(C)c3)CCC2)=O)CC1 C(=O)(C(C)C(O)C(C)C)NCC1(O)CCN(C(c2cnn(C(C)C)n2)=O)CC1 c1(C(=O)NCC2(NC(C(S(CCC)(=O)=O)C)=O)CC2)cc2ccccc2cc1O c1(C(=O)NCC2C(NC(c3cc(CC)nn3C)=O)CC2)cc2cc(F)ccc2o1 N(C1CCOc2cc(F)ccc21)C(C1CC1C1CC1NC(=O)OCC(C)(C)C)C c1(CNC(CN(C(=O)CSCCC#N)CCC)=O)cn(C)cn1 c1(CCNC(=O)NC2CC(C)OCC2)cc2ccccc2o1 C(CCC(C)C(=O)NCC1CCN(C(c2cc(O)ccc2C)=O)CC1)OC C1(C(=O)NC(CNC(CCC=C=C)=O)C)COCCC1(F)F Cc1cc(O)nc(C)c1C(N1CC(NC(=O)CSCC(F)F)CC(F)(F)C1)=O c1(C(N(CCNC(CCC(CC)OC)=O)C(C)C)=O)ncnc2c1OCCO2 N1(C(C(=O)NCCOCC)C(C)C2CCOCC2)CC2CC=CCC2C1 n1(CC)cc(Cl)c(C(=O)NCCCCC(C)NC(=O)CC(C)c2cnn(C)c2)n1 C1(CC(=O)NCc2scc(CC)n2)CC2(C1)CN(C(=O)CCCOC)C2 CC(CC1CCC1)C(=O)NCC1(CNC(C2CCC(CO)O2)=O)CC1 c1(OC)ccc(C(F)F)cc1C(=O)NC1COCCC1NC(C1CCN(C)C1=O)=O N(C(=NCC1CCNC(=O)C1)N(C)Cc1ccccc1OC)C(CC)C CCC(C)C(C(=O)NCC1(O)CCSC1)NC(C1CN(C(C)=O)C1)=O c1(N2CCCC(CNC(c3cc(Cl)c(Cl)nc3Cl)=O)C2)ncnc2sc(Br)cc12 C1(c2c(C(N3CC(OCC)C3)=O)c[nH]n2)CCCCN1C(=O)CC(C)C1CC1 N1(C(C(C)N(C(=O)C(C)(C)CO)C2CC2)=O)CCC2(CC2C)C1 C1(C(C)C)CCC(C(N2CC(CNC(c3csc(Cl)n3)=O)C3CC23)=O)CC1 N1(C(c2c(C)nc(C)[nH]2)=O)CC2CCC(C1)N(C(c1ccc(F)c(CO)c1)=O)C2 c1(CC2CC(n3cc(CCC(=O)N(CC(F)F)SC)nn3)C2)ccc(F)cc1Cl N1(C(c2ncc(OC)nc2)=O)C(C(N2CC(O)CC2CO)=O)CC2CCCC12 N1(C(C(=O)NC(CC)CSC)=O)CCC(NN)CC1 CC(C)CCC(O)C(=O)NCCOCCNC(=O)C(=O)N(C)C c1(C(C)C)ncc(C(N2CCN(C3CCCC3NC(C3CCO3)=O)CC2)=O)cn1 C1(C(N)=O)CCCCC1N=c1[nH]c(=NCc2cccc(F)c2Br)[nH]c2c1CCC2 Cc1nc(-c2cn[nH]c2)ccc1C(=O)N(C1(c2ccccc2)CC1(C)C)C1CC1 N1(C(C(CN(C)C)c2ccccc2)=O)CCCC(N(C(=O)C=CC2CC2)CCF)C1 C1(NC(c2ccn(C)n2)=O)C2CC(NC(C3COCC3(C)C)=O)CC12 N1(C(C(C)OCC#C)=O)CCCC(CC(=O)NCc2cc(C)cc(C)n2)CC1 CC1CCN(C(C2CCC(C)CC2)=O)CC1NC(C1COC(C)(C)C1)=O CC(CCCCCO)NC(C1CC2CCC1N2C(c1cc(=N)[nH][nH]1)=O)=O CC(O)C(C)C(=O)NCC1C(C)CCN1C(c1cccnc1F)=O c1(C(=O)NCCN(CCCCCC)C(C2SCCC2C)=O)c(C)cc(C)nc1C N1(C(C(N2CCC(=O)NCCC2)=O)=O)CCC2(CCOC2)C1 N1(C(C(C)N(C(c2cn[nH]c2)=O)CC)=O)CCC(C(=O)NC2CC2)C1 c1(C(=O)NCC2CN(C(c3c(CC)ccs3)=O)C(C)C2)cnn2cnnc2c1 c1(C(N2C3CCN(CC)C3CCC2)=O)cnn2c1OCC(C)(C)C2 c12ncccc1S2.C1(O)(C(=O)NC2(C)CC(NC(=O)CC#N)C2)CCSCC1 c1(C(N2CC3C(NC(C4COCCOC4)=O)(C3)C2)=O)ccc2c(c1)OCCCO2 N1(C(CSCC)=O)CC(NC(c2ccc(F)c(CSC)c2)=O)CC12CCOC2 C1(N(C(=O)CCCN2CCOC2=O)CCC)CCN(C(=O)CC2CCCC2)CC1 C1(=CC(N2C(C)CC(NC(c3n(CCC)nc(C)c3)=O)C2)=O)CCC(C)(C)CC1 C(=O)(CCCCC(N)=O)N1CC(CCNC(C(C(COC)C)C)=O)(OC)C1 O=C(C1=CC2CCCC12)N1CC2(C1)CN(C(C1(CCF)CCOCC1)=O)C2 c1(C(=O)NC(CNC(c2c(C)coc2C)=O)(C)C2CCC2)ccc(S(C)=O)cc1 C(=O)(C1=NOCC1)N1CCC(CCNC(C(C)c2ccon2)=O)C1 c1(SCC(=O)NC(C2CN(C(c3cnc(SC)s3)=O)C2)C)ccc(F)c(F)c1 C1(C(N2CCC(n3cnnn3)C2)=O)(CC)CCCN(C(c2cscc2SC)=O)C1 N1(C(C=CCCC)=O)CCCCCC1CNC(c1cc(NC)ccn1)=O C1(NC(Cc2ccc(C)s2)=O)CC(C(=O)N2CCCC2C(C)C)=CC1O CC1CN(C(c2cnc(C3CC3)nc2)=O)CC(C)N(C(C2CCCC2)=O)C1 c1(C(=O)NCC(C)CC(=O)N2CCCC2)cc(N2CCOC2=O)ccc1F C1(COC)(NC(C2CC2(Cl)Cl)=O)CCCN(C(c2ccc(NC3CC3)cc2)=O)C1 c1(C(=O)NCCCC2CCN(C(C(CC)(F)F)=O)CC2)cc2ccccn2n1 N1(C(c2ncc(NC)nc2)=O)CCC2CN(C(c3cncc(C)c3)=O)CC2CC1 c1(CC(=O)N(CCOCCN(C(C(c2cccnc2)OC)=O)C)C)ccoc1C c1(C(N2CC3C(CNC(CC=CCC)=O)(C3)C2)=O)ccc2c(c1)CCC2(C)C N1(C(c2c(C)ccc(C)c2)=O)CC2CC(NC(=O)CCc3nccn3C)CC1C2 C(C(=O)NC1CC(C(N)=O)C1)(C1=CCC2CC2C1)NC(=O)OC(C)(C)C Cc1ccc(Cn2nc(-c3cccc(C)c3)nc2C(c2cccc(Cl)c2)C)cc1 c12cnn(C)c1Cn1cc-2nn1.C1(CC(=O)N(CC)CC2CCCO2)COC(=O)C1 C(CNC(=O)CCC1CCCCC1)(CC(F)(F)F)NC(CCNC(N)=O)=O C1(F)(C(N2C(C(C)=O)CC2)=O)CCN(C(=O)C=C(C)C2CC2)CC1 Cc1ccc2n[nH]cc2c1C(=O)NCC(C)(C)NC(=O)CCC1CCOC1 N1(C(c2c(C)onc2)=O)CCN(C(=O)CSc2ccc(Cl)nc2)C(C2CCC2)C1 Cc1nc(C(C)C)ccc1C(N1CCC(=CCNC(=O)Cc2nccs2)CC1)=O c1(C(N2CC=CC(NC(C(COC)(C)C)=O)C2)=O)cc(O)cc(=O)o1 CCC(CC(=O)N1CC(CC(=O)NCCOC)C(C)C1)SC C#CCCC(O)C(=O)NCc1ccccc1CNC(c1ccccc1F)=O N1(C(CSC(C)C)=O)CC(CNC(=O)CCCNC(=O)C(C)(C)C)CCC1C C1(C(=O)NC(CCN(C(C(C(CC)O)C)=O)C)C(C)C)CCc2nncn2C1 c1(CNC(C2CCC(C(C)(C)C)CN2)=O)cccc(Br)c1O N1(C(C(C)NC(COC)=O)=O)CC(N(C(=O)Cc2ccc(Cl)nc2)C)C2(CC2)C1 c1(CCO)ccc(NNC(=O)C(F)(F)c2cc(Cl)cc(Br)c2)cc1 C1(OC)CN(C(=O)C(C2CCC2)NC(=O)CC2CC2(C)C)C1 n1(CC)ncc2c(N3CC(C)CN(C(c4ncn(C)n4)=O)CC3C)ncnc12 N1(C(C(F)=C(C)C)=O)CCc2sccc2C1CNC(=O)CCOCC1CCCO1 c1(C(N2CCC(O)(CCNC(C(CC)C)=O)C2)=O)cc(N)c(Cl)cn1 C(=O)(CC1NC(=O)c2ccccc21)N1CCC(CNC(C(C(CC)O)(F)F)=O)C1 N1(CC(=O)Nc2cccc(C)n2)CC2CCOC2(CO)C1 C(=O)(C(C)(C)S(C)(=O)=O)NCC1C2CN(C(C3(CC(C)C)CC(=O)C3)=O)CC21 C(CC(C)(C)CC(=O)OCCCN1CCN(S(C)(=O)=O)CC1)OC c1(CC(=O)NCC2C(NC(c3nc(OCC)oc3)=O)COC2)cc(F)ccc1F c1(OC)ccc2nc(C)nc(N3CCCC3C(=O)NCC3CCCO3)c2c1 CN1CCCC(C(C)(C)C(N2CCC(CF)(NC(=O)CS(=O)(=O)N(C)C)C2)=O)C1 C1(C(=O)NC2CC(CNC(=O)Cn3cnnn3)C2)(OCC)CCCC1 CC1CN(C)CCC1NC(C1CNC(=O)CN1C(c1ccc(CC#N)cc1)=O)=O c1(CCCNC(=O)NCC(C)Oc2cccc(F)c2)nc2ccc(Cl)cc2[nH]1 CN1CCC(C(=O)NCC(C)(CO)NC(c2cnc(Cl)s2)=O)c2ccccc21 C1(C#N)(C(=O)NCC(CNC(c2cncc(C#C)c2)=O)C)CCN(C)CC1 C(=O)(C(F)C(C)CC(C)(C)C)N1CCC(C)(CNC(CCCCOC)=O)C1 N(C(=NCC(=C)C)NCC1CCOC2(CCC2)C1)CC#C.C12(CCCSC1)OC2 c1(N(C)CCN2CCNC(=O)C2)[nH]c(=NC2C=CCC2)nc2scnc12 C1(CNC(c2nccc(SCC)c2)=O)CCCN(C(C2(C(=O)NC)CC2)=O)CC1 N1(C(C2N(C(C)=O)CCCC2)=O)CCN(C(=O)CC(=O)NC2CC2)CC1C1CC1 c1(OC)cc(C(=O)NC(C)CCCCNC(C2CCC(N(C)C)CC2)=O)ccn1 c1(C(N2CC(N(C(c3c(C)ccnc3)=O)C)C3(C2)CC3)=O)cc(O)cc(N)c1Cl c1(C(N2CCCC(C)(CNC(CC3CC(OC)C3)=O)C2)=O)ccc(S(C)(=O)=O)[nH]1 C1(NC(c2ccc(Cl)[nH]2)=O)Cc2ccccc2C1NC(=O)C(O)C(F)F N1(C(C2CN(Cc3ccc(C)s3)CC(F)C2)=O)CCc2nc[nH]c2C1 c1(CNC2C(C(=O)Nc3c(C)ncc(C)c3)C2)cc([N+](=O)[O-])ccc1C c1(C(N2CC(NC(=O)C(F)=CCCF)CC(C)(C)C2)=O)ccc([N+](=O)[O-])c(N)n1 c1(OC)cnc2[nH]c(C(N3CCOC(CNC(C4COC(=O)N4)=O)C3)=O)cc2c1 c1(CC(N2CC(c3ccccc3)C(F)(CO)C2)=O)cc(F)ccc1F C1(NC(CSCC)=O)CC2CCC1(NC(c1nc(C)sc1C)=O)C2 OC1(c2nc[nH]n2)CCN(N2CCOC(c3ccccc3F)C2)CC1 CN1C2CCC1CC(C(=O)NC1C=CCN(C(=O)CN3C(=O)CNC3=O)C1)C2 C(=O)(C(CC(F)F)C1CCC1)N(CCNC(C(CC)N(C)CC1CC1)=O)CC1CC1 c1(CC#N)cccc(C(=O)NC2(C(=O)NCC3CC3C3CC3)CC(O)C2)c1 C(=O)(NNc1nc2ccc(Cl)cc2s1)NC(c1ccnn1C)COC c1(C(N2CC(C(=O)NC(c3ccccc3F)CC)OCC2)=O)cc(Br)ccc1Br c1(N(CCOCC)C)cc(N(C)CCc2cccs2)nc(C(F)(F)F)n1 c1(NC(c2nc(NC(c3scc(C)n3)=O)sc2)=O)cnc(C)c(F)c1 CC1(C)CC(CNC(=O)C(C2CC2)C2CC2)N(C(=O)CCc2ccccn2)C1 c1(CC)cccc(OCC(=O)NCCC2CN(C(c3ncsc3C)=O)CCO2)c1 C1(NCC(CCCC)CC)CCSC2(CCC2)C1 C(CCCCCNC(C1CC=CC1)=O)NC(=O)CCn1cc(Br)cn1 CCC(C)C(C)(O)CNC(C1(CNC(c2nocc2Cl)=O)CC(C)(C)C1)=O c1(C(N2CCCC(C(C)NC(c3nnn(C)n3)=O)C2)=O)cccc(Cl)c1Cl N1(C(=O)OC(C)(C)C)CCC(C)(C(=O)Nc2nccs2)C1.C1C(=O)N1CCF Cc1ccc(C)c(OCC(N2CCC(C)(NC(=O)CC3CCOC3)C2)=O)c1 c1(C(N2CC(C(C)NC(=O)CC3CCOC3)OCC2)=O)cc(C#N)ccc1N C1(CNC(CC(=C)C)=O)CC(COC)N(C(C2CCCN(C(C)C)C2)=O)C1 N1(C(C2C3CC(=O)CC32)=O)Cc2[nH]nc(C(=O)NCC(C3CC3)N(C)C)c2C1 N1(C(C23CC(C)C2C3)=O)CCC(CO)(CNC(=O)CCC(C)(C)F)CC1 C(=O)(C#CC1CCCC1)N(C)CC1N(C(C(C)C(F)F)=O)CCCC1 N1(S(CC=C)(=O)=O)CCN(CC)CC1.C(=O)(CCCC1CCCCC1)N1C(=O)C1 C(=O)(C1OCCc2ccccc21)NC(C(C)C)CCNC(=O)CC=C(Cl)Cl CCC(C)C(C(=O)N(C)OCC(F)(F)F)N(C(=O)CC1COCC(C)O1)C CC(C)C(C#N)C(=O)N1CCCC(C(=O)NCC2CN3CCC2C3)CC1 C1(NC(CSCC(C)C)=O)CC2CCCC(C1)N2C(=O)Cc1csnn1 CCCC(C(N)=O)NC(C1CCCN1C(c1cc(C)oc1C)=O)=O C1(C)(C(=O)NCC2N(C(CC(C)C3CC3)=O)CCC2)CCCNC1=O C1(NC(CN(C)C(N)=O)=O)CN(C(C2CCCCO2)=O)C2(CCCCC2)C1 N1(C(CN(CC)CC)=O)CCN(C(=O)CC2CCOC2)C(CS(C)(=O)=O)C1 C1(OC)CCCCN(CC(N2CCC(C(C)N(C)CC#N)CC2)=O)C1=O C1(C(C)NC(C2C(CCC)CCC2)=O)CN(C(c2cnc(SC)s2)=O)CCO1 C1(C)(NC(C(CC)OC)=O)CCN(C(=O)CCc2ccc(OC)c(F)c2)CC1 c1(CC(=O)NC2(CC=C)CCN(C(=O)C(F)=C(C)C)C2)ccc(OCC)c(F)c1 C12(C(=O)NCCN(C(COCc3n(C)ncn3)=O)C3CC3)CC=CCN1CCC2 [N-]=[N+]=NC1CCN(C(=O)CC2CCN(C(c3cc(F)cc(F)c3)=O)C2)C1 N1(C(C2(CC)CCCC2)=O)CCCCC1CNC(c1cn(C)nc1C)=O CC1CCOC1C(=O)N(CC(C)CNC(=O)CC(=O)N(C)C)C c1(N2C(C)CC(CNC(c3cn(C(C)(C)C)nn3)=O)C2)ncnc2c1CCO2 N1(C(C(=O)N(C)CCN2CCOCC2)=O)CC(F)(F)C1C1(CN)CCC1 C#CCC(C)(CC)C(=O)NCCC(=O)NC1CC2C=CC1C2 N1(C(C2(COC)CN(C(=O)C(N=[N+]=[N-])C(C)C)C2)=O)CC=CC12CCCC2 c1(OC)cccc(CCC(N2CCC3CCC23CNC(=O)C(C)(Cl)Cl)=O)c1OC CCC(CC)(CC)NC(=O)CC1CCCC(NC(=O)COCCF)C1 C1(C(=O)OC)CCCC(CNC(=O)N(c2cccc(C)n2)c2ccc(C)cc2)C1 C1(NC(=O)C(CCC=CCF)N2CCOCC2)CCCC12CN(CC1CC1)C2 c1(NC(=O)CC2COCCN2Cc2ccccc2OCCO)ncc(F)cc1Cl c1(NC(CC)=O)cncc(C(N2CC=CC(NC(=O)CC3CCCOC3)C2)=O)c1 c1(CNC(C(COCC)C)=O)ccnc(C(=O)NCCC(=O)NC(C)C)c1 c1(CC(N2C(C)CC(NC(=O)C=Cc3cnc[nH]3)C2)=O)ccc2oc(O)nc2c1 n1(CC)nc(C)c([N+](=O)[O-])c1NCCC(C)(C)NC(=O)C(C)NC(C)=O CCS(=O)(=O)c1ccc(CCCN2CCCC(C)(C)C2C=Cc2cccs2)cc1 C#CC(CC(C)C)NC(=O)CC1(C)CCN(C(=O)C(C(C)C)SCC)C1 C1(OC)CN(C(=O)CCOc2ccccc2)CC1NC(=O)C=C1CCSCC1 c1(C(N2CC(CC)(NC(c3ccon3)=O)C2)=O)nccc2cc[nH]c12 CC(C)CCC(O)C(=O)N1CCC(C(=O)NCCCC(C)O)C(C)C1 C1(NC(=O)NC2CC3CCCC3C2)CC2C(O)C(O)CC12 C#CC(C)(C)C(=O)NC(c1ccc(F)cc1)CNC(=O)C(F)CC1CCC1 N1(C(c2c(C)cccc2)=O)CCCCC(CNC(=O)C(C)OC2CCCC2)C1 C1(C)(C(=O)NCc2c(C(=O)NC(CC)C(C)O)n[nH]c2)CC2C=CC1C2 N1(C(C)=O)CCC(CCNC(=O)CNC(=O)CN(C)C)C1.C12CCC(C1)C(=O)N2 c1(CC)nsc(CNC(=O)C(O)C2CN(C(c3ccsn3)=O)C2)n1 n1(C(C(=O)N2CC(OCCNC(CCCC#C)=O)C2)C)c(C)cc(O)cc1=O c1(C(C(=O)N(CCC#N)C(C)(C)C)NC(=O)OC(C)(C)C)ccc(Cl)cc1 n1(CCC)ncc(C(C(=O)NCCSC)N(C2CCC2C)C)c1C c1(NC2CCC(C(=O)NCC(C)CCl)C2)ncc2ccccc2n1 c1(C(=O)NC2CSC2)n[nH]c2c1CN(C(C1CCO1)=O)C2 Cc1cc(C(=O)NCC(=O)NCC(N2CCC=C(Cl)C2)=O)ncn1 c1(C(=O)NC(CC=C)C(=O)NC(c2cccnc2)CO)cc(F)ccc1F c1(C(N(C2CCN(C(CCC(=C)Cl)=O)CC2)C)=O)ccc(O)cc1F n1(CC(=O)NCCSC)cc(CCC(O)C2CC2)nn1 n1(CC(C)C)nccc1C(=O)NCCCCNC(=O)CC1CC1c1ccncc1 C(=O)(CC(C)(C)C#N)NC1C(CNC(C=CC(c2cn(C)nc2)=O)=O)CCCC1 Cc1ccn(CC(C)C(=O)NCCCC(C)NC(=O)CCSc2n[nH]c(C)n2)n1 Cc1ccc2c(C(N3CC(CCNC(=O)CCC4CCCCO4)C3)=O)n[nH]c2c1 N1(C(CCOC)=O)CCC2(CCC2NC(C23CC(C(F)(F)F)(C2)C3)=O)CC1 CC1C(C(=O)NCCCSCCO)CCCN1C(c1cncn1C)=O CC#CCC(C(=O)NCC(O)C(C)C)NC(c1ccc(=N)[nH]n1)=O c1(C(N2CCC(OCC=C)C2)C(=O)NC)cccc2c1oc1ccccc21 c1(C(=O)NC(C(C)NC(c2ccc(OC)cc2)=O)C(C)C)ccnc2ccsc12 C1(C(=O)NCCC(CNC(COCCCC)=O)OC)CC(C)(C)CCO1 n1(CC=C)cc(CNC(C2OCCC2NC(C2CCSCC2)=O)=O)nn1 C1(CNC(C(CC)n2cncn2)=O)CCCCN(C(c2cc(C)c(C)s2)=O)C1 c1(C(=O)OC)ncc[nH]c1=NCC1C(C)CCCN1C(C12CCC(C1)OC2)=O CCC(C)CCCCC(=O)NCC(C(C)(C)C)NC(=O)C(C)Cc1cnn(C)c1 C(=O)(CCCC(=O)N1CCC(NC(=O)CC2CC2(C)C)C1C1CC1)NCCC S(=O)(=O)(c1ccc(NCC2(CO)CCOC2)c(Br)c1)NCC1(C)CCCCCC1 C(CC)(CCCC(=O)N1CC(F)(F)CC1CO)NC(C(C1CCC1)OCC)=O c1(CC(N2CC(C)C(NC(C(C)C)=O)C(C)C2)=O)nn(C)c2ccccc12 C1(C(N2CCNCC2)C)CCCN(c2ccc(Br)cc2)C1=O C1(C(N2CCC(CNC(C(CC)OC)=O)(COC)C2)=O)CC2(C1)CC(F)(F)C2 C(C(=O)N1CCN(CCCCCNC(=O)CN(C)C)CC1)(C(C)C)N(CC)CC c1(C(N(C)CC2CCN(C(CSCC=C)=O)C2)=O)ccc(S(=O)CC#N)cc1 N1(C(CCN(CC)CC)=O)CCC2(NC(c3nc(CO)no3)=O)CCCC12 c1(CC(=O)N(CCNC(C2ON=C(C)C2)=O)C)cnc2cccnn12 C1(OC)CC(CNC(=O)CCc2cccs2)N(C(=O)C=CCN2CCCC2)C1 c1(OCCC(=O)NCC(C2CCOC2)NC(C=COCC)=O)cccc(Cl)c1 c1(C(=O)NCC(c2ccccc2)NC(=O)C2=CSCCO2)cnc2occc2c1 Cc1[nH]c(C)c(C(N2CC(NC(c3cccc(Br)c3C)=O)C3(CC3)C2)=O)c1C N1(C(CCOCCC)=O)CCC(COC)(NC(=O)CCNC(N)=O)C1 N1(C(Cc2c(CC)cccc2)=O)CCC(CNC(=O)C(C)C(C)(F)F)(OC)CC1 S(=O)(=O)(c1ccc(Br)cc1Br)NC(C12CCN(C(=O)OC(C)(C)C)C1C2)=O N1(CC(=O)NC)CC2CN(C(=O)CCOc3ccc(Cl)c(CO)c3)CC2C1 N1(C(C(C(C)C)C)=O)CC(C)(C)OCC1CNC(=O)C1=CCCC1 c1(C(N(C2CCCC(N(C(=O)CC3CCCC3)C)C2)C)=O)csc2ccccc12 Cc1c2ccc(C(=O)NC(C)Cn3cc(C)nn3)cc2nn1C.c1(O)ccccc1 c1(NC(c2c(NC(c3c(OC)csc3)=O)cccc2F)=O)n[nH]c2c1CCCC2 N1(C(CC(CNC(C(CCOC)OC)=O)O)=O)CCN(C)CC1CO N1(C(c2n[nH]c(C)c2Br)=O)CC2CC1CCN2C(C1C2CC3C(C2)C13)=O c1(C(=O)NC2C3CN(C(C(C)O)=O)C2C3)cc2cc(Cl)cc(Cl)c2[nH]1 N1(CC(c2ccc(C(C)=O)cc2)=O)CCC(O)(c2ccc(Br)cc2)CC1 N1(C(C2C(OC(C)(C)C)C2)=O)CC2CC(CNC(c3cncc(Cl)c3Cl)=O)C2C1 O=C1NC2(CO1)CC(C(=O)NC1CC(CNC(c3cccc4c3CCO4)=O)C1)C2 N1(C(C(CCC#C)NC(c2ccccn2)=O)=O)CCc2ncn(C)c2C1 N1(C(C=C2CCN(C)C2)=O)CCC(F)C(NC(c2cnns2)=O)C1 C1(CNC(C)=O)CN(C(C2COC3(CCC3)C2)=O)CCC1(C)C C1(C(C)O)CCC(NC(C2CCN2C(=O)CCc2ccncc2)=O)CC1 c1(N(C(C)CNC(C2CCCCC2c2cccnc2)=O)C)ncc2ccnc-2[nH]1 Cc1cnccc1NC(=O)CN1CCN(S(=O)(=O)C(C)C)CC1 C(CCCC(=O)NCc1ccoc1C(=O)NCC1CC1[N+](=O)[O-])SC C1(CC(F)F)CN(N2CC(C3CCCCC3)C2)C1 c1(C(=O)NCC(CO)NC(C(CCC)(C)C)=O)c[nH]c2cc(Cl)c(OC)cc12 N1(C(c2c(C)nc(C)o2)=O)CCC2(CC2)CC1C(N1CCC(F)(F)C(F)C1)=O N1(C(C2=CC(C)CC2)=O)CCCC2(C1)CN(C(=O)C(C)Cc1ccccc1F)C2 C1(C(=O)NCCOC2CN(C(C(C)N(CC)CC)=O)C2)CN2CCC1CC2 C1(CNC(c2cc(C(N)=O)oc2)=O)COCCN(C(C2CCCS(=O)(=O)C2)=O)C1 C12(C(=O)NCC(CCNC(C3(C)CC(C)=NO3)=O)OC)CCCC1CC(=O)C2 C1(Cn2cc(CCCC(C)=O)nn2)CC12CCN(C(=O)COC1CCCC1)CC2 C(=O)(C(O)CCCNC(C1CC(=O)OC1(C)C)=O)NCCN(CCCF)C C(C(F)(F)CC(=O)Nc1cccc(CCF)c1)N(C)C C1(F)(CNC(C(C)NC(C)=O)=O)CCN(C(=O)Cc2ccc(Br)cc2)C1 c1(CC)nc(C)c(C(=O)NC2(C)CCN(C(c3cnccc3C)=O)C2)s1 N1(C(CC(C(=C)C)O)=O)CCC2(CCCC2NC(=O)C=CCCC)CC1 C=C(C)CC(C(=O)NC1CCNC1=O)NC(=O)CC1CCCN1C C1(NC(Cc2nnc(C)s2)=O)CN(C(=O)C(C2CCCCC2)O)CC1C1CC1 N1(C(c2n(C)ccc2)=O)CC(CNC(c2cc3scc(Cl)c3[nH]2)=O)CC12CCC2 N1(C(C(C)Sc2scc(C)n2)=O)CCC2(CC1)CC(O)CNC2=O c1(C(=O)NCCN(C)C(C2OCCO2)=O)cc2nc[nH]c2cc1[N+](=O)[O-] c1(C(=O)NC2CCN(C(c3ccc(=O)n(C4CC4)c3)=O)C2)cccn2c(O)nnc12 Cc1ccncc1-c1cn(CC(N2CC(CO)C(CO)C2)=O)nn1 N1(C(c2ccn(CCC)n2)=O)CC2(C)CC1(C(=O)NCC(N1CCCC1)C)C2 CC1(C)C(C(=O)NC2CCCCC2NC(C23CC2CNC3=O)=O)CC1(F)F C(CCCC(=O)NC1(C2CCCN2C(=O)CO)CC1)OCCC=C C(=O)(CCN=c1[nH]ccs1)N1C(CNC(C2CC3CC3C2)=O)CC(OC)C1 c1(NCC(CO)F)nccc(=NCc2cc(O)nc(C3CC3)n2)[nH]1 n1(C(CC)C)nc(C(=O)NCCC(C)(C)NC(C2CCOC2)=O)cc1C C=CCC(CC)C(=O)NCCC(O)C(N1CCCC(CCC)CC1)=O c1(C(N2CCC(C3N(C(CSC)=O)CCCC3)C2)=O)cnn2cccc(Cl)c12 Cc1cc(NC(=O)C(=O)N(C(=O)OC(C)(C)C)CC2CC(C)CO2)ccc1Br CN1CCN(C(=O)COC2CC=CC2)CC1C(=O)N(C)Cc1cccnn1 N1(C(C2C(C)(C)C2)=O)CCCC(C)(C)C1CNC(c1sccc1CO)=O c1(C(N2CCCC(C)(NC(C(CC)NC(N)=O)=O)C2)=O)cnc2[nH]nnc2c1 N1(C(CNS(NC)(=O)=O)=O)CC(NC(c2ccsc2)=O)CC12CCCC2 C1(C(N2CCN(C(CCCCC)=O)CC2C2CCCC2)=O)CC2(C1)CC1(CC1)C2 c1(NC(C2C3CN(C(C(N4CCCC4=O)C)=O)CC32)=O)cc(O)ccc1F N1(CC)CCCC2(CCC2)C1C.C12CC(C1)CCNC2=O N1(C(C2C(C)CC(=O)N2)=O)CCN(C(=O)C(F)OC(F)(F)F)C2(CCC2)C1 c1(CC)nc(C)c(C(N2CCC(NC(=O)C(C3CCCO3)C3CC3)C2)=O)o1 n1(CCNC(C2(C(C)C)COC2)=O)cc(C(=O)NC(CO)CCO)nn1 C1(C(=O)NC(CC#C)C)CCC(C)CN1C(C1CC(C)(O)C1)=O CC(CN1CCOCC1)C(=O)N1CCC(OCCNC(=O)CC2CCOC2)C1.OCC N1(C(COCCNC(C(C=C)O)=O)=O)CCC(C)(O)C1 c1(OC)cc(C(=O)NC2CCCCC2C(=O)Nc2cnn(C3CC3)c2)cc(O)c1O C1(C)(CC)CC(NC(=O)CN(C)CC)CN1C(=O)CCSCC(F)(F)C(F)F C(=O)(C1CCCc2ccnn21)N(C1CN(C(=O)C(C)(C)C2CC2)C1)C c1(OC)ccc(C(N2CC(CCO)(NC(C3CCNC(=O)C3)=O)C2)=O)cc1C C(=O)(CCCCCC(C)(C)C)NCCCN(C(C(C)C(F)F)=O)C1CC1 c1(C(N2C(C(C)(C)C)C(NC(C34CCC3C4)=O)CC2)=O)cn2ccsc2n1 Cc1[nH]cc(C(=O)NCC(C)CNC(=O)C(C)(C)C(C)O)c(=O)c1Br C1(NC(=O)C2=CCSC2)CCC2CCN(C(=O)CC(O)C3CCCC3)C12 Cc1cncc(C(=O)NC2CCC2CNC(c2sccc2CC#N)=O)n1 c1(C(=O)NCC(C2CCC2)NC(CC(C)C)=O)cccc2nsnc12 CC1CN(C(=O)Cc2ccc3nonc3c2)CC(C)C1NC(=O)Cn1ncnn1 c1(CNC(CCSCCCC)=O)cn(C2CN(C(C3CC(=C4CC4)C3)=O)C2)nn1 C1(C(N2CCC(CN(C)C(=O)OC(C)(C)C)C2)=O)CC(C(=O)O)C(O)C1 N1(C(C(C)C2CC2)=O)CC2CCC1C1CN(C(c3cc(Cl)nnc3O)=O)CC21 C(C(C)(C)CCC#N)(c1nnnn1CCCOC)NC(CC=C)CC(F)F C1(C(=O)NC(CC)CNC(=O)C=CSC)(Cc2ccc(F)cc2)CCCCC1 N1(CCNC(=O)NCC(C#C)CC2CC2)c2ccccc2C(C)C1 c1(OC)c(C(N2CCCC(CN(C)C(C3(CCF)CC3)=O)C2)=O)cnn1C CCCCN=C(NCCc1cn(C)nc1C(F)F)NCC1CCC(C)(C)O1 C=Cn1nccc1C(=O)NC1C=CCC(C(=O)NC(C2CCCC2)CC)C1 N1(C(Cn2cc(CNC(c3cc(C)sc3N)=O)nn2)=O)CC(C)N(C)C(C)C1 N1(C(C=CCCC)=O)CCCN(C(C2CCOC2(C)C)=O)C(CO)C1 N1(C(c2c(COC)cc[nH]2)=O)CC(NC(=O)CCC2CCC(=O)N2)CC(F)C1 CCCC#CC(C)(C)NC(C1(C)CN(C(=O)CN(C)CCOC(C)=O)CC1C)=O C(=O)(C(C)(COC)CC)NCCN(C(c1cc(CCC)on1)=O)C(C)C C1(C(=O)NCCCN(C(C)C)C(c2cnc(C3CCC3)s2)=O)CNC(=O)CC1C C1(C)(C(=O)NCCOCCN(C(c2ccc(C)c(C)c2)=O)C)CC(C)OC(C)C1 c1(OC)cc[nH]c(=NCCC2CC(NC(=O)CC3CCCOC3)C2)n1 c1(C(N2CC(N(C(CC(=C)C)=O)C)C2)=O)ccc(OC)c2ccncc12 N1(C(C=CCC)=O)CC2CCC1CN2C(c1cc(Cl)cn1CC)=O c1(C(N(CCN(C(C)C)C(=O)C2CC2)C)=O)csc(CS(C)=O)n1 S(=O)(=O)(C1CCN(C(=O)NCC(c2ccco2)N(C)C)C1)NC(C)C C12(C(=O)NCC3(COC)CN(C(C)=O)C3)COC(Cc3ccnc(OC)c3)(C1)C2 c1(CC)cc(C(=O)NC2CCC(NC(=O)C(C)(C)n3cnnn3)CC2)cc(O)n1 CCC(C)(CNC(C1(C#N)CCCCC1)=O)C(=O)N1CCCC(C)CC1 C(=O)(C1=NN(C)C(=O)CC1)N1CCC(C)(CNC(CCCC(=O)N(C)C)=O)CC1 C1(C(N(CC(O)CF)C)=O)C2CC(O)C(C2)N1C(=O)CC(C)(C)C C(=O)(CCCCC(N)=O)NCC1C(C)CN(C(C2CC2c2ccccc2)=O)C1 CC1CCCC(C)CN1C(C1CCC2CCC1N2C(=O)OC(C)(C)C)=O c1(C(N2CCC(Cn3cc(C(C=C)(C)O)nn3)C2)=O)nc(Br)n2c1CCC2 C(=O)(N=c1cc[nH]c(C)c1C)C1C(NC(c2cnc(C)[nH]2)=O)CCCC1 C(=O)(CCC(C)(C)C#N)N1CCC(C(CCCN=[N+]=[N-])C)CC1C C1(CCC)CN(C(c2ccc(C(C)C)o2)=O)CC1C(N1CC2(CCC2)C1)=O C1(C(N2CC(C)C(NC(=O)C(CO)NC(N)=O)C2)=O)CCOC(=O)CC1 c1(CCC)cc(C(=O)NCC(C)N(C(=O)C(C)NC(=O)NC)CC)n(C)n1 CC1CCN(C(C2C3CCN2CC3)=O)CCN1C(=O)CCCN(C)C c1(-c2ccc(C(=O)NC)cc2)cn2cc(C(=O)NC(c3ccno3)C)ccc2n1 C(=O)(C(O)CCCCC)NCC(CC=C)C(=O)N1CCOC(COC)C1 C(=O)(C(C)CC(C)(C)C)NC12CN(C(c3cc(OCC)c(C)cc3)=O)C(C1)C2 C1(CC(=O)N(C(C)CNC(c2sccc2Br)=O)CC)CCCN(C)C1 N1(C(CC(C)(F)F)=O)CCC2(CCC2NC(=O)CSc2ccc(C#N)cc2)CC1 c1(C(N2C(C3(NC(=O)CC4=CCCC4)CC3)CCC2)=O)cc2c(O)cccc2[nH]1 C1(C)(CCC(=O)N(C2CCOC2)CC)CN(C(=O)CCn2cc(C)cn2)C1 S(=O)(=O)(c1ccc(=NCCC(C)O)[nH]c1)N1C(COC)COCC1 N1(C(c2cc(C)cc(C)n2)=O)CCN(C(=O)Cc2ccc(O)c(Cl)c2)C2CCC12 C1(C2(C(N3CC(C#C)(N(C)C)C3)=O)CC2)CN(C(=O)Cc2cc[nH]n2)CC12CC2 C(=O)(C(CC(C)C)N(C)C)N1C(CNC(CCc2onc(C)n2)=O)C(C)CC1 C(=O)(CCC(C)(C)F)N1CCCC(CN(C(c2c(C)n(CCO)cc2)=O)C)C1 N1(CC)CC(NC(c2c[nH]nc2CNC(c2ccc(O)cc2)=O)=O)C(C)C1 c1(NC(C2CCC(NCc3ccc(CO)cc3)C2)=O)ccc2c(c1)COC2 c1(C(=O)NCCC2C(C(=O)OC)C2(F)F)ccc2c(ccn2C(C)C)c1 CCC(CC(C)CO)NC(c1n[nH]cc1CNC(c1ccc(OC)nc1)=O)=O c1(C(N2C(COC)CN(C(=O)Cc3cncs3)CC2)=O)cnc2sccc2c1 C#CCC(C)(C(=O)N1CCCOCC1C)NC(C1CCC1OCC)=O C1(C2CCCO2)(C(=O)NCC(CNC(c2c(C)snc2)=O)(C)O)CCOCC1 Cc1cc(C(C)C(N2CCCC(N(C(=O)C(O)C3CCC3)C)CC2)=O)cc(F)c1 CCCCCC(O)C(=O)NC(C(=O)NC1CN(CC)C1)C1CCCC1 c1(CC(=O)NCC23CC(NC(C(C)=CC4CC4)=O)(C2)C3)cc(F)c(F)cc1F N1(C(c2ccc3ccoc3c2)=O)CCC2CCC(C1)N2C(C1C=CCC1)=O CCC(C)CC(=O)NC(CSC)C(=O)N1CC(CN(C)C)C1 Cc1nc(NCCCOC2CC2)cc(N(CCCOC(=N)O)C)n1 N1(C(C2C(c3n(C)cnc3)C2)=O)CCC2(NC(C3CC3(F)F)=O)CCCC12 N1(c2nccc(SC)n2)CCC2(CC(NC(c3cc(-c4cccs4)on3)=O)C2)C1 N1(C(CCC(=C)C)=O)CC(C)CCC1CNC(c1ccn(C(C)C)c(=O)c1)=O N1(C(CC(=O)OC)=O)CCCN(C(c2nccc(OC)c2C)=O)CCCCC1 c1(C(N(CC(CC)NC(=O)C(O)CN2CCCC2)C)=O)cccc2nonc12 C(CCN=C(NCc1ccc(Cl)nc1)NCC1CC2CCC1O2)OCC C1(C(=O)OC)(CO)CCN(C(c2cc(C3CC3)on2)C(=O)NCCCF)C1 C1(CNC(CCOCCN(C(=O)CS(C)(=O)=O)C)=O)CC(O)C(O)C1 C1=COc2cc1c(OC(F)F)cc2.N1(C(C)=O)CCC(C(=O)O)CC1 N1(C(c2ccn(C)c(=O)c2)=O)CCC2CN(C(C3(C4CCC4)CC3)=O)CC2CC1 N1(CCC(N2CC(CNC(C(C)OCCOCC)=O)C2)=O)CCC(C)CC1 c1(CN2CCC(c3n(C)cnn3)C2)c(-c2ccc(C=O)o2)cnn1C C(=O)(C(CNC(c1n[nH]c2c1COC2)=O)C(C)(C)C)NC(C(CC)(C)C)C Cc1cccc(F)c1CC(=O)N(CC(O)CNC(c1cc(Br)cn1C)=O)C c1(NC(c2nccc(C#C)c2)=O)nc2c(s1)CC(NC(=O)C(O)C(C)C)CC2 N1(c2c(C)cncn2)CCC(F)(F)C(C(N2CC(O)CC2CN2CCCC2)=O)C1 c1(NC(c2c(CNC(c3ncc(CC)cn3)=O)ccs2)=O)ccc(Cl)cc1C c1(CNC(CC(C(C)C)OCC)=O)nc2c(s1)CN(C(=O)C(O)CC)CC2 N1(c2ncn(C)n2)CCc2sc(-c3cccc(O)n3)nc2C1 c1(CN=C(NC(C=C)C)NC2CC3(CC3)C2)cccc([N+](=O)[O-])c1C Cc1cccn2c(CC(=O)NCCC(O)CNC(C34CC(F)(C3)C4)=O)cnc12 CC(C)CC(O)C(=O)NC1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)C12CC2 c1(C(C)=O)cc(C(=O)NC2CC2CNC(=O)CCCOc2cccnc2)co1 N1(C(c2cn(C)[nH]c2=N)=O)CCC(CNC(c2ccc(F)cn2)=O)C12CCC2 C1(F)(C(=O)OC)CC(C(=O)NCC2CC2CNC(=O)C(=O)NCC2CC2)C1 N1(C(CC2CC(=O)NCC2)=O)CC2(CCC(NC(=O)CCc3ncc[nH]3)CC2)C1 c1(OC)ccc2cnc(N(c3ncnc4cc[nH]c34)C3CNCC3O)nc2c1 C1(OCCC)CCCN(c2nnc(C3CCOC3)n2Cc2csc(CC)n2)C1 C(=O)(C1=CC(C)(C)C1)NC1C(CC(N2CC=CC(OC)C2)=O)C(O)C1 C1(N(C)C)(C(=O)NC2CCC(NC(=O)Cc3cc(C4CC4)on3)C2)CCCSC1 N1(C(=O)Nc2cocc2Br)CCCC(n2cc(C(c3ccccc3)O)nn2)CC1 C(=O)(CCN(OC)C(=O)c1coc(C(N)=O)c1)NCCC(CCC#C)O Cc1ccn(C(C)C(=O)N(C(c2ccccc2)CNC(C2(C)CC2)=O)C)n1 C1(C(=O)NCC(C(=O)NC2CC(OC)C2)OC)CCC2(CCC2)C1 C1(C(C)(O)CNC(=O)CCc2ccncc2)CCN(C(=O)CSCC(N)=O)CC1 C#Cc1ccc(C(=O)NCCCCC(CO)NC(=O)C(COC)OC)nc1 C1(Nc2nccc(CC(=O)OC)n2)CS(=O)(=O)CC1NC(c1c(C)coc1C)=O C(C(C)C(C)(C)C)C(=O)Oc1cc(C(C(=O)NC)N(CC)CC2CCCO2)no1 C1(C)(CCNC(CC=C(C)C)=O)CCN(C(=O)CC2CCCNC2)C1 C(=O)(CCP(C)(C)=O)NCC(CNC(c1snnc1C1CC1)=O)OC C(CC(C)C)(C(=O)NCCC(C)NC(c1cc(C)c(C(F)F)cn1)=O)OC C(=O)(C1=NOC(CC2(O)COC2)C1)N1CC(O)(CNC(c2c(C)nsc2C)=O)C1 c1(C(=O)NCCNC(C(c2cscn2)N(C)C)=O)nn(C)c2c1CCCC2 c1(CN(C(c2ccc(-c3cnn(C4CCCC4)c3)cn2)=O)CCO)cc(Cl)c(Br)s1 C#Cc1cn(C)nc1C(=O)NC1CCC(C)(CNC(c2ccnc(Cl)c2O)=O)C1 C1(C(=O)NCCN(C(c2cc(C)c(C)o2)=O)C(C)C)CC2(CCCCC2)S1(=O)=O C(=O)(C(O)CCCNC(C1CCCCC(=O)N1)=O)N(CCNC(C)=O)C C1(CNC(c2cc(CC)[nH]n2)=O)CCCCCN1C(=O)Cc1cc(C)cc(F)c1 C1(NC(C2CC(C#N)(OC)C2)=O)CCN(C(c2cc(N(C)C)ccn2)=O)C(C)C1 c1(NC(C2(C)CN(Cc3c(C)nccc3)C2)=O)cccn2cncc12 CCS(=O)CC(=O)NCC(C1CCN(C(c2ccnn2CC(F)(F)F)=O)CC1)C CN1CCC(C(N2CC(NC(c3cc(C(F)F)n(C)n3)=O)C(O)C2)=O)CC1 Cc1ccsc1C1CC1NC(C1CCCN1C(=O)NC1(c2ccccc2)CC1)=O c1(OC)c(C)cc(NC(C2CCCCN2C(=O)Cc2cc(C)n(C)n2)=O)cc1C n1(CCOC)c2nnc1C(OC)C1CCCN2C1.c1(C(=O)NC(C)C)nccs1 C1(NC(CCC#CC)=O)CC2CCC(C1)N2C(C1CCN(C)C1)=O N1(c2cc(NC(C(CCC)C)C)nc(C(C)C)n2)CCn2cnnc2C1 C1(CNC(C2C(=C)CC2)=O)C(C)CCCN1C(c1ccn(CCC)n1)=O c1(C(N2CC3C(CNC(=O)CC45CC(C4)C5)(C3)C2)=O)coc2c1C(=O)NCCC2 C(C(C)CC(=O)NCc1cn(C2CC2)cn1)NC(c1c(CC)ncs1)=O c1(CCCC)ncc(C(=O)Nc2ccc(=O)n(Cc3ccccc3Cl)c2)c(C)n1 CN1CCN(C(C2(OC3CC3)CC2)=O)CC1C(=O)NC1CCCCNC1=O CC1(C)CCC(CCNC(N2CCC(NC(c3ccc(Cl)cc3)=O)CC2)=O)O1 c1(OCC)c(C(=O)NC2CCOC(CNC(=O)Cc3cnns3)C2)cccc1F C1(NC(c2cc3ccc(O)nc3s2)=O)CN(C(=O)CC=C(Cl)Cl)C2(CCOC2)C1 c1(CNC(c2n(C3(C)CC3)nnn2)CCC2CCCOC2)ccc(C)c(F)c1F C(=O)(CCCC(=O)NC1CN(C(C2CC(O)CN2C(N)=O)=O)CC1O)NCC CCC(CCC(=O)NC1CCCC1CN=[N+]=[N-])NC(C1(C#N)CC1(C)C)=O c1(C(N2CC(NC(CCCOC(C)C)=O)C(F)CC2)=O)cc2n(n1)CCCN2 C=CCCC(C)(C)C(=O)N(C(C)C(=O)NCC1(CO)CCOC1)C1CC1 C1(c2n(C)c(N3CCC(C)(C4CC4)C3)nn2)CCC2(CCC2)CC1 C(=O)(C1=NOC(C(C)(C)C)C1)N1CC(CN(C)C(C2(O)CCSCC2)=O)C1 C12(C(=O)NC(C)COCC3CC3)CC(NC(c3ccnnc3)=O)(C1)C2 C1(N(c2ccc(C)c(O)c2)C(c2ccc(O)nn2)=O)CCCC12CCNCC2 C1(C(=O)NC2CC3(CC(NC(C(CC)OC)=O)C3)C2)CC2C=CCC(C1)C2 C#CC(CO)(CO)NC(C1CC(N(C)C(C2COCC(C)O2)=O)C1)=O c1(C(N2CC(C)C(C(=O)NCc3cccc(F)c3)CC2)=O)cc2ccccn2c1 N1(C(C2(CCC)CC2)=O)CCC2(NC(c3cc(C)n(C4CC4)n3)=O)CC2C1 CC1CCCN(C(C2(NC(c3nc(Cl)cs3)=O)CC(F)(F)C2)=O)C1C N1(C(C(=O)NCCCCCCOC)=O)CCc2c(CCSC(C)=O)cccc2C1 CC1(C)CC(C)(CNC(C2CC(O)C2)=O)CN1C(c1sccc1CC#N)=O CC1(C)CCN(C(C2CC(=O)C23CCCC3)=O)CC1.C(C)(C)(C)O N1(C(C(CC(C)C)OC)=O)CCC(NC(=O)CCC(C)(C)F)C12CCC2 c1(CC(=O)NC(c2ccco2)CC)c(C)nn(C(F)F)c1C Cc1nnc2cnc(C(=O)NC3CC(NC(=O)CC4CCN(C)C4)C3)cn12 N1(C(C2C(NC(C(CC(CC)C)C)=O)CCC2)=O)CCC2CN(C)CC2C1 C1(CNC(=O)CCC2CCCCO2)(NC(c2ccncc2F)=O)CCCCC1 C1(C(=O)NCC(=O)NCC(=O)OC)CC(=O)N(C)C1c1cnn(C)c1C C1(COCCOC)CCN(N2CCC(N3CCCC3C)CC2)CC1 N1(C(C2(C(F)F)CC(=C)C2)=O)CC(NC(=O)Cn2nc(C)c(Cl)c2C)CC(C)(C)C1 C1(CNC(C2CC(=C)C2)=O)(NC(c2csc(C(F)F)c2)=O)CCCCC1 c1(C(N2CCCC(C)(O)C2)=O)cc(O)nc2c1CN(C(C1C=CCS1)=O)CC2 O=C1NC(=O)C(CC(N2CC3CC2C3C(=O)NOCC2CCCC2)=O)N1 CC1(C)CCC(C(=O)NCCC2(O)CN(C(=O)CNC(=O)C3CC3)C2)C1 N1(C(c2cc(OC)c(Br)cc2)C(=O)NC2CCCC2)CC=CCC12CCCCC2 N1(c2n(CC3(C(C)(F)F)CCOCC3)nnn2)CCc2cc(O)nnc2C1 c1(C(N2CCC(C(N)=O)CC2)C(=O)NC(C(=O)OC)C)ccc2n[nH]cc2c1 C(=O)(C(C)CC(F)(F)F)N1CCC(C(C)(C)C)(CNC(CNC(C=C)=O)=O)C1 C1(C(=O)OC)CC(n2cc(C3(C)COC3)nn2)CN1C(=O)Cc1ccno1 CC1CCN(C(=O)Cc2cc(C3CC3)no2)CC1N(C(=O)CCc1nccs1)C C(=O)(C(C)P(C)(C)=O)NCCC(C)N(C)C(c1ccc(CN(C)C)cc1)=O C1(CC(N2C(NCCn3c(=O)cc(C)nc3)CCC2)=O)CCC2(CCNCC2)O1 c1(N2CCC(c3ccc(C#C)cc3)CC2)ccc2nc(Br)nn2n1 C(=O)(C(CO)C(C)(C)C)NCCC(CCNC(c1nc(C)oc1)=O)C C1(NC(C(=O)N(C(C)CS(C)=O)C)=O)CCCCC(P(C)(C)=O)C1 c1(C(=O)NCc2occ(C(=O)NCC=CCCOC)n2)nnc(O)nc1O N1(C(c2scc(OC)c2)=O)CC2(NC(=O)CN3CC4CC4C3)CC1(COC)C2 C=C=C(C)CC(=O)N1CC(CCNC(c2cnc(-c3ccccc3OC)[nH]2)=O)C1 Cc1cc(F)cnc1C(=O)NC(C1CCCC1)CNC(=O)CN1CCCCC1=O c1(C(N2CCCC(C)(CNC(C3(CF)CCC3)=O)C2)=O)cc(Cl)c(O)c(Cl)c1 N1(C(c2cccc(C)c2F)=O)C2CCC1CN(C(=O)Cc1cnn(C3CC3)c1)C2 C1(NC(CC(C)F)=O)CCC(CN(C)C(c2cccc(Cl)c2)=O)CC1 Cc1ccc(C(C)Oc2ccsn2)cc1.C(=O)(CC(C)(C)N(C(=O)CO)C)NC1CC1 C(CC)(CC(=O)N(C)Cc1cnc(C)cn1)NC(c1c(CC)cc[nH]1)=O c1(C(N2CCN(C(CC3CC(=C)C3)=O)CC2CCO)=O)ncn2ccccc12 C1(C(NOC(CC)C)=O)(NC(C2CCOC(C)C2)=O)CCCCC1 c1(C(C)C)cc(C(=O)N(C)CCNC(c2ccnc(CO)c2)=O)c(C(C)C)[nH]1 N1(C(c2[nH]nc(OC)c2Cl)=O)CC(NC(c2cnc(O)c(OC)c2)=O)CC(O)C1 c1(OC)ccc(F)c(NC2CC(C)N(C(=O)OC(C)(C)C)C2)c1 C1(NC(C(C)(C)C)=O)CN(Cc2ccccc2C(C)(C)C)CC1(F)F C1(C)(CN(C(c2cc(C)on2)=O)C)CCCC1NC(=O)C=CSc1nc[nH]n1 C1(C(C)C)CN(C(=O)CNC=O)CCCN1C(c1cccc(C2CC2(F)F)c1)=O C1(C=O)CC2(CCC2O)C1.N1(C(=O)C=CCF)CCCC(N(CCO)NC2CC2)C1 C1(CNC(C2C(CC)C2)=O)COC(C)(C)CN1C(=O)C=Cc1ccc(=N)[nH]c1C c1(N2CCC(NC(C(C(C)C)NC(N)=O)=O)C2C)nc(C#N)c(Cl)s1 O=C(C1=COCCC1)NC1(CNC(=O)C(C2CC2)C2CC2)CC2CCC1C2 C(=O)(CS(=O)(=O)CCOC)N1CC(CNC(COC(CC)C)=O)OCC1 c1(CCC(N2CCCCC(NC(C(F)=CC)=O)C2)=O)csc2ccccc12 N1(C(CNC(c2ccccc2)=O)=O)CCCCCC(Nc2cc(F)ncn2)C1 c1(CSC)cccc(N2CCCC(C(=O)NC(c3nc(=N)s[nH]3)C3CC3)C2)n1 N1(C(C2CC=C(C)CC2)=O)CC2CCC1CN2C(c1cc(C)ns1)=O N1(CC(=O)N(CC(CC)NC(C(C=C=C)C)=O)CC)C(=O)c2cccnc2C1=O N1(C(c2cc(OC)no2)=O)CC(CNC(c2cc(C3CC3)no2)=O)C(C)C1 C1(CC(=O)NC2(C#C)CC2)CCCN1C(c1ncccn1)=O CCCCCC(C)CC(=O)N1CC(C(=O)NC2CCC2(C)C)C(F)(F)C1 c1(-c2cnc(C(=O)NCc3c(OC)n(C)nc3)nc2)ccc(SC)cc1F Cc1cnn2c1CN(C(=O)C(CC(C)C)NC(=O)CSC1CC1)CC2 C1(NC(c2c(C)ncc(Cl)c2)=O)COC2(C1)CN(C(c1ncccc1Cl)=O)C2 Cn1cc2ccc(C(=O)NCC3(F)CC(NC(=O)C=CC4CCCO4)C3)cc2n1 C(=O)(C(CN(C)C)CC)NC(CCC)CNC(=O)CCN1CCOC1=O N1(C(C(CC(C)C)OC)=O)CCC(NC(c2cnc3[nH]cnc3c2)=O)C(C)(C)C1 C12(CNC(C3N(C)CCC3)=O)CCCCC1N(c1ccc(S(C)(=O)=O)cn1)CC2 N1(C(C(CCCNC(=O)CCC2CC2)O)=O)CCC(O)(C2CC2)CC1 C#Cc1cn(C)nc1C(N1CCN(C(=O)C(C)(C)C)CC1c1nccn1C)=O C1(C(=O)NCC2C3CN(C(c4n(CCC)ncc4)=O)CC32)CCCCC12CCC2 C#CCC(C)C(=O)NCCC1CCCN(C(C2CCC2(C)C)=O)C1 N1(C(c2cc3cscc3s2)=O)CCCC(C2CN(c3ncc(Br)cn3)C2)C1 c1(OCC)cccc(NC(=O)C(C)N(C(=O)CC2CSC2)C2CC2)c1 CCC(O)C(C)C(=O)NCC1(C(C)(C)C)CCN(C(=O)CC(C)(C)C)C1 N12CCCCC1C2=O.c1(CC(C)C)ncc(Cn2cc(CCNC(N)=O)nn2)[nH]1 Cn1c(=N)[nH]c2cc(C(N3CCC(NC(=O)CCn4ccnn4)C3)=O)ccc12 C(CC(C)C(=O)NCC=CCC(=O)NCC1(C)CCCC1)OC N1(C(c2cccc(=O)o2)=O)CC(C2CN(C(=O)C(c3ccccc3)C3CC3)C2)C1 C(CN=c1[nH]c2c(c(=NCCF)[nH]1)SCC2)N1C(CC)CCC1 c1(C(N2CC(C(C)NC(c3nccnc3N)=O)C2)=O)ccc(F)cc1Cl C(C)(CCI)(c1nnnn1C1CCCCC1)C(c1cccs1)=O.CCCC(C)N c1(C(=O)NCC(CC(C)C)NC(=O)C(C)C(F)(F)F)ccc(C(C)C)nc1O N1(C(C2(NC(C)=O)CCCC2)=O)C2CCC1CN(C(=O)CN(C)C(C)C)CC2 C(=O)(C1=CCC(NC(=O)CCS(C)(=O)=O)C1)NCC1C(C)C1C C1(C(C)(C)C)CCCN1C(=O)Cc1cnn(Cc2nc[nH]n2)c1 CC1(C)COC(C)(C(=O)Nc2ncnc(-c3ccccc3)n2)CO1 c1(COC)cc(C(=O)NCC(C)CNC(=O)Cc2csc(C)n2)n[nH]1 C(CC(F)F)(C(=O)N)N(C(c1c(NC)scn1)=O)C.C1(CO)(CO)CCN(C)C1 N1(C(C=CC)=O)CCCCC1C1(NC(C2(C)C=CCCC2)=O)CC1 C1(Cc2ccc(CNC(C3CN(OC(C)C)CC3CN)=O)o2)CCC(C2CC2)C1 Cn1cnc(C=CC(N2CCCC(CNC(C3CC3Br)=O)C2)=O)c1 c1(CC(=O)NC2CC(C)N(CC3CCS(=O)(=O)CC3)CC2)cn2c(n1)CCCC2 C(C(C(=O)N1CC(C#N)C1)C(C)(C)C)NC(c1c(C)cncc1C)=O N1(C(CN(C(C)=O)C)=O)Cc2ccccc2C(NC(=O)Cc2cnoc2)C1 N1(C(C=CCOC)=O)CC2CCN(C(=O)Cc3ccc(Br)c(Cl)c3)C2C1 c1(C(CCC)=O)csc(NC(=O)OC(C)(C)C)n1.C(=O)(C)NCCNC(C1CC1)=O c1(OC)ccc(Cl)c(C)c1C(=O)NCC1(F)CC(NC(=O)CC2(C)CCCO2)C1 CC1CN(C(=O)C#CC2CC2)CC1(C)CNC(=O)CN1C(=O)CCC1=O C1(C(=O)NCC2C(CC(=O)N(CCCO)C)C2)C2CC3C(C2=O)C13 CCCC(CNC(=O)Cc1n[nH]c(C)n1)C(=O)NC1(C)CCC(C)C1 CCC(C)(C#N)C(=O)N(CCCNC(=O)CCN1CCCCC1=O)C1CC1 CC1(C)CN(C2(c3ccccc3)CCC2)CC1C.C(C(=O)NCCOCO)C1CC1 C(=O)(C1Cc2ccccc21)NCCCN(C(CC(CC)OC)=O)CCO C1(CNC(CSC)=O)CC2(C1)CN(C(=O)CC1CCCC(F)(F)C1)C2 C1(CC)CN(C(=O)CC(C(F)F)NC(c2csc(C)n2)=O)CCCO1 c1(C(N2CC(NC(c3ccnc4ccsc34)=O)C2)=O)ccc2c(c1)SCCN2 c1(Cc2ccc(C(C)(C)C(=O)OC3C=CS(=O)(=O)C3)cc2)ccc(F)cc1F C1(CNC(c2c(SC)scc2)=O)CCN(C(=O)C(C)n2cccc2)CC1C C(C1CCC(C)CC1)=C(C)C(=O)N(CC(C)NC(c1cc(Br)c[nH]1)=O)C C(=O)(C(C)(C)C(C)NC(c1ccnnc1O)=O)NC(c1c(C)cccc1)C N1(CC(C)NC(=O)C=CC2CCC2)CCN(C(=O)CCC2CCC(C)O2)CC1 N1(CC(=O)Nc2cccc(F)c2Cl)CC2COCC2(CO)C1 CC(c1ccsc1)=CC(N1CCCC1C(C)(C)NC(=O)CC(O)C1CCCC1)=O N1(C(C2(C(C)(F)F)CC2)=O)CC2CC(NC(=O)Cc3cnccn3)C2C1 C1(O)(CNC(C2C=CCN(C(CN(C)CC)=O)C2)=O)CCC(C)(C)C1 C1(C(=O)NC2CN(C(c3cc(CC)ncc3)=O)CC(C)C2)CCn2nccc2C1 N#Cc1ccccc1C(N1CCCOC(CCNC(=O)CC(F)F)C1)=O C12(C(=O)NCC(CO)NC(=O)C(F)(F)c3ccccn3)C3CCC(CC13)C2(F)F c1(C(N(C(C)CNC(=O)C(C)(C)F)CC)=O)nc(C(C)C)ncc1Cl CC1=C(C(=O)N2CC3C(CC(=O)N(C(C)CC(C)C)C)C3C2)CCCO1 CC(C)P(=O)(CC(=O)N1CCC(NC(c2coc3c2C(=O)NCC3)=O)C1)C(C)C C1(C(=O)NCC(N2CC(C)(C(N)=O)C2)=O)CCCCC1F C1(N(C(c2c(C)csc2)=O)C)CN(C(c2c(Br)noc2C)=O)CC1F C1(F)(CNC(C(CC)n2cccn2)=O)CCC(CNC(=O)C(C)(C)F)CC1 N1(C(C2C(C)(NC(=O)CCC(N)=O)CCCC2)=O)C2CCC1CC(O)C2 N1(C(C(C(C)CNC(=O)CCCCCF)F)=O)Cc2cnn(C)c2C1 Cc1cc(C(=O)NC(C)CCNC(c2ccc(OCF)cc2)=O)c(N)cc1F C=CCCCC(=O)N1CCCC(C(C)(C)C(=O)NCC2(CCOC)CC2)C1 C1(CNC(C(n2ncc(C)c2)C)=O)CN(C(C2(P(C)(C)=O)CC2)=O)CC1(C)C C1(O)(CCNC(C2(C)CC(=C)C2)=O)CCCN(C(=O)C(C)C(C)(F)F)C1 N1(C(CNC(C(C)(C)n2cc(C(O)C3CC3)nn2)=O)=O)CCc2ccc(O)cc2C1 N1(C(c2c(C)cncc2)=O)CCCC12CCN(C(C1CCN(C)C1)=O)C2 C(CC(C)C(=O)NCc1ccc(C(=O)N(C(C)CC(C)C)C)nc1)OC C1(NC(C(C)NC(=O)NC)=O)CCC2CN(C(=O)C3=CCCCCC3)CC2C1 N1(C(C2C(C)CC(=O)N2)=O)CCCC2(C1)CN(C(C1CN(S(C)(=O)=O)C1)=O)C2 Cc1c(C(=O)NCC2CC(C)N(C(=O)CC3CCS(=O)(=O)C3)C2)sc2cncn12 c1(C(=O)NC2CC(NC(C3CC=C(C)CC3)=O)C(O)C2)c(C)nn2ccccc12 C#Cc1cn(C)nc1C(=O)NC1CCC(CCNC(=O)CN2CCC(O)CC2)C1 C#Cc1ccc(C(N2CC(CC(=O)NC3CC3)CC2(C)C)=O)cc1 CN1CC2C(C(=O)N(C(C)(C(=O)N3CC(OC(=N)O)C3)C3CC3)C)C2C1 c1(OC)cccc(C)c1C(N1CC(CNC(C2CC2(F)F)=O)C(O)C1)=O c1(CN2CC(C(=O)NCCOc3c(C)cccc3)SCC2)cccc(C#N)c1 c1(C(=O)NCC2(NC(C(C)NC(N)=O)=O)CCCCC2)ccc2nccn2n1 c1(C(N(C(C)CCNC(C2C3CCCCCC23)=O)C)=O)ccc2oc(=N)[nH]c2c1 C1(C)(CC)C=C(C(=O)N2CC(O)(CN(C)C(c3ncc(N)cc3Cl)=O)C2)C1 c1(CCNC(=O)CCC2CCN(C(=O)Cn3cnnc3)C2)ccncc1F O=C1NCCc2c(C(=O)NC3CCCC(CNC(C45CC(C4)C5)=O)C3)cncc21 C12(CNC(c3ccsn3)=O)CCCC1N(C(=O)CCC(F)F)CC2 C(=O)(C#CC1(C)CCCO1)N1CCCC(CNC(C(C(C)C)NC=O)=O)(CO)C1 C=CCC(CNC(C1(CN(C)C)CC1)=O)C(=O)NCC(O)C(C)C c1(C(=O)NC(CN(C(C(C)OCC)=O)CC)C)cc2n(n1)CC(F)C2 N1(C(c2c(OC)noc2C)=O)CC(NC(=O)Cn2cnnc2)CC(C)(C)C1 c1(CN2CCCC(NC(=O)NCc3cc(C)oc3)C2)ccc(C(F)(F)F)cc1 C(CCC(C(=O)Nc1c(C)cccc1C)N1CCCC1CC1CC1)OCC=C C1(C(=O)NC23CC(F)(C2)C3)CCCN1NC(=O)C12CCCC1C2 C1(NC(COCCC=C)=O)C=CCN(C(C23COC(CO)(C2)C3)=O)C1.OCC CS(=O)c1nc(Nc2cccc(OCc3noc(C4CC4)n3)c2)c(Br)cn1 C1(O)(C(C)NC(=O)COCC2CCOC2)CN(C(c2ncnn2C)=O)C1 N(C1CCCn2ncnc21)C(C(CC1CCC1)NC(C1N(CC)CCC1)=O)=O CCCCC(CC)CC(=O)NCC1CC2CC2N1C(C1CS(=O)(=O)C1)=O Cc1cc(C(N2CC(C)(NC(=O)CC(O)C3CCCC3)C2)=O)ns1 C1(CNC(c2ccn(CCF)n2)=O)(NC(C2CC3(CSC3)C2)=O)CCCCC1 C1(C(=O)OCC)(NC(=O)NCc2ccc(C)c(C)c2Br)CCC(F)(F)CC1 C1(NC(c2c(C)cccn2)=O)CC(F)(F)CC1NC(c1nsnc1O)=O c1(C(=O)NCCCCNC(C(C2CCC(=O)N2C)C)=O)cccnc1N C(c1cc(F)cc(F)c1)=CC(=O)NC(CC1CN(C(C(CSC)(C)C)=O)C1)C c1(C(=O)NCCC(CCNC(c2cccc(COC)n2)=O)C)cccn(C)c1=O c1(CC)ccc(CC)c(CNC(c2ccc(C(=O)OC)o2)=O)c1 Nc1cc(C(N2CCN(C(=O)CN3CC4CC4C3)C3CC23)=O)cc(F)c1Br C1(CC)CC(C)CN(C(=O)C(C2CCN(C(=O)CCOCC(F)F)C2)F)C1 c1(CC(C)(C)O)ccc(NC(=O)Cc2csc(Cl)c2)cc1 N1(C(c2cc(SC)oc2)=O)CC(C)OC2(CCN(C(c3cnn(CO)c3)=O)C2)C1 C(=O)(C(C)(C)C(C)(F)F)N(C)CC1CCC(CNC(C2CC2(C)Br)=O)CC1 C1(CCC)COCCC1NC(=O)C(C1(O)CN(C(=O)CNc2ccccn2)C1)F C(C(C)CC(=O)NC1CC1O)OC.C1(C(=O)O)CCN(C)C1 Cc1nccc(C(N2CC=CC(NC(c3nc(C4CC4)cs3)=O)C2)=O)c1N C1(C2CCC2)(C(=O)NC(C(C)(C)C)CNC(=O)CCc2ccc[nH]2)CC1(F)F CC(C)(C)CCC(F)C(=O)N1CC2(CCCCN2C(=O)Cc2cnns2)C1 C(=O)(C(C)(C)C(C)(C)C)NCCC(CNC(C1OCCC1(C)C)=O)OC N1(C(c2cc(C)nn2C)=O)CC(CNC(C2(C(F)F)CC(=O)C2)=O)OC(C)(C)C1 C1(NC(=O)C=Cc2ccccc2)CCCCN(C(=O)CN2CCCCCC2)CC1 C1(C(=O)OC)(N(C(c2cn(C3CC(C(=O)O)C3)nn2)(C)C)C)CCOC1 c1(OC)nc(=NC(C)c2nc(O)n[nH]2)[nH]cc1Br Cc1cc(C(=O)NCCN(C)CCNC(=O)C2=CCCC2)nn1C(C1CC1)C1CC1 C1(NC(C(CC=C)CC)=O)CC2CCC1CN(C(C1CCO1)=O)C2 CCCCC(CNC(C1CC1C(=O)OC)=O)NC(=O)C(Cc1ccccc1C)CC CC1CCC1C(=O)N(C1(CC(=O)N(C)CC2CC2(F)F)CC1)C N1(CC)CCCc2cc(CNC(=NCC3CCOCC3)NC3CC3C)ccc21 n1(C(C)C)ccc(C(N2CC(F)(C(=O)NCc3ncco3)C2)=O)n1 C12(CNC(Cn3c(CCC)nnc3S)=O)CCC(CC1)N2C(c1cc(C)no1)=O CC1CN(C(C2CC2C)=O)CCC1CNC(c1ccc(C2CCC2)cc1)=O C(=O)(C1=CCCS1)NC(c1ccccc1)C(C)NC(C1(CCC=C)CC1)=O CC1(C)CC(C(=O)NC2CCC23CN(C(=O)CN2CC4CCC2C4)C3)=NO1 c1(OC)cccc(C=CC(=O)NCC(C)(C(C)C)NC(=O)C(C)C(F)F)c1 C1(C(=O)NC2CC(NC(=O)C=Cc3ccccc3F)C2)CC2(CCOCC2)C1 C12(NC(=O)C=CBr)CCCC1N(C(=O)CCOc1ccc(F)cc1)CCC2 c1(C(N2C(CCNC(C(=O)NCC)=O)CCC2)=O)cc(F)cc(N)c1N c1(C(N2C(CNC(C(CC#C)O)=O)(COC)CCC2)=O)cc2ccncc2[nH]1 c1(CC(=O)NCC2(F)CCC(NC(C(C)OCC)=O)C2)c(C)cccc1C c1(C(=O)NCCCC(C)NC(CC=C)=O)ccc(OC)c(OC)c1Cl N1(C(c2n(CC)ccn2)=O)CCC2(CC1)CC2NC(=O)CC1CCC(=O)NC1=O C1(NC(c2c(C)snc2)=O)CCN(C(=O)CC2CCCC23CC3)CC(C)(C)C1 N1(C(Cc2c(C)cco2)=O)CCCC(NC(=O)CC(=O)NCC(F)(F)F)C1 C(N=c1cc(C2CCCC2)nc(Cl)[nH]1)C1CC(NC(c2cnn(CCO)c2)=O)C1 c1(C(N(CC(CN(C(C(C(CC)C)OC)=O)C)O)C)=O)nc2ccccc2s1 c1(NC(C2CCN2Cc2ccc(Br)nc2Br)=O)cnc2cc[nH]c2c1 Cc1[nH]c2ccccc2c1CC(=O)NC1CC(NCc2cn3cccnc3n2)C1 CC(C)(CNC(=O)CC1CC(O)C1(C)C)CC(=O)Nc1ccc(O)nc1 Cc1noc(C)c1CC(N1CCC(C(=O)NC2(c3cc[nH]n3)CC2)(CF)C1)=O Cc1nc[nH]c1CC(N1CCCC1CNC(=O)Cc1ccnn1C)=O N1(C(c2cc(C(=O)OC)no2)=O)CCC(O)(Cc2nc(C)no2)C1 N1(C(C23N(C(=O)CC4COCCO4)CC(C)(C2)C3)=O)C2CCC1CC(CO)C2 C(=O)(C1c2c[nH]nc2CCC1C)NCCC1CN(C(C(C)=C(C)C)=O)C1 C(=O)(C1CCCc2c1ncn2C)NC(=O)N(C1CC(NC(C)C)C1)C C(=O)(C1CCCc2ccccc21)CN1C(CNC(CCNC(=O)C=CCl)=O)CC1 C1(CO)CC2CC(C1)N(CCc1cn(CCCCCCO)nn1)C2 N1(C(C2(OCC)CCC2)=O)CC=CC(C(=O)NC(CSC)CC)C1 C(=O)(C1CCCn2cnnc21)NC1N(C(C(C)(C)C)=O)C2C(C1)C2 CCC(CC)(CC)C(=O)NCCC1CCCN1C(c1nc(Cl)c(Cl)s1)=O N1(C(C2CC(C)(CC)C2)=O)CCC(C)C(CNC(c2coc(C(C)C)n2)=O)C1 C(=O)(C(F)C(F)(F)F)NCc1ccc(C(C)NC(c2ncn(C(C)C)c2)=O)cc1 N1(C(CC(CC)N(C(=O)Cc2cccs2)C)=O)CCc2nc(C)[nH]c2C1 c1(C(=O)NCC2CC(C)N(C(C3OCCO3)=O)C2)sccc1S(C)(=O)=O C(=O)(C1CCc2nccn21)NCC=CCNC(c1cc(Cl)ns1)=O Cc1ccc(C(N)=O)cc1C(=O)NC1CC(NC(C2C3CCN2CC3)=O)C1 Cc1n[nH]c2cnc(C(N3CCCC34CCN(C(C3COC(C)C3)=O)C4)=O)cc12 C1(C2CN(C(=O)CS(N)(=O)=O)C2)(NC(CN(C)C(=O)C2CC2)=O)CC1 c1(CN(C(=O)C(=O)N(C2CCOCC2)Cc2nccs2)C)c[nH]c2ccccc12 N1(c2c(C)cc(C#N)cn2)CCc2cccc(C(N3CCCC(O)C3)=O)c2C1 C1(C(=O)NCC(CC)(C)CO)CCCCCN1C(=O)CCN(C)C C(=O)(CCCCC(N)=O)NC1CC(CCNC(CC2(C=C)CCC2)=O)C1 c1(CNC(N2CC(N3CCOC3=O)C2)=O)cc(-c2ccccn2)n[nH]1 Cc1nc2cccc(C(=O)N(C3(c4cn(CCO)nn4)CC3)C)n2n1 c1(OCC)ccc(-c2nc(C3CN(C)CCO3)nn2C2CCCCC2)cn1 N1(C(c2n(C)c(C(F)(F)F)cn2)=O)CC2CC(NC(c3nc(=O)n(C)[nH]3)=O)C2C1 C1(C(N(C)Cc2ncco2)=O)CN(C(C2CC2Cl)=O)CCO1 C1(NC(c2c(C)ccn2C)=O)(CNC(=O)CC2CCCC(O)C2)CCCCCC1 C1(NC(C2N(N=O)CCC2)=O)CC2CC1N(C(=O)COc1ccc(F)nc1)C2 N1(C(C2(SC)CCC2)=O)CC2CN(C(c3cccc4nc(C)nn34)=O)CC2(C)C1 c1(C(N2CC(NC(C(C)OCC)=O)C3(C2)CC3)=O)ccc2oncc2c1 N1(C(CC(C=C)(C)O)=O)CC2(C=C(C(=O)N(CCCC(O)CO)C)CO2)C1 N1(NC(C2CC(=C)C2)=O)CCS(=O)(=O)CC1.C12CC1C(=O)NC2 c1(C(=O)NCCN(CCOC)C(c2csnn2)=O)ccc(C)nc1 c1(OC)cc2ccccc2cc1C(=O)OCc1cc(Br)ccc1Cl C1(F)(C(=O)NCC(C2CCCCC2)NC(C2(CC)CCCC2)=O)CC=CCC1 C1(NC(C2C=CCC2)=O)CN(C(=O)CCc2nnc(S)nc2O)CCC1F N1(C(C2C(NC(C3C(C)(C)OCC3)=O)CCCC2)=O)CCN2CC(F)CC2C1 c1(C(N2CC(CCNC(C(C)=C(CC)C)=O)OCC2)=O)cccc(C#N)c1Br CC1=CCN(C(C2CC(C)N2C(=O)C=Cc2cscn2)=O)CC1 N1(CCC(=O)NC2CCC(CNC(c3ccc(C)s3)=O)C2)CCCCC1=O C12(NC(c3ncoc3C3CC3)=O)CCCC1N(C(=O)COc1cccnc1)CC2 N1(C(CSCC)=O)CC2(COC(CNC(c3cn(C)nc3C3CCOC3)=O)C2)C1 N1(C(C(COCC)NC(CC(OCC)OC)=O)=O)CC2(CCCO2)C1 c1(CNC(COCC)=O)ncoc1C1CN(C(=O)CSC)C1 Cc1nn(CCCNC(=O)C(n2cc(-c3cccc(F)c3C)nn2)C)c(C)c1C C#CCC(C(=O)N1CCC(CCC(=O)NCC(Cl)Cl)C1)C1CC1 C1(NC(C(CCC)=CCC)=O)CCCN(C(c2cc(C)nn2C)=O)CC1F c1(C(=O)NCc2c(C(=O)NCC34CCCC(CO3)C4)c[nH]n2)cccn2nccc12 c1(C(=O)NC2C(CNC(CC3C(CC(=O)OC)C3)=O)C2)cnc(OCC)c(C)n1 c1(C(=O)OCC)cccnc1NC1CC(C)N(C(=O)COCC2CCOC2)C1 N1(C(c2c(C)c(=O)cc[nH]2)=O)C2CC=C(C(=O)N(CC(C)N(C)C)C)C1CC2 C(=O)(CCC(=O)c1cccc(N)c1)NC(C)(C)CNC(C1(CCF)CC1)=O C1(C(=O)NCC2(O)CN(C(c3ncncc3OC)=O)C2)(COC)CCC(=O)N1 c1(C(N(CCC(C)NC(C2N(CC)CCCC2)=O)C)=O)nc(C)[nH]c2nccc1-2 c1(C(=O)NCC(CC=C)NC(c2csc(-c3ncc[nH]3)n2)=O)cnc(N)cn1 C(C(C)(Cn1cc(COc2ccc(N)cc2)nn1)CO)OC C1(CC=C)(C(=O)NC(CN(C)C)CC)CCN(C(C2CCC=CCC2)=O)C1 C12(CC(=O)OC(C)(C)C)CCC(CC1)OC2.n12nnnc1SC(=O)C2 c1(C(N2CC(C)C(NC(=O)C(C3CC3)C3CC3)C2)=O)ccc2nccn2c1 N1(C(CCC(=O)OCCC(C)C)=O)C2CCC1CN(C(C13CC(C)C1C3)=O)CC2 CCC(CC)(CC)NC(=O)CCN(C(=O)CC1CC(C)(C)CO1)CCO c1(CN2CCC(NC(C(C)O)=O)C2)cccc(Cl)c1F C(=O)(C(CC(=C)C)NC(C1CCCOCC1)=O)NCC(C=C)(C)C C1(C)(CC)C=C(C(=O)N(C(C)CN(C)C(c2sc(C)c(Br)c2C)=O)C)C1 c1(C(c2ncoc2-c2cccc(F)c2)CC)cnn(C(C)C(F)(F)F)c1C C1(N(C(c2ncn(CC)c2)=O)CCO)CCN(C(=O)Cc2ccsn2)CC1 C1(CC=C)(NC(=O)C=Cc2ccc(C)s2)CCCN(C(c2ccc(N)cn2)=O)C1 C1CCCC(=O)N(C(=O)Cc2ccc(Cl)cc2)C(CCl)C2(C(Cl)(C(=O)OC)C2)C(=O)O1 Cc1noc(C)c1CC(=O)NC(CCC1CC1)C(=O)NC1CN(C2CCC2)C1 C(=O)(C#CC1CCCC1)NC(C(=O)NC1(CCC)CC1)CCCOC c1(C(N2CC3CC3(C(=O)Nc3nc4sccc4s3)C2)=O)cc(O)nc(Cl)c1 C(=O)(C1=CCCOCC1)NCc1c(NC(=O)OC(C)(C)C)nccc1 C1(C(=O)NCC(C(=O)NCCC2=CCOCC2)N(C)C)CC2COCC2C1 c1(C(=O)NCCN(C(=O)CN2CCSCC2)C)ccc(OC(F)(F)F)cn1 c1(CC(N2CC(C)CC(NC(C(CC)SC)=O)C2)=O)cccc2sccc12 n1(CC(C)C)ncc(C(N2CCC(C)(NC(C3CC(F)C3)=O)C2)=O)c1C1CC1 Nc1cc(F)cnc1C(N1CCCCC(CNC(=O)CC2(C#N)CC2)C1)=O C1(c2cn(-c3c(OC)scc3)nn2)CN(C(c2ncccc2OCC)=O)CCO1 C1(NC(COc2c(C)cccc2)=O)CCN(C(C2C3CC4C(C3)C24)=O)C1(C)C N1(C(C(C=CCCC)O)=O)CCN(C)CC1CNC(C1CC=CCC1)=O C(C(CC(F)(F)F)NC(C1(O)CCSC1)=O)NC(COC(CC)CC)=O c1(C(N2CC(OCC(=O)NCC3C4CCCC34)C2)=O)cnc(S)nc1 C1(C(=O)NC(c2ccccc2Cl)CC)CC(C)CCN1C(=O)CCC(=O)OC C1(NC(C(C)NC(=O)NC)=O)CCN(C(c2ccn(C)c2C2CCC2)=O)C(C)C1 O=C1NCCN2CCN(C(C3CCCCC3(F)F)=O)CC12 CC1CC(C)(C(C)NC(C2CN(Cc3nccs3)C2)=O)C1 C1(C(N(CCOCCC(=O)NC(CC)C(=O)OC)C)=O)CCC(C)=C(C)C1 C1(NC(C(OC)OC)=O)CN(C(c2cc(Br)cs2)=O)C2(CCCC2)C1 Cc1cc(C)c(C(=O)NCC2CC3CCC2N(C(=O)C(O)C(F)F)C3)cc1C C1(C(=O)OC)CCCCC(NC(=O)NC2CCC(OC)(OC)CC2)C1 c1(NC(C2(F)CCN(C(C3(C)CCCC3)=O)C2)=O)cc(F)ccc1F c1(C(=O)NCC2N(C(CC3ON=C(C)C3)=O)CCC2C)n[nH]c2c1CCCCC2 Cn1nccc1CCC(N1CCCC1CN(C(=O)COc1cccnc1)C1CC1)=O c1(CONC(C(CC)n2nnc(-c3cccc(C)c3)n2)=O)ccc2c(c1)CCC2 N1(C(c2cc(OC)ncc2)=O)CC2CCN(C(=O)C(C)(C)O)C2C1 c1(CC(N2CC(OC)C(NC(C3(N(C)C)CCCC3)=O)C2)=O)ccc(C)nc1Cl C(=O)(C(O)C1CCCC1)N(CC(C)NC(=O)COC(F)F)CC C1(N(C(=O)Cc2cnoc2)CC#C)CCN(C(=O)C=Cc2cnc[nH]2)CC1 N1(C(CCC(=C)Br)=O)CCC2(CCN(C(=O)CCOCC)C2)C1 C(=O)(C#CC1CCCCO1)NCC1CC(C)(C)CN1C(=O)CC1CCC(O)C1 c1(CC)nn(C)c(Cl)c1C(=O)NC1C2CN(C(=O)CCC3CCOCC3)CC12 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C(N1CC(CN(C)C)C1)=O)C1CC1 C1(O)(C(N2CCC(CN(C(c3cc(C)sn3)=O)C)C2)=O)CCC(C)(C)CC1 c1(C(=O)NCC(c2ccc(F)cc2)OC)cc2c(N)cccc2s1 c1(Cc2onc(C(C)NC(C34CC(C(=O)O)(CO3)C4)=O)n2)cccc(OC)c1 N#CC1(C(=O)NC2COCCC2NC(c2cc(Cl)ccn2)=O)CCSCC1 c1(C(N(C(C)CNC(=O)C(C)NC(=O)CC(F)(F)F)CC)=O)cn2ccnc2s1 CN1Cc2ccccc2C(NC(=O)NCC=Cc2ccc(Br)cc2)C1 c1(C(=O)NC(C2CCN(C(CCC(=C)Br)=O)C2)(C)C)ccc([N+](=O)[O-])cn1 c1(C(=O)NC2(CF)CCN(C(CCC)=O)C2)ccc(P(C)(C)=O)s1 c1(C(=O)NCCN(C(=O)C(C)Cc2ccccc2Cl)C(C)C)cc(C#N)no1 C1(c2cn(CC3CNC(=O)O3)nn2)(NC(C=CC=CCC)=O)CCOC1 C1(CNC(C2CC(C)OC2)=O)CN(C(=O)C2=CCSC2)CCCO1 c1(OC)ccc(CC(=O)N(CCCCCNC(C2CCOC2C)=O)C)nc1 C1(COC)(CNC(=O)C(=Cc2cscn2)F)CCN(C(c2ccoc2Cl)=O)C1 c1(C(=O)NC2CC(C(C)(C)O)C2)cccnc1CNC(=O)C(C1CC1)C1CC1 Cc1cc(NC(C2CC3CC3N2Cc2cccc(CO)c2)=O)cnc1C N1(C(C2C(C(C)O)C2)=O)CCCC(NC(=O)Cc2cccs2)C1C C1(C(N2CC(NC(C3(CC)CC3)=O)C(OC)C2)=O)CN2CCN1C(C)C2 c1(C(=O)NCCOC2CCN(C(c3cn(C)c(O)n3)=O)C2)ccc(F)c(F)c1F Cc1cc(I)ccc1C(=O)NCC1COCCN1C(c1cccc(Cl)c1Cl)=O CC(C)C(CC(=O)N1CCC(N(C)C(C2SCCS2)=O)CC1)c1ccon1 c1(OC(C)C)ccc(NC(=O)N(C(CO)CO)Cc2ccccn2)cc1C#N c1(-c2n(C3C(C)OCC3)ccn2)ccc2[nH]ncc2c1 c1(C(=O)NC2C(NC(c3n[nH]c(C)c3Cl)=O)C2)c[nH]c2c(Cl)cccc12 C(=O)(C1=NN(CCO)C(=O)CC1)NCC1C(NC(C(CC)CC)=O)CCC1 N(C(=NCc1cccc(N(C)C)c1)NC1CN(C)CC1O)C(c1ccccc1)C N1(C(c2ccc(C)cc2)=O)CCCC2(C1)CN(C(c1cc(C3CC3)[nH]n1)=O)C2 C(=O)(C(C)(CNC(C1CCOC1C)=O)CC)N1CC(=CCC)C1 C(C(CC1CCCC1)C(=O)NCCCC(C)(F)F)NC(C1C(C(C)C)CCO1)=O N1(C(CC2CC(C(=O)OC)C2)=O)CCC(C)(C)C1C(=O)NCC(C)(COC)CC C1(CNC(=O)CSc2n[nH]c(O)n2)C2CCC(C2)N1C(=O)Cn1cncn1 N1(C(c2c(C)nn(-c3cnn(C)c3)n2)=O)CCCC(NC(=O)CC(C)CF)C1C N1(CC(=O)NCc2ccc(C(C)N)cc2)CCCCS1(=O)=O O=C(CC=C(Cl)Cl)N1CC2CC1(C(=O)NC1CSC1)C2 C1(C(N2CC(F)(CC)C2)=O)CC(F)(F)CN1C(=O)Cc1ccn(C)n1 c1(CN2CC(C(=O)Nc3nc(O)cc(OC)n3)OCC2)c(Cl)ccc(F)c1F N1(C(C2CC(=C)C2)=O)CCCCC1CCN(C)C=CCCC=CC(=O)O C1(F)(C(=O)NCC2(CO)CC(C)(C)C2)CCCN(C(=O)CCC2CCCO2)C1 C(C(C)(CNC(=O)CCCC1(NC(=O)CN2CC(C)(C)C2)CCC1)CO)OC c1(-c2cc(C)sn2)nc(-c2cccc(Cl)n2)nn1C1CCC1 c1(-c2ccc(NC(=O)Nc3nccc(OCC)n3)nc2)ccc2cncn2c1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(C(N2C(C)CC2)=O)CC12CCC2 Cc1ccc(C(N2CC3(CNC(=O)C(C)(C)C4CC4)CCC2CC3)=O)c(Cl)c1Cl Cc1cc(CNC(=O)C(=O)N(C)Cc2sccc2Cl)n(C)n1 N1(C(C#CC(C)(C)C)=O)CCCC1C1CCCN1C(=O)CCN1CCOCC1 Cc1ccc(-c2nc(C(=O)NC(C)C(C)NC(=O)C(C)(C)O)cs2)c(C)c1 c1(N2C(COCC)CCC2)nnc(-c2cccnc2)n1Cc1cncc(Br)c1 c1(C(N2CC(COC)(CNC(c3csnn3)=O)C2)=O)nnc(O)nc1O C1(NC(=O)CC2CCCOC2)CC2(C1)CC(CNC(C1(CO)CCCO1)=O)C2 N1(C(CCc2c(C)noc2)=O)CCCC(C)(NC(=O)C(C)Cc2cnco2)C1 N1(CC)CC(C(=O)NCC2CC3CC3N2C(=O)CCN(C)CCOC)CCC1=O Cc1cc(C)c2c(c1)C(N(C(=O)Nc1ccc(F)cn1)C1CC1)CCCO2 N1(C(CC(C=C)CC)=O)CCC2CCN(C(c3cn(C)nc3C(C)(F)F)=O)C2C1 c1(OC)cc(C(N2CCC(NC(=O)C(=O)NC3CC3)C2C)=O)ccc1OC(C)C C12(NC(Cc3ccc(C)c(Cl)c3)=O)CCCC1N(c1cncc(Cl)n1)CC2 C(=O)(CCCS(N)(=O)=O)N(CC(O)CN(C(=O)CC1C=CCCC1)C)C C1(OC)CC2CCC1CC2C(=O)NC(C)CN(C)C(C1CC(=O)NC1(C)C)=O C(=O)(C1=CCC(F)(F)CC1)OC(C)C(c1ccc2c(c1)OCO2)=O c1(C(=O)NC2CCC(NC(C(CO)N(C)C)=O)C2)cnc(Br)c(F)c1 N1(C(C2CN(C)C2)=O)CC(NC(C2CC3C(C2)C3(F)F)=O)CC(F)(F)C1 c1(C(=O)NCC=CCNC(CN(C)C(c2ccco2)=O)=O)ncc(F)cc1F O=C(C1=CCC(F)(F)CC1)NCCC1(O)CCN(C(=O)COCC2CC2)CC1 N1(CC(N2CC3CCC2(CNC(C2(O)CCC2)=O)C3)=O)Cc2ccccc2C1=O C(=O)(CC(C)CC(F)(F)F)N(CC(C)(C)CNC(c1ccnc(C)n1)=O)CC c1(CC)ccc(F)cc1NC(=O)CC(C)(C)NC(=O)CN(C1CCC1)C C1(NC(CC=C)=O)CC2CCC1N2C(=O)Cc1ccn(CC(F)(F)F)n1 C1(O)(CNC(=O)NC2CC(CF)C2)CCNC1 c1(OC)ccc(CN(C)C(C2CCN2C(=O)CC2CCCCO2)=O)cc1 C#CC1C(C(N2CC3CC3(CNC(c3ccc(C4CC4)cc3)=O)C2)=O)C1(C)C c1ccccc1.C(C(=O)NN(C)C(=O)OC(C)(C)C)N(C)CC1(CO)CC1 N1(C(CSCC#C)=O)CCN(C(c2cc(O)ncn2)=O)C2CS(=O)(=O)CC12 CC1CCC(NC(c2cccnc2C2CC2)=O)CN1C(C1C2CCCCC12)=O C#CC#CC(C)(C)NC(C1CN(C(C2CCC(OC)C2)=O)CC1CC)=O C1(NC(=O)CCc2ccsc2)CC2CCC1C(NC(=O)CSC1CCCC1)C2 N#CC1CN(c2nnc(C3CC4CCC3CC4)n2CCO)CCN1C1CC1 CC1=NOC(CC(=O)NCc2ccsc2C(=O)NOCC2(F)CCC2)C1 C1(N(C(CC(C)SC)=O)CCO)CCN(C(=O)CSCC(F)(F)F)CC1 C1(COC)CN(C(=O)C(F)C2CC(NC(=O)C=CC3CCCCC3)C2)C1(C)C N1(C(CNC(=O)NC)=O)CCCC(C)C1CCNC(c1nc(C(C)(F)F)cs1)=O C=C(C)CN=c1[nH]c(=NCCn2ccccc2=O)c2sccc2[nH]1 C=Cn1nccc1C(=O)NCC(C1CCC1)NC(=O)C(C)CC1CCCCC1 c1(OC)cc(NCC2CCCN2C(c2ccc(CN=[N+]=[N-])o2)=O)ncn1 N1(C(C(C2N(C(CC(COC)(C)C)=O)CCC2)(C)C)=O)CC2CCC(C1)C(=O)O2 c1(C(=O)NC2CCN(C)CC2)ccc2nccn2c1 CC1(C)CCOC(CC(=O)NCC(C)(C)NC(c2ccncc2Br)=O)C1 c1(CN2CCC(CNC(c3cc(C(C)(C)C)ncc3)=O)C2)cc(O)ccc1Cl C(=O)(CCCCNC(C1OCCC1C)=O)NC(COCC)(C)C C(CC(C(=O)N1CCOC(CCF)C1)NC(=O)CC1(CS(C)(=O)=O)CC1)SC CC(C)CC(O)CC(=O)NC1CCCN(C(=O)CNc2ccccc2C(N)=O)C1 C1(C(N(C(C)CNC(c2ccc(CN=[N+]=[N-])o2)=O)C)=O)CCCCN1CC(F)F C(=O)(C(C(C)C)C(C)C)NC1C(C(N(CC(C)(C)C)CCC#C)=O)CCCC1 CC(C)CCCCCC(=O)N1C2CCC1CC(CNC(c1cnn(C)c1F)=O)C2 c1(C(=O)O)ccccc1.C(=O)(NNC(=O)C1COCCO1)N1CCCC1 c1(CC)ccnc(-c2nc(CCc3ccccc3)nn2-c2ncnn2C)n1 C(CC(=O)NCCSCC(C)C)(C(F)(F)F)NC(C)=O.C1C(=O)NCCCO1 Cc1nc(C)c(C(N2CC(NC(=O)Cc3ccc(C(C)C)cc3)C(F)C2)=O)s1 n1(CC(N2CC(OC)C(NC(C3CC(C(F)(F)F)C3)=O)C2)=O)nc(C)c(C)c1C c1(CN2C(C(=O)Nc3nc(C)nc(Cl)c3)CC(C)C2)ccc(C)c(C#N)c1 N1(C(C2(C(=O)NC)CCC2)=O)CC2=C(C1)CN(C(C1(C)CC1(F)F)=O)C2 N1(C(CC2N(CC)CCOC2)=O)CC=C(CCNC(C2CCSC(C)C2)=O)CC1 CCC(C)(CNC(=O)C(C)SC)NCCSc1ccccc1 N1(C(C2CCN(CC(C)C)CC2)=O)CC2(CCN(C(=O)CC3CS(=O)(=O)C3)C2)C1 C(=O)(C1CCOc2ccccc21)NC1C2OCC(NC(=O)COC3CCC3)(C2)C1 CC(C)CCC(=O)NCc1cc[nH]c1C(=O)N(CC(N)=O)CC(C)C c1(C(N2CC(NC(C3(CCCF)CC3)=O)C(C(F)F)C2)=O)nccc2cc[nH]c12 N1(C(C(C=C)c2ccccc2)=O)CCC(CO)(Nc2ncnc(C(C)(C)C)n2)CC1 C(=O)(C(C)CC(C)(F)F)NCC(C)NC(=O)CN(C)C c1(C(=O)NCC(CO)NC(CC(CN(C)C)O)=O)cc(Cl)ccc1O N1(C(C(C(=O)NC)(C)C)=O)CCC(C2CC2)(NC(C2CCCN(C)C2)=O)C1 N1(C(C2N(C(=O)OC(C)C)CCC2)=O)CC2CC1C2NC(=O)C(C)(F)F N1(C(C(C)=CC)=O)CCn2ncc(CN(C(=O)CCNC(C)=O)C)c2C1 c1(C(C(=O)OC(C)(C)C)N(CCN=[N+]=[N-])CCOC)nc(C(=O)OCC)n(C)n1 N1(C(c2c(CC)nccn2)=O)CCCC(C)(NC(C2CCC(C)(CC)O2)=O)C1 c1(C(=O)NC(C)CNC(C2(CO)COC2)=O)cc2cc(Cl)c(Cl)cc2[nH]1 C#CC1CCN(C(C2CCCC(NC(c3[nH]ccc3COC)=O)C2)=O)C1 N1(C(C(=C)C(F)(F)F)=O)CC2(CCOCC2C(N2CC(SCC)C2)=O)C1 c1(C(C(=O)Nc2ccc(F)cc2)N(CCC)C2CC2)cnc(C)c(C)c1 CCC(F)(F)C(C)(C)CN1CCCC1Cc1ccc(C#N)cc1 c1(C(N2C(CNC(C3CC(=C)C3)=O)C(C)CC2)=O)cc(F)c2nc(C)cn2c1 C1(COC)(NC(=O)C(COC)OC)CCN(C(c2ccccn2)=O)C1 C1(NC(c2cncc(C)c2)=O)COC2(CCN(C(=O)CC3(O)CCCC3)C2)C1 c1(C(=O)NCC(N(C(C(C)CO)=O)C)C2CC2)cn(C)nc1C1CC1 CC1CCCN(C(=O)N(C(c2nc(-c3cccnc3)no2)C)C2CC2)C1 c1(OC)cncc(Br)c1C(=O)NCCN(C(=O)CCCOC(C)C)C c1(CC(=O)NC(C(CC)C)CO)c(C)cccc1Cl CON1CCC(CC(=O)NCC2(CNC(=O)C(F)CC3CCOCC3)CC2)CC1 CCC(CC(=O)NCC1CCN1C(=O)COC1CCC(C)CC1)SC Fc1cnc(Br)cc1CNCC1CCCCN1c1ccncc1 c1(CCC)cccc(CN=C(NCC(F)COC(C)C)NC(C)C2CC2)c1 CS(=O)(=O)C1CC(C(N2CCN(C(=O)COC3CCC3)CC2CO)=O)C1 CCC(CC(=O)N1CC(C(=O)NC(C2CC(F)(F)C2)C)C(C)C1)C(C)C C1(CNC(C2(CC#C)CCCO2)=O)CN(C(c2nc(C(C)(C)C)no2)=O)CC1C S(=O)(=O)(c1ccc(C(F)(F)F)cc1)N(C(CC(C)C)=O)CC1CCCCN1C(C)C c1(NCC2C(OCC)CC2)cc(=NCC(C)(C)n2ccnc2)[nH]cn1 CC(CC(F)F)C(=O)NCCC1CCN(C(c2cnc(C3CC3)[nH]2)=O)C1 C1(NC(CC2CC(=O)NC2)=O)CC2CC1N(C(=O)CC1CC(F)(F)C1)C2 c1(C(=O)NCC(CC=C)NC(c2ccn(CCO)c2C)=O)cccc2nncn12 Cc1[nH]nc2cc(-c3ncccc3-c3nccn3Cc3ncc(Br)cc3F)ccc12 C1(NC(=O)C(O)CC(F)F)CC2(CCN(C(=O)C(F)=CC3CC3)C2)C1 C1(C(N2CC(C)N(C(C3CN(C)C(=O)N3)=O)CC2)=O)CN=C2N=CNN2C1 Cc1ncc(N)cc1C(=O)NCC1CC(O)CN1C(c1ccc(CO)cc1F)=O c1(Sc2n(C)ccn2)ccccc1NC(c1c[nH]nc1CC#N)=O Cc1ccncc1CC(=O)N(CC(O)CNC(c1ccc(CC2CC2)s1)=O)C c1(CNCCC(=O)Nc2nn[nH]n2)cccc(C(F)C(=O)O)c1 n1(CCCS(C)(=O)=O)c(C(=O)N(CCC#N)C2CC2)cc2ccccc12 C1(NC(c2ccc3oc(O)nc3n2)=O)CCCC12CCN(C(=O)Cn1cccn1)C2 CN=c1ccc(Br)c(C(=O)NC(C)(C)CCNC(=O)C(F)C(C)(C)O)[nH]1 C1(C(=O)NC2(CC)CN(C(c3c(CC)nccc3)=O)C2)CC2CCCCN2C1 C#Cc1ccc(CC(=O)NC2CC3CCC2N3C(=O)CC2(NC(C)=O)CC2)cc1 C(=O)(C(C)(C)CS(N)(=O)=O)NCC1CC(NC(c2c(C)nc(C3CC3)cc2)=O)C1 CCC(N=c1[nH]c(=NCCC(C)OC)c2c(F)cccc2[nH]1)C(C)C Cc1ccc2nc(C(N3CCC(C)(NC(C4CCSCC4)=O)C3)=O)cn2c1 c1(OC)ccc(Cl)c(C(=O)NC2CC(C(=O)NCCOc3cccnc3)C2)c1F C(=O)(C(F)(F)C(F)F)N(CCCCCCNC(C(N1C(=O)CCC1=O)C)=O)C CC(C)(CNC(C1CC(CCO)C1)=O)CC1CN(C(c2snnc2C2CC2)=O)C1 CC1CCN(CCC(=O)NC2CC(NC(=O)C(C)Cc3ccc(F)cc3)C2)CC1 CC1CN(C(=O)C(C)NC(C2(O)CCOCC2)=O)CC(=O)N1 c1(CCOC)nc(C2CN(C)CCO2)nn1C1COC(C)(C)C1 N1(C(c2cc(C)cc(F)c2)=O)CCC2CC1CN2C(c1cc(C#N)cc(C)n1)=O N1(C(c2ccc(CC)[nH]2)=O)CCC(C)C1CNC(=O)C=C1CCCC1 C(=O)(CS(=O)(=O)CCO)NC(C1(O)CCN(C(=O)CC2CCC(F)(F)CC2)C1)C C#CCC(CC#C)C(=O)NCCOCCNC(=O)C(C)(C)C1CC1 C(=O)(C1=C(C)CCC1)N(C)CC1N(C(c2cc(CC(=O)OC)on2)=O)CCCC1 O=C(C1CCCc2nc[nH]c21)NC1CCCCN(C(c2cccc(CO)c2)=O)C1 CCC(C)C1C(=O)N1.n1(CC(=O)OC2CCC(O)C2)nc(-c2cccs2)oc1=O c1(C(=O)NC2CC3CN(C(CC=C(C)C)=O)C2C3)ccc(S(N)(=O)=O)c(C)c1 c1(SC)ccc(N)cc1C(=O)NCCC1(NC(=O)C(O)CN(C)C)CCC1 C=CCC(C)(C)C(=O)N(CCC(=O)N1CC(F)CC1C)OC CC1CN(C(=O)Cc2ccco2)CC1NC(=O)CCc1ccc(O)nc1 C1(COC)(NC(C2CSCCS2)=O)CCCN(C(c2ccc(C3CC3)cc2)=O)C1 CC1(C)CCCN(C(C2COCCN(C(=O)CC34CCCC3C4)C2)=O)CC1 Cc1nc(C2CC2)oc1C(=O)NC1CCCC(CNC(=O)CC(C)N(C)C)C1 c1(C(=O)NCC(CC)NC(=O)CC(O)CN(C)C)cc(N(C)C)ccc1N c1(C(C(=O)NCCOC)N(CC(c2ccccc2)(F)F)C)cnc(C)c(C)c1 N1(C(C(C)C(F)F)=O)CC2CCC1C1CN(C(=O)C=CS(C)=O)CC21 C(=O)(C(CC1CC1)NC(C1(COC)CN(C(C2OCCC2C)=O)C1)=O)NC O=C(C#CC1CCC1)N1CC(OCCNC(C2CCCN2CCCO)=O)C1 N1(CC(=O)OCC(C2CCCC2)C)CC(=O)CC(C)C1 c1(OC)ccc(SCC(=O)NCCC2CC(NC(=O)C3=CCOC3)C2)cc1 C(=O)(CC(C(F)F)n1ccnc1)NC1CC(F)(CNC(CNC=O)=O)C1 C(=O)(CC(F)(F)C(C)C)NCC1C(NC(c2cn(CCCC)nn2)=O)CCC1 c1(C(N2CC(NC(COCCOC)=O)C(C)(C)C2)=O)ccccc1S(=O)(=O)CC Cc1cn2c(CCC(=O)NC3CN(C(=O)C(C)CF)CCC3O)csc2n1 Cc1ccc(C(C)O)cc1NC(=O)NC1CCN(C(C)C)C1=O C(=O)(C(C)N=c1cc[nH]cc1)NCC1CCCN(C(C(C(C)C)(F)F)=O)CC1 c1(C(N2C3CC(C(=O)NC(C#C)(C)C4CCC4)C2CC3)=O)ccc2n[nH]cc2c1 C1(NC(c2cn(CC)nn2)=O)CCC(C(N2CCC2CF)=O)CC1 c1(C(N2CC(C)N(C(c3ccc(F)s3)=O)CC2)=O)coc2c(F)cc(F)cc12 C1(NC(=O)CCCc2ccccc2F)CCN(C(=O)C=Cc2nc[nH]n2)CC1F C=C(C)CC(C(=O)NCc1nnnn1C)NC(c1csnn1)=O C(=O)(CCCC(=O)N1CCCC1(C)CNC(C1CC12CCOCC2)=O)N(C)C c1(NC(C(N2C(Cc3c(C)cccc3)CCC2)=O)=O)cc(Cl)c(C#N)cn1 C=Cc1ccc(C(N2CCCC2C2CCN(C(C3(C)CCC(=O)NC3)=O)C2)=O)cc1 C(c1cscn1)=CC(=O)NCCN(CC(C)O)C(=O)CC1CCCN1C CCN=c1ccc(C(N2CCC(NC(C3CC(=C)C3)=O)C(F)C2)=O)c[nH]1 c1(CC(=O)NC2C(NC(C=CCC)=O)CC2)nocc1C c1(C(=O)NCC(CC=C)NC(C2(CC3CC3)CC2)=O)ccc2c(c1O)CCCC2 CC(CCC(C)(C)C)C(=O)N1CCC2(C(=O)NCC3(CN=[N+]=[N-])CC3)CCCC12 C(=O)(CC(C)CC(F)(F)F)N1CCC(C)C(NC(c2cc(C)cc(Cl)c2)=O)C1C n1(CC)cc(C#N)c(=NC(=O)C2CCN(Cc3c(C)[nH]c4ccccc4c3=O)C2)[nH]1 C(=O)(CC1CCc2ccccc21)N1CC(COC)(CNC(C2(F)CCC2)=O)C1 N1(C(C=COCC)=O)CC(NC(=O)C(N2C(=O)CCC2=O)C)CC(C)C1 C#CC1(NC(C2(F)CCN(C(=O)CN(C(=O)C(C)C)C)C2)=O)CCCOC1 n1(CC)c(C)cc(C(=O)NCC(C2CC2)NC(c2ccc(C)cn2)=O)c1C N1(c2nc(=N)nc(N(CCc3scc(C)n3)C)[nH]2)CCS(=O)(=O)CC(C)C1 c1(C(=O)NCCCCN(C(Cn2ncc(C)c2)=O)C)cccc2ccsc12 Cc1ncnc(N2CCC(NC(=O)Cc3ccoc3)C(C)(C)C2)c1C#N CCC(C(=O)NCc1cc(C(=O)NC2CC(C)(C)OC2(C)C)ccn1)C(F)(F)F c1(C(=O)NC2(CC)CCN(C(C(C=C)(C)C)=O)CC2)cc2c(nc1O)CCSC2 c1(CN(C2CC3CNC2C3)S(=O)(=O)CC2CC2)cccc(F)c1Cl Cc1c(C(=O)NC2CCN(Cc3cc[nH]n3)CC2(C)C)ccc(F)c1[N+](=O)[O-] CCCCS(=O)(=O)CC(=O)NC1CCN(C(=O)C(c2ccccc2)C)CC1CO C(=O)(C1CCCc2cncn21)NCCOCCN(C(=O)CC1(C)CC(F)(F)C1)C c1(OCC)cnc(C(=O)NCC2CCC(NC(C3CCC3C(F)F)=O)CC2)cn1 C(=O)(C(C)(C)CCF)NC1CC(NC(CN(C)C(=O)OC(C)(C)C)=O)C1 C=C(C)CC(C)C(=O)NCC1(NC(C2CC(CC)C2)=O)CCCCCC1 C1(C(N2CCC(NC(c3c(C)ccnc3C)=O)C(F)C2)=O)CC2(COC(=O)N2)C1 CCC1=NOC(C(=O)NC2CC(NC(C3COCCN3C3CCCC3)=O)C2)C1 N1(C(C(C)NC(=O)NCc2cccnc2F)=O)CCCCC1C(N)=O N1(CC)CC(CNC(c2ccccc2OC)c2nnnn2CCOCC)CC1=O C1(F)(C(=O)NCc2nn(C)c(=O)o2)CCCN(C(=O)CC2CC2(C)C)C1 c1(C(=O)NC(C)(CNC(c2ccncc2C2CC2)=O)CO)ccc(F)cc1F c1(C(CC(=O)NC(C2CN(C(c3cnn(C)c3)=O)C2)C)=O)ccc(O)cc1 N1(C(CCC)=O)CCC(CN(C(=O)COc2ccc(Br)cc2)C)CC1 N1(Cc2cccc(OC)c2)CCN(C(c2cc(C)oc(=O)c2)=O)C2(CC2)C1 N1(C(C(C(C)(C)C)SC)=O)CC2(CC(NC(=O)C=Cc3cnccc3C)CO2)C1 C1(C(N2CC3C(CNC(Cc4cc(C)sc4C)=O)(C3)C2)=O)CC(C2CC2)=NO1 C1(OC)(CO)CCC(C)(C)CC1.C12CC3(C1)CN(C3)C(=O)N2 N1(C(C2(NC(=O)C(F)C3CCCC3)CCSC2)=O)CCOC2CCC12 C1(C(N(CC(C)(C)NC(=O)C=Cc2ccccc2)C)=O)CNC(=O)CC1(C)C C=CCCCC(=O)N1CC2C(CNC(c3ccccc3NS(=O)(=O)CC)=O)C2C1 C(=O)(C1=CCCOC1)N1C(CNC(c2n(C)cnn2)=O)CCC1 CC1(C(=O)N2CC(NC(C34CC(F)(C3)C4)=O)C(O)C2)CCCc2ccccc21 c1(C(=O)NC2CC(F)(CNC(C3(C)CCCO3)=O)C2)ccnc(C(N)=O)c1 Cc1ccc(CN2CCC(OC3CCN(C(=O)C(O)CCNC)CC3)C2)c(C)c1 C(=O)(CCCCCCCC(=O)N(CCNC(=O)CC1=CCCC1)C1CC1)OC C(CCCCCCCO)=CC(C1CN2CCCC1C2)=O C=CCN(OC)C(=O)CC(C)CNC(=O)C=C(C)C c1(NC(C(C)Cc2ccccc2)=O)cnc(F)c(Cl)c1 c1(C(=O)NC(C2CN(c3nc(C)nc(O)c3)C2)C)ccc2c(c1)C(=O)NCC2 c1(CC(=O)N(C(C)C)CCN(C)C(c2ccoc2Cl)=O)cccnc1Cl C(=O)(C(C)C(O)C(C)C)N1CC(CC(=O)NCC2(CCOC)CC2)C(C)C1 N1(C(CN(C(CN2CCC(C)CC2)=O)C)=O)CCC(N=[N+]=[N-])CC1 CC(C)C(C)C(C)CC(=O)NC1CC2(CCN(C(=O)COC3CCC3)C2)C1 C1(CC)CN(C(=O)CC(C)(C)CC)CCN1C(c1cccn1CC)=O N1(C(c2cccc(C)c2Cl)=O)C2CCC1CN(C(c1cn(C)cn1)=O)C2 CC(C(=O)N1CCSCC1CCNC(c1csc(Cl)c1Cl)=O)C(C)S(C)(=O)=O CCS(=O)(=O)CC(=O)N1CCCCC(CNC(c2sc(C)cc2C)=O)C1 c1(C(=O)NC(CC2CN(C(CCCN(C(=O)OCC)C)=O)C2)C)cn(C)c(O)n1 c1(C(NOC(C(=O)OC)C)=O)cncc(CNC(=O)Cn2cncn2)c1 Cc1cc(C(=O)NC(CNC(=O)C(C)(C)c2cnco2)C(C)(C)C)ccc1F c1(N(CCNC(C2CC3CC3CC2C)=O)CC)ncc2c(ncn2C)n1 c1(NC(C2CC(NC(=O)OC(C)(C)C)C2)=O)nc2ccc3scnc3c2s1 C1(F)(CNC(c2c(C(C)C)cco2)=O)CCC(NC(=O)CCn2ccnc2)C1 O=S(=O)(C1CC2(CC(F)C2)C1)NCc1ccc(O)cc1 c1(C(N2CC(NC(=O)CC3CC4(CCC4)C3)(CF)C2)=O)cccnc1S Cc1cc(C(C)C(N2CCCC2C2(NC(C3CC(O)CN3C)=O)CC2)=O)c(C)o1 C1(NC(Cn2c(C)ccn2)=O)(CNC(=O)C=C2CCN(C)CC2)CCCCC1 C1(NC(C2(CC=C)CCCN2C(=O)C=CC(F)F)=O)CCC(C#N)CC1 c1(CN2CCN(c3cncc(OC)n3)CC2)ccc(CC(F)(F)F)c(F)c1 N1(C(C(C)(CCc2ccccc2)C(=O)O)=O)CCCNC(=O)C1C(F)(F)F c1(C(=O)NC(CC)C(=O)NCCN(C2CC2)CC)cnc(O)c(C)c1 N1(C(C(=O)NCCOCC)C)CC2CC(NC(c3cc4ccsc4s3)=O)CC1C2 c1(NC(=O)NCCc2cncc(OC)c2)ccc(F)cc1OCCC(C)C C(=O)(CC(C)C=C)NCC(CC=C)NC(c1cc(C)nn1C(F)F)=O c1(CCC(=O)NCCC(C)Nc2ncc(C)c(C)n2)ccc(C#N)cc1F c1(C(=O)NCC(C)(CC)NC(C2C(=C)CC2)=O)cncc(OC)c1C c1(C(=O)NCC2OCCCN(C(C3C(C=C)C3)=O)C2)cc(C)ccc1NCC C=C(C)C(O)CC(=O)NC1(C)CCC(NC(c2cncs2)=O)CC1 c1(CC(C(=O)N(CCN(C(=O)CCCN(C)C)C(C)C)C)C)cccc(Cl)c1 c1(C(=O)NC2C(NC(c3csc(CC(F)(F)F)n3)=O)CCC2)ccncc1O N1(C(C2(C=C)CCC2)=O)CCCC(N(CCO)C(c2ccoc2Cl)=O)C1 C1(COC)CN(C(=O)CC(C)(C)O)CCN1C(=O)Cc1cc(Cl)sc1Cl CC(CC(=O)NCC1CC(F)CN1C(c1cnc(C(F)(F)F)nc1)=O)P(C)(C)=O CCC(C)(C)C(O)C(=O)N1CCCC1C1CCN(C(=O)Cc2cnsc2)C1 N1(C(CCCNC(=O)OC)=O)CCC(O)CC1C(=O)NC1CCC(CO)C1 C1(NC(c2c(C)cc[nH]2)=O)C2CCC(C2)C1C(=O)NC1(CCO)CCOC1 C1(C(N(CC(C)OC)CC)=O)(NC(c2ccc(C(F)F)o2)=O)CCSC1 c1(CNC(=O)Nc2c(OC)c(Cl)ncn2)cc(Cl)c2ccncc2n1 C1(C(=O)NC2C(C)NC(=O)CC2)CC12CCOc1ccc(F)cc12 c1(C(=O)NC(C)CCCCNC(=O)Cc2cc[nH]c2)ccccc1N=[N+]=[N-] N#CC1(C(N2CC3CC3(CN3CCCC3)C2)=O)CCOC1.C12(CCCC1)C(=O)N2 Cc1ccc(F)c(C(=O)N(CCCNC(=O)Cc2nc(C)sc2C)C2CC2)n1 N1(C(C=C(CCC)C)=O)CCN(C(=O)COC(C)C)C2COCC12 c1(CC(=O)NC2CCC(C)(NC(C(CCC)OCC)=O)C2)ccc2nsnc2c1 N(C(=NCCCC1CCOC1)N1CCC2(CCCCCC2)C1)CC(CC)C(C)C C1(C(=O)Nc2c(CC)cc(O)cc2)CC2CC1CN(C(C1(C)CCOCC1)=O)C2 C(=O)(C1CCc2ccccc21)NCCCO.CC1(C)C2C1CNC2=O c1(N2CC(CN(C(C3(COC)CCCO3)=O)C)OCC2)ccc2nnnn2n1 N1(C(C2(CC#C)CCCO2)=O)CCC(NC(=O)Cc2cccc(OC)c2)C(O)C1 C(C(C)CC(=O)NC1C2CC1N(C(=O)C(n1nnnc1C(C)(C)C)C)C2)OC O=C(CC1=CCOCC1)NCC1(F)CCCN(C(c2ccc(C(F)F)o2)=O)C1 Cc1ccc(C2CC2C(N2CC(CNC(=O)CC(O)c3ccccc3)C2)=O)nc1 C1(NC(C(N2CC3CC3C2)C)=O)CCC(NC(c2cc(C(F)F)nn2C)=O)CC1 CN1CCC(C(N2CCCC(N(C(=O)CCN(C)CCO)CCO)C2)=O)CC1 c1(N2C(C)CN(C(=O)C3=CCSC3)CC(C)C2)nc2c(cc1Cl)C(=O)OC2 c1(C(N2CC3C(NC(=O)C(c4cc(F)ccc4F)O)C3C2)=O)cc(Cl)ncc1O c1(OCC)ccc(S(=O)(=O)NCCCC2COCCO2)cc1CC N1(Cc2ccn(CCC)n2)CCCC(C(=O)NC2CCNC2=O)CC1 C(CCCCC(=O)NC(C1(O)CCCCC1)C(N1CCN(CC)C(C)C1)=O)=CC C12(NCc3ccc(C#C)cc3)CCC(C(=O)NCc3cncs3)(CC1)CC2 Cc1ccc(C)c(C(N2CC3CC3(NC(=O)CSc3cn[nH]c3)C2)=O)c1O C1(NC(C(C)(C2(C)CC2)OC)=O)CCCCCC1NC(C1CCC(=O)O1)=O N1(CCF)CCCC(N=c2[nH]c3c(c(=NC4CCCOC4)[nH]2)COC3)C1 c1(C(=O)NC2C(O)CCN(C(C(CCCC)CC)=O)C2)ccc(C)cc1[N+](=O)[O-] c1(C(=O)OC)cc(C(=O)Nc2cn[nH]c2)c[nH]1 N1(C(Cc2cnc(C)[nH]2)=O)CC(NC(c2cncc(CO)c2)=O)CC1(C)C O=C(CC(O)C1CCCC1)NC1CCCC1NC(C12CC(F)(C1)C2)=O c1(C(N2CC(C(=O)Nc3cnc(C)c(Cl)c3)SCC2)=O)c(C)ccc(C)c1O Cc1oc(-c2ccco2)nc1CC(N1CCC(N(C)C(C2OCCC2C)=O)C1)=O Cc1ccc2oc(C(=O)NC(C)(C)CNC(c3cncn3C(C)C)=O)cc2c1 N1(C(c2cc(C)[nH]n2)=O)CC(CNC(=O)C(C2CCOCC2)C)CC1C N1(C(=O)NCc2c(C)cc(C)c(C)c2)CCC(O)CC(C)(C)C1 c1(COC)ccccc1C(N1CC=CC1CNC(c1conc1CC1CC1)=O)=O C(=O)(CS(=O)(=O)CC(C)C)N(CCNC(c1cn(CCOC)nc1)=O)C(C)C C1(NC(CN(C(COCC#C)=O)C(C)C)=O)CCCCC1CCC=C N1(C(c2c(N)csn2)=O)CCC(CC#N)C(F)(F)CC1 c1(N2CCCN(CCC)CC2)nccc(=NC2CCc3ccccc32)[nH]1 c1(C(=O)NCCC2(NC(CSCC=C)=O)CC2)ccncc1SCC C(=O)(C1=CCc2ccccc21)NCCC1(CNC(C2CC(=C)C2)=O)CC1 CC1(CNC(C2CC2(Cl)Cl)=O)CCN(C(=O)C=Cc2cncc(F)c2)CC1 C1(NC(C2C(OCC)C2)=O)COCCN(C(=O)C(C)(C)OC)C1 c1(NC(c2ccccc2)COCCCC)nccc(=NCCc2sccc2Br)[nH]1 c1(-c2ccc(C)cc2)csc(=NCC(C)c2ccc(N(C)C)cc2)[nH]1 c1(CNC(=NCC)NCc2ccnc(C)c2)cc(F)c(OC)c(F)c1 c1(C(=O)NCC(C)(CNC(=O)CCCN2CCCCC2)OC)ccnc(S)c1 C1(NC(C2(OCCOC)CC2)=O)CN(C(=O)CCc2ccncc2)CC1OC N1(C(C2CCCC(C)C2)=O)CCN(CCO)C(C)(C)C1 Cc1nc(C#N)c(NCCC(N2CCC(C)C2CNC(=O)Cc2cnc[nH]2)=O)o1 CC1CCC(NC(=O)C=CC2CCOCC2)CN1C(=O)Cc1csc(Cl)n1 N1(C(CC2N(C)CC=CC2)=O)CC2CC1CN2C(C1CNC(=O)O1)=O C(CCC(C(=O)NCCNC(N)=O)NC(=O)CC1NC(=O)NC1=O)OC c1(C(N2CCC(NC(CC(=O)NCC#C)=O)C2C(C)C)=O)csc2ccccc12 CCC(C#N)C(=O)N1CCCC(C(C)(C)C(=O)NCC(N2CCCCC2)C)C1 N1(CC)CC(CNC(=O)CC2(C)CCN2C(c2ccc(C)n2C)=O)OC1=O CCC(C)C(=O)C(=O)N(CCCNC(C1(CO)CCCO1)=O)CC CCCCC(O)C(=O)NC1CC2CC(NC(=O)COc3ccsn3)CC12 C1(C)(NC(C(CC(F)F)N(C(c2cnc(CC)s2)=O)C)=O)CCCCC1(C)C Cc1nc(=N)[nH]cc1C(=O)NC1CCC(CNC(C2CC(n3cccn3)C2)=O)C1 c1(Cn2c(C)ncc2)ccc(NC(=O)C(=O)NCCCc2ccc(Cl)cc2)cc1 O=C(C1CCCc2n[nH]cc21)N1CCC2(CC1)CN(C(C1CCO1)=O)C2 Cc1cc(N2CCCC(OC(=O)N(C)C)C2)nc(N2CCOC(C)CC2)n1 C(=O)(C1=CCCOCC1)N(CCC(=O)NCc1ccc(F)cn1)C1CC1 C=C(Cl)CCC(=O)NCc1ocnc1Cn1cc(Cn2ccnc2C)nn1 C(=O)(CCCCC1CC1)NC(C)C=CC(=O)NCC1CCC1(F)F c1(CC(N2CC=C(CNC(C3(C)CC3(Cl)Cl)=O)CC2)=O)ccc2nn[nH]c2c1 N1(C(CN2CC(NC(c3c(C)c[nH]c3)=O)C2)=O)CCC(OCC(F)(F)F)CC1 c1(C(=O)NCC(=C2CN(C(C3CCC(C(=O)OC)O3)=O)C2)F)cc(=O)cc[nH]1 Cc1nn(CC(F)F)cc1C(N1CCCC(N(C)C(C2CC2(Cl)Cl)=O)C1)=O N#Cc1cc(Br)cnc1NCC1CCCCN1C(C1CC12CC2)=O C(=O)(C(C)Cn1ccc(C)n1)NC(c1ncccn1)(CC)C N1(C(CC(C(=C)C)OCC)=O)CC2(CCN(C(=O)CN3CCC(O)CC3)C2)C1 N1(C(C(C)Cc2cnc[nH]2)=O)CCN(C(=O)C(C)(C)C2CC2)CC12CC2 C12(CC(=O)NC(C3CCN(C(CC=C(C)C)=O)C3)C)CCC(CC1)C2 CC(C)(CCCNC(C1CCSC1)=O)C(=O)NC1CCOC1C1CC1 C1(C(=O)NC2CCC(CCC(=O)NCCCC3CCCCC3)C2)CC(C2CC2)=NO1 Cc1cc(C(N2CCC(F)(C(=O)NCC3CNC(=O)CO3)C2)=O)cc(C)c1 C1(CNC(CCCCOC)=O)CC12CCN(C(c1ccnnc1O)=O)CC2 c1(CN(C(C(=O)NC2CCOC2)C(C)C2CCOC2)CC)ccc(Br)cc1 N1(C(CCn2ncc(C)c2)=O)CCN(C)C(C(=O)N(C(C)CO)C)C1 Cc1nc2c(o1)CCN(Cc1cc(C)c(C)c(C)c1)C2 N1(CC(=O)Nc2ccc(O)cc2)CCC2CC(C(=O)NCC3CC3(F)F)C2C1 C(C(N=c1nc[nH]n2cccc12)C(C)C)NC(CC1(C=C)CCOCC1)=O C(CCCCC(=O)NCCC1(C)CCN(C(=O)CN2CCC(C)C2)CC1)OCC C1(CNC(=O)NC2CC(=O)N(C3CCCCC3)C2)CNCCC12CCOC2 C(CN=C(NCN1CCCC1=O)N1CCC(Nc2ncccn2)C1)C1C(F)(F)C1 C12(CC)COC(C(=O)NC(C)CCNC(c3csc(CC(C)C)n3)=O)(C1)C2 c1(NC(C2C3CN(C(C=COCC)=O)CC32)=O)ccc(CC)c(CC)c1 c1(CCC)cc(C(=O)NCC(C)N(C)C(C2CSCN2C)=O)ccn1 c1(CCCN(C)CCF)nc(C2CC2)nn1C(C1CCOCC1)C1CCC1 N1(C(C2(NC(C(C)SCCCC)=O)CC(F)C2)=O)CCC(F)CC1 N1(C(c2nc(C)sc2)=O)CCCC(C)(CNC(C2(N3CCOCC3)CCCC2)=O)C1 C1(OCCNC(c2ccnn2CCF)=O)CCN(C(=O)CCCc2cnn[nH]2)C1 C(=O)(C(O)C(C)(C)C)NCCN(C(=O)CC1CC1)C(C)C c1(C(F)(F)F)ccc(OCc2ccccc2)cc1.n12ccnc1CCC2 C(C1=CCCN(C(=O)C(C)c2cc[nH]n2)C1)NC(C(C)CN(C)C)=O N1(C(CCCCCOC)=O)CCC2C(C1)CN2C(=O)C(C)C1CCC1 N1(Cc2ccccc2)CCC(C(F)(F)F)CC1C.C1(CC)(CCl)C2C(C)C1N2 c1(CN(C(CC)CN(c2nnc(C)n2C2CC2)C)C)ccc(S(N)(=O)=O)cc1 N1(C(CC2CC(CC)C2)=O)CCC(C(N2CCC(CCO)CC2)=O)CC1 N1(C(c2cncc(C)c2Cl)=O)CC2CC(NC(c3cnsc3)=O)CC(C2)C1 c1(C(=O)NCCN(CCC)C(C2CN3CCC2C3)=O)ccc(C)c(S(N)(=O)=O)c1 CC(C)(C)C#CC(=O)N1CCC(CCNC(c2cncc(SC(F)(F)F)c2)=O)C1 C(CCCCCCC(=O)N1CCC(C2CC2)C1CNC(c1cnc(Cl)s1)=O)SC Cc1ccc(CN2CCC(C(=O)Nc3cnnc(Cl)c3)CC2)cc1F N1(C(C(CCC)O)=O)CCCC(C)C1CNC(C1CC(C)=NO1)=O N1(C(C2(CSC)CCOCC2)=O)CCCC(NC(C2CC3(CCCC3)C2)=O)CC1 C(CCC(C)NC(C1COC(=O)O1)=O)NC(COCCOCC)=O N1(C(CCN(C)CC)=O)CCN(C(c2ccn(C(F)F)n2)=O)CC1CC(F)(F)F C1(C(C)N)CN(C(=O)C(N2CCCC2c2cccc(Cl)c2)=O)CCO1 CC1(C)C(NC(=O)CCN2CCCC2)CCN1C(C1CCC(=O)O1)=O C(=O)(CCCc1nc(C)no1)N(CC(CC)NC(C1CC(=C2CC2)C1)=O)C CCC(C)(F)C(=O)NCCc1ccc(CNC(=O)C(C)OC2CCOC2)cc1 c1(C(C)NCC2CCN(C)C2C)ccc(F)cc1OC(=O)N(C)C C1(CCOC)(NC(=O)CSc2ccc(C)cc2)CCN(C(=O)C#CC2CC2)C1 N1(C(COCC)=O)CC2(CCCCN(C(c3oc4ccccc4c3CC)=O)C2)C1 c1(C(=O)OC)ccc(CCC(=O)NC2CC(CNC(c3ccn(C4CC4)n3)=O)C2)[nH]1 C1(NC(Cc2ccc(C(C)=O)cc2)=O)CC(F)CN(C(=O)C=Cc2cncs2)C1 N1(C(C(CC=C)OC)=O)CCCC(O)(CCNC(=O)C(C)CSC)C1 c1(C(N(C)C)=O)ccc(C(=O)NCC(O)CCNC(=O)CCNC(=O)CO)cc1 C(=O)(C1=CCC(NC(=O)CCC2CC2(C)C)C1)NC1(CCC)CC1 N1(C(CC(=C=C)C)=O)CC2CCCC(N(C(=O)CN(C(=O)C3CC3)CC)C)C2C1 c1(CNC(=O)Nc2nc(C)c(N(C)C)cc2)ccc2[nH]ncc2c1 c1(CC)nc(C)cc(=NCC2CN(C(=O)CC(C)CC)CC23CCC3)[nH]1 C(=O)(CC1=CCOCC1)NCC(c1ccccc1Br)NC(C(CC)OC)=O Cc1cncc(CCC(N2CCCC2C2(NC(=O)C=CC3CCCC3)CC2)=O)c1 C=CC(CC)CC(=O)NC1CC2(C1)CC(NC(C1C(C(C)=O)C1(C)C)=O)C2 Cc1cc(C(=O)N(C)CC2CCN(C(=O)CC3CCCC(O)C3)CC2)[nH]c1C CO[Si](CCCN1CCC(C)CC1c1ccc(C)o1)OC C1(C)(CNC(C(CC(C)C)C)=O)CC(F)(F)CN1C(=O)CCC1CCC1 c1(SC)ccc(C(=O)NCC2(O)CCN(C(=O)CC3C=NN(C)C3=O)C2)cc1 C(=O)(C(O)CCCNC(=O)CC1C=CCCC1)NCC(CC)C#N N1(C(C2CC(C)(C)OCC2)=O)CCC2(CC1)CC2C(N1CC(C(F)(F)F)C1)=O C12(NC(C(CC)CC)=O)CCCN(C(c3cc(F)ccc3Br)=O)C1C2 N1(C(C(CCCC=C)C)=O)CCC2(CCC(NC(=O)C3=CCSC3)CC2)C1 C12(C(N3C(C)CCC(O)C3)=O)COCC1CN(C(c1cc3n(n1)CCO3)=O)C2 C(=O)(C#CC1CCOC1)NC(CC=C)C(=O)N1CCC(F)(C(N)=O)C1 c1(C(=O)NCC2N(C(CC3ON=C(CC)C3)=O)CC(O)C2)cc2c(C)cccc2o1 C1(OC)CN(C(c2cc(F)n(C)n2)=O)C(C)(CNC(c2cn(CCO)nn2)=O)C1 C1(C(N2CCC(O)(CNC(c3csc(CO)n3)=O)C2)=O)CCCC2(CCC2)C1 c1(C(=O)NCC2C(CNC(CN(CCC)C)=O)C2)ccc(OCC)c(F)c1F c1(C(=O)NC(C2C(C(=O)Nc3ncc(OC)nc3)C2)C)c[nH]c2ccccc12 C(c1ccc(Cl)nc1)=CC(N1CC(CNC(c2c(NC)cnnc2)=O)(OC)C1)=O CC1CCCC(C(N2CCC(OCCCNC(C3(O)CCSC3)=O)CC2)=O)CC1 c1(C(N2CCC(CCNC(Cn3c(=N)[nH]nc3)=O)C2)=O)ccc(O)nn1 C1(NC(C2CCC(CC)O2)=O)C2CCC1N(C(c1ccc(=O)n(C)c1)=O)C2 c1(C(N(C2CCN(C(COCCC=C)=O)C2)C)=O)cc(C)c(CC)nc1O C(=O)(C(O)CC(N)=O)NCc1cc(C(=O)NCC2(COCC)CCC2)n(C)n1 N1(C(c2ncc(C)cn2)=O)CCC(C)C(NC(c2ccc(C(C)C)c(C)c2)=O)C1 N1(C(c2cnc(OC)nc2C)=O)CCC2CN(C(C3CC(SC)C3)=O)CCC12 CCCCCCC(=O)N1CCN(C(C23CC2COC3(C)C)=O)C(C(C)C)C1 c1(NC(C2(CC)CCCO2)=O)cccc(NC(c2cc(F)n(C)n2)=O)c1 Cc1ccn2ncc(C(=O)NCCC34CCC3CN(C(=O)C3=CCSC3)C4)c2c1 c1(OCC(=O)NC2CC(OC)CN(C(C(CSC)C)=O)C2)cccc([N+](=O)[O-])c1 c1(C(=O)NCC2N(C(COC3(C)CCC3)=O)CC2)cnnn1C(C)C1CC1 c1(C(=O)NCC(C(C)(C)C)NC(=O)Cn2cccc2)cc2ccsc2s1 c1(C(N2CCC(NC(CC(C)F)=O)C2C(C)(C)C)=O)ccc2c(c1)OC(C)(C)O2 C12(CNC(C(N3CCC(C)C3)=O)=O)CCC(CC1)N(C(=O)CNC(N)=O)C2 S(=O)(=O)(c1cc(C)ccc1C)NCC(=O)NCCN(C(CC1C(OC)CC1)=O)C C1(CN(CC#C)C(C)C)N(C(=O)C(C)SC(C)C)CCCC1(C)C c1(C(=O)NC2CC3CC(NC(c4cn(CC)nc4)=O)C2C3)nccc2[nH]ccc12 N1(C(CCc2n(C)ncc2)=O)CC(C(N2CC3(CC=CC3)C2)=O)CCC1(C)C C1(Oc2ccnc(C3(C)CC3)n2)CS(=O)(=O)CC1O CC(C)CC(O)C(=O)N(C1CN(C(C2CCC(=O)NC2)=O)CCC1C)C Cc1nc2ccc(C(=O)NCCC3CCCCN3C(C3COCCO3)=O)cc2o1 C1(F)(C(N2CCC(CN(C(c3c(CC)cncc3)=O)C)C2)=O)CCC(C)CC1 c1(OC)nccc(C(N2CCC(NC(c3ccoc3C)=O)C(F)C2)=O)c1F C(=O)(C(C)C(C)C(C)(C)C)NCCC1CN(C(CCc2c(C)n(C)nc2)=O)C1 O=C1CCC(C(N2CC(F)(CNC(C3CCCN3c3cnccn3)=O)C2)=O)CN1 c1(OC)ccc(NC(N2CCCC(OC3COCC3n3ccnn3)C2)=O)cn1 C(=O)(CCCN=[N+]=[N-])NC1C(C)(OCCOC(C2(C(C)(C)O)CCC2)=O)C1 c1(C(N2CC(NC(c3c(C)ccc(Cl)c3)=O)C(O)C2)=O)ccnc2c1CC(=O)N2 N1(C(C(C)c2cccs2)=O)CC(CNC(c2cn(C)cn2)=O)C2(CCOCC2)C1 c1(C(N(C2CCCC(NC(C(C)=C3CC3)=O)C2)C)=O)ccc2sccc2c1 c1(C(=O)NCC2C(NC(C(COC)OC)=O)C2)cc(Cl)c(OC)cc1Cl C1(CCC)CN(C(=O)C2=CCCC2)CCN1C(=O)Cc1csc(S)n1 N#CCCCCC(=O)NCC1CCC(NC(=O)C(F)=CC2CC2)C1 c1(C(N2C(C)CC(CNC(CCCCC)=O)C2)=O)cc(C(F)(F)F)c(C)c(N)c1 C(C1CCN(C(C2CN(C)CCO2)=O)CC1)=CC(=O)N(C(C)CO)C1CC1 CCC(C)CCCC(=O)N1CC2(CCCC2)C1C(=O)NCC12CCC(CO1)C2 N1(C(C(C)(C)OC)=O)CCC(NC(=O)C(C)(Cl)Cl)C(c2ccccc2)CC1 N12CC(C)(CC1(C)C)C(=O)NCCOCC2=O.C1(CNC(=O)NC)CCC1 Cc1cc(C(c2nnnn2CCCF)NCc2cc(Cl)cc(Cl)c2)cc(C)c1Cl c1(CN(CCC)C)ccc(C(=O)NCC2CC2NC(C2CC2NC(C)=O)=O)o1 C1(C(=O)NCC(C)(C)NC(=O)C(F)CC2CCCCC2)CCCN(S(C)(=O)=O)C1 Cc1ccc(C(=O)N(C)CC2(O)CCCN(C(C3CCC(F)CC3)=O)C2)cc1Cl c1(CC)ccc(N)c(C(=O)N(CC(CO)(CO)NC(=O)CN2CC(C)C2)C)c1 c1(CN(C)CC2CCC(C)O2)ccc(CNC(=O)C(C)(C)Cc2cnn[nH]2)cc1 Fc1cc(F)c2[nH]c(=NC3CCCC(CO)C3)[nH]c(=NCc3cncnc3)c2c1 C1(C(N(CCNC(COC)=O)C2CC2)=O)CCN(Cc2cccnc2)CC1 C1(CN(C(CN(CCC)C)=O)C)CCN(C(=O)C(O)CF)CC1 Cc1cnc(C)c(NC(=O)C(=O)Nc2ccccc2N(C)Cc2ccncc2)c1 CCC(C)C(O)CC(=O)N1CCC(CC)(NC(=O)C=CC2(C)COC2)CC1 C1(C(N(CCNC(CC2CCC(C)CC2)=O)C)=O)CCC(N=[N+]=[N-])CC1 Cc1cc(C(=O)N(CC(=O)C(C)C)C(C)C)nn1-c1ccc(C(C)(C)C)cc1 CC1(C)Oc2cccc(C(=O)OCCc3cc(Br)cs3)c2O1 N1(Cc2cn(C)nc2)CC(C2CCCN(C(c3cn(C)c(C(F)F)n3)=O)C2)C1 N1(C(C(CC)SC)=O)CCC(CO)C(NC(c2oc(SC)cc2C)=O)C1 N1(c2snc(CC)n2)CC2CCC(NC(c3c(C)noc3C(F)F)=O)CC2C1 CC(C(=O)N(C)CCN(C)C(c1cc2n(c1)CCSC2)=O)C(F)(F)C(F)F CC1(C2CCCN(Cc3cccc(-c4ccsc4C(=O)O)c3)C2)COC(=O)N1 c1(COC)cccc(C(c2ccccc2Cc2nn[nH]n2)O)c1 C(=O)(C1CCOc2ccccc21)NCC1N(C(c2n(C)cnc2)=O)CCCCC1 CCCC(C(=O)OC)C(=O)NCC1CCC1NC(C1(n2cnnn2)CC1)=O c1(C(=O)NC2CC(c3cn(CC4CC(F)(F)CO4)nn3)C2)nccc(Cl)c1F Cc1noc(C)c1CC(=O)NCCC1CC(NC(=O)C(c2ccc(Cl)cc2)C)C1 c1(NC(C(C2CC(NC(C)=O)C2)F)=O)ccccc1-c1cc[nH]n1 N12CCCC1C2=O.C1(NC(=O)NCC)CSCSC1 N1(C(CC(C=C)C)=O)CCC(C2CC2)(CNC(=O)Cc2cccc(Cl)c2F)C1 C12(CC(=O)NC(CN(C(C(C)SCc3ccccc3)=O)C)C)COC(CF)(C1)C2 C(=O)(C1=CCC(C)CC1)N1CCC(C(C(N2CCCC(C(C)C)CC2)=O)(C)C)C1 C1(C(N2CCC(C(C#C)C)CC2)=O)CCN(C(C2C=CC=CC=C2)=O)C1(C)C c1(C(C(N2CCCC(NC(c3c(CC)occ3)=O)C2)=O)=O)cc(F)cc(Cl)c1 c1(CC(=O)OCC(CCC(=O)NC(C)(C)C)=O)cn2ccsc2n1 Cc1oc(CO)cc1C(N1CC(CNC(=O)Cc2nnc(O)s2)C2CC12)=O C12(COC)CC(C(=O)NC3(C)CCN(C(c4ccsc4C(C)=O)=O)C3)(CO1)C2 CCC(O)C(=O)NC(C(=O)NC(C)Cc1nncn1C)c1ccco1 C1(C(=O)Nc2c(CC)c(C(=O)OC)ccc2)CN(Cc2nnnn2C)CC(F)(F)C1 C1(CS(N)(=O)=O)CCCN1Cc1ccc(-c2ccccn2)o1 N1(C(COCCCOC)=O)CCCC1C1CCCN1C(c1cnc(SC)cn1)=O N1(C(CSCC(=O)OC)=O)CCC2CCCC12CNC(c1cnc(S)[nH]1)=O N1(C(c2ccnn2C2CCCCC2)C(=O)NC(CC)C)CCOCC1C(=O)OC c1(OC)ncc(Cl)c(C(N2CCC(NC(C3CCCC3(C)C)=O)CC2)=O)c1Cl CC1CCN(C(=O)COc2ccsc2)CC1CNC(c1ncn(C)n1)=O c1(CC(C(=O)N(CCN(C(C=C2CCC(C)C2)=O)C)C)=O)cccc(Cl)c1 C1(COC)(NC(C2CNC(=O)C2)=O)CCN(C(c2cc[nH]c(=N)c2)=O)CC1 S(=O)(=O)(c1cnc(NC2CSC2)c(Cl)c1)N1CCC(n2c(=N)nn[nH]2)CC1 O=C(C1=CCCCO1)NC(CCC1CCC1)C(=O)N1CC(N2CCCCC2)C1 C1(NC(C(C)Oc2ccccn2)=O)CC2CN(Cc3cc4n(n3)CCSC4)CC2C1 Cc1nccc(C(=O)NCC(C)(C)CC2CN(C(=O)C(=O)NCC3CC3)C2)c1C C1(NC(C(=O)NC(C)C)=O)CCC(C)N(C(=O)CC2CCC(C)(C)CO2)C1 c1(C(C)NC(C2CC2c2c(F)cccc2F)=O)c(F)ccc(Cl)c1F c1(C(N2CCC3(CC(NC(C45CCC4CC5)=O)C3)C2)=O)cnc2cccnn12 Cc1nc(C)c(C(N2CCC(CO)(NC(=O)CCC3(O)CCC3)CC2)=O)nc1C C(CC(CO)C(C)C)NC(C(C1N(C(C2C(CC)C2)=O)CCC1)(C)C)=O Cc1nc2c([nH]1)C(C(=O)NC1CCCC1NC(=O)CN(C)CCO)CCC2 C1(NC(C2CCOC2)=O)CCN(C(=O)C2=CCCC2)CC12CCC2 N1(C(c2n(C=C)nnc2)=O)CC2CC(C1)C2NC(c1ccc(C=C)cc1)=O c1(C(N2CCCC(CNC(CSCC)=O)C2)=O)cc2ccccn2c1 N1(C(C2(C(=O)OC)CC2C)=O)C2CCC1CN(C(=O)C(c1cc(C)oc1C)C)C2 C1(C(N2C(CCC#C)CCC2)=O)CC(C)CN(C(c2cnsc2)=O)C1 C1(CNC(c2cccc(C)c2)=O)CCCC2CN(C(=O)CC3CCCO3)CC12 N1(C(c2cc(CNC(c3c(C)ccc(C)n3)=O)sc2)=O)CCN(C)C(=O)C1C c1(C(=O)NCC2(F)CC(NC(C(C=C=C)C)=O)C2)cccc(CC)c1F N1(C(C(CC2CN(C(c3c(CC)nns3)=O)C2)F)=O)CC2(C1)CC(C)(F)C2 N1(C(c2c(C)[nH]c(C(=O)OC)c2C)=O)CC2=C(C1)CN(C(=O)C(F)=CC1CC1)C2 C12(NC(CN(CC#C)C(C3CC(N=[N+]=[N-])C3)=O)=O)CCC(CC1)C2(C)C N1(C(c2nc(C)sc2)=O)CC2CC2(C(N2CCOCC2C2CC2)=O)C1 C1(NC(c2cnn(-c3ccccc3)c2Cl)=O)CCCN(C(=O)Cc2cncs2)C1 N1(C(C(CCF)NC(c2ccc(O)nc2)=O)=O)CC2CCC1C(O)C2O c1(C(=O)NCCCC(=O)OC(C(C)(C)SC)=O)ccc(S(C)(=O)=O)cc1[N+](=O)[O-] c1(CC)cncc(CNC(=O)CC2CN(C(=O)Cn3c(C)ccc3C)C2)c1 N1(C(c2scc(OC)c2OC)=O)CC2COCCC2(NC(c2cnc(Cl)s2)=O)C1 C1(NC(C(C#C)(C)C)=O)CCC2CN(C(=O)CC(O)c3ccccc3)CC2C1 C1(NC(c2cccc3nsnc23)=O)CCC2CN(C(C3CCOC3)=O)CC2C1 c1(CN2CCCC(C(=O)Nc3c(C(N)=O)cccc3F)C2)c(O)cc(Br)cc1F C(=O)(C(C)C(C)(C)C)NCC(CCNC(CCCOC(C)C)=O)O C1(NC(C2C=CC(=O)N=N2)=O)CC2(CCN(C(c3cccc(O)c3Cl)=O)CC2)C1 C(=O)(CC(CC)CCCC)NCCC(CNC(C1(C)CC(=C)C1)=O)OC Cc1cc(F)ccc1NC(=O)C(=O)N(C1CC2CNC1C2)CC#N C1(NC(c2scc(C)c2)=O)CC(O)CN(C(=O)C(=O)Nc2ccc(Cl)cc2)C1 C1(C(N(CCC(=O)N(C)CC2(C(C)(C)O)CCC2)CCCO)=O)CCC(=O)C1 c1(CN2C(C(=O)Nc3cnccc3Cl)CC(C)C2)ccc(Br)cc1C(=O)O c1(OC)cccc(Br)c1C(N1C2CCC1C(CNC(=O)CC(F)F)C2)=O C1(C(N(CC(COCC)O)C)=O)CCCC(NC(c2cccnn2)=O)C1 N1(C(c2c(C)n(C)cn2)=O)CC(NC(C2(C(C)(C)C)CCC2)=O)CC(O)C1 CC(C)(C#N)CCCC(=O)NCCCC(O)C(=O)NC1(c2csnn2)CC1 C1(CCNC(C=C(CC)C)=O)CN(C(=O)C(O)CCC(C)C)CCS1(=O)=O c1(C(=O)OCCCOC(c2c(OCC)oc(C)n2)=O)cnc(F)c(F)c1 Cc1ccc(C)c(C(=O)NC2CCOCC2C(=O)NCc2nc(C)c(C)s2)n1 CCC(C(=O)NCC1C(C)CCN1C(c1cc(O)nc(O)c1)=O)C(C)O C(CC(F)F)(C(=O)N(CCCCN(C)C)C)N(C(CC(CC)C1CCC1)=O)C Cn1nc(C(N2CCN(c3ccc(F)cc3)CC2)C(=O)NC[Si](C)(C)C)cc1I N1(C(C=CCOCCOC)=O)CCCC12CCN(C(=O)CS(=O)(=O)C(C)(C)C)C2 C1(CN(C(Cc2c(C)cco2)=O)C)CCCN(C(=O)CCC2CCCO2)C1 n1(CCC)[nH]c(=NC(=O)C(F)(F)C(F)Cl)cc1C c1(C(N2CC(CN(C(c3n[nH]c(C)c3C)=O)C)OCC2)=O)cc2cnccc2[nH]1 c1(C(N2CCN(C(CC=C)=O)CC2)=O)c(-c2ccc(F)cc2)c(C)nn1C C1(CNC(c2cc(C)ncn2)=O)CN(C(=O)CCc2cscn2)CCC12CCC2 C(=O)(C1=C(Cl)CCC(C)C1)N1CC(COC)(NC(C2C3CC4C(C3)C24)=O)C1 CCCC(C)CCCC(=O)N(C1CCCC1)CCNC(c1c[nH]c(=N)cc1C)=O CC(C(=O)NCC(c1ccccc1)NC(c1cnc(C2CC2)[nH]1)=O)C(C)(F)F c1(C(=O)NCC23C(NC(c4c(C)nns4)=O)CC(CC2)C3)ccn2c1CCCC2 CC(C)(C)C1=NOC(C(=O)NCC(O)CCNC(C2CC=CC2)=O)C1 c1(-c2c(C)cc(N(C)Cc3c(F)ccc(C(C)=O)c3)nc2)ccc2c(c1)NCCO2 C1(NC(CC=CC=C)=O)CC(=O)N(C2CN(C(=O)CCc3cnccn3)C2)C1 N1(C(CCC=C)=O)CCN(C(c2cc(OC)c(Cl)cc2Cl)=O)C(C)C1C c1(CCCC(N2C(C(C)NC(C(CC)(C)C)=O)CCCC2)=O)ccc(C)c(C)c1 c1(CC)cc(C)c(C(=O)NC2(CNC(c3cc(C)co3)=O)CCOC2)o1 c1(NC)ccc(Cl)c(C(=O)NCCCN(C)C(C2CCC2F)=O)c1 N1(C(c2cc(C)n(C)n2)=O)CCC2(CCCN2C(c2ccco2)=O)C1 CC(CC(=O)NCC1CCN(C(=O)CSC2CC2)C1)C(=O)c1ccc(Cl)cc1 N1(C(c2ccn(C3CC3)c2)C(=O)NCC)CCC(NC(c2csc(C)n2)=O)CC1 c1(C2N(C(CC3(OCC)CCC3)=O)CCC2)ccccc1Cl.C12CC1NC2=O N1(C(C(CC)C2CCOCC2)=O)CCCC(C2CCN(C(=O)COC3CC3)C2)C1 c1(C(=O)NC2C(NC(c3c[nH]c(=N)s3)=O)CC2)cc(O)nc2ncccc12 c1(C(=O)NC(C2(CNC(c3cc(CCC)on3)=O)CC2)C)nc(C)sc1C c1(C(=O)NCC2CN(C(CC(=O)NC3CC3)=O)CC2O)cnn2ncccc12 C1(NC(C2CCN(C(CCc3cc(C)no3)=O)C2)=O)C2CCCCCC12 C(C)(CN=c1cc(C(=O)OC)nc(Cl)[nH]1)N(C(c1nccc(CC)c1)=O)C c1(OC)cc(CC(C)NC(=O)CCC2CCCNC2)cc(OC)c1OC c1(CC(=O)N(CC(C)O)CCNC(C2C(OC)COC2)=O)c(C)ncnc1C CCCC(CCNC(C1CCN(C(=O)C(CC)OC)C1)=O)C1CC1 CCCC(C)CC(=O)N1CCC(N2CC(C)(CNC(C3CCSC3)=O)C2=O)CC1 C#CC1(CC)COCCN1CC(=O)Nc1cccc(Cl)c1Cl c1(C(=O)NCC2N(C(c3cnn(C(C)C)c3N)=O)CCCC2)ncc(F)cc1F N1(C(c2c(C)nc(OC)s2)=O)CC2CN(C(c3cc(C)n(C)n3)=O)CCC12 N1(C(CC=CCC)=O)Cc2[nH]nc(C(N3CCC(C)(F)C3)=O)c2C1 Cc1cc(Cl)ccc1N(C(C)(C)C(=O)O)C(N1CCN(c2nccn2C)CC1)=O C12(C(N3CC(CNC(c4ccnc(OC)n4)=O)C3)=O)CCC(C)(C(=O)O1)C2(C)C CCC(C)(COCc1ccccc1)C(=O)N1CCC1NC(=O)CC=CC(C)(C)C CC1CN(C(C2CC3(C2)CC(F)C3)=O)CCC1CNC(=O)C(C)(C)C#N C1(NC(C(c2ccc(F)cc2)OC)=O)CCN(C(c2n[nH]c3c2COC3)=O)C1(C)C CCC(C(=O)N1CC(F)CC1CC(=O)NCc1cnc(O)c(F)c1)C(C)(C)CC c1(NC(=O)NC2(c3cccc(Cl)c3)CC2)cccc(F)c1Br N1(C(C(C)NC(c2cscc2Cl)=O)=O)CCC(C2CCC2)CC1 N1(C(=O)NCC(c2ccc(OC)c(OC)c2)C)CCC2(CC1)CN(C)C2 c1(C(C(=O)NCCn2cc(C(C3CCOC3)OC)nn2)CO)ccc(Cl)cc1 C1(NC(=O)CSC(F)F)(CO)CN(C(=O)C=CC2CCCO2)C1 c1(CN(C(=O)C(=O)Nc2ccc(N(C)C)cc2)C)ccccc1-c1ccccc1 c1(SCC(=O)N(CC(C)C)CCO)nc(Cl)c(=O)n(C)c1N N1(C(CCCCC(=O)NC)=O)CC(C2CCCN(C(C3CCNC(=O)C3)=O)C2)C1 C1(C(=O)NC2CCC(CNC(=O)Cn3cncn3)C2)(OCC)CCCCC1 c1(NCC(=O)NC(CCC)C(=O)NC)ccc(Cl)cc1Cl.C1C(=O)N1 c1(N(CCC#C)C)nnc(-c2ccccc2Cl)n1CCN1CCOCC1 CN1CCCC2CN(C(=O)NCCc3csc(C(F)F)n3)CCC12 N1(C(CCOC(C)=O)=O)CCC(O)(CN(C(C2CC2c2ccccc2Cl)=O)CC(C)C)C1 CC1(C)C(CNC(C2CC2C2CC2)=O)CCN1C(=O)CCN1CCCCC1=O O=C(C1=NOC2(CCOC2)C1)NC1CCCC12CN(C(C1CC(=C3CC3)C1)=O)C2 c1(CNC(CSCCCC)=O)cc(C(=O)OC)ccc1NCC N1(C(C2CCC(C(=O)OC)CC2)=O)CC(C(=O)OC)CC(CN)C1 C1(NC(N2CCCC(C(C)N)C2)=O)CCc2nn[nH]c2C1 N1(C(COC(C2C(Cl)(C(=O)OCC)C2)=O)=O)CCC(Cc2ccc(Cl)nc2)CC1 c1(C(N2CCC(NC(CCCc3nc(C)sc3)=O)C2C)=O)ccc([N+](=O)[O-])cc1 C1(NC(CC(CC)C)=O)CCCC(N=c2[nH]c3c(F)cccc3o2)C1 c1(OC)cc(C)c(CNC(=O)N(C)Cc2c(F)cccc2F)cc1OC CC1=C(C)CC(C(=O)NCCCN(C(=O)Cn2ncc(O)nc2=O)C2CC2)CC1 N#Cc1ccc(CC2CC2)nc1N1CCC(NC(=O)CC2CCCNC(=O)C2)C1 C(=O)(C#CC1(C)CCCO1)N(C(C)C(=O)NCC(=C1CCCCC1)F)C1CC1 C1(NC2CN(C(C34CC(CN3)C4)=O)C2)CCCC2CC12 c1(NC(C(=O)Nc2ccc(NC(=O)OC)cc2F)C)c(C)c2cnccn2c1C c1(C(=O)NC2CCN(C(CCN(C)CC)=O)CC2C(C)C)cccc2nn[nH]c12 c1(C(N2CCC(N(C(Cc3n(C)ncc3)=O)CCO)C2)=O)ccc([N+](=O)[O-])[nH]1 N1(C(C2(CCC=C)CC2)=O)CC2(CCC(CNC(=O)CCc3ccccc3)O2)C1 Cc1cccc2oc(=NCCCNC(=O)C(C)CSC(F)(F)F)[nH]c12 c1(OC)ncc(Cl)c(C(=O)N(CC(C)NC(c2c(C)nn(C)c2Cl)=O)C)c1Cl c1(C(=O)NC(c2cc(C)no2)C)cc(C)c(-c2cccs2)s1 N1(C(C(CC)C2CCC(=O)N2)=O)CC2(CCN(C(=O)C3=NOCC3)CC2)C1 C1(CNC(C2ON=C(C)C2)=O)C(C2CC2)CCN1c1ncnc2scnc12 C(C(CNC(=O)Cc1ccsn1)CO)NC(C1CC(SC)C1)=O N1(C(CCCC(C)=O)=O)CCCC2(CCCN2C(=O)C(F)CCC(C)(C)C)C1 C(=O)(CP(C)(C)=O)N1C(C(C)NC(c2ccc(Cn3nnnc3C)s2)=O)CCC1 N1(C(C(CC#C)C)=O)CCC2(CC1)CC(NC(c1nn(CC)cc1[N+](=O)[O-])=O)C2 CN1CCC(c2cn(CC3CCCN(C(c4nccs4)=O)C3)nn2)CC1 c1(CC)cccc(C(=O)NCCC(CNC(=O)CC2CCC3CC23)OC)c1 C1(CC#C)(C(=O)OCC2(O)CCC2)CCC1.C12(CCC1)C(=O)N2 c1(-c2c(C)cccc2)ccn2ncc(C(=O)Nc3cc(Cl)nn4ccnc34)c2c1 N1(C(CC(CC)OC)=O)CC2(C1)CN(C(=O)C(C(C)CC)N(C)C)CCO2 CCC(C)S(=O)(=O)Cc1nnc(N2CCC(c3nc(C)cs3)C2)n1CC1CC1 C1(NC(c2ccc(C)cn2)=O)CCCC12CN(C(C1CC3C(C1)C3(F)F)=O)C2 c1(CN(C)CC2(O)CCCN(C(C3CCCOC3)=O)C2)nc2ccccc2o1 C(CCC)(C(O)C(=O)N1CCCC1CNC(C)=O)NC(C(C=C)O)=O C1(C(C)NC(c2cc(C3CCOCC3)on2)=O)CN(C(=O)C#CC2CC2)CCO1 C1(C)(OC)CN(CC(=O)NCC2(CNC(=O)Cc3nccn3C)CCC2)C1 c1(C(N2C(C)CCC(CNC(C=CC)=O)C2)=O)cc2cncn2c(O)n1 Cc1cc2[nH]c(=O)c(C(N3CCC(CNC(c4n[nH]c(C)c4Cl)=O)C3)=O)cn2n1 CC1CN(C(=O)C#CC(C)(C)O)CCN1C(C1CCOC(C)(C)C1)=O c1(OC)ccc(CN2CCC(CCNC(=O)C(C)(F)F)C2)c(Cl)c1OC c1(CSC)cn(CC(F)CCNC(=O)C(C)(C)Cl)nn1 Cc1cn2cc(C(=O)NCC3CCN(C(=O)Cc4cn[nH]c4)CC3C)sc2n1 C1(C(=O)OC)CCN(C(=O)Cc2sc(COCC(C)C)nc2C)CCC1(F)F CCC(C(=O)N1CC2(CCC2NC(c2cocn2)=O)C1)C(C)(F)F C1(C(C)C)C(NC(=O)C=CC2CCCCC2)CCN1C(C1CC12CC(O)C2)=O c1(C(=O)NCC2CCN2C(=O)C(O)C2CCC2)occ2c1CCCC2 C(=O)(CCCCCF)NC1C=CCC(C(=O)NCC(C)(O)C2CCC2)C1 C1(C(=O)NC(CNC(c2ccc(Cl)cc2F)=O)C2CC2)CC(F)(F)C1(F)F C=CCCC(=O)NC.c1(CCC(=O)NC)nc(-c2nc[nH]n2)no1.C12(CC1)CCC2 c1(C(C)=O)ccc(C(N2CCC(C)C(NC(=O)C(O)C3CC3)C2)=O)c(F)c1 Cc1ccc2nc(C(=O)NCC(CO)NC(c3c(C)cncc3C)=O)cn2c1 c1(CC)nc(N2CCN(C(C3CCCSS3)=O)CC2)cc(C#N)n1 c1(OC)cccc2c1CN(C(=O)C(N1CCC(Nc3ccccc3)C1)=O)CC2 C1(NC(CS(C)(=O)=O)=O)COC2CN(C(=O)CCCCc3ccccc3)CC12 N1(C(c2ccc(OC)c(OC)c2Br)=O)CCCC2(C1)CN(C(C)=O)CCO2 N1(C(C2C(C)(CC)C2)=O)CCCC(C)(C)C1CNC(C1CNC(=O)N1)=O n1(CC(=O)NC2(CN(C(=O)Cc3nnc(O)s3)C)CC2)ncc(C#N)c1N N1(C2CCN(CC)C2=O)CCC2(CCN(C(=O)CC3CC4(CC4)CO3)C2)C1 C1(C(=O)NCC2(C(=O)NC(c3cncs3)C)CC2)CCCN1C1CC1 N1(c2ccnc(N3CC(C)C(O)C(C)C3)n2)CCc2c(CO)nn(C)c2C1 C(=O)(C1=CCSC1)NCCCN(CCCCNC(C1CCC(C)O1)=O)C N1(C(CCCC#C)=O)CCCC2C(CCCN2C(c2cc3c[nH]cnc-3n2)=O)C1 CC1CN(C(C2CC2(C)C)=O)CC1NC(=O)CSCc1cccnc1 C(C(C)(CC(C)C)NC(=O)C=CC1CCCN1C)NC(CCN(C(C)=O)C)=O CC#CCCC(=O)NC(C1(O)CCN(C(c2oc(C)nc2C(F)(F)F)=O)C1)C C1(C(CNC(=O)NC2CCC(CN(C)C)O2)(C)O)CC2CCC1O2 C1(C(N2CCC(NC(c3cnc(C)o3)=O)C2)=O)CC(=O)N(CC(F)(F)F)C1 Cc1c(Cl)nc[nH]c1=NCC1(CNC(=O)CN2CCS(=O)(=O)CC2)CCCC1 N1(C(C(C(C)C)C)=O)CCC(C2CN(C(=O)CN(CC(C)(C)C)C)C2)C1 c1(COC)ccccc1SC(C)C(=O)NC(=O)OCC(C1CCCO1)=O c1(C(=O)OCC)cnn(C2CCN(Cc3csc(C#N)c3)CC2)c1C C1(NC(COCC)=O)CCCCC12CCN(C(c1cc3cccnn3c1)=O)CC2 C1(CNC(C=COCC)=O)CCN(C(c2ccc(C(N)=O)nc2)=O)C1(C)C C1(C(=O)NCCCNC(c2coc(CO)c2)=O)CCCN(c2ccc(Cl)nn2)C1 N1(C(Cc2c(C(C)C)con2)=O)CC2CC(NC(c3n[nH]c(O)n3)=O)C2C1 Cc1cnc(S(C)(=O)=O)nc1N(C1CC1)Cc1ccc2c(c1)CNC2 c1(C(=O)NCC=CCNC(C2C(CC(C)C)C2)=O)cnc2c(c1)OCCN2 N1(C(CCNC(C)=O)=O)CCC(C=CC(=O)NC(C)C(C)n2cncn2)CC1 N1(C(C(CC=C)C)=O)C2CCC1C(NC(c1ccc(N3CCCC3)nn1)=O)C2 c1(C(N2CCCN(C(C3C(CC)CCO3)=O)CC2)=O)csc2c1CCCC2 C1(CC(=O)N(CCOCCC(N2CCC(=C)C2)=O)C(C)C)CCC(C)(C)C1 C1(NC(c2ccccc2)=O)CCN(C(c2cnnc(O)c2)=O)C12CCCC2 C1(CC)CC(O)CN1C(C1COCCC1NC(=O)C(C1CC1)C1CC1)=O c1(C(=O)NC2(C)CC(NC(=O)CO)C2)ccc(F)c(C(F)(F)F)c1F C1(OCC)CCCN(C(=O)CC2C3CN(C(C4(C5CC5)CC4)=O)CC23)C1 CC1CC(=O)NC(C(=O)NCC2(O)CN(C(=O)CNC(c3ccccn3)=O)C2)C1 c1(NS(C)(=O)=O)ccc(C(=O)NCCSCCCO)cc1F CC1CN(C(=O)CCSCC(N)=O)CCC1NC(C1CCCCS1)=O CC1(C)CNC(=O)N(CC(c2c(F)cccc2Cl)N2CCOCC2)C1=O C1(NC(CCC=CC(C)C)=O)CCN(C(=O)CSc2nc[nH]n2)CC1O C1(C(C(=O)N(CC)CC)(C)C)CCCN(C(=O)CN(C(=O)CNC(C)=O)C)C1 C(C(C)(O)CC(=O)NC(C)Cn1cnnc1)NC(CCN(C)CC)=O C1(CC(N2C(CN(C(C(C3CCC3)NC(C)=O)=O)C)CCC2)=O)CC2CCC1C2 C(CCCC(=O)N1CCC(C)(CCNC(=O)C(O)CC2CC2)C1)OCCC=C C(C)(C(=O)N1CCC(C(=O)NCCCC2CC(C)C2)C(C)C1)(C(C)C)OC C(=O)(CS(C)(=O)=O)N(CC(C)(C)CNC(=O)C(C1CCOC1)OC)CC Cc1cc(O)ccc1CC(=O)NCC1CC(NC(c2cnn(CC3CC3)c2)=O)C1 C#CCC(O)C(=O)NC1COCCC1NC(=O)COc1cccc(C(F)(F)F)c1 C1(CC)C(NC(c2cn(CC(=O)NC(C)C)nn2)=O)CCN1C(=O)C1=COCC1 N1(C(c2nnn(C)n2)=O)CC2(CCN(C(c3ccc4c(n3)OCCO4)=O)CC2)C1 N1(C(C(CC2CCC2)OC)=O)CCCC(C)(CNC(=O)CN(C(=O)C(C)C)C)C1 C(=O)(C(C(C)C)N1CCN(C)CC1)NC(CC)CNC(=O)CN(C)C(C)=O c1(C2C(C(N(C3CN(C(C4C(OC)CC4)=O)C3)C)=O)C2)nc2cccnc2[nH]1 CCC1=NOC(CC(=O)NCCCCNC(C2(C(=O)OC)C=CCC2)=O)C1 c1(CNC(c2cc(F)ncc2NCc2cc(O)cc(Br)c2)=O)cc(Cl)cc(Br)c1 C=CCCCCCC(=O)NCCC1CCN(C(c2cc(SC)c(Cl)cc2Cl)=O)C1 c1(OCC(CC(=O)OC)C)ccc(NC(c2cnc(Cl)s2)=O)c(C)c1 C=CC1(C(=O)NCc2ncc(CC)o2)CCN(C(=O)CCCC2CC2)C1 c1(OCCc2cn(C(C(=O)NCc3nnc(C)s3)C)nn2)ccc([N+](=O)[O-])cn1 c1(C(=O)NC(Cc2cnc(O)nc2O)C(=O)O)cccc2c(Cl)c[nH]c12 N1(C(C(C(C)C)=O)=O)CCCC(C2(NC(=O)C=C3CCN(C)CC3)CC2)C1 N1(C(C2CC(NC(C3CCCO3)=O)C2)=O)CCC(Oc2ccccc2Cl)CC1 c1(OC)cccc(CSc2nc(Cc3cnn(C)c3)nn2-c2ccnnc2)c1 c1(COC)ccc(C(=O)NC2CN(C(C3(OC)CS(=O)(=O)C3)=O)CC2C)cc1F n1(CCC)ccc(C(N2CCC(COCC)C2)C(=O)NCC)c1 N=c1[nH]c(N2CCCC(N3CCCC3=O)CC2)nc2c(Br)cc(Br)cc12 N1(C(C2CCC3(CCC3)CC2)=O)CC2CCCC(C1)N2C(C1CCCC(F)C1)=O c1(C(=O)NCC2C(NC(C3C(c4ccn(C)n4)C3)=O)CCC2)cc(F)ccc1N c1(N2CC(O)(C(C)NC(=O)C=Cc3cocn3)C2)ncnc2[nH]cnc12 c1(NC)ccc(C(=O)NCCN(CC(C)O)C(=O)CSC)cc1Br CCCCCCC(CNC(N1CC(F)(Cc2ccccc2)C2(CCC2)C1)=O)CC c1(CNC(=O)COCCNC(=O)C(c2ccc(O)cc2)C2CC2)ccc(O)cc1 Cc1nn(C)c(Cl)c1C(=O)NCC(C)N(C)C(c1coc(C(C)(C)C)n1)=O C1(N(C(CCC=CC)=O)C)CCN(C(C2CCCCN2C(=O)CC(C)C)=O)CC1 c1(C(N2CCC(CNC(C3(CF)CC3)=O)C2)=O)cc(O)nc(O)c1 N1(C(c2c(CNC(CC(CCC)C)=O)cco2)=O)CCOC(C)(C)CC1 C1(CNC(c2cnc(Cl)[nH]2)=O)CC(O)CN1C(=O)Cc1cscn1 Cc1c(C(=O)NC2CC2NC(=O)CCC(F)(F)F)cccc1F C1(NC(c2ccc(OC)cn2)=O)CC2CC(NC(=O)CCCc3ccsc3)C2C1 c1(C2C(C(=O)NC3CC(CNC(=O)CCF)C3)C2)cccc(Cl)c1 C1(C(=O)NC2CCC(OCC=C)CC2)C(C)OC(C)C1C CC1(C)COCCC1CC(N1CCCC(NC(=O)CN2CC3C=CC2C3)CC1)=O c1(C(=O)NC(C2CCN(C(c3cc(C(=O)OC)on3)=O)C2)C)ccccc1O c1(C(=O)NCC2CN(C(COCC=C)=O)C3C2C3)ccnc2c1CCO2 N1(C(C2CN(C(=O)COC3CCC3)CC(C)O2)=O)CCC2(CC1)CN(C)C2 C=CCCCC(C)(C)C(=O)NCC1OCCC1C(=O)NCCC1CCC1 C(=O)(C(F)(F)C(O)C1CC1)N(C)CCOCCNC(=O)CNC(=O)CC(F)(F)F C1(CC)C(C(=O)NCC(C)(C)C#N)CCN1C(=O)C=NOC c1(OC)ccc(C(=O)NC2CC2C(=O)NCC(=O)N(C)C)c(F)c1 c1(N(C(=O)C(C)CCc2ccc(OC)cc2)CCOC)ccc(F)c(F)c1 N1(C(C(C)OCC#C)=O)CC(CO)C2(C1)CN(C(C13CCC(C)(C1)OC3)=O)C2 C1(CNC(C(C(CC)C)OC)=O)CC2(CO1)CN(C(=O)C1=NOC(C)(C)C1)C2 Cc1cc(C(N2C(CNC(c3nnc(O)nc3O)=O)CC3CC23)=O)cnc1C c1(CC)nc(N2CCc3cc(CN)ccc3C2)c2c(F)cccc2n1 CCCCC(O)C(=O)N1CC2CC(NC(c3sc(C(C)(C)OC)nc3C)=O)C1C2 c1(NCc2scc(C(=O)NCCN3CCC(C)(C#N)C3)n2)c(F)ccc(Cl)c1F N1(C(Cc2nc(NC(c3ccc(F)cc3I)=O)sc2)=O)CCc2cnccc2C1 c1(C(=O)NC2C(CC)CN(C(=O)C3=C(C)OCC3)CC2)ccc2c(n1)OCCO2 C1(NC(CCOc2c(C)cccc2)=O)CCN(C(C2(CF)CCC2)=O)CC1C C(=O)(C1=CCOCC1)N(C(C)C(=O)NC1(CCCCOC(C)=O)CC1)CC c1(C(N2C(CCNC(C(CSC)(C)C)=O)CSCC2)=O)cc2cccc(O)c2[nH]1 c1(OC)ccc(F)cc1C(=O)NC1CC(C)N(C(c2ccc(CO)cn2)=O)C1 C1(CC(=O)N(CCCCC)C)CN(C(=O)COCCN(C)C)CC1C c1(C(=O)NC(CNC(c2cccc(NC(=O)OC)c2)=O)C)csc2ccncc12 N1(C(c2ccc(C#C)o2)=O)CCC(NC(c2nn(C)cc2Cl)=O)C(C(N)=O)C1 N1(C(C2ON=C(C(C)C)C2)=O)CCC2(CCN(C(=O)C(C)CCN(C)C)C2)C1 N1(C(CC2C(C)(C)OCC2)=O)CCC2(CC2C(N2CCC(c3cnco3)C2)=O)C1 Cc1ccc(O)cc1NC(C1OCCC1NC(C1CC12CCCC2)=O)=O C1(CC(C)C)CCCN(C(=NCCN2CCCC2)NCC2COCCC2(F)F)C1 C1(NC(=O)C=CC(F)(F)F)CN(C(=O)C=Cc2ccc(Cl)s2)CCC1F c1(-c2ccc(CNC(c3ccc(OCC)nn3)=O)cn2)ccc([N+](=O)[O-])c(C)c1 C1(CCC)CN(C(=O)CCCc2nnc(C)n2C)CCN1C(=O)C1=CCCCO1 c1(-c2c(C(=O)Nc3ccncc3NC3CCCCC3)cccn2)c(O)cccc1F C1(CNC(CCC#C)=O)CCN(C(=O)Cc2c(CC)cccc2CC)CC1CC N1(C(=O)OC)CC(N=c2[nH]c(=NCCCN3CCOCC3)[nH]c3ncn(C)c23)C1 C(C)(C(C(=O)N1CCC2CC12)NC(=O)C=CC1CCOCC1)OC CCCCCCC(=O)NC1CC(OC)CN(C(c2cc(C(C)(C)C)nn2C)=O)C1 c1(C(N2CCC(NC(c3cc(COC)no3)=O)C2C)=O)cccn2nccc12 C#Cc1cn(C)nc1C(N1CCC(O)(CNC(=O)C(C)=CC2CC2)CC1)=O c1(C(=O)OCC)cn2c(C3=CCN(C(C)C(=O)NC)CC3)cccc2n1 c1(C(N2CCC(NC(CC3CC(OC)C3)=O)C(O)C2)=O)cc(Cl)cc(Cl)c1N C1(C(=O)NC(CC)CN(C)C(C2CC(C)(C)CO2)=O)CC(=O)NC(=O)C1 c1(C(=O)NCCOC2CN(C(c3ccc(F)s3)=O)C2)cc2nc(F)ccc2o1 CN1CCN(S(=O)(=O)NC(CCSC#N)C(=O)OC(C)(C)C)CC1 c1(C(N2CCCC(C(C)NC(c3nc(C#C)sc3)=O)C2)=O)csc([N+](=O)[O-])c1 C(=O)(C(C)CC(F)(F)F)NCC(C(=O)NCc1c(C)nn[nH]1)(C)C C1(C)(NC(CCN(C(C(C=C)OC)=O)C(C)C)=O)CCC(C)(C)C1 N1(C(Cc2ccc(C)o2)=O)CCCC(C(=O)N(C(C)CC(C)C)C)C1C n1(CC)cnc2nc(N3CCC(C)(CO)C3)[nH]c(=NC(C)c3ccc(Br)nc3)c12 C=CC1(CC(=O)NC(c2ccsc2)C)CN(C(=O)Cn2ccc(C)n2)C1 C12(C(=O)NC3CC(CNC(C(C(C)C)OC)=O)CC3O)CC3CC1C2C3O c1(CC(=O)N(CCCNC(=O)CSCc2ccco2)C)cccc(F)c1F C1(C(=O)NC(c2ccccc2)CC2CCC2)CC2CC2N1C(c1sccc1Cl)=O C1(CC)CC(C(=O)NCC(C(C)C)NC(c2ccc(F)cc2)=O)CCO1 Cc1c(C(N2CC(C(O)C(N3CC(C)OCC3C)=O)C2)=O)[nH]ccc1=O N1(C(CC)=O)CCCC(C(=O)NCC2(F)CC(CNC(C3CCCN3C)=O)C2)C1 C=C1CC(C(=O)Nc2cnoc2)N(C(=O)C(c2ccccc2)O)C1 c1(C(=O)NCC(CO)NC(c2cc(C)[nH]c2C)=O)csc2ccccc12 CC(C(=O)NC1(C(=O)NCc2ccc(F)c(F)c2)CC(O)C1)S(N)(=O)=O C(=O)(C(O)CC(C)(C)C)NC1C(NC(CN(c2cccc(Cl)c2)C)=O)CC1 C(C)(C(=O)N1CCC1C(=O)NCc1cccc(F)c1C)(C(C)C)OC c1(C(=O)OC)cc(C(N2CCC(c3cn(CC4CC4)nn3)C2)=O)c(F)cn1 C(C)(CCCCNC(c1ccc(C(F)F)s1)=O)NC(CCc1scc(C)n1)=O c1(C(=O)OC)cc(NC(C23CC(CO2)C3)=O)nc2ccccc12 C1(C(N2CCC(C3N(C4CN(C)C4)CCCC3)CC2)=O)COc2ccccc2O1 C(C(C)(C)C1=CCCC1)NC(C1(CC)CN(C(=O)C(O)CC(C)(C)C)C1)=O C(=O)(C1=CCCOCC1)NC1CCC(C)(NC(=O)CC2CCC(C)(C)O2)CC1 c1(CC)sccc1C(N1CCCC1C(C)(C)NC(C1(C)CC(F)C1)=O)=O C1(C(=O)NCCC(C)(C)NC(c2cccnc2O)=O)CC2(C1)CC(F)(F)C2 c1(C(=O)NCC2CC(OC)CN2C(=O)CCC(N)=O)cc(C)nc(O)n1 Cc1nc2nccc(N(C)CC3CCCN3C(c3cn(C)nc3C)=O)n2n1 C(=O)(C(C)(O)C(F)(F)F)NCC(CC(=O)N(CC=C)CCO)O Cc1cc2ncc(-c3ccc(NC(c4cccc(O)c4O)=O)s3)cn2n1 C=CCC(C(=O)NC(C)CCCCNC(C1CN(C(C)=O)C1)=O)N(C)C C=C1CCC(C(=O)NCCN(CC(F)(F)F)C)CC1 N1(C(C(CC)NC(N)=O)=O)CC2(CCC2NC(c2csc(C(C)(C)C)n2)=O)C1 C1(C)(NCc2ccc(C(C)=O)o2)CCN(CCCN2CCC(O)CC2)C1 c1(C(N2C(CNC(c3n(CC)ccc3)=O)CC2)=O)cncc(OCC(F)F)c1 c1(C(=O)NCc2n(C)ccn2)cc(-c2nccs2)cn2ccnc12 c1(CNC(C(C=CC)O)=O)ccccc1CN(C(=O)C(C)OCC=C)C C1(CN(C)C(C2CCOC2)=O)CN(C(c2cccc(C(F)F)c2)=O)CC12CC2 C=CC(CC)CC(=O)NCC(c1cccc(C)c1)NC(c1ccoc1C)=O c1(C(N2CC(OC)(CNC(C3CCC34CCC4)=O)C2)=O)ccc(F)cc1Cl c1(NC(C)=O)cccnc1C(=O)NC1CC(CNC(C2CC2C(F)F)=O)C1 c1(C(N(C2CCN(C(C3CCCN3C(N)=O)=O)C2)C)=O)cc(C(N)=O)cn1C c1(C(=O)NCCC2(O)CCCN(C(c3cnco3)=O)C2)ccc2nccnc2c1 N1(c2c(C#N)cncc2)Cc2ccccc2C(CNC(C23CC(CO2)C3)=O)C1 c1(C(=O)NC(C(=O)NC2C(NC(C3(OC)CC3)=O)CC2)C)ccccc1F N1(C(C=CCC)=O)CCCC1C1CCCN1C(=O)C=Cc1c(C)coc1C c1(C(=O)NCC(CC)NC(=O)CN(C2CCCC2)C)cnc2cnc(Cl)cc2c1 S(=O)(=O)(c1cc(Cl)ccc1F)Nc1ccc2c(c1)CN(C(C(CC)(C)O)=O)C2 N1(C(c2cc(OC)no2)=O)CCC(O)(C2(NC(C3CCC(=O)N3)=O)CC2)CC1 N1(C(COCCC#C)=O)CCCN(C(=O)CCc2ccc(N(C)C)cc2)C(C)C1 N1(CC(=O)NCC2(F)CCCN(C(C(C(C)C)C#N)=O)C2)CCc2sccc2C1 Cc1nc(C(C)C)ncc1C(=O)NC(C)CC1CN(C(=O)C2=NOC(C)C2)C1 N1(C(=O)C=CCCN2CCCC2)CCC2(NC(=O)C(F)=CC3CC3)CCCC12 C1(N(C(=O)C=CCF)C)CCN(C(C2CCCN2C(=O)C(C)(C)C)=O)C1 N1(C(CC(=C)C)=O)CCCCC1CN(C)C(C1(CSC)CC1)=O Cc1nc2c(s1)CN(C(c1ccc(CNC(C3(C)CCC(C)C3)=O)cc1)=O)C2 C(=O)(C1=CCC(C(F)(F)F)OC1)N1CC(CNC(CCOC(C)C)=O)N(C)CC1 c1(C(C)NC(c2ccc(Cl)c(C(F)(F)F)c2)C)cccc(O)c1Cl C1(CN(C(CSCCC)=O)C)CN(C(C2CC2(CC)COC)=O)CCO1 n1(CCCC)cc(C(=O)NCC(CNC(C2(CO)CC(F)(F)C2)=O)CO)c(C)n1 Cc1cc(=O)n(C)cc1NC(=O)C(C1CCCO1)NC(c1ccccc1C#N)=O C1(NC(c2cnn(CC)n2)=O)CCCCC1NC(C1CCC(C(=O)OC)O1)=O CCC(CC(=O)NC(C1CCN(C(C2Cc3ccccc3O2)=O)C1)C)C(C)(C)C c1(Cn2cc(C3(O)CN(C(C4(C)CC4(Cl)Cl)=O)C3)nn2)ccccc1[N+](=O)[O-] c1(NC(CCC(=O)N2CCC(OCCNC(C)=O)C2)=O)n[nH]c(C(C)C)c1Br C(CC(=O)NC1CC(C(=O)OC)C1)(C(F)F)NC(C1CC(N(C)CC)C1)=O CC1CN(C(=O)Cc2ccc(Cl)s2)CC1NC(=O)CCc1cnc(C2CC2)o1 c1(C(=O)NCC2CN(C(C(C)c3ccco3)=O)C2)ccc(Br)cc1Cl C=C1CC2(C1)CC(C(=O)NC1CC(C)(NC(C3CC3(F)F)=O)C1)C2 N1(C(c2ccc(C(C)=O)o2)=O)CCOCC1C(=O)N(C)Cc1cnn[nH]1 N1(C(c2ccn(C)c2)=O)CC(O)CC1CC(=O)NCCOCC1CCC1 C1(CCNCC2(Cl)C(F)(F)C2)CSc2ccccc2O1 c1(C(=O)NC2(CNC(C)=O)CC2)ccc(C(=O)NCCn2cccn2)c(F)c1 Cc1cc(C(=O)N(C2CCC(NC(=O)CSc3ccc(O)cc3)C2)C)ncn1 Cc1cc(F)ccc1CC(=O)NC1CC2CCC1N2C(C1(F)CCCC1)=O N1(C(c2nc(C(=O)OCC)n[nH]2)C(=O)NCCCC)CCC(C2CC2)(N(C)C)C1 C(=O)(C(CC(C)C)NC(C1CN(C(C2CC(=O)CC(=O)N2)=O)CC1(F)F)=O)NC C(=O)(C(C)CC1CCC1)NCCCN(C(C(C)=C(CC)C)=O)C c1(C(=O)NC2CC(CNC(=O)Cn3nnnc3C3CC3)C2)cncnc1C1CC1 CC1CCN(C(c2[nH]ccc2C2CC2)=O)C(C)C1CNC(=O)CC1C=CCC1 c1(NC(CC)=O)ccccc1OCC.C1(C)C(=O)NCCCN1C CCCCC(O)CC(=O)NC(C)C(C)(C)C(=O)NOCCCO N1(C(c2cc(C)ncc2C)=O)CCC2OCCN(C(c3nn(C)cc3Cl)=O)C2C1 O=C1COc2ncc(C(=O)NC3CCN(C(=O)CC4C=CCC4)CC3F)cc2N1 C1(CC(=O)NC2C(CNC(c3nc(C)oc3)=O)CC2)CCC(=O)NC1=O C1(C(N2C(C(C)NC(=O)C=Cc3cnc[nH]3)CCC2)=O)CCC(C(C)(C)O)CC1 C(=O)(CP(=O)(C(C)C)C(C)C)NCCOCCNC(c1c(C)cc(C)cc1O)=O c1(N2CC(O)(C(C)NC(C=NOC)=O)C2)nc(C)nc2scc(CC(C)C)c12 C(=O)(CN=S(C)(C)=O)N(C)CC1N(C(COCCC=C)=O)CC(F)C1 C1(C(=O)NC(C)C(CO)NC(c2cc(N)cnc2Cl)=O)CCCC12CCC2 N1(C(c2cn(CCC)nc2)=O)CCC2CN(C(C3(F)CC3)=O)CCC12 C1(O)(CNC(C(CCOCC)NC(c2cn(C3CC3)cn2)=O)=O)CCC(C)(C)C1 c1(C(=O)NC(CNC(C(CC)(C)CO)=O)(C)C)cncc2c1CCNC2=O c1(-c2cnc(C(C(=O)OC)=O)s2)cccc(N2CCCC2=O)c1 c1(CCC(=O)N(CC(CC)NC(c2n[nH]cc2F)=O)C)cc(F)c(F)c(F)c1 N1(C(C2(COC)CC2(F)F)=O)CCC(O)(C(C)NC(c2cnc[nH]2)=O)CC1 N1(C(C(C=C)C)=O)CCC2(CCC2NC(c2ccc(OC)nc2)=O)CC1 C(=O)(CCCC(CC)NC(c1csc(CC)n1)=O)N(C)Cc1onc(CC)n1 C1(NC(CCCC=C)=O)CN(C(=O)C(O)C(C)C)CC1(C)C N1(C(Cc2cccc(C)c2)=O)Cc2ccc(NC(c3cncs3)=O)cc2C1 C(C(C(=O)NCCNC(C1CCCN1C)=O)NC(=O)OC(C)(C)C)OCC Cn1ncc([N+](=O)[O-])c1C(=O)NCCC(C)(C)NC(c1n[nH]cc1Br)=O c1(CNC(NC(C=C)C)=NCc2ccc(C)cc2C)c(O)nc(=O)n(C)c1N CC1(C)C(C(=O)NCCOC2CCN(C(c3cc(C4CC4)ncn3)=O)C2)C1C#N c1(-c2ccc(NCc3n(C)nc(I)c3)cc2)ccc2c(c1)CC2 C12(NC(C3(C)CCCN3C(C3CC3(Cl)Cl)=O)=O)CCCN(CCC1)C2 CN1CC(C2OCCO2)(N(C(C)(C)CC2CCC2)C2CC2)CCC1=O C=CCCCC(C(=O)N(CCC)CCC)NC(C1CC12CCC2)=O c1(OC)cccc2c(C(=O)NC3CCN(C(C4(C)CCNC(=O)C4)=O)C3)coc12 c1(C(=O)NC(CNC(C(c2ccccc2)SC)=O)CO)ccc(F)cc1Cl C1(CNC(C2(C(C)C)CCC2)=O)CC2(CC2)CN1C(C1CC2CC1CC2O)=O c1(OC)nc(=NC2CC(NC(c3c(Cl)ccc4c3OCO4)=O)C2)nc(OC)[nH]1 CC1(C)CN(C(C2(C)CCOC2)=O)CC(CNC(=O)CSc2cccs2)O1 C(=O)(C1CCCn2cnnc21)NCC1(CNC(=O)Cc2n[nH]cc2Br)CCC1 c1(C(N2CCCC(CNC(Cc3ccc(C)s3)=O)C2)=O)ccc2nnn(C)c2c1 N1(C(CNC(c2cc(OC)n(C)n2)=O)=O)C2CCCC1CN(C(=O)C=CCF)C2 c1(C(N(C2CN(C(=O)Cn3cccnc3=O)C2)C)=O)cnc2c(c1)OCCN2 N1(C(c2cc(Cl)sc2Cl)C(=O)NC2CC2)CCc2c(C(F)(F)F)n[nH]c2C1 C1(CNC(C(CC)OCC)=O)CC2CCC1N2C(=O)Cn1cnnc1O c1(C(=O)NCC2CN(C(c3c(CC)cno3)=O)C(C)C2)c(Cl)ccc(F)c1N C(C1CCCN1C)=CC(=O)N(C1CN(C(=O)Cc2n[nH]cc2Br)C1)C c1(-c2c(F)ccc(OCC)c2)ccc2c(c1NCc1cc(Cl)ccc1Br)OCO2 C1(NC(c2ccc(Br)o2)=O)CC2C1CCN2C(C1CC2(C1)CC(O)C2)=O CN1CCC(N=c2[nH]ccc(=NCCc3cnn(-c4ccccc4)n3)[nH]2)CC1 N1(C(C(Cc2cccc(OC)c2)O)=O)C2CCC1CN(C(C)=O)C2 C(=O)(CN=S(C)(C)=O)NCC1C(NC(C(c2nc(C)sc2)=O)=O)C1 Cc1cc(C(=O)NCC(C2CCC2)NC(C2(C)C=CCC2)=O)nn1CCO c1(NC(C(C)N(C(C2(OC)CCCOC2)=O)C2CC2)=O)cnc2ccccc2c1 C1(C(N2C(CC=C)CCCC2)=O)CC(O)CCN1C(=O)C(C)OCC C(CC(C)CCNC(=O)CCN(C)CCO)NC(C(c1cc(C)sc1)(C)C)=O C1(OC)CCN(C(C2(CCNC(c3ncsc3C)=O)CCCC2)=O)CC1C n1(C2C(C)CC2)c(-c2ccc(C#N)c(F)c2)csc1=Nc1cc(C#N)ccc1Cl C(=O)(CCCCC(N)=O)N1CC(C)C(CNC(=O)CC2(O)CCCCC2)CC1 CC(=Cn1ccnn1)C(=O)N1CC(C)C(C)(CNC(=O)COC2CC2(F)F)C1 CCC(CC)C(F)C(=O)NC1C2CN(C(=O)C(O)CC(C)(C)C)CC12 C1(C(=O)Nc2cnc(OC)c(F)c2)CN(C(=O)C(C)NC=O)CCC1(F)F CC1=C(CNC(C(C)(C)C)c2cnn(C)c2)S(=O)(=O)CCO1 C(=O)(C(C)(C)C(C)(C)C)N1CCCN(C(c2ccc(OCC=C)cc2)=O)CC1 C(=O)(C1=CCCC1C)NC(c1cccc(Cl)c1)CNC(CCCNC(C)=O)=O c1(OCCC(=O)NCCC2CC(C)C2)cccnc1 N1(C(C2(SC)CCC2)=O)CC2(C1)SCCC2NC(c1oncc1C)=O c1(C(=O)NC(CNC(C(C)NC(C)=O)=O)CO)ccn2ccnc2n1 CC1CCCC1(C)C(=O)N(C1CCN(C(c2cnc(CC(C)(C)C)o2)=O)CC1)C C1(C(=O)O)(NC(c2cnc(OC)c(C)c2)=O)CCc2ccccc2C1 CC(CCC(F)(F)F)(c1nnnn1C1CCOCC1)NC(c1ccccc1)C1CC1 N1(C(C(C)CNC(c2c[nH]nc2C2CC2)=O)=O)CCN(C)CC1C1CC1 C1(CC(=O)Nc2ccc(OCC)nc2)CN(C(=O)CCc2cccs2)CC12CC2 N1(C(c2cnc(CC)s2)=O)CCC(O)C(N(C)C(C2CC2C(F)F)=O)C1 C12(C(=O)NCC3CN(C(C4CCCN(CC)C4)=O)CC3C)CCC(C)(CC1)OC2 C1(C(=O)NCC2CCC(CNC(C(CC)F)=O)CC2)CC2CC2CC1C CC1CC(NC(=O)CCSc2ccccc2F)CN1C(=O)CC1CCC1(C)C C(C(CC(C)C)C(=O)NC1(C)CCCN(C(c2ccnn2C(C)C)=O)C1)OC C(=O)(CCCCCC(C)C)NC1C(OC)CN(C(c2n(CC)nc(C)c2)=O)C1 Cc1nc(Cl)[nH]c(=NC2CC(C)N(C(c3[nH]cc4c3CCCC4)=O)C2)c1Cl c1(C(=O)NC2(C(N3CC(C#N)(CC)C3)=O)CC2)cccc(F)c1OC N1(Cc2cc(C)cc(Br)c2O)CC2CCC1CN(C(c1nccnc1Br)=O)C2 c1(C(C)NC(c2cnc(OC)s2)=O)ccc(CNC(c2[nH]cnc2C)=O)cc1 N1(C(C(COCC)NC(C2CCS2(=O)=O)=O)=O)CC2(CC(C)CO2)C1 N1(C(COCC=C)=O)CCC2C(C1)CN2C(=O)C=CC1CCOCC1 c1(CC)ccc(C(N2CCCCC(N(C(=O)Cn3cc(C)cn3)C)C2)=O)c(C)c1 N1(C(CCSCC)=O)CC2(CCCCN2C(c2oc(CO)cc2C)=O)C1 C(=O)(C#CC1CCCC1)NC1CC(CNC(C(C)(C)SC)=O)C1(C)C C(C(C)(C)C(=O)NCCCCCN(C1CCCCCC1)Cc1cncs1)OCC C1(NC(C(C)OC)=O)Cc2ccccc2N(C(c2cnn(C(F)F)c2)=O)C1 C1(NC(c2c(CC)non2)=O)CN(C(=O)C=CCN2CCCC2)CC1O CC(C(=O)NCC(c1ccccc1)N(C(=O)Cc1cccs1)C)S(N)(=O)=O C(=O)(C(C)CS(C)=O)N(CC(C)(C)NC(c1c(C)nc[nH]1)=O)C N1(C(c2c(C)cco2)=O)CC(NC(c2cccc(C3(C)CC3)c2)=O)CCC(O)C1 C1(CC)(NC(=O)C(c2cnn(C(C)(C)C)c2)C)CCN(C(=O)CO)CC1 C1(C(=O)OC)(NC(c2c(O)cc(Br)cc2F)=O)Cc2ccccc2C1 CC1(C)OCCOC1C(=O)NCC1CC(NC(c2cc(C3CC3)[nH]n2)=O)C(O)C1 c1(SC)ccc([N+](=O)[O-])c(C(=O)NCC(CC(C)C)NC(=O)C2=CCOC2)c1 C(=O)(CCCCC(=O)NCC1CC(NC(c2cnc3c(c2)CCC3)=O)C1)NC N1(C(C(COCC)NC(=O)NC2CCC(=O)C2)=O)CC2CC1(C(F)F)C2 Cc1cc(=O)c(C(=O)NCC2CCCN2C(c2ccc(F)c(F)c2)=O)c[nH]1 c1(C(=O)NC2(CCCNC(C3CCCS3)=O)CC2)ccc2c(Br)cnn2c1 CCC(O)C(C)C(=O)NC1CCC(CNC(=O)Cc2cncc(C)c2)CC1 C1(CNC(C(C)OCCC#C)=O)CN(C(c2cc(Br)c[nH]2)=O)CC1C C(=O)(C(C)(C)CS(N)(=O)=O)N(CCN(C(c1cc(C(=O)OC)sn1)=O)C)C CC(C)C(O)CC(=O)NC1CCN(CCOCC(F)(F)C(F)(F)F)CC1C N1(C(C2C(c3c(C)ccs3)C2)=O)CC(CNC(=O)COCC(F)F)C(C)(C)C1 C1(CCC)CN(C(=O)C=Cc2ccsc2)CCN1C(c1nccnc1C)=O c1(C(N2CCC(C(N3C(C(C)C)COCC3)=O)C2)=O)n[nH]cc1[N+](=O)[O-] C1(C(=O)NC(CCC)CO)CCN(C(=O)C(C)N=[N+]=[N-])C1C CC1CC2CN(C(=O)CC(=O)NC3CC3)CC2N1C(=O)CN(CC(C)(C)C)C c1(OCC)ccc2[nH]c(=NCCCNC(=O)C(F)CC)sc2c1 C#CC1(C(=O)NC(C)(C)C#CC)CCN(C(c2[nH]cc(C)c2C)=O)CC1 c1(CNC(C2CC(NC(C3N(C)CC(O)CC3)=O)C2)=O)cc2cc[nH]c2cn1 C1(CNC(N2CCCC(N3CCCCC3=O)C2)=O)CN2CCCC2CO1 c1(C(N(CCNC(COc2ccn(C)n2)=O)C2CC2)=O)ccnc2ncccc12 C1(C(C)NC(c2cc(Cl)n[nH]2)=O)CCN(C(c2cnc(O)o2)=O)CC1 C(=O)(C1=C(C#N)CCC1)N1CCC(C=C)(C(=O)NC2CCC(N(C)C)C2)C1 C1(O)(CN(C(=O)CC(F)F)C)CCN(C(C2(CC3CC3)CC2)=O)CC1 c1(C(N2CCC(C)(NC(=O)CSCC(N)=O)CC2)=O)ccc2c(c1)CNC2=O Cc1nc(CC(=O)NCC(C2CCCC2)NC(C2CCCCS2)=O)[nH]c1C CC1CN(C(=O)COC(C)(C)CC2CCOC2)C(C)CN1C(c1csc(=N)[nH]1)=O N1(C(C(c2ccccc2)N(C)C)=O)CCC(NC(c2cnc[nH]2)=O)C(O)C1 C(=O)(CCN=C(NCc1ccc(OC)c(OC)c1)N1CC2CCN(C)C2C1)NC C1(NC(C(C)C(F)F)=O)CCCCN(C(=O)Cc2cc(Br)ccc2Cl)C1 Cc1ccc(C(=O)NCC(C2CCCCC2)NC(=O)CS(N)(=O)=O)c(C2CC2)n1 C(=O)(C(C(C)(C)C)N1CCNC1=O)N1CCC(C)(NC(c2c(C)nncc2)=O)C1 c1(CN2C3(c4nnc(Cc5sccc5)o4)CC(C2)C3)cc2c(cc1O)OCO2 c1(C(N2CC(CNC(c3c(OC)cccn3)=O)OCC2)=O)cc(C)cc(C)c1N Cc1cnc(CCNC(C2CC=CC(NC(=O)CCc3ccoc3)C2)=O)cn1 c1(C(N2C(CCC(N3CCC(OC)C3C)=O)CCCC2)=O)ccc(C#N)c(C)n1 CCC(C)C(O)CC(=O)N1CCCCC1C(=O)Nc1ccc(C)cc1C c1(CC)ccsc1C(=O)NC(CNC(=O)C(CO)OC)CO Cc1c(C(=O)NCCC2(O)CCN(C(=O)C(N3CCOCC3)C)C2)cncc1Cl N1(C(C(CCC)F)=O)CCN(C(=O)C(N2CCCCC2=O)C)C(C(C)C)C1 C(=O)(C(CC(C)C)OC)N1CC(NC(C2(CC=C)CCC2)=O)C(OC)C1 N1(C(c2nc(C(=O)NCC=C)sc2)=O)CCCC(CCC)(NC(=O)CC(C)F)C1 c1(C(=O)NC(CN(C(C(CC)OC)=O)CC)C)ccc2c(c1)CCCS2 CCCC(CC)NC(c1nnnn1C1CCCC1)c1ncc[nH]1 c1(COC(c2ccn(CCOC)n2)=O)cc(C)n(-c2cccnc2)c1C c1(C(N2C3CN(C(C(F)OC)=O)CC2CC3)=O)ccc2c(c1F)CCC2 c1(-c2cc(C(=O)OCc3cc(CC)ncc3)no2)ccc(F)c(F)c1 c1(OC)ccccc1C1(NC(c2csc(COc3ccc(Cl)cc3)n2)=O)CCC1 C1(CC(=O)N(CCN(C)C)CC)(NC(=O)CCn2cnnn2)CCCCC1 c1(CNC(C=CCC(C)(C)NC(C(C)n2cccn2)=O)=O)ccc(F)cc1F CC1CC(C(=O)NC2CCCC2C(N)=O)N1C(=O)CSc1nc[nH]n1 C1(C(N(CCCC(=O)NC)C)=O)CCC2CCC1N2C(c1ccc(C2CC2)o1)=O c1(CC)cc(NC(C2C3CC4C(C3NC(=O)CCCC#N)C24)=O)ccc1F C(CC(C(C)(C)C)NC(=O)CC1(O)CCC1)N(C(CC1CCN(C)C1=O)=O)C C(N=c1nnn(C)[nH]1)C1C(NC(C(C(C)C)OCC(C)C)=O)CCCC1 N1(C(CCOC)=O)CC2CN(C(C3CCCN(C(C)C)C3)=O)CCC12 c1(CCN(C2CC(C(=O)O)C2)C(C=CC)=O)ccccc1C(=O)Nc1ccccc1 c1(C(N2C(CNC(C(C3CCCC3)NC(C)=O)=O)CC2)=O)cc2n(n1)CCO2 c1(C(=O)NC(C)CNC(c2cccc(Cl)c2)=O)cc2sc(Cl)cc2s1 c1(C(N(CC(C)C(F)(F)F)C)=O)coc2c1CN(C(=O)C(=O)NCC1CC1)C2 c1(OCCNC(=O)NNC(=O)c2ccccc2)ccc(Cl)cc1F c1(C(=O)NC2(CC=C)CCN(C(C3CC(=O)NC(=O)C3)=O)C2)cncc(F)c1C C(=O)(CC(C)(C)CC(F)F)N1CCC(O)(C(C)NC(=O)CN(c2ccncc2)C)C1 c1(C(=O)Nc2ccc(C(=O)NCC)cc2C)cccc2c(C)csc12 c1(NC(c2c(C)nccc2)=O)c(C)ccc2ncccc12 C1(C(N2C(CCN(C(=O)CC3CC=CC3)C)CCCC2)=O)CCc2nnnn2C1 c1(OCC)cc(N2CCC(CO)(NC(=O)C(C)S)CC2)nc(C)n1 C(=O)(C1=C(Cl)CCCC1)N1CCCC(NC(=O)Cc2ccc(F)cn2)CC1 c1(C(C(=O)NCCC)N(C)Cc2csnc2C)ccc(OC)c(O)c1Br c1(C(N2CCN(C(=O)CCn3ccnn3)C(CF)C2)=O)cncc(Cl)c1Cl N1(C(c2c(C)nncc2)=O)CC2(C1)CN(C(C1CC3(C1)CC(O)C3)=O)CCO2 Cc1cc(F)c(Cl)cc1C(=O)NCC1CCN1C(=O)CC1CCC(C2CC2)O1 C(=O)(C(CC(F)F)N(C(=O)C(C)CN(C)C)C)N1CCC(C(=O)OC)CC1 N1(C(C(C)N(CC)CC)=O)CC2(C1)CN(C(=O)Cc1ccnn1C)CC2CO c1(C(N2CC(OCCNC(=O)CC3COCCO3)C2)=O)cc(Cl)ccc1F N(C1CCc2c(O)cccc21)C(=O)NCCc1nc(C(O)C2CC2)no1 c1(C(=O)NCC(CCNC(=O)CC(C)(C)C)OC)nccc(Cl)c1F N1(C(c2ncc(CC)s2)C(=O)NCC)CC2CS(=O)(=O)CC2(C#N)C1 CN1CCCC(OC(=O)Cc2coc(-c3ccc(Cl)cc3)n2)C1 c1(C(C(=O)Nc2cccc(NC(CC(C)F)=O)c2)(C)C)cccc2ccccc12 C1(N(C(C(C)OCC)=O)CC)CCN(C(C2(n3cncn3)CC2)=O)CC1 c1(OCC=C)cc(OC)ccc1C(=O)NC(C)CNC(=O)CC#N C1(OC(C)C(=O)N2CC(NC(=O)CCOC3CCOCC3)C2)CCOCC1 CCC(C)C(C)(O)CNC(=O)C(O)CNC(C12CC1CNC2=O)=O c1(C(=O)NCC2(C)CCC(NC(C(C=C)(F)F)=O)C2)cccc(Cl)c1O C1(CC)C(C(N2CC(O)CC2CNC(c2c(C)ncn2O)=O)=O)CCN1C Cc1cn2c(n1)CCC(N=c1nc3sccc3c(NCC(C)S(N)(=O)=O)[nH]1)C2 C1(NC(C2(Br)CC2)=O)C2CCC1CN(Cc1ccc(OC(F)(F)F)cn1)C2 C1(C(C)NC(=O)C=C2CC2)CCCN(C(=O)CCc2ccccc2Cl)C1 N1(C(C(C)S(N)(=O)=O)=O)CCCC(O)(Cn2cc(CCN3CCCC3)nn2)CC1 C1(OC)CCCC(C(=O)NC2(C)CC(NC(c3cc(C)[nH]c3C)=O)C2)C1 CCC(C)C(O)C(C)C(=O)NC1CC2(C1)CN(C(c1n[nH]cc1C)=O)C2 C(CO)(CCCCNC(C1(CCO)CC1)=O)NC(C1CC=C(C)CC1)=O C1(C)(C(N2CC(C)(NC(c3c(OC)cc(C)cn3)=O)C2)=O)OC(C)(C)OC1C C1(C(=O)NCC(CNC(C2(N(C)C)CCOCC2)=O)OCC)CCCCNC1=O Cc1onc(O)c1C(N1CC2C(CNC(C3CCC(C(F)(F)F)CC3)=O)C2C1)=O N1(C(CC2(OC)CC2)=O)CCCN(C(=O)C(F)C(C)C)CC1C c1(C(N2CC(NC(C3CSCCS3)=O)C2)=O)ccc(C(F)(F)C(F)(F)F)cc1 c1(C(NOC(c2ccncc2)C)=O)cc2c(s1)C(C)(C)CC2 C1(C(=O)NC2C(n3cc(C(CCC)=O)nn3)COC2)CC2(CC(C)=NO2)C1 N1(C(C(C)(C)O)=O)CCCCC(CNC(=O)Cc2ccsc2Br)C1 C1(CCCC)CN(C(c2cccn(C)c2=O)=O)CCN1C(c1nnccc1C)=O c1(CNC(C2CCN(CC)C2)=O)ccc(CNC(=O)C(C)c2cncs2)cc1F CC(C)(CC(F)(F)F)C(=O)NC1CN(C(=O)CCCF)CC(F)(F)C1 Cc1ncc(C)c(N2CCCC(CCNC(C3CC4(C3)CC(F)C4)=O)CC2)n1 C1(C(=O)NCc2ncn(C)n2)CC(F)CCN1C(C1CC(C)(C)CO1)=O c1(C(N2CCOCC(NC(CC=C=C)=O)C2)=O)ccc2ncc(=O)[nH]c2c1 n1(CC)nc(C)c(C(=O)NCCC2(O)CN(C(C3CC4CCCCC34)=O)C2)c1Cl C(c1cncnc1O)=CC(=O)NC1CC2CC1N(C(C1CCCOCC1)=O)C2 C1(NC(C(CC)C)=O)CCN(C(=O)C=CSc2ccccc2)C1C(C)C c1(OC)cc(C(N2C3CCC(C3)C2CNC(=O)C(C)CO)=O)ccc1O C(CCCCN(C(=O)CCSCC(C)C)C1CC1)NC(C(C)=C(CC)C)=O C1(CNC(C2(C)CCC(=O)NC2)=O)CC2COCC2N1C(c1ccccc1O)=O CC1CC(C(=O)NCCC(C)(C)NC(c2sc(C#N)cc2Cl)=O)CC(=O)N1 C1(CNC(c2c(C)cccn2)=O)CC2CCC(C1)N2C(C1CCCCN1C)=O C=CCCC(C(=O)NCCCN(C(=O)CC(O)C(C)C)C)NC(=O)OC(C)(C)C CC1(C)CCCNC1=O.C1(C(=O)NCCC2CCCC3CC23)CCOC1(C)C c1(C(=O)NC2(C)CC(NC(C3C(C=C)OCC3)=O)C2)cc(C)nc2[nH]nc(O)c12 c1(C(N(C2CCN(C(=O)C(O)CCC(C)C)C2)CC)=O)cc2cccnc2cn1 c1(CC)ccc(C)cc1NC(c1cccc(F)c1)c1nnnn1C1CCOCC1 C(=O)(CC(CNC(=O)C(CO)OC)C1CCC1)NC(C#C)CCC c1(N(CCOC)C)cc(N(C)CCOCCO)nc(COC)n1 c1(CC(=O)NCc2cnc(Br)s2)cccc2nonc12 C1(C2CC2)(NC(C(CNC(C(CC)NC(N)=O)=O)N(C)C)=O)CCOC1 C1(NC(c2cnn(CC)c2Cl)=O)CCN(C(=O)C(C)(C#N)CC)CC1F C1(F)(C(=O)NC2C(CC)CCC2)CCN(C(c2cncc(CO)c2)=O)C1 c1(OC)c(N2CCN(C(C3(Oc4ccc(F)cc4)CC3)=O)CC2C)ncnc1C C(=O)(C1=NOC2(CCOC2)C1)N1CC(CNC(c2cc(COC)on2)=O)OCC1 C1(CNC(c2c(NC)cnnc2)=O)CN(C(C2CNC(=O)C2)=O)CCN1C N1(CC)CCOC(C(=O)NCC2CCCCN2C(=O)COCC(C)(C)C)C1 C1(C(=O)NCCN2CC3CC3C2)CCOCCN1C(=O)CCC(F)(F)F N1(C(Cc2cccc(OC)c2)=O)CCC(N=c2ccn3ncc(C#N)c3[nH]2)C1 C=Cc1ccc(C(N2CCC(CC(=O)NCCC(O)COC)C2(C)C)=O)cc1 C1(CCC)(NC(C2CC(C)CO2)=O)CCN(C(=O)C=CC2CCC2)CC1 Cc1ccc(NC(c2sccc2CNC(C2(C)CNC(=O)C2)=O)=O)c(C)n1 c1(CC(N2C(CNC(C3C(C)C3)=O)CCCCC2)=O)ccc2c[nH]nc2c1 C1(C(=O)NC(C2N(C(c3c(CC)n(C)nn3)=O)CCC2)C)CCC=CCCC1 c1(C(=O)NCCC(C(N2C(COC)CCCC2)=O)O)c[nH]c2nccc-2c1 C1(CC)(CNC(C2(NC(=O)CN3CC=CC3)CC2(C)C)=O)CCC(=O)N1 C1(C(C)(C)NC(C2CC2(F)F)=O)CCCN1C(=O)CC1CCSC1 N1(CCC(=O)NCCCOCCNC(C(CC)F)=O)CCCC(N(C)C)C1 CCC(C)(CO)C(=O)NCc1ccnc(C(N2CCOCC2CO)=O)c1 C1(CNC(C(C)(C)C2CC2)=O)CN(C(=O)CC2CCC(=O)NC2)CC(C)(C)O1 N#Cc1ccc(S(=O)(=O)NC(CF)CF)cc1N1CCCOCC1 C1(NC(CC2(NC(C)=O)CC2)=O)CN(C(=O)C(C2CCCCC2)F)CC1C c1(OC)c(C(N2CCCCC2CNC(=O)CN(C)C(N)=O)=O)cccc1[N+](=O)[O-] CN1CCN(C(=O)C(CCF)NC(C2CNC(=O)O2)=O)CC1CO C1(C(=O)NC(CO)C(F)(F)F)CC12CCN(Cc1cccc(I)c1F)CC2 C1C(F)(F)CCC(=O)NCCC2(CCCCC2)c2cn1nn2.CC(F)CCCO C1(O)(C(=O)NCCCN(C(C(CC)(C)CO)=O)C)CCCC(C)(C)C1 C(=O)(C1CSc2ccccc21)N1CC(C2(NC(CC3CC(=O)C3)=O)CC2)C1 CCC(CC)CCC(=O)N1CC2CC1CN2C(c1ccc(NC(C)=O)cc1O)=O c1(OC)cc(C(=O)NCC2CC(C)N(C(c3cnn(C4CC4)c3)=O)C2)sc1Cl c1(C(=O)NC(C2CCOC2)CNC(c2cnc(SC)[nH]2)=O)cccc(F)c1C Cc1ccc(NC(=O)C(N2CC3CC3(C(=O)NCC3C(Cl)(Cl)C34CC4)C2)=O)cc1 C12(CCC(=O)N(C3CCCCC3)CCNC(=O)Cc3ccsn3)CCC(CC1)C2 N1(C(C2CCC2Oc2ccccc2)=O)CCCN(C(c2ccc(Cl)cc2)=O)CC1 N1(C(CC2(NC(C)=O)CC2)=O)CC2CN(C(C3(O)CCC3)=O)CC2(C)C1 N1(C(CCCC(=O)NC)=O)CC(C)CN(C(=O)CC2CCCCCCC2)CC1C C1(C(=O)NC(C)CCCNC(=O)C=Cc2nccs2)OCCOC1C C12(C(N3C(CCC#C)CCC3)=O)C(NC(c3nccnc3OC)=O)C3CC1C2C3 Cc1c(C(=O)NCC2(CO)CCN(C(=O)CCn3ccnn3)C2)cccc1O C(=O)(C(F)C(F)(F)F)NCCOCCC(=O)NCC(C)(O)C1CCC1 c1(N2C(CCNC(c3ccc(COC)[nH]3)=O)CCCC2)nc(C)nc2[nH]ccc12 N1(C(=O)NCC2(OC)CCCOC2)C2CCC1CC(c1cnn(C)c1)C2 CC1(CNC(c2cnc3n2CCC3)=O)CN(C(=O)CCC2CC2(Cl)Cl)CCO1 c1(C(N2CC(NC(COCC(C)C)=O)C(CC(C)(C)C)C2)=O)ccc(O)nc1Cl Cc1[nH]nc2ccc(C(=O)N(C3CCC(NC(c4ccc(F)nc4)=O)C3)C)cc12 c1(SC)cccnc1C(=O)N(C)CC1CCN(C(=O)C2=CCCS2)CC1 C1(O)(CNC(C(C)=CC)=O)CCCN(C(=O)C(C(C)C)NC(=O)OC(C)C)C1 c1(C(=O)NC2C(NC(C=C(C)C)=O)CCC2)sc2nccn2c1C C#CC1CCCCN1C(C1(OC)CCN(C(=O)CCc2cncs2)C1)=O C1(C(=O)NCC(CC)NC(=O)Cc2ccccc2F)CC1C1CCCC1 N1(COC(c2ccc(C(F)(F)F)nc2)C)CCC(O)(C(F)(F)F)C(O)C1 CC1CCC(CNC(=O)CC2CC(C)(C)C2)CN1C(=O)CCOCCN(C)C CC1(C)CN(C(C2(C3(C)CC3)CC2)=O)CCC1C(N1CC(C(N)=O)C2(CC2)C1)=O Cc1ccc(CC(N2CCC(N(C(=O)C(C)C3(O)CCC3)C)C2)=O)s1 C(=O)(CC(C)(C)C(F)F)NC1C(C(N2CCCC(OCC#C)C2)=O)COCC1 N1(C(C2(CC#C)CCCO2)=O)CCC(C)C(CO)C1.c12ncnc(OC)c1N2 CC1CN(C(c2cscn2)=O)CC(C)C1NC(=O)CN1CCN(C)CC1 N1(C(c2c(C)ccnc2C)=O)CC2COCCC2(NC(c2nn[nH]c2Cl)=O)C1 c1(CN2C3CN(C(C=C(C)C)=O)C(C3)C2)c(C)c(C(=O)C(C)C)n2ccccc12 c1(N(C)C)ccc(C(CNC(=O)COCc2nccn2C)C(F)F)cc1 C1(NC(CC=CC)=O)CCCC12CCN(C(c1cc(CC)on1)=O)CC2 C1(c2nc(CC3N(C)CCC3)nn2-c2cccc(Cl)c2)CCc2nncn2CC1 c1(C2(C(=O)OCC(=O)Nc3cnccn3)CC(F)C2)ccccc1F N1(CC(S(C)(=O)=O)NC(=O)CN=[N+]=[N-])CCC2(O)CCCCC2C1 C1(C(=O)NCCOCCC=C)CCN(C(=O)C#CC(C)(C)O)CC1O c1(C(N2CCC(NC(C(C=CC)O)=O)C(F)C2)=O)cc(N=S(C)(C)=O)ccn1 C1(NC(c2c(C)cno2)=O)CC2CC(C1)N(C(c1ccn3ccccc13)=O)C2 c1(C(N2C(CN(C(=O)C(F)(F)C3CCC3)C)CCCC2)=O)ccc(N)c(Cl)c1O C1(NC(C2C(C)(CC)C2)=O)CCC(N(C(=O)CCc2cn(C)nc2C)C)CC1 N(C1CN(C(C2(CO)CCOCC2)=O)Cc2ccccc21)C(C=NOC)=O c1(C(=O)NCC2CCN(C(C(CC)C(C)(F)F)=O)C2)cc2n(n1)CCNS2(=O)=O C1(CNC(CS(=O)(=O)NC)=O)CC(C)(C)CN1C(=O)C(=O)C(F)(F)F C1(NC(=O)Cc2c(F)cccc2F)CC2CC1N(C(=O)CC(O)C1CCCC1)C2 c1(N2CC(C)C(C)(CO)C2)ncc(S(=O)(=O)NCc2ccns2)cc1Cl CCC(CC(=O)NC(C1CCOCC1)C)NC(C1(COC)CCCC1)=O C1(C(=O)NC(C)Cc2ccncc2)(CNC(=O)CNc2ncccn2)CCCCC1 C1(C(=O)NC(C(C)C)CNC(C2C=CCCC2)=O)COc2ccccc2O1 Cc1cc(Cl)ccc1C(=O)NCCC(C)N(C)C(C1CCN(C)C1C)=O CCCCCC(F)C(=O)N1CC=CC1(C(=O)NCCCCCCCO)COC C1(COC(C2CCCOC2)=O)CCN(C(=O)C=Cc2ncc[nH]2)C(=O)CO1 n1(CC(=O)NCC2N(C(c3c(OC)n(C)nc3)=O)CC(F)C2)cc(C)ccc1=O N1(C(C(C)c2cccs2)=O)CCC(C)(C)C(C(=O)NC2(C)CC(C)(C)C2)C1 C1(C(=O)NC(C2(C(=O)NCCCCc3cnc[nH]3)CC2)C)CCC(F)CC1 CC1(C)CC(NC(=O)C(C)(C)N2CCOCC2)CCN(Cc2cccnc2)C1 C(CC(C)(C)C)(C(=O)N1CCCCC1CCC(=O)NCCCOCC(F)F)OC c1(C(=O)NCC(C)N(C)C(c2ccc(F)s2)=O)cccc(-n2cccn2)n1 C1(C(=O)NCCC2(CNC(C3(CC#C)CCC3)=O)CC2)CC2(C1)CC(F)C2 CN1CCC(CN(C(=O)CSc2ccnn2C)C)CC1 N1(C(C2CSCCS2)=O)CCNC2(CCNCC2)C1 N1(C(C)C)C(=O)CC(NC(=O)CCc2cccn2C)C1c1ccc(Cl)c(F)c1 c1(C(=O)OC(C)C(N2CCCC(N(C)C)C2)=O)sc2cc(Br)ccc2c1Cl c1(C(=O)OC)ccc(NC(=O)NCC2(c3cccs3)COC2)c(Br)n1 C(=O)(C(C)CC(C)C(C)=O)N1CC2C(C(=O)NCc3ncc(CC)s3)C2C1 CCCCC(C(=O)NCC1(F)CN(C(=O)Cc2c(F)cccc2F)C1)N(C)C N1(C(C2CCN(C(C(CC)C)=O)C(CC)C2)=O)CCC2CC1C(=O)O2 N1(C(CC(C)n2ccnc2)=O)CCN(C(c2cc(N)ccc2Br)=O)CC1C C#CC(C)CN=C(NC(C)C)N1CCC(c2ccc(OCC)cc2)C1 c1(C(=O)NC2CCC3CC2CN3C(=O)CCCCF)cnc(O)c([N+](=O)[O-])c1 CN1CC2(CCN(C(C3CCC4(CCNCC4)C3O)=O)CC2CO)C1 c1(-c2cc(C(=O)NCCCNC(C3C(C)(C(C)C)C3)=O)no2)ccccc1F C=CCC(C(=O)NC1(CNC(c2c(CO)cc[nH]2)=O)CCCCC1C)C(C)C c1(OC)cccc(C(O)C(=O)NCC(CO)NC(c2sccc2C(F)F)=O)c1 C(CC(C)C(=O)NC(CC1CC1)C(=O)N(C)Cc1cnnn1C)=CC N1(C(C(CC=C)(C)C)=O)CCC(C2CCN(C(c3coc(C)n3)=O)C2)CC1 Cc1nn(CC(=O)NC(c2nc(C(=O)NCC3C4COCC34)co2)C)c(=O)o1 C=C=CC(C)C(=O)NCc1ccccc1CNC(=O)CC(=C)Br C1(CNC(c2onc(CC)n2)=O)CN(c2nnn(C)n2)CCCO1 CC(C(=O)NCCCOCCOCCC1(C)CC1C)OC(C)(C)C.O c1(C(N2CCC(C(=O)NC(CCC#C)C3CC3)C2)=O)cc(COC)ccn1 C(C(CC1CC1)C(=O)NOCCCO)NC(C1CN(C)C(=O)C1)=O C1(CC(=O)NC2(C)CC2)CC(NC(c2ccc[nH]2)=O)C1(C)C N1(C(c2c(CC)cccc2)=O)CCC2(CCOC2)C(CNC(C2(C)CCC2)=O)C1 N1(C(c2c(C)scc2)=O)CCOC(CC(N2CCC(C(F)(F)F)C2)=O)C1 C(C(F)(C(=O)NC1CC2(CCCO2)C1)C(C)C)NC(c1cc(CC)[nH]n1)=O CC1(C)CCCN(C(=O)C#CC2CC2)C1C(=O)NC(CO)C(=O)OC C(=O)(C(C)(C)CNC(C1COC(CNC(=O)C(c2ccccc2)C)C1)=O)NCC N1(CC(O)C2(c3ccncn3)CC2)CCN(CCOC)CC1 c1(C)cccc(OC)c1.C12(C(N(C(CC)C)CC)=O)CC(n3cc(CCO)nn3)C1C2 C1(C(F)(F)F)(Cc2cn(C(C)C(=O)NCCCC3CCC3)nn2)CCCC1 c1(N(CCCNC(C2(COC)CCC2)=O)C(C)C)nccc(C#N)c1[N+](=O)[O-] C1(CCC2N(C(CCOCC#C)=O)CCC2)CCCCN1C(C1(Cl)CC1(F)F)=O C1(CC)C(C)CCCN1CC1(c2ccc(Nc3ccccc3)cn2)CCCCC1 C1(C(=O)NCC2(OC)CN(C)C2)N(C(=O)C2=C(C)CC2)CC12CCCC2 C(=O)(CCCC(=O)N1CC2CC1(C(=O)Nc1cc(C)cnc1O)C2)OCC c1(CC)ncc(C(=O)NCCC2CCN(C(=O)Cc3ccsc3)C(C)C2)c(C)n1 N1(C(C(CC#C)O)=O)CCN(C(=O)CC2CC(O)C2(C)C)C(C#C)C1 N1(CC(=O)N(C)CC2CC3CCC3C2)CCC2(CCCN(C)C2)CC1 C1(C(=O)NC(C(=O)NCC)C)CC1C1CN(C(c2cc(C)c(C)cn2)=O)C1 c1(C(N2CCCC(N(C(Cc3cnc(C)[nH]3)=O)C)CC2)=O)cc(N)c(Cl)c(O)c1 c1(C(C)(C)OC)nc(=NCC(C2CC2)NC(c2cnc3cnccc3c2)=O)s[nH]1 C1(CC)(CC)CC(NC(C2C(Cl)(Cl)C23CC3)=O)CN1C(=O)CNC=O c1(SC(C)C(N2CCC(NC(=O)COC3CCC3)C2C)=O)ccccc1Cl c1(CNC(=O)CC2CCCC(C(F)(F)F)O2)nc2cc3c(cc2[nH]1)OCCO3 C1(C(=O)OCC)CN(C(=O)Cc2ccc(Br)cc2[N+](=O)[O-])CC2(CCC2)O1 c1(C(N(C)CC2(CNC(C(C)n3cncn3)=O)CC2)=O)ccc(CO)s1 O=C(C1=CC2(CCN(C(C3CCSC3)=O)C2)C1)NCc1cc(CO)ccn1 CC1CN(C(C2(C)CC(O)CN2C(C23CSCC2C3)=O)=O)C(C)C(C)(C)O1 c1(C(N(C2CN(C(c3c(CC)nco3)=O)C2)C)=O)cccc(N2CCNC2=O)c1 C(C)(C(=O)C(F)(F)F)OC(C(CCN(C)C)NC(C)=O)=O C(CC(F)F)(C(=O)N(C)CCc1ncccn1)N(C(c1nc(C)oc1)=O)C C1(C#N)(CC(=O)NC(CN(C(C(C)OCC)=O)C)C)CCCCC1 C#CCCCCC(=O)NC1(C)CCN(C(c2cc(OC)ccc2N)=O)CC1 N1(C(CNC(c2c(CC)nn[nH]2)=O)=O)CCC2C(CCN2C)C1 C1(C)(CNC(c2cc(C)cc(O)n2)=O)COCCN(C(=O)C(C)C2CC2)C1 N1(CC2OCC(C)(C)C2)CCC2(NC(c3cc(C(F)(F)F)ncn3)=O)CCCC12 C1(CN(C2CCOC2)CCC#N)CCC2(CCCC2)C1 N1(C(c2c(CC)nccn2)=O)CCCC(NC(=O)CC2CC2CC)CC1 N1(C(C(=CC2CCCC2)C)=O)C(CC(=O)NCC(O)CC(F)(F)F)C2CCCC12 C1(CN(C)C(c2csnn2)=O)CCCCN1C(c1ncncc1Cl)=O c1(NC(C2N(C(C(C)OCC=C)=O)C(C)CC2)=O)ccc([N+](=O)[O-])cc1CO N1(C(C(F)=CC)=O)CCN(C(c2cc(C(N)=O)ccc2C)=O)C2CCCCC2C1 N1(C(CCOCC#C)=O)CC2CCC2(NC(c2cccc3sncc23)=O)C1 c1(C(=O)NCC2CC(NC(C(CC)N(C)C)=O)C2(C)C)ccc2c(c1)CCN2 N1(C(CC=CCC)=O)Cc2n[nH]cc2C1C(=O)NOCCC1CC1 c1(C(=O)NCC(CC(C)C)NC(=O)C(C)CF)c(O)cc(F)cc1F C1(CNC(c2ccccc2F)=O)CN(C(C2(O)CCC2)=O)CC1(F)F C1(CNC(CCCC#C)=O)CN(C(=O)CN2CCCCC2=O)CC12CCOCC2 C(=O)(N1CCCc2ccnn21)C12C(NC(=O)CC(Cl)Cl)C3CC1C2C3 C1(NC(C=CCCC)=O)C=CCC(C(N2CCOCC2CCC)=O)C1 C=C=C(C)CC(=O)NC(C)C(C(C)C)NC(c1cc(OC)n(C)n1)=O C1(C(N(C(C)(C)CC2CCC2)CCC)=O)(CCC(C2CC2)C2CC2)CC1(C)C C1(CN2CC(F)CC2C=O)CCC(CO)CC1.N1(CC)CCC(N2CCCC2)CC1 C=CCCC(C(=O)NCC1SCCS1)NC(=O)CCSCCC S(=O)(=O)(c1ccc(Br)cc1NC1(CO)CCOC1)N1CCCC(N(C)C)C1 c1(N2CCC(NC(CCC)C(=O)OC)C2C)nnc(C)cc1C(=O)OC(C)(C)C c1(C(=O)OCC2C=CCC2)cc2c(F)c(F)c(Br)cc2[nH]1 N1(C(c2cc(C(C)C)no2)=O)CCC(C(F)F)(CNC(C2C=CCCC2)=O)C1 n1(C2CN(C(C3(C)CS(=O)(=O)C3)=O)C2)ncc2c1CN(C(c1n[nH]cc1Cl)=O)C2 C1(C(=O)NCC2(NC(C3CCS3(=O)=O)=O)CCC2)(OCC)CCCCCC1 CC(C)C(O)CC(=O)N1CCC(C(=O)NOC2CCN(C)CC2)O1 c1(-c2c(NC(c3nccnc3Cl)=O)csc2)cccc2ncnn12 c1(NC(Cc2nc(Nc3ncc(C(=O)OC)s3)sc2)=O)c(Cl)c(C(C)C)nn1C Cn1cc(C(=O)N(C2CCCN(C(=O)CC3(C#N)CC3)C2)CCF)cc1Br C12(C(N(CCC)CC)=O)CCCC1CCN2C(c1occc1COC)=O N1(C(CCC=C=C)=O)CC2(CCN(C(c3cnc(Cl)s3)=O)CC2)C1 N1(C(c2c(C#C)c[nH]n2)=O)CCCOC(CCNC(c2cc(C)co2)=O)C1 O=C(C#CC1CCCCO1)NCC(C1CCC1)NC(c1ccc2sccc2c1)=O C#CCC(C(=O)OC)NC(=O)CC1C(NC(C2CC2(Cl)Cl)=O)CC1O c1(C(=O)NCC(C)C(=O)NC2CC(O)C(O)C2)cnc(S)nc1 c1(OC)c(C(=O)NC(C(=O)NC2C3CCCCC23)c2cccs2)cnn1C C1(C(=O)NC(C(=O)Nc2c(OC)ccnc2)(C)C)CC2COCC2C1 CC1CC(C(=O)N2CCC=C(CNC(C3CC(CF)C3)=O)C2)=NO1 C(N=c1nc(N2CCC(F)(c3cccs3)CC2)c2c([nH]1)CSC2)C1C(C)(C)C1 N1(C(C(C)CC(F)(F)F)=O)CCC2(CC1)CCN(C(C1CC3CCC3C1)=O)C2 C(C1=CCN(C(=O)C(O)CCN(C)C)CC1)NC(c1cc(C(C)C)[nH]n1)=O c1(C(=O)NC(CNC(CC(CC)SC)=O)C)cc(C)nc2c(C)cccc12 c1(NC(c2nc(CCOCC)oc2)=O)cccc(NC(=O)COC2CC=CC2)c1 c1(C(C(=O)NC2CC(F)(F)C2)N(CC(C)(C)C#N)C)nnn(C(C)(C)C)n1 C(CCC)(C(=O)N1CCC(N(CCO)C(C2CC(F)C(=O)N2)=O)CC1)=CCC CC(C)(CNC(c1cc(O)ncc1F)=O)CC(=O)NC1CNC(=O)C1(C)C C12(NC(c3cn[nH]c3)=O)CCOCC1CN(C(c1ccc(=O)n(CCO)c1)=O)C2 N1(C(C(CC2CN(C(COCC=C)=O)C2)F)=O)CCOC(COC(C)=O)C1 c1(C(=O)NCC2(OC)CN(C(c3cc(C)cc(C)n3)=O)C2)cc(Cl)c(F)cc1F C1(C(N(C2CCN(C(C3CCCOCC3)=O)C2)CCO)=O)CC2(C1)CC(F)(F)C2 c1(OC)c(C)cc(C(=O)NCC(O)CCNC(=O)C(C)n2cnnn2)cc1Cl C12(NC(C(CC)COC)=O)CC3CCC(C1C2)N3C(=O)CCc1c(C)n[nH]c1C CCCCCC(O)C(=O)N1CC(C(N2CC=C(COC)CC2)=O)C(C)(C)C1 Nc1ccc(C(=O)NCC2CC(NC(c3ccon3)=O)C2)c([N+](=O)[O-])c1 C1(NC(C(=O)NC(C)C)=O)CCCCN(C(=O)CCCC2(C)NC(=O)NC2=O)C1 N1(C(c2c(C)n[nH]c2)=O)CCN(C(C2CCCC2(F)F)=O)CC1c1cn[nH]c1 N1(C(Cc2ccc(C)o2)=O)CCCC(NC(=O)CNC(c2ccoc2C)=O)CC1 O=C1CC(NC(=O)C(c2cccnc2)NC(=O)CN2CCCC2)CO1 N1(C(=O)CC2=CCCC2)CC2COCC2(C(=O)NCc2ncoc2C2CC2)C1 C1(C(N(CCC(=O)NC2CCOCC2F)CC=C)=O)CCC(=O)N(C)C1 CCCCCC(C)(c1nnnn1C1COC1)NCC1CC2(CCC2O)C1 C(=O)(CCCC(=O)N1CC(C(=O)NCCC(C)CC)C(C)(C)C1)OCC CC1CN(C(c2cncn(C)c2=O)=O)CCCN1C(C1CCCCCC1(F)F)=O C1(CNC(CCNC(=O)OC)=O)CCCCN(C(C2C=C2C)=O)C1 c1(SC(C(=O)NCCN(C(C(C)=C2CCCC2)=O)C)C)ccc(F)cc1 C(=O)(C1=COCCC1)NC1C=CC(CC(=O)NCC2=NOC(C)C2)C1 c1(C(=O)NCCCOc2c(Cl)ccc(C)c2)nncc2ccccc12 Cc1nn(-c2cccc(F)c2)cc1C(=O)N(C)CCN(C)C(C1CC1[N+](=O)[O-])=O c1(C(=O)NCC2C(NC(C(C)OCCCC)=O)COC2)nccc(Cl)c1Cl C(=O)(CCCC=O)NCC(=O)NCCOCC.C1(C)(CC)CCCC1 N1(C(CCCSC)=O)CC2CC(CNC(c3ccc(=O)n(C)n3)=O)C2C1 C1(CNC(C(CC)N(C)C)=O)CN(C(c2cc(F)c(O)c(F)c2)=O)CC(C)(C)O1 c1(C(=O)NC2CC3CC2CN3C(c2cccc(=O)o2)=O)cc2c[nH]cnc-2n1 CCCC(CC(=O)OC)C(=O)NC1CCN(C(C2CCSCC2)=O)C1C Cc1cc(OC(C)C(=O)NC2CCOCC2NC(=O)C2=CCOCC2)ccc1Cl C1(COC)CN(C(c2ccncc2C(F)F)=O)CCN1C(=O)C(C)N1CCC1 C(C)(CSC)(C(=O)NC1(CO)CCC1)NC(C(C)OCCC=C)=O c1(C(=O)NCC(C)(C)CNC(=O)C(C)(C)c2cncnc2)cccc2c1OCC2 N1(C(CS(C(C)C)(=O)=O)=O)CCC2C(CCCN2C(C2CC(=O)C2)=O)C1 c1(CCC(=O)NC(CNC(CCSC)=O)C(C)C)ccc(C(C)C)cc1 CCC(F)(F)CC(=O)NCc1ncccc1C(=O)NCC1(CO)CC1(C)C N1(C(c2n(CC)c(O)nc2)=O)CC(CN(C(=O)Cn2nnnc2C)C)C2(CC2)C1 N#Cc1ccc(NC(C2CN(C(=O)Cc3ccc(Br)nc3)CCN2)=O)cn1 N1(C(CNc2ccc(C#N)cc2)=O)CCN(C(=O)CCn2ccnc2)CC(O)C1 C1(NC(C2CCN(C(C=CCN(C)CC)=O)C2)=O)CC2CCCCN2C1 Cc1ccc(C(N2CC3CC2CN3C(c2ccc(O)c(C(C)C)c2)=O)=O)c(C)c1 CCCCC(CCCC)C(=O)NC1(CNC(C2CC(F)CN2C)=O)CC1 C(=O)(C1=CC2C=CC(C1)C2)NCC1CC(NC(=O)C(N2CCCC2C2CC2)=O)C1 C(C(C)(O)CC(=O)NCC1(F)CCN(C(=O)C=CC2CCCN2C)CC1)OC c1(CC)cc(C(N2CCC(CO)(NC(=O)C(O)C(C)C)C2)=O)cc2c[nH]nc12 c1(OCC)ccc(C(N2CCCC2C(C)(C)NC(=O)Cc2ccno2)=O)cc1 CC1=C(C(=O)N2CC(C3CN(C(c4ccc(C)s4)=O)C3)C2)COCC1 C(CC)(CC)(CCNC(=O)CC1CCCC(C)(C)C1)NC(CC(=O)NCC#C)=O c1(CC)cc(F)c(C(=O)NCCNC(=O)CCc2cnc3ncccn23)cc1F CCC(C)(CO)C(=O)NCC1CCN(C(c2c(C)nn(CCCC#N)c2Cl)=O)C1 c1(C(N2CC(C(C)(C)O)C2)=O)c[nH]nc1CNC(=O)CCC1CC1(C)C N1(C(c2c(C)nc(COC)s2)=O)CC2CCC(C1)N2C(C1(OC)CC(CF)C1)=O CC(C)C(O)C(C)C(=O)NC12CC(CNC(c3cnc(O)cc3O)=O)(C1)C2 N1(C(C2(CC(C)C)CC2)=O)CCC(C)C(CNC(=O)CC2(C#N)CC2)C1 CCC(CC)CC(F)C(=O)NC1CC1NC(c1cccc(F)c1C)=O Cn1c(C(=O)NC2CC(NC(c3sccc3C#N)=O)CC2O)cnc1O C1(CCC)(NC(c2cc(-c3ccccc3)cs2)=O)CCCNC1 C=Cc1cncc(C(=O)N(CCNC(=O)C(C)CC(F)F)CCOCCO)c1 c1(N2CCN(C(C)C)CC2)nc(=NCCCCCCO)[nH]c2c(F)cc(F)cc12 C1(C)(C(=O)NC(CNC(c2c(C(C)C)[nH]cc2)=O)C(C)C)CC(C#N)C1 C1(C(N2CC(NC(c3c(NC)scn3)=O)(COC)C2)=O)CCC(=O)N(C)C1 c1(NC(C2CCN(S(Cc3cccc(C)c3)(=O)=O)CC2)=O)c(C)c(C)nn1C c1(OCCOC)ccc(-c2ccccc2N2CCC(O)C2)cc1 N1(C(COC(CC)C)=O)CCC(O)C(N(C(=O)C(C)Cn2ccc(C)n2)C)C1 c12ncc(Cl)c(n1)C(=O)N2.c1(C(N(CCCCC)C(=O)OC)C)ccncc1 CCCCCCCCN(C(=O)C(C(C)CC)N(C(=O)C(C)=C1CC1)C)C CN1CCC(NC(=O)CSCCNC(=O)CCc2cnccn2)C1=O CCCC(C1CC1)NC(=O)C(C1CCCO1)NC(=O)CNC(C1CC1C)=O.C1CCC1 Cc1cc(CNC(=O)CN(C(=O)CN2C(C)CCC2C)C(C)C)cc(O)n1 c1(C(=O)Nc2cc(I)ccc2F)n[nH]c2c1CN(C(c1ccc(O)nc1)=O)C2 N1(C(C(N)=O)=O)CCC2(CCCCN(C(C3CC4CC4C3)=O)C2)C1 C#CCCCCCC(=O)NC1CC2(C1)CC2NC(C12CC(C#N)(C1)C2)=O N1(C(CN(CC)CC)=O)CC(NC(=O)Cc2cc(Cl)ccc2Cl)CC1(C)COC N1(C(C2(CCC)CC2)=O)C(C(N2CC(C)OCC2CC)=O)CCC12CC2 C1(N(C(c2c(C)coc2)=O)C)CN(C(=O)CCCc2csc(=N)[nH]2)CC1O N1(C(c2c(OC)cccc2)=O)CCC(C2(NC(=O)C(C)P(C)(C)=O)CC2)CC1 C1(NC(C(C)NC=O)=O)CCCC1NC(C1CC1c1cccnc1)=O C(C)(CO)(CC(C)C)NC(COC1CC(NC(c2cc(C)sc2)=O)C1)=O Cc1sc(CC(=O)NC(CCN(C(=O)CNC=O)C)C(C)C)cc1Br C(=O)(C(C)(C)OC(C)C)N1CC(C(NOC(COC)C)=O)C1 Cc1ccc(C(=O)Nc2c[nH]nc2C(=O)NCCN(c2ccccc2Cl)C)cc1 c1(C(=O)NCC(CNC(C2CC3CCCCC23)=O)OC)cc(O)ccc1F c1(NCC2CC2)cc(OC)c(OC)c(O)c1.c1(NCCOC)cccc(OC)n1 C(=O)(CCCCCCCO)Nc1ccc(NC(=O)CCN2CCCC2)cc1F N1(C(C2CC(CC)C2)=O)CCC(NC(c2cc(CO)[nH]n2)=O)C1C(C)C c1(SC)ncccc1NC(=O)CC(O)CNC(c1cnc(C)s1)=O C1(C(=O)NC(CCCC)CO)CCCCN(C(=O)CC2CCC(C)CO2)C1 C(C(=O)NCC1(n2cccn2)CC1)(C(C)(C)C)n1cc(CC(C)O)nn1 C(=O)(C(C)CC(=O)N1CCC(C)C(NC(c2oncc2C)=O)C1)OC N1(C(C(C)Oc2cccnc2)=O)CC2(NC(=O)C(=CC3CCCCC3)F)CC1C2 C(=O)(C(C)(C)CC(C)C)NC1CCCC(NC(Cc2cc(C)c(CO)cc2)=O)C1 C1(C(=O)NC(CNC(c2ccc(C)s2)=O)C2CCC2)COCCN1C c1(C(=O)NC2C(C(N3C(C#N)C4CC4C3)=O)CCCC2)n[nH]c2ccccc12 N1(C(CN(CC)CC)=O)CCN(C)C(CNC(=O)C(CC2CC2)CC2CC2)C1 N1(C(C(C)=C2CCCC2)=O)CCC(C2(NC(c3cc(Br)n(C)c3)=O)CC2)C1 C1(SC)CCCCN(C(=O)C(C)(C)C(C)NC(=O)CC2CCCC2)C1 N1CCS(=O)(=O)CC1.C1(C(=O)OC)(OC)CCN(C(=O)NCc2cccc(Cl)c2)C1 C(CCCCCC(=O)N1CCCC12CCOC2)NC(=O)COCC1CCOC1 c1(C(=O)NC(C)CCCNC(c2ccoc2C(F)(F)F)=O)nc2ncccn2n1 CS(=O)(=O)c1cccc(S(=O)(=O)NNC(=O)CNCCOc2ccc(I)cc2)c1 C1(CNC(=O)Nc2c(OC)scc2)CCC(=O)N(c2ccccc2)C1 c1(CCN(C(Cn2cc(C(C)O)nn2)=O)CCn2cnnc2)ccccc1Cl Cc1sc2ccccc2c1C(=O)NCCCN(C(=O)CC1(O)CC1)C(C)C c1(CC)ccccc1C(=O)NC1(CC)CN(C(c2cccc(F)c2)=O)C1 C1(C(=O)NC2C(CNC(c3cc(C)no3)=O)COC2)CNC(=O)CC1(C)C c1(C(=O)NCCC(C)N(C(=O)CC(C)P(C)(C)=O)C)cc2ccc(Cl)c(F)c2[nH]1 N1(C(C(CC=CC)C)=O)CCC2(CC2)CC1C(=O)NCC1(CO)CC(C)(C)C1 C1(C(=O)NCCSCCC=C)CCN(C(=O)CCC(C)OC)C12CC2 C1(C(N(C2CCN(C(=O)C(c3ccc(Br)s3)=O)C2)C)=O)CCCN1C C(C(O)(CNC(C1CCC1NC(=O)C(C)(C1(C)CC1)OC)=O)CO)OC Cc1noc(N)c1.c1(-c2nc(C(C)SC)on2)cccc(NC(=O)OC(C)(C)C)n1 CC1CC(CNC(=O)CCCNC(C2OC3CCC2C3)=O)CC(C)C1 CCC(O)C(C)(C)C(=O)NCC(C)(C)CNC(C1(c2cccc(F)c2C)CC1)=O c1(C(N2C(CN(C(c3cnc(Cl)[nH]3)=O)CC)CCC2)=O)cnc2c(c1)CCC2 c1(C(C)=O)cnn(C)c1F.c1(C=O)sccc1OC(F)F.C12CC(C1)COC(=O)CO2 CC1(C#CC(=O)NCC2CCCC2NC(c2cc3ccsc3s2)=O)CCCO1 C(=O)(C1=NNC(=O)CC1)N(CCCNC(C1CC=CCC1)=O)CC c1(C(N(CCN(C(C2(CC)CCC(O)CC2)=O)C)C)=O)ccc2oc(O)nc2n1 C1(C(N(CCC(=O)N(C2CC3CCC2O3)C)C2CC2)=O)C2CCCCC12 C(=O)(C(C)(C)CO)N(CCNC(C1(C)CC1)=O)CC C1(CNC(C(C2CCN(C(c3cc(C(C)=O)on3)=O)C2)(C)C)=O)CCC(=O)NC1 N1(Cc2cn(CCN(C(=O)C(C)SC(F)(F)F)CC)nn2)CCS(=O)CC1 C(=O)(C(C)(CC)C(N)=O)NCC(CC=C)NC(=O)C#CC(C)(C)C C1(C(N2CC(NC(CSc3n(C)ncc3)=O)C2)=O)CCCN(c2cccs2)C1 CCCC(CC(=O)N1CCC(OC2(O)CC2)CC1)c1ccccc1 N1(C(C(C)n2cnnn2)=O)CC2(CCCCN(C(=O)C=CBr)C2)C1 C1(CNC(C=CCCC)=O)CCN(C(C2CCC(CCC)CC2)=O)C(C)C1 C1(C(=O)NCCOCCN(C)C(c2[nH]cnc2C#N)=O)CCc2nnnn2C1 c1(C(C)NCCN(c2cc(F)cc(F)c2)C(=O)C2CC2)ccc2c(c1)CNCC2 CCCCCCC(C)CC(=O)NC1(COC)CCN(C(c2oncc2C)=O)CC1 N1(C(CC(C=C)C)=O)CCCC(COC)(NC(=O)Cc2cccc(C)c2)C1 c1(OC)cccc(CC(=O)NC(C)C(C)NC(c2c(C(C)C)n[nH]c2C)=O)c1F C1(C(N(C(C)C(=O)NC(C)CC(F)(F)F)C)=O)(CO)CCCCC1 c1(-n2c(C(C)S(C)(=O)=O)nc(C(C)O)n2)ccccc1S(N)(=O)=O C(F)(F)(C(F)(F)F)OCCN(CC(=O)NC1CC12CC2)C(=O)CC1CCCCC1 CCC(CC(=O)OC)NC(C1CCCN1C(c1c(C)cnn1CC)=O)=O C#CCC(C)(C)C(=O)NCC12CCC1CN(C(=O)C(c1cccc(Cl)c1)(F)F)C2 CCC(C)CCCCC(=O)N1CCCC2CN(C(c3ccc(C(C)=O)s3)=O)CC12 N1(CC(N2CC=CC(NC(C(c3ccccc3Cl)C)=O)C2)=O)CCCNS1(=O)=O c1(SC)ccc(C)c(C(=O)NCC2CCCN(C(=O)Cc3c[nH]nc3C)C2)c1 CC(CC(=O)NCC(C)N(C)C(C1CSCCS1)=O)NC(c1ccccc1)=O C1(C(N2C(CNC(c3c(CC)con3)=O)CC(O)C2)=O)CCCCC(=O)N1 C1(C(=O)NC2CC(CNC(C3CCN(C(=O)OC)CC3)=O)C2)CC(=O)NC1(C)C N1(C(c2cc(C)c(F)cc2)=O)CCN(C(=O)Cc2c[nH]nc2O)C(C)C1C c1(C(=O)NCC(C(C)(C)C)NC(C2C(=C)C2)=O)ccc(OC)c(C)c1OC c1(N(C)CC2CCN(C(C3Cn4c(C)ncc4CC3)=O)C2)nc2ccc(Br)cc2o1 C1(O)(CN(C(c2cc(OC)ncc2)=O)C)CCN(C(c2cc(C)c(C)o2)=O)CC1 CCC(CC)(CCNC(c1cc(O)cs1)=O)NC(C1CC1C(=O)OC)=O CCC(CC)(C(=O)N1CC(NC(=O)CCOCC2CC2)C(C)C1)c1ccccc1 Cc1ccc(C(=O)NCCN(C(=O)C(C)N(C)C)CCc2ccccc2)n1C C1(C(=O)NCC(CC)O)CC(O)C(O)CC1CNC(c1ccc(C)cc1OC)=O c1(OC)ccc(C(=O)NC2CCCCN(C(C3(C#N)CCC3)=O)C2)c(OC)c1Cl c1(C(=O)NCC2CN(C(C3CC4CCC3O4)=O)CC2O)cc2cccnn2n1 Cc1cc(CNC(C2CCN(C(C3(Cl)CC3(F)F)=O)C2)=O)co1 N1(C(C(C(C)O)(F)F)=O)CC=C(C(=O)NCC2CC3CC2CC3O)CC1 C1(NC(C(CC)OCC)=O)CCC2(CC1)CCN(C(c1cc3occc3s1)=O)C2 N1(C(C(C2CN(C(C3(C4CC4)CC(=O)C3)=O)C2)OCC)=O)CCC2C(=O)NCC2C1 N1(C(c2cc(C)ns2)=O)CCN(C(=O)CCc2ccc(F)cc2)C(C2CC2)C1 O=C1NC(CNCC2CC2c2ccc(Cl)cc2Cl)=C(C(=O)O)C(c2ccccc2)N1 C1(C(=O)NC(CN(C(c2csc(C)n2)=O)CC)C)COC2COCC2O1 N1(c2nnc(C3CCC(C)O3)n2CC2CC2)Cc2ccccc2OC(C)(C)C1 c1(SCC(N2CC3C(NC(C=CC)=O)C(CC3)C2)=O)ccc([N+](=O)[O-])cc1 C1(F)(C(=O)NC(CNC(CCSCCCC)=O)CC(C)C)CC12CCCCC2 CC1C(C(=O)NCC2(O)CC(CNC(C3(C#N)CCCC3)=O)C2)=NOC1C c1(C(=O)NCC2(NC(C(CC#C)C3CC3)=O)CC2)[nH]c2ccccc2c1Cl c1(C(=O)NC2CN(C(CCc3c(C)n[nH]c3C)=O)C2)c(F)ccc2n[nH]cc12 CC1c2cc(F)c(F)cc2CCN1C(=O)CSCc1ccccc1F c1(C(=O)NC2CC(CNC(Cn3c(C)ncc3)=O)C2)coc2c1C(=O)NCCC2 N1(C(C2(c3cc(C)no3)CC2)=O)CCCC2CN(C(C3CCCO3)=O)CCC12 C1(CCOC)CN(C(=O)Cc2cn[nH]c2)CCN1C(c1cnc(C)n1C)=O C1(CC(N2C(C)(COC)CC2)=O)CN(C(c2cccnc2O)=O)CC1C C1(C(N2C(C)C(NC(=O)CCSC(F)(F)F)CCC2)=O)CCn2ncnc2C1 C1(CC)CN(C(=O)NCC2CCCCN2S(C)(=O)=O)CCO1 N#CC1(C(N2CCOC(CC(=O)Nc3cncc(F)c3)C2)=O)CCCC1 c1(N2C(C(=O)Nc3c(O)cccc3Br)C=CC2)ncnc2ccccc12 c1(C(=O)NC(CCCNC(CN(CC)CC)=O)C)cc(-c2cc[nH]n2)ccc1F C1(O)(CN(C)C(c2ncsc2C2CC2)=O)CCCC(C)(C)C1 N1(C(C23CC(C)(OCC2)C3)=O)C2CCC1CN(C(C1(C)CCCS1(=O)=O)=O)CC2 N1(C(CC=CC)=O)CC(NC(c2ccco2)=O)CC(C)(C)C1 C(C)(CCCCNC(C1CC1c1cccc(OC(F)F)c1)=O)NC(C=CCC)=O Cc1c(Cl)sc(Cl)c1C(N1CC(C(=O)NC23CCC(CC2)O3)CC(O)C1)=O N1(C(Cc2cc(C)sc2)=O)CCC(CCNC(C2CCC23CCC3)=O)C(F)(F)C1 C(=O)(C1Cc2ccc(F)cc21)NC1CC(C)N(C(=O)CC2(C)CC2(F)Cl)C1 c1(C(=O)Nc2nnc(-c3scc(C)c3)o2)sc2nc(C)nc(C)c2c1C c1(C(=O)NC2CN(C(c3c(C)nccn3)=O)CC(F)C2)coc2ccc(O)cc12 CCC(O)C(C)(C)C(=O)N1CCN(C(c2ccc(N)cn2)=O)C(C(F)F)C1 C(=O)(C(C)(C)C(C)O)NCC1CCCC(CNC(c2c(C)cnn2C(C)C)=O)C1 C(=O)(C1=CC2CCCC12)NC(CNC(CC1C(C)(C)CCCO1)=O)C1CC1 N1(C(CN2CCC(OC)C2)=O)CCC2CN(C(c3n[nH]c(C)c3C)=O)CCC2C1 c1(C(N2CC(CNC(C(CC=C)C)=O)(COC)C2)=O)cnc2n1CCOC2 c1(C(=O)NC(C)CN(C(=O)C(C)(F)C(C)(C)F)C)cccc(S(C)(=O)=O)c1 CC1OC(=O)NC1C(N1CC(CNC(=O)C(C)(C)c2ccsc2)C(O)C1)=O c1(CN(CCSC)CC)cc([N+](=O)[O-])cs1.C12(CC1)C(=O)NC2 C1(C(=O)NC2C(CNC(CCc3ccc(CC)cc3)=O)CC2)CC2C(C1)C2(C)C c1(C(=O)NC2C(CNC(c3on(C)c(=O)c3)=O)CCC2)cccc2oc(=N)[nH]c12 c1(CS(N)(=O)=O)cccc(S(=O)(=O)NC(C2CCCCC2)CN2CCC2)c1 N1(C(CCC(C)NC(c2occ3c2CCC3)=O)=O)CC(O)CC12CCC2 C1(C2(O)CCN(C(C3(C)CCCNC3=O)=O)CC2)(NC(CCCCC=C)=O)CC1 c1(C(N(CCNC(C(C)NC(CC)=O)=O)C)=O)cccc(C#CCO)c1 C1(NCc2nnc(CC)s2)CCOc2cc(Br)ccc2C1 c1(C(C)=O)ccc(N(C(=O)C(=Cc2ccc(OC(F)(F)F)cc2)C)CCO)c(F)c1 N1(C(C(c2n(C)ncc2)(C)C)=O)CC2CC2(CNC(=O)COC(C)(C)C)C1 C1(CC(N2CC(C)OCC2)=O)Cc2ccccc2CN1Cc1cccc(O)c1 N(C1CCc2c(Br)ccc(C)c21)C(c1cc(C)on1)C N1(C(c2nccc(CC)c2)=O)CC2CC1CCN2C(C1CC1(Cl)Cl)=O Cn1cnc2sc(C(=O)NCC(CNC(=O)Cn3cnc(=N)[nH]3)C(F)(F)F)cc12 CC1CCN(C(c2cc(Cl)sc2Cl)=O)CC1CNC(=O)CCC(C)(C)O c1(CCC(=O)NC2(CNC(COCCOC)=O)CCC2)cccc(F)c1Cl c1(N(C)C)c(NC(=O)NCCn2cnc(CO)n2)c(=O)c1=O N1(Cc2ccc(N(C)C)o2)CC2CCN(C(c3cc(Br)ncc3F)=O)C2C1 C1(c2cn(C(COCC)C(=O)NCCC(F)F)nn2)CC(C)=NN=C1C N1(C(C(C)(C2CC2)OC)=O)CCN(C(=O)CC2CCCC(OC)C2)CC1C CCCC(C)(C)CC(=O)NC(CC1CC1)CC(=O)NC1CCC(F)(F)CC1 C1(C(=O)NC2CC(O)(CNC(c3ccc(C)cc3)=O)C2)(CSC)CC(F)(F)C1 Cc1nc2cccc(C(N3CCN(C(C4CCC(C)(C)CC4)=O)C4CC34)=O)n2n1 CC1CC(=O)NCC1C(N1CC(=C(F)CNC(C2C(C)C2C)=O)C1)=O c1(Cn2ncc(C(C(=O)N(C(CC)CO)C)=O)c2)ccc(C(F)(F)F)cc1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CC(OCC(=O)N(N2C(C)CCC2C)CC)C1 CC1=C(C(=O)NCC2CC2NC(C2(CC3CC3)CCC2)=O)Cn2ncnc2N1C N1(C(C2(C)CC3CC3C2)=O)CCN(C(c2ccccc2Br)=O)CC(O)C1 Cc1nn(C(C)(C)C)cc1C(=O)N(C1CCCN(Cc2ccncc2Cl)C1)C c1(C(=O)NC2CCN(C(c3c(C)cc(CO)o3)=O)CC2)c(C)c(C)cc(C)c1C C1(F)(NC(=O)NCC2(C)ON=C(C)C2)CCCN(C(=O)OC(C)(C)C)C1 CCCC(C)(CCC)C(=O)NCC1CCCCC1C(=O)NCc1ncnn1C CCC1=NOC(C(N2CCCC2CN(C)C(c2cncc(O)c2)=O)=O)C1 C1(C(=O)NC2CC(C)(NC(C3CC3(F)F)=O)C2)CCC(C2CCCO2)O1 C(=O)(CCCCCCS(N)(=O)=O)N(CCC(C)NC(C1CSCCS1)=O)C C(CCC(=O)NC(C)CCNC(=O)CNC(=O)CN(C)C)=CCC=C C=C(CNC(c1cnn(C(C)(C)C)c1)=O)CCNC(=O)CC1OCCC1C N1(C(CCC#C)=O)CC2CCCC2(NC(c2cncnc2C2CC2)=O)C1 N1(C(C(C)c2cncs2)=O)CC2CC1CN2C(c1cn(CC(F)(F)F)nn1)=O c1(C(=O)NC(CNC(c2c(SC)scc2)=O)C(C)C)cc2scnc2[nH]1 c1(C(C)C)noc(C2CC2C(=O)NCCC(F)Cn2cc(C3CCCC3)nn2)n1 C1(NC(C=CCOC)=O)CCN(C(=O)Cc2ccc3c[nH]nc3c2)C12CCCC2 c1(-c2cnc(C(=O)Nc3ccc(C)c(F)c3)nc2)cnc2[nH]ccc2c1 C=CC(CC)C(=O)N1CC(C)(OCC(=O)NC(C)Cc2ccccn2)C1 C=CC(C)(C)CC(=O)NC(C(N1CCCCC(COC)C1)=O)C1CCC1 C1(CC(=O)Nc2ccc(NC(C(C)C)=O)cc2)CCCC2(CNC(=O)C2)C1 c12cccnc1CNC2=O.C1(CC(=O)NC2CC23CCC3)(N(C)C)CCCC1 C1(C(N(C)CC2(O)CCN(C(=O)C=CC(=O)N(C)C)C2)=O)COC(C)(C)CO1 N1(C(=O)CC2(Sc3ccccc3)CCC2)CCN(Cc2ccccc2I)C(=O)C1 C1(C(=O)NCCC=CC)CC2(CCN(C(c3ccc4cc[nH]c4n3)=O)CC2)C1 c1(CN(C)C(C2(CCCF)CC2)=O)cccc(CNC(=O)C=CC2CCOC2)c1 CC(=O)CCN=C(NCc1cc(F)ccc1Cl)N(C)Cc1ccc(Cl)s1 N1(C(CSCC#C)=O)C2CC=C(C(=O)NCc3cc(Cl)ccn3)C1CC2 c1(C2N(C(CC#N)=O)CCC2)ccc(Br)c(Cl)c1 C1(C(=O)NCCC(C)c2cn[nH]c2)(NC(C2CC=CC(O)C2)=O)CCC(C)(C)C1 c1(C(=O)NC2CC3CN(C(c4c(C)nccn4)=O)CC32)cnn2c1CC(C)CC2 c1(OC)ccc(CCC(=O)NCC23CC(NC(=O)CSC)(CO2)C3)cn1 N(C1=NCCCNC(=O)N2CCC(N1)CC2)C1C(C(=O)OC)C1.C(C)(C)(C)O.SC C1(CNC(C(CCC)CC)=O)CC2(CO1)CN(C(c1ocnc1C1CC1)=O)C2 c1(C(=O)NC(CC(C)NC(C2CC2(Cl)Cl)=O)C)ccc(=O)n(-c2ccccc2)n1 C(C(F)CCNC(=O)NC1(n2cc(CO)nn2)CC1)NC(=O)OC(C)(C)C C(=O)(C1CCCc2c(O)cccc21)NC(C)(C)CCCNC(c1ccc[nH]1)=O N1(C(=O)NCc2n(C)c(Br)cn2)CC2CN(C(=O)OC(C)(C)C)CC2C1 CCCC(C(=O)NCC(O)CCNC(c1sc(Cl)c(Cl)c1C)=O)C(C)C CC1(C)C(NC(c2c[nH]c(=S)cn2)=O)CC1C(=O)NCCCC(N)=O C1(NC(c2c(COC)cccc2)=O)CCN(C(=O)C(Br)=C(C)C)CC1C C1(C)(C(N2CC(c3cn(C(C4(OCC)CCC4)CO)nn3)(O)C2)=O)CNC(=O)C1 N1(C(C2CC(C)C2)=O)CC2CC2(CNC(c2ncoc2-c2ccccc2)=O)C1 C1(C(=O)NC2CC(C)(NC(C=C3CCN(C)C3)=O)C2)CCC(F)(F)C1O c1(C(=O)NC2CC3(C(NC(=O)CO)C3)C2)[nH]c2ccccc2c1Cl Cc1cc(NC(=O)NCC2=NOCC2)c2occc2c1 N1(C(CC2(CC)CC2)=O)CC2(CCC2)CC1CNC(=O)CN(CC(C)(C)C)C c1(C(=O)NC2CN(C(C3(CC#C)CCCO3)=O)CC2O)c(C)oc(C)c1C N1(C(c2c(CC)csc2)=O)CC2(CC(C(=O)NCCF)CO2)C1 c1(C(=O)NC2CC(C(C(=O)N(C3CCCC3)CC#CC)F)C2)oc(C)cc1C N1(C(c2ccc(CCC)s2)=O)CC2(CNC(=O)C(F)CN(CC)CC)CC1CO2 c1(C(N(CC(O)CCNC(=O)CNC(=O)Cn2cncn2)C)=O)ncccc1F c1(C(N(CCN(C(CCC=CC)=O)C)C(C)C)=O)cc(OC)cc(OC)c1 C1(C(=O)NC2CCN(CCO)CC2)CN(C(=O)COCCC(C)C)CC(F)(F)C1 N1(C(C(C)(CSC)NC(c2cc(CC)[nH]n2)=O)=O)CCC2(CNC(=O)N2)C1 c1(OCCC#C)ccc(C(N2CC(F)CC2CN(C)C(C2(C)CC2C)=O)=O)cc1 N1(C(CCCSC)=O)CCC2(NC(=O)C=Cc3ccc(OC(F)F)cc3)CC2C1 C=CCC(C)(CC)C(=O)N(CC(C)NC(=O)CN(C(=O)C(C)C)C)CC c1(OC)ccc(C(c2nnnn2CC2CCOC2)NC(CF)C2CCC2)cc1Cl C1(C(=O)NCC(C(C)(F)F)Cl)C2CC3C(C2NC(=O)Cc2ccc(O)cn2)C13 C1(NC(=O)CSC(F)F)CC2CCC1CC2NC(=O)Cc1ccc(O)c(Cl)c1 C#Cc1cccc(CC(=O)NC(C)CCNC(=O)Cc2ccccc2F)c1 c1(OC)cncc(C(N2CC(NC(=O)Cc3ccccc3F)C(CO)C2)=O)c1 c1(NC(C23N(C(c4ccc(OCN)o4)=O)CCC2C3)=O)cncc2ccccc12 n1(CC)ncc(Cl)c1C(N1CC(OC)C(NC(c2cccc(C)c2)=O)C1)=O N1(C(CC2CC(OC)C2)=O)CCCC(N(C)C(c2ccsc2C)=O)C1 CN1c2ccccc2N(CCNC(N2CCC(O)C2c2ccccc2)=O)S1(=O)=O C1(CNC(CC=C)=O)C2CCC(C2)N1C(=O)Cc1cccnc1O c1(C(=O)NCC2(NC(C34CC(F)(C3)C4)=O)COC2)ccc(SC(F)(F)F)cc1 c1(C(=O)NCC2N(C(C(C)SC)=O)CC(F)C2)c(O)nnc2c1COCC2 CC(C)CC(C)N(CCC(C)(C)CNC(=O)OC(C)(C)C)C1CC1 N1(C(C2CN(C(=O)NC)C2)=O)CCCC(NC(C2CC23CCOCC3)=O)CC1 Cc1nc(C)c(C(=O)NCC2CCCN2C(C2CC(C)OC2=O)=O)s1 c1(C(C)N(C)CCN(C(=O)C#CC2CC2)C)ccc2ccccc2c1 N1(C(=O)COc2ccsn2)CC2CCC1CN2C(c1cccc2nonc12)=O c1(C(=O)NC(COC)C(=O)NCc2cocn2)cc2ncccc2[nH]1 C1(CNC(C2C(OC)C2)=O)CCN1C(=O)CCC1CC1(C)C C=CCC(CNC(C1CC1C(F)(F)F)=O)NC(c1cnn(CC)n1)=O c1(C(=O)NC(CC)CNC(C2CC3(CSC3)C2)=O)cnc2scc(C)n2c1=O Cc1cccc2cc(C(=O)N(CC(C)N(C)C(C3CSCC(=O)N3)=O)C)cnc12 N1(C(c2ccc(CC)s2)=O)CCN(C(C)CNC(=O)Cc2ccc(F)cc2)CC1 C1(C(=O)NCC2CCC(CC)O2)CC=CCN1C(C1COCCC1C)=O Cc1cc(C)c2cc(C(=O)NC(C)CC(C)NC(=O)Cc3ccoc3C)[nH]c2c1 N1(C(c2cccc(F)n2)C(=O)NCCCOC)CCCC2(CC=CCO2)CC1 C1(NC(C(C)=C2CCC2)=O)CCN(C(=O)C(=O)C(F)(F)F)C12CCC2 C1(NC(CCCOCC=C)=O)CCOCC1NC(C12CCC(CC1)O2)=O N1(C(c2nccc(CC)c2)=O)CC(C)C(NC(c2cocc2C)=O)C(C)C1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CC(CNC(=O)Cc2nccn2C)C(C(F)(F)F)C1 N1(C(C(C)OCC(F)(F)F)=O)CCN(C(=O)CC2CC=CCC2)C(C(C)(C)C)C1 c1(C(=O)NCC(C(=O)OC)(C)c2ccccc2)c[nH]c2c(C)cccc12 C(=O)(N=c1[nH][nH]c2c1CN(C(=O)CCc1cccc(O)c1)C2)c1c(C)ocn1 c1(C(C(=O)N(CC(C)NC(C(CC)=CC)=O)C)C)ccc(C#N)cc1 c1(CC(N2CCC(Cn3cc(CC(C)C(=O)OC)nn3)C2)=O)c(Cl)cccc1Cl C(CCCC(C)NC(c1ccc(-n2ccnc2)cn1)=O)NC(C(C)SC(C)C)=O C1(NC(COC)(C(C)C)c2nnnn2C2CC(C(N)=O)C2)CC(C)(C)C12CC2 c1(C(=O)NC(C(=O)NC(CC=C)CC(F)F)c2ccoc2)ccn2ccnc2c1 c1(C(=O)NC(CC(C)NC(C2CCSCC2)=O)C)cc2nc[nH]c2cc1N c1(-c2cc(C(N(C3CCC(NC(C4CC(=C)C4)=O)C3)C)=O)sc2)ccc(F)cc1 C1(NS(CC)(=O)=O)CS(=O)(=O)CC1NC1(C)CN(c2ccccc2)C1=O C1(CCNC(Cc2ccc(C)o2)=O)C(C)CCCN1C(=O)CC1CCCC1 c1(C(=O)NC(c2c(C)noc2C)C)cc2ccccc2c([N+](=O)[O-])c1N C(=O)(C1=CC2(CCOCC2)C1)N1CCN(CCNC(=O)CC2CS(=O)C2)CC1 c1(CNC(C2C(CNC(c3ccc(C#C)o3)=O)OCC2)=O)ccc(C)c(O)n1 C#CC1(NC(C2(NC(=O)C(Cl)Cl)CC(F)C2)=O)CCOC1 C(=O)(C(F)(F)C(F)(F)C(F)F)N(CC(CC)NC(c1c(CC)cc(F)cc1)=O)C c1(C(N(CC(C)N(C(C2=NOC(C)C2)=O)C)C)=O)c(Br)ccc(F)c1N C1(NC(C(C)NC(C)=O)=O)CC(F)(F)CC1NC(=O)CC1(C)OCCO1 CCC(O)(CC)CCNC(C=CC1CCCN1C(=O)C(c1cnn(C)c1)=O)=O C1(CNC(C2CC(=C)C2)=O)CC2CN(C(C3CC3c3ccc(C)s3)=O)CC12 N(C1CCCc2c1cnn2CCO)C(CCCC)(C)c1nnnn1CCOC c1(C(=O)NCCC2CN(C(C(CCC)(C)CC)=O)C2)n[nH]c2ccc(OC)cc12 N1(C(C(C)=CC)=O)CC(C2CCN(C(=O)Cc3ccc(O)cc3Cl)CC2)C1 N1(C(CCCN(CC=C)C)=O)CCC2(CC(C(C(=O)OC)NCCCSC)C2)C1 c1(C(=O)NCC2(NC(=O)C=Cc3nccs3)CCOCC2)cc2cccnn2c1 C1(NC(C(C)OCCC(C)C)=O)CCCC1CC(=O)NCC(C)(O)CO C(=O)(CC(O)C(C)C)NCC(C)(C)OCC(=O)NC12CC(CC)(OC1)C2 c1(C(=O)NC2CN(C(Cn3c(C(C)C)nnn3)=O)CC3C2C3)cc(F)cc(N)c1F N1(C(C=CCOC)=O)CCC(C(F)(F)F)C(OC)C1.C12(CCC1)C(=O)N2 c1(SC)ccc(CN(c2nccc(C3CCCCC3)n2)CC(C)C)cc1 C(=O)(C1OCCc2c(O)cccc21)NC(CCN(C(CCCC)=O)C)C(C)C c1(-n2ccc(C)c2)ccc(C(=O)NCC2C=CCN2C(=O)Cc2cn[nH]c2)cc1 c1(C(c2nnnn2CCCOC)NC(C=C)C2CC2)csc(Br)c1 N1(C(C(C)N2CCC2)=O)CC2CCCC1C2CNC(c1ncccc1Cl)=O C(=O)(C1CCc2c[nH]nc21)N1CCC(NC(CC(n2ccc(C)n2)C)=O)C(F)C1 N1(C(CC(C)CF)=O)CCC2(CCOCC2)C(CNC(c2coc(CO)c2)=O)C1 n1(CCCC(=O)N(C2(CCO)CCCCC2)C)cnc(C#N)n1 c1(C(=O)OC(CNC(c2ccccc2)CC#C)C)ccccc1 C12(CCC(=O)OCCc3cc(C)[nH]n3)CCC1CN(C(=O)N)C2.C(C)(C)(C)O N1(CC)CC(C(N2CC(C(O)C(=O)N(C)CC3CCCS3)C2)=O)CC1=O N1(C(=O)C=Cc2ccsc2)CCCC2(C1)CN(C(C1C(F)(F)C13CC3)=O)C2 CN1CCCCC1C(N1CCCC(CCNC(=O)CCCN2CCCCC2)C1)=O Cc1[nH]c(=N)sc1C(=O)NCC(C)(C(C)C)NC(C1CCC(C)O1)=O N1(C(C(=O)NCC(=C)C)c2nccs2)CCCCC(CC(=O)OC)C1 c1(C(N2CC(N3CCNC3=O)C2)=O)cccc(CO)n1.N#CC1CC(N2CC2=O)C1 N1(Cc2nc(C)sc2)CCC2CN(S(=O)(=O)c3ccccc3C(=O)O)CC2C1 C(=O)(CC(C)(C)CC(F)(F)F)NCCC(CNC(c1ncn(C(C)C)n1)=O)(C)C c1(CCC(C)C)ccc(CN(C(=O)C(=O)NC2CCCC2CN)C)cc1 C1(C(=O)NC(c2ccccc2)CC)CCCN1NC(=O)C(C)OCOC CC(C)CCC(=O)C(=O)NC(C)CC(C)NC(C1CCCC(C)CC1)=O N1(C(C=CC(C)(C)SC)=O)CC2CCC2(CCNC(c2nc(C)ccc2F)=O)C1 Cc1cc(C(=O)NCC23CCC2CCN3C(=O)CCC(C)(C)C)nc(O)n1 CC(CCC(=O)NCC1CC(C#N)C1)NC(=O)CCc1nccn1C C12(C(N(CCCCN(C)C(C3COC(=O)O3)=O)C)=O)COCC1C2(F)F n1(CC)cc(Br)cc1C(=O)N(CC(C)NC(=O)CCn1c(C)ccc1C)C Cn1c(C(N2CC3CC(NC(=O)Cc4ccccc4)C2C3)=O)cc2ccccc12 c1(C(=O)NCCN(C(Cc2ccc(OC)nc2)=O)CC2CC2)c[nH]cc(Cl)c1=O C(=O)(C#CC1(C)CCCO1)NCC(CNC(c1c(F)ccc(C)c1)=O)CO Cn1nncc1CC(=O)NC(C1(O)CCOC1)c1ccccn1 CC1(C)C(NC(c2cnn(CCF)c2)=O)CCN1c1ccnc(Cl)n1 N1(C(COCCOCC)=O)CC2CCN(C(=O)C(c3ccc(F)c(C)c3)=O)CC12 O=C(C(F)(F)C(O)C1CC1)N(c1ccc(N2CCC2)nc1)C1COC1 C(C(=O)OC)(C(C1CC1)C1CC1)N(C1CCCNC1=O)CC1CC(F)(F)C1 N1(C(CCC)=O)CCCN(C(c2ccc(N(C(=O)CC)C)cc2)=O)CCC1 C1(CNC(N2C(c3cc(C)cc(C)c3)CCC2)=O)CCCC2(CCC2)C1O N1(C(C(CCSC)NC(CC(C)(C)OC)=O)=O)CCC(O)C(C)C1 N(C1CCCc2c[nH]nc21)C(C1N(C(CCSCCCC)=O)CC(O)C1)=O Cc1noc2cc(C(N3CCN(C)C(CNC(=O)CN(C)C)C3)=O)ccc12 N1(C(N(C2CC2(F)F)CC)=O)CCCCC1CF c1(C(N)=O)ccccc1S(=O)(=O)N1CC(CC(F)F)C1 O=C1OC2CC(C(=O)NC3CCCN(C(c4ncc5[nH]ncc5n4)=O)C3)CC2O1 N1(CC)CC(CNC(=O)C(C2CCCN(C(=O)CC=C(Cl)Cl)C2)C)CC1=O CC1CC(C(=O)NCC(C(C)(C)C)NC(=O)CC(C)C2CCCO2)CC1 c1(CCC)n[nH]c(=NCC2CC(NC(=O)C(O)CCSC)C2)s1 c1(C(=O)OC)coc2cc(C(=O)N(C3CC3)CC(C3CC(OC)C3(C)C)=O)[nH]c12 C(=O)(CC1=CCN(C)CC1)NC(C1CCN(C(C2CC3CC3C2)=O)C1)C C1(N(C(=O)C=CC=C(Cl)Cl)C)CCCC(NC(c2nonc2N)=O)C1 c1(C(C)C)cccc(N(C2CCC(C)(C)C2)C)n1.N12CCC(C1)NC(=O)C2=O c1(NC(C(CC=C)CNC(C2CC2=C)=O)=O)cccc2cccnc12 C1(NC(CCCN(C)Cc2ccoc2)=O)CCCN(C(c2c(C)ncs2)=O)CC1 C1(NC(COC2CN(C(C3CCC(C)(C)OC3)=O)C2)=O)CCn2nccc2C1 C#Cc1ccc(C(N2CC(CNC(C3CC(SC)C3)=O)C(C)C2)=O)cc1 c1(C(=O)NC(C(C)NC(c2cc(C)nn2C)=O)CO)c(O)cccc1F C1(C(N2CCC(=CCNC(CCC(C)OCC)=O)CC2)=O)CC2(C1)CC(F)C2 N1(C(C2C(CCC)C2)=O)CCOCC1CCNC(=O)CSc1nnnn1C c1(C(=O)OC)c(OCCC(N2CCC(OC(=O)N(C)C)C2)=O)sc2c1CCOC2 N1(C(C=C(CC)C)=O)CCN(C(=O)Cc2cnccc2OC)CCC1C C1(n2cc(Cc3ccc(OC)cc3)nn2)CC2CCC1(NC(=O)C(C)(C)SC)C2 C(=O)(CCCCCCCBr)NCc1nccc(C(N2C(C#N)C3CC3C2)=O)c1 c1(C(N2CCCCC(NC(C3CCS(=O)(=O)C3)=O)C2)=O)ccn2cnnc2c1 C1(NC(c2ncoc2C2CC2)=O)CC2(C1)CN(C(=O)C(F)CC1CCC1)C2 N1(C(c2nc(CCC)sc2)=O)CCC(C)C1CNC(c1cnc(C2CC2)s1)=O Cc1nc(C2CC2)[nH]c1C(=O)NC(C)CCCCNC(c1ncsc1C1CC1)=O Cc1coc(C(=O)N(CCC(=O)NCc2cscn2)CCO)c1 c1(C(=O)NC2CC(c3cn(CC(COCC)O)nn3)CC2O)cnc(C)nc1C C(CCNC(=O)CN(S(C)(=O)=O)C)(C(C)C)NC(C(C)=C1CCCC1)=O c1(OC)cc(Cl)c(C)cc1C(N1CC2CCC(N)C2C1)=O.C1(=O)C(C(C)C)N1 N1(C(C(=O)NCC(C)C)(C)CC2CCC2)CCC2(COC(C)(C)C)CCCCCC12 CC(C)CCCC(=O)N1CC2C(CC(=O)NC3CCCCC3O)C2C1 c1(C(C)(C)C)nc(=NCC2CCCCN(C(c3ncncc3Cl)=O)C2)s[nH]1 N1(C(C=COCC)=O)CC(C2CCCCN(C(c3c(C)ncn3O)=O)C2)C1 N1(C(C(N2CC(OC)C(N)C2)=O)=O)CCCOc2ccc(C)cc21 N1(C(c2cc(C(C)=O)on2)=O)CC=C(CNC(c2cc(C)cc(C)n2)=O)CC1 C1(NC(CCN(C)CC)=O)CC12CCN(C(c1c(OC)ccc(Cl)c1Cl)=O)CC2 Cc1cc(C#N)ccc1C(N1CCC(NC(=O)CSCCN(C)C)C1)=O N1(C(c2sc(C)c(O)n2)=O)CCCC(NC(=O)C(F)(F)C2CC2)C1C C1(C(N2CC(C)(NC(C(c3ccccc3F)C)=O)C2)=O)CCC(N=[N+]=[N-])CC1 c1(C(N(CC(C)NC(Cn2nc(C)c(C)c2C)=O)C)=O)cccc([N+](=O)[O-])c1 N1(C(C(Br)=C(C)C)=O)CCCCC1CNC(=O)CC(O)C1CCCC1 N1(C(Cc2c(C)ccnc2)=O)CCCOC(CNC(c2ccc(Cl)cc2F)=O)C1 C1(CC)(CO)CCN(C(c2cc(NC(=O)COCC(=O)NC)ccc2F)=O)CC1 N1(c2c(C)c(Cl)ncn2)CC(CNC(=O)C(C)(C)CC(C)C)OC(C)(C)C1 CCC(C)C(O)C(C)C(=O)N1CCC(c2cccc(F)c2)C1 C1(NC(CCC#N)=O)CCC(=O)NC1C1CCN(C(=O)Cn2cc(Cl)cn2)CC1 c1(OC)cnc(C(N2CCCC(O)(CCNC(=O)Cc3ccoc3)C2)=O)c(F)c1 N1(C(C(=O)NCCC)CC(C)SC)CC2CCC(C1)N2c1ccccc1 c1(OC)nc(C)ccc1C(=O)NCCN(C(c1cnns1)=O)Cc1ccccc1 c1(OC)c(CCNc2cccc(CN3CCCC3=O)c2)cc(Br)cc1F C(=O)(CC(O)C(C)C)NCC1(C(=O)NCc2ccc(OC)nc2)CCCO1 c1(OCC)ccccc1C(=O)NCC(O)CN(C(=O)CC1CC1(C)C)C c1(CC(=O)NCC23C(CN(C(c4cncc(NC)c4)=O)C2)C3)ccc(O)c(F)c1 N1(C(=O)C(=Cc2cccnc2)F)CCC2(CCN(C(c3cnccn3)=O)CC2)C1 C1(N(C(CCCn2c(C)ncc2)=O)Cc2cn(CC(=O)O)nn2)CCS(=O)(=O)C1 Cc1ccc(C)c(NC(C2CC2OCc2ccccc2)=O)c1.C12CN(C1)C2=O C1(NC(C(c2c(C)n[nH]c2C)C)=O)CC2CC(C1)CN(C(C1(O)CC1)=O)C2 C1(C(=O)NC(CC(=O)N2CC(COC)C2)COC)CCC(O)CN1C CC(CCCC(=O)NC1CCC(O)C1)c1ccccc1 CC(=Cn1ccnn1)C(=O)NCC(CO)NC(=O)CCC1CC1CC1CC1 C1(C)(CNC(C(c2ccoc2)NC(Cc2cn(C)nc2)=O)=O)CCCCC1 CC1CC(CNC(C2(C(F)F)CCC2)=O)CN1C(C1CC12CC(O)C2)=O C(=O)(CCCS(C)(=O)=O)NCC1(CO)CCN(C(CC(C)C(F)F)=O)CC1 c1(CC(=O)N(C(CNC(C(c2ccc(F)cc2)OC)=O)C)C)cccnc1O C=C(Br)CC(C)(C)C(=O)NC1CCN(C(=O)C(CCC)N(C)C)CC1 C(CCC(C(=O)NC1CCCC1F)NC(=O)C=CC(F)F)OC C1(CN(C(CCNC(CN(C(CC)=O)C)=O)=O)C)CC12CCOC2 CC1(NC(C2CCC3CCC23)=O)CCN(C(=O)CSCc2ccncc2)CC1 c1(CNC2C(CC=C)CCC2)n[nH]c2ccncc12 C=CCC(F)(F)C(=O)N1CCC(CO)(NC(=O)CNC(c2ccc(F)cc2)=O)C1 C1(NC(c2c(C)oc(CO)c2)=O)CC(O)CN(C(=O)CCCc2cnccn2)C1 C=Cn1nccc1C(=O)NCCC1(O)CCN(C(=O)CC2(OC)CCOCC2)C1 C1(C(N2CCCC(O)(CNC(C34CC(CO3)C4)=O)C2)=O)CC2(COCCO2)C1 N1(C(c2cc(C)oc2)=O)C(CNC(c2ccn(CC(C)C)n2)=O)CC2CCCC12 C1(C)(C(N2CC(O)(CCNC(C3(OC)CCC3)=O)C2)=O)CCCS1(=O)=O C(CCCCC(=O)NCC(C)N(C)C(C1(C)CCC(=O)NC1)=O)SC C1(NC(c2onc(C)n2)C2CCCCC2)CC2(CCC(CN)OC2)C1 c1cccc(C(=O)NCCN(C)C)c1.C1(C(=O)OCC)CCCC1CNC=O C(c1ccc(Cl)s1)=CC(=O)N(CC(C)N(C)C(c1cnnc(O)c1)=O)C CCCCC(C)CCC(=O)N1CCC(CF)(NC(C2CCC=CO2)=O)C1 C(=O)(C1CCCc2nc[nH]c21)N(C(C)CNC(=O)C(=O)NCC1CC1)C c1(C(=O)NCCCN(C(Cc2ccn(CC)n2)=O)CCO)cc(Cl)ccc1O n1(CC)ncc(C(=O)NCCC2CCC(NC(=O)CCc3cc(Cl)no3)C2)n1 C1(CNC(c2ccc(C(F)(F)F)o2)=O)CC2CCC1N(C(C1CC(F)C1)=O)C2 c1(-c2n(C3CCS(=O)(=O)C3)nc(CCO)n2)ccc2cccc(Br)c2n1 C(=O)(C(C)(CC)CCC)NC(CC=C)CNC(C12CC(C(=O)OC)(C1)C2)=O C1(NC(C(CNC(c2cn(CCC)nc2)=O)O)=O)CCS(=O)(=O)C1 C12(C(=O)NCC3N(C(C4CC(CC)C4)=O)CC(O)C3)CCC(N=[N+]=[N-])C1C2 c1(NC(N2CC(C=C)C(O)C2)=O)ccc2c(c1)nc(SCC)n2CC N1(C(C(C=C=C)C)=O)CCC2(CC1)CC2CNC(=O)N(C)C CCC(CC1CCCCC1)C(=O)N1CCC1CNC(=O)C(C)(C)NC(C)=O N1(C(CC2CC(NC(C3CCOCC3)=O)C2)=O)CCOC2CCCCC12 c1(C(=O)NCC2C(CNC(Cc3ccn(C)n3)=O)C2)cncc2ccsc12 c1(OC)ccc(C(N2CC(F)CC2COC)C(=O)NC2CC2)c(C)c1.C1(CS)CCCC1 C12(CC(=O)NCCOCC(=C)C)CCC1CN(C(=O)CC(C)(C)C)C2 c1(CC)[nH]c(-c2ccccc2)cc1C(=O)N(C1CN(Cc2ccccc2)C1)CC N1(C(Cc2cc(C)sc2C)=O)CCN(C(=O)CC2CCC(C)CC2)CC1C(C)C C=CCCCC(C)N=c1cc(C)[nH]c(=NCc2cc(OC)c(O)c(Br)c2)[nH]1 C1(C(C)C)CN(C(=NCCC(C)=O)NCC2(C)CC2(Cl)Cl)CCN1C C1(C(N2CC(CC)(OC)C2)=O)CCC(C)(C)N(C(=O)C(N=[N+]=[N-])C(C)C)C1 C(CNC(=O)C(c1ccnn1C)C)(C(C)C)NC(C1(CC)CC1)=O C1(C(N2CCCC(NC(C(=O)NCC(F)F)=O)CC2)=O)Cc2ccccc2CO1 C(=O)(C(CC=CC)NC(c1ncccn1)=O)NC(C#C)CC1CCC1 C(=O)(CC(O)C(C)CC)NC(C(=O)NC(CC)Cn1cncn1)CCN(C)C Cc1nc(C)c(C(=O)NCC(N2CCN(C(=O)CC3CCC(C)(C)C3)CC2)C)o1 N1(C(c2c(C)snc2)=O)CCCCC1CC(=O)NCCCC(C)O N1(C(=O)CC2CSCCO2)CC2COCC2(C(=O)NCc2ncccc2O)C1 C(N=C(NCC1CCCCO1)NCC(C)(CC)OC)c1c(CC)n[nH]c1 CC(C)(CN=c1[nH]c(NC2C3C=CC(C3)C2CO)nc2c1CCC2)c1ccsc1 c1(C(=O)NC23CCN(C(C4(SC)CCC4)=O)CC2C3)cc2cc(C)ccc2[nH]1 N1(C(c2n[nH]cc2C(F)(F)F)=O)CCCN(C(C2CCCS(=O)(=O)C2)=O)CC1 N1(C(C2CCCN(CC)C2)=O)CCC(C)(C(=O)NC2CCC(=O)NC2C)CC1 C1(N(C(=O)CC#N)CC2N(CC)CCC2)C(C)OCC12CCNCC2.c1cnco1 c1(C(N(C2CCCN(C(C3CSCCS3)=O)C2)C)=O)cn2c(n1)CCC2 C1(NC(C2N(CC)CCC2)=O)CC2CCC1C(NC(=O)CCc1ccncn1)C2 c1(C(=O)NCC(CC)(C)NC(=O)C(C)NC(C)=O)ccc(-n2ccnc2)c(C)c1 N1(C(CC=CCNC(CCCCC(=O)OC)=O)=O)CC2CC3CC2C1C3O C1(C(N2CCN(C(C3(C)N(C)CCC3)=O)CC2CO)=O)CC2C=CCC(C1)C2 c1(N(C)Cc2cccc(N)c2)nc(N2CCC(N3CCC3)C2)nc2c1SCC2 C1(NC(CS(N)(=O)=O)=O)CS(=O)(=O)C12CCN(C(=O)Cc1nncs1)CC2 N1(C(C2C(C(C)(F)F)C2)=O)CCC(CO)(CNC(c2cccc(Cl)c2)=O)CC1 C(=O)(C(C(C)C(C)(C)C)N1CCCC(C)(c2ccccc2)CC1)NCC=C N1(C(CCc2onc(CC)n2)=O)CC2(CCC2NC(=O)C(C)CO)C1 C(C1=CCCN(C(=O)C2=COCCO2)C1)NC(C1(CC=C)CC1)=O Cc1cc(CNC2CC2NC(=O)Cn2cccn2)no1 Cc1ccc(C(N2CCC(NC(c3cc(Br)n[nH]3)=O)C(CO)CC2)=O)c(N)c1C N1(c2ncc(OC)c(C)n2)CCC(F)(F)C(C(=O)Nc2cnc(C)nc2)C1 N1(C(Cc2nnc(C)s2)=O)CCCN(C(C2(C(F)F)CCCO2)=O)CC1C C1(NC(CC(c2nccn2C)C)=O)CN(C(=O)C#CC2(C)CC2)CC1C1CC1 CC1(NC(c2ccc(C#N)o2)=O)CCC(NC(C2CC3(CCOC3)C2)=O)CC1 C1(OC)CCCC(NC(=O)Cc2ccnc(-c3ccccc3)c2)C1 c1(NC(=O)CC2CN(C(C3CCC(F)(F)C3)=O)CCO2)cnncc1Cl c1(C(=O)NCCNC(c2c(CC)nns2)=O)cncc(O)c1Cl C1(N(C(CC2CC(SC)C2)=O)C)CN(C(=O)CCOC2CC2)CC1O N1(C(CC)=O)CCC2CCN(C(=O)Cc3cccc(Br)c3Cl)C2C1 C(C(CO)C(C)(C)C)NC(C1(C)N(C(c2ccn(C(C)C)n2)=O)CC=C1)=O C1(CNC(C(C)(C)F)=O)CN(C(C2CCSC2)=O)CC1C(F)(F)F C(CC(=C)Cl)(C(=O)NCC1CCC(C)C1)NC(C(CC#C)O)=O N1(C(c2cc(C)oc2C)=O)CCC(CNC(C2CC3(C2)CC(O)C3)=O)C(O)C1 C12(CNC(c3ccoc3)=O)CN(C(c3ccc4n[nH]cc4c3)=O)CC1CCO2 N1(C(C2(CC)CCCC2)=O)CCN(C(=O)CNC(=O)Cc2cnc(C)s2)CC1 CC1CCN(C(=O)C(=O)Nc2ccc(-c3cscn3)nc2)CC1CO n1(CC(N2C(CNC(C3CC(=C)C3)=O)CC(C)(C)C2)=O)[nH]cc2c(=O)ncnc1-2 c1(NC(C2CC(=C)C2)=O)cccc(NC(C23CC(C)(CO2)C3)=O)c1 N1(C(c2ccc(Cn3ncc(C)c3)o2)=O)CC(CCNC(=O)CCCF)C(C)C1 c1(CC(N2CCC(C3N(C(C(F)=CC)=O)CCCC3)C2)=O)c(OC)cccc1C c1(OC)cc(C)cnc1C(=O)NC1CCN(C(c2ccc(F)cc2C(F)F)=O)C1 N1(C(c2cnc(C)o2)=O)CCCC(O)(c2cn(CCC(F)(F)Cl)nn2)CC1 c1(OC)c(C(=O)NCC2(NC(=O)CC3CC4CC4C3)CCC2)csc1Cl C(=O)(CC(C(C)C)NC(C1CN2CCC1C2)=O)N(CCCO)CC C1(C(C)NC(c2cc(C(N)=O)no2)=O)CCCN(C(=O)CN2C(=O)CNC2=O)C1 c1(CC)onc(C)c1CNCc1csc(C)n1 CCC(C(=O)N1CCC(CN(C(=O)C(=O)N(C)C)C2CC2)CC1)C(C)O C(=O)(C(O)C(F)(F)F)NC(C(N1CCC(CN(C)C)C1)=O)(C)C c1(C(N(C2CCN(C(c3c[nH]c(=O)cn3)=O)C2)CCC)=O)cnc2ccsc2c1 C(=O)(C(C)(C)C(=O)NC(C1CCOC1)CNC(c1cc(Br)n(C)c1)=O)OC C(C1CCc2nccn21)NC(CC(CC1CC1)NC(C(C)(Cl)Cl)=O)=O C(C)(C(=O)NCC1(O)CCCN(C(=O)C(C)=C2CCCC2)C1)(C(C)C)NC(C)=O Cc1ccc(=N)[nH]c1C(=O)NC1CCCC(NC(=O)CCc2cn(C)nc2C)C1 C(CC(C)C)(C(=O)NC1CC(NC(=O)Cc2cc(Cl)n(C)n2)C1)NC(=O)OC Cc1ccncc1CC(=O)NC1C=CCN(C(C2CC(C(F)(F)F)C2)=O)C1 N1(c2nnc(-c3oc(OCC)c(C)n3)n2CC(C)C)CCC12CCCSC2 CC1=NOC2(C1)CC(C(=O)N(CCCNC(=O)CCc1ccccc1)C)C2 N1(CC(=O)NCC=CCNC(CCC(C)(C)F)=O)C(=O)NC(C)(C2CC2)C1=O c1(C(n2cc(NCC3COCC(C)O3)nn2)C)ccc(F)nc1Br CC(C(CO)NC(c1cnn(CCN(C)C)c1)=O)NC(=O)CSS(C)(=O)=O Cc1cc(C(=O)NC2(CF)CN(C(C3CCCCC3F)=O)C2)c(C)cn1 C(C(F)C(F)(F)F)NC(C(CC)N(C)CC)=O C1(NC(c2cn(CCN(C)C)nc2)=O)CC12CC(NC(C1CCS(=O)CC1)=O)C2 N1(CC(=O)OC2CCCCCC2c2ccccc2)C(=O)c2ccccc2C1=O C(CCCCCNC(c1nccn1C)=O)NC(C=CC(CC)C)=O C1(C(=O)NCC(CCOC)NC(C2CC3CC3C2)=O)(OC)CCOCC1 C(=O)(C(F)C(C)(F)F)N1C(CN(C(C(c2ccccc2)SC)=O)C)CCC1 c1(C(N2C(C(C)C)CN(C(C3CC3C)=O)CC2)=O)cc2oc(Br)cc2[nH]1 CC1CC=C(C(=O)NCc2cccc(NC(c3ccc(O)c(Cl)n3)=O)c2)CC1 C12(CNC(c3c(C)n(C)cc3)=O)CCCC1CCN2C(=O)CSCc1cccs1 CC1CC(C(=O)NCC2(CNC(c3ccc(C(C)(F)F)nc3)=O)CC2)CC(C)C1 N1(C(C2C(C(=O)OC)C2)=O)CCCC(O)(CNC(=O)Cc2[nH]cnc2C)CC1 C1(C(N2CCC(CC=C)(NC(=O)CC(C)F)C2)=O)CC(C(C)C)=NO1 n1(CC(=O)NCCN(CCC)C(C2CC23CC3(F)F)=O)ncc(O)nc1=O c1(C(=O)NC2CN(C(C3(CF)CC3(F)F)=O)CC2F)ccc2ccsc2c1 C1(C)(C(N2CCC(C)(OC)CC2)=O)Cc2ccccc2C1 n1(CC)cc(-c2n[nH]cc2C(=O)N(C2CN(C(C3CCN3CC)=O)C2)C)cn1 N1(C(c2c(C)cc(C)o2)=O)CCN(C(c2ccccn2)=O)C2COCC12 CC1CCN(CC(=O)NCCCC(CO)NC(C2CCNC(=O)C2)=O)CC1 C(=O)(CCCC(C)(C)C)NCC1CN(C(C2=CC(C)(CC)C2)=O)CC1(F)COC C=CC1CCN(C(c2cc(CNC(C3CC4CCC(C3)O4)=O)ccn2)=O)CC1 C=CCC(CC)C(=O)N(CCCNC(=O)C(CSC)Cc1ccc(F)cc1F)C C(C(=O)N(C1(C(=O)NC(C)CCCCO)CC1)C)(C(C)C)SC n1(CC(N2CC(CNC(=O)C=CC(F)(F)F)C2)=O)cc(F)ccc1=O c1(NC(C2CCC2)C)[nH]c(=NCc2nccc(C(F)(F)F)n2)nc2c1ncn2C C(=O)(C1=CC2(CCN(C(=O)CC3CC4C=CC3C4)C2)C1)NC(c1cn(C)cn1)C c1(NCC(c2cccc(OC)c2)NC)ccc(C(N(CC)CC)=O)cc1[N+](=O)[O-] c1(COCC)cc(F)ccc1CN1CCCC1CN(C)C CON(C(=O)C(CNC(C1CCC1C#N)=O)CC1CC1)C(C)C C(=O)(C(C(C)(C)C)NC(C)=O)N1C(C(N(CCCCC)C)=O)CC(C)C1 C1(NC(CCC2(C)CN(C(C3(CC=C)CC=CC3)=O)C2)=O)CCN(C)C(C)C1 c1(C(N2CCN(C(CCOC)=O)CC2)=O)ccc2nc[nH]c2c1F C1(CCNC(C(CC)CC)=O)CCN(C(c2ccn(CC)n2)=O)C(C)C1 Cc1cccc2c(C(=O)N(CC(C)O)CCNC(=O)Cn3cccc3)cnn12 C1(C(N2CC(O)(CCNC(CCS(=O)(=O)NC)=O)C2)=O)CN2CCN1CC2C N1(c2snc(C(=O)OC)n2)CCCCC(NC(c2cc(Cl)cn2C)=O)C1 C12(C(c3n(C4(C)CC4)nnn3)NCc3cnn(C)c3F)CCC(CC1)C2 N1(C(c2ccc(SC)o2)=O)CCCC(CCNC(=O)Cc2ccsc2)CC1 C(=O)(C(C)CC(F)F)NC1(C(=O)NC2(C)CC(=C)C2)CC(CO)C1 C12(C(=O)O)CCC(NC(=O)NC)(CC1)CO2.C12(CCCC1)NC2.C(C)(C)(C)OCC C(N=c1[nH]cnc2cc(C)[nH]c12)C1(F)CC(NC(C(C2CCOC2)OC)=O)C1 c1(C(=O)NCC2N(C(c3ccc(C)[nH]3)=O)CCCC2C)c([N+](=O)[O-])c(C)nn1C C1(C)(CNC(=O)NC(c2ccc(NC(C)=O)cc2)C)CCC(F)(F)CC1 C1(NC(c2cccn3ccnc23)=O)CN(C(C2C=CCS2)=O)C2CCCC12 C1(C(=O)NCC2C(C)(C)CCO2)CC12CCN(C(C1CCCC1)=O)C2 C1(N(C(=O)CCNC(=O)COC)CCC)CCN(C(C2(F)CCCC2)=O)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1C(CNC(C(C)OCCCCCC)=O)CC1 C1(NC(C(=O)NCC)=O)CCN(C(=O)CC2COCC2(C)C)CC1F N1(C(c2cc(C)[nH]c2C)=O)CC2CCC2(CNC(=O)CC2CCC3(CC2)CC3)C1 N1(C(C(F)=CC)=O)CCCOC(CCNC(=O)CSc2nncn2C(C)(C)C)C1 C1(O)(CN(C(C=C(CC)CC)=O)C)CN(C(c2cnn(C3CCC3)n2)=O)C1 c1(C(=O)OC)cccc(C(F)(F)C(=O)N(C)CCNC(c2ccc(C#N)s2)=O)c1 CC1(C)CC(NC(=O)CC2CCOCC2)CN(C(=O)CCc2cccnc2Cl)C1 C1(CNC(CSC(C)(C)C)=O)CC12CCN(C(=O)Cn1cnc(C#N)n1)CC2 CC(C)C(=O)C(=O)N1CCCCC1CCNC(=O)C=CCF N#CC1CN(C(C2CN(Cc3cc(Cl)ncc3Cl)CCC2O)=O)CCO1 C1(CNC(CC2(C)CCCC2)=O)CN(C(C2(C)CC2Br)=O)CCC12CCOC2 N1(C(C(CC)NC(N)=O)=O)CCC2CCCC12C(N1CCC2(CC1)N=N2)=O CC#CCCCC(=O)NCC1CCN1C(=O)Cn1nnnc1-c1ccsc1 Cc1nn(CCC#N)c(C)c1CC(=O)NC1(CNC(c2ccsn2)=O)CC1 N1(C(C(C)Cc2ccccc2F)=O)CC=C(CNC(C2(CC)CC2(F)F)=O)CC1 CN1CC(O)CCC1C(=O)NC1(C(=O)NC2CC(C(F)F)C2)CSC1 c1(C(N2CC3C(CNC(C4(C=C)CC4)=O)C3C2)=O)sc2cc(C)c(C)cc2c1C C=C(C)CC(C(=O)N1CCOC(C)C1C(N1CCC(C#N)CC1)=O)OC c1(C(N2C(CNC(=O)CCC(N)=O)CC(OC)C2)=O)nsc2ccc(C)cc12 CCC(C)C(CNC(=O)CC(CNC(C1CCC1C(C)(C)C)=O)C1CCC1)OC Cc1cccc2ncnc(N3CCCC(C4CC4NC(C4CC=CCC4)=O)C3)c12 c1(C(N(C)CC2OCCN(C(C(=O)NCC)=O)C2)=O)cccc2ncnn12 C(N=c1[nH]cnc(=N)[nH]1)C1CN(C(c2ccc(CSCC)cc2)=O)CC1C N1(C(C(C)OCC)=O)CCN(C(=O)CSc2nncs2)C(C2CCCC2)C1 Cc1ccc(S(=O)(=O)CNC(c2ccc([Si](C)(C)C)o2)=O)cc1 C1(NC(C(CN(CC)CC)F)=O)COC2(C1)CN(C(c1cc(C)cc(C)n1)=O)C2 c1(CNC(C2CC(C(C)C)C2)=O)ncc(C(=O)NCc2nncn2C)cn1 N1(Cc2cn(C3CN(C(C(CC)(C)CO)=O)CC3O)nn2)CCc2ccccc21 C1(NC(c2nccc(OC)c2)=O)CC2(C1)CN(C(=O)C(CC(C)C)OC)C2 N1(C(C=CSC)=O)CCCC(N(C)C(c2cn(Cc3ccccn3)nn2)=O)CC1 C1(CC=C)(C(=O)NCCC(=O)N(C)C)CCCN1C(=O)CC1(O)CCCOC1 c1(C(NC(C2(NC(C(C)SCC)=O)CC(F)C2)=O)CC)cc(C)cc(C)n1 c1(C(C)C)nnc(C=CC(N2CC(CNC(=O)C=Cc3cncs3)CC2C)=O)o1 Cc1nc(N2CCN(C(C3(O)CCOC3)=O)CC2CCO)c2c(C)c(C)sc2n1 C1(C(=O)NCC2C3CN(C(C(C)C4CCC4)=O)CC32)CNC(=O)CC12CCC2 C1(CNC(C(CCC)OC)=O)CCCCCN1C(c1ccnc(CO)c1)=O c1(NC2CCN(C(C(C)n3cccn3)=O)C2)ncc([N+](=O)[O-])c(=N)[nH]1 Cc1n[nH]c(=NC(CCN(C(=O)CC2CCCOC2)C)C(C)C)o1 C(=O)(CC1=NNC(=O)C1)N1C(C)(C)C(CNC(c2snc(O)c2Cl)=O)CC1 N1(C(COCC=C)=O)CCC2(CC1)CCN(C(=O)C(CC)(CC)CC)CC2 c1(C(=O)NC2CC3CN(C(C(CC)(C)O)=O)C2C3)ccc2c(n1)OCC(=O)N2 C(C#CC1CC1)NC(C(C1CC1)NC(CN(C)C(=O)C1CC1)=O)=O CC1CCC(C(=O)N(C)CCOCCCNC(=O)CC2CSCCS2)O1 Cn1c(C(=O)NC2(C)CCN(C(=O)Cn3cnccc3=O)C2)nnc1S N1(C(CC)C(=O)NC2CCC(CNC(=O)CCCSC)C2)CCN(C(C)C)CC1 C1(CC(=O)NCC2(C(=O)NCc3cc(C)no3)CCCO2)CCCN(C)C1 C12(NC(c3c(CNC(CC(C)(C)OC)=O)ccs3)=O)CCC(C1)OC2C N1(C(C(C)N=[N+]=[N-])=O)C2CCC(C2)C1C(N1CCCOC(CO)C1)=O C(CN=c1[nH]nco1)OCCN(C)C(c1[nH]ccc1C1CC1)=O N1(C(C=CC(=O)OCC)=O)C2CCC1CC(NC(=O)Cc1cccnc1OC)C2 c1(NCC2CC(C)NC(=O)C2)[nH]c(=NCC2CC2(F)F)nc2scnc12 C1(NC(c2cc(OCC)c(C)cc2)=O)CC(C(=O)O)C12CC(F)(F)C2 CC1OCCCC1C(N1CC(N2CCCC2)C1)=O.C1C(=O)N1 C1(NC(C)=O)CCCCN1C(=O)CCC1(C(=O)NCC(CC)NC(C)=O)CC1 C1(C)(C(N(CC(CN(C(C2(CC#C)CCCO2)=O)C)O)C)=O)CC(O)CN1C S(=O)(=O)(c1c[nH]ccc1=NCc1cn(C)nc1I)N1CC(C)SCC1 c1(C(C)=O)ccc(C(=O)N(CCCNC(=O)CN2CCC(C)CC2)CCO)cc1C C12(CNC(c3cc(CC)on3)=O)CCCC1N(C(c1occc1F)=O)CC2 O=C(C1=NOC2(CCCN(C(c3cnc(Br)o3)=O)C2)C1)Nc1ccc(Cl)cc1 c1(OC)cc(C(=O)NCCC2COCCN2C(=O)CC2CCCOC2)ccc1F C12(CNC(c3cc(Cl)c[nH]3)=O)CCCC1N(C(=O)Cc1ccc(O)c(F)c1)CC2 CCCCC(O)CC(=O)NCC(C)NC(c1cnn(CC(C)(C)O)c1C)=O Cc1cc(CC(N2CC(S(=O)(=O)NCCN(C)C)C2)=O)ccc1O C1(CNC(C2(C#C)CC2)=O)(CO)CCN(C(=O)Cc2nocc2C(C)C)CC1 N1(C(C(=O)Nc2cc3ncn(C)c3cc2)=O)CC=CCC2(CCOCC2)C1 c1(NC(c2c(CC)nc[nH]2)=O)ccc(Sc2ccc(Cl)nc2)cc1 C1(C(=O)NC23CC(NC(CN(CC(C)(C)C)C)=O)(C2)C3)CCCCNC1=O N1(C(C2N(C(C)C)C(=O)CC2)=O)CCC(CNC(C2CCC(O)CC2)=O)C(C)C1 N1(C(CCOC)=O)CC(NC(=O)CNC(=O)CNC(C)=O)C(O)C1 C1(C(=O)NC(c2cn(C)nn2)C)CN(C(C2CCCSC2C)=O)CC1C1CC1 c1(CC)nc(N2CC3C(NC(=O)C=C(C)C)C3C2)c(F)c(Cl)n1 CCCC(C)(O)CC(=O)N(CCC(=O)NCC(C)CC(C)C)CC C(C(=O)N=S1(=O)CC(O)(C2CC2)C1)c1cc(OC)c(Cl)c(OC)c1 C1(C(N2CCC(CC(F)F)C2)C(=O)N(CCOC)C2CC2)CC2C=CC1CC2 N1(CCCNC(CCC#C)=O)CCN(C(C2CC2C)=O)CC1 c1(C(N2C3CC(NC(C(CC)N(C)C)=O)C(CC3)C2)=O)cccc2cnccc12 c1(CC)n[nH]c(C)c1S(=O)(=O)NCC1COCO1 N1(C(C(CC)Sc2nc(=N)[nH][nH]2)=O)CCN(C(c2ccco2)=O)C(C(F)F)C1 C1(C(N2CCC(O)(C(C)NC(=O)Cc3ccc(Cl)cc3)C2)=O)COC2COCC12 CCCCC(C)C(=O)N1CC2CC2C1C(=O)N(C)Cc1cc(OC)no1 C1(NC(CC(C(C)C)C)=O)C2CCCC1CC(NC(=O)CCc1cnccn1)C2 C12(CNC(=O)Cn3cnnn3)CCCC1CCN2C(c1cc(Cl)cnn1)=O C1(C2CC2)(CNC(C(C)NS(CCC)(=O)=O)=O)CCN(C(=O)CCC2(C)CC2)C1 c1(C(C)C)ocnc1C(=O)N(CC(=O)NCCc1ccn(CO)n1)CC1CC1 C(CCCCC(=O)N1CC2(CC(C(N3CCS(=O)(=O)CC3)=O)C2)C1)=CC N1(C(CC=C)=O)CC23CCCCC2(C1)CN(C(c1ccc2n[nH]cc2c1)=O)C3 c1(CNC2CCC(CC(=O)NC(C#C)C)CC2)cc(F)cc([N+](=O)[O-])c1 c1(CNC(C(C)N(C(c2occc2C(=O)OC)=O)CC)=O)nn(C)cc1CO C(=O)(C1=CCCCO1)NCC(Cn1cc(-c2ncc(F)cn2)nn1)OC N1(CC)C(=O)CCC1CC(N1CCC1CC(F)C(=O)O)=O C1(NC(CCOC)=O)CC2CC(NC(=O)COc3cccc(C(C)=O)c3)C2C1 c1(CC)cc(C(=O)N(C(C)CCNC(C2(C#N)CC2)=O)C)nn1CCO Cc1cc(C(N2CCN(CCNC(=O)C(C)CN(C)C)CC2)=O)n2ncnc2n1 N1(C(=O)NCC2CC3(CC(=C)C3)C2)CCC2(CC1)CN(CC(=O)OC)C(=O)O2 N1(C(C2CN(C(c3oc(C)c(CO)c3)=O)CC2(C)C)=O)CC(C)CCC12CC2 c1(C(=O)NC2C(NC(C=C(C)I)=O)CC2)nc(C)ccc1F N1(C(C2(C#N)C(C)(C)C2)=O)CCCN(C(c2ncoc2C2CC2)=O)CCC1 CC1CC1N=c1[nH]c(=NCC23CC(C(F)F)(CO2)C3)[nH]c2cccnc12 c1(CNC(=O)NCc2c(C)non2)ccc(N2CCNC(=O)C2)c(F)c1 N1(C(C(CF)NC(C=CCN(C)CC)=O)=O)CC2CC1CN2C(C)=O C(=O)(C(CO)C(C)(C)C)NCCC1CCN(C(C2N(CCC)CCC2)=O)CC1 c1(C(N2CC(C)C(CNC(=O)CCCCO)CC2)=O)ccc(N=[N+]=[N-])cc1 c1(C(=O)NC(C)CCN(C(=O)C(O)CC(N)=O)C)n[nH]c2c1CS(=O)(=O)CC2 C(C(C)(C)CCNC(=O)C(C)C(F)F)NC(c1n(C(C)C)ncc1)=O C1(NC(Cc2c(CC)nn(C)c2CC)=O)CN2CCC1(F)CC2 c1(OC)ncc(C(=O)NC(CNC(c2ccncc2)=O)CO)cc1C c1(C(N2CCC(CNC(c3cc(OCC)n[nH]3)=O)C2)=O)cc2ccc(F)cc2[nH]1 C1(N(C(c2nc(CC)sc2)=O)C)CCCC(N(C)C(c2cccc(NC)n2)=O)C1 N1(CC(=O)N(C)CC)CCC(C2CCCN(C(=O)CCC3CCCO3)C2)C1 N1(C(CC2N(C(C3C(C)=CCS3)=O)CC(F)C2)=O)CCCCN(C)CC1 c1(C(N2CC(C)(C)C(NC(c3cc(Cl)ns3)=O)CC2)=O)coc2ccc(O)cc12 N1(C(c2c(C)ccc(N)c2)=O)CC2CC(NC(C3C(F)(F)C34CC4)=O)CC(C2)C1 c1(CC)cccnc1C(=O)N(CCCNC(=O)C(C)C(C)O)C c1(CC)nc(C)n(C)c1C(=O)NCC=CCNC(C1CS(=O)(=O)CCO1)=O CC1CCCN1C(C(=O)NCC1CCC1)C1CC1c1ccco1 C=C1CC2CC1CN2C(=O)C1=CCN(C(=O)CCNC(=O)COC)C1 N1(CC(=O)NC2C(NC(C3N(C(=O)OC(C)(C)C)CC3)=O)C2)CC(=O)NC1=O N1(C(c2cc(C)[nH]c2C)=O)CCC(C(N2CC3CCC(C2)N3C(C)C)=O)CC1(C)C N1(c2n(CCCOC)c(C3(O)CCCN(C)C3)nn2)CC2CNCC1COC2 c1(CC)cnccc1C(=O)NCCOCCOCCNC(=O)CS(=O)CC c1(C(=O)NC(C(=O)NCCC(=C)CNC(=O)C(F)OC)C)ccc2n[nH]cc2c1 n1(CC(=O)NCCN(CCOC)C(c2cc(=O)cc[nH]2)=O)nc(C)ccc1=O C12(CNC(C(CC=C)CC)=O)CCCC(CN1C(=O)COC(F)(F)F)C2 c1(C(=O)NC2CN(C(c3cc(C)n(C4CCCCC4)n3)=O)C2)cn2ccnc2s1 C(N=c1[nH]c(=N)[nH]c2[nH]cnc12)C1CC(OC)C12CCC2 C(=O)(C(C)C(C)S(C)(=O)=O)N1C2CN(C(c3ccc(CC)[nH]3)=O)C(CC2)C1 N1(Cc2cncc(OC)c2)CC2CCN(C(c3ccccc3C(C)(C)C)=O)C2C1 N1(C(c2c(CC)nc(C)[nH]2)=O)CC2CC(C)N(C(=O)C(n3cc(C)cn3)C)C2C1 CCCC(CCCNC(c1cccnc1)=O)NC(c1cccc(O)c1Cl)=O C1(C(=O)NCC2N(C(C3C(C(=O)OC(C)(C)C)C3)=O)CC=C2)Cc2cscc2C1 c1(NC(C(c2coc(C)n2)N(C2CCCCC2)C(C)=O)=O)ccc(SC(F)F)cc1 N1(C(C(C(C)C)C)=O)CCOCC(F)(CNC(c2ccc3nonc3c2)=O)C1 c1(OC)ccc(Br)cc1S(=O)(=O)NCC1CCCN(C(c2ccccc2Cl)=O)C1 Cc1cc(C(=O)NCc2nc(C)c(C(=O)NCC(O)C(C)(C)O)o2)c(C)cn1 C1(C(N(C2CC2)Cc2ccc(C3C(C)C3)o2)=O)COC2(CCC2)C1O CC(=O)CCCC(=O)NCC1(F)CCC(NC(=O)Cc2cc(C)[nH]n2)C1 c1(C(=O)NCCOC(CNC(C(CSC)C)=O)(C)C)ccccc1NC(N)=O c1(C(N2CCN(Cc3ccc(Br)cc3I)CC2)=O)cccc(Cl)c1Br c1(N(CCOC)CCNC(c2ccc(C(C)(C)C)cc2)=O)ncnc(Cl)c1CO Cc1sc(=O)n(CCC(=O)N(C2CCCN(C(=O)C(C#N)CC3CC3)C2)C)c1C N1(C(c2c[nH]c(=NC)o2)=O)CC2=C(C1)CN(C(C1CC3(CCC3O)C1)=O)C2 Cc1cc(C(=O)NC2CC(CNC(c3c[nH]cc(C)c3=O)=O)C2)ccc1Br c1(C(=O)NCCC(C)NC(c2cc(C)cc(C)c2O)=O)cccc(P(C)(C)=O)n1 C=CCC(CC(F)F)C(=O)N(CCCNC(=O)CC1(O)CCC1)C c1(CC(=O)N(C)CC2OCCN(C(c3c(C)[nH]nc3Cl)=O)C2)nc([N+](=O)[O-])n[nH]1 C1(CNC(C=Cc2ncc(C)[nH]2)=O)CN(C(=O)CCCc2cccs2)CCC1C C1(C(=O)NCc2cccc(NC(C3CCCO3)=O)c2)(CC)CCCOC1 C(CCC(C)(C)NC(=O)C=CC(F)(F)F)NC(C1C(C)C1)=O c1(OCC)nc(NC(CNC(=O)C#CC(C)C)C2CCC2)ncc1C N1(C(c2c(C)nn[nH]2)=O)CCOCCC1C(=O)NCC1(CF)CC1 c1(C(N(C(CNC(C(CCC)N(C)C)=O)C)C)=O)c(C)cc(C)nc1O CN=C(NCC1(C(=O)OC)CCCO1)N1CCC(C)(CC)C1 C(C)(CNC(=O)C(F)(F)c1cscn1)(CC)NC(C(C)NC(CC)=O)=O Cc1nc(S(=O)(=O)N2CC(O)C(O)C(C)C2)ccc1C(=O)O C=CC(C)(C)C(=O)N1CCC(C)(CNC(c2cccc(C(N)=O)n2)=O)C1 c1(CC)[nH]ccc1C(=O)NC1(CCC(=O)NCC2CN(C3CC3)C2)CCCC1 CC(C)CCCCC(=O)NCCC1CCCCN1C(c1ccc2nc[nH]c2n1)=O C1(C(N2CCCN(CCNC(CC3CC(SC)C3)=O)CC2)=O)CC2(C1)CC(F)(F)C2 CC1CN(C(=O)CCN(C(=O)CCC2OCCO2)CCO)CCC1N(C)C c1(C(=O)NC2C(O)(C(=O)OC)CCC2)sc2nccc(C)c2c1C N1(C(CN(C(C)=O)C)=O)CC(C)C1C(=O)NCCc1cscn1 N1(C(c2c(CNC(C3(OC(C)=O)CC3)=O)cnn2C)=O)CCCN(C)CC1C c1(OC)cc(O)ncc1C(=O)NC1CC12CC(NC(=O)C(C)N(C)C)C2 Cc1sc(C(=O)NC2CC(CCNC(=O)C=Cc3cnn(C)c3)C2)cc1Br c1(C(=O)NCC2CCN(C(C3C(C)(CC)C3)=O)C2)[nH]c2ccccc2c1C#N C1(C)(NC(C(=O)NCCS(=O)(=O)NC(C)C)=O)CC(F)(F)C1 C1(CC(=O)NCC2CCNCC2)CCN(C(c2cocn2)=O)CC1 CON1CCC(C(=O)NCC2(C(C)NC(=O)CSc3nncs3)CC2)CC1 Cc1cc2c(C(=O)NCC=CCNC(=O)CC3CC34CC4)cccc2o1 C=CC(CCC)CC(=O)NCCN(C(=O)C(C)CCC)CC O=S(=O)(c1cccc(=NCCC2CCCC2(F)F)[nH]1)NCCOCCF N1(C(CNC(=O)NC)=O)CCN(C(C2CCCC(C)(C)C2)=O)C(CO)C1 N1(C(CCCc2cc(C)no2)=O)CCN(C(=O)Nc2ccc(F)cc2Cl)C2CC12 C1(CC(=O)NCC(CNC(c2c(C)csc2Cl)=O)O)CC(C)(C)OC1=O c1(OC)ncc(C(=O)N(C)CC2CCCN2C(c2cc(Br)no2)=O)cn1 N1(C(C2CC(OC)C2)=O)CC2CC(C1)CN(C(C13CCC(CC1)C(C)O3)=O)C2 CCCCC(C(=O)N1CCN(C(C2CCN(CC)CC2)=O)CC1CC)NC(N)=O C1(NC(CCc2n(C)cnc2)=O)CCC2CC1CN2C(c1coc(O)n1)=O c1(C(=O)NCC2CC(OC)CN2C(=O)CC(C)SC)nccn2ccnc12 N1(CCCC2CCN2CCCOC(CCSc2n(C)nnn2)=O)CCCCCC1 C1(NC(N)=O)CCCN(C(=O)CCC2CCCN2C(c2cc[n+]([O-])cc2)=O)CC1 S(=O)(=O)(c1ccc2sccc2c1)N1C(C)(C)COCC1C(=O)O N1(C(c2n(CC)cnn2)C(=O)NCCCSC)CCC2CCC(O)C1C2 O=C(N=c1cc(-c2cccc(F)c2)o[nH]1)C(=O)NCc1nc(C2CCCO2)n[nH]1 C(=O)(CC(C)(C)CN(C)C)N(C(C(N1CC(C)C(CO)C1)=O)C)C c1(C(N2C(CC(=O)N(CCC#C)CC)CC2)=O)ccnc(OC)n1 c1(C(=O)NC(CN(C(C(C)OCCOCC)=O)C)CC)cc(O)cc(N)c1C CC(CC(=O)NC(C(=O)NCc1cc(O)cc(F)c1)C1CC1)C(F)(F)F CCCCC(C(=O)NCCSC)NC(c1ccc(C)c(O)c1)=O c1(CC)nnc2n1CCCC2C(=O)NCCC1CCCCN1C(C1CC(O)C1)=O c1(C(=O)NC(CNC(C=C(CC)C)=O)CC)c(Cl)cc(C#N)cc1Cl c1(C(C)(C)OC)cn(Cc2ncoc2CNC(c2cnc(C3CCC3)[nH]2)=O)nn1 c1(C(N2CCC(C)(NC(c3cn(C)c(=O)cn3)=O)C2)=O)coc2c1CCCC2 c1(C(N2CC(C)(OCC(=O)N(CCC)CCC)C2)=O)cnn2ccc(Cl)c(F)c12 C1(CC(=O)NCC(CC)CO)CCCN(C(C2CCC(C)O2)=O)C1 C12(NC(c3cc(Cl)c[nH]3)=O)CCC(CC1n1cc(CN3CCCSCC3)nn1)C2 C(=O)(CC(C)CC(=O)NC(CC1CC1)C(=O)NCCCC1(O)CC1)OC C1(NC(COCCC)=O)CCC(NC(=O)C=CC(c2ccccc2)=O)CC1 C1(CC)CC(O)CCN1C(=O)C(C1(O)CCC1)NC(c1cc(C#N)[nH]c1C)=O c1(C(N2CC(C(C)NC(Cc3cc(OC)no3)=O)C2)=O)ccn2ccnc2c1 C1(C(N(C2CCN(C(c3c(C)cno3)=O)C2)CCO)=O)CN(C)CC(C)O1 c1(OC)cc(C(=O)NCC2CC2NC(C2(F)CCOC2)=O)ccc1C(F)(F)F N1(C(C(C)NC(=O)NC)=O)C2CCC1CC(NC(C1(C(C)(F)F)CC1)=O)C2 CN=C(NCc1ccccc1)N1CCC(NC(c2nccc(OC)c2F)=O)C1 C1(N(C)C(c2ccc(CNC(c3sccc3Cl)=O)o2)=O)CNC(=O)C12CC2 C1(NC(c2cn(C(C)C)nc2)=O)CC2C(NC(c3ncc(C(F)F)s3)=O)C2C1 O=C1CCN(CC(=O)NCc2csc(CNC(C3CCCC(F)C3)=O)n2)C(=O)N1 c1(CSc2cccc(C(=O)NCC(=O)OC)c2)ncc(Cl)nc1Cl C1(COC)CN(C(c2ncc(N)cc2C)=O)CCN1C(c1cc(C)sc1C)=O c1(C(=O)NC2CN(C(c3c(N)cnc(SC)n3)=O)C2)cnn2c1CCCC2C N1(C(c2ccc(OC)c(C)c2)=O)CC2CCCN(C(C3CCCOC3C)=O)C2C1 N1(C(C(C(CC)O)C)=O)CCC2(CC1)CC(NC(=O)C(C)NC(=O)OC)C2 C(=O)(CC(C)(C)C)N(C1CC(NC(c2ccc(C(OC)OC)o2)=O)C1)C N1(C(c2c(C)nccn2)=O)CCCN(C(=O)C(CC(C)C)n2ccnc2)C(C)C1 C#Cc1cc(NC2(c3nnnn3CC3CC3)CCN(C)C2C)ccc1Cl C=C(C)C(CC(=O)NC(CCCNCC1CCN(C)C1=O)c1ccoc1)OCC N1(C(C2CC(C)OCC2)=O)CCOC2(C1)CN(C(C1(CC3CCC3)CC1)=O)C2 N1(C(C(OCC)OCC)=O)CCC(C)(C)C1C(N1CC(C)(C)C1CC)=O c1(C(=O)NCC(CO)NC(=O)COCCF)cc2ncccn2n1 n1(CCNC(C2(CC)COC2)=O)ccc(C(=O)NC(c2noc(C)n2)C2CC2)c1 Cc1cnc(C(=O)NC2(CO)CN(C(c3cnn4cc[nH]c34)=O)C2)c(C)c1 CC1CC(C(=O)NC(C)(C)C)CCN1C(c1cc(CN)on1)=O.C1(=O)CO1 C1(CC#C)(C(=O)Nc2cccc(Nc3nccc(OC)n3)c2)CCCOC1 n1(CC(=O)NC2C(NC(c3ccc(CC)s3)=O)CC2)nc(C)ccc1=O N1(C(CC(C)c2ccco2)=O)CCCCC(N(C)C(c2cnn[nH]2)=O)C1 CCC(CC(=O)N(CCC(=O)N1CCc2ncccc21)OC)C(F)F Cc1c(NC2COCCC2OC(F)F)ncnc1N1CC2CSCC2C1 C1(CC)CN(C(=O)C=Cc2cccnc2)CCN1C(C1CN(C(C)C)CCO1)=O N1(C(C=C(CCC)C)=O)CCN(C(c2c[nH]nc2C)=O)C2(CC2)C1 C1(OC(C)=O)CC2CC1CC2C(=O)N(C)OC c1(COC(C2(NC(=O)OC(C)(C)C)C(C)C2)=O)ccc(OC(F)F)cc1F c1(C(=O)NCCOCCN(C(C(C)NC(N)=O)=O)C)ccc(F)c(Cl)c1F CC#CCCCC(=O)NC1CCN(C(=O)Cc2c(C)nn(CC)c2C)C1C CCCCCCCCC(=O)NC1CN(C(=O)CC(CN(C)C)CC)CC1C CC1CN(C(=O)C(C)(C)C(C)NC(c2cccc(F)c2N)=O)CC(C)N1C c1(C(=O)NC2CCC(NC(C(C)OCCCC)=O)C2)c(OC)cccc1C N1(C(c2cc(CC)no2)=O)CCN2CCN(C(=O)C(=O)NC3CC3)CC2C1 c1(OC)cc(C(N2CCC(C(C)NC(=O)COc3ccon3)C2)=O)cc(C)n1 C(C(=O)N(OC)C1CCC1)C12C(CN(C(CC3ON=C(CC)C3)=O)C1)CC2 Cc1cccc2cc(C(=O)N(C3CN(C(c4ccncn4)=O)CC34CC4)C)oc12 C1(CC)CN(C(c2scc(C)c2OC)=O)CCC1NC(c1ccc(Cl)c(N)c1)=O N1(C(CC=C)=O)CC2CC1CCN2C(c1ccc(NC(=O)C(C)(C)C)nc1)=O c1(OC)cc(C(=O)OCC2(C)CCN(S(=O)(=O)Cc3ccccc3)C2)ccc1O C(=O)(C1=CCCCCC1)N(C1CCN(C(c2cccc3sncc23)=O)CC1)C C(CC(=O)NC1COCC1NC(C1CN(C)C1)=O)(C1=CCCC1)OCC CCC(C(=O)N1CCC(CNC(=O)CCCc2ccccn2)C1(C)C)C(C)(F)F C(c1cc(F)cc(F)c1)=CC(N1CC(C)CC(NC(C(C2CC2)OCC)=O)C1)=O N1(C(C2C(C(C)C)C2)=O)CC(=O)NCC1C(=O)NC(c1nc[nH]n1)C c1(C(=O)NCc2occ(C(N(C(C)C)Cc3ccco3)=O)n2)cnccc1C#N C1(O)(CCC)CCN(C(C23CC(C)(CN2C(=O)CCCCC#N)C3)=O)CC1 S(=O)(=O)(CC(=O)NC1CN(C(=O)C(C)(Cl)Cl)CC1O)N(C)C C1(CNC(c2cnc(CC)[nH]2)=O)CN(C(c2cc(O)ccc2F)=O)CC1(F)F N1(C(c2ccc(CSC)o2)=O)CCN(C(=O)C(C)c2ccon2)CC1CCO c1(C(N(C(C(=O)N(CC(=O)NCCC)C)C)CC)=O)cc(CO)[nH]n1 c1(C(=O)NCC2CN(C(C(F)=C(C)C)=O)C(C)C2)cccn2nnnc12 Cc1ccc2sc(SCC(N3CCN(c4ncc(C#N)cc4F)CC3)=O)nc2c1 C(=O)(C1=CCCCCC1)N1CCC(C(C)NC(C2CC(C)SCC2)=O)C1 N#Cc1c[nH]c(=NC2CCC(C(=O)NC3(C(F)F)CCCC3)CC2)c2sccc12 C1(NC(CC2C(C)(C)C2(C)C)=O)CN(C(c2cnsn2)=O)Cc2ccnn2C1 C1(CCC(=O)NCCCSC)COCCN1C(c1cc(C)[nH]n1)C(=O)NC C1(N(C(=O)C(F)n2cccn2)CCC)CCN(C(=O)CC#N)C1 C1(NC(C(C(C)C)(C)C)=O)CN(C(C2C=CC=CC=C2)=O)C2(CCOCC2)C1 C1(NC(C(C)Sc2ccccn2)=O)CCC(CNC(C2(F)CCC2)=O)CC1 CC1(C)CCCC1CCNC(=O)CCCn1cc(COc2ccc(F)cc2)nn1 C12(C(=O)NC(CNC(C3(CC4CC4)CC3)=O)C3CC3)CCC1CC2 c1(C(=O)NC2(CO)CCN(C(C3(F)CCS(=O)(=O)C3)=O)C2)csc2cncn12 c1(CN2CCCC(C(=O)Nc3nccc(OC)c3)C2)ccc(F)cc1C(=O)O C1(C(=O)NC2C3CN(C(c4n(CCC)nc(C)c4)=O)CC32)CNC(=O)CC1C C12(C(N(CCN(C(=O)Cc3ccnc(OC)c3)CC)CC)=O)COCC(C1)C2 N(C(=NCC1CCCC1(C)C)NC(c1ccccc1)C)Cc1nc(C)on1 N1(C(C(CC)N(C(=O)C(C)N(CC)CC)C)=O)CC2CC=CCC2C1 C(C1CCCN1C)=CC(=O)NC1CCC(NC(c2cc(C)on2)=O)C1 c1(C(N2CC3C(CNC(=O)C(O)c4ccsc4)(C3)C2)=O)ccc(=O)n(CCO)c1 c1(C(=O)NC(CCNC(Cc2nc(C)[nH]n2)=O)C)ccccc1OC1CC1 N1(C(c2c(C)cccc2)=O)CC2CCCC(C(=O)NC(C)(C)C3CC3)C2C1 c1(CC(=O)NC2C(NC(C3(NC(C)=O)CCCC3)=O)C2)ccc(F)c(Cl)c1 NC(=O)CC(C(=O)NCc1ccccc1)NC(c1n[nH]c(=N)[nH]1)=O CCCCCCC(COC)(c1nnnn1C1COC1)NCC(C)(C)OCCO c1(-c2cncc(-c3n(CC4(C5C(O)COC5)CC4)ccn3)c2)ccc(Cl)nc1 C1(C)(CNC(C(CNC(c2c(CC)noc2)=O)C)=O)CCC(=O)N1C C1(C)(C(=O)NCC(c2cccc(Cl)c2)NC(C(C)(C)OC)=O)CCCOC1 C(=O)(C1CCOc2c(F)cccc21)N(CCNC(c1c(C#C)cn(C)n1)=O)CC Cn1cnc(C=CC(=O)NCc2cccc(CNC(c3cc(Cl)cnn3)=O)c2)c1 C12(C(=O)NCCCNC(c3ccc(OCC(C)C)cc3)=O)CCCN1CC(O)C2 CC(O)(C(=O)NCC1CC2CC1CN2C(C1CC1C1CCC1)=O)C(F)(F)F C(C(C)(C)C#CC(=O)N(C(C)C(C)C)C)NC(COC)=O N1(C(CCC2CC(C)C2)=O)CCC(C(=O)NCC(c2ccsc2)C)C1(C)C n1(CCOC(c2nnnn2C2CC2)C2CC2)nccc1CC1CC1 N1(C(C2(COC)CCOC2)=O)CC(NC(c2coc(Cl)n2)=O)C2(CCOCC2)C1 c1(C(=O)NC(CCNC(c2c(C)n(C)nc2)=O)C)nccc2ccsc12 C1(CNC(C(COC)(C)C)=O)C(C2CC2)CCN1C(C1CC(C)C1)=O N1(C(Cc2ncc(C)o2)=O)CCC(NC(=O)C=Cc2ccc(Cl)s2)C(F)C1 CC(CC(C)(C)C)C(=O)NCC1CCC2CN(C(c3ncn4c3CCC4)=O)CC12 c1(C(N(C(CNC(CN(CCCCCC)C)=O)C)CC)=O)c(C)cnn1C(C)C c1(N2C(CCCNC(C3CCCCO3)=O)CCC2)ccc([N+](=O)[O-])cc1Cl CCCC(O)C(=O)NCCNC(C1CN(C(=O)CSc2nncs2)C1)=O Cc1nc2nccc(NCC3(C)CCN(C(c4nc(Cl)cs4)=O)C3)n2n1 c1(C(c2ccc(NC)cc2)NC(C2C(CCCC)CCC2)=O)ccc(C)cc1F C1(NC(=O)C(C2CCCC2)C2CCCC2)CCCC1CNC(=O)Cn1nccn1 C1(CC)C(NC(c2ocnc2C2CC2)=O)CCCN1C(C1CC(=O)N(C)C1)=O c1(C(=O)NC(CCNC(c2c(C)ncnc2O)=O)C(C)C)ccnc2[nH]nnc12 C(CC(CC)C(=O)NCC(C(C)C)NC(=O)CCc1cnc(O)[nH]1)=CC N1(C(C(C(C)C)OC)=O)CC2(COC(CNC(=O)Cc3[nH]cnc3C)C2)C1 n1(C(C(=O)NCCC(P(C)(C)=O)N2CCOCC2)(C)C)ccc2ccccc2c1=O N1(C(Cc2cc(C)no2)=O)CCCC2CN(Cc3csc(Br)n3)CC12 c1(OC)c(Cl)cc([N+](=O)[O-])c(Cl)c1C(=O)NCC1CCN1C(=O)OC(C)(C)C N1(C(CN(C)C(N)=O)=O)CCc2ccccc2C(NC(=O)C=CC2CCOC2)C1 c1(C(C(=O)NC)N(C2(C#N)CC2)C)ccc2c(c1Cl)OCO2 Cc1cc(C(=O)NC(C)C(CO)NC(C2COC(=O)N2)=O)cc(C)c1Br C1(NC(c2cccc(CC)c2)=O)CC(C2CCN(C(c3ccc(O)cn3)=O)C2)C1 Cc1ncc(CN2CCC(c3c[nH]cn3)CC2)n1-c1cnn(C)c1 c1(N(C(=O)CN2CCC3CCC23)C)ccc(-n2cccn2)c(F)c1 c1(SC)nc(NC(=O)NC(c2ccccc2Br)CF)cc(C#N)n1 c1(COC(=O)C(c2ccccc2Br)F)ccc(C(F)C(F)F)cc1 c1(C(N2CC(CN(C(C3C(C)OCC3)=O)C)C2)=O)cc(F)cc([N+](=O)[O-])c1 CN1CC=C(C(=O)NCCCNC(c2conc2C(C)(C)C)=O)C1 C1(CN(C(C2CC(C(=O)OC)C2)=O)C)CCCC(CNC(c2cc(Cl)no2)=O)C1 C1(C(=O)OC)CN(C(c2cc(-c3cn(C)cn3)on2)=O)CC1C(=O)OC C(=O)(C1=C(C)OCCS1)NCC1CCCC(C(=O)NC2(CCOCC)CCC2)C1 N1(CC(N2CC(CNC(C(C)=C3CC3)=O)C(C(F)(F)F)C2)=O)CCC(=O)NC1=O C=CCC(F)(F)C(=O)NC1CCCC1CNC(c1n[nH]cc1-c1ccccc1)=O CC1CCC(C(N2CC(F)(F)C2C2CC2)=O)N1C(C1CN(C)CCO1)=O C1(CNC(c2cncc(OC)n2)=O)CN(C(=O)C(F)C(C)C)CCN1C C(C(COC)C(F)(F)F)N(C(c1c(C(=O)OC)cn(C)n1)=O)C Cc1nc(C)c(CNC(C2CC(C)N2C(c2cc[nH]c2)=O)=O)s1 c1(C(=O)NCCCC(C)NC(=O)C=Cc2cnccn2)cccn2ncnc12 N1(C(c2cnc(C)nc2C)=O)CCC2(CC(C(N3CCOCC3C(C)O)=O)C2)C1 c1(C(N2C(C(=O)NC3CCC(OC)C3)CC(F)C2)=O)cc(F)cc(Br)c1 C(=O)(C#CC1CCCO1)N1CCCC(O)(CNC(c2c(OC)c(F)ncc2)=O)C1 N1(C(C=Cc2c(C)cccc2)=O)CCCC12CCN(C(c1nncs1)=O)C2 c1(OC)ccc(O)cc1NC(=O)CN(C1CC(C#N)C1)C(=O)C=Cc1cscn1 C12(C(N(C3CCN(C(C(C)n4cnnn4)=O)CC3)CCO)=O)CCCC1C2(F)F N1(C(CCC2(C)CN(C(=O)C=Cc3ccncc3)C2)=O)CC2CCC2(C)C1 N1(C(C(N2CC(C)C2)C)=O)CC(NC(c2cnc(-c3ccccn3)s2)=O)C(O)C1 C(=O)(C#CC1(C)CCCO1)N(CC(=O)NCC(C)O)CCC Cc1cc(C(=O)NCC2CCC(C)CN2C(=O)CN2CC(C)C2)nc(C)c1 CC1CN(C(=O)C(=O)Oc2cccc(OC)c2)CC1(C)CC1CCC1 C1(CN(C(c2ccc(CCC)[nH]2)=O)C)CCCN(C(c2cnc(C)s2)=O)C1 CC12COC(C(=O)NCC3CN(C(=O)CSc4n[nH]c(O)n4)CC3O)(C1)C2 N1(C(COCCCC)=O)CCC2C(NC(=O)Cc3c(F)cccc3Cl)C2CC1 C1(NC(c2ncn(C)n2)=O)CCCC(NC(=O)C(F)=CC2CC2)C1 C1(NC(Cc2c(OC(C)C)cccc2)=O)CN(C(C2C=C2C)=O)C2CCCCC12 N1(CC(=O)NCC)CCN(C(c2cc(Br)ncc2F)C(=O)NCC(F)F)CC1C CCC(C)C(C(=O)N(C)CCN(C)CCO)N(C)C(C1(n2cncn2)CC1)=O Cc1ccc2c(c1)C=C(C(=O)N1CC(NC(C3(CO)CCCO3)=O)C(C)C1)CO2 Cc1nc2c(C(=O)NCCCN(C(=O)C(C)CC3CC3)CCO)cccc2o1 CCCC(CNC(C1C2COCC12)=O)NC(=O)C=C1CCCCC1 c1(NC(C2=CCCN(c3ccnc(C)n3)C2)=O)c(Br)cc(Cl)cc1C#N N#Cc1cc(C(=O)NCC23CC2CN(C(c2ccc(O)nn2)=O)C3)c(F)cc1F C1(CNC(C(COC)OC)=O)CN(C(=O)C(F)(F)CO)CC1O CCCCC(=O)N1CC(C(=O)NC(C(O)CO)C2CC2)(CC)C1 CC1(C(=O)NC(C2CCCC2)CNC(c2ccnc(S)c2)=O)CC(C2CC2)=NO1 c1(C(=O)NC(CC)CNC(=O)Cn2nnc(=O)[nH]2)cc2ccc(F)cc2nc1C C=CCCC(C)(C)C(=O)NCC1CC2CCC1N2C(c1ccc(CO)cc1F)=O c1(C(=O)NC(c2ccc(C)c([N+](=O)[O-])c2)C)cc2c(nc1N)CCCC2 C1(C)(CC)CC(NC(c2n[nH]c3c2CCC3)=O)CN1C(c1ccnc(C)n1)=O C1(NC(=O)NC(c2n(CCC)cnc2)C)CCN(C(=O)OC)CC1 Cc1ccc(C(C)(C)C(N2CCC(CNC(C3CCOC(=O)N3)=O)CC2)=O)cc1 C(=O)(C(CO)C(C)(C)C)N1CC(N(C)C(=O)NCCNC(=O)C(F)(F)F)CC1(C)C C1(C(=O)NC(CO)C2CC2)C2CN(Cc3ccc(N4CCCC4)o3)CC12 C1(C(=O)NC2(C(NOC(CCC)CC)=O)CCOCC2)CC2(C1)CC2(F)F C1(C(=O)NCCCc2c(C)n[nH]c2)CCC(C(C)C)N1C(C1CC(C2CC2)C1)=O Cc1cc(NC(c2cnn(CCNC(=O)C(C)OCCC(C)C)c2)=O)c(O)c(C)c1 C1(C(c2ccccc2)NC2CC(F)(C(=O)OCC)C2)CCC(C)=C(C)C1 C(=O)(C(C)(C)C(F)(F)F)N1CCCCC(NC(C(C)Sc2ccc(C)cc2)=O)C1 CC1=NOC(C(N2CC(C)(NC(=O)CSc3cc(-c4ccccc4)on3)C2)=O)C1 C#Cc1cccc(OCC(=O)N(C)CCNC(=O)C(C)c2ccco2)c1 CCCC(CNC(=O)CC1CN(C(=O)CCCC2CCCO2)CC12CC2)CCC c1(C(N2CC(C)C(NC(=O)Cc3cccnc3)C2)=O)ccnc2c(F)cccc12 c1(C(N(CC(=O)NCC(F)Br)CC2CC2)=O)c[nH]ccc1=O N1(C(C(C2CCOCC2)C)=O)CC2CC2(NC(=O)CCc2ncccn2)C1 N1(C(C(COC(C)=O)C)=O)CCN(C(c2ccc(F)c(N)c2)=O)CC1CO S(=O)(=O)(c1[nH]c(=NCC(C)(C)C2CC2)ccc1Br)N(C1CCN(C)CC1)C1CCC1 C1(NC(c2ncc(OCC)nc2)=O)COC2(C1)CN(C(c1nncn1C)C)C2 c1(C(=O)Nc2nc(C(C)(C)C)[nH]n2)cc(N2CCNC2=O)ccn1 Cc1cc(=NC(=O)C2CN(C(c3cocn3)=O)CC2C2CC2)[nH]n1C1CC1 c1(C(=O)NC2CN(C(CC(C(C)C)O)=O)CC2N=[N+]=[N-])n[nH]c2ccc(Cl)cc12 C1(NC(CC(CC)O)=O)CCCCC12CCN(C(c1sccc1F)=O)C2 C1(C)(C(N2CCCC(C(C)NC(c3c(C)ccs3)=O)C2)=O)CCN(C)CC1 c1(C(=O)NCCNC(=O)C#CC2CC2)c(Br)ccc(C(F)(F)F)c1F c1(SCC2N(C(C(C(=O)OC)C)=O)CCOC2)cc(F)cc(I)c1 Cc1ccc(Cl)c(S(=O)(=O)Oc2cc(C)cc(C)c2)c1 c1(NC(C2(F)CCN(C(C3(CC=C)CCC3)=O)CC2)=O)ccc2nccn2c1 CC1CC(C)OC1C(N1CCCCC1C1CCCN(c2nccc(Br)n2)C1)=O c1(CNC(=O)NCC(c2ccco2)N(CC)CC)cnc(Br)c(F)c1 N1(C(CC2CC(=C)C2)=O)CCC(N=[N+]=[N-])(C(=O)Nc2cccnc2OC)C1 C1(NC(c2cnc3c[nH]nc3c2)=O)CC2CC(C1)N(C(C1CCCC(O)C1)=O)C2 c1(C(N2CCC(C)(C(=O)Nc3cncnc3)C2)=O)ccnc(Br)c1Cl C1(NC(C(C)Cc2ccccc2)=O)CCC(CNC(c2ccc(F)nc2)=O)CC1 C1(NC(C2CCN2C2CCCC2)=O)CCN(C(c2cn(C3CC3)nn2)=O)CC1F N1(C(CC2CC(OC(C)(C)C)C2)=O)CCN(CCNC(=O)CCF)CC1 c1(C(=O)NCCCCCN(C)C(C2C3CS(=O)(=O)CC23)=O)ccc(F)c(O)c1F CC(CC(C)NC(c1ccn(C2CCCC2)n1)=O)NC(=O)C(C)(C)C C12(C(=O)NC3CCC(NC(CC(C)(C)OC)=O)CC3)CCC(C1)c1ccccc12 CC1CN(C(=O)C(C)(C)C(=O)OC(C)(C)C)CCCN1C(=O)C(O)CC1CC1 C(CC(N)=O)(C(=O)NCC1(C)CCCCO1)NC(c1cc(CC)nn1C)=O c1(C(=O)NCc2ccccn2)csc2c1CCN(C(c1cccn1C1CC1)=O)C2 C1(C(=O)NC2CN(C(=O)CCn3ccc(C)n3)CC2O)(OC)CCCOC1 Cc1ncc(CCC(N2CC3(CC3)CC2CNC(c2nccs2)=O)=O)c(O)n1 N1(C(C2C(CC)OCC2)=O)CC2(C=C(C(=O)N(CCC(=O)OC)CC)CO2)C1 c1(CC)ncncc1C(=O)NCC1(F)CCC(NC(=O)C(C)(CO)OC)C1 C(=O)(CCCC#N)NCC(CC)NC(=O)Cc1nc(Br)sc1C n1(C(C)C)ccc2cc(C(N3CCOC4(C3)CN(C(=O)C3CC3)C4)=O)ccc12 C#CCCC(O)C(=O)NC(C)(CNC(c1ccc(C)n1C)=O)CC(C)C N(C)(S(=O)(=O)N1CC(C)CCC12CN(C(=O)OC(C)(C)C)C2)CCC(C)C c1(CN2CCCC(c3oc(COCC)c(C)n3)C2)cc(Cl)ccc1OCC(=O)O C1(C(=O)NCC(CC)NC(=O)C(c2cccnc2F)(C)C)CC(=O)N(C2CC2)C1 N1(C(CN2CC(C)(OC)C2)=O)CCC2CCCC12C(=O)NC1CCSC1C N1(C(c2cn(CC)nn2)=O)CC(NC(C2CC23CCOC3)=O)C2CCCCC12 Cn1cc(C(=O)NC(C)(C)CNC(c2ccccc2)=O)c(-c2cccc(F)c2)n1 c1(C(=O)NC(C)CCNC(C2CC(C)(O)C2)=O)nn(Cc2ccccc2)cc1Cl C1(C(N(CCC)CCNC(=O)Cc2c(F)cccc2Cl)=O)CCN2CCCC2C1 N1(C(C2C(C(=O)OC)C2)=O)CCC2(CCC(NC(=O)CN3CCCNC3=O)C2)C1 c1(NC(C2CCN(C(C3(Cl)CC34CCC4)=O)C2)=O)cccc2c[nH]nc12 N1(C(COC(C)C)=O)CCCC(CO)(NC(=O)C(c2ccc(Cl)cc2)=O)C1 CCC(C)(C(=O)NCC(C(=O)NCc1ccc[n+]([O-])c1)OC)OC c1(C(C(=O)OC)(C)C)cccc(-c2noc(CSCC3CCOC(C4CC4)C3)n2)c1 CCCC(CCCO)C(=O)NC(C1CN(C(=O)CC(C)(O)c2ccccc2)C1)C Cc1ccc(NC(=O)C(CC2CC2)NC(=O)CCF)cc1.C1C(O)CNC(=O)C(=O)N1 c1(CC(=O)NCCNC(C2C(C)C2)=O)ccc2sccc2c1 C(CC(CC)C(=O)N(C)CC1CN(C(c2ccc(C(C)C)cc2)=O)CCO1)=CC C=CCC(C)(C(=O)NC1(C)CCN(C(c2n[nH]cc2C2CCC2)=O)CC1)N(C)C C=CCC(CC(C)C)C(=O)NCC(C)(O)CNC(=O)CC1=CCOCC1 N1(C(C(=O)NCCC2CC2)c2ccco2)CCC(C2CCC2)C1 C(CC(CC)C(=O)NCC1CCC(C(N2CCC(C)C2CO)=O)CC1)=CC Cn1nnc(CNC(=O)CCC2CCCOC2)c1C(=O)NC1CCCC(CO)C1 C#Cc1cccc(C(=O)NC(C2CC(NC(=O)CC3CCCCO3)C2)C)c1 C12(CN)CCC(NC3CCC34CCNCC4)(CC1)CO2 CC(CCC(=O)NC1CCCC(CO)C1)NC(=O)CNC(=O)OC(C)(C)C N1(C(CCC2CC(OC)C2)=O)CCN(C(c2cn3ccsc3n2)=O)C2COCC12 C1(F)(C(N2CCC(CCNC(C3C(C)CCC3)=O)CC2)=O)CCN(C)CC1 c1(OCC(=O)NCC(C)(CO)NC(C2C(CCOC)C2)=O)cncc(Cl)n1 c1(C(=O)NCC#CCNC(=O)CC2CCC3CC23)c(F)ccc(F)c1F C(C(F)(F)C(=O)N1CCOC(CC(=O)NOCC(N)=O)C1)OC c1(C(c2n(CCC)nnn2)NCCCC2CC2(Cl)Cl)ncc(OC)cc1F c1(N(C2C=CCCC2)C)ccc2cc(S(=O)(=O)N3CCCC3)ccc2n1 C1(n2cc(CCCCC)nn2)CCN(C(c2nnc(CC)s2)=O)CC1O Cc1ccc(C(=O)NCC2CCN2C(=O)C=Cc2cc[nH]n2)cc1Br N1(C(CC(C)C2CC2)=O)CC2(CCN(C(=O)COC(F)F)C2)C1 C1(CNC(c2cncc(C)n2)=O)CC(C)(C)CN1C(=O)C(O)C(C)C c1(C(N2C(C)CCC(NC(C(C#C)(C)C)=O)C2)=O)ccc(F)c(F)c1F C1(C(=O)NCC2C(NC(CCNS(CC)(=O)=O)=O)CC2)CC(S(N)(=O)=O)C1 c1(NC(C2N(C(c3cnc(OC)nc3)=O)C3C(C2)C3)=O)c(OC)ncc(Br)c1C C1(NC(C(C)OCC2CCCO2)=O)CC2CN(c3nc(Cl)ncc3CO)CC2C1 N1(C(CC2OCCN(C(C3(CC(C)C)CC3)=O)C2)=O)CC2CCCCC2C1C C=CCC(C(=O)NCCC1=CCN(C(c2ccc(Br)c(C)c2)=O)CC1)C(C)C C#CC1CCC(CNC(C2C(C)CCN2C(c2nccn2C)=O)=O)CC1 C1(CNC(CSCC=C)=O)CCC2CN(C(=O)CC3CC(=O)NC3=O)CC12 CC1CC(C(=O)NC2CN(C(c3ccc(-c4cnn(C)c4)o3)=O)C2)CC(C)C1 Cc1ccc(C(=O)NC(CN)CC(C)C)cc1CO C#CCCCCN=C(NCS(C)(=O)=O)NC1CCS(=O)(=O)C1 N1(C(C=CC=CCC)=O)CCCC2(CNC(c3cn(C)c(C)n3)=O)CCCC12 Cc1nc2cc(-c3ccc4oc(C(N5CCCCC5CO)=O)cc4c3)ccc2s1 N1(C(C2(CC(C)C)CCCC2)=O)CCCC(CN(C)C(C2(CC#N)COC2)=O)C1 C(=O)(C(C)CS(C)(=O)=O)NC1CC2C(NC(c3c(CC)nccn3)=O)C2C1 C1(CNC(C2(C(C)C)CCC2)=O)CCCCC1C(=O)NCc1c(C)nsc1 c1(C(=O)NCCc2cc(C(N(OC)C)=O)no2)cc(O)ncc1F c1(CCCC(=O)NCC2N(C(C3N(CC)CCC3)=O)CC=C2)cc(C)ccc1C C1(c2cncc(OCC)c2)CC2CCCCC12 N1(C(C(C)N(C(c2ccc(C)o2)=O)C2CC2)=O)CCc2nocc2C1 C12(NC(=O)Cc3cscn3)CCCC1CN(C(c1ncsc1C(F)(F)F)=O)C2 C12(NC(C(N3CCSCC3)C)=O)CCOC(CNC(=O)C3=NNC(=O)C3)(C1)C2 C1(CC)CS(=O)(=O)CC1NC(=O)CCc1nc(CC(=O)NC(=O)C=NOC)no1 C1(C(N(C)CC2COCCO2)=O)CN(c2ccc(CS(C)(=O)=O)cn2)CCC1O N1(C(C(C)NC(=O)NC)=O)CC(C)(NC(c2coc(Br)c2)=O)C1 N1(CC)N=C(C(=O)N2CCCC2(CNC(=O)C2=CCCC2C)COC)CCC1=O C1(C(=O)NC2CCN(C)C2(C)C)CCN(C(=O)CCc2nc[nH]n2)C(C)(C)C1 C1(C(C)NC(CCC=CCC=C)=O)CCN(C(=O)C=Cc2ncc[nH]2)CC1 CCCCC(O)CC(=O)N1CCC(CCC(=O)NCC2(C)CC(O)C2)C1 C1(CCNC(c2cnn[nH]2)=O)(NC(C2CN(S(CC)(=O)=O)C2)=O)CCCC1 c1(C(N2CC(CC(C)NC(CN(CC)CC)=O)C2)=O)cnc(C)nc1C C=CCCCCCN(C(=O)CC(CNC(=O)CC1CCC(=O)N1C)OC)C C1(C(=O)NCCC=CC)CC2(CCN(C(=O)CCC=CC(C)C)C2)C1 CC1(C(=O)NCC(CNC(c2cnc(C3CC3)[nH]2)=O)CO)Cc2ccccc2N1 c1(C(=O)NCc2occ(C(=O)NCCc3cccc(F)c3)n2)cccc(F)c1O c1(C(=O)NC2CN(C(CC(=C)C)=O)C(C)C2)cccc(OC(C)C)c1F C(CCCC(C)NC(=O)CNC(c1cscn1)=O)NC(C12CC(OC)C1C2)=O C(=O)(C(CC(C)C)NC(C)=O)N(C1CCN(C(C2C=CCC2)=O)C1)CC N1(C(c2ncc(C)cc2F)=O)CC(CNC(c2c(C)nsc2N)=O)C2(CCC2)C1 C1(NCc2c(F)ccc(C(F)(F)F)c2F)CC12CCc1cc(Br)ccc12 C1(C(C)NC(=O)CC2OCCC2C)CN(C(c2ccncc2Cl)=O)CCO1 c1(C(=O)NC(CC(C)NC(=O)C(C)(C)n2ccnn2)C)ccc2[nH]ccc2c1 c1(C(N(CCCNC(c2cc(Br)c(C)cn2)=O)CC)=O)c(C)ccc(C)c1O C1(N(C(=O)CC2OCCO2)C)CCCN(C(C2(C3CCC3)CC2)=O)CC1 CC1(C)CC(=O)N(CC(=O)NCCCOCCNC(C2CC2(F)Cl)=O)C1=O C(=O)(CS(=O)(=O)CC(=O)NC1(CNC(=O)CCc2ncco2)CCOC1)OC C1(CC)CCCC1(C)C(=O)N(CCCC(=O)NC1CCOC1C(C)C)C C1(CC=C)(NC(c2occc2CNC(=O)C(c2ccn(C)c2)C)=O)CCOCC1 C1(N(C(=O)CCOC2CC2)C)CCCN(C(C2(C)COCCO2)=O)C1 C1(CC(=O)NCCCO)CN(C(c2cn(C3CC3)nn2)=O)CC12CC2 c1(C(=O)NC(C)CCN(C)C(C2CC3CC3C2)=O)cccnc1OC(F)(F)F c1(C(C)=O)cc(=NCC2CC(C)(C)CCC2NC(=O)Cc2cnsc2)[nH]cn1 CCCCCC(O)CNC(C1CCC2(CC2)N1C(=O)C(C)(C)COC(C)C)=O O=C(N=c1[nH]c(Cl)ncc1O)C1CN(C(=O)C2CC2)CCC1(F)F N1(C(C(CC)CCOC)=O)CC(C)(C)OCC1CNC(=O)CC(C)(C)C1CC1 C=CC(CC)CC(=O)NCC1(C(C)(C)C)CCN(C(=O)CCC2CCC2)C1 c1(NC(CN(C(c2ccc(OC)cc2)=O)CC)=O)ccc2cccnc2c1 Cc1nnc2n1CC(NC(=O)C(N1CC3CC4CC3C1C4)=O)CC2 C1(C(=O)NCCN(C(C)C)CC)CC2CCCC2C1.C1CCCC(CNC=O)C1 C1(NC(c2cc(C)on2)=O)CC2(C1)CC(C(N1C(C)CCCC1C)=O)C2 C(=O)(CC(C)(C(F)F)N(C)C)NC1CC(NC(c2c(C)scn2)=O)C1 Cc1nc(CC(=O)NCCCC2(NC(c3ccn(CCO)c3C)=O)CC2)c(C)s1 N1(C(C(C)NC(=O)C(C)(C)C)=O)CC(NC(C2CNC(=O)C2)=O)C2(CCOCC2)C1 c1(N2CCC(C)(C)C(CNC(=O)C=C3CCCC3)C2)nc2cccc(Br)c2o1 Cn1nc(C2CCC2)cc1C(N1CC2CC1C2CNC(C1CCCOCC1)=O)=O C(=O)(CCS(=O)(=O)N(C)C)NCC(CNC(C(C)Oc1ccc(C)cc1)=O)F C1(NC)CC(C)CN(CC2CC(F)(F)C2)C1 C(CN=c1[nH]c(Cl)nc2[nH]ccc12)(c1ccccc1F)NC(C(C)C1CC1)=O CCC(CC(=O)NCC1COCCN1C)N(C(=O)CN1C(=O)CCC1=O)C N1(C(C2(F)CCN(C(Cc3c(C)cccc3)=O)CC2)=O)CC2CCC(C1)N2C C1=CC=CC(=O)Nc2c1cccc2.C#CC(CCC)OCC c1(C(=O)Nc2cccc(NC(c3c(C)snc3)=O)c2)ncnc2c1ncn2C1CC1 CC(C)CCCOCC(N1CC(C(=O)OC(C)(C)C)C1)=O.c12cnc(s1)[nH]c2=O c12ccc(cc1)OC2.c1(C(c2nnnn2C2CC2)NC(C)C)ccccn1 C(=O)(N=c1ccn(C)[nH]1)c1cc(CNC(c2cncc(C)c2)=O)oc1 c1(C(=O)NCCCCCCNC(C2C(C)(C)C2(F)F)=O)ccc(Cl)cc1N c1(C(C(=O)NCC(C)(CO)NC(Cc2ccc(C)s2)=O)C)cn(C)nc1C c1(C(=O)NCC2(C(=O)NC(c3cn(C)cn3)C)CC=CC2)cc2cnccc2[nH]1 C1(C)(NC(C=C2CCN(C)CC2)=O)CCCN(C(C2CCNC(=O)C2)=O)C1 CC1CN(C(=O)C(=O)NCc2ccc(Cl)o2)CCN1C(=O)OC(C)(C)C C1(CC(=O)NCC2(NC(C34CCC3CC4)=O)CCC2)CCS(=O)(=O)C1 N1(C(C2(CO)CCN(C(C(CC=C)C)=O)C2)=O)CCC(CC)(CC)CC1 N1(C(c2c(C)noc2C)=O)CCC12CN(C(C1(C#N)CCCC1)=O)C2 Cc1ccc(F)c(CN(c2cc(N(C)C)nc(NC3CNCC(C)C3)n2)C)c1Br Cc1cc(=N)[nH]cc1C(=O)NC1CCC(C)N(C(c2ncoc2C2CC2)=O)C1 C1(C(N(C2(c3cc[nH]n3)CC2)C)=O)CC2CCCC2N1C(=O)Cn1c(O)nnc1O Cn1ncc(C(=O)NCCC2CC(NC(c3ccc(Br)o3)=O)C2)c1F C(=O)(NNC(=O)C1CCC(n2cc(-c3ccccc3F)nn2)C1)NCCOC C(=O)(C(C)(C1CCC1)NC(c1cc(Cl)ns1)=O)NC(C)CCO C(=O)(C1CCc2cccc(Cl)c21)NCC1C(C)C1 Cc1c(C(=O)NCC(C)CNC(=O)CCc2cn(C)nn2)nnn1C(C)C C(=O)(C(C)(C)CC(F)(F)F)N1C(CNC(c2cc(OC)ncc2Cl)=O)CCCC1 CC(C(=O)N1CC(F)(F)CC1CNC(C1CSCCS1)=O)S(C)(=O)=O c1(C(C(=O)OC)NC2CCCC2CN2CCCC2)cc(OC)cc(OC)c1 C(=O)(C(C)(C)CC(F)F)NCCCCCCN(C(=O)CC1CC(O)C12CCC2)C C1(C(N2C(CNC(=O)C(C)(C)CN(C)C)CC(OC)C2)=O)CCc2nc[nH]c2C1 C(=O)(CC(F)(F)CC)N1C(C2CCN(C(c3cnc(SCC)s3)=O)C2)CCCC1 C#Cc1cnn(CC(=O)NCC(CC(C)C)NC(C2(SC)CC2)=O)c1 c1(CC(N2CCC(C(N)CO)CC2)=O)ccc(Cl)c(I)c1 C1(C(=O)NCCC2C(C)CN(C(=O)CC3COCC3O)C2)CC(F)(F)C1(C)C c1(OC)cnc(Br)cc1C(=O)NCCS(=O)(=O)NC1CCCCC1 c1(C(N2CC(O)(C(C)NC(=O)C=CC3CC3)C2)=O)c(F)ccc(F)c1Cl c1(C(=O)NCCOC2CCN(C(CC=C(C)C)=O)C2)c(C)nn(C)c1Cl c1(Cn2cc(COc3c(C(N)=O)cccc3)nn2)cc(Cl)ccc1F c1(C(N2CC(CNC(C(C=C)(C)O)=O)C(C)CC2)=O)ccc2c(c1)CN(C)C2 c1(NC(C2C3(CCN(C(C(C)=O)=O)C3)C2)=O)nc(C)c(Br)nc1Br N1(C(=O)Cn2cc(CNC3CCNCC3)nn2)CCn2ncnc2C1 C1(CNC(COCCCOC)=O)CN(C(=O)CCN2CCOC2=O)CC1C(F)F C1(C(=O)NC(C2(C(=O)N(CCCC(C)(F)F)C)CC2)C)CC(O)CN1C S(=O)(=O)(CCCCS(=O)(=O)NC12CCCC1CS(=O)(=O)C2)NCC#CCOC C1(C(=O)Nc2c(C(=O)OC)ccc(C)n2)CCC2(CN(C(=O)CNC(N)=O)C2)O1 c1(OC)ccc(-c2nc(C(=O)NCC(C)CNC(=O)COC(C)=O)cs2)cc1 C1(F)(CNC(c2ccc(Cl)s2)=O)CN(C(=O)CCOC2CCCOC2)C1 C(=O)(C1Cc2ccccc21)NC(C1CN(c2nc(C)nc(Cl)c2C)C1)C c1(C(=O)NC2CCC(C(N(c3ncccc3N)C)=O)C2)cc2[nH]ccc2cc1Cl C1(CCNC(C2(CCC)CC2)=O)COCCN1C(C1CSCN1C(=O)CC)=O c1(OC)ccc(C(=O)NCCC(C)NC(C2(F)CCS(=O)(=O)C2)=O)cc1OC CCCCCCC(=O)NCCN(C(=O)C(c1c(F)cccc1F)C)CC N1(C(C(CC)C(=O)OC)=O)CCC2(CC1)C(NC(=O)C(C)C(C)O)CS2(=O)=O C1(N(CC=C(C)C)C)CCN(C)C1.C1(C(=O)N)(C(F)F)CCC1 C1(C(N(C(C(N2CC(CC)(CO)C2)=O)C2CC2)C)=O)CC=CCC1C n1(C(C)C)cc(C(N2CCN(C(c3cnccc3C#N)=O)CC2C)=O)ccc1=O c1(C(=O)NCC(=C)CCNC(C2CCC(=O)O2)=O)cc(C)nc2[nH]nc(O)c12 Cc1c(C(=O)NC(C)CNC(c2c(O)cccc2Cl)=O)sc2cncn12 C1(N(C(C(C)OCC=C)=O)C)CCCN(C(=O)Cn2cncn2)C1 N1(C(CN(C)C(N)=O)=O)CCCCC1CNC(=O)Cn1cnc(=N)[nH]1 C(=O)(C(O)CC(N)=O)NC1(C(=O)NC(C(C)(C2CC2)OC)C)CSC1 c1(N(C(c2nccs2)C)C2CC2)ccc2c(c1)C(C)CN2C(=O)OC.C(C)(C)(C)O C=C(C)CC(C)C(=O)NC1CCC(NC(c2cccc(-c3nc[nH]n3)c2)=O)C1 C#Cc1cnc(C(=O)NCCc2cc(C(=O)NCC(F)CO)no2)c(C)c1 c1(CNC(C2(F)C(C)C2)=O)ccccc1CN(C)C(c1cnn(C)n1)=O C1(CNC(COCCC#C)=O)CCCN(C(c2c[nH]nc2-c2cnn(C)c2)=O)C1 c1(N(S(CCCOC)(=O)=O)C2CCNCC23CC3)ccc2nc[nH]c2c1 c1(-c2c(C(=O)NCC(C)(C)NC(C(C)NC(C)=O)=O)cno2)cccc(Cl)c1Cl n1(CC(N2CC(CC(=O)NCc3c(C)nns3)C(C)C2)=O)ccc([N+](=O)[O-])n1 c1(CC)ccsc1C(=O)N(CC(=O)N(C1CC(CO)C1)C)C1CC1 c1(C(=O)NCC2(O)CC(NC(C(CCC#C)O)=O)C2)[nH]c2c(C)cccc2c1C c1(CCC(=O)NC(CN(C(c2csc(C3CCCO3)n2)=O)CC)C)cncn1C C1(CC(=O)NCCC(C)(C)NC(=O)CS(C)(=O)=O)COCCN1CC(F)(F)F c1(N(C)Cc2cccc(C)c2)nc(=NCCn2cnnc2)[nH]c2cc(F)ccc12 C(=O)(CC1=CCOCC1)NCC1CN(C(c2c(C)sc(C)c2C)=O)CC1C C(=O)(C(CC(C)CC)NC(c1ccc([N+](=O)[O-])[nH]1)=O)N(CCOCC)C c1(C(N2CC3C(N(C(C(CC)N(C)C)=O)C)C3C2)=O)cc2nc(C)[nH]c2cc1F CC1CC(C(=O)NCCCC(C)NC(C2C3CCC2CC3)=O)=NO1 c1(C(=O)NC(CNC(C2(CC)CCNC2=O)=O)(C)C)cc(OC)c(C)c(OC)c1 C(CCN=c1[nH]ncs1)OCCNC(C)(C)C(=O)OCC1CCN(C(C)=O)CC1 c1(OC)ccc(C(=O)NCC(C(C)C(C)C)NC(c2cccn2C)=O)nc1OC N1(C(c2c(C)onc2Br)=O)CCC(C2CCN(C(=O)C=C3CCC3)CC2)CC1 N1(C(C(C)(C)SC)=O)CCCC2(C1)C(NC(c1ncncc1Cl)=O)CCN2C C12(NC(c3c(-c4nc(C)sc4)c[nH]c3)=O)CCCC1N(C(=O)C(C)(F)F)CCC2 CCC(CN(C(=O)CN(C)C1CC1)CC)NC(=O)CCNC(c1ccco1)=O N1(C(CN(C)C(=O)C2CC2)=O)CC2(CC(NC(c3ccc(=O)n(C)n3)=O)C2)C1 C1(N(C(c2cnc(COC)s2)=O)C)CCCN(C(C2(CF)CC2)=O)CC1 CC1CCC(CNC(c2cc(Cl)c(Cl)[nH]2)=O)CN1C(c1ccncc1)=O N1(C(Cc2c(OC)ccc(Cl)c2)=O)CC(NC(=O)Cn2nccn2)C(C2CC2)C1 Cc1cc(C(N2CCC(C)N(C(=O)C3=CCOCC3)CC2)=O)n2ncnc2n1 CC1CC(CCNC(=O)C(C)(C)C2CCCC2)CCN1C(c1c[nH]cc1Br)=O C(=O)(C1=NOC2(CCC2)C1)N(C1CN(C(C2(C)CCCCO2)=O)CC1(C)C)C N1(C(c2n(C)nc(Br)c2)C(=O)NCCCNC(N)=O)CCOCCC1C1CC1 c1(CNC(C23CC(NC(c4cc(CC)n(C)n4)=O)(C2)C3)=O)c(F)cccc1F C#CCC(C)(C(=O)N1CC(C2(C)CC2)C1)NC(=O)CCCC1CCCO1 C1(=CC(=O)NC(CNC(=O)C(c2ccccc2)F)C2CC2)CN2CCC1CC2 CCC(C(=O)NCC1(CNC(=O)C(C)n2cccn2)CCC1)C1CCOCC1 C=CCCC(O)CNC(=O)C(F)CC1CN(C(C2(CCCC)CC2)=O)C1 C=CC(CCC)CC(=O)N1C(CNC(c2ccc(CN(C)C)cc2)=O)CC2CC12 CC(O)(C(=O)N1CCCC(F)(CNC(c2cnc(C(F)F)nc2)=O)C1)C(F)(F)F c1(N2CCC(C(=O)NCCNC(C(CSC)(C)C)=O)C2=O)ccc(Cl)c(Cl)c1 C(c1cc(OC)ccc1OC)=CC(=O)NC(CC)CNC(C1CCC(=O)N1)=O N1(C(C(CSC)O)=O)CCC(O)C(NC(C2COCCOC2)=O)C1 c1(C(=O)NCC(CNC(CC(COC)C)=O)OC)cc2sc(Cl)cc2s1 C1(C(N2CCC(F)(F)CC2)=O)CC2(CC2)CN1Cc1ccc(Cl)cc1C(=O)O S(=O)(=O)(c1ccc(N2CCC(CN(C)C)C2)nc1)NC(C)C(C)(C)C C12(NC(c3c(NCC)scn3)=O)CCC(CC1)N(C(=O)C(C)=C(C)C)C2 c1(OCCNC(C2CN(CC)C(=O)C2)=O)cc(Cl)cc(Cl)c1 C1(NC(C(C2CCOCC2)OC)=O)CC2CCC(C1)N2C(c1cc(C)n(C)n1)=O c1(C(=O)NC2CN(C(C(C(C)C)O)=O)CC2F)cn2cccc(Br)c2n1 Cc1nccc(C(N2CCC(C)C(CC(=O)NC3CCN(C)CC3)C2)=O)c1N N1(C(C(=O)Nc2ccc(OC)cc2OC)C)CCC2(CCCCO2)CC1 C1(C(=O)NCCC(CC)(C)NC(c2cnsc2)=O)CC2C=CCC(C1)C2 N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCc1cc(F)ccc1Br C(C(CC(C)C)C(=O)N1CC(F)(CNC(C2CCCN2c2nccs2)=O)C1)OC N1(C(c2c(OC)oc(C)n2)=O)CCN(C(c2cc(Cl)ccn2)=O)CC(C)(F)C1 C1(COC)CN(C(=O)C#CCNC(=O)CC2CC(O)C2(C)C)C1(C)C C=CCCC(CC(C)C)C(=O)NCC1CCCN(C(=O)C2=C(C)CCOC2)CC1 Cc1nc(N2CC3(CCCC3NC(C3CC=CCO3)=O)C2)c(F)c(C)n1 Cc1cc(C)n(C(C)C(=O)NC(C)(CNC(=O)CC2(C)CC2)C(C)C)n1 CC1=C(C(=O)NC2CCC(CNC(c3ccc(Cl)nc3Cl)=O)CC2)SCCO1 CCCCCCC(C)(C)C(=O)N1CCC(C(C)(C)NC(C2CN(C(C)C)C2)=O)C1 C(CC(C)(C)C(=O)NCC(C)NC(C1CCCN1c1ccncn1)=O)OC C1(CNC(COC)=O)CC(CNC(=O)CNC(C2CCC2)=O)CO1 C(=O)(C(F)(F)c1nccn1C)N(CCCNC(=O)C(C)OCOC)CC C1(N(C)C(c2cc(O)nn2C)=O)CN(C(C2(C)CCCS2)=O)CC12CC2 C1(C(=O)NC(C)CN2CCN(C(=O)C3=CCSC3)CC2)CCc2nncn2CC1 N1(C(C2COC(=O)O2)=O)CC2(CCC2)CC1CNC(c1cc[nH]c1C1CC1)=O C(CN=c1cc(C)nc(CO)[nH]1)(C1CCCC1)NC(C(C(CC)O)C)=O c12ccccc1NC(=O)C2.C1(CNC(C2C(CN(C)C)C2)=O)CCS1(=O)=O C1(C(=O)NCCC2N(C)CCC2)CN(C(=O)C(N)=O)CC12CCC2 N1(C(C(C)SCCCC)=O)CC2CC(C1)N(C(c1ccc(C)n1C)=O)C2 CC1CN(C(c2nn(C)nc2C(F)(F)F)=O)CCN1C(C1CCCCCC1)=O C(CCCCC(=O)NC(C)CCCC(=O)NC1(CO)CC(C)C1)=CC N1(C(C(CCC)C)=O)Cc2ccc(Br)cc2OCC1(C)C N1(C(CSCC#C)=O)CCOCC(F)(CNC(c2nnn(C(C)(C)C)n2)=O)C1 N1(C(c2nc(OC)oc2)=O)CC(OC)CC(NC(c2cnoc2CC(C)C)=O)C1 Cc1ccnc2c(C(=O)N(CC(C)NC(=O)C(F)(F)CN(C)C)C)cnn12 C(=O)(CCC(=O)NN(C)C)N1C(C)CC(NC(CCSCCCC)=O)C1 C1(NC(c2cc([N+](=O)[O-])n[nH]2)=O)C2COCC1CN(C(=O)C=CC1CCOC1)C2 C(=O)(C(O)CCS(C)=O)NC1CCN(C(C(c2c(OC)cccc2)OC)=O)CC1 CCC(CC)C(C(=O)NCC12CCC(CC1)N2C(=O)C(O)C(F)(F)F)OC c1(OC)ccc2cnc(N(c3ncnc4c3cnn4C)C3CNCC3O)nc2c1 C1(C(N2CCC(NC(COC)=O)C2C(C)(C)C)=O)CC(C)(C)OC(C)(C)C1 C1(C(N(CC(C)NC(C2SCCS2)=O)C)=O)CCCOC1C Cn1nc(CC(=O)O)cc1NC(N1CCCCC1CC(c1cccs1)=O)=O C1(C(=O)OC)CCCN(C(=O)C(c2ccc(Br)cc2)OC(C)C)C1C CC1CN(C(C2CCCNS2(=O)=O)=O)CC(C)N(C(=O)CCC2(O)CCC2)C1 c1(SC)nc(Cl)c(CNC2C(F)(F)CCN(C(c3ccc(O)nc3)=O)C2)c(Cl)n1 C1(N(C(CC2C(C)(C)C2)=O)CCO)CCCN(C(c2cnn(C3CCCC3)c2)=O)C1 C(=O)(C#CC1CCOC1)NC1CC(OC)CN(C(c2ccn(CC#N)n2)=O)C1 C(=O)(CC(CC)(C(F)F)NCc1cnc(-c2ccncc2)s1)OCC N1(C(C(CC)=CC)=O)CC(C)N(C(=O)COC2CN(C(C)=O)C2)CC1C CCC(O)CC(=O)NC1CCC(C(=O)NC2(C)CCCC2)C1 N1(C(=O)CCC2CCCO2)CCCC(OCc2ccc(O)nc2)C1 Cc1cc(=NC2CC(C(N)=O)C2)[nH]c(=NCCCc2nnnn2C)[nH]1 C1(CNC(CC(=C)C)=O)CCCN(C(c2ccncc2O)=O)CC1 n1(CC)ncnc1C(=O)NCC(C1CCCC1)NC(C1CCC(=O)N1)=O c1(OC)ccc(NC(=O)C(c2cn(C)nc2C)N(CC(C)OC)C)cc1 c1(CC)nc(C)oc1C(=O)NCCC(O)CNC(=O)CC(c1ccccc1F)C c1(-c2nc(CC)on2)cccc(C(=O)NCCN(CCC2CCOCC2)CC)c1 CCC(CC)C(C(=O)NCC1CN(C(C2CCCCCN2C)=O)CC1O)OC C1(C(=O)OC)(C(=O)NCC2SCC=C2C)CCCN(C(=O)OC(C)(C)C)C1 C1(C(=O)NCC(CC(=O)NCc2noc(C3CC3)n2)OC)CC(C(C)C)=NO1 Cc1nc(Cl)[nH]c(=NC2CCC(NC(=O)CCc3c(C)ncnc3O)CC2)c1Cl c1(C(=O)NCCC(=C)CNC(c2nnc(S)n2C)=O)c(C)ccc(C)c1N C(=O)(CCCN=[N+]=[N-])N1CCN(C2CCC(NC(C(C)N(C)C)=O)C2)CC1 C#CCCCCCC(=O)N1CCC(NC(=O)CCN2CCCCCC2)C1 C=CCC(CC=C)C(=O)N1CCCC1CCNC(C1CCCN1C1CC1)=O C1(C2CCCC2)(NC(COC2CCN(C(c3c(C)n(C)cn3)=O)O2)=O)CC1 C12(C(=O)NC(C3CN(C(c4cc(O)nc(O)c4)=O)C3)C)CCCCN1CCC2 c1(C(=O)NC2(C(=O)NCc3cnco3)C(C)C2)nsnc1O CCCCCC(C)(C)C(=O)NC1CCC(NC(=O)C(CC(C)C)N(C)C)CC1 C(CC(C)C)(C(=O)NCC(C1CC1)N(C)C(C1(c2ccccc2Cl)CC1)=O)OC CC1=C(C(=O)NC(Cn2cncn2)C(=O)N(C)CCN2CCCCC2)SCCO1 CC1(C)CCN(C(c2cccc3c2COC3)=O)CC1NC(=O)CC1=CCCCC1 C1(NC(=O)CCc2cccc(Cl)c2)CC(F)CN(C(c2nn[nH]c2Cl)=O)C1 C1(NC(C(CN(CC)CC)F)=O)CCN(C(C2CC(C)=NO2)=O)C1(C)C c1(C(N2CC(CC(CNC(C(CC)C)=O)(C)C)C2)=O)cc2cccc(N)c2cn1 c1(OC)ccc(C=CC(=O)NC2(CNC(C3CC(C)OC3=O)=O)CC2)cc1Cl N1(C(Cc2c(C)n[nH]c2C)=O)CC2(CCCCN(C(C3(C)COCCO3)=O)C2)C1 CCCCCCC(C)(CC)C(=O)N1CCCC(NC(=O)C(C(C)C)NC(N)=O)C1 N1(C(C=CCN(C)CC)=O)CCCC(NC(=O)Cc2c[nH]nc2O)CC1 C=CC(C)(CCOC)C(=O)N1CCCC(C(=O)NOC(C)C(=O)OC)C1 N1(C(C2CCC(CCC)CC2)=O)CCCC(CO)(CNC(C2CCN2CC)=O)C1 C1(C#N)(CCC(N2CC(CCNC(=O)OC(C)(C)C)C2)=O)CCC1 CCCCCC(=O)N1CC(COC)CC1CNC(C1CC1C(F)F)=O C1(NCCc2nnc(C3CN(C(=O)OC(C)(C)C)C3)o2)Cc2ccccc2CO1 CC1CN(C(C2CCSCC2)=O)CC(C(=O)NCC2(C)COCCO2)O1 C1(C(=O)NC(CCNC(c2c(C)nc(O)cc2)=O)C(C)C)CC12CCCCCC2 C(C)(CCC(=O)NCCC1(CNC(c2ccc(N)cc2)=O)CC1)OC C1(c2nn[nH]n2)(NC(=O)NCC(C(=O)O)C2CCCC2)CCC(F)(F)CC1 C=CCCCCCC(=O)NCC(c1ccccc1)NC(=O)C=CC1CC1 c1(C(N2C(CNC(C(C=C)O)=O)CC(OC)C2)=O)cccc(F)c1Cl CC1C2CCCCC2CN1C(C1CCN(C(=O)CN2CC3CC3C2)C1(C)C)=O C1(CC(N2CCCC(CF)C2)=O)C2CCC(C2)N1C(=O)CNc1ncccn1 Nc1c(O)ccc(Cl)c1C(N1CC2C(CNC(C3CCCN3C=O)=O)C2C1)=O Cc1cc(C(N2CCC2CNC(c2ccn(C3CCOCC3)n2)=O)=O)n(C)n1 C1(C(=O)NCCC(C)NC(=O)C(C2CCS(=O)(=O)CC2)(C)C)C(F)(F)C12CCC2 n1(CC)cc(C(=O)N(C)CC2CCCN2C(C2CC2CF)=O)cn1 CN=c1ccc(C(N2CCCC(CNC(=O)C=C3CCC(C)C3)CC2)=O)c[nH]1 CC1CN(C(C2CC23CCCC3)=O)CC(C(F)(F)F)O1 N1(C(c2cc(CC)no2)=O)CC(NC(C2Cc3nccn3C2)=O)CC(F)C1 C1(NC(C2(C(N)=O)CCC2)=O)CC2CC(C1)N(C(c1cccc(N)c1F)=O)C2 CC1CN(C(c2nc(Cl)cs2)=O)CCC1CNC(c1ccc(CO)c(F)c1)=O N1(C(CN(C)CC)=O)CC=C(C(=O)N2CC(CC(C)(C)C)C2)C1 n1(C(C)C)nccc1C(N1CCC(CN(C(=O)C(O)CC2CCCCC2)C)C1)=O c1(C(N2C(C(=O)NC(C)CSC)CC(=C)C2)=O)c(Cl)ccc(Br)c1Cl Cc1nc(COC(c2ccc(C(F)F)cc2)=O)nc2ccccc12 CCC(C)(C)CCCC(=O)NCC1CCCC1NC(c1nc(Cl)oc1C)=O C(C1CCOC1)=CC(=O)NCC(C)CN(C(=O)C=CSc1ccccc1)C c1(C(=O)O)cccnc1S(=O)(=O)c1n[nH]c(-c2ccc(NC3CCC3)cc2)n1 c1(C(=O)NC2(CNC(c3c(C)c(Br)no3)=O)CCC2)ccc2nnc(C)n2c1 N1(C(=O)CCC2CC2(Cl)Cl)CCC2C(NC(C34CCCN3CCC4)=O)CC12 c1(CC)ccc2[nH]c(C(=O)OCC(C3CCC4(CC4)C3)=O)c(C)c2c1 C1(C(=O)NC(CC)CN(C(=O)CC2CCC2)C)CCC(=O)N(c2ccccc2)C1 c1(OC)cc(N2CCCC2)ccc1C(=O)NCc1ncoc1C1CN(C(=O)CO)C1 C(=O)(C#CC1CCCCO1)NCC1(CCNC(CN2CCN(C)C(=O)C2)=O)CC1 c1(C(N2C(CNC(c3cc(C#N)c[nH]3)=O)CCC(C)C2)=O)ccc2cc[nH]c2c1 N1(C(C(CCSC)O)=O)CC(C2CN(C(C3COC4(CCC4)C3)=O)C2)C1 C1(C)(NC(CC(CC)OC)=O)CCCCC1C(=O)NC1CCCC1C#N C1(C2CN(C(=O)C(F)CC(C)C)C2)(NC(c2c(C)nsc2)=O)CC1 C(=O)(C1=CCOC1)NC(CC=C)CNC(C1CCC(CCCCC)O1)=O C1(CNC(CCc2cc(C)[nH]n2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C N1(C(C(CCNC(C(CC)COC)=O)O)=O)CCc2ncsc2C1 CC(CCc1cn[nH]c1)N=c1nc(N(C)CCC2CC2)c2ccccc2[nH]1 C1(C(=O)NC2(C(N(OC)C)=O)CC2)CC(N=[N+]=[N-])CN1C(c1cc[nH]c1C)=O CC1CCN(C(c2ccc[nH]2)=O)C(CNC(c2cc(Cl)ccc2Cl)=O)C1 c1(C(N(C2CN(C(C3CCCC3(F)F)=O)CC23CC3)C)=O)cc2ccccn2c1 O(NC(=O)C1CC(C(=O)NCC(CO)NC(C)=O)C1)CCOC C1(NC(c2c(CC)c[nH]n2)=O)Cc2ccccc2C1NC(C1CCCCC1F)=O C=C(C)CCC(C)NC(=O)CCC1CCC(NC(=O)C(C)N(CC)CC)C1 C=Cn1nccc1C(=O)N(C)CC1CCCN1C(C1(OC)CCCOC1)=O CC1(C(=O)NCC2CN(C(=O)CCNC(=O)CO)CC2C(F)(F)F)CC(C#N)C1 C1(C(=O)NCC2(O)CCN(C(=O)CSCc3ccncc3)C2)CC2CC1C1CC21 N1(C(COCCCC)=O)CCC(C2CC2)C1CNC(=O)C(C(C)C)n1cnnc1 c1(N2C(=O)CC(C(=O)N(CC(F)F)CCc3ccccc3)C2)cc(F)cc(F)c1 n1(CCOC)nc(C(=O)NCC2(C)CN(C(=O)COC(C)=O)CCO2)ccc1=O CC(CC1CCC1)C(=O)NCC(C1CC1)NC(=O)C(F)=CCCF N1(C(CNS(NC)(=O)=O)=O)CCC(NC(=O)Cc2cncnc2O)C12CCC2 c1(C(=O)NCC2CC(CNC(CCC(=O)NCC)=O)C2(C)C)cc(C)nc(C)c1 Cc1c[nH]c(C(=O)NC2COCC2NC(=O)CCC2CCN(C)C2)c1 CCC(CCC(=O)NC(c1nccs1)C)NC(c1ncncc1Cl)=O c1(C(=O)NCC(C2CC2)NC(C(COC)O)=O)cc(NC2CCCC2)ncc1Cl c1(C(C(N2CCC(NC(c3cn(CCC=C)nn3)=O)C2)=O)OC)ccccc1F CC1(CNC(=O)Cn2nnc(C3CC3)n2)COCCN(C(C23CCC(C2)C3)=O)C1 CCCCC(F)(F)C(=O)N1CC=C(C(=O)N(CC(O)CCC)C)C1 OC1CCc2ccccc2C1Nc1cc(N2CCC(F)(CO)C2)ncn1 C12(C(=O)NC(CC=C)(C)C)CCC(CC1)N(C(=O)C(O)C(C(C)C)OC)C2 c1(C(N(C2CCC(NC(C3(F)CC=CC3)=O)C2)C)=O)ccc2ccccc2c1O C(C(CNC(=O)Cn1cc(CN(C)C)nn1)C(F)(F)F)NC(CCC=C)=O c1(C(N2CCC(n3cc(CNC(CSC)=O)nn3)C2)=O)cc(C)ncc1Cl C1(C(C)CNC(=O)C=CCO)CCN(C(=O)C(c2ccc(Cl)cc2)(F)F)CC1 C1(NC(C=C=C(C)C)=O)C(CNC(=O)C(C2CCOCC2)C)CCC12CCC2 C1(C)(CC(=O)N(C2CCC2)C(C)C)CCN(C(=O)Cn2ncnn2)C1 CC1CN(C(=O)CCC2CC2)CC1CCNC(c1nncs1)=O C1(C2(O)CCN(C)CC2)(C(N2C(CN(C(C(F)=C(C)C)=O)C)CCCC2)=O)CC1 c1(COC)nc(C)c(C(=O)NC(CNC(C2CC(Cl)(Cl)C2)=O)C2CC2)s1 N1(C(C(C)(C)N(C)C(=O)OC2CCC2)=O)CC2(C1)CN(C(=O)OC(C)(C)C)C2 c1(C(=O)NCC(CCCC)NC(c2nc(C)ccc2F)=O)ccc2nn[nH]c2c1 O=S(=O)(c1cccnc1NC(C1CCCC1)CO)NCCn1cnnn1 c1(C(N2CC(NC(C(c3ccc(Cl)cc3)C)=O)C2)=O)cnn(C)c1F C#CCC(C(=O)N1CCCC(CCC(=O)NCC(F)Cl)C1)C1CC1 N1(C(C2CN(CCC)C(=O)C2)=O)CC2(CCN(C(=O)CS(N)(=O)=O)C2)C1 CC(C)C(CC1CCCC1)C(=O)Nc1ccc(Cn2cc(Cl)cn2)cc1 n1(CCC(=O)N(CCC)CCNC(C2(COCC)CC2)=O)c(C)csc1=O C(=O)(CCC(C)(C)O)N1CCC(c2ccccc2)(NC(C(C)CO)=O)C1 C1(C)(CC(=O)NCc2cc(C(=O)NCC(C)(C)OCCO)sc2)CCC(=O)N1 O=C(O)C1c2ccccc2CCN1Cc1cnn(CC2CCC2)c1 CC1CN(C(=O)Cc2cccnc2)CCC1NC(C1(F)CCOC1C)=O Cc1coc(CNC(=O)C(C2CCC2)NC(=O)OC(C)(C)C)c1 C1(C(N2CCC(CNC(C=C(C)C3CC3)=O)CC2)=O)OCC2COCCC12 C1(CNC(c2cnc(CC)[nH]2)=O)CCC(NC(=O)Cc2cnc(C3CC3)[nH]2)CC1 C1(CNC(N2CC(O)(CCC)C2)=O)CC1C1CCCC1 CC(C(=O)NCCN(C(=O)Cn1nnnc1-c1ccccc1)C1CC1)C(C)(F)F C1(CNC(C=CSC)=O)CCN(C(c2ncc(Cl)n2C)=O)CC1C C1(C(N(C(CC)CNC(=O)C=CC2CCC2)C)=O)CCC(=O)N1C C1(CNC(=O)C(c2ccccc2)F)CCCC(C(=O)NCCCF)C1 N(C1CCc2cc(CNC(C3CC(F)C3)=O)ccc21)C(=O)C(O)C(F)(F)F c1(C(=O)NCC(C)NC(C(=O)Nc2cc(C)ncn2)=O)cc(N(C)C)ccc1F c1(SC(c2cccc(C#N)c2)C)ccc(S(=O)(=O)N2CCOCC2)s1 Cc1ccc(C(=O)Nc2ccc(O)cc2C)c(-n2cc(CC3CCCC3)nn2)c1 C1(NC(C2(c3ccccc3)ON=C(C)C2)=O)CCCC(O)CC1 c1(C(=O)NC2CC(C(F)F)(NC(CC3CC(=O)OC3)=O)C2)n[nH]c2ccccc12 O=C(NN1CCc2ccccc2C1=O)C1CCCN(c2cnc(C3CC3)cn2)C1 n1(CC)cnc2c(N3CC(OC)C(F)C3)nc(=NCCCC#N)[nH]c12 N1(C(c2coc3c2CCCC3)=O)CCCC1C1CCCN1C(c1cc[nH]c1)=O C(Cc1cnc[nH]1)(C(=O)NCC1CCCSC1)NC(C1CC(=C2CC2)C1)=O CCC(CN(C)C)CC(=O)NCCN1CCCN(C(c2nocc2C)=O)CC1 CCC(C)C(CC(=O)NCC1CC12CCCCC2)NC(c1cc(C)oc1C)=O c1(SCC2N(C(=O)OCC)CCC2)ccnc(N2CCOC(C)C2)c1 c1(CC(=O)NCCN(C(c2c(C)cc(F)s2)=O)C)ccc(Br)cc1F c1(C(=O)NC2C(C)N(C(c3ccsn3)=O)CCC2)cc2c(=O)[nH]ccn2n1 C(=O)(C(C)CCC(C)(C)C)NC1(CNC(C=CCCC)=O)CCOCC1 C1(NC(c2c(C(C)C)onc2)=O)CN(C(=O)CN2CCN(C)CC2)CCC1C N1(C(c2c(SC)snn2)=O)CC(F)CC1CNC(c1cc(C)ncn1)=O C1(OC)CN(C(c2cc(Cl)cn2C)=O)CCC1NC(c1sccc1C1CC1)=O c1(C(=O)NC(C(C)NC(c2c(C#C)cnn2C)=O)C)cc(Cl)c([N+](=O)[O-])[nH]1 C(CN=c1[nH]c2cc(Cl)ccc2s1)C1CCN(C(c2c(C)nc(CC)o2)=O)CC1 N1(C(C)=O)CCC(Cn2cc(-c3cccc(OC)c3)nn2)C(CO)C1 c1(NCC2(O)CN(C(C(C)n3cncn3)=O)C2)ncnc2[nH]c3ccccc3c12 N1(C(Cc2nc(C)sc2)=O)CCCC2CN(C(C3(CO)CCCC3)=O)CCC12 c1(C(=O)OCC(=O)CCC2CCCC2)nnn(Cc2ccccc2)c1Cl c1(C(N(C2CC(NC(CC(=O)OCC)=O)C2)CC)=O)cc2cccnc2cn1 c1(C(=O)NC(C(C)C)C(C)NC(=O)C(C)(C)C(C)(F)F)cn2cc[nH]c(=O)c2n1 c1(C(=O)NCCC(C)N(C)C(C23CSCC2C3)=O)cnn2ccc(Cl)c(F)c12 CC(C)C(CN(C)C)C(=O)N(C(C)C(=O)N(C)CC1(O)CCOC1)C C1(C(=O)NC2CC(NC(C(C)CC3CC3)=O)C(O)C2)CC2(CCCC2)C1 n1(CCCC)nc(C)c(C(=O)NCC2CCCCC2Nc2cc(O)ncn2)c1Cl CCC(COC)C(=O)NCCC1CCCN1C(c1cc(CS(C)(=O)=O)c(C)s1)=O c1(C(=O)NCC2(O)CN(C(=O)CC3CCCCC3)C2)cccn(C2CC2)c1=O C1(NC(=NCCOC)NCCOCCOCC(C)C)CC2(CO1)CC(F)(F)C2 N1(C(Cc2c(C)scc2)=O)CCN(C(C2(CO)CC2(F)F)=O)CC2(CC2)C1 C1(c2nnnn2CCCC2CC2)(NC(CC)CC)CCCC(C(C)C)C1 C1(CC)CN(C(C2Cc3cscc3C2)=O)CCC1NC(C1OCCN(C)C1=O)=O N1(C(=O)N(C2CCC(C)CC2)CC2CC2)CC2CCC(C1)C2N1CCCC1 C1(CNC(C2(C)CCC2)=O)CN(C(=O)COCCc2cccc(F)c2)CCCO1 c1(SC)cc(=NC(=O)C2CC(C)CCN2C(c2ccn(C)c(=O)c2)=O)[nH]n1C c1(C(=O)NCc2ccc(C(=O)NCC(CO)OC)cc2)ccn2ncc(C)c2n1 CCCC(CNC(C1(C)CC(O)CN1C(=O)Cc1nocc1C)=O)CCC C12(CNC(=O)CN3CCOC3=O)CCC1CCN2C(c1ccc(CO)cc1)=O c1(CNC(c2cnn(CC3CCC3)c2)=O)occc1C(=O)O.C12CCCC1NC2 Cc1cc(NC2(N(C)C)CC2)ncc1S(=O)(=O)N(C(C)C(C)S(C)(=O)=O)C N1(C(C(C(C)C)CN(C)C)=O)CCOC2(C1)CN(C(=O)CC1CCC(C)(C)C1)C2 c1(CC2(C(=O)NCC(C)(F)CNC(=O)Cc3cncs3)CC2)ccc(O)cc1 Cc1cc(S(=O)(=O)N2CCCC(CN(c3ccc(O)nc3)C)C2)c(F)cc1Cl c1(-c2cccc(CC(=O)NCC3CCS(=O)(=O)C3)n2)c[nH]c2ncccc12 N1(C(C(CC)F)=O)CCC(NC(c2cc(C)n(C)n2)=O)C(O)C1 c1(NC(C2N(C(C3(C(=O)OCC)C(C#C)C3)=O)C3C(C2)C3)=O)ncc(Cl)cc1F c1(C(=O)NC2(CO)CCN(C(=O)CCCCC3CC3)C2)cnc2ccnn2c1 c1(CC(=O)N(C2CC3(CNC3)C2)C(C)Cc2ccccn2)c(Cl)cccc1Cl N1(C(C2N(C(C)=O)CCC2)=O)C2CCC1CC(N(C)C(C1CCS1(=O)=O)=O)C2 c1(OC(C)C(=O)NCC2COCC2NC(=O)Cc2csc(Cl)c2)ccccn1 CC1C2CCC(C2)C1C(=O)NCCC1(C(=O)N(C)CC2CC(O)C2)CCCC1 CC(C)(CCC#N)C(=O)N1C2CCC1CN(C(=O)CC1CNC(=O)C1)C2 n1(CCOC)c(N2CCCC(C(F)(F)F)C2)nnc1C(C)(C)C#N C1(C(N)=O)CCC(C(=O)NCCOCCNC(=O)Cn2nnc(=O)[nH]2)CC1 CC1(C)C(=O)NCC1NC(=O)CC=CCNC(c1ccsn1)=O Cc1nn[nH]c1CNC(C1COCC1NC(=O)C=CC(C)(C)C)=O C#CCC(C)(C(=O)N(C)CCC1CN(C)C1)NC(C1CC2OC1C1CC21)=O CCC(C)(C)C(O)C(=O)NCCC1(OC)CN(C(=O)C(c2cccc(C)c2)C)C1 C1(C(=O)NCC(C)(C2CC2)OCCOCC)CCC(C(=O)OC)CC1.C1C(=O)N1 N1(NC(=O)NCc2onc(N(C)C)n2)CCC=Cc2ccc(Cl)cc21 S(=O)(=O)(C1CC1C)N(C(=O)C(C)Oc1ccccc1)CCCC N1(C(C2CC3CCC2O3)C(=O)NCc2c(OC)cccc2)CCC2(CC1)CC2 C1(CC(=O)N(C)CC2(OCC)CCC2)CCCN(C(c2n[nH]cc2CC)=O)C1 c1(C(=O)NCC2(F)CN(C(c3cnc(C(F)(F)F)nc3)=O)C2)c[nH]nc1[N+](=O)[O-] CC(C)C(C)(C)C(=O)NCC(C)CNC(c1cnn(C)c1F)=O C1(C(=O)NCCCCNC(Cc2n(C)ccn2)=O)CCN2CCC1C2 C1(C2CN(C(c3ncsc3C(C)C)=O)C2)(NC(c2n(CCC)ccc2)=O)CC1 C1(C(=O)NCC2CCCCN(C(C(N)=O)=O)C2)CCn2cnnc2C1 C1(NC(c2c(OC)scc2)=O)CCCN(C(=O)CC2(n3cccn3)CCC2)CC1 C1(NC(c2cnc(OC)nc2)=O)CC(F)(F)CC1NC(=O)CCC(C)OC N1(C(c2n(C)ccn2)=O)CCCC(NC(=O)C(O)CCCc2ccccc2)CC1 c1(C(N2CCCC(NC(C3=C(C)CC3)=O)CC2)=O)cc([N+](=O)[O-])oc1C c1(CC)cc(O)ccc1NC(C12CC(CO1)N(C(c1cccn1C)=O)C2)=O CC1SCCN(S(=O)(=O)Cc2ccc(C3CC3)cc2)C1C CCCCC(O)CC(=O)NC1CC(C)(C(N2CC(c3nn[nH]n3)C2)=O)C1 c1(COC)nc(C(=O)NC(CO)C(C)NC(=O)C(F)OC)cs1 C1(C)(CC2CCN(CC(=O)NCCOc3ccc(C)cc3)CC2)CCC(O)CC1 c1(C(N(C(C)CCNC(C2CCC3CC3C2)=O)C)=O)ncc(Cl)nc1Cl N1(C(c2cnncc2O)=O)CCN(C(=O)Cc2cc(F)ccc2F)C(CF)C1 C1(C(=O)NC(C(=O)N(C)C)CO)(CF)CCN(C(=O)C=Cc2cnn(C)c2)C1 c1(NC(C2C(C(N(C)CC)=O)CC2)=O)ccc(CC(C)NC(=O)C=CCO)cc1 c1(CC(N2CCCC2CC2CCCCC2)=O)ccc(Br)s1 C(=O)(CCCCCCCNCCC1(CNC(C2(CC#C)CC2)=O)CC1)C1CC1 n1(-c2c(C)noc2)nc(-c2ccc(Cl)cn2)nc1C(C(C)C)C(F)F c1(OC)cc(OC)cc(C(N2CCOC(CF)C2)C(=O)NCC2CCOCC2)c1 C1(C(=O)NCC#CCC)CCCN(C(=O)C(=O)NOC)C1 C1(C(=O)NCCCCC=C)CCC2(CC2)N1C(C1CCCC1OC)=O N12CC(OC(C)(C)C1)CCn1cc(nn1)C2=O.c1(CC(=O)OCC)csc(C)n1 n1(CCC(=O)N(CCCN(CC(=O)N(C(C)C)C(C)C)C)C)cc(Cl)cn1 CC1(C)Cc2cccc(C(N3CC4(NC(C5CC(F)C5)=O)CC3C4)=O)c2O1 N1(C(CCC)=O)CCC(c2cccc(F)c2)C(NC(=O)Cc2ccsn2)C1 Cc1nc(C(C)(F)F)ccc1C(=O)NCC1(C)CCCN1C(C1CCCCO1)=O C=CCCCCCCC(=O)NCC(=O)NCCCc1ncco1 CCCCC(O)CC(=O)NC(C1(O)CN(C(=O)CSc2ccc(C)cc2C)C1)C Cc1cc(C)c(C(N2CCC(N(C(=O)C=CC(=O)N(C)C)CCO)C2)=O)s1 C1(C(NOCCOC(C)C)=O)C2CN(C(=O)CC3CC=CCN3C)CC12 N1(C(C(CCC)O)=O)CCC(C2(CNC(C3(O)COC3)=O)CCOCC2)CC1 CCCCC(C)CCC(=O)N(CCCNC(C1CN(C)CC(C)O1)=O)C CC1CCCN(C(=O)C=CCN2CCOCC2)C1CNC(=O)COCP(C)(C)=O C=C(Cl)CCC(=O)N1CC(CC(N2CC(CC)C(O)C2)=O)C(C)C1 N1(C(C(=O)NC(CCC(=O)OC)C)=O)CCC(S(=O)(=O)N(C)C)C1 C1(NC(C(COC)(C)C)=O)CN(C(c2ccnc(C(F)F)c2)=O)CCC1C c1(-c2cn(CCOCCNC(=O)CC3CC4CCC3C4)nn2)ccc2c(c1)CC2 C1(CC)CN(C(c2ccc(C)cc2Br)C(=O)NCC2CC2)CC(C)O1 C1(N(C(=O)CCSc2nccn2C)CC)CCCN(C(c2cnc(O)o2)=O)CC1 N1(C(c2ccc(NC(C)=O)cc2)=O)CCC(NC(c2nnccc2C)=O)C(C)C1 O=C1CC(C(=O)NCCOC2CN(C(c3cnccn3)=O)C2)c2cccnc2N1 C(C)(C)(CC(=O)NC1CN(C(C2CC(=O)N(Cc3ccccc3Cl)C2)=O)C1)OC N1(CC(=O)NCC=C)CC2(CN(C(=O)CC3CCCCO3)CCO2)C1 C1(N(c2nccc(N3CCCC(c4nnc(C)o4)C3)n2)C)Cc2ccccc2C1 c1(OC)cccc(C(=O)N(CC(CO)(CO)NC(c2ccncn2)=O)C)c1 n1(CC(=O)NC(CC=C)CNC(C2(CF)CCOCC2)=O)ccc(C)cc1=O C1(C(N2CCC(N(C(=O)C3=CCSC3)CCO)CC2)=O)CCCNS1(=O)=O c1(C(=O)NCC(N(C(=O)CC2C=CCC2)C)C2CC2)cn(C2CCCC2)nn1 c1(C(=O)NC2CCC(C(=O)NCCCO)OC2)cc(Br)cc(Br)c1 C1(CC(=O)N(C)CC2CCCCN2C(c2cnnn2C)=O)CC2(CCC2)CO1 C12(NC(C(CCCC)NC(C3CSCC(=O)N3)=O)=O)CC3CC(CC1C3)C2 C1(C(N2CCCC(C3(C)N=N3)C2)=O)C(C2CC2)CCN1C(=O)CCc1cnoc1 C(=O)(C(S(C)(=O)=O)C1CC1)NCCN(C(C)C)C(c1coc(C(C)(C)C)n1)=O Cc1c(Cl)ccnc1C(=O)NCC(O)CCNC(C1(C(C)C)CNC(=O)C1)=O CCC(CC(=O)N(C1CN(C(=O)C(F)(F)c2nccn2C)CC1(C)C)C)C(F)F C(C(C(=O)NCCc1nccs1)C(C)(C)C)NC(c1scc(C)c1)=O c1(CC(=O)NC(C(C)NC(CCCN(C(C)C)C)=O)C)cc(Cl)n(C)n1 c1(CCC)noc(CCC(=O)NCC2CCN(C(=O)C=Cc3cscn3)C2)n1 Cc1cc(C(=O)NC(C)Cn2cc(-c3ncc(C(=O)O)o3)nn2)on1 Cc1nc2cncc(C(N3CCCN(C(c4nc(O)sc4C)=O)C(C)C3)=O)c2[nH]1 N1(CC(=O)NC(c2ccccc2)C(=O)NCC2(C(=O)OC)CC2)CCOC1=O C1(CNC(C(C)P(C)(C)=O)=O)CC2(CO1)CN(C(=O)CCCCCF)C2 c1(C(N2C(C(C)NC(C3CCCCS3)=O)CCC2)=O)ccc(C(F)F)c(F)c1 CC1CCN(C(C2CC(F)(F)CCC2O)=O)CCN1CCC(=O)O N1(C(C)Sc2c(OCCOC)cccc2)C(=O)NC(CO)C1=O CC1CCCC=C1C(=O)NC1(C(=O)NC2CC(C(F)(F)F)C2)CCSC1 c1(CC(=O)NCCN(C(c2nccnc2C)=O)CC)ccc2nsnc2c1 C1(O)(CCNC(C(C#C)(C)C)=O)CCCN(C(=O)C(CCSC)NC(N)=O)C1 C1(C(=O)NCC(C2CCN(C(=O)Cn3cc(Cl)cn3)CC2)F)CCC2(CC1)CC2 c1(C(N2CC(O)(C(C)NC(=O)C(C3CCCCCC3)O)C2)=O)cc2n(c1)CCC2 Cc1nn(C)c(C)c1C(C)C(=O)NC1CCCC1NC(C1(C)CC1)=O c1(C(N2CCN(CCCNC(c3c(OC)ccs3)=O)CC2)=O)ncc(Cl)cc1Cl C1(N(C(=O)COC2CCOC2)C)CN(C(=O)C=C2CCCCC2(C)C)CC1(C)C c1(C(N2CCC(CN(C(=O)COC(C)(C)C)C)C2)=O)cnnc2ccccc12 n1(CC)cnc2c(NC3COC(C)(C)C3)nc(N3CCC(C(C)C)(CO)C3)nc12 c1(OC)ccc(CC(=O)N(CCCNC(=O)Cc2ccno2)C2CC2)cc1 Cc1cnc2ccc(C(=O)NC3CN(C(=O)CC(F)(F)F)C4CC34)cn12 CN1CC(C(=O)N(C2CCN(C(=O)CCCF)CC2)CCO)CCC1=O N1(C(c2nn(CC)c(O)c2)=O)CCCN(C(c2sccc2SC(F)F)=O)CC1C C(=O)(C1=CNC2=NCCC2=C1)N1CCC(CN(C)C(C2(C)CCCS2(=O)=O)=O)C1 N1(C(C(Cc2ccc(C)cc2)C)=O)CCN(C(=O)COc2ccsc2)C(C)C1 c1(NC(C2CN(C(C=CC)=O)CC2F)=O)ccc(Br)cc1OC(F)(F)F CCC(CC(=O)N1CCOC(CNC(C2CN(c3nnnn3C)C2)=O)C1)C(C)C C1(O)(C(C)NC(CC2(CSC)CC2)=O)CN(C(=O)C(N2CCOC2=O)C)C1 c1(C(N2CCC3CCC(C2)N3C(=O)C=C2CCCC2)=O)csc2c(O)ccnc12 C#CC(C)(C)C(=O)N1CC(CNC(c2c(C)ncn2O)=O)C(C)C1 C1(=O)CC(C)(C)C(=O)ONC(C2CCCCC2)CN1.C(CC(=O)OC)OCCC c1(C(=O)NCC2CN(C(c3c(COC)cc[nH]3)=O)CC2C)cc2ccncc2s1 N1(CCC(=O)NC(CC)CN(C(=O)C=C(C)C2CC2)CC)CCCCC1C N1(C(C(CC(C)C)OC)=O)C2CCC1CN(C(=O)Cc1cscn1)C2 c1(C(C)(C)CF)ncc(C(=O)NCC2CCN(C(c3nc(Br)c[nH]3)=O)C2)o1 Cc1ccc(C(=O)NC2(C)CC(NC(c3csc(S(C)(=O)=O)c3)=O)C2)cc1C#N C(CC)(CC(=O)NCC1(CO)CCC1)NC(C(C=C)O)=O C#Cc1ccc(CC(=O)NCCC2CSCCN2C(=O)C(O)C=C)cc1 N1(C(C(C)OCCN(C)C)=O)CCOC2(C1)CN(C(=O)C=CC1CCCO1)C2 N1(C(c2cc(OCC)ns2)=O)CC(NC(C2CC2[N+](=O)[O-])=O)CC(F)C1 C(CC(C)C)(C(=O)N1CCC(NC(=O)CCc2ccc(C(N)=O)cc2)C1C)OC c1(CC)noc(C)c1-c1cn(CC2CCCCC2O)nn1 C1(C(N2C(CC(=O)NC(c3c(C)noc3)(C)C)CCC2)=O)CCCC(=O)C1 C(C(F)(F)C(F)(F)F)OCCC(=O)NCC=CCNC(=O)CCc1ccccn1 c1(C(N(CCC)CCNC(C2(C)CCCCO2)=O)=O)cccc(C)c1C c1(C(c2n(CCCSC)nnn2)NCC(C)OCCO)ccc(S(N)(=O)=O)cc1Cl C(=O)(CC(CC(=O)O)C1CCCCC1)N1CC(c2ccn(CCOC)n2)C1 Cc1cc(C(N2CCC(C(=O)NC(c3ccccc3O)C)CC2)=O)sc1C O=C(C1=C2CCN=C2NC=C1)NC1CN(C(c2ccncn2)=O)CCC1CO c1(C(=O)NCC(CC)NC(c2cccc(N3CCCCC3)c2)=O)cn(C)[nH]c1=N c1(C(N2CC(N(CCC)C(C3CC3C(F)F)=O)C2)=O)ccccc1N=S(C)(C)=O C(=O)(C(CC(C)C)ONC(c1ccc(O)c(F)c1)=O)N(C(C)C(C)C)CC N(C1c2ccccc2CC1NC(c1cc(O)nc(O)c1)=O)C(C(C)(CO)CO)=O N1(C(C2CC(=O)NCC2)=O)CCC2(CO)CN(C(c3cnc[nH]3)=O)CC2C1 C=CCC(F)(F)C(=O)NCCOCCOCCCNC(C1CCCC1(F)F)=O C(=O)(C(C)(C)C(=O)N(C)C)NCC1(CNC(C2(OC(C)=O)CC2)=O)CC1(F)F CC(C)C(CCN(C)C(c1c[nH]cc(F)c1=O)=O)N=c1[nH]c2ccc(Cl)cc2s1 N1(C(C2CC(C#C)(O)C2)=O)C2CCC(C2)C1CNC(=O)CC(C)F N1(C(=O)C)Cc2ccccc2C1.C1(NC(C(F)=CCC)=O)CCNC(C2CC2)C1 c1(NC(=O)CNCC2(c3nn[nH]n3)CC2)cccc(F)n1 C(=O)(C(CNC(=O)C(=O)NCC(F)F)C(C)(C)C)N1CC(CC)SCC1 c1(C(=O)NCC2C=CCN2C(c2c(O)cccc2Cl)=O)nnc(O)cc1O CCCC(C)CC(=O)NC1CCCC(NC(=O)CSC(C)C)C1 c1(C(N2CCC(c3c(C)cccn3)C2)=O)n[nH]c2ccc(C(F)(F)F)cc12 c1(C(N(C)CC2CCN(c3nccc(C)n3)C2)=O)cc(=O)c2cc(F)ccc2o1 N1(C(C(=O)NCC(CC)(N)CC)=O)CC2CCC1CC2 c1(CN(C(=O)CCCN2CCCC2)C)ccc(CNC(C2(C)CCCC2)=O)cc1 C1(NC(CS(=O)(=O)N(CC)CC)=O)CC12CCN(C(C1CCCS1)=O)C2 C(=O)(C1CCCn2nccc21)N(CCNC(c1c(C)nn(C(C)C)c1)=O)C(C)C CC(C)C(C)C(C)CC(=O)NC1(CNC(=O)C#CC2(C)CCCO2)CCCC1 N1(C(C(CCCC)O)=O)CC2CCN(c3cc(C(F)(F)F)nc(C)n3)C2C1 c1(C(=O)NC2CC(NC(C3(OC)CCCC3)=O)C2)cc(Cl)ccc1C(F)(F)F c1(C(N2CC3CN(C(=O)C(F)F)CC3C2)=O)cnc2ccc(Br)cc2c1 Cc1cccnc1CCC(=O)Nc1nc(C2CCCC(C)C2)cs1 C1(N(C(=O)CCC2CC2(Cl)Cl)C)CC2CC1N(C(C1(CO)CCCC1)=O)C2 CC(=O)CCCCC(=O)N1CCCC1C(=O)NCC1CCS(=O)(=O)C1 N1(C(c2cccc(NC)n2)=O)CC(CNC(c2nc(C)c(C)s2)=O)CC(C)C1 N1(C(c2c(CC)nn[nH]2)=O)CC(NC(=O)Cc2csc(=N)[nH]2)C(C(F)F)C1 C1(OC)CN(C(=O)CCOCC(C)C)CC1NC(c1ccc(N)cn1)=O c1(C(=O)NC(c2cnn(-c3ccccc3)c2)CC)ccccc1OC N1(C(=O)OC(C)(C)C)CCC2(CCC(C(=O)OCc3nsc(CO)n3)OC2)CC1 c1(C(N2CC(CC(=O)NCc3ccccn3)C2)=O)cnnc2ccccc12 C(C1c2ccsc2CCN1C(=O)C(O)C1CC1)NC(CN(CCOC)C)=O N1(C(c2c(CNC(C(C)=C3CCCC3)=O)nccc2)=O)CCC2(C1)CC2(F)F CCC(C(=O)N(C)CCN(C)C(c1ccc(OC)c(N)c1F)=O)C(F)(F)F N1(C(=O)C(Cl)Cl)CC2(CO)CC1(C(N1CC(c3ncccn3)C1)=O)C2 S(=O)(=O)(c1ccc(=NCCCC(F)F)[nH]c1)NC1C(CC)CCCC1 CC(C)[Si](CC(C)(C)C)(CC(=O)N(S(C)(=O)=O)C)C(O)C(F)(F)F C=CC1(C(=O)NCC2(F)CCN(C(=O)C(C)N3CC(C)C3)C2)CCOCC1 C#CCCC(O)C(=O)N1CCC(NC(c2cnc(OCC(F)(F)F)c(Cl)c2)=O)C1 C1(NC(C2(OCC)CCC2)=O)CCCCCC1C(N1CCOCC1CO)=O c1(C(=O)NC2C(CO)CCN(C(c3ccc(CC)o3)=O)C2)cccc2ncnn12 C1(C)(NC(C(C(C)C)c2ccc(F)cc2)=O)CCCN(C(c2nncn2C)=O)C1 CCCC(C(O)C(=O)N=c1ccn(CC2CC2)[nH]1)NC(=O)C(CC1CC1)CC N1(C(c2cc(OCC)ncc2)=O)CCN(C(C2CCCOC2)=O)CC1C CCC(O)(CC)CC.c1(C(=O)N2C3CCC(C3)CC2=O)occ2c1CCC2 C1(CCC)CN(C(c2conc2C)=O)CC1C(=O)N(CCC(C)(C)C)C c1(CC(=O)NCC(CCCC)NC(C2CC2C(N)=O)=O)cc(C)ccc1O C1(C(=O)NCC2CN(C(C(C=C=C)C)=O)CC2C)(OC)Cc2ccccc2C1 C=C=CCCC(=O)N(C1(CC(=O)N(CC)CC2CCCC2O)CC1)C CCC(CC(=O)NC1(CN(C)C(C2CC(n3cnnc3)C2)=O)CC1)C(C)C CCCC(C(=O)N1CCC(N(C)C(c2ccc3c(c2)OCCN3)=O)C1)S(N)(=O)=O c1(C(N2CC(NC(C3C(C)C3)=O)C2)=O)nccc2cc[nH]c12 N1(C(c2ccc(C)cn2)=O)CCC2(CO)CN(C(=O)CCNC3CC3)CC2C1 CCC(C)(F)C(=O)NCCC1COCCN1C(=O)CCCOc1ccc(C)cc1 c1(C(C(N2CC(CNC(C3(CC=C)CC3)=O)C(O)C2)=O)O)cccc([N+](=O)[O-])c1 N1(C(C2CN(C)C2)=O)CCCC2(CCC2NC(=O)CS(C)(=O)=O)C1 c1(C(=O)N(CC2(F)CNC2)CC2(F)CCC2)ncnn2cccc12 Cc1ccnc(C(=O)NCCC2CCCN(C(=O)C(c3cccnc3)C)C2)c1N C1(C(=O)NCCCN(C(=O)C=C2CCOCC2)C2CC2)CCC2C(CC1)C2(F)F C1(C(=O)NCCC2(O)CCN(C(CC(C)=C(C)C)=O)C2)Cc2nccn2C1 C1(CNC(CC2(CN)CCC2)=O)CCC(OCC)CC1.C(=O)(CSC)NC(C)C c1(C(=O)NC23C(CN(C(CSCC(C)C)=O)C2)C3)ccc2c(c1)NC(=O)C2=O CC(Cl)(Cl)C(=O)NCC1CC(CNC(c2cnn(CCF)c2)=O)CO1 C(=O)(C1CC(=O)Nc2ncccc21)NC(CN(C(CC=CC=C)=O)C)(CO)CO Cc1nn(CC(=O)NC(CCNC(=O)C(C)CF)C(C)C)cc1Cl C1(NC(C(CSC)O)=O)CCN(CCNC(C2(F)CC2)=O)CC1 N1(C(COc2cn(C)nc2)=O)CCCCC(NC(=O)C=CC2CC2)C1 C(=O)(CC(O)CC(C)(C)C)N1CCC(CC=C)(NC(c2ncccc2Cl)=O)C1 N1(C(C(C)SCC)=O)CCc2sccc2C1CNC(c1cccc(CO)c1)=O c1(NC(C2CSC2)C)ncc(S(=O)(=O)N2CCCC(OCCO)C2)cc1Cl N1(C(CCCC(=O)OC)=O)CCN(C(c2ccc(F)cc2)=O)C(C)CC1C Cc1cc(C)c(C(=O)NCC23CC(CN2C(=O)CCC(=O)OC(C)(C)C)C3)[nH]1 c1(C(C)N(C)C(=O)NCC(O)Cc2cnsc2)ccccc1 C1(N(C(C2C(=C)CC2)=O)C)C2CN(C(=O)CCc3nnc(COC)o3)CC12 c1(C(=O)OCc2c(C)ccc(F)c2)c[nH]c2cc(F)c(F)cc2c1=O c1(OC)ccc(O)c(COC(C2CNCC2C(F)(F)F)=O)c1 c1(OCC(=O)NCC(C)(C)C(=O)N2CCCC(C(=O)O)C2)ccc(Cl)cc1CO C1(C(N2CCN(C(CN(C(C(CC)CC)=O)C)=O)CC2)=O)CS(=O)(=O)CC12CC2 C1(F)(CNC(CC(=C=C)C)=O)CC2CCC(C1)N2C(c1ccc(OC)nc1C)=O c1(C(N2C(CNC(Cc3c(C)scc3)=O)CCCC2)=O)cc(O)cc(F)c1 C(=O)(CCCC(C)(C)C#N)NCC1(C(N(CCOC)CCF)=O)CC12CCC2 Cc1c(Br)c(C(=O)NCC2C3CC2N(C(C2(F)CC=CC2)=O)C3)nn1C C(C)(CCP(C)(C)=O)(c1nnnn1CC(F)F)NCc1c(OC)cccc1Br N1(C(C(CC(C)C)NC(C)=O)=O)CC(C2CN(C(=O)Cc3ccns3)C2)C1 CCC(C)(C)C(=O)N1CCOC(CN(C(=O)CCSc2nccn2C)C)C1 C(C)(CCN=c1[nH]ccc(C#N)c1[N+](=O)[O-])NC(COc1c(C)cccc1)=O C(C(=O)NCC(C1CCCN1C(=O)COc1cnn(C)c1)(C)C)(C(C)(C)C)SC c1(OC)cc2c(cc1F)CCC2NC(=O)Nc1cccc(SC(C)C(=O)NC)c1 c1(OC)c(C(=O)NC2CN(C(=O)C=CC3CC3)CC2C)ccnc1Cl N(C1COc2ccccc21)C(c1cc(CNC(CC(C)N(C)C)=O)ncc1)=O c1(C(=O)NCCC2(O)CN(C(C(CCC#C)O)=O)C2)ccc(N)c2ccncc12 C1(C(N2C(CCC(=O)NC(CCSC)(C)C)CCC2)=O)C(C)(C)C1(F)F C1(C(=O)NC(c2n(C)ncc2)CO)CC12CCN(CC=CC1CCCCC1)CC2 c1(C(=O)NCC)cccc(NC(C2CCOC2C(N2CCN(C)CC2)=O)=O)c1 c1(NCC(C)OC)ncccc1S(=O)(=O)N1CCC(C(C)(C)C)C1 C(CC(C(=O)NCCSC(C)(C)C)NC(=O)CC1CNC(=O)O1)N(C)C c1(C(=O)OCC)cnc(O)c(C(N2CCCC2c2nc(C)co2)=O)c1 C1(N(C)Cc2c(C)nco2)CCN(C(=O)C(C)CSC(F)(F)F)CC1C c1(C(N2C(CCC)(Cc3ccccc3)CCC2)=O)cnc2c(c1)CCC(=O)N2 N1(C(CC(=O)NCC)=O)CC(O)CCC1C(N1CCC(C(C)C)CC1)=O c1(C(N(CCCNC(C2C(C)C2(F)F)=O)C)=O)n[nH]c2ccccc12 C1(NC(C(C)O)=O)CCC(C(=O)N(C(C2CCC2)=O)Cc2ccccc2F)CC1 C1(CNC(Cn2c(C(C)C)ncc2)=O)CC(NC(=O)Cc2ccon2)C1(C)C Cc1nc(Cl)sc1C(C(=O)NC1CCOC1)N(C(C)C)Cc1ncc[nH]1 N1(C(CCOC(C)C)=O)CC2(CNC(c3nc(Cl)sc3Cl)=O)CCC1CC2 CC1CCCN(C(C2CCCC23CC3)=O)C1CNC(=O)CCC(C)(F)F c1(CCNC(c2cnsn2)=O)ccc(CNC(C2CC3CC2C3)=O)cc1 CC1CN(C(c2ccc(SC(F)F)cc2)=O)CCN1C(=O)CC1COCCN1C c1(CC)ccc(C=CC(=O)NC2CCC2NC(c2occc2C)=O)cc1 C12(NC(C3CCCN(CCC)C3)=O)CCCC1N(C(C1CCOC1)=O)CC2 CC(C(O)C(=O)N(CC(C)(C)NC(c1ccc[nH]1)=O)C)c1ccccc1F C12(NC(C(CC)N(C(=O)C(C)(CC)C(N)=O)C)=O)CCC(CC1)C2(C)C Cn1cnn(CC(=O)NCCC2CN(C(c3cccc(Br)c3)=O)C2)c1=O c1(C(=O)NCCN(C(C2CC(OC)C2)=O)C(C)C)ccc(S(=O)C(C)C)cc1 CS(=O)c1ccccc1CC(=O)NC12CC1CN(C(=O)C(=C1CCCCC1)F)C2 CCCC(C)CCNC1(c2nnnn2C)CCN(c2ccccc2)C1 C(C(=O)N(C)CCNC(=O)CN(C)C(=O)OC(C)(C)C)OCCC CC(C)C(F)(F)CC(=O)NCCCCN(CCCNC(c1cnsn1)=O)C C1(CC(C)NC(c2[nH]cnc2C#N)=O)CCN(C(C2CC2C2CC2)=O)CC1 N1(C(CC2(C#N)CC2)=O)CCCC2(CC(NC(=O)C3=CCOC3)C2)C1 C(=O)(C1Cc2ccccc21)NC(CNC(c1c(C)nc(C(C)C)nc1O)=O)CO N1(C(Cc2c(C)nc(SC(F)F)s2)=O)CCC2(CC(C(=O)OC(C)(C)C)CO2)C1 c1(OC)cc(C#N)ccc1C(N1CCC2(NC(c3ccc[nH]3)=O)CCCC12)=O N1(C(C2CCN(C(=O)C3COCC(C)O3)O2)=O)Cc2cccc(C#N)c2C1 Cc1ccc(C(N2CCN(C(c3cn(C)ccc3=O)=O)C(CO)C2)=O)cc1Cl N1(C(c2c(OC)scc2)=O)Cc2n[nH]cc2C1C(=O)NC1COCCC1O N1(C(C(CC)(C)O)=O)CCC(C2CCN(C(C3CCC=CCCC3)=O)CC2)C1 c1(C(=O)NC2CCC(C)N(C(C3CC3F)=O)C2)cc(C#N)ccc1O N1(C(C=CC(C)C)=O)CCC(C)CC1C(N1CCC(CC(N)=O)C1)=O c1(CC)nn(C)c(Cl)c1C(=O)NCC1CCC1NC(C1CCC(=O)O1)=O N1(C(c2cc(C)sc2)=O)CCN(C)CC1CNC(C1CCC2CC12)=O N1(C(CC(C)C2CCCO2)=O)CCCC2CN(CC(N3CCNC(=O)C3)=O)CCC12 c1(CC(=O)OC)cccc(N(C(=O)C(N2CCNCC2)=O)C2CC2)c1 C1(C(=O)NCC2(C(N(CC)Cc3ncc[nH]3)=O)CC2)CCOC1(C)C C(C)(C(C)C(=O)NCC(N)=O)NC(c1cnc(OC)s1)=O c1(NCC(CNC(c2cnc(CC)[nH]2)=O)C)nc(C(C)CC)ccc1C#N c1(C(=O)NCC(C(C)C)NC(C2CCCC2(C)C)=O)cc2cccnc2[nH]1 C(=O)(C(C)(C)CC(=O)NCC1(CNC(=O)C(C)=C2CC2)CC1)OC N(C1c2ccccc2CC1O)C(C1C(C(N2CCC(OC)C2)=O)C1)=O c1(C(=O)NCC(CC)NC(c2ccc(COC)s2)=O)nc2ccccn2c1F C#CC1(NC(=O)CCCCCNC(C2CC2Cl)=O)CCCOC1 O=S1(=O)CCCCN1c1cccc(NC2CC3CCCC23)c1 C1(NC(c2c(C)snn2)=O)CCN(C(=O)Cc2cnns2)C1c1ccccc1 Cc1ccc(C(=O)NCCn2cc(CCN3CCN(C)C(CO)C3)nn2)cc1F c1(C(=O)NC2C(NC(C(CO)NC(N)=O)=O)CC2)ccc(Cl)c(S(C)(=O)=O)c1 CCC(C(=O)NC1(C)CCCCC1C(=O)NCc1nnn(C)c1C)C(C)(C)CC c1(OC)ncc(Br)cc1NC(C1CSCCN1C(=O)C(C)OC)=O C1(C(=O)NCCCN(C)C(C23CC(F)(C2)C3)=O)CC2OC(C)(C)OC2C1 N1(C(C(CC)N(C)C)=O)CC(CNC(=O)CC2CC3CC3C2)CC1C c1(CC(=O)NC2CN(C(Cc3ccc(C)nc3)=O)C(C)C2)cccc([N+](=O)[O-])c1 C(=O)(C1=C2CCN=C2NC=C1)NCCN(C(C1C(C(C)C)CCC1)=O)CC1CC1 C(c1csc(Br)c1)=CC(N1CCN(C(C2CCCS(=O)(=O)C2)=O)CC1)=O c1(N2CC(O)(C(C)NC(=O)CC3CCCS(=O)(=O)C3)C2)nccc(S(C)(=O)=O)n1 C12(CC)CN(C(=O)CCCN3C(=O)CCC3=O)C(CNC(=O)C(O)C3CC3)(C1)C2 c1(CC)nc(C)sc1C(N1CC2CC2(C(N2CCC(COC)C2)=O)C1)=O N#CC1CCCC(C(N2CC=CC2C(=O)Nc2ccsc2)=O)C1 CS(=O)(=O)CCC(=O)N1CC(F)(CNC(=O)C=Cc2ccco2)C1 CC(CO)(CCF)Nc1cc(N2CCCC(c3n[nH]c(CO)n3)C2)ncn1 Cc1cccc2cc(C(N3CC(NC(C4CC(=O)N(C)C4)=O)C(F)C3)=O)sc12 c1(N(CC=C)C(C2CN(c3ncc(C(N)=O)cc3Cl)C2)=O)cc2nc(C)ccc2o1 c1(C(=O)NCC2CCN2C(C2CC(C3CCC3)C2)=O)ccc2c[nH]nc2c1 C=CCCCC(=O)NCC1CC1CNC(C1CCN(Cc2cccnc2)CC1)=O c1(C2(C(=O)NC(c3ccc(C)o3)C(F)(F)F)CCCC2)ccccc1F Cc1ccc(OCC(=O)NC2CCN(C3CCCC3)C2)cc1 C1(NC(c2cncc(-n3ccnn3)c2)=O)C=CCN(C(C2CC2(F)F)=O)C1 N1(C(C(CCC)C)=O)CC(CO)C2(C1)CN(C(c1nnc(C3CC3)s1)=O)C2 CCC(C)CCC(=O)NCC1(O)CCCN(C(c2ccc(NC)c(F)c2)=O)C1 N1(C(C(CSC)(C)C)=O)CCC2C(CCN2C(=O)Cn2cc(C)cn2)C1 Cc1nc(N(C)C)sc1C(=O)NC1CC(C)N(C(c2cnn(C(C)(C)C)c2)=O)C1 n1(CCCC(=O)N2CC(N(C)C(C3C(C)(C)C3(C)C)=O)C2)cnc2ccccc12 N1(C(C2(C=C)CC2)=O)CCC(C(C)NC(c2cn(C)nc2C(C)(C)C)=O)CC1 c1(C(=O)NC(CCCC)CNC(=O)C=CC2CCCN2C)cc2scc(Cl)c2[nH]1 C1(C)(NC(C2N(C(=O)NC(COC)C)CC2)=O)CCC1 c1(CC=C)ccccc1C(=O)NC(C1(C(=O)NCC(C2CC(C)(C)C2)O)CC1)C C12(C(=O)NCC3(F)CCN(C(CC4(C)CCOC4)=O)CC3)CCCCC1OCC2 Cc1cc2[nH]c(C(N3CC4CCC4(NC(C4CC(C5CC5)=NO4)=O)C3)=O)cc2o1 C1(CC)CCCN(C(C2Cc3nccn3C2)=O)C1C(=O)NC1CCCCC1(F)F c1(OC)cn(C)c(C(N2CC(OCCNC(C3CCC4(CC4)C3)=O)C2)=O)cc1=O C1(NC(c2ncn(CC)n2)=O)CC2CCC1CN2C(C1CC(n2ccnc2)C1)=O C(=O)(C(O)CCCc1ccccc1)NC1CC(OC)CN(C(=O)CC(C)C)C1 c1(CC)nn(C)c(CC(=O)OC)c1CC(=O)NC1(CS(C)(=O)=O)CC1 C1(CNC(c2c(SC)n(C)nc2)=O)CC(F)(F)CN1C(c1csc(O)n1)=O c1(C(=O)NC2CCC(N3CCCS3(=O)=O)CC2)cc(O)c(O)c([N+](=O)[O-])c1 c12nc3ccccc3cc1CN1CC3CCN2C3C1.C(=O)CCN1CCC1.CO c1(CC=C)ccc(C(=O)N(C)CC2COCCN2C(C2CCCCO2)=O)cc1 C(C(F)C(=O)NC(C)CC1CCCCC1)C1CN(C(COCC=C)=O)C1 c1(NC(=O)NC(c2nc(C)sc2C)C)cnc2c(c1)C(=O)NCC2 O=C(CCCCc1cnn[nH]1)NCC1(F)CC(NC(C23CCCCC2C3)=O)C1 N1(C(=O)OC(C)(C)C)CCC2(CCC(C(=O)NCCCc3ccon3)O2)CC1 C1(C(=O)NC(c2ccccn2)CC)C=CC(NC(c2ccnnc2)=O)C1 CCC(CCO)NC(=O)C(C1CN(C(c2ncn(CC)n2)=O)C1)OC c1(C(=O)NCC2C(C)CN(C(c3c[nH]cc3Br)=O)CC2)nc2cnccc2s1 CCCC(CC(C)C)C(=O)N(C)C(C1CC(Oc2ccccc2)CN1CC)=O C1(C(N2CC(NC(=O)NC)C2)=O)CC2(CCN1C(=O)CS(C)(=O)=O)CC2 Cc1ccc(C(F)(F)F)cc1CNCCNC(C1CCCC1C)=O Cc1cccc(C(=O)NC2CCC(NC(=O)C(CO)NC(N)=O)C2)c1Cl CC(C(=O)N1CCCCC(CNC(=O)CN2CCC2)C1)C(C)S(C)(=O)=O CCC(C(=O)NC(C)CCN(C)C(C1(COC)CC1)=O)SC C1(C(N2CCN(C(C=C(C)C(F)F)=O)CC2C)=O)Cc2cccc(C)c2O1 N1(C(c2c(C)n[nH]c2C)=O)CCN(C(C2CC2c2ccc(Br)cc2)=O)CC1C#N C1(NC(C(C=C)(C)C)=O)CCCN(C(=O)C(C2CCCCCCC2)O)CC1 C(=O)(C1CCCc2nncn21)N(CC(CNC(c1c(C(C)C)nns1)=O)C)C N1(C(C#CC)=O)CCN(Cc2ccc(-c3ccc(N)cc3)cc2)CC1 CC(C)(CC(F)(F)F)C(=O)NCC(C)(O)CNC(=O)C=CC(=O)NC1CC1 N1(C(C2(OCC)CCCC2)=O)CCC(CCc2cn(C(C)C)nn2)CC1 C1(NC(c2cc(CO)[nH]n2)=O)CCN(C(C2CCOC2)=O)CC1O c1(C(=O)NCC(C2(O)CN(C(C(CCC)F)=O)C2)(C)C)ccc(C)c(C#N)c1 N1(C(C(C)C2CCC2)=O)CCOCC1CNC(c1cc(C(C)(F)F)n[nH]1)=O N1(C(C(C)(C)OC)=O)CC2CCC(C1)C2CNC(c1cccn1C(C)C)=O C1(CNC(COCCCC)=O)CCN(C(c2cnco2)=O)C12CCC2 C1(O)(CNC(C2C(C(C)C)(CC)C2)=O)CCCN(C(=O)CCCOC(C)C)C1 C1(O)(CNC(c2coc(C(F)F)n2)=O)CCN(C(C2CC(O)C2)=O)CC1 C1(C)(C(=O)NC(CC(=O)NC(C)C)C)CCN(C(c2ccnnc2O)=O)C1 Cc1nc2cc(CN3CC4(CC4C(=O)NCc4cccn4C)C3)ccc2s1 N1(C(COCCCC#C)=O)CC2CCCC(C1)N(C(=O)Cc1nn(C)cc1Cl)C2 C(=O)(C(Cn1cncn1)NC(c1ccncc1)=O)NCCC1CC(C)C1 C(C(C)(O)C(=O)N1CC2C(CNC(=O)C(F)(F)c3cnn(C)c3)C2C1)OC c1(C(=O)NCC(=O)N(C)CC2N(C(CC=CC=C)=O)CCC2)cc2c(s1)CCC2 c1(C(N(CCC(N2CC(CC)(CO)C2)=O)CC#C)=O)cccc(C)n1 c1(OC)c(Cl)nc[nH]c1=NCc1nnc2c(Br)cccn12 C(CC(CC)C(=O)NC(C(=O)NC(c1ccco1)C)c1ccco1)=CC C12(C(C)=O)CCC(C(N3CC4C(NC(=O)Cc5n[nH]c(C)n5)C4C3)=O)(CC1)CC2 C1(NC(c2c(C)snn2)=O)CCN(C(=O)C(F)(F)c2cncs2)CC1C(C)C c1(OC)cccc(-n2cc(C(C)N(C(=O)C(CSC)OC)C)nn2)c1 c1(N2CCCC(CNC(C)C)C2)nc(=NCC(C)(C)CC(C)O)[nH]c2c1CSC2 N1(C2CN(C(C3CC(=C)C3)=O)C2)CC(NC(c2ccncc2OC2CC2)=O)CC1=O N1(C(CCSCC)=O)CC2CC1CCN2C(c1ccc(-n2ccc(C)n2)cc1)=O N1(C(Cc2c(C)nc[nH]2)=O)CC(NC(c2cc(Cl)c(Cl)s2)=O)CCC1C C(=O)(CCC1=CCCCC1)N(C)C(C1COC(CC)C1)=O.C1(C)(C)CCCO1 c1(C(=O)NC2C(NC(C(C=C)(C)CC)=O)CCCC2)cccc2c1CCN2 C1(NC(c2cncc(C)n2)=O)CCCCN(C(=O)CCCn2ccnc2)C1 N1(C(c2c(COC)onc2)=O)CC2CCC1CN2c1ncnc(C(F)(F)F)c1Br C1(C(N2C(C(=O)O)CC(OCC)C2)=O)CC(=O)c2cc(F)ccc2O1 c1(C(N2CCC(C(C)(C)NC(CN(CCCCCC)C)=O)C2)=O)cnn(C)c1Cl c1(NC(C2C(CC)CCCN2C(C2CCCC(=O)N2)=O)=O)cn(C)c(=O)nc1O C1(C(N2CC(C=C)(O)C2)=O)CC2CCC(C1)N2C(=O)CC1CCC(=O)C1 C#CC1(C(=O)NCC2CCCN(C)C2)CCN(C(=O)CCc2nc[nH]n2)CC1 c1(C(N(C=O)CC2CCC2)C)ccc(F)cn1 c1(C(N(CCNC(c2c(OCC)ccs2)=O)C(C)C)=O)ccc([N+](=O)[O-])c(C)c1 c1(C(=O)NCC2CN(C(CSc3c(C)ccc(C)c3)=O)C2)cncc(N=[N+]=[N-])c1 C1(CNC(CCCNC(C)=O)=O)CCCC(NC(c2cc(C)n(C(C)C)n2)=O)C1 C(=O)(CC(C)CC(C)C)N1C(C)(CCC(=O)NCC=C)CCC1 C1(CC)CN(C(=O)CC2CCC3(CC3)CO2)CCC1NC(=O)C(C)=CC(C)(C)C C(=O)(C(O)(C(F)(F)F)c1cn[nH]c1)N(CC(CNC(CCSC)=O)O)C c1(CC)ccc(O)c(C(N2CCC(CNC(=O)Cc3cncn3C)C2(C)C)=O)c1 C1(CNC(CN(C)C)=O)CN(C(=O)Cn2cc(C(F)(F)F)cn2)CCC1(C)C c1(C(N(C(CCNC(c2ccc(CCC)[nH]2)=O)C)C)=O)ccc(Cl)c(N)c1 C(=O)(CCCC(C)(C)C)N1CCN(C(Cc2ccc(SCC)cc2)=O)C(CC)C1 C(c1cc2ccccc2o1)=CC(N1C2CN(Cc3nccc(OC)c3)C(CC2)C1)=O Cc1cccn2cc(C(N3CCC(NC(=O)CCSCC(C)C)C(O)C3)=O)cc12 C1(C(N2CC(CC=C)(NC(=O)CCc3cccnc3)C2)=O)CCC(N=[N+]=[N-])CC1 CC(CS(C)(=O)=O)C(=O)NCC(O)CNC(C1CCCCN1C(N)=O)=O C1(NC(C(CC)OC)=O)CN(C(=O)CCc2cn(C)nn2)CC2(CCC2)C1 c1(OCC)ccc(CC(=O)N(CC(C)(C)CNC(C2(C(C)C)CC2)=O)C)nc1 CC(C)CC(C(=O)NC(C(=O)N(C1(CO)CC1)C)C(C)C)C(N)=O CCC(CC)C(F)C(=O)NC1CN(C(=O)Cc2ccc(F)c(F)c2)C(C)(C)C1 N1(C(C(C2CC2)NC(c2cc(OC)ncn2)=O)=O)CCCCC(C)(F)C1 CCCCC(=O)C(=O)N1CC2CC(N(C(=O)C(C)C(C)C)C)C1C2 CONS(=O)(=O)c1ccc(C(=O)NCC=CCNC(C2(CO)CC=CC2)=O)cc1 C(=O)(CCC(=O)NCC1CCCC(NC(=O)C(F)(F)c2nc(C)cs2)C1)NC N1(C(c2cn(C3CCC3)nn2)=O)CCCC2(CCN(C(C3(O)CC3)=O)C2)C1 C1(C(=O)NC2CN(C(C3CCC(C)O3)=O)C(C)(C)C2)CCc2n[nH]cc2C1 c1(C=O)cc(O)c(Br)c(O)c1.c1(NCC2CCNC2)sc(Br)nc1Br c1(COC)cc[nH]c1C(=O)NOC(C)(C)C(=O)N(CCOC)CCOC N1(CC)CCN(CC(C)(C)NC(=O)C(n2cc(C(C)O)nn2)C)CC1 N1(C(CCc2onc(CC)n2)=O)CCC2(CC1)CC2NC(=O)CCOCC1CC1 N1(C(C(C(=O)OCC)OC)=O)CC=C(C(=O)NC(C)(CO)C2CCC2)C1 CC1(C)CCCCC1C(N1CCCC1CCCNC(C1(C)CC1(F)F)=O)=O c1(CC(=O)NCC2CN(C(c3cnccc3Cl)=O)CCO2)ccc(I)cc1 c1(C(N(C(CCNC(CC2C(CC)C2)=O)C)C)=O)cc(CN(C)CC)ccc1N C1(C(C)C)CN(C(=O)C=Cc2cscn2)CCN1C(=O)Cc1cc(O)nc(O)n1 Cc1nsc(C(=O)NCC2CCCN2C(=O)C=C2CCC2)c1N N1(C(c2ccc(C(C)C)o2)=O)C2CCC1C(CNC(=O)CCc1n[nH]c(=N)s1)C2 N1(C(N)=O)CCC(C(N2CCC(CCNC(c3cccs3)=O)C2)=O)CC1 C1(NC(c2c(C)[nH][nH]c2=N)=O)CN(C(c2nnn(C)c2C)=O)C2(CCOCC2)C1 N1(C(C2C3(CC(NC(CC4C(C)(C)OCC4)=O)C3)C2)=O)CC2CSCC2C1 c1(SCC)csc(CO)n1.C(CCOCCN(CCO)CC)N(C)C=O.C.OC c1(C(N2CC(CNC(COCCC#C)=O)C2)=O)cc(-c2ccn(C)c2)[nH]n1 c1(C(=O)Nc2ccc(NS(=O)(=O)CCCl)cc2F)cc(Cl)c(Cl)nc1Cl CCC(C)C(O)C(=O)N1CCCCC1C(=O)N(C)Cc1nc(C)cs1 CC1CN(C(C2CN(Cc3cccc(N(C)C)c3O)CCC2O)=O)CCN1C c1(C(=O)NC(CNC(C(COCC)C)=O)C2CCC2)ccc(-n2cnnc2)cc1 Cc1nc2ncc(C(=O)NCC3COCC3NC(C3(C)CCCO3)=O)cc2o1 C(=O)(CCC(=O)c1ccccn1)NC(CC)CN(C(=O)C(C)C)C Cc1cc(NC(C23CC2CCN3C(=O)C(C)CC#N)=O)cc(C)c1 c1(C(=O)OC)cc2ccccc2cc1S(=O)(=O)NCC1(C(N)=O)CC1 CCC(C)CCCCC(=O)NC(CNC(=O)CCc1nnc(C)n1C)C(C)(C)C c1(NCC2(OC)CCCOC2)nc(N(CC(F)(F)CC2CC2)C)cc(C)n1 c1(OC)cc(C)c(NC(C2CN(C(=O)C(=O)N(C)C)C3(CCC3)C2)=O)cc1Cl c1(NC)cc(Cl)ccc1C(=O)NCCOC1CCN(C(=O)C#CC(C)(C)C)C1 N1(C(CS(CC)=O)=O)CCN(C(c2ccc3c[nH]nc3c2)=O)CCC1C c1(C(=O)NCC2CN(C(CCCOCC=C)=O)CC2O)cn2cccc(F)c2n1 N1(C(COCCOC)=O)CCC2(C=C(C(=O)NCC3CC3CO)C2)C1 c1(C(=O)NC2CN(C(C(=O)NC)C)CC2(C)C)c[nH]c2nccc-2c1 C#CCC(C)C(=O)N1CCOC(CN(C)C(c2ccc(N(C)CCC)cc2)=O)C1 c1(C(N2CCC3CCC(C2)N3C(=O)C(O)C2CCC2)=O)cn2cccc(Cl)c2n1 N1(C(n2[nH]c(C(C)(C)C)nc2=S)C)CC(=O)N(CCOC2CCCC(C)C2)C1=O C1(CNC(C2N(C(C3C(=C)C3)=O)CC2)=O)CCC2(CC2)C1 C1(F)(NC(=O)CCCc2nnc(-c3ccccc3)o2)CCCCCC1 C#CCCCC(C)C(=O)NCC(C)N(C)C(c1ccc(C)cc1C)=O C1(C(=O)NC(COC)(C)CO)CCCN(C(=O)CCc2ccn(C)c2)C1 CC1(C)CCCC(CC(N2CCC(NC(=O)CCc3ccccn3)C2(C)C)=O)O1 c1(OCC(=O)NCC=CCNC(C2(c3ccncc3)CC2)=O)cccc(Br)c1 c1(C(=O)NCC2CC(C)(C)CN(C(C3CC3C#N)=O)C2)c(Cl)ccc2c[nH]nc12 C1(CC(N2CCC(CCOC)C2)=O)CCCCN1C(=O)CCC(=O)C1CC1 C(=O)(C1=CCC(F)(F)CC1)N(C1CCCC(N(C)C(c2cc(=O)n(C)o2)=O)C1)C N1(C(c2cc(OCC)ncc2)=O)CCC(NC(c2cnc(F)cc2C)=O)C(C)C1 C12(CNC(C(COCC)C)=O)CCC1CN(C(=O)COc1c(F)cccc1F)C2 C1(C(=O)Nc2c(C(N)=O)cnc(Cl)c2)COC2(CCN(C(C3(Br)CC3)=O)CC2)C1 C=CCCCCCC(=O)N1CCC(C(N2CCC3OCCC3C2)=O)C1C(C)C C(=O)(C1CCc2ccccc21)NC(C(=O)NC(CCC=C)(C)C)(C)CO N1(C(Cc2cn(CC)nc2)=O)CC2(C1)CN(Cc1ccc(Cl)c(F)c1)CCO2 C(=O)(CS(=O)(=O)CCO)N(CC(O)CNC(C1(SCC(F)(F)F)CC1)=O)C Cc1cc(C(=O)NCC(C2CC2)NC(C2CCCN2N=O)=O)c(N)cc1F Cc1cc(F)cnc1C(=O)NC(C(=O)NCc1cnc(O)nc1O)C1CCCC1 C(=O)(CCC(C)CCCC)N1C(C(=O)NCCCC#C)CC(C)C1 c1(C(=O)NCC=CCNC(C2C(COC)C2)=O)n[nH]c2c1CSCC2 c1(C(CNC(=NC)NCC2CCCO2)N(C)C2CC2)ccc(Cl)cc1 C1(C(=O)NCCCC(C)(C)NC(CC2(COC)CC2)=O)CC12CCC1(CC1)CC2 C(=O)(C1CC(=O)N(C)c2ccccc21)NCCCCC(C)NC(C=CC)=O N1(C(CSCCC)=O)CCCC(O)(CN(C(=O)C(n2cnc(C#N)n2)C)C)C1 c1(C(N)=O)cc(=NCC(O)CNC(=O)Cn2nccn2)[nH]cn1 C1(C(=O)NC2C(OC)C(O)C2)C(C)CCN1C(C1OCCC1(C)C)=O c12ccc(cc1)-c1cn(nn1)C(C)(C)CC(=O)N2.CC(F)(F)N(C)CC1CCC1 c1(-n2cc(CC3CCN(C(c4c(OC)noc4)=O)CC3)nn2)ccc(Br)cc1Cl C1(C(N2C(C)CC(NC(C3(C)CC(=O)C3)=O)C2)=O)C2C3CCC(C3)C12 c1(C(CN2C(c3nn(CC)nc3C)C(C)CCC2)O)cccc2c1OCC2 c1(C(=O)NC(CC(=O)NCC(C=C)O)C(C)OC)ccnc2cc[nH]c12 C1(C(N(C(C)C)CCNC(=O)COC2(C)CCC2)=O)CCS(=O)(=O)C1 c1(C(c2nnnn2C(C)(C)C)NCCN2C(C)CCCC2)cc(Cl)c(Cl)c(Cl)c1 c1(SCC)ccc(CC(N2CC(CCNC(c3nocc3Cl)=O)C(C)C2)=O)cc1 C12(C(=O)NC(C(C)C)CCNC(=O)C=C3CCOCC3)CCN(C1)S(=O)(=O)C2 C(=O)(C1=NN2CC(C)CN=C2N1)N1CCC(C)(CNC(CCCCCOC)=O)C1 C(CCCCC(=O)N(C1CCC(CNC(=O)CC2CSCCO2)CC1)C)SC c1(C(=O)OCC)cn(C)nc1C(=O)NC1CCN(C(=O)CCCOC(C)(C)C)C1 c1(SC)nc(C(F)F)cc(=NC(C)C2CNC2)[nH]1.c1(C=O)nc(F)ccc1Cl c1(C(N(C2CCOCC2)CC(=O)OCC)=O)ccc(OC)c(OCC)c1C(F)F N1(C(C(C)OCOC)=O)CCC(CCNC(C2CCOC2C)=O)CC1 CC1CCCC(CC(=O)N(c2ccccc2F)CCCCCN2CCCC2)C1 C(=O)(C1=NOC(CNC(=O)CCC(C)C)C1)NC(c1ccc(C)cc1)C S(=O)(=O)(c1cccnc1NCC1CC(C(F)(F)F)C1)N1CCC(CSC)C1 S(=O)(=O)(c1cnc(NCCCNS(C)(=O)=O)c(Cl)c1)NCC(C)(C)C(F)(F)F C1(NC(c2c(C)nc(C3CCC3)o2)=O)CCCC12CN(C(C1CCNC1=O)=O)C2 c1(CCC(=O)NCC(CNC(C(C)OCC(F)(F)F)=O)CO)ccc(O)nn1 N1(C(c2cc(C)[nH]c2C)=O)CC2CCC(C1)N2Cc1cc(O)ccc1F C1(CNC(C(C)=C2CCC2)=O)CC2(CCC2)CN1C(=O)CC1(C)CC1 C(C(CC(C)C)C(=O)N1CCCC(NC(c2ccc(C#N)cc2F)=O)CC1)OC C(N=c1nc(Cl)[nH]c(C)c1C#N)N1CC=C(CNC(Cc2nc(CC)sc2)=O)CC1 CC(C(=O)N1CCCC1CCC(N1CCCC(O)C1)=O)C(F)F C1(CC(=O)NC(C)(C)CCNC(=O)Cc2ccsc2)CC2CCC1C2 N1(C(c2ccc3sncc3c2)=O)CCCC1C1CCCN1C(c1ccsn1)=O C1(N(C(c2cncc(OC)n2)=O)C)CCN(C(c2c(C)noc2N)=O)CC1C C(=O)(C1=CCCCO1)N1C(C2CCN(C(CCc3c(C)cccc3)=O)C2)CCC1 c1(OC)ccc2c(c1)CC(C(=O)NC1CCC(NC(=O)Cc3cnc(C)s3)C1)O2 C(CC)(C(=O)NCC=CCNC(=O)CCc1nccn1C)OCC C(CC(C)(C)C(=O)NC1CC2CC1CN2C(c1cc(C2CCCC2)no1)=O)OC c1(C(=O)NCCN(C(C)C)C(C2CC3CCC3C2)=O)ccc2nc(CO)[nH]c2c1 N1(C(c2c(C)nc(Br)s2)=O)CC(NC(=O)C=C(Cl)Cl)CC(C)C1 N1(C(C(C)=CC)=O)CC(C2CCN(C(=O)Cc3ccc(C(=O)OC)c(C)c3)CC2)C1 c1(C2(O)CC(C(N3CC(NC(C4N(S(C)(=O)=O)CC4)=O)C3)=O)C2)ccc(F)cc1 c1(CC(C(=O)N(CCOC)CC2CCC3CC23)c2ncco2)c(C)cccc1Br C1(CN(C)C)CC(CN(C(=O)C(F)C2CCCC2)CC(=O)NC2CC2)C1 C1(CC(=O)Nc2nc(Br)cs2)CC2(C1)CN(Cc1cc(F)ccc1Cl)C2 S(=O)(=O)(c1ccccc1F)NCC(=O)N(CCCNC(C(C(C)C)NC=O)=O)C C(=O)(C#CC1CCCC1)N1CCCC(CCNC(c2noc(CC)c2C)=O)C1 C1(C(=O)NCC2CCN(C(C3(OC)CCCC3)=O)CC2)CC2(CCC2)CO1 N1(C(CN(C)C)=O)CCC(C(=O)Nc2cccc(F)c2F)C1(C)C C1(C(N2CC(OC)(CNC(c3cc(C(C)C)no3)=O)C2)=O)CCCC12CC2 CCC(CNC(=O)C=CCNC(C12CCC(CC1)C2)=O)C(C)C CN1CCN(CC(=O)NCc2ccccc2CN(C(=O)CC(F)(F)F)C)CC1=O c1(OC)ccc(Br)c(-c2noc(-c3cnc(O)c(C)c3)n2)c1 c1(CN(C(=O)NC(c2noc(C3CC3)n2)C)C)nc(Cl)cc(N)c1Cl C12(CNC(CCN(C(CC)CC)C)=O)CCC1CN(C(=O)C(C)S(C)(=O)=O)C2 CCCC(C)CCCC(=O)OCC(=O)N(C1CCOCC1)C(C)C N#CC1(NC(N2CCN(CC(N3CC4C(C3)C4(F)F)=O)CC2)=O)CCCOC1 N(C(=NCc1ccnn1C)NCC1CC12CC2)C(CC)CO CC1CN(C(=O)Cc2ccccc2F)CCN1C(C1CCC(C(C)(C)O)CC1)=O N1(C(C(CC(C)C)(F)F)=O)CCC2(CCC2CNC(=O)C2=CCCC2)CC1 N1(C(=O)CCC2CCCCC2)CCC2CN(C(=O)C(O)Cc3cnc[nH]3)C2C1 c1(NC(=O)Nc2cn(CCCl)nn2)cc2c(cc1F)NC(=O)CO2 c1(C(=O)NCc2c(CCNC(C(C)OCC=C)=O)ocn2)ccncc1N N1(C(COCC(=O)OC)=O)CCCCCC1CNC(C1CC(C)(F)C1)=O CCC1=NOC(C(=O)NC(CCN(C)C)C(=O)NC(C)C(=O)N(C)C)C1 c1(C(=O)NC(c2ccccc2)CNC(=O)COC2CC2(F)F)cnnc(O)c1 N1(C(CC=CC=C)=O)CC(NC(C2CC2c2ncccn2)=O)C(SC)C1 CCC(O)C(C)(C)C(=O)N(C)CC1CN(C(=O)Cn2ccc(C)n2)CCO1 C1(C(=O)NCC(COC)(C)O)CC(=O)CN1C(C1CCCN1C(C)=O)=O N1(C(C2(C)CCN(C)CC2)=O)CC2CCC(CNC(C3(C(F)F)CC3)=O)(C2)C1 N1(C(C(CCSC)NS(CC)(=O)=O)=O)CCCN(C(c2ccco2)=O)CC1CO C#CCC(O)C(=O)N(C1CCN(C(=O)CN(S(C)(=O)=O)C)CC1)CC C1(C(=O)NCC=CCNC(c2c(C)nn[nH]2)=O)CC2(CCCCC2)C1 C1(NC(Cn2cc(CC(OCC)OCC)nn2)=O)CS(=O)(=O)CC1O C(=O)(C(CO)NC(C1(NC(=O)CC2(OC)CCC2)CC1(C)C)=O)OC C1(C(N2C(CNC(c3cnc(CC4CC4)o3)=O)CCC2)=O)CCC(O)CC1 Cc1cccc(C(=O)NC2(C(=O)NCCN3CC4CC4C3)CCN(C)C2)c1F C(=O)(C1SCc2cccnc21)NCC(CNC(C=NOC)=O)F c1(C(=O)NC(CC)(CNC(=O)C#CC2CC2)CC)ccc(CO)cc1F Cc1cc(C(N2CCN(C(=O)CC3(O)CCCOC3)C(C)C2)=O)cn(C)c1=O N1(C(c2c(C)scn2)=O)CC(O)CC1C(=O)NCC(C)O C=CC(CC)CC(=O)N1CCC1C(=O)N(C)CCN(C)C1CC1 Cc1nc(CC2CC2)sc1C(=O)NCCC(C)NC(C1C(C)C1C)=O N1(C(C=CC(c2ccccc2)=O)=O)CCC(CCNC(C2CCS2(=O)=O)=O)CC1 c1(C(N2CCC(N(C(C3CC3c3cncn3C)=O)CC)C2)=O)cc(C)ccc1O N1(c2n(CC(=C)C)nnn2)CCN(C2CCCN(C(c3cncs3)=O)C2)C(=O)C1 c1(CN2CC3CN(C(CS(C)(=O)=O)=O)CC3C2)cncc2ccccc12 c1(CC(=O)NCC(C)N(C)C(c2ccc(C(C)(C)C)o2)=O)ncsc1Cl C1(NC(CN(C(COC)=O)C)=O)CC=CCC1C(=O)NC(C)(C)CCO c1(C(N2CCCC(N(C(C(n3c(C)ncc3)C)=O)C)C2)=O)cccc2c[nH]nc12 c1(C(=O)NCC2C(NC(C3(C)CCNC(=O)C3)=O)CCC2)cc(N)c(F)c(F)c1Cl C1(NC(CC2N(C)CCC2)=O)CCCCCC1C(N1CC(O)C1)=O Cc1ccc(NC(=O)CC2CN(C(c3cn(C)cc3C)=O)CCC2C)cc1C#N c1(C(=O)NC2CCN(C(C(CC=C)C(C)C)=O)C2C)cccc2c1CC(C)(C)C2 C#Cc1ccc(OCC(=O)NC23CC(NC(C4CC=CC4)=O)(C2)C3)c(OC)c1 N#CC1(C(=O)NCCC2CCCCN2C(c2cc(F)n[nH]2)=O)CCCCC1 CC1(C)CN(C(=O)Cc2ccc(Cl)s2)CC(CNC(c2cc(O)ncn2)=O)O1 c1(OC)c(C(=O)NC2CC(O)CN(C(C3CCS(=O)(=O)CC3)=O)C2)cccc1Cl C(=O)(C(C)CC(=O)N1CCC(F)(CNC(c2cc(F)ccc2C(C)C)=O)C1)OC C1(CNC(NC(C)C)=NCc2ccc(-c3nc[nH]n3)cc2)COCCC1(F)F N1(C(C=C(C)C(C)(C)C)=O)CC(NC(=O)C=CCF)CC12CCCOC2 C(CC)(CC(C)O)NC(C1CC(C)(NC(c2cnc(CC)s2)=O)C1)=O Cc1nc2ccccc2cc1C(=O)NC1C2CN(c3nc(Cl)c(C#N)s3)CC12 CC1CN(C(=O)C=CC(c2ccccc2)=O)CCN1Cc1ccc(F)nc1F C1(C(=O)NCC(C(=O)OC)C)CC(NC(=O)C2=CC(C)(C)C2)C12CCC2 CCCCC(F)C(=O)N1CCC(C(=O)N(CCCC)CCO)C(O)C1 c1(C(N2CCCC(NC(CCC3(C)CCC(=O)N3)=O)C2)=O)cnc2n1CCOC2 Nc1ccc2c(c1)N(C(C1C=CCS1)=O)CCC2 c1(CC)nnc(C)cc1C(N1CCC2(NC(=O)CCc3ccncn3)CC2C1)=O N1(C(C(CO)N(C)C)=O)CCN(C(C2CCC(C)(C)CO2)=O)CC1CO Cc1cccc(COCC(=O)NC(C)(CNC(=O)CSC2CC2)C2CC2)c1 C(=O)(CC(C)(F)F)NCC1C(NC(CC(=C)Br)=O)C1 Cc1cc(C(=O)N2C3(COC3)C2)ncc1F.c1(N)ccccc1.OC N1(C(C2(CNC(C3C(COC)CC3)=O)CCCO2)=O)CC2(C1)CN(C)C2 c1(CSCC(=O)NC(C2CCN(C(c3ccncc3)=O)CC2)C)ccccc1Cl CC1CN(C(C23CC2CNC3=O)=O)CC1CNC(c1nncs1)=O C1(NC(C(n2cc(Cl)cn2)C)=O)CN(C(=O)CCC#N)CC1O N1(C(C(C2CCCN(C(c3cnsc3)=O)C2)C)=O)CCN(C)CC(O)C1 c1(NC(C(=O)NC2CCC(CSC)CC2)=O)ccc(OC(C)C)c(Cl)c1 N1(C(C2C(C)CCO2)=O)CCC(F)(CNC(=O)CN(C)C(N)=O)C1 c1(OC)cccc2c1C(C(=O)NCC1(NC(=O)C3=CCCS3)CCOC1)CC2 n1(CCC)cncc1CNC(C1(NC(=O)C(C)c2ccsc2)CC(F)C1)=O C1(C(=O)OC)CN(c2ncnc3[nH]cnc23)CC12CCCC2 c1(CCC)cc(C(=O)NC2(CNC(=O)CCc3nc(CC)no3)CCC2)ccn1 Cc1cc(C(N2CCOCC2CC(=O)NCCn2ncccc2=O)=O)cc(O)c1 C1(NC(C2CCC(C)O2)=O)CN(C(=O)Cc2cnccn2)CC2(CC2)C1 C1(C#N)(C(N(CC(N2CCN(C(c3cc(C)oc3)=O)CC2)=O)C)=O)CCSCC1 c1(NC(C(COC)C)=O)cccc(NC(c2cc(OCCO)ns2)=O)c1 CC(C)C(C(=O)N1CCCC(NC(=O)Cn2cc(C(N)=O)nn2)C1)NS(C)(=O)=O S(=O)(=O)(CCC(=O)NC(C)CC1CN(C(C2(C#N)CCC2)=O)C1)NC c1(OC)ccc(CC(=O)Nc2ccc(NC(=O)Cc3cnns3)c(C)c2)c(F)c1 CCCCC(C(=O)NCC1=CCN(C(=O)CCc2cncnc2)CC1)C(C)C N1(CC(=O)NCC2OCC(CNC(C(C)(C)C3CC3)=O)C2)CCCCCC1=O CC1(CNC(=O)C(CC2CCCO2)NC(=O)CN2CCCCC2)CC2(CC2)C1 C1(C(=O)Nc2nc(C)cc(C)n2)CC2CCCCC2N1C(C1CCC1)=O c1(C(=O)NCC2(CNC(C3C(OC)CCCC3)=O)CC2)cnn2ccsc12 C(=O)(CCS(N)(=O)=O)NC1CCC(CNC(CCSCC)=O)CC1 C1(CC(N2CC(CN(C(C(C)C)=O)C)OCC2)=O)CC2CCC1CC2 N1(C(c2cc(CC)ccn2)C(=O)NCC)CCc2ccc(N(C)C)cc2C1 C(=O)(CC(C)(C)c1ccccc1)N(C1CN(C(=O)Cn2cc(Cl)cn2)CC1F)C c1(C(=O)NC23CCN(C(=O)CC4(CO)CC4)CCC2C3)cnnc2ccccc12 c1(C(N2C(C)CC(CNC(C3(C4CCC4)CC3)=O)C2)=O)cc(Cl)cc(Cl)c1N C(=O)(C1=CC(C)(CC)C1)NC1CC(CCNC(CCC#C)=O)C1 C12(C(N3CCC(N(C)C(C4CCC4)=O)C3)=O)CCCC(C)(C1)OC2 N(C(=NCCF)NC1CC1c1ccccc1Br)C(c1ncn(C)n1)C C(=O)(C1=Cc2cc(F)ccc2OC1)NCC1CC(C)(C)CN1C(C1CC1(C)C)=O Cn1ncc2cc(C(N3CCC(NC(c4ccoc4Cl)=O)C(F)C3)=O)ccc12 N1(C(COCCOCC#C)=O)CC(NC(c2nsnc2O)=O)CC1(C)COC CCCC(O)C(=O)N1CC(CC(=O)NC2CCCN2C=O)(OC)C1 C1(C(=O)NCC)(C(C)C)CCN(C(c2ccncc2OC)=O)C1.CCCN1CC1 N(C(=NCCCN1CCOCC1)NC(C)COC)CC1(OCC)CCC1 Cc1ccc2c(c1)CC(C(N1CCN(c3cc(C(C)C)ncn3)CC(O)C1)=O)S2 c1(C(=O)NC2C(C)CN(C(=O)CC3CC=CC3)CC2)cnc2c(=O)[nH]ccc2c1 Cc1nccc(C(=O)N(CC(C)CNC(C2(CC(F)F)CCC2)=O)C)n1 C(=O)(C(C)(C)C(=O)OC(C)(C)C)N(C1CCN(C(C2C(OCC)C2)=O)C1)CC C1(NC(C(=O)NCc2nnc(COc3ccc(F)cc3)s2)=O)CC2CNCC12 c1(CC(N2C(C)CC(NC(C3(C(N)=O)CC3)=O)C2)=O)cc2ccccc2oc1=O N1(C(COCc2ccc(C)cc2C)=O)CCC(O)C12CCCCCC2 C1(C(=O)NCC2CCC(C(=O)NC(CCOC)C(C)C)CC2)(CC)CCOCC1 c1(CC)ccc(C(=O)NC2(CO)CCCN(C(C3CC4(C3)CC4F)=O)C2)c(O)c1 Cn1cc2c(C(=O)NC3CN(C(c4cncc5c[nH]nc45)=O)C3)cccc2n1 N(C(=NCC(C)C)NCc1cc(-c2ccccc2)no1)C1CCCC(OC)C1 N1(C(CC(C=C)C)=O)CCC(C)CC1CNC(=O)Cn1cc(Br)c(C)n1 C12(CNC(c3c(CC)ncs3)=O)CC(CNC(=O)C(C)OC)(CO1)C2 c1(CC(N2CCN(C(C3CC(C)C3)=O)CC2CC(F)F)=O)ccc2nonc2c1 C(=O)(C(C)C(C)S(C)(=O)=O)NCC1OCC2(CN(C(c3cn(CC)nc3)=O)C2)C1 c1(CNC(N2CCN(S(=O)(=O)C3CCCCC3)CC2)=O)ccc2ccncc2c1 c1(OC(C)C)ccccc1C(=O)NCCN(C)C(C1(C(F)F)CC1(F)F)=O N1(CCN(C(=O)CC=CCNC(C2CC2C2CCCO2)=O)C)CCCCC1 C12(C(=O)NC(CNC(C(C(C)O)N(C)C)=O)C3CCC3)CCC(CO)(CC1)CC2 C1(NC(CSC(C)C)=O)CC2CCC1C(NC(=O)CS(C)(=O)=O)C2 Cc1ccc(CNC(C2CCC(C)C2)=O)nc1.C1(C(=O)N)CCC=CCC1 C1(C(N(CC(C)NC(C2(COC)CCC2)=O)C)=O)CCCCC1(C)C c1(C(=O)OCC2C(NC(C)=O)C2)cc(CC2CCC2)ccc1F C=CCC(C(=O)NCC1CN(C(=O)CCC(=O)OCC)CC1OC)C(C)C N1(C(COCC(C)C)=O)CCC(CNC(=O)CCC2CCN(C)CC2)C12CCC2 CN1CCCC(O)(CC(N2CCC(CCNC(c3cccc(Cl)c3N)=O)C2)=O)C1 C1(CCNC(c2cc[nH]c2C2CC2)=O)CCCN(C(=O)C=CC2CCCO2)CC1 N1(C(C(C)Cc2cccnc2)=O)CCC2(CC1)CC2NC(C1CC12CCCC2)=O C(=O)(CC(C)(C)C(C)=O)N(CC(=O)NC1CCOC1C)CC C1(C(=O)NCCCN(C(=O)Cc2cncc(C#N)c2)C(C)C)CC2CCC1CC2 N1(C(CCc2cc(C)no2)=O)CC2C=CCOC2C1 CN1CCC(=CC(=O)N(CCNC(C2(C)CC2F)=O)CC2CC2)C1 c1(CC)cc(C)ccc1NC(=O)C(C)N(C(C1CC=C(C)CC1)=O)C1CC1 C1(C(N(CCNC(c2cncc(C)c2)=O)C2CC2)=O)CCn2cc(C)nc2C1 C1(NC(=O)C2=COCC2)CCCCCN(C(c2cc(C(F)F)ccc2F)=O)C1 C1(C2CCN(C(=O)Cc3nnn(C(C)(C)C)n3)CC2)(NC(CCC2(C)CC2)=O)CC1 c1(OC)nccc(=NC2CC2c2cccc(C(F)(F)F)c2)[nH]1 C1(C(N2CC(=C(CNC(c3c(Cl)nsc3Cl)=O)F)C2)=O)Cc2ccncc2C1 C(=O)(CCCC(=O)Nc1cccc(CNC(c2cc(Cl)ncc2C)=O)c1)OCC c1(C(=O)N(C2CCN(C(c3n(CCOC)ncc3)=O)C2)C2CC2)ccc(Cl)c(O)c1 c1(C(c2ccccn2)Nc2nccs2)ccc(F)cc1.CC1C(=O)N1C C1(NC(C(CCC#C)O)=O)CCC2(CC1)CN(C(=O)COCC1CCCOC1)C2 c1(OCCC(=O)NCC2(F)CCN(C(C3CCCCO3)=O)C2)ccccc1F C(CC(C(=O)NCC1(CO)CCOC1)NC(c1cc(C)sc1C)=O)=CC c1(C(=O)NC2CCC(CC(=O)N(C)Cc3ncn(C)n3)C2)cccn2ccnc12 C1(C(=O)NC2CCN(C(C3C(=O)NCC3)=O)CC2)CC2CC1CC2O CCC(CC)CCC(=O)NCc1n[nH]cc1C(=O)N(C)Cc1cnc(C)s1 C(=O)(CCCCCC(C)C)N1CC(O)(C(C)NC(C(CC)OCC)=O)C1 Cc1nnc2n1CC(C(N1CC(CNC(=O)CC(C)(C)C#N)CCC1C)=O)CC2 c1(CC(=O)NCCN(C)C(c2cc(-c3ccco3)on2)=O)ccc(NC=O)cc1 Cn1cc([N+](=O)[O-])c(OCC(N2CC=C(CNC(C3CCC3)=O)CC2)=O)n1 CN1C(=O)c2ccccc2C1CC(=O)NCC12CCC(C1)N(C(C1CC1F)=O)C2 N1(C(C(C)SCC)=O)CC2(C1)SCCC2NC(=O)Cc1cccc(Cl)c1F c1(CC)occ(C(F)(F)F)c1C(=O)NC(C)CC(C)NC(c1c(Cl)cnn1C)=O c1(C(=O)NC2C3CCN(C(c4ccc(OC)cn4)=O)C32)cc2ccccc2cn1 c1(OC)ncc(C(=O)NC(C)(C)CCNC(C2(F)CC=CC2)=O)cc1C CC(C)C(C)CC(=O)NCC1CN(C(=O)CC2CC(C)OC2C)CCCO1 CC1(CNC(N2CC3CC(CO)(C3)C2)=O)Cc2ccccc21 C1(N(C(C=C(C)C(C)(C)C)=O)C)CN(C(c2ccnc(C(C)C)n2)=O)CC1O CC(C)(C)C(CCO)NC(=O)COC1CC(NC(C2CC(=C3CCC3)C2)=O)C1 N1(C(=O)COCc2ccccc2Cl)CCC(F)(CNC(C2(F)CCCC2)=O)C1 CC1(C)C=C(C(=O)NCCCCC2CN(C(c3ccco3)=O)C2)C1 N1(C(COCC#C)=O)CC(C)N(C(=O)CCCN2C(=O)CNC2=O)CC1C C(=O)(C(O)Cc1[nH]cnc1C)NC(CCNC(C(C)=C(CC)C)=O)C C(CC(C)(C)C(=O)NOC1CC2CCC1C2)NC(CC1CCC(C)O1)=O c1(C(N2C(C3(O)CN(C(CSCC)=O)C3)CCC2)=O)ccc2c(c1)CC(C)O2 C1(C(C(=O)NC2(C)CC2)N(CC(F)F)CC)CCC2CC1C2(C)C c1(N(C2CCCN(C(C3CCC(F)C3)=O)C2)C)ncnn2c(Br)ccc12 CC(C)CCCCC(=O)NCC1CC(CNC(=O)C=CC2CCOCC2)CO1 c1(CN2CCCC(NS(CCC)(=O)=O)CC2)cccc(S(C)(=O)=O)c1 CC(O)(C(=O)NCC(CNC(c1coc(O)n1)=O)CO)c1ccccc1 CCCCC(CC)C(=O)NC(c1ccccc1SCC)CNC(=O)C(=O)N(C)C CC1CCC(C(N2CC(CNC(=O)COC(C)(C)C(F)(F)F)(COC)C2)=O)CC1 C1(C(=O)NCc2c(C)ccnc2)CCN(C(C23CSCC2C3)=O)CC1C N1(C(c2n(CC)ccn2)=O)CC(NC(c2cccc(C#N)c2)=O)C(C2CC2)C1 c1(OC)ccc(C(=O)NCCCCNC(C2CC2OC)=O)cc1OCC(F)(F)F c1(OC)ccc(S(=O)(=O)NCC(=O)NCCCCC(C)(F)F)cc1 C(=O)(C1CCc2ccc(Cl)nc21)NC1CN(C(C2(CC(=O)OC)CC2)=O)CC1F CC1(C)CC(NC(=O)CCC2CCCCC2)CN1C(c1snc(O)c1Cl)=O C1(CNC(CC=C)=O)CN(C(c2cc(-c3ccccc3)ns2)=O)CCN1C CN1CCC(O)(CNC(C2(CNC(C3CCNC3=O)=O)CC23CCC3)=O)C1 c1(C(N(CCNC(=O)Cc2ccccc2O)CC)=O)cc(Cl)c2ccncc2n1 C1(OC)CCC2(C(=O)NC3CC(C)N(C(=O)Cc4nnn(C(C)(C)C)n4)C3)CC12 Cc1cn2cc(C(=O)NCC3CCCN(C(c4ccc(C)s4)=O)C3)ccc2n1 N1(C(c2cc(CC)n(C)n2)=O)CC(C(=O)NCCN2CCC2)CC(C)C1 N1(C(Cc2ccn(C)n2)=O)CCC(COC2CN(C(C3CC3(F)Cl)=O)C2)CC1 N1(C(C(CC)OCC)=O)CCC2(CC(NC(=O)CCCc3sccc3C)C2)C1 C#CC1CN(C(=O)C(F)C(C)CNC(c2cc(CC)sn2)=O)CCO1 C12(NC(CCc3ccnc(C)n3)=O)CCC(C1)N(C(=O)CN(C)C(N)=O)C2 C1(NC(=O)C=Cc2ccccc2F)CC2CN(C(c3ccc(F)cn3)=O)CC2C1 c1(C(N2CC3C(CNC(C=C4CCC(C)C4)=O)C3C2)=O)cc2c(s1)CCCCC2 c1(C(=O)NC2C(OC)CN(C(COCCOC)=O)C2)[nH]c2ccc(F)cc2c1Cl c1(C(N2CC(OCCNC(C3CC3C3CCCO3)=O)C2)=O)ccnnc1 C1(CNC(CC(c2cccs2)NC(N)=O)=O)CCCCCN1C(c1cnsc1)=O C(C(O)C(F)(F)F)NC(CCNC(=O)Cn1cnnc1O)=O CCCCCCCCCC(C)CC(=O)NC1CCC1NC(c1cc(Cl)c[nH]1)=O CC1=CC(C)CN(C(=O)C(=O)NC2CC(C)(C)CN2Cc2ccccc2)C1 C(=O)(C1=CCC2CCC1N2C(=O)CCCC1CCC1)NCC1=NOC(C)C1 CC(C)CCC(=O)NCCCCCC1CCN(C(C2(C)CCCS2)=O)CC1 c1(C(N2CCCC(CCNC(CP(C)(C)=O)=O)CC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 N1(C(C2C(=C)C2)=O)CCC(C(=O)NCc2nc(C)no2)(C(C)C)C1 CCCCCCC(C)(CC)C(=O)NCC(C)N(C)C(c1cc(C)n(C(F)F)n1)=O C1(C(=O)NC)CCC(N(C)C)C1.C1(N2C(=O)COC2=O)(CO)CCC1 Cc1nnc2cc(NC3CCN(C(=O)C(N4C(=O)CCC4=O)C)CC3C)ncn12 C1(C(=O)NC(c2occ(C(=O)NCC(C3CC3)SC)n2)C)CCCCCC1 N1(CCOCCCC)CCC(=O)N(CCON(c2cccs2)C)C1=O C=C1CC2(C1)CN(C(C1N(C(C3CC(O)C(F)C3)=O)CCC1(C)C)=O)C2 Cc1cccc(C(N2CCCC2(C)CNC(c2cn(C)c(O)n2)=O)=O)c1N c1(OC(C)C)cccc(C(=O)NC2CCCC2NC(C2C3COCC23)=O)n1 N1(C(C(C#C)(C)C)=O)CCC(C)(CNC(=O)C(C)CS(C)=O)CC1 C1(C(N(C)CC2(CNC(=O)C3CC3)CC2)=O)CCN(c2nccs2)CC1 C1(C(=O)NC(c2nc[nH]n2)C)(SC)CN(C(C2CC2(C)C(F)F)=O)C1 C1(CC(=O)N(CC(C)(C)N(C)C)C)CC2(CC2)CN1C(C1CCOCC1(C)C)=O c1(C(=O)NCCC(CNC(C(CC)NC(C)=O)=O)O)cc(Cl)c(OC)c(Cl)n1 c1(CC(=O)Nc2nnc(CCN)s2)ccccc1[N+](=O)[O-] c1(C(=O)NC2C(NC(c3nccc(CC)c3)=O)CC2)ccc2c(c1)N(C)C(=O)C2 n1(CC)ncnc1CNC(=O)C=CC(C)NC(c1ccc(SC)o1)=O C1(C(=O)NC(CCC)CNC(c2nccnc2C)=O)CC2(CC2)CN1C C(=O)(C1=NN2CCC(C)N=C2N1)N(CC)CC1CCOC1 C1(C(N(CC(C)N(C(=O)Cc2ccnn2C)C)C)=O)CCCN(S(N)(=O)=O)C1 C1(F)(C(=O)NC2CC3(CN(C(c4cc(C)c(C)s4)=O)C3)C2)CC12CCCCC2 c1(C(c2cccs2)C)nc(C(C)C(C)OCCO)no1 N1(C(c2onc(C)c2C)=O)CCCN(C(=O)C(C)Cn2ccnc2)CC1C c1(C(=O)NC(C2CCCN2C(=O)C(C)(C)n2cccn2)(C)C)ccnnc1Cl C1(CNC(c2csc(Cl)c2)=O)(NC(C2CCC3CCC23)=O)CCCCC1 c1(C(C(N2CCCC(CCNC(CC(=C)Br)=O)C2)=O)=O)c(C)nn(C)c1C N1(CC)CCOC(C(=O)NC(c2cnn(C)c2)C(=O)Nc2ccccc2Cl)C1 S(=O)(=O)(C1CC(c2ccccc2)C1)N1C(c2nnc(C(=O)OC)s2)CCCC1 C1(CNC(c2ccc(C(C)=O)o2)=O)CC(NC(c2ncoc2C)=O)C1(C)C c1(CNC(CC2N(C(C3C(OC(C)(C)C)C3)=O)CCC2)=O)cnc(O)c(F)c1 C1(C(C)NC(c2cocc2C(N)=O)=O)CCCN(C(=O)C(c2cnn(C)c2)O)CC1 n1(CC(=O)NCCOCCOC)cc(CNC(=O)CC2CCS2(=O)=O)nn1 N1(C(C2C(F)(C(=O)OC)C2)=O)CC(NC(=O)C(N2CCC(C)CC2)=O)C(C)C1 C(=O)(CCC1=CCc2ccccc21)NCCCC1(NC(CC2CN(C)C2)=O)CC1 c1(OCC)nc(N(c2ncc(Cl)nc2Cl)CC2(F)CCCNC2)ncc1OCC C12(NC(CC(C)(C)C)=O)CCCC1N(C(C1CC3CCC1C3)=O)CCC2 c1(C(N(C(C)CNC(=O)CCCN(C)C)CC)=O)cccc2oc(C)nc12 C1(C(N2C3CN(C(c4c(N(C)C)cccn4)=O)CC2C3)=O)CCn2cncc2C1 C1(C)(C(=O)NCC(CNC(CCSCC)=O)(C)O)CCC(C)CC1 CC(C)C(C(=O)NCC1(NC(=O)COCC2CC2)CCCC1)c1cn(C)nn1 Cc1sc(O)nc1C(=O)NC(CNC(C1CC1C(C)(F)F)=O)C(C)(C)C c1(C(N2CCC(C(=O)Nc3nc(C)c(Cl)nc3)C2)=O)ccc2c(c1)CNC2=O CCC(C)C(CC(=O)N(C)Cc1ncco1)NC(C1(C)CCCC1O)=O C1(C(=O)NC2CCCCN(C(CCc3c(C)ncs3)=O)C2)CCCCC1C1CC1 C1(CCNC(C(CC)=CC)=O)CC(OC)CN1C(=O)CC1C(=O)ON=C1C N1(C(CCC2C(C)C2)=O)CCC2(NC(c3coc(C4CCCC4)n3)=O)CC2C1 C=CCCC(C(=O)NC(c1ncn(C)n1)C)NC(c1sc(F)cc1C)=O C(=O)(CCC(=O)NN(C)C)NCC1N(C(C(C)=C(CC)C)=O)CCCCC1 CCC(CC(=O)NCC1(O)CCN(C(=O)CCCCN(C)C(C)C)C1)C1CCC1 C1(C(=O)OC)CCC(C)N(CCc2ccc(Cl)c(Cl)c2)C1 C1(C(=O)Nc2ccc(NC(C)=O)cc2)CCN(C(=O)Nc2ccncn2)CC1O Cn1c(C(=O)NC2CCCC2NC(=O)C(O)CN2CCOCC2)nnc1S c1(C(=O)NC2CC3(CC(NC(CCN(C)C)=O)C3)C2)ccc(Cl)c2ccccc12 c1(C(N2C(Cn3cc(C(C)(C)N(C)C)nn3)C=CC2)=O)cccc(N)c1Br N1(C(C2(CC)CCCN(C(C(CC(=O)OCC)C)=O)C2)=O)CCC2CC1C(=O)O2 c1(C(=O)NC2(CNC(C3C(C4(C)COC4)C3)=O)CC2)cc(Cl)c(F)cc1O c1(NC(C2CCN(C(c3ccc(C)cc3Cl)=O)CC2)C)ncnc2c1cnn2C c1(C(N2CC(NC(=O)CC3CC3)CC(C)C2)=O)ccccc1S(=O)(=O)N(C)C c12cccnc1NC(=O)C2.c12cn(nn1)CCCC2.CSOC c1(C(=O)NC2CCC(NC(CS(CC)=O)=O)CC2)nnc(O)nc1O CCCC(O)CC(=O)N1CCC(CCOC)(NC(c2ccno2)=O)C1 C1(NC(C(C=C)(C)C)=O)CC2(C1)CC(CNC(=O)C(C(C)(C)C)C1CCC1)C2 C1(CNC(CSCC=C)=O)CC2(CCCO2)C1.C1(c2ccco2)C(=O)N1 c1(OC)ccc(C=CC(=O)NCC(C(C)(C)C)NC(=O)C(C)N2CCC2)cc1 C(C(CNC(C1(NC(=O)CC(C)SC)CC(O)C1)=O)C(C)C)OC C(=O)(C(O)CCSC)N1CCC(C(=O)NC(COC)(C)C2CC2)C1 CN1CCN(C(C2CCCSS2)=O)C(CNC(=O)C(C)(C)CC#N)C1 C=CC(C)(O)C(=O)N1CCC(C)(NC(=O)Cc2ccnnc2O)C1 CCS(=O)CC(=O)NCCCCC1CN(CC(=O)NC2CC(C)(C)C2)C1 c1(OC)cc(C(=O)N(CC(CC)NC(c2cc(C3CC3)no2)=O)CC)ccn1.CC C1(N(C(c2cc(C(C)=O)[nH]n2)=O)C)CCN(C(c2ccnc(N(C)C)n2)=O)CC1 c1(N2CCC(CNC(c3n(C)ccn3)=O)CC2)ccn2ncc(I)c2n1 C1(CNC(C(C)OCCOC)=O)CC(F)CN1C(c1oc(C(C)C)nc1C)=O N1(CC(N2C(C(C)C)C(=O)N(c3ccccc3)CC2)=O)Cc2ccccc2C1=O Cc1ccc(C(=O)NC2CCN(Cc3ncccc3C)C2)c2ccccc12 C(=O)(C(O)C(F)(F)F)N1C(C)(CNC(c2c(CC)nn[nH]2)=O)CCC1 N1(C(CNC(C(C)(C)C)=O)=O)CCCC(F)(C(=O)NC(C)(C)CC(N)=O)C1 c1(C(=O)NC(C(C(C)C)NC(=O)C=Cc2ccoc2)C)c2c(nn1C)CCSC2 N1(C(c2cn(C)c(=O)cc2)=O)CC2(CC(NC(C3(C)COCC3(F)F)=O)CO2)C1 Cc1noc(C)c1C(=O)NC1CN(c2cc(-c3ccccc3)ncn2)CC1F N12CC=C(CNC1=O)CC2.C(C(C)(F)CC(=O)NC(C)(C)C)N(C)C N1(C(C(C(C)C)(C)O)=O)CCCC(C2CCN(C(c3ncnn3C)=O)CC2)C1 C1(=O)N=C2N=CN(N2)CCC(=O)N1.CC1(CO)CC=CCO1 N1(C(C(CCN(C)C)O)=O)CCC2CCCC12C(=O)NCC1CCCOC1(C)C C1(O)(CC(=O)NC(C(C)NC(=O)Cn2nnnc2C2CC2)(C)C)CCCOC1 C1(C)(C(N2CCC(CCNC(C(C)n3ccnc3)=O)C2)=O)CCSCC1 C1(C(=O)NCC(CNC(CCSC)=O)(C)C)(COC)CCOCC1 C(=O)(C1CNC(=O)c2ccccc21)NC(C)CC(C)NC(=O)CSCC#N N1(C(Cn2cccc(C)c2=O)=O)CC2(CNC(=O)Cc3cc[nH]n3)CCC1CC2 N1(C(CC2CC(=O)NCC2)=O)CCCN(C(=O)Cc2csc(NC=O)n2)CC1 N1(C(C(CCC)=CCC)=O)CC2(C1)CN(C(=O)CC1CC3CCC1O3)CC2CO c1(COC(=O)CC2(CO)CCOC2)ccc(COC2CNCCO2)cc1 CCC(CC)(CO)C(=O)N(CCC(C)NC(=O)CC(C)NC(C1CCCC1)=O)C CC(C)(C)C(=O)C(=O)N1CC(NC(c2ccc(F)c(Cl)c2)=O)CC1CO C1(C(CNC(C2(OC)CCSC2)=O)C)CCN(C(=O)CCC(=O)N(C)C)CC1 N1(C(CCC#CC)=O)CC(C)(C)OCC1CNC(=O)Cc1ccc(C(C)=O)s1 C1(CCOC)CCCCN1C(C1CCCN(Cc2cnc(=N)[nH]c2)C1)=O c1(CC)cc(C(=O)N(CCNC(c2nocc2C)=O)C(C)C)cc(F)c1 C#Cc1cccc(C(N2CC(NC(C3CCCCN3C)=O)C(CC)C2)=O)c1F c1(C(N(C(C)C(=O)NCC2(CO)CC2(C)C)CCC)=O)cccn1C1CC1 c1(CC)cc(CN(C2CCCN(C(=O)C3CC3)C2)C(=O)C#CC(C)C)cc(O)n1 c1(NC(C(CC2CN(C(CCC3CC(OC)C3)=O)C2)F)=O)cnn2c1CCCC2 C1(NC(C2C(C)(C)C(NC(=O)C=Cc3nccs3)C2)=O)CCC2(CCCC2)C1 Cc1oc(C)c(C(=O)NC(C)CNC(C2CC(n3ccnn3)C2)=O)c1C c1(NC(CC2CCN(C(c3cc(C)oc3C)=O)CC2)=O)ccc(CO)cc1F c1(CCC)ccc(CC(=O)N(C(C)CCNC(c2nnc(S)n2C)=O)C)cc1 C(=O)(C(C)S(C)(=O)=O)N1CCC(CN(C(c2cnsc2C)=O)CC)CC1 Cc1nc(CNC(=O)CCCN(C)C(C2CC(=O)CCO2)=O)sc1C C1(CCNC(CC(=C=C)C)=O)CCN(C(c2nn(C)c(N)c2C)=O)C(C)C1 c1(CCC(=O)NCC(CC=C)NC(=O)Cc2cncc(C)c2)cc(F)cc(F)c1 CON(CCC(=O)NCC12CC(F)(C1)C2)C(=O)C1(C(F)(F)F)CC1 c1(COCC(N2CC(CN(C(=O)C(O)Cc3cnc[nH]3)C)C2)=O)cccc(Cl)c1 N1(C(C=Cc2cc(C)no2)=O)CCC(CNC(=O)C(C)n2cncn2)C1(C)C N1(C(C)C)CC(C(N2CC3C(C2)N3C(=O)Cc2ccc(Cl)s2)=O)CC1=O Cc1ccccc1CNC(=O)COc1cccc(CCN2CCCC2)c1 CC(C)C(C(C)NC(c1cc(Cl)sc1Cl)=O)NC(c1cc[nH]n1)=O C(CC(=O)NCC(CNC(=O)CCn1ccnn1)OC)(C(F)(F)F)OC C1(CCC(=O)N(CC(O)CO)C)CCN(C(=O)COC2CCC2)C1 C1(CC(=O)N(C(CC)C2CC2)C)CCCN1C(=O)CCc1ncnn1C CC(C)(C)C(CNC(C1CC(O)CN1C(C1CCC2(CCC2)C1)=O)=O)CO Cc1[nH]nc(C(=O)NCC2CCC(C)CN2C(=O)C2=CCCCO2)c1[N+](=O)[O-] c1(CC(=O)N(CC(C)NC(C2CC2CC(C)C)=O)CC)ccccc1Cl C=CC(C)(C)CC(=O)NCC(CCOC)NC(=O)CC1COC(C)(C)CO1 C(=O)(C(C)(C)NC(=O)CC1CCCO1)N(CC=C)CCO c1(OC)cc(NCC2CCCC(NC(C3(C)CCC3)=O)C2)nc(C(F)(F)F)n1 CC(C)C(C)C(=O)NCCN(C(=O)C(C)(C)C1CCCCO1)Cc1ccccc1 C1(F)(CNC(C(=O)NC(c2nc(C)[nH]n2)C)=O)CCCOC1 CC1CCCCCN1C(c1cc(Br)cs1)C(=O)NCC(F)F N1(C(COCCC(C)C)=O)C(C(N2CC(C)(F)C2)=O)CC1C c1(C(N2CCC(NC(=O)Cn3nccn3)C(F)C2)=O)cc([N+](=O)[O-])ccc1Cl C1(NCc2onc(C(C)(F)F)n2)CCCC(C(=O)O)CC1 c1(C(=O)NC(C(c2ccccc2)NC(C2(COC)CC2)=O)C)sc(CO)nc1C N1(C(CC(C=C)C)=O)CCN(C(c2ccn(CCC(F)(F)F)n2)=O)CC1CF CCC(CC)(CC)C(=O)N1CCC(O)(CCCNC(=O)CN(C)C(C)C)C1 C1(OC)CCC(C(N2CC(CNC(=O)C(=O)NCC(F)(F)F)C2)=O)C1 N1(C(C(c2nccc(C)c2)(F)F)=O)CCC(CNC(=O)C=CC(C)C)C(F)(F)C1 c1(NC(C=CC=CC)=O)ccc(CC(=O)OCC)cc1.N12CC(C1)C2=O CC1CCC=C1C(=O)N1CCN(C)C(C(=O)Nc2cnccc2C2CC2)C1 Cc1cnc(C(=O)NCC2CC(NC(C3CC34CCC4)=O)C(O)C2)nc1 c1(CN2CC(NC(=O)Cc3scnc3-c3ccccc3)C2)cnc2n1CCOC2 Cc1ncnc(C)c1C(=O)N(C1CCN(C(=O)CCOC2CC2)C1)CCO N1(C(C(C)SC(C)C)=O)CCC2(CC1)CC(CNC(=O)C1=CCCC1C)C2 c1(CN2CC(Nc3c(OC)ccc(F)n3)CC(C(=O)O)C2)c(Cl)cc(O)cc1Cl Cc1cc(NC(=O)CC2CN(C(c3ncccn3)=O)CC2C)c(C)cc1F c1(SC(CO)Cc2cccs2)cccc(SC(F)(F)F)c1 C(CCCCC(=O)N1CC(F)CC1CNC(c1cnc(C2OCCO2)s1)=O)SC c1(CCC(=O)NC2CCCN(C(c3cccc(Cl)c3)=O)C2)ccc(O)nc1 C1(C(=O)NC2CN(C(CCC(=O)NC)=O)CC2C)CCc2nnnn2CC1 CC1(NC(c2cnc(-c3ccco3)s2)=O)CCN(C(=O)CNC=O)CC1 CC12CCC(C(N3C4CC3CN(C(c3ccc(C5CC5)cc3)=O)C4)=O)(CC1)CO2 c1(N2CCC(C=C)(CO)CC2)nc(=NCCCCS(C)=O)[nH]c2cc(C)ccc12 C=C(C)CC(C(=O)N1CC(C(=O)N(C2CC3CC3C2)C)CC(C)C1)OC c1(N(C)CC2N(C(=O)C=CC(N3CCCCC3)=O)CCC2)ncnc2scnc12 N1(C(CN(CCC)C)=O)CCN(C)CC1CNC(=O)CC1CCC1(C)C c1(C(N2CC(CN(C(c3occ(C)c3)=O)C)OCC2)=O)ccc(Cl)c(F)c1N S(=O)(=O)(c1ccc(NCc2ccns2)cc1Cl)N(CC1=CCSC1)C N1(CCc2ccc(C)cc2)C2CCCC1CC(NC(c1cc(Br)cc(Br)c1)=O)C2 c1(C(N)=O)ncc(C(=O)CN2CCCC2CCC(=O)OC(C)(C)C)s1 C1(CC(N2CCC(CCOC)(NC(C3CCC3C)=O)C2)=O)OCCCC1(C)C c1(C(N2CC(CNC(CC3N(C)C(=O)CC3)=O)OCC2)=O)c(O)ccc(Cl)c1F Cc1cc(CO)ccc1NC(C1CC(C)N1C(c1ccc(N)c(F)n1)=O)=O C(CN=C(NC1CC1C1CCCC(C2CC2)O1)N1CCC(O)C1)OC(C)(C)C C1(C(=O)NCC(CC)NC(=O)C(C)NC(c2ccoc2)=O)CC(=O)N(C(C)C)C1 n1(C(C)C)c(O)nc(N2CCCC2CCNC(C23CCCC(CO2)C3)=O)cc1=O C1(C(=O)NCCCCCCn2cc(C(CC)(C)O)nn2)CN2CCCN1CC2 C(=O)(CCCCC(N)=O)N1CCCC(CNC(C(c2ccccc2F)C)=O)CC1 C(=O)(C(F)CCC(C)C)N1CC(C(C(N2CCC(C)(COC)C2)=O)O)C1 c1(C(c2n(C(CC)C)nnn2)NCCC(CO)CO)cc(C(C)C)nn1C c1(C(=O)NCC#CCNC(C2C(CC)CCCC2)=O)cc2cc(OC)cnc2[nH]1 c1(C(=O)NCC2(NC(C3CC4CC(OC)C4C3)=O)CC2)ccnc2c1ncn2C CC1CN(C(=O)Cc2ccc(Cl)c(Cl)c2)CCCN1C(=O)C1=CC(O)CCC1 C1(C(=O)NCCC(=O)Nc2ccc(F)cc2Br)CC2CCCCN2C1 C1(NC(c2cnc(C(C)=O)s2)=O)CCCC(NC(C2CCCC2)=O)CC1 C(N=c1[nH]cnc(Cl)c1F)C1CCN(C(=O)Cc2cccc(C3CC3)c2)C1 N1(C(CC=C)=O)CCC(OCCNC(=O)CCC2CC2(Cl)Cl)CC1 c1(COC)ncc(C(=O)OC2CCCC(N(C)C)C2)c(C(F)F)n1 N1(C(C)C)CCC(C(N2CCCC(N(C)CC3CCC(F)(F)C3)C2)=O)CC1 N1(C(C2C(C=C)CC2)=O)C2CCCC1CN(C(=O)C(c1ccc(F)cc1)F)C2 C1(CC(=O)NCCC2CN(C(c3cnc(S)n3C)=O)C2)Cc2ccccc2O1 c1(CC2(C(=O)NCC(C)(C)CNC(=O)C(O)CC3CCCC3)CC2)ccc(Cl)cc1 N1(C(=O)C2=CCCC2)CCC2(CC1)CC2(CO)CNC(=O)COC1CC1 n1(CC(N2C(CNC(C(c3ccc(N)cn3)C)=O)CC2)=O)ncc2ncccc12 CCCCCCCC(F)C(=O)NC(C1CCN(C(=O)Cn2cnnc2O)CC1)C C=C=CCCC(=O)N1CC(CC(=O)NCC2(CC(C)C)CC2)C(C)C1 N1(C(C(=O)NC2CCOC2)C2CCSC2)CCCCC1c1cn[nH]c1 C1(C(N(CC(C)(C)O)CCC)=O)CC(CC)CCN1C(=O)C(C)CC(F)F C1(C2CCN(C(C3(N(C)C)CC3)=O)CC2)(NC(C2C(C)=C2)=O)CC1 C1(C(=O)NCc2n(C)ncn2)C2CC(O)C(C2)N1C(C12CCC(C1)C2(C)C)=O CCC(C)CC(C)C(=O)N1CC(CCCCNC(C2(O)CCOCC2)=O)C1 CCCCC(C)(F)C(=O)N(C)CCOCCC(=O)NCc1cccc(F)c1F C(=O)(C(C)CNC(C1(C(C)C)CC1)=O)N(C)CC c1(C(=O)NCCC(=O)NC(C)C)ccc(C(C)(C)C)nc1O C1(O)(C(C)CNC(c2ccc[nH]2)=O)CCN(C(=O)C(C2(O)CCOCC2)(F)F)C1 C1(C(=O)NCCc2ccc(C)cc2)CC(C)CCN1C(=O)CSC(F)F C1(CCC)(C(=O)NCC2COCCN2C(c2ccsn2)=O)CCNC1=O C(=O)(CCC(CC)CCC)N1CCC(C#C)(C(=O)NCC2CC(C(C)C)C2)CC1 c1(NC)cnc(Cl)cc1C(=O)NCCNC(=O)CCOc1ccccc1Br C1(C(N(C(C)C)CCNC(C2CC(O)C2)=O)=O)CCCC(=O)N1 CC(C)C1=NOC(C(N2CCCC(NC(c3cccnc3C(F)F)=O)C2)=O)C1 N1(C(=O)NC)CCN(C(C23CC(CO)(C2)C3)=O)CC1.C12CN(CCO1)C2=O C(=O)(C(C)CCCOC)NC(CC)(C)CNC(=O)C=Cc1ccsc1Br C1(NC(C)=O)CC(C)CN(C(=O)CNC(c2ccc(F)c(F)c2)=O)C1 N1(C(c2cc(C(=O)O)cc3c2cc[nH]3)=O)CCC(CO)C12CCOCC2 c1(C(=O)NC2CCC(CCNC(c3scc(C(C)=O)c3)=O)C2)nc(=O)n(C)[nH]1 N1(C(C(=O)NC2(C=C)CCOCC2)=O)CCC(C2CCC2)C1 C12(C(=O)NCCC(=O)NCC)CC(CN1C(=O)C(C(=O)OC)OC)C2 C1(N(C(=O)CCCC2CCOCC2)C)CCN(C(=O)CN2CC(=O)NC2=O)CC1 CCCCCC=CC=CC(N1CCC(NC(c2ccsc2Br)=O)C1)=O c1(CC)snc(C)c1C(=O)NC1CC(CO)N(C(=O)CCNC(=O)NC)C1 C1(C(N2C(C3(C)COC3)CCC2)=O)CCCC2(CCN(C(=O)OC(C)(C)C)C2)O1 n1(CC(=O)NC2C(CNC(CC(C)CN(C)C)=O)CC2)cc(F)ccc1=O CS(=O)(=O)c1csc(CNC(c2nc(C(F)(F)F)cs2)c2nnnn2CC2CC2)c1 C1(C(N(CC(CCC)O)C)=O)CCN(C(C2CC(OC)(OC)C2)=O)C12CC2 C1(CC(C)C)CCCCN1C(C1C=CCN(C(=O)C(F)F)C1)=O CCN(CC(C)Nc1cc(Cl)ccc1O)N1CCN(C(=O)OC(C)(C)C)CC1 c1(-c2ccn(C)c(=O)c2)ccc2c(C(=O)NCc3ncc(Br)s3)nsc2c1 C(=O)(C1COc2ccccc21)N1C2CC(CNC(C34CC(F)(C3)C4)=O)C1CC2 CCCCCCCCCCCn1nc(CCC2CCCC2)nc1-c1c[nH]cc1C c1(C(CO)NCc2nc(-c3cccc(F)c3)no2)ccc(F)cc1 n1(CC)ncnc1C(=O)NCC1C=CC(NC(=O)C(O)C2CCCC2)C1 c1(N(C)CC2CCN(C(=O)CC3CCCCN3C)C2)ccnc(Cl)n1 c1(C(=O)NCC2CN(C(C3(CC=C)COC3)=O)C2)ccc(Cl)nc1OC1CCC1 CC1CN(CC(=O)N(c2ccccc2)Cc2cccs2)Cc2c[nH]nc21 CC(C(=O)N1CCC(CC(=O)NC(C)(C)C(C)(C)O)C1)C(C)(C)C c1(C(=O)NCC2(CNC(C(CCSC)O)=O)CCCC2)nsc2ccc(C)cc12 C1(C(=O)NCC2CCC(C(=O)NC3(C=C)CCC3)CC2)CCOC(C)(C)C1 CCC(C)CCCC(=O)NC(CNC(=O)CNS(=O)(=O)CC)C(C)C c1(CNC(C23CCC(OC)C2CC3)=O)ccc(O)c(F)c1F C(N=c1[nH]c2c(c(=NC3CCC4CC4CC3)[nH]1)CCC2)c1nn(C)c(Br)n1 C(=O)(N1CCC(C(=O)NC2(CCF)CCC2)O1)C1C(OCC)CC1 N1(C(C2(SC)CCC2)=O)CC2CCCC(NC(c3ccn4ccccc34)=O)C2C1 N1(C(C(C(C)NC(COCC#C)=O)C)=O)CCC(C)(CO)CC1 CC(C)(C)CC(O)C(=O)NC1CCN(C(c2occ3c2CCC3)=O)C1C(C)(C)C C1(CN(C(C2C(CC)CCO2)=O)CC)CCN(C(=O)C2=C(C)CC2)CC1 c1(C(=O)NC2CCN(C(C3COCC4(CCC4)O3)=O)C2)c[nH]c2cccc(F)c12 C1(NC(CC2(COC)CCC2)=O)CCCC1C(C)(C)C.c12c[nH]nc1CNC2=O Cn1c(C(N2CC(NC(=O)C=CC3CCCO3)C(O)C2)=O)cc2cc(Cl)ccc12 C(=O)(CCCCCCC(=O)NCC(C)NC(C1CC(=O)N(C(C)(C)C)C1)=O)OC N1(C(=O)NC2C(C)OCC2)C2C=C(c3cccs3)CC1CC2 C(=O)(C#CC1CCOCC1)N1CCC(C(=O)NCC2CCOC2C2CC2)(CC)C1 c1(C(N(CCN(C(C)C)C(C2CCC(C)O2)=O)C)=O)ccccc1-c1ncc[nH]1 c1(C(N2CCSC(C(N3CCC34CCCCC4)=O)C2)=O)sc(Br)c2c1OCCO2 C1(C(=O)OC)CCC(C(=O)O)(NC(=O)Cn2cc(-c3ccc(C)cc3)nn2)CC1 CC(C)(C)CC(=O)NCCCN(C(=O)CCc1cccc(O)n1)CCO N1(C(CC(C)SC)=O)CC(CNC(C2(Oc3ccccc3)CC2)=O)CC1(C)C c1(CCNC(=O)NCCC2CC2(F)F)cccc(O)c1 CCC(CC)(CO)C(=O)NCC1CN(C(C2CCOC(=O)CC2)=O)CC1(F)F Cc1c(C(=O)NC2CN(C(=O)CCN3CCCCC3)C2)cno1 c1(C(=O)NCCN(C(C=C(CC)C)=O)CC(C)O)cccc(C(C)(C)C)c1 Cc1ncc(NC(=O)C(C2CC2)N(C(=O)C(O)C2CCC2)C)cc1C#N N1(C(C2C(CC)C(=O)C2)=O)CCOC(c2cccc(Cl)c2)C1 C1(NC(C23N(C(C(C(C)C)F)=O)CC(C2)C3)=O)CC(C)N(C)CC1C c1(CC)cc(=NC(=O)C2(CNC(=O)COC3CCOC3)CC=CC2)[nH]n1C c12ccc(cc1)o2.C1(C(=O)NCC=CCNC(C2C(OCC)C2)=O)(CC)CCC1 Cc1cc(Br)cnc1C(=O)NC(C1(O)CN(C(=O)C(C#N)C(C)C)C1)C N1(C(CCCC=C)=O)CC(NC(=O)CCC2CCCC(=O)N2)CC12CCCC2 C1(C(=O)NC2CC(C)(C(=O)OC)C2)CCN(C(C2CCCC2O)=O)C1(C)C CN(C)S(=O)(=O)NCC(=O)NCCC1CN(C(C2CCC=CCC2)=O)C1 c1(CN)ccc2ccc(C(N3CCN(C)C(CO)C3)=O)nc2c1 c1(C(=O)NC2(CCNC(CC(n3c(CC)ncc3)C)=O)CCC2)[nH]c(C)cc1C Cc1cc(Cl)cc([N+](=O)[O-])c1C(=O)N(CC(C)NC(c1cc(N)cc(F)c1)=O)C c1(-n2cc(C(C)(C)OC)nn2)ccc2c(c1)CCN(C(=O)C(C)(C)CF)C2 c1(SC)cccnc1C(=O)NCC1CC(NC(c2nn(C(C)(C)C)cc2Cl)=O)C1 n1(CC)ncnc1CN1CCC(CC(=O)N(CCC(C)(C)O)COC)C1 n1(CC(=O)NC(C(C)NC(c2cc(Cl)sc2Cl)=O)C)[nH]cc2c(=O)ncnc1-2 N1(C(c2cccc(NC(=O)OC)c2)=O)CCN(C(=O)C=CS(C)=O)C2CCC12 Cc1cccc(C)c1CNC(=O)C(=O)Nc1ncc(C(F)(F)F)cc1Cl c1(NC(CC)=O)ccc(C)c(NC(=O)NC(C)CN2CCOC2=O)c1 Cc1cc(C(=O)NC(c2ccnn2C)C(=O)NCc2ncc[nH]2)cnn1 C1(OCC)(CNC(=O)CNC(=O)C(C)C2CC2)CN(C)C1 C1(NC(=O)CCc2cncnc2O)CS(=O)(=O)CC1NC(c1cc(CO)[nH]n1)=O c1(C(N2C(CNC(=O)CN3CCCC3)C=CC2)=O)cc(Cl)c(Cl)cc1O c1(OC)ccc(S(=O)(=O)N2CC34CCCC3(CNC4)C2)cc1C(C)C c1(OC)cccc(Cl)c1CNC(C1CCCC1COC(=O)Nc1ccncn1)=O c1(C(N2CC(N3CCN(C(=O)CC4COCCO4)CC3)C2)=O)c[nH]cc(Cl)c1=O N#Cc1cccc(CC(=O)NC2CC(C(=O)O)C2)c1 C12(C(=O)NCC3CCN(CCC)C3)CC(CN1C(=O)Cc1cnn(C)c1)C2 c1(C(C)NC(=O)CO)cn(CC(N2CCCC2C2CCCOC2)=O)nn1.CCO N1(C(CC2C(C)OCC2)=O)CC2CCC(C1)N2C(=O)CC(C)(F)F c1(OCC)ccc(NC(=O)C(C)OC(=O)Cn2c(C)csc2=O)cc1 C1(C)(NC(c2ncc(NC)nc2)=O)CCCCC1C(=O)NCC#CCCO c1(NC(CC2CCCN(C(C#CC(=O)O)=O)C2)=O)cc2ccccc2cn1 c1(OC)ccc(C(=O)N(CCN(C)C(c2cn(C)nc2Cl)=O)C(C)C)nc1 CC1CCN(CCC(C)N(C(c2ccc(CN3CCCC3)o2)=O)C2CC2)CC1 c1(SCC(N2C3(CNC(c4c(C)nco4)=O)CC(C2)C3)=O)cc(F)cc(F)c1 N1(C(C2C(C(C)C)CCO2)=O)CC(C(=O)NC(CO)C(C)(C)C)C(F)(F)C1 c1(C(=O)NCC(CC)NC(=O)CC2CNC(=O)O2)ccc(=N)[nH]n1 c1(-c2ccn(C)n2)nc(C2CCN(C3CCOCC3)C2)n(CCCO)n1 S(=O)(=O)(c1cccnc1NCC1(C)COC(C)(C)C1)NCCCC(COC)(C)C N1(C(c2cnc(C3CC3)o2)=O)CCCCCC1CNC(C1(C(F)F)CC1)=O C1(Cc2cn(CC(C)NC(c3c(CC)nco3)=O)nn2)CCCCCC1 CC(CCc1cccc(F)c1)C(=O)NCC(C)(CO)NC(c1nc(=N)cc[nH]1)=O c1(C(=O)NC(CNC(C2(c3ccon3)CCC2)=O)CO)cc2ccccc2o1 C(C(C)C(C)(c1nnnn1C1CCOCC1)NCc1sc(Cl)cc1Br)OC N1(C(C2CCCC(OC)C2)=O)CCCC(F)(CNC(=O)C=CC(F)(F)F)CC1 O=C1CCCC(C(N2CCC(OCCNC(c3cccc(O)n3)=O)C2)=O)N1 Cc1cn2cc(C(=O)NCC3C(C)CCCN3C(=O)CCc3cnc[nH]3)nc2s1 N1(C(c2c(C)onc2)=O)CCN(C(=O)CC2CC2(Cl)Cl)CC(O)C1 N1(C(c2ncn(CC)c2)=O)CCC(C(=O)NCCCCC(C)(F)F)C(C)C1 c1(CCC)cc(C(=O)NCC2CC(O)CN2C(=O)C(C)C(F)F)c(C)o1 C1(CNC(C2N(CCC)CCC2)=O)CCCCN(C(=O)CCC2(C)CC2)CC1 C(=O)(C#CC1CCOC1)N(CCC(C)NC(c1ncc(C(N)=O)cc1Cl)=O)C C1(C)(C(=O)NCC2CN(C(c3[nH]cc(CC)c3)=O)CC2O)CC(C(C)(C)C)=NO1 N1(C(c2ccon2)=O)CCN(C(c2ccc(F)cc2F)=O)C(C2CCCC2)C1 c1(C(=O)NCCNC(=O)CC2CCCCO2)ccc(NC2CCCCC2)nc1 c1(C(=O)NCCC(C)NC(c2ccc(N)c(N)n2)=O)cnc2c(c1)CCCO2 c1(C(=O)NC2CCC(CC(=O)N(CCCC(=O)OC)C)C2)nc(C)c(C)s1 C1(C)(CNC(C2C(C)C2)=O)CN(C(c2ccc(F)cc2Br)=O)CCO1 N1(C(CSc2n(C(C)C)cnn2)=O)CC(CNC(=O)Cc2cc[nH]n2)C2CC12 CS(=O)c1ccccc1C(=O)NCCNC(=O)COC1CCN(S(C)(=O)=O)CC1 C1(NC(COCC)=O)CN(C(c2[nH]nc(C(F)(F)F)c2C)=O)CC(F)(F)C1 CN1CCC(C)(C(N2CC(O)(C(F)C(=O)NC3CCC4(C(N)=O)CC34)C2)=O)C1 CCCCCC(O)CC(=O)N1CCC(CC(N2CC(O)(C3CC3)C2)=O)CC1 c1(C(=O)NCC23C(CN(C(CC(C)SC)=O)C2)CC3)[nH]c2ccccc2c1C CCC(C)(CNC(=O)CCCOCc1ccccc1)NC(=O)CSc1cccs1 Cc1ccccc1C(=O)NC1(C(=O)NCc2cccc(Cl)n2)CCN(C)C1 CC(C)C(C)(C)C(=O)NC1C2CCC(C2)C1C(=O)NCc1c(F)cncc1F C1(C(=O)OCc2ccc(OC)nc2)CN(C)CCN1C(=O)CCOC(C)C C1(NC(c2cc(C)sc2C)=O)CC(F)CN(C(C2(C#N)CC3CC3C2)=O)C1 C(C(O)CCC(=O)OC(C)(C)C)NC(C1(NC(C(C)n2cccn2)=O)CC1)=O Cc1cc(C(N2CC(NCc3ccc(O)c(Cl)c3)CC(C)C2)=O)cnc1F C1(CNC(Cc2cc(C)on2)=O)CC2(CCN(C(=O)C=CCF)CC2)CO1 C1(CNC(COCCCCCC)=O)CCCN(C(C2CCC3CC3CC2)=O)CC1 N1(C(C(C(C)(C)C)O)=O)CCC2OCCN(C(c3cc(C(F)(F)F)on3)=O)C2C1 c1(C(=O)NC(C2(O)CCN(C(C3(C(F)F)CCCC3)=O)C2)C)cccc(Cl)c1F c1(CNC(COCCCOC)=O)cccc(CNC(c2ccc(Cl)o2)=O)c1 N1(C(C(C2CCOC2)NC(CC)=O)=O)CC(C)OC(C)(C)C1C N1(C(C(OC)OC)=O)CCC2CN(C(=O)CCCc3cncs3)CC12 c1(OC(C)C(=O)N(C(CNC(c2ccc(Br)o2)=O)C2CC2)C)ccccc1 c1(CC)ccc(F)cc1C(=O)NCC(C1CC1)N(C)C(c1ocnc1C(F)F)=O C=Cc1cncc(C(=O)NC(CN(C)C(C2CCN2CC)=O)(CO)CO)c1 Cc1oc(C)c(C(=O)NCCOCCCNC(=O)C(F)OC(F)(F)F)c1Br c1(C(=O)NCCOC2CN(C(c3c(C)cc(F)s3)=O)C2)cn2cccc(C)c2n1 C1(c2n(C)ncc2)CCCC1CN(C(C)(C)CC1CCOC1)CC1CC1 C=CCC(C(=O)N(C(CO)C1CC1)C)NC(C1CC2(CCC2)C1)=O C(N=c1[nH]cc2ncnc-2[nH]1)C1N(C2CCCN(C)C2=O)CCC1 C#Cc1ccc(CNC(=O)C(C)NC(=O)CC2CCOC2=O)cc1 N(C(=NCCC1(C)CC1(Cl)Cl)NC1CCCCC1)CC(C)(F)F c1(C(=O)NC(C2CCN(C(C(C)c3ccsc3)=O)CC2)C)nccc(N)c1Cl N1(C(C2(COC)CCCC2)=O)CCOCC(NC(C23CCCC2C3(F)F)=O)C1 C1(C)(C(N(C(C)C(=O)NC(C)C(=O)NO)CCC)=O)CC(F)C1 C1(OC)CN(C(c2ccc(C)s2)=O)CC1NC(c1nc(C)oc1C)=O C(c1nc2ccccc2o1)=CC(=O)NCC1CCCC(NC(=O)CC2(O)CC2)C1 C(C(C)(C)CC1CN(C(=O)CCC2CCCCO2)C1)NC(C(F)NS(C)(=O)=O)=O N1(C(C(c2ccccc2F)C)=O)CC2(C1)CN(C(=O)CN1CCCCCC1=O)C2 C1(NC(Cc2cc(C)on2)=O)CC2(NC(c3coc(C)n3)=O)COC1C2 c1(C2(C(N(CCNC(C3C(C)CCS3)=O)CC3CC3)=O)CC2)ccccc1F N1(C(c2c(C)nc(C)o2)=O)CC2C3CCC(C2C1)N(C(=O)C1=CCCC1(C)C)C3 Cn1cc(C(=O)N(CCNC(C2(c3ncccn3)CC2)=O)CCOCCO)nn1 C1(NC(CCc2c(C)nn(C)c2)=O)CCN(C(=O)Cn2cnc(=N)[nH]2)CC1O N1(C(C(C)S)=O)CCC(O)(CNC(c2cc(O)ccc2Cl)=O)CC1 c1(C(=O)NC)cccc(C(c2nnnn2C2CC2)NCCC2CC2)c1 C(C(C)(C)C(C)(C)C)NC(C1C(CNC(CCCCOCC)=O)C1(C)C)=O c1(CCCC(N2CC(O)(C(C)NC(C3CC3C)=O)C2)=O)ccc(Br)cc1 C1(C(C)C)(CO)CCN(C(=O)CC(C)NC(c2cnsn2)=O)C1 CC(CCCC(=O)NC1CCC(C(C)O)CC1)NC(c1cnn(CCO)c1)=O N1(C(=O)CC2CCCC2)CCC2CN(C(=O)C(c3ccccc3F)F)C2C1 N1(C(c2c(C)nn(C)n2)=O)CCN(C(C2COCCN2C)=O)C(CCO)C1 CCCCC(O)CC(=O)N1CC2CC2(CNC(=O)CCC(=O)N(C)C)C1 C(CC(C)C)(C(=O)NCC1CCCCCN1C(c1ccncc1F)=O)NC(C)=O c1(C(=O)NC2C(NC(c3cc(I)ccc3F)=O)C2)ccc(-n2cccn2)c(Cl)c1 C1(C(=O)NC23CN(C(c4n(C)cnc4)=O)C(C2)C3)CCOC2(CCCCC2)C1 c1(OCC=C)ccc(Cl)c(C(=O)NCCNC(C2(c3cccs3)CC2C)=O)n1 c1(CC)c(C(N2CCCC2C2(NC(=O)Cn3cc(C)cn3)CC2)=O)cccc1C CN1CC(C(=O)NCC(N2CC(CN=[N+]=[N-])C2)=O)CC1=O C=C(Cl)C(C)(C)C(=O)NC1COCC1CNC(c1cnn(C(F)(F)F)c1)=O C#CCCN=C(NCc1nccc(Cl)c1F)NC1CC(OCC)C1 c1(CCCCC(=O)NC(C)=O)ccc(OCc2ccccn2)c(OC)c1 N1(C(C(C)OC)=O)CC2CCC(CNC(=O)C(F)C3CCCC3)C2C1 C(=O)(C1=C(Cl)CCCC1)N1CC(O)(C(C(=O)NCC2(CC)CCCC2)F)C1 N1(C(CC2(C=C)CC2)=O)CCC(C2CC2)(CNC(c2ocnc2C)=O)C1 Cc1cnc(C=CC(=O)N(CC(C)NC(C2CCCOC2C)=O)C)[nH]1 N1(C(CCCC#C)=O)CCN(C(=O)C(N2CCOCC2=O)C)CC1c1cn[nH]c1 C1(C(=O)NCCN(C(c2[nH]cc(CC(C)C)c2)=O)C)CCCCN1C1CCCC1 Cc1cc(=NCC2COC(C)C2)c(F)c[nH]1 Nc1c(CN2CCOC(c3cccc(C(F)(F)F)c3)C2)cnn1C1CCOCC1 c1(N(C(C(CSC)(C)C)=O)C(C)CCCC2CCCCC2(C)C)ncnc2c1CCC2 N1(C(CC(C)OC)=O)CCCC(NC(c2cccc(OC(C)C)c2)=O)C1C N(C(=NCc1ccc(OCCO)cc1)NCCF)CC1CN(S(C)(=O)=O)C1 Cc1cc(CN2CCC(F)(CNC(c3cc(I)ccc3O)=O)CC2)c(F)cc1Br c1(C(N(CCCC(=O)NC(C)Cc2cccnc2)C)=O)ccc(F)nc1 CC(O)C(F)(F)C(=O)N1CCCC(N(C(=O)Cc2ccsc2Cl)C)C1 C1(CNC(C(C)(O)Cc2ccccc2)=O)CC2CCC1N2C(C1CC2(CC2)C1)=O c1(NC(C2CCN(C(C(F)=CCC)=O)C2)C)nc(C)ccc1C(=O)OC(C)C C(=O)(C1=CCOCC1)N(CC(N1CCCC(COCC)C1)=O)CC c1(C(N2CC(CNC(=O)CC3CC(F)(F)C3)C(O)C2)=O)cc2cc(F)ccc2[nH]1 C1(C(=O)NC2CCC(NC(c3c(C(C)C)ncs3)=O)C2)CC2(CCC2)CO1 C=CCCN=C(NCC1CC(COC)C1)NCC1C=CCCCC1 N1(C(C=CC(CC)C)=O)CCC(CF)(NC(=O)COC(C)=O)C1 O=S(=O)(c1cnccc1F)N1CCCC(c2ccccn2)C1 c1(OC)ccc(F)cc1C(=O)N(C1CCN(C(=O)C(O)C2CCCC2)C1)CCO C12(C(=O)NC(C)(C)CCNC(C3CC=CCC3)=O)CCC(CC1)C2 C1(C(=O)NCC2C(OC)CCC2)CN(C(=O)CSC(F)F)CCC1(C)C C=CCCCC(C(=O)N(C(C)C(F)F)C)NC(=O)CCc1cscn1 CC1OC2(CNC(=O)CC3CC4C=CC3C4)CC1(NC(=O)Cc1cccnc1)C2 CC1=CCN(C(=O)C(c2ccccc2)NC(=O)C(C)N2CCCC2)C1 C1(C(=O)NC2CC(C(=O)NCCCCOC)C2)CCCOC1 Cc1cc(CCCC(=O)N(C(C)CNC(=O)C(C)Cc2ccncc2)C)c(C)s1 C1(C)C(C)(C)OC(=O)COCCCN1CC(=O)NCC.CCCSC c1(C(N(C2CCC(NC(CS(CC)(=O)=O)=O)CC2)C)=O)cccn2c(O)nnc12 c1(OCC)cnc(N2CCN(C(c3nc(C)cs3)C(=O)NC(C)CC)CC2)nc1 N1(C(CN(C)CC)=O)CCC2CC(NC(c3cnco3)=O)CCC2C1 N1(C(c2ccc(SC)cc2)=O)CCN(C(=O)CCc2ccc(C)o2)C2CCCC12 n1(CC)nc(C)c(C(=O)NCC2C3CN(C(C4(C)CC4Br)=O)CC23)c1Cl C1(NC(CC(C(C)C)OCC)=O)CN(C(=O)C(COC)COC)CC(C)(C)C1 c1(C2(NC(c3n(CC#C)ccc3)c3nnnn3C3CC3)CC2)ccc(Cl)c(C)c1 C1(NC(c2cccc(C(C)(C)C)c2)=O)CC(F)CN(C(C2CC2(C)C)=O)C1 N1(CC)N=C(C(=O)NC2CCCC(CC(=O)N(CC(C)(C)SC)C)C2)CCC1=O c1(C(N(CC(CNC(CN(CCC#C)C)=O)C)C)=O)cc(OC)c(C2CC2)nn1 N1(C(C2C(C=C(C)C)C2(C)C)=O)C2CCCC1CN(C(=O)C=C(C)C)C2 c1(C(=O)NC(C)CNC(C2CC(C)C2)=O)cc2n(n1)CC(F)C2 N1(C(CCS(=O)(=O)N(C)C)=O)CCC(NC(=O)CC2=CCCC2)C(CO)CC1 C(=O)(CC(CCC)CCC)NCC(CNC(c1cn(CCCC)nc1C)=O)F c1(C(=O)NC(C2CCN(C(c3cc(C)nn3C3CC3)=O)C2)C)cnc(N)c(N)c1 N1(Cc2c(OC)cco2)CCN(C(=O)C=CC2CC2)C(C)C1 C(CNC(C1CCN(C)C(=O)C1)=O)(C(=O)NOCCCF)OC N1(C(c2csnc2C)C(=O)NCCCOC)CC(C)OC(C)(C(F)F)C1 C1(C(N(CCCNC(c2cc(CC(C)C)on2)=O)CC)=O)CCC(C)=C(C)C1 C=C=CCCC(=O)NCc1c[nH]nc1C1CCN(C(C2CCCN2CCC)=O)C1 c1(CC(=O)NCC=CCNC(C=Cc2n(CC)ncc2)=O)csc2ccccc12 c1(C(=O)NCCC2CCN(C(c3ccc(C(C)=O)[nH]3)=O)C2)sc(F)cc1Cl c1(NC2CN(C(C3(CC)CC3)=O)CC2C)cc(C)c([N+](=O)[O-])cc1Br N1(C(C=CCC2(NC(C(CCCC#C)C)=O)CCC2)=O)CC23CCC2(COC3)C1 N1(C(C(C(=O)OC)(C)C)=O)CC2CCOC(=O)C2C1.C12C3CN(CC13)CC2 C1(NC(CN(C(=O)OCC)C)=O)CC2CC1CN(C(c1cn(C)c(C)n1)=O)C2 N1(C(C2(SC)CCC2)=O)CC(NC(C2CNC(=O)N2C)=O)CC(C)(C)C1 C(=O)(C(F)(F)C(C)(C)O)NC(C(C)NC(=O)C(c1ccccc1)O)C c1(C(=O)NC(C(C)NC(C(CC)C)=O)(C)C)ccc2c(c1)CCCC(=O)N2 CCC(CC)C(C(=O)N1CCCC1CNC(=O)CCCCOC)N1CCOCC1 C1(C(=O)NCC2(F)CN(C(CC(=C)C)=O)C2)C2CCC1(c1ccco1)C2 Cc1cccc2c1OC(C(N1CCCCC1CNC(=O)Cn1ccc(=N)[nH]1)=O)C2 c1(NCCCNC(C(CC)CC2CCCC2)=O)cc([N+](=O)[O-])ccc1C(C)(C)C N1(C(C(C(=O)OCC)(C)F)=O)CCC2(CCCC2NC(=O)Cc2nc[nH]n2)CC1 CCC(C#N)C(=O)NC(c1cccnc1)C(=O)NCCc1ncccn1 Cc1ccc(CC(=O)NC2CCC23CN(C(c2cc4[nH]ccc4s2)=O)C3)c(C)c1 Cc1[nH]c(C)c(CSc2cn(CC3CNCCO3)nn2)c1C N1(C(C(C)C(F)F)=O)CCCC(C)(C)C1C(=O)NC1CCN(C)CC1(C)C c1(C(N(C2CCC(NC(=O)CC=C(Cl)Cl)CC2)C)=O)ccn(C)c(=O)c1 Cc1sc(S(N)(=O)=O)cc1C(=O)NC(C)(C)C(C)NC(C1CC=CCO1)=O N1(C(C(C=CCCC)O)=O)CCN(C(C2CCN(CC(F)F)CC2)=O)CC1 C1(C(N2CCC(=C)C2)=O)CCC(C)CN1C(=O)COCC(=O)NC c1(CC)ccc(C(=O)N(C)CC2(C)CCCC2NC(=O)C(O)C(C)CC)cc1F C1(C(=O)Nc2cn(C)nc2)CCCCCCN1C(c1cc(Cl)no1)=O C1(CCC)(NC(C2(COC)CCC(=O)N2)=O)CCCN(C(C23CC(F)(C2)C3)=O)C1 C1(CC)(NC(c2ccnc(C)c2N)=O)CCN(C(c2cc(C)cc(O)n2)=O)CC1 N1(C(C(C(C)C)O)=O)Cc2ccccc2CC1CNC(=O)C(C)(O)C(C)(C)C c1(OC)ccc(C(O)C(N2CCCC2c2ccc(O)cc2)=O)cc1OC c1(SC)nc(C)c(CCC(N2CC(NC(C3(O)CCCC3)=O)C(C)C2)=O)c(O)n1 c1(C(N(CCC(=O)NC(C)Cc2cnc[nH]2)CC=C)=O)cc(C)cs1 c1(OCCC)cccc(C(=O)NCCC(C)N(C)C(c2ccc(O)cn2)=O)c1 C(CC(F)(F)Cn1cc(C2CCCCCC2)nn1)NC(C(CC)n1cncn1)=O c1(C(C)=O)cccc(C(=O)NC2COCCC2NC(C2CC=CCC2)=O)c1 C1(C)(CNC(C(CN(CC)CC)F)=O)CCCN(C(C2CC(=O)CC(=O)N2)=O)C1 CN1N=C(C(=O)NC(C2CC=CCC2)C(N2CCC(N=[N+]=[N-])C(O)C2)=O)CCC1=O C=CCC(CC(C)C)C(=O)NC1CCN(CCNC(=O)CN2CCCCC2)CC1 c1(CC(=O)NC2(CC=C)CN(C(=O)C(C)NC(N)=O)C2)c(C)[nH]c2ccccc12 c1(C(=O)NCCC2(NC(C3C=C(C)CS3)=O)CCCC2)cc(O)ncn1 N1(C(C(C)OCCC=C)=O)CC(NC(=O)Cc2cncc(C)c2)C(S(C)(=O)=O)C1 CCCCC(C)C(=O)N(CC(O)CN(C)C(c1c(C)nn(CC)c1Cl)=O)C N1(C(CCC(C)(C)F)=O)CCN2C(=O)C(NC(c3cc(C(F)F)no3)=O)CC2C1 C(C(CO)(CO)NC(=O)C=CC1CCC1)N(C(=O)C(C)(O)C1CC1)C N1(C(C(C)NC(N)=O)=O)CC=C(C(=O)N2CCCN(C)CC2)CC1 C1(C(N2CC(OCCCCC)C2)=O)CC(O)CN1C(=O)CCCC1CCCC1 N1(C(COC)=O)CCCC(C)(C)C1CNC(C1CC1C1CC1)=O C(C(=O)N(C(C)CNC(=O)Cc1nc(C2CC2)n[nH]1)C)(C(C)C)SC N1(Cc2ccc(C(C)C)nc2)CCNCC2(CC2)C1 C(c1sccc1Br)=CC(N1CC(CCNC(C2C(C)CCS2)=O)C1)=O N1(C(C2C(C)SCCC2)=O)CC(C2CC2C(=O)NCC2(F)CC2)C1 c1(C(N2C(CCNC(C(CC#C)O)=O)CC(F)(F)C2)=O)ccn2cncc2c1 Cc1ccc(NC(c2c[nH]nc2CCNC(C2(C)CCCS2)=O)=O)c(O)c1 CC1CN(C(C2CSC2)=O)CC(C)CN1C(C1CCC(=O)N1C)=O C1(C)(C(=O)NC(CCC)C(=O)NC2CCOC(C)C2)CC2(CCC2)C1 C1(C(N2CCC(O)(CNC(CSCC(N)=O)=O)CC2)=O)CCN2CCOCC12 C1(NC(CSCC=C)=O)CCN(C(=O)C=Cc2ccnn2C)CC1C(C)C c1(C(=O)NCC(CC)NC(c2cc(O)n(C)n2)=O)ccc2ccccc2c1F Cc1cc(OC)ncc1C(N1CC2CC2(NC(=O)CCNC(C2CCC2)=O)C1)=O C12(NC(CCc3ccc(OC)c(F)c3)=O)COCCC1CN(C(=O)C(Cl)=CCl)C2 Cn1cc(C(=O)NCC(O)CNC(c2ccc(CCC#N)cc2)=O)n(C)c1=O C=Cn1nccc1C(=O)NCC(C(=O)NCC1CCCOC1)N(C)C c1(OC(C(=O)N(CC)Cc2cn(Cc3nccs3)nn2)(C)C)c(F)cccc1F c1(C(N(C)CCC2CCN(C(=O)C3=CC(C)(C)C3)CC2)=O)ncc(C#N)cc1Cl C1(C(N2CC(CC(=O)NCC3(C)OCCO3)(OC)C2)=O)CC(C)(C)CO1 C#Cc1ccc(C(=O)NC2(CO)CCCN(C(=O)CCNC(N)=O)C2)c(F)c1 c1(C(=O)NCC=CCC(N2C(COC)CCC2)=O)cc(Cl)ccc1-n1cnnn1 c1(CC)nc(C(=O)NCC(C2CC2)NC(c2cc(C(=O)OC)n[nH]2)=O)cs1 c1(SC)ccncc1NC(=O)C(N1CCSCC1CNC(=O)C(F)(F)F)=O CCCCC(C)CCC(=O)NC(CC)CC(=O)N1CCC(C)C1 c1(CCC(=O)NCCC2CCCN2C(=O)C=Cc2ccco2)cccnc1 c1(C(=O)NC2(CC(=O)NCC3(N(C)C)CCCC3)CC2)ccnnc1O c1(C(=O)NCC(C2N(C(C(C)NC(CC)(C)C)=O)CCC2)(C)C)nc(C)oc1C n1(-c2cccc(C)c2)cc(S(=O)(=O)N2C(C)CCC2C)cn1 c1(C(N2C(CN(C(=O)C(C)(C)O)C)CCC2)=O)ccc(-c2ncccn2)cc1 c1(COC)nc(C)c(C(=O)NCC(C)CNC(C2C3CCN2CC3)=O)s1 N1(C(C2N(CCC)CCC2)=O)CCC(C)(C(=O)NC2CC(CO)C3CC23)CC1 CCC(CC(=O)NCC1CC2CC2N1C(c1cnc(-c2cccs2)o1)=O)OC C1(CNC(C(C(C)O)C)=O)CC(C)CCN1C(=O)CN(C)C C1(C(N(CC(=O)NC)C)=O)CC(F)CN1C(C1CC1(C)C(F)F)=O C1(C(=O)NC2CCC3CCC23)(CNC(COCCOCC)=O)CC(F)(F)C1 N1(CCCNC(COCC(=O)NC)=O)CCOCC1 C=CC(CCC)CC(=O)NCC1(C(=O)NCc2ccc(OC)cc2)CC(C)(C)C1 CCCCCC(F)C(=O)N1CC(OC)CC1(C)CNC(=O)Cn1cccn1 C1(C(=O)NCc2ccc(C(N(CCOC)CC)=O)o2)CCC(F)(F)C1 CS(C)(=O)=Nc1ccc(C(=O)NC2CN(C(=O)CNC=O)C3(CCC3)C2)s1 c1(NC(C)=O)cccc(C(=O)NC2CCCC(NC(=O)Cc3nc(C)no3)C2)c1 C1(OC)Cc2ccccc2N(C(c2ccc(-c3cn[nH]c3)s2)=O)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)N(C(C)CN(C(=O)C1=CCC1)C)C C1(C(=O)NC(c2nc(=O)o[nH]2)C)CC2C=CC1N(C(=O)CCc1nc[nH]n1)C2 c1(C(=O)NCCC2C(C)CCCN2C(c2coc(Cl)n2)=O)nccc2ccsc12 c1(O)cccc(Cl)n1.c1(C(=O)OCCSCCNCC)ccccc1 c1(C(=O)NCC2C3N(C(C(C)OCCC=C)=O)C(CC3)C2)cnc2[nH]nnc2c1 CC(C)CCN=C(NCC1CCOC1(C)C)NC1CC(=O)N(CC(F)(F)F)C1 N1(C(CNS(N)(=O)=O)=O)CC(NC(=O)CCN2CCCC2=O)C(O)C1 C(c1cnn(C)c1C)=CC(=O)N(C)CC1N(C(CC(C)(C)OC)=O)CCC1 C1(C(=O)NCCC(C)N2CCC2)CC12CCN(C(=O)Cc1ccns1)C2 C(=O)(C(C)(C)CCC#N)N(C)Cc1c(CNC(C(F)=CCC)=O)cccc1 C1(NC(c2c(Cl)cnc(C)n2)=O)CCN(C(=O)C(=O)N=S(C)(C)=O)CC(C)(C)C1 CCCCC(CC(=O)N1CCC2(CSC2)C1)NC(c1cccs1)=O CC1CCN(C(=O)C=Cc2cscn2)CC1CNC(=O)CC(C)(C)CN(C)C C(=O)(C(C)CC(C)C(C)=O)NC(CCC(=O)NCCc1cn(CC)nn1)(C)C C12(C(=O)NC3(C=C)CCCCC3)CC(CCO1)N(C(C1CC1(C)CC)=O)C2 C1(CNC(CCC#CC)=O)COCCN(C(=O)C(C)N2CC(C)C2)C1 c1(C(=O)NCc2ccc(C(N3CCC(CC)C3)=O)s2)cccc(C)c1N c1(C(=O)NCCC(=C)CNC(=O)C(CCC)N(C)C)cc(C)cc(C)c1N c1(C(N2CCN(C(CC(C=C)C)=O)CC(C)C2)=O)cc2c(C)cccn2c1 C1(NC(C=Cc2c(C)ncs2)=O)(CO)CCCN(C(=O)CC(F)(F)Cl)C1 c1(OC)ccc(Cl)cc1CNC(=NCC1CC2CCC1CC2)NC1CCOCC1 C#CC1(O)CCCC(NCc2cc(Cl)ccc2Br)C1 C1(CNC(C2(OC)CCOC2)=O)CN(C(C2CCCOC2)=O)CC(C)(C)O1 C(=O)(C(C)C(O)C(C)C)N1C(C(=O)Nc2c(O)ncc(C)c2)CCC1C N1(C(C(C)N(C(=O)C=Cc2cc[nH]n2)CC)=O)CCC(O)(C(N)=O)C1 N1(Cc2ncc(C)o2)CCC(C)(C)C1C(=O)O C1(NC(c2n(CC)ccc2)=O)C2CC(NC(=O)C(n3ccnc3C)C)CC12 C1(O)(CNC(C2N(CC)CCOC2)=O)CCCN(C(=O)C=Cc2cn(C)cn2)C1 C=CCCCCCC(=O)N1CCN(C(=O)CCCS(N)(=O)=O)CC1CCC N1(C(C2(CNC(Cn3c(C)cc(C)n3)=O)CCCO2)=O)CCC(C2CCCC2)C1 c1(C(=O)NCCN(C(C(C)=C(CC)C)=O)Cc2ccccc2)c[nH]c(C(N)=O)c1 C1(CNC(CCN(C(CC)CC)C)=O)CC(O)(CNC(=O)C(=O)NCC)C1 C1(NC(C2(C)CC(C)C2)=O)CCC(F)(CNC(c2nc(C3CC3)cs2)=O)C1 Cc1nc(N(CCCNC(C2CC(=O)N(C(C)(C)C)C2)=O)C)cc2nncn12 C1(CNC(C2(N(C)C)CC2)=O)CCCCN1C(=O)CCc1cccnc1 C1(CNC(C=C(C)CCc2ccccc2)=O)C(C)CCN1C(c1cnsc1)=O C1(O)(c2onc(NC3CC(C)(CC)OC3=O)n2)CCC(C)(C)CC1 C#CCC(CC(=O)NCCC(O)CO)NC(C1CCC(=O)N(C)C1)=O C(CC1=CCN(C(=O)C=Cc2cccc(C(N)=O)c2)CC1)NC(CC=CC=C)=O N1(C(C2(CC)COC2)=O)CCCN(C(C2CCC3(CCC3)O2)=O)C(CO)C1 N1(C(C=CSC)=O)CC(CCNC(c2ccn(C)c(=O)c2)=O)OC(C)C1 Cc1ccc(C(=O)NCc2ccoc2C(=O)N(C2CCOC2)CCF)cc1C CCCC(C)(C)C(=O)NC(CN(C)C(c1cccn(CC(C)C)c1=O)=O)CC c1(C(N(CC(F)F)CCOC)=O)oc(CNC(c2cnsc2)=O)nc1C C1(C(N(C(C)CCNC(=O)C(c2ccc(Cl)s2)=O)C)=O)NC(=O)CC1C(F)(F)F c1(CC(N2CC(C)(NC(CC(C)n3cccn3)=O)C2)=O)cn2c(n1)CCCC2 CC#CCC(C(=O)NCc1cn(C)cn1)NC(=O)C=C(C1CC1)C1CC1 CC1(C)CCC(CNC(=O)C(F)n2ccnc2)N(C(=O)Cn2cnc(=N)[nH]2)C1 c1(N2CCCC(CCC)C2)nc(N(C)Cc2cccc(OC)n2)c2ccsc2n1 C12(NC(c3ncc(F)cc3F)=O)CCN(C(=O)C=CSc3nc[nH]n3)CC1C2 C12(C(=O)NCCCC(C)O)CCCC1CCN2C(c1ccc(C2CC2)cc1)=O C(=O)(CCCCC(F)(F)F)NC(CNC(C(CC(=C)C)OC)=O)C1CC1 c1(CONC(C2N(C(C)=O)CC2)=O)n[nH]c(C)c1C(C)C.C(C)(C)(C)OC(=O)NC c1(OC)cccc(CN2CCCC(C(=O)NC3COCC3O)CC2)c1C C(C(C)(O)C(C)C)NC(c1c(CNC(Cc2c(C)ocn2)=O)ccs1)=O c1(C(=O)NC2C(O)CCN(C(c3cc(CCC)[nH]n3)=O)C2)cc(Cl)cc(Cl)c1N c1(C(=O)NCC(CC)NC(=O)C(c2cncnc2)C)ncc(F)cc1C C1(NC=O)CN(C(=O)Cc2cnns2)CCC1(C)C.c1(OC)ncc(C=CC)cn1 Cc1cc(CCCC(=O)NCCC2CCC(NC(=O)CCOC(C)C)C2)c(C)s1 C1(C)(CC)CC(NC(=O)CSCCN(C)C)CN1C(c1ccc(C2CC2)o1)=O C1(CNC(CS(CC)(=O)=O)=O)CN(C(=O)CC2COC(=O)N2)C2COCC2O1 CCC(C)(CC(=O)N1CCOCC(NC(c2ccc(C)s2)=O)C1)C(=O)OC N1(C(c2nc(CCCCC)sc2)=O)CC(CNC(=O)C=CSC)C(C)C1 C1(C(=O)NC(CCC)C(F)(F)F)CCC(C)(C)N(C(C2CC23CC3)=O)C1 CC1CC(C(=O)NCC2CC(=C3CCC3)C2)N1C(C1CCOC1C1CC1)=O C(C)(C)(CCCNC(C1CC2CCCC12)=O)NC(CN(C)C(=O)C1CC1)=O c1(C(=O)NCCN(C(C2CCC(O)C2)=O)Cc2ccccc2)cnc(O)c(F)c1 c1(-c2c(OC)cccc2F)ccc2nc(C(=O)N(C)CCN(C)C)cn2c1 CC1CCN(C(=O)C(C)c2cccs2)CCN1C(=O)Cn1cc(Cl)cn1 C(=O)(CC(C(F)(F)F)N1CCOCC1)NCC(C)NC(c1cn(C)ccc1=O)=O c1(CNC(C2(C)CCN2c2ccnc(C(F)(F)F)n2)=O)ccc(Cl)c(F)c1 c1(CC)cc(C(N2CCC(O)(CCNC(=O)CN3CC=CC3)CC2)=O)cc(F)c1 c1(CC)cc(CNc2snc(C)c2C#N)cc(CC)c1 CCCCC(F)C(=O)NC1CN(C(=O)Cc2cnc(C)nc2O)CC12CC2 C12(C(=O)NCC3CC(C)N(C(=O)C=CC4CCC4)CC3)CCC(C1)C(C)(C)O2 Cc1ncc2c(n1)CCC(NC(C1OCCOC1(C)C)C)C2 N1(C(C(=O)Nc2cccc(C)c2)=O)CC2(C)CC1C2NC(C1CCCS1(=O)=O)=O c1(NC(C(=O)NC2C(CC)CC2)=O)cnn(CC(F)(F)F)c1 c1(N(C)C)ccc(-c2nc(C3CCCCC3)n(CCn3ccnc3)n2)cc1CO C1(OC)CC2N(C1)C2=O.C1(c2ncco2)(OC)CCCC1 Cc1cc(=O)ccn1CC(=O)NC(C)CC1CN(C(C23CCC(CC2)CO3)=O)C1 N1(C(CC2(OC)CC2)=O)CCC(C2(O)CCN(C(=O)CC3C=CCC3)C2)CC1 C(=O)(C(F)C(C)(F)F)NCCSCC(=O)NC(CC(=O)OC)C1CC1 C1(C(=O)NCC(C)N(C)C(c2cc(C3CC3)[nH]n2)=O)COCCN1C c1(C(=O)NCCC2(O)CN(C(Cc3c(C)scc3)=O)C2)ccc2nn[nH]c2c1 Cc1cccc2c(C(N3CC(C4CN(C(C5CCNC(=O)C5)=O)C4)C3)=O)c[nH]c12 C1(NC(C(CNC(c2c(CCC)n[nH]c2)=O)C)=O)CC2C=CC1C2 C1(OC)CCCC(CC(=O)NC(C)(C)CCNC(c2cc(CO)[nH]n2)=O)C1 CN1CCC(C(=O)NC2CCCC2NC(c2ccnc(CC(F)(F)F)n2)=O)C1=O CC(C)(COCC(F)F)C(=O)NC1CC1NC(C1CC(C(F)(F)F)C1)=O c1(CC)cc(C(=O)NCC2CCN(C(C3(C)CC=CCO3)=O)C2)c(C)nn1 O=C(Cn1cc(C#N)cn1)NN1CCCC1C(=O)NC1CCCC(O)CC1 c1(C(=O)OC(C)(C)C)ccc(C(=O)CN2CC3C(CN=[N+]=[N-])C3C2)cc1 CCC1=C(C(=O)N(CC(C)NC(c2[nH]ccc(=O)c2C)=O)CC)CCCO1 CCCCCC(O)C(=O)N1CCC(O)(CCNC(c2ccsc2OCC)=O)C1 c1(C(N2C(CNC(C(CC#C)C3CC3)=O)CCC2)=O)cccc2ncnc(O)c12 c1(C(=O)NC2CCN(C(C3C(=C)C3)=O)CC2O)ccc(S(=O)(=O)NC)nc1 C1(NC(=O)C(F)F)COCCC1NC(=O)CCSc1ccncc1 C1(CNC(C2CC(=C)C2)=O)CC2CN(C(c3n[nH]c(CC)c3Cl)=O)CC12 c1(C(=O)NCC(C)CN(C(=O)CCCC2CCCO2)C)cncn(C)c1=O C(CC(=O)N1CCOCC1C(C)O)(C(F)F)NC(C1CC(SC)C1)=O CC1(C)CN(C(C2(C)CC2)=O)CC(CNC(c2cc(C(F)(F)F)cc(O)n2)=O)O1 C1(CNC(Cc2c(-c3ccc(C)cc3)nc(C)s2)=O)CCCN(C(=O)C(C)O)CC1 S(=O)(=O)(c1cccs1)N(C)Cc1cc(-n2c(C)cc(C)n2)sc1.C12CON(C1)C2 c1(C(=O)OC)cnc(N(C(C23CCC(C2)OC3)=O)C2CC2)cn1.N1CCCC1C C(C(=O)N1CC(C)(C)C1Cn1cc(CCCCO)nn1)(C(C)(C)C)OC(C)(C)C N1(CC)C2CCC1CN(C(=O)CCCCNC(C1CS(=O)(=O)C1)=O)C2 N1(C(CCCCCN(C(CCOC(C)=O)=O)C)=O)CCC2(CCCN2C)C1 CCC(C)CC(C(=O)NCCc1csnn1)NC(=O)CC(=O)OC(C)(C)C CCC(C)(CCC(C)C)C(=O)NCC(C1CC1)NC(=O)CC1CCC(F)(F)CC1 c1(CNC(c2cc3occc3s2)=O)nc2c(s1)CN(C(C1CC(CF)C1)=O)CC2 C(=O)(C(CCCO)c1ccccc1)N1CCCC(CNC(=O)CCOC2CC2)C1 c1(C(N(C2CCN(C(c3ccc(CCC)s3)=O)CC2)CC#C)=O)cccc(O)n1 c1(C(=O)OCC)sc(SC)nc1NC(C1CC(NC(=O)Cc2nonc2C)C1)=O CC1=C(C)CC(C)(C(N2CC(NC(c3ncn(C)c3C)=O)CC(C)C2)=O)CC1 N1(C(C(C)OC2CCCCCC2)=O)CCC(N(C)C(c2ccnn2C)=O)C2(CC2)C1 c1(CN2CCC(F)(C(=O)NC(C3N(C)C(=O)CC3)=O)CC2)nccc2nc[nH]c12 c1(C(=O)NC(Cn2cc(CNC(CC=C=C)=O)nn2)C)cnc(CC)nc1C c1(OC)ccc(F)c(C(=O)NC2CC(NC(=O)CC(C)C)C2)c1F Cc1ccc(C(=O)NCC(=O)NCC(=O)NCCC(C)C(F)F)c(C)c1 Cc1noc(COCC(=O)NC(C)C(C)(C)NC(=O)COc2ccsn2)n1 C(=O)(C(CC(N)=O)NC(=O)CSCC)NC(CC=C)C1CC1 C1(C(=O)NCC2CC(NC(=O)CCc3ncco3)C2)CCC2C(C1)C2(F)F C1(NC(c2c(C)[nH]nc2C(F)(F)F)=O)CCCN(C(=O)C2=CCCCC2)CCC1 CC(C(=O)NCC1CCC2(CN(C(C3CNC(=O)O3)=O)C2)O1)C(F)(F)C(F)F N1(C(CCOCC(C)C)=O)CCC(C)(CCNC(=O)CCCCC2CC2)C1 Cc1ccc(I)c(C(=O)NCCCC2CC=CC2)c1 C(C)(C)(CC=CC(=O)N1CCC1)NC(C1CC(N(C)C)C1)=O C(CC1=CCN(C(=O)CNC(=O)C2CC2)CC1)NC(c1ccn(C(C)(C)C)c1)=O c1(C(=O)NC(CNC(COCC)=O)(C)C2CC2)oc(Br)nc1C(F)(F)F C1(NC(C=CC(C)=O)=O)CCCC1NC(=O)CCc1cscn1 O=C(C1=C(Cl)CCCC1)NCC1CC1NC(C1(c2ccccc2)CCOC1)=O C(=O)(C1=NNC(=O)C1)NCCSCC(=O)NCC(CCC)OC N1(C(C2C(C)(C(=O)OCC)C2)=O)CCCC(NC(C23CCC(CC2)OC3)=O)C1C C1(O)(C(N2CC(CC(=O)NCC(CC)(C)COC)C(C)C2)=O)CCCCCC1 c1(C(N2CC3C(C(=O)NCc4n(C)ncc4)C3C2)=O)c(Br)ccc2c1OCO2 N(C1CC(C)n2ccnc21)C(=O)NCc1cccc(-n2ccc(C)n2)c1C C1(C(N(CC#CC)C)=O)C2CC(O)C(C2)N1C(c1ccc(C)nn1)=O N1(C(C(C)(CO)OC)=O)CCN(C(c2cc(Cl)c(N)c(Cl)c2)=O)CC(CO)C1 O=C(C1CCc2c[nH]nc21)Nc1ccc(-n2ccnc2)c(F)c1 C(=O)(CCN=C(NC1CCN(CC(F)(F)F)C1)NC1CC(C)C1)NCC CC(C)C(CNC(=O)CC1CCCOC1)C(=O)N(C)CC1CC(F)C1 C1(CNC(=O)CC2CCOC2)OCCC1C(=O)N(C1CC1)C1CC1 Cc1cc(CN(C2CCN(C(=O)COC3CCOCC3)CC2)C)cc(F)c1 N1(C(C(C(=O)OC)(C)C)=O)CC2CCCC(N(C(=O)CC(C)C)C)C2C1 N1(C(C(C)Sc2cccc(OC)c2)=O)CC2(CC(NC(C3(Cl)CC3)=O)C2)C1 c1(CC)ncc(C(=O)NCC2CCCC2NC(c2cccn2C)=O)s1 CC(C)(C#N)CCCC(=O)NCC1CC(F)CN1C(=O)CCc1cccs1 c1(C(=O)NCC(=C)CCNC(C2CC(=O)N(C)C2)=O)cnc2c(c1)CCCC2 N1(C(CN(CCC)C)=O)CCCCC1CNC(=O)C(=O)C=Cc1cccs1 C=CC(C)(CCOC)C(=O)N(C)CCN(C)C(C1CN(C2CCC2)C1)=O C1(OC)CCCCC1S(=O)(=O)N1CCCC1c1cccc(I)c1 N1(C(COCC=C)=O)CCOC2(CCC(NC(=O)C(C)C(F)(F)F)CC2)C1 N1(C(CC=C)=O)CC2(C1)CN(C(C1CCCCN1Cc1cccnc1)=O)C2 CCC(C)(O)C(=O)NCC1(O)CCN(C(c2ccccc2-c2nnc(C)o2)=O)C1 C(=O)(C(CC)NC(C1CCOC1CNC(=O)Cc1cnsc1)=O)NCC C(CC)(C(=O)N(C1CC(C(N2CC(OCC(C)C)C2)=O)C1)C)OCC c1(C(=O)NC(c2ccc(F)cc2)CNC(C(CC)F)=O)c(S(N)(=O)=O)cnn1C C1(O)(C(=O)NC2CC(CNC(=O)Cc3ccc(Cl)cc3Cl)C2)CN2CCC1CC2 c1(C(N2CCC(C)(NC(=O)C(F)=C3CCCC3)C2)=O)ccnc2c(F)cccc12 c1(NC(=O)NCCC23COC(C2)C3)cccc(COc2ccccc2Cl)n1 C(CC(=O)NCCCn1cc(C)cn1)(C(C)(C)C)NC(COC(CC)C)=O CC1(C)C(C(=O)NC2(c3ccccc3OC(F)F)CCCC2)CC1O C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(NC(C(CC)n2nccc2C)=O)C(O)CC1 N1(C(C(C)CF)=O)CC(C)(C)OCC1CNC(C1(c2cccs2)CC1)=O c1(C(=O)NCCC(C(=O)NCC2CC(CC)C2)O)c(C)cccc1F C1(CS(=O)(=O)Nc2cn(C(C)(C)C)nc2)CCc2ccccc2CC1 N(C(=NCC1CCCCO1)NCC(c1ccncc1)(C)O)C(C)CC(F)F c1(NC(C)CN2CCC(O)C2)nccc(=NCC(C)(C)N2CCOCC2)[nH]1 N1(C(C(CC=CC)NC(=O)CCc2nc(O)n[nH]2)=O)CCC12CN(C)C2 N#CC1CN(Cc2cc3ccccc3o2)CCN1C(c1cc(O)nc(Cl)c1)=O c1(CC(=O)NC2C(NC(CNC(COC)=O)=O)CC2)ccc(C)cc1C Cc1cc(C)c(C(=O)NCC2CC3CC3N2C(=O)C(C)Cc2ccco2)c(S)n1 C(=O)(CC(C)C(C)(C)C)NC1CN(C(c2cc(C(N)=O)cc(C)c2)=O)C(CO)C1 c1(CC)cncc(C(=O)NC(CCOC)C(=O)N2CCC(CCN(C)C)C2)c1 C(=O)(C(C)(C)C(=O)NC(CNC(=O)C(COC)N(C)C)CC(F)(F)F)OCC C1(NC(c2ncc(C(C)=O)s2)=O)CCC12CN(C(=O)COC(C)C)C2 N1(C(c2sc(C)c(Br)c2)=O)CCCC(F)(CNC(=O)C(C)C)C1 N1(CCC)CCN(C(C(=O)NC2CCCCC2)C2CC2)C(C)(C)C1=O c1(C(=O)NC2CC(C)(NC(C(C(C=C)C)C)=O)C2)[nH]cc2c1CCS2(=O)=O c1(C(=O)NCCCCCCNC(C2(C)COC(=O)N2)=O)cccc2nccn12 C1(CC)CN(C(c2coc(Cl)n2)=O)CCN1C(C1C2CCCCC12)=O C=CC1(C(=O)NCCC(O)CCC)CCN(C(=O)C=CC2CCCCC2)CC1 Cc1ccc(C)c(C(N2CCC2(C)CC(=O)NCC2CCC(=O)O2)=O)n1 c1(NC(C23C(CN(C(CC(CC)O)=O)C2)C3)=O)cnc(Cl)c(Cl)c1 c1(C(=O)NC2CCN(C(C3(C=C)CCC3)=O)CC2O)cn2cc(C)sc2n1 n1(CC(=O)N(C)CC2CN(C(c3ccc(F)nc3)=O)C2)cc([N+](=O)[O-])cn1 c1(C(=O)NC(CNc2nccc(CC(=O)OC)n2)C)cc(C)cc(F)c1 CC(C)(C)C(CNC(C1CC(CNC(c2ccnnc2)=O)C1)=O)CO CC(CC(N)=O)C(=O)N1CC(C)(NC(=O)C(c2ccc(F)cc2)=O)C1 C1(CNC(c2c(CC)cccn2)=O)C(C)CCCN1C(=O)CC1CCSCC1 c1(C(=O)NC2CCC(N(C)C(c3nc(Cl)cs3)=O)C2)ccc2c(c1)CC(C)(C)O2 C1(CNC(c2ccc3ocnc3c2)=O)CC2COCC2N1C(c1ccncc1)=O N1(C(C2OCCN(C)C2)=O)CC(N(C)C(c2cn3c(n2)CCC3)=O)C(C)(C)C1 CN=c1ccc(C(=O)NC(CO)C(N2CC(O)CC2CO)=O)c[nH]1 C#CC(C)(C)C(=O)NCCCC(C)NC(=O)C#CCNC(=O)OC(C)(C)C N1(C(C2C(CC)N(C)CC2)=O)CCCOC(CCNC(c2[nH]c(C)cc2C)=O)C1 CCS(=O)(=O)CC=CCNC(=O)Cn1cc(C2(O)CCC2)nn1 N1(CC(=O)N(CC)CC)CCC(C(C)SC2C(C)C2(F)F)CC1 C(N=c1nnn(C)[nH]1)C1CCCC(CNC(COc2c(C(C)=O)cccc2)=O)C1 N1(c2cc(NCC3(CF)CC(F)(F)C3)nc(COC)n2)Cc2ccncc2C1 C(CCOCCO)(C(=O)NC1(C)CC(C)(C)C1)NC(C(F)=CCC)=O C1(NC(C2OCC(C)(C)OC2)=O)CC2CC1CN(C(c1nnc(O)nc1O)=O)C2 N1(C(C(F)=C(C)C)=O)CCCC12CCN(C(C1CC(=C3CC3)C1)=O)CC2 N1(C(C=CC(=O)OCCCC)=O)CCN2CCOCC2(CNC(=O)C(N)=O)C1 Cc1cc(C)c(C(=O)N(C(C)CCNC(=O)C(C)OCCN(C)C)C)o1 CS(=O)(=O)CC(=O)NCC(F)CNC(c1cocc1Br)=O C1(C(=O)NC(C(C)C)CNC(=O)Cn2ccc(C(F)(F)F)n2)CC(C)(C)CN1C c1(OCCC#C)ccc(C(=O)NCC(O)CN(C(=O)CC2C=CCCC2)C)cc1 N1(C(c2occ(S(N)(=O)=O)c2)=O)CCC2C(CCCN2C(c2ccc[nH]2)=O)C1 N1(OCCCCCCCCN(c2n(C)ccc2)CCO)CC2CC1C2N1CCNCC1 c1(C(N2CCN(C(CC3(C)CC(C)(C)OC3)=O)CC2)=O)cc2n(c1)CCOC2 Cc1ccn(C)c1C(=O)N(CCC(C)(C)NC(C1CC1(C)C(F)F)=O)C c1(-c2onc(C3(OC)CCCCC3)n2)cccc(C2CC2)c1F N1(C(CCC)=O)CC2CCC(CNC(c3cncc(OC(F)(F)F)c3)=O)(C2)C1 C1(NS(C(C)C)(=O)=O)CN(C(=O)CCN2C(=O)C=CC2=O)CCC1O C1(C(N2CCC(C(C(=O)NCc3cc(COC)on3)C)C2)=O)CCN(C)C(=O)C1 c1(OC)ccc(NC(c2c(F)cc(Cl)cc2Br)=O)cc1S(=O)(=O)N(C)C N1(C(C(C)NC(CC)=O)=O)CCC(O)(CCNC(c2oc(CO)nc2C)=O)CC1 C1(CNC(CCCCC)=O)CC2(CCN(C(c3cccc(F)c3O)=O)C2)CO1 C(=O)(C(C(C)NC(=O)C1=C(C)OCC1)C(C)C)N1CCOCC(CC)C1 C1(NC(C(N(C)C(c2cnns2)=O)C2CC2)=O)CNC(=O)C12CC2 C(C(C)CS(C)(=O)=O)N(CC(C)CNC(=O)CC(O)C1CCCC1)C N1(C(c2cc(C)ns2)=O)CC=C(CCNC(=O)C(c2ccccc2)N(C)C)CC1 C1(C)(NC(CN(CCOC)C(C2CCOC(C)C2)=O)=O)C(C)(C)C1(C)C N1(C(C2CC2C(=O)Nc2c(CC)nc[nH]2)=O)CC2CC2(C(=O)OC)C1 c1(CC)cn2c(n1)CC(C(=O)NCC1CN(C(=O)C(C)Cn3cccn3)C1)CC2 C(CC(=O)NCC1CCC(NC(c2nn(C)cc2Cl)=O)C1)(C(F)(F)F)OC CC(CC(=O)N1CCOC(C(C)NC(c2cnn(CCF)c2)=O)C1)C(F)(F)F CC(C(=O)NCCCCC1CN(C(C2CC(O)C2)=O)C1)c1ccco1 C(=O)(C(C(C)C)NC(=O)C(CCc1ccc(F)cc1)N1CCCCCC1)OC C(=O)(C(COC(C)C)NC(=O)CCc1ccoc1)NC(COC)C Cc1ccncc1CC(=O)NC1CCC(CNC(C2CC23CCC3)=O)C1 N1(C(c2cnc(OC)s2)=O)CC2CCN(C(c3cc(C)c(C)c(F)c3)=O)C2C1 C1(C(N(CCCNC(COCCC)=O)C)=O)CC(C(=O)OC)C12CCC2 CCC(C1CC1)NC(=O)CN(C(=O)CNC(=O)C1CC1)CC1CC1 C1(C(=O)NCCN(C)C(c2nccnc2N)=O)CCCCC(C)(C)C1 C1(F)(CNC(C2(CCCC)CC2)=O)CN(C(c2nnn(C(C)(C)C)n2)=O)C1 N1(C(CC(C)CF)=O)CCN(C(=O)CCc2ccccn2)CC1c1ccccn1 CCC(C)C(O)C(C)C(=O)NC1C2CC3C(C2)C13C(=O)NCC1CC2(CCC2)C1 c1(C(=O)NC(CC2CN(C(CCNC(=O)OC)=O)C2)C)cncc2c1CCCC2 N#CC1(C(N2CCC(CNC(C3CC3F)=O)CC2)=O)CCSCC1 C1(O)(CCNC(c2c(C)oc(Cl)n2)=O)CCCN(C(=O)CC2CC2C2CC2)C1 c1(CC)c[nH]nc1CNC(C1CC(CNC(=O)C(C)(C)NC(C)=O)C1)=O C1(CC(=O)NCC(C)CNC(c2nc(=O)n(C)[nH]2)=O)(CC)CCOCC1 N1(C(c2cc(Br)n[nH]2)=O)CCCCC(NC(C23CCC(CC2)CO3)=O)C1 N1(C(CC(=C=C)C)=O)CCC12CN(C(C1CC1c1ccco1)=O)C2 c1(NC(C(=O)NC(C#C)C2CCC2)=O)cc(F)ccc1OC(F)(F)F N1(C(C(CCNC(C(C)C2CC2)=O)(C)C)=O)C2CCC1CC1(C2)N=N1 Cc1nccn1C(C)C(=O)NCC1CCN(Cc2csnn2)C1 c1(C(=O)NCC2CN(CC3CCN(C(=O)C=CCO)CC3)C2)cc(Cl)cnc1O N1(C(CC)=O)CC(NC(=O)CCOc2cc(C)ccc2C)CC(F)(F)C1 c1(OCC)ccc(C(N2CC3(C2)CN(C(c2ccc(C(F)F)o2)=O)C3)=O)cc1C C1(CCNC(CN(CCC#C)C)=O)CCN(C(=O)C(CO)N(C)C)C1 N1(C(C(c2ccc(C)s2)C)=O)CC(C2CCCN(C(=O)CN3CC(C)(C)C3)C2)C1 c1(C(N2CCCC(n3cc(C4(O)CC4)nn3)C2)=O)ccccc1N1CCC(O)C1 C#CCC(CC#C)C(=O)NCC(CNC(C1CC(OCC)C1)=O)CO c1(C(=O)NC2C3CC(NC(=O)OC(C)(C)C)C(CC3)C2)cc2cccc(O)c2[nH]1 O=C(C1=CCCSC1)N1CCN(C(c2cnc(C3CCC3)nc2O)=O)C(CO)C1 C1(NC(CN(C(C)=O)C)=O)CS(=O)(=O)CC1NC(c1cncnc1C)=O CC(N=c1[nH]c2c(c(=NCC3(Cl)CC34CCC4)[nH]1)CCC2)c1nc(O)n[nH]1 c1(CC(=O)N(C(C)C(=O)NC(C)C(=O)NC2CC2)CCC)cnccc1OC C(C(O)C(F)(F)F)NC(C1(CC)CCCN1C(C1CCS(=O)CC1)=O)=O C(C(CC)CCO)NC(CCN(CC#C)C(c1cnn(C)c1C)=O)=O c1(OC)nc(C)ncc1C(=O)NC1CCCC(NC(=O)Cc2ccon2)C1 C1(C(=O)NC2CCC(NC(CC(CCSC)O)=O)CC2)CCc2nncn2C1 CC1CC(C)(C(=O)NCC(C)(C)CN(C(=O)C=C2CCCC2)C)CCO1 N1(C(=O)COCCF)CCC2CCCC(C1)N2C(c1ccc2oc(=O)oc2c1)=O C(CN=c1nc(N2CCOC(CCO)C2)c2c(F)cccc2[nH]1)c1c(C)ocn1 N1(C(CC(=O)NC)=O)CCC(NC(c2csc(O)n2)=O)C12CCCC2 N(C1CCC(Nc2ncc3ccsc3n2)c2ccccc21)C(C(C)NC(C)=O)=O CC(C)(O)CC(=O)N1CCN(C2CCC(NC(c3ccon3)=O)C2)CC1 c1(C(N2CCC(NC(C(F)=C(C)C)=O)C2C(C)C)=O)cc(F)c(F)c(Cl)c1F c1(C(=O)NCC(CC)N(C)C(c2cnncc2OC)=O)cc(C)c(=O)n(C)c1 Cc1nc(C(=O)N(C(C)CCNC(c2cc(-c3cccs3)[nH]n2)=O)C)n[nH]1 CC1(C)COC(C)(C(N2CC(NC(C3C(C)(C)C3(F)F)=O)C2)=O)CO1 C1(C(N(CCC#N)C(C)C)=O)CS(=O)(=O)CC1c1ccccc1 N#Cc1ccc(CC(=O)NCC2CC2CC(=O)Nc2cccc(CO)c2)cc1 N1(C(C2(C)CC2(Cl)Cl)=O)CCCN(C(C2(CO)CCC2)=O)CCC1 Cc1ccc(OC(C)C(N2CCC(NC(C3(N(C)C)CC3)=O)C2)=O)c(Br)c1 CCN=c1[nH]c(C)c(C(=O)NC(C)(CNC(c2cn3c(n2)CCCC3)=O)CO)s1 Cc1ncc(F)c(N2CCC(C(C)NC(c3ccccc3-c3nc[nH]n3)=O)C2)n1 O=S(=O)(c1ccc2[nH]c(=NCCCc3cncnc3)ccc2c1)NCC1CSC1 CS(C)(=O)=NC(=O)C(=O)N1CC2CC(NC(C3CC34CCC4)=O)CC1C2 c12cccc(c1)N2.c1(CN(C(=O)OCC(=C)C)C2CC2)ccccc1C c1(CC)ccccc1CC(=O)NC1(CO)CN(C(=O)CCCN(C)C)C1.C(C)(=O)OC C1(CNC(C2C(OC)(OC)CC2)=O)CC(F)(F)CN1C(c1cc(CO)oc1C)=O CC(C)(C)CC(O)C(=O)NC1CCC(NC(C2CC3(CCCC3)C2)=O)C1 c1(N2CC(C)C(CNC(c3cccc(CO)c3)=O)CC2)ccc(C#N)nn1 c1(CCCCC)ccc(NC(C2CC2C(N2CC3(CCC3)C2)=O)=O)c(C#N)c1 c1(OC)cccc2cc(-c3ccc(CN(C)C(C)C)s3)[nH]c12 N1(C(c2c(C(C)C)ocn2)=O)CC(NC(C2CCC2c2nc(S)n[nH]2)=O)C(C)C1 O=C(CS(=O)(=O)CCO)NC1CC1NC(c1ccc(-n2cnnn2)cn1)=O C1(NC(=O)CCc2ccco2)CN(C(=O)Cc2ccno2)CC1C1CC1 C1(CNC(C(C)=CC)=O)(OC)CCN(C(C2(CC)CC(C)(C)C2)=O)CC1 c1(C(C)C)ncc(C(=O)NC2(CCC(=O)NC(C3CCCO3)CO)CCCC2)o1 C1(C(=O)NCc2c(C)c[nH]n2)(NC(=O)CC2CCCCCC2)CCCC1C C1(C(N(C2CC(C)(NC(=O)OC(C)(C)C)C2)C)=O)CC(O)CCO1 N1(C(CC#N)=O)CCC(C2(NC(c3cc([N+](=O)[O-])c[nH]3)=O)CC2)CC1 N1(C(C(CC2CC2)OC)=O)CC2CCOCC2C1 C(=O)(CC(C)C(=O)N1CCCC1CNC(=O)CC=C(C)C)OCC C#Cc1cccc(C(=O)NCC23CCC2CCN3C(c2cc(C)on2)=O)c1F N1(C(c2cc(C)nnc2)=O)CC(C(=O)NC(C(N)=O)C2CCCC2)CC(C)(C)C1 CCC(C)(CCNC(=O)Cc1cnc(C)s1)NC(c1[nH]cc(C)c1C)=O CC(C)CC(F)(F)C(=O)N1CCCC(C(=O)NCCNC(=O)C(C)CF)C1 Cc1cnc(NCC2(C)CCCC(=O)N2)c(S(=O)(=O)NCC2CCC=CO2)c1 Cc1ccnc(C(N2CCC(C)C(CNC(=O)CC(=O)NC3CC3)C2)=O)c1O C(c1ccc(F)cc1)=C(C)C(=O)NCC(C)CNC(c1[nH]nnc1C)=O C1(CNC(C(CC=C)N(C)C)=O)CN(C(c2cnn(C)c2)=O)CCC1C N1(C(c2scc(C(N)=O)c2)=O)CCC(C2CC2)(CNC(C2CCCCO2)=O)C1 C1(NC(C2C(C)C2)=O)CN(C(c2ccc(Cl)[nH]2)=O)CC1Cc1ccccc1 C=Cn1nccc1C(=O)NC(C)(C)CCNC(c1nc(C2CC2)cs1)=O C1(CC(=O)NC)CN(C(c2cncnc2)=O)CCN1C(c1cnc(C2CC2)[nH]1)=O CN1CC2(CCN(C(C3CCN(C(c4cccc(Br)c4O)=O)CC3O)=O)CC2)C1 Cc1cnccc1C=CC(=O)NC1CN(C(=O)C(CCc2ccccc2)C(C)C)C1 c1(C(=O)NCC(CNC(C(CC2CC2)OC)=O)C)cncc2nc[nH]c12 N1(C(Cc2c(C)n[nH]c2)=O)CCC(C2OCCC2NC(=O)CCC2CCC2)CC1 Cc1ccc(C=CC(N2CC=CC2CNC(=O)C(C2CC(F)(F)C2)O)=O)cc1 c1(C(N(CCCCN(C)C(C2(C)CCCO2)=O)C)=O)cc(F)ccc1S(C)(=O)=O C(N=c1[nH]c(N2CCc3c(Br)cccc3C2)nc2c1COC2)c1cc(C)nn1C c1(C(=O)NCC(=C)C)ccc(NC(c2nc(C(N)=O)cs2)=O)cn1 C1(C(=O)NC2(C)CN(C(C(COC)N(C)C)=O)C2)CCCN(C)C1 N1(C(c2cccc(C)c2F)=O)CCC2CN(C(c3cc(C)n(C)n3)=O)CCC2C1 C1(CC(=O)NCCN(C(c2cncc(C(C)(F)F)c2)=O)CC)CCOC(C)(C)C1 c1(C(=O)NC2CCN(C(C(C3CC3)OCC)=O)CC2)ccc2[nH]cc(C#N)c2c1 C1(Cl)(C(N(CCN(C(=O)C(O)C2CC2)C)C)=O)CC12CCC2 N1(C(CC)=O)CCC(c2ccc(NC(=O)C(C)C3(O)CCC3)nc2)CC1 C1(C(=O)OC)C(C)CCN1C(C1C2CN(C(C3CCCN3C(C)C)=O)CC12)=O n1(CCC)cc(CCCNC(N2CC(c3ncc(C(=O)OCC)o3)C2)=O)cn1 CCC(CC)C(C)C(=O)N(C1CCCCC1NC(=O)Cc1c(C)nn(C)c1Cl)C C(CN=c1nc2c(ncn2C(C)C)c(NNCC2CC(N(C)C)C2)[nH]1)OCCC c1(CNc2c(C)cc(NC(=O)C(C)CN(C)C)cc2)c(C)sc2ccc(Br)cc12 C1(CNC(c2cnc(CC)nc2O)=O)CN(C(C2OCCCO2)=O)C2(CCC2)C1 Cc1cnc(Cl)nc1N1CCOCC(NC(C2C3CCCC23)=O)C1 C1(N(C(C=COCC)=O)CCOC)CCN(C(C2CN(C3CCCCC3)C2)=O)CC1 C(=O)(CS(=O)(=O)C(C)C)N(C1CN(C(c2nc(OC)c(F)cn2)=O)CC1(C)C)C c1(C(N(CC(C)NC(c2cocn2)=O)CC)=O)cc(C(N)=O)cs1 C1(C(=O)Nc2c(CC)nccc2)CCCCN(C(=O)CS(=O)(=O)NC)C1 N1(C(c2n(C)ccn2)=O)CC2(CCCC2CC(=O)NCC(N)=O)C1 N1(C(c2cnc(OC)nc2)=O)CCc2ccccc2C1CNC(=O)CSC(F)(F)F C1(CNC(C2C(OCC)C2C)=O)CCN(c2ccnc(COC)n2)C12CC2 N1(C(C(=O)NC(c2ccc(F)cc2)CF)=O)CC(O)C2(CC2)C1 C(=O)(C(O)CCCNC(C1CC2CC(=O)C1C2)=O)NCCCC(C)(C)C CC1CN(C(C2(c3cccs3)CC2)=O)CCN1C(C1CC1c1ccccc1)=O c1(C(=O)NC2C(C)CN(C(c3cnsc3)=O)CC2C)cc(O)c2ccsc2c1 C12(NC(c3cc(Cl)nc4n[nH]cc34)=O)CCCCC1CN(C(C1CCCO1)=O)C2 c1(C(N2C3CC(NC(C4C(C)(C)C4)=O)C2CC3)=O)cncc2ccccc12 N1(C(c2cc(CN(C)C)on2)=O)CCCC(F)(CNC(c2snc(O)c2Cl)=O)C1 c1(N(c2nc(C)cc(OCC)n2)C(c2csc(Br)c2)=O)ccc2c(c1)CNCC2.O Cc1cc(O)ccc1CC(=O)NC1(C)CC(NC(=O)C(C)(C)C2CCOC2)C1 CC(C)C(C)(C)C(=O)N1CCCC1CNC(c1cc(-c2cccc(F)c2)no1)=O N1(C(CC(=O)OC)=O)CCCCC(NC(=O)C(c2csc(C)n2)=O)C1 N1(C(C2CCC(F)(F)C2)C)CCC(O)(C#CBr)CC1 CC(O)C(F)(F)C(=O)NCC(CNC(C1SCCCS1)=O)C(F)(F)F N1(C(C(C2CN(C(c3n(CC)ccn3)=O)C2)OC)=O)CCOCC1CO C1(CNC(C2(C(=O)OC)CC2C)=O)CC2(C1)CN(C(c1nnn(C)c1C)=O)C2 CCCCC(C(=O)N(CC(C)NC(=O)C(C)(C)COCC)CC)C(C)C C1(C(C)OC)CN(C(=O)C(C)SC)CCN1C(=O)CC1CCN(C(=O)OC)CC1 CCCC(CCC)C(=O)Nc1ccc(C2CC2(F)F)cc1 C(CC(=O)NC(C)(CC)C1CC1)(C(F)(F)F)NC(c1c(CC)cccc1)=O c1(C(C)SCC(=O)Oc2cccc(C(C)NC(C)C(=O)O)c2)ccc(Br)cc1 Cc1cc(C(=O)NCCN(C2CCCC2)C(=O)CC2CC23CC3)c(O)nn1 c1(C(N2CC(CCNC(C(CC)=CC)=O)OC(C)C2)=O)cnc2ccnn2c1 C12(NC(c3ccc([N+](=O)[O-])o3)=O)COC(C1)C(NC(=O)C(F)n1ccnc1)C2 c1(OC)cnc2ccc(C(=O)NC3CS(=O)(=O)CC3NC(=O)CCCF)cc2n1 C(=O)(C(C(C)C)NC(=O)Cn1nnnc1C)N1C(CCCC)CCC1 Cc1ccc(C(C)C(=O)N2CC(N(C)C(C3CCOC3C)=O)C2)cc1 c1(-c2cn(CC(CCNC(=O)CCC3CCC3)F)nn2)ccc(C2CCC2)cc1 Cc1cnc(C(N2CC(NC(=O)C(F)CC3CC3)CC2C)=O)c(O)c1 c1(C(N(C2CCN(C(C3(C(C)(C)C)CCC3)=O)C2)C)=O)c(F)ccc2occc12 N1(C(C(C)SC(F)(F)F)=O)CCN(C(=O)CCCc2cccnc2)C(C2CC2)C1 N1(C(C2C(C(C)(F)F)C2)=O)CCC(NC(=O)Cn2nnc(C3CC3)n2)C(C)(C)C1 N1(c2nc(CC)cc(CC)n2)CC2CCC1C1CN(C(=O)C3CC3)CC21 C1(C)(CCC(=O)NCCC=CCCC)CN(C(c2ccc(C)o2)=O)C1 N1(C(C(C)OC2CCCC2)=O)CCCN(C(=O)COc2ccccc2)C(C)C1 C123CCC(CC1)(CC2)C(=O)N3.N#Cc1cncc(NC(C2CC2(F)F)=O)c1 c1(CNC(c2cn(C)nn2)C)cnccc1-c1ccccc1 S(=O)(=O)(c1ccc2c(c1)CCCC2)N1C(C)c2ccc(C#N)n2CC1 C1(NC(c2cc(OC)ncc2)=O)CC2CC(NC(C3(OC)CCOCC3)=O)CC12 C1(C(=O)NC2CCCOC2)(NC(c2ccc[nH]2)=O)CCCC1 c1(C(C)NC(c2cc(N(C)C)ccn2)c2nnnn2C)cc(F)c(Br)cc1F c1(OCC)nc(N(C)CC2CCCCN2C(c2occ3c2CCC3)=O)ncc1C C(=O)(CC(O)C(Cl)(Cl)Cl)NCCCCNC(c1cc(C(=O)OC)c(C)cc1)=O c1(C(=O)NCC2(C)CCCN(C(c3cnc(C)s3)=O)C2)ccc2c(n1)OCCO2 C(=O)(C(C)C(F)(F)F)N1CCC(C(=O)NCCCP(C)(C)=O)(CC)C1 Cn1nnnc1SCCCCNC(CC(F)(F)F)=O.C123CC(C1)(C2)C(=O)N3 C1(C(=O)NOCCOC2CC2)CCCN(C(=O)C#CC2CC2)C1 CC1CCCC=C1C(=O)N1CC(c2ocnc2CNC(=O)CN2CCC(C)C2)C1 C1(C)(C(=O)NC2C(NC(C(C)OCC(C)C)=O)CCCC2)CCN(C)CC1 c1(C(=O)NC2(C)CN(C(=O)CN3CCOCC3=O)C2)cc(C2CC2)oc1C1CC1 C1(NC(c2cn(CCOC)nc2)=O)CCN(C(=O)C(Br)=C(C)C)CC1C C(C(C)N=c1nc2scnc2c(NCC(Br)=C(C)C)[nH]1)OCC N1(C(c2cc(-c3nc(C)sc3)cn2C)=O)CCC(C)(NC(=O)C2=CCC2)CC1 C1(C(=O)NCCC2(COC)CC2)(CNC(=O)Cc2c[nH]nc2C)CC2(CC2)C1 C1(C)(NC(CC2CCCC(OC)C2)=O)CCN(C(=O)Cc2cncn2C)CC1 C1(CCNC(c2c(OCC)ccs2)=O)CCN(C(=O)C2=CCC2)C(C)C1 C1(NC(CN(C(c2cc(COC)on2)=O)CC)=O)CCC12CCCC2 CC1CCN(CC(=O)NCCCN(C(C)C)CC2CCCC(C3CC3)O2)CC1 C1(C)(NC(C(C)CF)=O)CCN(C(=O)CC2CCCC(C#N)C2)CC1 N1(C(c2c(C)ccc(Br)c2)=O)CC2CC1CCC2NC(=O)COC1CCC1 c1(C(N2CCC(NC(CCCNC(N)=O)=O)CC2)=O)n[nH]c2c1CCOC2 C1(Nc2nccc(C)n2)CCCN(C(=O)C(CO)c2ccccc2)CC1 C1(NC(CN(C(=O)CC2COCC2O)CCOC)=O)(CO)CC2CCCC12 N1(C(c2cnc(CC(C)(C)C)s2)=O)CCN(C(=O)C=C2CCCC2)CC1CO C(=O)(C(C)S(=O)(=O)c1ccc(F)cc1)NC1CCC(NC(CC(C)C)=O)C1 N1(C(c2cnn(CC)c2Br)=O)CC2CCC1C(CNC(C1COC1)=O)C2 CCC(O)C(F)(F)C(=O)NCC1CCC(NC(C2(S(C)(=O)=O)CC2)=O)C1 c1(NC(C2CCN(C(C3(C(C)C)CCC3)=O)CC2O)=O)c(Cl)cc(Br)c(Cl)c1Br CC(C)CCC(C)OC(N1C(C)(C(=O)NCc2ccccc2)CC1)=O CCC(C(=O)N1CCN(C(c2cn3c(n2)CCC3)=O)CC1CCOC)C(C)C c1(Nc2c(OCC)cccc2C)nc(Cl)c2c(n1)COC2 C(=O)(CC(C(F)(F)F)P(C)(C)=O)NC1(C)CN(C(C23COCC2C3(F)F)=O)C1 C1(NC(C2(C(C)(C)OC)CC2)=O)CC(C(=O)NOCCCN(C)C)CC1O C(=O)(CCC(C)C#N)N1CC(CNC(CC(n2c(CC)ncc2)C)=O)(OC)C1 C(=O)(C1OCCc2c(O)cccc21)NCC=CCNC(CCC(C)(C)C)=O c1(C(=O)NC2CC3CN(C(CNC(=O)NC)=O)CC32)ccc2cc[nH]c2n1 C1(C(C)NC(c2cnn(C)c2)=O)CCN(C(=O)COC(C)(C)C)C1 C12(C(=O)NC3C(NC(C4(CC#C)CC4)=O)CCOC3)CCC(N=[N+]=[N-])C1C2 C1(CCCC)(C(=O)NC2(CC(=O)NC(C)CSC(F)F)CC2)CCC1 O=S(=O)(c1ccc(NCc2c(F)cccc2F)c(Cl)c1)N1CCC2CC12 C(=O)(C1Cc2ccc(Cl)cc21)N1CCC(C(C)NC(COCCSC)=O)C1 N1(C(C2CCC(CNC(C3(OCC)CC3)=O)O2)=O)CC2CCCC2C1 C(=O)(CCC(=O)CC)NC(CCOCC)C(=O)N(C)CCC1CCCN1C c1(C(=O)NC2CC(NC(c3cc(C)c(O)nc3)=O)CC2O)ccc2sccc2c1 CC(CCCNC(=O)C(C)CO)NC(c1cnn(C2CCC2)c1)=O c1(OC)ccc(Cl)cc1CC(=O)NC1COCCC1NC(C1(C)CCC(=O)N1)=O N1(C(C=CC)=O)CC2(CCCC(CNC(c3cc(-c4ccccn4)[nH]n3)=O)O2)C1 N1(C(C(C=C)O)=O)CC2CCC(C1)N2C(c1ccc(C(C)C)cc1)=O c1(C(N2C3CC(NC(C(OC)OC)=O)C2CC3)=O)n[nH]c2c1CC(C)CC2 c1(OCC#N)ccc(CC(N2CC(CNC(=O)C=Cc3cncs3)C2)=O)cn1 C1(C(=O)NC(C)C2CC2)CN(C(=O)CSCCC#N)CC(C)(C)C1 O=S(=O)(c1ccc(N2CCC(Cc3ccccc3)C2)nc1)NCCN1CCCC1 CC1(C)CN(C(C2CCC3(CCC3)C2)=O)C(CNC(c2cnc[nH]2)=O)CO1 CC1CC(NC(=O)CC23COC(C)(C2)C3)CCN1C(=O)Cn1cc(F)ccc1=O n1(CCC(=O)NCC2N(C(c3nc(C)n(C)c3)=O)CCCC2)cc([N+](=O)[O-])cn1 c1(CCNC(C2C(C)C2C)=O)ccc(CNC(=O)C(F)n2cccn2)cc1 N1(C(Cc2cc(C)on2)=O)C2CCCC1CN(C(C1(C)CC(C)(C)C1)=O)CC2 C1(CNC(CCCCOC)=O)CN(C(C2C(C)C2C)=O)CCC1(C)C C1(C)(CCC)CCN(C(c2ccnc(CNC(=O)Cn3cccn3)c2)=O)C1 C1(C(N(CC#C)CC)=O)CCN(C(C2(CCC)CC2)=O)CCO1 c1(C(=O)NCC2OCCN(C(CC=CCC)=O)C2)ccc(I)c(F)c1 c1(C(N2CCCC(C)CC2)=O)ncn2cc(NC(=O)C(F)(F)Cl)ccc12 C(=O)(CCCCF)N(C(CNC(CC(C)N(C)C)=O)C)C CCC(C)(C)C(O)C(=O)NC(C)CCN(C)C(c1ccc(=O)oc1)=O c1(C(C)NCc2nc(C3(CCO)CCOC3)no2)coc2ccc(Cl)nc12 C(=O)(CC1=CCCCC1)N1CC(C)(C(=O)NCc2c(C)nco2)C(C)C1 C12(C(N3CC(CC)C(F)C3)=O)CCC(CC1)N(C(=O)C(CC)(CO)OC)C2 C1(O)(C(C)NC(C=CC(C)C)=O)CN(C(=O)C(c2ccccc2)NC(N)=O)C1 c1(NC(c2csc(NC(c3ccsc3)=O)n2)=O)cccc(S(=O)(=O)O)c1 Cc1ncc2n1CC(C(=O)NC1CCCN(C(=O)CNc3ncccn3)C1)CC2 C(=O)(C(O)C(F)(F)F)NC(CSC)(C)C(=O)N(CC(=O)NC(C)C)C Cc1cnc(NC(C)CC(N)=O)c(S(=O)(=O)N2CCCC(C(F)(F)F)C2)c1 CC(C)CCCC(=O)NC1CCC(CC(=O)NC23CCC(C2)OC3)C1 c1(OC2(C(N3CC(C)(NC(C4C5CCCC45)=O)C3)=O)CC2)cc(F)cc(F)c1 N1(C(C(C2CCN(C(C3(CC#C)CCC3)=O)C2)C)=O)CC2CC2C2CC12 C12(NC(=O)Cc3cccc(O)c3)COC(C1)C(NC(C1CCCC13CCC3)=O)C2 N1(CC)CCN(C(c2cccc(CN(CCCC(=C)C)C)c2)=O)CC1 C(=O)(C1CCc2c(Cl)cccc21)N1C(CNC(c2cnc(O)o2)=O)CC2CC21 C1(CC#C)(C(N2CCCC(c3ccccc3)C2)=O)CCCCC1.c12nnnn1C2 CCC(F)(C(=O)OC)C(=O)NCC12CCCC1CN(C(c1cc(C)ccn1)=O)C2 c1(OC)ccccc1-c1cn(-c2nc(C(C)C)c(C)o2)nn1 c1(N(C(=O)COCCC(C)C)CC)cccc(-c2c[nH]c(=N)s2)c1 C1(CCCCCNC(CCSCC)=O)CCN(Cc2cccnc2C)CC1 C1(C2CN(C(C(C)Cc3cnc[nH]3)=O)C2)CN(C(=O)C(C)N2CCCC2)CCO1 C1(NC(C=CC)=O)CCC(C)(CNC(c2csc(COC3CCC3)n2)=O)CC1 C(=O)(CS(=O)(=O)CCO)NC1(C)CCN(C(=O)COCCOc2ccccc2)C1 C1(C)(C(N2CC(NC(COCc3ncc(C)o3)=O)C(F)C2)=O)CCN(C)CC1 S(=O)(=O)(C1CCCCC1)N1CCC(NC(C2CN3CCC2C3)=O)CC1 N1(C(C(CC)SC)=O)CCC(C2CC2NC(=O)Cn2cc3ccccc3n2)CC1 C#CCC(C(=O)OCC)NC(=O)COC1CC(NC(C2CN(C)C(=O)N2)=O)C1 c1(C(c2ccccc2)N(C(=O)CCn2cccc2)C)nccn1C C(c1cc(C)ccc1OC)=CC(=O)NC1(CNC(C(CC)OC)=O)CCOC1 C(=O)(CC(CN(C)C)C(F)(F)F)NC1C(C)CN(C(=O)CSC(F)F)CC1 C(=O)(C(CNC(=O)C(c1cnn(C)c1)O)C(C)C)N(CCC#C)C N1(C(C(CC=CC)C)=O)CCCC12CCCN(C(=O)COC(F)(F)F)C2 C(=O)(CC(C(C)C)NC(c1ccncc1)=O)NC(C#C)CCC CC1CCC2(CC2)N(C(c2c(CNC(c3ccc(CO)s3)=O)nnn2C)=O)C1 CCC(C(=O)OC)C(=O)N1CC(F)CC1C(=O)NC1(CCOC(C)C)CC1 C=CC(C)CC(=O)N(C)CC1CC(F)CN1C(c1cc(C2CCC2)[nH]n1)=O C(CCC(=O)NCc1nc(C(=O)N(C2CN(C)C2)C)co1)OC(C)C c1(C(N2C(C)CC(NC(c3nn(C(CC)C)c(C)c3)=O)C2)=O)ccc([N+](=O)[O-])o1 C1(NC(=O)CC2CCOCC2)CCN(C(C2CC2c2ccccc2)=O)CC(O)C1 c1(C(=O)NC2CC(CCNC(c3[nH]cc(C)c3)=O)C2)sc(CC(F)(F)F)nc1C Cc1cc(NC(CCNC(c2cnn(C)c2C(F)F)=O)C(C)C)n2ncnc2n1 CCC(CO)C(=O)N(CC(O)CN(C(=O)CCc1ccccc1)C)C N1(C(=O)NC2CCCN(C(C)C(N)=O)C2)CCN(CC(F)F)C(C)C1 c1(C(=O)NC2CN(C(c3c(C)cnnc3)=O)C(C)C2)ccc2c(c1)CCCCN2 c1(CNC(=NCCC)NCCOC2CCS(=O)(=O)C2)ccc(S(N)(=O)=O)cc1C C1(C(=O)NCCN(C(=O)Cc2cnns2)CCOC)CC=CCC1C C1(NC(CCCCCOC)=O)(CNC(C2CCC(OC)C2)=O)CCC(C)(C)CC1 CC(C)CS(=O)(=O)CC(=O)NCCCCNC(=O)C(c1cc2ccccc2o1)C C(CNC(=O)CS(=O)(=O)NC)(C(C)(C)C)NC(C1N(S(CCC)(=O)=O)CCC1)=O C(=O)(C1=CCCCO1)N1CCC(O)(CCNC(c2c(C)c(C(F)(F)F)n[nH]2)=O)C1 c1(C(=O)NC2CC(NC(Cc3c(C)nccc3)=O)C2)c[nH]c2cc(F)c(F)cc12 C(=O)(N1CC(O)CCO1)C1(CCCN)CCCC1.CC(C)(C)OC(N)=O c1(C(=O)NC2C(CC)N(C(=O)COCC3CCOC3)CC2)ccn2ccnc2c1 C1(NC(C(CC)OC)=O)CC2(CCC(CNC(c3ccn(CCF)n3)=O)OC2)C1 N1(C(=O)COC2CCOC2)CCN(C(=O)C=C(Cl)Cl)C(CF)C1 c1(CN2C(CNC(c3ccc(NC(C)=O)c(Cl)c3)=O)CC2)cc(F)c(Cl)cc1F c1(C(=O)NC2CCN(C(C=C3CCC(C)CC3)=O)C2)ccnc2ccncc12 Cc1nc(C2CCN(C(=O)NCC3COCCN3C3CCCC3)CC2)[nH]c1C Cc1cncnc1C(=O)NCC1(CNC(=O)CC2CC(O)C2(C)C)CC1 C=C(C)CC(C(=O)NC1CCCC1CNC(C1(CSC)CCC1)=O)NC(C)=O C1(NC(C#CC)(C)C)CCN(C(=O)C(CC)OC)CC1 c1(C(N2CC(CNC(C3CCC(=O)NC3)=O)OCC2)=O)cc(Cl)ccc1Cl C1(NC(C=C(CC)C)=O)CCC(CNC(c2ncoc2-c2cnn(C)c2)=O)C1 N1(C(COc2ccc(OCC)cc2)=O)C2CCC1C(C(=O)NCCC1CC1)C2 c1(C(=O)NC2CCN(C(c3c(CC)nco3)=O)C(C)C2)ccc2c(n1)CCOC2 c1(C(C(=O)NC(C)C(=O)N(CC(C)(C)O)C2CC2)C)ccnn1C Cn1c(C(N2CCC2CNC(C2CC(CCO)C2)=O)=O)cc2c(O)cccc12 C1(C(=O)C(=O)NC)(OC)CCCC1.C(C)(C)C=CCNC(=O)OC(C)(C)C C1(CC)(CC)CCCN1C(C1COC(CNC(=O)CCCn2cccn2)C1)=O C(C)(CNC(=O)CCC1CCOC1)(CNC(=O)CCOC1CCC1)OC N1(C(c2c(OC)ccnc2)=O)CCCCC(NC(c2cn[nH]c2)=O)C1 C1(C)(CC(=O)N(CC(C)C)CC(=O)NC2CCSCC2)CCCCC1 C1(C(N2CC(C)C(C)C2C)=O)CC12CCN(C(=O)CC1C=CCCC1)CC2 c1(C2(C(=O)NC(C(CO)NC(C(CC)SC)=O)C)CC2)cncc(Br)c1 N1(C(C(CCCOC)C)=O)CC2(CCCC2NC(=O)C(=O)N(C)C)C1 c1(CCC(C)(C)C)nc(C2CCCCO2)n(C2COC(C)(C)C2)n1 C1(C(N2C(CNC(CCN(CCC(C)(C)C)C)=O)CC2)=O)C2CCCCCC12 Cc1nn(CC(=O)NC2CC(N(C)C(c3cc(C(C)C)[nH]n3)=O)C2)c(C)c1C c1(C(=O)NCC(C)NC(=O)C(c2cccc(F)c2)O)cccc2nn[nH]c12 N1(C(C(C)N(C)C)=O)CCC(c2n[nH]c(CNC(c3cnco3)=O)n2)CC1 C(C(CC(=O)N(CCCC(C)O)C)NC(=O)CCc1nc(C)no1)OC CC(C)S(=O)(=O)CC(=O)NC(c1ccccc1)CNC(c1cc(Cl)c(Cl)[nH]1)=O C1(n2cnnn2)(Nc2ccc(NC=O)cc2)CCCCC1 c1(OC)c(C(=O)N(CCCN(C(=O)C(OC)OC)C)C)csc1Cl N1(C(CNC(CC(C)(C)C)=O)=O)CCC2CC1CN(C(c1cnc(S)nc1)=O)C2 CCC(O)C(C)(C)C(=O)N1CCC(C(=O)NCC2(CO)CC23CCC3)O1 O(NC(=O)C(CCF)NC(=O)C=Cc1cncs1)CC(=O)N(C)C C1(C(C(=O)NC)N(C)Cc2cc(C)ncc2C(F)(F)F)CC(C)CC(C)C1 c1(CN2C(C)(C(N3CCC(C)(C(=O)OCC)C3)=O)CC2)c(F)c(F)cc(F)c1F c1(C(=O)NCC2CN(C(CC)=O)C2)sc2ncc(C(=O)OC)cc2c1C Cc1nc(C#N)cc(=NCC2CCCCN(C(c3cccc(O)n3)=O)C2)[nH]1 C1(C(=O)NC(C2C(C(=O)OC)C2)C)(OC)CCN(C(C2CCC(C)(C)C2)=O)C1 C(=O)(C(C)(CC)CO)NC(CCC)C(=O)NC1C=CCCC1 CC1(C(N2CCOCC(CNC(C3C=CC=CC=C3)=O)C2)=O)CCNC(=O)C1 C1(CNC(C(C(C)C)N(C)C)=O)CC2CCC(C1)N2C(=O)CCCC(=O)N(C)C C(=O)(CCCCC(=O)N1CCN(CC(=O)NC2CCC(=O)NC2)CC1)OC C1(C(N2C3C(NC(=O)C=Cc4ccc[nH]4)C(CC3)C2)=O)CCc2nc[nH]c2C1 [N-]=[N+]=NC1CCC(C(=O)NCC2(C(N)=O)CN(C(=O)CO)C2)CC1 C12(C(=O)NCCCOCCNC(COCC(C)C)=O)CCCC1C2Br c1(C(C)C)ccccc1C(=O)NC(C)C(C)(C)NC(=O)C=Cc1ccnn1C C=C1CCN(C(c2cn(C)c(=O)cn2)=O)C(C(=O)NOC(c2ccccc2)C)C1 N(C1=NC2CCCCC2S1)CCN(C(C)C)CC c1(C(C(=O)NC2(C)CC2)N(CC)Cc2ccncc2)cccc(F)c1C C1(N(C(c2ccc(OCCO)cc2)=O)CC)CCCN(C(=O)Cc2[nH]cnc2C)C1 N1(C(CN(CC=C)C(N)=O)=O)CCC(CC(=O)NCC(=O)NC)C1 O(N(C)C(=O)CNC(=O)C(C1CCN(C(c2nccn2C)=O)C1)F)CC C1(NC(=O)NC2(C=C)CCOCC2)CCC2(CCCC2)C1 C#CC1(C(=O)NC2CCCCC2CC(=O)NCC2CCOC2)CCCC1 C1(NC(c2cc(C3CCC3)[nH]n2)=O)CN(C(C2CC=CCC2)=O)CC12CCC2 N1(C(c2cccc(OC)c2)=O)C2CCC1CC(N(C(=O)C(C)(O)C1CCC1)C)C2 c1(C(=O)NC2CCC(N(C)C(C3CC(N(C)C)C3)=O)CC2)c[nH]cc(F)c1=O C1(CNC(C2CCCN(CC)C2)=O)CN(C(=O)C=CC2CCCC2)CC(C)(C)C1 C12(NC(c3c(CC)ncs3)=O)CC(CNC(=O)C(F)OC)(C1)OC21CCOCC1 c1(C(=O)NCc2cc(C)n(C)n2)cnn2cc(-c3ccc(O)cc3F)ccc12 c1(C(=O)NC2CC3CC(NC(CCC)=O)C2C3)cnc2c(C#N)cnn2c1 C(=O)(C(C)(F)CS(C)(=O)=O)N(CCCN(C(C(C)N(CC)CC)=O)C)C C(c1ccccc1F)=CCC(=O)NCC1C(NC(=O)C=C2CCC2)CCCC1 N1(C(c2cc(OC)c(F)c(F)c2)=O)CCCC(N=c2ccnc(C3CCC3)[nH]2)C1 CC1(C(N2CCC(c3cnn[nH]3)C2)=O)CCCN(C(C2CNC(=O)N2)=O)C1 C1(CC(=O)OCC)CCC2(CC1)CCN(C(c1cccc(Br)c1)C(N)=O)CC2 C1(CNC(CSC)=O)COCC1n1cc(CNC(=O)CCC2CCC(C)O2)nn1 C1(C(=O)OC(CC#C)C(=O)N(C(=O)CS(=O)(=O)C2CC2)CC)CCc2[nH]nc(O)c2C1 C1(NC(CCCNC(N)=O)=O)COCCN(C(C2CCC=CCC2)=O)C1 C1(C(=O)NCC(F)Cl)(NC(CCOC(C)=O)=O)CCCCC1 C12(C(N)=O)CCCCC1(n1cc(CN)nn1)CN(C(=O)CCS(=O)(=O)C1CC1)C2 C(=O)(CCS(C)(=O)=O)N(C1CCN(C(=O)C(F)(F)c2ccnn2C)CC1)CCC C1(CNC(C2(C)CCN(C(C)=O)C2)=O)CCN(C(=O)Cn2cncn2)C12CCC2 N1(Cc2c([N+](=O)[O-])ccc(OC)c2)CCc2c(C)cc(C)cc2C1 C1(NC(=O)NCC2C(C3CC3)C2(F)F)CC(CO)C12CCC2 N1(C(c2ccn(C(C)C)n2)=O)CC(CNC(c2cn(C)nc2C2CC2)=O)CC1C c1(C(=O)NCCCC(C)NC(C(F)=C(C)C)=O)ccc(=O)n(C2CC2)c1 C(=O)(C(C)(C)C(=O)NC1CCCN(C(=O)C(C)CC=Cc2ccccc2)CC1)OCC C12(CNC(=O)CSc3cccc(Cl)c3)CCC(CC1)N(C(C1(O)CCSC1)=O)C2 N1(C(C(Cc2cnc[nH]2)NC(c2c(C)nns2)=O)=O)CCC(O)CC(C)(C)C1 C1(NC(=O)Cc2nc(C3CC3)cs2)C2COCC1CN(C(=O)C1=COCCC1)C2 C12(C(=O)NC3CCC(CCNC(=O)CNc4ncccn4)C3)CCN(CC1)C2 N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCC2C(C1)NC(=O)CN2C(C1CCS1(=O)=O)=O CCC(CC1CCCCC1)C(=O)N(C)CC1CCCN1C(=O)COC(C)C C1(CNC(Cc2nc(C)sc2)=O)CN(C(=O)Cc2ccc(O)nc2)CCO1 C1(NC(C(C)C2CCCO2)=O)CS(=O)(=O)C12CCN(c1nnc(C#N)s1)CC2 C1(C(=O)NCC(CC)NC(c2c(N)ccc(CC)c2)=O)CCCC(F)(F)CC1 CCCC(C)(CC)C(=O)NC1CC2CN(C(=O)C=C(C)c3ccco3)CC12 CCCCC(CC(=O)N1CC=CC1(C)CO)NC(=O)CC#N N1(C(c2n[nH]c(C)c2Br)=O)CCCC(CCNC(C23CCC2C3)=O)CC1 N1(C(C=C(C)C)=O)CCC(NC(c2cc(Cl)ccc2Br)=O)C(CO)CC1 c1(C(=O)NCC2C(CNC(C(CC)=CC)=O)C2(F)F)ccc(C)nc1N C1(C(N(CC(C)NC(c2coc(Br)n2)=O)C)=O)CC(O)CN1C N1(C(C=CCN(C)CC)=O)CCOC2CN(C(c3ccc(S(C)(=O)=O)s3)=O)CC12 c1(C(=O)NC(C(C)C)CCN(C)C(C2(O)CC2)=O)cc(F)ccc1Cl C(CN=c1[nH]c(C)cc(=NC2CC2c2ccsc2)[nH]1)n1ncc(CC)c1 CC(C)CC(C)(O)C(=O)N(C)CC1CCN(C(=O)C=Cc2cn(C)cn2)C1 c1(SC(C(=O)N(CCNC(C2CC(OC)C2)=O)CC)C)ccccc1Cl C=CC(C(=O)N1CCC1CC(=O)NCc1cc(CC)co1)OCC c1(C(N(CC(CN(C(c2c(C(=O)OC)c[nH]n2)=O)C)O)C)=O)cc(C)cc(C)c1 Cc1nccc(Cl)c1C(=O)NCCN(C(=O)C(F)C1CCOC1)C C#Cc1cncc(C(=O)NC2CCN(C(c3cnc(Cl)[nH]3)=O)C23CC3)c1 c1(C(N2CCCC(CNC(CCCC(N)=O)=O)C2)=O)ccc(Cl)c(Cl)c1N Nc1ccc(C(=O)NCC(O)CNC(c2ccnnc2Cl)=O)cc1O N1(C(C(=O)N(C(CCCC)C)c2ccccc2)=O)CC(C)OC2(CCCC2)C1 c1(C(=O)NC2CN(C(c3cn(C)nc3Cl)=O)CC23CC3)cc(Cl)cc2c1CCC2 Cn1c(C(=O)NCC2CC(F)(CNC(=O)C(=O)NC3CC3)C2)cc2ccccc12 c1(NC(C2N(C)CCN(C(CC(=O)NCC)=O)C2)=O)cc(C)c(F)c(C)c1 C(=O)(C1=CC2(CCOC2)C1)N1CC(C)C(CNC(C2(c3cnn(C)c3)CC2)=O)C1 N1(C(C2(COC)CC2)=O)CCC(C)N(C(=O)Cn2[nH]cnc2=N)CC1 C1(NC(c2ccc(OCC)nc2)=O)CC(C)CN(C(C2CC3C=CC2C3)=O)C1 C(=O)(C1=CC2(CCN(C(c3cc(C4CC4)on3)=O)C2)C1)NCC(N)=O N1(C(c2c(CC)con2)=O)CCOC(C)(CNC(=O)C(C)OCC(C)C)C1 N#Cc1c(NCCCCNC(c2cscn2)=O)nnc2c1CCCC2 C1(CNC(CCNC(c2ccoc2)=O)=O)CCCN(C(C2CCCO2)=O)C1 N1(C(c2cc(C(N)=O)[nH]c2)=O)CCOCC1CCNC(=O)CC(F)(F)F CCC(CC(=O)NC1COCC1CNC(c1ccccc1NC)=O)SC C1(C(=O)OC)CCC(C(=O)NCC2(O)CN(C(c3coc(Cl)n3)=O)C2)CC1 N1(C(CCC#CC)=O)CCN(C(=O)C(C)Sc2nncn2C)C(CCO)C1 C=C(C)C(C)(O)C(=O)NC(CNC(c1ccc(F)cc1SC)=O)C1CC1 Cc1ccc(N)c(C(N2CCCC2C2CCN(C(=O)C(C)S(N)(=O)=O)C2)=O)c1 c1(OC)cc(CNC2CC(NC(c3ncc(Cl)cc3C)=O)C2)ccc1OC(C)=O C(C(=O)Nc1cccc(CNC(=O)Cc2cnoc2)c1)(C(C)C)NC(C)=O c1(C(=O)NCC#CCNC(c2ncn(CC)c2)=O)ccn2c(C)cnc2c1 CC(CC(N)=O)C(=O)NC(CNC(c1cccn(C(C)(C)C)c1=O)=O)CO N1(CC(C)C)CC(C(N2CCC(N(CCO)C(c3ccsc3)=O)C2)=O)CC1=O n1(C(CC)CC)ccc(C(=O)NC2CC2CNC(=O)CCc2nc[nH]n2)n1 N1(C(CC(COC)C)=O)CC2CCC2(NC(c2nc(-c3cccs3)oc2C)=O)C1 C(=O)(CCS(=O)(=O)c1ccc(F)cc1)NCC(C)(CNC(=O)C(C)C(C)C)OC C(CCCC(CO)NC(=O)C=C1CCCCC1)NC(c1c(NC)cnnc1)=O c1(C(=O)NCC(CN(C(c2nc(COC)oc2)=O)C)O)cc(F)cc2c1CCC2 N1(C(c2cccc(C(N)=O)c2F)=O)CC2(CC(NC(C3CC3C(F)F)=O)CO2)C1 c1(N2CC3CC(CNC(C(CC)(C)OC)=O)C3C2)cnc2ccccc2n1 c1(C(N2CC(F)CC(NC(=O)CC3CCCO3)C2)=O)cnc2c(c1)C(=O)CCC2 N1(C(Cc2ccc(OC)cc2C)=O)CCC(NC(=O)CSSC)C12CCCC2 N1(C(C2(C=C)CCC2)=O)CCN2C(=O)C(NC(=O)CCCc3ccsc3)CC2C1 C1(NC(C2(CCOC)CC2)=O)CCOC(C(=O)NC(C2CCCC2)CO)C1 C(=O)(CCCCCn1cc(CN2CCC(O)CC2)nn1)NCCC(=O)NC(C)C Cn1nc(C2CC2)cc1CC(=O)NCC1C2CC1N(C(c1coc(SC)c1)=O)C2 c1(CNCCN2CCN(C(C=CC)=O)CC2)c(Cl)cc(C)cc1Cl C1(NC(c2scc(OC)c2)=O)CCC12CCN(C(c1nccn1C)=O)CC2 C(=O)(C1=CC2C=CC(C1)C2)N1C(CONC(=O)COC2(C)N=C(C)SC2)COCC1 C1(CC)(NC(=O)C(C)NS(=O)(=O)CC)CCCN(C(=O)Cc2ccc(O)cc2)C1 C1(n2cc(C(N3CC(F)(CO)C3)=O)nn2)CCCN(c2ccccn2)C1 c1(C(=O)OC)cccc(C#Cc2cccc(NC(C3(NC(C)C)CC3)=O)c2)c1 CCCC(C)C(CO)NC(C1CC2(CC(NC(=O)CCOC3CCCC3)C2)C1)=O c1(C(=O)NCC(CC)NC(c2cc(=N)[nH]c(Cl)n2)=O)cncc(OC)c1C C1(OCC#C)CCCN(C(=O)C(C)CNC(=O)CSC(F)(F)F)C1 Cc1cc(N)ccc1C(=O)N(C)C(c1cn(-c2cccnc2C(F)(F)F)nn1)C C(C(C)(CC(C)C)NC(=O)C=C=C(C)C)NC(c1c(OC)nccc1)=O Cc1csc2c(C(=O)NCC(C)CC(C)O)cccc12 C(=O)(CC(C)C(C)C)NCC(CCCC)NC(=O)C=CCCC(C)C C1(O)(C(C)NC(=O)C(Cl)=CCl)CCN(C(c2cc(N)ccn2)=O)C1 c1(NC(C2(c3cccc(-c4c(O)cccc4O)c3)CC2)=O)nc2c(s1)CCCC2=O CC(C)C(O)C(O)C(=O)NCCCN1CC(C)OC(C)C1 C1(C(=O)NCCCC(=O)NC)CC(CNC(=O)OC(C)(C)C)CN1C(=O)C(C)C#N C(=O)(C1=C(Cl)CCC1)NCC1CC(=O)NC(=O)N1.CC12CCN(C1)C2=O N1(C(c2ccc(OC)cc2)=O)CCC2C(CCCN2C(C2(C)CC=CCC2)=O)C1 CC(C)C(C(=O)NCC(C1CC1)NC(c1cnc(CC(F)F)s1)=O)n1cccc1 N1(C(CC(C)C(C)(C)NC(=O)CCC(C)(C)C#N)=O)CCC2(CCOC2)CC1 C1(CCOC)(C(=O)NCCF)CCN(C(C2CC2C(N)=O)=O)CC1 Cc1ccc(N2CCCC(C(=O)NC3CC3NC(c3csc(O)n3)=O)C2)nc1 C(=O)(C(F)(CNC(=O)COC1CCOCC1)C(C)C)N1C(CCOC)CCCC1 c1(N2CCC(N(C(C3C(=C)C3)=O)CCC)CC2)ncnc2ccccc12 c1(C(N2CCCC(C(=O)NCC(CCCC)O)(CC)C2)=O)c[nH]c2cnccc12 c1(C(=O)NCCCN(C(C(c2ccccc2F)C)=O)C2CC2)nc(Cl)sc1Cl C(=O)(CC(=O)NC1CC1)N(C)CCn1cc(C2CCOC2)nn1 c1(C(C)C)nc2cccc(C(=O)NC(C)(C)CNC(=O)CC3CCC(C)O3)c2[nH]1 Cc1ncnc(C)c1CC(N1CCC(C)(NC(C23CCC2C3)=O)C1)=O C(CCN=c1[nH]c(N2CCc3oc(C)nc3C2)nc2c1CCCC2)NCCOC Cc1ccc(F)cc1CN(C1CCNC1=O)C(=O)NC(c1cccc(F)c1)CO CCCCC(C)CCC(=O)NC1CCC12CCN(C(=O)C(C)(C)CC(F)F)CC2 CCC(C)C(O)C(C)C(=O)NCC1CN(C(C2(O)CCCC2)=O)CC12CC2 C1(CNC(C2N(C(C(C=C)O)=O)CC(O)C2)=O)CCCC2(CC2)C1 C1(CCN(C)C(C2CCC(=O)NC2)=O)CCCCN1C(c1ncn(C)n1)=O c1(C(=O)CN2CCCC(C3CCCCO3)C2)ccc(I)cc1OC(F)(F)F c1(CN(CCC)CCNC(c2c[nH]nc2-c2ccccc2)=O)ccc(F)cc1F Cn1ccc2cccc(CNc3ccsc3C(=O)NC3CNC(=O)C3(C)C)c12 Cc1ncc(-c2noc(C(Cc3c(Br)csc3C)C3CC3)n2)c(C)n1 C(=O)(CC(C)C1CC1)NCCCN(C(=O)CNC(=O)C1CC1)CCC c1(CC(=O)NCC(C)CNC(=O)CCN(C)CCO)csc(-c2nc[nH]n2)n1 C1(NC(CC(C)(F)F)=O)CC(NCc2ccc(Cl)cc2)C12CCC2 N1(C(C(C(C)C)n2cccc2)=O)CCC(NC(=O)CC(C)n2cccn2)C(F)C1 N1(C(c2ccc(C)c(Cl)c2N)=O)CC(NC(C2(O)CCOC2)=O)CC2(CCC2)C1 C(=O)(C(C)(C)n1ccc(C)n1)N(CC(CNC(CC1(C=C)CC1)=O)O)C N1(C(=O)NCCOC2CCCC(C)C2)CCC(CC(=O)O)(CC2CC2)CC1 C#CCCC(C(=O)N1CCOC(CCC)C1)NC(c1cc(CC)no1)=O Cc1cc(C(=O)NCC(c2ccccc2F)NC(c2cscn2)=O)ccc1Cl c1(C(N(C2(CC(=O)NCCS(N)(=O)=O)CC2)C)=O)cc(C#N)c[nH]1 C1(F)(C(N2CCC(NC(=O)C(F)CC3CCC3)CC2)=O)CS(=O)(=O)CC12CCC2 N1(C(C(C)n2cccc2)=O)CCN(C(=O)C=C2CCCCC2)C2CCCCC12 N1(C(CCOCCOCC)=O)CCC2(NC(c3cnc(Cl)cn3)=O)CCCC12 C(=O)(C(Cc1cccc(Cl)c1)CCCO)NCC(=O)Nc1cc(N)cc(F)c1 CC1CCCCCCN1C(=O)C(C1CCN1C(=O)OC(C)(C)C)NC(N)=O C(=O)(CCS(=O)(=O)NC)N(CC(N1CCCC1)=O)C.C12CCCC(C1)N(CC(=O)O)C2=O C1(N(C(C(C(C)C)C)=O)C)CCCC2CN(C(C3CCCC3F)=O)CC12 C1(OC)CC(CNC(c2cccc(C)c2)=O)N(C(c2cc(C)sc2C)=O)C1 C(=O)(C(F)(F)C(F)F)N(C1CN(C(=O)CCc2ccccc2)CC1F)C N1(C(C=COCC)=O)CCC(=CCNC(C2ON=C(C)C2C)=O)CC1 C(=O)(C(C)(C)C(=O)N1C2CCC(C2)C1C(=O)Nc1cnn(C(F)F)c1)OC C1(CC(=O)NC2(CN(C(CN(C)CCO)=O)C)CC2)CCOC1(C)C C(=O)(CCC(C)NC(=O)Cc1sccc1C)N1CCC(COCC)C1 c1(CN(C(c2cccc(-n3cnnn3)c2)=O)CC23CC(CO2)C3)cncc(O)c1 C1(C)(CNC(C(F)OC)=O)CC(F)(F)CN1C(C1CC2(CC(=O)N2)C1)=O Cc1ccc(S(=O)(=O)N2CCC2(C)C(=O)Nc2cc(C(F)(F)F)nn2C)cc1C C(=O)(CCCC(=O)NC(C)C)NC(C(C(C)C)NC(=O)Cn1ccc(C(F)F)n1)C CC(C)CC(CC(C)C)C(=O)N(C)CCOCCNC(=O)C(C)(C)C1CCCO1 C1(CC(=O)NCCn2cncn2)CSCCO1 C(C)(CN=c1nc2c(cnn2C)c(N2CCOC(C)(C)C2)[nH]1)(C1CCOCC1)OC c12cc(no1)C(=O)OC2=O.c1(C(N(CCOC)C(C)C)=O)cn(CCCF)nn1 C(=O)(CCCOCCN(C)C)N(CC(=O)NCCCF)C(C)C N1(C(CC2N(C)C(=O)CC2)=O)CCN(C(=O)Cc2ccccc2Cl)CC1C1CC1 N(C(=NCCC(C)F)NC(C)Cc1ccccc1)Cc1nc(CC)sc1 Cc1cc(CNc2cc(Cl)ccc2NC(c2ccccc2Br)=O)c(C)n1C1CC1 N1(C(CN(C)CC)=O)CCN(C(C2C=CCCC2)=O)CC1CCO c1(C(=O)OCC)cc(Br)cc(F)c1NC(N1CCN(C(C)(C)C)CC1)=O C1(CNC(C2CC3(CSC3)C2)=O)CN(C(=O)Cc2ccnc(O)c2)CC12CC2 Cn1nccc1-c1cn(CC(=O)NCCC2(C(=O)C3CC3)CC2)nn1 CC(C)CCC(=O)N1CC(O)(C2CCCN2C(=O)CCNS(C)(=O)=O)C1 c1(CC(=O)NCC2(CN(C3CCCC3C)CC)CC2)cnn2c1CCCC2 N1(C(c2c(C)cc(C(=O)OC)o2)=O)CCCCC(NC(c2ccnc(S)c2)=O)C1 c1(C(N2C(C)(C(C)C)CC2)=O)ccc(CNC(=O)COC2CCCCC2)cn1 N1(C(C)=O)CC(O)CC1C(=O)NC1CN(C(=O)CO)CC1F CCC(CC(F)(F)F)C(=O)NCC1(C)CCN(C(c2ccc(C(F)F)nc2)=O)C1 c1(OC)ccc(CCNc2cc(NCC(n3cccn3)C)ncn2)cc1Br N1(Cc2nc(COC)sc2)CCC2C1CCCN2C(=O)CO N1(C(c2ccc(C)nn2)=O)CCC(C)(C)C(C(N2CCC(C(C)(C)C)CC2)=O)C1 C=CCC(C)(C)CC(=O)N1CCOC(C(=O)NC(C)CC2CCC2)C1 CC(C)(C(=O)NCC1CCC(NC(c2cc(C(F)(F)F)ccn2)=O)C1)C(N)=O S(=O)(=O)(c1ccc(C)c(C)c1)N1CC(NC(c2nc(C)oc2)=O)C(C#N)C1 C12(C(=O)NCCCCC3CN(C(=O)COCC(F)(F)F)C3)CCC(CC1)CC2 CC(O)CCCC(=O)NC1(CNC(c2n[nH]cc2Cl)=O)CCC1 c1(C(N2C3CC(NC(=O)Cn4ccnc4)C(C3)C2)=O)c[nH]c2ncccc12 c1(OC)ccc(SC)cc1NC1(c2nnnn2-c2cccc(Cl)c2)CCCC(C)C1 N1(C(C2(OC(C)=O)CC2)=O)CCN(C(=O)CC2CCCOC2)CC(C)(C)C1 CC(C(=O)NCC1CN(C(=O)CCC2CCCN2C)C1)C(F)(F)F C#CCC(C)C(=O)N1CCC(C)(CCNC(=O)CN2CC(=O)NC2=O)C1 CC1CCN(CCC(=O)NC23CC(CNC(=O)CC4CCCCC4F)(C2)C3)CC1 Cc1nn(CCO)cc1C(=O)NC12CC(CNC(=O)CC3(C)CC3(Cl)Cl)(C1)C2 C1(CNC(=O)CC2CCCCCC2)CN(C(c2nc(Cl)cs2)=O)CC12CCC2 N1(C(C(c2ccccc2Cl)OC)=O)CCC(CF)(NC(c2coc(Cl)n2)=O)C1 C12(NC(CCCN(C)C)=O)CCCC1N(C(c1cnc(C(F)F)cn1)=O)CCC2 c1(C(=O)NCC2C(C(N(CC)Cc3cccs3)=O)CCO2)cc(F)cnc1O CC1(C)CCC(C(=O)NC(C)(C)CNC(=O)CNC(c2ccoc2)=O)C1 c1(C(=O)NC23CN(C(C(CC)Oc4ccccc4)=O)C(C2)C3)nc(F)ccc1Cl c1(C(=O)NCC2N(C(C(CC)=CC)=O)CCCCC2)cnc2cnn(C)c2c1 C12CCCN(CC1)C(=O)C2.CC1(CCNC(=O)CC2CCOCC2)CC1(F)F CCS(=O)CC(=O)NCC(C)N(C(=O)CCc1ccc(OCCN(C)C)cc1)C c1(CCNC(c2c(Cl)nsc2Br)=O)ncccc1C(F)(F)F c1(OC)ccc2c(c1)OCC(C(=O)NC1CC1CNC(=O)CCC(C)(F)F)C2 C12(CNC(c3c(CC)ocn3)=O)CC(NC(c3ccnc(C(N)=O)c3)=O)(CO1)C2 [N-]=[N+]=NC1CC(C(N2CC(O)(C(F)C(=O)Nc3cnn(CCF)c3)C2)=O)C1 N1(CC(=O)N(C(=O)Cc2nnc3n2CCOC3)C)CC(C(C)(C)C)c2ccccc21 N1(C(CCC(CC)C)=O)CCC2(CCN(C(c3cscc3S(C)(=O)=O)=O)C2)C1 c1(C(N2CCC(C(CO)NC(=O)CC3CC3)CC2)=O)cc(F)ccc1O C(=O)(CN=c1cc[nH]cc1)N1CC(CC(=O)Nc2c(C)c(CO)ccc2)OCC1 Cc1cc(=NCCC#CBr)[nH]cc1S(=O)(=O)N1CCCC(C)C1C N1(C(C2(C)CCN(Cc3c(OC)c(Br)ccc3)C2)=O)CCC2(CC1)COC(=O)N2 Cc1oc(S(N)(=O)=O)cc1C(N1CC2(CCC(CNC(c3cnsn3)=O)O2)C1)=O CC1CCC(C(=O)NCC(C2CC2)NC(=O)C(c2ccc(Cl)cc2)O)CC1 Cn1c(C(=O)NC2CCN(C(c3cnc(S)n3C3CC3)=O)CC2)nnc1S CC(C)C(C(=O)N1CCC(C)C1)NC(c1ccc(F)cc1)=O N1(C(c2nc(OCC)oc2)=O)CCC(C)(COC(=O)C(COC(C)(C)C)OC)C1 CC(C)(C)CCC(=O)N1CC2(C)CC1(C(=O)NCC(=O)NCC1CC1)C2 N1(C(C2(N(C)C)CCC2)=O)CCC(N(C(C2C3CNC(=O)C23)=O)CC2CC2)CC1 c1(CC)[nH]nc(Cl)c1C(N1CC(O)(CCNC(=O)CCC2C(=O)ON=C2C)C1)=O c1(CC)nc(Cl)nc(N(C)CC2CCN(C(=O)Cn3ncnn3)C2)c1Cl c1(C(=O)NC(CN(C(CC(CC)SC)=O)CC)C)cccc(N)c1C N1(C(c2ccc(COC)[nH]2)=O)CCN(C(c2nnc(S)n2C)=O)C2CCCC12 C1(F)(C(N2CCC(C#N)C2)=O)CCN(C(c2cc(C(F)(F)F)cc(F)c2)C2CC2)CC1 C(c1ccc(F)c(F)c1)=CC(=O)NCCCCC1(NC(CCC#C)=O)CC1 c1(C(C2CCCC2)NC(=O)NCC2CCC(C(=O)OC)O2)ccc(C)cc1 c1(C(N2CC(CCC)N(C(=O)Cn3cncc3C)CC2)=O)cc(F)c(F)cc1N c1(C(=O)NC(C2CN(C(=O)CN3C(C)CCC3C)C2)C)cc(C2(Cl)CC2)n(C)n1 C1(C(=O)Nc2c(C(=O)OCC)ccs2)CCCCC1NCCc1nnc(C)n1C c1(C(=O)NC2(CNC(c3cncc(OC)c3)=O)CCC2)cc(I)ccc1F c1(CC(CC(=O)OC)C(=O)NC2CCOC2C)c[nH]c2ccc(Br)cc12 N(C)(C1CN(C(c2cc(C)on2)=O)CCc2ccccc21)C(CCCOCC)=O CC(CF)C(=O)NC(C1CCN1C(c1snnc1C1CC1)=O)C1CCCC1 c1(OC)cccc(F)c1NC(C1CN(c2ccnc(Br)n2)CCO1)=O c1(CN(C)C)ccc(S(C)(=O)=O)cc1.c1(-c2c(C)occ2)nc2n(n1)CC2 c1(CC(=O)NCCN(C(CCC(=C)Cl)=O)CCC)ccc(Cl)cc1F Cn1nccc1C=CC(=O)NC1CCC(C)(CNC(=O)COC(F)F)C1 N1(C(C2C(C)C2)=O)CCCCC(C2CN(C(c3occ4c3CCC4)=O)C2)C1 Cc1cnc(C(C)NCCOc2ccccc2)cc1Br.c1(N)cc(Cl)cnc1O c1(C(=O)OC(C)(C)C)nn[nH]c1C(F)(F)F.C12CN(C1)C(=O)NC2C C=CC1(C(=O)NCC23CCC(F)(CC2)C3)CCN(C(=O)CN2CC(=O)NC2=O)C1 C#CCC(C)(CC)C(=O)N1CCN(C(c2cc(F)c(F)cc2N)=O)C(C)C1 C1(CCC)(NC(c2cc(F)n[nH]2)=O)CCCN(C(=O)C=C(C)C2CCCCC2)C1 c1(C(N(C2CCN(C(=O)C(C)SC(C)C)C2)CC#C)=O)cccn2ccnc12 C1(NC(C2(CSC)CC2)=O)CCC(NC(c2cnc(-c3cnn(C)c3)s2)=O)C1 c1(C(N2CC(NC(C(C(C)O)N(C)C)=O)C(F)C2)=O)ccc2c(c1)C(=O)CCS2 c1(C(=O)NCCC(CCNC(C(C)=CC)=O)C)ccc(Cl)c(N)c1Cl C(CCC(C(=O)NCc1ccc(F)cn1)NC(c1ncccc1O)=O)OC C1(C(=O)OC(c2ccc(OCCF)cc2)=O)CCC2CC2C1 C(=O)(C(O)CC(C)C)NCC(=O)NC(CN(CC)CC)C N1(C(C=CC=CC)=O)CCOCC(NC(C2CC3(CC3)CN2C)=O)C1 Cc1cc(-c2nc(C(C)C)nn2C2CCOC2C)c(F)c(Br)c1 c1(C(C)C)ccc(N)c(C(N2CC(NC(=O)C=Cc3ccc(Cl)s3)C(C)C2)=O)c1 c1(CN(C)C(=O)Nc2ccc(O)c(F)c2)noc2c1CCCC2 c1(C(C)=O)c(CCC(N2CC(CNC(=O)CNS(N)(=O)=O)C(O)C2)=O)c[nH]c1C C1(C(C)C)CCOCCN1C(=O)NC1CCCCC1(C)C c1(C(=O)NC(CN(C(=O)CC2CC(OC)C2)CC)C)cc(C)c(C)o1 c1(NC(=O)C=Cc2ccc[nH]2)cc(O)nn1-c1ccccc1F c1(C(N(c2nnn(C3CCC(N)CC3)n2)C)=O)cc(Br)c2ncnn2c1 c1(C(=O)NCCNC(C(CC)=CCCC)=O)snc(O)c1Cl CC1ON=C(C(=O)NCC2CCN2C(=O)CCN2CCC(O)CC2)C1C c1(CNC(C2CN(C(CC3(OCC)CCC3)=O)CC2F)=O)ncc(F)cc1F c1(C(=O)NCC2CC(NC(C3CC4CC4C3)=O)C2)cnc2scnc2c1 c1(C(=O)NC(C)CNC(c2sccc2CN(C)C)=O)ccc2ccncc2n1 C#Cc1ccc(C(=O)NCCC2CCC(NC(C3CC(Cl)(Cl)C3)=O)C2)cc1 N1(C(C(CC)NC(=O)CSC(F)F)=O)CC(OC)C2(CC2)C1 C(=O)(C(N)CCC(C)(C)C)NC C1(NC(C2(C(C)C)CC2)=O)CC1C1CCN(C(c2cc(C(N)=O)[nH]n2)=O)CC1 CCC(C)CCCCC(=O)NC1CN(C(=O)CCc2csc(C)n2)CC1O C1(CNC(C(C(C)C)OCC)=O)CN(c2ncc(C#N)cc2C)CC2(CCC2)O1 Cc1[nH]nc(C(=O)NC2CCCC2NC(c2ccncc2Cl)=O)c1Cl c1(NCC2(CN)CC2c2ccc(Br)cc2)ccc(Cl)cc1F C=CC1(C(=O)NC2CC3C=CCC23)CCN(Cc2ccccc2)CC1 N1(C(c2c(F)ccc(OC)c2)C(=O)NC2CCC2)CCOc2ccc(F)cc21 CCN(N1CCC(n2cc(COC)nn2)CC1)N1CCc2ccc(Br)cc2C1 CC1CCN(Cc2nc(C3CC3)cs2)CC1NC(C1(c2ccccn2)CCC1)=O c1(OC)ccc(CC(N2CC(C(=O)OCc3ccncc3)OC2=O)=O)cc1F c1(C(=O)NC(CC(C)NC(=O)CN(C)C)C)sccc1S(N)(=O)=O CC1CCN(C(=O)CC2OCCC2C)CC1CNC(c1ncc[nH]1)=O C(=O)(C1c2c[nH]nc2CN1C(c1cnncc1O)=O)N1C(C)CNC(=O)C1 c1(OCC=C)ccccc1C(=O)NCCN(C(=O)C(O)C(C)OC)C(C)C c1(C(=O)NCCC2CN(C(=O)C3=CCCCO3)CCO2)cc2ccsc2c(O)n1 N(C1CN(C(=O)C2=C(Cl)CCOC2)CCc2ccccc21)C(C1C(C#N)C1)=O c1(C(=O)NCC(CC)NC(=O)C(C(C)C)NC(=O)CNC(C)=O)cncc(Cl)c1 C1(C(=O)Nc2ccc(Cl)nc2)CN(C(c2ccc(F)cn2)=O)CC1C1CC1 N1(C(c2c(CC)ncs2)=O)CCC(O)(CNC(C2CCC3CC23)=O)C1 C(CC(C(C)C)NC(=O)CCCn1cncn1)N(C(C1(NC(C)=O)CCC1)=O)C c1(C(N2CCN(C(C=C(CC)C)=O)CC2CF)=O)cc2cccc(F)c2s1 N1(C(C(CC(C)C)ONC(=O)C2CC=CC2)=O)CC2CCOC(=O)C2C1 C1(NC(Cn2ncc(C)c2)=O)CN(C(c2ccc(S(C)=O)cc2)=O)CC2(CC2)C1 C(C)(CCC(=O)N1CCC(CO)(NC(=O)C(CC2CCCCC2)OC)C1)OCC c1(CC(=O)NC(C2CCN(C(C3C(C)(C)C3)=O)C2)(C)C)cc(Cl)ccc1O Cc1cc(Cl)c(C(=O)NCC(C)(C)CN(C)C(C2(n3ccnn3)CC2)=O)cc1F N1(C(C(C)OCCC(C)C)=O)CCCC(C2CCCN(Cc3ncnn3C)C2)C1 C1(CNC(CC(C)(C)SC)=O)CCC2CN(C(=O)CC(C)c3cccnc3)CC12 C(=O)(C1=CC2CCC=CCCC12)N1CC(C)(CNC(=O)C(N)=O)OCC1 N1(C(C2C=CCC2)=O)CC2CCOC2(CNC(=O)C(F)(F)c2ccncc2)C1 C1(CC(N)=O)CCN(C(=O)CN2CCN(C(=O)C=Cc3cncs3)CC2)CC1 C1(n2cc(C(C)(C)SC)nn2)CC2CCCC(C1)N2C(=O)Cc1ccn(C(C)C)n1 C1(C(=O)NCC2(CN(C)C(c3cccc(OC(F)F)c3)=O)CC2)CCCC12CC2 C(=O)(C1=CC2C=CC1C2)N1C(CCNC(CSCC=C)=O)COCC1 C(=O)(C(C)Cc1ccccc1)NC(C1CCN(C(C2COC2)=O)C1)C C(=O)(CN=c1cc[nH]cc1)NC1C2CN(C(COc3c(C)cccc3)=O)CC1C2 C(CCCC(CO)NC(=O)CCc1cc(Cl)no1)NC(C1N(C)C(=O)NC1)=O c1(CNC(=O)OC(C)(C)C)cc(C#N)ccc1F.C12(C3CC3)CN(C1)C2=O N(C1CCCOc2ccccc21)C(C=C)C C(C(C)CC(=O)N1CC(NC(=O)C=CC(=O)N(C)C)C(C)C1)OC c12ccc(nn1)[nH]2.C(=O)(CC(C)(C)N(C)C(C)C)NC(CCCSC)=O CCCCCC(O)C(=O)N1CC=C(CCNC(C2(C)CC(=O)N(C)C2)=O)CC1 c1(N2CCC(c3scc(C)n3)C2)cc(Cl)ccc1-n1nccn1 C1(C(=O)NCCC2N(C(c3n(CC(C)C)ncc3)=O)CCSC2)C2CN(C)CC12 c1(C(=O)NCC2C(NC(C(CC)(C)OC)=O)CC2)cc(N)c(O)c(F)c1 c1(CC)nc(CC(=O)NCCCN(CCCn2cc(C)cn2)CC)cs1 c1(C(=O)NCCN(C(COC(CC)(C)C)=O)C(C)C)ccccc1NCCOC c1(C(N(C)CC2CCN(C(c3cc(C)on3)=O)C2)=O)ccc(C(F)(F)F)nc1 N1(C(C(C)OCC)=O)CCN2CC1OCC2=O.c1(CSCC(F)(F)F)cscn1 Cc1c(C(N2CC3(CC(CNC(C4CCCC4C)=O)C3)C2)=O)cccc1F Cn1nc(C(c2nnnn2C)NC(c2ccncc2)C2CCC2)nc1C1CC1 CCCC(O)CC(=O)NCC(C1CCC1)NC(c1c[nH]nc1-c1ccccn1)=O c12ccc(c(F)c1)CC(=O)N2.c1(OCCC(=O)NCC)ccc(Cl)cc1 c1(N2CCC(C)C2CNC(c2cc3c([nH]2)CCC3)=O)ncc2ncn(C)c2n1 c1(C(N2CCN(C(CC3C(CC)C3)=O)C(C)CC2)=O)cc2c(nc1O)CCC2 CC1CCN(C(=O)Cn2ncnn2)CC1CNC(c1csc(Br)n1)=O N1(C(C2CCN(C(C)=O)C2)=O)CCN(C(C2CCC3(CC2)CC3)=O)CC(CO)C1 C(CC(C)(C)C(=O)N1CCC(CNC(c2ncccc2N)=O)C(C)C1)OC N1(C(Cc2nnc(C)o2)=O)CCC2(CC1)CCN(C(C1CC3CC3CC1C)=O)C2 N1(C(C2(C(N(C)C)=O)CC2)=O)CCCN(CCNC(C2(C)CC2(F)Cl)=O)CC1 c1(C(=O)NCC2(OC)CCN(C(=O)CC(C)O)C2)ccc(C(C)=O)c(C)c1 c1(C(N2C(C(N3CCC(CCO)CC3)=O)CC(O)C2)=O)cnc2cc(Cl)ccn12 N1(C(C2(OC)CC(C)C2)=O)CCC(C)(CCNC(=O)CSc2n[nH]c(O)n2)C1 N1(C(C2(C)CCCC(F)(F)C2)=O)CCC2(CCCC2NC(=O)C2=CCOC2)CC1 C12(NC(C=C(CCC)CCC)=O)CCCN(C(c3ccc(F)c(N)c3)=O)CC1C2 c1(C(C(=O)OCCOCC(N2CC(C(=O)NCC(F)F)C2)=O)O)ccccc1.S C(C(CC(C)C)NC(=O)C(C)Cn1ccnc1)n1cc(-c2ccc(CC)s2)nn1 C1(C(=O)NC2C(NC(C3C(c4n(C)cnn4)CC3)=O)C2)CC(C2CC2)=NO1 Cc1cnoc1C(=O)NCC(C)N(C)C(C1CCC1C(F)F)=O N1(C(C2C(CNC(CSSC)=O)OCC2)=O)C2CCC1CC(F)C2 c1(C(C)C)ccc(C(N2CC(CNC(C3(Cl)CC3)=O)C2)=O)c(O)n1 CC1(C)CN(C(c2ncc(F)cn2)=O)CC1NC(C1COCC1(C)C)=O N1(C(C(CC)SC)=O)CCN(C(c2cccc(OC)c2OC)=O)C2COCC12 N1(C(CNC(CC(C)C)=O)=O)CC(C(=O)Nc2ccccc2CCO)CC1(C)C C1(C(=O)NC2C(NC(=O)CC3(O)CCC3)CCC2)CC1C1CCC1 C#Cc1ccccc1CNC(C1CC(CCNC(C2CCC2)=O)C1)=O n1(CCC)cc(C(=O)NCC2CC(C(=O)Nc3cn(C(C)(C)C)nn3)CO2)nn1 c1(C(N2C(CNC(c3ccsc3)=O)CC(OC)C2)=O)coc2c(F)cccc12 N1(C(C2(OC)CCCC2)=O)CCC(CCNC(C2(C)CCNC2=O)=O)CC1 c1(C(N2CC3C(NC(CC(CCC)C)=O)(CC3)C2)=O)cnc2c(c1)NC(=O)CS2 N1(C(COCC=C)=O)CCCCC(CNC(C23CCCC(CO2)C3)=O)C1 CCCCC(C(=O)NCC1CN(C(=O)C(C)(C)C(C)O)CCC12CCC2)C(C)C N1(C(Cc2c(C)ccc(C)c2)=O)CC2CCC1C(NC(=O)CCC1CCCO1)C2 CC(C1=NOC2COCC12)NC(=NCCCF)NCC(=O)NC(C)(C)C C1(CC)CN(C(=O)CCCn2ccnc2)CCC1NC(=O)C(c1cccnc1)O c1(C(=O)NCC(C)(CO)NC(C(CC(=O)OC)C)=O)cc2ccnc(Cl)c2s1 CN1C2CCC1CC(c1nnnn1CCCF)(NCC(CO)C1CCC1)C2 C=CC1OCCCC1C(=O)NCCN(C)C(C1CCN(CC(F)(F)F)C1)=O C1(N(C(c2cc(C)ns2)=O)C)CN(C(C2CC2(C)C)=O)CCC1O C1(CCCNC(=O)Cn2nnnc2C)(CNC(COCCCCC)=O)CCCC1 Cc1cc(C(=O)N(CCN(C)C)Cc2ccc(F)cc2)c2nccc(C)c2c1 N1(C(CC(C)(O)c2ccccc2)=O)CCCCC(NC(C2CC2F)=O)C1 N1(S(CCC(=O)OC)(=O)=O)CCN(C(=O)CCc2ccc(OC)cc2)CC1C#N N1(CCNC(C(CC2CC2)NC(C2(C#N)CC2)=O)=O)CCCNC1=O N1(C(CC2CC(=C)C2)=O)CC(C)(C)OCC1CNC(=O)C(C)n1cncn1 C(=O)(C(C)(C(C)C)NC(C)=O)N1CCC(CN(C(C=CCN(C)CC)=O)C)CC1 N1(C(c2c(C)n(C(C)C)nc2)=O)CCCN(C(C2CC3CC3C2)=O)CC1C C1(C(N2CC(OC)(CNC(C3C=CCCC3)=O)C2)=O)CC(=O)N(C(C)C)C1 C#CCCCC(C)C(=O)N1CCC(CN2CCN(C(=O)C=CSC)CC2)CC1 Cc1cn2ccnc(C(N3CCC3CNC(C3CCC(=O)N3C3CC3)=O)=O)c2n1 c1(NC(C2C3(CCN(C(c4cc(C)[nH]n4)=O)C3)C2)=O)ncc(I)cc1[N+](=O)[O-] CC1(C)CCCOC1CC(=O)NNC(=O)NCC(F)(F)F CCCC(C)(CO)NC(=O)CCC1CCCN(C(=O)C(C2CC2)C2CC2)C1 c1(C(=O)NCC2(CNC(C)=O)CC2(F)F)nn(C)cc1Cl c1(C(N(C)Cc2cccc(CNC(c3cnc(C)[nH]3)=O)c2)=O)cc(N)c(Cl)cn1 N1(C(C(c2cccs2)NC(=O)CSc2ncccc2F)=O)CCC(F)CC1 C1(NC(c2c(C)nc(CC)o2)=O)CC2CC1CN(C(=O)Cn1ncn(C)c1=O)C2 CC1CC(C(=O)NC(CO)(CO)CO)CN(C(c2cc(F)c[nH]2)=O)C1 N1(C(CSCCOC)=O)CCC(C)C(CC(N2CCC(C(=O)OC)C2)=O)C1 c1(OC)cc(=NC(=O)C2CC(=O)CN2C(=O)CCC(C)=O)[nH]n1C N1(C(C(CC2CC2)OC)=O)CCOC2CN(C(=O)Cc3ccc(F)cc3F)CC12 C1(CC(=O)N(C2CC=CC2)C)CN(C(=O)CC2(O)CCOC2)C(C)(C)C1 C=CCC(CNC(=O)CCCC1CCC1)C(=O)NC1CC(O)C(F)C1 CC1Cc2c(Cl)cccc2C1NCc1c[nH]c(=O)c2ccnn12 c1(C(=O)NCc2nc(CCC(=O)NCC3(CN)CC3)on2)cccc(F)c1F C(=O)(C1=C(Cl)CCCC1)NCC(C(=O)NC1C(OC)CCC1)N(C)C CC1CC(NC(C2C3COCC23)=O)CN(C(c2ccc(Br)cc2O)=O)C1 c1(NCCc2cc(C)no2)cc(NCc2csc(C(C)(C)C)n2)ncn1 CC1CCN(C(=O)CONC(c2cnnn2C)=O)C1C c1(CC(=O)NC(C)CNC(=O)C(N2CCP(C)(=O)CC2)C)ccc2nsnc2c1 C1(C(=O)NCCNC(C2CC(C)N(C)C2)=O)CCCC12CCC2 c1(C(N(CCC(C)NC(=O)CCCC2CCCO2)C)=O)ccnnc1O C1(NC(c2c(OCC)cccc2)=O)CCN(C(C2(C)COC(=O)OC2)=O)CC1C C12(NC(c3c(C)snn3)=O)CC1CN(C(C1CCCN(C(C)C)C1)=O)C2 c1(SCC)ccc(C(=O)NC2CCCC2NC(c2csc(C(=O)OC)c2)=O)cc1 CC(O)C(F)(F)C(=O)N1CCC(C)(CC(=O)NCCC#CCO)C1 c1(OC)ccc(C(=O)NCCC2CSCCN2C(=O)CC(O)C(C)C)nc1Cl c1(C(=O)NC(CC)CNC(=O)C(C)OCC(F)(F)F)c(Cl)ccc(OC)c1N CC(C(=O)OCC(=O)Nc1cccnc1-n1ccnc1)S(=O)(=O)C1CCOCC1 c1(C(N2C(C)C3CC2C3NC(=O)CNS(=O)(=O)N(C)C)=O)ccc2nn[nH]c2c1 C#CCCCCCCC(=O)NCC(CC(C)C)C(=O)NCCN(C)C(=O)C1CC1 N1(C(COC)=O)Cc2ccc(C(N3CCCOCC3)=O)cc2C1 c1(NC(C)=O)ccc(C(N2CCC(O)(CCNC(=O)C(C)CF)C2)=O)c(Cl)c1 c1(C(C)=O)cc(NC(=O)C(C)C(C)NC(=O)CN2CCCC2=O)ccc1F Cc1cc(C(=O)N(C)CC2(O)CCN(C(=O)CCC(N)=O)C2)cn1C N1(C(C(Cc2ncn(C)c2)O)=O)CCCCC(NC(=O)C=C2CCOCC2)C1 c1(C(=O)NCC(CNC(C(CC)n2ccc(C3CC3)n2)=O)O)nnc(O)nc1O N1(C(=O)OC(C)(C)C)CCC(NC2(C(N)=O)CCCOC2)CC1c1ccccc1 N1(CC(CCCC)CC)C(=O)CCN(CCO)C1=O.N(S(=O)(=O)NC(C)C)C(C)C O=C(C(O)CCNC(=O)C(O)C1CCCC1)N1CCC2CCC12 C12(NC(CC(CCC)C)=O)CCCC1N(C(=O)C(C)Oc1ccccc1)CCC2 C1(COC)CN(C(C2(C(=O)NCc3ccc[nH]3)CCC(=O)N2)=O)CC(C)(C)O1 c1(N2CCCCC(SC)C2)nc(N2CCN(C)C(CO)C2)c2c(n1)CCOC2 C1(NC(C(CC)CC2CCCC2)=O)CCSC12CN(C(C1CC(C#N)C1)=O)C2 c1(OC)cc(F)c(C(=O)NCC(C)CN(C(=O)C=C(C)Cl)C)cc1Br C1(NC(CC(C)(C)OC)=O)CCC2CC1CN2C(c1nc(C2CC2)oc1C)=O C1(CNC(C(C)OCCN(C)C)=O)(NC(C2CC23CCOC3)=O)CCCCC1 CC1(C)COC(CCC(=O)NC2COCCC2NC(=O)CC(C2CC2)C2CC2)C1 C1(CCCN(C(=O)CCOC2CCC2)C)CCCN1C(=O)CC(C1CC1)C1CC1 N1(C(C(CCC)OC)=O)CCC2(C1)CN(C(=O)C(C)=C1CCCC1)C2 C1(C(=O)NC2C(OC)C(O)C2)CC=CCC1NC(=O)CC1OCCO1 C(C(=O)N(C(C)C(=O)N(C(C)CO)C)C1CC1)(OC)OC CC1C(NC(=O)CNC(=O)C(F)(F)F)CCCN1C(c1ccnc(F)c1N)=O N1(C(c2ncc(-c3ccccc3)s2)=O)CC2CC1CN2C(=O)NCCCl c1(C(=O)NC2CN(C(c3scc(C#N)c3)=O)C2)ccc(F)c2c1CCC2 CC(CC(=O)N1CCC1CNC(C1CCOCC1)=O)n1cc(Br)cn1 C1(CC(=O)NC2CCCN(C(=O)CCc3ccnc(Cl)c3)C2)CC2COCC12 c1(C(N(C2CCN(C(=O)CCCn3cncn3)C2)CC)=O)sc([N+](=O)[O-])cc1Cl C1(OC)CN(C(c2cnn(C(C)(C)C)c2N)=O)CC1NC(C1(F)CC=CCC1)=O C12CCCN(C1)C(=O)c1cc(oc1C)-c1cccc(c1)N2C=O.CCO.OC c1(C(N2C(C)(C(=O)NC3(CCC)CC3)C=CC2)=O)ccc(C)cc1O CC1CCN(CCC(=O)NC(CNC(=O)CN2CCC(O)CC2)C2CCC2)CC1 n1(C2CC(C)C2)nnc2c1CN(C(=O)NC1CCC3(NC(C)(C)C)CCC13)CC2 C(CS(=O)(=O)C(F)F)NC(=O)NC1CCN(CC(=O)NC(C)(C)C)C1 c1(OC)cc(S(=O)(=O)N2CCOC(C)CC2)cc(C(=O)O)c1OC C(c1ccncc1)=CC(=O)NC1CC1NC(c1cc(C(F)F)ncn1)=O c1(CNC(=NCc2cccc(OC)c2)NC(C)C)ccc(Br)c(C)c1F c1(C(c2nnnn2CCSC)NCC(=C)F)cc(C)c(OC(C)C)c(C)c1 C1(CC#C)(C(=O)NCCN(CCN(C)C)CC)CCC1.C1(=O)C=CN1 c1(N2C(C3CCN(C(C(C)CN(C)C)=O)C3)CCC2)nc2cc(Cl)cc(Cl)c2o1 C1(c2nc(-c3cncc(OCC)c3)on2)CCOC12CCOCC2 C(c1ccccn1)=CC(=O)N(C(CN(C(C1(C(C)C)CCC1)=O)C)C)C C1(NC(CCC(=O)NC)=O)CCCCC1N=c1ccc(C#N)c(C)[nH]1 Cc1nn(CC(=O)NC23CC2CN(C(=O)COCCN(C)C)C3)c(=O)n1C Cc1ccc(F)c(C(=O)NC(c2cnn(C)c2)C(=O)NCc2cnccc2Cl)n1 Cc1cc(C(N2CC(O)(C(C)NC(=O)Cc3c(C)cccc3F)C2)=O)cc(Cl)c1 c1(OC)ccc(C(=O)NC2CCOCC2C(=O)NC2(CCO)CCCCC2)nn1 C12(CNC(C(CC)=CC)=O)CCC(CN(C(C3CCCCN3CC)=O)C1)C2 Cc1cnc(C(=O)NC(CNC(=O)Cc2ccc(Br)cc2C)C2CC2)c(F)c1 C(CC(=O)N(CC(O)CNC(c1nn(CC)cc1Br)=O)C)(C(C)C)OCC C1(NC(=O)NCC(=O)N(C)CCc2ccccn2)CCC2(CC1)CC2 CCC(C)CC(C(=O)N1CC(F)C(F)C1)NC(=O)C(OCC)OCC C=CC(C)(O)CC(=O)N1CCN(C(c2ncoc2-c2cccs2)=O)CC1CCO N1(C(C(c2ccc(F)cc2)C)=O)C(CNC(C2(Cl)CC2)=O)CC2CCCCC12 CCCC(CCc1ccccc1)C(=O)NCCCN(C(=O)C(CC)OC)CCO Nc1c(C(N2CC3(CCC3NC(c3cnn[nH]3)=O)C2)=O)ccc(Cl)c1Cl CC1CC(C(=O)NCCC2CC(NC(c3csc(C4CC4)n3)=O)C2)CCS1(=O)=O CON(C(=O)c1cccc(CNC(=O)CC(C)CN(C)C)n1)C1CCCC1 C1(CC)CN(C(=O)COCC2CCC2)CCN1C(c1cncc(C2CC2)c1)=O N1(C(C(COC)(C)C)=O)CCC2(CC1)CN(C(=O)C=Cc1ccsc1)CC2CO CC1(C)C(CNC(=O)CC23CCCC2C3)CCN1C(=O)CCP(C)(C)=O C(CC1=CCN(C(=O)CC2CCCC(=O)N2)CC1)NC(C1(C)CCCOC1)=O CC1(C(=O)NC2COCCC2NC(C2(O)CCC2)=O)COc2ccccc21 c1(C(N)=O)cccc(NCC(N2CC(O)(CCNC(C3OCCCO3)=O)C2)=O)c1 C1(NC(=O)C(c2ccccc2)O)CN(C(C2(c3ccno3)CC2)=O)CC1O C1(CNC(CCc2cc(C)n(C)n2)=O)CN(C(C2(C(F)F)CCC2)=O)CC1(C)C NS(=O)(=O)N1CC(C(N2CCN(C(=O)CC3CCC34CCC4)CC2)=O)C1 n1(CC(=O)N(C2CN(C(C3(N(C)C)CCC3)=O)C2)CCO)nc2n(c1=O)CCOC2 C1(C(C)C)CN(C(C2CCS(=O)CC2)=O)CCN1C(c1nccn1C)=O CCCC(CNC(=O)CCc1cc(Cl)ccc1O)CC(CC)CC C12(C(N3CCC(CN(C(=O)C(C4CCCCC4)F)C)CC3)=O)CCC(CC1)OC2 n1(CC)cnnc1CN(C(C(=O)NCc1ccoc1C)C1CCCC1)C n1(CCC(=O)NCCC(C)N(C(C2CC(OC)C2)=O)C)c(C)csc1=O C(CC)(C(=O)NCC(C)(O)CNC(c1cnc(C2CCC2)o1)=O)=CC c1(C(=O)NC(CNC(CC(C=C)CC)=O)C(C)C)cnc2nc(O)nc(O)c2c1 C1(O)(NCc2cn(C(C(=O)Nc3c(C)nn(C)c3)(C)C)nn2)CCCN(C)C1=O N1(CC=C)C(=O)NC(c2cnn3c2CNCC3)C2=C1CCNC2=O c1(OC)ccccc1C(CNC(=O)C(C)(F)F)NC(=O)CC1C=CCC1 C(=O)(C(CNC(C1(F)CCCCCC1)=O)C(C)(C)C)NC(c1ccc(C)s1)C C1(COC)CN(C(=O)C(N2CCC(CSC)CC2)=O)CCCO1 CC(CC1CCCC1)C(=O)NCC(C)CN(C)C(C1CC1(C)C)=O C(=O)(C1=NOC(C)(C)C1)NCC1CN(C(CC(n2ccc(C)n2)C)=O)C(C)CC1 c1(C(=O)NCC(CC=C)NC(C2(S(C)(=O)=O)CC2)=O)ccc(-n2ccnc2)nn1 C1(CNC(CC2N(CC)CCC2)=O)N(C(=O)CSC)CCCC1(C)C Cc1nc(NC2CN(C(=O)C3=CCOCC3)C2)c2cc[nH]c2n1 c1(NC(CC)CN(C)C)nc(N2CCCC(OC)C2C(=O)OC)nc2scnc12 C1(C(N2CC(OCCNC(C(C(C)C)n3cccc3)=O)C2)=O)CCC(C)C(C)C1 c1(C(=O)NC(C2CCN(C(=O)C=CC3CCCN3C)CC2)C)cnc2n1CCC2 N1(C(CCn2nc(C)c(C)c2C)=O)CC(C)CN(C(c2coc(Cl)c2)=O)CC1C c1(C(=O)NCCN(CCC)C(c2nnc(C)s2)=O)nccn2cc(C)nc12 Cc1cc(C(N2CCN(C(=O)CC3CCC4CC34)CC2CCO)=O)c(F)cc1N C1(CC(=O)NC(c2nc[nH]n2)C)CCCCC1NC(c1cc(=N)[nH][nH]1)=O Cc1cc(N)c(C(=O)N(C2CCN(C(=O)CC3CCC3(F)F)C2)C)cc1F c1(OC(C)CNC(=O)Cn2cc(NC(c3cc[nH]n3)=O)nn2)cc(Cl)ccc1Cl C1(NC(C(CC#C)CC#C)=O)CC(NC(=O)Cc2cnnn2C)C12CCOCC2 C1(CO)CCC(F)(F)C1.C12(CC1(F)F)C(=O)NCC1(CCC1)C(=O)NC2 N1(C(C2(OCC)CC2)=O)CCCC(CC(=O)NCCCN2CCCC2=O)C1 N1(C(CC2C(C)(C)C(O)C2)=O)CC2CCCN(C(c3ccccc3)=O)C2C1 c1(OC)ccc(C(C)C)c(C(=O)NC(C2CCN(C(=O)CO)CC2)C)c1 N1(C(c2c(C)nc(C)[nH]2)=O)CCN(C(=O)CCCn2ccnc2C)C2CCC12 C12(CNC(CN(C)CC)=O)CCCCC1N(C(C1Cc3cscc3C1)=O)CC2 c1(CC)cc(C(=O)NCC2CC(C)N(C(=O)CCNC(=O)CC(C)C)C2)n(C)n1 c1(OCC)cc(C(=O)NCCC2CCCN2C(=O)C(CC)OC)ccc1OC CCCCC(O)CC(=O)N1CCCC(N(C)C(c2cn3ccnc3cn2)=O)C1 N1(C(c2c(C)snc2)=O)CCC(NC(=O)CSCc2cccs2)C(C)(C)C1 n1(CCCOC)nc(-c2cc(SC)ccn2)nc1C1CC2(CNC2)C1 n1(CC)ccc(C(=O)NCC2CCN2C(C2C=CCC2)=O)cc1=O C(=O)(CCCCC(F)(F)F)N1CC(C)C(NC(c2coc(Br)c2)=O)CC1 c1(C(=O)NC2CC(NC(=O)CCc3cnoc3)C2)cccc(Cl)c1Br CCCCCC(C1CC1)NC(=O)NC1CCN(CCN(CC)CC)C1 Cc1ccc(Cl)cc1C(=O)NC1CC(CNC(=O)C(c2cccn2C)=O)C1 c1(CNC(c2c(C)noc2C(F)(F)F)=O)cccc2c1CCN(C1CC1)C2 C1(F)(C(=O)NCC2CC(=C)C2)CCN(C(=O)C(C)SC)C1 C(=O)(CCCC(=O)c1ccc(Cl)c(Cl)c1)NCCNC(C(C)(C)NC(=O)OC)=O CCC(CC(=O)NC1COCC1C(N1CC(OC(=O)NC)C1)=O)OC Cc1ccncc1CNC(=O)COC1CN(C(C2(C)CC3CC3C2)=O)C1 c1(C(=O)NC2CC(C)(CNC(=O)C3CC3)C2)ccc(-c2ccncc2)nc1 c1(CN=C(NC(c2ncn(C)n2)COC)NC2CCCC2)ccc(O)c(F)c1 C(=O)(CCCCCNC(=O)C(C1CCCCC1)F)N1CCC(C)(CC)C1 N1(C(C(C)NC(C)=O)=O)CC2CC(NC(c3[nH]c(C)nc3C)=O)C1C2 C=CC(CC)C(=O)NCCCOCCN(C(=O)CCCc1ccccn1)C c1(C(=O)NC2CCC(N(C)C(C3(C#N)CCC3)=O)C2)cccc(N2CCCC2)c1 C1(C(=O)NCCN(C(C=CC)=O)C)Cc2cccnc2C1 CCC(F)(F)C(=O)N1CC2CC2(CNC(=O)Cc2ccc(Cl)cc2)C1 c1(C(=O)NCC(C)NC(C2(CC#C)CCCOC2)=O)ccn2c1CS(=O)(=O)CC2 C(CCC1C(=O)O1)C(=O)C(n1cc(-c2ccc(C(C)=O)c(F)c2)nn1)C.CN N1(C(CCC=C)=O)CCN(C(=O)C(C)OCCc2ccccc2)C(CCC)C1 CC1CCC=C1C(=O)NCC12CC(CNC(=O)Cn3nc(O)ccc3=O)(CO1)C2 CC1(C(N2CC(F)(c3cn(C4CCCCC4)nn3)C2)=O)COC(=O)C1 N1(C(CCCOCCOCC)=O)CC(NC(C2CCC(CC)O2)=O)C(C)C1 C1(C(C)C)CCN(C(=O)C(=O)NCC=CC2CCCO2)C1 C1(NC(CCCCOC(C)(C)C)=O)COCCN(C(C2CC(O)C2)=O)C1 C(=O)(CS(=O)(=O)CC(=O)N(C1CCCC(NC(=O)CSC(F)F)C1)C)OC N1(C(c2n(C)ccc2)=O)CC2(C1)SCCC2NC(C1CC12CCCCCC2)=O C1(CN(C(C=CC(CC)=CC)=O)C)CN(C(=O)CSc2ccc(O)cc2)CCO1 c1(CC(=O)NCC2C(CNC(c3c(C)c(Cl)cnc3)=O)C2)cnn2ccccc12 c1(C(=O)NC2C(NC(c3nc(CC)sc3)=O)C2)cc(C)c2c(c1)CCCN2 C1(CCNC(COC(C)C)=O)CCCN(C(C2(F)C3CCCC23)=O)C1 C1(C(C)(C)CNC(C2(C(N)=O)CC2)=O)CCCN1C(=O)CCOc1ccccc1 N(C1c2ccccc2CC1NC(C1CCS(=O)(=O)C1)=O)C(=O)CCCCO C(=O)(CC(C)(F)F)N(CC(C(=O)NC(CCC)C1CC1)C)C C1(OC)CC(NC(C2CCCOC2)C2CC2)C1(C)C.C(C)(C)(C)OC(=O)O c1(C(=O)NCCC2CCN(C(c3nncn3C3CC3)=O)C2)ccc2c(c1)CCO2 C1(CC(=O)NCC(CC)O)C(NC(C2(CF)CC2)=O)CC1O N1(C(c2ccc(C)c(O)n2)=O)CCN(C(C2CC3CCC(C2)C3)=O)CC(C)C1 CC1CN(C(=O)CC2CCN(C)C2=O)CC2(CCN(C(C3(C#N)CC3)=O)C2)O1 CC(C)CCCC(=O)N1CC(N(C(=O)Cc2cscc2Br)C)C(O)C1 C(CCCCC(=O)NCC(CO)NC(=O)Cn1ccc(Br)cc1=O)OC C1(CNC(C(C)=C2CC2)=O)CCC(C)CN1C(c1cc(N2CCCC2)ccn1)=O C1(C(N(C)Cc2cc(C)on2)=O)CC2(CCN1C(=O)CC1CCCSC1)CC2 c1(C(=O)NC(COCC)C(=O)NCC(C)N=[N+]=[N-])ccc(C)nc1 C1(NC(c2c(C(C)C)n[nH]c2)=O)CC2CC1N(C(=O)C(C#N)C(C)C)C2 C1(NC(C(CC#C)NC(C2CC(=O)N(CC)C2)=O)=O)CC2(CCCC2)C1 c1(C(=O)NC2(CC=CC(=O)N(CC#C)CCOC)CCC2)ccc(CC)[nH]1 C(=O)(CS(=O)(=O)CCO)N1CCC(N(C(C(CCC)F)=O)CC)CC1 C1(C(N2CCC(C)(CNC(c3c(CC)nns3)=O)C2)=O)CC2OC1C1CC21 c1(CN(C(CC(C)n2cccn2)=O)CCO)cccnc1OCC(F)(F)F N1(C(C2CC(O)(CC#C)C2)=O)CCCC2C1CCCN2C(=O)CC(=C)C CN=c1nc(C(N2CCCOC(CNC(C3CC(CC)=NO3)=O)C2)=O)cc(C)[nH]1 N1(C(CCOCC)=O)CCC(NC(c2cnn(CC(C)C)c2)=O)C(F)(F)CC1 c1(C(N(C2CCN(C(C34CCC(OC)(CC3)C4)=O)C2)C)=O)ccnc2ncnn12 C=CCCCC(N=c1nc2sccc2c(NCCC(C)O)[nH]1)C1CC1 C12CN(CCO1)C(=O)C1(CC1)CNC2=O.C(=O)(C=CC)NCCSCC C1(CS(C)(=N)=O)(COC(C(C)OC2CCCCCC2)=O)CC(F)(F)C1 CC(C)C(C)CC(=O)NC1(CC(=O)NC2CC(=O)N(C)C2=O)CC1 C1(NC(CN2CCC(C)(O)C2)=O)CC(F)CN(C(c2ccc(F)c(N)c2)=O)C1 C1(NC(c2nnn(C)c2C(F)F)=O)CCCCN(C(=O)COC(C)(C)C)CC1 c1(NCCCC(C)NC(C(C)C2CCOC2)=O)nc(C(F)(F)F)ccc1C#N C1(OC)CC(C(N2CC3CC3(NC(=O)COCP(C)(C)=O)C2)=O)CC1OC CON1CCC(C(=O)NC2C3CCN(C(c4ccc(SC(F)(F)F)s4)=O)C23)CC1 C1(NC(=O)CCNC(C2CCC2)=O)CC2CC1N(C(c1nn[nH]c1Cl)=O)C2 N1(C(=O)Nc2ccc(C)nc2C)CCCC2C1CCN2S(=O)(=O)CC(C)C C1(C(=O)NC2CC(OCC)C2)CCC(CNC(c2ccncc2Cl)=O)CC1 C(=O)(CCCCNC(C1(C)CC1(F)F)=O)NC(Cn1ncc(C)c1)C Cc1ccc(C(=O)NCC2(C(=O)Nc3ccccc3)CC=CC2)cc1 c1(C(=O)NCCC2CC(NC(C(C)S(C)(=O)=O)=O)C2)ccc2c(n1)OCCO2 c1(C(N2CC(CNC(C(F)=CC)=O)CC2(C)C)=O)ccc2c(c1)NC(=O)CCS2 C1(CC)(CC)CC(C(N2CC(OCC(=O)NC(C)Cc3cn[nH]c3)C2)=O)C1 C1(NC(c2ccc(-c3ccccc3)o2)=O)CN(C(=O)C(F)CC2CC2)CC1O CCCC(C)(O)CC(=O)N1CC(C(C(=O)NC2(C)CC(O)(CO)C2)OC)C1 C#CC1(NC(c2ccc(CNC(c3[nH]cnc3CC)=O)o2)=O)CC2CCCC12 C1(C(=O)NCCC(=O)N(C)C2CC2)C=CCN(C(=O)CC2(O)CCOCC2)C1 C1(C(=O)NC2(CO)CCN(C(CC(C)(C)C3CC3)=O)CC2)CCC2(CCOC2)O1 c1(C(=O)NC2(CNC(c3c(C)coc3)=O)CC3CCC2C3)cn2ccccc2n1 c1(C(=O)NC(CC2CN(C(COCC=C)=O)C2)C)ccc(-c2ccco2)nc1O C1(CNC(COC(C)C)=O)CC2CCC1N(C(C1CC1(F)F)=O)C2 c1(C(N(CCN(C(=O)C(C)Cc2ccnn2C)C(C)C)C)=O)coc(N(C)C)n1 Cc1cc(CNC(=O)CONC(=O)C(C)n2[nH]cnc2=N)cnc1C S(=O)(=O)(c1cccc2cnccc12)N1C(C(=O)NCc2ccoc2)CC(O)CC1 c1(-n2ncc(C)c2)cc[nH]c(=NCCCOCCOC2(CO)CCCO2)n1 N1(C(C2CCC(C)(C)C2)=O)CC2CCC2(CC(=O)NC2CCOCC2O)C1 C1(C(=O)NCC(CC=C)NC(c2[nH]nc(OC)c2Cl)=O)CC2(C1)CC(F)(F)C2 c1(NC(=O)CN2CCN(Cc3sccc3Cl)CC2)ncc(C(F)(F)F)cc1F N1(C(CCC2(NC(c3c(OC)nsc3)=O)CCCC2)=O)CCCOC(CO)C1 CP(C)(=O)c1csc(C(N2CC(NC(=O)CN3CCCCC3)CC2CO)=O)c1 C1(CN(C(=O)CC2CCCC2)C)CCCN(C(C2CC2c2cncs2)=O)C1 C1(NC(CCNC(c2c(OC)cccc2)=O)=O)C=CC(C)(C)CC1 C1(NC(C2CC(C)(C)OCC2)=O)CCN(C(C2CC2(Cl)Cl)=O)CC12CCC2 CC1(C)CN(C(C2(n3cncn3)CC2)=O)CC1NC(N1CCC2CC12)=O N1(C(CCc2ccc(=N)[nH]c2)=O)CCC2C(NC(c3cn(CCO)nn3)=O)CC12 c1(C(=O)NC(C)C(=O)NCC(O)CN(C(=O)Cn2cnnn2)C)ccc(F)cc1 CC(C(CO)NC(c1cc(CN(C)C)c[nH]1)=O)NC(=O)CCC1CC(F)(F)C1 Cc1ccc(F)c(CNC(=O)CC(C2CC2)NC(=O)C(C)Cn2ccnc2)c1 O=S(=O)(c1ccc(N2CCCN(CC(F)F)CC2)c(Br)c1)NCC1CC1 c1(OC)ccc(CN(C2CN(C(c3cc[n+]([O-])cc3)=O)C2)C)c(OC)c1OC C(C(C)(O)C(C)C)NC(C1(NC(COCCCC)=O)CC(O)C1)=O c1(NC(C2CC23CCN(Cc2cc(F)cc(Br)c2F)C3)=O)ncnc2occc12 c1(C(=O)NCC2C(NC(CC=CC=C)=O)CCC2)cnn(C(C)C)c1Cl c1(C(=O)NCCC(C)N(C(=O)CC(C)CF)C)ccnc2c(F)cccc12 c1(C(=O)NC2(CNC(C3ON=C(C)C3)=O)CC2)cc(N)c(C)cc1C N1(C(c2cccc(CC)c2)=O)CC2CCC1CN2Cc1nccnc1C Cc1cc(F)c(C(N2CC3CC(NC(c4cnsc4)=O)C3C2)=O)c(F)c1 Cc1nc(C(=O)NC(C)C(C)NC(=O)CCCNC(N)=O)n2c1CCC2 Cc1[nH]nc2ccc(C(=O)NCC(C)NC(C3(C)CC(C(C)C)=NO3)=O)c(Cl)c12 N1(C(Cn2c(C)nnn2)=O)CC(C)(C)CC1CNC(c1cc(Cl)cc(Cl)c1)=O CC(CC(=O)NCC1(O)CC(CNC(=O)CC2CCC3(CC2)CC3)C1)C(F)F c1(C(=O)NCC2CCC(O)CC2)n[nH]c2c1CN(C(C1(CSC)CCC1)=O)CC2 C=Cn1nccc1C(=O)NC1(C)CN(C(=O)C(C)OC2COC2)C1 C#Cc1cc(F)c(C(=O)NCC23CCC(CC2)N3C(=O)C2CC2)cc1F Cc1nc(C(C(=O)NCCCF)N(C2CCN(c3ccccc3)C2)C)n(C)c1C C1(CNC(C(C(C)O)C)=O)CCCN(C(C2(C)C(C)(C)C2(C)C)=O)CC1 N1(C(C(C(C)C)NC=O)=O)CCC(Nc2ncnc(Cl)c2Br)C(C)C1 C(CC(C(C)C)NC(=O)CCOCC(F)F)N(C(c1cnc(C)s1)=O)C C1(N(C(=O)C=Cc2cccs2)CC)CCCN(C(=O)C(C)=C2CCC2)C1 C1(NC(C(COC(C)=O)C)=O)CCC(NC(C2CS(=O)(=O)C2)=O)CC1 Cc1nc(CCC(=O)NC2CC3C(NC(C4(C)CC=CCC4)=O)C3C2)[nH]c1C N1(C(c2c(OC)scc2)=O)CC(NC(=O)CC2(C)CC2(Cl)Cl)C(F)C1 c1(NCC(=O)NC2C(C(=O)Nc3ccc(C)cc3)CCC2)cc2ncccn2n1 CC(C)CC(C)(C)C(=O)N1CC(NC(c2ccccc2Br)=O)C2CC2C1 N1(C(C2CC(CC)C2)=O)CCC(C)N(C(c2csc(C)c2)=O)CC1 Cn1c(NC2CS(=O)(=O)CC2NC(=O)CC2CCCC2)c(C#N)c(=O)n(C)c1=O Cc1cc(N2CC(C)CN(C(c3nn(C)cc3C)=O)CC2C)ncc1[N+](=O)[O-] C1(CC)CCCCC1C(=O)NC1CC(CC(=O)NC2COCC2SC)C1 C1(CNC(=O)NCC2(CS(C)(=O)=O)CC2)(COC)CC=CC1 c1(C(=O)OC)cc(F)cnc1NC(=O)CC1CN(Cc2cc(Br)ccc2NC)C1 CCCCCCCCNC(CCCCCC1CCN(C(=O)CCS(C)=O)CC1)=O C(CCC(N)=O)(C(=O)N1CC(CO)C1)n1cc(C(CC)CC)nn1 c1(C(=O)NCCc2ncc(C)o2)oc(CNC(c2nocc2C)=O)cc1C C1(CC(=O)NCC2CCCC2C(N2CCC3(CC2)CC3)=O)Cc2ccccc2C1 c1(NC(C2SCCN(C(C(C)(C)OC)=O)C2)=O)ccc(Cl)c(C(F)(F)F)c1 N1(C(C(C=CC)O)=O)C2CCC1CC(O)(CNC(=O)COc1ccccc1Cl)C2 N1(C(c2cccc(OCC(=C)C)c2)C)C(=O)CN(CC2CCN2C(C)=O)C1=O C(=O)(CC(C)(C)C(F)F)N1C(C(C)C)C(C(N2CCN(CC(N)=O)CC2)=O)CC1 CC(C)CC(CNC(=O)CSC(C)C)NC(c1ccnc(N2CCOCC2)c1)=O c1(C(=O)NCC(C(C)C)NC(C2CCC(=O)N2C2CC2)=O)ccnc(C(F)F)c1 Cc1nc(C(N2CC(CNC(c3cc(O)n(C)n3)=O)C(C)C2)=O)ccc1Br N1(C(C2(CNC(c3ccnc([N+](=O)[O-])c3)=O)CC2)=O)CCN2CCCC2C1 C(=O)(CCP(C)(C)=O)NCC(CNC(c1nn(C)cc1C(C)=O)=O)OC CC(C)(C)CCC(=O)N1CC(NC(c2cc[nH]c2)=O)C(C(F)F)C1 N12CCN(CC1)CC2=O.c1(CNC2C(C(C)C3CC3)C2)ccc(O)nc1 C1(C(N2CC(O)(CCNC(C(n3c(C)ncc3)C)=O)C2)=O)CCC(=O)N1C1CC1 CC1CN(C(c2ccc(F)c(CCC(=O)O)c2)=O)C(C)C1C C12(CNC(C(CCC)OC)=O)CC(CO1)N(C(=O)CCCN(C)C)C2 N1(C(c2c(C)cno2)=O)CCN(C(=O)C(F)(F)C2(O)CCC2)CC(C)(F)C1 Cc1ncccc1-c1cn(CC(N2CCCC2n2nc(C(C)C)cc2C)=O)nn1 C1(OCC)CC2(C1)CC2C(=O)NC(C1CN(C(c2ccnc(O)c2)=O)C1)C c1(C(N2C(C)CC(NC(C=COCC)=O)C2)=O)c(Br)ccc(F)c1OC c1(C(N2CCC(C)C2CNC(=O)C=C(Cl)Cl)=O)cc(Cl)ccc1Cl C12(CNC(C3C(=C)C3)=O)CCC(N=c3[nH]nc(C(F)(F)F)s3)(CC1)CO2 CS(=O)c1ccc(CN(C=O)CC2(O)CN(C(=O)OC(C)(C)C)C2)cc1 C(=O)(C1COc2ccccc21)N1C2C(CNC(C(C)=CC3CC3)=O)C(CCC2)C1 c1(C(=O)NC(CNC(C2C(C)(C)CO2)=O)CO)ccc(Cc2nc[nH]n2)cc1 c1(CN(C(c2ccn(C(F)F)n2)C(=O)NCCC)C)cc(=O)n2cc(C)ccc2n1 n1(CC)cnnc1CNC(=O)NCC(C)(O)CC1CCCCC1 C1(C)(C(=O)NC(CC)CN(C(=O)C(C)NC(c2ccoc2)=O)C)CCCS1(=O)=O Cc1cc(NC(C2(NC(C3CCCCC3F)=O)CC2)=O)cc(O)c1 N1(CC(=O)N(C2CC2)CC)CC(C)C(=O)N(C)c2ccccc21 c1(OC)cccc(COCC(=O)N(C)CCNC(C2CCCC2(F)F)=O)c1 c1(N(C(c2c(I)cnn2C)C(=O)OCC2CC(F)(F)C2)CCOC)cccc(C)c1C C1(O)(C(C)NC(=O)CC2CC2C)CCN(C(C2C(c3ccccc3)C2(C)C)=O)C1 C(CCC(=O)NCCCCCNC(=O)Cc1csnn1)OCCOC Cc1ccc(NC(C23CCC(N)(CO2)C3)=O)cc1NC(c1ccccc1)=O c1(C(=O)NC2C(NC(Cn3cc(C(C)O)nn3)=O)CC2)coc2ccccc12 C1(CC)CCC1(c1nnnn1Cc1ccccc1)NCc1nc(C2CC2)no1 C1(CC(=O)N(CCCC(=O)N(C)C)C)CCCC(=O)N1 N1(C(CNC(=O)OCC)=O)CCC2(CCC2CNC(c2[nH]c(O)nc2C)=O)CC1 CCCC(C(=O)NC(C1CCCN1C(c1ccoc1COCC)=O)C)OCC N1(C(C2CN(CC)C(=O)C2)=O)CC2CC(CNC(=O)CN3CCC(O)CC3)C2C1 c1(N2C(CC)CCC2)ncc(C(N2CCC(C(C)O)CC2)=O)cc1C C1(CNC(c2nnc(CC)s2)=O)CC2(CCN(C(=O)C(O)C(C)(C)CC)C2)CO1 C1(O)(CN=c2ccnc(NC(c3ccncc3)C)[nH]2)CC2CCC1CC2 CCC(C)CC(=O)N1CC(CCNC(=O)C(F)(F)CC2CCCO2)C1 N1(C(C(C)Cn2cccn2)=O)CC2CCC1CC2NC(=O)Cn1cnnc1O CN1CCCN(C(C23CCCC2CCN3C(=O)Cn2[nH]cnc2=N)=O)CCC1 c1(C(=O)NC2COCCN(C(C3C(C)(CC)C3)=O)C2)cnn2c(C)cccc12 O=S(=O)(c1cnc(N2CCC(C3(C)N=N3)C2)c(Cl)c1)NC1CC1c1ccccn1 c1(CC)nc(NCC=CCNC(C23CCOC2CCOC3)=O)c(C#N)cc1C c1(C(=O)NC(C2CCCN(C(Cc3c(C)cccc3)=O)C2)C)ccc([N+](=O)[O-])o1 C1(C(=O)NC(CC=C)CNC(c2c(C)coc2C2CC2)=O)CCOC(C)(C)C1 C1(CCNC(C(c2ccc(F)c(F)c2)C)=O)CN(C(=O)C(C)(C)C)CCCO1 N1(CC(=O)N(C(CC)C(=O)N(C)CC2COCCO2)C)CC(=O)NC1=O c1(CNC(=O)NCCN(C(CC)CC)C)ccc(COC)cc1 c1(C(N(c2nc(-c3ccco3)cs2)C)=O)cccc(C(=O)NC2CC(=O)N2)c1 c1(Sc2nnc(C(=O)NCCOCCOC)s2)ccc(C#N)cc1C Cc1cc(F)sc1C(N1CC(OCC(=O)NCCC2COCCO2)C1)=O C=C(C(=O)NC1CC2(C1)CC(CNC(=O)C1CC1)C2)C(F)(F)F c1(CC)c(C(=O)NC2CN(C(=O)C=CC(C)C)CC2(C)C)cnc2cc(O)nn12 c1(NCCCC=CC)ncccc1S(=O)(=O)NCCc1cccs1 c1(C(N2CCC(c3c(C)cccn3)CC2)C)cccc2c1OCCC2 Cc1cc(O)c(C(=O)NC(C2CN(C(=O)CCC(=O)NC3CCCC3)C2)C)nn1 N1(C(CN2CC(C)(OC)C2)=O)CCC(CNC(=O)CN2C(C)CCC2C)C(C)C1 c1(CCC(=O)NC2C(C)CN(C(=O)CC34CCC(CC3)C4)C2)ccc(F)cc1F C(C(C)C(C)C(=O)NCCOCCN(C)C(c1ccn(C(C)C)c1)=O)OC c1(C(=O)NC(C(=O)NC(C)C(=O)NC2CC2)C2(O)CCC2)ccn(C2CC2)n1 CC(CNC(C1CC1(F)F)=O)C(=O)N(C)Cc1ncc[nH]1 C1(CC(=O)NCC(C#C)CC)CC2(CC2)CN1C(C1C(C(C)=O)C1(C)C)=O CC1(C)COCC(C(N2CC(NC(=O)Cn3cnc(Br)c3)C(O)C2)=O)O1 C(=O)(CCC(C)(F)F)N1CCC(C(F)F)(CNC(CCC=CCC=C)=O)C1 C1(C2CCN(C(c3ccc(CCCC)cc3)=O)C2)(NC(CCCCC=C)=O)CC1 c1(C(N2CC(CNC(=O)C=CI)C(C(F)(F)F)C2)=O)nccn2ccnc12 C1(C#N)(C(=O)NC(C(=O)N2CC(N(CC)CC)C2)(C)C)CCOCC1 C1(NC(c2ccc(N)c(F)c2)=O)CN(C(=O)CN2CC(=O)NC2=O)CC1C1CC1 c1(N(C(=O)C(=Cc2cn(C)cn2)F)C)cccc(CNC(=O)CN2CCCC2)c1 C(=O)(C(C(C)(C)C)NC(=O)CC1(NC(C)=O)CCC1)NC(CCC)CO N1(C(CCOC(C)C)=O)CCOCCC1C(N1CCC(CCF)CC1)=O c1(-c2cnc(SC)c(F)c2)ccc2cc(C(=O)NCCc3cccs3)[nH]c2c1 N1(CCC2N(C)CCC2)CCC(=O)N(CCc2ccccc2[N+](=O)[O-])C1=O C1(CNC(c2nc(COC)oc2)=O)CN(C(=O)C=CC(C)C)CCC12CCOC2 c1(C(N2CCCCCC2)C(=O)NCCCOC)ccccc1OC(F)F N1(C(c2n(CC)nnc2)=O)CCCC(NC(c2ccc(F)c(C)c2)=O)C1C c1(OC)ccccc1CNC(c1nc(-c2ccccc2CO)cs1)=O c1(C(=O)NC23CC(NC(c4c(N)ncc(O)c4)=O)(C2)C3)noc2ccc(Cl)cc12 c1(-c2nc(CCOC(COC)C)on2)ccc(C(F)(F)F)cc1 c1(C(=O)NCCN(c2ccccc2)C)ccc(NCC2CCSCC2)cc1 c1(C(=O)NCC(CC=C)NC(C2CC(C)(C)CO2)=O)sc(S(N)(=O)=O)cc1C C1(C)(NC(c2cc(CN(C)C)on2)=O)CCC(NC(C2CC(C(F)F)C2)=O)CC1 c1(C(N(CCCOCCN(C(c2c(C)csc2)=O)C)C)=O)cc(F)cc(C)c1N c1(C(=O)NC2CCC2NC(c2cnc3[nH]ncc3c2)=O)coc2c1C(=O)NCC2 C1(NC(c2cnc(C)[nH]2)=O)CN(C(=O)Cc2nc(-c3cccs3)oc2C)CC1C CC1CN(C(c2cc(CNC(=O)C(C)CC(C)(C)C)[nH]n2)=O)C(C)C(C)(C)O1 C(=O)(C(C)(C)n1ccnn1)NCC=CCC(=O)NCC1CN(C(C)=O)C1 C1(C)(CNC(C(C)=C(C)C)=O)CCCN(C(=O)C(C)CC(C)C)C1 C(=O)(CS(=O)c1cccc(OC)c1)NCC(=O)NCCCC(C)NC(=O)OCC CCN(OC)C(=O)CNC(C1C=CCN(C(=O)CN2C(=O)CNC2=O)C1)=O c1(C(N2C(CNC(C3N(CC)CC3)=O)CC(O)C2)=O)cc2n(n1)CCNS2(=O)=O c1(CCC(=O)OCC)ccc(NC(N2CCC(N3CCOCC3)C2)=O)cc1 C1(C)(CC(=O)N(CCC(C)O)C)CCN1C(=O)C(c1cnn(C)c1)O C12(OC)CCC(C(=O)N(C)CCNC(c3nnn(C)c3N)=O)(CC1)CC2 CCCC(CC)C(=O)N1CCC(CNC(=O)CC(C)(O)c2ccccc2)CC1 c1(N(CCCN(C)C(C2(n3cccn3)CCCC2)=O)C)ccc([N+](=O)[O-])c(O)n1 Cc1ccc2oc(C(N3CCCC(N(C)C(C4CCCN4C)=O)CC3)=O)cc2n1 C(c1ccc2c(c1)OCO2)=CC(=O)NC(C(C)NC(=O)CCNC(N)=O)C c1(C(=O)NCC2CC(C)N(C(=O)CC(F)(F)F)C2)cccc2nc(S)oc12 Cc1cn2nc(C(=O)N(C3CCN(C(C4(C)CCOC4)=O)CC3)C)cc(C)c2n1 N1(C(CNC(C(CC)C)=O)=O)CCCCCCC1C(=O)NC(CCO)C1CCCC1 N1(C(C2=NOC(C)C2)=O)CCC2(C1)CN(C(c1ccc(C(O)CF)cc1)=O)C2 c1(C(=O)NC2C(CCC)CN(C(=O)C(C)CC)C2)cc2ccccc2cn1 c1(CC)cc(C(=O)NCCC(C)(C)NC(=O)CC2CC(O)C2(C)C)cc(F)c1 Cc1c(C(=O)NCc2cc(C(=O)N(C3CCNC(=O)CC3)CC)on2)c[nH]c1C#N N1(C(c2cc(SC)c(C)o2)=O)CCCCC(NC(=O)CCCC2CCCCC2)C1 c1(CNCc2cnc(CC)s2)ccc(C=O)c(C)n1.C(C)(C)(C)OC=O N1(C(CCC)=O)CCN(C(C2CN(Cc3ncccc3Br)CCS2)=O)CC1 C(N=c1[nH]cnc2ccsc12)C1CN(C(=O)CCn2cnnn2)CC1C1CC1 C1(C(=O)NC(CC=C)CC=C)CC(C)(C)CN1C(=O)C(c1ccn(C)n1)C c1(N2CCC(C(C)C)CC2)nc(=NC2CCCC(C)C2)[nH]c2c1COC2 N1(C(c2c(COC)cc[nH]2)=O)CCN(C(=O)CN2CCNC2=O)CC1CCO S(=O)(=O)(c1ccc(NC(CC(C)C)C(N)=O)cc1Cl)N1C(CC)CCCC1 N1(C(C(C)NC(=O)NC2(c3cccs3)CC2)=O)CCCCC1C Cc1nc(C(=O)NC(CNC(c2nc(O)n(C)n2)=O)C2CCC2)n(C)n1 N1(C(C2(CNC(CN3CCC(C)CC3)=O)CCCC2)=O)CC2C(C1)C2(C)C C(=O)(C(C(=O)NC(C1CN(C(C2CC3(CC3)C2)=O)CCO1)C)OC)OC c1(C(N(CC(C)CNC(=O)C(C)(C)C(C)O)C)=O)ccc([N+](=O)[O-])c(Cl)c1 C#CCC(C)(C(=O)N(C)CCOC1CC1)NC(=O)C(O)CC1CCCC1 C(CCCC(C)(C)C)(C(=O)NC1CCOCC1)N(C(C)CC#N)C c1(C(=O)NCC2CN(C(CC(CC)SC)=O)C2)nc2sc(C)cn2c1C c1(C(=O)NCC23CC(NC(CS(N)(=O)=O)=O)(C2)C3)c(Cl)ccc(Cl)c1O C12(NC(COC)=O)CCN(C(=O)C=Cc3ccccc3C)CCC1C2 CC(C)(C)S(=O)(=O)Cc1noc(CCCN)n1 C1(C#N)(OC(C(COCC=C)c2ccccc2)=O)CCCOC1 C1(C(N2CC(CCc3cn(-c4ccc(Cl)cc4)nn3)C2)C)CC(C)(C)CCO1 Cc1cc(N)c(C)nc1C(=O)NC1CCN(C(=O)C(c2ccncc2)C)C1C N1(C(COCCOCCOC)=O)CCN(C(C2CC23CCC3)=O)C2COCC12 c1(C(=O)NC2CN(C(COCCC#C)=O)CC2C)ccc(OC)c(C(F)F)c1 c1(NC(=O)COc2ccc(CO)c(Cl)c2)ccc2c(c1)OC1(CCCCC1)O2 C1(C(N2CCCC(CCNC(=O)CC3(C)CC3)C2)=O)(COC)CCC(=O)N1 Cc1cc(C(=O)NCCC2CN(C(=O)C(F)CC3CC3)CC2C)nn1C(F)F C1(NC(CC=C(C)C)=O)CCCN(C(=O)COC2CCCC2)C1 C(=O)(C(C)(C#N)CC)NC(CC)CNC(=O)Cc1cc[nH]n1 C1(C(=O)NC(C(C)C)CNC(C2(Cc3ccccc3)CC2)=O)CCS(=O)(=O)N1 c1(C(N2CCCC(N(C(=O)C=Cc3scnc3C)CC)C2)=O)c(F)cccc1Cl N1(C(c2cc(C)[nH]n2)=O)CCCN(C(=O)C(C)N=[N+]=[N-])CC1 c1(C(=O)NCCN(CC(=O)NC2CCCC(C)C2)CCC)cccc(C)n1 c1(C(=O)NCCC2(O)CN(C(c3n(C)nc(O)c3)=O)C2)nnc(O)cc1O C1(OCC)CCN(C(=O)CC(C)NC(c2csc(CO)n2)=O)C1 CCC(C)(C)C(C)CC(=O)NC1(C)CN(C(c2ccc(NCC(C)C)nc2)=O)C1 C(=O)(CC(C(F)(F)F)C1CC1)N1CC(N(C(COCCC)=O)C)C2(C1)CC2 C1(NC(C(c2ccccc2)NC(=O)OC)=O)CCCN(c2ccc(C)cn2)C1 C1(CC)CN(C(=O)CCCC(C)NC(=O)C(C)CC(=O)OC)CCN1C Cc1ccc(NC(=O)C(C2CCN(C(=O)CC3CCC(C)(C)O3)C2)F)c(CO)c1 N1(C(C(CC)n2cccn2)=O)CCN(C(=O)CC2OCCCO2)CC1CF Cc1cccc2cc(C(=O)NCCOCCNC(c3ccc([N+](=O)[O-])[nH]3)=O)oc12 CCC(F)(F)CC(=O)N(C)CC1(CNC(C2CC(C(F)(F)F)C2)=O)CC1 N1(C(C(C=C=C)C)=O)C2CCC1CN(C(c1cnc3n1CCCC3)=O)C2 C1(C(N(CCCC)C)=O)CN(C(C2CC(O)(CC#N)C2)=O)C(C)(C)C1 C1(C(=O)NCC(CC)NC(c2ccn(CCF)n2)=O)CCCC(=O)CC1 Cc1ccc(O)cc1C(=O)NCC1CN(C(=O)CC2CC2)CC1C(C)C c1(C(=O)NCCCN(C(=O)CCCN=[N+]=[N-])C)ccc2n[nH]cc2c1 Cc1cc2ncn(Cc3cn(CCNC(=O)C(=O)CCC(C)C)nn3)c2cc1C C1(CC)CCC(C(=O)NCC2(OC)CN(C(C3CC(O)C3)=O)C2)C1 N1(C(c2c(CC)csc2)=O)CC2CCC2(CC(=O)NCCc2ncon2)C1 C1(CCC)CN(C(C2C3CC2N(C(=O)C(C)n2ccnc2)C3)=O)CCO1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CCCC(CCNC(=O)C2=CC(C)(C)C2)CC1 C(=O)(C1CCCc2nncn21)N1CCOCC(CNC(c2ccc(O)cn2)=O)C1 C1(C)(n2cnc([N+](=O)[O-])n2)CC12CCN(C(C)=O)CC2.CCC1CC(=O)CS1 C1(C(=O)OC)CC2(CCC2)CN1C(c1ccc(OCCOC)c(C(F)(F)F)c1)=O CC(CC(C)(F)F)C(=O)NC1CN(C(c2cc(N(C)C)cc(Br)c2)=O)C1 CCN=c1ccc(C(=O)NCCCC2CCCCN2C(C23CSCC2C3)=O)c[nH]1 c1(NC(N2CC3C(C(=O)OCC)(CNC3)C2)=O)nc2ccc(F)cc2[nH]1 N1(Cc2c(CC)con2)C(=O)CCN(Cc2ccc(Cl)cc2OCC)C1=O C=Cc1cccc(-c2cnccc2CN(C2CCS(=O)(=O)C2)CCO)c1 N1(C(c2cnc(OC)nc2C)=O)CC(NC(=O)C(C)N(C)C)C2CCCCC12 N1(C(=O)NCCCCCCCCCC)CCCC(O)(C2(C(=O)O)CCC2)C1 C1(NC(CNC(N)=O)=O)COC2(C1)CN(C(C1CCCS1(=O)=O)=O)C2 Cc1ncc(NC(C2CCN(C(C34CCC(C3)C4)=O)C2(C)C)=O)c(C)n1 S(=O)(=O)(c1ccc(Br)s1)NCCC(CNC(=O)OC)OC c1(C(N(C(CNC(CCC(=O)NC)=O)C)C)=O)cc(C)c(F)cc1N C1(NC(N(c2ccc(C#N)nc2)C)=O)CC2C(O)C(O)CC12 C1(C(=O)NCC2N(C(CN(C3CCCC3)C)=O)CC2)CCC12CCOCC2 C(=O)(C(C(C)(C)C)N(C)C)NCC(CC(C)C)NC(CCNC(C(C)OC)=O)=O c1(-n2cc(-c3c(OC)ccnc3)nn2)cc(C(=O)NCCCC(=O)O)ccc1Cl C1(NC(c2cnc(CC)[nH]2)=O)CC12CC(NC(C1CC1C1CC1)=O)C2 C(N=c1[nH]cnc(C)c1Br)C1OCC(CNC(C(CC)CCOC)=O)C1 N1(C(C=C(C)CNC(C23CCC(C2)C3)=O)=O)CCn2nccc21 c1(CC)c(C(=O)NC2(C)CCCC2NC(c2cnn(C(C)C)c2)=O)ccn1C Cc1nn(CCF)cc1NC(C1(CNC(C2CCCS2)=O)CCCC1)=O C1(C(=O)NOCc2cn[nH]c2)(CC=C)CCN(C(=O)CSC(C)(C)C)C1 C#CC1(C(=O)NCC2(OC)CCN(C(=O)CCC#CC)C2)CCCCC1 c1(OC(C)C(N2CC3CC3(C(=O)Nc3ccc(Cl)nn3)C2)=O)ccc(Br)cc1Br Cn1c(C(N2CCC3CC23C(=O)NCC2CCN(C(N)=O)C2)=O)nnc1S C1(CCNC(C=CC=CC)=O)CN(C(=O)CCC(=O)c2cnn(C)c2)CCCO1 N1(C(CCN(CCC)C)=O)CCCC(O)(CCNC(c2ccccc2OC)=O)C1 c1(C(N2CC3(N(C(c4c(CC)nn[nH]4)=O)CC3)C2)=O)cc2ccncc2o1 C1(NC(=O)Cc2cncnc2O)CN(C(C2CC=CC2)=O)C2(CCOCC2)C1 C(N=c1cc(C#N)nc(C)[nH]1)C1CN(C(C2(C(=O)OCC)CC2)=O)CC12CC2 C12(CNC(C(C)C3CC3)=O)CCCC1N(C(c1cc3n(n1)CCCC3)=O)CC2 C#Cc1cc(C(N2CC(O)CC2(C)C(=O)N(C)CC2CC2C)=O)ccc1C C(=O)(NNC(=O)N1CCCC(OC)C1)c1cc(OC)n[nH]1 C1(C(=O)Nc2ccc(OC)c(F)c2)CC2(CCC2)CN1C(=O)C(F)=CC1CC1 C1(CNC(C2(SC)CCSC2)=O)CN(C(C2CC(C)=NO2)=O)CCO1 N1(C(c2cnc(CC)s2)=O)CCC(NC(=O)CC(C(N)=O)NC(C)=O)CC1C C1(C(=O)NC(C)CCNC(c2cn(CCC3CC3)nn2)=O)CN(CP(C)(C)=O)C1 c1(-c2cc(C(=O)NC(CC)CN(C)C(c3occc3F)=O)n[nH]2)ccc(C)cc1 N1(CCC(N)=O)CCN(CC2CC(=O)N(CC(F)(F)F)C2)CC1 C(CC(C(=O)NC1CC=C(C)CC1)NC(c1ccoc1CC)=O)OCC c1(C(=O)NC(CNC(c2c(CCC)nco2)=O)CCOC)cncc(Cl)c1 C(C(CNC(=O)CC1COCCOC1)C(F)(F)F)NC(CC1N(C)CCOC1)=O C1(CC)CCCC(C)N1CCOCCOCc1ccccc1C C#CC1(C(=O)N(C2CC2C)C)CN(C(=O)C(=O)C(C)C)C1 C1(NC(CCN(C(CCC)C)C)=O)CCN(C(=O)CCc2cncc(C)c2)CC1 c1(CNC(C(C2CC2)OC)=O)ccc2c(c1)CCN(C(C1NC(=O)C3CC13)=O)C2 CC(O)C(C)(C)CNC(C1(NC(C2CN(C(N)=O)C2)=O)CCSC1)=O c1(CC)cccc(C(=O)NC(CO)C(C)NC(c2nc(C)oc2C)=O)c1 c1(C(=O)NC(C(C)NC(=O)C=Cc2ccsc2)(C)C)sc(Cl)cc1Cl CC1COc2ccc(C(N3CC4CCCC4(NC(C45CC(F)(C4)C5)=O)C3)=O)cc21 Cc1[nH]c(=NCc2cnccc2Cl)sc1C(=O)NCC1(O)CCCC1 CC1CNc2c(C(=O)NCC3CN(C(C4(N(C)C)CCC4)=O)CCO3)cnn2C1 N1(C(CNC(=O)NC)=O)CCC(NC(=O)Cn2ncnn2)C(C)C1 c1(C(N2CC(C)(NC(C(C=C)O)=O)C2)=O)cc(S(=O)(=O)N(C)C)c[nH]1 N1(C(C2CCC(=O)N2)=O)CCOC2(CCN(C(=O)COc3cncc(Cl)n3)C2)C1 N1(CC(=O)N(c2cc(Cl)cc(Br)c2)C)C(=O)N(C)C2(CCCCC2)C1=O CC1=NS(=O)(=O)NC=C1C(=O)N1CC2(NC(=O)C(n3cc(C)cn3)C)CCC1C2 N1(C(Cn2nc(C)oc2=O)=O)CC(CNC(C2(C)COC(=O)C2)=O)CC1(C)C N1(C(c2c(OC)c(Cl)c(Cl)cc2)=O)C2CCCC1CC(=O)NC2 c1(C(N(C)CC2CCCN(C(=O)COCC3CCC3)C2)=O)nccc2nn[nH]c12 N1(C(C2=NOC(C(C)(C)C)C2)=O)CC2(C1)SCCC2NC(=O)CCS(N)(=O)=O c1(CC)conc1CC(=O)N(C(C)CCNC(C1(c2cnn(C)c2)CC1)=O)C c1(NCc2cccc(C(=O)NCC(CC(N)=O)O)c2)nc2ccc([N+](=O)[O-])cc2s1 Cc1ncc([N+](=O)[O-])n1CC(N1CCC(CNC(=O)C(=O)C(F)(F)F)CC1C)=O c1(C(=O)NC(C(C)NC(C(CC)O)=O)(C)C)cc(F)cc(F)c1O C(=O)(C(Cc1cc[nH]n1)NC(C1CN(C(N)=O)C1)=O)NCC(C)(O)C1CCCC1 CCS(=O)(=O)CC(=O)NC(CC1CC1)C(=O)NC(c1nncn1C)CO c1(C(N2C(CNC(C3CC4C=CC3C4)=O)CC(OC)C2)=O)ccc2c(c1)COC2 CC1ON=C(C(=O)N(CC(C)(C)CNC(c2nn(C)cc2Cl)=O)C)C1C Cc1nsc(C(=O)NC(Cc2cn[nH]c2)C(=O)NC(c2cnn(C)c2)CO)c1N C(C(=O)N(C)CCNC(=O)CCc1c(C)noc1Cl)(C(C)(C)C)NC(C)=O C(C(=O)NNc1ccccc1S(C)(=O)=O)Sc1n(CC)c2c(n1)cccc2 N1(C(C2(SC)CC2)=O)CC=C(C(=O)NCCc2ccc(O)cn2)CC1 c1(C(N2CCC(CCNC(=O)CCOC3CCOC3)C2)=O)ccc2[nH]ccc2n1 C1(NC(c2c(C)cnn2C)=O)CC2CC1N(C(=O)C(O)Cc1cn(C)cn1)C2 C1(C(=O)NC2CN(C(=O)CCCc3nnc(-c4ccccc4)o3)C2)CC(F)C(=O)N1 N#Cc1c(-c2cn(CCCC(=O)NCc3ncc(F)cn3)nn2)cccc1N C(=O)(C#CC1CN(C(=O)OC(C)(C)C)C1)N1CC(NC(CCC)=O)C(C)(C)C1 C#CC1C2CN(C(=O)NCC(C(C)C)OCCO)CC12.C=O N1(C(CCc2n(C)ncc2)=O)CC(NC(c2n[nH]cc2F)=O)C(O)C1 C1(c2cn(CC)nc2)CS(=O)(=O)CCN1C(=O)NC1CCC(C(C)C)CC1 C=CC(C)(CC)C(=O)N1CC=CC(NC(=O)C=Cc2cn(C)nn2)C1 N1(C(CC=C)=O)CC(C(=O)N(C(C)C(C)C)CC)C(F)(F)C1 C1(C(C(=O)N(CC(C(C)C)C)C)C)CCN(C(=O)Cc2ccns2)CC1 C1(C(C)C)CN(C(C2CCC(F)(F)C2)=O)CCN1C(=O)CN(C1CCC1)C C1(C(N(C(CNC(c2nc(CC)sc2)=O)C)C)=O)Cc2cc(Br)ccc2O1 C1(c2n(CCCCCC)nnn2)(NCc2ccc(CC)cc2)CC(C)N(C)C1 Cc1cc(C(=O)NC2CCC(CNC(=O)CC3(C)OCCO3)C2)sn1 C1(NC(C2N(C(CC)=O)CCCC2)=O)CC2CN(C(=O)C(C(C)C)OC)CC2C1 C1(C(N2CCC(c3ccon3)C2)=O)CN(C(=O)Cn2cc(CO)nn2)CCO1 N1(CCSCC)CC(C)N(C(=O)CNC(=O)NCC#C)CC1C C(CC(C)(C)C)(C(=O)N1CC(F)CC1CC(N1CC(OCCF)C1)=O)OC C(C)(CNC(c1c(C)ncn1C)=O)(C(C)C)NC(CC1(OC)CCCC1)=O C1(CC(=O)N(CCN(C(C(C)SC)=O)C(C)C)C)CCCC(C)O1 N1(CCC)C(=O)NC(c2cc(Cl)cc(Cl)c2[N+](=O)[O-])C(C(=O)OCC)=C1C1CC1 CCC(C)C(C)(O)CNC(=O)C(C1(O)CCCCC1)NC(c1cc(C#N)n(C)n1)=O c1(CC(N2C(CCNC(C3(C)CSC3)=O)CCCC2)=O)ccc2c(c1)CCC2 c1(C(N2CC(CNC(c3c(C)cc(N)cn3)=O)C2)=O)cccn2c(O)nnc12 Cn1ncc(C(N2CCC(=CCNC(c3cc(Cl)cnc3O)=O)CC2)=O)c1C#N c1(NC2C(O)COC2)nc2ccc(Cl)cc2c(=NCC(F)(F)Cl)[nH]1 CCS(=O)(=O)c1ccc(C(C)NC(=O)CC23CCC(CC2)OC3)cc1 N1(C(CCCCC=CC)=O)CCC(C2CC2)C1CNC(=O)CC(Cl)Cl N1(C(c2c(Cl)ccc(C)c2)=O)CC2CCC(NC(c3cnc(O)n3C)=O)(C2)C1 c1(SC)ccc([N+](=O)[O-])c(-c2ccc(C3(C(N4CCC4CO)=O)CC3)cc2)c1 C=CC(C)CC(=O)NCc1cncc(C(=O)NCc2cc(C(C)C)n[nH]2)c1 Cc1ccc(O)cc1CNC(=O)C(C)CN(C(=O)CN1CCN(C)CC1)C c1(C(N2C(CCCNC(C(=O)NCC3CC3)=O)CCC2)=O)nc2ccccc2[nH]1 Cc1ccncc1N1CCC(C2CCCCN2C(=O)CSC(F)F)C1 N1(C(C2(O)CCN(Cc3ccc(C)s3)C2)=O)Cc2cccc(O)c2C1 CN1C(=O)CCC1C(=O)NCC1CCCC1NC(c1ocnc1C1CC1)=O c1(OC)cncc(C=CC(N2CCC(NC(=O)C(C)C3CC3)C(F)C2)=O)c1 N1(C(C(CCSC)O)=O)CCN(C(c2ncc(C#N)cc2Cl)=O)CC12CCC2 C1(SC)CN(C(=O)CC2CCCC(NC(=O)OC(C)(C)C)C2)CCC1(F)F CC1(C(=O)NC(C2CCCCC2)CNC(c2nc(=N)cc[nH]2)=O)CCC(=O)N1 Cc1cc(Cl)c(C(C)(C)NC(=O)C(=O)N(C2CCOC2)C)cc1F CC(C)CCC(O)C(=O)N1CCC(NC(c2cncc(C(N)=O)c2)=O)CC1C C1(CNC(c2c(C)nc[nH]2)=O)(NC(c2ccc(C(N)=O)[nH]2)=O)CC2CCC1C2 C=C(C(=O)N1CC(NC(C2(C(C)C)CCC2)=O)C(F)C1)C(F)(F)F c1(C(=O)OC)cccc(CN2CC3CN(c4ccccc4)CC32)c1[N+](=O)[O-] S(=O)(=O)(c1cc(C(=O)O)ccc1F)NC(c1ccc(N(C)C)cc1)C1CC1 C12(NC(CC(C)SC)=O)CCC(CNC(c3cnoc3C(C)C)=O)(CC1)OC2 c1(OC)ccc(C(=O)NCCC(C)(C)NC(C23CCCC2C3(F)F)=O)c(N)c1 n1(CC)ncc2c1CCC(C(=O)NNC(=O)Cc1cc[nH]c(=N)c1)C2 N1(C(=O)Cc2cc[nH]c2)CCC2CCN(C(c3cc4c(Cl)nccc4s3)=O)C2C1 c1(OC)ccc(C(C)NC(=O)C(n2cc(C(C)OCCOC)nn2)C)cc1C CC#CC1CCN(C(=O)CCOCCCNC(c2cc(C(F)F)[nH]n2)=O)C1 CCC(C)CCCCC(=O)NC1(CNC(c2ccc(C)s2)=O)CC1 c1(C(N2CCN(C(=O)Cc3nc[nH]n3)CC2CO)=O)cc2cc[nH]c2cn1 c1(C(=O)NCC2C(NC(c3cnc(C)[nH]3)=O)CCC2)c(C)cccc1N C1(NC(CC2CC(OCC)C2)=O)CCCN(C(=O)Cc2ccc(Cl)c(F)c2)C1C N1(C(C2CC(=O)N2)=O)CCCC(N=c2ccnc(C3CC3)[nH]2)C1 C1(N(C(COCCC(C)C)=O)C)CCC2CN(C(=O)C=Cc3ccncn3)CC12 c1ncccn1.CCC(C)OC.C1(=O)COCCOCCOCCNC1=O C1(CCC)(NC(=O)C=Cc2cnc[nH]2)CCCN(C(c2cc(CC)nn2C)=O)C1 N1(C(Cc2nc(NC(c3c(C)cccc3)=O)sc2)=O)CC(O)C(O)CC12CCC2 C1(C(=O)OC)CS(=O)(=O)C2CN(C(c3ccc(CO)c(F)c3)=O)CC12 N1(C(C(CC)(C#N)CC)=O)CCC2(CC1)CN(C(=O)CC=C(Cl)Cl)CCO2 N1(C(CSC(C)C)=O)CCC2(CC1)CCN(C(C1CC13CCC(F)(F)CC3)=O)C2 C1(C(N2CCCC(N(C(=O)Cc3ccn(C)n3)C)CC2)=O)CC2CCCCCC12 c1(OCC(N2CCCC(N(CCF)C(c3cn[nH]c3)=O)C2)=O)cc(F)cc(F)c1 CC1(C)CCC(CNC(c2cccn3nnnc23)=O)N(C(C2CC(CF)C2)=O)C1 c1(SC)nc(C)c(C(=O)O)s1.c1(OCC(=O)OC)cccc(C2CN2)c1 C(=O)(C(CC(C)(C)C)NC(=O)CC(O)CC(C)C)N(C)Cc1c(C)cccc1 CCCCC(C(=O)N1CCC(F)(F)C(CNC(c2cc(O)nn2C)=O)C1)C(C)C c1(C(=O)NC2CCC2NC(C2CCN(C3COC3)C2)=O)cccc[n+]1[O-] c1(C(=O)Nc2nnn(-c3ccc(C)cc3)c2C)[nH]c2ccccc2c1Cl C(=O)(C1CCCc2sccc21)N1C(CNC(=O)C=C2CCSCC2)CC(F)C1 S(=O)(=O)(c1ccccc1)NCC(=O)NC1C(C)CCN(C(c2c(C)nns2)=O)C1 c1(C(=O)NCCC(CNC(c2n(CCC)ccc2)=O)OC)cc(C(C)C)n(C)n1 C(=O)(CC(C)C(C)(C)NC(c1ncncc1N)=O)N1CCC(CCOC)C1 C1(CNC(C(CC=C)C)=O)C(O)C(O)CN1C(c1nc(Cl)sc1Br)=O CC(C)C(C)(O)C(=O)N1CCN(C(=O)C(c2ccccn2)O)C(CO)C1 N1(C(C2(CCCC)CC2)=O)Cc2nccn2CC(NC(C2CC(SC)C2)=O)C1 c1(SC)cnn(C)c1C(N1CCC(CO)(NC(=O)C=C(C)Cl)C1)=O N1(C(C(C)CC2CC2)=O)CC(CNC(c2ccncc2F)=O)OC2(CCC2)C1 C(=O)(C(C)(C)CC=C)N1C(C(=O)NCCNC2(CC#C)CCOCC2)CC2CC21 c1(C(=O)NC(c2cn(CC(C(=O)OCC)O)nn2)C)cc([N+](=O)[O-])c(C)cc1C Cn1ncc2c1CC(C(N1CC(NC(c3ccc(C(C)(F)F)cn3)=O)C1)=O)CC2 N1(C(CC(OCC)OCC)=O)CC(NC(=O)CCSC)CC(C)(C)C1 c1(OCC)ccc(CNC2CC2C(=O)Nc2ccc(F)c(C#N)c2)c(F)c1F C1(C(=O)NCC(CCCC)NC(=O)Cc2cc(C)cc(C)c2)CC(S(C)(=O)=O)C1 N1(C(C(C(C)C)OCC)=O)CCCC(CNC(c2nnn(C)c2C(F)F)=O)CC1 C1(NC(CC(=O)NCC(F)(F)F)=O)CC2CC(C1)N(C(c1cnc(Cl)[nH]1)=O)C2 C#Cc1ccc(C(=O)N(C2CN(C(=O)Cn3cccnc3=O)CC2F)C)cc1C c1(NCC2(C)CCOC2)ccc(S(=O)(=O)N2CCCCCC2)c(Cl)c1 C1(C2CC2)(C(=O)NC2CCN(C(c3nn(C(CC)CC)c(C)c3)=O)C2)CC=CC1 n1(CC(=O)NCC2(CCNC(c3cc(=O)cc(Cl)[nH]3)=O)CC2)ccc(O)nc1=O C1(NC(C2(CNC(C3OCC(C)(C)C3)=O)CC=CC2)=O)COCC1N=[N+]=[N-] C1(N=[N+]=[N-])(C(=O)NC2C(C)NC(=O)CC2)CCN(C(=O)Cc2ccccc2F)C1 c1(NC(CC)=O)cncc(C(N2CC(C(C)NC(c3cnc(CC)s3)=O)C2)=O)c1 c1(C(=O)NC(CNC(c2cccc(CNC(C)=O)c2)=O)C)ccc(F)cc1F N1(C(c2n[nH]c(=N)[nH]2)=O)CC23CCCCC2(C1)CN(C(=O)CC1CCOC1)C3 c1(C(=O)N=c2cc(C3CCCCC3)n(C)[nH]2)cnc(SC)c([N+](=O)[O-])c1.CO N1(C(CCC=CC)=O)CCOC(C2CN(C(c3[nH]cc(C)c3C)=O)C2)C1 C1(N(C(c2c(CC)cc[nH]2)=O)C)CN(C(=O)C(CC2CC2)OC)CC12CC2 c1(C(=O)NCC2C(C(=O)NCC(C)SC)CCC2)cn(C)ccc1=O c1(C(N2CCCCC(NC(C3C(=C)C3)=O)C2)=O)ccc2ccsc2c1 N1(C(c2c(CC)c(OC)ccc2)=O)CC(C2CCCN(C(=O)CC(C)SC)C2)C1 Cc1oc2cc(C(=O)NC(CNC(C3CC=CCC3C)=O)C(C)(C)C)[nH]c2c1C c1(C(C(=O)NC2(CNC(C(C(CC)O)C)=O)CCC2)=O)c[nH]c2cc(F)ccc12 N1(C(CNC(CC(C)C)=O)=O)CC2CC(NC(c3cnn(C(F)(F)F)c3)=O)C1C2 c1(C(=O)NC2(CO)CCN(C(CCCCC)=O)C2)cc(Cl)cc(Cl)c1F Cc1ccc2oc(N3CC4CCCC(NC(C5CC(C)(F)C5)=O)C4C3)nc2c1 C1(CNC(C(C)SCC)=O)CN(C(=O)Cc2ccccc2OC(C)C)CCO1 CCCCC(C(=O)NCC1(C)CCCN1C(c1ccccc1OC)=O)C(C)C Cc1cc(=NCc2nncn2-c2ccccc2)[nH]c(C)n1 C1(C)(CC)CCN(C(=O)C(C)Oc2ccc(N3CCCC3)cc2)C1 C1(OC)COCCC1N=c1[nH]c(N2CC(N3CCOC3=O)C2)nc(=N)[nH]1 c1(C(=O)NC2CCC(NC(CS(=O)(=O)NC)=O)C2)cc2c(s1)CCCC2 c1(OC)cccc(CC(=O)NC2CN(C(=O)CCc3cncs3)C3CC23)c1 C1(CCC)(NC(c2sccc2C)=O)CCCN(C(=O)C(C)(C)N(C)C)C1 C(CCCC(=O)NC(CO)C1CCC1)NC(C=CC(C)C)=O c1(C(=O)NCCCN(C(C2CCCC2C2CC2)=O)CC)cc(N(C)C)ccc1N c1(CC)[nH][nH]c(=NC(=O)N2CCN(C)CC2CN)c1-c1nn[nH]n1 c1(C(=O)NCC2(Cn3cc(CO)nn3)CC2)c(O)ccc(Br)c1Cl O=C(CCC1CCC1)NOC1CCCN(C(C2CC3C=CC2C3)c2cscn2)C1 N1(C(c2cnc(SC)nc2O)=O)CCC(NC(=O)C(C)S(N)(=O)=O)C12CCCC2 Cc1[nH]cc(C(=O)NC2CCCCCN(C(C3(F)CCCOC3)=O)C2)c(=O)c1Cl Cc1cc(C(=O)NCC(c2ccccc2)N(C)C(C2CC(O)C2)=O)c(F)cc1Cl N1(C(C=C(C)C(C)C)=O)CCC(NC(C2CCN(C(N)=O)CC2)=O)CC(C)(C)C1 C(=O)(C(F)CC(C)C)NCCC1N(C(Cc2c(OC)cccc2)=O)CC(OC)C1 N1(C(C2(CC(C)=O)CC2)=O)CC(C(N2CCC2(C)C(C)C)=O)CCC1(C)C N1(C(CC(C)(C)C#N)=O)CCC(F)(F)C(CNC(c2cc3c(o2)CCCC3)=O)C1 N1(C(c2cc(C)no2)=O)CCC=CC1C(=O)NCCCC1CCOC1=O c1(C(=O)NC2C(C)N(C(c3cc(CCO)on3)=O)CCC2)ccc2ccsc2c1 N1(C(C(C)OCCC=C)=O)CCN(C(=O)C2=NOC(C)C2)CC(C)(F)C1 c1(CC)ccccc1C(CNC(=O)C(C)n1ccnc1)NC(c1cnns1)=O C1(NC(CCCc2c(C)ccs2)=O)CCN(C(=O)C(C)N(C)C)C(C)C1 C1(NC(C2(C=C)CCOCC2)=O)CCC2CN(C(=O)C3=CCCOC3)CC2C1 c1(CNC(C2(CC)CCOC2)=O)nc(C)c(C(=O)N(C(C)C(=O)N(C)C)CC)o1 C1(C(=O)NCCSCCC=C)C(CC)CCN1C(=O)C(CSC)OC c1(CC)ccccc1C(CNC(=O)C(C)CN(C)C)NC(=O)CNC=O C#Cc1cncc(C(N2CCC(O)(C(C)NC(c3csc4nccn34)=O)C2)=O)c1 C1(NC(CCCCC)=O)CCN(C(C2CCN(CC(F)(F)F)C2)=O)CC1O c1(-n2c(C)ncn2)ccc(NC(c2ccc(C3(C)CCO3)cc2)=O)cc1 N1(C(c2csc(O)n2)=O)CC2OCCN(C(c3cccc4cncn34)=O)C2C1 c1(N(C)C)ccc(NC(=O)CCC2(NC(C3(O)CCSCC3)=O)CCC2)cn1 c1(C(N(CCNC(c2ccn(C)c2)=O)C2CC2)=O)cc(O)nn1C c1(C(N2CC(C(=O)NC3CCC(F)(F)C3O)(COC)C2)=O)cccc2nn[nH]c12 c1(C(=O)NC2C(NC(=O)Cn3cnnc3O)CC2)ccc(C2CC2)nc1O c1(C(N2CCC(C(C)(C)NC(c3cnn(C)n3)=O)C2)=O)cc(O)cc(=O)o1 C=CC1(CC(=O)NCC2(O)CCCOC2)CN(C(=O)C(O)c2ccsc2)C1 C1(C(=O)NC2CC(C)(NC(c3cc(C(CC)CC)no3)=O)C2)CCS(=O)(=O)N1C C1(CN(C)C)CN(S(=O)(=O)CCc2ccc(C(=O)O)o2)CCO1 C1(NC(C2CCC(C)O2)=O)CC2CCCC(C1)N2C(c1cc2cn[nH]c2cn1)=O c1(C(N2CCCC(N(C(C(CC#C)O)=O)CC)C2)=O)c(N)cc(OC)cc1F c1(C(=O)NC2(CC=C)CCN(C(c3cnnn3CC)=O)C2)cc(=N)[nH]c(Cl)n1 C(C(C)(C)CNC(=O)CN(C(c1cnccn1)=O)CC1CC1)SC C(CCC(=O)O)(C(N)=O)CC(N1C(c2ccc(C)cc2)C(C)C1)c1ccccc1 C1(C(=O)NCC2CC(F)(CNC(C3(C(=O)NC)CCC3)=O)C2)Cc2cccnc2C1 c1(C(c2ccncc2)Cc2n(CC)nc(-c3ccccc3Cl)n2)cccc(Cl)c1 C#CCC(C)(C)CNC(=O)CCOCCNC(=O)C(C)(C)n1cnnn1 CS(=O)(=O)c1cc(C(N2CCCOC(CNC(C3(C)CCC(=O)C3)=O)C2)=O)cs1 C1(C(=O)NC2C3CN(C(C4(C#N)CC=CC4)=O)C2C3)CCCN(S(N)(=O)=O)C1 c1(C(=O)NC2C(NC(c3c(C)ocn3)=O)CCOC2)c(Cl)cccc1[N+](=O)[O-] C=CC1(C(=O)NCC2(CO)CC23CCC3)CCN(C(C2CCC(=O)N2)=O)C1 C1(NC(C=NOC)=O)CCN(C(c2csc(-c3ccco3)n2)=O)CC1O N1(CCCNC(C2C(CNC(C3CN(C(C)C)C3)=O)CC2)=O)CCOC1=O C(CC(O)CNC(c1cncn1C(C)C)=O)NC(C(C)OCC#C)=O C1(C(C)NC(C2C(OCC)C2C)=O)CCN(C(C2CN(S(C)(=O)=O)C2)=O)C1 C12CCCN(C1)C(=O)c1ncccc1NC2=O.C(C(F)(F)F)C(N)=O C1(C(=O)NCC(CN(C(C(C)(C2CC2)OC)=O)C)(C)C)CN(CP(C)(C)=O)C1 N1(C(C2C(C)C2)=O)CCC(C2CC2NC(c2ccc(CN(C)C)s2)=O)CC1 N12CCC3C(C3C1)C2=O.C(=O)(CCCC1CC1C)NC1C(CCOC)C1 C(=O)(C(C)(C)N=[N+]=[N-])N1C(C(=O)NCCCCCN(C)CC)CCCC1 c1(CC(=O)NCC2C=CCN2C(c2ccc(O)c(Cl)n2)=O)ccc2c(c1)COC2 c1(C(=O)NCC(CC)(C)NC(=O)Cc2ccn(C)c2)cnccc1C(F)F c1(C(N(C2CCC(NC(=O)Cn3cnc(=N)[nH]3)CC2)C)=O)ccc2cccnn12 N1(C(C)=O)CCOC(C(=O)N(Cc2ccc(C)cc2)Cc2ccc(C)o2)C1 C(=O)(C#CC1CC1)NCCOCCC(=O)NC(C1CCC1)C N1(C2CN(c3ccnc(NC(CCC)C(C)C)n3)C2)CCCC(C)(O)CC1 N1(C(C2(N(C)C)CCC2)=O)CC2C(C(=O)NC3CCC(O)CC3)C2C1 c1(OC)ccc(C(F)(F)C(=O)NC2CC(NC(C3(O)CC3)=O)C2)cc1 C1(C2CCCN(C(c3ccc(Br)s3)=O)C2)(NC(=O)Cc2ccno2)CC1 N1(C(C2(C)N(C)CC(OC)C2)=O)C2CCC1CN(C(=O)CN1CC(C)(C)C1)C2 C1(C)(CNC(CNC(=O)NC)=O)CCN(C(C2(C(C)C)CNC(=O)C2)=O)C1 c1(C(=O)NC(CC)(C)CNC(=O)CC(F)(F)C(C)C)cnc2c(ccn2C)c1 c1(C(=O)NCCN(CCOCCO)C(C2CC2F)=O)cc(F)ccc1C1CC1 N12C(=O)NC(C3=C1CC(C(=O)O)NC3=O)c1c(F)ccc(F)c12.CCCC C(=O)(C(CC)(CC)C(C)C)NC1C(CNC(Cc2n(CC)ncc2)=O)CC1 C1(C(=O)NC(CCC)C)(NC(=O)Cc2ccc(O)nc2)CCN(C)C1 c12ccc(cc1)NC2C.Cc1ccc(C(C)NCc2cc[nH]n2)o1 C1(NC(C2(C(=O)OC(C)(C)C)CCCC2)=O)CC(F)CN(C(=O)CC2CC2)C1 N1(C(c2c(OCCOC)cccc2)=O)CCC(NC(C2C=CCC2)=O)C(F)C1 c1(C(C(=O)N(CC(CC)NC(=O)CN2CC(C)(C)C2)CC)C)ccccc1 c1(OC)ccc(Br)c(S(=O)(=O)NC(c2cccc(C(C)(C)C)c2N)=O)c1 O(Nc1nc(-c2ccccc2)nc2scnc12)CC(=O)NCCOO C(=O)(C(CO)N(C)C1CC1)N(CC(=O)NC(CC1CC1)C1CC1)CC#C c1(N2CCC(NC(CC(=O)OCC)c3ccccc3)C2=O)ccc(F)c(Cl)c1 N1(C(Cn2nnc(C)n2)=O)CCCC(NC(C2CC2F)=O)CCC1 c1(C(=O)NCC(CC)(C)NC(=O)C(c2cn(C)nc2C)C)cc(C)nn1C(F)F c1(C(N(CC(C)(C)CNC(C2CCCN(C(N)=O)C2)=O)C)=O)cc2c(s1)CCC2 C1(N(C(c2c(OC)csc2)=O)C)CCCCN(C(=O)Cc2cscn2)C1 CC(C)(C(=O)N1CCC(C(C)(O)CNC(=O)CC2CCCO2)CC1)C(F)F c1(C(=O)NC(C(=O)OC)c2cscn2)ccc(CN)c(Cl)c1 CC1(C)CCOC1C(=O)NC(c1cccnc1)C(=O)NCC(Cl)Cl N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCC(NC(c2cccnc2)=O)C(O)C1 c1(C(=O)NCC2CN(c3ncnc(C)c3Br)C(C)C2)cn2c(n1)COCC2 C1(C(C)C(=O)NCC2(Cl)CCC2)CCCN(C(C2(Cl)CC2)=O)C1 C12(C(=O)NCC(C)C(=O)NC(C)(C)CCCF)CCC(CC1)CC2 C1(NC(c2nc(C)sc2)=O)CC2CC1CN(C(=O)CC1CCCCC1(C)C)C2 C1(NC(CC2CC(=C)C2)=O)CC(O)(CNC(C2CCS2(=O)=O)=O)C1 c1(NC(=O)Nc2cnn(CCCC)c2C(C)C)nc2ccc(C(F)(F)F)cc2s1 CCC(CC)(CC)C(=O)NCC(C)(C)CNC(C1CC(=O)NC(CC(C)C)C1)=O C#CCC(CC#C)C(=O)N1CC2(CCC(CNC(c3cc(CO)oc3C)=O)O2)C1 C1(NC(C2CC2F)=O)CCCC2CN(C(=O)C3=CCS(=O)(=O)C3)CC12 Cn1ncc(C(N2CCCCCC2c2ccco2)=O)c1S(C)(=O)=O N1(C(c2ccn(CC)c(=O)c2)=O)CCN(C(=O)C(N2CCSCC2)C)CCC1C c1(C(C)C(N2CC(O)(CN(C)C(C3CC3(F)F)=O)C2)=O)ccc(Cl)c(Cl)c1 C12(CNC(C(C)NC(N)=O)=O)CC1CN(C(=O)CCOC1CCOCC1)C2 Cc1ccc(CC(=O)NC(C)CC2CN(C(c3cc(=O)c(C)c[nH]3)=O)C2)cc1C CCN=c1[nH]c(C(=O)NC2CC3CC(NC(C4CCC45CCC5)=O)C2C3)cs1 C(=O)(C(C)C(C)C)NCC1C(NC(CSCC(C)C)=O)C1 [N-]=[N+]=NCCCCC(=O)N1CCC(C2CC2)C1C(=O)N1CC(O)CCO1 c1(C(N(CC(C)NC(C=CCOC)=O)C)=O)ccccc1-c1nnc(C)o1 N1(C(C(COC)Cl)=O)CCC2CC(C1)CN(C(c1ccc(F)c3[nH]ccc13)=O)C2 N1(CCC(=O)NCC2(F)CC(NC(C3(F)C(C)C3)=O)C2)CCC(O)CC1 c1(C(C)C)nc(NCCN2C(=O)c3ccccc3C2=O)cc(=NC(C)CS(C)=O)[nH]1 C1(CC)(NC(=O)CC2CCCC(=O)N2)CCN(C(c2cnn(C)c2OC)=O)CC1 c1(C(N2CCC(NC(C(CC=C)CC)=O)C2C2CC2)=O)cnc2c(c1)COCC2 N#Cc1ccc(CSCC(=O)NC2CCN(C(=O)CCC3CC3(Cl)Cl)C2)cc1 N1(C(C=NOC)=O)CCC(CC(C)NC(=O)CC2CCC3CC23)CC1 C(=O)(CC(F)(F)C(F)F)NCCCN(C(CC(CCC)O)=O)CC1CCCC1 N1(C(C2CC(C)(C)C2)=O)CCCC(F)(C(N2CC3CCC3(CO)C2)=O)C1 N1(C(C(N2CCC(C)C2)=O)=O)CCC(N(C(=O)Cc2cccs2)C)CC1 C1(C(=O)NC2(COC)CC2)(NC(=O)C(c2ccccc2)F)CCN(C)C1 c1(C(=O)NCC(CNC(c2c(C)nn(CCO)c2)=O)(C)O)cc(F)ccc1N C1(C(=O)NCC2N(C(CN(C)C(N)=O)=O)CCCCC2)CCc2nn[nH]c2C1 CCC(C)CC(C)C(=O)NCCNC(c1ccc2c(n1)NCC2)=O Cc1onc(-c2ccsc2)c1C(=O)NCC(O)CNC(=O)CCN1CCC1 C1(F)(CNC(C(c2cncc(F)c2)C)=O)CCC(CNC(C2(O)CC2)=O)C1 C1(c2cccc(OC)c2)CC(F)(F)CN1Cc1ccncc1C#N N1(C(COCCOCC#C)=O)CC(C(N2CC(C#C)(OC)C2)=O)CC(C)(C)C1 N1(CC(=O)N(CC#C)C)CCCCC1.C1CS1 C12(NC(=O)C(c3cc(F)cc(F)c3)(F)F)CC=CC(C1)OC2 S(=O)(=O)(c1ccc(C(N2CCCC(CO)CC2)=O)cc1)NCCSC C1(C(=O)NC2CC(NC(c3nn[nH]c3Cl)=O)C2)(OC)CC(C)C1 C(=O)(C1=NNC(=O)C1)NC(CC(=O)NCCC=CC=C)CC1CC1 c1(OC)cc(C(N2CCOCC2C(N2C3CCCC2COC3)=O)=O)cc(O)c1O Cn1ncc(CC(=O)NCC2CCN(C(c3sc(F)cc3Cl)=O)C2)c1C(F)F C(C(C)C(C)C(=O)N1CCC(C)(CNC(C23CCC(OC)(CC2)C3)=O)CC1)OC C1(CNC(C2CN(CC(F)(F)F)C2)=O)COCCN1C(C1CCOC1C1CC1)=O c1(C(CNC(COCC)=O)NC(=O)C(=O)NCC2CC2)ccccc1 c1(CCNC(C(=O)NC(C#C)CCC)=O)cccc(F)c1F c1(C(N2CC(NC(=O)CCOCC(F)(F)F)C2)=O)ccn(C2CCOCC2)n1 CCC(C)C(O)C(=O)NC12CC(C(N3CCC(NC(C)=O)CC3)=O)(C1)C2 c1(CCC)cccc(C(=O)NCC(C2CC2)N(C(=O)C(O)C2CCC2)C)c1 c1(C2(C(=O)NCCC(C)(C)NC(=O)CO)CC2)ccc(Cl)nc1 Cc1ccnc(C)c1C(=O)NC1CC(C(F)F)(NC(C2CCC(C)O2)=O)C1 C1(C(=O)NC(CCNC(CCCCCC)=O)(CC)CC)CCN2CCCC2C1 Cc1cc(C(=O)NCC(C)(C(C)C)NC(C2CCC(C)CC2)=O)cn1C C(=O)(C(C)O)N(CCCOCCNC(CN(CCOC)C)=O)CC1CCOC1 c1(C(N(CCN(C(C2CCCN(C)C2)=O)C)C)=O)ccc(N)cc1O C(c1ccccc1C)=CCNC(=NCC)NC1COC2CC1C2 N1(C(c2cn(CCNC(CC3(N(C)C)CCC3)=O)nn2)=O)CC2CCC2(C)C1 c1(C(=O)N(C2CC2)CC2CCCN2C(=O)Cc2ccco2)cncc(Br)c1 c1(C(=O)Nc2cn(CCC(=O)OC)nc2)cccc(C)c1[N+](=O)[O-] N1(C(c2c(C)ccc(O)c2)=O)CC2OCC(NC(c3cc(Cl)cnc3C)=O)C2C1 C1(CCC)(NC(C2CC(=O)N(CC)C2)=O)CCN(C(=O)CC(C)SC)CC1 C(=O)(C(C)(O)C(C)c1ccccc1)NCC(CC(C)C)NC(=O)CN(C)CCO C(C(C)=Cc1ccccc1)(C(=O)NC1CCCC1)N(CCC)Cc1ccccc1 c1(C(=O)NCCN(C(C2(C(=O)OCC)CC2)=O)C)c[nH]c2nc(F)ccc12 C1(C(=O)NCCN(C(C(C2CCOCC2)OC)=O)C(C)C)CCC(C)O1 C=CCC(C(=O)N1CCSC(CC)C1)NC(C1CC2(CCC2)C1)=O CN1CCc2cc(C(=O)NCC3CC4(CCC4)CN3C(C3C=CCC3)=O)ccc21 C1(C(C)(C)C)(C(=O)OCc2ccsc2C(=O)OC)CCCCO1 c1(C(N2C3CC(NC(=O)CC4NC(=O)NC4=O)C2CC3)=O)cccc2nncn12 c1(OC(C)C(=O)NC2CC(CO)N(C(=O)C(F)C3CCC3)C2)cccc(Cl)c1 c1(N2CCC(C)(NC(c3nc(C)oc3)=O)CC2)ccc(Cl)c(C#N)n1 c1(-c2c(C)cc(SC)nc2)cnc2n[nH]c(C(=O)NCC3CCSCC3)c2c1 Cc1cncc(C(N2CCC=CC2C(=O)Nc2cncnc2O)=O)c1 N1(C(c2scc(C)c2)=O)C2CCC1CC(NC(c1nncs1)=O)C2 C1(C(C)NC(=O)Cc2cnsc2)CCCN1C(c1csc(Br)c1)=O c1(OCC=C)ccc(C(N2CCC(CF)(NC(c3csc(O)n3)=O)C2)=O)cc1 C(CCN(C)C(c1ccc(-n2ccnc2)nc1)=O)(C(C)C)NC(C(CC)C)=O CC(Cc1ccccc1)C(=O)N1CCCC1CC(=O)OCC(N1CCOCC1)=O C=C(Cl)C(C)(C)C(=O)N1CC(C(C)NC(=O)C(CC)N(C)Cc2ccccc2)C1 c1(C(=O)NCC2C(NC(C3(C)CC3)=O)CCCC2)noc2c(F)cccc12 C1(NC(C(C)Oc2ccccc2F)=O)CN(C(C2(C(F)F)CCC2)=O)CC12CC2 c1(C(N=S(C(C)=O)(C)=O)=O)ccc(S(=O)C(F)(F)F)cc1 N1(C(C(N2CCCCC2)C)=O)CC=CC(C(=O)NC2CC(=O)N(C)C2)C1 Cn1ncc2nc(O)c(C(=O)NCC(CNC(c3cccc(O)c3)=O)CO)cc12 CCC(C)CCC(=O)NC1(COC)CCCN(C(C2CCN(OC)CC2)=O)C1 N1(C(C2(CCC=C)CN(C(c3ccc(C#N)cc3)=O)C2)=O)CC(C)CCCC1C C(=O)(C1OCCc2ccc(Br)cc21)Nc1c(Br)ccc(N(C)C)c1 c1(CNC(c2cnc(C3CC3)[nH]2)=O)nnc(O)n1C1CC1 CC1CC(C)(C(=O)NCCCCCn2cc(-c3cccnc3)nn2)CC(C)O1 c1(OC)cc(C(N2CCC(CO)(NC(C3(n4ccnn4)CC3)=O)C2)=O)ccn1 c1(C(N2CC(CCC)N(C(=O)COCC(=O)OC)CC2)=O)cccc2sncc12 CC1=C(C(=O)N2CC(c3nc(C)no3)C2)SCCO1.C12CCN(CC1C)C2=O Cc1ccsc1C(=O)NC(C(=O)N1CCC1Cc1ccnn1C)C1CCCO1 c1(C(N2C(CNC(CC3C(C)(C)C3)=O)CCCCC2)=O)cc2c(Cl)cncc2s1 C12(CNC(CCSCC(C)C)=O)CC(NC(=O)CC3=CCOCC3)(C1)C(C)(C)O2 c1(C(N2CCC(CNC(c3[nH]cc(CC)c3)=O)C2(C)C)=O)cc(C)c(C)cc1C N1(C(c2cc(CSC)c(C)s2)=O)CCCC(O)(CCNC(c2ccco2)=O)C1 c1(CNCC)cc(O)c2ccccc2c1.C1CCN(C(=O)C2CC2)CC1 N1(C(C2C3(CC(NC(COC)=O)C3)C2)=O)C2CCC1CC(C)C2 c1(C(N(CCOCCNC(c2nc(CCC)oc2)=O)C)=O)ccc2nonc2c1 C1(N(C(=O)C=CC(F)F)C)CCC2(CCN(C(=O)CSCC3CCOC3=O)CC2)C1 C1(NC(=O)CSc2cn(CCCOc3ccccc3)nn2)CS(=O)(=O)CC1O C1(C(=O)OCCCN(C(C)CCO)C)C2CC2CN1C(=O)Nc1ccccc1 C#CCN(OC)C(=O)CC1(CNC(c2cc(=O)cc[nH]2)=O)CC1 C1(O)(CNC(CN(C(=O)CCCn2ccnc2)C(C)C)=O)CCC(C)(C)C1 CC1(C)CCC(C(=O)NCC(CNC(=O)CNC(N2CCCC2)=O)CO)OC1 C1(C(=O)NCC2CCN(C(C(C=CCCC)O)=O)CC2)(OC)CCC(C)(C)C1 C(=O)(C#CC12CC3CC(CC(C3)C1)C2)NCc1n(CCC)ccn1 C#Cc1ccc(CNC(=O)CC2C3CN(C(=O)C(C)NC(=O)CC)CC23)cc1 C(=O)(C1=CNC2=NCCCC2=C1)N(c1cccc(C(CC)C)c1)CC(=O)O N1(C(CC2CC(CC)C2)=O)CC(=O)NCC1C(=O)NCCC(O)C1CC1 N1(C(C(C)C(F)F)=O)CCCC(O)(CNC(=O)Cc2c[nH]ccc2=O)C1 N1(Cc2ccc3c(c2)C(=O)OC3)CC=C(c2ccccn2)CC1 C1(CN(C(c2c(C)n[nH]c2)=O)C)CCN(C(=O)C(C)(O)Cc2ccccc2)CC1 C1(C(=O)OCc2ncc(C(=O)OC)c(O)n2)Cc2cc(C)c(C)cc2O1 C(=O)(CC(C)C(=O)NCC1OCCC1C(=O)NC1(C)CCSCC1)OC C(=O)(C1CCCc2scnc21)NC(CCN(C(c1ccc(C)o1)=O)C)C CC(CNC(=O)C=CC(=O)NC1CC1)CNC(C1(CC#N)COC1)=O CN=c1cc(C(=O)NC2CCC(C)N(C(=O)CC(F)(F)Cl)C2)cc[nH]1 CCC(C)C(O)CC(=O)N1CCCC(CCC(=O)NC(C2CCC2)C2CC2)C1 Cc1cnn(C)c1CC(=O)NCC1CC1[N+](=O)[O-] c1(C(=O)NCC(CNC(c2ccc(C)o2)=O)C)cc(F)c(C(F)(F)F)c(F)c1 C1(O)(C(N(CCN(C(C(CC)Cc2ccccc2)=O)C)C)=O)CCCCCC1 c1(C(=O)NC(c2ccc(OC)c(Br)c2)C(=O)OC)ccc(C)c(I)c1 C1(NC(c2c(O)ncc(CC)c2)=O)CC2CCC1CN(C(C1CC(OC)C1)=O)C2 C(C(F)C(=O)N(C1(O)CN(C(=O)COc2cc(C)on2)C1)C)N(CC)CC CC(C)(CCC(=O)NC1COCC1CNC(=O)CCc1cn[nH]c1)[N+](=O)[O-] C1(NC(c2cn(CC)nc2)=O)C2CCCN(CC3CC(C)(C)C3)C2C1(C)C C12(NC(=O)CN3CCCCC3)CC1CN(C(c1cccnc1C1CC1)=O)C2 C1(C)(C(=O)NC2CC(NC(C34CCC(OC)C3CC4)=O)C2)CCC2(CC1)CC2 C1(C2CCOCC2)(CNC(CCC#CC)=O)CCN(C(=O)CCC(CC)CC)C1 CCC(CC)C(F)C(=O)N1CCOCC(C(=O)NCc2cc(OC)ncn2)C1 Cc1cc(=O)ccn1CC(=O)NCC1CCC(NC(C2(C#N)CCSCC2)=O)C1 N1(C(c2cnc(C)c(N)c2)=O)C2CCC1CN(C(=O)CCCC(C)(F)F)C2 C1(C(F)(F)F)CCC(N=c2nc(N3CCCCCC3)c3c([nH]2)CCCC3)C1 C1(C(c2n(CCSC)nnn2)NCC=CCl)CCCC(F)(F)CC1 c1(C(=O)NCCC2CCCN2C(c2cnc[nH]2)=O)cc2ccncc2s1 Cc1cc(C)nc(SCC(=O)N(C2CCN(C(C3CCOC3C)=O)CC2)CC)n1 C1(NC(C2(C(=O)NC)CC2)=O)CC(NC(=O)C(C)(F)F)C12CCC2 N1(C(C(CCC)F)=O)CCCC12CCN(C(C13CC(CCC)(C1)C3)=O)C2 C1(C(C(=O)NCCCCNC(C2(N3CCCC3)CCC2)=O)OC)CCCOC1 c1(OCc2ncc(C(=O)NC3C(NC(=O)OCC)CCC3)s2)cccc(CC)c1 c1(SCc2n(CC)ncn2)cccnc1N1CCC(C(=O)OC)C1 N1(C(COC(C)=O)=O)CCC2CCN(C(c3cc(C)c(Cl)s3)=O)CC12 C12(NC(CN(CC)CC)=O)CC1CN(C(c1nocc1Cl)=O)C2 C(=O)(C1=NOC(C)(C)C1)N1CCC(C)C(N(C(=O)C=CI)C)C1 c1(COCC)cn(CCNC(C(=O)NCCN(C)C)c2cscn2)nn1 Cc1cc(Cl)c(C(N2CCN(C(c3nn[nH]c3Cl)=O)CC(O)C2)=O)cc1F C(=O)(CCCC(=O)N1CC(CNC(=O)CNC(=O)OC(C)(C)C)CC1(C)C)NC c1(C(=O)NCC2C(NC(C3(C)CCCCO3)=O)CC2)cccn2nccc12 c1(C(N(CCNC(c2cc(CCO)on2)=O)CC)=O)cc(Cl)c2n[nH]cc2c1 c1(C(=O)NC2CCN(C(C=Cc3cnc(C)s3)=O)CC2)cccc2scnc12 c1(N2CCC(F)(C(=O)NC)C2)nccc(=NCC2CCOC2)[nH]1 C12(C(=O)NCC(c3ccccc3)NC(c3cc(Br)co3)=O)CCCC1OCC2 C(C)(C)(CC(C)C)NC(C=CC(C)NC(=O)CC1CCCN1C(=O)OC(C)(C)C)=O N1(C(C2C(C)OC(=O)N2)=O)CC2(C1)CN(C(C13CCC(CC1)CO3)=O)C2 C(=O)(CCCCCN=[N+]=[N-])N1CCC(C)(NC(C2OCC(C)C2)=O)CC1 c1(C(=O)NCC2(O)CN(C(C(CCOC)C)=O)C2)ncc(OC2CC2)cc1F C(C1CN(C(=O)CC2(OC)CCC2)CC1C(=O)NC(C)(COC)CC)=CC N1(C(CC(C=C)C)=O)CCC(C(=O)NCC2(O)CCCC2(C)C)C1(C)C c1(OCC)cc(C(=O)N(CC(=O)N(C)CC2CC2C)CC2CC2)[nH]n1 c1(C(N2C3(CNC(CC=CC=C)=O)CC(C2)C3)=O)cc2cc(Cl)ncc2[nH]1 CC(c1ccccc1)=CC(N1CC(O)(C(C)NC(=O)CCc2ccon2)C1)=O S(=O)(=O)(c1ccc(N2CCCC(OCC(F)(F)F)C2)cc1Br)N(CC(C)SC)C N1(C(C=C)=O)CCN(C(=O)Cc2ccc(OC)nc2)CC1c1ccc(CC)cc1 c1(NCCCC(N)=O)cc(NC2COCCOC2)ncn1 C1(C(N2CCC(N(C(C34COCC(C3)OC4)=O)CC)C2)=O)CC2CCCC(C1)C2 CN1C(=O)CC(C(=O)NCc2cn(C3CN(C(c4cscn4)=O)C3)nn2)NC1=O C(=O)(C1=NNC(=O)C1)NC1CC(OCc2cn(C)nc2)C1(C)C C1(CC(=O)NC2CC(F)(CNC(CCCCCOC)=O)C2)CCC2(CCC2)CO1 c1(C(=O)NC2CN(c3cc(OC)ncn3)C2)ccc(Br)cc1C(F)(F)F N1(C(C(=O)NCc2ncc(C(C)NC(=O)OC(C)(C)C)s2)=O)CCCC(O)CC1 N1(C(COCC)=O)CCC(NC(=O)CCC(F)F)C(C(C)C)C1 N1(C(CC(CC(C)C)NC(CC(CC)C(F)F)=O)=O)CCc2ccc(F)cc21 C1(C(=O)NC2CC(NC(CC(=O)NCCNC(C)=O)=O)C2)CCC(C)(C)C1 c1(OC(C)C)ncccc1C(=O)NCC(C)N(C(=O)CC1C=NN(C)C1=O)C C12(CCNC(c3c(C)nc(COC)s3)=O)CCC(CC1)N(C(C1(C)CC1F)=O)C2 C1(F)(CNC(=O)Cc2csnn2)CCCN(C(c2c[nH]c(=O)cn2)=O)C1 N1(C(CC)=O)CCN(C(=O)C(N2CCOCC2)OC)CC12CC2 N1(C(c2c(C)csc2Cl)=O)CC(CNC(c2cccnc2)=O)CC(C)(C)C1 C(=O)(C(C)C(O)C(C)C)NC(C(C)OC)C(=O)N(C(C)C(N)=O)C c1(OCC(=O)NCC2CC(NC(C=C(C)C(F)F)=O)CC2O)c(Cl)cccc1Cl C12(CNC(c3ccc[nH]3)=O)CCC1CCN2C(c1cc(=O)cc[nH]1)=O C1(CNC(c2c(C(C)C)c[nH]n2)=O)CN(C(=O)C(C)n2cncn2)CCC1(F)F C(=O)(C1=CC2(CCN(C(C3CCC(C)O3)=O)C2)C1)N1C(C(CC)O)CCC1 C12CC3(CCN(CC3)CC1)CO2.C(=O)(C(F)(F)C(F)(F)F)NCCCC(C)(C)C Cc1c(C(=O)NC2COCC2NC(C2(C#N)CCCC2)=O)nnn1C c1(NC(C2CCCN(Cc3ccc(Cl)nc3)C2)=O)cccnc1OC(F)F c1(C(=O)NCC2CCCN(C(CC(C)(C)OC)=O)C2)ccnc(C)c1Cl c1(NC(C(N2C(COCC)CCC2)CSC(C)=O)=O)ccc(F)cc1 CCCC(C(=O)NCC1(C)CCN(C(c2n[nH]c(=N)s2)=O)CC1)S(N)(=O)=O c1(C(c2c(C(C(CC)C)NC3CC(F)(F)CN3O)cccc2)=O)cc(F)c(F)c(F)c1 Cc1ncc(C(N2CCC(O)(CNC(c3cc(C)[nH]c3C)=O)CC2)=O)c(C)n1 c1(C(N(C(Cc2cccc(C)c2)C)C)=O)cncc2cccnc12 C(=O)(C1=CCCOC1)N1C(CC(=O)NC(c2nc(C)sc2)C)CCCC1 CCCC(C#N)C(=O)N1CCN(C(=O)C=CBr)C(CC2CC2)C1 c1(CC)nnc2n1CCCC2C(=O)NC(C1CN(C(=O)C(C)CC(C)C)C1)C C(=O)(C(CC(F)F)N(C(=O)C=CCN1CCCC1)C)N.C1(NC(C)=O)(CO)CCC1 c1(CC)ccc(OC)cc1C(N1CCCC1CCCNC(=O)C(C)CC1CC1)=O C(=O)(C(O)CCc1cnc[nH]1)NCC(C(C)C)NC(=O)C(F)(F)c1nccs1 c1(OC)ccc(N2CCC(CC(N3CCSCC3c3cnn(C)c3)=O)C2)c(Br)c1 N1(CCC(=O)NC2C(SC)COC2)CCC(C)CC1.C12CCCC1n1cc(nn1)C2 C(CCC(=O)N(CC(C)(C)CNC(=O)C(C)Oc1ccccn1)C)OCCC c1(OCCOC)cncc(C(N2CCCC(NC(C3CCCN(C)C3)=O)C2)=O)c1 c1(C(N(C)CC2(O)CCCN(C(COCCOC)=O)C2)=O)cc(N)c(C)cc1C N1(C(C=CCN(C(c2c(CC)nns2)=O)C)=O)CCN2CC(C)CC2C1 C1(NC(C2CCN(CC)C2)=O)CN(C(=O)Cc2cncc(C)c2)CC2(CCC2)C1 C(=O)(C1=C(Cl)CCOC1)NC1(CCOC)CCN(C(c2n(CC)cnn2)=O)C1 c1(C(=O)NC2CC(C)N(C(=O)C(c3ccccc3)F)CC2)c(F)ccc(F)c1N N1(CC)CCN(CC(N2CC(CCNC(c3nccn3C)=O)C(C)C2)=O)CC1 N1(C(C(C)=CC)=O)CCN(C(=O)Cc2cc(C)cc(C)c2)CC1COC C1(CCC)(NC(=O)CC(F)(F)F)CCN(C(=O)C(O)C(C)SC)CC1 C1(CNC(C(C)C2CCC2)=O)CCN(C(=O)Cc2cc(F)cc(Cl)c2)CC1O c1(CN2C(C(=O)Nc3c(C(C)(C)O)cccc3)CC(O)C2)c(Cl)cnc(Cl)c1Cl C(=O)(C1CCc2c[nH]nc21)NC1C(NC(CCc2ccc(=N)[nH]c2)=O)CC1 c1(CC)cnccc1C(N1CCC(C(C)(C)C(=O)N2CC(C(N)=O)C2)C1)=O c1(C(=O)NCCC(C)N(C(C(CC)CO)=O)C)ccc(OC)cc1Cl c1(C2OCCN(C(=O)Nc3nnc(C(C)N)s3)C2)cccc(Cl)c1Cl c1(C(N2CCC(C)C2CNC(=O)CSC(F)F)=O)ccc2occc2c1 N1(C(c2ccn(CCN(C)C)n2)=O)CCN(C(=O)Cc2cnn(C)c2)C2CC12 c1(C(=O)NC2CC(CNC(=O)C(O)C3CCC3)C2)ccc(=O)n2c1CCCCC2 N1(C(c2c(NCC)cccn2)=O)CC2(CCCC2NC(=O)C(C)CC)C1 C1(N(C)C(c2cnn(C)c2)=O)CCN(C(=O)C(c2ccccc2)F)CC1 c1(CC(=O)NCC23CC2CN(C(=O)CC2CCCO2)C3)ccc2c(c1)CCCC2 N1(C(c2ncn(C(C)C)c2)=O)CC(CNC(=O)CN2C(C)CCC2C)C(O)C1 c1(OC)coc(C(=O)NC2CCCC(NC(c3cccc(F)c3)=O)C2)cc1=O c1(C(=O)NCCN2CCN(C(C(C(C)C)(C)C)=O)CC2)cc2cccc(Cl)c2[nH]1 N1(CC(=O)N(C(C2CN(C(CN(CC(C)C)C)=O)C2)=O)C2CC2)C(=O)CCC1=O CCCC(O)CC(=O)NCC(CCNC(c1ccc(C(C)(C)C)s1)=O)C1CCC1 C1(CC(=O)N(C(CN(C(CNC(CC)=O)=O)C)C)C)CCC(C)(C)CO1 c1(NC(C=C(CCC)CCC)=O)ccc(NC(C2CCCC2O)=O)cc1C c1(-c2nc3c(cc2)O3)ccc(C#N)cc1N.Cc1cc(F)ncc1-c1ccccc1 c1(N(C)C)ccc(C(N2CC(F)(CNC(C3CC3(C)C(F)F)=O)C2)=O)c(F)c1 CC(CC(C)(F)F)C(=O)NC.C1(C)(C(N2CC3(C2)C(=O)NC3)=O)CCCNC1=O N1(CCOC(C)C)CC2CN(C(c3cc(CSc4ccccc4)on3)=O)CC2C1 C1(OC)CCOCC1NC(=O)CC1CC(C)N(C(=O)OC(C)(C)C)C1.c1nn[nH]n1 C1(CCNC(c2scc(C)c2)=O)CCCN(C(=O)CCC2CCCN2C)CC1 c1(CCC(=O)NC2CCN(CCC3CCOC3)C2)ccc(O)nn1 c1(C(N(CC(C)NC(=O)COC2CC=CC2)CC)=O)ccc(Cl)c(Cl)c1 CCCC(CNC(C1CCOC(C)(C)C1)=O)C(=O)N(C(C)C(=O)OCC)C N1(C(C(C)OC2CCOC2)=O)CCN(C(c2cc(CO)on2)=O)CC1CC(F)F C(=O)(C1=CCCOCC1)N1C(C)C(NC(=O)CNC(c2ccccc2)=O)CCC1 N1(C(C(C)N(C(C2CC2Cl)=O)CC)=O)CCC(n2cccn2)C1 C1(C(=O)NC(CNC(CC2CN(C(C)=O)C2)=O)C2CC2)CC(C)(C)CN1C C(=O)(C(CC1CCCO1)C(F)(F)F)N1CC(NC(C(=O)NCC)=O)C(C)C1 c1(C(N2CCN(C(CC(COC)(C)O)=O)C3C2CC3)=O)ccc2c(c1)CCCO2 C1(c2n(C(CC)C)nnn2)(NCCOc2ccc(F)c(Cl)c2)CCCSCC1 CC(C)(C)CCC(=O)NC1CC1NC(C1(F)CN(C(=O)OC(C)(C)C)C1)=O N1(C(C(CC)C2CCOCC2)=O)CCN(C(c2ccc(C)n2C)=O)CC(C)(F)C1 Fc1cc(CNC2(c3nnnn3C3CCOC3)CCOC2)c(F)c(F)n1 N1(C(C(CC=C)NC(C)=O)=O)CCC2(C1)CN(C(=O)CC1COCCN1CC)C2 c1(C(=O)NCC2OCC(CNC(C=CCOC)=O)C2)[nH]c(C)c(S(N)(=O)=O)c1C C1(C(=O)NC2CCC(NC(C(C)CN3CCOCC3)=O)CC2)CCC(=O)N(C)C1 Cc1ncccc1CC(=O)N(C(c1ccccc1)CNC(c1nocc1Cl)=O)C N1(C(CCc2ccc(N(C)C)cc2)=O)CCOC(C)(CNC(C2CC2CF)=O)C1 c1(N(C(c2coc(C)n2)C(=O)NCSc2cnn(C)c2)CC)cccc(OC)c1 N1(C(c2c(C)nn[nH]2)=O)CCCC(C(C)NC(=O)CCc2ccon2)C1 c1(OC(C)C(N2CCC(OC(F)(F)F)C2)=O)ccccc1-c1ccccc1 c1(CC(=O)NCC(CNC(Cc2ncc(C)s2)=O)F)cc(F)cc([N+](=O)[O-])c1 C(=O)(CC(C)(O)C(F)(F)F)NC1CC(CNC(C(CC=C)OC)=O)C1 c1(OCC)ccccc1OCC(=O)NC1CC(NC(=O)C(F)C2CCOC2)C1 c1(OCC=C)cccnc1C(=O)NCC(C)NC(c1cnc(OCC)s1)=O C(=O)(C1CCCc2c[nH]nc21)N(CCCNC(C(CCC(C)C)O)=O)C c1(NCC2C(C)CN(C(c3csc(O)n3)=O)CC2)ccc([N+](=O)[O-])cc1C(F)F N1(C(C(C=CC)O)=O)CCN(C(c2cc(O)cnc2N)=O)C(C)C1 C(=O)(C1=Cc2ccccc2OC=C1)NCC(CN(C(Cc1c(C)ccs1)=O)C)O c1(CNC(C(=O)NC(C2CCCCC2O)C)=O)ccc(S(C)(=O)=O)cc1 N1(C(C=CCOC)=O)CCCC(C2CCN(C(=O)C(O)CSC)CC2)C1 C1(NC(C(C(CC)C)=O)=O)CC2CC1CN(C(c1ccc[nH]1)=O)C2 C1(C(=O)NC(Cn2ncc(C)c2)C)CC(=O)N(c2cccc(C(F)(F)F)c2)C1 CN1C(=O)CSC1=CC(=O)NC1CCN(C(C2OCC2(C)C)=O)CC(O)C1 C(CCCC(C)C)NC(c1c(C(C)NC(c2cc(OC)no2)=O)noc1)=O c1(CC)ccc(NC(=O)CN(C(=O)C(C)CNC(C)=O)C)cc1 C(C(CC(C)C)NC(=O)CSC(C)(C)C)NC(C(c1cccs1)SC)=O c1(CC(CC(=O)NCC(C)(C)C)NC(C2CC2C(N)=O)=O)ccc([N+](=O)[O-])cc1 c1(SCC(N2CCC(C)(CNC(C3CCC(=O)N3)=O)C2)=O)ncnc2[nH]cnc12 N1(C(c2nnnn2C2CC2)C)CC2CCCN(C(C3CCC(=O)N(C)C3)=O)C2C1 CCCCCC(=O)NCC(N1CCC(N(C)C(C2CC3(C2)CC3F)=O)CC1)=O c1(C(=O)NC2C3CCN(C(CC(C)C(C)(C)C)=O)C32)nc2ccccn2c1F C(=O)(N=c1cc[nH]c2cccnc12)c1cc(C(=O)OC)cc(S(=O)(=O)OC)c1 Cc1ccc(C)c2[nH]c(C(=O)NC3CN(C(C4CCCC4)=O)C(C)(C)C3)cc12 N(C(=NCCOCC(F)(F)F)NC1CCCCC1)CC1CCC(=O)NC1 Cc1cc(C(=O)NCC2OCCC2C(=O)NC2CC3C=CC2CC3)ncc1N C1(NC(c2c(C(C)C)onc2)=O)C2CCC1CN(C(=O)C1=CC3C=CC1C3)C2 c1(NC(C2CCCN(C(C3(C)CCCO3)=O)C2)=O)ccc(O)c(F)c1 C1(NC(CNC(=O)OC)=O)CC(F)(CNC(C2CCN(C3COC3)C2)=O)C1 N1(C(C2(OCC)CCCC2)=O)CCCC(C2CCN(C(=O)CC3CC=CC3)C2)C1 C1(CC(=O)NCCCC(=O)NC2CC2)CC2(CCOCC2)CO1.N12CC(C1)C2=O N1(C(Cc2cc(OC)ncc2)=O)CCC(NC(=O)CN2CCSCC2)C(O)C1 N1(C(C)=O)CCCC(C(N2CCC(O)(CNC(=O)CSC3CC3)C2)=O)C1 N1(C(c2cc3ccc(F)c(C)c3[nH]2)=O)CCCC2C1CCCN2C(=O)C(C)C C1(F)(CNC(CC)=O)CC(NC(c2ncoc2C(C)C)=O)C1 C(=O)(CCCC(c1nnnn1C)NC1CCCCC1c1cccc(C)c1)OCC C=C1CCN(C(=O)CCC2CCC2)C(C(=O)NCCOc2cccnc2)C1 C1(NC(C(CCOC)NC(=O)CN2CCC(F)CC2)=O)C=CC(C)(C)CC1 c1(CC)ccc(CNC(C2(C)CC(NC(=O)Cc3ccccc3C)C2)=O)cc1 C1(CNC(C2C(C)C2)=O)CCCN(C(=O)CC2(CO)CC2)C1 C1(C)(C(=O)NCCCCCNC(CC(CCC)(C)O)=O)CC(C(F)(F)F)=NO1 C(CNC(C1CNC(=O)C1)=O)(CC(F)(F)F)NC(CS(=O)(=O)NC(C)(C)C)=O C1(CNC(=O)CC23CCCC2C3)C2CN(C(c3ccccc3)=O)CC12 c1(CC(N2CCC(N(CCC)C(c3ccc(F)o3)=O)C2)=O)ccc(F)cn1 C1(NC(C2(C)CC(C)C2)=O)CC2CC(C1)N(C(c1cc(C(N)=O)cs1)=O)C2 N1(C(C(C(C)C)OCC)=O)CCC(C2CCN(C(=O)Cc3cn(C)nn3)CC2)C1 S(=O)(=O)(c1ccc(NC2C(O)C3CCCC23)cc1)NC(c1cccs1)C N1(C(c2n[nH]c(C)c2Cl)=O)CCN(C(C2CN(C)CC(C)O2)=O)CC(O)C1 CC(C)CCC(O)C(=O)N1C2CCC1C(C(=O)NCC1CC(C)(O)C1)C2 CN1CCC(N(C(c2ccnc(-c3cccc(OC(F)F)c3)c2)=O)C2CC2)CC1 c1(-n2c(C)nnc2SC2CCCN(C(C)C)C2C(F)(F)F)ccc(Br)c(F)c1 CC(CN(C)C)CCC(=O)NCC1(O)CCCN(C(=O)COCCN(C)C)C1 Cc1cc(OCC(=O)NC2CC(C)(NC(=O)Cc3cncnc3O)C2)cc(C)c1 C1(CN(C(CCNC(=O)NC)=O)C)(NC(c2cc(C(C)(F)F)on2)=O)CC(=O)C1 c1(N(C)C)c(F)ccc(C(=O)NC2C3CCC2CN(C(C2(N)CC2)=O)C3)c1F CCCCCCC(C)(CC)C(=O)N1CCC(C(C)NC(=O)CCCC(C)C)CC1 CCCC(O)CC(=O)N1CCN(C(c2csc(CO)n2)=O)CC1C(C)C C12(C(N3CCC(C(C)(C)NC(c4cc(O)ncn4)=O)C3)=O)CC3CC1C2C3O c1(CN=C(NC(COC)C)NC2CC2(C)C2(C)CC2)ccc(C#N)c(F)c1 C1(NC(C2CCC(C)C2)=O)CC2CCCC(C1)N2C(C1CC(C)C1)=O C1(n2cc(-c3c(C(=O)OC)nccc3)nn2)CCC(C)(C)N(C(=O)C(F)OC)C1 C1(N=[N+]=[N-])(C(=O)NCCCc2nc(C)[nH]n2)CCN(C(=O)C#CC2CC2)C1 N1(C(C2C(C(C)C)CCC2)=O)CC(CNC(=O)CC(C)(F)F)C2(CC2)C1 C[S+](C)CCC(O)C(=O)N1CCCC1C(C)(C)CNC(=O)CCF c1(N(CCOC)C)[nH]c(=NCCS(=O)CCOC)nc2c1ncn2C(C)C CCC(C)CC(=O)N1CCCCC1C(C)Nc1cc(C(C)(C)C)ncn1 N1(C(CC(C)(C)C#N)=O)CCC2(CC1)CN(C(c1ccoc1Cl)=O)C1COCC21 Cc1cc(C(=O)NCCC2CC(NC(C3CC34CC4)=O)C2)c2ncccc2c1 c1(C(=O)OC)c[nH]c(C)cc1=NCC(CNC(=O)CCc1cnn[nH]1)C(F)(F)F C(=O)(CC1OCCc2ccccc21)NCC(C)NC(C1(CC#C)CCOCC1)=O N1(C(CCSCC)=O)CCC2(CCCCC2NC(c2nc(C)c(C)s2)=O)C1 C1(NC(c2cc(Br)n[nH]2)=O)CC1C1CCN(C(=O)COc2ccon2)CC1 C(=O)(C(O)CC(F)(F)F)NCCN(C(c1cncnc1-c1ccccc1)=O)CC c1(C(N2CC3(CN(C(CC(C)C4CC4)=O)C3)C2)=O)ccnc2[nH]ncc12 C=CCC(C(=O)NCCCOCCN(C(=O)C(C)C=C)C)c1ccccc1 CC1(C)CC2C(CN1C(=O)Nc1c(I)cc(Cl)c(Br)c1Cl)C2(F)F Cc1cccc(C(CNC(c2cscn2)=O)NC(c2ccnn2C)=O)c1 N1(C(C2CC(NCc3cc(C)sc3C)C2)=O)C2CCCC1COC2 C1(N(C(=O)CSc2ccccc2)C)CCN(C(=O)CCOCC2CC2)C1 N#Cc1ccc(S(=O)(=O)N2CCCC2CO)cc1NC1CCC(=O)NC1 N1(C(C(CC2CC2)OC)=O)CCC(COC2CCCO2)CC1 C1(C(=O)NC2C(=O)NCC2)CN(Cc2cc(F)c(Br)c(F)c2)CC(F)(F)C1 N1(C(CCCCC#C)=O)CCN(C(c2ccc(N)c(Cl)n2)=O)C2CCCCC12 C(CCC(C)C(=O)NC1C2CC1N(C(c1ccc(Br)c(O)c1)=O)C2)OC C(=O)(CCCC(=O)N1CC(C)(NC(C2CCC(NC(N)=O)CC2)=O)C1)NC C=C(C)c1ccccc1NC(=O)CCC1(C)CN(C(=O)CCN(C)CC)C1 C(CC(F)F)(C(=O)N(C)CC1(C)CCC1)NC(c1c(C)nn[nH]1)=O c1(C(=O)NCCN(C)C(C2COC(=O)O2)=O)cc(=O)c2ccccc2o1 c1(N(C)C)nnc(-c2cccc(N(C)C)c2)n1Cc1cccc(C(F)F)c1 C1(C(C)NC(C(F)=C(C)C)=O)CCCN(C(c2ccc(C(C)C)o2)=O)C1 C1(NC(CC(=O)NCC#C)=O)(CNC(=O)Cc2cnc(C)[nH]2)CCOCC1 C(c1ccc(C)nc1)=CC(=O)NCCN(C(C1CCCCN1CC(F)F)=O)CC C1(NC(c2c(C)cncn2)=O)CCN(C(=O)Cc2csc(Cl)n2)CC1C N1(C(C(C)n2cccc2)=O)CC2(C1)CN(C(=O)CSCCN(C)C)CC2CO N1(C(C(CC)F)=O)CCN(C(c2c(C(F)(F)F)coc2C)=O)C(C)C1 c1(C(=O)NC2(C(=O)OC)C(F)(C(=O)OCC)C2)ccc2ncn(C)c2c1 CN1CCOCC1C(=O)NC1CCOCC1NC(C1CNC(=O)O1)=O C1(CNC(c2nnc(O)nc2O)=O)CC(F)(F)CN1C(=O)C(C1CCOCC1)F C1(NC(CS(CC)=O)=O)CCCC12CCN(C(C1CC(F)(F)C1)=O)CC2 c1(C(N(CC(C)N(C(=O)CC2CC2(Cl)Cl)C)C)=O)cc(Cl)ccn1 C1(CNC(C2CC2C2CC2)=O)CCC2(CN(C(=O)C(F)=C3CCCC3)C2)O1 c1(NC(CN(C(C)C)Cc2cc(C)no2)=O)coc(S(C)(=O)=O)c1 C(C(C)(C)CCNC(=O)CCCC1(NC(C2(C#N)CCOC2)=O)CCC1)OC c1(CC(=O)NC(C(CO)NC(c2nc(CC)oc2)=O)C)cc(Cl)n(C)n1 CC(C)C(CNC(C1(NC(c2ccc(F)c(F)c2)=O)CC1C)=O)C(C)C c1(C(=O)NCCC2CC(NC(C3CC4CC4C3)=O)C2)cccc(OC2CC2)c1 C1(C(C)C)CC(C(=O)NCC2(CCNC(=O)C=C3CCCCC3)CC2)CCO1 c1(C(=O)NCCN(C(=O)C(C)C(F)(F)F)CC(C)O)coc2c1C(=O)NCCC2 C(CC(=O)N1CCCC(CCF)C1)(C(F)F)NC(c1cn(C)nc1)=O C#CCC(CC(F)F)C(=O)N1CCC2CCC(C1)N2C(C1(CC)CCNC1=O)=O S(=O)(=O)(c1ncccc1Br)NC1CC(OC(C)(C)C)C12CCC2 N1(C(C(C)C(=O)NOCCCN(C)C)=O)CC=CC1CN(C)C C(=O)(CC(O)CC(C)(C)C)N1CCC(O)(CN(C(=O)CCCC#N)C)C1 O=C(C#CC1CCCO1)NCC1CCCN(C(=O)CC2CC2)C1 C1(NC(C2CC(C)C2)=O)C2CC3C1C3C2C(=O)N(C)C(c1cnn(C)c1)C C1(C(=O)NCc2ccc(CO)o2)(COC)CN(C(=O)CC2(O)CCOC2)C1 C1(NC(c2cnc(CC)o2)=O)CCC(NC(c2ccc(O)cc2)=O)CC1 c1(C(N2CC(F)(C(N)=O)C2)=O)ccc(CNC(c2cc(CO)ccn2)=O)cn1 c1(CC(C)CCC(N2CCOC(c3nnn(C)n3)C2)=O)ccc(O)cc1 c1(C(CO)NC(CN(CCOC)C(C2CCC2C)=O)=O)c(C)cccc1Br C1(CC(N2CC(CC)N(C(c3csc(C)c3C)=O)CC2)=O)NC(=O)CN(C)C1=O c1(C(N2CCN(C(C3(CC)CCC3)=O)CC2)=O)ccc2c(n1)CCC2 C1(C)(COC)CC(NC(c2cc(OC(F)F)n(C)n2)=O)CN1C(=O)C#CC(C)C N1(C(C2N(CCC)CCC2)=O)CCC(N(C)C(C2CC2CF)=O)CC1 C1(C)(C(C)C)CN(C(=O)C(C2CC2)N(C(=O)C(c2ccccc2)C)C)CCO1 c1(CCC(=O)NC(CCC)(C)C)cnc2n1CCOC2 c1(-c2cn(CCC)nc2)ccc(C(=O)NC(C)C)c2[nH]ccc12 S(=O)(=O)(c1cccc(C(=O)N(C2CCOC2)CCO)c1)NC(C(C)C)CO Cc1nc(N2CCC(Oc3cccnc3)C2)ccc1F N1(C(=O)CCCCC2CC2)CC2=C(C1)CN(C(c1nsc3ccccc13)=O)C2 Cc1cccc(CC(=O)NCC2C=CCN2C(=O)COCCCC(C)C)c1Cl C1(C(=O)NC2C3CCC2CC3)CC2CCC(C1)N2 N1(C(CCOCC)=O)CCCN(CCCCNC(=O)C(=Cc2cnc[nH]2)C)CC1 C1(NC(C2CC(=O)CN2C(=O)CNC=O)=O)CNC(=O)C12CC2 C1(NC(CSCCCC)=O)CN(C(C2CC(n3ccnc3)C2)=O)C2CCCCC12 CC1(C(=O)NCCNC(C23CC(C2)C(C(F)(F)F)O3)=O)CCC(F)(F)C1 CC1=CC(C)CN(C(C2CCN(C(=O)C(C)(C)N3CCCC3)C2)=O)C1 C1(CNC(C(COC)OC)=O)COCCN(C(=O)Cc2cc[nH]n2)C1 Cn1nc2c(c1C(=O)Nc1ncco1)CN(Cc1ccc(F)c(F)c1Cl)CC2 N1(C(COCCC=C)=O)CC2(CC(CC(=O)Nc3ccc(Cl)c(C)c3)C2)C1 C1(O)(CCNC(CC2(OC)CCC2)=O)CCCN(C(=O)CC(C)n2ccnc2)C1 CCCCC(=O)C(=O)NCCCCC(=O)NCc1cc(F)ccc1F C(=O)(CC(C)(C)N(C(=O)CCOCC1CCOC1)C)NCCCOCC C(=O)(CC(C)C(C)(C)C)N1CC2C(C(N(C3CCCC3)CC#C)=O)(C2)C1 c1(C(=O)NCC2(NC(C3C(C=C)CC3)=O)CC2)cc(Cl)c(O)c(Cl)c1 C(CCCC(=O)N(C(C)CCNC(=O)C(C)C#N)C)NC(C)=O c12cccc(c1)OC2=O.C(=O)(C(O)CC)N(CCC)CCOCC1CCCO1 Cc1c(Cl)ccc(C(=O)NCC2C(C)CCCN2C(c2ccnnc2O)=O)c1N c1(OC)ccc(CC(=O)NC2CCOC(CNC(c3csnn3)=O)C2)c(OC)c1 Cc1cc(=NC2CCC(OC(F)F)CC2)[nH]c(CN2C3CCC2CC(O)C3)n1 c1(C(=O)NC(C)CC(C)NC(c2ccc(O)c(O)c2)=O)ncn2ccccc12 Clc1nc2ccccc2cc1-c1nc(-c2ccon2)no1 N1(C(C2(C#N)CCCC2)=O)CC2COCC2(C(N2CC3CCC3C2)=O)C1 c1(C(=O)NC2CC(CNC(C(C)SCC)=O)CC2O)ccnc2[nH]c(C)nc12 c1(OC(C)C(=O)NC(C2CCCN2C(c2cocn2)=O)C)ccc(CSC)cc1 C(c1ccccc1)=CC(=O)NC1CC(F)(CNC(c2ccc(C(N)=O)[nH]2)=O)C1 N1(C(c2csc(N(C)C(C)=O)n2)C(=O)NCCOC)CCC(C)(C(C)C)CC1 C=CCC(CNC(c1nnsc1N)=O)C(=O)NCCC1CCCC12CC2 c1(C(=O)NCC(CCOC)NC(=O)C(O)CCSC)ccc(OC)c2ccsc12 C#Cc1cccc(CC(=O)NC(C)(C(=O)NCC(=O)NOC)C2CCC2)c1 c1(OCCNC(C(=O)N(CC(c2ccccc2)(C)C)C)=O)ccc(C#N)cc1 Cc1cccc(Cn2nc(CC3CC3)nc2-c2nnn(C)n2)n1 C(=O)(CS(=O)(=O)Cc1ccc(Cl)s1)NC1C(CNC(COCCC#C)=O)C1 c1(C(=O)NC2CCN(C(C(=O)NCC)=O)C2C(C)(C)C)ccc(C(C)=O)c(F)c1 CCCCC(C)CCC(=O)NCC(n1cc(CCC#N)nn1)C CCC(CN(C)C)CC(=O)NCC(C1CCCCN1C(C1CCCC1)=O)(C)C CC(C)CC(C)(C)CNC(C1CCC(NC(c2cc(C(N)=O)[nH]n2)=O)C1)=O CC(CC(=O)N(C1CS(=O)(=O)C1(C)C)C)C(C)(C)NC(=O)CN1CC2CC2C1 c1(N(C2CC3CCCC(C2)N3)C(C(C)O)=O)nc(Cl)c2c(ccn2C(=O)NC(C)(C)C)n1 C1(COC)CCCCN(C(=O)CC2(NC(c3cn4c(n3)CCC4)=O)CC2)C1 c1(C(=O)NC(CC(C)NC(C(C)SCCCC)=O)C)cnn(CCO)c1N C1(C(=O)NC2CCCN(c3cc(C)nc(C4CC4)n3)C2)CCCC2(C1)CC2(F)F CC(C)CCC(C(=O)NC1CC(N2CCCC2)C1)NC(C1CC2(CSC2)C1)=O CCCC(CNC(=O)C1=C(Cl)CCOC1)C(=O)NOCC1(C)CCC1 c1(C(=O)NC(CNC(CCc2c(C(=O)OC)nco2)=O)C)ncnc2cc[nH]c12 N1(C(Cn2c(=N)nc[nH]2)=O)CCC2CN(C(C3CCc4nc[nH]c4C3)=O)CC12 N1(C(C(C)N(C(C)=O)C)=O)CCN(C(=O)CCc2cnccn2)C2COCC12 c1(C(C)=O)ccc(OCC(=O)NCC2CC2CNC(c2cnc(O)n2C)=O)cc1 N#Cc1ccc(CN2CC(O)CC2C(=O)Nc2cccc(Cl)c2F)c(F)c1 C1(CC(N2CCC(NC(c3cn(C)c(Br)c3)=O)C2)=O)CCCC2CCCCC12 Cc1c(NCC2(CCO)CCC2)ncnc1N1CCOC(c2cccc(F)c2)C1 C(C)(C)(CCCCNC(C1CCN(C)CC1)=O)NC(C(N1CCN(C)CC1)C)=O c1(C(N2CC(CNC(c3c(COC)cc[nH]3)=O)(OC)C2)=O)ccc2nncn2c1 CCCCC(O)C(=O)N(CCCN(C)C)CCNC(=O)C(C)(C)CS(C)(=O)=O CCCCC(CNC(=O)C=C(C)c1ccsc1)NC(c1ccc(C2CC2)cn1)=O C1(NC(CN(C)CC2N(C(COCCC(C)C)=O)CCC2)=O)CCCC(C)C1C C1(C)(C(N2CCCC(N(C(C3CC(C)C3)=O)C)CC2)=O)CCCCC1(F)F C(C(C)(C)C(=O)NC(C)CN(C(c1nn(C)cc1Cl)=O)CC)OCC Cc1c(C(=O)NC2CN(C(c3cnsn3)=O)CC2F)nn2ccccc12 c1(C(N2CCC(C)(NC(C(CC)C)=O)CC2)=O)ccc2c(c1)OCC2 c1(OC)cccc(S(=O)(=O)N2CC3C(C2)N3C(c2ccc([N+](=O)[O-])[nH]2)=O)c1 Cc1cnc2c(C(=O)NC3CN(C(c4sc(F)cc4Cl)=O)CC34CC4)cnn2c1 CC(C)C(CO)C(=O)N1CCCCC1CCNC(=O)COc1ccccc1O N1(C(CCN2CC(=O)NCC2)=O)CC2CCC1C2NC(c1sc(F)cc1Cl)=O N1(C(C)C)CCCC(C(=O)NC23CC(C2)N(C(=O)CSCC#N)C3)C1 O=C(C1=C(F)CN(C(c2ccc(Cl)cc2)=O)CC1)NCCC1(O)CCC1 c1(N(CCC#N)C)nc2cccc(F)c2c(=NC2CN(c3cccnc3)C2)[nH]1 c1(C(=O)NCC2C3CN(C(CNS(CC)(=O)=O)=O)CC32)cnc2ncc(Cl)cn12 C12(CCCC1C)C(=O)N2.c1(OC)csc(C(=O)NCCOC2(C)CCC2)c1 N1(C(C=CCOC)=O)CC(C)CN(C(=O)Cn2nc(Cl)ccc2=O)CC1C C1(C(N2CCC(CC)(Nc3ncncc3C)CC2)=O)CCOC2(CCCC2)C1 C1(C(=O)NCC2(CC)CCOC2)CCCCC1NC(=O)C(O)CSC c1(NCc2c(OC)cccn2)ccc(S(=O)(=O)N2CCCCC2C)cc1Cl C(=O)(CC(C)C(C)(C)C)N1CCC(C(C(=O)NCc2cc(C)sc2C)(C)C)C1 c1(OC)ccc(CN(C(C)C(C)C)CC2CCS(=O)(=O)C2)c(F)c1Br N1(C(c2c(C)n(C)nn2)=O)CCC(CNC(C2CCN(S(C)(=O)=O)C2)=O)C12CC2 C(C)(C)(CC(F)C(=O)NCC(C)N(C)C)NC(C(CC)N(CC)CC)=O N(C1CCc2cc(CNC(=O)C(C)C#N)ccc21)C(c1nn(CC)c(O)c1)=O c1(CCC)cc(NC(COC)C(C)(C)C)n2nccc2n1 c1(NC(C2C(C(=O)OC)C2)=O)ccc2nnsc2c1.N12CCCCC1C2=O c1(C(=O)NC2(CNC(C#CC(C)(C)C)=O)CCCCCC2)ccnc2[nH]ncc12 C1(NC(c2c(CC=C)cccc2)=O)CN(C(=O)CCC(=O)N(C)C)CC2(CC2)C1 S(=O)(=O)(c1ccc(Cl)c(C(=O)O)c1)N1C(C(=O)Nc2c(I)ccc(C)c2)CCC1 c1(C(N2CC(C)(NC(C=CC(=O)OCCCC)=O)C2)=O)n[nH]c(C)c1[N+](=O)[O-] c1(CO)cc(O)nc2c1CN(CCC1CCSC1)CC2 C=C=CC(C)C(=O)N1CC(CC(F)C(=O)NC2CCN(C)CC2)C1 c1(CC(=O)NC(c2ccccc2)CNC(c2c(C)noc2)=O)ccc(F)c(F)c1 c1(OC)c(F)cc(C(=O)NC2CC3CC2CN(C(c2ccc(C)o2)=O)C3)cc1Cl c1(C(N2CC(CCNC(C3CN(C)C3)=O)OCC2)=O)cccc2cnsc12 C1(C(=O)OC)CN(N2CCC3(CC2)COC3)C2COCC12 C1(CCC#C)CCCN1.c12coc(c1)CNC2=O.c1(C=O)cc(OC)no1 c1(OC)cccc(C(N2CC3CC(C2)N3C(C2(OC)CCC2)=O)=O)c1NC(C)=O N#CC1(C(N2CCC2C2CCC2)C2CC2)CCCO1 C=CC(C)(O)CC(=O)N1CCC2C(NC(=O)CCN3CCCC3=O)CC12 C1(NC(c2cccc(OC)c2C)=O)COC2(CCN(C(=O)C(F)OC)C2)C1 c1(C(=O)NCC(C)NC(C(C(=C)C)(C)O)=O)c([N+](=O)[O-])ccc(C)c1C N1(C(Cc2c(C)ncs2)=O)CCN(C)CC1C(=O)NC1CC(CF)C1 C1(NC(c2cncc(F)c2Cl)=O)CCN(C(=O)Cn2ccc(O)nc2=O)CC1O C#CCCCC(C)C(=O)N1CC2(CNC(=O)C(F)C3CCC3)CC1CCO2 c1(C(N2CCC(OCCCNC(C3CCC3F)=O)CC2)=O)ccc(F)c(Cl)c1 C1(CNC(C2(N(C)C)CCCC2)=O)C2CCC1CN(C(c1cc(C#N)c[nH]1)=O)C2 C1(CCNC(=O)CCc2ccncn2)CCCN(C(c2ccc(C3CC3)o2)=O)C1 C1(CNC(C2CCC(C(C)C)CC2)=O)CN(C(=O)C=Cc2ccsc2)CC12CC2 Cc1cc(C(=O)NCc2cc(C(=O)NCCNS(N)(=O)=O)cs2)c(C)[nH]1 c1(C(N2CC(CCNC(C3CCC3)=O)(OC)C2)=O)coc2c(F)c(Cl)ccc12 CC1(C(=O)NCC(O)CC(=O)NC2(CC(N)=O)CC2)CC(F)(F)C1 CCC(O)C(F)(F)C(=O)NCC1(CCNC(=O)C(=O)N=S(C)(C)=O)CC1 Cc1nc(C)c(CCC(=O)N(C)CC2CCCN2C(=O)C(C)(C)CF)c(O)n1 CC1C(NC(=O)CN2CSCC2=O)CCCN1C(=O)C1=NOC(C(C)(C)C)C1 CCC(CNC(=O)C=CC(C)(C)SC)(CC)C(=O)N1CCOC(CF)C1 N1(C(C(=O)Nc2cc(C#C)c(C)cc2)=O)CC(C2CCC2)CCC1C Cc1ccc(C(=O)NC2CC(CCNC(=O)C(C)c3cccs3)C2)c(C)c1 C1(N(C(CCc2cncc(OC)c2)=O)C)CCCN(C(C2CC2C(F)F)=O)CC1 c1(C(=O)OC)cc2cccc(NC(N3CCCCC3CC3CCC3)=O)c2cn1 c1(C(N2CC3C(COC)(C3)C2)=O)cc(-c2ccc(-c3cccs3)s2)cc(F)c1 c1(OCC)cccc(C(=O)NC2CCCC(NC(=O)Cc3ccoc3)CC2)c1N CC#CCCCC(C)(c1nnnn1CC1CCOCC1)NCC1CSC1 C1(CNC(C(CCN(C)C)NC(=O)CSc2nc[nH]n2)=O)NC(=O)OC1(C)C C1(NC(C2(C)CC2Br)=O)CN(C(=O)CCNC(=O)CO)Cc2nccn2C1 C1(C(N(CC(=O)NC)C)=O)CN(C(C)CC(C)(C)O)CCC1O N1(C(C2N(C(=O)OC(C)(C)C)CC(F)(F)C2)=O)CC2CCC(C1CO)N2C(N)=O C1(NC(CCCOCCOCC)=O)CCN(C(=O)CCF)CC1CC c1(C(=O)NC2CCCC2NC(C2CC3(C2)CC3F)=O)noc2c1COCC2 N1(C(C2CCN(C(CN(C)C3CC3)=O)C(C)(C)C2)=O)CCC2(CC1)CC2C#N CN1C(=O)CCC1(C)CNC(=O)CC(C)(C)N(C(=O)C=C1CCCCC1)C N12CCC3(CC(C3)C1=O)C2.N1(CCOCC)CCC(O)C(CN(C)C)C1 n1(CC)nnc2cc(C(=O)NC3CC3NC(=O)C(=O)NCC)ccc12 c1(C(=O)NCCN(C(CCC2C(C)C2)=O)CC2CC2)cccc(C#CCO)c1 N1(C(CCc2cncc(C)c2)=O)CC2(COC(CNC(=O)Cn3cncn3)C2)C1 c1(NC(C2CCCN(C(C(C)=C3CC3)=O)CC2)=O)cc(C)cc(C#N)c1 CC(CC(=O)NCC=C1CCN(C(=O)CC(C)(C)C(F)F)CC1)C(F)(F)F c1(COC)ncc(C(=O)NCC2CCC(NC(C3(C#N)CC3(C)C)=O)C2)c(O)n1 C1(CC(=O)NCCCCNC(=O)C(F)CC2CC2)COCCO1 Cc1cc(C(N2CCCCCC2CNC(=O)CN(C2CCSC2)C)=O)c(C)n1C c1(C(=O)NC(CC)CNC(c2cnc(COC)s2)=O)c(C)ccnc1O Cc1cnc(C(=O)NC2CCCC2CNC(=O)Cc2ncoc2C)cn1 C1(NC(c2ncc(CC)nc2)=O)(CO)CCCN(C(=O)C(C)(O)CC)C1 c1(C(=O)NCC(CNC(c2cccc(O)c2F)=O)OC)cc(F)cc2ccoc12 C(c1nc2ccccc2o1)=CC(=O)NCC=CCNC(=O)CC1CCCC1O c1(C(=O)NC(C(=O)NCC(CC)CC)C(C)C)ccc(C)c(C#N)c1 N1(C(c2ccc(C)o2)=O)CC(CNC(c2ccc(CS(C)(=O)=O)nc2)=O)C(C)C1 c1(C(=O)NC2C(CNC(C(C)(F)F)=O)C2)ccccc1OC(F)F C1(F)(CNC(c2cnco2)=O)CCN(C(c2cocc2Br)=O)CC1 C=CCC(C)(C)CC(=O)N1CCCCC(NC(C2COC3CCCCC23)=O)C1 Cc1cc(C)c(C(=O)OC(C)C(=O)Nc2ccc(Br)cc2)s1 c1(N(C(C2CCC(NC(c3ncc(F)cc3F)=O)C2)=O)CCC)nc(Cl)c(Br)cc1O CC1CCCN(C(C2CC23CN(C(C2CC=CCC2)=O)C3)=O)CC1 C12(C(=O)Nc3cccc(NC(c4cc(CF)on4)=O)c3)CC1CCC2(F)F CC1CCc2onc(C(N3CC(NC(c4cccc(S(C)=O)c4)=O)C3)=O)c2C1 c1(CC)cc(C(N2CCC(COC)(NC(c3cc(O)ncn3)=O)C2)=O)ccc1C C1(C(=O)NCC(CC)(C)NC(=O)C#CC2CC2)CC(C2CCOCC2)=NO1 c1(C(=O)NC2C(NC(C3CN(C(N(C)C)=O)C3)=O)CC2)ccc(F)o1 CC(CCC(=O)NCCOCCNC(c1ccco1)=O)S(C)(=O)=O c1(CC)nccn1CC(=O)NC(C(=O)N(C)CC1CCCCO1)C1(O)CCC1 N1(C(=O)OCC)CCCC(Nc2cc(C(F)(F)F)ccc2Br)C(F)C1 Cc1cc(C(=O)NCC2(F)CC(CNC(=O)CC3CC(O)C3(C)C)C2)c(C)[nH]1 C1(CC(=O)NC(C2CCCN2C(=O)CSCC(N)=O)C)C(C)(C)C1(C)C N1(C(C(C2CCCOC2)OC)=O)CCC(N(C(=O)C(C)O)CCO)C1 c1(C(C(=O)NCCC(CNC(C2CCOC2=O)=O)OC)F)cccc(C)c1 C1(CC)C(NC(c2nn(C)cc2Cl)=O)CCCN1C(=O)CCC1CCOC1 Cc1cc(C(N2CC(O)CC2C(N2CC(CC3CC3)C2)=O)=O)c(C)cn1 Cc1c(C(=O)NCC2CC(C(=O)NC3CC4CC4C3)=NO2)cccc1O Cc1cc(-c2nc(C3CCCCC3)nn2-c2cnn(C)c2)[nH]c1C c1(CC(N2CCC(N(C)C(C3CC3C(F)(F)F)=O)C2)=O)cc(O)nnc1O c1(C2(C)COC2)ccc(C2CN(C(N3CC(C4CC4)C3)=O)C2)cc1 C12(C(N(CCC)CCNC(C3CCCS3)=O)=O)CCC(N=[N+]=[N-])C1C2 c1(C(=O)NCCC2CCC(NC(CNS(CC)(=O)=O)=O)C2)cc2occ(C)c2[nH]1 C(F)(C(=O)N(C(C(=O)NCCCC1CCC1)C1CC1)C)=CCC c1(C(=O)NCC2C(NC(CCCN(C)C)=O)C2)ccc2c(c1)SCCN2 c1(C(N(CCCNC(C2=CC(C)CC2)=O)C)=O)cnn2cccc(Cl)c12 C(C(=O)NC1(CCO)CCC1)(C(C)(C)C)CNC(CCNC(=O)OC)=O N(C1CN(C(C2(c3ncccc3F)CCC2)=O)CCc2ccccc21)C(=O)CO Cc1nnc2n1CCN(C(=O)C(N1CCNC(C(F)F)C1)=O)C2C CN1CCCC(C)(C(=O)N(CCNC(c2cc(Cl)ncc2N)=O)C2CC2)C1 C1(C(=O)NC2(CN(C(=O)CCc3nccs3)C)CC2)CCCC(O)C1 C1(C(=O)NCCN(C(C2CC(OC)C2)=O)C2CC2)CC(C)(C)CCO1 c1(C(N2CCC(NC(C3C(C=C)OCC3)=O)C(O)C2)=O)ccc2c(c1)CCOC2 N1(C(=O)CC2(O)CCC2)CCC2C(CCN2Cc2n[nH]c3ccc(Br)cc23)C1 N1(C(C)CO)CCN(C(=O)Nc2cc(C)no2)CC1.c1(CN)cccnc1Br c1(C(=O)NC2C(NC(c3c(C)cco3)=O)C2)c[nH]c2cccc(C)c12 Cc1cc(Cl)c(Cl)cc1C(N1CCCC(NC(=O)CSc2nncn2C)C1)=O N1(C(C(CC)N2CCCC2=O)=O)CCC(O)(CO)CC1 c1(C(N2CC(CCNC(C3(C)COC3)=O)C2)=O)cc2cccnc2cc1F C(=O)(C(C)CC(C)(C)C)NC(CN(C(COCCCCOCC#C)=O)C)C N1(C(c2[nH]cc(C)c2)=O)CCCCC2(CCN(C(c3ccnc(C)n3)=O)C2)C1 c1(C(=O)NC2CCCC(N(C(CC(=O)OCC)=O)C)C2)cc(OC)cc(F)c1 C=CC1CN(C(=O)CNS(C)(=O)=O)CC1NC(c1ccccc1COC)=O C(=O)(CC(C)C(F)(F)F)N1CC(OC)C(NC(=O)CN2CCC(CO)CC2)C1 c1(CCC(=O)NC(CCCCNC(CCN(C(C)=O)C)=O)C)cc(F)ccc1F C12(C(N(C(C)CCNC(=O)CN(C)S(N)(=O)=O)C)=O)CCC(O)(CC1)CC2 c1(CC)ccoc1C(=O)NC1CC(NC(=O)Cc2csc(CCC(F)(F)F)n2)C1 C1(C(N(CC=C)CCO)=O)CCC(C)CN1C(=O)C=Cc1ccccc1 C(C)(CO)(C(=O)NC(c1nc(=O)o[nH]1)C)NC(C1C(C)=CCS1)=O N(C(=NCCC(C)=O)N1CCC(Oc2cccnc2)C1)CC(CC(=O)OCC)C c1(CC)cc(F)c(C(=O)NCC2COCC2NC(c2[nH]cnc2C)=O)c(F)c1 c1(-c2c(C(=O)NCCCN(C(CCCC)=O)C(C)C)scc2)ccc(C)cc1 C1(CC=C)(NC(=O)C(C)CCCC)CCN(C(=O)CO)CC1 c1(NC(C(=O)OC)Cc2ccccc2)ncnc(NC)c1N C1(CC)CN(C(=O)C(C)(C)SC)CCN1C(=O)C(C)C=Cc1ccccc1 C1(CNC(C2N(C(=O)NC)CCC2)=O)C(C)CCCN1C(c1ocnc1C)=O c1(C(=O)NC2CCN(C(=O)C3=NOCC3)C2)n[nH]c2cc(Br)ccc12 c1(C(=O)NCC(CC)NC(c2cnnc(Cl)c2)=O)cc([N+](=O)[O-])cn1C C(=O)(C1CC(=O)Nc2ncccc21)N1CCC(C(C)NC(c2ccco2)=O)CC1 CCC(C)(C)C(O)C(=O)N(C1CCCN(C(c2cc(C(N)=O)ccc2F)=O)C1)C c1(NC(c2cncc(F)c2)C)ccn(CC(F)(F)F)c(=O)c1 CC1CC(C)CCN(C(=O)CCC2(NC(c3sccc3C#N)=O)CCCC2)C1 N1(C(CC2(OCC)CC2)=O)CCC(NC(C2(C)CCCS2)=O)C1c1ccccc1 C(=O)(C1=CN=C2N=CNN2C1)NC1C=CCN(C(c2n(CC)ccn2)=O)C1 c1(C(N2CC(CNC(c3ccc(N)c(Cl)c3)=O)C(O)C2)=O)ccc2cccnn12 c1(C(=O)NC(C(=O)NCC2(C(N)=O)CC2)c2ccco2)cccc2ccoc12 C12(NC(=O)Cc3cnsc3)CC1CN(C(=O)CCc1ccon1)C2 C1(NC(CCc2cc(C)[nH]n2)=O)CN(C(=O)CCC(C)(C)N(C)C)CC2(CC2)C1 CCC(CC(=O)NCC1(NC(=O)C(CC)c2cccnc2)CC(F)(F)C1)SC c1(C(N2CCC(OCCCNC(c3n(C)ncc3)=O)CC2)=O)cccc(=O)n1C C1(NC(C(CCC)N(C)C)=O)CS(=O)(=O)C12CCN(C(C1(CF)CC1)=O)CC2 C=CC1CCCCN1C(C1CCCC(C)C1)=O c1(SC)cc(Nc2sc(OCc3ccncc3)nc2C)ncn1 N1(C(CC=CCC)=O)CCC(C)(C)C(CNC(=O)C(CC)SCC)C1 C1(C2CC2)(NC(C2N(C(C)=O)CCC2)=O)CCN(C(=O)Cc2ncccc2C)C1 c1(C(C)=O)cc(N2CC3CC(NC(=O)CC(C)C4CC4)CC3C2)ccc1[N+](=O)[O-] C1(C(=O)NC2(C(=O)NC(CO)C3(C)CC3)CCN(C)C2)CCOCC1(C)C c1(C(=O)NC(CNC(C(CC)CO)=O)CC(C)C)cnc(C)nc1COC Cc1csc(C(F)(F)C(=O)NC2CC(C)(NC(=O)C(n3ccc(C)n3)C)C2)n1 Cc1cc(C(=O)NC(C2CCCN2C(c2n[nH]c(C)c2O)=O)C)oc1C C1(C(C)CNC(=O)C(C2CCC2)C2CC2)CCN(C(C2(CO)CCCO2)=O)CC1 C1(NC(c2c(C)[nH]c(=N)s2)=O)CN(C(C2OCCN(C)C2=O)=O)CC2CC12 C1(C(N(C2(CC(=O)N(CC#C)C(C)C)CC2)C)=O)CCCCCN1C C1(C(=O)NCCC(C)(CC)NC(c2c(CC)nco2)=O)OCCCC1(C)C C1(CNC(CC2(C)CC2(F)Cl)=O)CC2(CCN(c3ncnc4[nH]cnc34)C2)CO1 C1(CC)(NC(=O)CC(F)(F)CC)CCN(C(c2cn3c(n2)CCC3)=O)CC1 C(=O)(C1=CCCC1C)N(CC(=O)NC(c1ncc(C)cn1)C)CC(C)C CC(C(=O)NCC(O)CCNC(=O)Cc1cc(F)cc(Cl)c1)C(C)(F)F N1(C(C(C)OCCOC)=O)CCC(NC(=O)C(O)C(C)(C)C)C12CCCC2 C1(NC(c2ccc(Br)cc2)(C)CO)C2C=CC1CC2 CCCC(C(F)(F)F)NC(C1(F)CCN(C(C2SCC=C2C)=O)CC1)=O C1(C2CN(C(=O)C=C3CCN(S(C)(=O)=O)CC3)C2)(NC(CC(C)(C)C)=O)CC1 Cc1[nH]nc(C(F)(F)F)c1NC(=O)CN1CCN(C(C)C(=O)N(C)C)CC1 c1(C(=O)NCC(CC)(CC)NC(c2c[nH]c(C(N)=O)c2)=O)ccc(OC)c(C)c1 N1(C(c2cn(CC(=O)OC)nn2)=O)CCC(NC(C2CCCC2)=O)C(C)C1 c1(C(C)N(C)C)nnc(N2CCCC(c3ccnn3C)C2)n1Cc1ccccc1 C(=O)(CCCCC(C)C)NCC(CN(C(c1cc(C)c(C)o1)=O)C)C N1(C(C2(C(C)C)COC2)=O)CC2(C1)CN(C(=O)COc1ccc(F)cn1)C2 c1(CC)nn(C)c(CC(=O)NCC2(CNC(c3ccsc3Cl)=O)CC2)c1Cl c1(CC(N2C(CNC(c3n(CC)ncn3)=O)C(C)CC2)=O)cc(OC)ccc1O c1(C(=O)NC(CCCNC(c2cc(OC)cc(F)c2)=O)C)cc(O)cc(N)c1Cl CC(CN(C)C)CCC(=O)N1CC(C)(C)CC1CNC(C1CC12CCSCC2)=O C(C(C)C)(C(O)C(=O)N1CC2(C1)CN(C(=O)CCNC(C1CCC1)=O)C2)OC C1(C(N2CCC(C=C)CC2)=O)CC12CCN(C(=O)CSCCC)CC2 S(=O)(=O)(c1ccc(NC2C=CCCCC2)c(Cl)c1)NC(C(C)C)CO c1(OC)cccc(C(N2CCC(NC(c3c(C)ncn3C)=O)CC2C)=O)c1C N1(C(C)=O)CC(O)CC1C(N1CCN(C2CN(C(C3CC4CCC3C4)=O)C2)CC1)=O C1(CCC(=O)NCC2(OC)CN(C)C2)CCN(C(=O)C(C)C2CCCO2)CC1 CCC(C)(CN=C(NCc1ccc(CO)cc1)NC1CCS(=O)(=O)C1)OC c1(C(N2CCN(C(c3cccc[n+]3[O-])=O)CC2CF)=O)ccc(O)c(F)c1F Cc1ccc(Cl)c(C(=O)NCC(C2CC2)NC(c2ccc(OC(C)C)cc2)=O)c1 C=CC(C)(C)CC(=O)N1CCC(O)(CCNC(=O)C(C)(CC)OC)C1 Cc1ncc2n1CCN(C(=O)C(C1(O)CN(C(C3CC4CCCC4C3)=O)C1)F)C2 Cc1nn(C)cc1C(=O)NC1CC(CC(=O)NCC2CCC(CO)O2)C1 C1(CC(=O)NCC2(CC)CCCC2)CN(C(=O)CSC2CC2)CC1C CC1(C)OC2(C(=O)NC3CCC3NC(c3c[nH]c4nccc-4c3)=O)CCC1CC2 CCC(CC(=O)NC(C)CN(C(=O)C=Cc1ccsc1C(F)(F)F)C)C1CC1 c1(C(=O)NC2CCC(C(N(C(C)C)CCF)=O)C2)cncc(Cl)c1 N1(C(c2[nH]nc(OC)c2Cl)=O)CCC2CCN(C(=O)CSC)CC2C1 C(C)(C)(CCC(=O)N1CCC2(CC1)CC2)NCC(C1CCOCC1)C C1(NC(C2C(C)(C)C2C#N)=O)CCCC12CN(C(c1cnc3[nH]ccc3n1)=O)C2 c1(C(=O)NC(CC)(CC)CCNC(C2(SC)COC2)=O)cnn2ccncc12 C=CC1(CC)COCCN1C(=O)C(n1cnc(C#N)n1)CC c1(NC2CCC(SCC)C2)cc(C)c(S(=O)(=O)NC2CCCCC2)cn1 Nc1c(C(=O)NCC2CC3CCC2N(C(c2cnsc2)=O)C3)ccc(F)c1F Cc1cc(N)c(C(=O)NCC(C)NC(C2CCCN2C)=O)nc1C N1(C(C(N2CCC(C)OCC2)=O)=O)CC2(CCCCC2)CC1C O=C(CC1NC(=O)NC1=O)NNC(=O)c1cccnn1 c1(C(=O)NCC(CO)NC(Cc2c(C)ccs2)=O)ccc2c(c1)COCCN2 Cc1cnncc1C(N1CCCC(C(=O)Nc2cccc(C(=O)O)c2)C1)=O CN1CC(C)(C(=O)NC2CN(C(=O)C=CCF)CC2F)CCC1=O C(C)(C)(C(C)CC(=O)N1CC(C)(C)C12CCC2)NC(c1c(C)nc(O)cc1)=O CC1CC(NC(=O)C=CCO)CN1C(c1cnc(S)n1C)=O C1(C(=O)NCCN(C(CCCOC(C)C)=O)CC(C)O)CC2CCCCC12 c1(C(=O)NCCSCCO)cccc(-n2cc(-c3cncnc3)nn2)c1 C(CN=C(NCC(C)(C)CC(F)F)NCc1cccc(C(C)C)n1)OC c1(CC)cc(C(=O)NC(C2CC=CCC2)C(=O)NCC(C)C(C)C)ccn1 c1(C(N2CCCC(Cn3ccnn3)C2)C(=O)NCC)cc(OC)c(OC)cc1C N1(C(C(C)n2cccc2)=O)CCCC(C2CC2NC(=O)Cc2cnn(C)c2)C1 CCC(C)CC(C(=O)NCCCC(=O)OC)NC(=O)CC1CCOC1C c1(OC)cc(CC(=O)NC2CC(C(C)NC(=O)CC3CC(C)=NO3)C2)on1 C1(C(C)NC(c2ccc(Cl)cn2)=O)CC(NC(c2cn(C3CC3)cn2)=O)C1(C)C C1(C(CO)N(C(C)=O)CC)CCN(C(=O)OC(C)(C)C)CC1.c1ncc[nH]1 CCC(O)CC(=O)NCCCC(=O)NCCc1cccnc1F C1(NC(c2c(C)scn2)=O)CC2C1CCN2C(c1cnc(=N)[nH]c1)=O c1(CNC(C2CC(CNC(C(C=C)(C)O)=O)C2)=O)cnc(O)c(F)c1 CCS(=O)(=O)c1ccc(F)c(C(=O)NC23CC2CN(C(=O)C2=CCCC2)C3)c1 N1(C(CCCN(C(C2C(C)CCCC2)=O)C)=O)CCC2CCCC2CC1 C1(CNC(C(C)CCO)=O)CC(F)(F)CN1C(c1nccnc1N)=O CCC(C)(O)C(=O)N(CCc1cn(-c2ccnc(C(=O)O)c2)nn1)C1CC1 C12(C(=O)NCC(CNC(=O)CCNC(=O)C=CCl)OC)CC3CC(CC1C3)C2 C1(C(C)C)CC(CC(=O)N(C2CCN(C(=O)CC=C(Cl)Cl)CC2)CCO)CCO1 C(N=c1[nH]c2cccc(F)c2s1)C1N(C(C2(F)CCC2)=O)CCCC1 c1(C(=O)NC2CN(C(c3c(CC)nc[nH]3)=O)C(C)CC2)nc2ncccn2n1 c1(C(=O)OC)c(C(=O)NC(CNC(C2CN(C(C)C)C2)=O)CO)n[nH]c1C C1(NC(=O)COCCOCCO)CN(C(C2(C#N)CCCO2)=O)CC1F c1(C(=O)NC(C2CCN(C(C(C(C)C)NC(N)=O)=O)C2)C)ccc(F)cc1N c1(C(=O)NC(C)CCCNC(c2ccc(C(F)(F)F)o2)=O)n[nH]c2c1CCOC2 c1(SC(c2cc(C)c(C)s2)CC)cccnc1NC(c1cccnc1)=O c1(NC(c2cc(C(=O)OCC)c(OCC)cc2)=O)ccc(F)c(O)c1F C1(N(C(Cc2ccc(C)o2)=O)C)CN(C(C2CC(F)(F)C2(C)C)=O)CC12CC2 C1(c2cc(C)no2)(C(=O)NC(CNC(C2(OC)CC(C)C2)=O)CO)CCOCC1 Cc1ccccc1-n1ccc(C(=O)NC(CNC(c2cnn(C)n2)=O)C(C)C)n1 C#CCCC(O)C(=O)NCCCN1CCN(C(=O)C(C)S(N)(=O)=O)CC1 c1(OC)cnc(F)c(C(N2CC(OC)C(NC(C3CC(C)=NO3)=O)C2)=O)c1 C1(NC(C2(C)CC2(F)F)=O)CN(C(c2nonc2N)=O)CC1c1ccccc1 Cn1nc(C(=O)NC2(C)CCC(NC(=O)CCC(C)(C)F)C2)cc1C#N c1(C(=O)NCC2N(C(C3NC(=O)OCC3)=O)CC2)ccc(=O)n(CCF)n1 Cc1ccc(N)c(C(=O)NCCc2ccc(CNC(C3CC3(F)F)=O)cc2)c1F n1(CCC)nnnc1C(c1cncn1C1CC1)NC1CC2(CC2)C1 c1(C(C)C(=O)NCC(CNC(=O)CSC2(C)CCCC2)CO)ccc(F)cc1F c1(C(=O)NC2C(NC(C(C)(CO)NC(C)=O)=O)COCC2)n[nH]c2c1CCCCC2 c1(C(=O)NCC2CN(C(C3C(C)(CC)C3)=O)C2)cc(F)c[nH]1 c1(C(=O)NC(c2cn(-c3nonc3C(=O)O)nn2)C)ccnc2c1cnn2C c1(CC(=O)NC2C3CN(C(c4cnco4)=O)CC23)cn2cc(F)ccc2n1 c1(NC(C2(C)CN(C(C(n3ccc(C)n3)C)=O)C2)=O)cc(F)cc(Br)c1 C1(OC)CCC2(CCN(C(=O)C(C)(C)CN(C(=O)Cn3ccc(C)n3)C)C2)C1 n1(CC)nccc1C=CC(=O)NCCC1(O)CCN(C(C2CC2C(F)(F)F)=O)C1 C1(C(=O)O)CCN(C(C2CCN2C(=O)C2CC2)=O)C1.C(C)(C)(C)N(CC=C)CC=O CC1(C(N2CCC(CC(=O)Nc3cccc(C(F)(F)F)c3)C2)=O)CCCCC1 c1(C(N2CCOCC(NC(C(C)S(N)(=O)=O)=O)C2)=O)ccc2c(c1)CCO2 C(CCCNC(C1(SC)CC1)=O)(C(=O)Nc1ccsc1)N(CC=C)C N1(C(C(C(C)O)(F)F)=O)CCC2(CCC2)C(NC(=O)CCn2ccccc2=O)C1 N1(C(c2cc(C)oc2C)=O)CCC(CC(N)=O)(NC(=O)CCn2ccnn2)CC1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CCC(CNC(=O)CCc2nnc(C)o2)C(C)C1 c1(C(=O)NC(CN(C(C(C)O)=O)C)(CO)CO)cnc2n(c1=O)CCS2 N1(C(=O)OC(C)(C)C)CCC(C2CC2)CC1.C1(=O)C(Cc2cncs2)C(=O)O1 Cc1cccc(NC(C)C(=O)NCC2(CNC(=O)CC3CCCO3)CCC2)c1 C12(NC(c3ccc(C)nn3)=O)CCC(C(=O)NCC(C)(C)C3CC3)(CC1)C2 C=C(C)C(CC(=O)NCCCOCCNC(c1ccoc1)=O)OCC N1(C(CCC(C)OC)=O)CCCCC(NC(=O)C=Cc2cnn(C)c2)C1 c1(C(=O)NCC2CC(NC(c3ccc(C)c(O)c3)=O)C2)cc2sc(Cl)cc2s1 C1(C(=O)NOCC2CCOC2)CCCCN(C(C2CN3CCC2C3)=O)C1 C1(CNC(C(CC(C)C)C)=O)CC2COCC2N1C(=O)CSCCC(F)(F)F C(=O)(C(F)CC(C)(C)NC(C1CC2C=CC1C2)=O)N(C1CCN(C)CC1)C N1(C(C2(CC=C)CC=CC2)=O)CCCC2(CCC(NC(=O)CNC=O)C2)C1 N1(C(CCC)=O)CCN(CCNC(C2CCC(=O)N2C)=O)C2(CCC2)C1 C1(CNC(CCCSC)=O)(NC(=O)CCOCCOCCCO)CCCCC1C c1(CC)cccc(C(=O)N(C)CC2CCCN2C(=O)CC2CCOC2)c1 c1(C(=O)NCC2N(C(C(C=CCCC)O)=O)CCOC2)cc2cncn2c(O)n1 CCC1=NOC(C(=O)NC(C)CNC(=O)Cc2coc(-c3ccccc3)n2)C1 c1(C(=O)NCC(C(C)(C)C)NC(C(CC)OCC)=O)n[nH]c2c1COCC2 c1(C(N2CC3C(NC(C4C(C(N)=O)C4)=O)(C3)C2)=O)cc2ccc(Cl)cc2c(O)n1 CN1CCCCC(NC(c2ccn(CCNC(C3(C#N)CC(=O)C3)=O)c2)=O)C1=O Cc1cc(C(=O)NCCNC(C2CC23CC3)=O)cc(C)c1C C1(OC)CC(NCC(C)OC)C12CCNCC2 c1(-c2cccc(-n3c(C)cc(C)n3)c2)ccc(S(=O)(=O)CCO)cc1 C1(C(=O)NC2CN(C(c3cc(CCC)on3)=O)C2)CC(F)(F)C12CCC2 C1(C(=O)NCC(C)(C)NC(=O)CC2CCC(=O)NC2=O)CCCCC(F)(F)C1 C1(SCC(=O)NC(Cn2cc(-c3ncc(C)cn3)nn2)C)CC=C(C(C)C)CC1 N1(c2nc(C#C)c(C)cn2)CCC(CC(N)=O)C(C2CC2)C1 Cc1sc(C)c(C(=O)N(C)CCNC(C2CCC3CC3CC2)=O)c1Br CC(O)C(C)C(=O)N(CCCCNC(C1(c2ccccc2)CC(F)C1)=O)C Cc1ccc2cccc(NC(=O)C(F)(F)CC3CCNCC3)c2n1 C1(NC(CCCC2C(C)C2)=O)COC2(CCN(C(c3cc[nH]c3)=O)CC2)C1 N1(C(C2CC3CCC2C3)C(=O)N(C2CCCC2)CC2CCCO2)CCCCCCC1 n1(CC)c(C(N2CC(O)(CNC(=O)C(F)n3ccnc3)C2)=O)cc2ccccc12 N1(C(C)=O)CCC(CN(C(=O)Nc2cnn(C)c2)C(c2nc(C)no2)C)CC1 c1(Cc2cnn(CC(O)C(F)(F)F)c2)c(F)cccc1F.CC1(C)CC(=O)N1 N1(C(CN(C2CCC2)C)=O)CCN(C(=O)Cc2cncc(Br)c2)CC1C1CC1 c1(C(=O)NCC2CN(C(c3c(C)nn(C(C)C)c3)=O)C(C)C2)ccc(O)cc1F Cc1ncc(CCC(=O)NCC(O)CCNC(c2nocc2Cl)=O)o1 N1(C(C2(CCCC)CC2)=O)CC2CC(C1)CN(C(=O)C(O)CN1CCOCC1)C2 N1(C(CSC(C)C)=O)CC(CNC(C2(C)COCC2(F)F)=O)CC1(C)C C(CNC(=O)C(C)=C1CCC1)(C(C)C)NC(C1(COC)CCC1)=O C1(NC(C23CC(CN(C(C4CCC(F)C4)=O)C2)C3)=O)CC2COCC(C1)C2 CC(C(=O)N1CC(CC2CCOCC2)CO1)SC(C)C(N1CCCCC1)=O C1(COC)(NC(c2ccc(-c3cscn3)cc2)=O)CCN(C(=O)CS(C)(=O)=O)C1 C(=O)(C(CN(C)C)NC(C1C(C)C1C)=O)NCCC N1(C(CC2CCN(C)CC2)=O)CC2(CC2)CC1CNC(=O)C1=CCCSC1 C(=O)(CC(O)CC(C)(C)C)NC(CNC(c1ccc(OC)cc1Cl)=O)(C)C(C)C N1(C(c2scc(OC)c2)=O)CC(NC(=O)CCC2CCCCO2)C2CCCC12 c1(CNC(COCC=C)=O)cncc(C(N2CCCC2CC(C)O)=O)c1 S(=O)(=O)(CCN=c1cccc(S(=O)(=O)N2CC(CO)OC(C(F)(F)F)C2)[nH]1)NC O=C(CCN(C(=O)CCn1ccnn1)CCCO)NCC(O)CC1CCC1 Cc1ccc(S(=O)(=O)N(C)C)cc1NC(=O)Nc1cnc2c(c1)CNC2=O C1(NC(C2(CCN(C)C)CC2)=O)CCCCC1CNC(=O)C=CC1CCCCC1 c1(C(=O)NCC(O)CC(=O)Nc2cnc(F)nc2)cnc(O)c(F)c1 C1(C(N(CC(C)(C)NC(c2cnc(C)nc2)=O)C)=O)COc2ccccc2O1 C1(C(=O)OC)C2CN(C(=NCCCCC(F)(F)F)NCc3ncc(Cl)s3)CC12 C1(CNC(CC=CC=C)=O)CN(C(=O)C(C)Cn2cccn2)CC2(CCC2)O1 c1(C(=O)NC2(CO)CCCN(C(CCOC)=O)C2)cccc(P(C)(C)=O)c1 c1(C(N(C(C(=O)NCCC(C)SC)C)C2CC2)=O)cc(C2CC2)no1 C1(c2cn(CCCC(=O)NC3C(N=[N+]=[N-])CCC3)nn2)CCC2C(CC1)C2(F)F N1(C(C2(C#N)CC3(CC3)C2)=O)CCN(C(C2CC(F)(CO)C2)=O)CC12CC2 C1(N(C(CC(CC)C2CC2)=O)C)CCCN(C(=O)CCOCC2CC2)CC1 N1(C(C23CCC(CN)(CC2)C3)=O)CCC(CNC(C2CC2C(F)F)=O)C12CC2 CC(C)C(=O)NCCC(C)N(C(=O)CCC1CCCC1)C C#Cc1cccc(C(=O)NCCC23CCC(C2)N(C(=O)C(C)=CC)C3)c1C C(CC1=CCN(C(C2CC2COC)=O)CC1)NC(c1ncc(OCC)nc1)=O Cc1nnc2n1C(C(=O)NCCCCCn1cc(C3(C4CC4)CC3)nn1)CC2 C1(S(N)(=O)=O)(C(N2CC(NC(CCNC(COC)=O)=O)C(C)CC2)=O)CCCC1 N1(C(CCCNC(C)=O)=O)CCN(C(c2cc(C(F)F)ncn2)=O)C(C)C1 c1(CC)ncc(Cl)c(C(=O)NCCCCCN(C(=O)C(C)(CO)NC(C)=O)C)n1 C12(CNC(C3CCCCS3)=O)CC1CN(C(=O)Cc1ccc(C(F)(F)F)cc1)C2 N1(C(CN(CC#C)C(C2CCN(C)C2C)=O)=O)CC2(CC(=C)C2)C1 c1(OC)cc(Br)cc(C)c1NC(=O)C=C1CCN(C(c2cc(Cl)ccn2)=O)CC1 CCCCCCCC(=O)NCC(C(C)C)NC(=O)Cn1cnc([N+](=O)[O-])n1 N1(C(C2CC(C)(C(=O)OC)C2)=O)CC(CNC(C2(F)CCC2)=O)OC2(CCC2)C1 C1(NC(c2cncc(C(C)C)c2)=O)CCC12CCCN(C(=O)CNC=O)C2 c1(CC)cc(NC(=O)C(CC2CCC2)NC(C2CC23CC3)=O)ccc1F C1(CNC(C2CCCN(CC)C2)=O)CCN(C(=O)C#CC2CC2)CC1(F)F C(=O)(CS(C)(=O)=O)N1CC(CCNC(=O)C(O)CC2CCOCC2)(OC)C1 N1(C(C2(Cl)C(C)(C)C2)=O)CC(C2CN(C(c3cc(NC(N)=O)ccc3Cl)=O)C2)C1 c1(C(N2CCN(C(COCCC(C)C)=O)C(C)C2C)=O)cnn2c1CC(F)(F)C2 Cc1cccn2cc(C(N3CCN(C(C4CCC(=O)C4)=O)CC(CO)C3)=O)cc12 C#Cc1ccc(C(N2CC(C(C)NC(c3cnn(C(F)F)c3)=O)C2)=O)o1 c1(OC)cc(F)cc(C(=O)NCC2(OC)CN(C(=O)C(F)(F)C3CC3)C2)c1N CCC(C(=O)NCC(C)C(N1CC(CO)C2(CCC2)C1)=O)C(F)(F)F c1(C(N2CCC(CCNC(c3ccco3)=O)C2)=O)cc(O)nc(O)c1 N1(CC)CC(C(=O)NCC(COC)NC(c2cn(C)cn2)=O)CC1=O CC(CS(C)=O)C(=O)N(CCCNC(=O)CCCCN1CCOCC1)CCO Cc1cc(F)cnc1C(N1CCN(C(=O)CC2CCC(C)O2)CC1)=O CC(C)C(C#N)C(=O)NC1(CNC(c2ccn(C(C)C)n2)=O)CCCCC1 C1(C(N2CCN(C(CN3CCC(C)(C)C3)=O)CC2)=O)Cc2nccnc2C1 C1(CNC(c2coc(Br)n2)=O)CCCN1C(c1c[nH]c(-c2ccccc2)c1)=O CC1CN(C(=O)COC2CCN(C(C3CC3Cl)=O)C2)CCC1N(C)C N1(C(CCC(C)O)=O)CCCC(CO)(NC(=O)COc2cccc(Cl)c2)C1 C1(C(=O)NC2CCCC23CC3)(CC)CCCN1C(=O)CCn1ccnn1 C(Cc1ccoc1)(C(=O)NCC(F)C1CCC1)NC(C1C=CCC1)=O Cc1cnc(C(=O)NCC23CC(NC(C4CCCCC4O)=O)(CO2)C3)cc1Br N1(C(CSCCC(C)C)=O)CCC2CCC(C1)N2C(=O)CC1CCCOC1 c1(C(=O)NC2CC3(CN(C(CC(C)SC)=O)C3)C2)cc2ccc(C)cn2c1 C1(C(C)(C)CNC(=O)CC2CC2)CCN(C(=O)COc2ccc(F)cc2)CC1 C1(C(=O)NC(C(=O)NC)C2CC2)C2CCC(C2)C1NC(=O)CS(=O)(=O)N(C)C C1(CC(=O)NCCCCN(C(c2ncn(CC)c2)=O)C)CC(OC)C1(C)C C1(CC(=O)NCC2(OC)CCC2)CCN(C(=O)CCc2ccccc2)CC1 CC(=O)CCCCC(=O)N1CC2CCCC2(CNC(=O)C(C)c2ccsc2)C1 c1(C(=O)NCC2N(C(c3c(C)sc(Cl)n3)=O)CC2)cnc2ncnc(O)c2c1 c1(N2CCCC3(NC(=O)C4=CCCCO4)C(C2)C3)ncnc2cc(Br)sc12 C(=O)(C1=C(F)CN(C(=O)Cn2[nH]cnc2=N)CC1)N(C(C)CC(N)=O)C CCC(C)CC(CO)NC(c1cn(CCNC(c2[nH]nnc2C)=O)cn1)=O C1(CC(=O)NCC(CC)NC(=O)Cc2cc(C(F)(F)F)n[nH]2)CCCC1O C(=O)(C1=CCCOCC1)NCC(CC(C)C)NC(=O)Cc1ccc2occc2c1 Cn1cnc2nc(=NCC3CSCCO3)[nH]c(NCCN3CC4CC4C3)c12 N1(C(C(C(C=C)C)C)=O)CC2(CCCCN(C(c3cnn(CCOC)c3)=O)C2)C1 C1(CC(=O)NC2(C(C)(F)F)CCC2)CCN(C(C23CC2CNC3=O)=O)CC1 C=CC(C)(CCOC)C(=O)OCC.C12(C)CCN(C1)c1cccc(c1)Cn1cc2nn1 C12(NC(CCCC)=O)CCCCCC1N(C(c1cnn(C(F)F)c1)=O)CC2 C(=O)(C(N)CCC(=O)O)NCCN(CC#N)CCN C(CC(C)(C)CC(=O)NC(COC)C(=O)NC(C1CCC1)C1CCC1)OC C(C(CC(C)C)C(=O)N1CC2CCCC2(C(=O)NCCC(C)N(C)C)C1)OC c1(C(=O)NC2(CCNC(CN(C(C)=O)C)=O)CCCC2)cc(C)cc(F)c1N N1(C(c2c(CC)noc2C)=O)CCC2C(C1)CN2C(=O)C(C(C)(C)C)OC c1(C(=O)NC2(CF)CCN(C(c3c(N)nccc3)=O)C2)cc2cccnn2c1 N1(C(CCc2scc(C)n2)=O)CCCC(NC(C2(C(F)F)CCCC2)=O)C1C N1(C(Cc2nc(C)oc2)=O)CCCN(C(C2CC(N(C)C)C2)=O)C(CO)C1 C(=O)(CC(C)(C)F)N1CC(O)(CNC(C(C)OCC2CCCO2)=O)C1 O=C(CCC(CF)CF)NCC1CCCCN1C(=O)Cc1ccc(CO)cc1 c1(CC)ncccc1C(=O)NCC1(C)CCCN1C(=O)CCC1CCCOC1 C1(C(N2C(C)CN(C(=O)C3=C(Cl)CC3)CC2)=O)CCCC2CCCN12 CC1=CCC(C(N2CCC(N(C(=O)CN3CCCOC3=O)CCO)C2)=O)CC1 CC1CC(N)CCN1Cc1ccc(=O)n(C)c1 C1(NC(C2(COC)CCOCC2)=O)CC2CCC1N(C(=O)C1=CCCSC1)C2 c1(NC(C2CCN(C(c3c(C)ccs3)=O)CC2)C)ncnc2sc([N+](=O)[O-])cc12 C1(C(=O)NCC(C(C)C)O)CC(C)(C)CN1C(=O)CC(Cl)Cl c1(-c2scc(C(=O)NCC(=O)OC(C)(C)C)n2)cncc2nc[nH]c12 N1(C(CC(C(=C)C)OCC)=O)CCC2(CCC2)C(CNC(C2CSC2)=O)C1 c1(C(=O)N)cnn2cnnc2c1.Cc1nc(C2C(C(=O)NC3CN(C(C)=O)C3)C2(C)C)n[nH]1 CCCCC(C)C(=O)NC1CCC(CCNC(=O)CSc2ccccc2)C1 Cc1cc(OCC(=O)N(C2CN(C(=O)C(C)OCC3CC3)C2)C)c(C)c(C)c1 C(C)(CNC(c1cnc(S)[nH]1)=O)(C(C)C)NC(CC1(C=C)CC1)=O Cc1nc(C(=O)NCCCN(C(=O)C(C)C(O)C(C)C)CCO)c2ccccn12 CCC(C(=O)N(CC(O)CNC(=O)CCC1CCCCCC1)C)C(F)(F)F c1(C(=O)NCC(CC)NC(=O)C(CSC)c2ccccc2)cn(C)c(=O)nc1O CC(c1ccco1)=CC(=O)NC(C)C(C)(C)NC(c1cnn(CCO)c1C)=O C1(ONC(c2n(CC)ccc2)=O)CCC(O)C1O.N12CCCC(C1)C(C)(C)C2=O N1(C(CCc2[nH]cc(C)c(=O)c2C)=O)CCC2CN(C(=O)OC(C)(C)C)C2C1 C(C(=O)NCC1CN(C(=O)COCC2CC2)CC1(F)F)(c1ccccc1)=C(C)C C12(C(=O)NCC3C(NC(C(C(=O)OCC)F)=O)CCCC3)CCC(CO)(CC1)C2 N1(C(CCC#C)=O)CCN(C(c2ccnn2C2CC2(F)F)=O)CC1CC(=O)NC C12(SCC)CN(N(CC(C)C)CCNC(=O)OC(C)(C)C)CC1(C)C2 C1(C)(NC(CCC(CC)NC(c2ccccc2C)=O)=O)CCC(C)=C(C)C1 C(=O)(C1=CCCC1)N(CC(=O)NCCC=C=C)CCOC N1(C(c2ccc3nc[nH]c3c2Cl)=O)CC2(CC2)Oc2ccc(Br)cc21 c1(CC(=O)NCC(CNC(C(CO)N(C)C)=O)CO)ccc(Cl)cc1F C#CCC(C)(C)C(=O)N1CC(O)(CN(C(=O)Cn2nnc(=N)[nH]2)C)C1 C1(NC(c2ccc(C3CC3)o2)=O)CC2(C1)CC(NC(C1CCC(F)C1)=O)C2 C1(NC(CC(CC)SC)=O)CC12CCC(NC(=O)CSc1ccccc1O)CC2 CC(CC(C)N=c1[nH]c(=NCc2c(Br)nnn2C)[nH]c2cccc(F)c12)C(F)F c1(SCC(=O)NC2CC(NC(C3C(C)(C(F)F)C3)=O)C2)ccncc1 C1(C)(C(=O)NC(C)CN2CCCCC2)CCCN1C(=O)Cc1ccco1 C=CCCN=C(NCc1csc(C(F)(F)F)n1)N1CCC(OC)C(C)C1 Cc1ccnnc1C(=O)NCc1ccc(CNC(=O)CN2CCCC2C)cc1 N1(C(CCNC(N)=O)=O)CC2CC1CC2CNC(=O)C=Cc1ccncc1 N1(C(C(c2n(C)ncc2)O)=O)CC2CC(C1)CN(C(C13CCC(C)(C1)OC3)=O)C2 C=CCCCCCCCC(=O)NCC1CC1NC(c1cc2sc(Cl)cc2[nH]1)=O N1(C(C2(N(C)C)CCN(C(c3cc(C)c(C)nn3)=O)C2)=O)CCC(F)(F)C(F)C1 c1(CC)cnn2ccc(C(=O)NC3CCOCC3NC(C3CC(C)(F)C3)=O)nc12 C(=O)(C1CCCc2nccn21)NC(CCC)CNC(c1cncc(C(N)=O)c1)=O C1(C(C(N2CC(O)(CC=C)C2)=O)(C)C)CCCN(C(c2cn(C3CC3)cn2)=O)C1 c1(SCC(=O)N(C(C)CCNC(=O)CNC(N)=O)C)ccc(Br)cc1 C(=O)(C1=NOC(C(C)(C)C)C1)NC(CC)(C)CCNC(C1CCC1OCC)=O C1(C(=O)NCCC2CCC(NC(CCc3n(C)cnc3)=O)C2)CCC2CC2CC1 C1(OC)(CNC(C2CCC2F)=O)CCN(C(c2cccnc2N(C)C)=O)CC1 CC1CN(C(C2(O)CC2)=O)CC2(CCN(C(c3nnc(Cl)cc3N)=O)C2)O1 N1(C(CSCC#C)=O)CC(C)N(C(=O)CC(C)(C)C)CC1C C1(CNC(C2C(CNC(c3c(C(C)C)ocn3)=O)CCC2)=O)CCCCN(C)C1 n1(CC)nc(C(=O)NC(Cc2cn[nH]c2)C(=O)N(C2CN(C(C)C)C2)C)c(C)n1 c1(OC)ccc(I)c(C(=O)NCC2CC(NC(=O)CNC(C)=O)C2)c1 C1(C2N(C(C(C)N(C)C)=O)CCC2)CCN(C(c2ncn(C)n2)=O)CC1 c1(C(N(CCCCN(C(C(C)=C(C)C)=O)C)C)=O)cnc2[nH]nnc2c1 N1(C(C(Cc2cn[nH]c2)NC(C(C=C=C)C)=O)=O)CCOCC(C)C1 c1(N2CCC(C)(NC(c3ccc(F)nc3)=O)CC2)nc2ncc(Cl)cc2o1 C1(C(=O)NC2(CC=C)CCC2)CCCCC1(C)NC(c1cccn1CCC)=O C(N=c1[nH]c(NC2CC3CC3C2)nc2c1CCCCC2)c1n(CC)ncn1 C#CCCC(C(=O)NC(CN(C)C)CCO)NC(C1C=CCS1)=O c1(CC)cc(C(=O)N(CC)CC2CCCCN2C(=O)CC(C)SC)cc(O)n1 CCC(C)(CC(=O)NC1COCC1NC(c1ccoc1C(C)C)=O)C(=O)OC N1(C(c2c(C)cc(CC)o2)=O)CCN(C(C2Cc3nccn3C2)=O)C2CCCC12 CC(C)(C)C(CNC(c1cnns1)=O)NC(=O)COc1ccc(Cl)cc1 C1(N(C(C(CC)OCC)=O)C)CCC2CN(C(=O)C=C(C)c3ccco3)CC12 CC#CCCCC(=O)N(C)CC1CCN(C(=O)C2=NOC(C3(O)COC3)C2)C1 C(=O)(C(CO)C(C)C)NCC(C(C)C)NC(c1cc(C)c(C)s1)=O Cc1ccc2c(c1)SC(C(=O)NC1CCCN(C(C34CCC(CC3)O4)=O)C1)C2 C1(Cl)(C(=O)NC2(C=C)CNC2)C2CCC(=O)C12 c1(NC(C2C3CN(C(c4c(CC)cccc4)=O)CC32)=O)cccn2cc(C)nc12 C1(NC(COCC=C)=O)CCCCCC1NC(c1c(C)nsc1NC)=O C1(NC(CCSC)=O)CC2CCC1N(C(C1CCC(CO)CC1)=O)C2 C(=O)(CC(C)C(=O)N1CC(CC(=O)NCC2(CCCO)CC2)CC1(C)C)OCC C1(C(=O)NCC2(O)CN(C(c3cc(C)nc(C)c3)=O)C2)CCc2ccccc2O1 N1(C(C(c2ccc(Cl)cc2)CC)=O)CC2COCCC2(NC(=O)CS(C)(=O)=O)C1 c1(C(=O)NC2CCCC(NC(c3ncc(C)cc3F)=O)C2)[nH]nc2ncccc12 C1(NC(c2ccc(CCC)[nH]2)=O)CCN(C(=O)C(C)CF)CC1 N1(C(CNC(C)=O)=O)CC(N(C(=O)Cc2cccc(C(N)=O)c2)C)C(F)C1 CC(Cl)(Cl)C(=O)NCCC(O)CNC(=O)Cn1nnc(C(C)(C)C)n1 C1(NC(=O)C#CC2CC2)CCC2CCN(C(=O)CSc3nc[nH]n3)C1C2 c1(N2CCC3(C)C(C)(C2)C3(F)F)nccc(=NCCCCC#N)[nH]1 CCCCCCCCc1cn(CC2CCCN2C(=O)CCC2CC2(F)F)nn1 c1(C(=O)NC2C(NC(C(CC#C)O)=O)CC2)ccc(CCCC)c(N)c1 c1(-n2c(C3CC(OC)C3)nc(-c3ccccc3)n2)ccc2ncsc2c1 CC(C)CCC(C(=O)N1CC2(C=CCO2)C1)NC(=O)CSC(C)(C)C S(=O)(=O)(c1cc(Cl)cc2cccnc12)NCC(c1ccco1)O C=CC(C)C(C)C(=O)N1CCC(C(C)NC(=O)Cc2nc(C)c(C)[nH]2)CC1 C1(NS(C)(=O)=O)CCCC1CNC(=O)Nc1csc(C(N)=O)c1 Cc1cc(N)cnc1C(N1CC(NC(c2ccnc(C3CC3)n2)=O)C2(CC2)C1)=O C(=O)(C1=NOC(C)C1)NCCCCC(C)NC(CC(=C=C)C)=O C1(C(C)NC(C2(C)COC2)=O)CN(C(C2CC2(c2ccccc2)C)=O)CCO1 CC(C)S(=O)(=O)CC(=O)NCC1CCC(N(C(=O)C(Cl)=CCl)C)CC1 c1(CC)cnc(C)c(NC(=O)C(c2cccs2)NC(C2CNC(=O)N2)=O)c1 S(=O)(=O)(c1ccc(Cl)nc1C)N1CC(F)CC(C(=O)NC(C(=O)OCC)C)C1 c1(NC(C(=O)N(CC(=O)OC)C)=O)cccc(N2CC=CC2)c1 c1(C(=O)NC2CCCN(C(CN(C3CCSC3)C)=O)C2)cccc2cc(O)ncc12 CCCCCCC(F)C(=O)N1CCN(C(=O)C(CO)N(C)C)CC1CCCC C1(C)(CNC(N2C(C)(C3CCCCC3)CC2)=O)CC=CCC1 c1(CC2(OC3CC3)CC2)ccc(CCC(N2CC(C(=O)NC)(COC)C2)=O)cn1 C(=O)(C(F)(F)CC(C)C)N(C)CC1(O)CN(C(C(C)(C)NC(=O)NCCC)=O)C1 n1(CCOC)nc(-c2ccn(C)n2)nc1-c1cc(CO)oc1C N1(C(CC2CCCCC(=O)N2)=O)CCN(C(=O)C=C(Cl)Cl)C2CCCC12 c1(CC)cccc(C(=O)NC2CC(C)(NC(c3c[nH]c(=NC)s3)=O)C2)c1F C1(C)(Cc2c(C(N3CC(C)OCC3(C)C)=O)cccc2)COc2ccccc2O1 N1(C(C)=O)CC2CC1CN2C(=O)CCOCCNC(c1nnc(O)nc1O)=O.OCO N1(C(c2c(CCC)nns2)=O)CCCCC1CNC(c1cc(C(C)(C)C)c[nH]1)=O c1(COC(C)C(=O)NCCOCCC(=O)O)nc2ccccc2s1 C=CCCC(C)(C)C(=O)NCC1CCC(C(N2CC(C)(C)C2COC)=O)O1 C1(C(=O)NC2C(NC(=O)CCc3ncc(F)cn3)COC2)CN2CCCN1CC2 C1(NC(c2csc(CO)n2)=O)C2CN(C(=O)CCc3ncc(F)cn3)CC12 C1(NC(C(CC#C)(C)NC(=O)CN2CCCCC2C)=O)CC(C)N(C)CC1C c1(C(N(C2CCCN(C(c3ncccc3O)=O)C2)C)=O)ccc(C2(C)CC2)cc1 N1(C(=O)NCc2ccc(CSC)cc2)Cc2cccn2C(C)C1 c1(CO)cn(C2CN(C(C3(CNC(C(c4ccccc4)C)=O)CC3)=O)C2)nn1 CC1CCCN(C(c2cn[nH]c2)=O)C1CNC(=O)Cc1csc(Cl)n1 c1(NCC2CCC(CC)O2)[nH]c(=NCc2ccc(N)cc2C)nc2scnc12 C1(CC)CC2(CC(NCC3CCC(c4nc(-c5cccs5)n[nH]4)CC3)C2)C1 c1(NC(c2n(C)cc(NCc3cccc(OC)n3)n2)=O)ncc(I)nc1Cl c1(C(=O)NCC(CNC(=O)CCn2ccc(C)n2)OC)ccc(Cl)[nH]1 C1(CC(=O)N(C(C(=O)N(CC(COC)O)C)C)C2CC2)CCCCC1 O=C1CCc2cc(S(=O)(=O)N3CCCC4(CO)CCCC34)cc(F)c2N1 C1(N(C(Cc2c(C)n(C)cn2)=O)C)CCN(C(c2cnc(S)nc2)=O)CC1C Cc1cnc2c(C(N3CCCC34CN(C(=O)C(O)C(C)(C)C)C4)=O)cnn2c1 CCS(=O)CC(=O)N(C)CCC1CCN(C(C2CC(F)C2)=O)CC1 c1(-c2ccc(CC)c(F)c2)ccn2cc(C(=O)NCc3noc(CC)n3)nc2c1 c1(C(=O)NCCC(C(C)C)NC(c2cn(CC)nn2)=O)cccc2c1C(=O)NC2 C(=O)(CCCCN(C(=O)C(C)NC(=O)NC)C)N(CCO)CC c1(N(C)Cc2ccc(Cl)cc2)ncccc1S(=O)(=O)NCCOC1CC1 N1(CCOC)C(=O)NC(c2cc(Br)cc(OC)c2O)C2=C1CC(C)(C)CNC2=O N1(C(C(COC)OC)=O)C(CNC(=O)C=Cc2cn[nH]c2)CC2COCC12 c1(OCC(=O)NCC2C3CCC(C3)N2C(=O)CC2CCC2)ccc(F)cc1F C(CCNC(=O)Cc1cncs1)(C(=O)NC(c1nn[nH]n1)C1CC1)OC C1(C(=O)NC(C2CCN(C(=O)CCc3nccs3)C2)C)CCC(NC(N)=O)CC1 N1(C(c2c(C)nn[nH]2)=O)C(C(N2CCN(CCN(C)C)CC2)=O)CC2CC12 C(=O)(CCCN=c1[nH]c(=NC(CC#N)C2CC2)[nH]c2cc[nH]c12)N(CCOC)CC C1(O)(CCNC(CN(C(C)=O)C)=O)CCCN(C(=O)CCc2cnn(C)c2)C1 c1(C(=O)NCCN(C(C2CN3CCC2(C)C3)=O)CC)occ2c1CCC2 C(=O)(CC(C)(C)NC(C1CCCC1(C)NC(C12CC(C(=O)OC)(C1)C2)=O)=O)OC CC1(C)CCN(C(C2CCC2)=O)CC1CNC(c1cn2ccnc2s1)=O c1(C(N(CCC)CCNC(=O)Cc2cnn(C(C)(C)C)c2)=O)c(C)cnnc1O Cc1csc(=O)n1-c1ccc(NC(=O)C(=O)NC2CCCOC2C(C)(C)C)cc1 C1(CC(=O)NCCC(CCNC(c2cc(C)ncc2)=O)C)CCn2cncc2C1 N1(S(C)(=O)=O)CCN(C(C2(F)CCN(C(=O)Cc3ccco3)C2)=O)CC1 CCC(CNC(c1cn(C2CC2)cn1)=O)(CC)NC(c1nnn(C)n1)=O C(CCC(C)C(=O)N1CCN(C(c2ccc(C(C)=O)cc2)=O)CC1CO)OC c1(C(=O)NCC(N(C)C(c2ccc(F)cc2CO)=O)C2CC2)ccc(C#N)cc1 CN1CCC(NC(C2CC2c2cnn(C)c2)=O)c2ccccc21 N1(C(CS(=O)(=O)N(CC)CC)=O)CCC(NC(c2cc(Cl)ccc2C)=O)C(O)C1 N1(C(C(C)NC(c2c(C)ccnn2)=O)=O)CCc2ccccc2C1 CCC(CN(C)C)CC(=O)NC(CNC(=O)Cc1cccnc1F)CCOC N1(C(C2(COC)COC2)=O)CCOC(C(=O)NC(CN(C)C)CC(C)C)CC1 C1(NC(CC=CC=C)=O)CC2CCC(C1)N2C(=O)C(C(C)C)NS(C)(=O)=O CC1CCc2c(C(=O)N(C3CC3)CC3CN(C(C4C5CNCC45)=O)CCO3)n[nH]c21 C1(CNC(C(CCC)F)=O)N(C(c2nncs2)=O)CCCC1(C)C c1(CC(N2CC(CC(C)NC(c3cnc[nH]3)=O)C2)=O)ccc(O)cn1 N1(S(CCC)(=O)=O)CCc2cccc(C(=O)Nc3cccnc3Cl)c2C1 c1(C(N2CCCC(N(C(C3CC3C(C)(F)F)=O)CC)C2)=O)c(C)nn(C)c1C c1(C(=O)NC2CC(CCNC(c3nc(C)sc3C)=O)C2)nc(C)n(C)c1C c1(CC)cccc(C(N2CCC(NC(c3ccc(C)c(O)c3)=O)CC2C)=O)c1F C1(OC)CCC2(C(=O)NCCCC3(NC(c4cc(O)n(C)n4)=O)CC3)CC12 C1(CNC(C(CC)OCC)=O)CN(C)CCN1C(c1cccc(F)n1)=O N1(C2C(C)(C)C2c2ccccc2)CCC(O)(c2cccc(F)c2)C1 C#CC1(C(=O)NCC2(CC)CCCO2)CCN(C(=O)COCCSC)C1 C(=O)(C1(C)CCCc2ccccc21)N(C)CC1N(C(CC=CCC)=O)CCCC1 n1(CCC(=O)NC2(n3nnc(C(=O)O)n3)CC(OC)C2)cnccc1=O c1(COC)cc(C(=O)NC2CCC(CCNC(=O)CCC3CCCCC3)C2)no1 O=C(C(F)(F)CO)NCC1CCCN(C(=O)CCOC2CCOCC2)C1 C(CC(=O)NC)N(C(=O)C(C)N(C(=O)Cc1cccs1)C)CC CCC(CCOC)C(=O)N(C1CCCN(C(=O)C(CC(C)C)NC(N)=O)C1)C C1(CCC#C)CCN(C(C2(CNC(=O)C(O)CCSC)CCC2)=O)CC1 C1(Cc2nnc(N3CCOCC(C)(F)C3)n2CCC#N)CCCC2CCCCC12 C(C(C)(CC)CO)NC(CN(CCOC)C(c1nc(C)sc1C)=O)=O c1(C(=O)NCC2C(CNC(c3c(C)occ3)=O)C2)cc(=O)n(C)cc1Br c1(CN(C(c2cc(C)ccc2C(F)(F)F)C(=O)NC)C)nc2c(s1)CCCCC2 N1(C(=O)Cn2cnnn2)CCN(C(=O)CN2CC3CC3C2)C2CC12 c1(NCC2CN(C(CNC(CC(C)(C)C)=O)=O)C2)ncc(S(C)(=O)=O)cc1Cl Cc1n[nH]cc1C(=O)N(CCCNC(c1ccc(COc2cnn(C)c2)o1)=O)C N1(C(c2cc(C)c(C)[nH]2)=O)CC2CC(CNC(C3(F)CCCCC3)=O)CC1C2 c1(N(CC(C)NC(C2(C)CCCO2)=O)C)nc(C2CCC2)ncc1Br c1(NC2(C)CC(NC(C(CC)OC)=O)C2)ncc(S(C)(=O)=O)cc1Cl C(C(C)(CC)CO)NC(C(CSCC)NC(c1cnsc1)=O)=O N1(C(c2c(CNC(C34CCC(OC)C3C4)=O)ocn2)=O)CC2CC3CC2C1C3 C1(C(N(C)Cc2nnc(CC)o2)=O)CCC(O)CN1C(=O)CC1(O)CCOCC1 CC1=NOC(C(=O)NCCCN(C(=O)CN(C2CCSC2)C)CC2CCCC2)C1 C1(CNC(C(CCC)C#N)=O)CN(C(=O)C(F)=C(C)C)C2(CCC2)C1 c1(CC)ccc(CCC(N2C(CNC(C3(C)CCC(=O)N3)=O)CC3CC23)=O)cc1 C1(OC)CN(C(=O)Nc2ccc(Oc3cnn(C)c3Br)cc2)C(C)(C(=O)O)C1 c1(C(N(CC(CNC(c2cc(C)oc2C)=O)C)C)=O)cc(F)c(N)cc1F N1(C(COC)=O)CCCCCC(NC2CCCN(S(=O)(=O)c3cccnc3)C2)C1 c1(C(=O)NCCC2N(C(CC=CC=C)=O)CC(F)(F)C2)cccc2c1ccn2C C1(C(N2C(C3CCN(C(=O)C=CI)C3)CCC2)=O)CCN(CCO)C(=O)C1 N1(C(C(C=C)O)=O)CCC2(CCC(NC(=O)COc3ccc(F)nc3)CC2)C1 C1(NC(C(Br)=C(C)C)=O)CCCCC12CCCN(C(C1CCC1(C)C)=O)C2 C12(NC(C(C(C)C)SCC)=O)CCOC(CNC(c3n[nH]c(C4CC4)n3)=O)(C1)C2 c1(SC)nc(=NC2CC(C)N(C(C3CN4CCC3CC4)=O)C2)s[nH]1 C1(CCC)CN(C(=O)CC(C)(F)F)CCN1C(=O)C1=CCSC1 c1(CCC(=O)NC2(C)CN(C(CNC(S(CC)(=O)=O)=O)=O)C2)c(C)noc1Cl c1(C(=O)NCCN(C(C=Cc2c(C)coc2C)=O)C2CC2)ccc2snnc2c1 CCCCCC(=O)NC1CC(C)(C(=O)N(C)Cc2csnc2C)C1 C1(NC(c2cnn(C)n2)=O)CCC2CN(C(c3ccc(O)nc3)=O)CC2C1 C1(C(N2CC(C)(C)C(NC(C3CC(F)(CO)C3)=O)C2)=O)CCc2ncncc2C1 c1(C(=O)OCc2ccc(Cl)s2)ccc(F)c2cccnc12 C12(C(N3CCC(CCNC(C(C)CC4CCCC4)=O)CC3)=O)CCC(CC1)CO2 C(CC(=O)NCC(C)N=[N+]=[N-])(CC(C)C)NC(c1ccc(C=C)cc1)=O n1(C(CNC(C(C)C2CCCO2)=O)C)cc(C(C2CC2)N(C)C)nn1 C1(CC(=O)OC)(NC(=O)C(N2CCCC(c3nc(C)c(C)s3)C2)=O)CCOCC1 c1(C(=O)NCCCCNC(C2(CC(C)C)CCC2)=O)cn(C)nc1C(C)C N1(C(C(C(C)C)SCC)=O)CCCC12CCN(C(c1nccc(C)c1O)=O)C2 CON(CCC(=O)NCCNS(C)(=O)=O)C(=O)C(C)Cn1cccn1 c1(CN(C)C)ccc(-c2nc(-c3cccnc3)nn2-c2ccc(F)cc2)cc1 C=CCCC(C(=O)OC)NC(C1CC(C)(C)CN1C(=O)C(CC)SC)=O CC1CCN(C(=O)CNC(c2cscn2)=O)CCN1C(c1ccn(CCF)n1)=O Cc1c(F)ccc(C(=O)NCCCCC(C)NC(=O)COCc2nc[nH]n2)c1N CCCC(C(=O)NCCN(C(C1CCC1(F)F)=O)CC)c1ccccc1 CC(Cc1ccc(Cl)cc1)CC(=O)N(C)CC1(NC(=O)CN(C)C2CC2)CC1 C(=O)(C1=CCC(NC(c2cc(F)ccc2F)=O)C1)N1C(CN(C)C)CCC1 c1(C(=O)NCC2C(NC(c3cc(SC)c(C)o3)=O)CCCC2)cc(C)cc(C)n1 N1(C(C(=O)NCC(=C)C)CCCOCC)CCN(C)c2cc(C)ccc21 C(=O)(CCC(O)C(C)(C)C)N(C1CN(C(CCc2cccc(OC)c2F)=O)C1)C c1(CC)nc(=N)[nH]c(=NCC2CN(C(=O)C(C)Cc3cccc(Cl)c3)CC2C)[nH]1 C(C)(C)(C(=O)NC(C)C(=O)NCC(O)Cn1cccn1)OC(C)C Cn1cc2c(n1)CCCC2C(=O)NCCOCCCNC(=O)CCC1CCCO1 N1(C(c2ncc(C)o2)C)CCC(NC(=O)NCC2CCCO2)CC1 N1(C(C(=Cc2ccco2)C)=O)CCN(C(C2CC3CCC2C3)=O)CC1C(C)C CON(CCC(=O)NC1CCNC(=O)CC1)C(=O)c1c[nH]cc1C C1(CNC(N)=O)CCCCN1C(=O)NCC1CNC(=O)N1 N1(C(CC#N)=O)CCC(C(F)(F)F)C(CNC(c2ccc(Cl)c(F)c2)=O)C1 C1(CNC(CC=C=C)=O)CCN(C(c2cccc(Cl)c2OC)=O)C12CC2 c1(C(N(CC(CC)NC(c2cc(C)sn2)=O)C)=O)ccc(=O)n2c1COCC2 N1(C(C2(C(=O)OCC)CCCC2)=O)CCC2(CCCC2NC(=O)CN(C)C)C1 N1(c2cc(NCc3ccc(Cl)cn3)nc(C)n2)CCC(C2CC2(F)F)CC1 c1(NC(=O)C(=O)NC2CCCNCC2F)cccc(C(F)F)c1Cl C1(C(=O)NC2(c3cccc(F)c3)CNC2)CC2C=CCC(C1)C2 C=CC(CC)CC(=O)N1CCOC(CNC(=O)COc2ccc(OC)c(C)c2)C1 C12(NC(CC3CC(OC)C3)=O)CCC(CN(C(=O)C(C)=C3CC3)C1)C2 C1(CCC)CN(C(C2CN(C3CCOC3)C2)=O)CCN1C(=O)Cn1nnc(C)n1 c1(C(=O)NC2CC(O)(CNC(C3(C)CCCCO3)=O)C2)cccc(N)c1Br CC1CN(C(=O)C=Cc2cccs2)CCCN1C(C1CC2CCC2C1)=O C1(NC(C2CCn3ccnc3C2)=O)CCN(C(c2ccccn2)=O)C12CCCC2 Cc1nc(F)ccc1CN1CCC2(CC2C(=O)NC2CCC(=O)NC2=O)C1 N1(CC(=O)N(C)CC2CCN(C(C3(C4CC4)CC3)=O)C2)CC2CCC1C2 CCC(C(=O)NC(C)(C)CCNC(c1cc(C(C)C)no1)=O)C1CCC(=O)N1 C1(NC(=O)C(O)c2cnc[nH]2)COCC1n1cc(-c2cnn(CCF)c2)nn1 c1(C(=O)NC(CNC(C=CSC)=O)C)ccnc2ccccc12 C=CC(CC)CC(=O)NCC1(CNC(c2scnc2C)=O)CCC1 C1(NC(Cn2cc(C(=O)NC)nn2)=O)COCCN(c2nnc(CC(C)C)s2)C1 N1(C(C(CC=C)NC(=O)Cn2nnc(C)n2)=O)CCSC(C)CC1 Cc1cc(C(N2CCCCC2CN(C)Cc2noc(C)n2)=O)c(C)c(C)c1 CC1CN2CCN1C(C(N1CCC(NC(=O)CN3CCCCC3=O)C1)=O)C2 C1(NC(CCN(C(C)=O)C)=O)C(C)CN(C(C2Cc3cscc3C2)=O)CC1C CCCCC(CCC)N=c1[nH]c(=NCCC(=O)N(C)CC)[nH]c2c1CC(C)CC2 C1(C(N(C)Cc2cc(C)no2)=O)CCN(C(C2CCC2(F)F)=O)C(C)C1 c1(COC)cc(CNC(CCCO)c2cccnc2)on1 c1(C(=O)NC(C(C)NC(C(CC=C)C)=O)CO)nc(OC)cc(OC)n1 N1(C(CNC(CNC(c2ccc(C(C)C)o2)=O)=O)=O)CCCC1(C)CC1CC1 c1(OC)ccc(C(N2CC(NC(=O)C=Cc3cn[nH]c3)C(C)(C)C2)=O)c(N)c1F N1(C(c2ccc(C(C)=O)cc2)=O)CCCC(NC(c2ccncn2)=O)C(F)C1 C1(CC=C)(NC(c2coc3c2COC3)=O)CCN(C(=O)Cc2nc(C)cs2)CC1 C(C1CCc2ccccc21)NC(c1n(CCC)nnn1)c1cc(CC)on1 C1(N(C(=O)CC(=O)OC(C)(C)C)C)C2CN(C(=O)C(F)CC3CC3)CC12 C=C(Cl)CC(C(=O)NCC12CCCC1CCO2)NC(C1CCCC(=O)C1)=O N1(C(c2n(CC)ccc2)=O)CC2(CCCC2NC(c2cn[nH]c2)=O)C1 C(=O)(C(=O)NOC)NC(CNC(C1(C(CC)=O)CC1)=O)CC C(=O)(C1=COCCC1)N(C)CCC1CCN(C(=O)C(F)(F)c2cnccn2)CC1 c1(NC)cncc(C(N2CC(CNC(c3cc(SC)oc3C)=O)C(C)C2)=O)c1 CC(C)CCC(O)C(=O)NCC1(CNC(=O)C(C2(O)CCCC2)F)CCCCC1 CCCC(CC(C)C)C(=O)NCc1cccc(CNC(C2CNC(=O)N2)=O)c1 C1(NC(CC(C)OC)=O)COC2CN(C(c3ccc(Cl)cc3Cl)=O)CC12 CC1(C)CC(=O)NCC1C(=O)NC1C2CC1CN(C(=O)COc1ccccc1)C2 C1(O)(C(=O)NC(C2CN(C(C34CC(CO3)C4)=O)C2)C)CC2CCC1C2 c1(C)ccc(Cl)nc1C.c12c(Cl)n[nH]c1C(c1n(CC(=C)C)nnn1)NC2.CCC c1(CNC(CCC=C)C2CCCO2)cc(OC(C)C)cc(OC)c1 C1(NC(C=C(C)CNC(C2CC3(CC3)C2)=O)=O)C(CO)CCC12CCC2 C1(NC(C2(C)CC(NC(C3CC(N(C)C)C3)=O)C2)=O)CC2CC1OC(=O)N2 c1(SCc2onc(-c3cc(OC)c(C)c(OC)c3)n2)cc2ccc(Cl)nc2s1 C=CC(C)(O)C(=O)NCCC(C(C)C)NC(c1ccn(C(C)(C)C)n1)=O C(CC(=O)NC1CCCN(C(c2cnc3c[nH]nc3c2)=O)C1C)(C(F)(F)F)OC C(=O)(CCC1CC1)NCCN(CC(C)O)C(C1CCN1C1CCCC1)=O N1(C(c2nccc(C)n2)=O)CCC2(CC1)CC2CNC(C1CC(=C2CC2)C1)=O C1(CCN(C(=O)CC(C)(C)O)C)CCCCN1C(=O)CC1CCCOCC1 c1(OC(=O)NCCOC(=O)NC)ccccc1C C1(C(=O)NCC2CCCC(C)O2)CN(C(c2cc[nH]c(=N)n2)=O)CC1(F)F C1(NC(C2CCC2(F)F)=O)CCC(C(=O)NC2CCCOC2)CC1 c1(OC)ccc(C(=O)NC2CCN(C(c3cc(CO)on3)=O)C2C2CC2)cc1F C1(CNC(c2nc(C)nn2C)=O)CC2OCCC2N1C(c1ccc(C)c(F)c1)=O C1(C(N2CC(C(=O)NC)C2)=O)C(O)CCN1C(=O)Cc1csnc1C Cc1ncnc(O)c1CCC(=O)NC12CC1CN(C(=O)C1=CCOC1)C2 c1(C(=O)NC2CN(C(c3ncn(C(C)C)n3)=O)CC2C)cccc(F)c1C#N CN1CC2CCCC(C1)N2C(=O)C(C1(C)CC1)NC(=O)CCC(=O)N(C)C Cc1nc2ncccc2cc1C(N1CCC2(CC1)CC2NC(=O)CCF)=O c1(C(=O)NCC(CC=C)NC(c2cc(CO)[nH]n2)=O)cccc2nc(CO)[nH]c12 Cc1ccc(C(C)(F)F)cc1C(=O)NC(C)CCNC(=O)C(=O)C(C)C c1(C(=O)NCC2(F)CC(NC(C(C)O)=O)C2)ccc(S(C)(=O)=O)s1 c1(-c2scc(CC(N3CC(NC(C(C)(C)OCC)=O)C3)=O)n2)ccc(O)cc1 C#Cc1cc(Br)cc(F)c1C(=O)NCCCCOCC(F)(F)F C=CCC(CNC(=O)Cc1coc(C)n1)NC(=O)Cc1cc(OC)no1 N1(C(c2nc(CC)oc2C)=O)CC(NC(=O)Cc2c(C)cccc2C)CC(O)C1 Cn1cnc(C(=O)NC2(CNC(C3CC3c3ccccn3)=O)CCOC2)c1 CCCC(C(O)C(=O)NC(C)CN(CCCC)C)NC(c1nccn1C(C)C)=O c1(NC(=O)CC2CCN(C(c3cc(Br)ccn3)=O)C2)nccn2c(Br)cnc12 CC1CN(C(c2cn(CCO)nn2)=O)CCC1NC(C12CCOC(C)(C1)C2)=O Cc1cccc2nc(C(=O)NC3COCCC3NC(c3csc(CO)n3)=O)cn12 c1(CC(=O)NC2CCC(N(C)C(C3CCCC3)=O)C2)ccc2c(c1)CCCS2 S(=O)(=O)(c1ccc(Cl)c(Cl)c1)NC(C(C)C)=O CCC(C)CC(C(=O)N1CCC2OCCC2C1)NC(=O)CN(C(=O)COC)C CC1(C)C(C(=O)NCC2(C)CC2(F)F)CCN1C(c1ccc(=N)[nH]n1)=O Cc1csc(C(C)NC(c2sccc2CNC(c2snnc2C)=O)=O)n1 N1(C(C(C)(F)F)=O)CCN(C(C2CCC(F)(F)CC2)=O)C(c2ccccc2Cl)C1 c12ccc(cc1)C1CCCN1C2.c1(C2C(C(=O)OC)C2)ccc(C(=O)O)cc1 CS(=O)c1cccc(C(=O)NCC2CCCCN2C(=O)C2=CCCC2)c1 c1(C(=O)NCC(CC=C)NC(c2ccc(CC)[nH]2)=O)cccc2c1nc(O)n2C CCCC(C)CCCC(C)NC(c1ccn(CC)n1)C C1(CC=C)(NC(=O)CNc2nccs2)CCCN(C(C2CCN(C)C2)=O)C1 c1(CCC(=O)NC(CNC(C(F)OC)=O)C(C)C)ncc(F)cn1 Cc1oc(CO)cc1C(=O)NC12CC1CN(C(C1(C(F)(F)F)CCCCO1)=O)C2 C(N=c1cc(C)nc(Cl)[nH]1)C1CCC(NC(c2c(CC)nc[nH]2)=O)C1 N1(C(C2C(C=C(C)C)C2(C)C)=O)CC2(CC2)CC1CNC(=O)C(C)O CCC(CC)(CC)C(=O)N1CC2CCC(CNC(=O)CC3(C)CCOCC3)C2C1 CCC(C)CC(=O)N1CCN(C(CNC(c2cc(C)c(C)s2)=O)C(F)F)CC1 c1(C(=O)NCC2(C(=O)NC(CCSC)C)CCC2)ccn2ccnc2c1 N1(C(C2CC(OC)C2)=O)CC=C(CC(=O)NC2CC(C)OC(C)C2)CC1 C#CCCCCC(=O)NC(C)CNC(=O)CCc1cccc(N(C)C)c1 Cc1c[nH]c(CNC(C2CCC2C(F)F)=O)c(C)c1=O C(CCCCCC(=O)NC1CN(C(=O)COCC(F)(F)F)CC2CC12)SC CC1CC(CCC(=O)NCC2CCC2C(=O)NCC2(c3ncco3)CCC2)C1 C(=O)(CCC(C)(C)C#N)N1CCCC(C(C)NC(c2c(O)cccc2F)=O)C1 c1(CC(=O)NC(C(C)NC(=O)C=CC(=O)N(C)C)CO)cc(F)ccc1Br N1(C(CC=C=C)=O)CC(NC(c2ccc(O)cc2)=O)C2(CCOCC2)C1 C1(C(=O)NCCN2CC(C)(C)OCC2)CCC2CCCCC2C1 Cc1ccc(COC(C)C(=O)NC2CCCC2NC(=O)C(=O)NCCCF)cc1 C1(C(=O)NC(COCC)C)(NC(c2nc(O)sc2C)=O)CCN(C)C1 Cc1ncc(Cl)c(C(=O)NC2(C)CCN(CCOCCC(C)C)C2)n1 C1(C(N2CC(C)(CC)C2)=O)CCN(C(c2ncccc2N)=O)C(C)(C)C1 C(=O)(CS(=O)CCC(F)(F)F)NCCN(C(C(C(C)(C)C)(C)O)=O)C1CC1 C1(CCNC(C(c2ccoc2)NC(=O)CN2CC3CC3C2)=O)CC2C=CC1C2 C(=O)(C(F)C(F)(F)F)N(CC(CC)NC(c1cc(CCCCC)[nH]n1)=O)CC C(=O)(CC(C)CNC(=O)CC1CC(C)(C)CO1)NCCc1nc(CC)[nH]n1 O=S(=O)(c1ccc(F)cc1F)N1CC2CCC(C1)N(Cc1ccc(Cl)c(I)c1)C2 N1(C(c2cc(C)c(C)nc2)=O)CCC(C)(C)C(C(=O)NCCC(C)(C)C)C1 N1(C(C2(NC(=O)Cn3nccn3)CCN(C)C2)=O)CC2CCC1CC2 C(=O)(C(C(C)C)OCC(C)C)NCCCCCNC(C1(CCOC)CCCC1)=O C1(N(C(=O)C=CC(C)C)CC)CCN(C(=O)Cc2ccnn2C2CCC2)CC1 N1(C(C(C)n2cncn2)=O)CC2(CNC(C3(C(C)(F)F)CC3)=O)CC1CO2 C(=O)(CCC(C)(C)C)NCCOCCO.c1(OC)cccc(N2CCCC2=O)c1 C(=O)(C1CC(N)c2ccccc21)N1C(CN)CC(C(=O)OC)C1 CCC(F)(F)C(=O)NC(c1ccc(OC)cc1)CNC(c1coc(Br)c1)=O c1(C(=O)NC2C(NC(C(C3CCOCC3)OCC)=O)CC2)cc(N)cc(F)c1 c1(OC)ccccc1NC(C1CCCCC1SC(c1ccc(C2CC2)cc1)=O)=O c1(C(=O)NC(c2nc(C(=O)NCc3ccc(Cl)cc3)co2)C)cncc(O)c1 C(=O)(C(C)CC(=O)N1CCOCC1CN(C(=O)C=Cc1ccccc1)C)OC C#CC1C(C(=O)Nc2ccc(N3CCN(C(C)C)CC3)cc2)C1(C)C C1(COC)CN(C(=O)CSCC(F)(F)F)CCN1C(=O)CC1C(C)(C)C1(C)C CC(C)(CCNC(=O)CCc1cnc(Cl)s1)NC(c1ccc(C2CC2C)o1)=O C1(C(=O)NC(C2CCN(C(C3(C)CCC3)=O)CC2)(C)C)CC2(CCCC2)CO1 c1(-c2cccc(NC(c3c(C)cc(OC)nc3)=O)c2)nnc2n1CCN(C)C2=O CCC(C)C(O)C(=O)NCCC1(O)CC(NC(=O)CCCc2csc(C)n2)C1 CCCCCCCCC(=O)N1CCC(NC(=O)CN2CCCC(CC)C2)C(O)C1 Cc1nn(C(C)C)c(NC2CC(C)N(C(=O)Cn3nnnc3C)C2)c1[N+](=O)[O-] c1(C(N(C)CC2CCN(C(c3ccc(CCC)[nH]3)=O)C2)=O)cc(C)n(C(F)F)n1 n1(CC)nc2c(c1C(=O)NC(C)C(C)NC(=O)CCC1CCCC1)CCCC2 Cc1cc(=O)ccn1CC(N1CCC(NC(c2snnc2C(C)C)=O)CC1C)=O CC1(C)CN(C(=O)Cn2ccc([N+](=O)[O-])n2)CC1NC(C1CC12CCSCC2)=O C1(C)(C(=O)NCC2(OC)CN(C(C3(C)CC3Br)=O)C2)CCC(C)(C)CC1 c1(CC)cc(N(C)CC2CCCN(C(=O)Cc3ccc(SC)cc3)C2)nc(C)n1 c1(C(=O)NCC2COCCN(C(c3c(C)coc3C)=O)C2)cc2ccccc2[nH]1 N1(C(C(C)CCN(C)C)=O)CCC(NC(c2nccnc2Cl)=O)C(C)(C)C1 C1(C(=O)NCCC(C(C)C)NC(c2ccc(C#N)cc2)=O)CCc2nncn2C1 N1(C(C2(C)CC(C)C2)=O)CCCCC1CCNC(c1cccnc1CO)=O CC(CC(F)(F)F)C(=O)NC1CC2CC(NC(C3CC(=O)CC(=O)C3)=O)C1C2 Cc1ccc(C(=O)NCC2CN(C(=O)CCCc3ccccc3C)C3CC23)cn1 c1(C(N(CCCNC(C2CC=CCC2)=O)CC)=O)cccc(C)c1I C1(C(=O)NC2C(NC(c3ccc(CC)s3)=O)CC2)Cc2ccccc2C1 C1(CNC(Cc2nnc(C)o2)=O)CC2CCC(C1)N2C(=O)Cc1ccnc(F)c1 c1(C(N(CCCN(C(C(=O)NCC)=O)C)C)=O)cc(-c2ccc(C)s2)[nH]n1 C(=O)(C(O)CC(C)(C)C)N1CCC(OC2CN(C(C(C(=C)C)(C)O)=O)C2)CC1 C1(CC)CN(C(c2cc(C)nn2-c2ccccc2)=O)CCN1C(=O)CNC(C)=O CCCCC(CC(=O)N1CCCC1(C)C1CC1)NC(c1nocc1C)=O C=CC1CC(NC(=O)CCC2CCCN2C(=O)CCC#CC)CCO1 C1(C(C)C)CN(C(=O)C=CCC(C)(C)NC(=O)CC(C)O)CC1C c1(OCC(=O)NCCCN(C(C2C(CCC)C2)=O)CC)ccc2c(c1)CCC2=O c1(C(=O)NCC2C(C(C)C)OCC2)cc(Cl)c(Cl)c(Cl)c1O C(C(F)(F)Cn1cc(-c2cscn2)nn1)NC(CCSCCC)=O Cc1nn(CCC(=O)N(C)CCNC(=O)C(c2ccccc2)C)c(C)c1C c1(N2C(C3CCN(C(C(CCC)OC)=O)C3)CCC2)ncnc2c1cnn2C c1(CCC(=O)NCC(CNC(c2c(C)ncs2)=O)F)c(C)nc2ncnn2c1C N1(C(COCCCCC)=O)CC(CNC(=O)CC2CSC2)(COC)C1 C1(C(=O)NCCCN(C(=O)CCOC2CCOC2)CC)CSCN1C(C)=O C1(C)(NC(C2C(NC(c3c(CCC)n[nH]c3)=O)CCO2)=O)CCC(C)=C(C)C1 C(=O)(C(C)CC(F)F)N1CC(CC(C)NC(c2ccc(CSC)o2)=O)C1 C1(CC)C(C(=O)NCCC(O)C(C)C)CCCN1C(=O)C(OC)OC c1(CC(=O)N(CCC)C(c2cccc(F)c2)c2nn[nH]n2)c(Cl)cc(Cl)cc1Cl N1(C(Cn2ccc(C)n2)=O)CC2CCC(C1)C2CNC(c1cc[nH]c1C)=O CCC(CC(=O)NCCC(C)N(C)C)N(C)C(c1n[nH]c(C)c1C)=O CC1(C(=O)NC2CCC3CC2CO3)CCN(C(c2cc3n(n2)CCO3)=O)CC1 CN1CC(=O)N(CC(=O)NCC2CC(O)CN2C(=O)C(F)=CC2CC2)C1=O CC1CN(C(C2(C#N)CCCOC2)=O)CCN1C(n1cc(C(F)F)ccc1=O)=O C1(C(C)Nc2ccc(Cn3cncn3)cc2)CC(C)(C)CN1Cc1ccncc1 c1(OC)cc(F)c(F)cc1C(=O)NC(C)CN(C)C(C1CCCC(=O)N1)=O C(CCCCCC(=O)NCC(c1ccccn1)C)NC(C1(CC=C)CCOC1)=O CC(C)(C)CCC(=O)NCC1CC(n2cc(CCC(CO)CO)nn2)C1 C(=O)(C1=CCC(F)(F)CC1)N(CCNC(c1c(N2CC(C)(C)C2)cccc1)=O)CCO c1(C(=O)NCCCCN(C)C(C2(CCO)CC2)=O)ccncn1 c1(C(N(CCOCC)Cc2ccnn2C)=O)ccn(C(C)C)n1 C1(NC(C(C)=C2CCC2)=O)CCC2(CCN(C(C3(C4CC4)CC3)=O)CC2)C1 N1(C(=O)NCc2oc(C(=O)OCC)c(C)n2)CCc2c(Br)ccnc2C1 C1(C(=O)NCC2CN(C(=O)COCC3CC3)C2)(SCC)CCOCC1 C1(NC(c2cc(I)ccn2)=O)CC2CCC1N2C(=O)C=C1CCC1 Cc1ccc2[nH]c(-c3ccc(C(C)NCc4nc(Cl)c(Br)cc4I)cc3)cc2c1 C(=O)(CC(C(F)(F)F)NC(=O)CCn1cccc1)NCCC(CC)CO Cn1ccc2sc(C(=O)NC3CCOCC3NC(=O)CN(C3CCCC3)C)cc12 N1(C(CCCOCCC)=O)CCOCC(CNC(=O)C(C)NC=O)C1 N1(C(Cc2nc(NC(c3cccc(C#N)c3)=O)sc2)=O)Cc2ccc(O)cc2C1 c1(NC(=O)NCC2CCOCO2)cccc(N2CCOC2=O)c1 Cc1cc(C=CC(=O)N(CC(=O)O)CC2CC(O)C23CCC3)ccc1F N(C(=NCCCF)NCCC1CCOC(C(C)C)C1)CCOC(C)(C)C c1(C(=O)OC)cccc(NC(=O)NC(C2CNC(=O)C2)=O)c1F C1(C)(CNC(C(C)(F)F)=O)CN(C2CCN(C(C34CCCCC3C4)=O)CC2)C1=O N1(C(C(C)CBr)=O)CCCC2(CCCN2C(c2cccnn2)=O)CC1 C1(C(=O)NCCCCN(C)C(C2C(F)(F)C23CC3)=O)CN2CCCN1CC2 c1(C(=O)NC2(CO)CN(C(C(C)OC(C)(C)C)=O)C2)ccc2scnc2c1 C(=O)(C(C)C(F)(F)C(F)F)NCC1(CCO)CN(C(c2c(OCC)con2)=O)C1 Cc1cc(=O)oc(C)c1C(=O)NC1CN(C(=O)CN2CCOC2=O)CCC1CO Cc1cccn2ncc(C(=O)NC3CN(C(=O)CC(C)C)CC3C#N)c12 C(=O)(CC(C)C(C)(C)C)NCC(C)CNC(c1cccc(N2CCCC2=O)c1)=O Cn1ccnc1CCC(=O)NCCC1(NC(C2(C(N)=O)CC2)=O)CCC1 c1(C(N2CC(NC(C(CC)(C#N)CC)=O)C(C)C2)=O)cnn2ccc(Br)cc12 CC(C)CC(C(=O)NC1CC(NC(=O)C(F)Cc2ccccc2)C1)C(C)C Cc1nc(C(=O)NCC(O)CNC(=O)C(C)c2ncco2)co1 N1(CC(=O)N(C(=O)Cc2ccon2)C(C)C)CCC(C2(C(F)(F)F)CCC2)CC1 N1(C(c2cccs2)=O)CCCC2(C1)CN(C(C1CC3(CCCC3)C1)=O)C2 c1(C(N2CC(NC(c3ncn(CC)c3)=O)(CF)C2)=O)ccc2cnoc2c1 CC1CCN(CC(=O)NC2CC2CNC(=O)C(C)Cc2ccnn2C)CC1 C1(n2cc(C(c3cc[nH]c3)C)nn2)CON(C(=O)C2CC2C(=O)OC(C)(C)C)C1 CC1(C)CCCC(C)(NC(=O)C(Cn2cccn2)NC(C2CS(=O)C2)=O)C1 c1(SCC(=O)N(CCN(C(=O)C(F)CCCC)CC)CC)nnc2ccccn12 c1(CC(N2CCN(C(CC=C=C)=O)CC2CO)=O)c(C)nc(C)nc1O N1(C(=O)CCc2cc(F)cc(F)c2)CCC(NC(C23CC(F)C2C3)=O)C12CC2 C1(C(=O)NCCCN(CC)CC)CCCN(C(c2cccc(C)c2O)=O)CC1 N1(C(CC2CC(OCC)C2)=O)CCC2(CC1)CC2NC(c1cc(C)c(C)[nH]1)=O c1(CN=c2ccn(C(C)(C)C)[nH]2)cnc2c(c1)NCC(=O)N2 N1(C(=O)CC2CCOCC2)CCC2CCC(C1)N2C(C1CCC(F)(F)C1O)=O Cc1n[nH]c(=NC2CC3CCCN3C2)s1 Cc1cnccc1CN(C(=O)C#CCNC(C1CCN(C)C1=O)=O)C c1(CN2CC(NC(c3cc(OC)ncc3)=O)C(F)C2)cc(Cl)ccc1Cl c1(C(N2CCCC(CNC(c3c(C)cnn3C)=O)C2)=O)cc(N)nc(Br)c1 C1(C(=O)NC2CC(CC(N)=O)C2)(CC)CCCN1C(c1cnc(C)s1)=O N1(C(CNC(C2C(C)C2)=O)=O)CC(N(C(=O)C=CC(F)(F)F)CCO)C(C)(C)C1 C1(C(=O)NC2(C)CCCN(C(CC(C(C)C)(F)F)=O)C2)CCOCC12CCCC2 N1(C(C(C)OCC)=O)C2CCC(C2)C1CC(=O)NCc1cc(F)cc(F)c1 C1(CNC(C(=O)NCC(C)(O)C2CCC2)=O)CCCSC1 c1(C(=O)NCC2CC(F)(CNC(c3cccnn3)=O)C2)cccc(C2COC2)c1 CC(C)C(CC(=O)N1CCN(C)CC1CNC(c1cc2c(s1)CCC2)=O)C(C)C C12(CNC(C3N(CC)CCC3)=O)CC(CN1C(=O)CC1CCOC1C)C2 N1(C(C(N2CCP(C)(=O)CC2)C)=O)CCC(C)N(C(=O)CCC(N)=O)CC1 c1(C(=O)NCC2C(C)CCN(C(CCC=C(C)C)=O)C2)ccc2nc[nH]c2c1F C=Cc1ccc(C(=O)N(CC)CC2CCN(C(=O)Cn3nccn3)CC2)cc1 c1(C(N2CCC(NC(CC(COC)C)=O)C(F)C2)=O)cc(C)c2c(c1)CCCN2 c1(CC(=O)NC(c2ccccc2)C(=O)N(CC)CC)ccc(Br)nc1 N1(C(c2cnc(C(C)C)o2)=O)CCN(C(C2(N(C)C)CC2)=O)CC1CC(=O)NC CCC(CC(F)(F)F)C(=O)NCCN(C(=O)Cn1cc(C(=O)OC)cn1)CC C1(C(N(CCCCC=C)C)=O)CCC(C)N1C(c1ccnc(CO)c1)=O N1(C(CCCC2(C)N=N2)=O)CCN(Cc2c(CO)cnn2C)CC1c1ncc[nH]1 c1(C(C)C)nn(C)c(Cl)c1C(=O)NC1CCCN(C(=O)C(O)CC(F)F)C1 C1(C(=O)NC2CC(C)CO2)CCCCC1n1cc(CC2(CC)CCC2)nn1 C(=O)(C1CCc2cccnc21)N1CCC(NC(c2ccc(N)c(Cl)c2)=O)C1 N1(c2cc(C)nc(CO)n2)CCC(C2CCCN(C(=O)CC(C)C)C2)C1 C(C(C(C)(C)C)NC(C1CC2CC2C1)=O)NC(Cn1cc(C(=O)OC)nn1)=O C1(C(=O)NC2(CC)CN(C(c3cc(=O)cc[nH]3)=O)C2)CC(=O)C12CCC2 c1(CC(=O)NC2CN(C(CCSc3n(C)nnn3)=O)C2)c(F)cncc1Cl N1(C(C(CCC)=C(C)C)=O)CCOCCC1C(=O)N(C)Cc1cccc(O)n1 n1(CC(=C)C)c(N(C)CCN2CCOCC2)nnc1CCC(F)(F)CO.C1CCC1 C1(N(C(=O)NC(c2ccc(C(=O)OC)cc2)C#N)C(C)C)CCC(CC)CC1 N1(C(COCCC)=O)CC2CCC2(CCNC(c2cccc(C(F)(F)F)c2)=O)C1 N1(C(CCc2nc(C)sc2)=O)CC2(CCC2)CC1CNC(=O)C(C)CC(C)C c1(C(=O)NC2(CO)CCN(C(C(C=CC)O)=O)C2)sc2ccccc2c1CC CCCN(OC)C(=O)C1CCC(C)N1C(=O)CCOC1CCCC1 CN1CC(NC(c2cc(CNC(=O)CCCN=[N+]=[N-])on2)=O)CCC1=O C1(C(=O)NCC(C)CN(C)C(c2cc(C#N)cs2)=O)Cc2ccccc2O1 C(C(CC(C)C)NC(=O)CNC(=O)NC1CC1)NC(Cc1ncc(CC)[nH]1)=O c1(NC(C2(CC)CCN(C(=O)C(CO)OC)C2)=O)ccc2c[nH]nc2c1 C(=O)(C(C)COC(C)=O)N(C1CN(C(C(C)OCC)=O)C1)C C1(NC(C(CC)NC(C)=O)=O)COC2C(NC(=O)CCc3ccoc3)COC12 Cc1ccc(C#N)cc1C(=O)NCC1CN(C(=O)C=Cc2cocn2)C1 c1(OC)ncc(C(N2CCCC2C(=O)Nc2ccc(I)c(C)c2)=O)cc1Br N1(C(C2C(CC(C)(C)C)C2)=O)CC(NC(C2CS(=O)(=O)C2)=O)CC2(CC2)C1 C(=O)(C(F)C(C)(C)O)N1CC(C(=O)NC(C2CCOCC2)C#C)(COC)C1 CCCCCCCC(=O)N(C)CCNC(=O)C(C)(C)Cc1cc2ccccc2o1 C1(CNC(=O)C2=CCC2)CC2(CCN(C(=O)CC3CCC4(CCC4)CO3)CC2)C1 C1(C#N)(C(=O)NC2CC(NC(C=C(CC)C)=O)C2)CCCO1 CC(C)(C(=O)NC1CCN(C(=O)C2CC2)C1)c1ccc(-c2cn[nH]c2)s1 c1(C(=O)NCCC2(OC)CN(C(=O)Cc3ncc(C)s3)C2)nc(C)c(C)[nH]c1=O N1(C(C2(F)CCC(C)CC2)=O)CC2CC(C)N(C(=O)CC(F)(F)C(F)(F)F)C2C1 CCCCN=C(NCCNC(c1ccoc1)=O)N(C)Cc1c(F)cccc1F C1(C(N2CCCC(NC(=O)CSC(F)F)(CO)C2)=O)C2C3CC4C1C1C2CC3C41 c1(C(=O)NCCC(C)N(C(c2c(C)occ2)=O)C)cc2cccnc2nc1O n1(CCC)cc(C(=O)N(C(CC)C(=O)NCCn2cncn2)C)nn1 N1(C(C=CSC)=O)CC(C)(C)OCC1CNC(=O)CNC(=O)CCCCO N1(C(c2ccn(CCN(C)C)n2)=O)CCN(C2CCN(C(=O)C3=CCC3)C2)CC1 c1(SCC)ccc(CC(=O)NCC(CC)N(C(=O)CP(C)(C)=O)C)cc1 c1(CC(=O)Nc2c(C)ccc(C(=O)OC)c2)cc(Br)cc(OC(C)=O)c1OC C1(C(=O)NCC2(CNC(Cc3c(C)nc(C)s3)=O)CCC2)CC2CCCN(C1)C2 C1(C(=O)NCCCOCCN(C(=O)CCc2ccoc2)C)CCC(F)C1 CC(C)CC(CNC(=O)C(C)Cn1ccnc1)C(=O)N1CC(O)CC1C(C)C CC1C(=O)NCCCN1N(C)Cc1ccc(OC2CC2)cc1 C1(C(=O)NCCN(CCO)CC)CN(C(C2CCCC(O)C2)=O)CCC1(C)C C1(CNC(CC(CC)c2ccccc2)=O)C2CCCC1N(C(=O)CCF)C2 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)N1CCCC(CN(C(CSCCC)=O)C)C1 N1(C(c2cnc(S)nc2)=O)CCC2CN(C(c3scc4c3OCCO4)=O)CC2C1 c1(NC(C(=O)NC(CC(=O)OC)C2CC2)=O)cc2c(C)cc(=O)[nH]c2cc1C c1(C(N(CCCNC(c2ncc(OC)nc2)=O)C)=O)cccc2c1C1CCC2O1 N1(C(CC(C)(C)C)=O)CCC(C2CC(NC(=O)CC3CC(n4cnnc4)C3)C2)C1 N1(C(CC)=O)CCN(C(=O)C(Cn2cncn2)NC(=O)CC(CC)SC)CC1 Cc1cc(C)c(C(=O)NC2CN(C(c3cccnc3F)=O)CCC2CO)c(=O)o1 c1(-c2nc(CC)sc2)nc(CCSC)nn1C1CCCN(C(=O)OC(C)(C)C)C1 c1(C(N2CCC(C(N(CCC=C)CC)=O)CC2)=O)cccc(C#N)c1C C1(N(C)C(c2ccc(O)nc2)=O)CCCN(C(=O)C(C)(C)c2cccnc2)C1 C1(C(=O)NC2CCCC(NC(CC3C(C)OCC3)=O)C2)C2CC3CC(C2)CC1C3 N1(C(C2ON=C(CC)C2)=O)CCCC(C)(C(=O)N(C)CCc2cnc[nH]2)C1 C1(C(=O)OC)CC2(CC(NC(c3nc(C4CNC4)cs3)=O)CCS2)C1 C1(C(=O)NCCC(C)C(F)F)CCOCCN1C(=O)CCC1CCOCC1 c1(NC(=O)NC2CC3CCC2(CNC(=O)C2CC2)C3)cccc(Cl)c1Cl C(=O)(CC(CNC(C1CC(O)C1)=O)C1CCC1)NCCC1(C)OCCO1 c1(C(=O)NCC2CCCN(C(C3(OC)CC3)=O)C2)ccc(=O)n2c1CCC2 N1(C(C2C=CC=CC=C2)=O)CCN(C(C2(c3ncco3)CC2)=O)CC12CC2 C1(NC(CN2CC(=O)NC2=O)=O)CC2CCC1(NC(c1cccnc1)=O)C2 c1(NC(C(=O)NC(c2ccc(Br)s2)C)=O)cnn2c1CCCC2 c1(C(C(N2CC(CNC(C3(C)CC(=C)C3)=O)C2)=O)C)ccc(N(C)C)cc1 C1(C(N(C)CCN(C)C2CC2)=O)CC2CCC(C1)N2C(c1ccc(F)cc1O)=O C1(C(N2CCCC2CN(C(=O)C(=O)NCCC(N)=O)C2CC2)=O)(CC)CC=CC1 Cn1nnc2cc(C(N3CC4(C3)SCCC4NC(C3CC=CCC3)=O)=O)cnc12 c1(CC(=O)NCC(C2CC2)NC(c2[nH]nnc2C2CC2)=O)ccc2ccoc2c1 C1(C(=O)NC(c2ccc(F)cc2)C(C)(C)C)C[Si](C)(C)CN1 c1(C(=O)NCC2CN(C(CC(C)OC)=O)C(C)(C)C2)nc2ncccn2n1 C1(C2CCN(C(C3(F)CCCC3)=O)CC2)(NC(c2ccc(NC)cc2Cl)=O)CC1 C1(C(N2CCC(O)(CNC(=O)CC(C)F)CC2)=O)(COC)CCCNS1(=O)=O c1(C(=O)NCC2C(NC(=O)CCc3csnn3)CC2)ccc(C(F)(F)F)o1 c1(NC(C)CC2CC2)cccc(NC(=O)NC(c2ccccc2)C)c1 C1(NC(c2c(Cl)cn(C)n2)=O)CC(O)CN(C(=O)CCSCC(N)=O)C1 N1(CCC)CCN(CCCCNC(=O)OC(C)(C)C)CC1.C12(C)CCCN1C2=O c1(C(N2CCC(N(C(CN(CC)CC)=O)C)C2)=O)cc(N2CCOCC2)ncn1 N1(C(C2(C=C)CCC2)=O)CCCC(C2CN(C(C3CCC(N(C)C)CC3)=O)C2)C1 c1(NC(C(c2cnccn2)C)=O)ccc(C(F)(F)F)c(O)c1 c1(C(CNC(C2CC(=O)NC2)=O)NC(C2CC(F)(F)C2)=O)ccccc1Br C(=O)(N=c1[nH]c(Cl)ncc1O)c1cc(-c2c(SC)c(F)cc(F)c2)[nH]n1 c1(OC)cc(C(=O)NCCOCCN(C)C(C2CCCC2C(F)F)=O)oc(=O)c1 CC(CS(C)(=O)=O)C(=O)N(C)CCOCCN(C)C(c1cnn(C)c1F)=O N1(C(c2c(C)nccn2)=O)CC2OCCN(C(=O)CC3OCCOC3(C)C)C2C1 CC1CCN(C(c2cnc3ccccn23)=O)CCN1c1nc(Cl)ncc1F C(CCC(=O)NCCCC1(NC(C2CC2c2nc[nH]n2)=O)CC1)OCCOC N(C1CCOc2ccc(F)cc21)CC1C(C)C1 C1(CNC(C2CCC(C)(C)O2)=O)CN(C(=O)C#CC2CC2)CCCO1 C(=O)(C#CC(C)(C)C)NC(C(C)C)C(C)NC(=O)Cc1csc(C2CC2)n1 CC1(C)CN(C(=O)CSc2ccccn2)C1C1CCN(C(=O)C2=CCCO2)CC1 c1(C(=O)NC2CC(NC(C(C=C)O)=O)C2)cccc(Cn2nccn2)c1 N1(CC)CCCC(C(=O)NCC2(O)CCN(C(C3(OC)CCCCC3)=O)C2)C1 CCC(CCC(=O)NCCC1CCSC1)NC(c1ccc(F)c(O)c1)=O Cc1cn2c(C(N3CCC(NC(c4nncs4)=O)C(C)C3)=O)c(Cl)nc2s1 C1(NC(C(C)NC(N)=O)=O)CN(C(c2cc(CN(C)C)c[nH]2)=O)CCC1(C)C CC1C(O)CC2CCC1N2C(=O)NC1(Cl)CCOCC1 N1(C(CCCCCC(C)C)=O)CCC2CCCN(C(=O)CCOCC(C)C)C2C1 N1(C(c2cc(C)c(O)nn2)=O)CCCC(C2CC2NC(=O)C#CC(C)(C)C)C1 n1(CCNC)cc(CN(C)C(=O)NCCOCc2ccco2)nn1 N1(C(C(C)=C2CCCC2)=O)CCN(C(=O)CCN(c2ccccc2)CC)CC12CC2 c1(OCC)cc2c(=NC(CN(C)C)CCO)[nH]cnc2cc1F c1(CC)nnc2n1CCCC2C(=O)NCCC1CS(=O)(=O)C1.C12(CC1)C(=O)NC2 c1(NC(c2ccc(OC)cn2)C)nccc(=NCCC(C)c2ccccc2)[nH]1 C=CCCCCC(=O)NCC(C1CC1)NC(C1(C(=O)N(C)C)CC1)=O C(=O)(CCS(=O)(=O)N(C)C)NCCC(C)NC(=O)CC1CCCCC1(F)F N1(C(C=CC=CCC)=O)CC2CC(C)N(C(c3ccnc(F)c3OC)=O)C2C1 CCN=c1[nH]cc(C(=O)NC2CCC(NC(=O)COCC3CCOC3)CC2)s1 C(=O)(C1CCC(=O)c2cccn21)NCCCC(C)NC(c1c(C)nc(C)o1)=O C(CC(CC)C(=O)N1CCN(C(c2cocc2C)=O)C(c2nccn2C)C1)=CC C=CC(C)N=c1[nH]c(N2CCC(C3CC(F)(F)C3)C2)nc2c1COC2 CCC1=NOC(CNC(=O)C(C)N(C)C(c2cn(C3CC3)nn2)=O)C1 c1(C(=O)OC)cn2cccc(NC(=O)Nc3cc(Cl)cc(Br)c3Cl)c2n1 C1(C(C)NC(=O)CSc2nncs2)CCCN(C(C2CCC(=O)C2)=O)C1 C(c1cc(F)c(F)c(F)c1)=CC(N1C(C(=O)NCC(=C)C)C=CC1)=O C(CC(C(=O)N1CC(CNC(=O)Cc2nn(C)cc2Cl)C1)NC(C)=O)SC C(CS(=O)(=O)c1ccc(Br)cc1)N(C1(CO)CCN(C)CC1)C1CC1 CCCC(O)C(=O)NC1CC(C)(CNC(=O)CC2CCN(C)CC2)C1 C1(S(C)(=O)=O)(C(=O)OC)CC(NC(=O)CC2CCC(C(F)(F)F)O2)C1 c1(CCNC(c2cnc(C)s2)=O)ccc(F)cc1Cl N1(C(c2cc(OCC)n[nH]2)=O)CCCC2(CCN(C(C3CC(F)C3)=O)C2)C1 C#CC1(NC(=O)COC2CN(C(c3cncc(C#N)c3)=O)C2)CCC(C)CC1 c1(NC(C(=O)NC(C#C)(C)CC)=O)ccc(C2CC2)c(C#N)c1 N1(C(C(C)N(C)C)=O)CC2(CNC(c3cnc(Br)s3)=O)CCC1CC2 N1(C(CC2CC(OCC)C2)=O)CCCC1(C)CNC(c1c[nH]c(=O)cn1)=O c1(CC)cc(C)c(-c2nc(-c3ccc(OC)cn3)nn2CCCOC)o1 C12(C(=O)NCC3N(C(=O)CCc4nc(O)n[nH]4)C4C(C3)C4)CCCC1OCC2 C1(CC)C(NC(c2ccc(N)c(F)n2)=O)CCCN1C(c1cnc(Cl)s1)=O C(=O)(C(C)(C)C(=O)N1CCOCC1CN(C)C(c1cncc(Cl)c1Cl)=O)OCC c1(OC)c(O)cc(C(N2CC3(CCN3C(c3cnccn3)=O)C2)=O)cc1O C1(CSC)CN(C(c2sccc2Cl)C(=O)NCCC2(C)CC2)CCO1 N1(C(c2c(Cl)ccc(OC)c2)=O)CC2CCC1C1CN(C(=O)C(C)C3CC3)CC21 CC1(C)CCCCC(C(=O)NCCC2CSCCN2C(=O)C(Cl)=CCl)C1 n1(CCC)cccc1C(N1CC(CC(C)NC(=O)C(C2CC(F)(F)C2)O)C1)=O Cc1cc(Cl)ccc1CN(C(C)(C)CC1CNC1)CCO C1(CCC)CC(C(=O)NCC#CCNC(=O)CCC2SCCS2)C1 C1(C(N(CC(CC)NC(c2c(C(F)(F)F)cnn2C)=O)CC)=O)CN(C)C(=O)N1 C12(C(C)NC(C34CC(CN=c5nn[nH]n5C)(C3)OC4C)=O)CCC(CC1)CC2 C(=O)(CC(C)(C)C(=O)NC1CN(C(c2ccn(C)n2)=O)CC1C(F)(F)F)OCC C(=O)(C(C)CCC(C)(C)C)N1CCN(C(C2(CC=C)CCC2)=O)CC1CCO CC1CC(NC(c2cncnc2)=O)CCN1C(c1ccc(C2CC2)c(F)c1)=O c1(C(N2CCC(C)(CNC(CNS(CC)(=O)=O)=O)C2)=O)cccc2[nH]ccc12 N1(C(C2(OC)CCC2)=O)CCC(C2CCN(C(C3CS(=O)(=O)C3)=O)C2)CC1 n1(CCC=C=C)cc(C(C)(C)CC)nn1.C12CCCN1C(=O)c1cnn(c1)C2 CC1CCN(C(c2cccc(CN3CCCC3)c2)=O)CCC1(F)F C(CCCCCC(=O)NCCCc1cn[nH]c1)NC(CC1C(C)C(=O)CC1)=O N1(C(c2ccc(C)nc2O)=O)CCC(NC(=O)C2=CCCOCC2)CC(C)(C)C1 S(=O)(=O)(c1ccc(CCN)cc1)N(C)CC1CCCCC1O C=CCC(F)(F)C(=O)N1CC(CN(C(=O)Cc2ccc(Cl)c(F)c2)C)C2(CC2)C1 C1(CCC(=O)N(CC(F)F)CC)CCN(C(=O)Cc2csnn2)C1 N1(C(C2(C)CCOCC2)=O)CC2(CCC(C(=O)NCC3(C4CC4)CCCO3)O2)C1 N1(C(CN2C(C)CCCC2)=O)CCC(C)N(C(c2cnn3ccn(C)c23)=O)CC1 c1(CNC(C2(C(C)NC(=O)Cc3ccn(C)c3)CC2)=O)ccc(C#N)cn1 O=C1CN(C(C23CCOC2CS(=O)(=O)C3)=O)c2cc(Br)cnc2N1 C1(NC(CC(C)OC)=O)CCC12CCN(C(=O)C=Cc1ccc(=N)[nH]c1)CC2 Cc1cc(=NCCc2cnc(O)nc2)[nH]c(=NCc2ccc(N(C)C)cc2F)[nH]1 S(=O)(=O)(c1ccc(Cl)cn1)N(C(CCO)C(F)(F)F)C c1(CNC(CCCn2cc(CCOC)nn2)=O)ccc(OS(C)(=O)=O)nc1 CC(CCCNC(=O)C(C)(C1CC1)NC(C1(CF)CC1)=O)NC(=O)OC(C)(C)C C(CC(O)C(=O)NC(Cc1cn[nH]c1)C(=O)NCC1(O)CCSC1)N(C)C CC(C)CCC(O)C(=O)N1CC2CCC1CC2NC(C1CN2CCC1CC2)=O N1(C(C(C)Oc2ccccn2)=O)CC2CC1CN2C(c1cc(I)cnc1Cl)=O c1(CC)ccc(C=CC(N2CCCC2CNC(=O)Cc2cnccn2)=O)o1 c1(C(N(C2CCN(C(C3(O)CC3(C)C)=O)C2)C)=O)ccc(Cc2nc[nH]n2)cc1 N1(C(c2cn(C)[nH]c2=N)=O)CCC2C(NC(c3ccnc4ncnn34)=O)C2CC1 CC1(C)CC1(O)CC(N1CCC(CNC(c2cnn(Cc3ccccc3)c2)=O)C1)=O N1(C(CC2CCC(=O)N2)=O)CC2CCC1CC2NC(c1cccc(O)n1)=O N1(C(C(CC)N(C)C)=O)CC(F)CC1CN(C)C(c1ncoc1Br)=O CN1CC(NC(c2ccc(CNC(C3CC(N(C)C)C3)=O)s2)=O)CC1=O c1(C(=O)NC(C)C(C)NC(c2c[nH]nc2C(F)(F)F)=O)cc2c(F)cccc2s1 c1(NC(C2CN(C(=O)CCc3ccco3)CCC2(F)F)=O)ccc2c(c1)CCC2 CC(CCCCNC(C1CC(C)(C)CO1)=O)NC(C1(c2cccnc2)CC1)=O C1(C(N2CCC(CNC(C3CC3c3ccccn3)=O)C2)=O)CCCC2(CC2)C1 c1(OC)cccc(C(N2CC3CC2C3CNC(c2csc(NC=O)n2)=O)=O)c1 N1(C(CC2ON=C(CC)C2)=O)CCCC(C(=O)NCC2(CCO)CC2)(CC)C1 N1(C(c2ccc(O)c(F)c2)=O)CCC2(CC1)CN(C(C13CCCCC1C3)=O)C2 C1(C(=O)N(CC(=O)NC)C)(CC)CCCN1C(=O)Cn1cnnn1 c1(-c2ccc(C)c(C)c2)ccc2c(C(=O)Nc3cc(Cl)cc(Br)c3C)n[nH]c2c1 CN1C(=O)CCC1C(=O)NCC(C1CC1)NC(c1cc(-c2ccccn2)no1)=O N1(C(CCC(CC)OC)=O)CCC2CCN(C(c3n[nH]c(C4CC4)c3Cl)=O)C2C1 Cc1cc(O)c(Cl)cc1C(N1CCC1CNC(=O)CN1CC2C=CC1C2)=O Cc1cc(NC(=O)C(c2cccnc2)NC(=O)Cc2cscn2)cnc1O N1(C(c2c(CC)nco2)=O)CCC2(CC1)CC2CNC(c1c(C)cncc1C)=O C=CC(C)(CC)C(=O)N1CC(O)(CCNC(=O)CCC2CCCOC2)C1 C(C(C)(C)CCCO)NC(C1N(C(c2c(CC)n(C)nn2)=O)CCCC1)=O C1(CNC(C2(CC)CC2(F)F)=O)CCN(C(=O)CC2CCOC2(C)C)CC1 N1(C(c2cnc(OCC)nc2)=O)CCC(NC(c2ccc(Cl)cc2F)=O)C(C)C1 Cc1cc(C(=O)NC2CCCC2CNC(=O)C(C2CC2)N(C)C)c(C)cn1 CC1CC(CNC(=O)Cc2ccc(C#N)nc2)CCN1C(c1cccnc1S)=O CC1(C)CC(NC(c2ccnc(OC3CC3)c2)=O)CN1C(c1[nH]cnc1C#N)=O Cn1nnc2c(NC3CC4CN(C(C5CC6(CCC6)C5)=O)CC34)ncnc12 N1(C(C2(CC#C)CCOC2)=O)CCC(C)(NC(=O)C(F)C2CCCC2)CC1 N1(C(=O)NCc2ccc(CC)o2)CCCCC1c1ccccc1Br C1(C(C)C)(C(=O)NCC2CC(C(=O)OC(=O)CSCC(F)(F)F)C2)CC(C)(C)C1 c1(C(=O)NC2CC(CNC(c3ccccn3)=O)C2)ccnnc1Cl c1(NC(c2ccc(Oc3ccccc3)c(Br)c2)=O)cc(F)c(F)c(Cl)c1F C1(CCNC(C2CC2(Cl)Cl)=O)CN(C(C2(C(F)F)CC(F)(F)C2)=O)CCO1 c1(C(=O)NC2CCC(C)(NC(C3CC4(C3)CC4F)=O)CC2)occ2c1CCCC2 N1(C(C2CC(C)(C)O2)=O)CCCC(C)(C)C1CNC(=O)Cc1ccccc1F n1(C(CC)C)nnnc1C(c1cnccn1)NCCCOCCCO c1(-c2n(CC(C)C3CC3)nc(-c3cncc(F)c3)n2)cc2c(s1)CCSC2 Cc1cnc(C(=O)NCC(C)(C)OCCNC(C2CCC2C)=O)c(C)c1 N1(C(C(CCOC)OC)=O)CCCC(C(=O)NCc2snnc2C)CC1 C1(NC(c2c(C)[nH]nc2C(C)C)=O)CN(C(C2(F)CC2C)=O)CC1N=[N+]=[N-] c1(C(C)=O)ccc(C(=O)NCC(C)CNC(c2cc(C)oc2C(F)(F)F)=O)nn1 C#CC1CCCCN1C(c1ccnc(CNC(C2(SC)CC2)=O)c1)=O C1(C)(C(N(CCNC(C2N(CCC)CCCC2)=O)CC)=O)CCN(C(C)=O)CC1 C1(c2cn(C(C)C(=O)NC3CCS(=O)(=O)C3)nn2)(OC)CCCCCC1 c1(C(N2CC(CC)C(C(=O)O)C2CC)=O)csc(=NC2CC2)[nH]1 O=C1CCCCC(NC(C2CCCCN(C(=O)COCC3CCCC3)C2)=O)C1 C(CC1=CCN(C(c2nncn2C)=O)CC1)NC(C=Cc1cnc(OC)nc1)=O n1(CC(C)O)cc(C(=O)NC2CCN(C(c3cc(N)cc(F)c3)=O)C2)ccc1=O C12(CC(=O)NC3CC(=C4CC4)C3)CCCCCC1N(C(=O)CN1CC=CC1)CC2 C1(NC(C2CC(SC)C2)=O)CCN(C(c2coc(C3CCCCC3)n2)=O)CC1C C1(F)(CNC(=O)CCC2CC2(F)F)CCN(C(C2(c3ccno3)CC2)=O)C1 c1(C(=O)NCCCN(C(c2cc(C)[nH]n2)=O)CC)cn(C)nc1C(F)(F)F C(=O)(C#CC1(C)COC1)N1CCN(C(C2CN(C)C(=O)N2)=O)C(CO)C1 c1(OC)cccc(C(=O)NCCCOCCN(C)C(C2C3CCCOC23)=O)c1F N1(C(Cc2c(C)non2)=O)CCOCC1CC(=O)NCC1(C)CCOC1 C1(C(=O)N(C2CC2NC(C23CSCC2C3(F)F)=O)CCO)CCC(F)(F)CC1 C=CCC(C)(C)CC(=O)NCC(O)CC(=O)NCC(C1CCC1)OCC N1(C(Cn2c(C(C)C)ncc2)=O)CCC(CNC(c2ccc(F)s2)=O)CC1C CCS(=O)(=O)CC(=O)N1CC(NC(c2c(C)cnn2C(C)C)=O)CC(C)C1 N1(C(C=C(CC)C)=O)CCN(C(=O)C(Cc2ccco2)C(=O)OC)CC1CC C1(NC(C(C(COC)C)C)=O)CN(c2nc(Cl)nc3c2CCC3)CC2(CCC2)C1 Cc1cc(C(C)C)ccc1OCC(=O)NCC(CO)NC(=O)C1=CCOCC1 N1(C(C(C=C=C)C)=O)CCC2(CCC(CNC(C3(C(C)C)CC3)=O)CC2)CC1 c1(C(=O)NCCC2CCN(C(c3nnn(C)c3N)=O)C2)nn(C)c2c1CCCC2 c12nc3cc(C(C)C)ccc3n1CC2=O.C=C1CC2CCC(C1)N2C(C1CNCCS1)=O C(=O)(CC1OCc2ccccc21)N(CCNC(C1(C=C)CCC1)=O)CCC c1(SC(C(=O)OC)CO)ccc(OC(C)C(=O)Nc2cccc(F)c2)cc1 C1CC(NCC2C3COCC23)C2(C1)CCN(Cc1ccccc1)C2 C1(CNC(C(CSC)C)=O)COCC2(CCN(C(=O)Cc3conc3C)CC2)O1 c1(C(N2CC(C)C(NC(=O)CCN3CCC3)CC2)=O)cc(Cl)cc(Cl)c1F C(CCCCC(=O)NC1CC(CCNC(=O)C(C)CF)C1)NC(=O)OC(C)(C)C c1(C(=O)NCCCCNC(=O)CN2CCC(O)CC2)cc2sccc2[nH]1 c1(C(N2C(CNC(COCCSC)=O)CC(O)C2)=O)ccc(C2CC2)nc1O c1(C(N2CCN(C(C(C)N3CCC3)=O)CC2CF)=O)ccc2occc2c1 C(=O)(CC(C)C(C)(C)NC(=O)C(C)NC(C)=O)N1CCC(CC=C)C1 c1(C(=O)NC2CN(C(C(C=C)(C)CC)=O)CC(C)C2)nccc2ccccc12 C1(CNC(C(C)C2CCCC2)=O)CCC(NC(C2(C(N)=O)CCC2)=O)C1 C1(C(=O)NCCN(CCOC)C(c2cc(OC)no2)=O)(C(F)F)CCCC1 N1(C(CCC(=O)N(C(C)C)C)=O)CCN(C(c2cccc(O)c2)=O)C2CCC12 C(=O)(C(C)CC(N)=O)NCC(C)=CC(=O)NC1C(=O)OCC1CO C(C)(C)(CC(=O)NCC1(C)CCN(C(=O)CC2CC(F)(F)C2)C1)OC C1(NC(C=Cc2cn(C)nc2)=O)C2CC3C(C2)C13C(=O)NCC(F)CO C=CC1(C(=O)N(C)Cc2csnc2C)CCN(C(=O)CC(C)C(F)F)CC1 C(CC(=O)N(CCN(C(c1csc(C)c1)=O)CC)CC)(C(C)C)OCC c1(C(=O)NCC(=C)CCNC(C2SCCCS2)=O)ccc(-n2cc(C)cn2)cc1 N1(C(c2ccc(CC)s2)=O)CCC2CN(C(c3ccccn3)=O)CC2CC1 N1(C(c2cccc(CCC)c2)=O)CC(F)(F)CC1(C)CNC(=O)C=CCO N1(C(C2(C)C(CC)CCC2)=O)CC(NC(c2cnn(C)c2)=O)C(C)(C)C1 N1(C(c2n(C)c(O)nc2)=O)CCCCC(CNC(C2(S(N)(=O)=O)CCC2)=O)C1 n1(CC(=O)N(C(C)CNC(C2CC2(F)F)=O)C)cnc2c1CCCC2 c1(OC)nc(C(N2CCN(C(c3cc(OC)ccc3F)=O)C3CC23)=O)cc(O)n1 c1(CCC(=O)NC2CCC(CC(N3CC(O)C(F)C3)=O)CC2)cccc(Br)c1 C(CCC(C)(C)C(=O)N(C)CC1CC1C)NC(C=CCCC)=O C(=O)(C(C)(C)C(=O)NC)NC1CN(C(CC(CC)SC)=O)CC1C c1(CN2C(C)(C(=O)Nc3ccc(I)c(F)c3)CCC2)ccc([N+](=O)[O-])cn1 N#Cc1cc(C(N2CC(NC(c3cccn3C3CC3)=O)C3CC23)=O)ccc1F C(CCCCCN(C)C(C1CC1CCC)=O)NC(C1(CC#C)CCOC1)=O N1(C(CCN(CCC)C)=O)CCC(CC(=O)NC(C2CCOC2)CO)CC1 c1(C(C)C)cc(C(N2CCC(NC(C3(C#N)CCOC3)=O)C2)=O)nn1C c1(-c2ccn(C)n2)ccc(Cl)c(NC(N2CCCCC2C(N)=O)=O)c1 N1(C(C=CC(C)NC(=O)C(c2cccnc2)O)=O)CCC(C2CC2)CC1 C1(C(N(C)C)=O)CCCN(C(=O)C(=O)NCC2CNCCN2C)C1 N1(C(C=CCC)=O)CCN(C(=O)CCC(C)(C)C)CC1C(C)C C1(N2CCOCC2)(CC(=O)NC(C(C)NC(=O)C2CC2)C)CCCC1 N1(C(CCC)=O)CC(N(C(=O)CCCCNC(c2ccccc2)=O)C)C(F)C1 C1(C(N2CC(NC(C(CC=C)OC)=O)C3(C2)CC3)=O)OC(C)(C)OC1(C)C C1(CNC(c2cnc3[nH]cnc3c2)=O)CCC2(CN(C(c3cn[nH]c3)=O)C2)O1 C(=O)(CCCCCF)NCC(C(=O)NCC(N(OCC)C)=O)C n1(CCN(C(C23CC(CO2)C3)C)C(=O)NC(C)(C)C)c(=O)cnc2ccccc12 C(=O)(C(C)(C)C(C)(F)F)N(CC(C)C(=O)NC(C)C(=O)NO)C N1(C(c2ncn(C(C)C)n2)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC1C(F)F C1(F)(NC(C(C=C)c2ccccc2)=O)CCS(=O)(=O)C1.C12CCC(C1)CNC2=O c1(C(c2nnnn2CCCOC)NC(COC)C)c(C)c(C#N)n2ccccc12 C1(C(N2CC=C(C)C2)=O)N(C(c2ccc(O)cc2)=O)CCC1(C)C C12(CNC(C(C)Oc3ccccc3)=O)CCC(CN(C(=O)CCCC(F)F)C1)C2 N1(C(Cn2cc(C(=O)OC)nn2)=O)CCC(C2CC2)(CNC(=O)CC(C)(F)F)C1 Cc1cnc(N)c(C(=O)NC2CCOCC2NC(c2coc(C)c2)=O)c1 C1(O)(C(N2CCC(CCN(C(=O)C(F)C3CCC3)C)CC2)=O)CCC(C)(C)CC1 C12(NC(c3nc(C)sc3)=O)CC(CNC(=O)CC(C)C(F)(F)F)(C1)OC2(C)C C1(N(C(C2(COCC)CC2)=O)C)CCC(OC)CC1.C12CCC(C1)CNC2=O C1(CC(=O)NC(C#C)(C)C2CC2)C(NC(=O)COCc2ccccc2)CC1O c1(C(C(N2CC(C(C)NC(c3c(C)scn3)=O)C2)=O)C)cccc(F)c1 C1(CC(C)C)CCC(NC(=O)CCCN(C)C(c2c[nH]nc2C2CC2)=O)C1 c1(C(N(C)CC2CCCN2C(C2CC(CF)C2)=O)=O)ncncc1F c1(OC)nc(C(=O)N(CC(C)NC(c2ccc(C(C)(C)C)cc2)=O)C)ncc1F N1(C(CC(C)C)=O)CC(CNC(C2CN(c3ccccc3F)C2)=O)OC2(CCC2)C1 c1(OCC)cc(N2CCC(CNC(c3nc(Cl)sc3Cl)=O)C23CC3)nc(C)n1 CN1CC(C(N2CCC2(C)CC(=O)NCC(C)(C)C2(O)CCC2)=O)CCC1=O C1(C(NOC(C)(C)CO)=O)CN(C(=O)C(C)(C)CC#N)CC1(F)F Cc1ccc(C(=O)NCCc2n[nH]cc2C(=O)NC2CC2(C)C(F)F)nc1O N1(C(C2N(C(CCC(C)N(C)C)=O)CCC2O)=O)CCn2ccnc2C1 C1(CC(=O)NC(CC=C)CNC(c2ccnc(Cl)c2O)=O)CC2(CCCC2)CO1 N1(CCNC(C2(CCCC)CCCC2)=O)CCN(C(=O)CC2(O)CCCC2)CC1 C1(CC)CCCN(C(=O)C(CNC(=O)C=Cc2ccc(C)cc2)C(C)C)CC1 c1(C(=O)NC2C(C)N(C(=O)C(CCO)N(C)C)CC2)[nH]nc2ncccc12 C1(OCC)CC(=O)NC2OCCC2C(=O)NCCCO1.C1(COCC)CC1 c1(OCC)cncc(CNC(N2CCC(O)(c3ccc(F)cc3)C2)=O)c1 c1(C(=O)NCC2N(C(C(CC)(C)C)=O)CC2)c(C)nn(CC(F)(F)F)c1C N=c1[nH]c(=NCCc2cc(Cl)ccc2Br)[nH]c(=NC2CCN(CC(F)F)C2)[nH]1 c1(C(=O)NCC(C)(CO)NC(c2c(CC)nc(C)[nH]2)=O)cccc2c1ncn2C Cc1nnc(O)c(C(N2CCCC(CNC(=O)C=CC3CCOC3)C2)=O)c1C c1(NC(c2cncnc2)=O)cnc(Cl)cc1C(N1CCSCC1)=O c1(C(N2CC3CN(c4ncc(OC)cn4)CC32)=O)ccc(C#N)c(F)c1 c1(NC(c2c(F)ccc(Cl)c2Cl)=O)cc2c(cc1Cl)OCCO2 C(CC(C(C)(C)C)NC(=O)CCc1c(Cl)cccc1Cl)NC N1(C(CCC(CC)NC(=O)CC(O)CC)=O)CCC2CCCC2CC1 C(C(CC(F)(F)F)NC(=O)CC1CCCCCO1)NC(CC=C)=O c1(C(N2CCC(CCCO)C2)C(=O)NCC(=C)C)ccc(C)c(Br)c1C C=CCCCCCC(=O)N1CCN(C(=O)C(C)n2cnnn2)C(CC)C1 Cc1cnncc1C(=O)OC(C)(C)C.N12CC(F)(F)C1C1CN(C1)C(=O)NCC2 C1(CCC(=O)N(CCCCNC(=O)Cc2cnc[nH]2)C)CCCC(O)C1 C(=O)(CCCCC(N)=O)N(C1CC(NC(c2cn3c(n2)CCC3)=O)C1)C N1(C(C(C)(C)n2cnnn2)=O)CC2CCCC(NC(C3CC3C#N)=O)C2C1 C1(CC)CN(C(C2CCCN2C(C)C)=O)CCN1C(=O)CCc1nnc(S)n1C c1(CNC(CC=CCC)=O)cccc2c1CN(C(=O)CCCc1cnn[nH]1)C2 C1(OCC)(CN(C)C(C2CCC2CNC(=O)C=CC2CC2)=O)CCC1 C(=O)(C(C)C(C)NC(C1(C)CCCN1C)=O)N1CC(COC(C)=O)C1 c1(C(N(C2CCCCC2)CCNC(C(COC)(F)F)=O)=O)nccc(Cl)c1Cl Cc1cnc(CN2CCCC(O)(CNC(C3C4COCC34)=O)C2)cc1Br C(=O)(C(C(=O)N(C(C)C(=O)N(C1CCCC1(C)O)C)C1CC1)OC)OCC C1(NC(C(C(C)C)C)=O)CCSC12CN(C(c1ccc(O)cc1C(F)F)=O)C2 c1(NC(=O)NCCN(CC=C)C)ccnc(F)c1OC Cc1csc(CNC(c2csc(CNC(=O)C(C3CCOCC3)O)c2)=O)n1 C#CCCCCC(c1nnnn1CCCCCC)NCC1CCC(CC)O1 c1(C(=O)NCCC2CC(C(N(CC(C)C)C3CC3)=O)C2)cnc2ccccn12 c1(C(=O)NCC(CC=C)NC(=O)C(C)CN(C)C)cnncc1C(F)(F)F S(=O)(=O)(c1ccc(N2CCN(C3CC3)CC(C)C2)c(C#N)c1)NCCCC#N Cc1ncc(CC(=O)NC2(C)CCCN(C(c3cc(CO)oc3C)=O)C2)c(O)n1 C1(NC(CCSC)=O)CC(C)N(C(=O)CC2C=CCC2)C1 Cc1cc(C(N2CCCC(N(C)C(C3(F)CCOC3)=O)CC2)=O)c(O)c(C)c1 C(CCCC(=O)N1CCC(C(F)C(=O)NOCC2(F)CCC2)C1)(OC)OC c1(C(=O)NCCC(C)NC(c2cc(C)c(C)o2)=O)ncc(C(N)=O)cc1Cl C1(C(=O)NCC(n2cccn2)C)CCCCC1CNC(C1CN(C)C1)=O c1(CC(=O)NCCOC2CCN(C(CNC(CC)=O)=O)C2)ccc(Cl)c(C)c1 C#CCC(C)(C(=O)NCC1CC1(Cl)Cl)NC(=O)CCOC1CCC1 C1(C(=O)NCC(C(C)C)NC(CC2(C(=O)OC)CCC2)=O)CC2C(C1)C2(C)C C(C)(CC(=O)NC(CO)C(C)NC(=O)CCc1cnn(C)n1)OC Cc1cc(C)c(C(=O)NC23CC(CNC(=O)CC(O)c4ccccc4)(C2)C3)o1 C(C(C)(C)CC(=O)N1CC(CF)(NC(=O)CC(C)F)C1)OC N(C(=NCCCF)NC(CO)C1COC1)C(C1CCCCC1)C C12(CNC(C3(S(N)(=O)=O)CC3)=O)CC(CO1)N(C(C1CCCC3(CC3)C1)=O)C2 C1(C(N(C)CC2(CNC(C3C4CCCC34)=O)CC2)=O)COc2ccccc2O1 C1(NC(c2cnc(-c3cccs3)s2)=O)CCN(C(=O)C2CC2)CC12CCC2 c1(C(=O)NCC2N(C(CC(N3CCCCC3=O)C)=O)CC=C2)cc(Cl)ccc1Cl c1(OC)ccc(C(=O)NCC(C2CC2)NC(=O)CC2CC3(CC3)CO2)c(C)n1 CCCCC(=O)C(=O)NC1CCC(CNC(=O)CCc2ccccc2C(N)=O)C1 Cn1ncc2c1CCC(C(=O)NCC1CCN(C(C3CC=CC3)=O)CC1(F)F)C2 Cc1nc(N2CCC(C)C(NC(=O)COCC3CC3)C2C)c(F)c(C)n1 c1(NC(C2CN(Cc3c(Cl)cc(Cl)cc3Cl)CCS2)=O)nccn2c(Br)cnc12 C1(NC(CSCCCC)=O)CCCCN(C(=O)C=Cc2cccnc2C)C1 C1(NC(C(C2CCC(=O)N2)C)=O)CCN(c2cc(Cl)nc(C3(C)CC3)n2)CC1F C1(C#N)(C(=O)NCC2(C(=O)NC3C(CC(C)C)C3)CCC2)CCCCC1 N1(C(c2cccc(C)n2)C(=O)NCCC#N)CCN(S(=O)(=O)N(C)C)CC1 C1(CNC(C(=O)NCC)=O)(NC(c2ncccc2N)=O)CC2CCC1CC2 C#CCC(C(=O)NCC(C)(O)CNC(c1cccc(C(N)=O)n1)=O)C1CC1 C=CCCCC(C(=O)N(C)Cc1nnnn1C)NC(=O)CCCOC(C)C CCC(CC(F)F)C(=O)N(C(C)CCNC(c1ccc(SC(C)C)cc1)=O)C c1(C(=O)NC2CCN(C(C3C(CC)C3)=O)CC2)coc2c1C(=O)CCC2 C1(C#C)(C(N(CC#C)CCO)=O)CCN(C(C2CCCC(C)CC2)=O)CC1 C1(N(C)C)CCN(CC(=O)N(C)Cc2cccc(Cl)c2)CC1.N12CCC(C1)C2=O CN1CCC(C(=O)NCC2CCC(NC(C3CCCNC3=O)=O)CC2)CC1 c1(CC(=O)NC(COCC#C)C(N2CCC(C#C)C2)=O)cc(C)nn1C C(C)(C(=O)NC1CC(C(F)C(=O)NCCCOC(=N)O)C1)NC(=O)OC N1(C(c2c(NC)nccc2)=O)CC2CCC(CNC(=O)CCCOC(C)C)C2C1 C(=O)(CS(=O)(=O)C1CC1)NCCCCn1cc(CN2CCN(C)CC2)nn1 n1(CCC)ccc(=NC(C)(CC(OC)OC)c2nnnn2C)[nH]1 c1(OC)cccc(CCC(=O)NC(CNC(c2ncsc2C(C)C)=O)C(C)C)n1 N1(C(CC(=C)C)=O)CCC2(CCOC2)C(CNC(C2CCSC2)=O)C1 C1(CNC(=O)Nc2sc(Cl)cc2Br)CCCC(C(F)(F)F)C1 C1(CNC=O)(O)CCSC1.C1(C(=O)NC(C(=O)OC)C)SCC=C1C C1(NC(C(C)CN(C)C)=O)CC2CC1N(C(=O)CCN1CCNC(=O)C1)C2 CCC(CC)C(=O)N1CCCC(CC(=O)NOCc2ccccc2)C1 C1(NC(c2cnc(SC)nc2)=O)CC2CN(C(c3nc(C4CC4)cs3)=O)CC2C1 C1(C(=O)NCC(C(C)O)C)CN(C(=O)CC2CNC(=O)O2)CCO1 c1(C(=O)NC2(C3N(C(C4COC(=O)O4)=O)CCC3)CC2)cnc2ccoc2c1 c1(N2CC(C)C=C(C)C2)nc(N(C)Cc2ncc(Br)cn2)nc2c1ncn2C(C)C c1(C(=O)NCC2CCN(C(c3cn(C)nc3)=O)CC2)cnc2ccccn12 C(=O)(C(O)C(C)(C)C)N1CCC(CN(C(CC(C)O)=O)C)C1 N1(C(CS(CC)=O)=O)CC(CNC(c2ccc(OC)c(OC)c2)=O)C(C)(C)C1 c1(C(=O)NCC(CN(C(C(C2CCOC2)OC)=O)C)C)cc2c(F)cccc2s1 C1(C(=O)NC2(CN(C(COCC=C)=O)C)CC2)CC(=O)NC(CC)C1 N1(S(C)(=O)=O)CCC(CC(=O)OC(C(F)(F)F)C2CC2(C)C)CC1 C(=O)(C(C)CC(C)(C)C)N1CCN(C(C(C)N(C)C)=O)CC1C1CCC1 C1(CC(=O)NC2(C(N3CC(O)C(O)C3)=O)C(C)C2)CC2(CCC2)C1 C1(C(F)F)CC(NCCc2ccsc2Cl)CO1 N1(C(CCC=CCC=C)=O)CCCC(CNC(=O)CCNC(=O)NC)C1 C1(CNC(=O)COCCCF)(CNC(C2CCCCO2)=O)CC12CCC2 N1(C(C#CCNC(c2cccc(O)n2)=O)=O)CCC2(CCCCC2)C1 c1(C(=O)NC2C(CNC(CC(=O)OC)=O)CC2)ccc(SC)c([N+](=O)[O-])c1 C1(C)(CNC2(C(N)=O)CCCCC2)CCN(c2ccc(C(C)C)nn2)CC1 CCC(C(=O)NCCOCC(=O)NC1CCn2cncc2C1)C(F)(F)F N1(C(C2CCN(C)C2)=O)C2CC1CN(C(c1cncc(C3CC3)c1)=O)C2 C(CCC)(C(=O)N1CCC(C(=O)N(CCC(=O)OC)C)C1)=CCC c1(CCC)nc(C)c(C(N2CCC(C)(NC(=O)C(O)CSC)C2)=O)s1 C#Cc1cccc(CCNC(=O)C(C)(C)NC(c2ccccn2)=O)c1 c1(C(N2C(CCNC(CC3CC(OC)C3(C)C)=O)CCC2)=O)ccc(N)c(Cl)n1 N1(C(c2ccc(OC)s2)=O)CC2CN(C(=O)C(C)Cc3ccc(Cl)cc3)CC2C1 c1(N(C2CCN(C(Cc3cncc(C)c3)=O)C2)C)nn2cc(C)nc2s1 Cc1nnc(NCCN(C(=O)C=C2CCC(C(C)(C)C)CC2)C)c(C#N)c1C N1(C(C(CC)C#N)=O)CCC2(CC1)COC(CNC(=O)CCc1cc(C)on1)C2 N1(C(C(C)C2CC2)=O)CCCC(CCn2cc(N)cn2)CC1.n12cc(nn1)C2 C1(N(C(=O)Cc2nc(Cl)cs2)CC2CC2)CCCN(C(=O)COCC(F)(F)F)C1 CCCCC(CO)NC(C1(NC(=O)CC2CSCCO2)CC(F)C1)=O C#CCC(CC(F)F)NC(C1(C(C)C)CCN(C(c2cc(CO)ccn2)=O)C1)=O C(=O)(C1=CC2(CCOC2)C1)NC1(C2CCN(C(C3(C(C)C)COC3)=O)C2)CC1 CC(C(=O)NC(C)(C)CCCNC(c1cc2c[nH]cnc-2n1)=O)C(C)C(C)(C)C C1(C(=O)NC2CCN(C(CCc3ccn(C)c3)=O)C2)CC(C)(C)OC1(C)C c1(NCC23C(CN(C(c4cc5ncccn5n4)=O)C2)C3)ccc(Br)cc1[N+](=O)[O-] c1(C(=O)NC2(CCOC)CCN(C(C3CC(=O)N3)=O)C2)ccc2[nH]ccc2n1 C(=O)(C#CC(C)(C)O)NCCCN(C(=O)CCNC(=O)C=C(C)C(C)(C)C)CC N1(CCC(N2C(CCNC(C3(C)CCCC3)=O)CCC2)=O)CCCCCC1 C1(C(=O)NC2(C3CCCN3C(=O)C(F)n3cccn3)CC2)CC12CCCC2 C1(C(=O)NC2C(c3n(C)ncc3)C2)CN(C(C2CC3CCC2CC3)=O)CC12CC2 C1(C(NC[Si](C)(C)C)=O)CN(C(c2ccc(CN3CCCC3)o2)=O)CCO1 CCCC(C(O)C(=O)N(CC(c1nn[nH]n1)C)C)NC(=O)C(CC(C)C)OC C1(C(=O)NCC#CC(=O)OC)CCCN(C(C2C=CCC2)=O)C1 N1(C(=O)CSc2ccncc2)CC(C2CN(C(C3CC4(CCC4)C3)=O)C2)C1 O=C1CCC(N2CCC(CC(N3CCC(C(=O)O)CC3)=O)C2)CN1 CC1C2CC(C2NC(=O)CCn2cncn2)N1C(=O)C(C)S(C)(=O)=O C1(C(=O)NCC(C)CN(C)C(c2cc(F)cc(Cl)c2O)=O)CCC2(CCC2)CC1 C1(C(=O)OC(c2cc(C(F)(F)F)no2)C)CC2(CCC(=O)CC2)C1 CC1CN(C(C2CCC(=O)N(C3CC3)C2)=O)CCC1NC(C1CCS(=O)(=O)C1)=O C1(=O)C(C(C)C)N1.c1(CC(=O)NC(CCN(CC)CC)C)nccn1C CC1CN(C(c2cc3sccc3s2)=O)CCN1C(c1n[nH]cc1C1CC1)=O C1(C(=O)NCc2snc(CC)n2)CC(NC(c2ncccn2)=O)C1(C)C C(=O)(C1=C2CCN=C2NC=C1)NCC1CN(C(c2c(C)c(CO)ccc2)=O)C1 CCCCCC(O)C(=O)NCCCCCC1CCN(C(=O)C=C(C)Cl)CC1 c1(C(N2CCC(CNC(c3ccc(CC)s3)=O)C2)=O)cc(Cl)n(C)n1 c1(SC)nc(=NC23CCCC2CN(C(c2cn4cc(Cl)cnc4n2)=O)C3)s[nH]1 c1(NC(c2n(C)ncc2)=O)sc2c(c1C(=O)NC1CCCCC1(F)F)CCCC2 C#CCCCCCC(=O)N(CC(C)(C)CNC(=O)CC1CCCNC1=O)CC c1(C(=O)OC)cccc(C(N2CCC(C(C)O)C2)C(=O)NCCCN(C)C)c1F C1(C(=O)NCCCCN(CC)CC)CCCCN1C(C1CCC1(C)C)=O N1(C(=O)NCCCNC(C)=O)CCC(c2nc(C(F)(F)F)cs2)CC1 C1(NC(c2c(C(C)C)onc2)=O)CCCC(NC(c2occc2F)=O)C1 c1(OCC)cc2c(cc1F)N(C(=O)NCCC1=CCN(C)CC1)CCC2 CCC(CC)CC(F)C(=O)NCCC(CNC(=O)CCc1cccnc1F)OC C(C(C)C(=O)NCC(C)CNC(=O)CNC(C1CCCC1)=O)SC C(=O)(CCC(CC)NC(=O)CCc1cncs1)N(CC(=O)NCC)CC C1(C(=O)NCCCCCNC(CC=CCC)=O)Cc2cccnc2C1 c1(C(=O)NCC2N(C(C(C3CC3)SC)=O)CCC2)n[nH]c(C)c1O c1(CC(=O)NC2CC(CC(N3CC(CC(C#C)C)C3)=O)C2)nonc1C C#CC1(C(=O)N(C)CC2CC23CC3)CN(C(=O)NC)C1 Cc1nn(C)c(CNc2cc(OCC(=O)O)cc(F)c2)c1I C1(CCO)CCN(N2CCC34CCCC3(C2)C4(F)F)C1 N1(C(c2cc[nH]c2C2CC2)=O)CC2CCN(C(c3n[nH]c4c3COCC4)=O)C2C1 N1(C(c2c(C)cc[nH]2)=O)CCC(CN(C(C2CC2C(F)F)=O)C2CC2)CC1 c1(C(=O)OC)conc1CSC1CN(C(=O)NC(C)C)C1 c1(C(N2CC(NC(CCCCC#C)=O)C(O)C2)=O)cc2sc(Cl)cc2[nH]1 C(=O)(CC(O)CC(C)(C)C)NCC(CN(C(=O)COC(=O)C1CC1)CC)(C)C C1(CCNC(CSc2nc(C)[nH]n2)=O)CSCCN1C(=O)CN(C)C(N)=O C(=O)(CCCCC(=O)NC(C(=O)NC(C)(C)CCN(C)C)C1CCOC1)OC c1(C(=O)NCC(C)(CO)NC(C(c2cnn(C)c2)C)=O)cc2c(s1)CCC2 N1(C(C(C)(F)F)=O)CCN(Cc2cccn3ccnc23)C(CO)C1 C(CN=c1[nH]c(N2CCC(N=S(C)(C)=O)C2)nc2c1CSC2)N(C(C)C)C C1(NC(CC=CC=C)=O)CCOC(C(=O)NC2(C(N)=O)CC(C)C2)C1 n1(CC)cnc2c(NCCC3CC(C)(C)C3)[nH]c(=NCCC(C)S(C)=O)nc12 C1(NC(Cc2cccc(OC)c2F)=O)COC2(C1)CN(C(c1cccnn1)=O)C2 CCCCC(O)C(C)C(=O)NC(C1CC=CCC1)C(N1CCC(C)(F)CC1)=O C1(NC(=O)COc2cn[nH]c2)CCCN(C(c2cccc(C(F)(F)F)c2)=O)C1 c1(C(C(=O)NCCCCCC)N(CC(C)(C)OC)C)cnc(C)cn1 C1(NC(CC2(C)CCC2)=O)CCN(C(=O)C(F)(F)C(O)C2CC2)CC1O C(=O)(C(CN=c1ccc(S(C)(=O)=O)c(C)[nH]1)C1CC2(CCC2)C1)OC N1(C(C(C(C)C)O)=O)CCN(C(c2cccc(CCO)c2)=O)C(C#N)C1 C(=O)(C(CC(C)C)NC(c1cn(CCNC(=O)CCC2CC(C)C2)cn1)=O)NC CC(CC1=CCCCC1)NC(C1(NC(=O)CN2CCCC2)CC(F)C1)=O C1(C(=O)NCCCSCC)CN(C(c2ccnc(CC)c2)=O)CC1F CC(C(F)(F)C(F)(F)F)=CC(=O)NC(C)(C)C(C)NC(=O)C=CC1CCC1 c1(CN=C(NCC)NCC2(CO)COCC3CCCN23)cnc2c(F)cccc2c1 N1(C(c2cc(Cl)c(Cl)s2)=O)CCN(C(=O)COC(F)F)C(c2ccncc2)C1 CC1CC(=O)NCC1C(=O)NCC(C)(C)C(=O)NCC1C2CCCOC12 c1(C(N2C(=O)NC(C(C)C)C2=O)C)cc2ccccc2o1 C#Cc1ncc[nH]c1=NNC(=O)c1csc(-c2ccccc2F)n1 CC1CC(CC(N2CC(F)(CNC(=O)Cc3ccccc3F)C2)=O)CC(C)(C)C1 C=CC(C)(CC)C(=O)NCC1CCC1NC(c1c(OC)noc1C)=O Cc1ccc(C=CC(=O)NCCCCC(=O)NC2CCCC2CO)o1 c1(C(=O)NCC2(O)CC(C(=O)NCCC3CCCOC3)C2)cccc2occc12 c1(OC)ccnc(C(=O)NCC(C)(C)NC(c2n[nH]c(C)c2O)=O)c1F C1(NC(CN(C(C)C)C)=O)CC2CC(NC(C3CN(C4CCC4)C3)=O)CC12 c1(CCC(=O)NCC2N(C(C3CCC(C)O3)=O)C3C(C2)C3)ccc(Cl)cc1F N1(C(C2CCOC2)=O)CCCC2CN(C(C3(n4cccn4)CCC3)=O)CCC12 Cn1cc(C(=O)NC2CC(n3cc(CCCCCC(=O)O)nn3)C2)cc1C#N C1(CNC(COCCSC)=O)CC12CCN(C(=O)C(C)CC(F)F)CC2 CC1(C)c2[nH][nH]c(=NC(=O)c3cn[nH]c3)c2CN1Cc1ccnc(F)c1Cl c1(C(N2C(C(N3CC(C)(CC)C3)=O)CSC2)=O)cccc(F)c1 N1(C(C2N(C(CC(C)SC)=O)CCC=C2)=O)CC(O)C(O)C1CO C1(C)(NC(c2cccc(C)n2)=O)CCCN(C(=O)COc2cccc(Cl)c2)C1 C1(NC(C2(C#C)CCCC2)=O)CN(C(=O)CC(=C)C)C(CC)(CC)C1 C12(C(N(C)Cc3nncs3)=O)CCCC1N(C(=O)CCCn1cccc1)CC2 CCCCC(CNC(c1ccnc(C)c1)=O)NC(c1cc(Br)sc1C)=O N1(C(c2nc(C(C)OC)oc2)=O)CCCC2C1CCN2C(=O)CCCS(N)(=O)=O c1(C(N2C3C(NC(C4CCCOC4)=O)C(CC3O)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 c1(C(=O)NC(C2(O)CN(C(C3C(C=C)OCC3)=O)C2)C)[nH]c2ccccc2c1C C1(NC(=O)CC=CCNC(=O)CC2CCC(=O)N2)CCc2nncn2C1 N1(C(C(=O)NCCOCC)C2CC2C)CCCC1c1ccsc1 C1(NC(c2n(CC)ccn2)=O)CCN(C(c2cc(C(F)(F)F)nn2C)=O)C(C)C1 C1(C(C)C)(CNC(C2CC2OC(C)(C)C)=O)CC1 c1(C(=O)NCC23N(C(c4ccc(C)c(C)n4)=O)CC(C2)C3)c(C)nc2sccn12 N1(C(c2nccc(C#C)c2)=O)C2CCC1CC(C(=O)NCC1CCCCC1C)C2 c1(OC)cccc(C)c1C(N1CC2CC1CC2NC(c1ccns1)=O)=O C1(C(N2CC(CCNC(c3ccc(CO)s3)=O)C2)=O)CCCC1C1CC1 c1(C(=O)NCc2c(Cn3cc(CSC)nn3)nco2)cc2cnn(C)c2s1 c1(C(=O)NCC2(CNC(C3C(C)CC(=O)N3)=O)CCCC2)cnn2c1N(C)CC2 CCCS(=O)(=O)CC(=O)NC1CC(F)(CNC(c2ncccc2OC)=O)C1 CC(C)CC(C(=O)N1CC2CCN(C(c3coc(C(F)(F)F)c3)=O)C2C1)C(C)C N1(C(C=CC(=O)OCC)=O)CC2(CCC(NC(c3nn(C)c4c3CCC4)=O)C2)C1 N1(C(Cc2c(C)n[nH]c2)=O)CC(F)CC1CNC(=O)CC1CCOC1=O N1(C(CN(C)C(=O)OC)=O)C(CC(N2CC(Cc3ccco3)C2)=O)C2CCCC12 C1(C(C)(C)NC(C2CCCC2O)=O)CCN(C(c2c[nH]c(C(N)=O)c2)=O)CC1 C1(C(=O)NC2(CCCNC(c3cn(C(C)C)nn3)=O)CC2)CC(C)CC(=O)N1 N1(C(c2c(C)csc2)=O)CC2(CC(C(=O)NC34CC(F)(C3)C4)CO2)C1 CCC(C)CCCC(=O)NCC(O)CCNC(c1cscc1C#N)=O c1(C(N2C(CNC(C(C=C)(C)C)=O)C(C)CC2)=O)cnc(C)[nH]c1=N N1(c2ccc(S(=O)(=O)NC(CCSC)C)cc2F)CCCC2(CCC(=O)NC2)C1 CCCC(CC(C)C)C(=O)NC1CCN(C(c2ccc(N3CCCC3)cc2)=O)C1 N1(C(C(C(C)(C)C)c2cccc(C)c2)=O)CC2C(C1)C(F)(F)C2(F)F C1(C(N(CC(C)N(C)C(c2cc(C3CCC3)no2)=O)C)=O)CN2CCCN1CC2 N1(C(C(C)=C2CC2)=O)CC(C)CN(C(c2cnc3n2CCCC3)=O)C(C)C1 c1(CCCC(=O)NC(c2ccc(C)cc2)COC)ccc(Cl)cc1 Cc1ccc(C(=O)Nc2ccc3c(c2)CN(C(C2CCCS2)=O)C3)c([N+](=O)[O-])c1 Cc1ccc(NC(=O)C(C)CN(C)C(c2n[nH]c3c2COC3)=O)cc1C C1(S(C)(=O)=O)(C(N(CC(CNC(Cc2c(C)ocn2)=O)O)C)=O)CC1 C(C(N=[N+]=[N-])C(=O)NCC1(OC)CN(C(=O)C(C)C(=O)OC)C1)OCC N1(C(C2N(C(c3cc(OC)no3)=O)CC2)=O)CCCC(C(N)=O)C1 N1(C(C=C(CCC)C)=O)CCC2(CC1)COC(CNC(=O)CN(C1CCC1)C)C2 C1(C(=O)NCCC(=O)NC(C)(C)C)CCCN1C(C1CCCN1C(N)=O)=O C1(Cn2cc(-c3c(C(C)C)n[nH]c3)nn2)CCN(C(C2(F)CCOC2)=O)C1(C)C c1(C(=O)OCCC2CCN(C(=O)OC(C)(C)C)C2)cnc(N)c(Br)c1 N1(C(CN(CCOC)C(C2CCSC2)=O)=O)CCCC(CCF)C1 CC1(C)CCc2c1n[nH]c2C(=O)NCC1(F)CN(C(C2CCCCC(=O)N2)=O)C1 N1(C(Cc2ccc(C)nc2)=O)CCN(C(=O)CCCCC2CC2)C2CCCCC12 C#Cc1cccc(CC(N2CC(NC(=O)C=CC(C)C)CC2(C)CC)=O)c1 N1(C(CCC2C(C)C2)=O)CC(C)CN(C(c2ccccc2SCCO)=O)CC1C c1(C(=O)OC)ccncc1NC(=O)CC1CCCN1C(c1cc(Br)ccn1)=O C(c1cscn1)=CC(=O)NC1CC(CNC(C2OCCCO2)=O)C1 C1(NCc2c(COC)occ2)CC(N(C)C)C1(C)C O=C(CCCCC(F)F)N1CCC2CN(C(=O)C(F)C(F)(F)F)C2C1 N1(C(CSCCOC)=O)CC(NC(=O)CCc2nc(C)c(C)[nH]2)C(C2CC2)C1 c1(NC(C(C)(C)CCNC(C23COCC2C3)=O)=O)cnc2ncnn2c1 c1(C(N2CC(NC(C(C)S(N)(=O)=O)=O)C(O)C2)=O)cc2c(cc1Cl)OCO2 Cn1ncc(C(N2CCC(CCNC(C3(C)CCCCC3)=O)C2)=O)c1C(C)(F)F c1(C(=O)NCC2CC(NC(C3CN(CC)C(=O)CC3)=O)C2)cc(Cl)c(F)cc1C C1(C(=O)NC2C(NC(c3c(C)ncn3O)=O)COCC2)CCc2ccnn2C1 c1(C(=O)NCC2CN(C(=O)CO)CCO2)ccc(S(=O)(=O)NCC2CCCO2)cc1 C(C(C(=O)NC(C1CCCCO1)(C)C)NC(C1CCCC1O)=O)N(C)C N1(C(C(C)OCC=C)=O)CC2CC(NC(=O)CCCCC(C)C)CC(C2)C1 c1(CNC(CC(C)NC(C2CC2C(=O)N(C)C)C)=O)cnc(C)cn1 C1(C(N2CCC(C)(F)CC2)=O)CCCN1NC(=O)Cn1cc(CO)nn1 Cc1onc(CO)c1C(N1CCN(C2CCC(NC(=O)CCS(C)=O)C2)CC1)=O c1(C(N(C2CN(C(c3c(C(C)C)c[nH]n3)=O)C2)C)=O)cccc2ncccc12 c1(CNC(C2(NC(Cc3cc(C)sc3)=O)CC2)=O)cncc(O)c1 NS(=O)(=O)N1CCCC(C(=O)NC23CCCC2CN(C(C2CCCCC2)=O)C3)C1 c1(CN2C(CNC(C(c3ccccc3)C)=O)CCC2)c(I)ccnc1O C(C)(C(C)(C)C)=CC(N1CC(OCCNC(C=CC(CC)C)=O)C1)=O c1(CCOC(C(CCC)OC)=O)cc(F)ccc1F c1(OCC)ccc(C(=O)NC2CCCN(C)C2)cc1[N+](=O)[O-] c1(CN(C)C(C2(N(C(=O)CCc3nc[nH]n3)C)CCC2)=O)nnc(O)o1 C1(N(CC(=O)N(C2CCCC2)CCC#N)CCO)CC(O)(CSc2ccccc2)C1 c1(C(N(C(CNC(C2(C(=O)NC)CC2)=O)C)C)=O)cc(C(F)F)ccn1 Cc1sccc1C(=O)NCC(CO)NC(=O)Cn1ccnc1C c1(NC(C2CCC(C3CC3)N2)=O)c(Cl)c(Cl)cc(Cl)c1Cl C(=O)(C(C)(C)C(=O)NCC1CC1CNC(=O)CN1CCS(=O)CC1)NC c1(C(N2C(CNC(CCc3c(C)n(C)nc3)=O)CC2)=O)[nH]nc([N+](=O)[O-])c1Cl C(CNC(=O)CC1(c2ccccc2)CC1)(CC(C)C)NC(CC=CC=C)=O c1(C(N2CCN(CC3CN(C(C(C=CC)O)=O)C3)CC2)=O)c(C)ccnc1N c1(C(N2CCCC(C(C)NC(c3ccc(C)o3)=O)C2)=O)cn(C)c(=O)c(C)n1 c1(C(N(C)CC2CCCCN2C(C2CCC2(C)C)=O)=O)ccc2[nH]c(=N)sc2c1 c1(CC(=O)NC(C)(C)COCCCNC(c2ccoc2)=O)cccc(F)c1Cl c1(C(=O)NCC2CCN(C(C(C(C)C)NC=O)=O)C2)ccc2c(c1)OCCO2 c1(C(N2CCC(CNC(c3ccc(C)s3)=O)C2(C)C)=O)cccc2scnc12 C1(O)(C(C)NC(C(CC)N(C)CC)=O)CCN(C(C2(CO)CCC2)=O)C1 C1(NC(c2c(C)ccs2)=O)CC(C)CN(C(c2ccc(C(C)C)s2)=O)C1 C(CCOCC(C)C)(C(=O)NC(C)(C)CO)NC(COC(C)=O)=O.C(C)C c1(CNC(c2n(C(C)(C)C)nnn2)c2nc(Cl)cs2)cc(O)nc2ccccc12 C(=O)(CC(C)C(=O)NC1CC2(C1)CN(C(=O)C(C1CCCCC1)C)C2)OCC N1(C(C2(CNC(C(C=CC)O)=O)CC3(CC3)C2)=O)CC2CCC2(OC)C1 c1(C(N2CC(CC=C)(C(N3CCC3CC(C)(C)C)=O)C2)=O)ccc2cncn2c1 C1(CC(=O)NC2CC(N(C(CCSCCCC)=O)C)C2)COCC(C)(C)O1 C#Cc1ccc(C(N2CCN(C(C3CCC(=O)N3C3CC3)=O)C(CC)C2)=O)cc1 C1(C(N2CC3(CC(CNC(COC(CC)(C)C)=O)C3)C2)=O)OC(C)(C)OC1(C)C N1(CC(=O)NCC2N(C(c3cnc(C(C)C)s3)=O)CCC2)CCC(C)(C)C1 c1(C(N2C(C(C)(C)NC(C3CC4CC4C3)=O)CCC2)=O)cnc2[nH]cncc1-2 c1(OC)ccnc(F)c1C(=O)NCC1CC1NC(=O)Cc1ccncc1 S(=O)(=O)(CCC(=O)NC1CS(=O)(=O)CC1NC(=O)C1=CCCC1)NC C(=O)(CCCCC(N)=O)NC1CC(CCC(=O)NC(CC)C(C)O)C1 C1(C(=O)NC(c2cnnn2C)C)CCc2nnc(Br)n2C1 N1(Cc2nc(-c3ccc(F)cc3)on2)CCc2ccc(Cl)cc21 c1(CCOC(CNC(C2C(CCC)C2)=O)(C)C)ccc(SC)cc1.C(C)=O CC(=O)CCCC(=O)NCC(C)N(C(=O)C(Cc1ccccc1)n1cnnn1)C C1(CNC(C2CCCN2C2CC2)=O)CCCN1C(=O)CC(O)C1CCCC1 c1(C(=O)NCC(=O)NCC=C)ccnn(C)c1=O CC1(C)CC(CC(N2CC=CCC2)=O)N(C(=O)C#CC2CC2)C1 c1(OC(C)C(N2CC(C)(NC(=O)C(F)(F)CC3CCCO3)C2)=O)ccc(Cl)cc1 N1(C(c2ccc3c[nH]nc3c2)=O)CCC2CCCN(c3cc(F)ncn3)C2C1 C(=O)(C(C)(CCC)CCC)N1CC(NC(c2n(CCC)nnc2)=O)C(CO)CC1 C(=O)(C1CCCn2cnnc21)OC(C)(C)C.N12CCN(CC1)C(=O)N(C)CC2 CC(C)CC(C(=O)N(C)CC1CCCN1C(=O)Cc1c(F)cccc1Cl)C(C)C N1(C(C(CCC)N(C)C)=O)CC(N=[N+]=[N-])CC1C(N1CC2(CC2)C1)=O c1(OC)ccc(C(=O)N(C(C)CN(C(=O)CCCc2cc(C)no2)C)C)cc1 c1(C(=O)NCC2(CNC(C3(CF)CC3(F)F)=O)CC2)cc2n(c1)CCOC2 C1(CC(=O)NC2(CNC(=O)C(O)C3CC3)CCCC2)COCCO1 c1(OC)ccc(S(=O)(=O)CCC(=O)N2CC3C(NC(=O)C(C)C(C)O)C3C2)cc1 CC(=O)NNC(=O)C(C)NCC1CNC(C)C1 C(C)(CNC(=O)CCSc1ccc(F)cc1)(CC(C)C)Nc1ncc(C)cn1 C(=O)(C(F)CC(C)(C)NC(=O)C(C1CCOCC1)F)N(C)CCn1ccnc1 N1(C(C(F)(F)C2(OC)CCC2)=O)CC2(CNC(=O)CC3(C)CCCC3)CC1CO2 c1(C(=O)NC2CC(NC(C=CC)=O)C23CCC3)occ2c1CCCC2 C(CN=c1[nH]ccc(=NC2CC3(CCC3)C2)[nH]1)c1c(C)[nH]c2ccc(F)cc21 c1(NC(c2cn(C(C)CCOC)nn2)c2ccccn2)cc(C#N)no1 C1(C(N2C(C(C)O)CC2)=O)CCN(C(=O)CN(CC(C)(C)C)C)CC1O C12(CNC(c3c(CCC)occ3)=O)CC(CN1C(C1CC3CC3C1)=O)C2 N#Cc1cncnc1C(=O)NCCOCCNC(c1cccc(=O)o1)=O C(=O)(N(CCC(=O)OC)OC)C1N(C(=O)C(=O)NOC)CCC(=C)C1 c1(CC)cc2c(CC(=O)NCC3CCC(NC(=O)C(Cl)=CCl)C3)csc2s1 N1(C(CCC#C)=O)CCCN(C(=O)CC2CCCN2CC)C(C(C)C)C1 O=C(C1CCc2c[nH]nc21)NCC1CCCCN(C(=O)C2CCc3c[nH]nc32)C1 CC1CCc2ncc(C(=O)NCC3C4CN(C(=O)CCc5cn[nH]c5)CC34)n2C1 C1(NC(C2C(C)CC(C)O2)=O)CCN(C(c2ccc(O)c(F)c2F)=O)CC1(C)C c1(CN(C(=O)Cc2c[nH]nc2O)C)ccccc1CNC(c1ccoc1)=O Cc1cc(C(=O)N(CC(=O)NC2CCCC(N(C)C)C2)C2CC2)nc(C)c1 c1(C(=O)NCC(C)(C2CC2)NC(CCOC)=O)ccc(C)c(OC(F)F)c1 CC1COC(C(=O)NCC(C)CN(C)C(c2cnn(Cc3ccccc3)c2)=O)C1 C(=O)(N(CCC(=O)NOC(C)C(=O)OC)OC)C1C(CCC)CCC1 c1(OC)cccc(O)c1CN(C)CC1CCCN(C(=O)C=CC(C)C)C1 C1(NC(CCN(C)CC)=O)CC2CN(C(C3(C4CC4)CC3)=O)CCN2C1=O c1(CC(=O)N(CCN(C(C2CC2F)=O)CC)CC)ccsc1Br C1(CC)CN(C(=O)C=C2CCC2)CCC1NC(=O)CC1(c2cccc(Cl)c2)CC1 N1(C(c2c(C)cc[nH]2)=O)CC2(NC(=O)C(C)Cc3ccccc3Cl)CC1C2 Cc1cc(CC(=O)NC2CC2CNC(=O)CN(C)C2CC2)nn1C C1(NC(CSc2cc(C)on2)=O)CS(=O)(=O)CC1NC(=O)CSc1nccn1C C(=O)(C(O)CC(N)=O)N1CC(C(C)NC(=O)Cn2ccc(C3CC3)n2)C1 C(=O)(CC(C)(C)N(C)C)NC1(CC=C)CN(C(c2ccc(SC)o2)=O)C1 c1(NC(C2(c3cccc(Br)c3)CCC2)=O)ccc(Cl)cc1C(=O)C1CC1 N1(C(C(C(C)C)NC(CCCC#C)=O)=O)CCC(NC(C)=O)C(C(N)=O)C1 C1(CC(=O)N(C(C)C)CCNC(=O)CCC2CCCN(C)C2)OCCCC1(C)C C12CC3CCC(C1)N3C2=O.C(=O)(CC(C)(C)Cc1ccccc1)NC(C)C N1(C(CC(=C)C)=O)CCC2CCN(C(c3cc(C)nc(O)n3)=O)CC12 c1(OC)ccccc1C1(C(N2CCOC(C(O)CO)C2)=O)CCC1 C(c1cn(C)nn1)=CC(=O)NCC(C)N(C(C1N(CC)CC1)=O)CC C1(C(NOCC=C)=O)CC12CCN(C(=O)C(C)(C)CC(F)F)CC2 CCCC(F)(F)C(=O)NC1CC(C)CN(C(c2ccncc2NC)=O)C1 C(=O)(N=c1cc(Cl)cn[nH]1)C1CCCC(NC(c2cncc(OCC)c2)=O)C1 C1(C(=O)NCC(CC=C)NC(=O)CSc2nncn2CC)CCN(C(C)C)CC1 N1(CCCNC(C2C(C)(C)CC(F)(F)CC2)=O)C(=O)C2C3C=CC(C3)C2C1=O C(C(CNC(C1CN(C2COC2)C1)=O)C(F)(F)F)NC(CN1CCN(C)CC1)=O CC1(CC(=O)NC2CC(NC(C3C=CCC3)=O)C2)CCS(=O)(=O)N1 c1(-c2cc(C(=O)NC(C(C)NC(=O)Cc3ccco3)C)no2)ccccc1O Cn1nncc1C(=O)NCCOC1CCN(C(=O)CCNC(N)=O)C1 c1(OC)c(C(=O)NC(CNC(C2CC(=O)NC2(C)C)=O)C2CCC2)c(C)nn1C N1(C(C2CCC(=C)CC2)=O)CC2(COC(CNC(c3ccccc3)=O)C2)C1 C=CCCC(C)(O)c1nc(-c2ccccc2)nn1C12CC(C(F)F)(C1)C2 N1(C(CC2(COC)CC2)=O)CCC(C)C(NC(C23CCCN(CC2)C3)=O)C1C N1(C(c2ccc(C#N)o2)=O)Cc2occ(C(=O)NC3CCC(CO)C3)c2C1 c1(CC)nc(C)c(C(N2CCN(CCN(C(=O)C#CC(C)C)C)CC2)=O)s1 N1(C(c2nc(C)nn2C)=O)CCC2(CC1)CN(C(=O)C(=O)NC(C)C)C2C(C)C C(=O)(C1=NOC2COCC12)NCC1N(C(Cc2c(F)ccc(OC)c2)=O)CC1 C(CCCC(C)(C)C(=O)NNC(=O)CNc1cccc(F)c1)NC(CC=C)=O c1(OCC(C)(C)C(=O)NCCCCCCOCCCC(=O)O)ccc(F)cc1F C12(CNC(c3c(C)scc3)=O)CN(C(c3cc(F)c[nH]3)=O)CC1(C(F)(F)F)C2 N1(C(C2(NC(CC(=O)NCC#C)=O)CCOCC2)=O)CC(CO)OC(C)C1 N1(C(C(C)OC2CCOCC2)=O)CC(O)CC1CN(C)CCN(C)C n1(CCCNC(=O)Nc2ccc(N(C(C)=O)CC)cc2)cc(C#N)c(O)nc1=O N1(C(C2(OC)CCOC2)=O)C(C(N2CCC(N3CC(O)C3)C2)=O)C2CC(O)C1C2 C1(CC(=O)N(CC(=O)OCC)C(C)C)CC(C)N(C(c2ccc(C(C)=O)o2)=O)C1 C1(C(N2CC(F)CC2CNC(C2(C3CC3)CC2)=O)=O)CC2(CCOC2)C1 C#Cc1ccc(NC(=O)CC(O)CNC(c2occc2COC)=O)c(C)c1 Cc1cccc(C(N2CC(CCNC(C3CCCN3C(C)C)=O)C(C)C2)=O)c1C C1(CC=C)(NC(C2CCOCC2)=O)CC2CCC(C1)N2C(C1(C)CCCO1)=O Cc1cnc(N2CCCC(CC(=O)NCC3CCN(C)C3=O)C2)nc1C C(=O)(CC1=CCCCC1)NCC1CC(NC(C(c2c(OC)cccc2)(F)F)=O)C1 N1(C(C)=O)CCCC1(C)C(N1CC2CC2(NC(=O)C(F)=C(C)C)C1)=O CCC(CC)CC(=O)NC(C1CCN(C(C2(CC)CCCC2)=O)CC1)C Cc1cc(C(=O)NC(C2CN(C(C3(c4ccno4)CC3)=O)CCO2)C)nc(O)c1 Cn1c(C(=O)N(C2(C(=O)NCCC3NC(=O)NC3=O)CCC2)C2CC2)nnc1S N1(C(C2CCC(CNC(c3c(C(C)C)n[nH]c3)=O)C2)=O)CCC2(CCN(C)C2)C1 c1(C(=O)NC(C(C)NC(Cc2ccc(C(C)=O)s2)=O)C)ccc(F)c(F)c1N N1(C(C(C)C2CCCO2)=O)CCC(NC(=O)Cc2cnc(C(F)(F)F)s2)CC1C C1(C2CCOCC2)(C(=O)NC2CN(C(C=C(C)C3CC3)=O)CC3C2C3)CC1(F)F N1(C(Cn2c(C)ncc2)=O)CCC(F)(F)C(NCc2cc(I)ccc2O)C1 c1(OCCC)cccnc1C(N1CCC1CNC(=O)Cc1ccccc1F)=O C(CCC(=O)NCc1ccc(C(=O)NCCCCCSC)o1)=CCC=C Cc1nc(C(N2CCC(CN(C)C(C34CCN(CC3)C4)=O)C2)=O)ccc1[N+](=O)[O-] c1(OC)cnc(C(N2CC(CCNC(C3(C)CCNC3=O)=O)C2)=O)c(OC)n1 N1(C(C(C)SCCCC)=O)CCN(C(=O)C(c2ccc(F)c(F)c2)C)C(C)C1 C(C(F)(F)CCC(=O)NCC(c1ccccn1)C)n1cc(C(=O)OCC)nn1 c1(C(=O)NCC23N(C(CC4CC(=C)C4)=O)CCC2CC3)cccc2nncn12 Cc1cccc(C)c1C1(C(=O)NC(C)CCNC(=O)CC2CCCCO2)CC1 N1(C(CN(C(C)C)C)=O)CCCC2(C1)CN(C(C1CCCSC1)=O)CCO2 Cn1ccc2nc(N3CC4CC3CN4c3ncnc4[nH]ccc34)nc(Cl)c12 N1(C(CC2(OCC)CC2)=O)CCCC(NC(C2CCC(C)(C)OC2)=O)CC1 CC1CN(C(c2cc3ccccc3[nH]2)=O)CCCN1C(=O)CC(C)(C)Cl C1(CNC(c2occ(C)c2)=O)CN(C(=O)C(F)(F)c2ncccn2)CC1(C)C C1(N(C(=O)C(c2cn(C)nn2)NC(=O)C=Cc2ccsc2)C)CCCC(O)C1 C1(C(=O)NCCOCC)CCN1C(=O)Cc1ccon1 c1(C(N2CCC(NC(COCC(=C)C)=O)C(F)C2)=O)oc2ccc(F)cc2c1C C(=O)(C1=C(C)OCCS1)NCC(CC(=O)NCC(=O)N(C)CC)C C1(O)(CNC(CC2C(C)(C)C(O)C2)=O)CCN(C(=O)CC2CC(C3CC3)C2)CC1 C=CCC(F)(F)C(=O)N1CC(CNC(=O)CCC2CC2(F)F)C(C)C1 C(C1CSc2ccccc21)NC(c1cc(C(C)(C)C)c(O)cc1)=O C12(CC(=O)OC(C(=O)OC)C3CCC3)COCC(C1)C2 c1(OC)ncc(C(=O)NC2(C)CCN(C(=O)C(C)c3cncs3)C2)cn1 N1(C(COc2cc(C)on2)=O)CCC2(CCC2)C(NC(C2CC3C=CC2O3)=O)C1 CC1(C)OCC(C)(CNC(c2ccccc2)C(=O)N2CCCC2)O1 C(=O)(C(CO)C(C)(C)C)NC1C2CC(NC(CCCOCCOC)=O)CC21 c1(CN(CCN(C(=O)CC2(OCC)CCC2)C)CC)cc(-c2ccoc2)nn1C CCC(C)C(O)C(=O)NC1(CC(N2CC(CC(F)(F)F)C2)=O)CC1 C#Cc1ccc(C(N2CCCC2CCC(=O)NCc2conc2C(F)(F)F)=O)o1 c1(C(=O)NCC2CCC(NC(c3c(N)cc(Cl)cc3)=O)C2)cnc2[nH]cnc2c1 c1(N(C2CN(C(C3CC=CCC3)=O)C2)C)ncc2ccc(Br)cc2n1 C1(C(C)(C)NC(c2cc(C)oc2)=O)CN(C(C2(c3ccno3)CC2)=O)CCO1 c1(CC(C(=O)NCCC(C)NC(=O)CC2SC(=N)NC2=O)C)ccc(Cl)cc1 c1(C(=O)OC)ccc(F)cc1CNC(=NCCSC)NCC(C1CCCCC1)C N1(c2[nH]c(=NCC3CCCC3C)cc(C)n2)CCc2c(cnnc2O)C1 c1(C(N2CCC(C)(NC(=O)C3=CCS(=O)(=O)C3)C2)=O)cc2c(o1)CCCNC2=O S(=O)(=O)(c1c(C)nn(C)c1C)N1C2CN(c3ncnc(CC)c3F)C(C2)C1 N1(C(c2c(CNC(C(C)NC(=O)NC)=O)noc2)=O)CCC12CCSCC2 N1(c2nc(=N)nc(N3CCCC(CC(C)C)C3)[nH]2)CC(C)OC(C)(C)C1 C1(C(=O)OC)CCOC1C(=O)NCC=CCC1CN(C(=O)Cc2cncn2C)C1 C(C(CC(C)C)C(=O)NCCc1cc[nH]n1)NC(CCCC)=O C#CCCCC(C)C(=O)N1CC=CC(NC(C2(O)CCCCC2)=O)C1 N1(C(C2(CC)CCNC2=O)=O)CC2CC(NC(=O)C=C(C)C(C)(C)C)C1C2 C(CC(C(=O)NC(C1CCCCC1)CNC(c1n[nH]cc1F)=O)NC(N)=O)SC C1(NC(=O)C=CC=C(Cl)Cl)CC2CC(NC(c3cncc(F)c3Cl)=O)C2C1 N1(C(CC2(C=C)CCC2)=O)CC(C)N(C(=O)Cc2cnn(C(C)C)c2)C(C)C1 C1(CNC(C2(C(C)C)CC2)=O)CC(C(=O)NC(C)Cc2cccs2)=NO1 C1(CN(C(=O)C(C)(C)CN(C)C)CC)CCN(C(=O)C(c2ccn(C)n2)C)CC1 c1(C(=O)NC2CN(C(C=Cc3cnc(C)s3)=O)CC2C)cc([N+](=O)[O-])ccc1C C1(CC(=O)NCCCOCCN(C(=O)CC2CCC2)C)CCc2sccc2C1=O C1(NC(c2c[nH]nc2F)=O)CCN(C(c2ccc(O)cc2Cl)=O)C(C2CC2)C1 C1(C)(CC(=O)N(C)CC2CCCCN2C(C2(CF)CC2)=O)CCS(=O)(=O)N1 c1(OCC)ccc(C(=O)NCCCN(c2cn(C3CCOCC3)nn2)CC)cc1 c1(C(=O)OCC(=O)NCCNC(=O)OC)c(OC)cncc1Br c1(N(CC(c2ccc(OCCC(C)C)cc2)=O)C)nc2ccc(O)cc2s1 C(=O)(C(C)CC(C)C(C)=O)NC1CC(CCC(=O)NC(CC#CC)CO)C1 C(CN=C(NCC(F)F)N1CCC2(CCC(O)CC2)CC1)c1nnc(C(C)C)s1 N1(C(Cn2c(C)nnn2)=O)CCCC(C(C)(C)C(=O)NC(C)CCC(C)C)C1 c1(CCC)nnc(SCCCC(=O)O)n1CCCN N1(C(C(CC)C#N)=O)CCOCC(C)(CNC(=O)Cc2cccc(Cl)c2)C1 C(=O)(C(C)(CSC)NC(=O)C(C)CCOC)NCC(CC)n1cccn1 C1(CNC(c2cc(Cl)no2)=O)CN(C(C2CCC3CCC(=O)N23)=O)CC12CCC2 C1(CN(C(C2C(C(C)NC(c3ccc(O)cn3)=O)C2)=O)C)OCCC1(C)C C1(CNC(c2c(CC)nn[nH]2)=O)CCC(C)N(C(C2CC(C(=O)OC)C2)=O)C1 C1(CNC(=O)CCOCC2CCCO2)C(C2CC2)CCN1C(c1ccccn1)=O C1(CN(CCCC)Cc2cccc(C(=O)Nc3ccncn3)c2)CCS(=O)(=O)C1 CC1CN(C(c2cnc(S)[nH]2)=O)CC1NC(=O)Cn1cc(C(F)(F)F)nn1 C(=O)(C(C)(C)C(C)(F)F)NC1CC2CC(NC(C3CCC(C)CC3)=O)C1C2 C=CCC(C)(C)CC(=O)NC1COC2(CNC(C3CCOC3(C)C)=O)CC1C2 c1(CNC(=O)NC(c2ccc(F)cc2F)CC)ccc2c(c1)ncn2C C(=O)(C(c1ccccc1)=Cc1ccccc1)NC1(CN(C)C(C2CC2Cl)=O)CC1 c1(CC(C)C)nc(C(=O)NCC2(CN3CCOCC3)CCC2)cs1 Cc1ccc(CCCNC(c2n[nH]c3c2CCC3)=O)c(O)c1 C1(C(C(N2C(CN(C(C(C=C)C)=O)C3CC3)CCC2)=O)O)CCCCCC1 c1(NC)snc(C)c1C(=O)NCC1CC(CNC(C2CC3CCC3C2)=O)CO1 c1(C(N2CCC(C(C)NC(C=C(C)C3CC3)=O)C2)=O)ccc2c(c1)OCO2 C12(C(=O)NCC3(C(N)=O)CN(C(C(C(=O)OC)(C)C)=O)C3)CCC(C)(CC1)OC2 C(CCCCCCC(=O)N1CC(CNC(=O)CC2CC(C)C2)C2(CCC2)C1)SC C12(C(=O)NCCCN3CCN(C)CC3)CC(CO1)N(C(c1cnc(O)[nH]1)=O)C2 Cc1cc(C(C)(C)C)cc(C)c1CN1CCC(C(C)N)CC1 C1(=O)C(CC(C)C)ONC(=O)C2CCC(C2)N1.C(=O)(CCC(C)N(C)C)OC C1(C(C)C)CN(C(c2ccc(CNC(=O)C(C)(C)c3ccno3)o2)=O)C1C(C)C C(=O)(C(C(=O)NC1(CNC(=O)C(F)CC(C)C)CCCC1)C(C)C)OCC N1(C(c2c(C)nc[nH]2)=O)CCN(C(c2ccc(Cl)s2)=O)C(CO)C1 N1(C(CCC(=C)Br)=O)CC2CCC(C1)C(NC(=O)C(C(C)(C)C)OC)C2 C1(C#N)(N2CCC(OCC=C)C2)CCCCCCC1 C1(NC(=O)Cc2cncs2)CC2CCC1CC2NC(C1CCc2nc[nH]c2C1)=O c1(C(=O)NC2C(NC(c3cn(CCC(C)C)nn3)=O)CC2)cnc(N(C)C)nc1 c1(OCC)ccc2nc(O)n(C(C3CCOC3)C3CCC3)c(=O)c2c1 C1(C(=O)NCCn2ncc(CC)c2)C=CCN(C(c2cnsc2C)=O)C1 c1(C(N(C)CCN(C(=O)C(C2CCCCC2)F)C)=O)cc(-c2cc[nH]n2)ccn1 N1(C(C2(CC=C)CC2)=O)CCCN(C(c2ccc(F)c(C(=O)CC)c2)=O)C(C)C1 N1(C(C(C(C)(C)C)OC)=O)CC(NC(C2(C3CC3)CC(=O)C2)=O)C(C2CC2)C1 C1(C(N2C(C(C)NC(C=CCCC)=O)CCC2)=O)CCCCCS1(=O)=O c1(CN2CC(NC(c3cccc(OC)c3)=O)(CO)C2)ccc(Br)nc1Br c1(C2CCC(=O)N2)ccc(CCC(N2CCCC2CO)=O)cc1 C12(CNC(Cn3c(C)c(Cl)cn3)=O)CCC1CCN2C(=O)CSCCC#N c1(CC(=O)N(CCCN(CC(COC)O)C)C)nnn(C(C)(C)C)n1 c1(CNC(=O)Cc2cncs2)ncccc1CNC(c1ccnnc1)=O Cc1cc(NC2CCCCCCC2)ncc1S(=O)(=O)N(CCO)Cc1ccsc1 C(C)(C#CC(=O)N=c1cc(C)n(C)[nH]1)NCC(C(CC)CC)OC c1(C(=O)NC(CC)CN(C)C(C2CNC(=O)C2)=O)sc2ncn(C)c(=O)c2c1C [SH](=O)(=O)c1ccc(Br)c(C#N)c1.c1(N2CC(N(C)C3CC3C)C2)ncc(F)cn1 Cc1ccc(C(=O)NCc2csc(CNC(C3COC(=O)O3)=O)n2)c([N+](=O)[O-])c1 CC(C)S(=O)(=O)CCC(N)C(=O)NC1CCCC1c1ccc(Br)cc1 C1(C(=O)NC2(C)CCCC2O)CC1C1CN(C(=O)Cc2cscn2)C1 C1(C(N(C)CC2CCCN2C)=O)CC(F)(F)CN1C(C1CCCC1)=O c1(C(=O)NC2(C)CC(NC(c3ncoc3C3CC3)=O)C2)cncc2c1CCC2 c1(C(C(=O)NCCCF)N(CCCN(C)C)C)ccc(SC(F)F)s1 C#CC1(O)CC(C(=O)NCC2(O)CN(C(C3C(C(F)(F)F)C3[N+](=O)[O-])=O)C2)C1 C1(C#N)(C(=O)NC2(C)CCN(C(C34COCC3C4)=O)C2)CCS(=O)(=O)CC1 c1(C(N2C(C(C)NC(C(C)=C(CC)C)=O)CCC2)=O)ccc2[nH]ccc2c1 C1(C(N2CCCC(N(C)C(C3CC(O)C3)=O)CC2)=O)CCCC2(CCC2)O1 CCC(C)CCCC(=O)NCC1CC1CC(=O)NCC(C)C(C)CC C1(NC(Cc2[nH]n(CC(C)C)c(=O)c2)=O)CCCN(C(=O)CN2CCCC2)CC1 c1(CNC(Cc2ccc(CNC(C=C(C)C)=O)cc2)=O)ccc(F)nc1F c1(CC)cccc(C)c1NC(=O)CNC(=O)CC1C=CCCC1 C1(C(=O)NCC(C)(C2CC2)NC(c2ncc(Cl)cc2Cl)=O)CC(=O)CC12CCC2 C1(C(N(C)Cc2cccc(CNC(=O)Cc3ccco3)c2)=O)CC(=O)OC1(C)C N1(C(c2cnc(OC)nc2)=O)CCCC(F)(CNC(=O)C(CO)OC)CC1 CC(CCC(=O)NCC1(CC(N)=O)CC1)NC(=O)C(C)(O)C1CC1 CCCC(C)(C)CC(=O)N1CCCCC(C(=O)NC2CCCC2(C)C)C1 C1(C(N(C)CC2CCOCC2)=O)CC12CCN(C(c1cnn3c1OCC3)=O)CC2 n1(CC)ncc(C)c1C(=O)N(CCCCN(C(=O)CC1OCCO1)C)C N1(C(=O)Cc2ccc(F)cn2)CC2CN(C(C3(c4cccc(Cl)c4)CC3)=O)C2C1 C1(NC(CCOCCNC(C2(CCCC)CC2)=O)=O)C=CC(C)(C)CC1 c1(C(=O)OCC)cc(COC(c2cc(-c3csc(C)n3)cn2C)=O)oc1C N1(C(c2scc(C)c2)=O)CCOC2CN(C(=O)CC(C(C)C)C(C)C)CC12 c1(C(=O)OC)nc(=NCCc2ccc(C(=O)O)cc2O)c(Cl)c[nH]1 c1(C(=O)NC2CCC(C)(CNC(CCN(CCC)C)=O)C2)nc(C)c(C)nc1C c1(CNC(C=C(C)C)=O)ccc(CC(F)(F)F)nc1 Cc1ncc2n1CCC(C(N1CCCC1CCNC(=O)CC(C)O)=O)C2 C12(C(=O)NC(CNC(c3ccc(C(=O)OC)nc3)=O)C)CCCC(C1)C(=O)N2 S(=O)(=O)(c1sc2cccc(Cl)c2c1C)N1CCN(C2(C(=O)OC)CCC2)CC1 N1(C(C2(C)CC=CCC2)=O)CCCC2(CCN(C(C3CCNC3=O)=O)C2)C1 C1(CNC(c2cncc(C)c2)=O)CN(C(c2ccccc2)=O)CCC12CCC2 Cc1oc(CO)cc1C(=O)NC(C1CCCC1)CNC(c1ccc(N)cc1)=O N1(C(C(C)SC)=O)CCC(C2CC2NC(c2ccc(F)c3c2OCC3)=O)CC1 C1(C2CCCN(C(c3nnsc3C(F)F)=O)C2)(NC(C(C)=C2CCC2)=O)CC1 C1(C(=O)NC2C3CC(NC(c4c(Cl)cn(C)n4)=O)CC32)CCn2ncnc2C1 Cn1nc(C(N2CC3(C2)CN(C(=O)C(C)(F)F)CC3CO)=O)c2cc(Br)ccc12 N1(C(c2cc(C)sc2C)=O)CCCC(C)(C)C1C(N1CC2(CNC(=O)C2)C1)=O C1(C(=O)NCC(C)(C)C2CCCC2)CSCCN1C(c1ccc(Cl)o1)=O C1(F)(C(N2CC(O)(CCNC(C(C)NC(=O)NC)=O)C2)=O)CC2(CCC2)C1 c1(NC(C2CN(C(=O)C=Cc3cccs3)CCO2)=O)cnc2ccccc2c1Cl c1(OC)cccc(-n2nnnc2C(c2cc(C)sc2C)NCC2C(C)C2C)c1 N1(C(C2CCCN(C(Cc3n(C)ccn3)=O)CC2)=O)CC2CCCC(O)C2C1 Cn1cc(C=CC(=O)NCC2COCC2NC(C2CC3C=CC2O3)=O)nn1 C1(O)(Cn2cc(C(C)O)nn2)CCN(C(=O)Cc2ccnn2C)C1 O=C(CCC1C(=O)Nc2ccccc21)NC1CCCN(C(=O)CO)CCCC1 CC1(NC(=O)Cc2cccc(C(F)F)c2)CCN(C(=O)Cc2csc(=N)[nH]2)C1 C(CC(=O)NC(c1ccco1)CO)OCCN(C)C(c1ccco1)=O C(=O)(C1CCCc2nc[nH]c21)N1C(C2(NC(c3ncn(CC)c3)=O)CC2)CCC1 C1(NC(c2cc(C(C)=O)sc2)=O)CCC(NC(C2(C)CC3(CC3)C2)=O)CC1 c1(C(N2CCC(O)(CN(C(CSCC=C)=O)C)C2)=O)ccn2nnnc2c1 C(=O)(CCCC(C)C)NCC1CCCN(C(Cc2c(C)nc(C3CCC3)s2)=O)C1 N1(C(c2c(SCC)cccc2)=O)CC2CC(C1)N(C(C1CC13CC(F)(F)C3)=O)C2 CC#CCCC(=O)NCC(O)CN(C)C(c1cnn(CCOC)c1)=O Cn1ncc2c(C(N3CC(NC(=O)Cc4cc(F)ccc4O)C3)=O)ncnc12 C1(COC)(NC(c2sccc2F)=O)CCN(C(c2nnn(C)c2C(F)F)=O)CC1 C1(OC)CC(CNC(=O)CCC2(C)CCC(=O)N2)N(C(c2cc(Cl)cn2C)=O)C1 c1(CC(=O)NCC(CCOC)NC(C2(F)CCCC2)=O)ccc2c(c1)CC(C)O2 CC1OCCN(C(C2CC23CC(NC(=O)Cc2cnsc2)C3)=O)C1C O=C(C(Cn1cccn1)NC(C1CC12CCC2)=O)NCCCc1nncs1 c1(C(=O)NCC(C2CC2)NC(C(CC)O)=O)ccc(Cl)cc1C(F)F Cc1cc(C(=O)NCC(C)(CO)NC(c2cc(C3(C)CC3)n[nH]2)=O)cc(F)c1 C1(OC)CC(CNC(=O)CC23CCC(CC2)C3)N(C(=O)C=CCN2CCC2)C1 N1(C(=O)CC2COCCOC2)CC2OCCN(C(=O)C3CCc4nccn43)C2C1 c1(C(N2CC(N(C(C(C)n3ccnc3)=O)C)C2)=O)ccc(Cl)c2ccccc12 C(=O)(CC(C)(C)C(C)=O)NC(CC#CC)C(=O)NC1CON(CC)C1=O c1(C(C(C)C)NC(C2N(C(C(C)=C3CC3)=O)CSC2)=O)cc2ccccc2o1 Cc1nnc2c(C(N3CCC(NC(c4ccc(F)cc4)=O)CC3C)=O)cccn12 CCC(C(=O)NC(C)CNC(=O)CCC1CC1(F)F)n1cccn1 C1(CC)C(NC(c2cc(Br)ccn2)=O)CCCN1C(C1COCCC1C)=O C(C(C(=O)NC1(c2ccccc2)CC1)C(C)C)NC(CC1CC(=C)C1)=O CC1CCN(C(C2(CO)CCCC2)=O)CC1NC(C1C2CN(C)CC12)=O Nc1ncc(Br)nc1C(=O)NCC#CCNC(c1ccccc1C1CC1)=O Cc1c(Br)c(C(=O)NC2CCOCC2NC(=O)C(C)(C)C(N)=O)nn1C CCCC(CC(=O)NCCC1(C)CCCC1)NC(c1cc(C(C)=O)[nH]n1)=O C(C(F)(C(=O)NCCC1(C)CC1)C(C)C)NC(CC1CCC(C)CO1)=O C1(C(=O)NC2CC(C(C)NC(C(c3cnn(C)c3)OC)=O)C2)CC2(CCO1)CC2 C=C(Cl)CCC(=O)N1CCCC1C1(NC(c2cnoc2C)=O)CC1 C1(c2nnnn2C(C)C(=O)OC)(Nc2ncc(CC)s2)CC2(CCCCCC2)C1 Cc1cc(C(=O)NC2CCC2NC(c2cnn(C3CCC3)c2)=O)cc(Br)c1 C(=O)(CCC(=O)N(CC)CC1CN(C(=O)COCC(F)(F)F)CCO1)NCCC C(C(CC(C)C)C(=O)NC(C)(CNC(c1csc(F)c1)=O)CC(C)C)OC C(CC(O)CC(=O)N(C(C)CNC(c1n[nH]c(C)c1Br)=O)C)SC c1(OC)ccc(CCC(N2CC(NC(=O)C(=O)NC(C)C)C(O)C2)=O)cc1Cl C=CCC(CC=C)N=c1cc(NCC2CCCSC2)nc(COC)[nH]1 C#Cc1ccnc(C(=O)NC2(C(=O)NCC(C)(CO)CO)CC(F)C2)c1 C(C)(CCCCNC(C1(N(C)C)CCOC1)=O)NC(c1ccc(C(C)C)s1)=O N1(C(C=Cc2ccc(SC)s2)=O)CCN(C(c2coc3c2COC3)=O)C(C)C1C n1(CCCOCC)c(N2CCOC(C3CC3)C2)nnc1-c1ccncc1 C1(NC(c2c(CC)cco2)=O)CN(C(c2cnn(C)c2C)=O)CC1OC C1(F)(SCCNC(C(C2CC2)OC(C)(C)C)=O)CCN(C(=O)Cc2cscn2)C1 C=CCC(C)(C)NC(=O)CC(C)N(C)C(c1csc(C)c1)=O c1(C(N2CC(O)(C(C)NC(C(C)N(C(C)=O)C)=O)C2)=O)ccc(Cl)c(N)c1 N1(C(C(C=C)C)=O)CCC2(CCC(NC(=O)C=CCO)C2)C1 c1(SC)ccc(O)c(C(=O)NCC2CCN2C(C2(CC3CCC3)CC2)=O)c1 c1(CC)nc(C)[nH]c1C(N1CCCC1C(C)NC(=O)C=CC(C)(C)C)=O C1(OC)CC(CNC(c2cc(C)n(C(CC)CC)n2)=O)N(C(=O)CNC(N)=O)C1 Cc1cc(N2CCC(CNC(C3CCCCC3C3CC3)=O)C(C)C2)ncc1C#N CCC(C)CCCC(=O)N1CCC2C(C1)CN2C(c1cc(Cl)cc(Cl)c1OC)=O c1(-c2c(OC)ccc(F)c2)cc(C(N2CCCOCC2)=O)cc2c[nH]nc12 CC(C)(CCCCNC(=O)C1=CCCC1)C(=O)NNC(=O)C1CCCO1 N1(C(C2(C)CCC(F)(F)C2)=O)CCN(C(c2c[nH]c(=N)nc2C2CC2)=O)CC(O)C1 C12(CNC(CC(C=C)C)=O)CCCC1CN(C(c1[nH]ccc1C1CC1)=O)C2 C(CC(F)F)(C(=O)N(CC(C)C#N)C)NC(c1c(CC)ncnc1)=O c1(OC)cc(C(=O)NCC2CC2NC(c2cnoc2C)=O)cc2c(C)c(C)[nH]c12 N1(C(c2c(C)cnn2C)=O)CCC(NC(=O)CC(C)c2cnn(C)c2)C(CO)C1 c1(C(=O)NCC(CNC(C(CC#C)C2CC2)=O)(C)O)cnc(O)c2ccccc12 CC1CN(C(=O)CCCN=[N+]=[N-])CCN1C(=O)CN1CCCCS1(=O)=O c1(C(=O)NC2CC(NC(c3nn(CC)c(C4CC4)c3)=O)C2)ccc2n[nH]cc2c1 c1(NC(C2N(C(C3N(C)CCOC3)=O)CC=CC2)=O)ccccc1N=[N+]=[N-] c1(NC(CC2(C)CN(Cc3cc(C)c(Cl)nc3)C2)=O)c(C#N)oc2ccccc12 CC(C(=O)NCCCCNC(c1ncccc1O)=O)S(N)(=O)=O C12(C(N3C(CNC(C4CCC(=O)N4)=O)CCCC3)=O)CCCC1OCC2 C12(NC(c3c(CC)nc(C)o3)=O)CCCN(C(c3cc(Cl)cn3CC)=O)CC1C2 C1(C(=O)NCC(C)N(C2CC2)CC)CCCN(C(=O)CNC(=O)OCC(C)C)C1 CC1CCCCC1(CO)CNC(c1nnsc1SC)=O.N1(CC=O)CC2CC2C1 N1(C(C2(CC(C)C)CC2)=O)CCC(O)(CN(C(=O)C#CC(=O)N(C)C)C)C1 C12(C)CCCN(C1)C(=O)CCNC2=O.CC1CC(C(=O)NCc2ccoc2)CO1 N1(c2n(CCCC#C)nnn2)CCN(C(CC)CC)CC1 Cn1ccc(C(=O)NC(Cc2ccco2)C(=O)NCc2cscn2)c1 C=CC(CC)CC(=O)N1CC2CC(CNC(c3nc(C)c(C)s3)=O)C2C1 N1(C(CC2(C)CC2)=O)CCC(NC(C2CCN2S(C)(=O)=O)=O)C12CC2 c1(C(=O)NCCCCC2(NC(C(OC)OC)=O)CC2)cc(O)ccc1Br c1(C(=O)NC2CC(NC(c3cn(CC(F)(F)F)nn3)=O)C2)cnn2ccncc12 N1(C(C(C)N2CCC2)=O)CCCOC(CNC(=O)CCc2nc(O)n[nH]2)C1 c1(CNC(=O)OC)ccc(C2CC2)o1.C12(CC(C[Si](C)(C)C)C1)c1nnnn1N2 c1(C(N(CC(C)NC(C2CCCC2CF)=O)C)=O)n[nH]c2c1CCCCC2 c1(CC)cc(C(=O)N(CC(C)NC(c2cc(CO)n(C)n2)=O)C)oc1CC CCC(CC)(CO)C(=O)NCCCCNC(C1(C)CCC(C)C1)=O c1(C(=O)NCC2C(NC(Cn3c(C)cnc3)=O)CCC2)cccc2cc[nH]c12 c1(OC)cc(Cl)ccc1C(N1CCC2(NC(c3cc(Cl)c(C)cn3)=O)CC2C1)=O N1(C(CC(CC)C)=O)CC(C)C(C)(CNC(c2c(Cl)nn(C)c2C)=O)C1 N#Cc1ccnc(N2CCN(CCCCCNC(c3cc(Br)c(Cl)s3)=O)CC2)c1 C1(C)(C(=O)NCC(C(=O)NCCC(=O)N(C)C2CC2)(C)C)C(C)(C)C1(C)C c1(C(=O)NC(CC(C)NC(c2ccc(OC)nc2F)=O)C)ccn2ncnc2c1 C1(CC(=O)NCCCC(=O)N(CCCO)C)CC(C2CC2)C1 c1(OC)ccc(CC(=O)NCCNC(C2COCCO2)=O)c(Cl)c1 CCC(CC(=O)N1CC(O)(CNC(=O)CC(F)(F)C(F)(F)F)C1)C(C)(C)C c1(NCCN2CCC(O)(C(=O)Nc3ccc(C#N)cc3)C2)cccc2c1CCC2 CC(C(=O)N1CC(CC(N)=O)C1)n1ccnc1 c1(OC)cc(CC(N2CCN(C(C3C(OC)CCC3)=O)CC2CO)=O)ccc1Cl C(=O)(C(F)C(F)(F)F)NC(CCNC(c1c(C)oc(CO)c1)=O)C(C)C CC(C(=O)N1CCN(C(c2cccnc2C(F)F)=O)CC1CCO)C(C)(C)C Cc1ccc(CCC(=O)NC(c2cn(C(c3ccccn3)C)nn2)C)cc1Cl C1(C(=O)NCC2CCCN2C(C2CCC2)=O)CCCCC12CC2 CC1(C)Cc2[nH]nc(C(=O)NCCCNC(c3cncc(N(C)C)c3)=O)c2C1 CCCC(O)CN(C)C(C1(CCNC(=O)C(COC)OC)CCC1)=O CN1CC(C(=O)NCC2CC2CNC(c2cnc(C3CCC3)s2)=O)CC1=O c1(C(=O)NC(CNC(C2(C)CCC2)=O)C2CCC2)cc2n(c1)CCSC2 C1(CCOC)(NC(c2sccc2F)=O)CCN(C(C2CC(=C(F)F)C2)=O)C1 C(CN(C(=O)C(C)=CCCC(C(=O)N)OC)C)(C(C)C)OC C(=O)(C#CC1CCCOC1)N1CC2C(NC(c3cc(OC)c(F)cc3)=O)(CC2)C1 c1(COCC(CN2CC(CCNC(C3(COC)CCC3)=O)C2)O)ccc(Cl)cc1 Cc1cccc(N2CCC(C(=O)NCCN(C(=O)C(O)C3CC3)C)C2=O)c1 CCC(C)(CC)C(=O)NCCC1CCCCN1c1ccnc(CCOC)n1 S(=O)(=O)(c1ccc(Cl)c(F)c1Cl)NC1CN(C(=O)OC(C)(C)C)C1 c1(C(N2CCN(CCCNC(C3C4CN(C)CC43)=O)CC2)=O)cc(=O)n(C)cn1 Nc1cc(Cl)cc(Cl)c1C(=O)NC1CC(NC(c2noc3c2CCCC3)=O)C1 c1(NC(C2C(C(=O)NC(c3ccccc3F)C)C2)=O)ncccc1Br c1(NC(c2csc(C(=O)Nc3ccc(F)cc3O)n2)=O)cc(Br)ncc1F c1(CC(N2C(CNC(c3n(CC)cnn3)=O)CC2)=O)ccc2c(c1)OCO2 C(=O)(C1=CC2CCC(C1)C2)NC(CCC)CNC(c1n[nH]c2c1COC2)=O C1(CNC(CCSCCC)=O)C(C)CCN1C(=O)C(CC1CCCC1)N(C)C N1(C(CC(C)n2cc(Br)cn2)=O)CCOC(C(C)(C)C)C1 Cc1onc(C2CC2)c1C(=O)NCCNC(C1(C)CC=CC1)=O C(C)(C)(CCC(=O)N1CCOCCC1C(=O)NC(C)CC1CCC1)OC c1(C(=O)NCC2N(C(C(CC)O)=O)CCOC2)cnc2ncccn12 Cn1cccc1NC(=O)C(CO)NC(=O)C(=O)NC1CC1 c1(CC=C)c(NC2CN(C(C)C)C2)ncnc1Cl Cn1cc(NC2CC(C(=O)NC(CO)CCF)C2)cn1 c1(C(=O)NCc2cccc(CN=c3ncc(Cl)c[nH]3)c2)ccn2ccnc2n1 C1(CNC(CNC(CCC)=O)=O)CCc2nc(NC(=O)CC)sc2C1 c1(CC(=O)N(CCC)CCNC(c2cc[n+]([O-])cc2)=O)ccc(C)c(F)c1F Cc1cnc2nccc(N3CCC4(CCC(CC(=O)N(C)C)C4)C3)c2c1 c1(C(N(C)CC2(NC(=O)CC3CCCC(=O)N3)CC2)=O)cc2cccc(F)c2s1 CCC(C)(C)C(C)CC(=O)NCC1(O)CN(C(=O)C(n2nccc2C)C)C1 c1(C(=O)NC2(CCNC(C3C4CCCCC34)=O)CC2)ccc2ccoc2c1 Cc1cc(Cl)cc(C)c1C(=O)NC1CCCCC1NC(C1(CF)CCC1)=O N1(C(C=CC)=O)CC(C(=O)NC(C)(C)CCCC)C2(CC2)C1 C1(C(=O)Nc2cc(F)c(C(=O)NC3CC3)c(F)c2)CCC2C(CC1)C2(F)F c1(CC)cccnc1C(=O)NCC1(F)CCN(C(=O)Cc2ccccc2OC)C1 C1(CC(N2C(C)C(NC(=O)CC34COCC(C3)C4)CC2)=O)CCCC(C)(C)C1 c1(C(N2CCC(N(C(=O)Cc3ccnc(Br)c3)C)C2)=O)c(Br)cc(Br)c(O)c1Br C(=O)(CC(C)(C)C#N)NCC=CCC(=O)NC1(CC=C)CCOC1 C1(NC(C(C)(C)OCC)=O)CN(C(C2CCCN(C(C)C)C2)=O)CCC1F c1(CCC2CCCC(C(=O)NC(=O)Cc3ccccc3I)C2)ccc(Cl)cc1Br C(N=c1[nH]c(N2CC(C)OC(C)C2)nc2cccnc12)c1cnc(CC)s1 N1(C(C(C)Cc2ccccc2F)=O)CC2=C(C1)CN(C(=O)C=C1CCOCC1)C2 C(=O)(C(F)(F)CC(C)C)NC(C1CCN(C(C(C2CCCCC2)OC)=O)C1)C n1(CC)ccc(C(=O)N(C)CC2CCCN2C(C23CCCC(CO2)C3)=O)cc1=O C1(NC(C2(CCCC)CC2)=O)CN(C(c2cnncc2OC)=O)CC1C c1(OC)cc(C(=O)NCC2CC(NC(=O)CC3CCCS(=O)(=O)C3)C2)cc(F)c1 c1(C(N2C(C)(CNC(C3CC(F)(CF)C3)=O)CCC2)=O)cccc(=S)n1O C1(C(N2CC(CC)S(=O)(=O)C(C)C2)=O)CCN(C=CC(=O)C(F)(F)F)CC1 CC1OC(=O)NC1C(=O)NCCC1(C)CCN(C(=O)C=C2CCCCC2)C1 c1(C(=O)NCC2(C)CCC(NC(C=C(CC)CC)=O)C2)cc2ccccc2[nH]1 N1(C(C2CC2(F)F)=O)CCCC(NC(C2(F)CCCC2)=O)CC1 C1(C2CC2)C(=O)N2CCC(O2)C(=O)N1.N1(CC)CCc2cccc(F)c21 N1(C(C(C)(C)OC)=O)CC(C)(C)C1C1CCN(C(=O)CCCc2ncco2)CC1 N1(CC(=O)NC2CC(NC(=O)C(F)(F)C3CC3)C2)CC2CCC1C2 C(=O)(CCC(=O)N1CCC(C)C1CNC(=O)C(F)=C(C)C1CC1)NC n1(CC)cnc2c(N3CCCC(CCO)C3)nc(=NCc3ccsc3)[nH]c12 c1(NC(c2cccc(N)n2)=O)c(Cl)cc(F)cc1Cl c1(C(=O)NC2C3(CC(NC(CNC(CC(C)C)=O)=O)C3)C2)ccc(N(C)C)cc1 c1(OC)cccc(-n2nnnc2C2(N(C)Cc3nc(C)no3)COC(C)C2)c1 Cc1cc(Cl)ccc1NC(c1cc(CCNC(=O)C(C2CCCCC2)O)on1)=O N1(C(Cc2c(C)nn(C)c2)=O)CC(S(=O)(=O)c2cccc(F)c2)C1 S(=O)(=O)(c1cccc(=NCCCCCO)[nH]1)NC(COCC)C(C)C C1(N(C(=O)C=CCOCC(F)(F)F)CC#C)CCN(C(c2cnoc2)=O)CC1 Cc1cc2occ(C(N(c3cc(OC4CCOCC4)ncn3)C)=O)c2cc1C CCC(C)(CC)C(=O)NCCC1(CNC(=O)C(C2CCCC2)OC)CC1 CC(C)CCCC(C)NC(=O)CCN(CCO)C(c1nc(Cl)cs1)=O CCCS(=O)(=O)c1ccc(C(=O)NCC(C)NC(=O)CCCC(C)(C)C)cc1 C1(NC(c2cc(CC)on2)=O)CCC(NC(=O)CC2CCCN2C)CC1 C1(CC(N2CCOCC2)=O)CCN(N2CC(c3nnc[nH]3)C2)CC1 C1(NC(c2c(C(C)C)ccs2)=O)CC(C)CN(C(=O)Cc2csc(Cl)n2)C1 Cc1nnc(=NCC2CCCC(NC(C3CC4CCCC(C3)C4)=O)C2)[nH]c1C N1(C(N)=O)CC(O)CC1C(=O)NC12CC1CN(C(c1cc(C3CCC3)[nH]n1)=O)C2 C1(CNC(CN(C)C(c2cccs2)=O)=O)C2CN(C(=O)CN(C)C(N)=O)CC12 C1(C(N(C)CC2(NC(CSC)=O)CC2)=O)CC(=O)N(C)C1c1ccc(Cl)c(F)c1 c1(C(N2CC(OC)C(NC(=O)C(C)(C)C(F)F)C2)=O)ccn2nccc2n1 CN(C(=NCC1CCOC1)NC1CCS(=O)(=O)C1)Cc1ccc(F)cc1Br c1(OC)ccnc(F)c1C(=O)NC(C)CNC(c1n[nH]c(C)c1F)=O Cc1cc(NC(C2CC(NC(c3ccc(C(N)=O)[nH]3)=O)C2(C)C)=O)cnc1O C12(NC(N3CCC(c4cccc(OC(F)(F)F)c4)C3)=O)CC3CC(CC(C3)C1)C2 C1(C(=O)OCCCNS(CC)(=O)=O)NCCC12CCC2 Cc1nc(C)c(C(=O)NC2COC3(C2)CN(C(c2cnc(C)[nH]2)=O)C3)c(C)n1 C1(NC(Cn2c(C)c(Cl)cn2)=O)CCCCN(C(=O)CC23CCC(C)(C2)OC3)C1 CCCC(C#N)C(=O)NCCc1ccc(CNC(=O)C(O)C(C)C)cc1 C1(C2CCCCC2)(C(N2CCC(CNC(C=C(C)C(F)F)=O)C2)=O)CCCCC1 C(CC(C)(C)C)(C(=O)NCC1(OC)CCN(C(=O)CC2CC3CC3C2)C1)OC C1(CC)CCCCCCN1C(C1(CC)CCCN1C(c1nccc(C)c1N)=O)=O c1(CC)nc(C(N2CC(CNC(=O)Cc3cc(OC)no3)CC2C)=O)c(N)s1 CCC(C)(C(=O)N1CC2CN(C(=O)Cc3csc(C(C)(C)C)n3)CC2C1)C(N)=O C1(C(=O)O)CC(n2cc(Cn3ccnc3)nn2)CN1C(C12CCCC1C2)=O C1(N(C(c2c(C)noc2N)=O)C)CCCN(C(C2NC(=O)CC2C)=O)CC1 N1(C(c2c(CNC(C(C)O)=O)cco2)=O)CC(O)CC1CO c1(CN2CC(CC(=O)NC(C3CC(F)(F)C3)C)C2)cc(Cl)cc(Br)c1 c1(CC(=O)NC(c2cccc(F)c2)CNC(C2(CC)CCC2)=O)nn(C)cc1Cl n1(CC(=O)NC2CN(C3CN(C(CC(=O)NC)=O)C3)C(=O)C2)cnc([N+](=O)[O-])n1 n1(CCC)ccc2cc(NC(=O)Nc3cnn(CCC(=O)OC)c3)ccc12 C(=O)(C#CC1CCCC1)N1CCC(C(=O)NCC(COC)(O)CO)C(C)C1 Cc1c(NC(C)C)cccc1C(=O)N(C1CN(C(=O)CCc2cn(C)nn2)C1)C N1(C(C2CN(C(C3OCCC(C)(C)C3)=O)CC2(F)F)=O)CC(C2CC2(F)F)C1 c1(CC)c(C(N2CC(CC(C)NC(C3(C)CC4CC4C3)=O)C2)=O)csc1C N1(C(c2c(CC)cco2)=O)CCN(C(c2cocn2)=O)C(c2cccc(F)c2)C1 N(C(=NCCOC(F)(F)F)NCC1CCC1)CC(c1cc(F)cc(Cl)c1)O Cc1oc(C(C)C)nc1CCCNC(=O)OC(=O)OC(C)(C)C.C(=O)(C(C)C(C)C)N C(=O)(C(CCS(C)=O)NC(=O)OC(C)(C)C)N1CCC(Oc2c(C)cccc2)C1 C1(F)(CNC(C(C2CC(NC(C3CCCCC3)=O)C2)F)=O)CCOCC1 C1(NC(CN(CCOC)C)=O)CN(C(C2(CF)CCOCC2)=O)CC1S(C)(=O)=O C1(CC)CCCC1C(=O)NC1CC1CNC(=O)C(C1CCCCC1)F N1(C(CSCC=C)=O)CCC(NC(c2cnc(C(F)(F)F)cc2C)=O)C(O)C1 C(C(C)(C)CNC(c1nc(Br)c[nH]1)=O)N(C)C(c1cccn1C1CC1)=O c1(C(=O)OCc2c(C)ccs2)ccc([N+](=O)[O-])c(N)n1 N1(C(Cc2cc(OC)c(O)cc2F)=O)C2CCCC1CN(C(C1(F)CC1C)=O)C2 c1(OCC2C(N(C)S(N)(=O)=O)CCC2)ccc(Br)cc1 c12cccc(c1)OCC(=O)N2.N1(C(C)=O)CC(CCO)(NC(=O)CSC(F)F)C1 c1(C(N2CCC(C(C)(C)C)(CNC(CC3(C)CC3)=O)C2)=O)cc(=N)[nH]c(Cl)n1 C(=O)(C1=CCCC1)NCCC(CNC(C1C(c2ccccc2)C1(C)C)=O)OC c1(NC(=O)NCC2C(CC(C)(C)C)C2)ncc(Cl)cc1Cl c1(N(C)Cc2cccc(F)c2)nc2c(c(=NCc3ccccn3)[nH]1)COCC2 C1(C(=O)OC)CCCC(C(=O)NC2(C)CN(C(c3cc(N)cc(O)n3)=O)C2)CC1 CCCC(CC)C(=O)N(C)CCOCCC(=O)N(C)CCC1CCCO1 C1(C(N2CC(CC(C)NC(C3C=CCC3)=O)C2)=O)CC2(C1)CC1(CCC1)C2 N1(C(C)C)CCN2C(=O)C(NC(c3ccn4cnnc4c3)=O)CC2C1 CN1CC(O)CC1C(=O)NC(c1cccnc1)C(=O)NCCC(O)C1CCCC1 N1(C(C2C(=C)CC2)=O)C2CCC1C(CNC(c1cc(C)sn1)=O)C2 c1(C(C)Oc2ccc(C(F)(F)F)cc2)csc(=NCC2CCCS2)[nH]1 CCCCCC(C)CC(=O)NCC1CN(C(c2nccc(C)n2)=O)CC1C c1(C(N2C(CO)CC(NC(c3nccc(C)c3)=O)C2)=O)nccc(C#N)c1F c1(C(N(CC(C)NC(c2ccn(C(CC)CC)n2)=O)C)=O)cccc(OC)n1 C1(C(=O)NCc2c(C(=O)NC3(CC=C)CCOC3)[nH]cc2)CC(O)C(F)C1 C(=O)(CC(CCCC)NC(=O)CN1CCCCC1=O)NC(CC=C)CC Cc1cc(C(=O)NC(C)C(CO)NC(c2nnn(-c3ccccc3)n2)=O)ncn1 CCCCCC(=O)NCC1(NC(=O)CC2CCCN2CC)CC(OCCC)C1 Nc1cc(Cl)c(Cl)cc1C(N1CCN(C(C2OCC3CCCC23)=O)CC1CF)=O c1(C(N2CC(C)C(NC(c3cncc(Br)c3)=O)C2)=O)ccc(Cl)cc1F C(=O)(CCCN=[N+]=[N-])NCC1(CNC(CS(Cc2ccc(C)cc2)(=O)=O)=O)CC1 C(=O)(CCCC(C)(C)C#N)N1CCC(NC(C(C)P(C)(C)=O)=O)C1C(C)(C)C C1(F)(C(=O)NC2(C(C)C)CC2)CCCN(C(C2CCCC3(CC3)C2)=O)C1 CN1CCC(N(C(=O)C(=O)NC2CC2)C(c2nn(C(C)(C)C)cc2Cl)=O)CC1 N1(C(C(C)(F)F)=O)CC2COCC(C1)C2NC(C1COC2(CCC2)CO1)=O C(=O)(C(C)(O)C(F)(F)F)NCC1(CNC(c2cccc(C#C)c2)=O)CC12CCC2 C1(CNC(C2N(CC)CCOC2)=O)CN(C(C2CCCCS2)=O)CCN1C C(=O)(CC1OCc2ccccc21)NCCCNC(c1cnc(C)nc1C(C)C)=O CCCC(CCC)CC(=O)NC(CNC(C1CC1CCOC)=O)CO C1(C)(CNC(C=CCOC)=O)CCN(C(=O)C(C)N(C)C(=O)OC(C)(C)C)C1 N1(C(CCC2CC(OC)C2)=O)CC(NC(c2nccn2C(C)C)=O)CC12CCC2 c1(NC)c(C(=O)N(C2CCCN(C(=O)C=C(C)C)C2)C)cccc1F C(C1CCOc2ccccc21)NC(=NCCCF)NCCN1CCCCC1 c1(C(=O)OCC)ccoc1C(=O)NCC(C)N(C)C(c1ccnn1C1CCC1)=O N1(C(CCCNS(C)(=O)=O)=O)CCC(NC(=O)C(c2ccccc2)F)C12CC2 C1(NC(CC2CCC(C)C2)=O)CCN(C(C2CCCC2)=O)CC1(C)C c1(C(=O)NCCNC(C2(C=C)CCOCC2)=O)ccc2nc[nH]c2n1 N1(C(=O)COC(F)F)CCCC1C1CCCN1C(c1cc(F)c(F)c(Cl)c1F)=O n1(CC(=O)NC(CN(C)C(c2ccnn2C(F)F)=O)(C)C)cnc(C#N)n1 c1(C(=O)NC2CC(NC(C(CC)OC)=O)C2)cc(C)c2ccccc2n1 C1(CCC)CCCN(C(=O)C(C)(C)CN(C(=O)CCCN(C)C(C)=O)C)C1 C(C(C)C(=O)N1CC(C)(c2cn(Cc3cnns3)nn2)C1)OCC c1(C(N2Cc3c[nH]nc3C2)C(=O)NCC=C)noc2cc(Br)ccc12 N1(C(C2C(COC)C2)=O)CCC(C)N(C(c2cnc(COC)[nH]c2=N)=O)CC1 C(=O)(C1=C(Cl)CCCC1)NCC1CC(C)CN(C(c2csnc2Cl)=O)C1 C1(C2CCN(C(c3nn(C)c(Cl)c3Cl)=O)CC2)(NC(c2c(C)ncnc2)=O)CC1 c1(C(C)(C)OC)nc(C)c(C(=O)NCC(C2CC2)NC(C2CC(C)(C)CO2)=O)s1 C(C(=O)Nc1nc(C2CC(F)(F)C2)cs1)(C(C)C)NC(C)=O N1(C(c2c(CC)n[nH]c2)=O)CCN(C(=O)CN2CCCNS2(=O)=O)C(CCO)C1 N1(C(c2cncc(COC)c2)=O)CC2CCC2(CNC(=O)C(C)(C)CO)C1 N1(C(CC=C=C)=O)CCN(C(CNC(=O)CCCCN2CCCC2)C(F)F)CC1 c1(C(N(C2CCN(C(=O)C(C)NC(=O)C3CC3)C2)CC)=O)cnc(CO)nc1C C1(CC)CN(C(=O)Cn2cc(-c3ccc(CC)s3)nn2)CCC1CC(N)=O N1(C(CCN(CCCCC)CC)=O)CCc2cccc(O)c2C1 C1(NC(COCCC)=O)C=CCC(C(N2CCCC(C)C2)=O)C1 CC(C)(C)C(=O)C(=O)N1C(CC(N2CCC(C(C)(C)O)CC2)=O)C2CCCC12 C(=O)(CC(C)P(C)(C)=O)NC(c1cn(-c2cc(OC)cc(Br)c2)nn1)C C1(Nc2c(C(=O)OCC)cccn2)CN(C(=O)CC2C=CCCC2)C(C)(C)C1 N1(C(C2(C)CC(C)OCC2)=O)CCC2(CCCN(C(c3csnn3)=O)C2)CC1 C1(NC(C2(CC)CCC2)=O)CC(=O)N(C2CN(C(C3CCCC3C)=O)C2)C1 C#Cc1ccc(C(N2CCC(NC(=O)C=CC3CCCCC3)C2(C)C)=O)cc1C C1(NC(C(C)NC(=O)Cn2cncn2)=O)CC2CCC1(NC(c1cncs1)=O)C2 c1(C(=O)NC(CCC)CNC(=O)C(O)CN(C)C)ccc2nonc2c1 Cc1cc(C#N)ccc1C(N1CCC(F)(F)C(CNC(=O)CC2CCCO2)C1)=O N1(C(COc2ccc(C)cc2F)=O)CCC(C)N(C(c2cc(C#N)no2)=O)CC1 c1(C(=O)NCCCN(C)C(c2nccc(C#N)c2F)=O)cnc2cccnc2c1 C1(NC(CC(C)(F)F)=O)COC2(C1)CN(C(C1CC3CCC(C1)C3)=O)C2 C(C)(CCCC(=O)NC(C)CCC(F)(F)F)NC(CN(CCOC)C)=O c1(C(N(CCC(C)NC(c2ccc(C(=O)OC)nc2)=O)C)=O)cc(C)ccc1F C1C(N=c2cc(C)nc(SC)[nH]2)O1.c1(OC)ccccc1NC1CCC(SC)CC1 C1(C(=O)NCC2C(C(N(C3CC=CC3)C)=O)CC2)CCC(=O)C1 c1(OC)cccc(OC)c1NC(c1cccc(NC(c2c(C)n[nH]c2C)=O)c1)=O c1(C(=O)NC(CN(C(CCCOCC=C)=O)CC)C)ccnc2ccsc12 CCCC(CC(=O)Nc1cc(C)ccc1C)NC(=O)C=Cc1ccc(C)o1 N1(C(c2nn(CC)c(C)c2)=O)CCC2CCC(C1)N2C(C1(O)COC1)=O C1(C(=O)NC(C)Cc2nc[nH]n2)(NCc2ccccc2)CCOCC1 N1(C(c2c(C)csn2)=O)CCC(NC(c2c(C)cncc2C)=O)C(C)C1 N1(C(c2cnn(CC)c2Cl)=O)CCOC2(CCN(C(C3CC(F)CN3C)=O)C2)C1 CC1C(NC(=O)CSC(=N)N)CCCN1C(=O)C=Cc1cccn1C C1(c2ccccc2)(NC(C2C(C)(C(C)C)C2)=O)CN(C(c2n[nH]c(=N)[nH]2)=O)C1 C1(CNC(C2OCC(C)(C)C2)=O)N(C(=O)C2=CCCCC2)CCC1(C)C c1(CN2CCC(CNC(=O)C(F)F)C2)cc(C(F)(F)F)cc(F)c1 c1(C(N2C(CNC(C(C(=O)OC)C)=O)CC(O)C2)=O)csc2c1CCCC2 C(=O)(N=c1[nH][nH]c2ncc(Br)cc12)C1N(C(CC(CC)O)=O)CCC1 c1(C(N2CCCN(Cc3ccc(OC)cc3Br)CC2)=O)nc2ccc(F)cn2n1 c1(C(=O)NCC(CNC(c2c(C(C)C)con2)=O)CO)cc(C#N)ccc1N C1(CNC(C(C)(C)CNC(=O)CCOC2CCC2)=O)CC(O)C12CCC2 C(CCC(C)C(=O)N1CCC(N(CCO)C(c2csc(C#N)c2)=O)C1)OC C(N=c1ncc2ccccc2[nH]1)C1C(NC(Cn2cc(C(C)C)nn2)=O)C1 c1(C(=O)NCC#CCNC(C(C)c2ccsc2)=O)c[nH]c2ccccc2c1=N C1(C(=O)NC2C3CN(C(c4n(C=C)nnc4)=O)CC32)Cc2ccccc2C1(C)C CC1(C)NC(=O)CCC1NC(C1CCCCC1(C)NC(C1CC(=O)CCO1)=O)=O c1(C(N(C(C)CNC(=O)CC2CC2)C)=O)cc(F)c(C2CC2)cc1F N1(CC(C)(C)C)CCC(N(C2CCSC2)CC2CCCO2)CC1 S(=O)(=O)(c1cc(-c2nn[nH]n2)ccc1F)C(N1C2COCC1CC(CO)C2)C N1(C(c2c(C)nns2)=O)C(CNC(=O)Cn2ccnc2C)CC2CCCCC12 C1(CC#C)(C(=O)NCC2CCCC2NC(=O)COc2ccccn2)CCCCO1 C=CCCCCC(=O)NCC1CCCC1(F)F CCCCCC(C)(CC)C(=O)NCCC1CCCN(C(C2CCS2(=O)=O)=O)CC1 Cc1cc(C(=O)NC(C)CNC(=O)C(F)n2ccnc2)cc(NC2CC2)n1 C(N=c1[nH]c(=NCCCCN2CCC2)[nH]c2c1CCCC2)C1NC(=O)C(F)(F)C1 N1(C(c2nc(CCC)oc2)=O)CC(C(=O)N(C2CCC2)C)C(C)(C)C1 c1(C2CCN(C(C(=O)NCC3CC3)c3ncco3)CC2)nnc2n1CCCC2 C1(CNC(C(F)=CCC)=O)CCCC1C(=O)NCC(C)(C1CC1)OC C1(N(C(CCCC#C)=O)CC)CC(F)CN(C(=O)CCc2ccc(C)nc2)C1 C1(NC(c2ccco2)=O)CCCCN(C(=O)CC(O)c2ccccc2)CC1 C=CC(CC)CC(=O)N1CCSCC1CCNC(=O)CCc1cn(C)nc1C C1(NC(C(C)(C)SC)=O)CCCN(C(=O)CSc2cc(F)ccc2F)CC1 C12(CC)COC(C(=O)NC3CN(C(=O)C(=Cc4c[nH]cn4)F)CC3OC)(C1)C2 c1(OC)ccc(NC(C2CC(OC)CN2C(c2cc(Br)cs2)=O)=O)c(C)n1 Cc1nc(N2CCN(C(=O)C(C3CCCO3)C3CC3)CC2C)cc2nncn12 C1(CNC(C(CCOC)C)=O)CC2(CC(NC(=O)C(C)n3ccnc3)C2)C1 N1(C(CC2CCN(Cc3cnn(CC)n3)C2)=O)CCCC1(C)C(=O)OC N1(C(=O)NC2C(c3n(CC)ccn3)OCC2)CCC(C)(c2ccc(Cl)cc2)CC1 c1(CN(C)CC2CCN(C(=O)C(c3ccccc3)F)CC2)ccc(Cl)nc1 C(=O)(C(C)(C)CC(=O)OC)N(C1CC2CNC1C2)CC.C12CCCC1(C)NC2=O C(CN=c1ccc(C(N2CCC(O)(CCNC(C3CC3F)=O)C2)=O)c[nH]1)OC N1(C(CCC)=O)CC2CCCC(C1)N2C(c1nc2c(C(F)(F)F)cccc2s1)=O N1(C(c2cc(OC)nn2C)=O)CC(C)CCC1C(=O)N(C1CCCC1(F)F)C C(=O)(C1=NN(C)C(=O)CC1)NC(CCNC(CC(=O)OC)=O)C N1(C(c2c(C)cc(C(F)F)o2)=O)CCC(F)C(NC(c2ncncc2Cl)=O)C1 C(=O)(C(C(C)(C)C)n1ccnn1)NCC(CNC(C1CC(OC)C1)=O)C c1(NC(C)CNC(=O)C(c2cccc(Cl)c2)C)ccc(S(C)(=O)=O)cc1[N+](=O)[O-] N1(C(C2(OCC)CCC2)=O)CC2CCC1C1CN(C(=O)CN(C3CCC3)C)CC21 C1(C(=O)NCC(C(C)(C)C)NC(C2CNC(=O)N2)=O)CC2CS(=O)(=O)CC2C1 c1(C(N2C3CN(Cc4ccc(O)cc4Br)CC23)=O)cc(Cl)nc(Cl)c1 N1(C(C2N(CC)C(=O)CC2)=O)CC2=C(C1)CN(C(C1CC(C)(C)CO1)=O)C2 C1(C)(C(N2CCC(NC(C3(COC)CCOCC3)=O)C2)=O)CCC12CCC2 c1(C(N2CC(C)C2C(=O)NOCCC(F)F)=O)c[nH]c(C#N)c1 C(=O)(C(C)(F)C(=O)N1CC2(NC(c3ncccc3F)=O)CCC1C2)OCC Cc1cn2cccc(C(N3CC4(C)CC3C4NC(=O)CC3CCCOC3)=O)c2n1 N1(C(=O)NCC(c2nncn2C)C)CCOc2cc([N+](=O)[O-])ccc2C1 CCCC(O)CC(=O)NCC(c1ccccc1)NC(C1SCCCS1)=O c1(C(=O)NC2CCN(C(C(C)(CO)OC)=O)C2)ccc([N+](=O)[O-])c(C#N)c1 c1(C(=O)NC23CN(C(CCOC(C)C)=O)C(C2)C3)cc(Br)cc2c1OCC2 CC(CC(N)=O)C(=O)N1CCC(NC(=O)CCc2nncn2C)C1(C)C CC(C)CC(O)C(C)C(=O)NCc1ccsc1C(N1CC(C(=O)NC2CC2)C1)=O S(=O)(=O)(c1ccc(=NCC(C)CCCC(C)C)[nH]c1)NCCC c1(C(N2CCC(NC(Cc3c(C)cccc3F)=O)C2)=O)ccc2c(c1)CC(=O)N2 N1(C(C#CC(=O)N(C)C)=O)CCC2(CC(NC(=O)C=Cc3cncn3C)CO2)C1 N1(C(C#CC)=O)CCC2C(CCN2C(c2ccncc2Cl)=O)C1 c1(NC(C2N(C(C3(OCC)CCCCC3)=O)CC2)=O)cccc(COC)c1O C=Cn1cc(C(COCc2ccccc2)N(CC(c2ccco2)O)C(C)C)cn1 c1(C(=O)NCc2c[nH]cc2C)cnc(C(C)C)nc1N(C1CCCN(CC)C1)C c1(N2C3(CNC(c4cc(C)cc(C)c4)=O)CC(C2)C3)ccc(Br)c(C)c1[N+](=O)[O-] c1(C(N(CCOCCNC(C=CC=CCC)=O)C)=O)cc(C)c(F)c(C)c1 c1(C(=O)NC(CCOCC)CO)cc(C)n(-c2ccc(OC)cc2)c1C c1(C(=O)NCCC(C(=O)N(C(C)C)CC2CC2)O)ccc2occc2c1 S(=O)(=O)(c1cccc(-c2ccc3ncsc3c2)c1)NS(=O)(=O)CC(F)(F)F C1(N(C)C(c2cc(Cl)c(Br)s2)=O)CCCC2CN(C(=O)C(C)(O)C(F)(F)F)CC12 Cc1cc(C(=O)NC2(C(F)F)CCCN(C(=O)OC(C)(C)C)C2)nc(C)c1 c1(CC(=O)NCC(=O)NCC(=O)Nc2cccc(OC(F)F)n2)ccc(O)nc1 C1(C(C)=O)CC(CC(=O)NCCN(C)C(c2cccc(Cl)c2)=O)C1(C)C CS(=O)(=O)c1cccc(CC(=O)NCCN(C(=O)CCC2CCCO2)C2CC2)c1 C(N=c1[nH]c(=N)[nH]c(Cl)c1[N+](=O)[O-])C1OCC(CNC(c2c(C)oc(C)c2C)=O)C1 N1(C(CC2(C=C)CCC2)=O)CC(NC(c2oc(CO)cc2C)=O)C2(CCC2)C1 C(=O)(C1Cc2ccc(Cl)cc21)NCC(N(C(=O)C(F)C(C)(C)O)C)C1CC1 c1(C(=O)NC2CCN(c3nccc(OCC)n3)C2(C)C)cnc2c(c1)CCCO2 C(=O)(CS(=O)(=O)N(C)C)N(CC(C)NC(C1(c2ccccc2)CC1(Cl)Cl)=O)C C1(CCC(=O)NCCN(C(C)C)C(C2CC(=O)N(C)C2)=O)CC(C)(C)CO1 CCCCC(O)CCC(=O)N1CCCC(NC(=O)CN(CC(=O)NCC)C)C1C N1(C(CC)=O)CC(F)(F)CC1(C)CNC(C1CCN(CC(C)C)C1)=O CC(C)C(O)C(C)C(=O)N1CCN(CCNC(=O)C(F)=C2CCC2)CC1 C1(C(N(CC(C)CNC(C2(CF)CCC2)=O)C)=O)(Cc2cnn[nH]2)CC1(F)F c1(C(=O)NCCNC(C2CC(C3CC3)=NO2)=O)cc2cc(Br)cnc2o1 c1(CC)cc(F)ccc1OC(=O)CONC(=O)Cc1cccc(OC)c1Cl Cc1ncc(NC(C2CCCN2C(=O)CCCC2CCCO2)=O)cc1C#N N1(C(=O)CSc2cccc(F)c2)CCCC(C2CCN(C(c3ccns3)=O)C2)C1 c1(C(=O)NC(C(CC)C)C(=O)O)cc(C)cc(C=O)c1 C1(NC(C(C(C)C)F)=O)CN(C(c2ncc3ccccn23)=O)CC1C1CC1 c1(C(=O)OC)cc(Br)c2nc(NC(c3c(Cl)cnn3C3CCCC3)=O)sc2c1 c1(C(=O)NC(CC)CNC(c2nccc(Cl)c2F)=O)cc(N)c(F)cc1F C1(C)(C(N2CC(CC)OCC2)=O)CCN(C(=O)CCc2ccc(C)cc2C)CC1 N1(C(CCOC(C)=O)=O)CCC(NC(c2ncoc2C)=O)CC1C1CC1 N1(C(C2C(CC)C2)=O)CC2C(CNC(c3cc(C)sc3C)=O)C2C1 C1(NC(C2(CC(F)F)CCC2)=O)(CNC(=O)C(O)C2CC2)CC(CO)C1 c1(CC)nc(C)c(C(=O)NC2CCOCC2C(=O)NCc2cc(OC)no2)o1 C1(C(=O)NC(C(C)NC(=O)CC2(N3CCCC3)CC2)=O)CCC1C#N C1(NC(=O)NCC(C2(OC)CCC2)OC)COC2(CCOC2)C1 C1(NC(C(CC=CC)C)=O)CCC(O)CN(C(c2cc(CCC)ccc2N)=O)C1 C1(CCC(=O)N(CCCNC(CSNC2CC2Cl)=O)CCC)CCCCC1 C(CCCCC(=O)NCC1CC1C(N1CCC(c2cnn[nH]2)C1)=O)OCC C(C(=O)NC(CO)C(C)NC(=O)CCCF)(C(C)(C)C)c1cccc(C)c1 CC(C)C(C#N)C(=O)N1C2CCC1(CNC(c1n[nH]cc1C(F)(F)F)=O)CC2 Cc1csc2ncnc(Nc3cccnc3C(N3CCOCC3C(C)C)=O)c12 c1(C(C)NC(CCOCCNC(C2(CC)COC2)=O)=O)ncc(C)cn1 CC1=C(c2ccco2)CN(C(=O)CC2(CN(C)C)CCCCC2)CC1 c1(C(N2CCC(C)C(NC(C3CCC(F)C3)=O)C2)=O)cc[nH]c2nccc1-2 N1(C(c2n(CC)cnn2)=O)CCCC(C2CN(C(C3(F)CCC3)=O)C2)C1 c1(C(NNC(CC2(C)CC2)=O)=O)cc(F)c(Cl)cc1F.c1ccc(F)cc1 c1(C(=O)NC(C)CC(C)NC(=O)C(Cl)=CCl)ccc(Cn2cccn2)cc1 C=CC1(C(=O)NOCCc2ccccc2)CCN(C(=O)C2=CC(C)(CC)C2)C1 O=C(CCCC(F)F)NCC(CNC(c1cn(CC2CCOC2)nn1)=O)CO C1(NC(CC2CCN(c3cc(C(C)C)ncn3)C2)=O)CCCS(=O)(=O)C1 C1(NC(c2nc(C(C)C)sc2)=O)CN(C(C2CCCCC2(F)F)=O)CC12CC2 c1(NC(C(CSC)NC(C(CCC)OC)=O)=O)cccc2c1OCO2 c1(CC(=O)OC(C(=O)O)C2CCCO2)ccc(Br)s1 N1(Cc2cccc(C(=O)OC)c2)CCc2c(OC)ccc(OC)c2C1 C1(NC(=O)CC2CCC3CC23)CC2CC(C1)N(C(C1CC3(C1)CC(O)C3)=O)C2 C(=O)(C(C)CCC(C)(C)C)N1C(CNC(C(C(CC)CC)C)=O)(COC)CCC1 c1(C(N2CC(C3(NC(C(CC)F)=O)CC3)C2)=O)ccc2cncc(Br)c2n1 C1(CC(=O)NCc2ccc(CC)s2)CC(C)(C)CN1C(c1nc(C)sc1C)=O C(=O)(C(C)(C)C(F)(F)F)NC(C(C)C)CNC(C1CCC(O)CN1C)=O N1(C(C(C)(C)Cc2ccc(Cl)cc2)=O)CCC(O)C(NC(=O)CCc2cnoc2)C1 C12(NC(CCCC)=O)CC(CNC(c3c(Cl)sc(C)c3C)=O)(C1)OC2C C1(C(N(C2CC(CCNC(C3C4CC(=O)CC34)=O)C2)C)=O)(CF)CC(F)(F)C1 c1(NC(C(CCCNC(C2CCC2(F)F)=O)O)=O)ccc2c(c1)CCC2 c1(C(=O)NCC2C(CNC(COC(C)=O)=O)C2)ccc(C)c2c1CCC2 c1(C(=O)NC(C2CCCCC2)CNC(C(C)C2CC2)=O)cccc2occc12 C(=O)(C(O)CCC(F)(F)F)N1CCC(OC)(CNC(=O)CC(C)C2CCCC2)C1 C1(CNC(C2CC3CC3N2C(=O)OC(C)(C)C)C)COC2(CCOCC2)O1 C=CCCCCCCC(=O)N(CCCC(=O)N(CCC=C)CC)C c1(C(=O)NCC(C)(CO)NC(C(CC)CC)=O)cnc2onc(C3CC3)c2c1 c1(C(=O)NC(C(N2CC(O)(C(=O)OC)C2)=O)C2CCCO2)ccc(O)cn1 c1(C(N2C(C(=O)NCc3ccc(Br)s3)CC(O)C2)=O)cc(Cl)cnc1Br C(=O)(CC(C)(C)CC(=O)NC(C)CC(C)NC(C1(NC(C)=O)CCCC1)=O)OC C1(NC(C(C)S(C)(=O)=O)=O)COC2(CCN(C(=O)Cc3ccc(F)cc3)CC2)C1 c1(C(=O)NC(CNC(C(CC)C2CCOCC2)=O)C)ccccc1COC Cc1cnc(C#N)c(-c2cnc(CC(=O)Nc3ccnc(Br)c3)nc2)c1 c1(NCCCCSC)nccc(=NCCCc2nncn2C)[nH]1 C12(C(N3CCC(CNC(c4c(C)noc4C)=O)C(C)C3)=O)CCCN(CCC1)C2 c1(C(N2CC(F)(CC)C2)=O)cc2c(F)cc(Cl)cc2[nH]1 c1(C(=O)NC)ccc(F)c(CNC(=O)NCCOC)c1.N12CCCCC1C2=O C(C)(C(=O)NC(CNC(c1sccc1-n1cccc1)=O)CO)(C1CC1)OC Cc1ccc(CCC(=O)NC2CCC(NC(c3cnn(CCF)c3)=O)C2)cc1C N1(C(c2c(CC)nco2)=O)CCC(CNC(=O)Cn2nc(CC)cc2C)C(C)C1 CC1C(NC(=O)C2=NOC(C)(C)C2)CC2CCC1N2C(=O)COCC1CCCO1 Cc1nc(C(C)C)ccc1C(N1CCCN(C(=O)CNC(N)=O)CC1)=O Cc1cc(C(N2CC(NC(=O)C(C)NC=O)C(O)C2)=O)c(O)cc1F N1(C(C2CC(SC)C2)=O)CCCC1Cn1cc(COCC2CCCO2)nn1 N1(C(CCC(CC)OC)=O)CCC(NC(=O)CC(F)(F)CC)CC(O)C1 C12(NC(c3c(C)oc(C(C)C)n3)=O)CCC(C1)N(C(=O)COC(C)(C)C)C2 C1(SC)CN(C(=O)C(C)n2cnnn2)CC1NC(=O)C(C)(C)c1cscn1 c1(NC(C2C(c3n(CC)cnn3)OCC2)=O)cc(C)oc(=O)c1 C1(CNC(C2CCN(C)C2)=O)CN(C(C2(CCN(C)C)CC2)=O)C2COCC2O1 c1(OC)nccc(C(N2CC(NC(C3(CF)CCC3)=O)CC2C)=O)c1F C(CC(F)F)(C(=O)NCC12CC(CCO1)C2)NC(c1c(CC)cncc1)=O C12(NC(CNC(C)=O)=O)CC3CC(C1)CC(CNC(C1CCCN1N=O)=O)(C3)C2 CCC(COC)C(=O)N1CC(CC(=O)NC2C=CC(C(=O)NC)C2)C(C)C1 CC(C)CC(C(=O)NCC(O)CN(C)C)ONC(=O)CCn1cccc1 c1(C(N2CCCC2c2nc[nH]n2)=O)csc(-c2ccc(C(F)(F)F)o2)n1 c1(CCC)nc(C)c(C(=O)NCC2CCCN(C(=O)CC(C)n3ccnc3)C2)o1 c1(CCNC(c2ccc(C(N(C)CC)=O)cc2)=O)c(Cl)cccc1Br Cc1nnccc1C(=O)NCCCN(C(C1CC2C=CC1O2)=O)C(C)C N1(C(c2cc(OCC)ncc2)=O)CCCC2(NC(C3CCC(C)(C)O3)=O)CC2C1 C1(N(C(CSCC=C)=O)C)CCC(CNC(=O)C(C)=CCC)C1 C12(C(=O)NCC3(C)N(C(C4C(C(C)O)C4)=O)CCC3)CCCCC(=O)N1CCC2 C(=O)(C#CC1CC(F)(F)C1)NCC(CC(C)C)NC(c1c(CC)c[nH]n1)=O N1(C(c2ccc(NS(C)(=O)=O)cc2)=O)CCC(CO)(NC(=O)C=C2CCC2)CC1 n1(CC)ncc(C(N2CCCC(N(CCO)C(c3n[nH]c(C)n3)=O)C2)=O)c1Cl N1(C(C2(Cl)C(C(C)=O)C2)=O)CC(C(=O)NOC2CCOC2)C(C)(C)C1 CC1(C)C(CC(N2CC(O)CC2CNC(c2cnco2)=O)=O)C1(C)C CC1CN(CCN2CCC(N(C)Cc3nccn3C)CC2)CCO1 c1(CC)nocc1C(=O)NCC1(NC(c2cn(CC3CC3)nn2)=O)CCOC1 C(=O)(C(C)N=[N+]=[N-])NC(C=CC(=O)N(C(C(C)SC)C)C)(C)C c1(C(N2C3(C(=O)NC4C(CC)CCCC4)CC(C2)C3)=O)nccc2[nH]ccc12 C(=O)(CC(CNC(c1ccccc1Cl)=O)OC)N(CC)Cc1sccc1C C(CCCC(=O)N1CCCC(C(C)NC(c2ccc(CN(C)C)[nH]2)=O)C1)SC c1(CN2CCC(C(C(=O)NCC)NC(=O)OC(C)(C)C)CC2)ccc(F)cc1F c1c2ccc(o2)c(=O)c(=O)c1.C1CCCC1O.C12CC(C1)N(C)C(=O)N2.CCO c1(NCCC2(CO)CC2)[nH]c(=NCc2cc(Cl)nc(=N)[nH]2)nc2scnc12 C1(O)(CC(=O)NCC(CC)(C)NC(=O)CCCc2cc(C)no2)CCCCCC1 C1(C(=O)NC(CNC(C2C(CC)CCCC2)=O)C(C)(C)C)C(C)OC(C)C1C N12CCCC(C1)OC2=O.n1(C(C(=O)NC)C)cc(C(N(C)CC)C)nn1 C(C)(N=c1[nH]c(=NCC(C)c2cccc(C(F)(F)F)c2)[nH]c2cc[nH]c12)c1c(C)non1 C1(C(CC)O)CCCCN1C(=O)C(CNC(=O)C(C)=C1CCCC1)OC CCC(C)C(CC(=O)NC)NC(c1cccn2nnnc12)=O C1(C(=O)NC2(C)CN(C(c3sc4ncn(C)c4c3)=O)C2)CCCCC12CC2(F)F C1(C(=O)NC2CC(C)(C)N(C(=O)Cc3ccoc3)C2)CC2CC(C1)CC(F)(F)C2 C1(C(N2C(C(=O)Nc3cncc(Cl)c3)CCCC2)=O)CCc2nc[nH]c2C1 C(=O)(C(CC)CCCC)NC12CN(C(C3(C=C)CCC3)=O)C(CC1)C2 c1(C(=O)NC(CC)C(=O)NC)ccc(CNC(=O)C(C)OCC2CC2)cc1 n1(CC)ccnc1C(C)NC(=O)C(=O)Nc1nc(C2CCCCC2)ns1 c1(OC)cc(C(N2CCCCC(CO)C2)=O)cc(-n2cccn2)c1 c1(C(=O)NC(CC(=O)N(CCCCCC)C)C2CC2)ncccc1N c1(CCCNC(CN(CCOC)C(C2CCCC2)=O)=O)cnn[nH]1 Cn1nnc2cc(C(=O)NC3(C4CCCN4C(C4CCCS4)=O)CC3)sc12 C(C1COC(C)(C)O1)=C.C1(C(=O)NC(C(C)C2CCC2)=O)(CN)CCCC1 O=S(=O)(c1cn[nH]c1)N1CCC(n2cc(C3NCCS3)nn2)CC1 C1(C(N2CC(=C)C2)=O)CC(NC(=O)CCN(C)C)C1(C)C c1(C(N2CC(COC)(NC(C3C=CCC3)=O)C2)=O)ccc(F)c(C(F)(F)F)c1F C1(CNC(Cc2n(C)nnc2)=O)CCC(C(=O)NCCCCCCF)CC1 CCC(CNC(=O)C(C)Nc1ccccn1)(CC)NC(=O)Cn1nc(C)cc1C c1(C(=O)OC)cnc(NC2CCCN(C(=O)C=CCN(C)C)CC2)c([N+](=O)[O-])c1 CCC(CCCC(=O)N1CCC(F)(C(N)=O)C1)NC(c1nc(C)oc1C)=O c1(CC(=O)NCCC(C)NC(C(COC)(C)O)=O)c(C)[nH]c2ccnn2c1=O C(=O)(C1CCCc2ccnn21)N1C(CCNC(CNS(NC)(=O)=O)=O)COCC1 N12CC(C)(C(F)(F)C1)C2=O.c1(OC(C)C)ccccc1OCC(=O)OC(C)(C)C C(=O)(CCCCN(C)C(C)C)NCC(COC)NC(=O)COC1(C)CCOCC1 c1(OCC(=O)NC(C(CO)NC(CC=C(C)C)=O)C)c(C)cc(Cl)cc1C c1(C(N(CC(O)CN(C)C(C2CCCC2CF)=O)C)=O)cc(C(N)=O)cc(F)c1 Cc1nc(N2CCC(C)(C)C(CNC(c3ccc(O)nc3)=O)C2)c2cc[nH]c2n1 c1(C(N(CCN(C(CC(C)OC)=O)C(C)C)C)=O)c[nH]c2cc(C)ccc12 N1(C(CCC)=O)CC(C)CCC1CNC(=O)CCc1ccc(OC)c(C)c1 c1(C(=O)NC(c2ccccc2)C(=O)NCC2CC(C)C2)ccc(=O)n(C)c1 C(C(C(=O)NC(C(C)C)C(C)C)C(C)(C)C)NC(c1c(CC)csc1)=O N1(C(C2N(C)CCC2)=O)CCC(F)C(NC(=O)CC#N)C1 c1(NC(C)=O)ccc(C(=O)NCC(O)CNC(C2CCCCN2C(N)=O)=O)cc1 C1(NC(c2c(C)n(C)cn2)=O)CC2CC(NC(C3CC3c3ccccc3)=O)C1C2 CC(C)(C#N)CCCC(=O)NCCCC1CCCCN1C(C1CCNC1=O)=O c1(N2CCCC(NC(CCC=C(C)C)=O)CC2)nc(C(F)F)nc2ccccc12 c1(C(C(=O)NCC)N(C(c2ccc3c(c2)OCO3)=O)CC)cnc2c(c1)CCC2 C=C1CC2(C1)CC(C(=O)N(CCNC(=O)CS(C)(=O)=O)C1CC1)C2 C1(CNC(C(CSC)O)=O)Cc2ccccc2CN1C(=O)CC1CSCCS1 C1(NC(C=COCC)=O)CN(C(c2sc(Cl)cc2Cl)=O)CCC1CO C1(NC(C(CCC)OC)=O)CC2CCC(C1)N2C(C1CCCCC1OC)=O N1(C(CONC(c2c(OC)nccc2)=O)=O)CC(CO)C2(CC2)C1 C1(C(=O)NCCOc2ccccn2)CC12CCN(c1cc(C(=O)O)ccn1)CC2 C1(CC)CCCCCCN1C(C1CCN(C(c2csnc2Cl)=O)C(C)C1)=O N1(C(c2c(CC)noc2C)=O)CC2(CCNC(=O)C(C)C3CC3)CCC1CC2 N1(C(c2ncc(C)c(Cl)c2)=O)CC(NC(C2CNC(=O)C2)=O)Cc2ccccc21 C1(CC)CCC(C(=O)NCCCN(C(c2cc(Br)n[nH]2)=O)CC)O1 Cc1cc(F)c(C(N2CCNCC2)=O)cc1-c1cccc(SC(C)(C)C)c1 c1(CC)ccc(C)cc1NC(C1(C(C)C)CCN(C(=O)CCC2CC2C)C1)=O C1(C(N2CCC3CN(C(c4ccnn4C)=O)C3C2)=O)(OC)CCC(F)(F)CC1 C1(NC(C(C)CO)=O)CN(C(c2cc(C3CC3)cs2)=O)C2(CCC2)C1 c1(C(=O)NCC2N(C(C3C(CC)C3)=O)CCC2)cnccc1Cl CC1C(O)CCCN1C(=O)CCC(C)(C)NC(=O)CC1CCCC12CC2 c1(C(=O)NCC2CC(NC(C3CC(O)C(F)C3)=O)C2)cc([N+](=O)[O-])cnc1O N1(C(C2(CN(C)C)CC2)=O)C2CCCC1CN(C(C1CC(O)CN1C(N)=O)=O)C2 c1(C(=O)NCCN(C(C(C)OCCC=C)=O)C)cnc2nccnc2c1 C1(C(=O)O)CCCCC1n1cc(Cn2cc(CC3CN(C(N)=O)C3)nn2)nn1 C(CCCCC(=O)N1CCCN(CCO)CC1)N(C(C(CCC)NC(N)=O)=O)C CN=c1cc(C(N2C3CCC(C3)C2C(=O)N(C2COC(C)(C)C2)C)=O)cc[nH]1 CC1(C)CCCC(C(N2CC3(CCCCN3C(=O)CCNC(N)=O)C2)=O)CC1 N1(C(C2C(C)OCCO2)=O)CC(NC(=O)CCOCC2CC2)C(C)(C)C1 C=CC(O)C(=O)N(C)CCN(C)C(c1cnc(N(C)C)o1)=O c1(C(=O)NC2CC(C(=O)Nc3c(C(C)=O)ccc(F)c3)C2)cc(F)c(Br)cc1Cl c1(C(=O)NC2CCCN(C(c3nc(C)sc3)=O)C2)cc2n(n1)CC(C)NC2=O CCCC(CCC)CC(=O)NC1C(C)CN(C(c2ccsc2)=O)CC1C c1(C(N2CC(C)(NC(c3cc(CCO)on3)=O)C2)=O)[nH][nH]c(=N)c1Br N1(C(C2(C)CCC2)=O)CCCC(O)(CNC(c2cncc(C#N)c2)=O)C1 CC1OC2(C(=O)NCC3(CCNC(C4(C)CC4(F)Cl)=O)CC3)CC1C2 CC(C)CC(CNC(=O)CC1(C)CCCCC1)C(=O)NCCn1ncccc1=O C=CC1COCCN1C(C1CNC(=O)CN1C(c1cc(C)c(C)o1)=O)=O n1(CC(N2CC(C)N(C(C3CCCN3N=O)=O)CC2)=O)nc2ccccn2c1=O Cn1ncc(C(=O)NCC2CN(C(=O)CC3CC3)C3(CCC3)C2)c1S(N)(=O)=O N1(c2cn(C)nc2)CCCC(NC(c2cn(C3CCCCC3)nn2)=O)C1=O CC(C)C(C(=O)NCC(CNC(=O)C(CO)N(C)C)CO)C1CCC1 C(C)(CNC(=O)COC1CN(C(=O)COC2CCC2)C1)(C1(C)CC1)OC c1(-c2cn(C(C(N3CC(C#C)OCC3)=O)CCC)nn2)ccc([N+](=O)[O-])nc1 N1(C(CC=CC)=O)CCCC(C)(CNC(c2cc(-c3ccoc3)on2)=O)C1 C1(C#N)(C(=O)NCCC2N(C(c3n(CC)ccn3)=O)CCCC2)CC2C=CC1C2 c1(C(=O)NCC2(NC(C(CC)O)=O)CCC2)cc2c(s1)CCC(C)C2 Cc1ccc(-c2cn(C3CN(C(=O)CN4C(=O)CSC4=S)C3)nn2)c(F)c1 C1(NC(c2ccc(CC)[nH]2)=O)CN(C(c2ccc(N)c(Cl)c2)=O)CC2(CC2)C1 N1(C(C(C)CO)=O)CCCN(C(c2cc(C3CCCO3)n(C)n2)=O)CCC1 c1(N(CCOCCN(C)C(c2ccc(Cn3ccnc3)o2)=O)C)ncnc(=N)[nH]1 CC1CN(C(=O)CCCCn2ccnn2)CCC1CNC(c1cc(CF)on1)=O CCCCC(C(=O)NCCC[Si](C)(C)C)NC(c1ccccc1CC#N)=O Cc1cccc(C)c1NC(=O)C(=O)NC1CCC1C CCCCC(C)C(=O)NCCN(C(=O)CCC(=O)c1cc(Br)cs1)C c1(-c2cc(NC(C)=O)c(C)cc2)nc2c(s1)CCN(C(C1(O)CCOCC1)=O)C2 C1(C(=O)NCC(CN(C(=O)CC(F)(F)F)C)O)NC(=O)C2CC12 N1(C(c2ccc(C)s2)=O)CC(C(=O)NCCCN(CC(C)C)C)CC12CCC2 c1(NC(=O)Nc2cc(C3CCOC3)ccn2)cc(F)ccc1Br c1(C(=O)NC(CNC(C2(COC)CC2(F)F)=O)C(C)C)ncc(C)cc1C CCC(C)(C)C(=O)C(=O)N1CCCCC1C1CCCN(C(c2ccc(C)s2)=O)C1 Cc1ccc(NC(=O)CSC(F)F)cc1S(=O)(=O)Nc1ccc(Br)cc1 c1(CN2CCC(C)(NC(CC3N(C)CCC3)=O)CC2)nc2cccc(F)c2[nH]1 c1(C(N2CCC(OCCF)C2)=O)cn(CCNC(=O)C(F)n2ccnc2)nn1 C1(F)(C(=O)NCC(N2CC(C)C2)c2ccco2)CC(N(C)C(C2(Br)CCN2)=O)C1 c1(OC)ccc2c(c1)C(NC(=O)C(c1ccc(F)c(Cl)c1)C)CC2 C1(NC(=O)Cc2noc(CO)n2)CC2CCC1(CNC(c1cccs1)=O)C2 Cc1nc2c(N3CC4CCC(C3)N(S(=O)(=O)CC3CC3)C4)ncnc2[nH]1 N1(c2ccnc(NC(C)Cc3ccco3)n2)CCCC2(CCOCC2)C1 C1(CC(=O)NC(CCC2CC2)C(=O)NC(CO)CCC2CC2)CCCC12CC2 c1(C(=O)NCC2N(C(C(COC)COC)=O)CC2)sc2ccc(F)cc2c1C N#Cc1ccc(C(=O)NC2(CNC(C3Cc4cscc4C3)=O)CCCC2)c(F)c1 CC1CCN(C(c2cc(C(F)F)cs2)=O)CC1NC(c1cc[nH]c1C1CC1)=O C(=O)(C(C)(C)C(C)O)NCC1C(CNC(c2ccc(SCCC)cc2)=O)C1 C1(NC(c2nn(CC)nc2C)=O)CC2CC(NC(=O)Cn3cc(C#N)cn3)C1C2 C1(C)(C(=O)NC2C(C(=O)NC(c3nc(=O)o[nH]3)C)OCC2)CCCN1C c1(NC2CC(CCNC(=O)C=Cc3ccccc3)C2)cc2nncn2cn1 N1(C(C2N(CCC)CCC2)=O)CCOCC(CNC(c2ccc(=O)n(C)n2)=O)C1 c1(OC)ccc(C(=O)N(CC(O)CN(C)C(c2cccc(O)c2Cl)=O)C)c(Cl)n1 C(C(=O)N1CCC1CNC(C1(N(C)C)CCCOC1)=O)(C(C)C)c1cc(C)no1 N1(C(c2cc(CCC)nc(O)c2)=O)CC2CCCC(NC(C3CC(C)C3)=O)C2C1 S(=O)(=O)(c1cnc(Cl)n1C)NCC(COC)Cl C(=O)(CC(C)NC(=O)N(C)CCN(C(=O)CCc1cnn(C)n1)C)NC(C)C C1(NC(c2cnc(C(C)C)o2)=O)C2CC3C(C2)C13C(=O)NCCn1cc(C)cn1 CCC(C(=O)OC)C(=O)NC1CN(C(=O)CC2(O)CCCN(C)C2)CC1C N1(C(c2c(CC)ncs2)=O)CC(CNC(c2c(C)nn(C)c2C)=O)C(C)(C)C1 C1(CNC(C(C2CCCC2)NC(C)=O)=O)CN(C)CCN1C(=O)CCC1CC1(F)F c1(COC)cncc(C(=O)NC2(CNC(C3(C)CC3(F)Cl)=O)CCC2)c1 C1(CNC(c2cnc(C)s2)=O)CN(C(c2coc(Br)n2)=O)CCC12CCOC2 N1(C(c2c(COC)ccs2)=O)CC(NC(=O)CSc2ccc(O)cc2)CC(O)C1 C1(C(=O)NCCc2cc(C(=O)NCCn3nncc3C)no2)(CC)CCCO1 N1(C(CCNC(C2(C)CCSCC2)=O)=O)CCc2ccccc2C1 CCC(C)(C)C(C)CC(=O)NC1CN(C(c2ccc(Br)c(F)c2C)=O)C1 C=CCC(CC=C)C(=O)NC(C(=O)NC(C)Cc1nncn1C)C1(C)CC1 c1(C(=O)NCC(N(C(=O)CC2CC2(Cl)Cl)C)C2CC2)ccn(CC(F)(F)F)n1 CON1CCC(C(=O)N(CCCNC(C2(C)CCN(C)C2=O)=O)C2CC2)CC1 c1(C(=O)NCC(C)(C)NC(=O)COC2CCOC2)cc2ccc(F)cc2[nH]1 C(c1ccccc1F)=CC(=O)N(CCCCCC)CCNC(=O)CC1(O)CCC1 C(=O)(C(C)(C)CN1CCCCC1)NC1N(C(C2(COC(C)(C)C)CC2)=O)CCC1 N1(C(c2c(C)ncc([N+](=O)[O-])c2)=O)CCC(C2CCCN(C(=O)CO)CC2)CC1 C#CCCN=C(NCc1nc(C(C)(F)F)cs1)N1CC(C)CC(C)(C)C1 C(C(O)CCNC(C1CCCC1C)=O)NC(C(OCC)OCC)=O Cc1nc(-n2nc(CCCO)nc2-c2cscc2Cl)n(C)n1 C(=O)(C(C)CCNC(C1CCC(C)N1C(=O)CCn1cnc(=N)[nH]1)=O)OC C1(N(C(C(C)Cc2cnc[nH]2)=O)C)CCCCN(C(=O)Cn2cccc2)C1 CC1CCCN(C(C2(CNC(c3cnn(CCN(C)C)n3)=O)CCCCC2)=O)C1 N1(c2c(OC)cnc(Cl)n2)CCCC2(NC(c3ccc(C(C)(C)C)[nH]3)=O)CC2C1 Cc1ccc(CCNC(=O)CNC(c2nc[nH]n2)=O)nc1 Cc1cc(NC(C2CC(C)(Nc3ccncn3)C2)=O)c(Cl)cc1Cl S(=O)(=O)(c1cnn2ccc(=NCC(c3cccs3)N(C)C)[nH]c12)N(C)CC C(C)(C)(C(=O)NCC(C)CNC(=O)CN1CC2CC2C1)OC(C)C C(=O)(CCCN(C(=O)C(C)(C1CCC1)NC(C1CCN1C)=O)C)OCC N1(C(C(C)N(CC)CC)=O)CC(C)(C)OCC1CNC(=O)CSC(F)F C1(CC(=O)NCCC2CC(NC(c3ccsc3Cl)=O)C2)CC2CC2C1 O=C1CC(C(=O)NC(Cc2cc[nH]n2)C(=O)NCC2CC23CCC3)CC(=O)N1 N(C(=NCCC(=O)NC)NCc1cnc(C)s1)CC(=C)C c1(C(=O)NCCC2([N-]C3CC3)CC2)sc(Br)cc1C.C1(C2CC2)C(=O)CO1 C1(NC(c2cnc(C(C)(C)C)s2)=O)COC2(CCN(C(=O)CC3CCOCC3)C2)C1 C(CC(C(=O)Nc1cnc(SC)nc1)NC(=O)C(F)F)OCC c1(C(N2C(C)(CNC(c3ccc(Br)o3)=O)CCC2)=O)nc2ccccn2c1F C(=O)(CCC(CC)OC)N(CCCC(=O)N(C(C(CC)(C)C)C)C)C c1(C(=O)NCCCOCCNC(C2C(C)OCCC2)=O)cccc2[nH]cc(Cl)c12 Cc1cc(C(=O)NCC23CC2CN(C(c2ccoc2Cl)=O)C3)cc(C)c1F C1(CNC(C2C(C(C)O)C2)=O)(NC(c2cnc(Cl)[nH]2)=O)CCCC1 N1(CC(=O)N(C)CCNC(c2cn(C3CCCC3O)nn2)=O)OC(C)(C)CC1=O C1(C(=O)NC(C2(O)CCN(C(c3cc(C)sn3)=O)C2)C)CN(C)CCN(C)C1 c1(C(N(C)CC2CCN(C(=O)COCC3CCC3)C2)=O)cc2ccoc2cc1F C(=O)(C1=C(Cl)CCOC1)NC1CCN(C(C(C)CC(F)F)=O)C1(C)C c1ccc2c(c1)CCCC2CNCc1nnnn1-c1ccc2c(c1)OCCO2 C(=O)(C1=CCSC1)NCCC(=C)CNC(c1csc(C(N)=O)n1)=O c1(C(=O)NC2CCC(NC(c3c(CC)ccs3)=O)C2)cccc2c1COCC2 c1(C(=O)NC(CC)CN(C(=O)CC(C)C(C)C)C)ccc2cnsc2c1 c1(CNC(c2ccc(-c3ncco3)cc2)=O)nc2ccccc2n1C(F)F C1(C(=O)OC)CCCCN(C(=O)C(c2cccnc2)NCCC(F)(F)F)C1 c1(N2CC(CCCCN(C(C(C)O)=O)CCO)C2)c(Cl)cncc1[N+](=O)[O-] C1(CNC(c2ccc(OCC)cc2)=O)CCN(C(c2cc(F)c[nH]2)=O)CC1C c1(C(=O)NC(COCC)C(=O)Nc2ccc3c[nH]nc3c2)ccc2occc2c1 N1(C(C2C(C)=C2)=O)CCCC(C2CN(C(c3ccc(S(C)=O)cc3)=O)C2)C1 C1(CNC(CC(C(C)C)C)=O)CN(C(=O)Cc2ccns2)CCC1(F)F N1(C(c2ccc(SCC)cc2)=O)CC(NC(=O)CNC(=O)NC)CC(O)C1 c1(NC(CNC(=O)C=CSCc2ccco2)C2CCC2)nccc(CC(=O)OC)n1 C(=O)(C(C)(C)C(=O)N(C)CC1CCCC(NC(c2ncn(C(C)C)n2)=O)C1)NC CCC(CC(=O)N1CCC(N(C)C(C2CCNC2=O)=O)C1)OC Cc1nnc2n1CC(C(N1CCC(C)(NC(c3cc4ccccn4n3)=O)C1)=O)C2 S1(=O)(=O)c2cc(Br)ccc2ON1.C12(C(=O)OC)CCC(CCCC(=O)O)(C1)OC2 C(=O)(C(F)CCC(C)(C)C)NCC(CCC)NC(c1cccc(CC#N)c1)=O Cc1nc(C(F)(F)F)ccc1S(=O)(=O)NCCCS(=O)(=O)CC N1(C(c2c(COC)noc2)=O)CCOCC(NC(c2cnccc2C)=O)C1 C1(C(=O)OC)C2C=CC(CC2)C1C(=O)NCC1(c2ccccc2)CCOC1 CC(C)(C)C(O)CCC(=O)NC1CC(CNC(C23CCC(C)(C2)OC3)=O)C1 c1(C(C(=O)N(C(C=CC(C)(C)C2C(C)C2)=O)CC(F)F)(C)C)cccc(Cl)c1 c1(C(=O)NC2C(NC(c3ccc(Cl)s3)=O)C2)cnc2n1CCCC2 C1(C(N2CCC(NCCOCCNC(COCCC)=O)C2)=O)CCC(C)(C)OC1 C1(CC(=O)NC2CCN(C(=O)C=Cc3cccnc3)CC2)CCCC(=O)N1 N1(C(COC2(C)CN(C(C3CCCCC3F)=O)C2)=O)CCC(C)(C)CC1 N1(C(CCC(=O)NC)=O)CC2(CC(C(N3CC4(CC(C(F)F)C4)C3)=O)CO2)C1 c1(OC)ccc(C(=O)NC2(C(=O)NCCC3(OC)CCC3)CC2C)o1 N1(C(CN(C)C2CC2)=O)CC2CC(C(=O)NC3CN(C4CCC4)C3)C(C2)C1 CC(CNC(=O)CCc1cncs1)(CO)NC(=O)CC1(C)CCOC1 c1(C(N2C(C(N3CCCC(C)C3)=O)(COC)C=CC2)=O)coc2ccccc12 CCC(C)CCCCC(=O)NC1CC2CN(C(c3cc(Cl)ccc3N)=O)CC12 C(=O)(C1c2ccnn2CCN1N1CC2(C1)OCC1CC21)OCC C(=O)(C(C(C)(C)C)C1CCCCC1)N(C1CCCCN(C(C2CC(O)C2)=O)C1)C C(CC(=O)NCC(C)C)NC(C=CC(C)N(C)C)=O Cc1ccc(C(N2CCC23CCOC3)=O)c(N)n1 C1(C(=O)NCC2(NC(COCCCC)=O)CC2)Cc2nccn2C1 C1(CC)CN(C(=O)CN(C2CCC2)C)CCC1NC(c1cc(OC)no1)=O C(=O)(CCS(N)(=O)=O)N1CCCC(N(C(Cc2c(C)n(C)cn2)=O)CCO)C1 c1(C(=O)NC(C2CCCN2C(c2ccccn2)=O)C)ccc([N+](=O)[O-])cc1 CC1OC2CCC1(C(=O)NCCOCCN(S(=O)(=O)Cc1ccon1)C)C2 C(=O)(C(O)CCNC(=O)C=C(C)c1ccco1)NC(C#C)(C)C1CCCC1 C(=O)(C(F)C(C)CNC(C1CC2(CCC2O)C1)=O)N(C)Cc1ccc(C)cc1 CCCCC(CNC(=O)CCOc1cccnc1)NC(=O)COC1CC1(F)F C(C(F)(F)CC(O)CO)N(C(c1cc(C2CC2)ns1)C(=O)NCCCSC)C c1(C(=O)NC(C)CCCNC(=O)C=CSCc2ccco2)cc2c(ncn2C)[nH]1 N1(C(C(CCC2CCC2)NC(c2c(C)csc2)=O)=O)CC2(C=CCO2)C1 c1(CN2C(C(=O)NCC(C)(C)CC3CC3)COCC2)cc2ccccc2nc1O C(=O)(CCC(=O)NC1CC2(C1)CC2NC(=O)Cn1nnnc1C)NCC c1(C(N2CC3(CC(NC(=O)CO)C3)C2)=O)cn2ccnc2cn1 C1(C(=O)NC(C)CNC(C2CC(n3cnnc3)C2)=O)CCOCC1(C)C c1(C(=O)NC2CCN(C(CC(CC)O)=O)CC2F)cc(Br)cc2c1cnn2C n1(CC(=O)NC2CCCC(NC(c3cc(OC)ncc3)=O)C2)nc(O)ccc1=O CC(c1cnn(C)c1)=CC(N1CCCC(N(C(=O)CC2CCSCC2)C)C1)=O N1(C(CCN(C)CC)=O)CCOC(C(N2CC(C(=O)N(C)C)C2)=O)CC1 c1(CC(CN(C)Cc2cc(C3CC3)n[nH]2)=O)ccc(C(F)(F)F)cc1 O=C(C1=CCCS1)NCc1ccc(CNC(c2cc(F)cs2)=O)cc1 c1(C(N2CCC(OCCNC(c3nccc(N)c3)=O)C2)=O)ccnc2c1CCO2 C1(CN(C(COC(C)C)=O)C)CCCC(CNC(C2(C3CC3)CCC2)=O)C1 C(=O)(CCP(C)(C)=O)NC1CC(N(C)C(C23CC(c4ccccc4)C2C3)=O)C1 c1(C(=O)NC2CC(SCC)C2)[nH]ccc1COC.c1(CC(=O)N)ccccc1 CC(C)C(CN(C)C)C(=O)NCC1(CNC(=O)C2=CCCC2)CCOCC1 N(C(=NCCC1CC1)NC1CC1(C)C(F)F)C(C)C.C1(C)CC1C C(=O)(N1CCC(NCCN2CCCC2)O1)C1C(C)CC1 c1(C(=O)NC2CCCN(C(C3(N(C)C)CCC3)=O)CC2)cccc2c1OCO2 C1(NC(C2(COC(C)C)CC2)=O)CCC(NC(=O)CCCC2CCOCC2)CC1 c1(C(=O)NCCC(C)N(C)C(c2cccnn2)=O)c(O)cnc2ccccc12 C(=O)(CCC1=CCCCC1)NC(C(C)C)CC(=O)NCCc1ccccn1 c1(-c2cn(Cc3ccc(OCC)nc3C)nn2)cnn2c1CNCC2 C1(CC(=O)NC2(CN(C(c3cc(C)no3)=O)C)CC2)CC(C)(C)OC1=O C(=O)(CCCC(=O)c1ccccc1)NCCC(=C)CNC(=O)C(C1CC1)OC N1(C(C2CCC(C)N(C(=O)OC(C)(C)C)C2)=O)CCN(C)Cn2nccc21 S(=O)(=O)(c1cnn2ccc(N3CCN(CCF)CC3)nc12)NCCCC=C c1(C(N2CC3=C(CN(C(C4N(C)CCC4)=O)C3)C2)=O)cnn2c1OCC(F)C2 c1(CC)onc(C)c1CNC(C1C2CN(C(=O)C(C)(C)OC)CC12)=O C(=O)(CCCCCNC(C)=O)N1CC(C(C(=O)NCCc2cccnc2)OC)C1 C(=O)(CCCC(=O)NC1CC2(C1)CC(NC(C1CC3(CCCC3)C1)=O)C2)OC c1(C(=O)NCCC2CCCN(C(c3ccccc3O)=O)C2)c[nH]nc1[N+](=O)[O-] N1(C(CC(CC#C)NC(=O)CC2CCCN2C)=O)CCCC(F)(F)CC1 n1(CC(=O)NC2C3CN(C(C(C)SC)=O)C2C3)ccc2ccccc2c1=O C(CCC(C)(C)C(=O)Nc1cncc(F)c1)NC(C1C(C)C1)=O c1(-c2nc(CC)on2)ccc(CN2CCC(C(=O)Nc3cncnc3Cl)C2)cc1 N1(C(C(C(CC)C)=O)=O)Cc2ccc(CNC(=O)CCS(N)(=O)=O)cc2C1 N1(C(c2cc[n+]([O-])cc2)=O)CC23COCC2(COC3)C1 CCCCC(CC)CC(=O)NCC1CN(C(c2cccc(OC)n2)=O)CCC1C CC(C)CCCCC(=O)NC1CCC(CNC(=O)Cc2cnns2)C1 C(=O)(C(CC(C)C)ONC(=O)C=C=C(C)C)N(CCCOC)CCO c1(SC)cc(F)ccc1C(=O)NC1CN(C(=O)C(C(C)C)N(C)C)CC1SC Cc1cnc(C)c(NC(C2C3CC3CN2C(=O)C(C)NC(c2cccs2)=O)=O)c1 C(=O)(C(C)(C)C(=O)NCC1CC2(CC(NC(=O)C(C(C)C)SC)C2)C1)NC N1(C(C(C)NC(=O)NC)=O)CCCC2C1CCN2C(=O)Cn1cc(C(C)O)nn1 N1(C(C(CNC(C(C)(C)OCCC)=O)CCC)=O)CCC2(COC(=O)N2)C1 c1(SC)ccccc1CN1CC(NC(=O)Cn2cc(-c3ccc(CN)s3)nn2)C1 c1(NC(=O)CC2(OC)CN(C(=O)Cc3cscn3)C2)ccc(OC(F)(F)F)cn1 c1(C(=O)NC(CNC(CCC=C=C)=O)(CC)CC)cnc2n1C(C)CCC2 c1(OC)cc(CNc2cccnc2C(=O)NC(c2cnccn2)C)cc(Br)c1O c1(CC)cc(C(N2CCOCC2CNC(=O)C(C)n2cccn2)=O)c(C)o1 C1(CNC(c2c(NC)cncc2)=O)CN(C(=O)CCC(C)(C)N(C)C)CC1(C)C N1(C(C2C(C)OCCC2)=O)CC(NC(c2cc(Cl)n[nH]c2=N)=O)CC(F)(F)C1 N1(CCCNC(=O)NCc2nc(-c3ccncc3)cs2)CCCC1=O [N-]=[N+]=Nc1ccc(C(N2CC3C(CNC(C4CCSC4)=O)C3C2)=O)cc1 c1(C(=O)NCCNC(C(CN(C)C)O)=O)ccc(F)c(Sc2cccc(Cl)c2)c1 N1(C(COCC=C)=O)CCCC(NC(C2C(C)C2(F)F)=O)CC1 N1(C(C=C(CCC)CCC)=O)CC(=O)N2CCOCC2(CNC(=O)CC(C)F)C1 c1(OC)ccc(CCC(N2CCC3(NC(=O)CC=C(Cl)Cl)CC3C2)=O)cc1OC Cc1nn(C(C)(C)C)cc1C(=O)NCCOCCCN(C)C(C1CC=CC1)=O C(=O)(CC1OCc2ncccc21)NC(C#C)C(C)OC C1(NC(c2csc(-c3ncccc3Cl)n2)=O)C=CCN(C(C2CC=CCO2)=O)C1 c1(N(CCC)Cc2ccncc2)[nH]c(=NCCC2CCCCC2)nc2sccc12 CC(C)(C(=O)N1CC2CCC1C(NC(=O)C=Cc1ncc[nH]1)C2)C(F)(F)F O=C(C1=CC2(CN(C(c3ccncc3F)=O)C2)OC1)NCC1CC1(Cl)Cl C1(CNC(CCc2cnn(C)n2)=O)CCCCC1NC(c1cc(C(F)F)[nH]n1)=O C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NCC(C)CNC(=O)CCOC1CCC1 n1(CCCC(=O)NC2CCN(C(C(C)(C)c3cncnc3)=O)C2)cnc(C#N)n1 C1(NC(C(C)SCC)=O)CCCN(C(c2cc(C)ccc2O)=O)C1C C1(C(=O)NCC2N(C(c3c(C)ccc(C)n3)=O)CCC2)Oc2ccccc2C1C c1(C(N2CCC3(C(C(=O)NC(CCC)C(=O)OCC)C3)C2)=O)ccc(F)cc1C CC1(C)CCN(c2ncc3ccnc-3[nH]2)CC1CNC(=O)CCCC1CC1 CCC(C)(C)CC(=O)NCC1(c2cnn[nH]2)CCN(C(=O)C#CC2CC2)C1 c1(C(=O)NC2CC(C)(NC(C(C)OCCCC)=O)C2)ccc2c(c1N)CCCC2 Cc1cc(C(=O)NC2CCC2NC(=O)CCc2ccon2)c2n[nH]cc2c1 C(=O)(C(S(C)(=O)=O)C1CC1)NC1C(NC(c2c(OC)n[nH]c2)=O)CCOC1 C1(C)(C(N2CC(C)C(NC(=O)CCS(C)(=O)=O)C2)=O)CC(O)CN1C C1(NC(C(CCN(C)C)NC(=O)C(F)CC2CCOC2)=O)CC2(C1)CC(C#N)C2 c1(OCC)ccccc1CN1CCC(CNC(=O)CCc2ccc(Cl)cc2)CC1 C(=O)(C(C(C)(C)C)NC(c1ccc(CO)nc1)=O)N1C(CCC#C)CCC1 CCC1=C(C(=O)NCCC2CC(NC(c3cn(CCO)nc3C)=O)C2)CCCO1 C(=O)(C1=NN(c2cccc(F)c2)C(=O)CC1)NCC(Cc1ccc(OC)cc1)C c1(C(N(C2CCN(C(c3ncsc3C)=O)C2)CCC)=O)ccc2ncsc2c1 CC1CN(C(C2CN(CC(F)(F)F)C2)=O)CCN1C(=O)Cn1cncn1.C1CC1 CCCC(C(=O)N1CC2CCC1CN2c1cc(Cl)ncn1)C(C)C c1(C(=O)NCC(C)NC(C(N2CCCCC2=O)C)=O)cc(-n2cnnc2)ccn1 N1(C(c2cnc(C)nc2C2CC2)=O)CCCC2C1CCN2C(=O)CC1CC12CC2 C1(CC(=O)OCC(C)(C)S(C)(=O)=O)CCc2ccccc2C1 S1(=O)(=O)c2ccc(cc2)N1CC(C)(C)N.C(C(N)=O)NC(=O)C1CC1 C1(C2(O)CN(C(C3CC3CN(C)C)=O)C2)(CNC(C2OCCC(C)C2)=O)CC1 n1(CC)cc(-c2cnc(C(N3CCC(N4CCN(C)CC4)C3)=O)cn2)ccc1=O c1(OCCC)ccnc(C(=O)NCCNC(C2CC2c2ccc(Br)o2)=O)c1 CN1C(=O)COc2ccc(-c3nc(C4(C)CCCO4)no3)cc21 C1(CCN=C(NC(C=C)C)NCC2(C)CCC(=O)N2)Cc2ccccc2C1 CCC(C)C(C(=O)NCC(C)(C)NC(C1C(F)(F)C12CC2)=O)NC(=O)OC c1(CC(=O)NCC2C(NC(CCN(CCCCC)C)=O)C2)cn(C)nc1C(F)F C1(NC(CCCNC(=O)OCC)=O)CCCC(CC(=O)NC2CCCNC2=O)C1 C1(CC(=O)OC)CCCCC1C(=O)NC1CCN(C(=O)CCc2ccn(C)n2)C1 c1(C(N2C(C)CCC(NC(=O)C=CCOCCOC)C2)=O)ccn2cnnc2c1 N(C(=NCC1CCCNC1=O)NC1CCOCC1)Cc1onc(CC)n1 c1(C(=O)OCC)ccnc(F)c1NC(=O)CCC(N)=O C1(CCNC(c2nc(C)[nH]n2)=O)CCCN(C(=O)C(C2CCOCC2)F)C1 N1(C(C(C)NC(C)=O)=O)CC(CNC(=O)Cc2cncc(C)c2)C(O)C1 C(=O)(C1=NOC(C)C1)N1CC(C=C)(CC(=O)N(C)Cc2ccon2)C1 C=CC(C)CC(=O)NCC1CCCC(CNC(=O)CCSCc2ccccc2)C1 C=CCC(CC)C(=O)NCCC1CCC(NC(=O)COCCOCC)C1 N1(C(c2c(OCC)nccc2)=O)CCC2CC1CN2C(c1nnc(O)nc1O)=O N=c1[nH]c2ncc(C(N3CC4CCCC4(NC(=O)CC4(CO)CC4)C3)=O)cc2s1 c1(C(=O)NCC(=C)CCNC(c2nccn2C)=O)onc2ccccc12 C(=O)(C(CC1CC1)NC(=O)C(C)N)OC C(=O)(C(C(C(C)C)NC(=O)OC(C)(C)C)N1CCC(C)C1)NCCSC C1(NC(COCCCC)=O)CN(C(C2CCC3CC23)=O)C2(CCC2)C1 Cc1nc(CNC(=O)NCC2CCOC(C)C2)nc2c1CCCC2 c1(C(=O)NC2C(CNC(Cc3nc(C)sc3)=O)C2)cc(S(N)(=O)=O)sc1C C(=O)(CCCC(C)(C)C#N)N(CCC(=O)NC1CCCC(O)CC1)C CC1CCSCCN1C(C1C=CCCN1C(=O)CC1(C)CCOC1)=O C=CCCC(CC(C)C)C(=O)N1CCC(OCCNC(=O)C(CC)(CC)CC)C1 C(=O)(C(C)CC(=O)c1ccccc1)c1ccc(CCCCCC)cc1 c1(CN(C(=O)NCc2c(OC)c(Br)cc(Br)c2)C)cc(C)cc2c(C)c(C)[nH]c12 C#CCCCCCCC(=O)N1CCCC1C=CC(=O)N(CC(C)O)C CC1CN(C(c2cncc(O)c2)=O)CC1C(N1CCOCC1C(N)=O)=O c1(C(N2CC(C(C(=O)N(C)CCN(C)CCO)OC)C2)=O)ccc(Cl)o1 c1(OC)cc(C(N2CCC(NC(=O)C(C)C)C2)C(=O)NCCSC)c(F)cc1Cl N1(C(c2c(N)cnc(Cl)c2)=O)CCCC2(NC(=O)Cn3ncnn3)CCCC12 N1(C(C(CC=C)C)=O)CCC(NC(=O)CCC(C)(C)F)C(C)C1 C1(CNC(C(C)(C)N2CCCC2)=O)CC(F)CN1C(=O)C=CCN1CCCC1 c1(C(=O)NCC2(OC)CCN(C(C3C=CCC3)=O)C2)ccc(C)c2ccccc12 C(=O)(CS(=O)(=O)C1CC1)N1CCCC(NC(c2c(Cl)nc(OC)s2)=O)(CO)C1 CCC(CC(=O)NC(CC(=O)N(C)CCc1cnn(C)c1)C1CC1)C1CC1 CC1CC(C(=O)NCC2(C)CSC2)CN(C(c2nnc(S)n2C)=O)C1 c1(OCC(=O)N(CCNC(C2CC(Cl)(Cl)C2)=O)CC)ccccc1Br S(=O)(=O)(c1cc(C)cnc1NCC1(CO)CC2CCC1CC2)N(CCCSC)C C1(C(N2CC(O)(CCNC(C=C(CC)C)=O)C2)=O)CC2C=CC1C2 C(=O)(C1=CCN(C(=O)OC(C)(C)C)C1)NC(C1N(C(C2C(C)C2)=O)CC1)C1CC1 c1(C(N2CCN(C(c3ccc(C)nn3)=O)C3C2C3)=O)cnc2ccccn2c1=O CC(C)(CO)C(=O)NC1CC(NC(C2CCNC2c2ccccc2)=O)C1 n1(CC(=O)N(C2CCN(C(=O)CC(C)F)C2)CCC)nccc1-c1ccccc1 c1(OCC)cc(C(=O)NC(C)(C)C(C)NC(C2CC23CC3)=O)on1 c1(CC(=O)NCCOCCCNC(C2C(C(N)=O)CC2)=O)c[nH]c2cnccc12 CCCC(CCNC(C1(CC)CCN(C(=O)CCSC)CC1)=O)CCC C(CCC(C)(C)NC(=O)CCc1scnc1C)NC(CSCC#C)=O C1(NC(c2c(CC)scc2)=O)CN(C(=O)C(c2ccc(F)c(F)c2)O)CC12CC2 c1(C(=O)NC(CC)CN(C(=O)C(O)CF)CC)ccc2c[nH]nc2n1 CC12COCC1CN(C(=O)C(=O)Nc1cncc(F)c1)C2 N1(C(C(n2cc(CC(CC)C(=O)O)nn2)C)=O)CCC(C(F)(F)F)(C(=O)O)CC1 C1(C(N2CCC(OCC(C)C)C2)=O)CN(C(=O)CC2CC(C)=NO2)CC(C)(C)C1 C1(C(C)=O)CCN(C(=O)CNc2cccc(OC(=O)CC3CCCC3)c2)C1C c1(CC2CN(C(CCCNC(=O)OC(C)(C)C)=O)C2)cc(I)ccc1Cl N1(C(C(C)OCC(C)C)=O)CC2CC1CN(C(=O)Cc1noc3ccccc13)C2 C1(N=[N+]=[N-])(C(=O)NCC2(CNC(C3C(C)CC3)=O)CCC2)CCOCC1 c1(OC)ccc2cc(C(=O)N(C)Cc3nc(CC(F)(F)F)no3)sc2c1 COC1CCOc2c(OCN3CCC(F)(F)C4(CCOC4)C3)cccc21 N1(C(=O)C(O)c2cnc[nH]2)CCCN(C(C2(N3CCOCC3)CCCC2)=O)CC1 C1(C)(CNC(C2(SC)CC2)=O)CCCN1C(=O)CCN1CCC1 C(=O)(CCC(C)CN(C)C)NC(CC)C(N1CCC(OC)C(F)C1)=O N1(C(C(F)=CCC)=O)CCC2(CC1)CN(C(c1nocc1Br)=O)C2 C1(CC(=O)NCC(CN(C(C2(F)CC(C(=O)OCC)C2)=O)C)C)CCC12CCC2 Cc1nsc(CN(C(=O)C(C2CCN(C(c3cncn3C)=O)C2)F)C)n1 C1(C2CCN(C)CC2)(NC(C(c2cccc(C)c2)N)=O)CC1 n1(CC)ccc(C(=O)NCC2(NC(c3cc(C(F)F)no3)=O)CCOC2)n1 C1(CC(=O)N(C(c2ccccc2)C(=O)NC(COCC)CO)CC)CCN(C)C1=O CC1CCn2ncc(C(N3CCN(C(c4cnccc4Cl)=O)C(CF)C3)=O)c2C1 C1(NC(C(C)CC2CC2)=O)CC2(C1)CC(NC(=O)C(c1cccnc1F)(C)C)C2 N12CCC(CC1)NC2=O.C1(C(C)(C)C)(NCCOC(C)C)CCCC1 N1(C(C(CC#CC)NC(C2CC(C)=NO2)=O)=O)CCCN(C)C(=O)C1 C1(C(=O)NC(CNC(C)=O)(C)C)CCCCCC1NC(=O)C1=CCSC1 n1(CC)cc(C(=O)NC(CNS(C)(=O)=O)C(=O)NCCSC)nn1 N#Cc1cc(S(=O)(=O)NCC2CCCCC2)ccc1NCc1c[nH]c(=N)s1 N1(C(CCC(C)O)=O)CC2(CCOCC2)CC1CNC(c1ccccc1Cl)=O N1(C(c2c(C)cns2)=O)CCCC(Cn2cc(C3CCCC(C)C3)nn2)C1 CC1CN(C(=O)NCC(F)(F)CN2CCOCC2)C(C)CCO1 c1(C(N2CC=CC(NC(c3nc(C)c(C)s3)=O)C2)=O)cccc(OC(C)C)c1Cl CCCC(C(O)C(=O)N1CC(N(C)C)C(C)C1)NC(=O)Cc1ccc(C)o1 C1(NC(C(C2CC(NC(C=NOC)=O)C2)F)=O)CCCCC1N=[N+]=[N-] N1(C(C2CC(C)C2)=O)CC2(CCCCN(C(=O)C#CC3CCOC3)C2)C1 c1(NC(=O)OC)ccc(C(=O)NC2CC(CNC(=O)Cc3csc(C)n3)C2)cc1 [N-]=[N+]=NCCCCCC(=O)NC(C1CC=CCC1)C(=O)NCCCn1cnnn1 CC1=NOC(C(=O)N(CC(C)N(C(=O)CCOc2cccnc2)C)C)C1 N1(C(C(CCOC)NC(=O)C(C)OC)=O)CC(F)CC(F)C1 C1(NC(CCNC(CC(C)C)=O)=O)CN(C(c2cc(Cl)ccn2)=O)CC1O C1(C(=O)NC(CNC(c2cc[nH]c2C2CC2)=O)C2CC2)(OC)CCC12CCC2 C1(C(C)C)CN(C(=O)C=CC2CC2)CCN1C(c1ccc(N)cc1O)=O N1(C(Cc2cc(C)cc(F)c2)=O)CCCN(C(=O)C(O)CC(N)=O)C(C)C1 N1(C(C(C2CCCC2)NC(C)=O)=O)CCC2(CCN(C(C3CCCCO3)=O)C2)C1 C(=O)(CCCC(=O)N1CCOC(C(C)NC(=O)CNS(C)(=O)=O)C1)N(CC)CC c1(CC)cnc(O)c(C(N2CC(NC(=O)CC3CCOC3(C)C)C3(CC3)C2)=O)c1 c1(CN2CCC(C)(C(=O)NCC(C)OC)CC2)cc(F)c(Cl)c(F)c1 N1(C(c2c(C)ccs2)=O)CCCCC1CC(=O)NCCOc1ccccc1 N1(C(CC2C(C)OCC2)=O)CC(O)(C2(CNC(=O)CCC(F)(F)F)CC2)C1 C1(NC(c2csnn2)=O)CC2CN(C(=O)C(c3ccc(Cl)nc3)(F)F)CC2C1 c1(NC(C23CC(C(NC4=NCCS4)=O)(C2)C3)=O)ccc(-c2ccccc2)nc1 C1(NC(C=NOC)=O)CC(C)CN(C(=O)CCc2csc(=N)[nH]2)C1 CC1(C)CN(C(C23CC(C#N)(C2)C3)=O)CCC1C(=O)NOCCCC1CC1 C1(C(N2C(CN(C)C)CCCC2)=O)CCC2(CC2)N1C(c1ccc(=O)n(C)n1)=O c1(CNC(c2sc(C)c(O)n2)=O)c(C)nn2c1CN(C(c1sccc1Cl)=O)CC2 c1(CC)cnccc1CNC(=O)CC1(NC(c2conc2C(=O)OC)=O)CC1 n1(CCC(=O)N(CCN(C)C)CC2CC2)cnc2c(N)ncnc12 O=C(CCC1=CCCCC1)NCC1CC2CCC(C1)N2C(=O)CN1CCCCC1 C#CCCC(O)C(=O)Nc1ccccc1.C12CCCN1C2 C=CCCCCCC(=O)NC12CCC(C1)N(C(=O)CN(S(C)(=O)=O)C)C2 C12(C(=O)OCC)CC3CC(CC(NC(c4ccc(C)c(Br)c4)=O)(C3)C1)C2 C1(C(=O)NCC(C)NC(c2ccc(CF)cc2)=O)CSc2ccccc2O1 Cc1c(C(=O)NCC2(NC(C3CCN(C)C3)=O)CC3CCC2C3)cncc1N c1(C(=O)NCC2CCCN(Cc3c(C)nc(Cl)cc3)CC2)cc(C#N)ccc1O c1(C(C)C)nc(N(C2CN(C(=O)CC3CC3(C)C)C2)C)cc(C(C)(C)C)n1 C1(NC(CC2N(C)CCCC2)=O)CN(C(c2c(O)cccc2Cl)=O)CCC1(C)C C12(C(=O)NCC3OCC(CNC(=O)CCn4cncn4)C3)CCC(CC1)OC2 O=C1CCCC(CC(=O)NCCCCNC(c2csc(Cl)n2)=O)N1 Cc1ccc(C(=O)NCC2CCCCC2NC(c2nc(C)n(C)n2)=O)c(N)c1 CCC(C(C)Cc1ccccc1)Nc1cccc(-c2nc(O)n[nH]2)c1 C1(C(=O)NCCC(C)NC(=O)CSCCC(F)(F)F)OCCOC12CCC2 O=C(C1=CS(=O)CCC1)NCC1CC(F)CN1C(C1CCCN1c1nccs1)=O N1(C(C(CC)O)=O)CCc2c(C(=O)NCc3cnc(C(F)(F)F)nc3)n[nH]c2C1 C=CC(CCC)CC(=O)NCC1CCCN(C(C23CCC(C2)OC3C)=O)C1 c1(NC(C2N(C(c3c(C)cc(C)o3)=O)C(C3CC3)CC2)=O)ccc2nc[nH]c2c1 C1(C2CCN(C(c3cn4ccsc4n3)=O)C2)(NC(c2cc(C)c(Cl)s2)=O)CC1 c1(C(=O)NC2CN(C(c3cc(C)c(C)s3)=O)C2)coc2c(C)cccc12 N1(C(CC(CC)(F)F)=O)CCCC(C2CN(C(c3cc(F)c(F)cc3O)=O)C2)C1 C1(C(=O)OC)N(C(C2C3CC3CN2C(=O)COCC(C)C)=O)CC1(C)C C(=O)(CN=c1ccc(Cl)n[nH]1)NC1CC(NC(=O)CC2CN3CCC2CC3)C1 C(N=c1[nH]c(=N)[nH]c(Cl)c1[N+](=O)[O-])C1OCC(CNC(C(C)OCCCC)=O)C1 N(C1CC2(CCN(C(C3(Cl)CC3)=O)C2)Oc2ccccc21)C(c1nnc(C)s1)=O C1(C(N(C2CC3CC2N(C(=O)C(C)(C)C#N)C3)C)=O)CCOCC1(C)C N1(C(C2C(CC(C)(C)C)C2)=O)CCC(NC(c2ncccc2Cl)=O)C12CCC2 C1(NC(CCCOCC)=O)CC2CN(C(=O)CC3CCCN(C(C)C)C3)CC12 C1(CC(N2CC(O)(C(C)NC(=O)CNC(c3ccoc3)=O)C2)=O)CCCC(O)C1 N1(C(C)=O)CCC2OCCN(C(c3ncn4cc(-c5ccnn5C)sc34)=O)C2C1 C=CCCCCCCCCC(=O)N1CCN(C(=O)CCSCCCC)C(CC)C1 Cc1nccnc1C(C)NC(=O)C(c1ccoc1)NC(C1CC=CC(O)C1)=O N1(C(CCCOCC)=O)CCSCC1CCOCC1C(c2ccccc2)C1C Cc1cscc1NC(=O)C(CN(C)C)NC(C1COC(=O)N1)=O c1(COCC(N2CC(NC(C3(SC)CC3)=O)C(O)C2)=O)nc2ccccc2s1 N1(C(c2ccc(CNC(c3c(C)cc(C)o3)=O)cn2)=O)CCCC(C#N)C1 c1(CCC(=O)N(CC(C)CNC(=O)CNS(C)(=O)=O)C)nc2ccccc2o1 c1(C(=O)NCCCC(C)NC(c2c(C)coc2C)=O)coc2c(Cl)cccc12 C(CC(C)C(=O)N1CCC(C(=O)NCc2nc[nH]n2)(C(C)C)C1)=CCC N1(C(c2c(CC)c[nH]n2)=O)CCCC(C)(C)C1CNC(c1scc(C)c1Cl)=O CC1C(O)CCCN1C(=O)CC1(NC(c2cccnc2)=O)CCC1 C(=O)(C(C)(C)C)NC(C1CCCN1C(=O)Nc1ccc(CN2CCCC2)o1)C CCCCC(C)(F)C(=O)NC1CCC(NC(c2cccc3scnc23)=O)C1 C1(N2CC(C(=O)OC)C(C(=O)O)C2)CCC2CCCC1C2=O C(=O)(C(C(=O)NCC(F)CNC(c1cc(F)ccc1CC)=O)C(C)C)OCC c1(C(C)NC(=O)C(F)C2CCNC2)ccc2nc[nH]c2c1 Brc1cc2c(N3C4CN(Cc5cccc(-n6ccnc6)c5)CC34)ncnn2c1 c1(C(=O)Nc2c(NCC)ccc(Cl)c2)ncc2ccccc2c1O C(=O)(C1CCCc2nncn21)NC1(C)CN(C(C2COC3COCC23)=O)C1 C1(C2(O)CCOCC2)(C(N2CC(CNC(C(CC)=CC)=O)C(C)(C)C2)=O)CC1 C#CCCCCC(=O)NC(C)CN(C(C1CC(=O)N(CCC)C1)=O)CC c1(C(N2C(CC)CN(C(C3(CC(C)C)CC3)=O)CC2)=O)ccc2c(c1)CC(C)O2 c1(C(=O)OC)ccc2ccccc2c1-c1ccc(C(N2CC(O)C2)=O)c(C)n1 C1(CNC(CC)=O)C(C)CCN1C(C1CC(C)(O)C1)=O CC12CC(NC(C3CCC3)=O)(C1)C1(CN(C(=O)CC3CN4CCN3CC4)C1)O2 C1(OC)CN(C(=O)C2=CCSC2)C(C)(CNC(c2ccc(C(C)C)nc2)=O)C1 C(=O)(CS(=O)(=O)CCOC)NC(C(=O)NC(CCCC)CO)C1CCC1 Cc1cc(C(=O)NC(CO)C(C)NC(c2sccc2F)=O)nn1C(C)C1CC1 C1(C(=O)NC2(COC)CCN(C(=O)Cc3sc(C)cc3C)C2)CC12CCSCC2 N1(Cc2c(OC)nccc2)CCC(C2=NOC(C(=O)N(C)C)C2)CC1 c1(C(C)(C)C)nc2ccc(NC(=O)C3CCc4snnc43)cc2[nH]1 CC(C)CC(=O)NCCC(N1CCCC1C(C)NC(C1CCCN1C(C)C)=O)=O CC(C)C(C(=O)NC1(CNC(C2CC(n3ccnc3)C2)=O)CC1)NC=O C1(C(=O)OC)CCN(C(=NCC2CC2C(F)(F)F)NC(c2ccccc2)C)CC1 C(=O)(CC(CC)NC(=O)Cn1cc(C#N)cn1)NCC(=O)NCC c1(C(=O)NC2CC(N(C(C=CCN(C)CC)=O)C)C2)ccc(CO)c(F)c1 C(CCSC)(C(=O)NC1CC1NC(C1(C(=O)Nc2ccccc2)CCC1)=O)OC N1(C(CSc2nc(C)cc(C)n2)=O)CCC2(CCN2)CC1 C(C(=O)NCC1CCCCN1C(=O)COCCOCCO)(C(C)C)OC C(c1cc(C)c(C)cc1C)=CC(N1CCN(C(CCNC(C)=O)=O)CC(O)C1)=O C1(C(N2C(C)C(NC(=O)CN(C)C)CC2)=O)CCCCC1(C)C c1(CC)ccc(C(=O)NCC(C)(C)NC(=O)CCCSC)cn1 Cc1cc(=NC(=O)C(=O)NCC2CCCN2C(=O)Cc2ccc(F)c(N)c2)[nH]o1 c1(OC)cnnc(C(=O)NCC2(NC(=O)C(c3ccccc3)C)CCOCC2)c1 c1(N(C)CC2CCCN(C(CS(CC)(=O)=O)=O)C2)ncnc2c1nnn2C1CC1 c1(OC)ccc(C(F)(F)F)cc1C(N1CCC(OC)CC1C(=O)O)=O C1(N(C)C(C2CC3CC3C2)=O)CCCN(C(c2ccc(CNS(C)(=O)=O)o2)=O)C1 c1(C(=O)NC2CC(NC(=O)CSc3ccncc3)CC2O)c(Cl)cncc1Cl C(CCCCC(=O)N1CCCN(C2CC2)CC1)NC(COC1(C)CCCC1)=O C1(c2n(CC=C)nnn2)(NC2CCCC2SCC)CCC(CC)CC1 CC1CCCn2ncc(C(=O)NC3CC(O)(CCC(C)(C)C)C3)c21 C1(NC(c2oc(CC)c(C)c2)=O)CCN(C(=O)CC2CCCC(C)(C)O2)C1(C)C N1(C(CSC)=O)CCCC(C2CCCN2C(=O)C=CC(=O)Nc2ccsc2)C1 CC1CNCCC1N(C)C(=O)Nc1cccc(CNS(=O)(=O)C2CC2)c1 N1(CC)CCCC(C(N2CC(CC(=O)NCC(C)(COC)CO)(OC)C2)=O)C1 C1(CNC(c2c(C)cncc2)=O)CN(C(c2coc(Br)n2)=O)CC12CC2 c1(C(N2C(C(N(C3CCOCC3)C)=O)CSCC2)=O)cc(O)nc(O)n1 c1(OC)nc(Cl)cnc1NC(C1C(O)CCN1C(c1cccc(F)c1I)=O)=O N1(C(C2(CC(C)=O)CC2)=O)CCCC(N(C(=O)CN2CCCC2C)C)CC1 c1(C(N2CCC(N(C(CSCC(C)C)=O)CCO)C2)=O)nccnc1C(N)=O C1(NC(n2c(C)csc2=O)=O)CC(NCC(N)=O)C12CCC2 CCCCC(C(=O)Nc1cc(Cl)ccc1O)NC(=O)C(CN(C)C)CC C(=O)(CC(O)c1cnc(Cl)s1)NC1(CNC(CC2CC(OC)C2)=O)CCC1 N(C1=NCCCNCC2CCN1C2)C(C=C)C.C1(COC(=O)OC)CCCC1 N1(C(C23CC(CC)(OC2)C3)=O)CC2CN(C(=O)OC(C)(C)C)C(CO)C2C1 C1(CC(N2CC3CC2(C(F)F)C3)=O)C2CCCC2N1C(=O)C(O)CN1CCCC1 c1(C(N(C2CN(C(=O)C3=NNC(=O)CC3)C2)C)=O)cc2c(F)ccc(F)c2s1 c1(C(N2C(CCNC(C(COC)C)=O)CSCC2)=O)cc2cc(C)ccc2[nH]1 C1(CC#C)(C(N2CCC(O)(CNC(=O)C(C(C)C)NC(C)=O)C2)=O)CC=CCC1 c1(C(N2CC(C)C(NC(=O)CC3CC3(Cl)Cl)C2)=O)ccc(N)c(F)c1F Cc1cc(C2CC2)ccc1-c1c[nH]nc1C(N(C(C)C)C1CC1)=O c1(NC(C2CC(F)CN(Cc3ccc(O)cc3Cl)C2)=O)cccc([N+](=O)[O-])c1I C=CCC(CC)C(=O)Nc1cccc(NC(=O)Cc2cnc(C)o2)c1 CCCC(CNC(C1COCC(C)O1)=O)C(=O)N1CCC(C#N)C1 C12(C(N3CCC(C)(CNC(C(C(C)C)NC=O)=O)CC3)=O)CCOC1CCOC2 c1(OCCC(=O)NCCCNC(c2c(C(=O)OC)csc2)=O)ccc(F)c(F)c1 Cc1sc(C(N2CC(NC(c3ccn(C4CCOCC4)n3)=O)C(C)C2)=O)nc1O C(=O)(CC(O)CNC(c1cccn1C(C)C)=O)NC(C=C)(C)C N1(C(CNC(=O)NC)=O)CC2CC1CCN2C(=O)C(C)Oc1cccc([N+](=O)[O-])c1 CCC(C)C(C)CNC(c1cn(CCNC(=O)Cc2cc[nH]n2)cn1)=O c1(C(=O)NC(CN(C(C2(C(C)(C)OC)CC2)=O)C)C)cn2cccc(F)c2n1 c1(C(N2CCCC(NC(c3ccc(CC)c(N)c3)=O)C2)=O)cc(S(C)(=O)=O)cs1 C1(C)(C(=O)NCC2N(CC)CC2)CC(O)CN1C(=O)C1=COCCC1 c1(C(=O)OC(N(CCNC(CCCCC=C)=O)C)=O)cc([N+](=O)[O-])ccc1NC C12(Nc3c(C)cncn3)CCCCC1CN(C(C1CC1C)=O)C2 C=CCC(CC)C(=O)N1CCC(C)(NC(=O)CCCc2ccc(C(C)C)nc2)C1 N1(C(C2C(C)C2)=O)CC(NC(C23CCC(C)(CC2)CO3)=O)CC12CCCOC2 N1(S(CCCC)(=O)=O)CC2CN(Cc3cccc(C(C)(C)C)c3O)C2C1 C(C)(CCC(=O)NCC1CN(C(C2CC(F)C(=O)N2)=O)CCO1)OC c1(OC)nc(C)cc(=NC2CCN(C(c3conc3C)=O)C(C)C2)[nH]1 CC1=C(C(=O)NCC2(C)CCC(NC(=O)CCN3C(=O)CCC3=O)C2)CCCC1 c1(C(=O)NC(CNC(=O)C#CC2CCOC2)C2CCC2)ccc2nc(O)oc2c1 Cc1cc(CC(C)NC(c2[nH]ccc2CNC(=O)Cn2nccn2)=O)n[nH]1 C1(NC(c2cnn(C(C)C)n2)=O)CCCCC1NC(c1c[nH]nc1F)=O C1(C(=O)NCC(CNC(CC2(CC)CC2)=O)(C)O)CC(=O)N(C2CCCCC2)C1 N1(C(C(C)C2CC2)=O)CCC(CF)(NC(=O)CN(CCCF)C)C1 C12(C(=O)NC(CC)CNC(C3CC34CCC4)=O)CCC(OC)(CC1)C2 Cc1ccc(CN2C(C(=O)Nc3ccc(CC#N)nc3)CC3CC23)cc1Br c1(C(=O)NC(C=CC(=O)NCC2CCN(CCC)C2)C)cc(O)cc(=O)o1 C1(C(N(CCCCNC(c2cc(C)nn2C)=O)C)=O)CC(C)CCC1C(C)C c1(CC2(NC(C(CCCC)NC(=O)CC3CC3)=O)COC2)ccc2c(c1)OCO2 C(=O)(C(C)C(F)(F)F)NCC1(NC(C(c2ccc(C)cc2)C2CC2)=O)CC1 CCCC(C)(C)C(=O)NCC1CCN(C(c2c(C)nn(C)c2Br)=O)CC1 c1(C(N2CC(CCC)C(NC(c3ccc(O)nc3)=O)C2)=O)cnc2ccnn2c1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1CCC2(CC(CNC(C(N)=O)=O)C2)CC1 C=C(C)CC(C)C(=O)N1CCC(OCCNC(C2CN(S(=O)(=O)CC)C2)=O)CC1 c1(C(=O)NC(C)C(CO)NC(=O)CCc2cccs2)cc2n(n1)CCC2 C1(C(=O)NCC2(O)CN(C(C=CC(=O)N(C)C)=O)C2)CCCN(c2nccs2)C1 C(C1=NOC2(CCC2)C1)NCCNC(=O)NC1(c2cc(Cl)ccc2F)CC1 c1(C(N2CCC(C)(NC(C3CC34CCCCC4)=O)C2)=O)ccc2ncnn2n1 C1(C(=O)NC2CC(n3ccnn3)C2)C2CCC1(c1ccc(C(F)(F)F)cc1)C2 C1(C(N(C2CC23CCN(C(=O)CCOC2CC2)CC3)C)=O)CCc2cnn(C)c2C1 N1(C(C2C(C)(CC)C2)=O)CC2CCC1C1CN(C(=O)C(C)(C)CF)CC21 c1(OC)ccc(OC)c(C(F)(F)C(=O)NCC(O)CNC(C2(C)C=CCC2)=O)c1 Cc1c(Br)ccc(C(=O)NCC(c2ccc(Cl)s2)O)c1F C(=O)(C(C)CC(N)=O)NC(C)C(=O)NCC1(O)CN(C)C1 N1(C(C2N(C(C3(CCCC)CCC3)=O)CCCC2)=O)CCCCC(C(N)=O)C1 c1(C(N2CCCC(F)(C(=O)OC)C2)=O)ccc2c(c1)C(C1CCOCC1)C(=O)N2 c1(C(N(CC(CC)NC(c2ncncc2F)=O)CC)=O)cccc2cncn12 CC1CC=C(C(=O)NC2CCN(C(C3COC(=O)C3)=O)C23CCC3)CC1 c1(C(=O)NC2CN(C(CCC3N(C)CCC3)=O)CC2O)cn2cccc(Cl)c2n1 n1(CCC)cc(Cl)c(C(N2CC(NC(c3nccn3CC=CC)=O)C(C)C2)=O)n1 N1(C(c2c(CC)nccn2)=O)CC(C)(C)CC1C(=O)NCC1COCCN1C CC(O)C(C(=O)N1CC(O)(CNC(=O)CC2(C)CC2(F)F)C1)NC(N)=O c1(NC(c2cc(CC)n(C)n2)=O)ccc(NC(=O)C=Cc2ncc(C)[nH]2)cc1C c1(NC(=O)NC2(CC=C)CCCNCC2)c[nH]c2ccccc12 CC1(C)CCCCC1CC(=O)N(CCNC(c1cc(C(N)=O)[nH]n1)=O)CC1CC1 C(=O)(C(C)(C)C(C)(C)O)NC1CCCC(NC(CSc2n(C)ccn2)=O)C1 N1(C(C2N(CC)CC2)=O)CCOCC(NC(=O)C(c2ccccc2C)C)C1 CN=S(C)(=O)c1ccc(C(=O)NC2CC(N(C(=O)C3=NOCC3)C)C2)cc1 CC(C)CC(C(=O)NC1CC(C)(CNC(=O)C=C(Cl)Cl)C1)C(C)C N1(C(c2c(C)cc(C)s2)=O)CC2CCC1C(NC(c1ccc(F)cc1)=O)C2 C1(C(N2CC(OCCNC(c3c(C)snn3)=O)C2)=O)CC(O)CN1C c1(NCCCCCC)ccc(S(=O)(=O)NCC2CC(CC(N)=O)CO2)c(Cl)c1 N1(C(c2cc(CC)on2)=O)CCCC(CC(=O)NC(C)CCn2cncn2)C1 C(=O)(C(O)CC(F)(F)F)NC(C1CCN(C(C2CC(=O)CCO2)=O)CC1)C c1(OCC)ccccc1CCCC(C)N(C)Cc1sc(C(=O)NCSC)c(C)n1 C1(NC(c2c(C)nc(Br)o2)=O)CC(C)CN(C(c2cnccc2Cl)=O)C1 C1(NC(C2(Nc3sccc3C(F)F)CC2)=O)CCCCC1C(F)(F)F c1(CC(=O)N(C(CNC(C(C2CCC2)OC)=O)C)C)coc2c(Cl)c(Cl)ccc12 Cc1cn(C)cc1C(=O)NC1CC(OCC(=O)NCC2CC(O)C2(C)C)C1 C1(NC(c2cccc(C)c2Br)=O)CC12CCN(C(=O)Cc1cnc[nH]1)CC2 CCC(C)C(C(=O)N1CCC(Nc2nccc(C(F)(F)F)n2)C1)OC N1(CC(=O)NC(C(N2C(CNC(=O)NC)CC2)=O)C2CCCC2)CCCCC1C C1(C(N(CCC#C)CC)=O)C2CC(O)C(C2)N1C(=O)C(c1ccc(C)o1)C Cc1nc2cc(C(=O)NCCCCCCNC(=O)COc3ccsn3)[nH]c2s1 NC1CCC(F)(F)CC1C(=O)NCCCNC(=O)Nc1ccccc1 Cc1nn(C)c(Cl)c1-c1cn(CCCNC(C2CC3CC2CC3=O)=O)nn1 c1(OC)ccc2oc(CN(CC(=O)Nc3nn[nH]n3)C)cc2c1 Cc1cc(C)c(C(N2CCC3(NC(c4oc(C)cc4C)=O)CCCC23)=O)c(O)c1 Cc1cc(NCCCCC2CN(C(=O)C3=CC4CCCC34)C2)n2ncnc2n1 c1(C(=O)NC(C2CC(NC(c3cc(C)c(C)o3)=O)C2)C)ncc2ccccn12 c1(-n2cc(CCC(C)=O)nn2)cccc(CCNC(C2(C)CCCN2C)=O)c1 c1(C(N(C2CCCN(C(C(CC)F)=O)CC2)CC)=O)cccc2[nH]ccc12 C(=O)(CC(C)N1CCCC1)NC(C1CCCCC1)CNC(C(F)=CCC)=O C(CNC(c1cnc(C2CC2)[nH]1)=O)(CC(F)(F)F)NC(Cc1cccc(C)c1)=O C1(C(=O)NCC(C2CCC2)NC(CCNC(=O)NC)=O)CCc2nc(C)[nH]c2C1 Cc1ccc2c(c1)CC(C(=O)NCC13CCC(CC1)N(C(c1ccsc1)=O)C3)S2 c1(C(=O)NCCCNC(c2cc(C(C)=O)sc2)=O)cc(O)nc2c1CCCC2 c1(C(=O)Nc2c(Cl)nc(C)c(Br)c2)cccc(S(=O)(=O)NCC(C)O)c1 C1(NC(COC(C)C)=O)CC2CC1N(C(=O)CC1CCCC(=O)C1)C2 c1(NC(C(=O)N(CCC#C)CC)=O)ccc(Oc2ccc(F)cc2)nc1 Cc1ocnc1CC(=O)NCCOC1CN(C(C2CC(=O)C2C(C)(C)C)=O)C1 CC1(C(N)=O)CCN(C(=O)C(CCF)NC(=O)Cc2ccsn2)C1 C12(CNC(CSCCCC)=O)CCCC1CCN2C(=O)C(=Cc1ccncc1)C C(=O)(CCC(C)(C)OC)NCC(C(C)(C)C)NC(C1OCCN(CC)C1)=O C1(CN(C(CCC=C)=O)C)CCCCN1C(=O)C(CC)OC1CCCC1 c1(C(=O)NC2CCC(N(C)C(c3cnccn3)=O)C2)cnc(O)c2c1NCCC2 C=Cc1ccc(C(N2CCCC(NC(=O)C(CC)=CC)C2C)=O)cc1 c1(C(N2CC(F)CC(NC(C(C)S(C)(=O)=O)=O)C2)=O)ccc([N+](=O)[O-])cc1O N1(C(c2c[nH]cc2Br)=O)CC2(C1)CN(C(c1ccc3c(c1)CCO3)=O)CCO2 CC1CCN(C(c2cccc(C3CCOCC3)c2)=O)C1(C)C Cn1cnc2c1CCC(C(=O)NC(CNC(=O)CSCCC#N)C(C)(C)C)C2 C1(CNC(CCCCC)=O)CC2CCC(C1)N2C(=O)COCC(F)(F)F c1(SC2C(CC(=O)N(C(=O)CCC3(C)CC3)C)CCCC2)ncnc2[nH]cnc12 c1(CCNC(c2ccc(Cl)s2)C)ccc(F)c(Br)c1 Cc1ncc(C(C)NC(C2CCC(NC(C3COCCO3)=O)C2)=O)s1 S(=O)(=O)(C1CN(C(=O)CCC(N)=O)C1)N1CCN(C(CC2(COC)CC2)=O)CC1 Cc1ccc(C2=NOC(CNC(=O)NNc3cc(C)nc(Cl)c3)C2)cc1 CCC(O)C(=O)NCC1CC(CNC(=O)CC2CCN2C(=O)OC(C)(C)C)C1 C1(CNC(C(C)(C)CF)=O)CN(C(c2cc3ncccc3s2)=O)C2CCN1C2 N1(C(c2n(C)cnc2)=O)CCC2CN(C(c3ccc(C(F)(F)F)s3)=O)CCC2C1 c1(OC)ccc(O)c(NC(=O)CONC(=O)CC(O)C2CCCCC2)c1 C12(NC(c3c(C)nsc3)=O)CCOCC1CN(C(=O)CCc1ccc(Cl)nc1)C2 c1(C(C)C)nn(C)c(Cl)c1C(=O)NCCCN(C)C(C1CC(N(C)C)C1)=O C1(NC(c2cnc(C)nc2)=O)C(CNC(=O)Cc2ccc(C)s2)CCC12CCC2 C1(C(N(C)CC2(NC(=O)CN3CC4CCC3C4)CC2)=O)COc2ccccc2O1 Cn1cccc1C(=O)C(=O)NCC1CC1NC(C1(CC2CC2)CCC1)=O Cc1ncncc1C(=O)NC(C(=O)N1CCC(C(F)F)CC1)C(C)C Cc1cncnc1C(=O)NC(CC(N1CC(CO)CC1CO)=O)C1CC1 CCCCC(CCCC)NC(C1CCC(C)N(C(c2cccc(O)c2F)=O)C1)=O C(=O)(C(C(C)(C)C)Sc1ccccc1)NCC1(NC(CN(S(C)(=O)=O)C)=O)CC1 c1(OC)cc(C(N2CC(CNC(c3ccnn3CC(F)F)=O)CC2C)=O)n(C)n1 C1(CNC(c2n(CC)nnc2)=O)CC(F)(F)CN1C(C1CNC(=O)N1C)=O c1(NC(C2(C)CCN(C(c3c(C)cnnc3)=O)C2)=O)c(O)cccc1O Cc1[nH]nc(CO)c1C(=O)N(CC(C)C(=O)NC(C1CCC1)C1CCC1)C N#CC12CC(C(N3CCC(CCNC(=O)CSCc4ccccc4Cl)C3)=O)(C1)C2 c1(NC(C2CC2C(=O)Nc2cnccc2CO)=O)nccn2ccnc12 N1(Cc2nccc(C(=O)OC(C)(C)C)c2)CCN(c2cnc(F)cn2)CC1 C1(C(=O)NCC(C)(CO)NC(=O)OC(C)(C)C)CC2(CCC2)CCO1 C(c1ccc(Cl)cc1)=CC(=O)N(C)CC1N(C(c2nc(CC)oc2)=O)CCC1 N1(C(COCC(C)C)=O)C(C)C2CC1C2NC(C1CCOC1)=O C1(NC(c2c(OC)nn(C)c2)=O)CCCN(C(=O)CCc2cnc(N)cn2)CC1 C(c1cccc(F)c1F)=CC(=O)NC1(C2CN(C(Cc3ncc(C)s3)=O)C2)CC1 C(CC(=O)Nn1nnc2c1CCCC2)NC(C(C)NC(=O)NC)=O Cc1occc1C(=O)NC1CCC1CNC(=O)C(c1cccnc1)O c1(OC)n[nH]c(C(=O)OC(C)(C)C)c1I.C12CC(CN1C)C(=O)OC2 C1(CC(=O)NCC2CN(C(c3c(C)ocn3)=O)C(C)C2)CC(C)(C)OC(C)(C)C1 c1(C(=O)NC(CNC(CCOCCC)=O)(C)C2CCC2)cncc2ncn(C)c12 N1(C(c2cnc(OCC)s2)=O)CCCCC1C1CCCN1C(c1ccnn1C)=O N1(C(C2CCCC2)C)CC(CN)C(C)(C)C1 N1(C(N(C)C)=O)CCC(NC(C2CC2CNC(=O)CC2(C)CC2)=O)CC1 C1(CC)(CC)CC(NC(c2cc(Cl)no2)=O)CN1C(=O)Cn1cc(C)cn1 C(=O)(C(CC)C(=O)NC(C)CCNC(=O)CCc1ccc(C)nc1)OCC C(=O)(C(F)CC(C)(C)NC(=O)C=CC(C)CC)N1CCC(N(C)C)(COC)C1 C(=O)(C1CCCc2scnc21)N1CCC2(CN(C(c3cccc(F)c3Cl)=O)C2)C1 C1(CC(=O)N(C(C)C)CCN(C(=O)CCC2CC2(F)F)C)CNC(=O)O1 c1(CC(=O)NC2C(NC(c3c(OC)n[nH]c3)=O)CC2)cc(O)nc(O)n1 C(=O)(C#CC1CCCC1)NC(CC=CC)C(=O)NC1CCOCC1(C)C O=C(C#CC1CCOCC1)NCCC12CCC1CN(C(c1cnn[nH]1)=O)C2 C=CCCC(O)CN(C(=O)C(C)(CO)NC(c1cccc(F)c1)=O)C C1(F)(CNC(c2c(C)cc(CC)o2)=O)CCN(C(c2c(C)ccnc2O)=O)CC1 C1(C(=O)NC(C(=O)NC(c2onc(C)n2)CO)C2CCCC2)C2CCC(C2)C1C Cc1cc2ccc(C(=O)NC(C3CN(C(c4nnc(C(C)C)o4)C)C3)C)cn2c1 C1(C(=O)NC(C)(C)C)CCCN(C2C=CCCCC2)C1 C1(C(=O)NC(c2ccccc2)CCN(C)C(C2CCSCC2)=O)CCCCC1(F)F c1(C(=O)NC(CC)CNC(c2cccs2)=O)cc(Br)cc([N+](=O)[O-])c1 C1(NC(C=CC=CC)=O)COC2(C1)CN(C(C1(C)CC1)=O)C2 N1(CCSC)CCCCC1C(=O)N(C)Cc1ccc(-n2cccc2)cc1 C1(CNC(C(OC)OC)=O)CN(C(c2ccc3c(c2)CC3)=O)CC1(C)C O=C(C1=NN2CCCN=C2N1)NCC(O)CNC(c1nnn2c1CCCC2)=O N1(C(C(=O)NCCCSCC)C2(CC)CC2)CC2CCCN2c2ccccc21 C1(CS(=O)(=O)N(CC(=O)OCC)Cc2ncc(Cl)s2)(CF)CC(F)(F)C1 C1(NC(c2ncn(CCNC(C3(CC)CCCC3O)=O)c2)=O)C2CCC(F)(F)C12 CC1(C)CCCC(C(=O)NC(C(=O)NCC(C2CCCC2)O)C2CC2)C1 C#Cc1cncc(C(=O)NCC2CC2CNC(=O)CCC2CCC(=O)N2)c1 C1(N(C(C)=O)CC)CCCN(C(=O)C(C)(C)C)C1.c1(C(C=O)(F)F)ncccc1F C1(C(N2CC(O)(C(=O)OC)C2)=O)CC(C)CN(C(c2ccc(O)cc2)=O)C1 N1(C(c2scc(C)c2)=O)CC(CNC(c2ccccc2-n2cccn2)=O)CC1C c1(CN2CC(CC)N(C(c3ccc(F)c(I)c3)=O)CC2)ccc(N)c([N+](=O)[O-])c1 C1(CC(=O)NCC(=C)F)CN(C(c2cnc(C)[nH]c2=N)=O)CC12CC2 C(c1cccc(F)c1)=C(C(=O)NC(C)CCN(C)C(C1CCCS1)=O)F c1(CC)cccc(OC2CCCC(NC(C=CC=NC(=O)CS(C)(=O)=O)=O)C2)c1 C1(CNC(=O)CCc2cncnc2)CC2(CC(NC(C3CCCCO3)=O)C2)C1 CCC(CC)C(F)C(=O)NCC1CCCCCN1C(C1CCCCS1(=O)=O)=O N1(C(c2c(C)ocn2)=O)CCOCC(CNC(c2nccn2C)=O)C1 C(C(C(C)C)NC(c1cc(I)sn1)=O)NC(COC(C)C)=O N1(C(C2CC(N3CC(O)C3)C2)=O)CCCC1CCNC(C1CSCCS1)=O c1(NC(C2N(C(C)=O)CCC2)=O)c(CNC(=O)COc2ccsn2)nnn1C S1(=O)(=O)c2ccc(cc2)CCC(C)NC(=O)C1.C(=O)(CCCSC)OC.[nH]1cnnn1 CCCC(C)(CC)C(=O)NC1CCC1NC(c1coc(C2CCCCC2)n1)=O CC1CN(C(C2(NC(=O)C=CCN3CCC3)CCC2)=O)C(C)C(C)(C)O1 C1(NC(CNC(C(CC)C)=O)=O)C2CN(C(=O)C(=C3CCCCC3)F)CC12 N1(C(=O)Cn2cc(Br)cn2)CC2CCC(C1)N2C(=O)Cc1ccn(C(F)F)n1 c1(C(=O)NCCN(CCC)C(c2ccsc2OC(C)=O)=O)cc(=O)c(OC)cn1C c1(NC(C2(CNCc3cc(Br)ccc3F)CC2)=O)cnccc1[N+](=O)[O-] C(C#CC(=O)NCC1CCCC1NC(=O)CC(=O)C1CCCC1)(OCC)OCC c1(NC2CN(C(=O)Cc3ccnn3C3CCCC3)C2)ccc([N+](=O)[O-])cc1Cl CC(C)C(CNC(c1cnns1)=O)NC(=O)CSCCCc1ccccc1 C1(CC(=O)N(C(C)C(=O)NC(C)(C)C)CCC)CC=CCN1C c1(C(N(CCC(C)NC(=O)CC(C)C(F)(F)F)C)=O)cc(F)cc2cccnc12 c1(NC(c2c(CNC(C(C)OC(C)(C)C)=O)occ2)=O)ccc(CO)cc1 N1(C(C)=O)CCC(C)(C(=O)COC(C)=O)C1.N12CCN(CC1)C2=O.C(C)(C)(C)O C(=O)(C(C)(O)CC(F)(F)F)NCCN(C(COCCCC)=O)CC(C)O c1(C(=O)NC2CCN(C(C=Cc3cn(C)nn3)=O)C2(C)C)snc2ccccc12 C(CCCCC(=O)NCc1ccc(C(=O)OC)cc1N)OCC C1(C(=O)NC(C)CCc2ccc(F)cc2F)CCN(CC(N)=O)CC1(C)C C(=O)(C(C)(C)CS(C)(=O)=O)N(C1CCN(C(C2CCC(O)CC2)=O)CC1)C N1(Cc2c(OC)cco2)CC2CCC(C1)C2NC(c1cc2cnccc2[nH]1)=O N1(C(Cc2ccc(C)nc2Cl)=O)CCC2CN(C(C3SCCS3)=O)CC12 c1(C(=O)NC(CC(C)NC(COCC#C)=O)C)cn(C(F)F)c(C)n1 n1(CC)ccc(CNC(=O)C=CC(C)(C)NC(c2ccco2)=O)n1 CCC(CNC(C1(C)CCCO1)=O)(CC)NC(=O)CCSCC(C)C c1(C(N2CC(O)CC(NC(C3(OC(C)C)CCC3)=O)C2)=O)cc2cnn(C)c2s1 Cn1ccc2cc(-c3ccc(NC(=O)OC(C)(C)C)nc3)cnc12 C12CCC(CC1)CNC2=O.C1(CC(=O)NCCC(C(C)O)C2CC2)C=CCC1 C(N=C(NCC(C)(C)C)NC1CC(OC)(OC)C1)C1(C(=O)OC)COC1 c1(C(N2CC(NC(=O)Cc3cncs3)CC(C)C2)=O)cc2ccc(F)cc2o1 c1(C(=O)OCC)cc(I)c(NC(c2cscc2-c2cccnc2F)=O)cc1Cl C1(CNC(C2C(C(=O)OC)C2)=O)CN(c2ncc(C(F)F)cn2)CCC1(F)F c1(NC(=O)NC(C)CCCOc2cccnc2)ccc2c(c1)ncn2C c1(C(N2CC(C(C)NC(C=CC)=O)C2)=O)ccc2ccc(O)nc2c1 CC(C)(C(=O)NCC1(F)CCCN(C(=O)Cc2cn[nH]c2)C1)C(N)=O C1(OC)CC(C(=O)NCCC2CC(NC(C3(C#N)CCC3)=O)C2)CC1OC c1(NC(CNC(C(CC)CN(C)C)=O)=O)cnc(Cl)nc1C C12(NC(=O)CN3CC=CC3)CCC(CC1NC(=O)C(O)(C1CC1)C1CC1)C2 C1(NC(CCC2(C=C)CC2)=O)CC(CNC(C2CCCN2CCC)=O)C(O)C1 c1(CC(C(=O)NCC(CNC(c2cn(CC=C)nc2)=O)C)C)ccc(Cl)c(Cl)c1 c1(-c2ncn(C)n2)ccccc1C(N1CCC(CCNC(c2cocn2)=O)C1)=O Cc1c(C(=O)NCC#CCNC(=O)CC2(CO)CCOCC2)cncc1N N1(C(C2(CC)CC2)=O)CC2CCN(C(c3cccc(C)c3NC(C)=O)=O)CC2C1 C1(CNC(C(C)NC(=O)C2CC2)=O)CN(C(=O)C2=CC(C)C2)CCCO1 O=C(N=c1nc[nH]n2cc(Br)cc12)N(C1CC2(CNC2)C1)C1CCCC1 Cc1nn(C)cc1C(C)NC(=O)COC(C)(C)CNC(C12C=CC(CC1)C2)=O C=CC(C(=O)NCC1CCN1C(c1ccc(F)s1)=O)NC(=O)OC(C)(C)C c1(C(=O)NC2C(CO)CCN(C(c3c(C)nn(C)c3)=O)C2)cccc2cncn12 CC1(C)CCN(C(=O)CSCC(N)=O)CC1NC(c1ccn(C2CC2(F)F)n1)=O c1(C(=O)NCC2OCC(CNC(CCC=C(C)C)=O)C2)cc2sccc2n1C N1(C(C2CCN(CC)CC2)=O)CCCC(C)(C(N2CCC(C)(CO)C2)=O)C1 c1(C(=O)NC(C2CN(C(COC(CC)(C)C)=O)C2)C)nn(CC)cc1Cl CCCCC(C(=O)NC(c1n[nH]c(CO)n1)C)NC(=O)COCC(=O)NC C(C)(CCCNC(=O)CCC1CCOCC1)NC(C=C(C)C(C)C)=O c1(C(C(=O)NC(CC)C)N(C)CC2CC2)ncn(C)n1 N1(C(C2(Cl)C(C(C)=O)C2)=O)C2CCC(C2)C1CC(=O)NCCOCC(F)(F)F c1(C(N2CCC3CN(C(CCCOC)=O)CC3C2)=O)coc2c(F)cc(F)cc12 C1(C)(C(=O)NC2CCN(C(CSCC=C)=O)C2C2CC2)CCC(F)(F)C1 c1(OC)ccc(O)cc1C(=O)NCC1CN(C(=O)CCc2ccon2)C1 C(CCF)(C(=O)NCC1C(C)(C)C1(F)F)NC(C=CCCC(C)C)=O c1(NC(C(C)=O)=O)n[nH]c2c1CN(C(c1cc3ccoc3cn1)=O)C2 N1(C(Cc2nc(CC)sc2)=O)CC2(C1)CN(C(=O)C(c1cnn(C)c1)OC)C2 c1(C(N2C(CN(C(C3CCCN3C3CC3)=O)CC)CCC2)=O)c(C)noc1C c1(C(=O)NCC(CC)NC(C2CSC(C)=N2)=O)cc2c(nc1O)CCCC2 N1(C(C=CC(C)(C)C)=O)CC2CCN(C(=O)COC3(C)CCC3)C(C2)C1 C1(OC)CN(C(C)=O)CC1NC(c1c(Cl)cnn1C)=O C1(C(=O)NC(CCC)C2CCCC2)CC2(CCN(C(c3cnccc3C)=O)C2)C1 Cn1nc(Br)c2c(NC3CC(NC(=O)CN4CCCCCC4)C3)ncnc12 CC(C)C(O)CC(=O)NCCC(C)NC(C1(C)CCN(C)C1=O)=O N1(CC(=O)NCC(C(=O)NCC(C)(C)COC)OC)CC2CCC1C2 C(C1=C(C(=O)OC)C(c2nnc(Br)s2)NC(=S)N1CCC(C)C)OC c1(OC)ncccc1CC(N1CCC(N(C)C(c2nn(C)cc2C)=O)C1)=O c1(C(N2CCC(NC(CSCC)=O)CC2C2CC2)=O)ccc2c(C)noc2n1 N1(C(c2occ(C(=O)OC)c2)=O)CCCN(C(=O)C(CN(C)C)C(C)C)C(C)C1 N1(C(c2cn(CCNC(c3c(C)snn3)=O)nc2)=O)CCC12CCN(C)C2 N1(C(CC2C(C)(C)CCO2)=O)CCC(C(=O)NC(CO)C2(O)CC2)C12CCC2 C1(C(=O)NC2(CO)CC(CO)C2)CCCN(C(C2CCOC2)=O)CC1 CCC(C(=O)N(CC(O)CN(C(=O)Cc1cn[nH]c1)C)C)Sc1nc(=N)[nH][nH]1 C1(NC(c2ccc(OC)c(F)c2)=O)CCN(c2ncc(C)cn2)CC1(C)C C1(C(C)(C)C)CC(CNC(c2cccc(Br)c2)=O)CN(C(=O)CCCF)C1 S(=O)(=O)(c1cc2c(cc1C)OCO2)Nc1ccc(NCC)cc1C N1(CC(=O)NCc2ccn(CCOCCOC)n2)C(=O)C(C)C(C)C1=O C#CCC(C)(C(=O)NC1CCCCCC1O)NC(C1CCC(C)(C)OC1)=O c1(C(=O)NC2C(NC(Cc3cnn(C)n3)=O)CCCC2)c(F)cccc1[N+](=O)[O-] c1(C(=O)NCC2CC3(CC(NC(c4ccsn4)=O)C3)C2)ccc2nnc(S)n2c1 C(c1ccncc1)=CC(=O)NC1C(NC(COCc2cc(C)no2)=O)CCC1 O=C1CC(N=c2ccnc(NCc3ccc(Br)cc3F)[nH]2)CN1c1ccccc1 N(C1CCc2cccc(F)c21)C(c1c[nH]c2nc(Br)ccc12)=O C1(NC(C(CC)SC)=O)CC2CC1CN(C(C1(C)CCC(OC)CC1)=O)C2 CC1CCC(C2OCCO2)N(C(=O)NCc2ccc(-c3ccncc3)cc2)C1 c1(CN2C3C(C(N4CCC5(CCC5)C4)=O)C(C3)C2)ccc(F)c(Br)c1F c1(CNC(C(c2cscn2)N(C2CC2)CC2CCN(C)C2)=O)ccccc1F c1(N(C)C)cc(C(=O)NC2CC(CNC(C3SCCS3)=O)C2(C)C)ccn1 C1(CC)CN(C(=O)C(C(C)C)N2CCN(C)CC2)CCN1C(=O)CCSC CCCCCCC(C)CC(=O)NC1(CNC(C2CCCCCC2(F)F)=O)CC1 c1(CNC(C2(C)N(C(C(C)N(C)C)=O)CCC2)=O)cccc2c1CCCC2 C1(NC(=O)C(C2CC2)C2CC2)CC2CCC1N(C(=O)CCc1ncccn1)C2 N1(C(C(CCC)F)=O)CCCCC2(CCN(C(=O)CCNC(=O)COC)C2)C1 N1(C(c2ccc(SCCC)cc2)=O)CCCC(CC)(NC(=O)COC)C1 N1(C(c2scc(C)c2)=O)CC(C(=O)Nc2cscc2C)CC(C)(C)C1 C1(SC)CCCC1N=c1nc(N2CCn3nccc3C2)c2c([nH]1)c(C)nn2C Cc1ccc(C(=O)N(C2CCCN(C(=O)C(C)Cc3cnc[nH]3)C2)C)c(N)c1Cl N#CC1CC2(CC(NC(C3CCC3NC(=O)C3=CCCSC3)=O)C2)C1 Cn1cc(NC(c2ccnc(C(F)F)c2)=O)cc1C(=O)NCCC1CCCC1 c1(C(N2CCN(C(C=CC(C)C)=O)CC2CF)=O)cc(=NS(C)(=O)=O)cc[nH]1 C(=O)(CCCCCCn1cc(-c2conc2CC)nn1)N(C(CCC)C)C N1(C(C2(CC)CCCC2)=O)CC2CS(=O)(=O)CC2(NC(=O)Cc2cnsc2)C1 c1(C(=O)NCC(CNC(C(OC)OC)=O)O)cc(F)c(F)cc1C(F)(F)F c1(NC(C2N(C(C(CC)OCC)=O)CC2)=O)ccccc1OCCCN(C)C C1(NC(=O)OC(C)(C)C)CC2CCCCC2C1.C12CC(CCO1)NC(=O)N2 C(C)(C)(C(C)CC(=O)N(C)Cc1nnc(O)o1)NC(C(C)CC(N)=O)=O Cc1ccc2cc(C(=O)NC3CCN(C(C4CC(O)C4)=O)CC3F)cn2c1 CCC(CC(=O)NC1CCC(C(=O)NCCC(=O)NC(C)(C)C)CC1)C(C)C C1(C(=O)Nc2cccs2)CCCCCN1C(c1ccncc1C(F)(F)F)=O C1(NC(c2c(C)nccn2)=O)CCN(C(=O)CCc2cc(F)ccc2F)CC1O C(=O)(CC(C)C(=O)N1CC(NC(c2ccccc2SC)=O)C(O)C1)OC c1(OCC)cc(C)ccc1-c1ccc(C(=O)NCc2cccc(C)c2O)c(C)n1 Cc1cnc(C(C(=O)N(C)C)N(C(C)C(=O)NCCOC(C)(C)C)C)n1C Cc1nc(C)c(NC(c2ccccc2)C(c2ccccc2)NC(C2CC3CC3C2)=O)o1 C1(N(CC(N2CCC(C(=O)N(CC(C)(C)C)CCO)CC2)=O)C)CCS(=O)(=O)C1 c1(NC(C2CC(C)N2C(C2C3CCC(F)(F)C23)=O)=O)cc(Cl)ccc1O N1(C(C2(C#C)CCC2)=O)CC(NC(C2COCCN2CC(F)(F)F)=O)C(O)C1 c1(C(N(C2CCCC(N(C(CN(C)CC)=O)C)C2)C)=O)cccc2sccc12 Cc1cnc(C(=O)N(C2CCCC2)CCNC(c2csc(Cl)n2)=O)cc1C c1(CCC(=O)NC2CC(F)(CNC(C3CC3F)=O)C2)ccc(Cl)cc1Cl c1(C(N2CCC(C)(CNC(C=CC=CCC)=O)C2)=O)cccc2nc(C(F)F)sc12 N1(CC2CC(=O)C23CCC3)CC2C3CCC(O3)C2C1 c1(C(=O)NCCOCCCNC(=O)CCC2CCOC2)ccc(OC(F)F)nc1 c1(OC)ccc(OC(F)F)c(CN2CCOC3CC23)c1.c1(N)cccc(OC)c1 Cc1nc2c(c(O)nn2C)c(C)c1CC(N1CCN(C(N(C)C2CC2)=O)CC1C)=O c1(OC)n[nH]cc1C(N1CCC(C(F)C(=O)NCC2(n3nccn3)CC2)C1)=O Nc1ccc(C(=O)NC2(CNC(C3CCC3)=O)CC(F)(F)C2)c(F)c1F c1(C(=O)Nc2cc(C(=O)OCC)sc2C)cc(F)ncc1OC c1(C(N2CC3C(NC(CCN(C)CC)=O)C3C2)=O)cccc2c1CCC(=O)N2 c1(C(=O)NCC2=CCN(C(C(CC)(C)OC)=O)CC2)c(C)ccc2n[nH]cc12 C#Cc1cc(C(=O)NC2CC2NC(C2(C(F)(F)F)CCCCO2)=O)cc(F)c1 c1(C(=O)NCC(c2ccc(Cl)c(Cl)c2)C)ccc(F)cc1C1CC1 Cc1cc(F)ccc1C=CC(=O)NCCC1CCN(C(=O)C=CCO)C(C)C1 N1(C(C(C)(C)C2CCC2)=O)CCC2(CC(C(=O)NC3CCc4c[nH]nc4C3)C2)C1 CCC(CC)(CC)C(=O)N1CCCCCC(NC(=O)C(c2ccccc2)C)C1 N1(C(C(C)NC(=O)NC)=O)CCCN(C(c2cc(C#N)on2)=O)CC1 CC1(C)CCC(C(=O)NC2CCN(C(=O)CCc3nnc(C(F)F)o3)CC2)C1 Cc1nnc2n1CCC2(C)C(=O)N1CC(C2(NC(C3CC3C(F)(F)F)=O)CC2)C1 c1(CNC(=NCC)NCCOCC(F)F)cnc(C)cc1C CCCCC(C(=O)N1CCC(C(N2CC3C(C)C3C2)=O)C1(C)C)C(C)C C(C(C)(CO)CC=C)NC(C1C(NC(C(C=C)OC)=O)COCC1)=O Cc1ccn(C(C)CC(=O)NC2CCC2CNC(c2ccc(C(F)F)s2)=O)n1 Cc1n[nH]c(C)c1CC(C)C(=O)N(CCN(C)C(C1NC(=O)CC1C)=O)C(C)C c1(C(=O)NCC2N(C(C(C)(C)NC(C=COC)=O)=O)CCC2)cnc2n1CCC2 c1(C(C(=O)OC)N(C)Cc2nc(CC)sc2)ccc(F)c(F)c1 C(C(C)(C(=O)NC(=O)COCCN(C)C)NC(C)C)SC.C1C(C(C)C)CN1 c1(C(N2CC=CC(NC(c3nccc(C)n3)=O)C2)=O)cnc2scnc2c1 C1(CS(=O)(=O)N(C)CC2(F)CCCC2)CC(C)(C)CO1 CCC(CC)C(C(=O)N1CCC(O)C1C(N1CCOCC1CO)=O)OC c1(C(=O)NCCN(C(=O)CCc2csc(C)n2)CC)ncc(C)cc1OC c1(C(=O)NC2C(NC(CCSCC(C)C)=O)C2)cnn2ccncc12 C1(CC)COC(C)(C)CN1C(=O)CCN(CCCO)C(=O)Cc1ccns1 CC(C)(F)CC(=O)NC1CCC(NC(=O)C(c2ccc(C(F)(F)F)cc2)F)CC1 CCCCCCC(C(=O)NC1CCOCC1NC(c1n[nH]cc1C)=O)NC(C)=O N1(C(c2cccn3ccnc23)=O)CCN(C(=O)CC2CC2)C2CCCCC2C1 N1(C(C2(CC)CCCO2)=O)CC(C(N2CC(C(C)C)C2)=O)CCC1(C)C C1(C(=O)NC2CC(CC(=O)N(CC(C)C)CCN(C)C)C2)CC12CCC2 c1(C(=O)NCC2CC(NC(c3ccc(C(C)=O)s3)=O)C2)ccc(Cl)nc1 C1(C(=O)NCCC2(C)CCOC2)(OC)CCN(C(c2nnsc2C)=O)C1 N1(C(C(CC)(C)OC)=O)CC(CNC(=O)C(C)(C)CCSC)C(F)(CO)C1 N1(C(C(C)NC(=O)C(C)(C)C)=O)CCC2C1CCCN2C(=O)C(F)=C1CCCC1 C1(CNC(c2nc(CCC)oc2)=O)CN(C(c2ccc(C)nc2N)=O)CCN1C n1(C(C)C)ncc(C(=O)NC2CCC(CNC(c3nsnc3O)=O)C2)c1F C1(C(=O)OC)CCC2CN(C(C)=O)CCC2C1.c12ccc(cc1)s2 C(CCCCCCC(=O)NCCCN(C)C(C1COC(=O)N1C)=O)SC N(C1COCc2c(Br)cncc21)C(C1CN(c2n(C)ccn2)C(=O)C1)=O Cc1oc(CNC(=O)CCn2cncn2)nc1C(=O)NCc1cnns1 c1(C(N2CC(NC(C3(OC)CCCOC3)=O)C(C)C2)=O)nc2nc(C)ccn2n1 CN1CCC(OC(=O)C(c2ccc(Cl)cc2)(C)C)C1(C)C C1(NC(c2cc3c([nH]2)CCC3)=O)CN(C(C2CC23CCCC3)=O)C2CCCCC12 N(C(=NCC(C)C)N(C)Cc1nc2c(s1)CCCC2)CC1(OC)CC(CC)C1 C(=O)(C(O)CCC(C)C)NC(C1N(C(CCc2cc(C)no2)=O)CCC1)(C)C C1(O)(CNC(C2CCC(=O)N2)=O)CCCN(C(=O)CCc2cnoc2)CC1 C1(NC(C(C)C#N)=O)CN(C(=O)C=CCOc2ccc(F)cc2)CC1OC C1(NC(c2ncsc2Br)=O)(CNC(C2(O)CC2)=O)CCOC1 CC(O)C(C)(C)C(=O)NCC(C1CCCCC1)NC(c1ccccn1)=O c1(C(=O)NC(C(CCC)C)C(=O)O)coc2c1N(C)C(=O)CCC2 Cc1cc(C(=O)NC2CC(C(=O)NCCc3ccn(C)n3)C23CCC3)cc(C)n1 C1(C(N(CCC(N2CCC2(C)CC)=O)CC#C)=O)CCC(C)=C(C)C1 C1(NC(COCc2cc(C)on2)=O)CN(C(=O)C(C)N2CCC2)CC1N=[N+]=[N-] c1(C(=O)NC23C(CN(C(=O)CCn4cc(Cl)cn4)C2)C3)ccc2ocnc2c1 c1(OC)c(C(=O)NC2CN(C(=O)C(c3ccccc3)O)CC2(C)C)cccc1Cl N1(C(CC2N(CC)CCC2)=O)CCOC(C(C)NC(=O)CNC(=O)OC)C1 N1(C(C=C(C)C)=O)CC(NC(=O)C#CC2(C)CC2)CC12CCCOC2 C1(C(=O)NCC(CC)Nc2ncncc2OC)CN(CP(C)(C)=O)C1 Cc1ccnnc1C(=O)NC1CCCC(CNC(=O)CCC2(C)CC2(F)F)C1 C1(CNC(CC2N(C)C(=O)CC2)=O)CN(C(c2ccncc2Cl)=O)CCN1C C1(NC(CC2CCC(C)CO2)=O)CC12CCN(C(C1(C(F)(F)F)CCC1)=O)CC2 c1(C(N2C(COC)(CNC(=O)CC3CC3)CCC2)=O)cc2c(OC)cccc2s1 c1(C(C)C(N2CCC(N(C(=O)Cc3cnns3)C)C2)=O)ccc(Cl)c(Cl)c1 C1(C(=O)OC)CCC(C(=O)NCC2CCCN2C(=O)CSc2ccccn2)CC1 c1(CC)nc2cc(NC(c3cc(C(C)(C)C)c[nH]3)=O)ccc2o1 c1(CC)ccc(N2CC(C(=O)Nc3ccnc(OC)c3)CC2=O)cc1 C1(CC(=O)NC(c2ccccc2F)CNC(C(CC#C)C)=O)CCC(C)(C)CC1 C1(CCCCNC(C2C(C(C)C)CCC2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)CC1 c1(C(=O)NCC(C)N(C(c2ccc(F)cc2F)=O)CC)cccn2cnnc12 C1(CNC(Cc2cccc(CC)c2)=O)CC(C)(C)CN1C(C1CC(OC)C1)=O c1(C(=O)NCC(CN(C(C(CC)c2ccccc2)=O)C)O)n[nH]c2c1CCOC2 c1(-c2ccc(CCSCCC)cc2)ccc(Cl)c(C(=O)O)c1N N1(C(c2ccc(C)cc2F)=O)CCN(C(C2CN(C)C2)=O)C(C)CC1C CN=c1[nH]c(=NCc2cccc3ncn(C)c23)[nH]c(=NCc2cscc2Cl)[nH]1 N1(Cc2ccc(CC)cc2)CCC(C(=O)Nc2ccc(I)c(Cl)c2)C(O)C1 c1(NC(C=CC(C)NC(C(CC=CCC)C)=O)=O)cccc(F)c1F c1(CC)cc(C(N2CC(N(C(=O)CN3CCCCC3)C)C(O)C2)=O)ccn1 c1(C(C2CCOCC2)CC)nc(-c2ccncc2)nn1-c1nccn1C Cc1ccc(C2CC2C(=O)NCc2ccc(N3C=CC=C(F)C3)cc2)cc1 c1(C(=O)NCC2CCCCC2NC(C23CC(C2)C3)=O)cc2n(n1)CCCC2O C(=O)(CC(C)CC(C)(C)C)N1CC(N(C(Cc2cc(C)on2)=O)C)C(C)(C)C1 C(=O)(CC(O)CN(C(=O)C(F)(F)c1cnn(C)c1)CCO)OC C1(NC)CCC(C(=O)NCCC(O)CNC(=O)C=C(C)C(F)F)CC1 c1(-c2scc(C(=O)NC(C)CCCNC(=O)CCF)n2)ccc(Cl)cc1 C(c1cnc2ccccc2n1)=CC(N1C(CN(C(=O)COC2CC2)C)CC(F)C1)=O c1(CNC(=O)N(c2ccccc2)C2CC2)ccc(C(F)(F)F)cc1Br c1(C(=O)NCC(CO)NC(CCCC#CC)=O)cc2ccccc2cc1O N1(C(C(C2CN(C(C(C)C3CCC3)=O)C2)O)=O)Cc2nncn2C(C)C1 N1(C(c2c(CC)csc2)=O)CCOC(C(C)NC(=O)CNc2cccnc2Cl)C1 C(C)(C)(CCCC(=O)NCC1CC1[N+](=O)[O-])NC(C1(COC)CCCO1)=O C1(C(N2CC2C)=O)(COC)CC=CC1.C(=O)(C(=O)NC(C)C)NC(C)C C1(NC(C(CC2CC2)NC(c2cn(C)nn2)=O)=O)CN2CCC1C2 n1(CC)ccc(C(=O)NC(C)(C)CN(C)C(c2cc(C)c[nH]2)=O)cc1=O c1(C(N2CCCC(N(C(c3csc(O)n3)=O)CC)C2)=O)c(F)ccc(C)c1F C1(C(=O)O)(N(c2ccccc2)C(Cn2cc(CC=C)nn2)=O)CCOCC1 c1(NC(C2CC3(CC(NC(C(COC)N(C)C)=O)C3)C2)=O)c(C)ccn(C)c1=O C(=O)(C1=CCCOCC1)NCC(CC(=O)N(CC(C(=O)NC)C)C)OC Cc1nonc1CC(C(=O)O)N(c1ccn(-c2ccccc2)n1)CC(=O)N(C)C C1(NC(C2(COC)CCC2)c2nn[nH]n2)CCC(P(C)(C)=O)C1 c1(C(N2C(Cc3cn(Cc4cn(C)nn4)nn3)CCC2)=O)nc[nH]c2nccc1-2 C(CNC(C1CCCSC1)=O)(CC(F)(F)F)NC(=O)C=CC1CCCC1 n1(C(C)C)cc2cccc(CNC(=O)NCC3CNC(=O)CO3)c2n1 CC(CS(C)=O)N=c1[nH]c2c(c(=NCCc3cc(O)n(C)n3)[nH]1)COCC2 N1(C(c2ccc(SC)o2)=O)CCC(C)C(CNC(=O)C(O)C(C)C)C1 c1(N(C(C)=O)C)nc2c(s1)CN(C(C(=O)NCCC(=O)N(C)C)C1CC1Cl)CC2 c1(N(C(C2CCC(OC(C)=O)C2)=O)Cc2cncnc2)n[nH]c2cc(C)ccc12 CC1CC(NC(c2c(Cl)n[nH]c2C2CC2)=O)CN(C(=O)C(C2CCOCC2)O)C1 c1(OCC(N2CC(CNC(c3n(C)nnc3)=O)C2)=O)ccc(C(N)=O)cc1 C1(CC(=O)NC2C(NC(=O)CCCc3ccsc3)C2)CCC(=O)NC1=O Cc1ccc(C(=O)Nc2ncc(CCNC(=O)C(C)(C)O)s2)cc1Br N1(C(c2cc(OC)n[nH]2)=O)CCCCC12CC(NC(c1cc(C(F)F)cs1)=O)C2 N1(C(C2CCC(=O)O2)=O)CCC2(NC(c3ccc(Br)nc3O)=O)CCCC12 C1(O)(CNC(C(CCC)O)=O)CCN(C(c2cnnn2C)=O)CC1 c1(C2(O)CCC2)ccc(Cl)cc1.C(=O)(C(O)CC1CCNC1)N1CC(SCC)C1 C(=O)(C(CCC(C)C)NC(c1scnc1C)=O)NCc1nnc(C)o1 N1(C(COCC)=O)CCC2(CCC(NC(c3c(SC)cnn3C)=O)C2)CC1 c1(CNC(CCC)=O)c(C)nn2c1CN(C(C1CCS1(=O)=O)=O)CC2 N1(C(C2CCCC(C)C2)C(=O)NCC(C)C)CCC(C)c2ccccc21 CS(=O)(=O)C1(C(=O)NCC2CCC(NC(=O)C(C3CCOCC3)=O)C2)CC1 Cc1cncc(CNC(C2CC(NC(C3CC(F)(CF)C3)=O)CCO2)=O)c1 N1(C(c2cc(OC)nn2C)=O)CC2(C1)SCCC2NC(=O)CN1CC2CC2C1 C1(F)(C(N(CCOCC#C)C)=O)CCCN(C(C2(OC)CCOC2)=O)C1 c1(NCCc2ccc(F)cc2)ncc(Cl)cc1CN1CC=CC1 O=C(CC1NC(=O)c2ccccc21)OCC=CC1CCCCC1 C1(C(N2CCN(C(=O)CCCF)C(c3ncc[nH]3)C2)=O)CC12CCCCC2 n1(CC(=O)N(C(CNC(C2(C)CC(=C)C2)=O)C)C)ncc(O)nc1=O c1(C(=O)NCC2CN(C(C3C(F)(C(=O)OC)C3)=O)C2)cc2n(n1)CCCO2 c1(C(N(CCNC(CC2CC(=C)C2)=O)CCOC)=O)cc(C)nc(C)n1 c1(C(CC2CC2)OC(c2cccc(C(C)=O)n2)=O)ccc(F)c(Cl)c1 N1(C(C2(F)CCCC2)=O)CCN(C(C2CC2C(F)(F)F)=O)C(c2ccccn2)C1 N1(Cc2c(CC)onc2C)CCCC(CO)(NC(c2cc(C(C)C)n(C)n2)=O)C1 c1(CNC(C(CNC(C2COC(=O)N2)=O)OC)=O)cc(C)cc(F)c1 Cc1cnn(C)c1C(=O)NCC(C)CC(=O)N1CCC(c2nn[nH]n2)C1 C1(C(=O)NC(CC)CNC(C2(CCOCC)CCCC2)=O)C(C)(C)C1(C)C N1(C(C=Cc2cc(C)on2)=O)CCC2CN(C(=O)C(O)CC(C)C)CC2C1 N1(C(CC=C)=O)CCc2ccccc2C1CNC(c1ncccc1C)=O c1(C(=O)NCC(CNC(C(C)SC)=O)C)cc(-c2cccnc2)nn1C CN=S(C)(=O)c1cccc(C(N2CCCCC2CNC(c2nccn2C)=O)=O)c1 C1(CC(=O)N(CCN(C(c2cc(CSC)[nH]n2)=O)CC)CC)CC(O)C12CCC2 C1(NC(C=CC(CC)=CC)=O)CCN(C(=O)C(C)(C)n2cccn2)CCC1CO c1(C(=O)NCc2c(C(N3C(CC#C)CCCC3)=O)nco2)ccc(F)cc1F C1(C(=O)NCC2(CC)CCOC2)CCCCC1CNC(c1nc(C)oc1C)=O C(=O)(CC(O)CC(C)(C)C)NCC12N(C(C(C)NC(CC)=O)=O)C(CC1)CC2 C12CC3(C1)CC3C(=O)N2C.C1(C(N(C(CO)C2CC2)C)=O)C(C#N)C1(C)C c1(C(=O)NCCC(CNC(C(C#C)(C)C)=O)O)cc(N)ccc1Cl C(=O)(C(C(C)(C)C)NC(C)=O)N(C)CC1N(C(CNC(C)=O)=O)CC(F)C1 N1(C(c2c(C)nco2)=O)CCN(C(=O)C(CN(C)C)C(C)C)C(CC(F)F)C1 C(=O)(C(F)CCC(C)C)NCC1(OC)CCN(C(C2CC(C(C)C)=NO2)=O)C1 CC(CNC(C1CCC1(F)F)=O)(Cn1cccn1)NC(=O)CSC(F)F C(C(=O)NCC1(O)CN(C(C2(O)CC(C)(C)C2)=O)C1)(C(C)C)n1cc(C)nc1 N1(C(C2C(=O)NCC2)=O)CC2(NC(c3cn4ccsc4n3)=O)CCCC2(F)C1 N1(C(C=CCCC=C(C)C)=O)CCOCC1CCNC(=O)CC1(O)CCCOC1 CN1C(=O)CSC1=CC(=O)N(C)CC1CCN(C(C2CCCC(=O)N2)=O)C1 C1(CC=C)(NC(=O)C(C)C(C)O)CCCN(C(c2c(Cl)cnn2C)=O)C1 c1(NC(C(=O)NCC2CCCN2)=O)cc(C(F)(F)F)cc(Cl)c1 C(CC(C(C)C)NC(=O)C(c1cccc(F)c1)O)N(C(C1C(CC)C1)=O)C N1(c2cc(C(=O)OCC)ncn2)CC2CC1CN2CCc1ncn(-c2ccccc2)n1 c1(C(N2CC(OC)CC(NC(C(CC=C)CC)=O)C2)=O)ccc2oc(C)nc2c1 N1(NC(CC(=O)NC(CCN(C(c2ccncc2)=O)CC)C)=O)CCN(C)CC1 CCC(CC(=O)N1CCOCC1CNC(=O)C(F)OC(F)(F)F)CC(C)C C1(CN(C(=O)CCCN(C)C(C2CCCO2)=O)C)CCCOC1 N1(C(C2(COC)CC=CC2)=O)CCC2C(CCN2C(=O)CC(C)(C)C2CC2)C1 C1(C)(C(=O)NCC(CCC)NC(c2cc[n+]([O-])cc2)=O)CCN(C)C1 c1(C(N2CCC(CN(C(=O)C=C3CCC3)C)C2)=O)cc(F)cc2ccncc12 c1(C(N2C(C)C(NC(=O)Cc3csnn3)CC2)=O)cc2cccnc2s1 C1(CNC(c2c(C)oc(Cl)n2)=O)CN(C(=O)COC2(C)CCC2)C2CCCCC12 c1(C(=O)NC2CCC(CC(=O)NC(c3ccc(C)cn3)C)C2)cc(C)cc(O)n1 C12(CNC(c3ccc(C(F)F)cc3)=O)CC1CN(C(C1C(F)(F)C13CC3)=O)C2 C1(OCCNC(C2(CCC)CC2)=O)CCN(C(=O)CC2CCCO2)C1 C#CC1(C(=O)NCCCCCCOC)CCN(C(c2cnc(N)cn2)=O)C1 C(=O)(C(CNC(c1cnnc(O)c1)=O)C(C)(C)C)NCc1ncn(C)c1 Cc1cc(C)c(CNC(=O)CC2(C)CCN2C(C2CCCC(=O)CC2)=O)cn1 C=CCC(C)(C)C(=O)NC(CNC(c1ncsc1C)=O)C(C)C(C)C C1(CNC(c2ccc[nH]2)=O)CCN(C(=O)CC2CCSCC2)CC1(F)F c1(C(N2CCC(NC(CNC(=O)NC)=O)(CO)C2)=O)ccc2c(C)noc2c1 C(C)(C(CC(=O)NCC1CNC(=O)C1)NC(=O)C(F)(F)C1CC1)OC CC(C)(CC(=O)N1CCOCC(F)(CNC(C2CCC=CCCC2)=O)C1)C(F)F CCC1=C(C(=O)N2CC(CNC(c3[nH]c(C)cc3C)=O)CC2C)SCCO1 c1(CC(N2C(C(C)(C)NC(C(CC)F)=O)CCC2)=O)ccc2nonc2c1 c1(C(N(C(CCNC(C(C=C)(C)C)=O)C)C)=O)cc2cc(F)cc(F)c2nc1C CCC1=C(C(=O)N2CCCC(CN(C(=O)C(O)C(C)C)C)C2)SCCO1 O=S(=O)(Cc1cc(Br)ccc1Cl)C12CC(C1)C2 C(=O)(C(F)(F)C(C)O)NCC1C(NC(c2c(COC)cco2)=O)C1 c1(NCC(C)NC(=O)NC(COC(C)(C)C)CF)ccccc1 c1(CC(=O)N(CCOCCN(C(C(C)OCCCC)=O)C)C)cc(CC)nn1C c1(CCC(=O)NCC2(OC)CCN(C(COC)=O)CC2)cnc2ncccn12 CC1(C)OCCC1C(=O)NC1CCCC1NC(C1(C#N)CCCC1)=O n1(CC=C)cc(C(=O)N(C(C)(C(=O)NCCN(C)C(N)=O)C2CC2)C)cn1 c1(OCC)cc(C(N2CC(N(C)C(=O)OC(C)(C)C)C(F)C2)=O)ccn1 N1(C(c2cc(C)c(C)[nH]2)=O)CC2CCN(C(=O)C=CC3CCCO3)CC(C2)C1 O(NC(=O)C(C)C(C)NC(c1ncn2ccccc12)=O)CCOCC#C c1(OC)ccc(C(=O)NC2CCN(C(c3cc(C)n(C(F)F)n3)=O)CC2)nc1 C(=O)(C(C)(F)CC1CCCC1)NC1C(CNC(CCCn2c(C)ncc2)=O)C1 C(=O)(C(F)C(C)(F)F)N(CC(C(N1CC(C)(COC)C1)=O)C)C N1(c2ncc(C(=O)OC)s2)CCN(CC2CCN(c3ccc(F)cc3)C2=O)CC1 c1(C(=O)NCC2N(C(CC=CC)=O)CCC2C)cnc2c(cnn2CC(C)C)c1 C=CCC(C)(C)CC(=O)NC1(C(N2CCCC(COC)C2)=O)CSC1 C(=O)(C1=CCCN(C(=O)COCC2CCCC2)C1)N(CCOC)C c1(C(N(C2CCN(C(c3c[nH]nc3OC)=O)C2)CC)=O)cc(C)n(C)c1 C(=O)(C#CC1(C)CCCO1)N1CCCC(NC(C2(C)CC=CC2)=O)CC1 C1(NC(CC2C=CC(NC(c3c(NC)scn3)=O)C2)=O)CCCCC1C(N)=O c1(C(=O)NC2(CCC(=O)NC3CC3c3cccs3)CC2)cccc(CO)c1Cl C(=O)(CC(CC)CCCC)N1C(C(=O)Nc2nccc(SCC#C)c2)C2CC2C1 N1(C(c2occ(C)c2C)=O)CC(C2CCCN(C(=O)C(C)(C)C3CC3)C2)C1 N1(C(=O)CCc2cnc[nH]2)CC2(CCCCN2C(C23CCC(CC2)OC3)=O)C1 c1(OC)cc(Cl)ccc1C(=O)C(=O)NCCC(C)NC(c1ccc[n+]([O-])c1)=O c1(CC(=O)NCC=CCNC(C2CN(C)C(=O)N2)=O)cn2c(n1)CCCC2 CCCC(CNC(C1(NC(=O)CC(C)(C)OC)CC(F)(F)C1)=O)CCO C(N=c1cc(C)nc(N2CCC(C3CCCO3)CC2)[nH]1)C1(CC)CC1 C(=O)(C1=NOC2COCC12)NC1(CC)CN(C(c2csc(-c3ncc[nH]3)n2)=O)C1 C(=O)(C(C)Cn1ccc(C)n1)NCC(C)(C)NC(C1CC(=C)C1)=O c1(NCc2n(C(C)C)ncn2)[nH]c(=NC2CCCC2C(N)=O)nc2scnc12 n1(CC)c(C)c(C(N2CC(C(=O)O)CC(O)C2)=O)c2cc(OC)ccc12 c1(C(=O)NCC2(O)CC(NC(CCC=C(C)C)=O)C2)ccc(Br)c(C)n1 C1(CC(=O)N(C2CCN(C(c3ccc(C)nc3)=O)CC2)CC)CCC(C)CO1 c1(OC)ccc(F)cc1NC(C1CC1NC(c1nc(C)no1)=O)=O N1(C(CC(=O)NC)=O)C2CCC1CC(NC(=O)COCC1CCCOC1)C2 N1(C(CCN(C(C)=O)C)=O)CCC(OCCNC(C2CC=C(C)CC2)=O)CC1 C(CN=c1[nH]c(C)cc(=NC2CC(C)C2)[nH]1)n1ccc(C(=O)OCC)n1 C12CCN(CC1C)C2=O.c1(CNC(CC=C)=O)ccccc1OCC(N)=O C(=O)(CC1=CCN(C(c2cc(C(C)C)no2)=O)CC1)N1CCC(OC(C)=O)C1 Cc1nn(C)cc1CC(=O)NCC#CC(N1CCCC2CC12)=O O=C(CCC(=O)NC1CCCC1)NCC(CO)NC(=O)CC1CC2(COC2)C1 Cc1[nH]c2ccccc2c1CC(=O)NC1CC(NC(=O)C(C)(C)C#N)C12CCC2 C(C(C)(CC(C)C)NC(c1cc(C(C)C)oc1C)=O)NC(C(CC)C#N)=O C1(O)(CNC(CC(C)OC)=O)CC2CCC(C1)N2C(=O)C(=O)N=S(C)(C)=O C1(NC(C(COC)C)=O)CN(C(c2ccc(O)c(Br)c2)=O)CC12CCC2 c1(C(N2CC(NC(CNC(c3ccc(C)s3)=O)=O)C2)=O)oc2c(C)cccc2c1C c1(NCC(CC)(C)CC)[nH]c(=NCCC2(C)CC2(F)F)nc2c1cnn2C(C)C N1(C(c2scc(C(C)=O)c2)=O)CC(C)OC2(CCN(C(C3CCCC3)=O)CC2)C1 C(=O)(C1CCc2nccn21)N1CCC(CC(=O)NC(C(C)C)C)C1 N1(C(C23CCC(C)(C2)CO3)=O)CC2(COC(CNC(=O)Cc3ccc(Cl)s3)C2)C1 C1(C(N(C2CCCN(C(c3cnn(C)c(=O)c3)=O)C2)CC)=O)CC(=O)N(OC)C1 c1(OC)ccccc1C(C)C(N1CC(CNC(c2c(C)coc2C)=O)C(C)C1)=O O=C(Nn1nnc2c1CCCC2)C1CC=CCN1C(C1CS(=O)C1)=O N1(C(CC(C)N(C)C)=O)CCCC(NC(=O)CS(=O)(=O)NC(C)(C)C)CC1 CCCC(C)(O)CC(=O)NCC(C)NC(C1CC(=O)N(C(C)C2CC2)C1)=O CC1(C)CNCC(CNC(=O)C(=O)Nc2cccc(OC3CC3)c2)O1 c1(CC)c(NC(=O)NC(C)(C)CO)cnn1C1CCCC1 c1(C(=O)NC(C)CN(C)C(C2CC2C(F)F)=O)cc2cc([N+](=O)[O-])ccc2[nH]1 c1(CC(=O)NCC(C)NC(C(C)NS(CCCC)(=O)=O)=O)nc2ccccc2s1 Cc1cc(C(=O)NCC2CCN(C(C3CC(F)C(=O)N3)=O)C2)cc(Cl)c1 N1(C(CN(C)CC)=O)C2CCC1CC(CNC(c1ccsn1)=O)C2 Cc1cc(C(N2CC=CC2(C)C(N2CCOC(CC3CC3)C2)=O)=O)cc(F)c1 N1(C(CCC(=O)NCCC)=O)CCC(O)(CCNC(=O)C(C)NC(C)=O)CC1 c1(C(=O)OC)coc(C=CC(=O)NCCC2CCCN2C(=O)C=CC2CC2)c1 N1(C(c2cnn(C3CC3)c2)=O)CCOCC1CO.c12ncc(cn1)COCCO2 C1(CC)CCCC(NC(c2sccc2CNC(c2cccn2C2CC2)=O)=O)C1 n1(CC)cc(CC(N2CC(CNC(c3cc(C(C)=O)on3)=O)C2)=O)cn1 C1(C(=O)NC(CCNC(C2(COC)CCC2)=O)C)CSc2ccccc2O1 C(=O)(CCC(C)NC(c1ccn(C)n1)=O)NC1(C(=O)NCC#C)CC1 CC1C(O)CCCN1C(C1(C)C=CCN1C(=O)CSC1CCCC1)=O C(C#CC(=O)N1CCCc2nccn21)NC(C(C)C1CCCO1)=O c1(N2CCC3(CCCN(C)C3)CC2)nc(=NC2CCOC2)[nH]c2c1SCC2 C(=O)(C1=CCN(C(=O)OC(C)(C)C)C1)N1CC2C(NC(CC(=O)NC)=O)(C2)C1 C1(NC(C2(CC)CN(C(=O)COc3ccn(C)n3)C2)=O)CCOC1(C)C C12CN(CCC1F)C(C)(c1cccs1)C(=O)N2.C(C(=O)NC(C)C)(C(C)C)SC N1(CC(=O)N(CCC)Cc2ccc(OCCC)cc2)CCOCC1(C)CC C1(CNC(c2ccc(Cl)s2)=O)(CNC(=O)C(C2CCCCC2)O)CC12CCC2 c1(C(c2nnnn2C2CCOC2)NCC2C(C(=O)OC)CC2)cc(C)ccc1Cl C(=O)(C(CCSC)NC(=O)CC1COCCO1)N(CC(C1CCC1)OC)C CCCCCCCCCC(=O)NC1CN(C(c2cnn[nH]2)=O)CC2CC12 Cc1cc(F)ccc1CC(N1CCCCC(CNC(C2(C)CCNC2=O)=O)C1)=O c1(C(=O)NC(CCOC)CNC(C2CC23CC3)=O)ccc(C)c([N+](=O)[O-])c1 C(CC(C)(C)C(=O)N1CCC(NC(=O)C(O)CC2CCOCC2)C1)SC C1(C(=O)NC(C)CCNC(c2ccncc2O)=O)CC2CCCCCC12 C1(C(=O)NCc2ccc(C(=O)NC3C=CC(CC)C3)nc2)CC2CC(=O)C1O2 C(=O)(C(CC)CC(F)F)N1CC(CC=C)(N(C(c2cc(=N)[nH]cc2Br)=O)CC)C1 c1(C(=O)NC(CNC(c2c(Cl)c(C)n(C)n2)=O)C(C)(C)C)cn2c(n1)CCCC2 C1(C(=O)NCC2(COC)CN(C(=O)CC3CCCO3)C2)CC2CC(O)CC(C1)C2 N(C1CCSc2ccc(F)cc21)C(C(=O)N(CCCOC(C)C)C)=O N1(C(c2ccnc(C(C)C)n2)=O)CCN(C)C(CNC(=O)C=C2CCC(C)C2)C1 N1(CC(=O)NCCC(=C2CN(C(C(C)OC3CCCC3)=O)C2)F)CCC(F)CC1 C=C(C)C(C)(O)C(=O)NCC1(NC(c2sc(COC)nc2C)=O)CCOC1 c1(OC)cccc(OC)c1CC(c1ccc(C)nc1C)c1nnnn1C.N c1(OC)ccc(OC=CC(=O)NCCCN(C(C2CNC(=O)C2)=O)C2CC2)cc1 C1(C(=O)NC(C(C)C)C(=O)N(C)CC2CCN(C)C2)CC2(CC2)CN1C C#CC1CN(C(c2cc(C)sc2C)C(=O)Nc2ccccc2OC)CC1O c1(OC)cc(-c2cn(CC3CCCN3C(C3SCCS3)=O)nn2)ccc1F Cc1ccc2c(c1)CCC(C(=O)NCCN(C)C(C1CCC(C)O1)=O)O2 N1(C(c2c(OC)csc2)=O)C2CCC1CC(NC(c1n[nH]c3c1CSCC3)=O)C2 c1(C(=O)NC2C3N(C(c4cn(CCC)nc4)=O)C(CC3)C2)ccc2c(c1)CCC2 c1(CCN(C2CCN(c3cc(C)ncn3)CC2)C)ccc(Cl)cc1F c1(N(CCC#C)C)ncccc1C(=O)NCC(C)NC(C1CCN(C)CC1)=O CCCCC(C(=O)NC(C)COCC)NC(=O)Cc1cccn1C N1(C(CC=C)=O)CCCC(N(CCO)C(c2ccc(OC(F)F)cn2)=O)C1 N1(C(c2nc(C(C)C)oc2)=O)CC2OCCN(C(C3(C)CCC(=O)N3)=O)C2C1 c1(C(N(CCCNC(CCCSC)=O)C)=O)cccc(C(F)F)c1F N1(C(C2(OC)CCC2)=O)CC=CC(NC(=O)CCCn2cccn2)C1 C(=O)(C(C)(C)CC(F)F)NC1CCN(C(CC(COC)(C)C)=O)C(C)C1 C1(CC(C)(C)C)CN(C(C2CCC3(CC3)C2)=O)CCN1C(c1csc(C#N)c1)=O CC1C(NC(c2cccc(=O)o2)=O)CCCN1C(c1cc(C(F)(F)F)ccn1)=O Cc1ccc(O)c(CC(=O)NCC2CCC(NC(=O)C(C)(C)CC3CC3)C2)c1 C1(NC(C2(CC=C)CC=CC2)=O)CCN(C2CCCN(C)C2=O)CC1O N#CC1(CCC(=O)NCCC2(C(=O)NC3CCCOC3)CC2)CCC1 N1(C(CCCCC)=O)CCC(NC(c2ccc(OC)cn2)=O)C(CO)CC1 C(=O)(C1COc2ccccc21)NCC1(O)CCCN(C(COCCCCC)=O)C1 C1(CC(=O)NC2CC2NC(c2ccn(CC3CCCO3)n2)=O)CCCNC1=O c1(CC(=O)NCC(CC)NC(=O)Cn2cc(CN(C)C)nn2)nncn1C N1(C(C(COC)N(C)C)=O)CCN(C(c2cc(O)n(C)n2)=O)C(CC(C)(C)C)C1 C1(CC(=O)NCC(C#C)CC)CC(NC(=O)Cc2cccc(F)c2)C1(C)C C=CCCCC(C(=O)NC(C)(C)CC=C)NC(c1nccnc1N)=O C12(NC(C3CC(SC)C3)=O)CCCC1N(C(=O)CC1CCC(O)C1)CCC2 Cc1nc(Br)cnc1NC(=O)Cc1ccc(F)cc1 C(=O)(C(O)CC(F)F)N1CC(CNC(CC2(C(F)(F)F)CC(=O)NC2)=O)C1 N1(C(c2ccc(SC)s2)=O)CCC(NC(=O)CC2CCN(C)C2=O)C(CO)C1 Cc1cc2cc(C(N3CC4ON=C(CNC(C5(O)CC5)=O)C4C3)=O)[nH]c2cc1Cl c1(C(N2CCC(CN(CCC3=CCCCC3)CC)CC2)=O)cnn2cccnc12 c1(C(=O)NCC2(CN(C(CCCOC)=O)C)CC2)cc(F)c(C(C)C)cc1F C(=O)(C1=CCCCC1C)NC(C)CCCNC(C1(C)CC=CC1)=O N1(C(CCC=CC)=O)CC2CC2(CNC(c2cn(C)nc2COC)=O)C1 c1(OCC)ccc(C(=O)Nc2ccc(-c3cccnc3C)s2)c(F)c1 Cc1noc(Cl)c1CC(N1CCC(C)(CNC(C2(C)CC(C)(C)C2)=O)C1)=O CN1CC=C(CC(=O)NCC2(NC(c3cccc4c3C(=O)NC4)=O)CCC2)CC1 C1(NC(c2nc(C)c(C)s2)=O)CN(C(C2(C(N)=O)CC2)=O)CCC1C C(=O)(CCC(CF)CF)N1C(C(=O)NCCCC(=C)Cl)CCOCC1 C1(NC(C(F)=C(C)C)=O)CC2CCC(C1)N2C(c1ncc(C(F)(F)F)cc1N)=O C1(CC(=O)N(C(C)CCNC(C23COC(CF)(C2)C3)=O)C)CCS(=O)(=O)CC1 CC(O)CCCC(=O)NCC1CN(C(=O)CSCc2cccnc2)CCO1 c1(C(C)=O)ccc(C#N)cc1.C123CC(C1)N(C2)C(=O)N3CC(C)(C)C C1(N(C(CC2(C=C)CCC2)=O)C)CCCN(C(C2CCC(CCCCC)O2)=O)C1 C=C(C)CC(=O)NC(C)(CNC(=O)C(C)COc1ccccc1)CC N1(C(CCC)C(=O)OCc2ccc(F)cc2F)CC(=O)NC2(CCCC2)C1 CN1CCCC(C(=O)NCC(C(F)(F)F)N2CCN(C(c3cnsc3)=O)CC2)C1 C1(C(N(C(CCCC)C)C)=O)C=CCN(C(C2(C(C)C)CC2)=O)C1 C=CCC(CC(C)C)C(=O)N1CC2CC1CN(C(=O)C(C)(C)COCC(F)F)C2 N(C(=NCCCCN(C)C)NC1CC2CCC(C1)N2C)C(C=C)C C1(C)(CNC(C(Cc2ccc(C)cc2)C)=O)CN(C(C2CC(F)(F)C2)=O)CC1C Cc1cc(OCCCC(=O)NCC(C)CNC(C2CC3CCC3C2)=O)ccc1Cl c1(COCC)nnc(N2CCC(N(c3ccsc3)C)CC2)n1CSc1ccco1 C(=O)(C1CCc2c(Cl)cccc21)N1CCC(C(CNC(C2(CC)CC2)=O)F)CC1 CC1(C)CN(C(=O)C=CC(F)(F)F)CC1C(N1CCC(C)(O)C1)=O Cc1c(C(=O)NCC2CC2NC(=O)CN2CCCC2=O)cnn1C1CC1 C(=O)(C1Cc2ccccc21)NC(C1(O)CN(C(c2c(N)ncc(C)c2)=O)C1)C c1(C(C)NC(c2n(CCC)nnn2)c2ccsc2Cl)ccc2c(c1)CCCC2 c1(CC)cccc(NC(=O)NC(C)CC2CCN(C)CC2)c1C CC1CC(CNC(C2CC(=O)C2)=O)CCN1C(=O)CN(C)C1CC1 c1(CN2C(CNC(c3c(C)ncs3)=O)CCC2)cccc(S(C)(=O)=O)c1 CN1CCCC12CN(C(C1CC=CCN1C(=O)COC1CCC1)=O)C2 c1(N(C(=O)Cc2cc[nH]c2)C2CC2)ccccc1.N12CCC(C1)C(=O)NC(C)C2=O C1(CC)(NC(C2CCC(O)CC2)=O)CCN(C(=O)C(n2cc(C)cn2)C)CC1 C1(COC)CCN(C(C2CC23CCN(C(=O)CC2(O)CCC2)C3)=O)C1(C)C c1(CC)nc(C(=O)NC(C(N2CCC(C(N)=O)(C)C2)=O)C2CC2)c(C)o1.C(N)=O CCC(C)C(CO)CN=c1[nH]c(=N)[nH]c(=NCCCc2nc3ccccc3[nH]2)[nH]1 CC1(C)C2CCC1(C(=O)NC(C)(CO)C(=O)NCC(O)C(F)F)C2 CON(CCO)C(=O)C1CCCCN(C(=O)CC2CNC(=O)O2)C1 C12(CCCN1C(=O)CC1CCCN(C)C1)C(=O)NC2.C1(CCC)CC(N(C)C)C1 C1(CNC(CN(C2CCCC2)C)=O)COCCN1C(=O)C(C1CCOCC1)=O N1(C(c2cc(CCC)n(C)n2)=O)CCCC2C1CCN2C(c1cncc(C)c1)=O CCCC(C)(O)CC(=O)NCCC1CN(C(c2ccc(N3CCC3)nc2)=O)C1 N1(C(C(c2ccnn2C)C)=O)CCCCCCC1C(=O)NC1(CO)CCOCC1 C1(COC)CC(CNC(C23CSCC2C3)=O)N(C(=O)CC2CCSC2)C1 S(=O)(=O)(c1cc(C(=O)NCC2(O)CCN(C(=O)C(O)C(C)C)C2)co1)NC Cc1nc(N2CCC(c3cccc(F)n3)C2)c2cnn(C(C)(C)C)c2n1 C1(C)(C(N(C(C)CNC(=O)Cc2csc(NC(=O)OC)n2)CC)=O)CC(C#N)C1 C1(NC(C(CSC)O)=O)C2CN(C(C3CCOC3c3ccc(Cl)cc3)=O)CC12 c1(C(=O)NC2CCC(NC(C(CC)C(C)O)=O)CC2)cccc2c1OC(F)(F)O2 Cc1cc(CC(N2CCC(Cc3ccn(C)n3)C2)=O)on1 C1(CCOC)CC(Oc2ccccc2)CCN1 C1(CC(=O)N(c2ccccc2)C2CC2)CCN(Cc2c[nH]nc2-c2ccco2)C1 C#CCC(O)C(=O)NCCCCNC(=O)Cc1cnc(C(F)(F)F)s1 c1(NC2CCCC(C(=O)Nc3ccc(OCC)cc3)C2)ncnc2n[nH]cc12 N1(C(CC)=O)CC(N(C(=O)C(C(C)O)NC(=O)OC(C)(C)C)CC)C(C)(C)C1 N1(C(C2C(NC(c3c(C)cccc3)=O)CCC2)=O)CC2CC=CCC2C1 Cc1cc2[nH]c(C(N3CCCCC3CNC(=O)C(C3CC3)N(C)C)=O)cc2s1 N1(C(C2(C#C)CC2)=O)CCCC(CNC(c2nccnc2C)=O)C1 CCCC(CCCNC(=O)CCC(C)OC)NC(c1c[nH]c(Br)c1)=O N1(CCNC(c2cc(F)cc(F)c2Br)=O)CC2CC(C1)C1CCCCN1C2 CCCC(C(O)C(=O)N1CCCC1C1CCCC1)NC(=O)CCCC(=O)C1CC1 C1(NC(c2c(OCC=C)cccc2)=O)CN(C(=O)CCCC(C)C)CC1C=C c1(SCC(=O)N(C)CC2(NC(=O)CCC3CCOC3)CC2)cccc(C(F)F)c1 C1(CC(=O)NC(COCC)C(C)C)CC(O)CN1C(c1cscc1CC)=O N1(C(CC(=O)Nc2nccs2)=O)CCC2(CCC(NC(c3cc[nH]n3)=O)C2)C1 N1(CC(=O)NC(c2ccccc2F)CNC(C2(O)CCOC2)=O)CCCCC1=O c1(NCCCC(=O)NC2(N)CC[Si](C)(C)C2)ccc([N+](=O)[O-])cc1 N(C(=NCCCOc1ccncc1)NCc1ccco1)CC1C(CO)CCCC1 C(=O)(CC(F)(F)CC)N(C(CC(=O)NCC1CN(CC)C(=O)O1)CC)C N1(C(c2ccc(Br)cc2)C(=O)NC(CC)(C)C)CCCC(O)(c2ccsc2)CC1 N1(C(C(c2c(Cl)cccc2Cl)C)=O)CCN(C(c2c[nH]nc2F)=O)C2(CC2)C1 C(=O)(C1=CCCCCC1)NCC1C(C(=O)NC2C(c3n(C)ncc3)OCC2)C1 c1(C2CCN(C(N3CC(C)(C)OCC3)=O)CC2)ccc2ccccc2n1 c1(C(=O)NC2CCN(C(CC3CC(=O)NCCC3)=O)C2)cccc2oc(O)nc12 C1(C)(C(N(CC(C)(C)CNC(C2CC2C(C)(C)C)=O)C)=O)CC(C)(C)C1 c1(C(=O)NCC(CO)NC(=O)CSCc2ncc[nH]2)sc(F)cc1Cl c1(OC)ccc(CCNC(=O)C(=O)NCCC2CCC(N)C2)cc1 N1(C(C2(C)CC=CC2)=O)CC2C3CCC(C2C1)N(C(c1cnn2c1CCC2)=O)C3 C(=O)(CCCCN(C(=O)CC(C)NC(=O)CC1NC(=O)NC1=O)C)NC C1(NC(C2COC3COCC3O2)=O)CCCC2(C1)CC(O)C2 C1(C(=O)NC(CN(C(=O)C(C)(c2ccccc2)N(C)C)C)(C)C)CC(C)(C)O1 c1(C(c2n(CC=C)nnn2)NCC2(C3CC3)CCC2)c(Cl)ccc(F)c1Cl c1(CCC)cc(C(N2CC(O)(CNC(=O)C3=CCSC3)C2)=O)ccc1Cl CCCC(O)CC(=O)NCC1(COC)CCN(C(C)C(=O)NCCC(C)C)CC1 N1(C(C2(C(=O)OC)CC2)=O)CCC(C(=O)NC2CC2(C)C)=C(F)C1 c1(C(N2CCC(NC(C(C)=C(CC)C)=O)C(F)C2)=O)c(N)ccc(F)c1C C1(O)(C(N2CCC(NC(c3cc(OC)ncc3)=O)(CF)C2)=O)CCCCCC1 c1(N2CC(NC(C(C)CNC(=O)OCc3ccccc3)=O)C2)nc(Cl)c(C#N)s1 N1(C(c2c(OC)scc2)=O)CC2CCC(C1)N2C(=O)Cc1ccc2c(c1)COC2 Cc1[nH]nc(C(=O)Nc2ccc(CCS(C)(=O)=O)cc2)c1F c1(CN2CC3(C(C(=O)Nc4c(OC)nccc4)C3)C2)cc(I)c(C)c(I)c1 C1(NC(c2c(C)nn(CC(F)F)c2)=O)CCC(C)(CNC(c2csnn2)=O)CC1 C1(NC(C2CCCC2)=O)CN(C(c2c[nH]cc(Cl)c2=O)=O)CCC1CO C1(N(C(C(C)NC(=O)NC)=O)C)CCCN(C(=O)CC(C)NC(N)=O)C1 C12(COC)CC(CNC(=O)C(CCO)N(C)C)(CN1C(=O)CCC(=O)N(C)C)C2 N1(CC)CC(C)OC(C)C1.C1(=O)C(=O)NCCOCC2CC2C(=O)NCCCN1 c1(OC)c(CC(=O)NCC2CC(O)CN2C(=O)C(C)NC(C)(C)C)cccc1F c1(C(C(=O)NCCC2CC2)N(CCCCC=C)C)ncccc1Br Cc1c(C(N2CC=CC(NC(c3conc3C3CCC3)=O)C2)=O)cnn1CCO c1(C(=O)NC(C(C)NC(c2ccc(C#N)s2)=O)C)onc2c1CCCC2 c1(C(N2CC(O)(C(C)NC(=O)CC3(N4CCCC4)CC3)C2)=O)cnn2ccccc12 CN1CC2(CC2)CC1C(N1CCC(O)C1C(N1CCC1(C)CCO)=O)=O C1(O)(CN(C(=O)CSc2nc[nH]n2)C)CCN(C(=O)C(C)(C)C2CCCCO2)C1 c1(C(N2CC(C)C(CC(N3CC(N4CC(F)C4)C3)=O)C2)=O)cnc2ccccn12 C(=O)(CCS(=O)(=O)C(F)(F)F)NC(C1CN(C(=O)CC2CCC(=O)C2)C1)C O=C(C1CCc2ccccc21)NC1C2CC1N(C(c1cscc1C(F)(F)F)=O)C2 C(=O)(C(C(C)C)N(C)C)NC1CC(CCNC(c2ccn(CC(C)C)n2)=O)C1 c1(NC(C2CCN(c3cc(-n4cncn4)ncn3)C2)=O)ccc(F)c(C(=O)O)c1 C1(c2nc(C)c(C)c(C)n2)CCN(N2CC(N(CCC(F)(F)F)C)C(C)C2)CC1 C(=O)(C(C)(C)CC(F)F)NC1CN(C(C(C)OCCC=C)=O)CC(O)C1 C12(C(N(CC(CN(C(C(C)(C)OC)=O)C)O)C)=O)CC3CC(CC(C3)O1)C2 c1(C(=O)NC2C(N(C(C(C=C=C)C)=O)C)CCCC2)cc(C)cc([N+](=O)[O-])c1N c1(CNC(=O)Cc2c[nH]nc2C(=O)NC2CC2CO)ccc(OC)cc1OC CC(C)(C)C(C(=O)NC1(CNC(C2(CO)CC2)=O)CCCCC1)C(O)C(F)(F)F C1(CC)CCC(CNC(C2(NC(C3CC4(CC4)C3)=O)CC(O)C2)=O)O1 CC1COc2c(C(=O)NC3CC3CNC(c3snnc3C3CC3)=O)cnn2C1 C(=O)(C(C)S(N)(=O)=O)N1C(C(=O)NCC2CN3CCC2CC3)(COC)C=CC1 N1(C(c2ncn(CC)c2)=O)CCC(C)CC1C(=O)NCC1(CC)CCOC1 n1(CC(=O)OC2CCC2c2ccccc2)c(=O)ccc2ccccc12 c1(OC)ccc(CN2CCSCC2C(=O)Nc2ncccc2Br)c(Cl)c1 c1(OC)cc(CN=c2[nH]nc(C(F)F)o2)cc(C)c1 c1(CC(N2CC3CCC2CN3C(c2cccnc2)=O)=O)cc(F)ccc1[N+](=O)[O-] C=CCCC(F)(F)C(=O)NC1CC(F)(CNC(=O)Cc2cc(F)ccc2Cl)C1 CCC(C)(C)CC(=O)N1CC(CNC(c2ccc(C(C)C)nc2C)=O)C(C)(C)C1 C1(C(=O)NCCC2(CNC(=O)CC3OCCO3)CC2)COc2ccc(Cl)cc2C1 C(c1c(C)nn(CC(C)C)c1Cl)=CC(=O)NC(CNC(c1cc(C)no1)=O)CO Cc1cc(Cl)c(C(N2CCN(C(=O)CCC(F)(F)F)C(CO)C2)=O)cn1 c1(C(N2CC(CNC(C=C(C)Cl)=O)C(C)C2)=O)nc(C)ncc1Cl C1(CC(=O)NC(c2ccco2)CNC(CSC)=O)COC(=O)N1 c1(C(C(=O)OC)(C)C)ccc(F)c(C)c1.C12(CC(C)(C)C1)CN2 C1(C(N(CCCOCC(=O)NCC2(CO)CCC2)C)=O)C2CCC(C2)C1(C)C c1(C(N2CC(C)C(NC(=O)COCC3CCCC3)C2)=O)nc2ccccn2n1 C1(C(=O)NC2(C)CS(=O)(=O)C2)CCC(C(C)NC(C(C)OCCC=C)=O)CC1 C1(NC(c2cn(C)nc2C2CC2)=O)CN(C(c2ccccc2)=O)C(C)(C)C1 c1(C(N2CC(OC)C(C(=O)O)C2)=O)cc2sc(C)nc2[nH]1 C1(CNC(C(=O)Nc2cccc(-c3cn(C)nc3)c2)=O)CCC2(CC1)CC2 C(=O)(CCCCC(F)(F)F)N1C2(CC2)C1=O.C(=O)(CCCCC)O.C1(NC(C)=O)CCCCC1 CC1CN(C(C2C3CC4C(C3)C24)=O)CC1(C)CNC(c1cnc(C(C)(C)C)[nH]1)=O C12(C(N3CC(NC(C4CC(C)C4)=O)C(C)C3)=O)CCCC(C)(C1)OC2 c1(NC(=O)NC(C#C)(C)C2CC2)cc(CC(=O)OC)ccc1Br N1(C(C(CC(C)C)=O)=O)C2COCC1CC(NC(C1CC3CCC1C3)=O)C2 C=CC(C)(C)CCCNC(=O)C(C)(C1CC1)N(C(=O)CCCCSC)C C(C(COC)CC(=O)NCCOCCCNC(=O)CCC1CCCC(=O)N1)OC C(C(C(=O)NCCCCCN(C(=O)CCCc1nncn1C)C)OC)OC C1(C)(C(=O)NCC2(COC)CN(C(c3nnn(C)c3N)=O)C2)CCC(=O)N1 N1(C(C=CCN(CC)CC)=O)CCC(C)(NC(c2ccnc(OC)n2)=O)C1 C1(c2n(CCCF)nnn2)(NCc2ccc3nncn3c2)CCC2(CC1)COC2 Cc1cncc(CC(=O)NCC2(F)CCN(C(=O)C(c3cc(C)oc3C)C)C2)c1 Cc1cn2cc(C(=O)N(C(C)CN(C)C(c3cc(N)cc(F)c3)=O)C)ccc2n1 CCC(C)C(=O)C(=O)NCCn1ccc(C(=O)NCc2cnn(C)c2C)c1 N1(C(C(C)SC(F)(F)F)=O)CCn2nc(CNC(c3cccc(O)n3)=O)cc2C1 c1(C(N2C(C)CC(CNC(c3c(C)cccn3)=O)C2)=O)ccc(F)c(O)c1 c1(C(N2CC(CCCCNC(CSc3nc(C)[nH]n3)=O)C2)=O)cnn(C)c1Cl c1(CC)[nH]nc(C(=O)N(c2nccc(C)n2)C2C3CNCC23)c1F N1(CC(=O)NCC(=O)Nc2cc(Cl)cc(Cl)c2)CCN2CC(F)CC2C1 c1(NC(C)CCNC(=O)C(C)(O)c2ccccc2)cc(C2CCCCN2)ncn1 c1(C(N2CCC(CNC(C(C)(O)C3CCC3)=O)C2)=O)cc(N)nc(Br)c1 C(CCC(=O)NCC(C)NC(c1nnsc1-c1ccccc1)=O)OCCC C1(C(=O)NCCNC(C(C)c2ccco2)=O)CCCCS1 CC(C)C(CN(C)C)C(=O)N1CCC(CO)(CNC(=O)CC2CCSC2)CC1 c1(C(=O)NCc2cnn(C)c2Br)ccc2ccccc2n1 O(C1(OCC)c2cccnc2CCC1NC(=O)C=NOC)CC.C1CCN1 CC1CC(C(N2CCC(O)(C(N)=O)CC2)=O)CN(C(c2cnn(C)c2)=O)C1 C1(CNC(c2cnccc2Cl)=O)CN(C(c2nc(C3CC3)cs2)=O)CC12CC2 C1(NC(=O)CC23CCCC2C3)CCC(NC(c2cncc(F)c2)=O)CC1 Cc1ccc(S(=O)(=O)N2CC(C(F)(F)F)C(F)(c3ccccc3)C2)c(C)c1 c1(SCC(=O)N(C2CCC(NC(=O)CCCN3CCCCC3)C2)C)ccccc1 c1(NC(CCC=C)(C)c2nnnn2C2CC2)cnc2c(O)cccc2c1 CC(C)C(C(=O)OC(C)(C)C)NC(c1[nH]nnc1C1CCN(C(=O)C2CC2)C1)=O CC1(C)CCCN(C(=O)CC2CCCC3CC23)C1C(=O)NOCC1CCOCC1 C1(NC(c2c(OC)cnnc2)=O)CCN(C(=O)CCc2ccncc2)CC1O C1(C(=O)NCc2cccnc2O)CN(C(=O)CCN2CCCCC2)C2(CCC2)C1 C1(CCC(=O)NCC2C(NC(C(C)O)=O)CCC2)CCCCN1C C#CCC(CC#C)C(=O)N1CCN(C(c2cccc(O)n2)=O)C(CS(C)(=O)=O)C1 C(=O)(CCCNC(=O)NC1CCCCC1)NCC(C)(C)NC(C1CC1(Cl)Cl)=O CN1CCOC(C(=O)N(C)CC2COCCN2C(C2CCCC23CC3)=O)C1 N1(C(c2cn(C)nc2O)=O)CCCN(CCCCNC(C2CCCC2O)=O)CC1 C(=O)(C(C)(C)C(=O)NCc1cncc(C(=O)NOCC(C)C)c1)OCC Cc1ccc(N(C)C(C)C)c(C(N2CCCC(C)(CNC(c3cc[nH]n3)=O)C2)=O)c1 N1(C(CC(=O)NCC)=O)CCCC(C)(C)C1CNC(c1ccc(N)cc1OC)=O C1(C(=O)N(CCCn2ccnc2)C2CC2)CSCCN1C(=O)Cc1ccco1 c1(C(=O)NCC2N(C(CCC(=O)OC(C)(C)C)=O)CCCC2)ccc(F)cc1F c1(CC)cc(F)ccc1C(N1CC(CCNC(=O)CC(F)(F)Cl)OC(C)C1)=O c1(N(CC(C)NC(C2(c3cc(C)on3)CCC2)=O)C)ncnc2cc(Br)sc12 C12(NC(C(C)=C(C)C)=O)CCCC1CN(C(=O)Cc1csc(-c3ccoc3)n1)C2 C1(C)(NC(c2cnc(COC)s2)=O)CCN(C(c2cccc[n+]2[O-])=O)C1 C1(CNC(C(C)CN(C)C)=O)CCC2(CN(C(=O)Cc3cscn3)C2)O1 C1(NC(C(CC#C)C2CC2)=O)CN(C(=O)CCCCC2CCCCC2)CC1(C)C N1(C(CN(C)C)=O)CC2CCC2(CNC(C2(Cl)CC23CCC3)=O)C1 c1(C(N2CC(NC(C(CC)O)=O)C(C3CC3)C2)=O)cc2nc(Cl)ccc2o1 c12cc([nH]n1)CNC(=O)CONC2=O.c1(C(C)C)[nH]nnc1C1CC1 c1(C(N2CCCC(NC(CCC#C)=O)C2C)=O)ccc(C(F)(F)F)c(Cl)c1Cl N1(C(C(C)(F)F)=O)CCC2(CCC(CNC(c3ccnnc3S)=O)OC2)CC1 Cc1cc(C(=O)NCCCCN(C)C(C2(C)CCCNC2=O)=O)cc2c1CCC2 C1(NC(c2scc(C(C)=O)c2)=O)CC(NC(C2CCC(=O)NC2)=O)C(O)C1 CC(c1ccccc1Cl)=CC(N1CCC(CF)(NC(=O)C(O)C(F)(F)F)C1)=O C1(C(=O)NC2CC2)CCN(C(=O)CCOCC2CC2)C12CCC2 N1(C(C(CC)c2ccccc2)=O)CCN(C(C2CC(O)CN2C)=O)C(C(C)C)C1 c1(NC(C2CN(c3ccc(F)cc3)C(=O)C2)=O)nccc(Cl)c1I c1(NC(c2ccccc2-n2cccn2)=O)cc(Cl)ccc1CO c1(C(N2CCN(C(=O)CCc3cnc[nH]3)C(CC(F)F)C2)=O)csc2nnsc12 N1(C(CC(C)(C)F)=O)CCCC2(C1)CN(C(c1nccnc1C(N)=O)=O)C2 n1(CCCOCC)c(N2CCOC(c3ccccc3C)C2)nnc1-c1ccco1 N1(C(CC2CCC(C(C)C)CC2)=O)CC2(CCN(C(=O)CN(C)C)C2)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)NC1CC(OC)CN(C(C2(C#C)CCCC2)=O)C1 c1(C(=O)NC(C2CCN(C(=O)CCC3(C)CC3)CC2)C)ccnc(C(C)(C)O)c1 C(=O)(C(C(C)CCC(=O)OCCSC)N(CCC(=O)OC)C)NC c1(OCc2cccc(C)c2)cc(CC2(n3ccc([N+](=O)[O-])n3)CC2)c(Br)cn1 c1(CC(=O)NC2(C(=O)NC(C#CC)(C)C)CC2(C)C)c(C)noc1C C(=O)(C#CC1CCOCC1)N(C)CCN(c1ncc2c(n1)COC2)C O(N=C1CCCCCC1)CC(N1C(C)CC(CNC(c2ccsc2C#N)=O)C1)=O C(=O)(CCCC(F)(F)F)N(C1CC(NC(c2ccc(C(CC)(C)C)cc2)=O)C1)C C(=O)(C(CC)C(F)(F)F)N1CC(N(C(CCC#C)=O)C)C2(C1)CC2 C1(C(N2CCC(N(C)C(C3CC4CCC(C3)O4)=O)C2)=O)CCC2(CC1)CC2(F)F N1(C(C)C(=O)NCCNC(C2(C)CC2(C)C)=O)C(=O)CCC1=O c1(C(N2C(CC(=O)NC3(CSC)CC3)CC(C)(C)C2)=O)cc(C#N)ccc1N Cc1ncc(Br)cc1C(=O)NCC1(O)CCN(C(C2CN(C)CCO2)=O)C1 c1(OCC)cc(CN2CCOCC2(C)CC)cc2c1OCCO2 c1(C(C(F)(F)F)NCC(=O)NCc2ccccc2)cc(Cl)cc(Cl)c1 Cc1c(C(N2CCN(C(C3CCC(=O)NC3)=O)CC(O)C2)=O)cnc2ncnn12 C(=O)(CC1=CCN(C(=O)C(F)(F)C2CC2)CC1)NC1CC(C)OC1=O Cc1cc(C(=O)NC2CCCN(C(c3csc(=N)[nH]3)=O)C2C)cc(C)c1F C1(CC)CN(C(c2cnc(Cl)c(Cl)c2)=O)CCC1N=c1cc(C)nc(OC)[nH]1 c1(C(=O)NCC2N(C)CCN(C(c3cnc(S)nc3)=O)C2)cc([N+](=O)[O-])nn1C C(=O)(CCC1CCc2ccccc21)N1CC(NC(=O)CCCCCF)C2(C1)CC2 N1(C(c2cncnc2)=O)CC(C2CCN(C(c3ncncc3Br)=O)CC2)C1 Cc1ccc2ncn(CC(=O)NC3CCCC3NC(c3ccnc(S)c3)=O)c2c1 c1(C(=O)NC2CC(NC(CCCNC(C)=O)=O)C2)cc2sc(Br)cc2[nH]1 c1(C(=O)NCC2CC(NC(c3ccc(CC)cc3)=O)C2)cc2cc(C)ccc2s1 C1(c2nnnn2C2(C)CC2)(NC(c2nccs2)(C)C)COC2(CCOCC2)C1 C(=O)(CCC(C)S(C)(=O)=O)N(C1CCCN(C(C=C(C)C)=O)CC1)C CC(C(=O)N1CC(N(C)C(C2CC3(C2)CC3F)=O)C1)C1=CCCC1 Cc1cnc(Br)cc1NC(C1CC(F)CN1C(c1cc(Cl)ccc1Br)=O)=O c1(C(N(C)CC2N(C(C=CCCC)=O)CC(F)C2)=O)cc2c(s1)CCSC2 N(C(=NCCCC1CCOC1=O)NCC1CNC(=O)O1)CC(C)C C1(C)(NC(C2(NC(CC(C)OC)=O)CC2)=O)CCCC1(C)C C(c1nccs1)=CC(=O)NCC1(O)CC(CNC(=O)C(c2cccnc2)O)C1 Cc1cc(C(=O)NC(C)(C)CC(=O)NCC(C)C(C)(F)F)ccn1 C(=O)(CCCC(F)(F)F)NCC12CCC(NC(c3cnc(CC)s3)=O)(C1)CO2 CC(C)C(CCN(C(=O)CC(C)C1CC1)C)NC(c1cc(C(C)(F)F)on1)=O c1(C(C)C)cccc(C(=O)NCCNC(=O)NC(=O)CC(C)n2cccn2)n1 c1(CN(C)C(c2cnc3cc(F)ccn23)=O)cn2cc(Cl)ccc2n1 c1(C(c2nnnn2CCCSC)NC(C=C)C2CCC2)csc(CCC)n1 Cc1ccc(CCC(=O)NC(C)(C)C(=O)NCC2CCN(C(C)C)C2)o1 CN1CCN(C(C2C3CCCC23)=O)CC1CNC(c1ccnn1CC(F)F)=O CCCCCC(O)C(C)C(=O)NCC1CC(NC(C2(C3CC3)CC2)=O)C1 CCCCN=C(NCCOC1CCS(=O)(=O)CC1)NC1CCOCC1F N1(C(Cc2c(C)scc2)=O)CCN(C)CC1C(=O)N(C)Cc1ccns1 C(CCC(C)NC(=O)C=C1CC1)NC(C(C)NC(C1CCCC1)=O)=O CCCC(CCC)C(=O)N1CCN(C(C2CCCCC2)=O)CC(O)C1 c1(SC)ccc(C=CC(=O)NCCCC(C)NC(=O)CN(C)CCO)cc1 C=CCC(CC=C)C(=O)N1CC(NC(c2cc(C(=O)OC)ccn2)=O)CC1C C1(C2(C(=O)NC(C)(C)CCCN(C(=O)COCCCF)C)CC2)CCCCO1 C1(C)(COC)CCCN(C(=O)C(CC2CCC2)NC(c2cc(C(N)=O)co2)=O)C1 N1(C(c2cc(C)[nH]c2C)=O)CCCC(NC(c2coc(O)n2)=O)C1C N1(C(C2C(C=C)CC2)=O)CCC2(CCCN2C(=O)Cc2cccc(F)c2O)C1 N1(C(C=CCOC)=O)CC2CC(NC(=O)C(C)P(C)(C)=O)C1C2 C12(C(=O)NCC3CCC(CNC(C(C)(C)F)=O)CC3)CCC(CC1)CO2 c1(CC(=O)NC2CC(F)(C(=O)O)C2)nsnc1O N1(C(c2cc(C(=O)OC)oc2)=O)CC2C(CNC(C3(C(N)=O)CC3C)=O)C2C1 Cc1cc(N)c(C(N2CCC(NC(=O)CC3COCCOC3)C(O)C2)=O)cc1C C1(CNC(c2on(C)c(=O)c2)=O)CC2CCC1N(C(=O)COC1CCCOC1)C2 N1(C(C#C)=O)CCC2(CC2C(=O)NC2(C)CC2)C1 C(=O)(C(O)CCC(C)C)N(CCCNC(C1C(C)(C(=O)OCC)C1)=O)CCO CC1=CCC(C(=O)NC(C)C(=O)N(C)Cc2cc(C)nn2C)CC1 c1(C(=O)NC2CN(C(C3CC34CC(O)C4)=O)CCC2O)cccc2c1CCC2 c1(-c2cncc(SC)c2)ccc2c(C(=O)NCC3CCCCC3)noc2c1 N1(c2ncnc(OC)c2OC)CCn2ncc(CNC(=O)C=C(C)C)c2C1 C1(C(N2C3CC(c4cn(CC(=O)O)nn4)C2CC3)=O)Cc2ccncc2C1 C(C(C(F)(F)F)N1CCN(C(c2cn[nH]c2)=O)CC1)NC(C=CCOC)=O c1(OC)cccc(C(N2CC(CC(C(=O)C(F)(F)c3nccn3C)C)C2)=O)c1C CCC(CCCC(=O)NC(C)Cc1ncn(C)n1)NC(C1(O)CCCC1)=O N1(C(c2ccc(C)cc2Cl)C(=O)NCC(F)F)CCC(C2CCCC2)C1 N1(C(c2c(OCC)cccc2)=O)CCC(C)(C)C1CNC(=O)Cn1ccnc1C CCCCCCCCCCCn1nc(-c2nccs2)nc1C1CC1C C1(C(=O)Nc2n(CC)ncc2)CN(C(c2cc(Br)cc(F)c2C)=O)CC(F)(F)C1 CCCCCCCCCC(=O)N1CCCC(CNC(=O)C(F)CC(C)C)C1 O=C1CCCC(C(=O)NC2(C(=O)NCC3(F)CC3)CCCCC2)N1 C=CCC(CC(=O)N(C1CCNC1=O)CC)NC(=O)CCCc1ncco1 c1(SC)ccc(OC(C)C(=O)N(CCCCNC(=O)Cn2cc(Cl)cn2)C)cc1 CC(c1ccco1)=CC(=O)N(CCCNC(c1ccnc(C2CC2)n1)=O)CCO C1(O)(CNC(CCOCC)=O)CCCN(C(=O)CNC(c2cccc(C)c2)=O)C1 c1(C(=O)Nc2nc(C(N3CC4CCCC4C3)=O)cs2)ccc(O)c(Br)c1 CC1(NC(C2CCS(=O)(=O)C2)=O)CCN(C(C2CC(C(=O)O)C2(C)C)=O)CC1 C1(C(=O)NCC(CC)CC(C)C)CCCN1NC(=O)C(C)(C)COC c1(NC2CCN(C(CN(C(=O)OCC)C)=O)C2)ccnn1Cc1ccccn1 C1(C(N(C2CCCC2)CC(=O)O)=O)CCCC1c1nc[nH]n1 C(=O)(C1=CCCOC1)N1CC(CCC)C(C(N2CCC3CC23)=O)C1 N1(C(C(C(=O)OCC)OC)=O)CCC(C(=O)NCC(CC)CCO)C12CCC2 c12cc(no1)C(=O)NC1CC3(C1C3)NC(=O)N1CC2C1.C(C)(C)(C)O.CS CCCC(C)(C)CC(=O)NC12CCC(NC(C3CC(C4CC4)=NO3)=O)(CC1)C2 c1(NC(C)=O)ccc(NC(CC2(NC(=O)NCCCl)CCCCC2)=O)c(Cl)c1 C12(NC(C(C)C(F)(F)F)=O)CCCCC1CN(C(c1cnc3n1CCCC3)=O)C2 C1(C2CCC2)(C(N2CC(O)CC(NC(c3c(C)nncc3)=O)C2)=O)CC1(F)F CC#CCCC(=O)NCC=C1CCN(C(c2cccc(SC(F)(F)F)n2)=O)C1 CC(C)CC(CNC(=O)Cc1cscc1Br)C(=O)OCC(=O)OC(C)(C)C c1(OC(C)(C)C)ccc(OCC(O)CCOC(C2CC(CC(=O)OC)C2)=O)cc1 C1(C(N2CCC(CNC(CCc3nnc(CC)o3)=O)C2)=O)CC2(C1)CC(F)(F)C2 C1(C)(COC)CC(NC(c2coc(C)n2)=O)CN1C(=O)CSC(C)C C(=O)(C1CCCn2nccc21)OCc1nccc(C)n1 CC1(C)C(NC(C2CCCCN2N=O)=O)CCN1C(c1csnc1Cl)=O N1(C(c2ccc(OCCSC)cc2)C(=O)NC)CC2C(C(F)(F)F)(C1)CS2(=O)=O N1(C(COC(C)C)=O)CCN(C(C2CCCC(F)(F)C2)=O)CCC1C c1(C(=O)NC(C2CN(C(C(C)=CC)=O)C2)C)ccc(NC(C)=O)cc1Cl N#Cc1c[nH]c2cccc(C(=O)NCC3CCC3NC(=O)C(F)CC3CC3)c12 N1(CC)CCOC(C(=O)N(C(C)CN(C(=O)CCC(=O)c2ccccn2)C)C)C1 C(C(C)(O)CC(=O)N1CCN(C(c2cnc(F)c(C)c2)=O)CC1C)OC CC(C)(CO)C(CO)NC(=O)C(Cn1cncn1)NC(c1csc(Cl)c1)=O C(=O)(C(C)C(F)(F)C(F)F)NCC(CC)(CC)NC(c1cn2c(n1)COCC2)=O C1(CC(N2CC(CN(C(C(C=C)c3ccccc3)=O)C)C2)=O)CC2CCC1C2 C1(NC(c2ccno2)=O)CCOC12CCN(c1nnc(C(F)F)o1)CC2 c12cccnc1S2.N1(CC(=O)NCCCNC(CSC(=N)N)=O)CCSCC1 CCC(CC(=O)N(C)CCc1cccs1)NC(=O)CN1CC(OC)C1 c1(C(N(C)CC2N(C(CNC(=O)OC)=O)CC(F)C2)=O)cc(N)cc(F)c1 c1(C(=O)NCC2CCN(C(c3nccc(N)c3)=O)C23CC3)ccc2c(c1)COB2O Cc1nc(C)c(C(=O)NC2CCC(CNC(C3CSCCS3)=O)C2)nc1C N1(C(c2cncc(SC)c2)=O)CCC(C2(NC(c3ccn(C(F)F)n3)=O)CC2)C1 C(N=c1cc[nH]cc1S(=O)(=O)NC1CC2(CCCCC2)C1)C1CCCC(C)C1 C(C(CC(=O)NCC1CCC(C)C1)NC(C1CCCC(=O)C1)=O)OC Cn1ncc(C#N)c1C(N1CC2CC(NC(=O)C=CC3CCCCCC3)C2C1)=O N1(C(C(=O)NC(CC)(C)C)c2cnsc2)CCC(C2CCCOC2)CC1 n1(CC)nnc2cc(C(N3CCC(C)CC3CNC(C3CC3C#N)=O)=O)ccc12 N#Cc1cc(NNCc2ccc(Br)s2)ncn1 C(C)(CNC(=O)CC1C=CS(=O)(=O)C1)(C(C)C)NC(CCC#C)=O Cc1cc(C)c(C(=O)NCC2(CCNC(C3(C(F)(F)F)CCOCC3)=O)CC2)o1 C1(CCC(=O)NC2(C(=O)OC)CCOC2)CCCCN(C(=O)C(F)=C(C)C)C1 C1(NC(CC(COC)(C)O)=O)COC2(C1)CN(c1ccnc(C3CCCC3)n1)C2 N1(C(C(C(C)C(F)(F)F)F)=O)CCCC2(CCN(C(c3cccn3C)=O)CC2)C1 C=C(C)CC(C)C(=O)N1CC(NC(c2cc(NC(C)=O)ccc2N)=O)C2(CC2)C1 c1(C(C(=O)NCCOCCCN(C)C(c2cn(C)nc2O)=O)F)ccc(F)cc1 CC1CCCc2cc(C(N3CC(NC(=O)CP(C)(C)=O)C(CC4CC4)C3)=O)nn21 c1(OC)ccc(C(=O)NCC=CCNC(C2(C3CCC3)CC2)=O)c(OC(F)F)c1 Cc1cc(Cl)c(C(N2CCC(CC(C)NC(c3ncoc3C)=O)CC2)=O)cn1 N1(C(CC2CCN(C)CC2)=O)CCC2C(CCCN2C(C2CC2C(F)(F)F)=O)C1 c1(NC(N2CCCC(O)C2)=O)cc2ccccc2nc1Br C1(CC)C(C(=O)NCCN(C(=O)C(c2ccc(Cl)cc2)N(C)C)C)CCN1C c1(C(=O)NCC(C(C)C)NC(=O)Cn2nccn2)cncc2sccc12 c1(-n2cc(C(N(CCN(C)C(c3ns[nH]c3=O)=O)C)=O)nn2)ccccc1Cl CC1CCC(NC(=O)CC23CCC(C)(C2)OC3)CN1C(c1cc2scnc2[nH]1)=O c1(C(N2C(C)CC(NC(CCNC(=O)NC)=O)C2)=O)cnc2[nH]ccc2n1 C(=O)(CCC1=CCCCC1)N1CCCCC(N(C(=O)C(F)C2CCCC2)C)C1 C(CNC(c1c[nH]nc1Cl)=O)(C(=O)NC1CCC1)N(C)C C1(CNC(c2n(C)ccc2)=O)N(C(=O)CCc2cnccn2)CCC1(C)C c1(C(=O)NCCCN(C)C(c2cnn3c2NCCC3)=O)cnc2[nH]nnc2c1 C1(CNC(C(=O)NC)=O)C(C)CCCN1C(=O)CCSc1ccccc1Cl c1(OC)ccc2[nH]c(C(=O)NCCC(C)=O)cc2n1.C1CCSN1C(C)=O c1(C(=O)NC(CNC(CC2ON=C(CC)C2)=O)C)nccn2ccnc12 C1(NC(C2(SC)CCC2)=O)CCC(O)CN(C(C2(CO)CC(C)(C)C2)=O)C1 c1(C(=O)NC(CNC(c2ccc(CC3CC3)s2)=O)C2CC2)nccc2occc12 N1(C(C(CC)C(=O)OC)=O)CCC2CC(C1)CN(C(c1cc(C)sc1C)=O)C2 Cc1cc(C(=O)NC2CCC(NC(=O)C=Cc3cccs3)CC2)nc(O)c1 C1(CC(N2CC(NC(CN(C)C)=O)C(O)C2)=O)Cc2cc(C(F)(F)F)ccc2O1 N1(C(c2ccc(Cl)s2)=O)CCC2(CCCCN(C(C3(C(F)(F)F)CCO3)=O)C2)C1 CCCCCC(C)CC(=O)NC1CCOC(CNC(=O)C2=CCCS2)C1 N1(C(c2cnc(C(C)C)s2)=O)CC2CC1CCC2NC(=O)COc1cnn(C)c1 c1(OC)ccccc1COC(C)C(=O)N1CC(N(C(=O)C(=O)NC2CC2)C)C1 c1(C(N2C(CNC(c3cn(CCO)nn3)=O)CCCC2)=O)cncc2c1CCC2 c1(CC(=O)N(CCC(C)NC(=O)CC(=O)N(C)C)C)ccc([N+](=O)[O-])c(N)c1 N1(C(CCOCC#C)=O)CCN(CC2CCCN(C(c3cnn(C)n3)=O)C2)CC1 C1(NC(c2c(CC)noc2)=O)CC(F)CN(C(=O)CC2(O)CCCN(C)C2)C1 c1(C(N2C3(CN(C(c4cccc(I)c4Cl)=O)C3)CC2)=O)cc(F)c(Br)cc1F C(=O)(C1=C(F)CN(C(=O)CCOCC2CC2)CC1)N(C1CCC1C(C)(C)C)C CC1CC(C2CN(N3CCC4(CCNC4)CCC3)C2)=NO1.C1CC1 N1(C(C(C=C)O)=O)CC(NC(c2ccc(O)c(Cl)n2)=O)CC(C)C1 c1(NC(C2C(CNC(C3C(C)=CCS3)=O)CCCC2)=O)cnc(F)cc1C N1(C(C(=O)Nc2cccs2)c2cncs2)CCN(C(C2C3COCC23)=O)CC1 C(N=c1[nH]c(Cl)ncc1Br)C1CCCCN(C(c2cn(C3CCC3)nn2)=O)C1 c1(C(N2CCC(NC(C3(C=C)CCC3)=O)C(O)C2)=O)ccc(S(=O)(=O)N(C)C)o1 Cc1cccc2cc(C(=O)NCCC3CCCN(C(c4cscn4)=O)C3)nn12 CC(C)(C(=O)N1CCC(NC(c2csc(C3CC3)c2)=O)C1)C1CCCCO1 C1(NC(C(C2CCOCC2)NC(c2ccc(CC)s2)=O)=O)(CO)CC(F)(F)C1 c1(C(=O)NCC2CC(NC(C3CC34CC4)=O)C2)nc(N2CCOCC2)ncc1Cl C1(CNC(c2c(C)cc(CNC(C3(CSC)CC3)=O)o2)=O)CCC2(CC2)CO1 N1(C(C2CCN(C(=O)C3(CCN=[N+]=[N-])CC3)O2)=O)CC2CCC1C(O)C2 N1(C(C(C=CCCC)O)=O)CCC(C)(C)C(NC(=O)C(C)NC(C)=O)C1 C1(F)(CNC(CN(C)C)=O)CCCN(C(C2CC2(F)F)=O)C1 C1(N(C(=O)C(C)(C)C)C(C(=O)N(C(C)C)C(C)C)=O)CCC2CCCC1O2 N1(C(CCCC#CC)=O)CCC2CCN(C(c3ccc4oc(O)nc4n3)=O)CC12 c1(C(N2CC(C)(C)C(NC(C3CC3C(F)F)=O)CC2)=O)nnc2ccccc2n1 c1(CNC(C2CCN(C(c3cnn[nH]3)=O)CC2)C)cnc(C(F)F)nc1 C1(CC=C)(C(=O)NC(C)C(C)n2cccn2)CCN(C(c2ccccn2)=O)C1 Cn1ccnc1CCC(=O)NCCC1(NC(c2cc(F)cs2)=O)CCCC1 C(CC(F)F)(C(=O)N1CC(CO)CC1CO)NC(C(C)n1cnnn1)=O C(CC(=O)N1CCC(C(N(CC(=O)NC)C)=O)O1)SCC N1(C(CN(CCC)C)=O)CC2C(CC(=O)NCCNC(=O)NC)C2C1 C1(C(C)C)OCCC1C(=O)NCCCCNC(c1cc(C2CC2)no1)=O C1(CNC(C(C)c2ccco2)=O)CC(=O)N(C2CN(CCC3CC(F)(F)C3)C2)C1 c1(C(N(CC(CN(C(C(C)CO)=O)C)O)C)=O)ccc(F)cc1[N+](=O)[O-] CCCC(CC)CCC(=O)NC1CN(C(c2cc(N)cnc2Cl)=O)C1 c1(N2CCCC3(NC(c4cnc(C)o4)=O)C(C2)C3)c(C#N)cccc1[N+](=O)[O-] C(=O)(C(F)C(C)(C)O)NCc1ccc(C(N(CCC(C)O)C2CC2)=O)o1 C(=O)(C1=NOC(C)(C)C1)N1CCC(C#C)(C(=O)N(CCC(C)C)CCO)C1 CC(C)C(C(=O)NCC1CCCCCN1C(=O)COCc1ncnn1C)C(C)C C1(C(=O)NC2(C(=O)NC3C(C)COCC3)CCCCC2)CCCC(C#N)C1 C1(C(N(C)CC2CCCN(C(c3ccc(COC)o3)=O)C2)=O)CC12CCCCC2 N1(CC)CCCC1C(=O)NC(CNC(c1cc(C)c[nH]1)=O)CCOC CON(CCC(=O)NCC1(C)CCC(C)(C)CC1)C(=O)CN1CCCC(C)C1 c1(CC)nc(C)c(C(=O)NCC2CCCN2C(=O)C(C)(O)CC)s1 c1(OC)nc(=NCCCN(C(=O)C2=NN(C)C(=O)CC2)C)nc(OC)[nH]1 c1(C(=O)NC2C(CC)N(C(c3nc(C)sc3C)=O)CC2)nccn2nccc12 C1(CC(=O)NC2CC(Nc3cc(O)nc(O)n3)C2)Cc2ccccc2O1 C(=O)(CC1CCCc2ccccc21)NC(CNC(Cn1nnc(C)n1)=O)C CC1=C(C(=O)N2CCC(O)(c3ccc(-c4cnn(C5CC5)c4)cc3)CC2)CCC1 C1(NC(c2c(CC)ncnc2)=O)CCN(C(C2SC3C=CC2CC3)=O)CC1O C(=O)(C(C(C)C)C(C)C)NC1CN(C(c2cnc(OC)c(C)n2)=O)C(CO)C1 Cc1cc(NC(C2CC(O)CN2C(c2cccc(F)c2Cl)=O)=O)ccc1Br C1(C(N2CC(C(N)=O)(CNC(C(C)OCCC=C)=O)C2)=O)COCCOC1 C12(C(=O)NCC(CC)O)CC(CO1)N(C(C1CCCCO1)=O)C2 C1(CNC(CCCCSC)=O)CC(NC(c2nccn2C)=O)C12CCC2 N1(C(CC(=O)N(C)C)=O)CC(O)CCC1C(=O)NCCC1(C)CCOC1 C1(NC(CN(CC)CC)=O)CC(C(=O)N(CC(=O)NCC(C)C)C)C12CCC2 c1(C(=O)NC23CC(CNC(C(CSC)O)=O)(C2)OC3C)cccn2cc(C)nc12 c1(-c2nc(CSC)nn2-c2nc(C)nn2C)cccc2c1ncn2C c1(C(=O)NC2C(C)(C)C(C(=O)NCC3(CO)CC=CC3)C2)ccc2c(c1)CCC2 C(C(C)(CC(C)C)NC(C1CC=CCC1C)=O)NC(c1occ(C(=O)OC)c1)=O c1(CC(N2CC(C)C(NC(=O)C(F)(F)C3CC3)CC2)=O)cccc2ccsc12 C1(NC(Cn2nnc(C)n2)=O)CCN(C(=O)CCOC(C)C)C12CCC2 c1(CC(=O)N(CCCN(C(C(C(C)C)OCC)=O)C)C)ccc(Cl)cc1C S(=O)(=O)(c1ccc(C(=O)OCc2ccc3c(c2)OCO3)cc1)N1CCC(C)(C)C1 c1(CC)nc2cc(S(=O)(=O)N3C(C)CC(c4ccccc4)C3(C)C)ccc2o1 O=C1CC(NC(C2CC3CC2CC3NC(=O)CC2CSCCO2)=O)CC(=O)N1 c1(NC(C(n2ncc(C)c2)C)=O)cccc(CNC(C2CC3CCC2O3)=O)c1 C1(C(=O)NCC2(OC)CN(C(c3csc(=N)[nH]3)=O)C2)CC2C=CC1CC2 Cc1cccc2[nH]cc(C(=O)NCCNC(=O)CCCCc3cccc(O)c3)c12 C1(C(=O)NCC2N(C(c3ccsc3)=O)CC(C)(C)OC2)CC2CCC(C1)C2(F)F N1(C(C(CC)Cl)=O)CC2(CCC(N3CCC4(CNC(=O)O4)C3)CC2)C1 c1(C(=O)NCC(C)NC(C2CCCC(=O)CC2)=O)ccc(F)c(Cl)c1F CC1(C)CCOC1CC(N1CCC(NC(c2cccnn2)=O)C1)=O c1(C(N2CC3C(CNC(c4c(C(C)C)ccs4)=O)(C3)C2)=O)ccc(Cl)c(O)c1N c1(CC)[nH]nc(C(=O)N(C)CCN(C(c2ccnc(C)n2)=O)C(C)C)c1[N+](=O)[O-] C(C)(CO)(C(=O)NC(CC1CCC1)CO)NC(CC(C)N(C)C)=O C#Cc1cccc(C(=O)OCC(=O)NC2CCc3nccn3C2)c1C#N C1(C(N(CCCCN(C(C(C)CC2CCC2)=O)C)C)=O)CC(C2CC2)C1 C(=O)(N1CC(O)CO1)C1CN(C(C2CCN(C)CC2)=O)CC1F c1(C(N2CCC(O)(C(=O)NC(CC)COC)CC2)=O)c[nH]c2ccc(F)cc12 C1(CNC(CSCC(N)=O)=O)CN(C(c2ncncc2Cl)=O)C2(CCOCC2)C1 N1(C(c2cc(CC)ncc2)=O)CCC(C(=O)N(OC)C(C)CC)C(C)(C)C1 C1(CNC(c2cc(CC)nc(O)c2)=O)CC12CCN(C(=O)C1=CCOCC1)CC2 c1(CNC(C2(C)CCCS2)=O)nnn2c1CCCC2 N1(C(CC2CCCN(C(C(C)n3cccc3)=O)C2)=O)CCc2ccsc2C1 c1(C(=O)NCc2ccc(-n3c(C)ncc3)cc2)cc2n(n1)CCCN(C)C2=O C(=O)(C(CNC(C12C(=O)C3CC1C2C3)=O)C(C)(C)C)N1CCC(N(C)C)C(O)C1 Cc1cc(=NCCc2cnn(C)c2)[nH]c(=NCc2nc(Br)ccc2C)[nH]1 CN1CCC(C(N2CC(O)CC2CC(=O)NC2(C)C(C)(C)C2(C)C)=O)CC1=O N1(C(C2CCCOC2)C(=O)NCCCF)CCCC(CO)CC1 C1(C(=O)NCCCN(C(CC(C)C)C)CCO)CC(=O)N(C(C)(C)C)C1 Cc1[nH]c(-c2ccccc2)cc1C(=O)NCC1CC(NC(=O)CCF)C1 C=Cc1cncc(C(=O)NC(C)CCCCNC(=O)C(C)(C)C)c1 Cc1cc(Cl)ccc1C(=O)NC1CCC(CNC(c2cc(O)ccc2F)=O)C1 CC1CC(=O)NC1C(=O)Nc1cnn(CC(F)(F)F)c1C1CC1 c1(Oc2ccc(OCC)cc2)cc(C)ccc1C(N1CCOCC1)=O c1(OCC)ccc(-c2nc(CCOC(C)C)n(C(C)C(F)(F)F)n2)cc1 C=C1CC(C(=O)NC(C(O)CO)C2CC2)(CNC(c2scnc2C)=O)C1 c1(NC(c2cccc(CC)c2)=O)ncc(F)cc1C#N C1(CNC(c2nnnn2CCOCC)CCC)CC(C)(C)CC(C)(C)C1 C12(C(N3CC(NC(c4ccn(C)c4)=O)C4(C3)CC4)=O)C3C4C1C1C2C3C41C N1(C(C2(CSC)CC2)=O)CC(CO)C2(C1)CN(C(c1cnc3[nH]ncc3c1)=O)C2 c1(COC)ccoc1C(N1CCC(N(C(C2CC(n3ccnc3)C2)=O)CC)C1)=O NC1CCCC2(CC(C(N3CCN(c4nc(O)cs4)CC3)=O)C2)C1 c1(CN2CC(CNC(c3c(C)ocn3)=O)OCC2)ccc2nc[nH]c2c1 C=CCCC(C)(C)C(=O)NCC12CC1CN(C(=O)Cc1cc(C)[nH]n1)C2 C1(CCC(=O)NC2(CCOC)CC2)CCCN(C(=O)CCn2ccnc2)C1 C1(CNC(COCC(C)C)=O)CCN(C(c2ccc(F)cc2)=O)CC1(F)F Cc1cc(=NCCCCC(C)NC(=O)C2=CCCCCC2)c([N+](=O)[O-])c(C)[nH]1 N1(CC#C)CCCC1C(N1CC(COC)(NC(c2ccno2)=O)C1)=O C(=O)(CCCCCC#N)NC1C=CC(CC(=O)N(CC#C)CC2CCCO2)C1 c1(C(=O)NC(CCCNC(C=C(CCC)C)=O)C)cc(C(N)=O)ccc1OC c1(CCC=CC(=O)NCCCC2(NC(=O)CNC(N)=O)CC2)ccccc1 CC#CC1CCN(C(C23CC(CO)(CN2C(C2CCCC(O)C2)=O)C3)=O)C1 CCCCC(CC)(c1nc(CS(C)(=O)=O)no1)c1nnnn1CCOC(C)(C)C C1(C(=O)NCCC2CCCN2C(=O)Cc2c(F)cncc2Cl)C2CC(F)(F)CC12 c1(OC)cccc(F)c1C(=O)NC1CCC1NC(=O)C(C)OCC(F)(F)F N1(C(Cn2cccc(N)c2=O)=O)CCC2CCN(C(C3CCC3)=O)C2C1 C1(N(S(=O)(=O)C2CCN(C(=O)OC(C)(C)C)C2)C(C)C)CCCCN(C)C1=O C12(NC(c3scc(C(C)=O)c3)=O)CC1CN(C(=O)C(C(C)C)NC(N)=O)C2 C12(C(=O)NC(CCC)c3ccco3)CC(CO)(CN1C(c1cc(OC)n[nH]1)=O)C2 Nc1nccnc1C(=O)NCC1(C(=O)NCCCc2ccccn2)CC1 CC1C(=O)Nc2ccccc2N1C(=O)C=Cc1ccc2c(c1)OCO2 c1(N2CCOCC(NC(C3N(C)C(=O)NC3)=O)C2)nc2c(cc1C#N)CCCC2 c1(CC(=O)N(C)CC2CCN(C(C3C(C=C)CC3)=O)C2)c(C)cccc1Cl N1(C(C(CC)C(C)C)=O)C2CCC1CC(N(C(=O)C1=CCCS1)C)C2 C(=O)(C(F)CCC(C)(C)C)NCC(C)N(C(c1cc(SC)oc1)=O)C N1(C(CC2(OC)CCOCC2)=O)CCN(C(C2CN(C)CCO2)=O)C(CCO)C1 CC1(C)C(CC(=O)NC2(CC(=O)Nc3cncc(CO)c3)CCCC2)CC1O c1(C(=O)NCC(C)N(C(CC(=O)NCC#C)=O)CC)nc(C)n(C)n1 c1(C(=O)NCC(CNC(c2cn3c(n2)CCC3)=O)F)ccc(F)cc1F C#CCC(C)(CC)C(=O)N1CCC(C)(NC(=O)C=C2CCC(C)C2)CC1 CCCC(C)CC(=O)NCC(C)(C)CN(C(C1(C(C)(F)F)CCOCC1)=O)CC C(CCC1CCC1)(C(=O)NCc1cnccc1C)NC(CN1CCC(OC)C1)=O c1(C(N(C2CCCN(C(CC(C(C)C)O)=O)C2)CCO)=O)nnn2c1CSCC2 C(C(C)(CNC(C1(CCNC(=O)CN2CCNC(=O)C2)CCC1)=O)CO)OC c1(NC(CCC2N(C(c3nn(CC)c(C)c3)=O)CCC2)=O)cc(C)cc(C)c1O N1(C(C2(N(C)C)CC2)=O)CC2C(CNC(=O)CC3C=CS(=O)(=O)C3)C2C1 C1(O)(NCc2cc(C)sc2)CCN(CCNC(=O)OC(C)(C)C)C1 c1(COC)cccc(C(=O)NC(C)C(N2CCCC2C2(OC)CC2)=O)c1 N1(c2nnc(CCC)s2)CCCC(C(=O)N(CCCCn2ccnc2)CC)CC1 Clc1ccc(CNC2(c3nnnn3CC3CCCCCC3)CCOC2)nc1 C1(COC)(CNC(=O)C(C(C)C)NC=O)CCN(C(C2CC3(CSC3)C2)=O)CC1 c1(C(N(C)CCNC(C2(C)CCOC2)=O)=O)cc2cc(Cl)c(Cl)cc2[nH]1 c1(N(C(CNC2CC(OCC)C2(CC)CC)=O)C)cnc(C#N)c(Cl)c1 C1(NC(=O)Cn2ccnn2)CC12CCC(NC(C1COCCO1)=O)CC2 CCC(C)(CC)C(=O)N1CC2CC2(NC(c2cnn(C)c2OC)=O)C1 c1(OC)c(C(=O)NC2CCCCN(C(=O)C(O)CSC)C2)cc(Cl)cc1Cl c1(NC(=O)Nc2nccn2C(F)(F)F)nc(C2CCCOC2)cs1 N1(C(c2ccc(OC)o2)=O)CCC(C(O)CNC(=O)CN2CCCC2C)CC1 c1(C(=O)NC(CC=C)CNC(=O)CC2CCC(=O)NC2)cc(C)nc(C)n1 CCCCCCC(C)C(=O)NC(Cn1cncn1)C(=O)NCc1c[nH]ccc1=O N1(C(C(=O)NCCCSC)C2CC2(C)Br)CCc2cnccc2C1 c1(C(C(=O)NC(C)C(F)F)NC(CC=C)=O)cnn(C)c1O c1(OC)ccc2c(=NCC3CCC(F)C3)[nH]c(=NCCc3ccccn3)[nH]c2c1 CCCC(C(=O)NCC1CCN(C(=O)C(c2cnn(C)c2)OC)CC1)N(C)C N1(C(c2cn(CCC)nn2)=O)C(C(=O)NCC2CCC(=O)O2)C2CC(O)C1C2 c1(C(N2C(CNC(CCC(C)SC)=O)CCC2)=O)ccnc2[nH]nnc12 c1(CC)ccccc1C(=O)NCCOCCN(C)C(C1(CCO)CC1)=O C(=O)(C(C)CS(C)(=O)=O)NCC1CCCCN(C(c2ccn(CCC)n2)=O)C1 C1(C(N2CCC(C)(CNC(=O)Cc3nccs3)C2)=O)CC1C1CCCCC1 N1CCCC(O)C1C.C#Cc1ccc(CN)s1 c1(N2CC(CN(C(c3ccc(CC)[nH]3)=O)C)OCC2)ncc2ccsc2n1 C=CCCC(C)(C)C(=O)NCCC1CCCN(C(c2cccc3c[nH]nc23)=O)C1 C(=O)(C1CCc2c[nH]nc21)N1CCC(C=C)(NC(=O)CNC(=O)C(F)(F)F)C1 CC1CCOC(C(=O)Nc2cccc(NC(=O)Cc3nc[nH]n3)c2)C1 c1(CC)nn[nH]c1C(=O)N(CCC(=O)NCC1CSC1)CCCO c1(C(=O)NCCCOC(=N)O)ccc2c(n1)CN(C(=O)CCOC1CC1)CC2 C(CO)(C(=O)NCCC1CC(F)(F)C1)NC(=O)C=CC(F)(F)F c1(CC)ccc(C(C(=O)NC2CCCC2)N(C)CCOc2ccccc2C)cc1 C1(CC)CN(C)C(=O)CN1C(=O)C(CC(F)F)N(C(=O)Cn1nccc1C)C C1(NC(C(C)CC2CC2)=O)CC=C(C(=O)N2CCCCCCC2)C1 C1(CC(=O)NCC(C=C)O)CCN(C(C2OCCC2(C)C)=O)C1(C)C CCC(C#N)(CC)C(=O)NCC1CC1CNC(=O)CCN1CCNC(=O)C1 Cc1cc(C(=O)NC2CC(CNC(=O)CN3CCC(F)CC3)C2)nc(C)c1 c1(OCC)cccc(CC(=O)N(C)CC2CN(C(c3ncsc3Br)=O)C2)c1 c1(C(N2CCC(CCNC(CC3(C=C)CC3)=O)C2)=O)c(C)oc(C)c1Br C1(CC(=O)OCC)CCCN1C(=O)CC1CCN(C(=O)Cc2cncnc2)C1 N=c1ccc(C(N2CCCCC2C2CCCC2NC(=O)C(F)=CC2CC2)=O)n[nH]1 C1(SC)CN(C(=O)C2=CCCS2)CC1NC(=O)C(C)c1ccco1 c1(C(=O)Oc2ccc(-c3ccc(OC)cc3)cc2)cccc2c1NC(=O)CC2 C1(NC(C(C)CN(C)C)=O)CN(C(=O)CO)CCC1c1ccccc1 C1(N(C(=O)COCC(N)=O)CC)CCN(C(c2ccnn2C(C)CC)=O)C1 CC1=C(C(=O)N2CC(N(C(=O)C(n3cc(C)cn3)C)C)C3(CC3)C2)CCCC1 C1(COC)(NC(=O)C(C)Sc2ccncc2)CCC(F)(F)CC1 C1(C(=O)NC2CCC(C)(CNC(CCCOC)=O)CC2)CS(=O)(=O)CC12CCC2 C1(C(=O)NCC(C)OCC#C)CCN(C(C2COCCN2C)=O)CC1C N1(C(C(C=C)OC)=O)CCCC2C1CCCN2C(=O)C(=O)NOC N1(c2nnc(-c3c(C)n(C)nc3)n2CC2CC2)CCOC2CCCCC12 CCC(CN(C(=O)C(O)C1CCCC1)CC)NC(=O)CCSCC(C)C C1(CC)CCCN(C(C2CC23CC(NC(C2(COC(C)C)CC2)=O)C3)=O)CC1 C#Cc1ccccc1CC(N1CCCC(F)(CNC(=O)C(CC)OCC)C1)=O CCCC(CCCNC(C1CC2C=CC1CC2)=O)NC(c1nnn(C)c1C)=O C=CC(C)(C)C(=O)NCCCCN(C(=O)C(CNC(=O)OC(C)(C)C)CO)C CC1OC2CCC1(C(=O)NCC1CCN(C(c3cncc(Cl)c3)=O)C1)C2 N1(C(C(CC=C)C)=O)CCN(C(C2CC(F)(CO)C2)=O)C(c2cn[nH]c2)C1 c1(C(=O)NC(COCC)C(=O)NCCS(=O)(=O)NC)coc2ccccc12 CCC(C(=O)NC1(c2ccccc2)CN(C(=O)CCCCCO)C1)C(C)C CC1(C)CN(C(C2CCC(C(N)=O)O2)=O)CC1NC(=O)CC12COC(CF)(C1)C2 c1(C(=O)NC2CCCC(NC(CC3ON=C(C)C3)=O)C2)cc2ccsc2s1 N1(C(C(C)OC(C)=O)=O)CCCC(C)(C)C1C(=O)N(C)Cc1ccon1 C1(CCNCC(C)Oc2ccc(Cl)c(Cl)c2)CC2(CCC(F)(F)CC2)C1 N1(C(COC(C)=O)=O)CCC2(CC1)CCN2C(c1ncccc1Br)=O CC1(C)CCC(CNC(=O)Cn2cccn2)N(C(=O)Cn2cc(F)ccc2=O)C1 N1(C(CCCOCCC)=O)CCOCC1CCNC(c1ccnn1CCOC)=O Cc1nc(C)c(C(=O)NC(C(N2CC(C)(CF)C2)=O)c2ccoc2)s1 c1(Nc2cccc(C(=O)NCC(CC)C)c2)cc(C)nc(C2CC2)n1 C1(NC(c2cc(C)ns2)=O)COC2(CNC(=O)C(C)CN(C)C)CC1C2 C1(C(=O)NC(CC)CNC(=O)CCc2cnn(C)c2)CCCC(=O)O1 N1(Cc2ccc(N(C)C)nc2)CCC(F)(F)C(NC(c2cc(Cl)c(Cl)s2)=O)C1 C1(NC(c2ccc(C#C)cc2OC)=O)CCN(C(=O)CCOC)CCC1(F)F C=CC(C)(CC)C(=O)NCCC1CCN(C(c2cnc(C(C)=O)s2)=O)C1 c1(C(=O)NC(C2CCCN2C(=O)Cn2ccc(C3CC3)n2)C)cc(C2CC2)cs1 N1(C(C2(NC(=O)OC(C)(C)C)C(C)C2)=O)CCN(C(=O)C=CCBr)CC1 CCCC(C(=O)NCC1(C)CCN(C(=O)Cc2cncs2)C1)c1cccc(Cl)c1 C(=O)(C1=NOC2COCC12)NC1C(NC(c2c(C)nccn2)=O)CCC1 C1(NC(c2cnc(CCCC)s2)=O)CCCC12CN(C(=O)C(C)(C)N(C)C)C2 c1(C(=O)OCC)ccc(C(=O)NCCCC(C)NC(C2CCOCC2)=O)cc1 N#Cc1ccc(C(C(F)(F)F)NC(N2CC3CC2(C(F)F)C3)=O)cc1 C1(C(=O)NCC2C(C)OCC2)CC12CCN(C(c1cccn1C)=O)C2 N1(C(COCC)=O)CCC(N(C)C(C2CCCN(Cc3ccccc3)C2)=O)CC1 C1(CC(=O)NC2(CO)CN(C(C3CC3C3CC3)=O)C2)CCCCCCC1 C(C(F)(F)C(=O)NCC(CCOC)NC(c1cnc(O)n1C)=O)OC C(=O)(C(O)P(C)(C)=O)NC(C(C)C)CNC(C1CC2(CSC2)C1)=O Cc1cc2sc(C(N3CCCC3CCNC(c3cncs3)=O)=O)cc2s1 c1(COC(C)C)nccc(=NCCCC2CCCC2NC(C)(C)C)[nH]1 c1(CC(C(=O)OC)NC(=O)CC2CCCC2(C)C)ccc(Br)nc1 c1(C(N2CC(C(=O)NCCSCC)SCC2)=O)cccn(C2CC2)c1=O N1(C(C2(C)N(C(C=Cc3ncn(C)c3)=O)CC(O)C2)=O)CC2CC=CCC2C1 CC(C)(O)C(F)C(=O)N1CCC(C(C)(C)NC(=O)CCC2OCCO2)C1 c1(C(=O)NC2CCN(C(c3c(C)oc(C#N)c3)=O)C2)cc(S(C)(=O)=O)ccc1Cl c1(C(N2CCC(CNC(CCC(=C)Cl)=O)C2)=O)ccn2cc(C)nc2c1 N1(C(C(C)(C2CC2)SC)=O)CCN(C(CNC(=O)C=CC(C)C)C(F)(F)F)CC1 C(=O)(C(C)(C)CC(F)(F)F)NCC1CN(C(c2c(C)ccnn2)=O)C(C)C1 C(c1cnc(O)nc1O)=CC(N1CCC(N(C(=O)C(O)C(F)(F)F)C)C1)=O c1(C(=O)NCC(C(=O)NCCN(CCC)CC)O)cc(=O)cc[nH]1 C(CC(C)(C)C)(C(=O)NCC1(C)CCCN(C(C2(n3nccn3)CC2)=O)C1)OC Cc1ccc(OCCCN)cc1.N12CCC(C1)N(C)C(=O)C2.c1cc(C)sn1 C(=O)(C(C(C)C)c1ccc(F)cc1)N1CCC(N(C(C(C2CC2)OC)=O)CC)C1 C(=O)(CS(=O)CCC(F)(F)F)NC(C1CCCC1)CNC(CCC=C)=O C1(CNC(C2(CC=C)CC2)=O)(CO)CCN(C(C2CC2OC(C)(C)C)=O)CC1 C12(NC(C(C)Cc3ccccn3)=O)CCOCC1CN(C(C1OCCCO1)=O)C2 C1(OC)CCN(C(=NCC(C)SC)NC(C2CC2)C2CC2)CC1(C)C Cc1cc(Br)cc(C(=O)NC2CN(C(=O)C=Cc3cncs3)C2)c1F C1(O)(CNC(c2ccc(CC)o2)=O)CCN(C(c2nc(C)oc2C)=O)C1 c1(C(=O)NCC(C)(CC(C)C)NC(CS(CC)=O)=O)c(C)ccc(C)c1N C(CCN(C)C(C1CCCC1OC)=O)(C(C)C)NC(c1cc(CC)no1)=O N1(C(Cc2cc(C)no2)=O)CCC2(CCN(C(c3c[nH]c(C(C)(C)C)c3)=O)C2)C1 C(=O)(C(CNC(C)(C)CNC(C)=O)c1ccccc1)OCC C(C(=O)N1CCC(C(C)NC(c2ccc(=N)[nH]c2)=O)CC1)(C(C)C)SCC c1(CC(=O)NC2CCCC2CNC(C2CCCC3CC23)=O)ccc(O)c(F)c1 c1(C(N2CCC(NC(C=CCN(C)CC)=O)C2)=O)cc(Br)n2c1CCC2 c1(NC(c2ccc(-c3ccc(NC(C)=O)cc3)nn2)=O)ccc(F)nc1F c1(OC)nc(C)ccc1CN1CCCC(NC(=O)CCC(=O)SC)CC1 c1(CC(=O)NC(CNC(C(CC)n2cncn2)=O)COC)ccc(C)cn1 Cc1c(C(N2CC3(CC(NC(C4CC4Cl)=O)C3)C2)=O)oc2cc(Cl)ccc12 C1(NC(C=CC(CC)=CC)=O)CC2CCC(C1)N2C(C1CC1(C)C)=O c1(OCC)ccc(OCC(=O)N(C(C)CNC(=O)C(F)n2ccnc2)C)cc1 c1(CCN(C2CCCC2)CC(C)O)cccc(Cl)c1 O=C(CCCCC(F)F)NC1(CO)CCN(C(=O)Cc2ccc(F)cn2)CC1 c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)CC2F)cc(C)c(Cl)c(C)c1 c1(OC)ccc(Cl)c(Cc2noc(-c3ccsc3OC)n2)c1 N1(C(Cc2cnc(C)s2)=O)CCC(C2CC(NC(c3nc(Cl)cs3)=O)C2)C1 N1(C(c2cc(C)[nH]n2)=O)CCCC1C1CCCN1C(=O)CN1CCN(CC)CC1 c1(CCC(=O)NCC2CN(C(Cc3cnc(C)o3)=O)C(C)C2)cccc(C#N)c1 N1(C(C2C(C(C)O)C2)=O)CCC2CCC(C1)N2C(C1(CO)CC1(F)F)=O c1(CC)cccc(C(=O)NC2CCC2NC(=O)CCCN(C)C(C)=O)c1 C(CN=c1[nH]c2c(c(=NC(C)c3c(Cl)cccc3Cl)[nH]1)COC2)OC1(C)CCC1 C1(NC(C(COC)NC(C)=O)=O)CCC(NC(c2nnsc2C)=O)CC1 Cc1cc(C(F)F)ncc1C(=O)NC1CN(C(c2cnco2)=O)CCC1CO CC(CC(N)=O)C(=O)N1CCC(CO)(NC(=O)C(=O)NCC2CC2)C1 C(CC(F)(F)C(=O)NCCC1CCC2(CCC2)O1)n1cc(CNC(C)=O)nn1 c1(C(=O)NC2CCN(C(c3ccco3)=O)CC2)cc2ccc(Cl)nc2s1 c1(C(c2nnnn2C2CC2)NC(c2nc[nH]n2)C)nn(C)c2c1CCCC2 c1(C(=O)NCCN(C(=O)C(CO)C(C)(C)C)CC)cc2scc(Cl)c2[nH]1 C(=O)(C(C)C(C)(C)C)NCCC(C)(C)NC(C(c1cccnc1)C)=O n1(CC(=O)NC(C)C(C)NC(=O)Cc2cncn2C)nc(C(F)F)cc1C1CC1 c1(C(=O)NC2CC(NC(C(C3CCOCC3)C)=O)C2)cc(N)c2ccccc2n1 c1(C(=O)NC2CN(C(Cc3ccc(OC)cc3)=O)CC2C)ccc(Br)cc1F C1(O)(C(C(=O)N(C(C)C(F)F)C)NC(=O)C(C)O)CCCCC1 Cc1cc(Br)ccc1S(=O)(=O)N1CC2C(C1)N2C(=O)CCc1c(C)nn(C)c1C c1(C(N2CC(NC(C(CC=CC)C)=O)(CO)C2)=O)ccn(C(C)C)c(=O)c1 c1(-c2cn(C)nc2)ccc(C(=O)OC2CC3CCC2C3)cc1 c1(C(C)Nc2ncnc(NCc3c(C)nco3)c2C)ccc2c(c1)CCCO2 O=C(C1=CC2CCCC12)NC1CCCCC1NC(c1ccc(CO)nc1)=O C1(NC(=O)CC(F)F)CCCOC1C1CCN(C(c2ccoc2Cl)=O)CC1 N1(C(CCc2ccn(C)c2)=O)CC(NC(=O)CN2CCC(C)(O)C2)C2(CCC2)C1 c1(CCC(=O)NCC(CC)NC(c2ccn(C)c(=O)c2)=O)c(O)nc(=N)[nH]c1C c1(CNC(=O)NC2CCN(C(c3ccsc3)=O)CC2)ccnc(Cl)c1 CCC(Cc1ccc(C)cc1)N=c1ccnc(NCc2cocn2)[nH]1 C1(CNC(c2ccc(CCC)[nH]2)=O)C(C)CCN1C(C1(COC)CCC1)=O N1(C(C(CCC)NC(N)=O)=O)CCC(NC(=O)CCCC2CC2)C12CC2 c1(C(N2C(C(=O)NC(CC)C(C)O)CC(C)C2)=O)c(C)cc(OC)cc1C c1(C(=O)NCCCC2N(C(CC(=C)C)=O)CCC2)cc(Br)ccc1OC c1(C(N2CC(C)C(NC(C3CC(=C(F)F)C3)=O)C2)=O)cccc2nc[nH]c12 N1(NC(=NCCCCOC)NCCNC(C)=O)CCS(=O)(=O)C2(CCCCC2)C1 c1(CN(C)C)ccccc1COC(=O)CCc1ccn(-c2ccccc2)n1 c1(OC)cc(C#N)cc(Cl)c1OC(=O)C(O)CC(=O)O N1(C(C2N(C(C)C)CCC2)=O)CCCC(C(=O)NCc2nc[nH]n2)CC1 C1(CC(=O)NC(COC)C)CCCN(c2nccc(-c3sc(C)nc3C)n2)C1 Cc1ccc(CNC(=O)C(N2CCC(N(C)C(c3cc(Br)co3)=O)C2)C)cc1 CC(C)C(O)CC(=O)N1CC2(CCN2C(=O)CCC(C)(F)F)C1 c1(NC(C)=O)cc(=NCC2CN(C(c3ccnc(CN(C)C)c3)=O)C2)[nH]c(C)n1 c1(C(N2CCCC(NC(CCc3cnn(C)n3)=O)C2)=O)c(F)ccc(N)c1F c1(NCCC2CCCN(C(CC(COC)(C)O)=O)C2)nc[nH]c2ncnc1-2 C1(CNC(CCc2n(C)ncc2)=O)CC(C)(C)CN1C(=O)C(O)C1CC1 N1(C(C2CCCCC2)=O)CC(C(=O)O)Cn2nccc21 c1(CC(=O)NCC2C(C)(C)CN(C(C3CC34CC4)=O)C2)cccc2ccoc12 C1(C)(CC)CC(NC(=O)CNC=O)CN1C(=O)CC1CNC(=O)O1 C(=O)(C1=CCCCO1)NCC1(F)CN(C(c2c(C(=O)OC)cccc2)=O)C1 CCC(C(=O)N1CC(N(C)CCNC(C2(c3cc(C)no3)CC2)=O)C1)NCC C1(OC)CC2(C1)CC(N=c1[nH]c(=NCC34CC(CCO3)C4)[nH]c3c1CSC3)C2 CC(C)CCCC(C)C(=O)N1CCN1C c1(NC(C2N(C(=O)Nc3ccc(C)cc3)CC(O)C2)=O)cnc(Cl)c(Br)c1 c1(CC)nc(N(C)CC2CCCN2C(c2ccc(CC)s2)=O)cc(C#N)n1 C#CCCCCCCC(=O)N1CCC(F)CC1C(=O)N(C)Cc1cccs1 C(CCCC(CO)NC(C1(OC(C)C)CCC1)=O)NC(c1onc(CC)c1C)=O N1(C(c2cc(C(C)=O)[nH]n2)=O)CC(NC(c2cnn(C)n2)=O)C(C)(C)C1 c1(OC)cc(F)cc(C=CC(=O)N(CC(C)O)CCOCc2cc(F)ccc2C)c1 c1(N2CC(NC(C(CN(CC)CC)F)=O)C(C)CC2)ncc(C#N)cc1Cl Cc1c(NCC2CN(C(C)C)CCO2)ncnc1N1CCOC(C2CCOCC2)C1 C1(CNC(CN2CC(C)C2)=O)CC(F)CN1C(=O)C(C)OCCN(C)C CC1(C)CN(C(=O)C(N2CC3CCC2CC3Br)=O)CC(CC(N)=O)O1 CN=S(C)(=O)CCOC.N1(C)S(=O)(=O)NC2C(C(=O)OC)C2C1=O C1(C)(C(N2CCC(N(C(C(CCOC)C)=O)CCO)C2)=O)CCCCCC1 c1(C(=O)NC(CCNC(CCN(CCC)C)=O)C(C)C)cc2ccnc(Cl)c2[nH]1 C12(C(=O)NC3C(CNC(CCC(C)OCC)=O)CCC3)CC3CC(C(=O)N1)C2C3 C1(C(=O)NC2(C(C)C)CC2)CC(NC(C2(n3cccc3)CC2)=O)CCO1 n1(CC)ccc(C(N2CCCC2CC(=O)NCC2CC23CC3)=O)c1C N1(C(C(C)CC2CC2)=O)CC(F)CC1C(=O)NCCS(C)(=N)=O c1(OC)c(Br)ccc(C(c2nnnn2C)NCCc2cc(O)nc(SC)n2)c1F N(C1CCc2c(F)ccc(F)c21)C(=O)NCc1c(C(C)(F)F)cccc1 N1(C(c2c(C)csc2)=O)CC2(C1)OC1(C)CC2(NC(=O)C(C(C)C)N(C)C)C1 C1(OC)CN(C(c2cccn2C2CC2)=O)CC1NC(=O)CS(=O)(=O)NC(C)(C)C C1(C(=O)NC(CNC(C2C(C)(C(=O)OCC)C2)=O)CC)CNC(=O)N1 N1(C(C2(C#N)CC(C)C2)=O)CCC=C(CNC(=O)CC(C)C(F)F)C1 C1(NC(=O)C=C2CCOCC2)CCSC12CN(C(c1cccc(C(F)F)c1)=O)C2 N1(C(c2c(Br)ccc(C)n2)=O)CC(S(=O)(=O)CC(F)(F)F)C1 O=C(CC(C(F)(F)F)c1cc(Cl)cc(Cl)c1)OCCC1CCCCC1 C1(C(=O)NCc2cc(CO)ccn2)C2CCN(C(=O)COCC3CCC3)CC12 c1(OCCC)ccc2c(c1)OCC(CN1CC3C=CC1C(C(=O)O)C3)=C2 c1(CN2CCCC(CNC(c3nc(C)c(C)s3)=O)C2)ccc(C#N)c(F)c1 C=CC1(C(=O)N(C2CC(CO)C2)C)CCN(C(C2C(C#N)C2(C)C)=O)CC1 C1(NC(C(C2CCN(C(c3cccc(O)c3)=O)CC2)C)=O)CN(C)CC12CC2 c1(OC)cc(Cl)cc2[nH]c(C(=O)NC3(CNC(=O)C=CCF)CCC3)cc12 CC1CCN(C(c2cccc3oncc23)=O)CCN1C(c1ncccn1)=O N1(C(CNC(=O)OC)=O)CCC(CC(C)NC(C2(CO)COC2)=O)CC1 N1(C(CCCCCCCC)=O)CCC2OCCN(C(C3CCCCN3C)=O)C2C1 C1(C(N2CC(O)(CNC(c3n(C)nnc3)=O)C2)=O)CCc2n[nH]cc2C1 Cc1cc(-n2ccnc2)ccc1C(=O)NC1CN(C(c2cnns2)=O)CC1O C1(NC(=O)NC2CCN(Cc3ccccc3)C2=O)CCc2n[nH]cc2C1 Cc1ccc(C)c(CCCC(=O)NCCC(O)CNC(C2(C)CC2(F)F)=O)c1 c1(C(=O)NC2CCC(NC(C3CC(C(=O)OC)C3)=O)CC2)cc(F)cc(F)c1 C(=O)(CCC(C)(C)NC(c1ncncc1Cl)=O)NCC(C)CC1CCC1 N#Cc1ccc(CCC(=O)NCc2ncsc2-c2ccccc2)cc1 C1(NC(CC(COC)C)=O)CN(C(c2cc(OC)no2)=O)CCC12CCC2 n1(CC(=O)NC2CCC(NC(C(CC=C)C)=O)CC2)cnc2c1CCCC2 N1(Cc2c(C)nc(CC)o2)CCC2C(CCCN2C(=O)CCc2cnn[nH]2)C1 C1(NC(CCCOCC)=O)COCCC1C(=O)NC1C=CCCC1 C(=O)(N=c1[nH][nH]c(C)c1C)C12CC(NC(c3cccc(OC(C)=O)n3)=O)(C1)C2 N1(CC(C)SC)C(=O)CN(CCCCn2cnnc2)C1=O C=CC1(NC(=O)CCN(C(=O)C(=O)NC(C)C)C(C)C)CCOCC1 c1(C(C)CC(=O)NC2CCCC2NC(=O)CC2(C)CC2)ccccc1F c1(C(=O)NC(C2CCCN2C(=O)CCc2cc(Cl)no2)(C)C)coc2c1COC2 c1(C(N2C(C)CC(CNC(C3(C)COCCO3)=O)CC2)=O)nccn2ccnc12 C1(CNC(CC(COC)C)=O)(NC(c2nnc(S)n2C)=O)CC2CCC1CC2 CC1(C)CN(C(C23CCC(CC2)CC3)=O)CC1CNC(c1n[nH]cc1Cl)=O CC(=O)n1cc(CNCC(c2ccc(O)c(O)c2)C)c2ccccc12 CCC(C)CC(C(=O)NC1(C)CN2CCC1CC2)NC(=O)CCCC(C)C N1(C(c2cc(Br)ncc2F)=O)CCN(C(=O)CC2CCCC2)C(CO)C1 Clc1ccnc(N2CCCC(OC3CC3)C2)c1I c1(C(=O)NC2CN(C(CCc3nnc(C)n3C)=O)C(C)C2)cccc2nc[nH]c12 c1(C(=O)NCc2c(CNC(C=CSC)=O)cncc2)ccc(C(C)=O)c(F)c1 N1(CCCC(=O)NCC23CC2CN(C(=O)Cc2cncnc2)C3)C(=O)CNC1=O N1(C(C2CC(=O)CC(=O)C2)=O)CC2CCC1CN2C(=O)C(O)c1ccsc1 C1(CC(=O)NC2CCN(C(c3ccc(F)cn3)=O)CC2F)CCCC2(CCC2)O1 c1(C(=O)NC2CN(C(C(CC)N3CCCC3=O)=O)CC2O)cc(F)ccc1Br c1(C(=O)NC(C2CC3(CCC3)C2)C)ccc2c(n1)CN(C(C1CC(F)(F)C1)=O)CC2 C1(O)(C(C)NC(COCCCCOCC#C)=O)CN(C(=O)C(F)CC2CCC2)C1 C#CC1CCCN1C(C1COCC1NC(c1ccc(Cl)cn1)=O)=O c1(C(=O)NC(C2(O)CN(C(COCC#C)=O)C2)C)cc(F)cc(Br)c1 c1(OC(C)C(=O)NC2CC(OCC(F)(F)F)C2)cc(C(F)(F)F)ccn1 c1(C(N2CCN(C(C3N(CC)CCC3)=O)C(C(C)C)C2)=O)cc(C#N)c(C)cn1 CCC(C)C(C)C(=O)N1CCC(CNC(c2cc(C3CCCC3)[nH]n2)=O)C1(C)C C1(CC)CNC(=O)CN1C(=O)CCC1CCCCN1C(c1n[nH]cc1C)=O c1(OC)cnc(C(=O)N(C2CCN(C(=O)C3=COCC3)CC2)C)nc1 Cc1c(C(=O)NC2CC3CCC2N3C(=O)C(C)C#N)oc2ccc(Br)cc12 N1(C(C(C)NS(C)(=O)=O)=O)CC(NC(C2(C)CCCCC2)=O)Cc2ccccc21 N1(C(C2OCC(C)(C)C2)=O)C2CCC1CC(C(=O)NC1CCCC(C(N)=O)C1)C2 c1(C(=O)NCC2C(NC(c3cc(Br)co3)=O)CC2)cccc2[nH]ncc12 N1(C(c2cc(C)cc(O)n2)=O)CCCN(C(=O)Cc2cc(Cl)cc(Cl)c2)C(C)C1 C1(CC)CN(C(=O)NCC2CCCN2C)CC1CO c1(C(=O)NC2C(C(=O)NCCOCC#C)CC2)cccc(C)c1O c1(C(N(CCC(C)NC(=O)COC2CCOC2)C)=O)ccc(C(F)F)c(F)c1 N1(C(c2c(C(=O)OC)[nH]nn2)=O)CCC(C2(O)CCOCC2)CC1 c1(C(CO)NC(=O)COC2CCC2)cccc(OCc2ccccn2)c1 N1(C(C(CCC)N(C)C)=O)CC(NC(C2CCC3(CCC3)CC2)=O)C2CCCC12 c1(-c2nnc(C(C)(C)OC(=O)CCc3ccnc(Br)c3)o2)ccc([N+](=O)[O-])cc1 C(=O)(C(C#N)C(C)(C)C)NC(C)CCNC(=O)CCS(C)(=O)=O C1(C(=O)NCC2(Cl)CC2(F)F)(CC)CCN(C(c2cc(C)nc(O)n2)=O)CC1 N1(C(C2CCCC(F)C2)=O)CCN(C(=O)Cn2nnnc2C2CC2)C(CCO)C1 c1(C(=O)NCC2N(C(C(C=C)OC)=O)CCC2)ncc(C#N)cc1C Cn1ncc(C(N2CCCCC2CCNC(c2ccc(Cl)nc2)=O)=O)c1C1CC1 N1(C(Cc2c(O)ccc(C)c2)=O)CCC2CN(C(c3ccccc3C)=O)CCC12 CC1(C)C(C(=O)OC(C)(C)C)CCN1CC#Cc1cccs1 Cc1nc(C)c(C(=O)N(C2CCCN(C(C3(C(C)C)CC3)=O)C2)CCF)[nH]1 CC(C)C(F)(CNC(c1cc(F)cnc1O)=O)C(=O)NCc1cnccc1C#N c1(OCCCc2n(C)nnn2)cccc(-c2ccon2)c1 CC(C)(C)CCCCC(=O)NC1CCC(NC(=O)CC2CC(=O)C2)CC1 c1(OC)ccnc(OC)c1C(=O)N(CC(C)C)Cc1cn(C(C)CO)nn1 Cc1nc2c(C(=O)NC3CCN(C(C4CCCCC4O)=O)C3)ccnc2[nH]1 C(c1cn(C)c(=O)n(C)c1=O)=CC(=O)NCC(CC=C)NC(c1csnn1)=O c1(C(N(C2CCCN(C(=O)CCC(=O)OC(C)(C)C)C2)C)=O)ccc(CO)nc1 c1(C(=O)NCC(CC)NC(C2CCCN2C(C)C)=O)cccc2occc12 CC(C)C(C(=O)NCCCC1(O)CC1)N(C(=O)Cc1ccccc1)CCO c1(NC(=O)NCC2C(CCC)C2)ccc(OC)nc1Br C=CCC(C(=O)NCC=CC(=O)N(C(C)CO)C)NC(C)=O c1(CNC(C2(NC(c3c(CC)c[nH]c3)=O)CCCCC2)=O)ncc(F)cc1F CCC(CC)(C(=O)N1CCC(C)(C)C(C(=O)NC2(CCF)CCC2)C1)C(C)C Cc1cc(Cl)c(C(=O)NC(C2CCOC2)CNC(c2cnc(S)[nH]2)=O)cn1 C(=O)(CC1=CCCCC1)NCC12N(C(=O)C(C)(C)F)CC(COC)(C1)C2 C=CC(C)(C)C(=O)NCCN(C(=O)Cc1cnccc1C(F)(F)F)C N1(C(CCCCC(=O)NC)=O)CCC(NC(=O)C=Cc2cnc[nH]2)C2(CCC2)C1 C(CC(C)(C)C(=O)N1CCC1C1CCC1)NC(C(SC)SC)=O Cn1cnn(CCC(=O)NCC2COCCN2C(=O)C2=NOCC2)c1=O Cc1cccc2c1CN(C(=O)C(c1ccoc1)NC(=O)CC#N)C2 c1(CC)ccc(C(=O)NC23COC(C2)C(NC(=O)C(C(C)C)SC)C3)cc1Cl c1(-n2cc(CN(C)C(c3cc(Cl)sc3Cl)=O)nn2)ncc(Cl)cn1 C1(NC(C2CCC3CC3CC2)=O)CCCCN(C(c2n[nH]cc2[N+](=O)[O-])=O)C1 CCC(C(c1nnnn1C)NCCC1(c2ccccc2)CCCCC1)C(C)C c1(C(N(CCC(=O)NCC(=O)NC(C)C)C2CC2)=O)sccc1C#N C1(OC)CC(NC(c2cccc(F)c2)=O)CN(C(=O)CN2CCCC2)C1 Cc1noc(C)c1CC(=O)NC1CCC1NC(=O)CC(C)(F)F C1(CN(C(c2c(OC)c[nH]n2)=O)C2CC2)CCCCN1C(=O)CCNC(C)=O c1(SCC)ccccc1C(=O)NCC1CCC(NC(=O)Cc2cccnc2Cl)C1 C1(NC(COCC)=O)CC12CCN(C(=O)CCC1CC(C)(C)CO1)CC2 c1(C(N2CC(C)(NC(c3cccc(OC)c3F)=O)C2)=O)cc(S(N)(=O)=O)co1 C(C(C)(C)CC(=O)NC1CCOC1(C)C)NC(C=Cc1ccc(C)o1)=O C1(CNC(Cc2c(C)ccs2)=O)CC2CC2N1C(=O)CCCC1CCCCC1 N1(C(COC2CCN(C(C(CC=C)N(C)C)=O)C2)=O)CC(O)C2(CCCC2)C1 c1(C(=O)NC2CC(CNC(C(C)S(N)(=O)=O)=O)OCC2)cc2ccccc2s1 C1(C#N)(C(=O)NCC2CC(COC)CN2C(C2(F)CCOC2)=O)CCSCC1 c1(C(=O)NCC2CC(NC(C(CC)N(C)C)=O)CC2O)cn2c(C)cccc2n1 CCCC(CC)C(=O)NCC1(F)CC(NC(c2cc[nH]c2C2CCC2)=O)C1 Cc1cc(C)c(CNC(N2CCOCC2c2cn[nH]c2)=O)s1 c1(OC)ccc2c(c1)CCC2C(=O)N1CCC(CO)(NC(=O)CCCC(C)C)C1 c1(CC(=O)NC2CC(NC(c3c(C)cc(F)s3)=O)C2)c(C)nn(C(F)F)c1C CC(C)C(CC(=O)N1CCCC(C)(CNC(c2cnco2)=O)C1)c1ccon1 c1(C(=O)NCCC(C)N(C)C(c2ccn3ncccc23)=O)ccc(Cl)c(N)c1Cl C1(Cn2cc(C(C)OC)nn2)C(C2CC2)CCN1C(=O)Cc1c(C)cccc1Cl CCC(c1cccc(Cl)c1)=CC(=O)NC1CN(C(c2occc2F)=O)CCC1C n1(CC(=O)OC)cnc(C)c1C(=O)NC1CCOCC1NC(=O)C(C)CSC N1(C(c2cn(CC)nc2)=O)C(C)CN(C(=O)C(F)(F)CO)CC1C c1(C(=O)NC(CC)C(C)O)cn2c(n1)CN(Cc1ccnc(C(=O)OC)c1)CC2 C1(C(=O)NCCC(C)NC(c2cc(C3CC3)ncn2)=O)(COC)CCC(=O)N1 C(C(C)(C)CN(C(=O)CCc1cnc(C)s1)C)NC(C1(OC)CCC1)=O CC(C)CC(CNC=O)CC(=O)N1CCC1CNC(c1cscc1S(C)(=O)=O)=O C1(CC=C)(C(=O)OC)CCCN(C(c2cnn(-c3cc(C)ccc3F)c2N)=O)C1 C(C(C(=O)NCCCOCCN(C)C(c1ccc[nH]1)=O)c1ccccc1)SC C1(C(c2cc(CC)no2)NCc2cnccn2)CCCCCC1 N1(C(C2C(CNC(C(C)=CCC)=O)CC2)=O)CC2(CCN(C)CC2)C1 N1(C(C(CC=C)C(=C)C)=O)CCC2(COCCN2C(=O)C(C)(C)COC)C1 N1(C(C(CO)NC(C(C)C)=O)=O)CCC(=CCNC(C2CC23CCOC3)=O)CC1 CC1(C)CC(NC(=O)Cc2ccoc2)CN1C(c1cc(C(=O)NCCO)[nH]n1)=O Cc1cc(S(=O)(=O)NCC2CCCC2NC(=O)C(F)(F)F)c(C(=O)O)cc1Br Cc1csc(Cl)c1C(=O)NCC1(CO)CCN(C(C2(CC(C)C)CC2)=O)C1 C1(NC(C(=O)NC(C)C)=O)CC2CCC1N2C(=O)CCCCCN(C)C N1(C(CCOC)=O)CCC=CC1C(=O)NCCCOCC(F)F N1(C(COCCCC)=O)CC2COCC2(C(=O)NC(C)CCC(F)(F)F)C1 Cn1ncc2c1CC(C(=O)NCC1COCCN1C(c1cn(C3CC3)nn1)=O)CC2 C(CC(=O)NCc1ccc(OC(F)F)cc1F)(C(C)C)C1C(C)CNCC1 Cc1nc2n(n1)CCC(C(=O)NC(c1cn(C)nn1)C(=O)O)C2 CC(C)(C#CC(=O)N1CC2CCCC1C2CO)CNC(c1cccc(O)c1F)=O Cc1ccc2c(c1)C(NC(C1(N)CCC1)=O)CCCN2Cc1ncco1 CC1NC(=O)CCC1NC(C1CC(O)(CNC(C2CC3(CC3)C2)=O)C1)=O c1(C(=O)NCCN(CCCCCC)C(=O)C(C)C2CC2)c[nH]c2cccc(C)c12 c1(CC(=O)NCC(O)CCNC(c2cc(O)ncn2)=O)ccccc1Cl C1(c2nnnn2C2CC2)(NCc2c(N(C)C)ccc(Br)c2)Cc2ccccc2C1 C1(C(=O)NCCC2N(CC)CCC2)CN(C(c2nnc(S)n2C)=O)CC1C c1(CN2CCN(c3ncc(SC)cn3)C(C#N)C2)ncnc2cc(I)sc12 C#Cc1ccc(C(=O)NCCN(C(=O)C(c2ccc(C)s2)C)C(C)C)c(F)c1Cl N1(C(C(C=C)(F)F)=O)CCN(C(c2cccn2C(C)C)=O)C(CS(C)(=O)=O)C1 NS(=O)(=O)c1ccc(C(=O)Nc2ccc(I)c(F)c2F)nc1 Cc1cc(CC(N2CC(c3cn(-c4nccc(C)n4)nn3)C2)=O)cc(F)c1 C(c1cccc(O)c1)=CC(=O)N(C)CCN(C)C(c1cncc(C(F)F)c1)=O C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC1C(OC)CN(C(c2nc(CCC)sc2)=O)C1 CCC(C(=O)N1CC(C(C)(C)O)(CNC(=O)C(F)n2cccn2)C1)NC(C)=O c1(C(=O)NC23C(CN(C(CC4(NC(C)=O)CC4)=O)C2)C3)cc2c(Cl)nccc2o1 Cc1cc(C#N)nc(N2C3CCC2(CNC(=O)C(c2ccc(Cl)s2)C)CC3)n1 C(=O)(N1CCCc2nncn21)C1CCN(C(Cc2cnc(C)s2)=O)CC1(C)C C(C)(C(C)C(=O)NCCCS(C)(=O)=O)NC(C1CC(O)(CC#C)C1)=O c1(CN(C(C2N(C(C=CCN(C)CC)=O)CCC2)=O)C)ccc(C)cn1 c1(OCCC(N2CCC(C(C)NC(C3N(CC)CC3)=O)C2)=O)cccc(C)c1 Cc1ccc(C(N2CCCC2Cn2cc(CNC(C3CC3(F)F)=O)nn2)=O)nn1 Cc1cc2sc(C(=O)NC(C3CCCN3C(C3CC34CCCC4)=O)(C)C)cc2s1 c1(CC(N2C(CN(c3nc(Cl)c(C#N)s3)C)CCCC2)=O)ccc2c(c1)CCO2 c1(C(=O)NCC(CC(=O)NC2CC=C(C)CC2)(C)C)cccc2c(C)coc12 N1(C(C(C)N(C(=O)Cc2cccc(C)n2)CC)=O)CCOC(C)(C(C)C)C1 c1(N(C2CCN(C(c3cc(C)ncn3)=O)C2)C)nc(C(C)C)nc2[nH]ccc12 C=CC1(C(N2CCC(N(CCC)C(C3CC4(C3)CC(O)C4)=O)C2)=O)CCCCC1 N1(C(C(C)c2cccs2)=O)CC2C(NC(c3c[nH]c(C(F)(F)F)c3)=O)C2C1 C1(CC(=O)NCCN(c2nc(C(=O)OC)ns2)CCC)CCCC(F)(F)C1 Cn1cc(S(N)(=O)=O)c(C(=O)NC2CN(C(=O)COC3(C)CCCC3)C2)n1 c1(CC)cc(C(=O)NC(CNC(c2ccnn2COC)=O)CC(C)C)c(C)nn1 Cc1nn2ccccc2c1C(N1CC(CCNC(c2ccc(F)cc2O)=O)C1)=O c1(OC)ccc2c(C)c(C(=O)Nc3cnn(C(C)C(C)C)c3C)oc2c1 c1(C(C(=O)NC2C(C)CN(C(c3cnn(C4CC4)c3)=O)C2)=O)ccc(F)c(F)c1 C1(C(N2CCC(N(CCC)C(c3oc(CO)cc3C)=O)C2)=O)CCS(=O)(=O)CC1 C1(NC(c2cnc(OC)nc2)=O)CC(O)CN(C(=O)CCc2nc(C)no2)C1 C(=O)(C1Cc2ccc(F)cc21)NC1C(OC)CN(C(c2c[nH]cc(C)c2=O)=O)C1 C1(CC(N2CCC(CN=c3[nH]ncs3)(CO)CC2)=O)CC2(CCC2)CO1 C1(C(N(CCCNC(C(C)SC)=O)CC2CCCC2)=O)CCN(S(C)(=O)=O)C1 c1(CC(=O)NCC2CC(NC(C(CCC)N(C)C)=O)C2)cc(C)cc(C)c1 C1CCN=C2NC(=NCC(=O)N1)Nc1cc[nH]c12.c1(C(=O)OC)ccccc1 c1(CCCn2cc(CCS(C)(=O)=O)nn2)c[nH]ccc1=O.C1(=O)C(CO)N1CC Cc1ccc(CC(=O)NCC2CCN(Cc3ccccc3OC(F)F)C2)cc1 CCC(C)(C)C(O)C(=O)N1CCOC(C(=O)NCC(Cl)C(C)(F)F)CC1 C1(NC(CC(=C)Br)=O)CN(C(=O)CNC(=O)CC2CCCC2)C2(CCC2)C1 N1(C(C(C)(C)OCC(F)(F)F)=O)CC(NC(C2CC3(CCCO3)C2)=O)C(C)(C)C1 C(=O)(C(C)(F)c1ccon1)N(CC(C)NC(C1CSCCS1)=O)C C#Cc1ccc(CC(=O)N(CC(=O)Nc2cnn(C(C)(C)C)c2)CC2CC2)cc1 C(=O)(CC1=NNC(=O)C1)NCC(C)NC(c1ccc(CNS(CC)(=O)=O)cc1)=O N1(C(C(C)CO)=O)CCCCCC1C(=O)NOCC1(C)CC1 N1(C(C)C(c2cnn(C)c2)=O)CCCCC(C(=O)O)C1 c1(C(=O)NC2C3(CC(NC(=O)Cc4cccc(F)c4)C3)C2)cc2ccccc2[nH]1 c1(C(N2CCC(C(C)(C)NC(c3c(C)coc3)=O)C2)=O)ccc2ncsc2c1 CC1(C)CC(Cc2nc(-c3cc[nH]n3)nn2CC2CC2)CN(C(=O)OC(C)(C)C)C1 C1(C(=O)NC2CN(C(=O)C3=C(Cl)CC3)CC23CC3)Cc2ccccc2S1 Cc1ccc(O)cc1C(N1CCC(C)C(NC(c2ccc(C3CC3)nc2)=O)C1)=O N1(C(C(C=C)CC)=O)C2CCC1C(C(=O)NCCCN(C)C(C)=O)C2 c1(C(N2CC3(CN(C(C4(C)C(C)(C)C4(C)C)=O)C3)C2)=O)c(N)cccc1[N+](=O)[O-] c1(OC)ncc(C(N2CCCC2C(C)NC(c2cc(C)nc(O)c2)=O)=O)cc1Cl N1(C(CC)=O)CCC(C)C(N(C(=O)CSCc2ccc(Br)cc2)C)C1 Cc1nn(C)c(C(=O)NC(c2ccccc2)CNC(c2cc(Cl)n(C)n2)=O)c1Cl Clc1ccc(OCCN(c2cc(-c3ccccc3)ncn2)C2C3CNCC23)cc1 c1(C(=O)NC2(C)CC(NC(Cc3cc(C)on3)=O)C2)nc2ccc(Br)cn2n1 C(C(C(=O)NC1CCCC(C)C1)C(C)(C)C)NC(C1(COC)CCCC1)=O C1(C(N2C(C)CC(CNC(c3c(C)n[nH]c3C)=O)C2)=O)C2CC3C(C2=O)C13 C1(C(N2CC3C(CC(=O)NCCc4nc(CC)[nH]n4)C3C2)=O)CC(=O)OC1(C)C N1(C(C2(CC)CC2(F)F)=O)CCC(N(C)C(c2cc(CS(C)(=O)=O)on2)=O)CC1 C1(CC(N2CC(=CCC)C2)=O)CCCN(C(C2(C)CCOC2)=O)C1 C1(C(=O)Nc2c(C)cc(CC)s2)COC2(C1)CN(C(=O)OC(C)(C)C)C2 CCC(CC)(CC(=O)N1CCCC(NC(=O)CCC(C)O)CC1)C(N)=O Cc1ccc(-c2ccccn2)cc1NC(C1CN(C(=O)CN(C)C)CCO1)=O C(C)(C)(CCCN=c1[nH]cc(Cl)c(C)c1C#N)NC(COCCCOC)=O C(=O)(C(C(C)C)NC(C1CCCOCC1)=O)N1CC(C)(CC=C)C1 c1(C(=O)NCC2(CO)CCN(C(CC3C(C)CCO3)=O)C2)nnc(O)nc1O c1(C(=O)NC(CNc2nccc(OCCC)n2)(C)C2CC2)cccc2scnc12 C=CC(C)(CCOC)C(=O)N1CCN(C(c2cccc(CN(C)C)c2)=O)CC1C Cc1cc(N)c(C(=O)NC(CCNC(c2ocnc2C)=O)C(C)(C)C)nc1C C(=O)(CCC(C(C)C)NC(=O)CC1CCN(C)CC1)Nc1cncc(C#C)c1 N1(C(CCC=C)=O)CCC2C1CCCN2c1ncc2ccccc2n1 C(C(Cc1ccccc1)C(=O)O)NC(c1ccc(C(F)F)cc1)=O C1(CC(=O)NCC(C(C)C)(C)F)N(C(C2CCCCCN2C)=O)CCC1(C)C C12(NC(Cc3cccc(C(=O)OC)c3)=O)CCN(C(c3nccn3C)=O)CC1C2 c1(-n2cc(CCC(=O)Nc3ncc(CC)s3)nn2)ccc(F)cc1F c1(OCC)ncccc1C(=O)N(CCCCCNC(c1nnn(CC)c1C)=O)C C(=O)(C(C)(C)CN1CCN(C)CC1)NCC(C(C)C)NC(=O)CNS(N)(=O)=O C1(CC)CN(C(=O)C(=Cc2cccs2)C)CCC1NC(c1ccc(Cl)nc1N)=O S(=O)(=O)(c1ccc(Br)cc1F)NC(C1CCCN(C(C=CC=CC)=O)C1)C C1(C(=O)NC2C(CNC(CC(C)(O)C3CC3)=O)CCCC2)CCCCCCC1 C1(C(N(c2ccc(F)cn2)C)=O)CC2(CCCC2)C1 C1(NC(CSc2c(OC)cccc2)=O)CCC(C)N(C(=O)C2=CCCOC2)C1 C(=O)(C1=Cc2ccccc2C1C)NCC1N(C(CCc2cc(C)on2)=O)CC=C1 C(=O)(C(C)CC(C)CC)N(c1ncccc1C(F)(F)F)CC=C N1(C(C(CNC(C23CCC(CC2=O)C3)=O)OC)=O)CCCCN(C)CC1 c1(NC(C2CCN(c3snc(C)c3C#N)C2)=O)c(C(F)(F)F)nc2n1CCCC2 C(C(C(=O)N(C)C)C(C)(C)C)NC(CS)=O.CC(C)CCC=CCCOC N1(C(c2nc(C)n(C)c2C)=O)CCN(C(c2cc(F)c(F)c(F)c2)=O)CCC1C c1(CNCC(=O)NC(c2ccc(O)cc2)C(F)(F)F)ccc([N+](=O)[O-])cc1F S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1CCC(F)(C(=O)Nc2cncc([N+](=O)[O-])c2)C1 CCCS(=O)(=O)CC(=O)NCC1CCC1NC(=O)CCCCC=CC C(c1cccc(F)c1)=C(C(=O)NC(C)CCNC(=O)C=Cc1cnc[nH]1)F c1(C(N2C(C(=O)NC(C3CCCC3)C#C)CC(C)(C)C2)=O)ccc2c[nH]nc2c1 CC1CN(C(=O)COC2CCCOC2)CCCN1C(c1cncc(Br)c1)=O c1(C(N2CC(CNC(c3cnsn3)=O)C3C2C3)=O)n[nH]c2nccc(Cl)c12 c1(C(N2CC(N(C(CCc3cccc(OC)c3)=O)C)C2)=O)cnc2scc(C)n12 C1(C(=O)NCCC(=O)NCC(C)C)(NC(C23CC(F)(C2)C3)=O)CCC(C)(C)C1 C1(C)(CNC(C2(OCC)CC2)=O)CCCN(C(C23CC(CC(F)F)(C2)C3)=O)C1 c1(C(=O)NCC(C)(O)CNC(=O)COCc2ccncc2)ccc2cccnn12 C(N=c1[nH]c(=NCCN2CCCC2C(N)=O)[nH]c2ccsc12)c1cccc(C)c1 C(=O)(C1CCc2nccn21)N1CCCC(CN(C(=O)C(C2CCCCC2)O)C)C1 c1(C(=O)OC)ccc(NC(C)CCNC(=O)Cn2cnccc2=O)nc1 C1(C)(C(=O)NCC(C2CC2)NC(CN(S(C)(=O)=O)C)=O)CCCN1C C(C)(CCN=c1[nH]c2ccc(Br)cc2o1)NC(C1(C)C(CC)CCC1)=O Cn1[nH]c(=NC(=O)NCC(c2ccncc2)O)cc1C1CCCC1 Cc1ccsc1CC(=O)NC1CC(C)(CNC(=O)CCn2cccn2)C1 N1(CCCCCNC(C2(CC=C)CCCC2)=O)CCN(C(=O)C(O)C(F)F)CC1 S(=O)(=O)(c1ccncc1)N1CC(C)C(NC(c2cc(Br)ncc2F)=O)C1 Cc1cc(CNC(C2(NC(c3cnc(C)s3)=O)CC(F)C2)=O)c(C)s1 C(=O)(C1CCc2c[nH]nc21)N1CCN(C(CNC(CNS(NC)(=O)=O)=O)=O)CC1 C(=O)(CCN=c1[nH]c2ccccc2s1)N1CCC(O)(CNC(C(C)(C)F)=O)CC1 c1(C(=O)NC2(C(=O)OCC)CCC2)ccc(NCC2(F)CCOC2C)cn1 C=CC1(C(=O)NC2C=CCCCC2)CCN(C(=O)Cc2nccn2C)C1 N1(C(C2(CC=C)CCCC2)=O)CCC2CCN(C(=O)Cn3nnc(C)n3)CC2C1 CCCC(C)CCCC(=O)NC1CCCN(C(c2cccc(N)c2)=O)CC1 c1(CC)nn(C)c(CC(N2CCC(O)C(NC(=O)C=C(Cl)Cl)C2)=O)c1Cl O=C1CC2C(C(=O)NC3CCCN(C(=O)CCOCC4CCC4)C3)C2C1 c1(C(N2CCC(OCCNC(C(C(COC)C)C)=O)C2)=O)ccc2nn[nH]c2n1 Cn1cnnc1C(CO)NC(c1ncoc1CNC(c1cncs1)=O)=O CCC(O)C(C)C(=O)NC1CC(OCC(=O)NC23CC(F)(C2)C3)C1 N1(C(C2CCCS2)=O)CCN(C2CCN(c3cc(C(F)F)ncn3)CC2)CC1 CC(C)C(CC(=O)N1CCCC(C)(CO)C1)NC(=O)CC=Cc1ccccc1 C1(C(=O)NC(CN(C(CCOCCOC)=O)C)C)COC(C)(C)C1 c1(C(N2CCC(C)(C(N(CC(C)OC)C)=O)C2)=O)cc2c(=O)[nH]c(C)cn2n1 Cc1cn2c(n1)C(C)CC(C(=O)NC1CN(C(c3ccn(C(C)C)n3)=O)C1)C2 N1(C(CCCOCCC)=O)CCC2(CNC(=O)CN(C)C3CC3)CCCCC12 c1(C(N2CCCC(NC(c3ccco3)=O)C2)=O)ccc(-c2ccncc2)nc1O C12(C(N3C(C)(C)CC(NC(C4SCCS4)=O)C3)=O)CCCCC(F)(C1)C2 c1(C(N2C(C(=O)NCc3cc(C)sc3)CC2)=O)ccc(SC(C)C)cc1 C1(CNC(Cn2c(C)nnn2)=O)CC(F)CN1C(C12COCC1C2)=O N1(CC)CCCc2cc(CNC3CCCN(C(C)C(=O)NCC(C)C)C3)ccc21 C(=O)(C1CCOc2c(F)cccc21)NCC(C(C)C)NC(=O)C(F)(F)C(F)(F)F C(CC(CC)C(=O)NC1CN(C(=O)COc2cccnc2)CCC1O)=CC CC(C)(CC(F)C(=O)NC1CC(CO)C2CC12)NC(C1C=CCCC1)=O C(=O)(C(C)(C)CC(F)(F)F)NCCCC(C)NC(C1CCC(C)(C)CO1)=O c1(C(=O)NC2CC(NC(C(CC)CC(F)F)=O)C2)cnc2ccncc2c1 c1(NC(=O)C(=O)NC2CC2)cccc(OCC(=O)NCCc2cc[nH]n2)c1 c1(C(N(C2CN(C(C34OC(C)C(CC3)C4)=O)C2)C)=O)ccc2nc(CO)[nH]c2c1 c1(C(=O)NCC2(O)CN(Cc3c(C)nccn3)C2)cc(O)nc2ccccc12 C#Cc1ccc(CN2CC(C)OC(C)C2)cc1OC(F)(F)F c1(NS(C)(=O)=O)ccccc1C(=O)NCCNC(c1nccnc1Cl)=O c1(OC)c(C(=O)NC2CC3(C2)CC3NC(=O)C(C)O)cc(Br)cc1F c1(-c2cc(C)nnc2)cnc2cc(C(N3CCCCC3C(N)=O)=O)ccn12 N1(C(C(C(C)C)SCC)=O)CCN(C(=O)C(F)=CCCF)CC(O)C1 C12(C(N3CCC3CC(=O)NC3CCN(C(C)=O)C3)=O)CC3CC(CC(C3)C1)C2 CCC(C)(O)C(=O)NCC(C)CNC(=O)C(c1ccc(SC)s1)=O Cc1ccc(C(=O)NCC2CCCCN(C(c3cnnn3C)=O)C2)cc1O C(c1c(O)nc(=O)n2c1CCC2)=CC(=O)NCCOc1ccc(Cl)c(Cl)c1 c1(C(=O)NC2C(NC(C3C(c4c(C)ccs4)C3)=O)COC2)nn(C)cc1Cl C(c1ccccc1)=CC(=O)NC(C)(CNC(C1CC1c1ccoc1)=O)CO C1(C(N(C2CCNC2)CC)=O)CC(=O)N(Cc2ccccc2)C1 O(C=CC(O)(CNC(=O)NCC(C(F)(F)F)C1CCC1)C(F)(F)F)CC N1(C(C2(COC)CC2)=O)CCCC(O)(CN(C(=O)Cc2c[nH]nc2O)C)C1 O=[N+]([O-])c1ccccc1C(O)CNc1cnc2ccnn2c1 c1(N(C)C)ccc(CNC(=O)C(=O)NCCN2CCNC(=O)C2)cc1 c1(C(=O)NCC2CCC2NC(C(CC)C)=O)ccc(COc2ccccc2)cc1 c1(C(N(CCNC(=O)Cc2cnsc2)CC2CC2)=O)ccnc2ncccc12 C1(C)(C(=O)NCc2c(C(=O)NC(c3ncccn3)C)c[nH]n2)CC(F)(F)C1 CC1CC(CNC(=O)C=CCNC(C2(CO)COC2)=O)CCO1 C12(C(=O)NCCCNC(C)=O)CC1CN(C(C1CCC(CO)CC1)=O)C2 Cc1cc(C(=O)NC2(CCO)CCOC2)sc1-c1cccc(Cl)c1 C(C1CCN(C(C2(C#N)CCOC2)=O)CC1)=CC(N1C(C)(C(=O)NC)CCC1)=O c1(-c2ccc(CC3CCN(Cc4c[nH]c(=N)s4)C3)cc2)cccc2ccnn12 C(=O)(CCS(=O)(=O)CC(C)C)N1CCN(C(CCCCCOC)=O)C(CO)C1 c1(C(=O)NCCCCN(C)C)cccc(-n2cc(COC(=N)O)nn2)c1 C1(CC(=O)NC(C)CCCNC(=O)CC2(N(C)C)COC2)CCC12CCC2 N1(C(c2cnn(C3CCC3)c2)=O)CC2(C1)CN(C(c1cc(Cl)nc(Cl)c1)=O)C2 c1(C(=O)NCc2nnco2)ncncc1Cl Cc1c(O)c(=O)ccn1CC(N1CC(NC(C2CC2(C)C)=O)C2(CC2)C1)=O N1(CC(c2c(CN)c3c(s2)cccc3Br)=O)CCN(C)c2ncccc2C1 C1(C(N(C(CCNC(C(C)NC(N)=O)=O)C)C)=O)CC2C=CCC(C1)C2 N1(C(Cc2cnc(C)[nH]2)=O)CC2(C1)CN(C(c1coc(C(F)(F)F)n1)=O)CCO2 c1(CC(=O)NC(C2(O)CN(C(=O)COC3CCOC3)C2)C)ccn(C(F)F)n1 CC1(C)CN(C(C2CCS2(=O)=O)=O)CCC1NC(c1ncnc(O)c1Cl)=O C1(OCC)CCN(C(=O)NC(C2CCN(C)CC2)C2CC2)CC1C c1(C(=O)NCC2CC(NC(C(N3CCSCC3)C)=O)C2)occ2c1CCC2 CC(CC(=O)NN1CCCC1C(N1CCCC1C1CCOC1)=O)C1CCCC1 c1(C(N2CC(SC)C(NC(c3cnn(CCO)c3)=O)C2)=O)nc(C)c(C)nc1O C(=O)(C1CCCc2nn[nH]c21)N1CCN(C(C=Cc2c(C)nccc2)=O)C(C)C1 c1(C(C)NCC(=O)OCC(F)(F)F)ccc(OC(c2cnnc(O)c2)=O)cc1 S(=O)(=O)(c1ccc(C(=O)N(CC(C)NC(=O)C2=COCCO2)C)cc1)NC c1(C(N2CCC(CC(=O)NC3CCCN(C4CC4)C3)C2)=O)nc(Cl)ccc1Cl CCCCC(C(=O)N1CCCCC(CNC(C2(OC(C)C)CCC2)=O)C1)N(C)C Cc1c(F)ccc(C(N2CCC(C)C2CNC(c2cnccn2)=O)=O)c1N C(CC(C(N)=O)NC(C1(CNC(=O)C(C)SC)CCCCC1)=O)OC C1(NC(c2cnc(C)[nH]c2=N)=O)CN(C(=O)C=C2CCC(C)CC2)CC(C)(C)C1 C1(N(C)C)(C)CCN(c2ccccc2)CC1.c1(N2CCC(N)C2)cc(Cl)ccc1C C=CC1(CC(=O)N(CCCNC(c2cc(C(C)(C)C)n[nH]2)=O)C2CC2)CCC1 C(=O)(CCCCCS(N)(=O)=O)NC1C(CN(C)C)CCCC1 c1(CNC2C(C)CN(C(=O)C(C)(C)F)C2)ccc2c(c1)CCO2 c1(OCC)ncc(C(=O)NCC(C)(F)CNC(=O)Cn2nnc(C)n2)s1 N1(C(C2CCC(CC)CC2)=O)CCC2CCN(C(=O)Cc3cnccc3C)CC12 C(CCCCC(=O)N1CCC2CCC12)OCC.C12(CC)CN(C1)C2=O c1(C(=O)NC2(CC=C)CCN(C(=O)C(C)CCO)C2)ccc(Cl)c(F)c1F N1(C(C=CCOC)=O)CCOC(C)(CNC(C2CCN2C)=O)C1 C(=O)(CS(=O)(=O)C1CC1)N1CCCC(CNC(Cc2c(C(=O)OC)scn2)=O)C1 C(=O)(CCC(C)(C)C#N)NC(CNC(c1n(CC#C)ccc1)=O)C1CCC1 CN1CCN(C(=O)CCNC(c2cnc(Cl)n2C)=O)C(CO)C1 c1(CC)nc(C(=O)NC(CNC(c2cnc(C3CC3)[nH]2)=O)C2CCC2)co1 C12(NC(C(CO)N(C)C)=O)CCCC1N(C(=O)Cc1ccc3c(c1)OCO3)CC2 C(CCCCC(=O)N1CCCC(CO)(NC(=O)C=CC2CCCO2)C1)SC c1(C(=O)Nc2ccc(NS(N)(=O)=O)cc2)cc2c(cc1F)NCCC2 C(C(O)CC(=O)N1CCC(CN(C(=O)CC2CCC(O)C2)C2CC2)C1)N(C)C N1(C(C(CCC(C)C)NC(C2CC3(CC3)CO2)=O)=O)CCC2(CCCCO2)C1 CC1CN(C(C2CCCC23CCC3)=O)CC1(C)C(N1C2CCC1CC2)=O C(C1CN(C(C2(CC(C)C)CCC2)=O)CC1C(N1CC(OCCO)C1)=O)=CC C1(NC(c2nccc(OC)c2)=O)CCN(C(c2ccc(Cl)cc2C)=O)CC1CO CCCC(CNC(C1(C)CC(F)(F)C1)=O)C(=O)N1CC(N=[N+]=[N-])C1 C(c1cccc(F)c1Cl)=CC(N1C(C)(C)C(CNC(=O)C=CC(F)(F)F)CC1)=O C1(NC(C2(COC)CCCO2)=O)CCN(C(=O)Cc2cncc(C)c2)CC1CO c1(C(c2n(CCOC)nnn2)NCC2(COC)CCC2)cccc(F)c1F C1(NCCN(C(=O)Cc2ccc(C)s2)CC)CCCCN1C(c1[nH]ccc1C)=O C1(CC)CC(O)CN1C(=O)C(CNC(C1(OC)CCCOC1)=O)CC1CCCC1 C1(NC(C2(C)CC2(F)F)=O)CN(C(C23CC(C2)C3)=O)CC1C#N C1(NC(CS(CC)(=O)=O)=O)CC2CCC1CN2C(=O)C(C)(F)C(F)(F)F C1(C(N2CCCN(C(CCC(CC)OC)=O)CC2)=O)CCc2nc(O)[nH]c2C1 N1(C(C(c2cn(CC)nc2)=O)=O)CC(CNC(=O)C2CC2)N2CCC1C2 N1(c2nnc(C)s2)CCN(C)C(CNC(C2(CCF)CC2)=O)C1 C1(NC(c2ccc(OC)c(Cl)n2)=O)CN(C(=O)C(C)(C)N(C)C)CC2CCCC12 C1(NC(C2C(C=C)C2)=O)CCCN(C(c2cccc(-c3nnc(C)o3)c2)=O)C1 c1(C(C(=O)NCC2CCOC2)N(C)CC2C=CCC2)ccnn1C N(C1CCCn2cnnc21)C(C(C(C=C)C)C)=O Cc1ncn2c(NC(=O)CSC3CC3)ccnc12 N1(C(=O)C2CC2)CCCC(C(N2CCC(n3cncn3)C2)=O)C1 N1(C(CCCn2cc(-c3n(C)ncc3)nn2)=O)CCCc2c(F)cccc21 C1(NC(C=C(C)C(C)(C)C)=O)CCN(C)C12CCCN(C(C1CCSCC1)=O)C2 C1(CNC(CCC#C)=O)C(C)CCCN1C(=O)Cc1cscc1Br C1(N(C(=O)CNC=O)C)CCCCN(C(C2(O)CC2(C)C)=O)C1 C1(CNC(C(C2CCC2)OC)=O)CC(O)CN1C(c1cn(CC(F)(F)F)cn1)=O C1(C(=O)NC(C)CC(F)(F)F)CN(C(=O)C(C)(C)CN(C)C)CCC1(C)C C1(CNC(CN(C(=O)C=Cc2cn(C)nn2)CC)=O)CC2(CCC2)CO1 c1(-c2c[nH]c(=NCc3cc(OC)c(Br)nc3)s2)cc(O)c(F)cc1F c1(CNC(CC2CC(NC(CNC(CC)=O)=O)C2)=O)nnn(C)n1 N1(C(C2(C)CC(C#N)C2)=O)CCC(NC(C2CC23CCCC3)=O)C(O)C1 C1(C(=O)NC(CC)CO)(CO)CCN(C(=O)N(C)C)C1 N1(C(c2cccc([N+](=O)[O-])c2)=O)CCC2(C1)CN(C(C1CC1F)=O)CCO2 N1(C(C2C(NC(C3C(CCOC)C3)=O)CCO2)=O)CC(C)(C)C1C1CC1 C1(O)(CNC(c2c(C)nc[nH]2)=O)CCN(C(=O)CCc2cnccn2)C1 C(c1ccc(C)nc1)=CC(=O)N(C)CC1(O)CCN(C(C(C(C)C)OC)=O)C1 CCC(CC(=O)N1CC2CC(NC(C3(C(F)(F)CC)CC3)=O)C(C2)C1)C(C)(C)C c1(C(=O)NCC2C(NC(C3C(C)(C)C3)=O)CCC2)cnc(O)c([N+](=O)[O-])c1 c1(C(=O)NCCCC(C)NC(=O)CN2CCOCC2)cc2ccccc2[nH]1 c1(C(=O)NCC(CNC(CNC(CC(C)C)=O)=O)C)cccc(N(C)C)c1 C1(C(N2CC(N(C)CCO)C2)=O)CCCC(NC(C2OCCC2(C)C)=O)CC1 c1(COC(F)(F)F)ccc(SS)cc1.C1CCC(=O)NCC(C)CNC(=O)N1.CC=O Cn1ccc(-c2nc(C(=O)NC3CC(NC(=O)CCF)C3)cs2)n1 C(=O)(C(C)(C)CCC(=O)OCC)NC1C(CNC(COCCC=C)=O)C1 Cc1nccn1CCC(=O)NCC1(C(=O)NCCCO)CCC1 C1(CNC(CC2CCC(C)(C)CC2)=O)CC(C)(C)CCC1NC(=O)CCC(F)F N1(C(CCC(=O)OCC)=O)CC2CC(NC(c3cc(OC)ccc3F)=O)CC1C2 c1(COC)nocc1C(=O)N(C)CC1CCN(C(=O)CSC2CC2)C1 c1(NCC2(CNC(CN=S(C)(C)=O)=O)CC23CCC3)ccc([N+](=O)[O-])cc1 CCN=c1ccc(C(=O)NC2CCOCC2NC(=O)CC2(N(C)C)CCC2)c[nH]1 C1(C(N2CCC3C(NC(c4cnc(SC)n4C)=O)C32)=O)CCC(=O)N(C)C1 N1(C(c2ccc(C)nc2)=O)CC2CCC1CC2NC(=O)CC1=CCOCC1 CCCC(CC1CCCC1)C(=O)NC1CC(CNC(C2CC3(C2)CC3(F)F)=O)C1 N1(C(c2nc(C)[nH]c2)=O)CC(CNC(=O)CONC(=O)OC(C)(C)C)CC1C CC1CCC(NC(=O)OC(C)(C)C)CN1C(=O)NC1(C)CS(=O)(=O)C1 O=C(CC1C(=O)Nc2ccccc21)NCCC1(O)CN(C(C2(O)CCC2)=O)C1 C(=O)(CCCCCC#N)N(C1CCCCN(C(c2ccccc2C(F)F)=O)C1)C O=C1CCCC(C(N2CCCCC2C(=O)NCCc2cccnc2O)=O)CC1 c1(C(c2n(CCC)nnn2)NC(C)C(=O)NCCOC)cc(Cl)sc1C C(=O)(C(C#N)C(C)(C)C)NC1(CO)CCCN(C(c2cc(OC)c(O)nc2)=O)C1 c1(C(N2CCC(CNC(CCc3scc(C)n3)=O)CC2)=O)sc(C)c(C)c1C N1(C(C2(C)CC(OC)(OC)C2)=O)CC(NC(c2cccn(C)c2=O)=O)CC(O)C1 N1(C(C(CCC)OC)=O)CCN(C(c2cc(=O)c(OC)co2)=O)C(COC)C1 c1(C(N(CC(N2CCC(CCC)C2)=O)CC)=O)ccn2cncc2c1 n1(C(C(=O)NCC(CN(C(CNC(C)=O)=O)C)(C)C)C)nc(C)c([N+](=O)[O-])c1C N1(C(=O)OC(C)(C)C)CC2CCN(C(=O)CC3CCCCCC3(F)F)CC2C1 C1(OC(c2cc(COC)no2)=O)CCC(C)CC1.C1(C)C(=O)N1 C=C1CCCN(C(=O)CC2(CNC(=O)C(C3CCCCC3)O)CC2)C1 c1(C(N2C(CN(C(C3CC(C)OC3=O)=O)C)CCC2)=O)cncc2c1CCC2 N1(C(C2N(C(=O)OC)CCC2)=O)CCC(O)(CCNC(C2CNC(=O)N2)=O)CC1 c1(C(N(CCN(C)C(c2cnc(S)nc2)=O)C)=O)cccc2c1COCCN2 c1(CN2CCC(CNC(c3cn(C(C)(C)C)nc3)=O)C2)cc(Br)cc(F)c1O CCC(C)CCCC(=O)NCC=CCC(=O)NC(C)(CO)C1CCCC1 N1(C(Cc2cc(C(=O)OC)sc2)=O)CCC2(CCN(C(=O)C=CSC)C2)C1 CCCC(C(=O)NCCCNC(N)=O)NC(=O)C(c1ccco1)OC C1(C(C)C)C(NC(c2coc(O)n2)=O)CCN1C(=O)COc1ccc(O)cc1 CC(C)CCC(O)C(=O)NCC1CN(C(c2ocnc2C2CC2)=O)CCC1(F)F N1(C(C2(C(C)NC(c3cc(C#N)c[nH]3)=O)CC2)=O)CCOC(C)(C)C1 C12(NC(c3c(C)cccc3C)=O)CCC(NC(C3CCOCC3)=O)(CC1)CC2 c1(SCCN(C(C(=O)NC2CCN2)=O)CC2CCCC2)ccc(Cl)cn1 n1(CC)nc(C(C)C)cc1C(=O)NCC1CCN1C(C1CCCCO1)=O C(CS(=O)(=O)CC(=O)NC1CC(CNC(=O)C(C)C(C)C)C1)OC N(C1CCCc2cccc(F)c21)C(c1ncc(Br)cn1)C c1(C(=O)NC2CCCN(C(CC3(NC(C)=O)CC3)=O)C2C)ccc2oncc2c1 CC(C)CCC(O)C(=O)N1C(C)CCC1C.n12cc(nn1)CCC1CC2C1 Cc1csc(=NCC(=O)NC(CNC(=O)CCC2CC2C)CO)[nH]1 n1(CC(N2CCCCCC(NC(C(COC)O)=O)C2)=O)ccc2cc(F)ccc12 C1(N(C(C(CC)C)=O)C)CC2CC1N(C(=O)CCCCN1CCCC1)C2 n1(CC#C)cccc1C(=O)NCCN(C(=O)C(C)Cc1ccccn1)CC(C)O c1(NC)scnc1C(=O)NCC(C)(O)CNC(=O)CNS(N)(=O)=O C#CC1(O)CC(C(=O)N(C)CC2CCCN(C(=O)C(c3cncnc3)C)C2)C1 C1(C(N)=O)CCCN(C(=O)CCCCNC(=O)CN2CC(=O)NC2=O)C1 CC1(C(=O)NCCC23CCC(C2)C(=O)N3)CC2CCC(C1)S2 c1(C(C(=O)NC2CC(CCNC(CCN(C(C)=O)C)=O)C2)(C)F)ccc(F)cc1 C(N=c1[nH]c(=NCCS(=O)(=O)CCOC)[nH]c2c1COC2)c1n(CC)ncn1 O=C1NCC2CN(C(=NCCCN3CCC3)NCCn3cc(Br)cn3)CCN12 C1(N(C(=O)C(F)=C2CCCC2)CC)CCCN(C(c2csc(C3CC3)n2)=O)CC1 CC1CC(CNC(C2CC2C2CC2)=O)CN1C(c1ncccn1)=O c1(C(=O)NC2CCN(C(c3ncn(C)n3)=O)C2)csc2ccc(C(F)(F)F)cc12 S(=O)(=O)(CCC(=O)N(CCCNC(=O)C#CC(C)(C)O)CCO)NC C(=O)(CC(C(F)F)C(C)(C)C)NC1CCC(C)N(C(c2cccc(O)c2)=O)C1 C(C(C)CN=c1cc(C2CC2)nc[nH]1)NC(C(C)C1CC1)=O c1(C(=O)NCC2CCN(C(=O)NC(=O)C(Cl)(Cl)Cl)C2)ccc(C(F)(F)F)c(Cl)c1 C(CC(F)F)(C(=O)NCC1(O)CCC(C)C1)NC(c1c(C)csn1)=O C12(NC(CN(C)C(=O)OC(C)(C)C)=O)CCC(CC1)N(C(=O)Cn1cncn1)C2 N(C(=NCC1CCCO1)N1CCC=C(c2ccco2)C1)CC(O)C(F)(F)F C1(NC(c2ccc(C(F)(F)F)s2)=O)CCN(C(=O)Cn2cccc2)C12CC2 C1(C(=O)N(CC(C)NC(c2sc(-c3ncc[nH]3)nc2C)=O)C)(OC)CS(=O)(=O)C1 c1(C(N(CC(C)N(C(=O)CCOc2ccc(F)nc2)C)C)=O)[nH]cc2c1CCC2 c1(C(C(=O)NCCOCCCn2cc(C(CSC)C)nn2)F)cccc(C)c1 Cc1ccc(C)c(N(C(=O)C(C)C(C)NC(c2cc(=N)[nH][nH]2)=O)C)c1 C1(C(C(=O)NCC(=O)OC)C)CCN(C(=O)C(C)(C)c2ccno2)C1 c1(-c2c(C(=O)NCC3CCC(CCC)CC3)n[nH]c2)ccc(S(C)(=O)=O)cc1 Cc1cccc(CCNC(C2CC(C)N2C(=O)CC2CCCC2O)=O)c1 N1(C(c2cc(O)ncn2)=O)CCN(C(=O)C(c2cccc(Cl)c2)CO)C2CCC12 N1(CC2(N(C)C)CCN(C)CC2)CCCN(Cc2nn(C)cc2I)CC1(C)C CC1=CCN(C(=O)C(C2CCCC2)NC(c2c[nH]c(=N)o2)=O)C1 C=CCC(C(=O)N(C(CNC(=O)CNC(=O)OC(C)(C)C)C1CC1)C)C(C)(C)C c1(OC)ccc(O)cc1C(=O)NCC1CCN(Cc2cncc(C)n2)C1 c1(C(=O)NC2(C(N3CC(C(=O)N(C)C)C3)=O)CCN(C)C2)ncc2ccccn12 c1(C(N2C(CCN(C(CCCCC)=O)C)CCCC2)=O)c[nH]c2cccnc12 c1(NC(COC(C)(C)CNC(C2CC3CCC2C3)=O)=O)ccc([N+](=O)[O-])[nH]1 C1(CS(=O)(=O)NC2(c3ccccc3)CC(C)(CC)C2)(C(F)(F)F)CCCCCC1 C1(NC(=O)CCn2cccn2)CCC(NC(c2cnc(C3CCC3)o2)=O)CC1 N1(C(c2cc(C(C)=O)oc2)=O)CCCCC1CN(C)C(c1ccncc1)=O C12(NC(C(COC)C)=O)CCCC1N(C(c1n[nH]c3c1CCCCC3)=O)CCC2 c1(C(=O)NCC(CC)NC(=O)C(C)SC(F)(F)F)ccc(F)cc1SC C(=O)(C1CCCc2ccnn21)NC1C(CNC(C2OCCN(C)C2)=O)CCCC1 N(C(=NCCc1ccco1)NCC(c1ccccc1)F)Cc1n(C)ncc1 N1(C(C=CC(CC)C)=O)C2CCC1CC(NC(c1cccc(Cl)c1C)=O)C2 C(C)(C)(C(=O)NCc1ccc(C(=O)NCc2ncc(C)s2)s1)NC(C)=O C(C)(CCCC(=O)N1CC(N2CC(O)C2)C1)NC(C(C)N(C(C)=O)C)=O c1(C(=O)NC2(C)CC(NC(=O)CC3C=CS(=O)(=O)C3)C2)cccnc1SC(F)F Cc1cc(C(=O)NC2(C)CC(NC(=O)C(C)C(O)C(C)C)C2)c(O)cc1F c1(C(N2C(C(=O)NC3CC(C(=O)OC)C3)C3CCC2C3)=O)ccc2[nH]ccc2c1 N1(C(CC(C=C)CC)=O)CCC(C)(C)C(CNC(C2(C)CC(O)CN2C)=O)C1 c1(C(N2CCCC2Cc2cccs2)=O)ccc(F)c(C(F)(F)F)c1Cl C1(NC(C(C)SC(F)(F)F)=O)CC2CCC1N(C(=O)Cc1ccn(C)n1)C2 n1(CC(=O)NC(CCNC(C2(C)C(C)C2)=O)(C)C)ncc2ccccc12 N1(C(c2c(CC)con2)=O)CCCCC2(C1)CN(C(=O)C(C)C(C)CC)C2 c1(C(=O)NCC(C(C)C)Nc2cccc(C(=O)OC)n2)cnc(OC)c(Cl)c1 c1(OC)cnc(C(N2CCCC2CC(=O)NCCCO)=O)c(F)c1 CCCCC(CN=c1nc(OC)cc(OC)[nH]1)NC(c1ccc2nc(O)[nH]c2n1)=O N1(CCNC(C2C(c3cncc(C)c3)C2)=O)C(=O)c2ccccc2C1=O C1(CCNC(C2CC23CCCC3)=O)CC(F)(F)CN1C(=O)C1=CSCCO1 N1(C(C)C)N=C(C(=O)NC2C=CCN(C(c3cc(O)n(C)n3)=O)C2)CCC1=O C(=O)(CCCCC(C)(C)OC)NCC(c1c(OC)cccc1)N(C)C C1(C(N(C(C)CNC(c2ccc[nH]2)=O)C)=O)CC(=O)N(C2CCC(C)CC2)C1 N1(c2sc(C(=O)OC)c(C)n2)CC2CCN(C(=O)OC(C)(C)C)C2C1 C12(C(=O)NCC3(O)CC(NC(c4ccccc4)=O)C3)CC3CC(CC1C3)C2 CCC(C)C(O)C(=O)N(C)CCOCCN(C(=O)CN1CCCC(N(C)C)C1)C N1(C(C2(NC(c3cc(C)n(C)c3)=O)CCCC2CO)=O)CCOC(C)(C2CC2)C1 c1(C(N(CC(C)NC(C2(CC=C)CCOC2)=O)C)=O)ccc(C(F)F)nc1O CC1(C(=O)NC2(C#N)CCC2)CC12CCN(C(CCC(=O)O)C(=O)O)CC2 C1(C(=O)NC2CCN(C(=O)CCOC3CCC3)CC2O)CCn2c(O)nnc2C1 N1(C(c2c(C)ncn2O)=O)CC2CCC2(CNC(c2c(F)cncc2Br)=O)C1 CCCCCCCC(=O)NCC1(NC(c2ccn(C)c(=O)c2)=O)CCCCC1 CC(CC(=O)N1CCC(CNC(=O)C(C)(C)c2ccns2)C1)C1CCCO1 c1(OC)ccccc1C(C)C(=O)NC1CC(CO)N(C(C2CC(C(N)=O)C2)=O)C1 CC1(C(=O)NCC2CC3CN(C(C4CC(O)C4)=O)CC23)C2Cc3ccccc3C12 c1(C(C(=O)NCC(=C)CCNC(=O)C=CC(=O)N(C)C)C)c(Cl)cccc1Cl Cc1[nH]c(C)c(C(=O)NCC2CCC(NC(=O)C(C)(C)C(F)F)C2)c1C c1(C(C)=O)cc(C(=O)NCC2(F)CC(NC(=O)COc3ccccc3)C2)oc1C c1(NC(C(C2N(C(C(CC)OCC)=O)CCC2)(C)C)=O)ccc(F)c(CO)c1 C1(CC(=O)NCCN(C(=O)C#CC2CC2)C)CCC2(CCOCC2)CO1 c1(N(C)Cc2nc(=N)[nH][nH]2)nc(N2CCC(n3cncn3)C2)c2ncn(C)c2n1 CC1CN(C(=O)CNc2ccccc2Cl)CC1NC(=O)CC1CC(=O)NC1=O C(=O)(C(C#N)C(C)C)N(C)CC1N(C(c2cc(C)nn2C(F)F)=O)CCC1 C(=O)(C(CCCC(C)C)N1CCC2(CC1)CC(O)C2)NC C1(C(=O)NCCC(=C)CNC(c2ccc(N3CCCC3)nn2)=O)CCS(=O)CC1 N1(C(c2cc(CC)[nH]n2)=O)CCC(NC(=O)CC(=O)NC)C1(C)C N1(C(c2cc(C)n(C(C)C)n2)=O)CCCC2(C1)CN(C(=O)CCC1CCOC1)C2 C1(NC(CCc2cn(C)nn2)=O)CN(C(C2CC23CC3)=O)CCC12CCC2 c1(C(c2nnnn2C2CCOC2)NCCC2CC(C)C2)cccc([N+](=O)[O-])c1 S(=O)(=O)(c1ccc(F)c(C)c1)NCC(C(=O)OCC)(F)C(C)C c1(C(=O)OC)cc(C)n(CC(=O)N(C)CCNC(c2nncs2)=O)n1 CC(O)CCCCCC(=O)N1CCN(C(c2cccn2C(C)C)=O)C2(CC2)C1 c1(NC2CCCC(NC(C(C(C)C)C)=O)C2)cccc(F)c1[N+](=O)[O-] c1(SCCC(=O)OC)cnc(N(C)C)nc1.n12nccc1NC2=O N1(C(c2cnc(C(C)C)n2C)=O)CCN(C(=O)C=CCN(C)C)C(CF)C1 C1(C)(C(N(C)CC2CCCCC2O)=O)CN(C(=O)CCC(CF)CF)C(C)(C)C1 c1(C(N2CCC(CN(C(c3c(C#C)cnn3C)=O)C)C2)=O)cccc2ncsc12 c1(OC)c(N2C3CCC2CC3)ncnc1C.C(=O)(CC(C)(C)C#N)NCC1C(=O)N1 C12(CNC(CNC(N)=O)=O)COC(CNC(=O)CCc3nccs3)(C1)C2 Cc1nn(CCO)c(C)c1C(=O)NCC1CCCC1NC(C1(C)CC=CCC1)=O N1(C(C2C(OC(C)=O)C2)=O)CC2C(CNC(C3CCCN3C)=O)C2C1 Cc1nncc(C(=O)NCCN(C)C(C2CNC(=O)N2)=O)c1C c1(OC)ccc(Cl)c(C(=O)NC2CC3CCC(C2)N3C(=O)CN(C)C(C)C)c1F N1(C(C2N(C(C(C)N=[N+]=[N-])=O)CC(C)CC2)=O)CCCC(C)(C#N)C1 c1(OC)ccc(F)c(C(=O)NC2(C)CCCN(C(c3cc(C(C)=O)cs3)=O)C2)c1 C12(NC(N3CCCC3=O)=O)CC1CN(C(=O)COc1ccc(Cl)cn1)C2 C(=O)(CCCCCF)N1C(CCNC(C(C)Oc2ccccc2F)=O)CCC1 C1(O)(C(=O)NC2CCN(CCC)C2)CCN(Cc2cc(OC(C)=O)ccn2)CC1 CCCCCCC(CC)C(=O)NCCCC1CCCN1C(C1CC2(CSC2)C1)=O C(C(CC)(CC)C(=O)NCc1cccnc1)NC(C1N(CC)CCC1)=O C12(CNC(C(C)C3CCC3)=O)CN(C(=O)CCc3ccc(N)cn3)CC1CCO2 c1(C(N(C(C)C)C2CC2)=O)cc(CNC(C2CCCC2F)=O)nn1C CC1(C)CC(C(N2CCSCC2CCNC(c2ccns2)=O)=O)CCO1 c1(OC)cccc(F)c1CN1CCSCC1C(=O)NCCCSC c1(C(N2C(CNC(C3CCCS(=O)(=O)N3)=O)COCC2)=O)cn2ccccc2n1 c1(CNCc2ccc(-c3cc(OC)cc(COC)c3)nc2)ccc(C)c(C#N)c1 C(=O)(CN=c1[nH]c(=NCCCSC)c2ccccc2[nH]1)N(CC)CC C1(C(N2CCCC(CNC(c3nnc(O)nc3O)=O)C2)=O)Cc2ccccc2C1 C(=O)(C1CCOc2ccccc21)N1CC(NC(c2c(C)oc(Cl)n2)=O)C(C)CC1 c1(OCC(=O)NC2CC(C)(NC(c3c(CC)oc(C)c3)=O)C2)ccc(C)cc1C c1(C(N(C2(C(=O)NCC3CC(O)C(O)C3)CC2)C)=O)ccc(O)nn1 C1(=O)CCS(=O)(=O)N1c1ccccc1.C1(C(C)=O)CCCCC1N1CCCC1=O.C1(C(=O)O)CC1 CON1CCC(C(=O)N(C2(C(=O)NCC(C)(C)C3(O)CCC3)CC2)C)CC1 c1(C(=O)NCCN(C(c2ccn(CCC)n2)=O)C2CC2)ccc(C2CC2)nc1C Cc1nc(NC(C2CCN(C(C3CCCN(C)C3)=O)C2)C)c2cc[nH]c2n1 C1(C2CCC2)(C(N2CCC(CN(C(C3C(CC)OCC3)=O)C)CC2)=O)CCC1 CC1CN(C(=O)CC2N(C(=O)CC3CCOCC3)CCC2(C)C)CCCO1 C(=O)(CCCn1cccc1)N(C(c1ccccc1)Cc1ccccc1)C(C)C c1(C(=O)NCC(C(C)C)N(C)Cc2cccc(NC)c2)cc2c(nc1N)CCC2 CC1CCCC(CCNC(=O)CC2CCCC2NC(C2CCC2)=O)C1 Cc1cc(C(=O)NCCC(C(C)C)N(C)C)ncc1F.C1CCOCC(=O)N1 c1(C(=O)Nc2ccc(C(C)N)cc2)cn2ccc(-c3ccccc3Cl)cc2n1 C(=O)(CN=c1[nH]c2ccccc2s1)N1C2CN(C(C3(C)CCOC3)=O)C(CC2)C1 N1(C(c2cc(C)c(C)s2)=O)CC2(CC(C(=O)NCC(=O)NCC3CC3)CO2)C1 N1(C(c2cccc3c2CCO3)C(=O)NCCC)CCCCC12CCOC2 C1(NC(C(C=CCCC)O)=O)CC(C)N(C(=O)C(CC)n2ccnc2)C1 c1(OCCC(=O)NCCOCC(N2CC(OC3COC3)C2)=O)ccccc1F c1(C(=O)OC)sc(N(C2CCC(NC(=O)CC3(C)CCCCC3)CC2)C)nc1Cl C1(C(=O)NCC2(NC(c3cc(C)[nH]n3)=O)CCCCC2C)CC2(C1)CC(C#N)C2 N1(C(C2CCC(C(=O)NCc3ccc(C)o3)CC2)=O)CC2CCC(C1)N2C C(CCCCCCO)NC(=O)C(C1CC1)NC(C1CC12CCCCC2)=O c1(CC)nccnc1C(=O)NC(C1CCCCC1)C(=O)NCC(O)CO c1(NCCO)cc2cccnc2s1.C12CCN(CC1O)OC2=O.c1(C)ccncc1 c1(CNCC2N(C(=O)Cc3ccc(Br)nc3)CCOC2)cccc(O)c1O Cc1cccc(Cl)c1C(=O)NC1CCN(C(c2cc(Cl)nnc2Cl)=O)CC1F N1(C(c2cnc(C3CCOC3)s2)=O)CCN2CC3(CC3)CC2C1 CCC(CC(=O)N1CC(C(C)NC(C2CC(O)CN2C(N)=O)=O)C1)OC Cc1cc(=O)oc(C)c1C(N1CC2CC2(NC(C2CCCN2S(C)(=O)=O)=O)C1)=O c1(CC(N2CC(N(C(C3C(CCC)CCC3)=O)C)C2)=O)c(C)nc(CC)nc1C c1(C(=O)NCCC2CCCN(C(c3cn(C)nc3)=O)C2)cc(N)c(Cl)c(O)c1 C(N=c1nc2c(c[nH]1)COC2)C1(CNC(C2CCC(C)C2)=O)CC1 c1(C(=O)NC(CN(C(CC=C)=O)C)CC)cc(Br)ccc1C N#CC1(C(N2C3CCC2C(CNC(c2sccc2C2CC2)=O)C3)=O)CCOCC1 c1(C(=O)NCC(CNC(C(C=C)O)=O)C)c(F)c(C)cc(N)c1F c1(NC(C2C(O)CCN(Cc3c(OC)ccc(Br)n3)C2)=O)c(O)cccc1C#N c1(OC)ccc(C(=O)NCC23CC2CN(C(=O)CN2CCC(C)C2)C3)cn1 C1(NC(c2nc(SC)sc2)=O)CN(C(C2CCOC(C)(C)C2)=O)CC1(C)C c1(C(=O)NC(C)C(C)NC(c2cc(O)cc(Cl)c2)=O)ccc2nccn2c1 C12(C(N3C(C(C)(C)NC(CCC=CC(C)C)=O)CCC3)=O)CCC(N=[N+]=[N-])C1C2 N1(C(CSc2nc(C)[nH]n2)=O)C2CCC1CC(CNC(C1CCCS1)=O)C2 C(=O)(C#CC1(C(F)(F)F)CC1)NC1CCCN(C(c2cc(C)sc2C)=O)C1 C1(CNC(CC(=O)NCC)=O)CCC12CN(C(=O)CC(c1c(C)noc1C)C)C2 C1(CC(=O)NC(C2CN(C(C(C)Cc3ccco3)=O)C2)C)CC=CCN1C c1(C(=O)NCCC2CCC(NC(c3c[nH]c(=NC)o3)=O)C2)[nH]nc2ncccc12 Nc1cc(F)c(Cl)cc1C(=O)NC1CC2(C1)CC(NC(=O)C(F)=CCCF)C2 CCC(C(=O)N(C(CNC(=O)CC1CCOC1)CC)C1CC1)N(C)C N1(C(CCC=CC)=O)CC(C(=O)Nc2cc(O)ccc2C)C2(CCC2)C1 N1(CC(CC)CC)CCC2CC(C(=O)N(CC)Cc3cc(C)ccc3C)C2C1 c1(C(N(C2CCN(C(=O)C(C)c3ccon3)C2)CCC)=O)ccnn(C)c1=O c1(CN(C(c2nnn(C(C)(C)C)n2)C(=O)NCC)C)cc(Br)ccc1F c1(C(N2CCCC(F)C2)=O)cc2c(C(F)(F)F)cccc2s1 N1(C(c2cccc(C3CC3)c2)C(=O)NCC)CC(C)OC2(CCC2)C1 C(=O)(C1=NN2CCCN=C2N1)NCC1CN(C(c2cc(C)c(Cl)s2)=O)CC1(C)C Cc1nc(Cl)cc(Cl)c1C(N1CCCC1(C)C(=O)Nc1c(Br)ccc(F)c1F)=O N1(C(C2CC(=C)C2)C(=O)NCc2cccs2)CCc2cc(F)ccc2C1 Cc1cc(C(=O)NC2CC3CC2N(C(c2nc(C)oc2C)=O)C3)cc([N+](=O)[O-])c1 N1(C(=O)NC(CCOCC=C)=O)CCCN(C(=O)CSCC(=O)OC)CC1 c1(C(N2CCC(C)C(NC(=O)C3=CCS(=O)(=O)C3)C2)=O)ccc(S(N)(=O)=O)o1 C(C(=O)NC1CCOC1)(C1=CCSC1)N(N1CCCCC1)C(C)=O c1(NC(CCC)C)ncnc(N(C)Cc2c(OC)cncc2Cl)c1C c1(C(=O)OCCN2CCS(=O)(=O)CC2)ccc2c(c1)nnn2O CC(O)C(C)(C)C(=O)N1CC=CC(NC(=O)C2=CC(C)(C)C2)C1 Cc1csc(C(N2CCCCC2c2ccco2)C(=O)NCCC2CC2)c1C N1(C(c2cnc(CC)[nH]2)=O)CC2CC(NC(=O)Cc3conc3C)CC2C1 C12(NC(CCn3ncn(C)c3=O)=O)CC3CCC(C1C2)N3C(=O)CO CC(C)CC(C(=O)NCCCC1CCCC1)ONC(C1C2(CC2)C12CC2)=O N1(C(c2ccc(CC)s2)=O)CCC2(CC1)CC2C(N1CC(CO)C(CO)C1)=O c1(C(=O)NC2(C)CCC(NC(C3CN(C4CC4)C3)=O)CC2)cc2nc[nH]c2cn1 Cc1nc(C)c(C(=O)NCCC2(O)CN(C(C3CCCCN3CC(F)F)=O)C2)[nH]1 C1(C(N2C(C3(C(=O)NC(C=C)C4CC4)CC3)CCC2)=O)C2CCCCCC12 c1(CC(=O)NC2(CO)CN(C(C(COC)(C)C)=O)C2)c(N)nc(C)nc1O N1(C(CC(C)SC)=O)CC2(CCCC(CNC(=O)CCN3CCCCC3)O2)C1 C1(C(N)=O)(OCCCCCC)CCN(C(=O)N(CCC=C)CC(=O)O)CC1 N1(C(c2cn(C)nn2)C(=O)NCC2CCCO2)CCC(N2CCC(F)CC2)CC1 C=CCC(C)C(=O)N(CC(=O)NCC(C)(CO)OC)CCOC C12(NC(COCCC=C)=O)CCC(OC)C1C2.C1(=O)CCC2CC(C2)N1 C1(C(=O)NCC2N(C(CC(C)O)=O)CC2)CCCCC1c1nc[nH]n1 c1(NC(C)=O)ccc(C(N2CC(NC(c3snnc3C3CC3)=O)C3CC23)=O)nc1 Cc1cc(C(N2CCC(C)C2CNC(c2ccc(CO)nc2)=O)=O)sc1C CC(C)CCC(=O)N1CC(O)(CNC(=O)C(O)Cc2cnn(C)c2)C1 N1(C(CN(CC)CC)=O)CCN(C(=O)C(C)OC)CC1c1ccc(OC)cc1 C#CCCCC(C)C(=O)NCCC1CCN(C(=O)CN(C)C(=O)C2CC2)CC1 c1(CC)nc(-c2ccc(-c3nccn3CCO)s2)c2n1CCCC2 C1(CN(C)C(C2(C)CC2C(F)(F)F)=O)CCCCN1C(c1cc[nH]n1)=O N1(C(c2nc(C(C)=O)sc2)=O)CCC(NC(=O)C(C)CC2CCC2)C(C)(C)C1 CC1(C)CN(C(C2(C)CC2Br)=O)CC(CNC(c2ccn(C(F)F)n2)=O)O1 c1(C(=O)NC2CN(C(C(C)OCOC)=O)CC2C2CC2)ccc(Cl)cc1[N+](=O)[O-] N1(C(C2=CCN(C)C2)=O)CCC2(CC2)CC1C(=O)NCCCc1cn[nH]c1 N1(C(C2(CC#C)CC2)=O)CC2(CCN(C(=O)C(CSC)OC)CC2)C1 CCCC(C)CC(=O)N(C(C(=O)NC1CC(COCC)C1)C1CC1)C N1(C(C=CCOC)=O)CCOCC2(COCCN2C(=O)C(O)CCSC)C1 CCCCC(F)C(=O)NCC1(C)CN(C(=O)CCn2ccccc2=O)CCO1 Cc1nc(NC2CCCCC2O)cc(N(C)Cc2ccccc2Br)n1 C(CC1=CCN(C(C2(C3CC3)CC2)=O)CC1)NC(CC1CCN(C)CC1)=O CC(C)C(CC(=O)N1CCCC(NC(C2CSc3ccccc3O2)=O)C1)C(C)C CCCC(CC)C(=O)NCCN1CCN(C(C2CCCN(C(=O)OC)C2)=O)CC1 N(C1CCc2cc(CNC(=O)C(C)(C)CO)ccc21)C(C1(OCC)CC1)=O C1(CNC(CCCSC)=O)CCCC2(CN(C(=O)Cn3cnc([N+](=O)[O-])c3)C2)O1 C=C(C)C(C)(C)C(=O)NCC1CCCN(C(=O)CC2COC(C)(C)CO2)CC1 C1(CNC(c2cc(C)[nH]c2C)=O)CCC(C)CN1C(c1ncsc1C)=O C1(N(C(CC=C(C)C)=O)C)CN(C(=O)CN(C)C(=O)OC(C)(C)C)CC1(C)C N1(CC(=O)NC2CCCN(C(C3C4CCCC34)=O)CC2F)CCc2ccccc21 c1(N2CCC(n3ccnc3)CC2)nc2c(c(=NCCCC3CC3Cl)[nH]1)COCC2 C=C1CCN(C(c2nccnc2C)=O)C(C(=O)NC(CCC)CCO)C1 CCCCC(CNC(C1(C)CCCC1C)=O)NC(=O)C1=NOCC1 c1(OC)ncnc(C(N2CCCC(NC(C3(C)CCN(C)C3=O)=O)C2)=O)c1F Cc1ccc(Cl)c(CNCC2(F)CCC(C(=O)O)C2)n1 c1(NC(c2c(NC(C)=O)ccc(Br)c2)=O)c(Br)cc(Cl)cc1Br CC(C)C(O)C(F)(F)C(=O)NCC1CN(C(=O)CN(C)C(=O)C2CC2)CC12CC2 CC1C(C(=O)Nn2cccn2)CCCN1C(=O)COCc1nc[nH]n1 C1(C(=O)NCC(C2CCCC2)OC)CCCN(c2ccc(C(N)=O)cn2)C1 CC(C)CCCCCCN(C1CCOCC1C)C1CC1 C1(C(N2CCC(CNC(C(C)OCCC#C)=O)CC2)=O)CC(C2CCCC2)C1 CC1(C)c2ccccc2CN1CC(=O)NC(c1ccccc1)=O C1(N(C(c2cncc(CC)c2)=O)C)CC2CCC1CC2.c12ocnc1C(=O)NC2 C1(N(C(=O)C(C2(O)CCCC2)F)C)CCN(C(c2cnnc(O)c2)=O)CC1 c1(C(=O)NCC(C(=O)NC(c2c[nH]ccc2=O)C)(C)N(C)C)ccc2c(c1)CC2 c1(C(=O)NCC(C)NC(=O)CSCCN(C)C)cccc2nnn(C)c12 C(=O)(C(C)(C)C(C)(C)C)NCC1CC(C)CN(C(=O)CC(C)(C)N(C)C)C1 C1(NC(=O)OC(C)(C)C)CC(C(N2CC(O)CC2C2CCCOC2)=O)CCC1O n1(CC(=O)NC2CN(C(c3c(OC(C)C)nncc3)=O)C2)ccc(=O)c(O)c1C CS(=O)(=O)C1(C(=O)NC2CN(C(C3CCCC3)=O)CC3CC23)CCC1 CC1CC(C(N2CC(CN(C)C(C3COC3)=O)C2)=O)CCS1 C(CC(C(=O)N(C)CC1CCCC2CC12)NC(c1cnc(C)s1)=O)OCC N1(C(c2ccc(N(C)C)cn2)=O)CC2CCC(NC(=O)CCNC(=O)CO)(C2)C1 C12CCCN(C1)CCS(=O)(=O)N(CCO)C2=O.c1(C2CCOCC2)ccc(Cl)cc1 CC(CCC(C)(C)C)C(=O)N1CCC(n2cc(C(C)N(C)C)nn2)C(O)C1 C1(C(N2CC(C)CC(NC(c3c(C)occ3)=O)C2)=O)CC2(C1)CC1(CC1)C2 N(C1CCCc2n[nH]cc21)C(CC(CC1CC1)NC(c1ccc(C)nn1)=O)=O C1(CC(=O)NC(C(=O)N(CC)CC)C)CCCN1C(c1cnccn1)=O C1(N(C)C)CCCCC1C(=O)NCC1(F)CN(C(=O)Cn2nnc(C3CC3)n2)C1 C1(CNC(CCCC=C)=O)CCC(C)(C)CN1C(=O)CC1CC1OC c1(C(=O)NC2CN(C(C=C(C)Cl)=O)C3(C2)CCOC3)cncc2ccc(F)cc12 C1(C(C(N2CC(CNC(C(C)n3cccn3)=O)(CO)C2)=O)O)CCS(=O)(=O)CC1 C1(C)(CNC(C=C(C)CNC(c2ccnn2C)=O)=O)CC2CCC1C2 C#CCC(CC(=O)N1CCC(O)C1C)NC(=O)CCc1nncn1C Cc1ccc(C(=O)NCCCNC(C2CCCC3(CCC3)O2)=O)cc1C#N c1(C(N2CCCC(CC=C)(NC(C3CC3CCC)=O)C2)=O)nc2ccccc2[nH]1 C1(NC(Cc2cnc(C)[nH]2)=O)CC2CCC1CN(C(C1CCCO1)=O)C2 C1(C(C)(C)CNC(C2(O)CC2(C)C)=O)CCCN(C(=O)Cc2c[nH]ccc2=O)C1 N1(C(COCCC)=O)CCN(C(=O)CCC2CCCN(C)C2)C(CC(C)(C)C)C1 C1(NC(c2cc(Cl)no2)=O)CC(C2CCN(C(=O)CN3C(=O)CNC3=O)C2)C1 c1(C(=O)NC(CC(=O)OC)C2CCCCC2)ccccc1P(=O)(CC)CC [N-]=[N+]=NC1CC(C(N2CCC(OCC(N3CCCC3C(=O)N(C)C)=O)C2)=O)C1 C1(CCCCCNC(C(CSC)OC)=O)CCN(C(=O)C(C)(O)C2CC2)CC1 c1(N2CCCCC(CNC(c3c(C)ccs3)=O)C2)ncnc2c1nnn2C(C)C N1(C(c2c(COC)scc2)=O)CCC(NC(=O)C(c2ccccc2C)C)CC1 c1(C(N2CC(NC(=O)C(F)=CCCF)C(CO)CC2)=O)cnc2c(c1)CCCO2 c1(C(=O)NC2(CCNC(C(n3cc(Cl)cn3)C)=O)CC2)ccc(O)c([N+](=O)[O-])c1 Cc1cc(F)sc1C(=O)N(C1CCCN(C(=O)C(F)(F)c2ccncc2)C1)C Cc1cc(C(C)(C)C)ccc1C(N1CC2CC2(NC(=O)C2=COCCO2)C1)=O C1(CCNC(c2ccsn2)=O)CCCN(C(c2coc(CO)c2)=O)C1 C1(C(N2CCCC(C)C2CNC(=O)CC2=CCOC2)=O)CCc2nncn2CC1 n1(CC)cnc2nc(=NCc3nnc(CO)s3)[nH]c(NCC3CC4(CC4)C3)c12 C#CCC(CC(F)F)C(=O)NCCN(c1nc(-c2ccccc2C)ns1)CC C1(NC(=O)CC2C=CCC2)CN(C(C2CCN(CC(F)F)CC2)=O)CC1C(F)F C1(C(=O)NC(C)CN(C)C(C2CNC(=O)N2)=O)CCCC2CC12 c1(CC)ccoc1C(=O)NC1CCC1NC(c1cc(COC)on1)=O Cc1cc(CN2CCNCC2C(=O)Nc2ccc(OC(F)F)cc2Cl)cc(O)n1 c1(OC)c(C(=O)NC2CC(NC(C3CN(C(C)=O)C3)=O)C2)ccc2c1CCC2 C=CC(C)(C)C(=O)NC(CNC(C1(c2cc[nH]n2)CC1)=O)CCCC N1(C(C(C)SC)=O)CCCOC(CNC(=O)Cc2ccc(NC(C)=O)cc2)C1 N1(C(CCCCC#C)=O)CC2CS(=O)(=O)CC2(CNC(=O)Cc2cnoc2)C1 n1(CC)cc(CC(N2CCC(NC(c3cnnn3C3CC3)=O)C2)=O)nn1 c1(C(N2C(CNC(c3c(C)nc(CCC)o3)=O)C(C)CC2)=O)ccc(F)nc1F N1(C(C(COC)NC(C)=O)=O)CCCC2(CCN(C(c3ccncn3)=O)C2)C1 c1(C2CCN(c3nnc(CCC)n3CC)CC2)cc(O)nc(C)n1 C1(C(=O)Nc2cc(OCC)ncn2)CCCN(C(C2CCCC23CC3)=O)CC1 CC1CCn2ncc(C(N3CC(O)(CCNC(c4ocnc4C4CC4)=O)C3)=O)c2C1 N1(C(CC2(OC)CCC2)=O)CCC(C(N2CCSCC2)=O)C12CCC2 CS(=O)(=O)C1(C(c2cccs2)OCCO)CCCC1.C12CCCN(C1)C(=O)OC2=O Cc1cccc(C(=O)N(C)CC2(O)CCN(C(C3CCC(C)CC3)=O)CC2)c1O N1(C(CC2(NC(C)=O)COC2)=O)CCC2CCC12.C12(CC1)C(=O)N2 Cn1ccc2cccc(CN3CCC(C#N)(NC(c4cc(I)ccc4Br)=O)C3)c12 c1(C(N(C(C)CCNC(=O)CCc2nc(O)n[nH]2)C)=O)ccccc1O C1(C(=O)Nc2cc(C)sc2C)(C)CC2CCC1CC2.C(=O)(NC1CC1)N Cc1cc2cc(C(N3CCN(C(C4CCC=CCC4)=O)CC3C)=O)oc2cc1C O=C(C1=CC2(CNC2)OC1)Nc1ccc(C(F)(F)F)c(Cl)c1 c1(C(=O)OC)ccnc(N(C(Cc2ccc(O)cc2)C(N)=O)C)c1I Cc1ccc(C=CC(N2CCC(=CC(=O)Nc3ncc(F)cc3Br)CC2)=O)cc1 C(CCCCC(=O)N1CCC1CC(C)(C)C)N(C(c1cn(CC=C)nc1)=O)C C(=O)(CC(C)(C)n1cc(-c2cc(C(=O)O)cs2)nn1)NC(C)C c1(CC(=O)N(CC)CC2CCN(C(C3(O)CCOC3)=O)C2)cccc(C(N)=O)c1 C1(CC)CNC(=O)CN1C(=O)C(C)(C1CC1)N(C(=O)C(C)n1ccnc1)C N1(Cc2c(C(=O)OCC)ccs2)CCC2CN(C(c3sccc3C)=O)CCC12 C1(CC=C)(C(=O)N(C(C)C(C)SC)C)CN(C(C23CSCC2C3)=O)C1 c1(C(=O)NCCC(=C)CNC(C2(O)CC2)=O)cncc(C(C)(C)C)c1 C=CCC(F)(F)C(=O)NCCC1CCCN(C(=O)C(C)C(C)(F)F)C1 CC1(C)CCC2(CC1)CC2NC(N1CCOC(C(F)(F)F)(C(=O)O)C1)=O CCC1=C(C(=O)NCCC2CCCCN2C(c2ccn(C)n2)=O)SCCO1 Cc1c(C(=O)NCC2(NC(C3COCCN3C)=O)CCC2)nn(C)c1N C(=O)(CC(C)(c1cccs1)N(C)C)NCC1N(C(CCC2C(C)C2)=O)CC1 C1(NC(C2COC3(C2)CN(C(=O)COCCO)C3)=O)CCc2ccccc2C1 C=CC1(C(=O)NC(C)CC(C)NC(C2CCC(CO)CC2)=O)CCOCC1 c1(CNC(C2(C(C)C)N(C(CC(=O)OC)=O)CCC2)=O)cn(C)nc1C(N)=O C=CCC(C)(C)C(=O)N1CCC(CNC(c2ccc(C(C)(C)C)[nH]2)=O)(OC)CC1 Cc1cc(C(=O)NCCCCC(C)NC(=O)CC(C)c2ccccc2)ccc1O C(C(=O)Nn1nnc(C)c1C)N(CCN1C(=O)CC(C(=O)OC)C1)C1CC1 C(=O)(CC(C)C(C)C(C)C)NCCNC(c1c(SCC)cc(Br)cc1)=O C1(NC(C(C)CN(C)C)=O)CC=C(C(=O)NCCc2cccc(O)n2)C1 c1(-c2nc(-c3ncc(N)nc3)nn2CC2CCCO2)cc2c(F)cccc2[nH]1 N1(C(=O)CC2=CCCCC2)CC2C3CCC(C2C1)N(C(=O)CNS(=O)(=O)C1CC1)C3 N1(C(C2N(CC)CC2)=O)CC(C)(C)CC1CNC(=O)Cc1c(C)cccc1F N1(C(=O)Cc2ccncn2)CCC(F)(C(=O)NC2(C(O)CO)CCC2)CC1 CC(C)(C(=O)NCC(=C1CN(C(c2coc(O)n2)=O)C1)F)C1(C)CC1(F)F c1(OC)ncc(C)c(C(=O)NCC(C)CNC(C2CC(=O)N(C)C2)=O)c1Cl c1(CN(CCNC(c2cc(OC)c(O)c(I)c2)=O)CC)c[nH]c2cc(F)ccc12 C1(C)(C(N(C(C2CCCO2)C)C)=O)CN(C(C23CSCC2C3)=O)C1 C1(C(=O)NCCN(CCCCCC)C(=O)CC(=O)OCC)CCN(C(C)C)CC1 c1(C(N2C(C(C)NC(c3cnoc3-c3ccoc3)=O)CCC2)=O)c(Cl)cnn1C N1(CCC(=O)N(CCC)CCNC(=O)C(C2CCC2)OCC)CCCS1(=O)=O C1(C)(CNC(CC2C(OC)COCC2)=O)CCN(C(=O)C(F)C(C)C)CC1 N1(C(C2CC(NC(COC)=O)C23CCC3)=O)CCCC(C)(C)CC1 C1(COC)(NC(c2cc(C)ccc2Cl)=O)CCCN(C(C23CC(C2)C3)=O)C1 CN(C)NC(=O)CCC(=O)NC1(C(=O)NC2CC(c3ncc[nH]3)C2)CC(F)(F)C1 Nc1cc2c(cc1C(=O)NCC1CN(C(=O)CNC=O)CC13CCC3)CCC2 N1(C(C(CC)C#N)=O)CCCC(O)(CNC(c2cnc(-c3cnn(C)c3)s2)=O)C1 CC(C)C1(F)CNC(=O)C2(CC2)CNC1=O.C1(CO)(CC2CC2)CC1 C1(NC(c2cn(CCC(C)C)nn2)=O)C2CCN(C(C3CC=CCC3)=O)C12 c1(C2CN(C(C(N3CCC(O)CC3)C)=O)C2)ncc(C2CCC2)cn1 C(C)(c1ccc(OC)cc1)=CC(N1C(C)CC(NC(CCCC)=O)C1)=O N1(C(=O)C(C2CCCCC2)O)CC2CCCC2(CNC(C23CCC(CC2)C3)=O)C1 c1(OC)[nH]c(=N)nc2sc(C(=O)NC(C)C(C)NC(=O)C=Cc3ccco3)cc12 c1(CN2CC(NC(C3CCC4(CC3)OCCO4)=O)C2)ccc2ncccc2c1 N1(C(C(CC=C)CNC(=O)C(C)(O)CCN(C)C)=O)CCCC(C)(C#N)C1 c1(C(=O)NCC(CC)NC(C2(CF)COC2)=O)cscc1S(C)(=O)=O CC(C)CC(CN=c1[nH]nc(-c2ccon2)s1)c1ccccc1 c1(CN2C(C(=O)Nc3cnc(OC)c(C)c3)CCC2)cc(C)c(F)c(F)c1 c1(NC(CN2CCN(Cc3cc(C)[nH]c3C)CC2=O)=O)ncnc2scc(C)c12 N1(C(C(C)CO)=O)CCC(C(F)(F)F)C(NC(C2(C#N)CCCOC2)=O)C1 c1(C(=O)NCC2C(CNC(C(CC(C)C)O)=O)C2)cc2c(C(F)F)nn(C)c2s1 c1(C(N2CCCC(NC(c3cnsn3)=O)CC2)=O)cc(F)c(F)cc1O C(=O)(C1CCCn2nccc21)NC(CCCC)CNC(c1cc(Cl)cs1)=O c1(C(=O)NCCN(C(C23OCC(COC)(C2)C3)=O)C(C)C)cccc(N)c1O c1(CNC(c2n(C(CC)(C)C)nnn2)(C)CCOCCBr)cncc(Br)c1C N1(C(CC2N(C)CCCC2)=O)CC2CCC1CN2C(=O)CS(N)(=O)=O CON(CCC(=O)NCCc1ccc(C)s1)C(=O)Cc1ccc(C)cc1 N1(C(N2CC(C(=O)OCc3ccccc3)C2)=O)CC2CC2(NC(=O)CC2CC2)C1 C(=O)(C1=CCc2ccccc21)NCC=CCNC(C1(OC)CCC(C)C1)=O C(=O)(C(N=[N+]=[N-])C(C)C)N1CC(F)CC(NC(C(CC)COC)=O)C1 CC(CC(=O)NC1CC2C1CCN2C(c1nncs1)=O)C(F)F c1(CC)cnoc1C(=O)NCC(C)C(=O)N(C)Cc1ccnn1C C(=O)(CC(C)C(C)C)N1CC(CC#C)(C(=O)N(C)CCOC(C)=O)C1 N1(C(CN(C(C)=O)C)=O)CCC2(COC(CNC(c3ncc(Cl)cc3F)=O)C2)C1 N1(C(C(C2(C)CC2)NC(CCOCCC)=O)=O)CC(C2CC2(F)F)C1 C1(CNC(c2c(COC)ccs2)=O)(NC(c2cc(F)n(C)n2)=O)CCCCC1C c1(C(C)C)ccc(Cl)cc1C(=O)NCCCN(C(=O)CCCCCF)C(C)C C(=O)(CC(C)C(=O)NCC(C)CC(=O)NC(c1ccnn1C)CC)OCC CCCC(CC)C(=O)NCC1(CC(N)=O)CCN(C(=O)CC2CC(SC)C2)CC1 C(=O)(C(F)C1=CCCCC1)NC1CC(NC(C(C)N(C)C)=O)C12CCC2 c1(CN(C2CCCC2(C)C)CC)ccc2oc(=O)n(C)c2c1 c1(C(N(CCCCCNC(C(CC)CC)=O)C)=O)ccc(F)c(S(C)(=O)=O)c1 C1(C(=O)NCc2cc(Br)cs2)CC(O)CN1C(=O)CCCc1ccc(Br)cc1 Cc1ccc(OCCCCC(=O)N2CCCC(C(=O)NCc3nn[nH]n3)C2)cc1 c1(OC)c(CSc2nnnn2-c2ccc(F)cc2F)cccc1Cl CCC(C)CCC(=O)NC1CN(C(=O)Cc2cnn(C(C)C)c2)CC1C Nc1nccnc1C(=O)NCC(CC1CC1)C(=O)NC1CCN(C(N)=O)C1 c1(NC(=O)COCC2N(Cc3c(OC)nccc3)CCCC2)cc(C)ccc1Cl C12(C(=O)NCC(COC)NC(=O)CC3(COC)CC3)CCC(CC1)CC2 N1(C(C2C(CC)C2)=O)CCOCC1CCNC(c1n[nH]c(COC)c1Cl)=O C1(O)(CCNC(C2CCC(=O)C2)=O)CCCN(C(C2(c3cc[nH]n3)CC2)=O)C1 Cc1nc(C(=O)NC(C2CCCN(C(c3cc(Cl)cnn3)=O)C2)C)c(C)s1 N1(C(c2n(CC)ncc2)=O)CCCC(NC(=O)CS(N)(=O)=O)C1C c1(OC)ccc(CC(N2CC3C(NC(=O)CC4CCCN4C)C3C2)=O)cn1 N1(C(c2c(C)nsc2)=O)CCCN(C(=O)C2=CCOCC2)CC1C c1(C(=O)NCC(C(C)C)NC(=O)C2=CCCS2)cnc2n1C(C)CCC2 C(=O)(C(F)CCC(C)C)N1CC(CC(=O)NCC)OCC1 C1(NC(CC=CCC)=O)C(C)CN(C(c2cccc3cnsc23)=O)CC1C CCCC(CC)C(=O)N1CCC(N(C)C(c2cc(-c3ccccc3C)on2)=O)C1 c1(C(=O)NCC23CC(NC(C(C(=O)OC)C)=O)(C2)C3)cccc2c1COCC2 C(CCc1ccccc1)(C(=O)O)NC(Cc1cn(CCOC)nc1)=O c1(C(=O)NCC(CC)NC(=O)Cc2ccoc2)cc(C(N)=O)cn1C N#Cc1cc(F)c(NC2CCCN(C(=O)Cn3ncnn3)C2)c([N+](=O)[O-])c1 c1(C(N(C)CCN(C)C(C2CC=CCC2)=O)=O)cc(F)ccc1F CCCC(O)CC(=O)N1CC(NC(C23CC(CC)(CO2)C3)=O)CCC1C CC(C)C(C(=O)N1CCC(C(=O)NCC2CNC(=O)C2)O1)NC(N)=O C1(OC(C)C)CCN(C(c2nc(Cl)cs2)C(=O)NC(C)(C)C)C1 N1(C(c2c(CC)nn[nH]2)=O)CCC(CNC(C2CC(=C3CCC3)C2)=O)C(C)C1 C1(NC(CC(C)(C)SC)=O)CCC(O)CN(C(C2C(C)C2(F)F)=O)C1 Cc1c(C(=O)NCC(C)(C)CNC(c2ccon2)=O)csc1Br c1(C(N(CCC)CCNC(C2CC3CC2C3)=O)=O)ccc(SC2CCC2)cc1 N1(C(c2ncn(C)c(=O)c2)=O)CC2CCC1CN2C(C1OCCC1(C)C)=O c1(C(=O)NCCN(CCCC2CCOC2)CC)csnc1Cl N#Cc1c[nH]c2ccc(C(=O)NCCN3CCNC3=O)cc12.N12CCSC(C1)C2=O N1(C(CCCCCN(C(C(C)c2ccco2)=O)C)=O)CCOCC(C)(C)C1 N1(C(CN2CC(CC)C2)=O)CCC2(NC(=O)CCc3ccon3)CCCCCC12 Cc1ccc(F)cc1C(=O)NCC1CCN1C(c1scnc1Cl)=O c1(C(=O)NC2CN(C(C(CC)O)=O)CC2(C)C)c[nH]c2cc(F)c(F)cc12 c1(C2C(NC(C(N3CCC(C(C(=O)OCC)F)C3)=O)=O)C2)ccc(F)c(Cl)c1 C1(C(CC)CC)CC(NC(=O)NC2CC(=O)N(c3ccc(OC)cc3)C2)CCO1 C(C)(C(=O)NCC1CCN(C(c2ccno2)=O)C12CC2)(C(C)C)NC(C)=O N1(C(c2ccc(OC)cn2)=O)CC(C(=O)NCc2csc(O)n2)C2(CC2)C1 N1(C(COCCOC)=O)CCC(C)CC1CNC(C1CCCCCN1C)=O c1(SC)ccc(CC(N2CC(OC)CC2CNC(=O)COC(F)(F)F)=O)cc1 c1(OC)ccc(C)c(C(N2CCC(C)N(C(=O)C(O)CSC)CC2)=O)c1N C1(NC(c2cn(C)[nH]c2=N)=O)C2CCCN(C(c3csnn3)=O)C2C1(C)C c1(C(N2CCN(C(c3c(O)ccc(Cl)c3F)=O)CC2)=O)cnc2ccccc2c1 c1(CC)ccc(-n2ccc(-c3cccc(C4(C#N)CC4)c3)n2)cc1 Cc1ccccc1C=CCNC(N1CCCC1c1cccc(F)c1F)=O N1(C(C(c2cccc(Cl)c2)C)=O)CC2C(CNC(=O)CC3(CO)CCC3)C2C1 Cc1c(C(N2CCOCC2CCNC(=O)C=CC2CC2)=O)cc(C2CC2)n1C C12(CC(=O)N(C3CCCCC3NC(c3c[nH]nc3C(F)F)=O)C)COCC(C1)C2 C1(C)(CC(=O)NCCSCC(C)C)CCN(C(c2ncnn2C)=O)C1 C1(NC(C=Cc2cncc(OC)c2)=O)CN(C(=O)CCC(C)C)CCC1(C)C CCCCN=C(NCC(=O)NCC1CC1)NCC1(C)CCC(=O)N1 C#Cc1ccc(C(=O)NCc2ccnc(C(=O)NCC=C(C)C3CC3)c2)cc1C c1(N2CCC(C(C)NC(=O)CN3CCCC3=O)C2)nc2ccc(Br)cc2o1 Cc1c(C(=O)NC(CNC(c2cc([N+](=O)[O-])n[nH]2)=O)CO)sc2ccc(F)cc12 Cc1cc(C(=O)NC(C)C(CO)NC(=O)CC2CC2)c(C)n1-c1ncccn1 C1(NC(COCC(C)C)=O)CN(C(c2ncsc2Br)=O)CC1C N1(C(CSCCOC)=O)CCC1CC(=O)NCCC(CCO)C1CCCC1 Cc1cn2cc(C(N3CCC(c4cc(C)[nH]n4)C3)=O)cc2c(C)n1 C1(NC(c2c(C)csn2)=O)CC2CC1CN(C(=O)CN(CC(C)(C)C)C)C2 C1(CC(N2C(CNC(c3cc4ccncc4[nH]3)=O)CC2)=O)CCn2cncc2C1 c1(C(NOCC(N2CC(C(=O)O)C2)=O)=O)noc2cc(Br)ccc12.CC(C)COC(F)F O(C1CCCc2ccccc21)CC(=O)NC1(CCNC(C2CCC2)=O)CCCC1 c1(N(C)CC2CCCN(C(C(CC=C)(C)C)=O)C2)nnc(C)c(C)c1C#N CCC(CC)(CO)C(=O)NCc1cn(CC(=O)NCC2CCC3(CC2)CC3)nn1 N1(C(C2(C)ON=C(C)C2)=O)CCC2(CC1)CC(NC(C1CC1CN(C)C)=O)C2 O=C(CCC[N+](=O)[O-])NCC1CCCC1NC(c1cc(Cl)ccc1F)=O C1(OC)CCCC(C(=O)N(C)CCNC(=O)C(C)(C)c2ccnn2C)C1 c1(-c2c[nH]c(=NC)s2)ccc(NC(C)CC(C)=O)c(OC)c1 C(=O)(C(C)(C)CCCNC(C1CCOC(C)(C)C1)=O)NC(COC)C(=O)OC C1(CC(=O)NCC(CNC(C2CC(CC)(CC)C2)=O)O)NC(=O)CNC1=O Cc1cc(C(=O)NCC2(O)CCN(C(C34CC5CC3C4C5O)=O)C2)cc(=O)n1C C1(NC(C(Br)=C(C)C)=O)CN(C(=O)CSc2ccc(C)cc2)CC2CC12 c1(CCC)ccc(N)c(C(=O)N(CCC)CCNC(C2CCCN2CC)=O)c1 N1(C(C2N(C=O)CCC2)=O)CC2(C1)CN(C(c1ccc(-n3cncn3)nc1)=O)C2 CC(C)CCC(C(=O)N1CCC(C)(CO)C1)NC(=O)C(=O)CC(C)C N1(CC(=O)NC2CN(C(C(C3CCC(=O)N3)C)=O)CC2C)C(=O)C(C)C(C)C1=O C(=O)(C1=CCCCCC1)NC(C(=O)N1CC(CCC)OCC1)CCCOC N1(C(C(COCC)n2cc(CN)nn2)=O)CCC(n2cccn2)CC1 C1(C(N(CCNC(Cc2cc(C)ns2)=O)C(C)C)=O)C(F)(F)C12CCC2 C1(COC)(CNC(=O)CC(C)SC)CN(C(=O)CCCN(C)C(C)=O)C1 c1(CCC(=O)NC2CC(NC(CC(C)c3ccco3)=O)C2)ccc(F)cc1F N1(C(c2nc(CC)sc2)=O)CCC(O)(C(C)CNC(c2cnc(Cl)[nH]2)=O)C1 c1(OC)ccc2[nH]cc(C(=O)NC3CCC(NC(=O)C(C)(F)F)C3)c2n1 N1(C(c2nn(CC)c(C3CC3)c2)=O)CC2(CCCN(C(=O)C(N)=O)C2)C1 c1(CCNC(c2coc(CNC(C3CCC4CC34)=O)c2)=O)cccc(F)c1 C(CCC(O)CO)N(C)C(C1C=CCN(C(c2cc(F)c[nH]2)=O)C1)=O C(CCC(C(=O)N1CC2CC1CN2C(C)C)NC(=O)CCc1cnn[nH]1)OC N1(C(C2CC(C(=O)OC)C2)=O)CCCCC1CN(C)C(C1COCCO1)=O c1(CNC(C2C(CC)C2)=O)ccc2c(c1)CCN(C(c1c(C)cncc1F)=O)C2 CN1CC(C(=O)NCCC2CCCNC2)c2ccccc2C1=O C1(CC)CN(C(C)=O)CCC1NC(c1conc1CSc1ccccc1)=O N1(C(C2CCC(C(C)C)CC2)=O)CC2=C(C1)CN(C(c1cccc(N)n1)=O)C2 C=CCCC(F)(F)C(=O)N1CC2CCC2(CCNC(=O)CCc2cnc(O)[nH]2)C1 C12(CNC(C(CNC(C)=O)(C)C)=O)CC(CO1)N(c1nccnc1F)C2 C(=O)(CC(COC)NC(=O)CC1CCC(C)(C)C1)N(C(C)C(=O)OC)CC Cc1onc(C2CC2)c1C(=O)NC(C)C(C)NC(=O)C=Cc1cc[nH]c1 C1(NC(CCCc2onc(CCC)n2)=O)CC(C)N(C(=O)CCC=C(C)C)C1 N1(c2ccc(-c3sccc3)nn2)CCCC(O)(C2CC2)C1 C1(CNC(CCS(C)=O)=O)CC2CCC1N2C(C1(c2ccc(F)cn2)CC1)=O C1(C=O)CCCCN1C(c1ccoc1)=O.C1(NC(C(=O)OCC)C)(CF)CCC1 c1(NCc2c(OCC)nccc2)cc(=NCC(C)c2cc(F)cc(F)c2)[nH]cn1 N1(C(CCOC(C)=O)=O)CC(F)CC1CN(C)C(C1CC1c1ccccc1Cl)=O CC1(C)CC(C(=O)NCC2CC3(C2)CC(O)C3)CN(C(=O)C(C)(C)N(C)C)C1 C=C(C)C1OCCC1C(=O)NCC1(NC(=O)C(n2nccc2C)C)CCOCC1 c1(C(=O)NCC(CNC(C(CSC)OC)=O)C)ccn2c1CS(=O)(=O)CC2 C1(C(=O)NCc2nnc(C)o2)CCN(C(c2cnc(Cl)n2C)=O)CC1O C1(S(N)(=O)=O)(C(N2CC(COCC)C(NC(C3(CC4CC4)CC3)=O)C2)=O)CCC1 C1(C(N2CCC(C(N3C(C#C)CCC3)=O)(C(C)C)C2)=O)CCC2(CC1)CC2 CCC(CC)CCC(=O)NCC(C1CC1)NC(c1ccc(F)c(F)c1N)=O C1(C2(NC(CNC(CCC)=O)=O)CC2)CCCN1C(=O)C(c1csc(=N)[nH]1)=O C1(N(C(c2ccncc2C)=O)CC)CCCN(C(c2cc(Cl)no2)=O)CC1 c1(OC)cccc2c1CN(C(=O)C(c1cccc(Br)c1)O)C2.C12CC(C1)NC2=O C1(CNC(COCC#C)=O)CC(C)N(C(=O)Cc2ccccc2O)C1 c1(CC(=O)NC2CCCN(C(c3nccs3)CNC(C)=O)C2)ccc(Br)cc1F C1(C(=O)NCC2(C)CCCN2C(=O)CCCC2CCC2)CC2CCCCN2C1 C(=O)(C1=C2CCN=C2NC=C1)NC(C)(C)CNC(=O)Cc1cn2ccsc2n1 Cc1cc(C(N2CCOCC2)=O)ccc1NC(c1ncc(C(C)C)o1)C C1(C2N(C(C(C=C)O)=O)CCC2)CCCN(C(=O)COC(C)C)C1 O=C1CC(C(=O)NC2CC(c3ccccc3)(CNC(=O)COC(F)(F)F)C2)CN1 C(CNC(=O)C=C1CCOCC1)(CC(F)(F)F)NC(Cn1c(C)cc(C)n1)=O C1(O)(CC#C)CC(C(=O)NC(C)CCCNC(=O)C(CC)SC)C1 Cc1cccc2c1CC(C(N1CCC(CNC(C3CCSC(C)C3)=O)C1)=O)N2 n1(C(CC(=O)NC(CNC(c2ccc(CC)o2)=O)C2CCC2)C)nc(C)cc1C c1(C(N2CCN(C(C(CSC)C)=O)C(C(F)F)C2)=O)cc2c(F)cc(F)cc2[nH]1 N1(C(C(F)=CC)=O)CC2CCCC2(NC(c2cc(=O)n(-c3ccccc3)[nH]2)=O)C1 N1(C(=O)CCN2CCCC2)CCCCC(C(=O)NC2(c3cccnc3Cl)CC2)C1 c1(C(N2C(C(C)NC(c3cscn3)=O)CCCC2)=O)nc2ccccc2cc1Cl C1(CC)CCCN(C(=O)CN(C)CC)C1C(=O)NCC1CC(O)C(O)C1 c1(CC(N2CC(CC=C)(NC(=O)C(O)C3CCCC3)C2)=O)c[nH]c2ccccc12 C1(CC)CN(C(=O)CCC#N)CCN1C(C1CC=CC1)=O CN=c1cc(C(=O)NC2(CN(C)C(C3(C4CCCO4)CCC3)=O)CC2)cc[nH]1 N1(C(c2cc(CC)on2)=O)CC(C2CC2)(C(=O)N(C2CCOC(C)C2)C)C1 c1(C(C)NC(C2CC2c2cc[nH]n2)=O)cc2ccccc2[nH]1 CN1CCCCC(C(N2CC(NC(=O)CCOC3CC3)C(F)C2)=O)C1=O N1(C(CCC(C)OC)=O)CCCCC(NC(=O)CC2CCOC2)C1 C1(C(=O)Nc2cnc(Cl)nc2)COCCC12CN(C(c1ncc[nH]1)=O)C2 c1(C(N(C2CCN(C(C3CC3C#N)=O)C2)C)=O)ccc(OC2CCCC2)cc1 S(=O)(=O)(c1cccs1)NCCC(=O)NCCNC(C=C(C)C(C)(C)C)=O C1(NC(=O)CCc2nncs2)CC(F)CN(C(c2sccc2SC(F)F)=O)C1 N1(C(CCCOC)=O)CCCC(F)(CNC(=O)CC(c2ccc(F)c(F)c2)C)C1 c1(C2(C(=O)NCCCC3N(C(C(C)NC(C)=O)=O)CCC3)CC2)ccccc1F c1(C(=O)NCC2C(CNC(C(C)SC(C)C)=O)C2)cnn(CC(F)F)c1 CN1C(=O)CCC(CNC(=O)NCCCc2ccc(Cl)s2)C1c1cnn(C)c1 Cc1c(Cl)ccc(C(N2CCN(C(c3nccc4occc34)=O)CC2C)=O)c1Cl N1(C(C(CC)SC)=O)CCC2(CC1)OCCC2NC(c1ccnc(O)c1)=O c1(C(=O)NCC2CN(C(CCC#CC)=O)C(C)(C)C2)cccc2nccn12 C1(F)(C(=O)OCC)CCCN(C)C1.C(C1C(=O)O1)OCC N1(C(C(C)(C(C)C)OC)=O)CC2(CCC(NC(=O)Cc3cnccc3C)CC2)C1 c1(C(N(C2CCN(C(c3nnn4c3CSCC4)=O)C2)C)=O)cc2ncccn2n1 C1(OC)(CNC(C2(NC(c3ccc(C)[nH]3)=O)CCOCC2)=O)CCCCC1 C1(COC)(NC(=O)C(O)C2CCC2)CCN(C(=O)C(C)(C)C)CC1 C1(CC(=O)NCC2CN(C(c3cn(C(C)C)nc3)=O)CC2C)OCCCC1(C)C C(=O)(C(F)CCC(C)C)NCCN(C(c1c(C)nc(CC)o1)=O)C CCC(C)C(O)C(C)C(=O)N(CC(=O)NCCc1cc[nH]n1)CC1CC1 N(C1CN(C(=O)C2=COCCC2)Cc2ccccc21)C(C(N1CCOCC1)C)=O c1(CC(=O)NCC2N(C(c3c(CC)cno3)=O)CCOC2)cnn2c1CCCC2 CC1CC(CNC(=O)CCCCN(C)C(C2CC(O)C2)=O)CC(C)O1 C12(NC(C(C)CO)=O)CCC(NC(c3ccncc3N)=O)(CC1)C2 C(=O)(CC(C(F)F)c1cccc(F)c1)NC1CC(NC(c2c(C)n[nH]c2C)=O)C1 Cc1c(C(N2CCN(C(=O)C(C(C)O)N(C)C)CCC2C)=O)ccc2c1CCC2 CC1CN(C(=O)CC(O)C2CCCC2)CCC1NC(C1(S(C)(=O)=O)CC1)=O CC1CC(NCc2cc(CS(=O)(=O)NC)on2)(Cc2ccccc2)C1 N1(C(C2C(COC)C2)=O)CC2OCCN(C(c3nnc(C)s3)=O)C2C1 N1(C(C(C)OCC#C)=O)CCCCC(NC(=O)CC2C(=O)N(C)N=C2C)C1 C1(NC(C2(COC)CCCO2)=O)CN(C(=O)CCc2nccn2C)CC1C c1(C(=O)NC2C(NC(c3cnc(COC)s3)=O)CC2)c(C)ncc2ccccc12 C1(CC(=O)NC2C(NC(C(COC)OC)=O)CS(=O)(=O)C2)Cc2ccccc2N1 C(=O)(C#CC(C)(C)CNC(C1CC2CC(=O)C1O2)=O)NCc1ccc(C)cc1F c1(OCC(=O)NCC(CC)(C)NC(c2cnn(C)c2F)=O)ccc(C)cc1F Cc1cccc2[nH]cc(CC(=O)NCC(C)(C)CNC(=O)CC(C)C(C)C)c12 N1(C(CC2ON=C(C)C2)=O)CCOCCC1C(N1CC(F)(CO)C1)=O c1(C(N2C(C(=O)NCc3ccc(Br)o3)CC2)=O)cccc(Cl)c1O N1(C(c2n(COC)ncc2)=O)CC2(C1)CN(C(=O)CCc1ccc(Cl)s1)C2 c1(C(=O)NCC2(CNC(C(C)OC)=O)CCC2)cc(Cl)sc1NC(C)=O c1(C(=O)NC2CC(F)(CNC(c3ccc(CC)[nH]3)=O)C2)cc2nn[nH]c2cc1F C(C(O)CCC(F)(F)F)NC(C1C(CC(C)(C)C)CN(C(=O)OC(C)(C)C)C1)=O c1(SCC)cncc(C(=O)NC(C)C(C(C)C)NC(=O)CC2CSC2)n1 N1(CC=C)C(=O)c2ccc(C(N3CCC(C4(N)COC4)CC3)=O)cc2C1=O c1(C(C)C(=O)NCCCCNC(C2CC2C(C)(F)F)=O)cccc(Br)n1 C(=O)(C1=CC2(CCOC2)C1)NCc1c(C(=O)Nc2c(OC)cccc2)cccn1 c1(C(=O)NCC(C)N(C(CC(CC=C)(C)C)=O)C)cc2cccc(C)c2s1 N1(C(CCNC(CC(C)C)=O)=O)CCCCC(CCC(=O)NC(C)C(C)O)C1 N1(C(C(c2ccccc2)N(C)CC)=O)CC(O)(CN(C)C(C2CCC(C)O2)=O)C1 c1(NC(C2(c3ccc(Cl)cc3)CC(C)C2)=O)cccc(C(C)(F)F)n1 c1(C(N2CCC(NC(C34COCC3C4)=O)C(O)C2)=O)cccc2sccc12 N1(C(C(CC)(C)C)=O)CC2CC1CN2C(=O)CNS(=O)(=O)NC CCCCC(C)C(=O)NCC1CC2CCC1N2C(c1cc(C)n(C(F)F)n1)=O C1(C(=O)NC(C(=O)N(C)C)CO)C2CCC(C2)N1C(C1CC(N=[N+]=[N-])C1)=O c1(C(=O)NCC2C3N(C(CC4(OC)CC4)=O)C(CC3)C2)cccc2oncc12 N1(C(C2C(CC)C2)=O)CCCCC12CC(NC(c1ccnn1C1CC1(F)F)=O)C2 c1(CCC)nc(C(=O)NCc2ccc(C(=O)NC(CC)C(N)=O)s2)co1 CC1CCN(C(C(=O)NCC(F)CNC(c2nc(Cl)cs2)=O)C(C)C)CC1 N1(C(C2(CC#C)CCOC2)=O)CCC(CN(C(=O)CC=C(Cl)Cl)CC)CC1 c1(-n2c(C)ncc2)ccc(C(=O)NCC(O)CNC(c2cnc(Cl)[nH]2)=O)cn1 N1(C(C2CC(C)(CC)C2)=O)CC2CC2(CNC(c2cc(C)c(C)[nH]2)=O)C1 Cc1nc(F)ccc1CNc1ccsc1C(N1CCCC(Br)C1)=O Cc1cc(NC(C2CN(C(=O)CN3CC(C)(C)C3)CC23CC3)=O)c(C)cc1F c1(OC)ccn2c(C(=O)NC3(C)CCN(C(C4OCCCO4)=O)CC3)cnc2c1 N1(C(C2=C(C)OCC2)=O)CCC2C(C1)CN2C(c1ccccc1OCC1CC1)=O N1(C(CCCc2onc(CCC)n2)=O)CC(=O)NCC1C1CCCCC1 c1(C(=O)NC(CC(C)NC(CNC(=O)NC)=O)C)cc2ccccc2s1 N1(C(CC(CCC)C)=O)CC(CNC(=O)Cc2ccnn2C)OC2(CCC2)C1 Cn1cc([N+](=O)[O-])c(C(=O)NC2CCN(C(c3cnc(S)nc3)=O)CC2O)n1 c1(C(N2C(C(=O)NC(C(C)F)C)CCCCC2)=O)ccc2[nH]nc(Cl)c2c1 N1(C(C2N(C(CCCC)=O)CSC2)=O)CC2=C(C1)CN(C(c1ccc(N)cc1Cl)=O)C2 Cc1cnc2n1CCC(C(=O)NCCC1=CCCCC1)C2 Cc1cc(Cl)cc(C(N2CCOC(CN(C)C(C3(C)CCOCC3)=O)C2)=O)c1N CC1(C)NC(=O)C2(CCN(C(C(=O)NC3CCOC3)c3cc[nH]n3)CC2)O1 C1(C2(O)CCN(C(=O)C3=C(Cl)CCC3)CC2)(NC(=O)CCCCCF)CC1 N1(C(C(C)O)=O)CCC2CC(NC(=O)C(C)(C)OC(C)C)CCC2C1 C1(C(=O)NCCCN(C(c2cnn(C(C)C)c2)=O)CC)(CC)CNC(=O)C1 C(=O)(C1=CC2(CCN(CCC(F)C3CCC3)C2)C1)C(c1cccn2nccc12)=O C1(NC(COCCC#C)=O)COCC1NC(=O)C=CC(c1ccccc1)=O N1(C(c2[nH]ccc2C2CC2)=O)CC2CC1CN2C(C12CCCC(C1)OC2)=O N1(C(c2c(C)cc(Cl)nc2)=O)CCC2C1CCCN2C(c1conc1C)=O C1(CC(=O)N(c2ccn(C(C)C)n2)C)CC(C)(C)CN1C(C1CCOC1)=O Cc1nn(C)c2ncc(C(=O)N(CC(CO)(CO)NC(c3cn[nH]c3)=O)C)cc12 N12CCCC(C1)Cn1nnnc12.C(C)(C)(C)OC(=O)OCCNCCOCC N1(C(COc2ccc(C#C)cc2)=O)CC2CCN(C(=O)C(C)CC(F)(F)F)C(C2)C1 C1(CC(=O)NCC2C(CC(=O)NC(c3cnnn3C)C)C2)CCC(=O)CC1 N1(C(C2(SCC)CCC2)=O)CC2CC(NC(=O)Cc3csc(CC)n3)C2C1 CC(O)C(C)(C)C(=O)N1CCC(C(F)C(=O)NCC(C)(C)C(C)(C)O)C1 C1(CN(C(c2ccn(CC)c2)=O)CC)NC(=O)NC1=O.C(=O)CCCOCN=C(C)C C1(C(N(CCO)CC)=O)CN(C(c2cc(Cl)cs2)=O)CC(C)O1 N1(C(C(C)OCCN(C)C)=O)CCCCC1CNC(c1cnn(CC(F)F)n1)=O NC(Cc1ccc(F)cc1)CC(=O)Nc1ccc(C(N2CC(O)C(O)C2)=O)cc1 C1(C(N(CCC(=O)NC2CN(CCC)C(=O)C2)C)=O)CCC2(CCC2)C1 CCCC(CCC)CC(=O)NCCOCCN(C(=O)C1=CCCC1C)C C(=O)(CCCC(F)F)N1CCC(F)(CNC(CNC(CCC(C)C)=O)=O)C1 C1(NC(CCCCC)=O)CN(C(c2c(C(F)(F)F)cnn2C)=O)CC1N=[N+]=[N-] c1(C(=O)NC2CCN(Cc3ncnn3-c3ccccc3)C2)cc2ccccn2c1 N1(C(c2c(C)nn[nH]2)=O)CCCCC1C1CCCN1C(c1cc(O)cc(=O)o1)=O c1(C(N2C(C(C)NC(CC3ON=C(C)C3)=O)CCC2)=O)ccc(F)c(C)c1N C1(NC(c2cc(C(N)=O)[nH]c2)=O)CCCCC1CNC(=O)COC1CCCCC1 Cc1ccc(C2CCN(CC3CCN(C)C(=O)C3)CC2)c(Cl)c1 CC(CC(N)=O)C(=O)NCC12CC(CO1)N(C(=O)CCN1CCC(O)CC1)C2 C1(c2n(CC)cnn2)CCCN(C(c2ccsc2Cl)C(=O)NCCCF)C1 N1(C(C(n2cc(C(C)N(C)C)nn2)C)=O)CCC(C(N2CCSCC2)=O)CC1 C1(NC(Cc2c(C)nccc2)=O)CN(C(c2cc(C#N)ccn2)=O)CC2(CC2)C1 C1(C(N2C(CNC(N)=O)CCC2)=O)(CO)CCN(C(c2ccon2)=O)C1 c1(C(N2CC(C)C(CNC(c3ccc(Cl)cn3)=O)CC2)=O)cccc2ccoc12 c1(C(=O)NCC(C)(C2CCC2)NC(CSCCOC)=O)coc2c1C(=O)CCC2 Cc1c(NC2CCCN(CC(N)=O)C2)ncnc1N1CCCC(C#N)C1 c1(C(N2C(CC=C)CCC2)=O)cnc2ccc(C(F)(F)F)cn12 Nc1cccc(C(F)F)c1C(N1CC=CC(NC(C2CCCC3(CC3)C2)=O)C1)=O C1(C2CCCO2)(C(N2CC(NC(c3ccc4sccc4c3)=O)C2)=O)CCCO1 C1(C(N2CCC(CCNC(C(CC#C)(C)C)=O)C2)=O)CCOC2(CCCCC2)C1 c1(CNc2c(C(=O)NCCC3CCCCCC3)n[nH]c2)cccc(Br)c1[N+](=O)[O-] c1(CNC(c2n(CCCOC)nnn2)c2cc(C3CC3)cs2)cnc(F)c(C)c1 N1(C(C2N(C)C(=O)CC2)=O)CCC(C)(C)C(C(=O)NCc2nccn2C)C1 N1(C(Cc2cccc(OCC)c2)=O)CCC2(C1)CN(C(C1C3CCCC13)=O)C2 C#CCC(CC#C)C(=O)NC1CCOCC1NC(c1cccc(CC)c1O)=O N1(CCCCC)CCC(O)C(CNC(c2c(Br)c(C)nn2-c2ccccc2)=O)C1 C1(C(C)NC(C2(CO)CCOC2)=O)CCN(C(C2CCC(=O)O2)=O)CC1 c1(C(=O)NC2(CNC(C(C)SC(F)(F)F)=O)CC2)csc([N+](=O)[O-])c1 c1(C(=O)NC2COCC2NC(C2CC23CCOCC3)=O)cc2ccccc2s1 N1(C(Cc2ccccc2)=O)CCCC1CC1CC(SC)C1 c1(NC(=O)CONC(C2CC23CCOC3)=O)ncc(F)cc1F c1(CN2CCN(C(C3(C)N(C)CC(OC)C3)=O)CC2)ncc2cc(Cl)ccn12 C(=O)(C(C)(O)C(C)(O)C(=O)O)Nc1cn(C)c(=O)cc1 n1(CCC(=O)N(c2cccc(Cl)c2C#N)C)ccc2cc(Cl)ccc12 C1(C(C)CC2CC2)C(=O)Nc2cccc(c2)N1C1CC1.C(CCOCC)NCC C#CCCC(C(=O)NCC(C)CC)NC(c1cnn2c1OCC2)=O C(C(C)(CC)C(C)O)N.C(CCCC(=O)NC1CCCC1)OCC CCC(C)CC(C(=O)N1CCC(C(=O)N(C)C)C1)NC(=O)Cc1cccnc1 C1(C(N2CC(N(C)C(c3csc(-c4ccoc4)n3)=O)C2)=O)CCCCC1(F)F Cc1nc(-c2cc[nH]n2)sc1CC(=O)NCCC1(C)CC1(F)F C1(C)(CNC(CN(C)CC)=O)CN(C(=O)CCN2CCC(N(C)C)CC2)CCO1 N1(C(C2(CC)CCC2)=O)CC2CCN(C(c3cc(C(F)F)ccn3)=O)C2C1 c12cccc(c1)OC2.C1(C(N(CCOC)CCO)=O)C(C)C1C C#CC1CN(C(=O)COC2CC=CC2)CCN1C(c1csc(O)n1)=O C(N=c1[nH]cnc(I)c1C)C1C(OC)CN(Cc2ccccc2)C1 N1(C(C2N(N=O)CCCC2)=O)CCCC2(NC(=O)CN3CCCCC3)CCCC12 C1(C(=O)NCC2(F)CC(NC(c3occc3Br)=O)C2)Cc2ccccc2O1 Cn1c(C(=O)NCC2(C)CCN(C(=O)CCc3cccnc3)C2)cnc1S CCS(=O)(=O)c1cccc(C(=O)NC(CNC(=O)C(CSC)OC)C(C)(C)C)c1 C1(CS(=O)(=O)NCc2cn(-c3ccccc3)nn2)CCCC12CC2 C1(NC(CC(C=C)C)=O)CN(C(c2cccc(=O)n2C)=O)C2(CCC2)C1 C1(N(C(C)=O)CC)CC2CC1CC2O.c12cncc(c1)-c1cn(nn1)CCCO2 N1(C(C(c2ccccc2)SC)=O)CCC(CO)(NC(c2nocc2Cl)=O)C1 c1(OC)ccc(C(=O)NC(C)CNC(C2(O)CC2(C)C)=O)c2cnccc12 C1(C(=O)NCCCC(C)=O)C2CC2CN1C(=O)CN1CCCC1=O c1(NC)ccc(C(=O)NC(CNC(=O)CCc2cccnc2)CO)cc1 CC1CCN(C(=O)CC(O)CN(C)C)CC1CNC(C1(C)COC(=O)OC1)=O C1(NC(C2OCC(C)C2)=O)C2CC1N(C(c1ccc(CO)o1)=O)C2 N1(C(C(=O)NC2C(C)(CO)CC2)=O)CCC(c2ccccc2)C(O)C1 C1(=CCNC(C2C3CCCC23)=O)CCN(C(=O)CC2CC=CC2)CC1 CC1CN(c2cc(C(F)(F)F)nc(Cl)n2)CCC1NC(=O)C(F)n1cccn1 Cc1cc(C(=O)NCC(O)CNC(=O)CC2CC3(CC3)CO2)cc(N)c1O CC(O)CC(=O)N1CC(CO)(NC(c2ccc(-c3ccncc3)s2)=O)C1 C1(CNC(=O)CSCC(F)(F)F)CCN(C(=O)CCc2ccccn2)C12CCC2 c1(-c2n(CC)ncc2)cnc2cc(C(C3CC3)NCCC(C)(C)COC)ccn12 C1(F)(CNC(=O)COCc2cccnc2)CCN(C(=O)C(C2CCOCC2)O)C1 N1(C(CC2(N(C(C3(C)C(CC)CCC3)=O)C)CC2)=O)CCCC2(CC(O)C2)C1 N1(C(CCCC)=O)CCC(NC(=O)Cn2ccc(Br)n2)C(F)C1 c1(C(=O)NCCCCCCNC(C(C(C)C)F)=O)ccc([N+](=O)[O-])cc1C(F)F c1(C(N2CC(CC=C)(NC(c3csc(CO)n3)=O)C2)=O)cc2c(F)cccc2s1 c1(NC(C2NCCN(C(C(CC)C)=O)C2)=O)cc(F)cc(F)c1Cl c1(OC)ccc(C2CCCN2C2CN(C3COC3)C2)cc1 C1(NC(C2(OC)CC2)=O)CCCCN(C(=O)CC2(O)CCCN(C)C2)C1 C1(C2CCN(C(c3cncc(Cl)c3)=O)C2)(NC(c2cnc(Cl)s2)=O)CC1 c1(C(=O)NC(CO)CF)cnc(O)n(C2CC2)c1=O N1(C(C2C(C=C)CC2)=O)CC(F)(F)CC1CCNC(C1CC(O)C1)=O C(=O)(CCS(C)(=O)=O)NC(CN(C(C1CCCS1)=O)CC)C N1(C(C2C3CC(NC(c4c(CC)cc[nH]4)=O)C(C3)C2)=O)CCCC(N=[N+]=[N-])C1 N1(C(C(C)NC(=O)Nc2cc(C)nc(C3CC3)n2)=O)c2ccccc2CC1C C=C(C)CC(C(=O)N(C(C)C(=O)NC1COC(C(F)F)C1)C)OC C1(N(C(C(C)(C2CCC2)OC)=O)C)COCC1(C)C.c12cc(on1)C(=O)NC2 CCC(C)CC(=O)NCCCN(C(C1CC2CC1C2)=O)Cc1ccccc1 c1(C(=O)NCC(C)(CC(C)C)NC(C(CCC)O)=O)cnc2cc(C)ccn12 C1(N(C(c2cc(COC)no2)=O)C)CCC(NC(=O)Cn2cnnn2)CC1 C1(NC(CSCC#C)=O)C2COCC1CN(C(=O)CCCc1cnccn1)C2 N1(C(CN(C(C)=O)C)=O)CC(NC(=O)CSCc2ncc[nH]2)C(C)(C)C1 N1(C(C(C2CCC2)OC)=O)CCC(CO)C(NC(=O)Cc2ccc(O)nc2)C1 C1(C(N(C2CC2)CC)=O)CC2CC2N1C(=O)Cc1cc(C)cs1 C(=O)(C(C)CN(C(=O)CN1CCSCC1)C)N(CC(C)O)CC N1(C(CS(C(C)C)(=O)=O)=O)CCC2(CCCC(CNC(c3ccns3)=O)O2)CC1 c1(OC)cc(Cl)ccc1CN1CCC(CO)(NC(=O)C(C)OC)CC1 C1(CNC(CC=C)=O)CC2(CCN(C(c3ccc(C(=O)C(C)C)[nH]3)=O)C2)CO1 c1(C(=O)NC(CN(C(c2c(OC)nc(Cl)cc2)=O)C)C)c(Cl)ccc(C)c1N Cc1cc(Cl)ncc1CC(N1CC(N(C(=O)CCCn2c(O)nnc2O)C)C1)=O C12(CC(=O)NC)CCC1CN(C(C1(Cl)CC1C(C)=O)=O)C2.C12CCN(C1C)C2=O CC1C(NC(=O)C=Cc2cccc(F)c2)CC2CCC1N2C(C1COC(=O)N1)=O C=CCC(C)(O)C(=O)NC1CCC(CNC(=O)CC2COCCN2C)CC1 N1(C(COCC#C)=O)CCN(C(=O)C(c2ccc(F)c(Cl)c2)C)CC1CO c1(C(=O)NC2C(CNC(C(C)SC)=O)CC2)nscc1Br C1(N(C(C=C=C(C)C)=O)C)CN(C(=O)C=Cc2ccnn2C)CCC1O CC1CC(NC(c2coc(CC3CC3)n2)=O)CN1C(=O)CC1CC(F)C1 c1(NC(C2SC3C=CC2C3)=O)cnc2n1CCC2 C(CC(C(C)(C)C)NC(c1nccnc1N)=O)N(C(C(C)CC1CCC1)=O)C c1(OC)ncnc(C)c1NC(=O)CC1(C)CCN(C(=O)Cc2ncoc2C)C1 C1(NC(c2nc(C(C)C)sc2)=O)CCN(C(c2c[nH]cc2C(C)(C)C)=O)CC1O n1(CC)cnc2c(NCCNC(C)CCOC)[nH]c(=NCCC#N)nc12 N1(C(c2n(CC)ncc2)=O)CCN(C(c2ccc(C#N)c(Cl)c2)=O)CC(CO)C1 C12(CNC(Cc3ccc(CCC)cc3)=O)CCC(CC1)N(C(=O)C(C)(C)O)C2 Cc1c(C(=O)OCC(=O)CC(C)c2ccccc2)noc1-c1ccccc1F N1(C(CC2N(C)CCCC2)=O)CCCC(F)(CNC(c2cc(CO)on2)=O)C1 N1(C(C(CC)n2cccn2)=O)CCN(C(=O)C(F)(F)Cc2ccccc2)C(C)C1 N1(C(CCNC(=O)OC)=O)Cc2ccc(CNC(c3sc(C)cc3C)=O)cc2C1 C1(CC(=O)NCCCC(C)NC(=O)CC2CCCNC(=O)C2)CCC2(CCC2)O1 N1(C(c2ncncc2Cl)=O)CCCC1C1CCCN1C(c1ccccc1CO)=O Cn1nc(C(=O)NCC(C2CCCCC2)NC(C2CC2(F)F)=O)cc1C1CC1 CC1=NNC(=O)C1CC(=O)NCCNC(=O)CC1CC=CCN1C c1(CC(=O)NCC2CCCCN(C(CSCC(C)C)=O)C2)ccc2nn[nH]c2c1 C1(NC(c2c(O)cc(C)nn2)=O)C2CC3CN(C(c4cnn(C)c4N)=O)C1C3C2 N1(C(C(CC)(C)O)=O)CCCN(S(=O)(=O)CC2CC2C(=O)OC(C)(C)C)CC1C CCCCC(C(=O)NCC1CCOC1)N1C(C)CCC1C C(C(O)CC(=O)NCC1CCC(O)CC1)NC(CCCN(C(C)C)C)=O C(c1ccc(C)cc1C)=CC(N1CC(OC)(CNC(c2ncccn2)=O)C1)=O C1(NC(c2cn(C(C)C)nc2)=O)CCC2(C(=O)NC(C)C(=O)N3CCCC3)CC12 C(=O)(C(C)(C)CC1CCOCC1)NCC1C(NC(CCOC(CC(C)C)C)=O)C1 Cn1[nH]cnc1=NC(=O)C1CC(F)CN(Cc2ccc(OC(F)(F)F)cc2Cl)C1 C1(O)(C(N(C(C)CNC(=O)CCC2CCOC2)C)=O)CCCC(C)(C)CC1 c1(C(N2CC(C)(NC(c3sccc3CO)=O)C2)=O)nccc2c[nH]nc12 Cc1nn(C)c2sc(C(=O)NCC(O)CNC(C3C4CCCOC34)=O)cc12 C1(C(=O)Nc2nc(Cl)ccc2Br)CCC2(CN(C(=O)CCc3cnc[nH]3)C2)O1 C(=O)(C(C)(C)S(C)(=O)=O)N1CCC(CN(C(c2ccc(OC)s2)=O)C)C1 N1(C(C=C(C)C2CC2)=O)CCC(CNC(c2cc(C(N)=O)[nH]n2)=O)C1 Cc1cc(C)c(C(N2CCCC(C(C)NC(c3csc(C)c3C)=O)C2)=O)c(=O)o1 C1(CCC)CN(C(=O)Cc2cc(C)no2)CCN1C(=O)C(C(C)CC)N(C)C c1(CNC(=O)NCC(c2ccccc2Cl)C(C)C)cc(=O)n(C)cn1 N1(C(c2c(C)cc(F)cn2)=O)CC2CCN(C(c3sccc3C)=O)CC2C1 c1(OCC)ccc(C(N2CCOCC(NC(=O)CC3=CCCC3)C2)=O)cc1OC C12(C(N(C(C)CCO)CCOC)=O)CC(n3cc(C(C)(C)O)nn3)C1C2 c1(SC)cc(C(=O)NCCCCCN(C)C(C23CC(C)C2C3)=O)oc1C C(CC(C)CCNC(=O)CC1CCCS1(=O)=O)NC(COCc1ncc(C)o1)=O c1(CC(=O)NCC(CO)NC(C(C)OC)=O)nnc(S)n1C N(C(=S)N1CC(CO)C(C)C1)C(c1ccccc1)C C1(NC(C(C=C)c2ccccc2)=O)(CNC(C2CCC2C(N)=O)=O)CCOCC1 N1(CCCc2c(C)nn(C)c2)CCC2(CCCC2CNC(=O)OC(C)(C)C)C1 C1(C(=O)NC2OCCN(C)C2)N(C(C2CCC3(CC3)C2)=O)CCCC1(C)C CC1(NC(=O)Cc2csc(-c3cccnc3)n2)CCCN(C(=O)C(O)C2CC2)C1 c1(C(=O)NC2CC(CNC(C3CC3Cl)=O)C2)cc(C(C2CC2)=O)on1.N1CCCCC1 c1(C(=O)NCC2CCC(NC(Cn3c(CCC)ncc3)=O)C2)ccc(C)c(N)c1 C1(C(N(C2CCN(C(c3ccoc3C3CC3)=O)C2)CC#C)=O)CCCC(=O)N1C c1(OC)cncc(C(N2CCC(CN(C)C(c3ccc(N)c(N)n3)=O)C2)=O)c1C c1(C(N(CCCNC(Cc2c(CC)con2)=O)C(C)C)=O)csc(C)c1N S(=O)(=O)(c1cc([N+](=O)[O-])cc(C)c1Cl)N(C1CCCN1CC)C(C1CCCS1)=O C1(NC(C(CSCC)NC(c2c(CCC)nco2)=O)=O)CC(C)(OC)C1(C)C C12(CNC(CC(CN(C)C)O)=O)CC(CO1)N(C(=O)COCCSC1CCC1)C2 c12ccc(cn1)NC(=O)CO2.c1(CNC(C=C(COC)C)=O)ncnn1C(C)C C(=O)(CC(C)CC(=O)N1CC(CC(N2CC3(CCC(=O)N3)C2)=O)C(C)C1)OC c1(C(CNC(c2c(CC)ccs2)=O)NC(c2c[nH]cc2CC)=O)ccccc1F c1(C(N2CCOCC2CC(c2ccccc2)O)=O)ccc2c(c1)CCO2 CCC(C(=O)N1CCCCC(CNC(c2cc(C(C)C)n(C)n2)=O)C1)C(F)(F)F c1(C(N(CCN(C(C(C)Sc2ccccc2)=O)C)C)=O)ccc(Cl)cc1C(F)F N1(C(C(CC)C)C(=O)NCC2CCOC2)CCc2ccncc2C1C CC(C)C(CNC(c1ccc(C(N)=O)[nH]1)=O)C(=O)NCC(C)(C)CC1CC1 C12CCN(CC1)C(c1cn(C(C)C)nc1C)C(=O)NC2.C(C(C)C)OC(C)=O N1(C(CC(COC)C)=O)CCCCC(N(C(=O)COc2c(C)occc2=O)C)C1 N1(C(C(C(C)C)O)=O)CCCN(C(C23C4CC(CC24)C3(F)F)=O)C(C)C1 C1(NC(C(C)NC(N)=O)=O)CN(C(c2nc3ccccc3[nH]2)=O)CC1C1CC1 C12(CC(=O)NCC(C(C)C)NC(=O)CCS(C)=O)CC3CC(C1)CC(F)(C3)C2 CC1CN(C(c2ccc([N+](=O)[O-])s2)=O)CCC1NC(C1(N(C)C)CCCCC1)=O C(=O)(CCCC(CC)CC)NC1C(NC(CC(CC=C)(C)C)=O)CCC1 C1(NC(C(C=CC)O)=O)CN(C(=O)COCc2ccc(C)cc2)CCC12CCC2 C1(CC(=O)N(CCNC(C(c2ccccc2)OC(C)=O)=O)C)CCOC1(C)C Cc1cc(C)c(S(=O)(=O)N2CCc3[nH]nc(C(N4CNC(=O)C4)=O)c3C2)c(C)c1 c1(OC)cc(C)cnc1C(N1CC2(CC2)CC1CNC(=O)CCC1CCOC1)=O c1(CN(CC(O)CO)Cc2ccc(-c3n(C)c(O)nn3)cc2)ccc(F)c(Br)c1 c1(C(N2C(CNC(CCOCC)=O)CC(F)(F)C2)=O)ccc(C#N)c(Cl)c1 N1(C(C(C)SCC)=O)CCC(NC(=O)Cn2nc(C(F)F)cc2C2CC2)C(F)C1 C(=O)(CC1=CCN(C(=O)C(C)(F)C(=O)OC)CC1)N1CCC(CC)C(F)C1 c1(CC)c(C(=O)NC(CNC(c2nn(CC)nc2C)=O)CO)cccc1F CCCCCCC(F)C(=O)N1CCC(CCNC(c2ccc(COC)s2)=O)CC1 Cc1ccc(C#N)cc1C(=O)Oc1cccc(Br)c1F c1(C(C)=O)cc(C(=O)NC2CN(C(c3cnc(S)n3C)=O)C2)ccc1O Cc1cnc(C(=O)NCC(N2CCN(C(C3SCCC3C)=O)CC2)=O)nc1 C1(NC(C2CC3C=CC2O3)=O)C=CCN(C(C23CC(C2)C(C(F)(F)F)O3)=O)C1 N1(CCN(C)CCc2n[nH]c(=N)s2)CCOCC1(C)C N1(C(C(COC)O)=O)CC2CCCC(NC(C3CN4CCN3C(C)C4)=O)C2C1 N1(C(C(CC=C)C)=O)CC2(CCC2)CC1C(N1CC(S(N)(=O)=O)C1)=O S(=O)(=O)(c1ccc(I)cc1Br)NC(C(=O)OC)Cc1nccn1C CC1ON=C(C(=O)NCC(O)CCNC(c2ccccc2NS(C)(=O)=O)=O)C1C N1(C(Cc2c(SC)cccc2)=O)CCN(C(C2COC(=O)N2C)=O)C(C)C1 c1(OC)nc(C(N2CC(NC(=O)C(N3CCNC3=O)C)CC(O)C2)=O)ncc1F CC1CN(C(=O)Cn2nnc(=O)[nH]2)CC1NC(=O)Cc1cc(Cl)sc1Cl C1(C)(C(=O)NCC2C(C)CN(C(c3c[nH]c(=O)cn3)=O)C2)CCC2CC2C1 C(=O)(C(C(C)C)n1ccnc1)NC1C(CNC(c2c(OCC)scc2)=O)C1 n1(CC)nc(C(=O)N(C2CCC(NC(=O)C(=O)NCC(F)(F)F)C2)C)cc1C N1(C(C(C)NC(CC)=O)=O)CCC2(CC1)CC(C)N(C(c1cc(F)n[nH]1)=O)C2 N1(C(C2(CC)CCC2)=O)CC2CCCC(C1)N2C(c1cnc2c(c1)CCCC2)=O c1(OC)ccc(C(C)(C)C)cc1C(=O)NC1CN(C(c2ncoc2C)=O)CC1F C1(O)(CN(C(=O)Cn2ccc(O)nc2=O)C)CCCN(C(C2CC=CCC2)=O)C1 c1(CCNC(CCSC)C(=O)NC(C)(C)C)ccc(Cl)c(C)c1 N1(C(C(C(=O)OCC)F)=O)CCCC2(NC(=O)C(C)S(C)(=O)=O)CCCC12 O=C(C1CCCn2c(Br)cnc21)N1CC(NC(C23CC(F)C2C3)=O)C1 c1(C(=O)NCCN2CCN(C(c3nccc(C)c3)=O)CC2)cccc2occc12 C(=O)(C(C#N)C(C)(C)C)N(C(C(=O)NC(C(=O)OCC)C1CC1)CC(F)F)C c1(C(N(C(C(=O)N(C(CC)C)C)C2CC2)C)=O)csc(C)c1C c1(C(N2C(C)CC(NC(=O)C(C)(C)c3nccs3)C2)=O)ccc(C(N)=O)c(Cl)c1 C1(N(C(CCOCC)=O)C)CC2CCC(C1)N2C(c1sccc1S(C)(=O)=O)=O N1(C(C2(CC=C)CCN(C(c3cocn3)=O)C2)=O)CCCC(C)(OC)C1 C1(CNC(C(C(C)C)NC(C)=O)=O)COCCN(C(c2n[nH]c(C3CC3)n2)=O)C1 S(=O)(=O)(c1ccc([N+](=O)[O-])cc1)N1CCN(C(=O)NCc2nnc(CC)s2)CC1 C(=O)(C(CO)C(C)(C)C)NC(C(C)(C)O)C(=O)NCCn1ccnc1 C(C(=O)N1CCCCCO1)C1N(CC(=O)NC(CC)(C)C)CCCC1 CCCC(CNC(=O)CCOC(C)C)C(=O)Nc1cnc(Cl)nc1 C12(C(=O)NC(CC#C)CC#C)CCCC1CCN2C(C1CC(O)CN1C)=O c1(C(=O)NCC2(NC(=O)CCn3cccn3)CCOC2)ncnc2sccc12 N(C1CCOc2cc(F)ccc21)C(C(=O)NCCSC1CC(C)(C)NCC1)=O c1(CC)nc(C(=O)NCC2C3CN(C(C4(SC)CCC4)=O)CC23)c(C)o1 C1(C)(CCCC(=O)N(C(CC)C)C(c2cnc(OC)c(C)c2)=O)NC(=O)NC1=O C(=O)(CC(C)C(C)(C)NC(C1CC12CCCC2)=O)N1C(C)(CCC)CC1 Cn1cc(Cl)c(CC(N2CC3CC3(NC(C3CC3(F)F)=O)C2)=O)n1 c1(NC(=O)OC(C)(C)C)ccc(CC(=O)N)cc1.C1C(F)(F)CC(=O)N1.C1CC1 N1(C(=O)CC2CCCC2O)CCC(C2CCCCN2)CC1 N1(C(CCSCC(C)C)=O)CCC(NC(C2CCS2(=O)=O)=O)C(F)C1 N1(C(C(c2cncnc2)C)=O)CCC(CNC(c2ncoc2-c2ccon2)=O)C1 C1(S(C)(=O)=O)(C(=O)NCC(C2CCCN2C(=O)CC2CCCCC2O)(C)C)CCC1 Cc1ccccc1-n1c(SC2CCCN(CC(CC(=O)O)SC)C2)nnc1C c1(-c2cn(CCNC(CCc3cncc(OC)c3)=O)nn2)ccc(C#N)c(F)c1 O=C(N=C1CCN(c2cccc(Cl)c2)N1)c1cc(F)ncc1Br C(=O)(CCCC(F)(F)F)NC1CC(C(N2CCC(C(C)C)CC2)=O)C12CCC2 C1(CNC(C2CC(CC)C2)=O)CN(C)CCN1C(c1cc(Cl)n[nH]1)=O c1(C(=O)NCCN(C(C2(C(C)C)CCC2)=O)C)cn2c(n1)CCC(C)C2 Cc1cc(CC(=O)NCC2(NC(C3COCC3(C)C)=O)CCCC2)ccc1O S(=O)(=O)(c1ccc(F)c(C(=O)OC)c1)N1CC2C(CNC(CC=CCC)=O)(C2)C1 N1(C(C(C2CCCOC2)OCC)=O)CCC(NC(=O)CCc2cnoc2)CC1 C1(C#N)(C(=O)NCCCCC(C)NC(=O)C(C)(C)c2ccno2)CC2(CCC2)C1 N1(C(C(N2CC(C)C2)C)=O)CC2(CC(C(=O)NCC3(C#N)CC(C)(C)C3)CO2)C1 C1(CC#C)(C(N2CCC(C)(COC)C2)=O)CCN(C(=O)C=Cc2ccc(C)o2)C1 Cc1nc(NC(=O)CC2CCN(C(=O)Cc3cccnc3Cl)C2)sc1Cl c1(C(N2CC3CCN(C(=O)CCN4CCC4)CC32)=O)cc2ccc(Cl)cc2[nH]1 Cc1cc(O)n2ncc(C(=O)NC3CCCN(C(=O)C(=O)NC4CC4)CC3)c2n1 N1(C(=O)OC(C)(C)C)CCCC(C(=O)NC(C)C(C)(C)c2ccccc2)C1CO CC1(NC(=NCC2CCCCC2)NC2CC(C)(F)C2)CCCOC1 c1(CC(=O)N(C)CC2(O)CCN(C(C(C)=C(CC)C)=O)C2)cc(F)ccc1F N(C)(C1CS(=O)(=O)c2ccccc21)C(c1cncc(OC)c1)C(=O)NCC(F)F C(=O)(C(CNC(c1cnsn1)=O)C(C)(C)C)N1CCC(OC)C1(C)C C(=O)(CC(CC1CC1)NC(=O)C(C)C1CC1)NCc1cn(C(C)C)nc1 c1(C(=O)NC2CC(C)N(C(=O)CCSc3nnnn3C)C2)ccc(N)c(Cl)c1 Nc1cc(F)ccc1C(=O)NCC(O)CNC(=O)CS(=O)(=O)NCC1CCCO1 N1(C(COCC(=C)C)=O)CCC(CO)C(NC(=O)C=Cc2nccs2)C1 c1(NC(=O)NC(CCO)C2CCCC2)ccc2ccc(O)nc2n1 N1(C(c2c(C)ccnn2)=O)CCC(C)CC1CNC(=O)COCc1nc[nH]n1 CCC1=C(C(=O)NCCC(CNC(=O)C2=CCCC2C)OC)CCCO1 C1(NC(c2ccc(SCC)nc2)=O)CCN(C(=O)Cc2cnns2)CC1O c1(C(N(CCCCNC(C2CC2c2ccccc2)=O)C)=O)cc(Br)cs1 c1(CSCC(=O)NCCCOCCNC(C2CCCS2)=O)cccs1 N1(c2n(CCC3CC(O)C(O)C3)nnn2)Cc2cnn(-c3ncccn3)c2C1 N1(C(=O)NCC2CCCSC2)CCCC(O)(c2ccccc2)CC1 N1(C(CC(C(=O)OC)C)=O)CCC2(C1)CN(C(=O)C(C)(C)C1CCCO1)C2 CCCCC(O)CCC(=O)N(CCN(C)C(c1ccc(N(C)C)cn1)=O)C(C)C c1(N(C)C)cc(CN2CC3CC3(C(=O)NCCCc3ccccc3)C2)ccn1 C1(NC(C(COC)O)=O)C=CCN(C(C2(CC3CC3)CCC2)=O)C1 c1(C(=O)NC2CC(F)(CNC(Cc3cc(C(C)C)no3)=O)C2)c(Cl)nn(C)c1Cl C1(CC(=O)NCCN(C(C)C)C(c2cc(Br)cs2)=O)CCC(C)(O)CC1 Cc1cccc(C(=O)NCC(C)N(C)C(C2CCC(C)(C)OC2)=O)c1C#N c1(C(=O)NC(C(C)NC(=O)Cc2nnn(C(C)(C)C)n2)(C)C)ncc[nH]c1=O C(CC(C)(C)CNC(C1CC(CN(C)C)C1)=O)NC(c1cc(CC)on1)=O N1(C(CC2CC(SC)C2)=O)CCCC(C(=O)NCC23CC(CCO2)C3)CC1 O=C1CC(C(F)(F)F)C(C(N2CC(NC(c3nocc3Br)=O)C2)=O)N1 c1(N2CC(CNC(c3cccc(C(=O)NC)c3)=O)C2)nc2ccc(OC)nc2s1 C1(C(=O)NCC(c2ccsc2)C)CC(O)CCN1C(=O)CCc1ncnn1C Cc1cc(=N)[nH]cc1C(N1CCCC(NC(=O)CNC(c2ccsc2)=O)C1)=O C(C(C(=O)NC1(CO)CC=CC1)C(C)(C)C)NC(CC(C)n1cccc1)=O c1(OC)ccc(C(CF)NC(C2(CF)CCN(C(=O)OC(C)(C)C)C2)=O)cc1 N1(c2cc(C)c(C#N)cn2)CCOC2(CCC(NC(=O)C3=CCC3)CC2)C1 N1(C(C)=O)CCC(C)(C(=O)NCC2CCN(C(c3sc(C)cc3OCF)=O)C2)C1 C(N=c1[nH]c(=NC2CC(C)(CO)C2)c2[nH]ccc2[nH]1)c1c(OC)c(C)ccc1 C1(CSC)(Nc2nc(Br)sc2C)CCC(C)CC1 N1(C(C2N(C)CCC2)=O)CCOC2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CC12 c1(NC(c2c[nH]nc2C(=O)NCC2CCCCO2)=O)cc(C(F)(F)F)ccn1 c1(N2CCN(C(c3sc(C)c(Br)c3)=O)C3C2C3)ncnc2cc(F)ccc12 N12CCC(CC1)C(C)(O)CNC(=O)C(=O)N(CC#C)CC2=O.C(C)(C)(C)NC(C)=O c1(C(=O)NC23CCC(NC(C(C)CC4CCC4)=O)(CC2)C3)cc2cccnc2[nH]1 N1(C(C(C=CC)O)=O)C2CCC1C(F)C(NC(c1cc(C)cc(C)c1)=O)C2 C=Cc1cnn(C)c1C(=O)NCC1CN(C(C2(c3cc[nH]n3)CCC2)=O)CC1O N1(C(c2c(OC)scc2)=O)CC2CCN(C(c3cc(C)ccc3C)=O)CC12 c1(C(=O)NCCNC(=O)Nc2scc(C(=O)NC(C)C)n2)c(Br)nnn1C Cc1nccc(Cl)c1C(N1CCN(CCN(C(=O)CCCCCF)C)CC1)=O CC1CC(CC(=O)NC23CCN(CC2)C3)CN1C(=O)CC(C)(C)C1CC1 Cc1nc(O)c(C(=O)NC2CN(C(c3ccc(CO)cc3)=O)CC2C)cc1Br c1(OCCC(C)C)ccc(CNC(C2C(C(C)NC(=O)C(C)(C)C)C2)=O)cc1 CCCS(=O)(=O)CC(=O)NC(C)CC(C)NC(c1ccc(C2CC2(F)F)cc1)=O c1(C(N(CC(=O)NC2COCC2O)CCOC)=O)ccsc1C#N CC(=O)C(C)CC(C)C(=O)NC1CCC(CNC(=O)C2=CCSC2)CC1 C1(C(N2C(COC)CN(C(=O)CC3(C#N)CC3)CC2)=O)Cc2ccccc2S1 Cc1cc[nH]c(=N)c1C(=O)NCC(CNC(c1cnn(C)c1CF)=O)C(F)(F)F C1(C2(NC(C3C(=C)CC3)=O)CC2)CCCN1C(c1nnn(C)n1)=O C(=O)(C1=CC(C)(CC(=O)OCC)C1)C(C1CC(F)(F)C1)C#C C(CN=c1[nH]c(Cl)c(C#N)s1)C1C(C)CCN(CCCCCCC(=O)N(C)C)C1 C1(CC)NC(=O)C2=C1N(c1c(F)cccc1F)C(=S)NC2c1c(C)ccnc1O Cc1cc(C(=O)NC2CC3CN(c4cc(C5CC5)ncn4)CC23)cc2nn[nH]c12 CC1OC2CCC1(C(=O)NCCC1(NC(=O)CCc3cnoc3)CCCC1)C2 N1(C(COCC#C)=O)CCCCC12CN(C(=O)C1=CS(=O)CCC1)C2 c1(CC(=O)NC2CCN(C(C3(C)CC3)=O)CC2)ccc2sccc2c1 c1(CC)nn(C)c(C(N2C3CN(Cc4cccc(C)c4C)CC23)=O)c1Br c1(OC)ccc(C(C)NC(c2nnnn2C2CCCC2)(C)CC2CCC2)c(C)n1 Cn1cc(C#N)cc1C(N1CCN(C(=O)C(O)CC(F)F)CC1CCO)=O N1(C(C(CC=CC)CC)=O)CCC2C(C1)CN2C(c1nn(C)cc1Cl)=O N1(C(CCCC(CC)NC(c2nc(C)c(C)s2)=O)=O)CCC2(CCOC2=O)C1 C1(C(C(N2CC(C(C)NC(C3C(C)(CC)C3)=O)C2)=O)F)CCC(=O)CC1 N1(C(CN(C2CC2)CC)=O)CC2CCCC2C1C(=O)NCC1CCCC(C)CC1 c1(C(N2CC(CNC(c3cc(C(CC)C)no3)=O)(OC)C2)=O)cnnc(CC)c1 [N-]=[N+]=Nc1ccc(C(N2CCOCC(F)(CNC(C3CCC3)=O)C2)=O)nc1 N1(C(c2[nH]cc(CC)n2)=O)CC2(C1)CN(C(=O)C(C(C)C)N(C)C)C2 c1(C(=O)NC2CCN(C(C3(OC)CCCC3)=O)C2)ncc(C(F)F)cn1 c1(NC(CC2(C)CN(C(c3cc(Br)ncc3Cl)=O)C2)=O)cccc2cc[nH]c12 N1(C(c2cccc(OC(C)C)c2)=O)CCCCC12CN(C(C1(F)CC1C)=O)C2 C(=O)(CC1=CCOCC1)NCCC(CNC(c1ccc(N(C)C)cc1)=O)OC CC1CN(C(C2COCCN2C(c2cccc(O)c2)=O)=O)C(C)C1C c1(C(N2CCCCC(N(C(CC=C=C)=O)C)C2)=O)cnc2n1C(C)CCC2 CCCCCC(O)C(=O)NC1CC(C(=O)NCC2(CC)CCC2)CC1O Cc1nc(Cl)[nH]c(=NC2CCCN(C(C3(C4CCC4)CCC3)=O)C2)c1Cl C#Cc1cccc(NC(=O)C(CCF)NC(C2CCCN2CCC)=O)c1 N1(CC)CCCC(C)C1CN(c1cccc(N)c1I)C(CC(OC)OC)=O N1(CC(C2CCOC2)OC)CC(N(C)C)C(C)(C)C1 c1(C(=O)NC2CC(O)(CNC(C=COCC)=O)C2)cc(CC)c(C)s1 c1(NCC(=O)NC(CNC(C(COC)C)=O)C2CCC2)cccc2ccccc12 C1(N(C(C(C)N(C(CCC(C)SC)=O)C)=O)C)CCCC(C)C1C C1(CNC(c2c(CC)cns2)=O)CN(C(=O)Cc2cc(C)cs2)CC1(F)F c1(C(=O)NC2CCC(NC(c3n(CC)nnc3C)=O)C2)cccc(Cl)c1F C1(NC(c2c(CC)nc(C)o2)=O)CCC2CC1CN2C(c1ccncc1Cl)=O CC1=C(C(=O)N2CC(CNC(c3cn[nH]c3)=O)C(F)(F)C2)Cc2ccccc2O1 C1(Nc2nnc(C)c(C)n2)CCN(C(=O)Cc2cc(C3CC3)on2)CC1(C)C c1(NCc2ccc(N)c(Cl)c2)ccc(S(=O)(=O)N2CCC3CC3C2)c(Br)c1 c1(OC(C2CCCN(C(c3cncn(C)c3=O)=O)C2=O)=O)cn2ccncc2n1 C1(CNC(=O)CC2CCOC2)CC2CCC1N(C(=O)Cc1sc(O)nc1O)C2 c1(C(=O)NCC(CN(C(C(CC#C)O)=O)C)O)c(F)ccc(Br)c1F N1(C(C=C(CC)CC)=O)CC(OC)CC1CNC(c1cn(C2CCC2)nc1C)=O C1(O)(C(N2CCC(C(C(=O)NCc3ncc(C)s3)C)C2)=O)CCOCC1 CP(C)(=O)c1ccc(C(=O)NC23CC2CN(C(C2CC24CCOCC4)=O)C3)nc1 Cn1nnc2cncc(C(=O)NCCOCCCNC(C3(F)CCCC3)=O)c12 c1(CC)oc(C)cc1C(N1CC(O)(CNC(=O)CC2CSCCO2)C1)=O N1(C(C2(C)CCOC2)=O)CCC2(CCC2)C(NC(=O)Cc2ccsc2)C1 C(=O)(C#CC1CCCOC1)N(C1COC2(C1)CN(C(=O)CCOCC(F)F)C2)C C(=O)(CC(F)(F)C(=O)O)N1CCCC(CCNC(c2cn3cccnc3n2)=O)C1 CC1(NC(c2cnc(N)c(CO)c2)=O)CCN(C(=O)C=CC2CCCO2)CC1 C#CCCCCCCCC(=O)N1CCC2(CCC2)C(NC(=O)C=CBr)C1 C1(NC(c2cc(C)nn2CCO)=O)CC2CCC1CN(C(=O)CCC(F)(F)F)C2 C=CCCC(CC(C)C)C(=O)N1CCC(F)(CNC(C2(CC(F)F)CC2)=O)C1 N1(C(C(CSC)OC)=O)CCCC(O)(CNC(c2ncnc(O)c2F)=O)C1 c1(C(=O)NCCOCCN(C)C(c2ccc(C#N)s2)=O)cnc2c(c1)CNC2=O c12ccc(cc1)CC(=O)N2.c1(C(COC)N(C)C)cnn(C)c1 c1(C(=O)NC(CN(C(c2cc(C)ncc2C)=O)C)C)cc2c(C)ccc(C)c2[nH]1 c1(C(=O)NC2C(NC(CN(C(=O)OC)C)=O)CCC2)c(C)ccc2n[nH]cc12 C1(NC(C(C)(C)OCC)=O)CCCC12CCN(C(C1CC1C1CCCC1)=O)CC2 N1(C(C2CC(C)CN2C(=O)CCN2CCN(C)CC2)=O)CC2C3CCC(C3)C12 CC(C)C(CNC(=O)C(C1CCCCC1)C)C(=O)N1CCCCC1CC(N)=O C1(C(=O)NC23CC(CNC(CCCOCC=C)=O)(C2)C3)CCCC(F)(F)C1 c1(OC)ncc(NC(C2(C)CCN2C(=O)COC2CCCC2)=O)cc1C C1(NC(c2c(C)onc2-c2ccccc2F)=O)CCCCN(C(=O)C2CC2)C1 n1(CC(=O)NCCC2(OC)CN(C(=O)C(O)C(C)C)C2)c(C)c(C)sc1=O c1(C(=O)OC)cc(NC(=O)NCc2ccc(-c3cnco3)cc2)c(Cl)c(Cl)c1 N1(C(c2c(C)cnc(F)c2)=O)CCC2CN(C(=O)C(C)(C)NS(C)(=O)=O)CC12 CC1CCCCN1CC(=O)NCCC(=O)NCCc1ccc(F)cc1 C(=O)(CCCS(=O)(=O)N1CCCC1)NC1C(C)N(C(=O)CN2CCCC2C)CC1 c1(OC)cc(C#N)ccc1CN1CCCC(NC(c2sccc2C)=O)C1 N1(C(C(C2CCC2)OC)=O)CC(CNC(C2(CSC3CC3)CC2)=O)OC(C)(C)C1 c1(C(=O)NCC2(CNC(CC3CC(C)C3)=O)CC2)ccc(=O)n(C)c1 Cc1c(C(=O)NC2CN(C(C3CCCS3)=O)C2)ccc(Br)c1Cl N1(C(C(C)OCC#C)=O)CCC2C(C1)NC(=O)CN2C(c1cccc(CF)c1)=O N#Cc1ccc(CC(=O)NC2CCC(NC(=O)C(=O)NCC(F)F)C2)c(F)c1 C1(C(=O)NCC2CCN2C(c2cc(F)c(F)cc2Cl)=O)CCCC2(CCOCC2)O1 C12(C(N(CCC#C)CC)=O)CCCC1CCN2C(=O)CC1(OCC)CCOCC1 CC(c1cnn(C)c1)=CC(=O)NCC1CC(F)CN1C(c1ccc(C2CC2)o1)=O S(=O)(=O)(c1cccnc1NCC(C)(C)n1ccnc1)NC1CC(C)N(C)CC1 N1(C(C2(CC=C)COC2)=O)CCN(C(=O)CC(O)C2CC2)C(C)C1 c1(OC)ccc(S(=O)(=O)N2CCOCC2)cc1NC(c1ncccc1F)=O c1(CC(=O)NC2CC(F)CN(C(C3CC4(C3)CC43CC3)=O)C2)ccc(F)cc1Cl CC1CN(C(c2nn[nH]c2Cl)=O)CC1NC(=O)C(C1CC1)N(C)C C1(OC)CN(C(=O)Cc2ccns2)CC1NC(=O)CCn1ccnc1 CC1(CNC(C2(C)C=CCC2)=O)CCN(C(c2cc(Br)no2)=O)C1 N1(C(COCCC)=O)Cc2nccn2CC(NC(c2nc(Cl)oc2C)=O)C1 Cc1ncsc1C=CC(=O)NC(C1CCCN1C(=O)C(C)CC1CC1)C N1(C(C2C(CNC(=O)C=Cc3cncs3)CC2)=O)CC=CC12CCOCC2 C1(C(=O)NC(CCC)CCO)CCCC(NC(C2(C3CC3)CC2)=O)CC1 C(CN=[N+]=[N-])(C(=O)NC(C)CN1CCCC1=O)NC(CCC(=O)NCC)=O N1(C(c2c(CC)sc(=N)[nH]2)=O)CCN(C(=O)C2=CC3(CCOC3)C2)C2CCCC12 c1(C(=O)NC(CC)CNC(c2cc(OC)n(C)n2)=O)c(C)ccc(Cl)c1O c1(C2C(F)C2)nc(Cc2cccs2)nn1C1CSC1.c1ccc(Cl)nc1 c1(C(=O)NC2(CC=C)CN(C(c3cnnn3C3CC3)=O)C2)ncsc1S(N)(=O)=O N1(CC)CC(NC(=O)CN(C(=O)C(C)N(C(C)=O)CC)C2CCC2)CC1=O c1(CCC(=O)NCCNC(CC2CCC(C)O2)=O)cncc(F)c1 C(CC(C(C)C)NC(=O)C=CCN1CCOCC1)NC(C(C)=C1CCCC1)=O c1(CC)cccc(C(=O)NC(C2CCN(C(=O)C=CC(C)C)C2)C)c1F c1(C(N2CCCC(NC(COC)=O)C(F)C2)=O)n[nH]c2c1C(=O)NCC2 c1(C(C)=O)ccc(C(=O)NCC2CCCN2C(c2cncc(F)c2)=O)cc1 C123CN(CC1CCO2)C3=O.CN1CCCC(CC(=O)NCC2CN(C(N)=O)C2)C1 c1(C(=O)NC(CNC(C(C)OCC=C)=O)CCOC)cc(F)c(OC)cc1F C1(NC(c2cccc(C(=O)N(CCO)CCO)c2)=O)CCOC12CCS(=O)(=O)CC2 c1(C(=O)NCC(C2CC2)NC(C)=O)ccc(Oc2ncccn2)cc1 c1(OCCC(=O)NC2CN(C(C(F)=C(C)C)=O)C(C)C2)cccc(Cl)c1Cl N#CC1CN(C(=O)CCOC2CN(C(=O)CCC3CCOCC3)C2)C1 C12(C(=O)NCC(C)S(C)(=O)=O)CC(CN(C(=O)C(F)C(F)(F)F)C1)C2 CN=c1[nH]c(C(=O)NCC2CCCC(NC(=O)CSCC(C)C)C2)cs1 C1(C)(NC(C=C(CCC)C)=O)CC(NC(=O)C(c2ccccc2)OCC)C1 C(=O)(C1CCCc2ccccc21)N1C(C(=O)Nc2nc(Br)cs2)COCC1 C1(C(N2CC(CN(C(=O)CS(N)(=O)=O)C)OCC2)=O)CCc2cc(F)ccc2O1 C1(C(C)NC(C=COCC)=O)CCN(C(=O)CN2CCOCC2=O)CC1 N1(C(C(=O)Nc2ccccc2)=O)CC(C2CCCN(C(c3cscc3F)=O)C2)C1 c1(C(N(CC(CC)NC(C2CC23CC(O)C3)=O)CC)=O)ccnc(Cl)c1 N1(C(CC2(OC)CCC2)=O)CCOC(CNC(=O)C(C)(C)NC(=O)C(F)(F)F)C1 CCC(CC)CC(=O)NC1C=CCN(C(=O)Cc2nc(-c3cccs3)oc2C)C1 C1(NC(CC=C)=O)C=CCCC1C(=O)NCC(O)C(C)C N1(C(C)=O)CCC(CNC(=O)CSCc2n[nH]c(=N)s2)CC1 N1(C(C(CCOC)C)=O)C(CNC(C2C3CCC2CC3)=O)CC2CCCC12 N1(C(C(C)=C2CCC2)=O)CC(NC(=O)CCOc2cccnc2)CC1(C)C C(CC(C)(C)CNC(c1ccc(OC(C)CC)cc1)=O)NC(CCC=C)=O c1(N2CC(C)C(CNC(C3(C)CCC3)=O)CC2)nc(O)c2ccccc2n1 C1(CN(C(=O)CCCc2ccsc2)C)CCCN(C(=O)Cc2ccon2)C1 C(=O)(CCCS(N)(=O)=O)NCCC1N(C(C2OCCN(C)C2)=O)CCSC1 c1(CC(C(=O)NCCNc2ncc(C)nc2)N)ccc(Cl)cc1C(F)(F)F N1(C(C2CCCC2)=O)CCCC(O)(CCNC(C23CCCC2C3)=O)C1 Cc1ccc(C(F)F)cc1C(N1CC(F)(CNC(=O)CCC2CC2(Cl)Cl)C1)=O c1(-c2n(-c3ccc(OC)cc3)nc(-c3ccn(C)n3)n2)cccc(Br)c1C C1(C(=O)OCC)COCCC1NC(c1cc(CCOC)[nH]n1)=O.C12(CC1)C(=O)N2 C(=O)(CC(C)C(C)(C)NC(=O)C1CC1)NC(C)CCF C1(CNC(C(CC=C)C)=O)CN(C(c2ns[nH]c2=O)=O)CCCO1 CC1=C(C(=O)N(C(C)CNC(c2cc(-c3cccnc3)on2)=O)C)CCCC1 C1(C)(CNC(C2(CC=C)COC2)=O)CCCN1C(=O)CC=CCC N(C(=NCCCC(F)(F)C(F)(F)F)NCC(C)(C)C)CC1(C)CCN(C)C1 C(CC(=O)NCCN1CCNC1=O)(C(F)F)NC(C1CCC(OC)CC1)=O c1(C(=O)NC2C(C)CCN(C(C3(C#N)CC=CC3)=O)C2)cc2cccc(Cl)c2o1 c1nccnc1N(C(C1(C(=O)OCC)CC1)=O)C.N1(C=O)CCC(OCC)C1 C(CS(=O)(=O)CC(=O)N1CC(CC(=O)NCc2ncc(C)cn2)CC1C)OC c1(CC)nnc(C)cc1C(=O)NCC1CCC(NC(C2COCC(C)(C)O2)=O)C1 CCC(C)C(C(=O)NC1CC(F)(CNC(=O)Cn2cc(C3CC3)nn2)C1)OC c1(C(=O)NCCCCN(C)C(C2(C3CCC3)CCC2)=O)ccc(O)cc1C(F)F N1(C(CCOC(C)=O)=O)CCC(C(N2CCC(CCO)C2)=O)C(C)(C)C1 c1(CNC(C23C(CN(C(c4ccc(C)cc4)=O)C2)C3)=O)ccc2nc(Cl)sc2c1 C1(NC(C(CNC(CC2OCC(C)(C)C2)=O)(C)C)=O)CC2CCCCN2C1 C(CCC(C)C(=O)N1CC2CC1(C(=O)NC(C1CCC1)C)C2)OC Cn1nnc2c1C(C(=O)N1CC3C(CNC(=O)CC4CC(F)C4)C3C1)CCC2 CC1CC(CNC(C2CSCCS2)=O)CCN1C(C1CCCCC1(C)C)=O c1(C(N2CCC(CNC(C(C)SCC)=O)(OC)C2)=O)cc(C)c(C(N)=O)cn1 N1(C(C(CC)NC)=O)CC2CN(C(c3ccc4c(c3)CCC4)=O)CC(C1)O2 C=C(C)CC(=O)NC1CC1CNC(=O)CC1CN(C(=O)OC(C)(C)C)C1 C1(C(=O)NC(CNC(C=CCCC=C(C)C)=O)(C)C)CCCN(S(C)(=O)=O)C1 N1(C(c2c(C)n[nH]c2)=O)CCC(C(N2CC(c3ccncc3)C2)=O)C(O)C1 C(=O)(C(C)(C)C(=O)NCC(c1ccccc1)CNC(=O)C(C)(C)CO)OC N1(CC(C)OC)C(=O)CCN(CC2CN(CCOC)CCO2)C1=O CCC(CCOC)C(=O)N1CC(O)CC1CNC(C1(CC2CC2)CC1)=O C(C)(N=c1nn[nH]n1C)c1c(CN(C(C)C)C(C2CCCC(F)(F)C2)=O)cccc1 N1(C(c2n(CC)c(O)nc2)=O)CCCC(NC(c2ncc(Cl)cc2O)=O)CC1 CCCCCC(C)(CC)C(=O)NN(C(=O)CCNC(N)=O)C1CC1.C12(CC1)CC2 N1(C(C2N(C(c3scc(C#N)c3)=O)CCC2)=O)CCn2nccc2C1 c1(CC)cc(C(=O)NCC(C)C(=O)NC(C)CN2CCCC2=O)ncn1 C1(NC(NNC(c2cccc(C)c2F)=O)=O)CCCC2(CCOC2)O1 C1(NC(C2(COC)CCCCC2)=O)CCN(C(=O)CCC2CC2(Cl)Cl)CC1O C(=O)(CC1=NNC(=O)C1)N(CC1N(C)CCN(c2ncc(C(C)=O)cn2)C1)CC c1(OCC)c(CNC(C2CCCCN2Cc2ccc(NC)s2)=O)cc(C)cc1Br C(=O)(CCCC(F)(F)C(F)(F)F)NCC1CC(C)N(C(=O)C(Cl)=CCl)C1 CC#CCC(CO)NC(=O)C(C)(C)C1CCCN1C(=O)CCn1cccc1 CC1CCCC1C(=O)NCCOCCCNC(c1cn(C(C)(C)C)cn1)=O N1(C(C2(C(N(C)C)=O)CC2)=O)C2CCC1CC(NC(C1CC(=O)NC(=O)N1)=O)C2 N1(C(=O)OCC2N(C(=O)OC(C)(C)C)CC(F)C2)C(=O)C2C=CCCN2S1(=O)=O N1(C(C)C(=O)NCCNC(N2CCOC(CO)C2)=O)CCc2ccccc21 n1(C(C)C)ncc(C(=O)N(CC(C)CNC(=O)CC(C)F)C)c1N C(=O)(C1=CCS(=O)(=O)C1)N1CCCC(C)C1CNC(=O)CC1CCOC1 c1(NC(COC)C)ncnc(N(C)Cc2cc(F)ccc2F)c1C C12(NC(C(CC(N)=O)O)=O)CCOCC1CN(C(c1onc3ccccc13)=O)C2 c1(C(N2CCC(C(C)NC(c3ccsc3C(F)F)=O)C2)=O)ccc(Cl)c(N)c1 N1(C(=O)C2=CCCS2)CCN2C(=O)C(NC(C3(F)CCCCC3)=O)CC2C1 N1(C(Cc2c(C)occ2)=O)CCCC(C(N2CCC(CC3CCC3)C2)=O)CC1 c1(N2C(C)CCN(C(CS(CC)=O)=O)CC2)ncnc2c(Br)nn(C)c12 c1(C(N2CCC(CN(C(c3c(C)cco3)=O)C)C2)=O)cnc2[nH]cc(C)c2c1 CCC(C(=O)NC(CC1CCC1)C(=O)NCC(F)CO)NC(N)=O c1(N2C(C)CC(NC(c3cccc(C(C)(F)F)n3)=O)C2)cc2nncn2cn1 CN1CC(CC(=O)N2C3CCC2CN(C(C2CCC(=O)N2)=O)C3)c2ccccc21 C(=O)(C1Cc2ccccc21)N1CC2CC(Nc3ncc(Cl)c(C)c3C#N)C2C1 N1(C(C(C)=C2CCCC2)=O)CCC(NC(c2cc(C)cnn2)=O)CC1C C1(C(N2CC(CCCCN)C2)=O)(CCl)CC1(F)F.C(C(F)(F)F)C1(C(=O)NC2CC2)CC1 c1(C(c2ccccc2Cl)N(C)C)nc(-c2ccc(Cl)s2)nn1C1(C)CC1 CC1(CC(=O)NC(CO)C(=O)Nc2ccn(C3CC3)n2)CCOC1 c1(C(=O)NC2CCN(CC(=O)Nc3ccc(Br)cn3)CC2)c(F)ccnc1Cl c1(C(=O)NCC(CNC(C(COC)(C)O)=O)C)nn(C)c2c1CS(=O)(=O)CC2 C1(C(CNC(CCN(CC)CC)=O)O)CCN(C(C2(C)CC2(C)C)=O)CC1 N1(C(C2=CCC(NC(C3(COC)C=CCC3)=O)C2)=O)CCC(OC)C(C)(C)C1 N1(CC(=O)N(CCCNC(=O)CC2CSCCO2)C)CCCCCC1 Cn1c([N+](=O)[O-])cnc1C(=O)NCC1CC(F)(CNC(=O)CN2CCSCC2)C1 N1(C(C2C3C(NC(CC4C(C)=NNC4=O)=O)C4C(C3)C42)=O)CCCC(C)(O)CC1 c1(C(=O)NC(CCN(C(C(CCSC)OC)=O)C)C(C)C)cc(C)c(C)cn1 C12(CNC(C(n3cc(-c4c(CC)cccc4)nn3)C)=O)COCC(COC1)O2 C1(C(N(C)CC2CCN(C(c3cc(C#N)on3)=O)C2)=O)CCCCCS1(=O)=O c1(C(=O)NCCCNC(C2N(S(CC)(=O)=O)CCC2)=O)cc(Cl)c2n[nH]cc2c1 c1(OC)cnc(C(=O)NCC2CC3CC2CN3C(c2cnn(C)n2)=O)c(OC)n1 C1(NC(c2c(C)ncn2C)=O)CN(C(=O)C=CCN(C)C)CCC1C(F)(F)F Cc1c(C(N2CCC(NC(=O)COCCO)C2C)=O)cnn1C(C)(C)C C(=O)(C1=C(Cl)CCC1)NC1(CCO)CN(C(c2ccc(OC(CC)C)cc2)=O)C1 C(=O)(C1CCSc2ccccc21)N1CCCC(N(C)C(C2CC3CC2C3)=O)C1 O=C(CCCCOC1CCCC1)NCC1CC(NC(C23C=CC(CC2)C3)=O)C1 Cc1ccc(C)c(CN2CCOCC2CC(=O)NCC2CCCCO2)c1 Cc1cc(F)c(C(N2CCC(C(C)NC(c3ncc(F)cn3)=O)CC2)=O)c(Cl)c1 C1(CNC(CCC=CC)=O)CCC12CCN(C(=O)C(CN(C)C)CC)CC2 C1(CC)COCCC1Nc1ccc(N(C)C(=O)OC(C)(C)C)cn1 C1(NC(C2N(C(C)=O)CSC2)=O)CN(C(c2nccnc2C)=O)CC1C c1(CC)c(OC)cccc1C(N1CCN(C(=O)C=CC(C)(C)SC)CC1)=O C1(C)(C(=O)NC(CCCC)CNC(=O)COC(C)=O)CC2CCC1O2 C(=O)(C(CC(C)C)C(N)=O)N1C(C(C(=O)NCC(=C)CC)(C)C)CCC1 C1(C(c2cn(C)nn2)=O)CCCCC1C(N1CCCC(CS(C)(=O)=O)C1)=O C1(NC(C(CC)OC)=O)CN(C(c2cnn(CN(CC)CC)c2)=O)CCC1(C)C C1(C(N2CC(NC(c3n(CC)cnn3)=O)C(O)C2)=O)CCCCC12CCC2 c1(CC)ccc(C(N2CCC(C)C(NC(c3cnc(C4CC4)s3)=O)C2)=O)cc1F C12(C(N(C(C)CC3CC3)C)=O)CCN(C(=O)CNC(=O)C(C)(C)C)CCC1C2 C1(C(C)C)CN(C(=O)CCC#N)CCN1C(c1cc2c(s1)CCC2)=O c1(SCCC(=O)NC2C(OC)CN(C(C3CC(C#N)C3)=O)C2)cc(F)ccc1F N1(C(C(C)=C2CCCC2)=O)CCC2(CCCC2NC(=O)C=CC(=O)NC2CC2)C1 C(C1=CCN(C(C2(C)CC(F)C2)=O)CC1)NC(c1n(CCC)ncc1)=O N1(C(CCCn2c(C)csc2=O)=O)C2CCC1CN(C(=O)Cc1ccnn1C)C2 N1(C(c2ccc(CN=[N+]=[N-])o2)=O)CCC(CNC(c2ccncn2)=O)C(F)(F)C1 c1(C(=O)NCC2(NC(c3ccc(F)c(F)c3)=O)CCC2)nc2cccnc2s1 c1(C(N2C(C)CN(C(=O)C(C)(C)F)CC2)=O)ccc(S(=O)(=O)NC2CC2)cc1 C(N=c1[nH]nc(C(C)(C)C)o1)C1CN(C(c2cnc(CC(C)C)s2)=O)C1 C1(C(=O)NC2CN(C(c3csc(C)c3C)=O)CC2C)CN2CCCN1CC2 Cc1cccc(CCNC(=O)C(C2CC=CCC2)NC(=O)C(C)c2cc[nH]n2)n1 C(=O)(CC(C)C(=O)N1CCC(OCC(=O)NC2CC2c2ccco2)C1)OC O(NC(=O)C(C1CCC1)NC(C1CCC(F)(F)C1)=O)CCC(C)C S(=O)(=O)(c1ccc(C(N2CCCC2C2(O)CC2)=O)cc1)N(CCOC)CCO C(=O)(CC(C)(C(F)F)N(C)C)NC(C1(O)CN(C(c2cnc(CC)[nH]2)=O)C1)C CCCC(C)(C)CC(=O)N(C1CN(C(=O)C=Cc2cncc(CO)c2)CC1O)C CCCCCC(C(=O)NCCOCC)N(C)CCNC C1(NC(C=CC(=O)OCCCC)=O)CCC(C)N(C(c2ccnc(OCC)c2)=O)C1 C(=O)(C(CNC(c1ccoc1Cl)=O)(CC)CC)NC(C#C)C N1(C(CC(CNC(CC2CC(SC)C2)=O)(C)C)=O)CCC(C2CCCC2)C1 c1(C(=O)NCC2COCCN(C(C(CC)SC)=O)C2)cc2c(cc1Cl)NCC2 C1(CNC(C2CCN(C(CC)=O)C2)=O)CCCCN1C(=O)Cc1nc(=N)[nH][nH]1 O=C(CCCCC(F)(F)F)NC1CCCN(C(C2CC(F)(F)C2(F)F)=O)C1 C(=O)(C(C)(C)C1CCCC1)N1C(C(N(CC(=O)NCc2cccs2)C)=O)CC1 CCC(CC)(CC)C(=O)N(C1CCCC1)CCNC(=O)C(F)CC1CCOCC1 CCC(CCC(=O)N(C1CN(C(=O)Cc2ccc(O)nc2)C1)C)OC C(=O)(C1=C(C)OCC1)NC(CNC(C(CC)N1CCCC1=O)=O)CC(C)C c1(C(=O)NC2C=CCC(C(=O)NCC=C=C)C2)nc(C)ccc1C C(=O)(CCC(C)CC)NCCN(CC(C)O)C(c1c(CC)noc1)=O Cc1cc(=NC2CCN(C3CCNC3=O)CC2C)[nH]c(Cl)n1 c1(C(CC(=O)O)C)cccc2ccccc12.C(=O)(CCCCCF)OCC N1(C(CCn2c(C)cc(C)n2)=O)CCCC(C)C1CNC(c1ccc(CO)o1)=O C(=O)(C(F)(F)CC(C)C)N(C)CC1N(C(c2c(C)ccc(OC)c2)=O)CCC1 C1(CC(=O)NC2(CSC)CCC2)CN(C(c2cncc(OC(C)C)c2)=O)CCO1 CC(CCCNC(=O)CCC1OCCO1)NC(=O)C(c1ccccc1)O C1(NC(c2cc(C(F)(F)F)ns2)=O)C2CCC1N(C(c1ncncc1Cl)=O)C2 CC(CC(F)F)C(=O)NCc1ncccc1C(N1CCCC1C(N)=O)=O C1(N(C)C(=O)OC(C)(C)C)CC2CC1CN(C(=O)C=CCN1CCCC1)C2 C1(C(=O)NC2CCC(C(=O)OC)C2)CCN(C(=O)CC2CC(C3CC3)C2)CCO1 C12(NC(CCN(C(C)=O)C)=O)CC3CC(C1)CC(NC(=O)CC1OCCO1)(C3)C2 CCC(C)C(CC(=O)NC1(CO)CCSC1)NC(c1cncs1)=O C1(C(N2CCCC(O)(CN(C(COCC(C)C)=O)C)C2)=O)CC2(C1)CC21CCC1 C(CCCOC)(C(=O)N1CC=CCC1)NC(C1CC(CCC)C1)=O C#Cc1ccccc1CNC(=O)CN(C(=O)C(CC)N(C)C)C1CC(C#N)C1 CC(CCN=c1[nH]c2c(c(=NCCCCc3ncc[nH]3)[nH]1)CCCC2)N(C)C N1(C(CCCC)=O)CCc2nc(CNC(c3cc(C)nc(O)n3)=O)sc2C1 C1CC2(C1)CCOC2CNC1(c2nnnn2C2CCCC2)COCCOC1 c1(OC)ccc2c(C(=O)N(C(C)CCNC(=O)CC3CC3(Cl)Cl)C)c[nH]c2c1 C1(C)(NC(COCC(C)C)=O)CC(NC(=O)C=Cc2ncc[nH]2)C1 CC1(C)Cc2ccc(C(=O)N=c3ccn(CCN4CCOCC4)[nH]3)cc2O1 c1(C(=O)NC(C)C(C)NC(c2cnc(C3CCCCC3)s2)=O)cc(C(F)F)n[nH]1 C(=O)(C(C)(CCC)CCC)NC(CN(C(CC(C=C)(C)C)=O)C)C c1(C(N(C2CN(C(C3COCC(C)(C)O3)=O)CC2O)C)=O)ccn2cnnc2c1 c1(OC)ccc(C)cc1CC(=O)NCCCC(C)NC(C1COC(=O)O1)=O O=C(CC1CCc2ccccc21)N1CC(O)C(O)C1 c1(CC(=O)NCC(C2CCC2)NC(CC(=C)Br)=O)ccc(C)c(Cl)c1 C1(C(N2CCC(O)(C(C)NC(CCSC)=O)CC2)=O)CCc2cc(F)ccc2O1 Cc1ccc2c(N3CCCC3(C)CNC(=O)CC3CCCCN3C)ncnc2c1 CC(C)(C)CC(=O)NCCCNC(C1C2CCC(=O)C12)=O C1(NC(CCSCC)=O)CN(C(C2(CCOC)CCCC2)=O)CC2CC12 c1(CNS(=O)(=O)CC2CC(F)(F)C23CCC3)ccc2c(c1)CCCO2 C1(CC(=O)NC2C3CC(NC(C(CCC)=CCCC)=O)CC32)CC2(CCC2)CO1 c1(CNC(c2n(CCC)nnn2)c2ccnn2C(C)CC)cccnc1Br C1(CC(=O)NC2C3(CC(NC(c4c(CC#N)ccs4)=O)C3)C2)CC(=O)NC(=O)C1 c1(OCC)ccc(NS(C)(=O)=O)cc1NC(=O)CC1CCCCN1CC(F)(F)F C1(C(=O)NCCN(C(c2ncccn2)=O)CC2CC2)CC(F)(F)CS1 N1(C(C2(C)C(C)OC(C)(C)O2)=O)CCOC2(C1)CN(C(=O)CCC(C)(F)F)C2 N1(C(=O)C2=NN(c3ccc(Br)cc3)C(=O)CC2)CCC2CCC(O)CC2C1 Cc1cc(NC(=O)CCc2nc(C)c(C)[nH]2)ccc1NC(C1(O)CC1)=O C(=O)(C(O)CC(F)(F)F)N1CCC(CCNC(c2cc(N)cc(O)c2)=O)C1 CCCCC(CC)CC(CC)N1CCCC1CCC1(O)CCN(C(=O)OC)CC1 CC1C(NC(c2ccc(N)cn2)=O)CCN1C(c1ccnc(-n2cncn2)c1)=O N(C(=NCC1(O)CCOC1)NCC1(c2cccs2)CCCCC1)C(CC)CC C1(C)(C(=O)NCCC(C(C)C)OC)CCCN(C(c2cc(C)cc(F)c2)=O)C1 C1(COC)(NC(=O)CC=C(C)C)CCN(C(=O)C(C)NC(=O)CC(F)(F)F)C1 N1(CC(=O)N(C)CC2CCCC2)CCN(CCc2cnccn2)CC1 N1(C(CC2C(CNC(C(C(=O)OCC)OC)=O)C2)=O)CCOCCC1CC C(CCCCC(=O)NC1CCCC1CNC(C12CCN(CC1)C2)=O)SC c1(N(CC(=O)NCC2(NC(=O)C(O)C3CC3)CCC2)C)cccc([N+](=O)[O-])c1 C(=O)(C1CCCc2ncnn21)NC1C2CN(C(c3c(N)cncn3)=O)CC21 Cc1cccc(C(=O)NCCN(C)C(C2CCC3CC3CC2)=O)c1Cl CC1CCCC(CCNC(C2CCC(NC(=O)C3=COCC3)C2)=O)C1 C1(CC#C)(C(N2CC=CC(NC(c3snc(O)c3Cl)=O)C2)=O)CC=CCC1 C1(NC(c2csc(Cl)n2)=O)CC12CCN(C(c1cccc(CCO)c1)=O)CC2 C=C1CC(C(=O)NC(C)CN2CCOCC2)(CNC(C2CC(OC)(OC)C2)=O)C1 c1(CCC(=O)NC(c2cn(CC3(CO)CC3)nn2)C)ncc(C(C)(C)C)o1 N1(C(C(=Cc2ccccn2)C)=O)CCOC2(CCC(NC(=O)C(N)=O)CC2)C1 C1(O)(c2onc(COc3ccc(OCC)cc3)n2)CCOCC1C1CN(C(C)=O)C1 N1(C(C(C)c2cc[nH]n2)=O)CCC(CCC(N2CCCC(CC3CC3)C2)=O)CC1 CCC(CCC(=O)NCCC1COCC1O)NC(C1(F)CCCCC1)=O c1(C(N2CCC(CN(CCOC)C)C2)C(=O)NCCCSC)cc(Cl)ccc1F c1(COC)csc(C(=O)NCC(C2CCCC2)NC(=O)CCCNC(N)=O)c1 c1(C(=O)NC2(C)CN(C(c3nccc(C(=O)OC)c3)=O)C2)ccc(Cl)c(C)c1 C1(CC(=O)NCCN(CCC)C(C)C)(NC(=O)CC2CCNC2=O)CCCCC1 c1(C(C)=O)cocc1C(=O)NC(C)C(=O)NCCP(C)(C)=O Cc1nn(C2CCOC2)cc1C(=O)NCCNC(=O)C(C)(C)c1ccn(C)n1 c1(C(=O)NC2CCN(C(CNC(=O)NC)=O)C23CC3)cccc2c1CCC(=O)N2 C12(NC(C(C)Sc3ncccn3)=O)CCCC1N(C(=O)CCC(C)(C)O)CC2 C1(NC(CCOC(C)C)=O)CN(C(c2cccc(N)c2O)=O)C2(CCC2)C1 c1(CC)ncc(C(=O)NC2CCC2CNC(=O)C(C)CC2CCCCC2)cn1 O=C(C(Cc1cccc(Cl)c1)=NO)NC1CCC1NC(c1coc(Cl)n1)=O c1(CC)ccc(OCCC(=O)NCC=CCNC(C2CNC(=O)N2)=O)cc1 CC1(n2cncn2)CC=CCC1.C1(C2CCCO2)(CN2C(=O)CSCC2)CCC1 C1(c2nnnn2C(C)(C)C)(NCC(C)OC)CCC(O)(C(F)(F)F)CC1 C(=O)(CC(C)CC(C)(C)C)N(C(CC(N1C(C=C)COCC1)=O)CC)C C(CCC(=O)N(C(C)C(=O)N(C(C(N)=O)C1CC1)C)C1CC1)=CC n1(CC)ncc(C(=O)NC2CCN(C(=O)C(C(C)C)n3cnnc3)CC2)c1Cl C1(CNC(C(Br)=C(C)C)=O)CC2(CO1)CN(C(C13CC1COC3(C)C)=O)C2 N1(C(C(CC(=O)OC)(C)C)=O)CCC2(CC1)CC(NC(=O)CC1(C)CC1)CCO2 c1(C(=O)NC2C(NC(C(n3c(C)ncc3)C)=O)CCC2)ccc(NC(N)=O)cc1 C(=O)(C(CC(C)C)NC(C1CCCC1C1CC1)=O)NCC(=O)OCC c1(C(N2CC3(C(NC(C=CSC)=O)CCS3)C2)=O)ccc2ccccc2c1 C1(C(N2CCC(N(C(c3c(C)nc[nH]3)=O)CCO)C2)=O)CC2(C1)CC21CC1 Cc1c(Br)ccc(NCCC=C(Cl)Cl)c1[N+](=O)[O-] C1(NC(C(C)NC2(C3CC3)CC2)=O)CC(C)CC(C)(C)C1 N1(C(COCCC)=O)CC(CNC(c2nccc(Cl)c2F)=O)CCC1C CC1(NC(c2ccc(CO)cc2)=O)CCN(C(c2n[nH]cc2C2CC2)=O)CC1 Cc1cnc2c(C(=O)NCC(C(C)(C)C)NC(c3cn(C)cn3)=O)cccc2n1 Cc1nc(C)c(CC(=O)NC2CCC(NC(c3ncncc3Cl)=O)C2)s1 CS(=O)(=O)c1ccc(C(N2CCC(CNC(=O)CCCCN3CCCC3)C2)=O)o1 C1(CC)CN(Cc2cccnc2F)CCN1C(c1ccnc(F)c1Cl)=O C(=O)(C1CCc2snnc21)NCC1N(C(c2c(CC)ccs2)=O)CCCC1C N1(C(C(CCOC)(C)C)=O)CCC(C2CCN(C(=O)CN3CC4CC4C3)C2)CC1 c1(C(=O)NC2CCN(C(c3ccco3)=O)CC2F)cc2ccc(Cl)cc2o1 C1(F)(CNC(CC(CC)C2CCC2)=O)CCCN(C(C2(C)CCCN2C)=O)CC1 c1(C(N2CC(c3ccccc3)(C(=O)NCC)C2)=O)cn(CCOC)nc1C C(=O)(CC(C)(C)CC(F)F)NCC1N(C(c2c(C)nsc2)=O)CC=C1 CC(C(=O)NCC(O)CNC(c1cnoc1)=O)N(C)C N1(C(CC2N(C)CCCC2)=O)CCOCC(CNC(c2cnoc2C2CC2)=O)C1 C1(C(=O)NC(CCN(C(c2ccc(CCC)s2)=O)C)C)COCCN1CC C1(CN(C(C(C)(C)SC)=O)C)CN(C(C2COC(C)(C)C2)=O)CCO1 N1(C(CC(=O)Nc2ccccc2Br)=O)CCC(F)(F)C(NC(c2cscn2)=O)C1 CCC(C)(C(=O)N1CC(CC(C)NC(=O)C(O)C2CC2)C1)OC c1(C(=O)NCC2C(NC(C(C3CCC3)OC)=O)CCC2)ccc([N+](=O)[O-])c(O)c1 C1(C(=O)NCC(=O)Cc2ccccc2)(Cn2cc(CO)nn2)CCOCC1 Cn1cc(C=CC(=O)NCC2CCCCC2NC(c2ccc(Cl)[nH]2)=O)cn1 C(=O)(C1CCCc2c[nH]nc21)NCC1CN(C(=O)CSCCC#N)CC(C)(C)O1 CC(CN=c1ccnc(NCc2c[nH]nc2C(C)(C)C)[nH]1)C(F)F N1(C(C(CC#C)C2CC2)=O)C2CCC(C2)C1C(=O)NCC1(O)CCCCC1 C(=O)(C1CCc2c[nH]nc21)NC1C(NC(c2nc(OC)c(F)cn2)=O)COC1 C(C)(CCC(=O)N1CCOC(CNC(=O)C(=Cc2cccnc2)C)C1)OCC C(C)(CCC(=O)N(CCCNC(C1CCCSC1C)=O)CC1CCCC1)SC C1(CNCC)(OC(c2cc(C(F)(F)F)ccn2)=O)CCC(C(F)F)CC1 c1(OCC(=O)OCc2cnc(C(F)(F)F)s2)ccc(S(=O)(=O)C(F)(F)F)cc1 N1(C(C=C(CC)CC)=O)CCC(C(N2CC(C)(CO)C2)=O)C(C)C1 C1(CNC(C2(C(=O)OCC)CC2)=O)CN(C(c2ccc(SC)o2)=O)CC12CCC2 c1(N2CCC(CNC(CCc3c(C)n(C)nc3)=O)C2)ccc(S(C)(=O)=O)cn1 c1(C(=O)NC2C(O)CCN(C(c3n(CC)ccc3)=O)C2)nc2cccnc2s1 C12(C(=O)NC3CC(F)(CNC(c4c(C)csc4)=O)C3)CC(C)(C1)OC21CCC1 Cc1nc(C2CC2)sc1CC(=O)NC1CC(CNC(=O)CSCCN(C)C)C1 CCCC(CCCO)C(=O)N1CCC(CCC)(NC(=O)CCCC(=O)NCC)CC1 C1(C(=O)Nc2ccc(SCC(=O)OC)cc2)CC2CCCC1(N)C2 C(Cc1ccccc1)(C(=O)NCC(CO)NC(c1cnco1)=O)NC(CCC)=O C1(NC(c2ccccc2SCCO)=O)COCCN(C(C2C(F)(F)C23CC3)=O)C1 c1(C(N(CCC(=O)Nc2cn(CC=C)nc2)C2CC2)=O)nnc(O)nc1O C(=O)(CCCN=[N+]=[N-])NC(CC(=O)NCc1c(C)cn(C)n1)CC1CC1 c1(C(N(CCC)CCNC(c2cnc(C)nc2)=O)=O)c(Cl)nn(C)c1C N1(C(c2cc(C(CC)C)no2)=O)CCC=C(CNC(=O)CCCCN(C)C)C1 N1(C(CC2N(C)CCC2)=O)CCNC(C(=O)Nc2cnsc2)C1 c1(N)cccc(C#N)c1.S(=O)(=O)(CC(=O)NCCN(C(=O)C(F)OC)C)N(CC)CC c1(C(=O)NC2CC(CNC(Cc3n(C(C)C)cnn3)=O)C2)nc(OC)ccc1Cl C(=O)(CS(=O)(=O)CC(F)(F)F)N(CCC(C(C)C)NC(=O)C(C)N(C)C)C C1(C(=O)NC2(C3CN(C(C4CSCCS4)=O)C3)CC2)CC12CCC(F)(F)CC2 c1(OCCC)ccc(CC(=O)NC2(CNC(=O)CCc3cc(C)on3)CC2)cc1 c1(C(N(CC(CN(C(c2c(C)coc2)=O)C)O)C)=O)cc2ccccc2[nH]c1=N N1(C(CC2N(C(C)C)CCC2)=O)CC2CC1CCN2C(c1ccc(F)c(Cl)c1)=O c1(C(=O)NCC2(CO)CCN(C(C(CC#C)O)=O)CC2)cc2cccnn2n1 O=C(CCSC1CNCCOC1)NN=c1cc[nH]c2ccccc12 Cc1cncc(-c2cn(CCCC(=O)NC(c3nc(=O)o[nH]3)C)nn2)c1 c1(NCC2CN(C)C2)ncc(S(=O)(=O)NC2COc3cc(Cl)ccc32)cc1Cl CCCC(C(=O)N1CCCC2(NC(c3cn4c(n3)CCC4)=O)CC2C1)C(C)C C1(C(=O)NCC(CCCC)NC(c2ccnnc2O)=O)Cc2nnc(C)n2C1 C1(NC(C2ON=C(C)C2)=O)CCOCC1NC(=O)C=Cc1sccc1C C1(C)(CCC(N2CCC(OCC=C)C2)=O)CCCN1C(=O)CCC=CC N1(CC23CC(C)(OC2)C3)C(=O)CCN(Cc2nc(C(F)(F)F)n[nH]2)C1=O C1(CC)CCOC1C(=O)NCCN(C(=O)Cc1nncs1)CCOCCO c1(CC)ccc(NC(C2CCC2CNC(c2cc(CC)[nH]n2)=O)=O)c(C)c1 N1(C(CC(C(=O)OC)(C)C)=O)CCC2CN(c3nccc(C)n3)CC2C1 N1(C(C(c2ccncc2)C)=O)CCCC1CNC(c1cnn(C2CCC2)c1)=O c1(C2(NC(CN(C)CC3CCN(C(c4cn[nH]c4)=O)C3)=O)CC2)cccc(F)c1 c1(C(N2C(CNC(CCCC=C)=O)C=CC2)=O)coc2c(Cl)cccc12 O=C(CCCn1cncn1)NCC(C1CC1)NC(C1CSC1)=O C(=O)(CC1=NN(C)C(=O)C1)N(C1(C(=O)NCCOCC(=O)OC)CCC1)C1CC1 C1(CC)C(=O)NCCCN1C(C1C=CCN(C(C2(C#N)CCCO2)=O)C1)=O C1(NCc2c(Cl)nccc2)CC(N=c2nc[nH]n3cccc23)C1 c1(C(=O)NCC=CCNC(C(n2ccc(CO)n2)C)=O)ccnc(C(F)(F)F)c1 C12(C(N3CC(C(C)NC(=O)Cn4ccnn4)OCC3)=O)CCCC1CCC2 c1(C(=O)NC2(C(=O)NCC(C)OCCO)CSC2)cncc(F)c1 Cc1cc(C(=O)NC2(C(=O)NCC3=NOC(C)C3)CC(O)C2)sc1C N1(C(C2(C)CCOCC2)=O)CC2CCC(NC(C3CCCNS3(=O)=O)=O)(C2)C1 c1(C(=O)NC2CN(C(c3ccoc3C(F)(F)F)=O)C2)cc(C2CCOCC2)[nH]n1 CC1=C(C(=O)N(CCCNC(=O)CC2CC3(CC3)C2)CCO)CC1 C(=O)(C1=CCOCC1)N(CC(C)NC(c1n(C(CC)C)ncc1)=O)C C1(CCNC(c2c(C)cccc2)=O)CN(C(=O)COCC(F)F)CCCO1 S(=O)(=O)(c1ccccc1F)N1CCN(CCC)C(=O)C1 N1(C(C(F)=CC)=O)CCC(NC(C2CCSCC2)=O)CC(C)(C)C1 c1(C(N2C(CC(=O)Nc3c(C)ncc(Cl)c3)CCC2)=O)cn2cc(F)ccc2n1 c1(C(=O)NC(C2CN(C(C(C)n3cccc3)=O)C2)C)ccccc1CCN(C)C c1(C(N2C(CCNC(c3ccoc3C)=O)CC(OC)C2)=O)cncc(Cl)c1C C1(C(=O)NCCCN(C)C(=O)OC(C)(C)C)(C(=O)NCC2CC2F)CCCC1 N1(C(C2ON=C(C)C2)=O)CCCCC12CN(C(C1(C)CCCNS1(=O)=O)=O)C2 C(=O)(CC(C)CC(C)(C)C)NC(CCC)C(O)C(=O)NCc1cn(CC)nn1 C1(N)CCN(C(c2cccc(Cl)c2)=O)CC1C.C=CCN(CC=C)C(C)C N1(C(C(CO)NC(CCCSC)=O)=O)CC2C=CCC(C2)C1 c1(C(=O)NC2CN(C(CCC(=O)NCC)=O)C(C)CC2)cc2cccc(Cl)c2o1 C1(C(C(=O)N(C)Cc2cn(-c3cccc(CO)c3)nn2)F)CCS(=O)(=O)CC1 n1(CC(=O)NCC(C)CNC(=O)C(F)n2cccn2)cc(Br)c(O)nc1=O c1(C(=O)NC2CN(C(CC(C)F)=O)CC(O)C2)ccc2c(c1)C=CCC2 O=C1CCC(C(=O)N(C2CCN(C(C3CCCSC3)=O)C2)CCO)=NN1 C1(CCCNC(CN(CC(C)(C)C)C)=O)CCCN1C(=O)CSC1CCCO1 N1(C(=O)NCCSCCSC)CCOC(c2ccc(OC)cc2)C1 C1(NC(C2(CCC)CC2)=O)CCCCN(C(=O)C(CC)OC)C1 N1(C(CCCOC(C)C)=O)CCCCC1CCNC(c1nc(Cl)sc1Cl)=O C1(C(N2CC(CNC(c3cc(C)nc(C)c3)=O)C2)=O)CC2(CCCC2)CO1 C1(C(=O)NCC2CC(F)CN2C(C2(C3CCC3)CC2)=O)CCc2[nH]nc(O)c2C1 c1(C(=O)NC(C)CC2CN(C(c3coc(O)n3)=O)C2)cnc(N(C)C)cn1 c1(C(N(CCCN(C)CC2CCOCC2)C)=O)ccc2c(c1)CC2 c1(CC)cc([N+](=O)[O-])ccc1C(=O)Nc1cccc(NC(=O)C2=CSCS2)c1 CC(C)C(C)(O)C(=O)N1CC2CCC2(CNC(=O)Cn2ncc(Br)n2)C1 N1(c2nc(SC)nc(C)c2)CCc2cccc(C(=O)NC3CCS(=O)(=O)C3)c2C1 c1(C(N2C(C3CCN(C(C4(C)CCNC4=O)=O)C3)CCC2)=O)cc(N)ccc1Cl C(=O)(C1CCc2c(Cl)cccc21)N1CCC(COC)(NC(=O)CSC2CC2)C1 Cc1nc2ccc(CN3CCC(C4CCCN4C(=O)CCCC(N)=O)C3)cc2s1 C(=O)(C(C)(O)CC(F)F)N1CC(CNC(C(=O)N(C)C)=O)OCC1 C1(CNC(c2c(CC)ncnc2)=O)CN(C(c2nccn2C(C)C)=O)CCC1C Cn1nc(C(=O)NCC2(O)CCN(C(C3(CO)CC3(F)F)=O)C2)ccc1=O c1(C(N2C(CNC(c3c(SC(C)C)cccc3)=O)C=CC2)=O)ccc(O)c(Cl)n1 C1(C(=O)NCc2ccc(C)s2)(CC)CCCN(C(c2ccccc2O)=O)C1 c1(CN(C(=O)C(=O)NC(CN(C)C)Cc2ccccc2)C)cc(Cl)c(Cl)c(Cl)c1 c1(CNCC2CCCN(C(c3c(C#N)ccnc3)=O)C2)ccc(F)c(F)c1Cl c1(NC(CO)CCN2CCCCC2)nccc(N2CCCCC2)n1 c1(C(=O)NC2CCN(C(=O)C3CC3)C2)c(F)cncc1Br Cc1ccc(F)c(C(=O)NC2CC(F)CN(C(c3cc(Br)cnc3Cl)=O)C2)c1 c12cc(CC)ccc1Cn1c(nnn1)C(c1ncc(CC)s1)N2.C1(CC)CCC1 c1(CCC(N2CC3C(CNC(C)=O)C3C2)=O)cccc2cnccc12 C1(OC)CCCN(c2cc(N3CCC(c4cccc(Cl)c4)C3)ncn2)C1 c1(C(N2CC(CNC(C=C(COC)C)=O)OCC2)=O)cccc2c1NC(=O)C2=O C(=O)(C1CCCc2cncn21)NC(CN(C(=O)Cc1ccnc(Br)c1)CC)C c1(CN2CCN(CCN3C(C)(C(=O)OC)CCCC3)CC2)ccc(C#N)c(C)c1 N1(Cc2c(F)cc(-c3sccc3Cl)cc2)CCC2(CCC(O)C2)CC1 C(C)(CC(=O)NC1CCN(C(c2ccoc2)=O)C1(C)C)(C(F)(F)F)N(C)C N1(C(CC2(COC)CC2)=O)CCC(C)(CCNC(=O)C(C)CN2CCCCC2)C1 c1(CC(=O)NCCC(C)CO)nnc(-c2ccncc2)n1CCCN c1(C(=O)NCC(CCNC(Cn2c(=O)ccc(C)c2)=O)O)cccn2ccnc12 c1(C(=O)NCCC2CN(C(c3csnc3Cl)=O)CCO2)cc2c(Cl)cccn2n1 N1(C(c2c(C)ocn2)=O)CC(C)(C)CC1C(N1CCC(F)(CF)C1)=O c1(C(N2CCOC(CNC(c3cccc(F)c3)=O)C2)C(=O)O)cccc(F)c1 CC1CN(C(=O)CCn2ccnn2)CCC1CNC(=O)C(F)(F)C1(O)CCC1 Cc1ccc(CC(=O)NCC2(F)CN(C(=O)C(C)Oc3cccnc3)C2)c(Cl)c1 C1(C)(CNC(C2CCCN(C(c3c(C)n(C)nn3)=O)C2)=O)CC2CCC1C2 C(CC(O)C(=O)NCCNC(C1CCCCN1C(C1CCCCCC1)=O)=O)SC c1(C(=O)NCC(C)NC(=O)C(C(C)(C)C)NC(N)=O)cnc2ccccc2c1 c1(C(=O)NCCCN(C)C(c2cnns2)=O)cc(C2CC2)nc2ccc(Cl)cc12 C(C(C)C)(C(C)(C)C#N)NC1CC(C)(SC)C1 c1(C(=O)OC)ccc2nc(C(=O)NC3(CN(C(C)=O)C(C)C)CC3)c(F)n2c1 c1(OC(C)C)ccc(F)cc1C(=O)NCC12CCC(CC1)N2C(C1CC1(F)F)=O c1(N(CC(CC)OC)C)ncc(S(=O)(=O)NCC2COCCN2C)cc1Cl N1(C(c2ccc(N)c(N)n2)=O)CCC2CN(C(c3cc(C(F)F)cs3)=O)CC12 c1(C(N2CCCC(CCNC(CNS(C)(=O)=O)=O)C2)=O)cc(Cl)c(F)cc1F CCCCC(C)CCC(=O)NCC1CC(CC(N2CCC(C)(CCO)C2)=O)C1 CCCCCC(C)(C)C(=O)NC(C1CCCCN1C(c1cnncc1O)=O)C N1(C(N(C)C)=O)CC(NC(=O)CC(F)(F)Br)C(C)C1 Cc1ccc(C(F)C(=O)NCC(CNC(=O)CN2CCSCC2)CO)cc1 N(S(=O)(=O)N1CCN(C(C2CCN(C)C2c2ccccc2)=O)CC1)(CC)CC C(C(C(=O)N1CC2(CNC(=O)O2)C1)C(C)(C)C)OCCOC C1(C2CCOCC2)(NC(C2C(C)(C)C(NC(c3cc(Cl)ns3)=O)C2)=O)CC1 CC(C)C(C#N)C(=O)N1CC(NC(=O)CC(c2cccc(F)c2)O)C1 c1(C(C)C)conc1C(=O)NC1CN(C(c2ncoc2-c2cccs2)=O)C1 C1(NC(CN(C(CC2(C(C)OC)CC2)=O)CCO)=O)CN(C2CCC2)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCN(C(C=Cc2scc(C)n2)=O)CC1 O=C1CNC(=O)C(CC(N2CCC2CNC(C2CC=CCC2)=O)=O)N1 c1(NC(C2C(OC)CCC2)=O)ccc(NC(=O)Cc2cc[nH]c(=N)c2)cc1C Cc1cnsc1C(=O)NC(C)(CNC(C1CN(c2nnnn2C)C1)=O)C1CCC1 C(=O)(C(O)CN1CCCC1)NC(CNC(C1(SCC)CC1)=O)C1CC1 c1(C(N2CC=CC(NC(C(CCCC)C)=O)C2)=O)cnn2cccc(Cl)c12 [N-]=[N+]=NC1CCC2(C(=O)NCC3CCC(CNC(=O)C(O)C(F)(F)F)CC3)CC12 c1(CNC(C(C)(F)F)c2ccccc2)ccc2c(c1)NC(=O)CS2 c1(C(=O)NC(CCOC)CNC(C2CC3CCC3C2)=O)n[nH]c2c1COCC2 O(P(C)(=O)CNC(C1CCCN(C(=O)Cc2ccccc2C)C1)=O)CC Cc1ccc(Cl)c2[nH]c(C(=O)NCC3COCCN3C(=O)C3=CCOCC3)cc12 N1(C(C2CCC(=C)CC2)=O)CCC2CN(C(C3CC(C(C)(C)C)=NO3)=O)CC12 c1(CC(N2CC(C)C(NC(CNC(C)=O)=O)C(C)C2)=O)c[nH]c2ccc(C)cc12 c1(C(=O)NCC2C(NC(CN(C)C)=O)CC2)csc(-c2ccoc2)n1 c1(C(=O)NCCCCNC(C2CCN(C(=O)NC)C2)=O)ccncc1Cl Cc1cn2c(n1)CC(C(N1CC3(CC3)CC1CNC(c1coc(Cl)n1)=O)=O)CC2 c1(OC)cc(C=O)c([N+](=O)[O-])cc1OCc1nc(C2CCCCO2)no1 C1(NC(CCCCNC(N)=O)=O)CCC2CN(C(=O)C(=Cc3cnc[nH]3)F)CC12 c1(C(=O)NCC(=O)NC2(C)CN(C(=O)C(F)(F)CC3CC3)C2)ccc(F)cc1 c1(CCC)cc(C(=O)NCCCCN(C)C(C2CC3C=CC2C3)=O)n(C)n1 C(=O)(C(C(C)(C)C)N(C)C)N1CC(Cn2cc(C(C)(C)OC(C)=O)nn2)C1 C1(CN(CC(C)(C)C)C)CCCN(CCc2csnn2)C1 c1(NC(C2(C)N(c3nc(C)cc(C(=O)OC)n3)CC2)=O)nccc2[nH]ccc12 C1(NC(c2c(O)nnc(C)c2C)=O)CCSC12CN(C(=O)CC1CCCCO1)C2 c1(C(N2CCN(C(c3c(COC)nn(C)c3)=O)CC2)=O)cnc2c(c1)CCCC2 C(=O)(C(C(C)C)N1CCCS1(=O)=O)NC1CCN(C(c2c(CC)csc2)=O)C1 C(=O)(C(C)C(O)C(C)C)NCCCC(CCC)NC(=O)Cn1cnnn1 c1(CC)ccc(C)cc1C(=O)NCC1(C)CCN(C(=O)CCNS(=O)(=O)CC)C1 c1(SC)nc(Cl)c(NC(C2CCCN2C(c2cc(Br)c(C)c(Br)c2)=O)=O)c(Cl)n1 CCC(C)C(O)C(C)C(=O)NC1CCC1C(=O)Nc1cccc(O)c1 N1(C(C(c2ccc(F)cc2)C)=O)CC(NC(c2ccnn2C)=O)CC2(CC2)C1 n1(CCC)cc(C(=O)NCCCN(C)C(C2(COC)CC2)=O)nn1 C1(OC)CCCN(C(C2(C)CC3CC3C2)=O)C1 C1(C(=O)OC)CCN(C(=O)C(C2CCN(C(=O)C=C3CCOCC3)C2)C)CC1 c1(NC(N2CCC(CC(=O)OC)C2)=O)ccc(Br)cc1Cl N1(C(C2(C)COC2)=O)CC2CC2C1C(=O)NCCN1CCCC1=O N1(CC(c2cccc(OC)c2)=O)CC2(CCCC2)C1C(C)C Cc1ccc2c(c1)CN(c1nccc3sc(C)nc13)CCO2 N1(C(CC(=O)NCC)=O)CCC(C(N2CCC3CCC23)=O)(CO)C1 C(=O)(CC(O)CC(C)(C)C)N1CCN(C(Cc2ccc(C)o2)=O)CC1CCO N1(C(CC)C(=O)NC(C)C)CCC2(CC1)CC2NC(C1CC=C(C(C)C)CC1)=O C1(CNC(C(c2ccccc2)C)=O)CCCN1C(=O)CCn1cccn1 C1(COC)(NC(c2ccc[nH]2)=O)CCN(C(c2cnc(O)n2C)=O)CC1 C1(CC)CN(c2ncccn2)CCN1Cc1cc(Br)cs1.c1ccc(C(C)C)cc1 C(CC(=O)NCC1CC(C)(C)CN1C(c1cc(Cl)n(C)n1)=O)(C(C)C)OCC N1(C(c2ccnn2CC(F)F)C(=O)NCCC(=O)OCC)CC(C)S(=O)C(C)C1 c1(CC)c(C(=O)NCC(c2ccccc2)NC(=O)CC(F)(F)F)nnn1CC C1(NC(C2(CC)CC2)=O)COC2(CCCN(C(=O)C=Cc3cncc(F)c3)C2)C1 N1(C(c2ccn(CF)n2)=O)CCC2(CCCN2C(c2ccc(C(F)(F)F)o2)=O)C1 N1(C(C(C=C)C)=O)CC(NC(=O)CC(C)CN(C)C)C(F)C1 Cc1cccc2cc(C(=O)NC3CCCC3c3cccc(Br)c3)nn12 C(CCC(C(=O)NCCC1CC1)N1CCC(c2nnn(C)n2)CC1)OCC=C N1(C(C2CC(C#C)(O)C2)=O)CCC(C)C(CNC(=O)C(N2CCCC(C)C2)=O)C1 C1(NC(CCc2cc(C)on2)=O)CCC(F)(CNC(=O)C(=O)NCC(F)(F)F)C1 c1(NS(C)(=O)=O)cc(C(=O)NC2CC(F)(CNC(=O)CCC(F)(F)F)C2)ccc1F C(CC(N)=O)(C(=O)NC1CCC(CNC(N)=O)CC1)NC(CNC(CC)=O)=O C(CCCCC(=O)NC(c1cnc(C)s1)C)NC(C1CC=C(C)CC1)=O N1(C(CC(=O)OC)=O)CCC2(CCC(NC(C3(C)CC(C4CC4)=NO3)=O)CC2)C1 C1(CCN(C)C(C2CC2(C)C)=O)CCCCN1C(=O)CCc1cnco1 Fc1cc(-n2nc(-c3ccc(Cl)cn3)nc2-c2n[nH]cc2Br)ccn1 c1(C(=O)NC2C(C)CN(C(=O)CC3CCCOC3)C2)ccccc1[N+](=O)[O-] Cc1cnn(C)c1CC(=O)NC(C)CC(C)NC(=O)Cc1cc[nH]c1 CCCCC(CCCC)NC(=O)C(CC(C)(C)C)OC.N12CC(OC)CC1C2=O Cc1c(C2C(C(=O)N=c3[nH][nH]cc3Br)C2)ccc(-c2cnn(C3CCCC3)c2)c1F C(=O)(C1=CC2(CCOC2)C1)Nc1cccc(NC(C(C)Cc2cnco2)=O)c1 N1(C(C(CNC(C2(CC(C)=O)CC2)=O)N(C)C)=O)CCCC(O)C1 Cc1c(C(=O)Nc2cccc(-n3cc(-c4c[nH]nc4C(=O)O)nn3)c2)cnn1C C(=O)(CCCCC#N)NCCOC1CN(C(C(C2CCCN(C)C2)(C)C)=O)C1 CCN=C(NCC1C(C)C1(F)F)NCC1(C2CC2)CC1 C1(NC(C2(COC)CCC2)=O)CCN(C(=O)CNS(=O)(=O)C2CC2)C1 CC(C)CC(C)CNC(=O)C(O)CCNC(c1cn(CCO)nn1)=O C1(C(N(CCCCNC(=O)CCNC(c2ccoc2)=O)C)=O)CCCC12CC2 c1(OCC)ncc(NC(=O)C(C2CCCN(C(=O)CC3(N(C)C)CC3)C2)C)cn1 C1(CNC(CN(C)C(N)=O)=O)CCCC1C(=O)NC1CCC(N(C)C)C1 C1(CNC(C(COC)(C)O)=O)N(C(c2sc(C)cc2Cl)=O)CCC1(C)C C1(C(=O)NC2(CNC(c3n(C(C)C)ccc3)=O)CC2)CC(c2ccncc2)=NO1 N(C(=NCCN=c1cncc[nH]1)NCC1(CO)CCCC1)C(COC)C C1(C)(C(N2C(CCC)CN(C(=O)C(C)C(C)(C)C)CC2)=O)CCC2(CC1)CC2 CCC(C)C(CC(=O)N(C1CC(C(N)=O)C1)C)NC(=O)CC1CCCO1 C(=O)(C(C(C)(C)C)C1CCCC1)NC(CNC(CC1(OC)CCCCC1)=O)C CC(C)S(=O)(=O)C(C)C(=O)N1CCOCC1CNC(c1cnc(S)[nH]1)=O C(=O)(C1c2ccccc2CN1Cc1cc(Br)ccc1OC)N(CC=C)CC1CC1 c1(OC)nccc(C(=O)NCC(CO)NC(=O)CNC(=O)CC(F)(F)F)c1F N1(C(CC=C=C)=O)CC2(C(N3CCC(CC)C3)=O)CC1CCO2 c1(C(=O)NCC(C)CN(C(=O)Cc2cncs2)C)ccnc(S)c1 C1(NC(C2CC(C)(NC(C(c3ccn(C)n3)C)=O)C2)=O)C=C(C)CCC1 CCC(COC)C(=O)N1CCC(OCC(=O)NCC2(O)CC=CC2)C1 N1(C(C2N(C)CCC2)=O)CC(F)(F)CC1(C)CNC(=O)C(C)(C)C(N)=O n1(C(C)C)ncc(C(N2CC(N(C(=O)CCC3CC3)C)C(F)C2)=O)c1N C1(C(=O)NC2(CNC(c3ccsc3C(F)F)=O)CCOC2)CC2COCC2C1 O=C(CCCC#Cc1ccccc1)NC1CC1NC(C1CC12CC2)=O C12(NC(=O)NCCS(=O)(=O)NCC3CC3)CC1COC21CCC1 C(=O)(C(C)(C)n1ccnn1)NCCN(C(=O)Cc1cnc(C(F)(F)F)s1)CC c1(OC)ccc(C)nc1C(N1CCN(CC(C)(C)NC(C2CCCS2)=O)CC1)=O CC1=C(C(=O)NC2COCC2CNC(c2oc(CO)nc2C)=O)C(C)(C)CCC1 N1(C(c2c(NCC)cccn2)=O)CC(C)N(C(=O)C(C)=C2CC2)CC1C Cc1cc(C(=O)NCC2(C)CCCN2C(=O)C(F)F)c2cc(Br)ccc2n1 C#Cc1cccc(CC(=O)NC(CC(=O)NC(C)(CO)CO)C(C)OC)c1 c1(CC)cc(C(=O)NC2CC(CNC(C3CC4CCC3CC4)=O)C2)cn(C)c1=O N1(C(c2ccc(C)c(Cl)c2Cl)=O)CCC2CN(C(C3(C)CC3(F)F)=O)CC2C1 Cc1cc(C(=O)NCCCC(C)NC(=O)CC2CSCCO2)cc(C)c1C#N N1(C(CCCNC(CC=C)=O)=O)CC(NC(=O)C(CC)CCC)C2(CCCC2)C1 CC1CCC(C(=O)NCC(C)(C)N(C)C)O1.C12CC1CC(=O)N2 N1(C(C(CC)N(C)C)=O)C(C)CC2CN(C(C3CCC(C(=O)OC)CC3)=O)CC12 c1(CN(C)C(C2C(CNC(=O)CCc3ccnn3C)C2(C)C)=O)ncccn1 c1(OC)cc(C)c(C(=O)NC2CCOCC2NC(=O)CN2CCC(O)CC2)cn1 N1(C(CCC2(C)CC2(F)F)=O)CC2(CCC2NC(=O)Cc2nnc(O)s2)C1 C1(NC(C2N(C(C)(C)C)CC2)=O)CCC(CC(=O)NC2(C(O)CO)CC2)CC1 c1(C2N(C(C(C3CC3)NC(C(C)n3ccnn3)=O)=O)CC2)ccccc1 N=c1[nH]c(=NCC2(CO)CCCCC2)[nH]c(=NCCC(O)C2CCC2)[nH]1 CCC(C)CCC(=O)N1CC=CC1(C)C(=O)N(C)CC1CCSC1 Cc1nc(C)c(-c2ccc(CN3CCCC3(C)c3ccccc3)s2)s1 C1(C(=O)NC(CC=C)CO)CC(C)(C)CN1C(c1ccc(F)s1)=O C1(C)(CCNC(C2CCC(C)(CC)O2)=O)CCN(C(c2nc(=N)cc[nH]2)=O)CC1 CC1COC2(C1)CN(C(=O)C1=CCN(C(C3COCC3C(N)=O)=O)C1)C2 N1(C(c2c(C)cc(C)s2)=O)CC2CCC(C1CO)N2C(=O)C(C)n1cccn1 C1(COC)(CNC(c2cc(C)ns2)=O)CCCN1C(c1nc(O)sc1C)=O O=C1CN(C(C2(C(=O)O)CCOCC2)=O)CCN1Cc1ccccn1 c1(C(C(=O)NCCC)N(C(C)C(=O)OC)C)sc(Br)nc1Cl C1(C(N(CC(C)CNC(=O)C(C)(C)OCC(F)(F)F)C)=O)COCC2(CCC2)O1 Cc1nc([N+](=O)[O-])cn1CC(N1CC2CCC1C(NC(=O)CN(C)C(N)=O)C2)=O c1(C(=O)NC(C(C)C)CCNC(C2(S(N)(=O)=O)CC2)=O)ccc(N)c(Cl)c1 c1(C(=O)NC(CCC)C)c(C)[nH]c(C(=O)ONC(=O)C(C)NC)c1C C(=O)(CCCC(C)(C)CC)NC(CC)CNC(=O)Cn1nnc(C)n1 CC(CO)(C(=O)N1CC(c2cc(O)no2)C1)NC(C1COCOC1)=O c1(C(N2CCCC(NC(COC(C)=O)=O)CC2)=O)ccc(Cl)c2ccccc12 C(=O)(CC(F)(F)F)Oc1ccccc1.N12CCCC1CNCC=CCNC2=O N1(C(c2cnc(C)s2)=O)CC(NC(=O)Cc2coc3ccccc23)C(C2CC2)C1 CC1CC2CN(CCN)CC2N1C(=O)C(N1CCc2ccccc2C1)CCC1CC1 CCC(CC)(C(=O)N1CCC(O)(CN(C)C(c2nnn(C)c2N)=O)CC1)OC CCCCCC(O)CC(=O)N1CCOCC1CN(C(=O)C(c1ccccc1)C)C C1(C(=O)NC23CC(C(=O)NCC(CC)CO)(C2)C3)CCC=CCC1 C(CCC(=O)N1CCCC1CCCNC(=O)COCC(F)F)NC(C)=O N1(CC)CCC2=C(C1=O)C(c1ccc(Br)cc1Br)NC(=O)N2CCF c1(OC)ccc(NC(C2CCCCC2NC(C2(C(F)(F)F)CCC2)=O)=O)nc1C C1(F)(C(=O)NCCCCCNC(C(CC)=CCCC)=O)CCCCC1 Cc1cc(C(=O)NC(C2CCN(C(c3occc3C)=O)C2)C)cs1 c1(C(=O)NC2CCC(CNC(C3CC(N(C)C)C3)=O)C2)cncc(F)c1Cl CCC(C)(O)C(=O)NC1CCN(C(=O)C=CC2C(C)C2(Cl)Cl)CC1 C1(NC(c2c(C)[nH]cc2)=O)CCOCC1C(=O)NOCC(C)(C)O C1(O)(CN(C(CCC=C)=O)C)CCCN(C(C23CCC(CC2)C3)=O)C1 c1(C(=O)NC2CCN(C(C3C(F)(F)C34CC4)=O)C2C2CC2)cc2cccn2cn1 N1(C(C(C2CCC2)NC(CCCOCC)=O)=O)CC(N(C)C)C(C)C1 N1(C(C(C2(O)CN(C(=O)CCc3nncs3)C2)F)=O)CCC(F)(F)CC1 c1(COC)cc(CN2CCC(O)CC2C(=O)NCC2CNC(=O)CO2)cc(Br)c1 C(=O)(C1CCc2cc(F)ccc21)NCCOCCN1CCN(C(C)=O)CC1 C1(C)(C(=O)NCC(CN(C(CC2N(CC)CCC2)=O)C)(C)C)CCOCC1 c1(C(C)C)ccc(C(=O)NCCCCN(C(=O)Cn2cncn2)C)cc1[N+](=O)[O-] C1(OC)CC2(C1)CC(C(=O)NC(CNC(=O)CN1CCC(CO)CC1)CO)C2 C1(C)(C(N(C(C)C)CCNC(c2c[nH]ccc2=N)=O)=O)CCCC1(F)F C1(CN(C(=O)CC2CC(c3ccccc3)C2)C)COCCN1C(C1CCCO1)=O CC1=NOC(C(=O)NCCOCCN(C)C(c2cccc(CF)c2)=O)C1C c1(C(N2CCN(CC=C)CC2)=O)coc2c1CN(C(=O)CC1CC(O)C1(C)C)C2 c1(C(=O)NCC(CN(C(CC)=O)C)C)nc(OC)ccc1C Cn1nc(C(=O)NCC2CCC2NC(=O)COC(=O)CO)c2cc(F)ccc12 C#CCC(C)(C)C(=O)NC1CC(O)CN(C(c2cnncc2C)=O)C1 C1(CC(=O)N(C(C)C)CCN(C)C(c2csnn2)=O)CC2(CC2)C1 C1(C(=O)NC(CC=C)C(=O)N2CC(CO)C(O)C2)CCC(C)(O)CC1 C1(NC(C2(CC)CCN(C(C3C4CCCCC34)=O)C2)=O)CCC(=O)NC1C CC1C(N(C)C)CCN1C(=O)CONC(c1ccncc1)=O C1(C(=O)NC(CCCC)CNC(C2CNC(=O)N2)=O)C2Cc3cc(Cl)ccc3C12 N1(C(C(C)Sc2ccccc2)=O)CCC(CCNC(c2snc(Cl)c2Cl)=O)CC1 Cc1ccc(SCC(=O)NCCC(O)CNC(C2C3CCCCC23)=O)cc1 C(N=c1ccn2nccc2[nH]1)C1N(C(c2ccc([N+](=O)[O-])s2)=O)CCC1 C1(NC(COC(CC)C)=O)CC2CCC1(C(=O)NCC1C(C)(C)C1(C)C)C2 C(N=c1nc(N2CCC(c3ccncc3)C2)c2c([nH]1)CCCC2)C1(C)CC(C)C1 C(=O)(C(CNC(c1cc(C)cc(F)c1)=O)CC(C)C)NCc1cc(CC)on1 C1(NC(C(CC=C)C)=O)CCCN(C(C23CCC(C2)OC3)=O)C1C C1(C(N(C)Cc2c(C)cncc2)=O)CN(C(c2cn(C)cn2)=O)C(C)(C)C1 c1(CC)nc(C)[nH]c1C(=O)NCCC1CC(NC(c2ccc(C3CC3C)o2)=O)C1 C1(CNC(C2C(C(=O)OC)C2)=O)CN(C)CCN1C(C1(CSC)CC1)=O n1(C(C)(C)C)nnnc1C(C)(CCc1ccccc1)NCCC12CCCC1C2 c1(OC)cc(CC(=O)NCc2cc(C(C)(C)C)ccn2)c(F)cc1O C1(NC(=O)C=Cc2cccnc2)CCN(C(C2CC3(C2)CC(O)C3)=O)C12CCC2 N1(C(=O)OC(C)(C)C)CCN(Cc2ccccc2)CC1Cc1snc(Cl)c1Cl C1(C(N2CCC(C(=O)N(C)CC3CC3(C)C)(OC)C2)=O)CC2(CC2)CN1C C(=O)(C(=O)NCCC(=O)N(C)Cc1nc[nH]n1)NC(C)C CC1CCN(C(=O)CN(C2CCSC2)C)CC1N(C(=O)CC1(N(C)C)CCC1)C C(=O)(CC(C)CN=c1[nH]c(=NCc2c(C)cc(C)n(C)c2=O)[nH]c2c1SCC2)NC Nc1cc(C(=O)NCCC2(O)CN(C(C3CCC(C(N)=O)C3)=O)C2)cnc1Cl C1(NC(CCC(CC)NC(C2CC2(F)Cl)=O)=O)CCC(=O)N(C)C1=O N1(C(C2(CC#C)CCCC2)=O)CCCC(C(=O)NCCC(=O)N(C)C)CC1 Cc1ccc(C)c2[nH]c(C(=O)OCCCC(Cl)Cl)cc12 N1(C(C(CN(C)C)NC(c2nc(Cl)cs2)=O)=O)CC2C(C1)C2(F)F N1(C(C=C(CC)CC)=O)CCC(N(C(=O)COCC(F)(F)F)CCO)C1 C1(CNC(C=C(COC)C)=O)CC2CCC1N2C(c1csc(C(C)(C)C)n1)=O c1(NC2(CNC(CC=CC=C)=O)CCCC2)nc(C)nc2c1cnn2C C(=O)(C1=CCC(F)(F)CC1)N(C(C)C)CCN(C(=O)CCC1CC1)C C1(NC(CCCCC#C)=O)C2CC(O)C1N(C(C1CCCC(O)C1)=O)C2 N1(C(c2n(CC)nnc2)=O)CCCC2CN(C(c3cccn4ncnc34)=O)CC12 C1(C(=O)NC2C(C(C)(C)C)C2)OCCC1NC(C1CC2(CC2)C1)=O C(C(C)NC(=O)C=Cc1cncs1)(C(C)C)NC(COCCCOC)=O C1(C(=O)NCC2N(C(CCC(=O)NCCC)=O)CC(OC)C2)CCCCS1(=O)=O C(c1ccc(Br)s1)=CC(=O)N(C(C)CNC(=O)CC1OCCCO1)C C1(NC(C2N(S(C)(=O)=O)CCCC2)=O)CN(C(=O)C2=COCCC2)CCC1(F)F C12(C(=O)NCCC(CNC(=O)C3=CCCCC3)O)CCC(CO)(CC1)CC2 C1(NC(c2n(CC)nnn2)c2cnn(-c3ccc(C)cc3)c2)CC12CC(O)C2 N1(C(c2cn(CCCC)nc2C)=O)CC2CC1CCN2C(C1CCN1CC)=O c1(C(=O)NC(CCN(C(C2(CC)CCNC2=O)=O)C)(C)C)cn2cccnc2n1 N1(C(C(SC)SC)=O)CC2(C(=O)NCC(N3CC=CC3)=O)CCC1CC2 N(C(=NCc1ccc(OC(F)(F)F)cc1)NCC1CCSC1)C(CC)C c1(C(=O)NCC(C2CC2)NC(C(=O)NCCOC)=O)cc(S(C)(=O)=O)cnc1O CC(C)CC(F)C(=O)NC(C1CN(C(=O)C(F)(F)F)CC1(C)C)C1(O)CCCC1(C)C C1(CC(=O)N(C(CC)CNC(c2ccn(C(C)C)n2)=O)C)CN(CC)CCO1 c1(CC(=O)NC2CCC(NC(c3ccc(CC)[nH]3)=O)CC2)c(C)nc(O)nc1O CC(Cc1cnn(C)c1)C(=O)NC(c1nc(C2CC2)n[nH]1)C c1(C(=O)OC)ncc(C(=O)NCC2COCC2NC(C2(F)CC2)=O)s1 c1(OC(C)C(=O)NC2CC(Cn3cc(CC(C)O)nn3)C2)ccccc1Cl C(CC(C)C(=O)N1CCC(N(C(=O)CCC=C(C)C)CCC)C1)=CC N1(C(C2CN(CCC)C(=O)C2)=O)CCC(CNC(=O)CCF)C12CCC2 C(=O)(C1=CCOCC1)N1CCC(NC(c2n[nH]cc2C2CCC2)=O)C1 n1(CCC(=O)NCC2CCC(NC(C(COC)N(C)C)=O)C2)ccc(O)nc1=O c1(C(=O)OC)cccc2c1CCCC2NCC(C)(C)OCC(=O)OC Cc1cc(F)cc(C(=O)N(C)CCN(C(=O)CC2=CCOCC2)C(C)C)c1N N1(C(C2C(C(N)=O)CCC2)=O)CCC(=CCNC(C2CC(=O)N2)=O)CC1 c1(CN(C=O)CC(=O)N(CC(F)F)C2CC2)ccc(F)c(Cl)c1 C=CCC(C)(CC)C(=O)NC1CC2(C1)CC2C(N1CCCCCCC1)=O C(=O)(CC(O)C(C)C)NC(CC)CNC(C1CC2CC1C2)=O N1(C(CCOCCOCC)=O)CCOCC1CNC(c1cc(C)nn1C1CC1)=O C1(C(=O)Nc2ccc(OC(C(=O)OC)C)cc2)Cc2nccnc2C1 Cc1ccc(C(C)(C)CC(=O)NCC23CC2CCN3C(=O)CC#N)cc1 C(CC(C(=O)N(C)Cc1ccc(C)cc1)NC(C1CC1(C)C)=O)SC N1(C(C(CC)=CC)=O)CC(C(=O)NCC2CC2)C(CC)C1.C1C(=O)O1 C(CCCCC(=O)NC(CNC(=O)CC(O)Cc1ccccc1)C(C)C)OC C1(CNC(c2c(C(=O)OC)cccc2)=O)CCN(C(=O)C(C)(C)CSC)CC1O N1(C(CN(C(COC)=O)C)=O)CCN(C(=O)CCNC(=O)C=CCl)CC1C Cc1ccc(NC(=O)N(c2ccccn2)C2COC2)c(CO)c1 N1(C(C(C)(N(C(c2[nH]cc(C)c2)=O)C)C2CC2)=O)CCC2(C1)CC2(F)F CCCCS(=O)(=O)NC(C)C(N1CCC(NC(=O)COC(C)=O)C1C(C)(C)C)=O CCCC(CC(C)C)C(=O)NCC(C)(CNC(=O)Cc1ccccc1C)OC C12COCCN(C1)C2=O.C1(N(C(=O)C(=O)Nc2ccccc2)C)CCCC1C n1(CCC)nccc1C(=O)N(C1CCC(NC(=O)C(F)(F)c2cnccn2)C1)C c1(CNC(C2(CNC(c3ccccn3)=O)CCC2)=O)ccccc1O Cc1ccc(C)c(OCCCOC(c2c(CN)n[nH]c2C)=O)c1 CCC(C)(CC)C(=O)NCC1CC(F)(F)CN1C(=O)CNS(=O)(=O)NC C(N=c1cc(C(C)=O)c([N+](=O)[O-])c[nH]1)C1CCCN(C(C2C(C)(CC)C2)=O)C1 c1(CC)ccc(C(=O)NC2CCC(CNC(C3(C)CC=CCC3)=O)C2)cc1C C1(CNC(CC2C(C)(C)C2(C)C)=O)CC2COCC2N1C(=O)Cc1cnsc1 N1(C(C(C)=CC)=O)CC2(C1)CN(c1ccc(NC(=O)OC(C)(C)C)cn1)C2 Cc1cscc1C(=O)NCC(C1CC1)N(C(=O)Cc1ccc(Br)s1)C c1(C(N2C(CNC(=O)CCC3CC3)CC(OC)C2)=O)c[nH]c2ccc(O)cc12 CCC(C)CCC(O)CC(=O)N1CCN(C(C2(N(C)C)CC2)=O)CC1C c1(C(=O)NC2C(C)CCN(C(CCOCCOC)=O)C2)n[nH]c2c1CCCCC2 c1(COC)nc(N(C)CC2CCCN(C(=O)CCn3cc(Cl)cn3)C2)cc(C)n1 C1(NC(C(CC)n2nccc2C)=O)COCCN(C(c2cc(C3CC3)[nH]n2)=O)C1 N1(C(Cc2c(C)nc[nH]2)=O)CCOCC1CCNC(C12CCC(C1)OC2)=O c1(NC(C2(CC=C)CCCN2C(=O)C(C)CCCOC)=O)cc(C)ccc1C c1(CNC2CCC(NC(c3c(C)cc(F)cc3C)=O)C2)ccc2nccnc2c1 C12(NC(=O)Cc3ccno3)CCCC1CN(C(c1cc(C(F)(F)F)on1)=O)C2 Cc1cc(C(=O)N(C(C)C(=O)NCC2(N(C)C)CCOC2)C)c(N)s1 C1(C(N(CC(=O)NC2CC(F)C2)CCC)=O)CCCCC1OC c1(C(=O)NC(CNC(C(C)SC)=O)CC(C)C)ccn2cccc2c1 CC1CCN(C(=O)CC(C)(C)C2CC2)CC1CNC(=O)CNC(=O)C(C)(C)C C1(C2CCCCN2C(=O)Cc2ccco2)(CNC(CC(C)SC)=O)CCOCC1 CC(C)CC(C(=O)NCCCCNC(C1CCCN1C=O)=O)N1CCCCC1=O c1(OC)c[nH]c(C(N2CCC(N(C)C(C3CCC(=O)C3)=O)C2)=O)cc1=O C1(NC(c2c(C)sc(Cl)n2)=O)CCN(C(=O)C(C(C)C)N(C)C)CCC1(F)F Nc1cccn(CC(=O)NC(CNC(C23CSCC2C3)=O)CC(F)(F)F)c1=O C1(C(=O)NCC(CNC(c2ccnn2C2CCCC2)=O)O)Cc2ccccc2N1 N1(C(Cn2ccc(C(=O)OC)n2)=O)CCC(F)C(NC(c2cc(Cl)c[nH]2)=O)C1 C1(NC(C23N(C(C(CCC)N(C)C)=O)CC(C)(C2)C3)=O)CC(C)(C)OC1(C)C N1(C(Cc2ccc(C)o2)=O)CCC(O)C(NC(=O)Cc2sc(C)nc2C)C1 C1(CNC(Cc2c(C)occ2)=O)CCCC(NC(C2CC2c2cccnc2)=O)C1 C1(C(=O)NC2CC(NC(c3cc(SC)oc3)=O)C(O)C2)CCC(=O)N(C)C1 C(=O)(NN1CCCC1N(C(C)=O)C)c1cc(C(N2CCCC(F)CC2)=O)[nH]n1 n1(C(CC(=O)NC(CC)CNC(=O)CCN2CCC2)C)nc(C)cc1C c1(C(N2C(COC)(CNC(=O)CC(C)C(C)C)CCC2)=O)ncn2ccccc12 C1(C(=O)NC(CCC)C2CCCC2)(CNC(=O)COC2CCC2)CC(C)(C)C1 c1(NC(C)C)cc(C(=O)N(C)CCN(C(=O)C2=COCC2)C(C)C)ccc1F CCC(C)CCCCC(=O)NC1CC2CC1N(C(C1(C(F)F)CCC1)=O)C2 C1(O)(CCNC(C(C)c2cccs2)=O)CCN(C(=O)Cc2nncn2C)CC1 c1(C(CC)NCC(C)C(F)F)ccccc1OC c1(C(=O)Nc2nc(C)c(CN)s2)cc2n(n1)CCCC2 C1(CC#C)(C(=O)NC(CNC(=O)C(=O)NC2CC2)CCC)CC=CCC1 c1(CNC(CC2C(CC)C2)=O)ccc(C(=O)NCCC2(C)CCOC2)s1 C1(C(N2CCC(CCCNC(C(C3CC3)OC)=O)CC2)=O)CC2OC(=O)OC2C1 c1(C(=O)NC(C)CCNC(C2(C)CCCC2(F)F)=O)n[nH]c2ccccc12 c1(C(N(CC(C)NC(=O)CC(O)C2CC2)C)=O)cc(C(N)=O)co1 C(=O)(C1CCN(C)c2ccccc21)NCC(C)NC(C1(COC)CCCO1)=O N1(C(=O)C=CSc2nc[nH]n2)CCC2(C1)CN(C(C1(F)CCCOC1)=O)CCO2 NS(=O)(=O)c1ccc(F)c(C(N2CCC(C3CC3)(NC(=O)C=CCO)C2)=O)c1 CCC(CN(C)C)CC(=O)N1CCC(CNC(C2CCCCN2C(C)C)=O)C1 c1(C(=O)NCC(C2N(C(C3CC(C)(F)C3)=O)CCC2)(C)C)ccnc2cc[nH]c12 c1(CCC(=O)NC(C)CCN(C(=O)C(C)NC(N)=O)C)ccc(N(C)C)nc1 c1(C(=O)NCCN(CCC)C(c2cccc(CC)c2)=O)ccc2nccn2c1 Cc1c(C(=O)NCC2(C(=O)NC3CCCC(O)C3)CC=CC2)[nH]ccc1=O c1(C(N2CC(NC(c3cc(C)n(C)n3)=O)C(C)C2)=O)ccc([N+](=O)[O-])cn1 C1(C(C)NC(Cc2c(C)con2)=O)CCN(C(=O)C(C(C)C)n2cccc2)CC1 C1(NC(c2cc(C(F)(F)F)ccc2F)=O)C2CC(O)C1N(C(c1cnns1)=O)C2 C1(NC(c2c(CC)c(C)sc2)=O)CC2(C1)CC(NC(c1ccnn1CC)=O)C2 C1(CC=C)CCCC1NC(C1CC1CNC(=O)CC1CCSC1)=O C(=O)(C(O)(C(C)C)C(F)(F)F)N1CC(CCNC(C(C=C)(C)C)=O)OCC1 C(CCCC(C)NC(=O)C(COC)NC(C)=O)NC(COCCOC)=O C=CC(CC)CC(=O)N1C2CCC1C(CNC(C1(NC(C)C)CC1)=O)C2 N1(CC)CCOCC1C(=O)NC1(CCCC(=O)N2CCC(C(C)C)C2)CCC1 C1(CC)CCC(C(=O)NC(C(=O)NCCNS(C)(=O)=O)c2ccoc2)O1 c1(C(=O)NC2C=CC(CC(=O)NCC3(CO)CC(C)(C)C3)C2)cncc(C#N)c1 N1(C(C2C(C)CCS2)=O)CCC2(CCC(NC(=O)CCC3(C)CC3)C2)C1 c1(OC)cc(Cl)c(C(=O)NC2CN(C(C3CCCCC(F)(F)C3)=O)C2)cc1Cl C1(CC(N2CC3C(CNC(C4(CCC=C)CC4)=O)C3C2)=O)CCCCC1(C)C CC1(C)C(C(N2CC=C(CCNC(c3ccnnc3Cl)=O)CC2)=O)CCS1(=O)=O C1(OC)CC2CC(NC(=O)C(C)N(C(=O)CCc3cnn(C)c3)C)CC12 CCCC(C)(C)C(=O)NCC(C)NC(=O)C(C)(O)CCC C=CCCCCC(=O)N1CCOCC1C(=O)NC1CCC(O)C1 CC1(C)C(NC(c2ccc(Cl)cc2)=O)C2CCCN(C(=O)C(F)n3cccn3)C12 CN1CCN(C(C2CCN(C(=O)c3cc([N+](=O)[O-])n[nH]3)O2)=O)CC(O)C1 C1(NC(=O)CCc2cncnc2)COC2(CCN(C(=O)C=CCF)CC2)C1 C1(CC(=O)NCC=CC(=O)NCC(C)CC2CC2)COCCO1 N1(C(C(=O)NC(C)C)=O)CCCC(CCNC(=O)C(c2cncn2C)N(C)C)C1 c1(C(=O)NCC(C)N(C(=O)C2=CC(O)CCC2)C)c[nH]c2cc(F)c(F)cc12 C1(NC(CC=Cc2ccc(C)cc2)=O)CCC(O)CN(C(=O)C(F)(F)C(F)F)C1 Cc1ccc(C(N2CCC(OCCNC(=O)CCC3CCC3)C2)=O)c(N=[N+]=[N-])c1 C1(C(N2CCC(C)(CNC(=O)CCc3cc(Cl)no3)C2)=O)CCCCC1(F)F c1(C(=O)NC2C(NC(c3ccco3)=O)COC2)ccc(N2CCCC2)nc1 c1(N2CC3C(F)(F)C3C2)nc(N2CCCC(C3CCC3)CC2)nc2ccccc12 C(=O)(C1=CC2C=CC1C2)NCCOCCNC(C(C)S(N)(=O)=O)=O CC1CC(NC(=O)CCC=CBr)CCN1C(=O)CC1CC2(CC2)CO1 N1(C(C(N2CCN(C)CC2)(C)C)=O)CC2CN(C(=O)Cc3cn[nH]c3)CC2(C)C1 CC(=O)C(C)CC(C)C(=O)NC12CCC1CN(C(=O)CCCC(C)C)C2 c1(C(N(C(CN(C(CC2N(CC)C(=O)CC2)=O)C)C)C)=O)cnc(C)c(C)c1 n1(CC(=O)NCCCN(C(CC=C=C)=O)C)ccc(=O)n(C)c1=O C(=O)(C1=CCCOCC1)NC1C2(CCN(C(c3c[nH]c(=N)s3)=O)C2)C1 c1(SCCCOC(C2(C(=O)OC(C)(C)C)CCCO2)=O)ccc(F)cc1 C1(C)(NC(CCN(C(=O)CSC)CC)=O)CCC(C)C1 C(N=c1[nH]c(=NCCC(C)F)c2[nH]ccc2[nH]1)c1[nH]nc(CSC)n1 c1(C(C(N2C(CCNC(CSCC)=O)CCCC2)=O)=O)c[nH]c2cc(F)ccc12 C1(NC(CC(C)CN(C)C)=O)CC2CC1CN(C(=O)CC1CSCCO1)C2 c1(C(N2C(COC)(CNC(C3CC34CCOC4)=O)CCC2)=O)ccc(C)cc1C C1(CCN(C(C2C(=C)CC2)=O)C)CCN(C(C2CCC(F)(F)C2)=O)CC1 C(=O)(CCCC(C)(C)C)N1CCCC(CC)(NC(=O)C(C)OCC(C)C)C1 C1(NC(C(CCC)=CCC)=O)CC2CCC(C1F)N2C(c1ccc(O)cc1F)=O C1(NC(=O)Cc2ccco2)CC(NC(C2CCCO2)=O)CC1O C(CC1CCc2ccccc21)N1CCC(NC(Cc2n(C)cnc2)=O)C(F)C1 C(c1ccccn1)=C(C(=O)NC(CC=C)CNC(=O)COC1CC(F)(F)C1)C Cc1c(NC(c2n[nH]cc2Br)c2nnnn2Cc2cccs2)cncc1Br N1(C(c2cc[nH]c2)=O)CC(C)CCC1C.C12(CC1)C(C)NC2=O C1(NC(c2cnc(Cl)c(Br)c2)=O)CC2CCC(C1)N2C(c1cncc(O)c1)=O Cc1nc(SC(F)(F)F)sc1.c1(CC2CCN(C(C)=O)C2)cccc(O)c1 N1(C(CCCSCCCC)=O)CCN(C(=O)CC(C)CN(C)C)CC1CO CC(F)(F)CCC(=O)NC1CN(C(c2cc(Br)c(C(F)F)s2)=O)CC1O N1(C(C2C(NC(C3(CCOC)CCC3)=O)CCCC2)=O)CC(C)CC(C)C1 C=CCC(CNC(=O)CCc1cc(C)on1)C(=O)N(CC(C)C)CCC C1(C2=CCN(C(=O)Nc3ccc(F)cc3C)CC2)(C(=O)OC)CCOCC1 Cc1ccc(F)c(C(F)(F)C(=O)NC(C)CC(C)NC(=O)CCC(=O)N(C)C)c1 C(=O)(CCCCCCn1cc(CN2CC3CC3C2)nn1)N(CCCO)C(C)C Cc1cn2c(n1)CC(C(=O)NCCOCCNC(c1cc(F)cs1)=O)CC2 C1(C)(C(=O)NCC2(CCNC(CN(CCOC)C)=O)CC2)C=CCCC1 CC(F)(C(=O)NCC(O)CCNC(=O)CCCn1ccnc1)c1ccon1 c1(C(N2C(CNCc3ccc(C)s3)C=CC2)=O)cccc(S(F)(F)(F)(F)F)c1 CC1CC(C(=O)N(C2CN(C3CC3)C2)C)CN(C(=O)CCC2OCCO2)C1 c1(C(N2CCC(O)(CNC(CSCC=C)=O)C2)=O)ccc(Cl)cc1CC CC(C)S(=O)(=O)CC(=O)N1CCCC1CN(C(=O)C(C)(C)N1CCCC1)C Cc1cnc(C(N2CCCC(F)(CNC(=O)C(C)OCCC(C)C)C2)=O)c(C)c1 c1(OC)ccc(C(=O)C(=O)NC2CCC(NC(=O)C(Br)=C(C)C)C2)cc1 Cc1cccc(C(F)(F)C(=O)NC2CC2CNC(C2COC(=O)C2)=O)c1 c1(OC)cc(C)nc(N(C2CC3(CNC3)C2)Cc2cnc(Cl)c(C)c2)n1 C1(C)(C(=O)NCC(CC)(C)O)CCN(C(=O)Cc2cc(C)no2)C1 C(=O)(CC(C)CC(C)(C)C)N1CCN(C(CC(C=C)C)=O)C(C)CC1 C(=O)(C(C)(F)C(C)(C)F)NCC1(C)CCCN(C(c2cc(CCC)on2)=O)C1 c1(N2CCC(C(=O)NCCS(=O)(=O)O)CC2)ccnc(C(=O)NC2CCCC2)n1 N1(C(=O)CCc2ccc(Br)nc2)CCC2C1CCCN2C(=O)Cc1cncnc1 CC1CC(C(=O)NCC2CN(C(c3ccnc(CO)c3)=O)C2)C(C)O1 C1(C(N(CC(=O)NC(C#C)C(C)OC)C2CC2)=O)C2CN(C)CC12 C1(NCCNC(c2ccc(C3CC3)o2)=O)CC12CCN(C(=O)CC1CC1(F)Cl)CC2 N12CC3(CC(C3)C1=O)C2.N1(C(c2ccn(CC)n2)=O)CCCC(N2CCCC2)C1 C(=O)(C1=CCCCC1)NCCC(=O)Nc1c(C(F)(F)F)nc(C)s1 C1(CNC(C(CC)SC)=O)C(C)CCN1C(C1CC(N(C)C)C1)=O N1(C(Cn2cccc(C)c2=O)=O)CC(C)CN(C(=O)C2=CCCCO2)C(C)C1 C1(NC(CN(CCC#C)C)=O)CC12CCN(C(=O)C=CSCc1ccco1)CC2 C12(C(N(CCNC(=O)CCCC(N)=O)CC)=O)CCCC(CCC1)C2O N1(C(C(c2cn(C)nc2)=O)=O)CCC2(NC(c3ccc(Cl)s3)=O)CC2C1 N1(CC(=O)NCC2CC(NC(c3ccnn3CC3CCC3)=O)C2)CCCC(O)C1 C1(NC(C2C(C)CC(C)O2)=O)CCN(C(c2cocn2)=O)CCC1CO C1(NC(C2(N(C)C)CCCCC2)=O)CC(C2CCN(C(c3ccoc3)=O)CC2)C1 c1(C(=O)NCC(CNC(C2(C(F)F)CC(=C)C2)=O)O)cn(CC)nc1C1CC1 C12(NC(Cc3n(C)ncc3)=O)CCCC1N(C(c1cn[nH]c1)=O)CCC2 c1(OC)cc(C(=O)N(CC(C)NC(c2ccc(OC3CCC3)cc2)=O)C)ccn1 C(N=c1nc(N2CCC(CC3CC3)CC2)c2c([nH]1)CCOC2)C1CC(C)(C)C1 c1(NC(C(CCSC)N(CC(C)(C)C)CC2CC2)=O)ccccc1SC N1(C(C2CN(C(C3CC(C)(CC)C3)=O)CC2(F)F)=O)CCCC(C2CC2)CC1 C(C(O)CC(=O)N(CCNC(c1ccc(F)o1)=O)CC1CC1)N(C)C Cc1cc(C)nc(SCC(=O)N(C)CCNC(c2cc[nH]c2C)=O)n1 C=CCCC(O)CN(C)C(C1(CO)CCN(C(=O)Cn2cc(C#N)cn2)C1)=O C1(F)(CNC(C2(CC#C)CCC2)=O)CCN(C(c2ccnn2C2CC2(F)F)=O)C1 C1(CC(=O)NCCCN(C)C(C2COCC2C(F)F)=O)CCCS1(=O)=O CCCCC(O)CCC(=O)N1CC(N(C)C(C2COCCN2C2CCCC2)=O)C1 CC(C)CCCCC(=O)NCC1CC1NC(c1c(Cl)cnn1C1CCCC1)=O CCCC(C(O)c1ccccc1)Nc1ccc(C(C)(F)F)cn1 CCC(C)(C(=O)NC1CC2CCC1N(C(c1cncc(Cl)c1)=O)C2)C(N)=O CC(C)(CF)C(=O)NC(CNC(c1cnn(-c2ccc(Br)cc2)c1)=O)C1CC1 C(=O)(C1=C(C#N)CCC1)N1CCC(CN(C(=O)CC2(N(C)C)CC2)CC)CC1 C1(NC(C=C(C)Cl)=O)CCOCC1NC(c1ccc(CCNS(C)(=O)=O)cc1)=O C#CCCC(O)C(=O)NCCCN(C1CCCC1)C(c1cc(COC)no1)=O C1(COC)(NC(c2cc(CCO)on2)=O)CCN(C(C2CC=CCC2C)=O)C1 c1(C(=O)NC2CC(CNC(C(C)OCC)=O)C2)ncc(C(N)=O)cc1Cl CCCC(C(=O)N1CCOCC1C1CCC1)NC(=O)Cn1ccnn1 N1(C(c2ccn(CC)c2C)=O)CC2CC(C(=O)NC3CCCCC3C)(C2)C1 C1(C)(C(=O)NCCN(C(c2c(C)cccc2)=O)C)COC(C)(C)O1 c1(C(=O)NCCCn2cc(CC(=O)OC)nn2)ccc(I)cn1 N1(C(c2occ(C)c2)=O)CCCCC1C1CCN(C(c2ncc(C)cn2)=O)C1 O=C1CCc2ccc(NC(C3CCN(C(c4ccc(OC(F)F)cn4)=O)C3)=O)nc2N1 c12nnsc1C(=O)N(CCc1ccccc1)CCNC2=O.c1(CC)cccnc1 C(C(=O)NCC1CCN1C(c1ccc(SC)o1)=O)(C(C)C)NC(CCCOC)=O C1(C(=O)NCC(C)CN(C)C(c2noc3ccccc23)=O)CC2C=CCC(C1)C2 c1(C(=O)NC2(CCNC(CCCOC(C)C)=O)CCC2)cccc([N+](=O)[O-])c1N C1(CNC(C(CC)C)=O)CCC(F)(CNC(c2ccc[n+]([O-])c2)=O)CC1 C(=O)(C(C)C(O)CC(C)C)NCCCCCNC(CCCc1cc(C)no1)=O N1(C(CN2C(C)CC2)=O)CCOC2CN(C(c3cc(CCO)on3)=O)CC12 Cc1cc(C)c(C(=O)NC2CC(CCNC(=O)CCOc3ccccc3C)C2)[nH]1 c1(CNC(c2ncn(CC)c2)=O)cnn(C)c1C(=O)NCCC1CCC(C)C1 C1(CCNC(C(C)SCC)=O)CCCCN1C(=O)CCC1C(=O)ON=C1C C(CC1CCc2ccccc21)NC(=NC)NC(C(CC)(CC)CC)C1CCCC1 c1(OC)cncc(C(=O)NC(CO)C(=O)NCC(C)C(C)(F)F)c1 CCCCC(CC)OCCNC(C)(C)C.C(COCCO)OC(C)=O O=C1CCC2CN1CC(CSc1cccn1CC(F)(F)F)O2 c1(C(=O)NCC2N(C(COCC=C)=O)CCCC2C)nnc2n1CC(=C)S2 C1(CC(N2CCC(NC(c3ccoc3Cl)=O)C2C2CC2)=O)CC2CCC1CC2 Cc1nn(C)nc1C(=O)NCCC1CN(C(c2conc2C2CCC2)=O)CCO1 c1(C2CC(C(=O)NCC3(NC(CN(CCC#C)C)=O)CC3)C2)ccc(O)cc1 C(C(=O)NC1(CNC(c2c(C)cccc2N)=O)CC1)(C(C)(C)C)OC N1(C(C(CCOC)C)=O)CCOCC(NC(C2(COC)CC=CC2)=O)C1 c1(C(N(C(C)C(=O)NC2CCCCC23CC3)CC)=O)cc2cccn2cn1 c1(C(=O)NC(C(=O)OCC)CS(C)(=O)=O)ccc(F)c2ccncc12 c1(C(=O)NC(CC)CNC(C2(OC)CCC(C)(C)CC2)=O)cn2ccc(C)cc2n1 c1(C(=O)NC2CN(Cc3c(C)scn3)CC2C#N)ccc2cccnc2c1 c1(CNC(C(c2cnn(C)c2)C)=O)nc(C(=O)NC(c2ccncc2)(C)C)co1 C(=O)(C(C)P(C)(C)=O)NCCCC(C)NC(c1nc(OC)oc1)=O C(C(=O)N1CC(C(F)(F)F)C(CNC(C2CC(O)C2)=O)C1)(C(C)C)OC N1(C(CC2CC(OC)C2)=O)CC(NC(C2(C)CC3CC3C2)=O)C(SC)C1 N1(C(c2c(F)ncc(OC)c2)=O)CCC(C2CCN(C(=O)CCC(=O)NC)C2)C1 C(=O)(C(CC)ONC(=O)C1(COC)CC1)N(CC(=O)NCC)C1CC1 C1(Cn2c(N3CC4CC(CC4)C3)nnn2)C(F)(F)C12CCOCC2 C1(C(=O)NC2(C)CCCN(C(C(C)C)=O)C2)CCn2nnnc2C1 c1(C(=O)NC(CCCC)CNC(=O)CSCC(C)C)ccc(COC)cc1Cl CCC(CC)CC(F)C(=O)NC1COCCC1NC(c1c(C)ncnc1C)=O n1(C(C)C)[nH]nnc1=NC(=O)NCCOC(N)=O c1(COC(C2C3CCC2(c2ccnn2C2CCCCC2)C3)=O)ccccc1F c1(-c2n(CC)c(S)nn2)cc(CN2CCC(CC(N)=O)C2)ccc1C c1(OC)ccc(OC)c(C(N2CCC(CN(C(=O)CCC3CC3(C)C)C)C2)=O)c1 c1(C(C(=O)NCC(CC)N(C(=O)CNC(=O)CN(C)C)C)O)ccnn1C CCCCC(CC)CC(=O)N1CCOCC1CNC(c1cc2n(c1)CCOC2)=O c1(CSCCC)ccc(C(N2CC(N(C(=O)CCCC3CC3)C)C2)=O)o1 CN1C(=O)C(F)CC1C(=O)NCC1CC(NC(C2C3CCCCC23)=O)CCO1 C1(C(CNC(CSCCCC)=O)(C)O)CCN(C(=O)Cn2c(C)csc2=O)CC1 c1(C(N2C(CCNC(C3C(COC)C3)=O)COCC2)=O)nccc2[nH]ccc12 C1(CC(=O)N(C2CN(C(c3cc(C#N)on3)=O)CC2O)C)CCOC(C)(C)C1 C1(CCNC(C2C3CCCCC23)=O)CCCN(C(=O)CN2CCCC2=O)C1 C1(C(N(C23CC(C2)C3)CC)=O)CN(C(=O)CC2C=CCC2)CC1C(C)C c1(NC)cncc(C(=O)NCC2(CCO)CCCC2)n1 c1(SC)ccc(Br)cc1C(=O)NC1CC(NC(=O)Cc2cnn(C)c2)C1 C(=O)(C(C)N1CC(NC(=O)OC(C)(C)C)C1)OC.C1(OC)CN(C2CC2)CCN1 C(=O)(CCCC(=O)N1CC2CC(NC(=O)CSCC3CCCO3)C2C1)NCC C=CC1OCCC1C(=O)NC1CC(NC(c2cccc(OC(C)(C)C)c2)=O)C1 C1(NC(C(CCO)N(C)C)=O)(CO)CCN(C(C2CCN2S(C)(=O)=O)=O)CC1 C1(NC(C(C)(C)CO)=O)CN(C(=O)CCc2cc(F)ccc2F)CCC1CO CC(C)CC(CNC(C1CCCSC1C)=O)C(=O)NCCN1CC=CCC1 c1(C(=O)NC(C(C)C)C(C)NC(=O)CN2C(=O)CNC2=O)nccc(N)c1Cl c1(OC)ccc(S(C)(=O)=O)cc1C(N1CC(NC(=O)CC(O)C(C)C)C1)=O c1(C(N(CC(C)NC(C2CC(Cl)(Cl)C2)=O)CC)=O)c[nH]c2cccc(Cl)c12 c1(C(N(CCNC(=O)CCC2OCCO2)CCOCCO)=O)c[nH]cc(Cl)c1=O N1(CCC)C(=O)CCC1C(=O)NCC(C)(C)CNC(=O)CSc1cccc(C)c1 N1(C(C(C)OCCOCC)=O)CCC(CNC(c2cnoc2C)=O)(COC)CC1 Cc1cncc(CC(=O)NCCCN(C(=O)C=CC(=O)N(C)C)C(C)C)c1 C1(CCOC)CN(C(=O)C(C)C)CCN1Cc1ncccc1O C12(NC(=O)CC3C=CCC3)CCC(CC1n1cc(C3(O)CC3)nn1)C2 c1(C(N2CCCC(F)CC2)=O)nnc2ccc(-c3ccncc3F)cn12 N1(C(C=CCNC(CC2CC(SC)C2)=O)=O)CCC(C=C)CC1 C(=O)(CC(C)(C)CCOC)NC1C(NC(C(CC=CC)C)=O)COC1 C(CC(=O)NCC1(F)CCOC1)(C(C)(C)C)NC(C=C(C)CN1CCCC1)=O N1(C(C2CN(CC)C(=O)C2)=O)CCC(C)C(CC(N2CCC2CF)=O)C1 C1(C(N2CC(OC(C)C)C2)=O)CN(C(=O)CCCN(C)C)CC1(C)C c1(C(=O)NC2(CCC(=O)N(CC(C)(C)C)CC)CCC2)cccc(CO)c1 C(C(C)(F)C(C)(C)F)NC(C1C2(CC(NC(C(CCC)C)=O)C2)C1)=O c1(C(N(C)CC2CCN(C(C=C(C)Cl)=O)CC2)=O)noc2c1CC(C)(C)CC2 c1(OCC)ccc(C(=O)Nc2ccoc2CNC(c2coc(C(F)F)c2)=O)cc1 Cc1cc(COC(c2nc(C)c(-c3ccccc3)s2)=O)nnc1C c1(CC)cc(C(=O)N(C(C)CNC(C2CCC(NC(C)=O)CC2)=O)C)cc(Cl)c1 C1(NC(CCCCC)=O)CCN(C(C2CCN(S(C)(=O)=O)C2)=O)CC(O)C1 CC1(NC(=O)CCC2CCCCC2)CCN(C(=O)C=CC(=O)NC2CC2)CC1 Cc1cnncc1C(=O)NC1CCC(N(C)C(c2ccc(OC(C)C)cn2)=O)C1 c1(C(N(CCN(C(C(F)=CC)=O)CC)CC)=O)ccc(COc2ccccc2)s1 N1(C(CCCN(C)C)=O)CC(O)CC1(C)C(N1CC(C2CCCO2)C1)=O C(=O)(C(CC=C)CC(C)C)NC1(C(N(CC(CCC=C)O)C)=O)CC1C CC(O)C(F)(F)C(=O)NCCN(C(c1cc(CO)cn1C)=O)Cc1ccccc1 Cc1ccc(C(=O)NCC2(O)CCN(C(=O)C3=NOC(C)C3)C2)c(Br)c1 C1(C(N(CC(C)O)CC)=O)CCN(C(=O)CCSC)C1 C1(CNC(C=C(C)Cl)=O)(CO)CC12CCN(C(C1CC(CCO)C1)=O)CC2 c1(C(=O)NCCNC(CCCN(CCCC)CCCC)=O)ccc(S(N)(=O)=O)s1 c1(OC)ncc(C(N2CCN(C(c3ccncc3Cl)=O)C3CC23)=O)nc1C C#CCC(C(=O)NC(C)(C(=O)NC(CC1CC1)CC1CC1)C1CCC1)C1CC1 C12(NC(c3ccc(CN(CC)CC)o3)=O)CCCN(C(c3cnc(C)s3)=O)C1C2 c1(CN2C(C(N3CCOCC(O)C3)=O)CC3(CC3)C2)c(F)ccc(O)c1F C1(CC(=O)NC(C)CC2CCOC2)CN(C(C2CC2C(C)(C)C)=O)C(C)(C)C1 C1(C(=O)NCC2(NC(=O)CC3(n4ccnc4)CC3)CCC2)C2CC2C2CC12 C1(NC(COCC=C)=O)CC(C2CCN(C(=O)C(C)(C)CF)C2)C1 C1(C2CCN(C(c3cnc(S)[nH]3)=O)C2)(NC(c2cnc(C)s2)=O)CC1 Cc1ncncc1C(=O)NCC1CN(C(=O)Cc2ccc(Br)s2)CCO1 NC(=O)CCCCC(=O)NCC1CCCN1C(C1CC(c2ccc(O)cc2)C1)=O C(=O)(C1SCc2cccnc21)N(CCC(C)NC(c1cccc2ncnn12)=O)C C1(CNC(c2ccc(CC)nc2)=O)CC2(C1)CN(C(C1CCN(C)C1C)=O)C2 Cc1cc(C(N2CCCC(C)(NC(=O)COC3CCOC3)C2)=O)ccc1[N+](=O)[O-] c1(C(=O)NCC(C(C)C)NC(=O)C(=O)C(C)(C)C)cc2c(o1)CCCNC2=O c1(C(C(=O)NCC(CC(C)C)NC(=O)CC2(C)CC2)C)cn(C)c2ccccc12 CC1CCCN(C(=O)Cn2cnnc2O)C1CCNC(c1cc(Br)no1)=O c1(C(=O)NC(C)CC2CCN(C(c3n[nH]cc3Cl)=O)CC2)ncc2ccccn12 N1(c2cc(OC)c([N+](=O)[O-])cc2)CC(C)CN(C(=O)CCC(C)(C)C)CC1C N1(C(C2(COC)C=CCC2)=O)CCOC2(C1)CN(C(C1C=CCS1)=O)C2 N1(C(c2ccc(C(C)=O)s2)=O)CC(NC(c2cnc(C)nc2CO)=O)CCC1C C1(CC)CC(C(N2CC(NC(c3cnn4ccsc34)=O)CC(C)C2)=O)CC(=O)N1 N1(C(C=C(C)C)=O)CCC2CN(C(=O)C=Cc3cccc(OC(F)(F)F)c3)CC12 c1(CC)nc(C(N2CCC(C(N3CCCC3C)=O)(CC)C2)=O)c(C)o1 Cc1[nH]nc(Cl)c1C(=O)NC(C)CCN(C(=O)CCCC1CCCC1)C c1(OC)ccc2c(C)c(C(=O)NC3CC(C)(NC(c4coc(C)c4)=O)C3)[nH]c2c1 CC1CN(C(=O)C2=CCCC2C)CCC1C(N1CCOCC1)=O c1(OC)cc(C)c(C(N2CCN(C(=O)CC3C=CCCC3)CC2C)=O)c(C)c1 N1(Cc2nc(CCC)on2)CC2(CC(NC(=O)C(C3CCCC3)OCC)CO2)C1 Cc1ncc(Cl)c(C(N2CCN(C(=O)CCc3ccc(N)cn3)CC2C)=O)n1 CCCCCCC(C)C(=O)NC1(C)CC(NC(c2ccc(C(C)(C)C)cn2)=O)C1 c1(C(C)(C)N(C)C)cn(CCCNC(=O)C(CC)NC(C2CCCCC2)=O)nn1 N1(C(c2cnc(CC)s2)=O)CCC(F)(C(=O)N(C)Cc2sccc2C)CC1 N1(C(C(C2CCC(C)(C)CC2)C)=O)CC2CC(C1)N(C(=O)C(=O)N=S(C)(C)=O)C2 CC1CCOCCN1C(C1CC(O)CCN1C(c1cccc[n+]1[O-])=O)=O c1(NCCCc2cncc(OC)n2)ccc(CNC(=O)OC(C)(C)C)c(Cl)c1 C1(NC(c2onc(C)c2C)=O)COC2(CCN(C(=O)CCN3CCCC3=O)C2)C1 CC1CN(C(C)C(=O)N2CC(CC(C)NC(=O)COCC(F)(F)F)C2)C1 CC(C)C(O)C(C)C(=O)N1CC2CC(C(=O)NC3CC(CO)C34CCC4)CC2C1 c1(C(N(C2CCN(C(=O)COCc3nnc(C)s3)C2)CC)=O)cnnn1C(C)C c1(CC(C)NC(=O)NCC(c2cccc(Cl)c2Cl)C)c[nH]c2cc(F)c(F)cc12 C1(NC(C(C)Sc2ccccc2)=O)CCN(C(=O)Cc2cnn(C)c2)C12CCC2 C1(NC(C2(C=C)CCC2)=O)COCCC1NC(=O)C(C)NC(C1CCC1)=O C1(CC(=O)NCCCCN(C)C)CC2(C1)CN(C(=O)CCc1ccoc1)C2 C(CNC(=O)CC1COCCO1)(CC(=O)NOCc1ccccc1)OC N1(C(C(CCSC)OC)=O)CC(C2CN(C(=O)Cc3ccoc3C)C2)C1 c1(NC(C)=O)cnc(O)c(C(N2CC3(CC(NC(=O)C=C(C)Cl)C3)C2)=O)c1 c1(C2(NC(C=Cc3cn(CC)nc3)=O)CCC2)ccc(C#N)cc1 c1(C(C(=O)NCCC2CCCC2)NC(=O)OC)ccccn1 N1(C(CCN(C)CC)=O)CCN(C(=O)Cc2ccc(S(C)=O)cc2)C2(CCC2)C1 CCN=c1[nH]cc(C(=O)N(C2CCCN(C(=O)CCCC)C2)C)s1 N1(C(c2cc(C)n(C)c2)=O)CCCC2C1CCN2C(=O)Cn1cnc(C#N)n1 n1(CC)nc(C)c2cc(C(N3CC(CN(C)C(C4CC4C(C)C)=O)C3)=O)sc12 C12(C(=O)OCC)CN(C(=O)C(=O)N(CC(C)C(F)(F)F)C)CC1CCCO2 CCC(CC(=O)N1CCN(C)C(C(=O)NC(CC)(CC)C(C)C)C1)C(F)F c1(C(=O)NC2CCCC(NC(c3c(CC)cco3)=O)C2)cccc2[nH]ccc12 Cc1c(C(N2CCC3C(CCN3C)C2)=O)cc([N+](=O)[O-])cc1Br O=C1CC(NC(C2(NC(C3CCCC3C(F)F)=O)CC2)=O)CC(=O)N1 C1(CC)C(C(=O)NCC(C)(C)NC(c2ncccc2C)=O)CCN1C c1(C(=O)NC2C(N3CCN(C(CC(C)F)=O)CC3)COC2)cc(S(C)(=O)=O)co1 C1(C(=O)NCCOCCNC(CN2C(C)CC2)=O)Cc2ccc(F)cc2O1 Cc1nncc(C(N2CCOCC2C(N2CC(CC(C)(C)C)C2)=O)=O)c1C c1(C(N2CC(CC(N3CCC(O)CC3)=O)C2)=O)ccc2c(n1)OCCO2 c1(CN(C(=O)C=CC2CCOC2)C)cccc(CNC(C2CCC(=O)N2)=O)c1 c1(CC)nc(Cl)c(CC)c(=NCCC(C)NC(C2(O)CC3CCC2C3)=O)[nH]1 C1(O)(CCNC(c2nncc(C)c2)=O)CCN(C(C2CC(=O)N(C)C2)=O)CC1 C1(NC(COCC(=O)NC)=O)C2CCC(C2)C1C(=O)NCCCCNC(C)C c1(N2CCN(C(c3ccc(C)cc3C)=O)CC2CCO)nc(O)c2c[nH]nc2n1 c1(C(=O)NC(c2ccccn2)C)ccc(Cl)nc1NCc1ccc(I)o1 Cc1cc(C(=O)N(C2CC(NC(c3cc(C)c(C)[nH]3)=O)C2)C)c(C)s1 N1(C(C(C)(N(C(c2c(C)occ2)=O)C)C2CC2)=O)CC(C2CC2)C1C1CC1 CON=CC(=O)NCCC1CCN(C(c2c[nH]nc2-c2ccc(Cl)s2)=O)C1 C#Cc1ccnc(C(=O)NCC2CC(C)N(C(C3CCC(N(C)C)CC3)=O)C2)c1 n1(-c2cn(CC)nc2)nc(-c2ccccc2CO)nc1C1CNC(=O)N1C N1(C(CC2(OC)CCC2)=O)CC(NC(=O)C(=O)Cc2ccc(F)cc2)CCC1C Nc1ccc(C(=O)NCc2csc(C(=O)NCC3(CO)CC4CC4C3)c2)nc1 C(=O)(CCCCC(=O)OC)NC(CC#C)(C)C(=O)NCCC(=O)NCC Cc1ccc(-n2cc(COC3CCN(C(C4CCC(N(C)C)C4)=O)C3)nn2)cc1 CC1(C)CN(C(=O)C=CBr)CC(C)(C)C1NC(=O)CC1CCC1(C)C C1(NC(CCOCCOC)=O)CC(C)(CNC(=O)CC2(OC)CC2)C1 C1(C(N2CCN(C(C)CNC(C3CC4(CCC4)C3)=O)CC2)=O)(CC)CCNC1=O C1(NCC#CC)CC(NC(=O)CCn2cc([N+](=O)[O-])cn2)C12CCC2 C1(C(=O)NC2(CNC(C3C(COC)CC3)=O)CC=CC2)CC12CCCCC2 Cc1ccc(C(=O)N(CCC(C)NC(=O)C=CC2CC2)C)c(N)c1Cl C(=O)(CC(C)(O)COC)NCC(C1CC1)NC(C1(COCC)CC1)=O C1(CNC(c2cc(OC)nn2C)=O)CCCC2(CN(C(=O)CC(O)C3CC3)C2)O1 C1(C(N(CC(C(=O)OC)C)C)=O)(NC(=O)C=Cc2cocn2)CCC(C)(C)C1 CN1CC(NC(C2COCCN2C(c2cccs2)=O)=O)C(C)(C)C1 C1(C(N2CC(CNC(C#CC(C)C)=O)C2)=O)Cc2nccn2C1 Cc1ccc(I)c(CNC23CC(NC(=O)Nc4ccc(I)cc4)(C2)C3)c1 C1(C(N2CC(CN(C)C(c3ccn4ccnc4c3)=O)C2)=O)OC(C)(C)OC1(C)C C(=O)(C1CCCn2ccnc21)N1CC2CC(NC(C3CCOC3)=O)C2C1 CCCC(CCC)CC(=O)NCC1CC1NC(c1cc2c(nn1)CCC2)=O C(=O)(C(F)(F)CCn1cc(CC(C)O)nn1)N(C(CCSC)C)C c1(C(=O)NCc2ccc(-c3c(O)cccc3O)cn2)ccc2c[nH]nc2c1 Cc1ccc(CNC(=O)N(CC(=O)NCC2(C)CCC2)C)o1 C=CCC(C)C(=O)NCc1csc(C(=O)N(C)Cc2c(C)noc2C)c1 C1(C(N(CCCC)CC)=O)(CC)CCN(C(=O)C(C2CCCCC2)F)C1 C1(NC(N2C(C(C)(C)C)CC(C)(C)C2)=O)C2CCC(C2)C1(C)C CC1(CNC(C2CC3CCCCCC23)=O)COCCN(C(C2(C#N)CCC2)=O)C1 c1(CNC(c2ccc(COC)[nH]2)=O)cccc(CNC(C2(C#N)CC2C)=O)c1 c1(C(N(CCNC(C2C(C=C)C2)=O)CC)=O)ccc(C(F)F)nc1 N1(C(C2(C=C)CCCC2)=O)CCC2(CC(C(=O)NC3CCC(=O)NC3(C)C)C2)C1 c1(C(=O)NCC2N(C(c3n[nH]c(CC)c3Cl)=O)CC(O)C2)ccc(F)c(Cl)c1 CC(C)C(CC(=O)NCCN(C(=O)CCc1cncs1)C(C)C)c1ccon1 N1(C(CC2N(CC)CCOC2)=O)CC2(COC(CNC(=O)CC(C)C(C)C)C2)C1 c1(OC)ccc(O)c(C(=O)NC2CN(C(C34CC(C3)C(C)O4)=O)CC2C)c1 N1(C(C2(CC#C)CC2)=O)CCN(C(=O)C(C2CCC(=O)CC2)F)C(CCC)C1 C(CCCC(=O)NCCC1(NC(=O)CCC(=O)c2ccc(N)cc2)CCC1)SC N1(C(C(C(C)C)SC)=O)CCN(C)C(CNC(c2ccc(F)c(F)c2)=O)C1 C1(c2n(CC)nnn2)(NCc2ccc(C(=O)OC)o2)CCN(C2CC2)C(C)C1 C1(COCCOC)CCN(C(=O)C(C)(O)c2ccccn2)C1 C(=O)(CCC(=O)NCCCCCN(C(=O)CNC(c1ccccc1C)=O)C)OC C1(NC(c2cc(CCC)on2)=O)CN(C(C2(CC)CCC2)=O)CCC1O N1(C(C2CCCCC2O)=O)Cc2occ(C(N3CCOCC3C(F)F)=O)c2C1 CC(C)(C(=O)N1CC2CCC1C(NC(=O)CCCCN1CCCC1)C2)C(F)(F)F N1(CCCC)CCCCC1C(=O)NCC(C)(C)CNC(c1ocnc1C1CC1)=O CC1(NC(=O)C=CCC(C)(C)NC(C23C(=O)C4CC2C3C4)=O)CC2CCC1C2 C1(c2nnnn2CC(F)F)(NC(c2ccccc2)CC)CCC=CCC1 N1(C(c2c(CC)occ2)=O)CCC2(CC(NC(=O)CSC(C)C)CO2)C1 CC(C)(C)C#CC(=O)N1CCC(CCNC(=O)Cc2ccc(F)c(F)c2)C1 N1(C(c2ccc(N(C)C)cn2)=O)CCCCCC1CNC(C1CCC1CF)=O CC(C)(C)S(=O)(=O)CC(=O)NC(C1CCOC1)CNC(=O)CCC(F)(F)F c1(C(=O)NCC2C(CNC(C(c3c(C)cncc3)C)=O)C2)cc2c(ncn2C)s1 c1(C(N(C2CCN(CCC3CCCO3)CC2)CC#C)=O)cccc(Br)c1 c1(CC(=O)NCCC2CN(C(Cc3cc(C)no3)=O)C2)ccnc(Cl)c1F N1(C(c2ccnn2C)C(=O)NC(C(=O)OC)C)CC(O)CC(O)C1 Cc1ccc2c(c1)SC(C(=O)NC1CN(C(C3(Cl)CC3)=O)CCC1C)C2 N1(C(C2CCN(C)CC2)=O)C2CCCC1CC(NC(C1CCCCS1(=O)=O)=O)C2 CC1(C(=O)NCc2cc(Cl)cc(Br)c2)CCN(C(=O)Cn2nccn2)CC1 C(F)(F)(C(F)(F)F)OCC(=O)NCC1(F)CCC(NC(=O)C=CCO)C1 C(=O)(C(C(C)NC(=O)CC1CCC1)C(C)C)NCC1CN(CC)C(=O)O1 c1(C(N2CCC(CNC(C3(CC=C)CCC3)=O)C(C)C2)=O)cnn2ccccc12 N1(C(Cc2cn(CC)nn2)=O)CC2(CNC(=O)Cc3ccccc3)CCC1C2 C1(CNC(C2C(CC)CCN2C(=O)CCCN(C)C)=O)OCC2CCC1C2 C(C1c2ccsc2CCN1C(c1ncc(C(F)F)cc1Cl)=O)NC(=O)C1=CCC1 N1(C(CC2N(C(C(C)SC)=O)CCC2(C)C)=O)CCC2(CC(F)C2)C1 Cc1ccc(C(C)C)cc1C(N1CC(NC(=O)CC2COCCO2)C(C)(C)C1)=O CN1CC(C(=O)NC2CC(F)CN(C(=O)C=C3CCOCC3)C2)OCCC1=O C1(C(N2CCCN(CC=C)CC2)=O)C2CC(O)C(C2)N1C(C1CC1(C)C(F)F)=O c1(C2(OC(=O)CNC(=O)Nc3ccccc3C(F)(F)F)CC2)ccccc1Br O=C(C1=C(F)CN(C(c2ccncc2O)=O)CC1)N1CCCCC1CCCO C(=O)(Nn1cnnc1CC)C1N(C(C(CC=C)CC)=O)C(C2CC2)CC1 C=CC1CN(C(=O)C(C)(O)C2CCC2)CC1NC(C1COCCOC1)=O Cc1cnccc1C(C)C(=O)NCC(C)(O)CNC(=O)COC1CC1 c1(C(c2n(CCCSC)nnn2)NCCn2cc(C)cn2)snc(OC)c1Br C1(CNC(COc2ccn(C)n2)=O)CCCCC1C(N1CCCC(C(N)=O)C1)=O C#CCC(C)(C(=O)NC1(C2CCCCO2)CC1)NC(c1cn(C)c(C)n1)=O CC1=C(C(=O)N2CC(N(C)C(C3CC(=C4CC4)C3)=O)C2)S(=O)(=O)CCO1 C1(NC(C2(C)CC3CC3C2)=O)CN(C(=O)CC2CCCC2)CCC1F C1(C)(OCC(=O)N(C2CCN(C(C3CCC4(C3)N=N4)=O)C2)CC)CCOCC1 C(=O)(C1=NOC(C)C1)N1CC(OC)C(C(=O)N(C)Cc2cccnc2)C1 c1(OCC(=O)NC2CC(N(C)C)C(O)C2)cc(Br)cc(F)c1F Cn1cc(C(=O)NC2CCN(C(C3OCCCC3(C)C)=O)CC2O)ncc1=O C(=O)(N=c1[nH]n(C)c2nccnc12)c1c(C(=O)OC)ccs1 c1(OC)cnc(C(=O)NCCC(C)NC(C2CC2C2CCCO2)=O)cn1 O=C(O)CCC(Cc1ccccc1)NS(=O)(=O)CC1OCCO1 CCC(CC(=O)N(C)Cc1ccccc1CNC(=O)CCOCC(F)F)C(F)F Cc1n[nH]c(C)c1C(=O)NCC1C(C)CCN1C(=O)C(=O)Cc1ccc(Cl)cc1 CCC(N=c1[nH]c2c(c(=NC(C)c3ncc[nH]3)[nH]1)COC2)c1c(C)noc1C C(=O)(C1=CC2(CCOC2)C1)NC(CC#C)(C)C(=O)NC(CC)C(=O)OC c1(N(C(=O)N(C2CC=CC2)C)CC)ccn(C)n1 c1(C2N(C)CC2)ccc(S(=O)(=O)N2CCOCC2)cc1.C1(=O)NCCN1 C1(C(=O)NCc2cc(C)sc2)C(C2CC2)CCN1C(c1cc(Cl)n(C)n1)=O c1(CCN(C)C(=O)NC(c2cccs2)CC2CC2)nn[nH]n1 c1(N(CC(C2CC2)OC)C)nc(=NCCC2(C(F)F)CC2)[nH]c2c(F)cccc12 c1(CC)cc(C(N2CCC(CN(C)C(C3(C#N)CCOC3)=O)C2)=O)cn(C)c1=O C12(C(=O)NCC3CCCSC3)CC(C(F)(F)F)(CO1)C2 C=C=CCCC(=O)NCC1CCN1C(c1cc(SC)c(C)o1)=O CC1CCN(C(c2cc(CO)[nH]n2)=O)CC1CNC(=O)C(C)(C)N1CCOCC1 N1(C(CCn2cnc(=N)[nH]2)=O)CC2C=CC1C(C(=O)NCCC1CCC(=O)N1)C2 c1(C(N2CCC(CCNC(=O)CCOCC(F)F)C2)=O)ccc(F)c(O)c1F C1(NC(c2cnsn2)=O)CC2CC(C1)N(C(=O)CN1CCOCC1)C2 C1(NC(c2scc(C)c2C)=O)CS(=O)(=O)C2CN(C(=O)CN(C)C(=O)C3CC3)CC12 C(=O)(CCCCCC#N)N(C(CCNC(c1c(C)ccc(C)c1)=O)C)C CCC(C)(C)C(C)CC(=O)N1CC(NC(c2ncn(C(C)(C)C)n2)=O)CC(C)C1 c1(CC)cccnc1C(=O)N(CCCNC(=O)C=C1CCC(C)CC1)C C1(C(=O)NCCc2ccccn2)CCN(N2CCCCCCC2)CC1 Cn1nnc(C(N2CCCCC2Cn2cncn2)=O)c1C(F)(F)F C1(CNC(C(CC)F)=O)CCN(C(c2ccc[nH]2)=O)CCC1(F)F C(CS(=O)(=O)CC(=O)NCC1CC1NC(=O)CN1CCC(C)(C)C1)OC c1(OC)ccc(C(=O)C(N2CC(NC(C3(F)CC=CC3)=O)C3CC23)=O)cc1 c1(CN(C(COCCC#C)=O)CCCNC(=O)CC2CCCN2C)ccccc1 C1(C(=O)OCCSC(C)(C)C)CCCCN1C(C1CCCC1c1ccccc1)=O c1(C(N2CCC(N(C(=O)C(C)CF)CCC)C2)=O)c(C)cc(Cl)cc1C N1(C(c2c(C)nc(C)o2)=O)CC(NC(=O)CC2NC(=O)CNC2=O)CCC1C N1(C(C2C(C(=O)OCC)C2)=O)CCC(C)(NC(=O)COCCc2cccs2)C1 C(=O)(N=c1ccc(CC)n[nH]1)NCCc1ccc(OCC)c(C(F)(F)F)c1 C#Cc1ccc(CC(=O)NCC2(O)CCN(C(C3CS(=O)(=O)CCO3)=O)C2)cc1 C(C)(C)(CC(F)C(=O)NC1CCCCN(C)C1=O)NC(CC(=O)NCC)=O c1(C(N2CCN(C(C(COC)(F)F)=O)CC2)=O)c(C)cnc2ccccc12 N1(C(c2cc(C)cc(O)c2)=O)CC2(CCN(C(c3c(C)ncn3O)=O)CC2)C1 c1(CN(C(=O)Nc2c(CC)n3c(n2)CCC3)C)nc(C)c2ccccc2n1 C1(CC)CN(C(C2CC3CCC(C2)O3)=O)CCN1C(=O)C=CC(C)C C1(CNC(C=CS(C)=O)=O)CN(C(C2CC(=C3CCC3)C2)=O)CC2(CCC2)O1 c1(CC)cc(=NCC2CCN(C(C3CC4CC4CC3C)=O)C2)[nH]c(COC)n1 C(=O)(CCCC(C)(C)NC(=O)C(=O)NOC)NC1C(C=C)COC1 c1(OCCNC(C23CCCCC2C3)=O)ccc(Br)cn1 c1(CC(N2C(C)CN(C(=O)CCC(C)CN(C)C)CC2)=O)cnn2c1CCCC2 c1(C(N2CCC(CCC(=O)NC(c3cnn[nH]3)C)C2)=O)ccn(C)c(=O)c1 c1(C(=O)NC(CNC(COC(CC)C)=O)C2CC2)ccn2ncc(Br)c2n1 C=CCN=C(NCCS(=O)(=O)CC)NCc1ccc(C#N)s1 Cn1ncc2ccc(C(=O)NCC3CC4CCC3N4C(c3cnns3)=O)cc12 C1(N(C)C(c2ccon2)=O)CCCC(NC(c2ocnc2C(F)F)=O)C1 Cc1c(CC(N2CC(CCNC(=O)C=CC(F)(F)F)C(C)C2)=O)ncn1C C1(C(=O)NCC2(CC)CC(C)(C)C2)CCCCCCN1C(=O)C(C)CC(N)=O C=CCCC(F)(F)C(=O)NCC1CCC(NC(=O)C(N2CCC(C)C2)=O)CC1 Cc1nn2c(c1OCC(=O)NOCC1CCOC1)CCCC2C C12(CC(=O)NCC3(SC)CCC3)CCC1CN(C(c1ncccn1)=O)C2 C=C(Cl)CC(C(=O)NCC(O)COCC)NC(=O)CC(C)CC Cc1ccc(C(=O)N(CC(C)CNC(C2CCN(C)C2)=O)C)c(N)c1Br C1(C(=O)NC(C)CCCNC(=O)CCCc2ccsc2)NC(=O)CC1C N1(C(c2nccc(CC)c2)=O)CC2CCN(C(=O)C(F)=CC3CC3)CC12 c1(C(N(CCCOCCN(C(CSC)=O)C)C)=O)c(-c2ccncc2)noc1C C=CC1(CO)CCN(C(C2CN(C(c3ccc(CC)nc3)=O)CC2(F)F)=O)CC1 CN1CCC2C(CCN2C(C2CCC3(CC3)N2C(C2(C)CC(F)C2)=O)=O)C1 c1(CNC2C(CNC(C3CC4CC4C3)=O)CCC2)ccc(Cl)nc1Cl c1(CC)nc(N2CCC(CCNC(c3ccnc(F)c3Cl)=O)C2)c2ccsc2n1 C1(C(N2CCN(CC3CCCO3)CC2)=O)CC2(CCOCC2)CCO1 C(=O)(C(C)N=c1cc[nH]cc1)N1CC(NC(Cc2ccc(C)s2)=O)C2(C1)CC2 c1(C(N2CC(C)(NC(c3ccnc(C)n3)=O)C2)=O)cc2cc([N+](=O)[O-])ccc2o1 N1(C(C2C(COC)C2)=O)CC=C(CC(=O)N2CC(C(=O)OC)C3(CC3)C2)CC1 C1(CC(C)C)CC(c2nnnn2C2CC2)(NC(C)(C)C2CC2)C1 c1(NC(C(c2ccc(F)cc2)(C)O)=O)cccc(-c2cnco2)c1 c1(C(=O)NC2C(C)N(C(C3CCC3)=O)CCC2)nnc2ccccn12 N1(C(c2cncc(NC)c2)=O)Cc2occ(C(=O)N(C)Cc3ccnn3C)c2C1 N1(C(C2CCCC23CC3)=O)CCN(C(=O)Cc2nc[nH]n2)C(c2ccccn2)C1 c1(C(=O)NCC(Cc2ccccc2)N(C(CC=CC=C)=O)C)c(F)cccc1F CCC(CC)C(C)C(=O)NCC(C)CC(=O)NCC(c1cnn(C)c1)=O N1(C(CCCCCSC)=O)CC2CN(C(=O)C(O)C(C)C)CC2(C)C1 CC(CN(C)C)CCC(=O)NC1CCN(C(c2cnsc2)=O)C1 Cc1cnc2n1C(C(=O)NCCN(C(=O)CN1CCC(C)C1)CC1CC1)CCC2 C(C)(C(=O)NCC(C1(O)CN(C(=O)Cc2nn(C)cc2Cl)C1)(C)C)(C(C)C)OC N1(C(c2ccc(C(C)=O)s2)=O)CCOCC1CNC(=O)CSC(C)(C)C C1(NC(C(C)(C)c2cnsc2)=O)CC(F)CN(C(C2(F)CC2)=O)C1 Cc1ccc2cc(C(N3CCC(NC(=O)CC4(C)CCC4)C3)=O)[nH]c2c1 C1(N(C(c2cc(F)c[nH]2)=O)CC)CCCN(C(C2CC2Br)=O)CC1 c1(C(=O)NC(CNC(c2ccc(C#N)o2)=O)CO)c(Cl)cccc1Cl c1(C(=O)NC(c2ccc(SC)cc2)C(=O)OC)cnc(S(C)(=O)=O)s1 N1(CC(N2CC(COC)(NC(=O)CCN3CCC3)C2)=O)CCC(O)CC1 C(CS(=O)(=O)CC(=O)Nc1c(C(=O)NCC2CC2)cccc1C)OC c1(C(c2n(CCC)nnn2)NC2(CC)CCC2)cccc(C2CC2)c1 C(=O)(C#CC(=O)N(C)C)N(CCNC(C1CCC(C)S1)=O)CCF N1(C(C2CCCOCC2)C(=O)NCCCOC)CCCSCC1C c1(SC)ncc(CNc2cccc(OCC(C)(C)C)c2)n1C C(C(C)(C(C)C)NC(c1cnc(O)s1)=O)NC(C1C(c2ccc(C)s2)C1)=O C(=O)(C1CCc2c[nH]nc21)NC1C(CNC(c2c(C)nn(CC)c2C)=O)COC1 Cc1c(C(=O)N(C(C)C(=O)OCc2ccccc2)CCF)cnn1C C1(C(=O)NCc2ccns2)(OC)CCN(C(C2CCC3CC23)=O)C1 C1(C(C(=O)NCCC2(NC(C(=O)NCC)=O)CCC2)OC)CCCOC1 N1(C(Cc2ccc(C)nc2)=O)CCCC2(NC(C3(F)CCCCC3)=O)CCCC12 C(=O)(C1=CC2(CN(C(C3(OC)CC(C)C3)=O)C2)OC1)NCCSCCC=C N1(C(c2c(CC)noc2)=O)CC2CCC(C1)N(C(C1OCCO1)=O)C2 CCC(C)(C)C(C(=O)NCC(CC)(CC)NC(c1cnoc1C)=O)OC N1(C(=O)C=CC2CCOC2)CCC2CN(C(c3ccccc3O)=O)C2C1 C(C)(N=c1[nH]c(N2CCC3(CCC3)C2)nc2cc[nH]c12)c1c(C)nc(C)[nH]1 c1(OC)ccc(COCC(=O)NC(C)C(C)NC(C2(C)CCOCC2)=O)cc1 CCC(C)CCCC(=O)N1CC(NC(C2CC(OC(F)(F)F)C2)=O)C(C)C1 c1(OC)cccc(C(C)C(=O)NCC2CC(O)CN2C(c2ccnn2C)=O)c1 N1(C(c2c(C(C)C)ocn2)=O)C2CCCC1CN(C(C1CC3(CCC3)CO1)=O)C2 C1(CNC(C2(C)CCCC2)=O)CCCC(NC(C2CCN(C3CC3)C2=O)=O)C1 C(CC)(CCCC(=O)N1CCC(CC)C1)NC(c1cc(CCC)[nH]n1)=O C1(C(N2CCC(C)N(C(c3n[nH]c(=N)s3)=O)CC2)=O)CC12CCC(F)(F)CC2 c1(C(N2CC3CC2CC3N2CC3(COC3)C2)=O)nc2cccc(F)c2[nH]1 c1(OC)cc(N)c(C(=O)NC2CCCCC2NC(C2CC2C(C)(F)F)=O)c(F)c1 N1(C(c2ncn(C(C)C)c2)=O)CCOCC(CNC(=O)C=Cc2cc[nH]n2)C1 N1(C(C2CCN(C(C)=O)CC2)=O)CCC2C1CCN2C(C1CCCSC1)=O c1(C(=O)NCC2(C)CCN(C(CC(=C=C)C)=O)C2)ccc(F)c(C)c1C#N CC1CC(C)OC1C(=O)NC1CC(NC(=O)CC2CCC(=O)N2)C1 C1(C(=O)NCC2(NC(C(C)=CC)=O)CC2)CN(C(=O)OC(C)(C)C)CC(C)(C)C1 C1(C(=O)NCC=CCNC(c2c(C(F)(F)F)ncn2O)=O)CCC2CC1CO2 c1(C(=O)NCCN(C)C(C2(F)CC=CCC2)=O)ccc2c(c1)CCCO2 Cc1cnc(C=CC(=O)NC2COCC2NC(=O)CC2(O)CCCC2)[nH]1 C1(CNC(C(C(C)C)NC=O)=O)CCCCN(C(=O)C=C2CC2)CC1 CN1CCN(C(=O)CC2(C)CCOC2)CC1CNC(C1CN(C(N)=O)C1)=O C1(CNC(C(C)OCC#C)=O)CC(C)CCN1C(=O)COCCOCC n1(CC)ncc2cc(C(=O)N(C3CN(C(=O)CC(C)C)CC3(C)C)C)cnc12 C1(CC)CN(C(=O)C(C2CCCN(C(=O)CC3OCCO3)C2)(C)C)CCO1 Cc1nc(C(F)(F)F)ccc1C(=O)NC(C)C(C)NC(c1csc2nnsc12)=O Cc1ccc(CC(C)=CC(CCCC)=O)cc1.c1(CCC(=O)NC)csc(Cl)n1 C1(C(=O)NC2(CNC(c3scc(COC)c3)=O)CCOC2)(CC)CCNC1=O O(N(C)C(=O)C(C1CC=CCC1)NC(=O)C(F)CCC)CC(=O)OC S(=O)(=O)(c1ccc(I)cc1F)NC(C(C)(F)c1ccccc1)=O N1(C(c2sc(C)c(O)n2)=O)CCCC(CNC(C2CCC3(CC2)CC3)=O)CC1 N1(C(C2CC(OCC)C2)=O)CCC(NC(=O)COCC)C(CC)C1 c1(C(N2CCCC3CCN(C)CC23)C(=O)NCCOC)nc2ccccc2nc1C N1(C(CN(C(C)=O)C)=O)CCCC(C)(C)C1CNCCNC(C1CCCSC1)=O C(c1cn(C2CN(C(C3CC(C)(C)CO3)=O)C2)nn1)=CC Cc1cn2c(n1)CCC(C(=O)N(C1CCCN(C(c3cnc(C#N)s3)=O)C1)C)C2 C1(NC(CCc2ccc(OC)cc2)=O)CC2CC1N(C(c1cc(CO)[nH]n1)=O)C2 n1(CC#C)cnc(S(=O)(=O)N=S(C)(=O)Cc2ccccc2)c1 n1(NC2CCn3ncc(C(=O)OC)c3C2)ncc2c1C(NCCOCC)CCC2 N1(CC(=O)NCCN(CC(C)O)C(=O)CC2(O)CC2)CCOCC1=O C(=O)(CCCC(C)(C)C)N1C(C)(C(NOCCC(C)O)=O)CCC1 C(C)(C)(CCCNC(=O)CC1C=CC(NC(=O)CN(C2CCC2)C)C1)OC N1(C(c2ccn(CC#C)c2)C(=O)NC2CC2)CCN(CC)C(=O)C1C c1(NC(C2(O)CCN(C(CCC=C(C)C)=O)C2)=O)cc(Br)cc2[nH]ncc12 C#Cc1ccc(C(=O)NC2COCCN(C(c3[nH]ncc3C#N)=O)C2)cc1 CC(CO)CCCNC(=O)CSCCNC(C1OCCC1(C)C)=O c1(C(=O)NC(CNC(c2cc(SC)oc2)=O)C2CC2)ccc(Cl)c(N)c1 N1(C(C2(C=C)CCCC2)=O)CCC=C(C(=O)NCC2CCCC(=O)N2)C1 c1(C(=O)NC2(C)CN(C(CNC(C3C(C)C3)=O)=O)C2)ccccc1SC(F)(F)F N1(C(C2(C)CC(C)=C(C)CC2)=O)CCCCC(S(C)(=O)=O)C1 c1(C(=O)NC2C(NC(c3c(C)cc(C)[nH]3)=O)C2)ccn2c(Br)cnc2c1 N1(C(c2c(CC)nc(C)nc2)=O)CCC2CN(C(c3cn(C)nc3SC)=O)CC12 C1(C(=O)NCCCN(C(=O)CC2CC2(C)C)C(C)C)CC12CC(C)(C)C2 N1(C(C=CC(CC)C)=O)CCOCCC1C(=O)NCc1cccc(OC)n1 C1(C2(NC(=O)CSC3CC=CC3)CC2)CCCCN1C(=O)C(F)CC1CCOC1 C1(NC(C(CC)n2cncn2)=O)CCC(N=c2[nH]c(C#N)c(Cl)s2)CC1 N1(C(C(=O)NCCCCNC(C(C)Cc2cnn(C)c2)=O)C)C(=O)CCC1=O N1(C(C(C)(C)O)=O)CCCC2(NC(=O)Cc3ccc4c(c3)CCO4)CC2C1 C#Cc1ccc(C(N2CCC(O)(C(=O)OC)CC2)C(=O)NCCC2CC2)c(F)c1 C1(C(N2C(CNC(C3(C)CCCS3(=O)=O)=O)CCC2)=O)CCCC12OCCO2 n1(CC(=O)N(CCCN(c2nncs2)C)C)cnc2ccccc12 C(CCC)(CCCNC(=O)CN1CCCNC1=O)NC(COCCCCC)=O C1(NC(CS(=O)(=O)NCC)=O)CN(C(c2cc3c(s2)CCC3)=O)CC2(CCC2)C1 N12CCC(CC1)NC(=O)OCc1cccnc12.C(=O)(COCCOCCO)OCC n1(CC(=O)NC(CC(=O)N(C)C2CC2)C(=O)O)cnc2ccccc12 C1(CNC(CCCC)=O)CN(C(C2(C)CC(C#N)C2)=O)CC1(F)F N1(c2c(C)cc3c(c2)OCO3)CCC2(CC1)Cc1ccccc1NC2=O C#CCCC(O)CCNC(c1cnc(CNC(=O)C(C)n2ccnc2)nc1)=O C1(OC)CC(CC(=O)N(C)CCN(C(=O)C=Cc2cnc[nH]2)C(C)C)C1(C)C N1(C(C2CC(=O)N(c3cccc(Cl)c3Cl)C2)=O)CCC(c2nn[nH]n2)C(F)(F)C1 N1(Cc2cnc(CCC)s2)CCN(C(C2CN(C)CCO2)=O)C(CC)C1 N1(C(C=Cc2nc(C)sc2)=O)CCCC(NC(=O)CC2CCCCCO2)C1C C1(NC(CCCC(=C)C)=O)CN(C(=O)COC2CCCCC2C)CC1C1CC1 c1(NC(=O)CCc2cccnc2)ccc(C(N2CCC2)=O)cn1 C(=O)(C1OCCn2ccnc21)N1CCCC(CC=C)(NC(=O)Cn2nccn2)C1 CCCN=C(NCCCOCC1CC1)N1CCC(F)(c2ccc(F)cc2)C1 CCC(CCC(=O)NCC(C)S(C)(=O)=O)NC(c1cn(CC)cn1)=O C1(C(=O)NCCCN(C(C2C(C(N)=O)CC2)=O)CCO)CCCN1c1nccs1 CC1CN(C(C2CCC(N(C)C)C2)=O)CCC1C(=O)NC(c1ncc[nH]1)C c1(C(N(C2CCN(C(=O)C=CCn3cncn3)C2)CCC)=O)ncc[nH]c1=O c1(C(=O)NC2C(NC(c3c(CC)cco3)=O)CCC2)cccc2c1CCC2 c1(C(=O)OCC)cc(C(=O)NCCCN(C)C(c2occc2Cl)=O)[nH]n1 c1(NC(=O)CCC2CCCO2)c[nH]nc1CCNC(C1(CS(C)(=O)=O)CCC1)=O C1(CNC(c2cc(C)ncc2)=O)CCCN(C(c2cc(F)cnc2Cl)=O)CC1 Cc1ncc(C(N2CCC(C(F)C(=O)NCC3C4CCCC34)C2)=O)o1 N1(CCN(C(=O)CCN(C)C(c2ccsn2)=O)C)CCOCC1 Cc1ncnc(C(=O)NC(c2ccccn2)(C)C)c1C Cc1ccc(NC(C2C=CCN(C(C3CCCO3)=O)C2)=O)c(F)c1 C1(C(N(CC(O)CF)C)=O)CC2(CCC2)CN1C(c1cc([N+](=O)[O-])n[nH]1)=O c1(C(=O)NC2CC(NC(CCC)=O)C(O)C2)nc(C(F)(F)F)ccc1N C(C(CN=c1nc(C(C)C)cc(C)[nH]1)C(F)(F)F)CNC(CC1(CSC)CC1)=O N1(S(CC(C)C)(=O)=O)CCN(C(=O)C(C)(C)N(C)C)CC1CO C(C)(C)(CCC(=O)NC1CC2CCC(C1)O2)NC(C(CCC)=CCC)=O c1(C(N2CCC(F)(CNC(=O)COC3CCOCC3)C2)=O)c(F)cccc1Cl CCCCCC(O)C(=O)NCCC(C)N(C)C(c1cccn1CCC)=O C1(C(=O)NC2CCCC2C(=O)NC2CC2c2ccc(Br)cc2)CCc2nc[nH]c2C1 C1(C2CCN(C(C3CC(C4CC4)=NO3)=O)CC2)(NC(C(C)(C)C2CCC2)=O)CC1 c1(C(=O)NC(C)(C)CCCNC(=O)C=CC2CCOC2)ccc(N)c(F)c1 C(C(C)(C)C(=O)N1CC(CNC(c2nc(C3CCCCC3)no2)=O)C1)N(C)C CC1(C)CN(C(C2COC3(C2)CN(C(C2CC2C(C)(F)F)=O)C3)=O)CCCO1 N1(C(c2cccc(OCCC)c2)=O)CCC2(NC(c3cc(C)no3)=O)CC2C1 C(=O)(C1=C(C)CCOC1)NCC(C(=O)NC(CCCC)CC)CC1CC1 N1(C(C(C2CCC2)OCC)=O)CCC2(CCCN2C(=O)C=CC2CCCO2)CC1 c1(C(N2CC(CN(C(C3(COC)CC=CCC3)=O)C)C2)=O)cc([N+](=O)[O-])c[nH]1 C1(CNC(C2(OC)CCOC2)=O)COCCN(C(=O)CC2OCCCO2)C1 C=CCCCCCCC(=O)N1CCC2C(CCN2C(=O)CC(O)C(C)C)C1 C1(NC(CCSCCC)=O)CCOC12CCN(C(C1CC(C#N)(OC)C1)=O)CC2 c1(CCNC(=O)C(F)Oc2ccc(F)cc2)nccc(-c2ccccc2)n1 N1(C(C2(OCC)CC2)=O)CC(NC(C2CCc3nncn3C2)=O)C(C2CC2)C1 N1(C(c2c(OC)csc2)=O)CCCC(CNC(c2ccc(CN(C)C)[nH]2)=O)CC1 C1(NC(C2N(C(CC)=O)CCCC2)=O)CCC2CCN(C(=O)COCCO)C1C2 C1(c2ccc(OC)cc2Br)NC(=S)N(c2cccc(C)c2)C2=C1C(=O)NC(C)C2 C12(O)CCCN(C1)C2=O.N12CCC1C2.C1(CNC(=O)OC(C)(C)C)CCCC1 C(C1CCCc2nccn21)NC(N(c1ccsc1)CCOC)=O Cc1nonc1CC(=O)NC(C)(C)C=CC(=O)N(C1CC2(CC2)C1)C c1(OC)ccc(C(=O)NCC2(NC(c3nnn(C(C)(C)C)n3)=O)CCC2)s1 C1(CNC(c2ccn3c2CCCC3)=O)CC2(CO1)CN(C(=O)CC1CC1(Cl)Cl)C2 Cc1nc(N2CCN(C(=O)CC3CC=CCN3C)CC(O)C2)c2ccsc2n1 N1(C(COCCC)=O)CCC(N(C(=O)C(C)(C)OCCOC)C)CC1 C1(NC(C2C(C)(C)C2(C)C)=O)CN(C(=O)C2=NNC(=O)CC2)C2(CCCOC2)C1 CC(C)CC(C)C(=O)N1CCC(C(CO)NC(=O)CC2C=CCCC2)CC1 c1(C(=O)NC2CN(C(C3(F)CC3)=O)CCC2F)cc2cccnc2o1 c1(C(C(=O)NCCCSC)N(C2CN3CCC2CC3)C)cn2cc(Br)ccc2n1 Cc1nc(C(=O)NCCCOCCOCCNC(C2(C)COC(=O)C2)=O)[nH]c1C N1(C(CS(=O)(=O)NC)=O)CCN(C(=O)C(C2CCCCC2)O)C2CCCCC2C1 C12(CNC(C(C)c3cncs3)=O)CC1CN(C(c1csc(Cl)n1)=O)C2 CC#CCC(CO)NC(=O)CCN(C(C1CCCCCC1)=O)CC CCC(CC)(CCNC(C1CCCC(O)C1)=O)NC(c1cc(C(F)F)no1)=O C(=O)(CCCCC(C)(C)C)N1CC(O)CC(NC(C2(CC)CCC(O)CC2)=O)C1 N1(C(c2n(CC)nc(C)c2)=O)CCCC2(CCN2C(=O)Cc2nnc(C)s2)C1 CCC(CC)C(C)C(=O)NCC(F)CNC(c1ncoc1-c1cnn(C)c1)=O C1(C(=O)NC(CNC(c2ncc(C)cc2O)=O)CC(C)C)CCC2CCCCN12 C(CC(=O)NC1CC2C(NC(c3nnn(C)c3CC)=O)C2C1)(C(C)C)OCC c1(CC)ccc(OC2(CO)CCOC2)cc1N=c1nc(OCCO)[nH]s1 C1(NC(=O)CCc2ccsc2)CCC(O)CN(C(=O)CN2CCCS2(=O)=O)C1 C1(C)(NCc2cccc(Br)c2Cl)CC(NCC)c2ccccc2O1 C1(CC(N2CC3C(CNC(c4cnc(C)n4C)=O)C3C2)=O)CCCCC12CC2 CC(C)(C#CC(=O)N1CC(N2CCCC2)C1)CNC(c1cnc2ccccn12)=O c1(C(N2CCC(CN(C(=O)CSc3ccccc3)C)CC2)=O)ccn2ccsc12 C=CCCCCCC(=O)NCC1CCCCCN1C(C1CNC(=O)N1)=O N1(C(CC2(F)CN(C(=O)OC(C)(C)C)C2)=O)CC(OOC(=O)C(C)(C)C)C2CC12 C1(CSCCNC(=O)NC(CCCC)C)CCCN1S(=O)(=O)N(C)C C(c1c(Cl)cccc1Cl)=CC(=O)NC1CN(C(c2cn(CC=C)nc2)=O)CC1O C(=O)(C1=COCCC1)NC1CC(F)(CNC(C2(CC)CCCC2O)=O)C1 N1(C(C(C)OC)=O)CCOC(CNC(=O)CC2CC(C)=NO2)C1 C=CC1(C(=O)NCC2CN(C(=O)OC)C2)CCN(C(c2ccnn2CC)=O)C1 C1(NC(C2CC(C)SCC2)=O)CCN(C(c2cc(O)nn2C)=O)CC1F N1(C(Cc2c(Br)cn(C)n2)=O)CCCCC(NC(C2(C)CC=CCC2)=O)C1 C#CC1(F)CCN(C(C2C3CC3CN2C(=O)C(C)OC)=O)CC1 C(=O)(N=c1[nH][nH]c2cc(F)ccc12)c1c(OCCOC)nccc1 C=C(C)CCC(c1nnnn1CC(F)F)NC(C)C(C)C C(=O)(C1=NOC2COCC12)NCC1(CNC(CC(CCC)C)=O)CCC1 CC(C)CC(F)C(=O)N(C1CCCCC1N(C(=O)CCSc1ccccn1)C)C N1(C(CC(C)C2CC2)=O)CC2(CO)CC1(C(=O)NCC1CC13CCCCC3)C2 c1(C(N2CCC(O)(C(CNC(C(F)=CC)=O)C)C2)=O)cc(C)cc(C)c1N Cc1ccc(NNC(=O)c2cccc(S(=O)(=O)NCc3ccco3)c2)cc1F c1(OC)cnc(F)c(C(N2CC(CCNC(C3C4CCCCC34)=O)(OC)C2)=O)c1 c1(CC)ccc([N+](=O)[O-])cc1C(=O)NCC1CC1NC(c1cnc(Cl)c(N)c1)=O N1(C(CN(C2CCOC2)CCC)=O)CCCC(O)(CC)C1 C1(C(C)C)CCCCCN1C(=O)CS(C)(=O)=O.c12cccc(c1)CN2 CC(CS(C)(=O)=O)C(=O)N1CC2CCC1CC2NC(C1(CO)CC1)=O c1(C(=O)NCC(C)NC(c2ccns2)=O)csc(-c2ccoc2)n1 Cn1nc(C(=O)NCC2CC3(CCN(C(C4(Cl)CC4)=O)C3)CO2)c2ccccc12 N1(C(CCC2N(C(Cc3c(C)n(C)cn3)=O)CCC2)=O)CCCC2(CCOC2)C1 c1(C(=O)NC2(CNC(c3cc(N)cc(F)c3)=O)CCC2)c[nH]c2nccc(Cl)c12 C(=O)(C1CCCc2nc[nH]c21)N1C2CN(C(C(CC)F)=O)C(CC2)C1 C(=O)(CCCC(C)(F)F)NC(CC(C)NC(c1n(CC)ccc1)=O)C N1(C(c2cc(OC)c(Br)c(OC)c2)=O)CC2CC(C1)CN(C(=O)CC(C)(C)O)C2 c1(C(=O)NCCN(C(=O)C(=Cc2cccnc2)F)CC)ccc(O)c(C(C)=O)c1 N1(C(C(CCF)NC(C(C(C)(C)C)OC)=O)=O)CCC2(CCC2)CC1 C1(C(=O)NC(CC)(CO)CO)CCCN(C(c2ccccc2Br)=O)CC1 S(=O)(=O)(c1cc(Br)c(F)cc1F)N1CCC(C(=O)NC(C#C)(C)C)CC1 N1(C(CC(=C=C)C)=O)CC2(CCCN(C(=O)C(C)CC3CCC3)C2)C1 C1(CNC(CN(C)C)=O)CC2CCC1N2C(c1ncc(C(F)(F)F)s1)=O C1(C(=O)Nc2c[nH]nc2C2CCOCC2)NCCC1C1CCC1 Cc1ccc(C(=O)NC2CCN(C(C3(C)CC4(CC4)C3)=O)CC2F)cc1F CN1C(=O)NCC1C(=O)NCC1CN(C(C2CC(n3ccnn3)C2)=O)CC1O CC1CCN(C(C2C3CCCC3CN2C(=O)CCc2ccncc2)=O)CC1(F)F C1CCCC(=O)C1.C(CCNC(=O)CNC(=O)CNC(=O)C1CC1)N(C(C)C)C C(C)(CCC(=O)NC(CNC(=O)CN(CC(=O)NC1CC1)C)C(C)(C)C)SC c1(COC(CNC(CCCOCC)C)=O)ccc(-c2ccccc2F)n1C n1(CC(=O)N(C)C)cc(C(=O)NN2CCCC2)nn1.C12CCN(C1)C(=O)CN2C C1(NC(C(CSC)CC)=O)CN(C(C)(C)C)CCC1(C)C c1(C(=O)NCC2OCCC(NC(CCC(=C)Br)=O)C2)ccc(F)c(C)c1 C12(NC(c3ccc(OC)cn3)=O)COC(C1)C(NC(=O)C=Cc1ccc(C)o1)C2 N1(C(C(CSC)C)=O)CC(CNC(=O)Cc2cc[nH]n2)CC(C)C1 c1(CNC(C=CC(CC)C)=O)cc(C(N2CC(OCCO)C2)=O)ccn1 c1(CC)ccc(C)c(C(N2CC3CC(N(C(=O)C(C)(C)CC4CC4)C)C2C3)=O)c1 C(=O)(C(C)(C)C(F)c1ccccc1)NC1C(OC)CN(C(=O)CC2(O)CCC2)C1 C1(C(N(CCCNC(=O)C(C)Sc2ccccn2)CC)=O)CC=C(C)CC1 N1(C(C2C(C)OC(C)C(C)C2)=O)C2CCC1CC(CNC(=O)Cc1ccon1)C2 C=C1CCN(C(=O)CC(C)n2ccnc2)C(C(=O)NCC(O)C=C)C1 c1(C(N2CCCCC2c2ccc(Cl)nc2)C(=O)NC2CC2)cc(Cl)c(Br)cc1F N1(C(c2cn(CCCC#C)nn2)=O)CCC(NC(=O)C(C)(C)CC#C)C(C)C1 c1(NC(CC2C(CNC(c3ccc(OC)cc3)=O)C2)=O)cnc(OC)cc1C C(=O)(C(CC)C(C)C)NC(CNC(c1cncc(NC(CC)=O)c1)=O)CCOC N1(C(N(CCCNCc2ccc(Br)cn2)CCC)=O)CC(COC)OC(C)(C)C1 N1(C(C(CC)(C)CNC(=O)CNC(C2CC2C)=O)=O)CC2NC(=O)OC2C1 c1(C(C(=O)NCCCC2CC2)N(C)CCc2cccc(O)c2)nccc(Cl)c1Cl N1(C(C(C=C)(F)F)=O)CC(C2CCN(C(=O)Cc3cn(C)nc3C)CC2)C1 C1(NCc2ccc(OC(C)C)cc2Cl)CCCCC12CCNCC2 N1(C(C(CC)OCC)=O)CCCC(CNCc2ccc(CC)cc2)CC1 C1(C(=O)NCC(C2CCN(C(C3CCN(C)C3)=O)CC2)C)CCCCC1O CC1CCCCN1C(=O)CC(C)NC(c1cncc(CO)c1)=O Cc1cccn2c(C(=O)NC3CC3CNC(c3ccc4[nH]ccc4n3)=O)cnc12 C1(NC(C=CC(C)NC(=O)CC2CC=CCC2)=O)CC2CCC(C1)C2O Cc1cc(C(=O)N(C)CC2CCCCN2C(=O)CCn2ccnc2)c(C)o1 C1(C(N(CCN(C(CCc2c(C)ncs2)=O)C)C)=O)CCC(=O)CC1C C(=O)(C(F)CC(C)(C)NC(=O)OC(C)(C)C)N1CC(CC)C(C)C1C N1(C(CC2CC(OCC)C2)=O)CCC(NC(c2coc(Cl)c2)=O)C1(C)C N1(C(C2N(C(CC(CC)C)=O)CC=C2)=O)Cc2cnn(C)c2C1 c1(OCC)n[nH]cc1C(=O)NCC1(NC(=O)C(O)CN2CCOCC2)CCOC1 CC1(C)C2CCC1(C)C2C(=O)NCC1CCCN(C(c2cc3n(n2)CCC3)=O)C1 C1(C(C)NC(c2c(CC)c[nH]n2)=O)CCN(C(c2ccc(C)s2)=O)CC1 c1(C(N(CC(CNC(C(CC)(C)COC)=O)O)C)=O)ccc(OC)c(OC)c1C C(CCN(C)C(c1cccc(CC(C)C)c1)=O)(C(C)C)NC(C(CSC)O)=O N1(C(C2CN(C(N(C)C)=O)C2)=O)CCC(F)(C(N2CCOC(C(N)=O)C2)=O)CC1 Cc1c(C(N2CC(n3cc(-c4ccncc4)nn3)C(C)C2)=O)cnn1CC(F)F C1(CCCC)CCC(C(=O)NCC(C)(C)NC(=O)C(CC)SC)CC1 CC(C)C(C)C(=O)N1CCC(C)(CNC(=O)CCc2cccc(O)n2)C1 C1(CNC(C2CC(SC)C2)=O)(CNCCC2CCCCO2)CC=CC1 N1(C(=O)Nc2ccc(OCC)cc2)CCN(C(=O)CCCCOC)C(CO)C1 c1(C(=O)NCC(C)CNC(C2CC3CCC2CC3)=O)cc2ccsc2s1 N1(C(CCC(=C)Cl)=O)CC2CC1CN(C(c1cccc(-c3cnn(C)c3)c1)=O)C2 C1(O)(CNC(CC(=O)NCC#C)=O)CCN(C(=O)CS(=O)(=O)NC2CC2)CC1 C1(CC)(NC(c2ccc(C)nc2OC)=O)CCN(C(c2cnc(C)[nH]2)=O)CC1 CCCCCCCCCC(C)CCNC1CCC(C)C(C)(C)C1 N1(CC(=O)N(CCCCCNC(c2ccncc2)=O)C)C(=O)CC(C)(C)C1=O S(=O)(=O)(c1cccs1)N1CC2(C(C(=O)Nc3cc(C)nn3C(C)C)C2)C1 C#CCC(COCC)NC(=O)NCc1cnoc1C(C)C C1(C(N2C(C(C)C)C(NC(=O)CCc3cscn3)CC2)=O)OCCOC12CCC2 C1(C(N(CC(=O)NCCc2cnnn2C)CCOC)=O)CCC(C)(CC)O1 c1(CC(C(=O)NC2CC(N(C(=O)CN3CCCC3=O)C)C2)O)ccccc1Cl c1(C(=O)NC2CC3CC(NC(=O)Cc4nc[nH]n4)C2C3)ccc(O)nc1Cl c1(C(=O)NCC2C(NC(CCCC(=O)OC)=O)C2)cc2n(n1)C(C)CCC2 c1(CC(=O)NCCC2(CNC(C3(C(=O)OCC)CC3)=O)CC2)ccc(Cl)cc1F c1(CC(=O)NC2CC(CNC(c3c(C(C)C)ccs3)=O)C2)c[nH]c2cnccc12 C12CC3(C1)CC(C3)N2CC(=O)NC12CCC1C2.CC1(C)CN(CC(F)(F)F)C1 C1(NC(CC(=C)C)=O)CC(CNC(c2cc(CC)ccn2)=O)C(O)C1 N1(CC(=O)NCC2CC2Nc2ncc([N+](=O)[O-])cn2)Cc2ccccc2C1=O CC1(C(=O)NCCOC2CCN(C(c3csc(O)n3)=O)C2)COC(=O)C1 CC1C(NC(=O)CN2CCCCCC2)CC2CCC1N2C(C12CC(C)(CO1)C2)=O n1(CC)ncc(Cl)c1C(=O)N(C(C)CCNC(=O)C(C#N)=CC1CC1)C C1(C(=O)NC2C=CC(C(=O)NCCC3(COC)CC3)C2)COCCC1C c1(C2C(C(N3CC(O)C(O)C3O)=O)CC(=O)N2)ccc(Br)cc1F C1(C(N2CCC(SC)C2)C(=O)Nc2ccccc2C)C2(CCC2)C12CCC2 C(N=c1[nH]c2c(s1)CC(C(=O)O)CC2)c1cccc(NC(C2=NOC(C)C2)=O)c1 Cc1cncc(CNC(C2(CNC(=O)C(C)c3ccco3)CC3(CC3)C2)=O)c1 CCCC(O)C(=O)NC1CCN(C(=O)Cc2cnn(C)c2)C1CC c1(C(=O)NCC2(F)CCCCN(C(COC(C)=O)=O)C2)nccn2nc(C)cc12 N1(C(c2c(C)occ2)=O)CCC(C)C1CNC(C1CC2CCC1O2)=O C(CC(CNC(=O)CCc1cnco1)NC(=O)CSC(C)C)OC CN(C)NC(=O)CCC(=O)NC12CCCC1N(C(C1C3CCCC13)=O)CC2 C1(CN(CCOC)CCNC(=O)CCc2cc(OC)no2)CCC(C)(C)C1 Cc1csc(=O)n1CC1(C(=O)Nc2ccc(-c3cccc(O)c3)o2)CCC1 N1(C(C23CN(C(CC4CC(=O)NC4=O)=O)C(C2)CO3)=O)CCC2(CCCOC2)C1 CC(CCC(=O)NC1COC(=O)C1)NC(=O)CCN(C)C C(=O)(N=c1[nH][nH]cc1C(N)=O)C1CCN(Cc2cccc(OC)c2O)CC1 n1(CC)ccc(C(=O)NCC(C)(C)CN(C)C(C2(C#N)CCCO2)=O)cc1=O N1(CC(=O)NCC2CCCN2C(=O)C=CC2CC2)CCNC(=O)C1 CCCC(CCCNC(=O)CC1C=CCC1)NC(c1cn(CC(N)=O)nn1)=O N1(C(c2cc(C)c(C)s2)=O)CCC(C2CC2)C1C(=O)NC1(CO)CCC1 C(C(C)C(=O)N(CCC(=O)NC1CC=C(C)CC1)OC)N(CC)CC CC(CN(C)C)C(=O)NCCOCCOC1CC(CNC(=O)COC2CCC2)C1 CC(=NO)c1cc(C(=O)N(C2C3CN(C(=O)Cn4cccn4)CC23)C)cnc1O n1(CC(N2CCCN(C(=O)CNc3ncccn3)CC2)=O)cc(F)ccc1=O C(=O)(CCC(=O)C(C)(C)C)N1C(C(N2C(CC=C)CCCC2)=O)CN(C)CC1 N12CCC3C(C3C1)C(=O)NC(CC#C)C2=O.c1(COC)ccnc(O)c1 c1(CC(N2CC(N(C(CC3(OC)CCC3)=O)C)C(F)C2)=O)ccc(F)cc1Cl c1(C(=O)NC(CC2CCOC2)CO)cnc(N2CCCCC2)s1 C(=O)(CCC(F)(F)Cn1cc(-c2ccc(F)cc2)nn1)N1C(COC)COCC1 C1(NC(C(CNC(c2ncn(C)c(=O)c2)=O)(C)C)=O)CCn2nnnc2C1 c1(NC(C(c2n(CC)nnn2)N2CCCC2)(C)C)cc(CO)ccc1C C1(N(C(C(C2CC(F)(F)C2)OC)=O)C)CCCN(Cc2ncccc2O)CC1 C1(CC)CN(C(=O)CC2CC2(Cl)Cl)CCN1C(c1cc(C#N)cs1)=O C1(C(=O)NCC(C)OCC#C)CN(C(=O)C(F)C2CCCC2)CCC1(C)C C(=O)(C(C(C)(C)C)n1ccnn1)NC(C)C(C)(C)NC(c1cnn(C)n1)=O C(=O)(C1=COCCC1)N1C(C(=O)NC2CC(F)C2)CC(O)C1 N1(CC(=O)NCCNC(C(C)(C)NC(=O)OC(C)(C)C)=O)CCCOC1=O c1(OC(C(=O)N(C(C)CNC(c2ccncc2)=O)CC)C)cc(C)c(F)cc1F C1(NC(C(CSC)OC)=O)CCCC2CN(C(c3ccc4c(c3)OCO4)=O)CC12 C1(CCNC(C(CC=C)(F)F)=O)CCN(C(=O)CCSCC(N)=O)CC1(F)F N1(C(CN(C(=O)OC)C)=O)CCC(C(=O)NCC2CCCO2)(CO)C1 C(=O)(C1CCCc2c[nH]nc21)NC1(C)CN(C(c2ncc(C)nc2)=O)C1 CC(C)CCC(=O)NCC(=O)NC1(CNC(C2C3CC3C3CC23)=O)CCC1 C#Cc1ccc(F)c(C(=O)N(C2CN(C(=O)CC3CCCC(=O)N3)C2)C)c1 CCCCCC(O)CC(=O)NCC1CCN1C(c1sccc1-n1ccnn1)=O C(C)(C)(CCC(=O)NC1(C(=O)NCc2cnccn2)CC1)OC CC1CCN(C(C2CSCCS2)=O)CC1CNC(C1CSCC(=O)N1)=O c1(C(N2CC(C)(NC(C(C)CN3CCCCC3)=O)C2)=O)nccc2ccccc12 Cc1cc(=NC(=O)CC2CC3CCC2N(C(=O)OC(C)(C)C)C3)[nH]n1CC(N)=O Cc1csc(CC(N2CCCC2C(C)(C)C(=O)NCc2cnc(C)s2)=O)c1 C1(C(=O)NC2CCCSCC2)CCC2(CC2)N1C(C1CC(F)(CF)C1)=O N1(C(Cc2c(OC)cccc2)=O)CCC2(CCC2)C(CNC(=O)CC2CCC2)C1 CC(C)(C(=O)Nn1cc(CC2C(CCNC=O)CCC2)nn1)N1CCCCC1 C1(C(C)NC(C2C3CCCC23)=O)CCN(C(C2CCCN2C(N)=O)=O)C1 c1(CC(N2CCC(O)(C(C)NC(COC)=O)CC2)=O)ccc2c(c1)CCN2C CC(=O)C(C)CC(C)C(=O)N1C2CCC(C2)C1C(=O)N(CC(C)O)CCO N(C1CN(C(C2CC2F)=O)Cc2ccccc21)C(c1c(C)nn(CCC)c1C)=O C1(C(=O)NC2CSC2)CN(C(C2CN3CCC2CC3)=O)C2(CCC2)C1 N1(C(c2c(CC)onc2C)=O)CCC(C(=O)NC2CCCNC2=O)C(C)(C)C1 c1(OC)ccc(Br)cc1CNc1cn(C)c(C(N2CCC(C(F)(F)F)C2)=O)n1 Cc1cc(OCC(=O)NCC(O)CNC(c2c(C)cncc2C)=O)ccc1F C(c1cccc(C#N)c1)=CC(=O)NCCN(C)C(C1(C2CCC2)CC1(F)F)=O C(CN=c1[nH]c(N2C3CCC2CC(F)(F)C3)nc2c1CSC2)(C1CC1)OC C1(C(=O)NCCC(C)CCNC(c2cnns2)=O)C2Cc3cc(Cl)ccc3C12 C1(C(N2C(C(=O)N(C)Cc3sccc3C)(CC)CCC2)=O)CCCC(=O)N1C N1(C(C2C(CC)C2)=O)CCN(C(c2nnc(O)nc2O)=O)CC1C C1(O)(CN(C(=O)C(F)F)C)CCN(C(=O)C(F)=CCCF)CC1 N1(C(CCC=C)=O)CC2CC2(CNC(=O)Cc2cccc(I)c2)C1 c1(CC)ccc(NC(=O)CC(C)n2ccnc2-c2ccc(C(=O)OC)s2)c(OC)c1 CCC(CN(C)C)CC(=O)N1CC(C)C(C)(CNC(=O)CCC(=O)N(C)C(C)C)C1 N1(C(COCCOC)=O)CCC(CNC(=O)CC2CC(C)=NO2)C1 C(=O)(C1CCCn2nccc21)NCCCC(C)NC(c1ccc(C)c(CO)c1)=O C1(N(C(c2cnn(C(C)C)n2)=O)C)CN(C(c2cocn2)=O)CC1F C(=O)(C1Cc2ccccc21)NCC1(F)CCCN(C(Cn2cnc(C#N)n2)=O)C1 c1(C(N(C2CCN(C(=O)C(Cl)=CCl)C2)CCC)=O)ccc(C2CC2)cc1F C12CC(O)CN(C1)C2=O.c1(C(C(=O)C(Cl)(Cl)Cl)=O)ccc(Cl)c(Cl)c1.C12CN(C1)NC2=O c1(N2CCCC(=C)C2)nc(N2CCS(=O)(=O)C(C)C2)nc2c1CCCCC2 Cc1c(C(=O)NCC(C(C)C)NC(C2(O)CCC(C)CC2)=O)cccc1C1CC1 N1(CCCC(=O)NCC(CNC(=O)C(C)OC(C)C)OC)CCc2ccccc21 c1(C(=O)NC2CCOC(C(=O)NCC3(O)CCC3)C2)cc2cnccc2[nH]1 c1(C(N2C(C)CN(C(CC)=O)C(C)C2)=O)cccc2c1CCS2(=O)=O c1(C(=O)NCC(C)(C2CCC2)NC(Cc2c(C)nc[nH]2)=O)cc(C)n(C(C)C)n1 C1(F)(C(N2CC(O)(C(C)NC(Cn3c(C)ccn3)=O)C2)=O)CCOCC1 C(=O)(CC(C)(C)C1OCCO1)N.C1(=O)C#CCCCN1.c1(C2(C)CC2)ccccc1 c1(C(=O)NCC2C(CNC(c3c(C)nsc3)=O)C2)cnn2c(C)ccnc12 c1(C(=O)NCC2C(NC(c3cccc(NC(N)=O)c3)=O)C2)cccn2cncc12 CC1C(NC(=O)C(N2CCCCC2=O)C)CCCN1C(=O)CC12CCC(CC1)C2 C1(C(=O)NCC2(OC)CN(C(c3c(SCC)cccn3)=O)C2)CCCC(C)CC1 C(=O)(CC(CC)C(C)(C)C)N1C(C2(C(=O)NC(CC#C)CCOC)CC2)CCC1 C(=O)(CN=c1ccc(Cl)n[nH]1)N1CC(CNC(=O)C=Cc2cocn2)OCC1 C1(NC(C2CCOC2)=O)C2CC(O)C1N(C(c1c(Cl)nsc1Cl)=O)C2 C(C(C(=O)N1CCC(c2nn[nH]n2)C1)C(C)C)NC(C(CC)C#N)=O C1(CCNC(C2CC2(Cl)Cl)=O)(NC(C(N2CCSCC2)C)=O)CCOCC1 C1(C(=O)NC2CC(CC(=O)NC3(CCCC)CC3)C2)(C(F)F)CCCC1 c1(OCCC)cc(F)ccc1NC(N1CCCC1C(C)(C)CO)=O CC(C)C(F)(CNC(=O)CN(C)C1CC1)C(=O)NCc1csc(O)n1 C(=O)(C#CC(C)(C)O)NC(c1n(C)ncc1)C(N1CCOC(C)(CO)C1)=O Cc1nnccc1C(N1CC=CC(NC(=O)CCc2ccsc2)C1)=O C1(CNC(C(CCC)CC)=O)CC2(CO1)CN(C(=O)Cc1ccsn1)C2 C1(C(N(CCNC(C2CC(C(F)(F)F)CO2)=O)CC)=O)CC(=O)NC(=O)C1 C1(CC#C)CN(C(=O)CCN(C(c2c(CO)n[nH]c2C)=O)C(C)C)CCO1 N1(C(C(C(C)O)(F)F)=O)CCC(C2CC2)(NC(c2snc(Cl)c2Cl)=O)C1 C(=O)(CCCC(=O)NC1CN(C(=O)CNC=O)CCC1c1ccccc1)N(C)C C(=O)(CN=c1cc[nH]cc1)NCCN(C(c1cc(C2CC2C)on1)=O)CC C1(C(=O)NCC2(C(=O)OC)CCC2)CCCCN1C(c1n[nH]c(C)c1Cl)=O N1(C(C(CC)O)=O)CC(CN(C(=O)C2=C(C)CC2)Cc2ccccc2)C2(CC2)C1 CC1(NC(=O)C(C2CCOCC2)O)CCCC1NC(=O)C(O)CC1CCCC1 c1(C(=O)NC(COC)CNC(C2CCC2)=O)cc(C)c(C)o1 CC1OC2(C(=O)NCC3(O)CN(C(C4(CF)CC4(F)F)=O)C3)CCC1CC2 c1(CCC(=O)OCc2ccc(-c3ccccc3)o2)ccnn1CC1CCC1 C(=O)(C(C)(C)C(=O)N(C)C)N1CCC(C(C)NC(Cn2nnc(C)n2)=O)CC1 c1(SC)ccccc1CC(=O)NCC1CC1CNC(c1cnc(Cl)s1)=O c1(CC)[nH]c(=N)sc1C(N1CCC(N(C(C2CC(F)(F)C2)=O)CC)C1)=O C(=O)(C(C(C)(C)C)SC)NC1(CNC(COCCCC)=O)CCCCC1 N1(C(C=CCC)=O)CC2(C1)C(NC(=O)C(F)=C(C)C1CC1)CCS2(=O)=O N1(Cc2cncc(C)c2)CCCC2(CCN(C(=O)C(C)Cc3ccccc3)C2)C1 c1(OC)cccc(I)c1C(N1CC2(CC(C(=O)Nc3ncc(F)cc3Br)C2)C1)=O c1(N(C)Cc2cccc(C(C)C)c2)ccc([N+](=O)[O-])cc1-n1cnnn1 c1(C(N(CC(CNC(c2n(CCC)ncc2)=O)O)C)=O)ccc(Br)nc1O c1(C(=O)Nc2scc(C(=O)OCC)n2)cnc2c(-c3ccc(F)cc3)cnn2c1 C1(C(N2C(CCNC(=O)Cn3cccn3)CSCC2)=O)CC2CCC(C1)O2 C1(OC(C(=O)NCC(CNC(c2n(C(C)C)nnc2)=O)F)C)CCCCCC1 Cc1ccc(CNc2ccc(F)c3cnccc23)c2ccccc12 CC1CCC(CNC(c2cc(N)c(Cl)cn2)=O)N(C(c2cc(C(F)F)no2)=O)C1 c1(C(=O)NCCCN(C(C(CC)c2ccccc2)=O)C)ccc(F)c2c1CCC2 N1(C(CCC=CC)=O)CCC(NC(c2noc(C3CC3)c2C)=O)CC1C1CC1 C1(NC(C)CCCc2cccnc2)CCc2nnc(-c3cccc(F)c3)n2C1 Cc1cc2c[nH]nc2cc1C(=O)NC1CC1NC(c1csc(Cl)n1)=O C1(NC(C2CCCC(OC)C2)=O)CC2CCC(C1)N2C(=O)C(C)CS(C)(=O)=O C1(C(=O)NC2CCN(CCc3ccns3)CC2)C2CCCCCCC12 CCN=c1cc(-c2nc(N3CCCCCC3)no2)cc[nH]1 C(=O)(C1=CC2(CCOCC2)C1)N1CC(CN(C(c2c(C)cncn2)=O)C)OCC1 c1(C(=O)O)cn2c(n1)CC(C)CC2.c1(NC(C(=O)N(C)CC)=O)ccsc1C(F)(F)F c1(C(=O)NCC(CC(C)C)NC(CCC)=O)cc(N2CCCC2=O)ccc1Cl c1(C(N2CC(C)C(NC(C3CC34CCSCC4)=O)C2)=O)n[nH]c2ccc(O)cc12 C1(CC(=O)NCC(C)(C)C2CC2)(NC(=O)Cc2cnsc2)CCCCC1 c1(C(=O)NCC2CCCCN2C(c2scnc2Cl)=O)nccnc1C(F)(F)F CN(CCCC(=O)NCC(C)(C)NC(C1CN(C(=O)N(C)C)C1)=O)N=O N1(C(CNS(NC)(=O)=O)=O)CC2CCCC(N(C)C(C3CSC3)=O)C2C1 Cc1csc(C(C)C(=O)NCCC2(NC(C3CCC(C)O3)=O)CCC2)n1 C(=O)(CCCCCCCS(C)(=O)=O)NC1C(CC)N(C(C2CC3CC3C2)=O)CC1 C1(C(=O)NCCCC(=O)OC)CC2(CCCC2)CO1 C1(C(=O)NC(C)Cc2nn[nH]n2)CCN(C(=O)CC2CCCOC2)C(C)(C)C1 N1(C(C(=O)NC(c2ccc(C(C)(C)C)cc2)C)=O)CCCC(C)(C)CC1 CC1(C)CC(C(N2CC3C(NC(=O)CCn4ccnc4)C3C2)=O)C(C)(C)O1 C1(NC(CC2CC(=O)NC2)=O)CC2CC1CN(C(c1cc(F)c(Cl)cc1F)=O)C2 N1(C(C2C(C(=O)OC)C2(C)C)=O)CCCC(O)(CNC(=O)CC2CC=CC2)CC1 c1(C(=O)NC2C(CNC(c3n[nH]cc3F)=O)C2)cc2ccc(Br)c(F)c2[nH]1 N1(C(CN(C2CCCCC2)C)=O)CCN(C(=O)CCc2cnc[nH]2)C(CF)C1 c1(C(N(C2C(C)CCN(C(C(C)(C)OCC)=O)C2)C)=O)cccc2nc(Cl)cn12 c1(C(N2CCC(COC)(NC(C3CC3[N+](=O)[O-])=O)C2)=O)ccc(F)c(F)c1N N1(Cc2c(C)cc(Br)cc2)CCC2CN(C(=O)CCN(C)C)CC2C1 C1(NC(C2C(C)(C)C2)=O)CN(C(C2(C)CCCCNC2=O)=O)CC12CCOCC2 C(=O)(CC(O)CCCC)NC(CC(=O)N(C(CC#C)C)C)C N1(C(Cc2nc(C)oc2)=O)CC2(CC2)CC1Cn1cc(CCCCCCO)nn1 CCCCC(C)(F)C(=O)NCC1(CNC(=O)CC(C)(C)C(F)F)CCCCC1 C1(C(=O)NC(CCSC)C(=O)N(C)Cc2cncn2C)CC(=O)NC1(C)C c1(C(=O)NC2C(NC(c3cc(CSCC)on3)=O)CC2)c(C(C)C)n[nH]c1C c1(COCC)nc(N(CCCNC(c2sncc2C)=O)C)cc(C)n1 C(=O)(C1CCc2nccn21)NC1C2(CCN(C(C=CC=CCC)=O)C2)C1 CC1(C(=O)NCc2ccc(C(=O)Nc3cncc(Cl)c3)s2)CCCC1O c1(C(=O)NCCCOCCC(=O)NC(c2nnnn2C)C)coc(C2CC2)n1 c1(SCC(N2CCC(N(C(c3ccncn3)=O)CC)C2)=O)cccc(F)c1 C1(COC)CN(C(=O)CC(=O)N(C)C)CCN1C(=O)CCN1CCCC1 C1(C(=O)NCCC(C)NC(c2ccc(C(F)(F)F)o2)=O)(OCC)CCCC1 C1(CCC=C(C)C)NC(=O)CCN(CC(c2ccccc2C)O)C1=O C(=O)(CC(C)CC(=O)NCC1CC(NC(C2CCN(C(=O)CC)C2)=O)C1)OC CCC(CCCC(=O)NC1CCC2CC1CO2)NC(c1cscn1)=O c1(-c2nc(-c3nccc(Br)c3)nn2C2CCOC2)cccn2ccnc12 C12(C(N3CCN(C(CC(CC)O)=O)CC3C)=O)CC(CO)(C1)OC21COC1 c1(CC(N2CC(C)(NC(c3cc(Cl)nnc3Cl)=O)C2)=O)ccc(F)cc1[N+](=O)[O-] C=CC1(C(=O)NC(C)CC(C)NC(c2cc(CCCCC)[nH]n2)=O)CCCCC1 C(=O)(C(O)CC(F)(F)F)NC1C(C(=O)NC(C2C(C(=O)OC)C2)C)C2CCC1C2 C(CCC(=O)N1CCCC1CNC(=O)CC1(C)CC1)OC(C)C c1(C(N(CC(C)NC(=O)CS(=O)(=O)C2CC2)C)=O)cnc(C(F)(F)F)c(C#N)c1 C1(CNC(CCCC)=O)CN(C(=O)C(CC#N)c2ccccc2)CC1SC N1(CC(C)(C)C)CC2(CC(NC(=O)CC3(c4ccccc4)CCC3)C2)C1 N1(C(c2ccc(OC)nc2)=O)CCN(C(c2ccc(C)c(F)c2)=O)C(C2CC2)C1 CC1=C(C(=O)NC(C)(CNC(=O)Cc2ccoc2)C2CCC2)SCCO1 C1(C(C)NC(=O)C(c2ccccc2)F)CCCN(C(C23CSCC2C3)=O)C1 C1(C(=O)NC(C)CCC2CC2)(CNC(c2occc2CN(C)C)=O)CCCC1 N1(C(C=CC(C)(C)SC)=O)CCCN(C(c2cnc(NC(C)C)cn2)=O)CC1C c1(C(=O)NCCNC(C=C(C)C2CC2)=O)ccc(=O)n(-c2ccc(F)cc2)n1 C1(C(=O)NC2CC(CNC(c3cc(O)cc(O)n3)=O)C2)CCC2(CCOCC2)O1 c1(OC)cc([N+](=O)[O-])ccc1S(=O)(=O)N1CC2C(C(N3CCOCC3)=O)C2C1 Cc1nn(C)c2nc(C3CC3)cc(C(=O)NCC(C(=O)O)C3CC3)c12 N1(c2ccc(F)cc2C(=O)C(C(C)C)C(C)C)C(C(F)(F)F)(OC)CC(C)C1 c1(C(N2CCCC(CCNC(=O)CC3CCCCO3)C2)=O)cc2ncccc2o1 C(=O)(C(C)C(O)C(C)C)NC1CN(C(CCc2cncc(C)c2)=O)CC1O Cc1nc(N(C2CC2)C(C2(c3ccccc3)CC(=O)C2)=O)nc2ccccc12 CCCC(C)CN(C)C(c1c[nH]nc1CCNC(=O)CCc1cc(C)[nH]n1)=O c1(C(N2C(C(N(CCCSC)C)=O)CC2)=O)snnc1C C1(NC(C(C)CO)=O)CCC2CN(C(=O)C=Cc3cnn(C)c3)CCC2C1 c1(C(N(CC(C(=O)N(CC)Cc2cccs2)C)C)=O)c[nH]c2cnccc12 CC(C)(CNC(c1nc[nH]n1)=O)CC(=O)NC(CO)CC(F)(F)F CN1CCn2ncc(CNC(N3CCC(NCCO)CC3)=O)c21 c1(C(N(C2CCC(NC(CCC(=O)NC)=O)C2)C)=O)cc(F)cnc1O Cc1cc(C(N2CCCC(CCNC(c3ncnn3C)=O)C2)=O)c(C)cc1Br c1(C(=O)NC2(CNC(c3nn(C)c(F)c3)=O)CCC2)ccc(C#N)c(O)c1 C1(NC(c2ccc(C(F)(F)CF)cc2)=O)C2CC(CN(C(=O)CO)C2)C1CO N1(C(C2(C=C)CCC2)=O)CCN(C(c2ccc(CCC)cc2N)=O)C(CC)C1 c1(C(C)NC(=O)CC2(O)CCC2)nccc(O)n1.C12(CSC1)C(=O)N2 C1(CNC(=O)CC(=O)NC2CC2)CCCN(C(=O)CC2CC3(CC3)CO2)CC1 C(C(CO)CC(C)C)NC(CN(C(C1(CC)CCOC1)=O)C)=O Cc1nc(C)c(C(N2CCN(C(C3CCN(CC(F)(F)F)C3)=O)CC2)=O)o1 N1(S(CCCC#C)(=O)=O)CCCC2(CCN(c3ccccc3)C2)C1 c1(C(N2CCC(N(C(C(C)SC)=O)C)C3(C2)CC3)=O)c(F)ccc2c1OCC2 N1(C(CC)CC)C(=S)NC(c2ccccc2)C2=C1CCN(C1CCCCC1)C2=O c1(OC)cnc(C(=O)NC(CC2CC2)C(=O)NCCCC(C)(F)F)cn1 c1(C(N2C(CCNC(C(C(C)C)C)=O)CC(F)(F)C2)=O)[nH]nc([N+](=O)[O-])c1Cl CCCCC(CCC)NC(=O)CCC(C)NC(=O)CCc1nncn1C c1(C(N2CC(NC(CCc3nnc(C)n3C)=O)C2)=O)cc2c(o1)CCCNC2=O N1(c2snc(C(=O)OC)n2)CCC(C)(NC(C2CC(F)(CO)C2)=O)C1 N1(C(c2c(C)c(N)ccc2)=O)CC2CC(NC(=O)C(F)CC3CCC3)CC2C1 Cc1ccc2sc(NC34CC(NC(C5CC6C(C5)C6(C)C)=O)(C3)C4)nc2c1C C1(NCCOC)CCCC(CNC(=O)C(C)CCOC)C1 N1(Cc2ccc(CC)cc2)CCC(F)(F)C(C(=O)Nc2cnc(Cl)c(Br)c2C)C1 c1(C(=O)NC2(C)CCN(C(C(CCO)N(C)C)=O)C2)cc2ccc(F)cc2o1 C12(CNC(CCc3n(C)cnn3)=O)CCCC(CN(C(=O)CCC(C)(C)C)C1)C2 CS(=O)(=O)CCC(=O)COC(c1cc(Br)c(F)cc1Br)=O C1(O)(C(C)C)CCN(C(=O)CCN(C(C2CCC(=O)C2)=O)C2CC2)C1 C(C(C)C(C)C(=O)NC1CC1CNC(c1cscc1C)=O)OC N1(Cc2ccc(C)[nH]2)CCC2(CCCC2C(=O)Nc2cc(O)c(Cl)cc2F)C1 c1(C(=O)NC(CC(C)NC(c2ccn(C(F)(F)F)n2)=O)C)ccc(F)c(Cl)c1 c1(OC)ccc(CC(=O)NCC(C(=O)O)C2CCOC2)c(Br)c1 C(C)(CCC(=O)N(C)CC1COCCN1C(c1occc1Cl)=O)OCC N1(C(C(CC(C)(C)NC(C(C)OCCN(C)C)=O)F)=O)CC2(CCC(=O)NC2)C1 C1(CNC(C(C(C)C)OCC)=O)CCN(C(c2cc(OC)ncn2)=O)CC1O N1(C(C(C)Nc2ccoc2)=O)CC(c2ccccc2)(NC(=O)COCCO)C1 N1(C(c2c(SC)ncs2)=O)CC(n2cc(C3CN(C)CCO3)nn2)C(C)C1 C1(NC(=O)OC(C)(C)C)C2CC(O)C1N(C(=O)C(=O)NCCCCCO)C2 c1(C(=O)NC(C(C(C)C)NC(=O)CCc2csc(=N)[nH]2)C)cc2ccccc2s1 c1(OC)ncccc1C1CCN(CCn2cc(C3CCCCO3)nn2)C1 c1(CNC(CC2C(C)C2)=O)nnn(C)c1C(=O)N(CCn1cncn1)C1CC1 CCC(CC)(CC)NC(=O)CCC1CCN(C(=O)CCC(C)SC)C1 c1(OC)cc(C(N2CC3CCN(C(=O)CC4CC4)CC3C2)=O)cc2cccnc12 C(=O)(N=c1[nH][nH]c2c1CCCC2)C1N(C(c2cc(OCC)c(Br)cc2)=O)CC=C1 C1(O)(C(C(=O)NC(CC#CC)C)(F)F)CCN(C(=O)OC(C)(C)C)CC1 CN=c1cc(C(N2CCCC2C(=O)NC2(C(C)O)CC2)=O)cc[nH]1 C#CC1(NC(C2CN(C(=O)C(CCC)NC(N)=O)CC2CCC)=O)CCCCC1 Cc1c(Cl)ccc(C(N2CCC(C(C)NC(C3CNC(=O)N3)=O)CC2)=O)c1Cl c1(C(N(C2CCN(C(=O)CC3C=CCCC3)C2)C)=O)ccnc2c1ncn2C Cc1cc(C(=O)NCC2CC(NC(c3ccc(C(N)=O)[nH]3)=O)C2)ccn1 CCC(CC)CCC(=O)N1CCC(C(=O)NC2CN(C(N)=O)C2)O1 c1(OC)ccc(C(=O)NCC=Cc2nnc(C(C)C)o2)c(F)n1 CCC(CC(=O)NCC(C)NC(=O)OC(c1ccccc1)=O)NN1CCCCC1 C(=O)(C1=CCCC1C)NC(C(=O)Nc1c(C)ccnc1)(C)C1CCC1 N1(C(CNC(CC)=O)=O)CC(NC(c2coc(CO)c2)=O)C(C)C1 c1(C(N2CCOC3CC23)=O)ccc(OCC2CC2)cc1 Cc1cc(F)sc1C(=O)NCC(O)CNC(=O)CCc1ccncc1Br N1(Cc2c(C)cccc2O)CCC2C1CCCN2C(c1coc(Cl)n1)=O N1(C(CSc2ccc(OCC)cc2)=O)CCC2CCN(C(=O)C3=CCC3)CC12 C1(CC(=O)NC2CCC(c3cc[nH]n3)O2)CN(C(c2ccco2)=O)CCO1 CCC(CNC(=O)CCCCCNC(c1c(C)noc1C)=O)CC(C)C n1(C(c2nnnn2C)C)cc(C2NC(=O)Nc3c(N(C)C)cccc32)cn1 c1(N(CC(CC)C)C)ccc(S(=O)(=O)NC(CC(C)C)CS(C)(=O)=O)cc1C#N O=C1CC(CC(=O)N2CC3CC2CN3C(c2ccn3ncnc3c2)=O)=NN1 C(C)(CC(=O)NCC1(C)CCN(C(=O)C(C)(C)CO)CC1)(C(F)(F)F)N(C)C C12(C(=O)NCCC(C(C)C)C)CC(CO1)N(C(=O)CC13CCCC1C3)C2 c1(C(C)(C)C)ccc(O)c(C(=O)NC2CC2C(=O)NCCCc2ccccc2)c1 N1(C(C2(CSC)CCC2)=O)CCC(NC(c2cc(Cl)ns2)=O)C(O)C1 c1(C(=O)N(CC2CC(NC(C3C(C)C3)=O)C2)C2CC2)cccn1C1CC1 N1(C(CC2N(C(=O)COc3ccccc3)CCOC2)=O)CCC12CCCOCC2 C1(C(=O)NC2CCC(C(N)=O)C2)(OC)CCN(C(=O)C(O)CCl)C1 N1(C(CCc2c(C)nn(C)c2)=O)CCOCC(CNC(=O)C(C)CN(C)C)C1 C(CCCC(=O)NC1CN(C(C2CCCN(CC(F)F)C2)=O)C1)NC(N)=O CC(C)CC(C)C(=O)N1CCC(F)(CNC(=O)C(C)(C)C2CCCO2)CC1 C12(C(N(CCNC(c3noc(CC)c3C)=O)C3CC3)=O)CCOC1CS(=O)(=O)C2 Cc1cc(C(=O)NC(c2nc(C(N3CC(n4cc(CO)nn4)C3)=O)co2)C)co1 C(=O)(C1CSc2ccccc21)NC(CNC(c1c(C)c(O)ccc1)=O)C1CC1 C(=O)(CCCCC(C)(C)C)N1CC(CC)N(C(=O)CCOC)CC1 c1(CC(=O)NC2CCC(NC(C(F)OC)=O)C2)cn(C)c2ccccc12 c1(COC(C)C)ccc(C(=O)NC2CC(NC(C3CC4CC4C3)=O)C2)cc1 c1(NC2(CCNC(C3N(S(C)(=O)=O)CC3)=O)CCCC2)cc(O)nc(O)n1 c1(OC)c(C(N2CCC2CNC(C2(CS(C)(=O)=O)COC2)=O)=O)c(C)nn1C c1(OC)ccc2cc(-c3c[nH]nc3C(=O)Nc3cn(C)cn3)ccc2c1 C1(N(C)C(C2CNC(=O)C2)=O)CCCCN(C(C2(F)CC=CC2)=O)C1 N1(C(CN2CCC(C)C2)=O)CCN(C(=O)CCC2CCCN2C)CC12CC2 Cc1cc(C(=O)NCC2CCCN(C(c3nc(O)sc3C)=O)C2)ncc1C(N)=O C(=O)(CCCCCS(N)(=O)=O)NCCCCC(CO)NC(C1(COC)COC1)=O c1(OC(C)C)cccc(C(=O)NC2CC(NC(C3(O)CCCCCC3)=O)C2)c1F N1(C(C2N(C)CCC2)=O)CCC2(CC2NC(=O)CC2CCCCO2)C1 C1(NC(c2c(C)ncn2C)c2n(CCCOC)nnn2)COC2(CCCCC2)C1 C12(CNC(c3nc(Cl)cs3)=O)CC(CN1C(=O)C=C(C1CC1)C1CC1)C2 c1(NCc2c(C)c(Br)ccc2)[nH]c(=NC(C)c2ccc(F)cn2)nc2sccc12 CC1=C(C(=O)N2CC(C)(NC(C3CCN3C(C)(C)C)=O)C2)SCCO1 c1(NC(c2nc(CNC(=O)C(F)(F)CO)n[nH]2)=O)ccc(-c2nn[nH]n2)cc1 CCC(CCC(=O)N(C)CCc1nccs1)NC(C1CC2(CCCO2)C1)=O c1(C(=O)NCC2=CCN(C(C3C(C(=O)OC)C3)=O)CC2)cccn2ccnc12 C1(C(N)=O)(NC(C(C)(C)C2CCCN2C(c2cnc(Cl)s2)=O)=O)CCOCC1 C1(C(N2CC(NC(CC(C=C)(C)C)=O)C2)=O)CCc2nc(C)cn2C1 c1(C(=O)NCC2C(NC(Cc3scc(C)c3)=O)CC2)n[nH]c(C)c1Cl c1(-c2n(CC3CC(C)C3)nc(CC(C)C)n2)cc2cc(F)c(F)cc2[nH]1 C(=O)(CC(C)C(F)F)NCC(Cc1ccccc1)N(C(C1C(CC)C1)=O)C C1(CNC(c2c(C)cccc2)=O)COCCN(C(=O)CC2NC(=O)NC2=O)C1 c1(C(=O)NC(C(=O)NCC(C)(C)C2CCC2)Cn2cncn2)cc2n(n1)CCC2 N1(C(C(C)c2ccco2)=O)CC(C(N2CCOC(C)(C)C2)=O)CC1(C)C CN1C(=O)OCC12CCN(Cc1nn(C)cc1S(N)(=O)=O)C2 c1(C(N2C(CNC(c3nn(CC)nc3C)=O)CCCC2)=O)cc(Cl)ncc1N C(=O)(N=c1[nH]ccc2cc(Cl)ccc12)C1C(NC(c2ccc(C#N)cc2Br)=O)C1 C1(O)(CCNC(c2ccnc(Cl)c2F)=O)CCN(c2ncncc2I)CC1 N1(C(c2c(C)cco2)=O)CCCC(C(N2CCCC(CS(N)(=O)=O)C2)=O)CC1 C1(CNC(c2c(C)cn(C)c2)=O)CCN(C(=O)CC2CC(=O)NC2=O)C1(C)C c1(C(N2CC(C)(C)CCC2C)C(=O)NCCC2(C)CC2)ccc2nc(C)oc2c1 Cc1ccncc1C(=O)NC1CC1NC(=O)CC1CCCCCC1 C(CCSC)(C(=O)NCC(C(F)(F)F)N1CCN(C(=O)C2=COCC2)CC1)OC N1(C(C2CC(=C)C2)=O)CC2CN(C(c3cc(CC)ccn3)=O)C2C1 C(=O)(CCCCNC(N)=O)NCC1N(C(C(c2cccnc2)OC)=O)CC1 N1(C(CN(C(C)C)C)=O)CCC(O)(CNC(=O)CN2C(=O)CSC2=S)CC1 C(=O)(C(CC(F)F)NC(c1c(O)cccc1F)=O)NC(C(C(=O)OC)C)C c1(C(=O)NC2CC(N(C)C(C3(n4cccn4)CC3)=O)C2)cc(=O)cc[nH]1 N1(C(CN(C2CC2)CC)=O)CC(N=[N+]=[N-])CC1C(=O)Nc1cnn(C(F)F)c1 C1(NC(=O)C(c2ccc(Br)cc2)=O)CN(C(c2cc(F)ccc2Cl)=O)CC1(F)F C1(C#N)(CNC(C2(C)C=CCN2C(=O)CC2CCCC23CC3)=O)CCCCC1 O(NC(=O)C(C)C(C)NC(c1c(C)ncnc1C)=O)CCCC c1(C(N2CC(CCNC(c3cc(CC)no3)=O)OCC2)=O)cc(C)c(F)cc1Cl CC1(C)CCN(C(c2csc(Cl)c2)=O)CC1CNC(c1cc(Cl)ncc1O)=O c1(-c2cc(C(N3CC(CNC(CC(C)C)=O)C3)=O)n[nH]2)ccc(SC(C)C)cc1 c1(C(c2nnnn2CC(F)F)NCc2ncn(C(C)C)n2)ccncc1F C(CC)(C(=O)NC(C)CN(C(c1csc(-c2ncccn2)n1)=O)CC)OCC Cc1[nH]nc(C(=O)N(C(C(=O)NCCCCCCO)C2CC2)C)c1Cl N1(C(c2cnc(CC)nc2O)=O)CCC2(CCC2)C(NC(=O)CCS(C)(=O)=O)C1 c1(C(N(CCCCN(C(C(=Cc2ccco2)C)=O)C)C)=O)cc(Cl)c(C)cn1 Cn1nc(NCC2(C)CN(CC3CC3)C2=O)cc1-c1ccc(OC(F)(F)F)cc1 C1(NC(C(CC)N(C(CCC=CCC=C)=O)C)=O)CCCC(CO)C1 CCC(C(=O)N(C(C)CO)CC)NC(=O)COc1ccccc1 CCCCC(CNC(=O)COC1(C)CCC1)NC(C1(CC(C)C)CCC1)=O C1(NC(=O)CCn2ccccc2=O)C2CC(CN(C(c3cocn3)=O)C2)C1CO c1(CC)cc(C(=O)NC(CNC(C2CCSCC2)=O)(CC)CC)nn1C c1(C(=O)NC(CC)CN(C(=O)Cn2cccn2)C)cc(F)c(OC)c(Cl)c1 C1(NC(C2CN(C(C)C)C(=O)C2)=O)CC2CCC1N2C(c1cccc(N)c1F)=O C1(OC)CCCC1C(=O)NCCN(CCCN(C)C)C(C1(CC(F)F)CC1)=O N1(C(Cc2cccc(C)c2)=O)CC(CNC(C2CCC=CCC2)=O)CCC1C n1(CC(=O)NC(CC)CNC(c2snc(Cl)c2Cl)=O)nc(C)c(Cl)c1C C=CC(C)(O)C(=O)NC(C1CCN(C(=O)CC2(c3ccccc3)CCCC2)C1)C n1(CC(=O)NC2(COC)CN(C(C3C(COC)C3)=O)C2)c(C)cc(C)nc1=O C1(CCC(=O)NCC(C)N(C(=O)CSCCOC)CC)CCC(=O)N1 CC1CCCC=C1C(=O)NC1CC2(C1)CC2C(N1CCCC1(C)C)=O Cc1nc(C(C)C)ccc1C(=O)NCc1c(F)cncc1Cl C12(C(=O)NCC(CNC(c3c[nH]cc(C)c3=O)=O)F)CC3CC(C(=O)N1)C2C3 Cc1cn2c(CCC(N3CCN(C(C4CCC4C)=O)CC3C(C)C)=O)csc2n1 c1(C(=O)NCC2N(C(c3ccc(C)nc3)=O)CC(F)C2)cccc2c1OCCN2 C1(NC(C(c2cccc(OC)c2)(C)C)=O)CCN(C(=O)CCCOC)CC1F c1(CC)ccc(C(=O)NCCN(C(=O)CN2CCCC2CO)C)nc1 CC(C)C(O)CC(=O)NCC1(F)CCN(C(=O)CC2CC(C(F)F)C2)CC1 C1(CCNC(C2(CC=C)CC=CC2)=O)CSCCN1C(c1csc(C#N)c1)=O N1(Cc2cccc(OCC(C)N)c2OC)CC(C)OC2(CCOCC2)C1 C(=O)(C(C)(CC)CCC(C)C)NC1CCN(C(C=C(CC)CC)=O)CC1 N1(C(c2c(CC)non2)=O)CC2CCN(C(=O)C=C3CCN(C)C3)C2C1 C12(NC(C(C)NC(CC)=O)=O)CCC(CN(C(=O)C=CC3CCCCC3)C1)C2 C1(NC(C(CCC)C#N)=O)CC(O)(C2CCN(C(C3CC34CC4)=O)CC2)C1 c1(C(N(C)CC2CC(F)CN2C(=O)C(F)CC2CCC2)=O)ccc2cncn2c1 c1(C(=O)OC)nc(NC(C2CCC(NC(=O)C(C)(C)NC(C)=O)C2)=O)sc1C C(CCC(C)C)(C(=O)NC1(CF)CCN(C(C2(C)CCC2)=O)C1)NC(C)=O N1(C(N(CC(C)(F)F)C2CC2)=O)c2ccccc2CC1C(=O)OC(C)(C)C c1(C(C)C)cnn(C)c1C(=O)NC1CC(C)N(C(c2cccc(=O)o2)=O)C1 c1(C(=O)NC(C(=O)OCC)Cc2cccc(C)n2)cnn2ccc(C=O)cc12 C1(NC(CCOCCN(C(C(c2cnn(C)c2)C)=O)C)=O)CC2CCCC2C1 CCC(C)C(=O)C(=O)N1CC2(C(=O)NCC(CO)OC)CC1CO2 C1(N(C)C)(CNC(c2ccc(CC#N)cc2)=O)Cc2ccccc2C1 C(C1C(C)C1(Cl)Cl)=CC(=O)N(CCC#C)C C(=O)(C(C)C(F)(F)F)N1CC(CNC(c2c(C)nsc2C)=O)OCC1 C1(CCC(=O)NC2(CC(C)C)CC2)CCCN(C(=O)C(N2CCNC2=O)C)C1 CC(C)(F)C(C)(F)C(=O)N1CCCC1C(=O)NCC1C=CCOC1 Cc1c(C(=O)NC2CC(NC(c3ccoc3C3CC3)=O)C2)ccc2c1OC(F)(F)O2 n1(CCC)ncc(C(=O)NC2(CNC(=O)CSc3n[nH]c(=N)s3)CCCC2)c1C c1(C(=O)NCC#CCNC(C2CCCC(OC)C2)=O)ccc([N+](=O)[O-])cc1Cl c1(CNC(=NCC)NCc2ccc(Br)c(C)c2O)ccc2c(c1)CNCC2 C1(NC(c2cc(C)nnc2)=O)CC2CC(NC(c3cc(C)c(C)o3)=O)CC2C1 CC1(C)CN(C(=O)CCCN2CCCC2)CCC1NC(=O)C=CC1CC1 C=CC1(CC2C(NC(C)=O)C2)CN(C(c2ccn(CCF)n2)=O)C1 N1(C(C2(COC)CCCO2)=O)CCN(C(c2cncc(COC)c2)=O)CC12CC2 c1(C(C)NC(CN(C(C)C)C)=O)nocc1C(N1CCC(C(F)F)C1)=O C1(NC(C2CCN(C)C2)=O)CC2CN(C(c3cc4ncccn4n3)=O)CC2C1 N1(C(c2cccc(OC)c2O)=O)CCCN(C(c2nnsc2C(F)F)=O)CC1C C(=O)(CCCCC(C)CC)N(C1CCN(C(C2(F)CCCC2)=O)CC1)CC#C C=C1CCN(C(=O)CCC(=O)CC)C(C(=O)NC(c2cccnc2C)C)C1 C1(CCNC(C2C(C=C)C2)=O)CCCN(C(c2cc(C)c(C)s2)=O)CC1 C(CC(COC)N=c1[nH]c2c(c(=NC(C)c3cnn(C(C)C)c3)[nH]1)COC2)OC CC1CN(C(c2ccc(N(C)C)nc2)=O)C(C)CN1C(C1CCC(=O)N1C)=O Cc1cc(C)c(CN(C)C(c2nnsc2C(F)F)=O)cn1 O=C(C1=CC2(CN(C(=O)CC3CSC3)C2)OC1)Nc1ncc2c(n1)CCC2 N1(C(c2c(NC)scn2)=O)CCOC(C(=O)NC2CN(C)CC2C)C1 C1(NC(c2c(C)nn(CC(F)F)c2)=O)CCN(CC2CCOC2)CC1O c1(OCC)ccccc1C(=O)NC(C1CCN(C(c2ccc(Cl)nn2)=O)C1)C CC1(C(=O)NCC2(NC(c3ccc(CC(F)(F)F)cc3)=O)CC2)CC2CCC1C2 N1(C(C(C)c2ccsn2)=O)CC2CN(C(=O)C=CBr)CC2C1 CCCCCCCC(=O)N(C1CC2CC1N(C(c1ccc3nccn3c1)=O)C2)C C1(NC(c2c(C(C)C)nco2)=O)CC2C(NC(=O)C(c3ccccc3)C)C2C1 C(=O)(CC(C(F)(F)F)NC(c1snc(C)c1N)=O)NC(CC=C)CO c1(C(N2C(CN(C(CC(CC)OC)=O)CC)CCC2)=O)ccc(S(N)(=O)=O)cc1 c1(C(CNC(=O)NCCn2c(C)cc(C)n2)=O)ccc2c(c1)ncn2C C1(CNC(C=CSC)=O)CCN(C(=O)COC2CC=CC2)C1(C)C Cc1c(N(C(=O)C(CNC(c2cnc(=N)[nH]c2)=O)C(C)C)C)cccc1F C(CC(F)(F)F)N(C(N1CCC(N2CC(F)C2)C1)=O)CC Cc1ccc(C(=O)NC2CCN(C(C3CCCCC3F)=O)C2)c(F)c1 C1(CNC(c2c(C(C)(C)C)c[nH]n2)c2nnnn2C2CC2)CCS(=O)(=O)C1 C(=O)(C(CNC(C1CC1[N+](=O)[O-])=O)CC1CCCC1)N(CCCCC=C)C N1(C(=O)CC(F)F)CCCOC(CNC(c2cc(N3CCOCC3)ncn2)=O)C1 C1(NC(c2cn(C3CC3)cn2)=O)CCN(C(=O)CCc2cnc(O)[nH]2)CC1F Cc1cc(C(C)N)cc(C)c1.C(=O)(N(CCO)CCOCCNC=O)C1CC1 c1(CC)ccnc(C(=O)NC(Cc2ccco2)C(=O)Nc2cnn(C(F)F)c2)c1 C1(CNC(C=NOC)=O)CC(F)(F)CN1C(C1CCC(C(N)=O)O1)=O S(=O)(=O)(c1ccc(NC(CO)CCC(C)C)cc1Cl)NCCN(C1CC1)CC C1(N(C(CCCN(C)C)=O)C)CCCN(C(C2(F)C3CCCC23)=O)C1 C1(N(C(=O)C(C)(O)C2CCC2)C)CCC(NC(=O)Cc2cncnc2)CC1 Cc1ccc(CN(C(c2cn(CC(F)(F)F)nn2)C(=O)NCC2CC2)C)cc1 c1(C(=O)NCC2CCN(C(C(C(COC)C)C)=O)CC2)c(SC)nc(O)nc1C C1(C(NOCC(=O)N(C)CC2COCCO2)=O)OCCC1(C)C Cc1ncc(S(N)(=O)=O)cc1C(N1CC(NC(=O)COCCCF)C(O)C1)=O C1(CNC(c2cn(CC)nc2)=O)CC2(CCN(c3cc(S(C)(=O)=O)ncn3)C2)CO1 N1(CC)CC(NC(c2nnnn2C2CCC2)(C2COC(=O)C2)C)CC1=O N1(C(c2c(C)noc2)=O)CCN(C(C2C=CCC2)=O)C(c2cc(F)ccc2F)C1 c1(C(=O)NC(CCC)CNC(=O)CNC(N)=O)cnn2cccc2c1 CCC(CC(=O)NCC(CC)NC(c1cnn(C(F)F)c1)=O)OC N1(C(c2cc(CSC(C)C)on2)=O)CC=CC(NC(=O)C(C)(C)SCC)C1 O(N=C1CCCCCC1)CC(N1CC(CNC(CSC)=O)N(C)CC1)=O c1(C(=O)NCC(C)NC(C(c2ccccc2)OC)=O)cnc2c[nH]nc2c1 c1(C(N2C(C(N(C)Cc3cc(C)no3)=O)CC2C)=O)cccc2c1CCC2 C1(C)(C(=O)NC(C(=O)OCC)(C)c2ccccc2)CCCCC1 C1(CNC(C(=O)NC(C)C)=O)CC2CCC1N2C(=O)CNc1ccccn1 C1(C2CCN(C(C3(Cl)CC3(F)F)=O)CC2)(NC(C(CC)OC)=O)CC1 N1(C(C2N(C(C)=O)CCC2)=O)CC2CC(NC(=O)CC3CC4(CCC4)CO3)C1C2 O=C(CS(=O)(=O)CCCc1ccccc1)NC1CCNC12CC2 Cc1cnc(C(=O)N(C(C)(C)CC(N2CCC(C#N)CC2)=O)C)c(F)c1 c1(OC)cccc(C=CC(=O)NC2CCCC2C(=O)N(C)C)c1OC(F)F CC1CC2(CCC2)CN1C(C1CCC(CNC(=O)Cc2ccccc2O)O1)=O N1(C(C2(CC)CCCC2)=O)CC2CCN(C(c3cncc(Br)c3)=O)C2C1 C1(C2CC2)(CNC(CCCCNC(C)=O)=O)CCN(C(=O)Cn2cc(C)cn2)C1 C1(C(=O)N(C(C)CC(C)C)C)(COC)C=CCN1C(C1SCCS1)=O c1(C(N2CCC(NC(COCCSC)=O)C2)=O)cc(C(F)(F)F)ncc1N N1(C(c2c(CC)n(C)nn2)=O)CCOCC(F)(CNC(c2cncc(Cl)c2)=O)C1 C1(NC(=O)C=CC2CC2)CCN(C(=O)C(c2cccc(F)c2Cl)(F)F)C12CC2 c1(NC(CNC(CC(=O)OC)(C)C)=O)ccc(S(=O)(=O)N2CCCCC2)cc1 CC#CCCC(=O)NC1CN(C(=O)C(c2cnccc2C)(C)C)CC1C N1(C(CC)CC)CC(C(=O)NCCCNC(=O)C(C)Cc2ccnn2C)CC1=O c1(C(=O)NC(CNC(C2CN(CCC)C(=O)C2)=O)CC)cc2ccccn2c1 N1(C(CC(CC)O)=O)CC(S(=O)(=O)N2CCN(C(C3CCCN3CC)=O)CC2)C1 N1(C(CC2CCN(C(N(C)C3CC3)=O)C2)=O)CC2CCCC1C2OCCO c1(C(=O)NCC2COCCN(C(C3CCS3(=O)=O)=O)C2)n[nH]c2c1CCOC2 C(=O)(CCCCC(F)(F)F)N(C1CCN(C(C2CCC(C#C)CC2)=O)C1)CCO C1(CNC(=O)Cc2ccsn2)CCCCC1NC(c1ccc(NC=O)cn1)=O C(CCCC(=O)N(C1CCSC1)C)n1cc(-c2onc(C)n2)nn1 C(=O)(C1=COCCO1)N1CC=CC(NC(c2[nH]cc(C(C)(C)C)c2)=O)C1 CC1(C)CC=C(C(=O)NCC2CC(NC(c3csc(Br)c3)=O)C2)CC1 C(=O)(CS(=O)CCC(F)(F)F)NCCN(C(=O)CN1CCCNS1(=O)=O)CC C(CC(C)C(=O)N(CC(O)CNC(=O)CS(=O)(=O)NC)C)=CCC C1(CN(CCOC)C)CCN(N2CCC3(CC2)CNC(=O)N3C(C)C)CC1 N1(C(Cc2ccc(C)o2)=O)CCC2CN(C(C3CCS(=O)(=O)C3)=O)CCC12 c1(C(N2C(CNC(C(c3ccccc3)OCC)=O)CC2)=O)cc(F)n(C)n1 CC(CC(=O)NCC(O)CNC(C1CCCN1C(N)=O)=O)CSc1ccccn1 C1(CNC(C2(CF)CCN(C(c3nc(=N)[nH]cc3)=O)C2)=O)C2CCCCCC12 C(C(=O)N=c1c(Br)c[nH]cc1Br)C1OCCN(C(c2cc(C#N)c(F)cc2)=O)C1 n1(C(C)C)ncc(C(=O)NCC2CC(CNC(=O)CCN3CCCC3=O)C2)c1N c1(CC(=O)NC(CC(C)NC(C(C)NC(=O)NC)=O)C)cccc(C(=O)OC)c1 N1(C(C=CC)=O)CCC(CC(=O)N(C)Cc2ccc(C)cc2)CC1 c1(C(=O)NC(C)C(C)(C)NC(c2cnn(C)c2C#N)=O)cnc2c[nH]nc2c1 N1(C(CC(CC)C(C)(C)C)=O)CC(=O)NCC12CCNC2 N1(C(=O)OC(C)(C)C)CC2CN(C(=O)Cc3cnn(C4CC4)c3)CC2(C(=O)O)C1 c1(C(=O)OC)cc(C)c(NC(c2c(C)nn(-c3cccc(Br)c3)c2Cl)=O)cc1F CCC(CC(F)F)C(=O)NC1CC2CN(C(=O)C(CC)N(CC)CC)CC2C1 c1(C(=O)NC(CC(C)NC(Cc2cn(CC)nc2)=O)C)c(C)nsc1C C1(CNC(CC(C)O)=O)CN(Cc2c(F)cccc2F)CCC1(F)F C1(CC(=O)NC2CC(C#C)C2)(NC(c2c[nH]ccc2=O)=O)CCCCC1 c1(NC(N2CC(c3c(NC(C=NOC)=O)c[nH]n3)OCC2)=O)ccc(O)c(F)c1 N1(C(c2c(CC)onc2C)=O)CCCC2(NC(c3cn(C4CC4)cn3)=O)CC2C1 Cc1ccc(C=CC(N2CCC(C(C)C(=O)NCCc3cnc(C)o3)C2)=O)o1 C=C(CNC(c1nc[nH]c1C(C)(C)C)=O)CCNC(C1(C)CCCO1)=O c1(NC(CC2(C)CN(C(C3CCCC(O)C3)=O)C2)=O)nccc2cccc(F)c12 O=C1Cc2c(C(=O)NCC3(F)CN(C(C4CC5CCC(C4)O5)=O)C3)cccc2N1 C1(C(=O)NC(CN(C(C(C=C)C)=O)C)Cc2ccccc2)Cc2nnc(C)n2C1 c1(C(N2CCCC(NC(=O)C=Cc3cncs3)C2)=O)cccn2nccc12 c1(CC)sc(C(N2CCC(C(C)(C)NC(=O)CC(=O)N(C)C)C2)=O)cc1C c1(CC(CN(C(=O)C(O)C2CC2)C)NC(C2(c3cccs3)CC2)=O)ccccc1 Cc1ccc(CN2CCCC(N(C)C(c3ccccc3Cl)=O)CC2)c([N+](=O)[O-])c1 C1(C(C)NC2(c3nnnn3C)CC3CC3C2)CCC2(CCOCC2)C1 C(=O)(C#CC1(C)CCCO1)N1CC(NC(CCOC(C)=O)=O)C(O)C1 c1(C(N2C(CCNC(C3ON=C(CC)C3)=O)CSCC2)=O)cc2c(s1)CCCC2 C1(C(=O)Nc2cccc(NC(C(C(C)C)F)=O)c2)COc2cc(Cl)ccc2C1 C(=O)(C(O)C1=CCCCC1)NC1C2(CN(C(Cn3nc(C)oc3=O)=O)C2)SCC1 CCCCC(CN1CCCC1c1nnc(NS(=O)(=O)NC)n1CC1CC1)CC N1(C(c2ccn(CC(C)C)n2)=O)CCCN(C(=O)CC2CC3CC3C2)CC1C C(=O)(C(CC(=O)N1CCCN(C(=O)COCCO)CC1C)C(C)=O)OC c1(CNC(C2CC(C)OC2)=O)cc(C(=O)O)ccc1F CC1CN(C(=O)CCCCn2ccnn2)CCC1NC(=O)CC1CCCCC1 c1(C(C)=O)cc(C(=O)N(CCCN(C(=O)CNC(c2cscn2)=O)C)C)oc1C C1(OCC(=O)Nc2ccc(SC(F)(F)F)cc2)CC2CSCC2C1 CC(C)CC(C(=O)NC1CCCCC1NC(=O)CN1CCOCC1=O)C(N)=O c1(C(=O)NC2CN(C(c3c(CC)occ3)=O)CC2C=C)cc2c(=O)[nH]ccn2n1 Cn1ncc(C(=O)OCCSCc2nnnn2C)c1-n1cccc1 c1(C(N2CC(C(N3CC[Si](C)(C)C3)=O)(SC)C2)=O)cnnc(O)c1 c1(NC(C2CC(F)CN2Cc2cc3ncccc3o2)=O)cnccc1[N+](=O)[O-] CC(=O)CCCC(=O)NC(C)C(c1ccccc1)NC(c1ccnc(Cl)c1N)=O CC(=O)CC(C)(C)C(=O)NC1COCCC1C(=O)NC(C)CN(C)C(C)C N1(C(c2nc(C)sc2)=O)Cc2ccccc2CC1CNC(=O)Cc1ccns1 C1(C(N2CC(CNC(=O)C=Cc3cncs3)C2)=O)CC2CCCCC2O1 c1(C(=O)NCC(CO)NC(c2ccc([N+](=O)[O-])o2)=O)cn2c(n1)CCC2 c1(OC)ccc(C(=O)N(C)Cc2ncc[nH]2)nc1Cl c1(CC)[nH]nc(C(=O)NCCC2(O)CN(C(=O)C(=Cc3cccs3)C)C2)c1C C1(NC(c2n(C)ncc2C2CCC2)=O)CC2CN(c3ncc(F)cn3)CC2C1 c1(N(C(C(C)S)=O)C)ccc(-c2cccc(CN(CCC)C)c2)cc1.NC c1(OCC)ccc(C(=O)NCC2(O)CCN(C(=O)C(c3ccccc3)O)C2)cn1 CC(C)(CNC(C1COCOC1)=O)C(=O)NCC12CC(CCO1)C2 C12(NC(C3CCN(C)C(=O)C3)=O)CCCC1CN(C(c1ccsn1)=O)C2 N1(C(C2ON=C(C)C2C)=O)CCC(CCNC(C2(N(C)C)CC2)=O)C(F)(F)CC1 Cc1cc(F)c(C(=O)NC2CC23CC(NC(c2c(C)nn(C)c2F)=O)C3)cc1F C1(CNC(N(C(c2nc[nH]n2)(C)C)C)=O)(NC(=O)OC(C)(C)C)CCC1 CCCCC(CC)CC(=O)N1CCC1CNC(c1cc(F)cc(F)c1F)=O C1(NC(CC(c2scc(C)c2)O)=O)CCC2(CC1)CN(C(c1cocn1)=O)C2 CCC(C(=O)NC1(CNC(c2ccc(CS(C)(=O)=O)cc2)=O)CC1)C(C)C N1(CC(N2CCC(N(C(C3CCS3(=O)=O)=O)CC)C2)=O)CC(=O)NC1=O C(=O)(C1CCCn2nccc21)NC1C(NC(CCCN(C)C)=O)CCC1 CC1(C)CN(C2CCN(CC(F)(F)F)C2=O)c2ccc(C(=O)O)cc21 c1(C(=O)NCC2(F)CC(NC(=O)CCc3ccccc3O)C2)ccccc1O C1(CNC(C2C(CN(C)C)C2)=O)N(C(C2(C(N)=O)CC2)=O)CCC1(C)C C(c1ccncn1)=CC(=O)NC(C1CCN(C(c2ccnn2CCF)=O)CC1)C N1(C(C(c2scc(C)n2)C)=O)CCC(NC(=O)C(C)(C)F)C(O)C1 c1(OC)nc(NCCNC2CCCCC2)ncc1C.C1(C(C=O)OC)CCCCO1 CC1(F)CCN(c2nnc(-c3ccc(Br)s3)n2CCc2sccc2OC(F)F)C1 C1(CC#C)CN(Cc2cc(C)n(C)n2)C12CCC2 CC1(C)CCCCC1CC(N1CCC(NC(=O)C2=CCC2)C12CC2)=O C1(O)(C(C)NC(C2(CN(C)C)CC2)=O)CCN(C(=O)C(F)(F)C(C)O)CC1 c1(NC(CCCC#CC)=O)c2c(nn1-c1cccc(Cl)c1)CCC2 Cc1c(Br)noc1C(=O)NC1CCCCC1NC(=O)COC(F)F Cc1sc(C(=O)NCC2(C(C)(C)C)CCN(C(C3(O)CCC3)=O)C2)c(C)c1C CCC(C)(CC)C(c1nnnn1CC1CC1)NC1(CCC(=O)OC)CCOC1 C(C(C(F)(F)F)N1CCN(C(c2cnc(Cl)s2)=O)CC1)NC(C1CC=CCC1)=O N1(C(c2c(C)cc(F)s2)=O)CCCCC1C1CCCN1C(c1cc[nH]c(=N)c1)=O CC1(C)CN(C(c2n[nH]cc2Cl)=O)CCC1C(=O)NCC1CCC(F)(F)C1 N1(C(CN(C)Cc2ccc(F)cc2)=O)CC(NC(c2ccoc2)=O)C2(CCC2)C1 c1(CC(=O)NCC(C(C)C)N(C)C)ccc(Cl)cc1Br CCCC(C)(O)CC(=O)N1CCN(C(=O)CN2C(=O)CCC2=O)C(C(C)(C)C)C1 Cc1c(C(=O)NC(C)CNC(=O)CCc2ccoc2)[nH]c2c(Cl)cccc12 Cn1cnc(N(CCNC(c2c(C(F)(F)F)cnn2C)=O)CC2CC2)c(Br)c1=O N1(CC)CCCC(N2CCCC2)C1.C1(C)CCNC(=O)N1 C1(N(CC(=O)OC)C)CC12CCN(S(=O)(=O)c1ncc[nH]1)CC2 N1(C(CC)=O)CCC(C(=O)NC(C)CCN(C(=O)COc2ccccc2)C)C1 C(=O)(CC(C)(C(F)(F)F)N(C)C)NC(CNC(C=C(CC)C)=O)(C)C1CC1 C(=O)(CC(C)(C)F)NCC(C)NC(c1c(SC)csc1)=O N1(Cc2ccn(C)n2)CCC(C)(CNC(=O)C(O)c2ccco2)CC1 C(=O)(C(Cc1ccco1)NC(=O)CC1CCC(=O)C1)N(CC(C)SC)C N1(C(c2ccc(C)o2)C(=O)NCCn2cncn2)CCN(CCCO)CC1 c1(C(=O)OC)cncn1CC(=O)NCCN(C)C(C1CNC(=O)N1)=O c1(OC)ccc(F)c(-c2cn(CC3CCN(C(=O)CCC(C)O)C3)nn2)n1 C1(CC)CN(C(=O)C(C)(C)CNC(=O)CCCC2CCC2)C(C)CO1 c1(N(C)Cc2ccco2)nc(NCCCF)c2ncn(C)c2n1 C1(C(=O)NCc2cc(OC)no2)CCC(C)(C)N(C(=O)C(C2CCCCC2)=O)C1 Cc1cc(Cl)cc(C)c1C(=O)NC(CNC(=O)Cc1csc(S)n1)C1CC1 CCCCC(O)CC(=O)NC(C1CCCN1C(c1cc(C)c(Cl)s1)=O)C c1(C(=O)OC)c(C(N2CC(NC(c3c[nH]nc3OCC(F)F)=O)C2)=O)n[nH]c1C Cc1ccc(C(=O)NC(CC2CCC2)C(=O)N2CCC2(CO)CO)c(F)c1 C=CCN=c1[nH]cc(C(N2CC(NC(c3c(OC)ncnc3OC)=O)C2)=O)s1 N1(C(c2[nH]c(=N)sc2)=O)CCC(NC(C2CCCNS2(=O)=O)=O)C12CCCC2 N1(C(CC2(OC)CCC2)=O)CCOCC(CNC(c2ccc(C(C)C)nc2)=O)C1 c1(NC(C2CC(NC(C3CC3(F)F)=O)C2)=O)c(Cl)cc(Br)cc1[N+](=O)[O-] c1(C(=O)NCc2c(C(=O)NC(c3onc(C)n3)C)c[nH]n2)n[nH]c(C)c1Cl c1(OCC)nccc(C)c1C(=O)N(CCCNC(C1CCC(C)S1)=O)C N1(C(C(CC)C)=O)CC(C)(C)C(NC(=O)CC2CCCN(C)C2)C(C)(C)C1 CC1CCN(c2ccc(CNC(=O)CC(C)(C)C3CC3)cn2)CC1 n1(CC)cnc2nc(=NCc3cc(Cl)sc3Cl)[nH]c(NCC3CN(C)CCO3)c12 C1(C)(C(N2C(C)CC(CNC(c3cc(C)n(C(C)C)n3)=O)C2)=O)CCN(C)C1=O c1(SCC(=O)NC2C=CCN(C(CN3CCN(C)CC3)=O)C2)cc(F)ccc1F C1(CNC(c2c(C(C)C)ccs2)=O)CCN(C(c2ccoc2Cl)=O)CCC1(F)F N1(C(CC=CCC)=O)CCC(C(=O)NCC(CC)CCO)C(C)C1 c1(NCC(n2cccn2)C)ccc(S(=O)(=O)NC(C)CS(C)(=O)=O)cc1Br S(=O)(=O)(c1ccc(N2CCC(OCCO)C2)cc1Br)N1C(CCC)COCC1 c1(OC)cc(C(N2CC(O)CC2C(=O)Nc2ccc(SC)nc2)=O)cc(F)c1 C1(C(N2CC3OCCC23)=O)CCCN(Cc2cccnc2)CC1 c1(SC(C)C(=O)Nc2ccc(Cl)cc2)ccc(N=NC2CC2)cc1 C1(CC(=O)CN2CCC(NC(C3CCC(SCC)CC3)=O)C2)CCC(C)(C)CO1 S(=O)(=O)(c1ccc(=NCC(O)CF)[nH]c1)N1CCCC(OC)(CO)C1 S(=O)(=O)(c1ccccc1C1CC1)NCCCCCC(=O)OC C1(C2CC2)(CNC(c2c(C)cccn2)=O)CCN(C(=O)C2=CCCC2)C1 c1(CNC(C(SC)SC)=O)cc(C(=O)NCC2CC2(Cl)Cl)n[nH]1 C(C(=O)NCCNC(=O)CC1(C(F)(F)F)CCC(=O)NC1)(C(C)(C)C)OC C1(NC(C(CSC)(C)NC(C2CC3(CC(=O)C3)C2)=O)=O)CCOC12CCOC2 S(=O)(=O)(c1ccc(F)c(C(=O)NC(C)CNC(=O)C(F)n2cccn2)c1)NCC N1(C(COC(CC)(C)C)=O)CC2CCC1C(C(=O)NCC1CCCCN1C)C2 C(=O)(NNC(=O)C1CCOC1C(C)(C)C)NC1C(c2cn(C)nc2)C1 c1(C(=O)NCC2C3CN(C(C4(F)C(C)OCC4)=O)CC32)cccc2cc[nH]c12 N1(C(CC2C(C)(C)C(NC(=O)CSc3cn[nH]c3)C2)=O)CCCC2(C1)N=N2 Cc1nn(CC(=O)NC(c2cn(Cc3ccno3)nn2)C)c(C)c1[N+](=O)[O-] C(C(F)(C(=O)NCCC1C=CCC1)C(C)C)NC(C1(C#C)CCCCC1)=O c1(N(C)C)ccc(NC(=O)CC2C=CC(NC(=O)CC3CSCCO3)C2)cc1 C#CCCCC(=O)NC1CCC(NC(=O)C(C(C)C)n2cc(Br)cn2)C1 Cc1ccsc1C(C(=O)NCCCC1CC1)N(CC(F)Br)C C#CC(CC(C)(C)C)NC(C1CCN(C(=O)C2(SC)CC(=O)C2)O1)=O c1(C(=O)NCC(C)NC(=O)C2=CCOC2)ccccc1S(=O)(=O)N1CCOCC1 Cc1ccc(Cl)cc1C(N1CCC2(CC2C(=O)NCc2ccsc2)C1)=O c1(C(N2CCCC(CCNC(=O)CC3(CO)CC3)C2)=O)cn2ccc(F)cc2n1 C(=O)(C1=CCCC1C)N1CCC(NC(C=CC=CC)=O)(CO)C1 S(=O)(=O)(c1ccccc1)NCC(=O)N(C)CC1(NC(c2cc(Cl)cnn2)=O)CC1 c1(CN2CC(CNC(c3ccnnc3O)=O)C2)c[nH]c2cc(Cl)ccc12 CCCCC(C)C(C(=O)NCC(c1ccccc1)OC)N1CCC(O)CC1 C(=O)(CC1=CCOCC1)NCCOCCCNC(C(CCCC)ON=C(C)C)=O N1(C(C=Cc2c(C)nsc2)=O)CCCCC(N(C(=O)C(O)Cn2cncn2)C)C1 C1(NC(C2CCC(=C)CC2)=O)CC2CC(C1)N(C(c1cc(O)nn1C)=O)C2 c1(C(=O)NC2CN(C(CCc3ccc(C)o3)=O)CC2(C)C)ccc2ncnn2c1 C1(NC(c2cc(Br)n[nH]2)=O)(CF)CCN(C(C2CCN(CC(F)(F)F)C2)=O)C1 N1(C(C=NOC)=O)CCCCC1C1CCCN(C(c2nccnc2C(N)=O)=O)C1 c1(CCC)onc(C)c1C(N1CC(C(N)=O)(CNC(=O)CC(C)NC(N)=O)C1)=O c1(C(N2CCCC(NC(=O)CCF)C2)=O)cncc(Br)c1Cl N1(C(C(CCC)N(C)C)=O)CCN(C(C2OCCCO2)=O)C2COCC12 c1(CC(N2CCCN(C(C(CC)n3cccn3)=O)CC2)=O)ccc(F)cc1Cl C(=O)(CC(=O)NCC1CC(NC(c2ccc(NC(=O)C3CC3)s2)=O)C1)OC N1(C(C2C=CCN(C(=O)CCn3cccn3)C2)=O)CCCC(C2CCC2)C1 N1(C(CCC(N)=O)=O)CCC(F)(F)C(NCc2c(O)cc(O)cc2O)C1 c1(C(=O)NCC(CC=C)NC(=O)CN2CCOCC2)cncc(OC)n1 CCC(C)(C)C(=O)N1CC(CCNC(C2CC(SC)C2)=O)C(C)C1 O=C(C1CCOc2ccc(Cl)cc21)N1CC2(CO)CC(C(=O)O)(C1)C2 CC1CN(C(=O)CC(C)(F)F)CC2(CCN(CC(O)COc3ccccc3)C2)O1 Cc1cc(C(N2CC(NC(C3(C(C)C)CC3)=O)C3CC23)=O)sc1C c1(C(=O)NCC=CCNC(C(C)Oc2ccc(C)cc2)=O)cc(C#N)[nH]c1C CC1(C)CNC(=O)C1NC(=O)Nc1cccc(OCCC(C)(C)O)n1 CCCC(C(=O)N1CCC(c2nc[nH]n2)C1)NC(C1CCC(CC)O1)=O C1(C(=O)NCC(C)NC(c2nn(CC)nc2C)=O)CC2CC1C1CC21 C(CCCO)(c1ccccc1)NC(=O)NCC(COC)O C1(NC(C2(C)CC(=C)C2)=O)CCC(CNC(C2CC2C(=O)OC)=O)CC1 S(=O)(=O)(c1cccc(Cl)c1C#N)Nc1n(C)nc(-c2ccccn2)c1 C1(C(N(CCCCC)CCO)=O)CCC(C)(C)N(C(=O)CC2C(=O)NN=C2C)C1 c1(C(N2CCOCC(F)(CNC(C(=O)N(C)C)=O)C2)=O)cc2ccc(O)cc2[nH]1 C(C)(C(C)C(=O)OC)NC(C(COC)NC(=O)C=CC(F)(F)F)=O N1(C(c2ccc(N)c(F)n2)=O)CC2CC1CCC2NC(C1CCCC1O)=O CC1CCN(C(c2ccc(Cl)c(F)c2)=O)CC1NC(=O)CN1CCCNC1=O Cc1ccc(SCC(=O)NCCCN(CCO)C(C2CCC(OC(C)C)C2)=O)cc1 C1(NC(C(C=C)O)=O)(CF)CCN(C(c2ocnc2C2CCC2)=O)C1 C1(c2nnnn2C)(NC(CCCN(C)C)=O)CCCOCC1 c1(OCCC)cccc(C(=O)N(C)CC2CN(C(c3ocnc3C3CC3)=O)C2)c1 c1(C(N(CC(C)NC(c2ncn(CC)n2)=O)CC)=O)ccc2c(c1C)CCC2 N1(C(C(CC)N(C)C)=O)C2CCCC1CC(NC(=O)CCC(C)O)C2 C1(NC(=O)NCCOCCC#C)CCOC(C(C)C)C1 C1(CN(C(C(C)Cn2cccn2)=O)C)COCCN1C(=O)CS(=O)(=O)N(C)C C1(C(N(C)CCNC(=O)C#CC(=O)NC2CCCC2)=O)CCc2nnc(O)n2C1 S(=O)(=O)(c1cc(Cl)ccc1Cl)Nc1c(C(=O)Nc2nc(SC)nc(O)c2)scc1 c1(C(=O)NCC2C(CNC(c3cc(OC)nn3C)=O)C2)cc2c(ccn2C)s1 N1(C(C2C(C3CN(C(C4(C)CCNC4=O)=O)C3)C2)=O)CC(O)C2(CCCC2)C1 CCCCC(F)C(=O)N1CCCCC(CCC(=O)NC2(C)CC3(CC3)C2)C1 CC(C)(CC(F)F)C(=O)NCC1CC2COCC2N1c1ccc(Cl)cc1[N+](=O)[O-] c1(C(N2CCC(CC=C)(NC(c3cc(=O)n(C)o3)=O)C2)=O)cc(C)ccc1F CC(C)(C(=O)N1CC(=C(F)CNC(=O)CN2CCNC2=O)C1)c1cncnc1 C1(CNC(C2CC23CCOCC3)=O)CCN(C(C2(CCF)CC2)=O)CCC1(F)F C1(CNC(C2CCCS2)=O)CN(C(=O)CCC2CCCCO2)CCO1 C1(C)(C(=O)NCCCCN(C(CCc2cnc(C)o2)=O)C)CCCCCCC1 N1(C(CCCCOC)=O)CCN(C(=O)C(c2cc(F)cc(F)c2)C)CC(O)C1 c1(C(=O)NC2CN(C(Cc3cnc(C)s3)=O)C(C)CC2)cnc2c(Cl)cccn12 N1(C(CCc2ccnc(C)n2)=O)CC2=C(C1)CN(C(=O)C=Cc1ccn(C)c1)C2 C12(C(N(c3c(C)ccs3)CCC(C)CO)=O)CCC(CSc3ccccc3)(CC1)CC2 N(C(=NCCCP(C)(C)=O)NCc1ccc(OC)c(C)c1)C1N(CCC)CCC1 C1(CN(C(=O)C(F)=CCCF)C)CCN(C(=O)CC2CNC(=O)C2)CC1 N1(C(C(CCCC#C)C)=O)CCC2(CCN(C(=O)CCOC3CCC3)C2)C1 N1(C(C)C)CCCCC1C(N1CCC(C)(NC(c2cnsc2)=O)C1)=O CN1C(=O)CCCC1C(N1CCC(O)C1C(=O)NC1CC(Cl)(Cl)C1)=O CCCCCCCCNC(=O)C(=O)NC1CN(C(=O)N=CC(C)(C)SC)CC1C N1(C(CC(C)n2cccn2)=O)CCC2(C(=O)NCC3CC4(CCC4)C3)CCCC12 N1(C(C=NOC)=O)CCCC12CCN(C(c1noc3c1CN(C(C)C)CC3)=O)C2 c1(C(=O)NCCC2(O)CN(C(c3cc[nH]c3)=O)C2)ccc(-c2cscn2)cc1 CCCCC(O)C(=O)N(C1CN(C(C2CC2c2ccccc2N(C)C)=O)C1)C C1(NC(C2CC3(CCC3O)C2)=O)CC2(CCC(COCc3ccccc3)CC2)C1 N1(C(CSC(C)C)=O)CCN(C(=O)CCc2cccc(F)c2)C(CC(F)(F)F)C1 CCC(CC(=O)N1CCN(C(=O)CCCOC)CC1CC)CC(F)(F)F C(=O)(N=c1nc[nH]s1)C1N(C(C(Cc2ccccc2)NC(=O)OC)=O)CC1 c1(C(=O)NC23CCCC2CN(C(c2coc(O)n2)=O)C3)oc2ccccc2c1Cl C1(NC(C(=Cc2ccccc2)C)=O)CCCCN(C(=O)CCOC2CC2)C1 CCC(C)C(O)C(C)C(=O)NC1CN(C(C2(C)CCC(=O)C2)=O)CC1O C1(NC(C=C(CC)C)=O)CC(C2CCN(C(=O)CCN3CCCC3=O)C2)C1 N1(C(C(C)S(C)(=O)=O)=O)CC2(CCN(C(c3ccc(C4CC4)o3)=O)CC2)C1 C(CCCN=c1[nH]c2c(c(=NC(C)CN3CCCC3)[nH]1)CCC2)=CC c1(C(=O)NCC(C)NC(=O)CCc2ccncc2)nn(C)cc1[N+](=O)[O-] C1(C(C)(C)NC(c2ncn(C)n2)=O)CCN(C(=O)CCC2(C)CCC(=O)N2)CC1 N1(C(C(C)(C)N2CCOCC2)=O)CCC(O)(CNC(=O)C2=CCOC2)C1 CC1(NC(=O)COC2CC2)CCCCC1C(=O)NCC1(F)CCC1 c1(C(=O)Nc2ncccc2Br)cc2ccc(-c3cc(C4CC4)cnc3F)cn2c1 N1(C(C(C)=C(C)C)=O)CC(F)(F)CC1CNC(c1n[nH]cc1C(F)(F)F)=O C1(CC)C(C(=O)NC(c2cscn2)CO)CCCN1C(=O)Cc1ccc(F)nc1 C#CCCC(O)C(=O)N1CC2(C1)CN(C(C1CCN(C)C1=O)=O)C2 N1(C(c2c(C)snc2)=O)CC(CO)C2(C1)CN(C(c1ccc(N)c(F)n1)=O)C2 C1(C(N(C)Cc2ncnn2C)=O)CCC2CCC1N2C(C1C2CCCC12)=O C1(CNC(c2c(C)nc(C)s2)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1C C1(NC(c2c(C)nccn2)=O)CC2(NC(=O)Cc3cnsc3)COC1C2 N1(C(C2N(C(C(C)OC(C)=O)=O)CC=CC2)=O)C2CCC1CC1(CC1)C2 CCC(CC(F)F)C(=O)N1CC2(CCN(C(=O)C(C)Cc3c(C)n[nH]c3C)C2)C1 N(C1CCCc2ccoc21)C(C(C(C)NC(=O)CCC1(C)N=N1)(C)C)=O N1(C(C2(COC)C=CCC2)=O)CC2CCCC(C1)N2C(c1ccsc1Cl)=O C(=O)(C1CCCc2nn[nH]c21)NCCCN(CC)Cc1ccc(F)cc1 N1(C(C(CCO)N(C)C)=O)CC(CNC(c2coc(C(N)=O)c2)=O)CC12CCC2 C12(CNC(C(=O)NCC(=O)N(c3ccncc3)C)=O)CCC(CC1)CC2 c1(CCC(=O)NC2CC(C)(NC(CN3CCC(C)(C)C3)=O)C2)ccc(F)cc1Cl c1(CC(=O)NC2C(NC(CC(C=C)C)=O)CCC2)cccc(S(=O)(=O)CC)c1 N1(C(C(C)CC2CC2)=O)CCC2(CC1)CC(NC(c1cc(Br)cn1C)=O)C2 N1(C(C(C(C)OC)NC(C(CCC)CC)=O)=O)CCN2C(=O)OCC2C1 c1(OC)cc(C(CC(=O)O)NC(C2(c3cc(O)cc(Br)c3)CC2)=O)c(Br)cn1 c1(C(=O)NC2C(N(C(c3c(C)n(C)nc3)=O)C)CCCC2)c(C#N)cnn1C CC(C)CCCN=c1[nH]c(N(C)CCOCc2ccccc2)nc2c1COCC2 C1(N(C(CS(=O)(=O)NCC)=O)C)CCCN(C(=O)CCc2c(C)noc2Cl)CC1 C1(c2onc(COC(C)C)n2)CCCCN1C(=O)N(C(C)C(F)F)C c1(C(=O)NCC2(F)CN(C(C3CN(CC)C(=O)C3)=O)C2)cnc(C2CC2)nc1C Cc1cc(C(N2CCC3C(NC(=O)CCc4ccc(Cl)cc4)CC23)=O)cc(O)n1 C1(F)(CNCCc2nccc(C)n2)CCC2(CC1)CC2 C1(CNC(C2(C)CCCC2O)=O)CC2(CC(NC(c3n[nH]c4c3COC4)=O)C2)C1 C12(NC(C(C)C)CNCc3ccccc3)CC(c3ccccc3)(C1)C2F C1(C(=O)NCC2N(C(CCN(CCC)C)=O)CC(F)(F)C2)CN2CCC1(C)CC2 Cc1ccc(C(C)C(=O)NCC=CCNC(=O)COC2CCOCC2)s1 C1(CNC(N(CC(CC)(C)OC)C)=O)CNCC(OC)C1 C(=O)(CCCCCCCC1CC1)N1C(CNC(CN(C(C)=O)C)=O)CC1 c1(C(N2CC(CC(C)NC(C3CC3c3cnc[nH]3)=O)C2)=O)cnc2[nH]ncc2c1 CC(CNC(C1CCCCS1)=O)C(=O)N(C1(CO)CC1)C C1(C(=O)NCc2nc(C)c(C)[nH]2)CC2(CCC2)CN1C(=O)CC1CCC=CCC1 N1(C(C2CN(C)C2)=O)CCN(C(C2CCCN2C=O)=O)C2(CCC2)C1 CC(COC1CCCC1)N=c1cccc(S(=O)(=O)NCc2nccc(=N)[nH]2)[nH]1 CP(C)(=O)C(CC(=O)N1CC2C(NC(=O)Cc3ccccc3O)C2C1)P(C)(C)=O C12(CNC(c3nc[nH]n3)=O)CC(CO1)N(C(C1CC(C(F)(F)F)C1)=O)C2 c1(C(N2CCOCC(F)(CNC(CC(C=C)C)=O)C2)=O)cnn2c(N)ccnc12 C1(NC(c2c(C#C)c[nH]n2)=O)CCCN(C(c2coc(Br)n2)=O)C1C N1(Cc2cccc(C(C)C)c2)CC2(CCC(C(=O)Nc3ccc(Br)c(I)c3)O2)C1 N1(C(C(CCO)NC(COCCCN=[N+]=[N-])=O)=O)C2CCC1COC2.C(CO)N CC1(C)CCC(NC2COCCC2CCC#N)(NC(=O)OC(C)(C)C)C1 N1(C(C2C(OC)CN(C(c3nn(CC)nc3C)=O)C2)=O)CCC(N=[N+]=[N-])C1 c1(CC(=O)NC(CC(C)NC(c2c(C)occ2)=O)C)ccccc1Cl C(C(C(=O)NOCC(=O)Nc1ccc([N+](=O)[O-])cc1)C(C)C)NC(C)=O C1(c2c(C)n(C)nc2)C(NC(N2CCOCC2CNC(N)=O)=O)CCC(=O)N1C n1(CC)nc(C(N2CCCC2(C(=O)N(C)Cc2cnn(C)c2)CC)=O)cc1C c1(OC)cc(C(=O)NC2CCC2C(N2CCCC2Cn2ccnn2)=O)ccn1 C1(OC)CN(C)C(C)(C(N2CCC(F)(CNC(=O)Cc3ccc(C)s3)CC2)=O)C1 n1(CC)ncc(C(=O)NCc2cn(CC(C)NC(C3CN(C(C)=O)C3)=O)nn2)n1 c1(C(=O)NCCC(C)NC(=O)C(C)CO)cnn2c1C(=O)NCC2 C1(C(N2CCCCC(NC(c3cnc(C)nc3C)=O)C2)=O)C2(CCC2)C12CCC2 C1(C(C)NC(c2ccn(C(F)F)n2)=O)CCCN(C(c2cccc(=O)o2)=O)C1 C1(C(=O)NCCOCCCNC(C(C)O)=O)COC2(CCC2)C1 c1(C(=O)NC(C(=O)N(C)CC)(C)C)ccn2ccccc12 Cc1nnccc1C(=O)NCC1CCC(NC(C2CCCCC2O)=O)CC1 c1(C(N2CCN(C(CNC(=O)C#CC3CCC3)=O)CC2)=O)cc(F)c(F)c(F)c1 CC1=CCC(C(=O)NCc2nocc2C(=O)NC2CCC(F)CC2)CC1 C(=O)(C#CC1CCCCC1)N1CCC(C(N(CC(F)(F)F)CC)=O)CC1 c1(C(C(=O)N(CC(C)OC(F)F)CC(C)C)NC(COC)=O)cnn(C)c1 N1(C(CSC)=O)CCC(CCN(C(=O)C(CCSC)N(C)C)C)CC1 c1(C(N2C(CNC(CN(CCCCCC)C)=O)CC2)=O)cccc(N)c1 CC(C)(C)C#CC(=O)N1CCC(OCCCNC(c2cnc(F)c(F)c2)=O)CC1 c1(C(=O)NCC2CC(NC(c3cc4n(n3)CCC4)=O)C2)ccc([N+](=O)[O-])s1 c1(C(N2C(C3CCN(C(Cc4cnc(C)[nH]4)=O)C3)CCC2)=O)ccc(C)c(C)n1 N1(C(C(CCC)O)=O)C2CCC1CC(CNC(=O)C(C)(C1CC1)NC(C)=O)C2 c1(C(=O)NCc2cnn(C)c2C(N2CCC3C(O)CC23)=O)occ2c1CCC2 N1(C(C=C(CC)CC)=O)CCC(CNC(c2cnn3c2CCC3)=O)C(F)(F)CC1 C1(NC(c2ccc3c(c2)COC3)=O)CC2CN(C(C3(CCF)CCC3)=O)CC2C1 C(=O)(C(C)S(N)(=O)=O)NC1CCC(NC(C2C(OC)(OC)CC2)=O)CC1 C1(C(N(CCC(=O)N(CC)Cc2ccoc2)C)=O)CCCCC1 C(=O)(C1=C(Cl)CC1)N(C(C)CNC(c1cc(-c2ccccc2O)[nH]n1)=O)C N1(CCNC(C2(C(=O)OC)CC2)=O)CCCC(NC(=O)C(C)CSC(F)(F)F)C1 c1(C(N2CC3C(NC(C4CCCN4C4CCCC4)=O)(C3)C2)=O)cc(O)ccc1O N1(CC)CCCCC1C(N1CC(n2cc(CCSC)nn2)C(O)C1)=O c1(C(N2C3C(NC(C4CSCCS4)=O)CC(C3)C2)=O)cccc2c1CCCC2 c1(-c2scc(C(C(=O)NC3(C)CC3)N(C3CCCC3)C)n2)cccc(Br)c1 S(=O)(=O)(CCC(=O)N1CC(CNC(=O)C=Cc2cncn2C)CC1(C)C)NC C(=O)(CC(C)(C)C#N)N(C)CC1CC(F)CN1C(=O)CC1COC2CC1C2 c1(NC(C(C)(C)C(=O)OC)c2n(CCCC)nnn2)ccc2c(c1)C(O)CCC2 c1(C(N2CC(NC(C34CC(C(=O)OC)(C3)C4)=O)C2)=O)ccc(N(C)C)c(F)c1 C1(NC(C(CC)N(C)C)=O)CN(C(=O)Cn2cnc3c2CCCC3)CC2(CC2)C1 Cc1nccc(C(=O)NCc2ccccc2CN(C)C(C2CC23CC(O)C3)=O)n1 C1(NC(C2(CC#C)CCCCO2)=O)CC2CCC1N2C(c1cc(F)cnc1O)=O c1(C(=O)NC2C(OC)CN(C(=O)CC3(C)CC3)C2)cnc(N)c(CO)c1 CCC(CC(=O)N1CCCC1(C(N1CCCC1CN(C)C)=O)CO)C1CCC1 c1(OC)ccnc(C(=O)NC(CNC(=O)CC(C)(C)OC)C2CCC2)c1C c1(C(=O)OC)cn(C)cc1C(N1CC2(CC2C(=O)OC)C1)=O c1(OC)cc(C(=O)NCC2=NOC3CN(C(=O)CSC)CC23)ccc1[N+](=O)[O-] C(=O)(CC(C(F)(F)F)N(C1CCC1)C)N(C)CC1(SC)CCC1.C1(=O)CN1 N1(C(CC2CC(=C)C2)=O)CC(CNC(C2(CC)CCNC2=O)=O)C(C)C1 N12CC3(CCC(CC3)NC(=O)c3cc(n[nH]3)C1=O)C2.c1(COC)ccc(F)cc1 C12(CC(=O)N(C3CCCN(C(C4C5C6CCC(C6)C45)=O)C3)C)CNC(=O)C(C1)C2 N1(C(CC(C)C(F)(F)F)=O)CCc2sc(CNC(c3ccncc3)=O)nc2C1 c1(NC(CC2(C)CN(c3ncccn3)C2)=O)ccccc1N1CCCC1 N1(C(c2cncc(Cl)c2)C(=O)NC2CC(F)(F)C2)CCOCC2(CCC2)C1 N1(C(c2c(CC)non2)=O)CC(C(=O)NCCC#CCO)CC12CCC2 c1(COC)cc(C(=O)NC2CC(C(=O)N(C3CC4CC4C3)C(C)C)C2)n[nH]1 c1(C(N2CCC(C(C)NC(c3cc(Cl)on3)=O)C2)=O)cc[nH]c(=N)c1[N+](=O)[O-] C1(CC#C)CCCN(C(C2CC=CCC2C)C(=O)NCCC(=O)OCC)CC1 c1(C(=O)OC)ccc(-c2nc(C)cs2)cc1NC(=O)NCc1cnc(Cl)cn1 CCCC(C)(C)CC(=O)NC1CCC(CNC(=O)C=CSc2ccccc2)CC1 Cc1nc(C)n(CCCCC(=O)NC(C)C(C)(C)N2CCCC2)n1 N(C1CCOc2c(Br)cccc21)C(C1CC2(CCCC2)CO1)=O C1(C)(c2cn(CCNC(C(C)C)=O)nn2)CCCN1C(C1COC(C)(C)C1)=O c1(C(NOCC(=O)NC(Cn2ncc(C)c2)C)=O)ccc(C#N)cc1 C12(CCNC(c3cc(C(=O)OC)on3)=O)CCC1CN(C(c1ccco1)=O)C2 C12(CNC(C(C(CC)C)O)=O)CCC(CC1)N(C(c1cn3ccnc3s1)=O)C2 O=C(C1OCCc2ccccc21)N1CCC(C2CCCN2CC2CCCC2)CC1 C=CC(CC)CC(=O)N1CC(C(C(N2CC(F)CC(F)C2)=O)OC)C1 c1(OC)nc(N2CC=C(CCNC(C3(C(C)C)CC3)=O)CC2)nc(C)c1F C(C(CNC(c1coc(Br)n1)=O)CO)NC(c1cnn(C2CC2)c1)=O N1(C(c2c(C)cn(CC)n2)C(=O)NCc2ccc(F)cc2)CCC2(CCCO2)C1 C(=O)(C1CCc2cc(Br)ccc21)N1CCC(NC(C2(CC=C)CC2)=O)C1C C1(OCC#C)CCCCN1C(=O)C(N1CCC(N(C)CCOCCOC)C1)=O CC1(C)CCC1CC(=O)OCC1CCCC1CCc1ccccc1 C12(NC(c3cc(C)nn3C)=O)CCCC1N(C(c1cnn[nH]1)=O)CCC2 c1(C(=O)NC(C(=O)NC(CCOC)C)C2(C)CC2)ccc(C#N)c(C)n1 C(CO)(CCC(=O)NCCN1CCCOC1=O)NC(=O)OC(C)(C)C C1(C(=O)OC)N(C(=O)CCCc2csc(=N)[nH]2)CC12CCOCC2 C1(CC)CN(C(C2(C)CCCC2C)=O)CCC1NC(C1(C#N)CC2CC2C1)=O Cc1cc(C(=O)N(C2CN(C(=O)C(C)C3CCCC3)C2)C)cc(C)n1 N1(CCNC(c2n(CC)nnc2)=O)CCCN(C(=O)Cc2ccc(O)nc2)CC1 C1(CNC(C2=C(C)CCC2)=O)CC2(CO1)CN(C(C1COCCN1C)=O)C2 c1(C(=O)NCC)cnc(CNc2cccc(Oc3ccc(Cl)cc3)c2)nc1 c1(C(N2CCCC23CCN(C(C2CC(O)C2)=O)C3)=O)cc2ccncc2c(O)n1 C(=O)(C(F)(F)C(C)(C)O)N1C(C=CC(=O)N(C2CNC(=O)C2(C)C)C)CCC1 C1(CNC(C(C(COC)C)C)=O)N(C(=O)C(=O)C(C)(C)C)CCCC1(C)C C1(NC(CCCCN(C(C)=O)C)=O)CC(CNC(C2COC2)=O)C12CCC2 N1(C(C(=CC2CCCC2)C)=O)CCC(C(=O)NCc2nnc(C)o2)CC1(C)C CC1(C)CN(C(C23CC2CN(C(c2cc4ncccc4[nH]2)=O)C3)=O)CCC1O CC(C)C(CC(=O)NCC1CCN(C(c2cnnn2C2CC2)=O)C1)C(C)C Cc1cc(C(=O)NC2CCCN(C(=O)CC3(C)CC3(F)F)CC2)ncc1F CC1CC1(F)C(=O)NCCCN(C(=O)Cn1cnnc1)CC1CCCC1 c1(C(N(C2(C(=O)NC(CC=C)CC=C)CCC2)C2CC2)=O)cc(C)cc(O)c1 C1(CC)CC2CC2CC1C.c12ccc(nc1)C(=O)N1CCC(CCO)(C1)C2 c1(C(=O)NC(C2(O)CN(c3cc(OC)ncn3)C2)C)cccc2nc(O)[nH]c12 C1(NC(C=CC(CC)=CC)=O)CN(C(c2cc(Br)oc2C)=O)CC1OC c1(C(=O)NC2CN(C(Cc3ncc(CC)[nH]3)=O)C2)c(O)nc(C)c([N+](=O)[O-])c1C C(=O)(CCCCCF)NC1C(CNC(C23CC(C)(C2)C3)=O)CCCC1 Cc1cc(C(=O)NC23CCC(C(=O)N(C4CCCC(O)C4)C)(CC2)C3)cc(O)c1 c1(C(N(C)CC2CN(C(c3cccc(C#N)c3)=O)C2)=O)cnc2[nH]ncc2c1 C(C)(C)(CCCO)N(C)C(=O)NC1CCC1C(=O)OC(C)(C)C C1(C(=O)NCC2(COC)CN(C(c3[nH]nnc3C)=O)C2)CCCC2CCCN12 C12(C(=O)NC(C=C)(C)C)COCC1CN(C(c1cccc(OC)c1)=O)C2 CC1(CNC(c2cnc(Br)s2)=O)CCCN1C(c1ccoc1Cl)=O C1(CNC(CN2CCC(C)CC2)=O)CC2CCC1N(C(=O)C(C)c1ccsc1)C2 C#CCC(CC(F)F)C(=O)NC(c1nocc1C(=O)NC1CCC2(CC2)C1)C Cc1cccc(C=CC(=O)N(C)CC2(NC(c3cn4ccnc4s3)=O)CC2)c1 N1(C(C(C(C)(C)C)NC(CCN(C)CC)=O)=O)CC2CCC(C1)C(=O)O2 CC1(C)C(NC(c2nnc(O)o2)=O)CC1CNC(c1coc(OC(F)F)n1)=O c1(NC)ccnc(C(=O)NCC2(C)CC(NC(c3conc3C(F)(F)F)=O)C2)c1 CCCC(C)(C)C(=O)N1CC2(CCN2C(C2(C)CCN(C)C2=O)=O)C1 N1(C(c2n(CC)ncn2)=O)CC(CNC(c2ccsc2OC)=O)CC1C Cc1cccc(Br)c1NC(C1CC(NCc2ccc(N3CCCCC3)cc2)C1)=O C1(CC(=O)NCC(C(=O)NC)O)CCCN(C(=O)Cn2nccn2)C1 CCCC(C)(O)CC(=O)NC1CC(O)CN(C(C2C3CCC2(C)C3(C)C)=O)C1 Cc1ccc2c(c1C)OCC2NC(N1CCCC(NC(=O)NC2CC2)C1)=O c1(N2CC3C(CNC(=O)COC4CCCC4)C3C2)nc2cc(F)ccc2o1 CCC(CNC(C1(CO)COC1)=O)(CC)NC(=O)CNc1nccc(OC)n1 C1(C)(NC(C2N(CC)C(=O)CC2)=O)CCCN(C(=O)Cc2nocc2C)C1 N1(c2n(CC=C)c(-c3cccnc3)nn2)CCC2(CC1)OCC1CC21 N1(C(C(C(CC)C)O)=O)CCc2ccccc2C1CNC(c1ccon1)=O c1(C(C)C)cccc(C(=O)NCC2CCN(C(=O)Cn3cccn3)CC2)c1 CCC(Cc1cn(CCOC)nn1)C(=O)NC1CCN(CC2CC2C(=O)O)CC1 C=CCC(C)(C)CC(=O)NC1CCSC12CN(C(=O)CCC1(O)CCC1)C2 Cc1nn(CC(=O)NC(CCF)C(=O)N2CCC(CCO)C2)c(=O)o1 C1(NC(C2(OC)CCCC2)=O)CCCN(C(c2cccnc2S)=O)C1 N1(C(=O)CC(F)(F)F)CCC2CCN(C(c3occ4c3CCCC4)=O)CC2C1 C(=O)(CCCCCCc1ccccc1)N(CCC(C)NC(c1cnco1)=O)C Cc1ccc(F)c(OCC(=O)NCC2(O)CCN(C(c3ccc(C#N)s3)=O)C2)c1 c1(CC(=O)N(CCCNC(=O)CC2CC3COCC23)CC)cc(C)cc(F)c1 CCC(C)C(CC(=O)N1CC2CC(F)CC2C1)NC(=O)C(C)(C)n1ccnn1 Cc1ccsc1C(N1CCC(C(C)(C)C(=O)N)C1)=O.C(F)C(=O)C1CC1C C(=O)(C(CC(C)C)C(C)C)NCC1C(NC(Cn2c(=O)ccc(C)c2)=O)CCC1 C(=O)(C1CCCc2cncn21)NC1CC(CNC(c2cnc(C)[nH]c2=N)=O)C1 c1(C(N(C)CCC2CC3CCC2O3)=O)cccc(S(=O)(=O)NCC(N)=O)c1 CC(C)CC(C)C(=O)NC(C)(CO)C(=O)N(C)CCc1ccccn1 CC(C)(C#CC(=O)C1CC2CC(C)CC(C1)C2)C(=O)NCc1cccc(Cl)c1 C1(CNC(CCC(C)SC)=O)CN(C(c2ccnc(C3CC3)n2)=O)CC12CCC2 C(=O)(CS(=O)(=O)CCOC)N1CCCCC(N(C(C=CCCC)=O)C)C1 C1(NC(C2C(CC)C2)=O)CCN(C(c2cc(C(F)(F)F)n(C)n2)=O)CC(C)(C)C1 CCC(C)(C#N)C(=O)NCC1CCCCC1NC(c1cc(C(C)C)nn1C)=O N1(C(C=CC(CC)C)=O)CCC(C(N2CC(N=[N+]=[N-])C2)=O)(C(C)C)C1 C1(CC=C)(NC(c2cc(Cl)ccn2)=O)CCCN(C(C2(SC)CC2)=O)C1 C(CCC)(C(=O)NCCC1(CNC(=O)C=CCN(C)C)CC1)=CCC C1(OC)CN(C(c2c[nH]c(C#N)c2)=O)CC1NC(C1(C)C=CCC1)=O C=C=C(C)CC(=O)NC1CC(CNC(c2ccn(-c3cccs3)n2)=O)C1 c1(N(C2CCN(C(C(c3ccc(Cl)cc3)C)=O)CC2)C)cc(=O)n(C)cn1 N1(C(C(COCC)(C)C)=O)CCC2CC2(C(=O)NCc2ncnn2CC)CC1 N1(C(CC=C)=O)CC(C2CN(C(C3COC(=O)O3)=O)C2)C1 S(=O)(=O)(c1cn(C(C)C)nc1C)N(CCN(C)C)Cc1c(C)ccs1 N1(C(C(COC)CC(C)C)=O)C2CCCC1CN(C(c1cn[nH]c1)=O)CC2 C(c1ccc([N+](=O)[O-])cc1)=C(C)C(=O)NC(C(C)C)c1nn[nH]n1 c1(C(N2CCC(C(=O)Nc3ccccc3CO)C2)=O)cnc(Cl)c(C(F)(F)F)c1 c1(C(=O)NC2CC(NC(c3ccns3)=O)C2)cnn(C(F)(F)F)c1 S(=O)(=O)(c1ccc(NCC2C3CC4CC(C3)CC2C4)c(C#N)c1)NCCC(C)C S(=O)(=O)(c1ccc(C)c(C)c1)NCC(=O)NCC(CNC(CCCC(C)C)=O)C C(=O)(C(C)(C)C(C)(C)C)NCC1(F)CCC(CNC(CN2CCC(C)C2)=O)CC1 CCC(C)(C)C(C)CC(=O)N1CC(CNC(=O)CCc2cnn(C)c2)C2(CC2)C1 C12(C(N(C3CCN(C(=O)C4=C(Cl)CC4)CC3)CC#C)=O)COCC1C2(F)F c1(C(=O)NCC(CNC(=O)CCn2cccn2)O)ccnc2ccncc12 Cc1ccc(CNC(N2CCC(C(c3ccncc3)O)C2)=O)cc1C C1(C)(CNC(CSC)=O)CCCN(C(c2ccc(C(F)(F)F)cc2N)=O)C1 N1(CC(=O)N(CC(CC)NC(c2ccsc2SC)=O)CC)CCCCC1 C1(CNC(CC2(O)CC(C)(C)OC2)=O)C2CCCC1N(C(C1CC(=O)C1)=O)C2 C1(NC(CCC(C)C)=O)CCC2CCN(C(c3cc(NC(N)=O)ccc3Cl)=O)C12 c1(C(=O)NC(C2CCCC2)CNC(c2c(C)cn(C)n2)=O)cc(F)c(F)cc1F C1(OC)CC(NC(C)=O)CN(C(=O)CCSC)C1.C12CCCCN1C(=O)C2 C1(C(=O)NCCCOCCN(C(=O)C(O)(C2CC2)C2CC2)C)CC1C1CCCC1 CCCC(O)C(=O)NCCN(C)C(c1nnsc1C)=O C1(CN(C(C2(C#C)CC2)=O)CC)CCN(C(C2CCOC2C)=O)CC1 N1(CC(N2CC(NC(CC(C)F)=O)C(O)C2)=O)CCC(=O)NC1=O C(N=c1ccc([N+](=O)[O-])c(OC(C)C)[nH]1)C1N(C(C(C=C)(C)O)=O)CCC1C CC1CCN(C(c2cccc(-n3ccnc3O)c2)=O)CC1CNC(=O)CC1CC1 C(CCCCCNC(C12CC1CN(C(=O)CNC(N)=O)C2)=O)N(C)C CCCCC(=O)NCC(C1CCCC1)NC(=O)CC(C)n1cccn1 C1(CC(=O)NCC(N2CCN(C(C3CC(F)(F)C3)=O)CC2)=O)CCCOCC1 C1(C#N)(C(=O)NC(C)C(C2CCCCC2)NC(=O)CN(C)CCO)CCCO1 c1(C(=O)NC(CN(C(c2nc(CC(C)C)sc2)=O)C)C)cnn2ccncc12 C1(CNC(C(C(C)C)CO)=O)CCN(C(=O)Cc2cc[nH]n2)CCC1(F)F Cc1ccc(Cl)c(C(=O)NCC2CCN(C(c3cc(Cl)n(C)n3)=O)C2)c1 c1(-c2n(-c3ccc(OC)c(OC)c3)nc(C3CCC3)n2)cc(Br)c(F)cc1Cl S(=O)(=O)(c1ccc(NCc2cncc(F)c2)c(Cl)c1)N1CCCCC(SC)C1 n1(CC(=O)NCC(c2cccc(C)c2)NC(C2C=CCC2)=O)nc(C)c(Cl)c1C N1(C(Cc2ccn(CC)n2)=O)CCCCC1C(N1CC(N(CC(C)C#N)C)C1)=O Cn1c(=O)oc2c(C(=O)NCC3CCN(C(=O)COCP(C)(C)=O)C3)cccc12 CN1CCC(C)(C(=O)NCCOC2CCN(C(c3ccc(N)cc3Cl)=O)C2)CC1 CCCCC(CNC(=O)CC(c1ccccc1F)C)NC(c1cc(CC)on1)=O c1(C(CC(=O)NC(CC(C)NC(C2CC(=C)C2)=O)C)C)ccc(C)cc1 N1(C(N2C(C)COCC2)=O)CCCC(n2ccnn2)CC1 C12(NC(C(C)Sc3ncccn3)=O)CCC(CC1)N(C(=O)C=CC(F)(F)F)C2 c1(N(CC(CN(C)C(C2CSCCS2)=O)O)C)nc(Cl)ncc1C1CC1 N1(C(CN(CC(C)C)C(C2CC(F)(F)CS2)=O)=O)CCCOC(C2CC2)C1 c1(COC)cc(C(=O)NCC2CC(CNC(=O)CSc3nccn3C)CO2)n[nH]1 c1(SC)ccc(-c2nc(C(O)C(F)(F)F)n(CC(C)CO)n2)nc1 c1(NCCC(C)(C)NC(C2C(CC)OCC2)=O)nc(C)nc2sc3c(c12)CCC3 CP(C)(=O)c1cccc(C(=O)NCC=CCNC(C2CCN3CCCC3C2)=O)c1 Cc1nc(CC(C)C)c(C(=O)NC(C2CN(C(=O)CC3CCCO3)C2)C)s1 C=C(Cl)C(C)(C)C(=O)N(CCCCCCNC(=O)C(C)(C(C)C)NC(C)=O)C Cc1cc(Cl)cc(C(=O)NC2(CCNC(C3(C)CC3F)=O)CC2)c1O C1(C(=O)NC2(CCNC(=O)CC3(O)CCC3)CCC2)(OC(C)C)CCOC1 CC(C)CC(CNC(=O)OC(C)(C)C)NC(=O)Cn1cnnc1 N1(C(C(C)OCC=C)=O)CC2CN(Cc3c[nH]c4cnccc34)CC2C1 c1(NC(c2ccc(CCC(N3CCN(C(C)=O)CC3)=O)[nH]2)=O)c(C)ccnc1Cl N1(C(C(CC)C(F)(F)F)=O)CC2CCN(C(C3(CF)CC4(CCC4)C3)=O)CC2C1 CC(=NO)C1CC(C(=O)NCC(C(C)(C)C)NC(=O)C(C)(F)F)C1(C)C C(=O)(C(C)(C)C(=O)N1CCC(C2OCCC2NC(C2CCCN2C)=O)CC1)NC C=CC(CCC)CC(=O)N(C)CCC1CCCCN1C(=O)CCCc1cccs1 C1(NC(=O)NCc2n(C)c(-c3ccc(F)cc3)nn2)CC2CCCC2C1 c1(CSc2n(CC=C)c(CCn3cncn3)nn2)nnc2n1CCCC2 c1(C(N(C(C)CN(C)N(C)C(C2CCN(C)CC2)C)CC)=O)ccccc1SC c1(C(C(=O)NCC(C)CN(C)C(C2CC3CC2C3)=O)(C)C)ccc([N+](=O)[O-])cc1 c1(C(N2CCCC(CN(C(C(C)N(C)C)=O)C)C2)=O)ccc(N)c2ncccc12 C(=O)(CCCCCCS(N)(=O)=O)NC1CCN(C(Cc2cc(C)sc2)=O)CC1F CC(CN=[N+]=[N-])NC(=O)CNC(C1CC(C)(C)C1)=O N1(C(c2c(SCC)ncs2)=O)CC2CC(C)N(C(=O)C(CC)CC)C2C1 c1(CN(C(C(C(CC)C)O)=O)C)cnn2c1CN(C(c1cncc(F)c1)=O)CC2 CC1(C)CN(C(c2c(O)cc(O)cc2O)=O)CCC1NC(C1(C)COC1)=O c1(CCC)ccc(C(C(C)C)CNC(N2CCC(N3CCCCC3)C2)=O)cc1 c1(C(C)OC(c2c(C)nc(C3CCCC3)s2)=O)ccc(Br)c(F)c1 N1(C(c2c(C)non2)=O)CCC(O)C(C(=O)N(c2ccccc2)C2CCOC2)C1 Cc1cc(C(C)C(=O)NCC2CC2CNC(c2cccc(C(C)C)n2)=O)c(C)o1 C1(CC(=O)N(CCC(=O)NCCN2CC=CC2)CCCO)CCC(=O)N1 CC(CNC(C1CC2(CC2)CO1)=O)CC(=O)NOCc1ccc(F)cc1 C1(CC)CCN(C(c2cc(C(C)=O)c[nH]2)=O)C1C(=O)N(CCN=[N+]=[N-])CC C1(N(C(=O)CNC(=O)NC2CC2)C)COCCN(C(=O)C=CC(F)F)C1 N(C(=NCCN1CCCC1)N1CCC2(CC1)C(F)(F)C2(F)F)C1CCC(SC)C1 C(=O)(CC1OCc2ncccc21)NC1(C)CC(NC(=O)C=C2CCC2)C1 C1(CNC(C2CCC(OC)C2)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)C12CC2 c1(C(C)NC(C(=O)N(CC)Cc2cccs2)=O)ccc(O)c(F)c1 C1(C(=O)NC(COCC)C(=O)NCC(F)(F)F)COCCN1CC C1(C)(C(N(CCCCCC)CCNC(=O)C(CO)NC(=O)C(C)C)=O)CCCCC1 N1(C(C(C)SC)=O)CC=C(CCNC(=O)CSCc2nnc3ccccn23)CC1 c1(NC(C(CC(C)C)NS(C2(CC)CC2)(=O)=O)=O)cccc([N+](=O)[O-])c1C C1(CNC(C(C(=O)OCC)F)=O)CN(C(=O)Cn2cc(C)cn2)CC12CCC2 CCCC(C(=O)NCCC(=O)OCC)N1CC(O)(Cc2cccnc2)C1 C1(C#N)(CC)CCN(C(=O)C(F)C(C)CNC(C2(O)CCSCC2)=O)CC1 Cc1cc(C(N2CCC(CNC(c3cncc(Cl)c3Cl)=O)C2)=O)c2n[nH]cc2c1 C1(NC(c2ccc(N)cn2)=O)CC2CC1CN(C(C1CCCCNC1=O)=O)C2 C=CC(C)(CC)C(=O)NC1CC(CCNC(=O)CC(C)c2ccco2)C1 c1(N(C)C)nccc(=NC(=O)C2CC(F)CN(Cc3ccc(CBr)cc3)C2)[nH]1 N#CC1(C(N2CCOC(CNC(=O)COCCO)C2)=O)CC2C=CC1C2 c1(C(=O)NC(CN(C(CC2C(C)=NNC2=O)=O)C)C)cc(O)ccc1C N1(C(c2n(C(C)C)ccc2)=O)CCN(C(C23CCCC2CC3)=O)CC(C)C1 N1(Cc2c(-c3c(OC)nccc3)cnn2C)CCC(N(C)CCO)C(C)C1 c1(C(=O)NCCOCCC(=O)NCC(COCC)C)cc(C#N)cn1C C1(C)(CNC(c2c(C(=O)OC)[nH]cc2)=O)CCCN(C(=O)C(F)(F)C2CC2)C1 c1(CC)noc(CC)c1Cn1c(N2CCCC(CCC(=O)OCC)C2)nnc1C C(=O)(CC1=CCN(C(c2cc(F)ccc2O)=O)CC1)N(CC(N)=O)CC(N)=O CC(C)C(CCC(=O)NC1COCC1CO)NC(c1cc(O)nn1C)=O C=CCC(C)(C)C(=O)N1CC2(CC(CCNC(=O)C=CSCc3ccco3)C2)C1 C(C(CC(F)(F)F)NC(c1cc(C)nn1C1CC1)=O)NC(C1N(CC)CCC1)=O N1(C(C=COCC)=O)CCC2(COC(CNC(c3ccc4ncnn4c3)=O)C2)C1 C12(C(=O)NCC3(NC(C(C)n4ccnn4)=O)CCCC3)CCC(N=[N+]=[N-])C1C2 c1(NC(CN2CCN(OC)CC2c2nn[nH]n2)=O)cccc(Cl)c1C C1(CC(=O)NCC2(NC(C(=O)N(CCOC)C3CC3)=O)CCC2)CC(O)C1(C)C C(=O)(CCCCCCC(=O)NC1CN(C(c2cn(C)nc2Br)=O)C1)OC N1(C(C2N(C(C)=O)CCC2)=O)CC2(CCCN(C(=O)COCCOCCO)C2)C1 c1(C(=O)NCC2C(NC(=O)CCF)CCC2)cnn2cccc2c1 c1(C(N2CCCC(CN(C)C(c3ccoc3)=O)C2)=O)c[nH]c(=N)c2[nH]ccc12 c1(CCC(=O)NC2CCCN(C(c3cc(C)nnc3)=O)C2)nc2cnccc2[nH]1 c1(CC)nc(N2CCC(CF)(NC(=O)CC(C)C(C)C)C2)[nH]c(=N)n1 C12(C(N3C(C(=O)NC)CC3)=O)CCN(C(=O)CN(C)C)CCC1C2 C(=O)(C(CC)CCOC)NCc1ncc(C(=O)NCC(CCC)OC)cn1 c1(CC)oc2ccccc2c1C(N1CC(NC(=O)CCn2cnnn2)C(C)C1)=O c1(C(=O)NC(C(CO)NC(COCCC)=O)C)ccc2nc(Cl)nn2c1 c1(OC)ncnc(C(=O)NC2CCC(C)N(C(C3CCC4(CCC4)C3)=O)C2)c1F C1(NC(C(COC)OC)=O)CCCC2CN(C(C3C=C(C)CS3)=O)CC12 C1(CCNC(C2CC(C#C)(O)C2)=O)CCCN(C(=O)C=C(C)C(C)(C)C)CC1 c1(C(=O)NC2CC3C(NC(=O)CCn4cccn4)C3C2)cc2cccnn2c1 N1(C(CSCCC#N)=O)C2CCCC1CN(C(=O)CC1CCCCC1F)C2 c1(C(C(=O)NCCNC(C2C(C(C)C)(CC)C2)=O)C)cccc(OC)c1 N1(C(c2cc(C)on2)=O)CCC2CCCC12C(N1CC(C)CCC1C)=O C1(N(C(C2CCCN2S(=O)(=O)CC)=O)CC)CCN(C(=O)CP(C)(C)=O)CC1 CC(N=c1ccn2ncc(S(=O)(=O)N(C)C)c2[nH]1)c1cccnc1O N1(C(c2coc(SC3CC3)c2)=O)CC2=C(C1)CN(C(c1cccnc1)=O)C2 c1(C(N2CC(C)N(C(C3(CN(C)C)CC3)=O)CCC2)=O)c2c(nn1C)CCOC2 C1(CNC(c2cnc(OCC)s2)=O)CN(C(=O)C(C)=C(C)C)CC(C)(C)C1 C(=O)(CCCC(F)(F)CO)NC1CC(CNC(c2ccn(CCN(C)C)n2)=O)C1 C1(CNC(C(CCC)OCC)=O)CN(C(=O)CCn2cccn2)CCC1(C)C C1(CNC(C(COC)(C)C)=O)CN(C(c2cc(C)cc(C)c2C)=O)C2(CCC2)C1 N1(C(C2CN(C(N(C)C)=O)C2)=O)CCN(C(C2CCC=CCC2)=O)CC(O)C1 c1(C(N2CCOCC2CC(N2CC(c3ncc[nH]3)C2)=O)=O)cccc(O)c1 c1(C(=O)OC)ccc(NC(=O)C(C)(C)NC(=O)OC(C)(C)C)c(COC(C)=O)n1 c1(C(N2CCC(C(N3CCC(CCOC)C3)=O)(C(C)C)C2)=O)cc(C)nnc1O C1(CN(C(c2nncs2)=O)CC)CCN(C(=O)CCN2CCCC2)C1 C1(C(=O)NC(C2(CNC(C3(c4ccno4)CC3)=O)CC2)C)CCCN(C)C1 CC1CCC=C1C(=O)N1CCCC1C(C)NC(=O)CN1CCC(=O)NC1=O c1(OCC)ccc(CN(CCCO)C(c2cccc(-n3cnnn3)c2)=O)cc1 N1(C(C=CCCC)=O)CCC2(NC(c3cc(O)cc(Cl)c3)=O)CC2C1 c1(C(N(C2CCN(C(=O)C(C)(C)C(O)CC)C2)CCC)=O)ccn2cnnc2c1 C1(CNC(c2c(CCC)occ2)=O)N(C(c2cncc(O)c2)=O)CCCC1(C)C Cc1[nH]nc(C(=O)N(CCCNC(C2(C)CC(F)(F)C2)=O)C)c1[N+](=O)[O-] N1(C(C)C)CCCC(C(=O)NC(C)CC(C)NC(=O)Cc2cc(C3CC3)on2)C1 C(=O)(C1=NN(C)C(=O)CC1)N1CC(NC(c2nc(OCC)sn2)=O)(COC)C1 C1(Oc2n3c(ccn2)nnn3)CCC2(CCCOC2)C1 C(N=c1cc(NCCC#CCO)nc[nH]1)c1cn(CC(C)C)nn1 c1(C(=O)NCC2CC(OC)CN2C(=O)C(C)n2ccnc2)c(C)cnnc1O C1(C(N(CCOC)C(C)C2CC2)=O)CCN(C(c2cccc(CC#N)c2)=O)CC1C CC(C)C(C(=O)NCC1(C(C)NC(=O)CC2CCCC23CC3)CCCC1)N(C)C N#Cc1ccc(C(=O)NC2CC23CC(NC(c2ccc(OC(F)F)cn2)=O)C3)s1 c1(OCC)cccc2[nH]c(C(=O)OCC(=O)OCc3ncc(Br)cc3C)cc12 c1(OC)ncc(C(=O)NCc2ccc(C(=O)NOCCO)nc2)cn1 C1(CC(=O)NCC(c2cccs2)O)(NC(c2ncn(C(C)C)c2)=O)CCCCC1 c1(C(N(C2CN(C(c3c(OC)cnc(F)c3)=O)C2)C)=O)cc(F)c(F)c(O)c1F N(C(=NCc1ccccc1CC(N)=O)NCC1CC(OC)C1)C(C)C c1(C(=O)NCC2(C)N(C(CC=CC=C)=O)CCC2)ccc2cc(Br)ccc2n1 c1(C(=O)NC2C3CC(O)C2N(C(C2CCC(F)CC2)=O)C3)cccc2nn[nH]c12 n1(CC(=O)N(C)CC2N(C(C(C=C)C)=O)CCC2)nc(C)oc1=O C1(C(N2C(CCC)CCC2)=O)CSCCN1C(=O)CCCC1CCCC1 C(=O)(CCCCC(F)F)NCC1C(CNC(c2nccc(OC)c2)=O)C1 C1(CNC(COC2(C)CCCC2)=O)CC(C(F)(F)F)CN1C(C1CC1C(F)F)=O CN=c1[nH]cc(C(=O)N(CCCC(=O)NCCC(O)C(=O)OC)C)s1 c1(C(N2CCC3CN(Cc4ccc5n[nH]cc5c4)CC23)=O)cc(F)cc(F)c1Br c1(C(N2CCN(C(C(C)OC)=O)C(CO)C2)=O)cc2c(Br)cccc2cn1 c1(N2C(C(=O)NC(COCC)C)CCC2)ncc(C)c(OC)n1 c1(NC)c(C)cccc1C.N12CCN(CC1)C(=O)C2c1cc(C2CC2)on1 C(C(F)(F)C(=O)NCC1(CCNC(C2CCCSC2)=O)CC1)N(C)C CC1CC(C#N)(C(=O)NCC2(CNC(=O)CCCc3cncs3)CC23CCC3)C1 c1(CCS(N2CCC(OCC(C)C)C2)(=O)=O)ccc(Cl)cc1 N1(C(C(C(=C)C)(C)C)=O)CC(CNC(=O)CCOC2CCOCC2)C2(CCC2)C1 C1(NC(C=Cc2ccc(SC)s2)=O)CN(C(=O)C(C)CC(F)F)CC1(C)C N1(C(C(CC)(C)CC)=O)CCC(C(=O)Nc2ccc(SC)cc2)=C(F)C1 N1(C(C(C)S(C)(=O)=O)=O)CCCC2(C1)CN(C(C1Cc3n[nH]cc3C(=O)N1)=O)C2 n1(CC)nnc(C(N2CCOC(C(=O)NCCC3CCCCC3)C2)=O)c1C C(C(=O)NCCNC(c1cccnc1NC)=O)(C(C)C)OCC C#CCC(C(=O)NCC1(SC)CC1)NC(C1CC(C2CC2)C1)=O N1(C(c2cncc(NC)c2)=O)CCN(C(=O)C(O)C(C(C)C)OC)CC(C)(F)C1 C(=O)(C(C)(F)CC1CCCC1)NC1C(NC(CCC=CC)=O)C1 N1(C(C2(CC)CN(C(c3ccccc3Cl)=O)C2)=O)C2CCC1CC(=O)NC2 c1(C(N2CCCC(F)(CNC(C3=CC(C)(C)C3)=O)C2)=O)cc(O)ccc1[N+](=O)[O-] c1(NC(C2CC(OC)CN2C(C2CCCSC2C)=O)=O)ccc(C)c(F)c1 c1(OC)ccc2nc(N(CC(C)CO)C)[nH]c(=NCC3(OC)CCSCC3)c2c1 C1(CCNC(CCOC)=O)CN(C(=O)C(c2ccccc2F)F)CCCO1 C12(CNC(CCCSC)=O)CC(NC(=O)CCn3cnccc3=O)(CO1)C2 CN=c1[nH]c(C(=O)NC2CCCCC2NC(C2CC2C)=O)cs1 C(CN=c1[nH]c(=NCc2cncn2C2CC2)c2sccc2[nH]1)c1[nH]ccn1.C1CC1 C1(C(=O)NCCn2cc(C(C3CCCCC3)N(C)C)nn2)(OC)CCCOC1 c1(CNCC2(O)CCCN(C(=O)OC(C)(C)C)C2)c(F)ccc(F)c1O C(=O)(C(C(C)(C)O)NC(=O)COC(C)(C)CNC(=O)C(C)CN(C)C)OC c1(CNC(C2(CC#C)CCC2)=O)nc(CNC(=O)CC2CC(C)C2)cs1 c1(CNCC(=O)N(CCCNC(=O)C(F)NC(N)=O)C)ccc2ccccc2c1 N1(C(C=CC)=O)CCC(C(N2CCCC(NC(=O)C3CC3)C2)=O)C1(C)C C1(NC(C(C)SC(C)C)=O)(CCNC(c2ccn(CCO)c2C)=O)CCOCC1 c1(CNC(c2c(C)nc[nH]2)c2nnnn2C)ccnc(Cl)c1Cl c1(C(=O)NCC2(CN(C(=O)CN3CCCC3CO)C)CC2)ccc(=N)[nH]c1 Cc1cc(C(N2CC(CNC(C3COCC(C)(C)O3)=O)C2)=O)cc(C)c1C c1(C=O)cc(C)ccc1Cl.C1(CCC)CN(C(C2(CC)CCC2)=O)CC1O C(C(COC)C(=O)NC1CN(C(c2ccc(Cl)cn2)=O)CC1OC)OC c1(C(N2CCC(CC(=O)NC(CC#CC)C)CC2)=O)cccc(C)c1C#N c1(SC)cc(F)ccc1C(=O)NC(C)CCCNC(C1(C)CCCS1)=O C12(C(N(C3CN(C(c4ncc(Cl)nc4Cl)=O)CC3(C)C)C)=O)CC1COC2(C)C Cc1cccc2[nH]c(=NCC(C(C)(C)C)NC(=O)C(c3ccccc3)O)oc12 C1(N(CCC)C(C23CCC2C3)=O)CCN(C(c2sccc2SC)=O)CC1 CC1(C)C=C(C(=O)NCCCN(C(C23CC(CCO2)C3)=O)C2CC2)C1 c1(CCC)[nH]ccc1C(=O)NCc1n[nH]cc1C(=O)N(C(CC)C(C)C)C1CC1 C12(C(N3CCC(CNC(C(C)(C)C4CCC4)=O)C3)=O)CC3CC1C2C3 C1(NC(C23OC(C)C(C2)C3)=O)CCCN(C(=O)CCP(C)(C)=O)CC1 c1(-c2c(C(N3CC(C(CC(=O)OC(C)(C)C)O)C3)=O)nco2)c(Cl)cccc1Cl CN=C(NCCC(=O)OC)N1CCC2CN(Cc3cccc4c3OCC4)CC2C1 N1(C(c2c(OC)nsc2)=O)CCN(C(C2CCN(C)CC2)=O)C(CCO)C1 N1(C(C(CCC)N(C)C)=O)CCN(C(C2CCSC2)=O)CC1CC(F)F N1(C(CNC(CC)=O)=O)CC(O)CCC1C(N1CCC(C)C1COC)=O CCC(C)(C)C(C)CC(=O)N1CC=CC1CNC(c1nccc2ccsc12)=O C(CN=c1cccc(S(=O)(=O)NC2CC(CO)C2)[nH]1)c1nnc(C)n1C N1(C(CN(N2CCCCC2)C(C(c2cnn(C)c2)C)=O)=O)CCC(=C(F)F)CC1 C1(c2nc(COC)on2)CC(F)(F)CN1C(=O)CC(C(C)C)n1cccc1 N1(C(CCSCC(C)C)=O)C2CCC1CC(NC(C1CCOC1=O)=O)C2 Cc1oc2cc(C(=O)NC3(C4CCCN4C(=O)C(O)C(C)(C)C)CC3)[nH]c2c1C c1(CNC(C(CC)n2ccnc2)=O)cccc(C(=O)N(CCO)CCN(C)C)c1 C1(NC(COC)CNC(=O)OC(C)(C)C)COCCN1CC CC1OC(C)CC1C(=O)N(CCCn1cc(-c2ccnn2C2CCC2)nn1)C1CC1 c1(SCC(=O)NCCCN(C(C=CC=CCC)=O)C(C)C)nc2ccccc2[nH]1 N1(C(C(C)OCCC=C)=O)CCOCC(CNC(c2cc(C(C)C)on2)=O)C1 c1(N2CCCC(COC)C2)cc(S(=O)(=O)N2CCSC(C(C)C)C2)ccc1C#N c1(CCC(=O)ON2CC(c3ccccc3)C2C(=O)O)ccncn1 CC1(C)COCCC1C(=O)NCCC(O)CNC(=O)Cn1cncn1 CC1CCC(CNC(c2ccn(C)c(=O)c2)=O)CN1C(=O)CC(C)(C)N(C)C C1(C(=O)NCC(C)=CC(=O)N(C2CCOC2)CCF)CCSC(C)C1 C1(c2occc2)N(Cc2nnc(-c3cccc(Br)c3)o2)CC12CCC2 C1(CC=C)(NC(C2CC(n3cnnc3)C2)=O)CCN(C(C2CCS2(=O)=O)=O)C1 N1(C(C2CCCCC2O)=O)CCCC(C2CN(C(C34COC(CF)(C3)C4)=O)C2)C1 c1(CC)sccc1C(=O)NCCOC(C)(C)CNC(C1OCC1(C)C)=O CCC(C(=O)NC1CCN(C(c2cc(C)ccc2F)=O)CC1O)C(F)(F)F c1(NC)ccc(F)cc1NC(C1CSC(C)C1)=O C(C(O)C(=O)N(CCCNC(c1cc(-c2ccccc2)[nH]n1)=O)C)N(C)C C=CC1(C(=O)NCC2(C)CNC(=O)O2)CCN(C(=O)Cc2ccc[nH]2)C1 N1(C(C=CCC)=O)CC2(CCN(C(c3c(C)nn(CC)c3Cl)=O)C2)C1 N1(C(C(C)=C(C)C)=O)CC(NC(c2cnc(C(C)(C)CF)o2)=O)C2(CC2)C1 c1(C(N2C(NC3(CNC(=O)C(F)(F)F)CC3)CCCC2)=O)cc(Cl)c(Cl)c(Cl)c1O C1(NC(CCNC(CC(C)C)=O)=O)CC12CC(NC(=O)Cc1ccc(Cl)cc1)C2 c1(C(=O)NC2(CO)CN(Cc3cccc(OC)c3)C2)ccc([N+](=O)[O-])c(O)c1 N(C1CN(C(=O)C(O)C2CCC2)Cc2ccccc21)C(C(C(C)C)(C)C)=O C1(NC(CCNC(=O)NC)=O)CCC2(CC1)CCN(C(=O)Cc1ccc(C)s1)C2 c1(SCC(=O)NC2(C)CCCN(C(c3cnc(Cl)[nH]3)=O)C2)ncnc2[nH]cnc12 N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCN(C(c2cc(O)cs2)=O)CC(C)C1 N1(C(CCC=C)=O)C2CCC(C2)C1CNC(c1csnc1Br)=O C1(NC(COC2CC(NC(c3[nH]n(C)c(=O)n3)=O)C2)=O)CCCCC1(C)C c1(C(=O)OCC(C2C(C(=O)OC(C)(C)C)C2)=O)cc([N+](=O)[O-])cc(Br)c1F c1(C(=O)NCC2C(NC(c3c(C)snc3)=O)CCC2)ncc(F)cn1 c1(N(C)C)ccc(C=CC(=O)NC23COC(C2)C(NC(=O)C2=CCSC2)C3)cc1 c1(NC(=O)CCN2CSCCSC2)ccc(C(N2CCC2CO)=O)cc1 N1(CC(N2CCC(NC(CN(CCC)C)=O)CC2C)=O)CCN(CC)C(=O)C1=O C(=O)(C(C)(C)C(C)NC(=O)CCCC1CCCC1)N(CCCC=C)CC N1(C2C(=O)N(Cc3nccs3)CC2)CCCC(S(=O)(=O)N2CCCC2)C1 N1(C(C(F)=CCC)=O)CCC(C)C1C(=O)NCCNC(C)=O C12(CNC(C=NOC)=O)CCC(CC1)N(C(c1cnc(C3CCC3)nc1O)=O)C2 CC(=O)CCC(=O)NC(CO)C(=O)NC(CCN(C)C(C)=O)=O c1(C(=O)NC(CC)C)cn(C)nc1Nc1ccc(C(C)CC)cc1 C(CNC(C1(SC)CCC1)=O)(CCNC(C1C=CCC1)=O)OC C(c1ccncn1)=CC(=O)NC(C1CCN(C(c2c(CC)c[nH]n2)=O)C1)C C=C(C)CN=C(NCC1CCN(C)C1)NCC1(c2cccs2)CCCCC1 N1(Cc2c(Br)cc(OCC)c(O)c2)CCC(C)(O)C(O)C1 C1(NC(CSCCC(C)C)=O)CCN(C(=O)CNC(=O)C(F)(F)F)CC1F c1(C(N(C(CCNC(Cn2c(C)nc(C)n2)=O)C)C)=O)nc(C)n2c1CCCC2 C(c1ccc(=N)[nH]c1)=CC(=O)NC1CCC(CCNC(C(CCSC)O)=O)C1 N1(C(C2CCC(C)(CC)O2)=O)CCN(C(=O)Cc2ccc(Cl)nc2)CC(O)C1 C12(NC(C3(C)CCCN(Cc4cc(F)ccc4F)C3)=O)CCC(C#N)(CC1)CC2 Cc1noc(C)c1CCC(=O)NCC1CN(C(=O)C=CC(C)C)CCO1 C1(CC(N2CC(C3CCN(C(C4CCCCO4)=O)C3)C2)=O)CCCNC1=O C1(CNC(c2c(C)ocn2)=O)CC2(CCN(C(=O)C3=CCCO3)C2)CO1 N1(C(c2cc(C)nc(C)c2)=O)CC2CC(C1)N(C(C1CCN1C1CCCC1)=O)C2 C1(F)(CNC(C(C2CCOC2)OCC)=O)CN(C(C2(C3CC3)CC2)=O)C1 C1(C(N(CCC(C)(C)NC(C2(O)CCCCC2)=O)C)=O)C2CC3C(C2)C13 Cc1ccc(-c2ccsc2C(=O)NC2CN(C(=O)C3=CCSC3)C2)cc1 c1(CNC(=NCC)NCCCCC(C)C)cc(Br)c(OC(F)F)cc1F CC1CC(=O)NCC1C(N1CCCC(NC(c2cc(C3CC3)[nH]n2)=O)C1)=O n1(CC)ncc(C(=O)NC2CCC(NC(=O)C=Cc3ccc[nH]3)CC2)c1C CCCC(C)(C)C(=O)NCC(CC(=O)NCCCn1cnnc1CC)C1CCC1 CC1CCN(C(=O)CCCN(C)C)C(CNC(=O)CC2CC(O)C23CCC3)C1 C1(CCCC)CCCN1C(C1(C)CN(C(c2cnc(OC)s2)=O)C1)=O Brc1ccc(-c2ccc(N(Cc3ccccc3)Cc3nccn3C3CC3)nc2)cc1 C1(C(N(CCCC)C(C)CC)=O)CCCCC1NC(c1ncccc1O)=O C#Cc1ccc(CNC(N2CCN(c3ccc(CC)cc3)CC2)=O)cc1 C1(CC)CCC(C)N(C(c2nc(CNC(c3cnc(C)c(C)c3)=O)oc2C)=O)C1 CC1CN(C(=O)CN2CCC2)CCC1CNC(c1c[nH]nc1C(F)F)=O c1(C(=O)NC2(C)CCN(C(C3=C(C)CCC3)=O)C2)ccc2cccc(O)c2c1 C(=O)(C(CCC)OC)N1CC(CC#C)C1.C12(CCCO1)C(=O)N2 c1(C(=O)NCC2N(c3nnc(CC(C)C)s3)CCC2)cccc2[nH]ncc12 C(=O)(C1CCCc2nn[nH]c21)NCCCOCCNC(=O)CCOCC1CC1 c1(OC)cc(C(N2CC3CN(C(c4conc4C)=O)CC3C2)=O)c(OC)cc1Cl C(=O)(CC(C)C(C)(C)C)N1CC2(C(NC(c3n(CC#C)ccc3)=O)CC2)C1 c1(C(N(CCOCCN(C(CSC(C)C)=O)C)C)=O)cn(C(C)C)nc1C1CC1 C12(CNC(c3c(C)snn3)=O)CC(NC(C3CCC(=O)N3)=O)(CCO1)C2 CS(=O)(=O)c1cc(NC(c2cc(C#N)c(N)cc2O)=O)cc(C(F)(F)F)c1 C1(NC(C2(S(N)(=O)=O)CC2)=O)COC2(C1)CN(C(=O)C(F)n1cccn1)C2 c1(CNC(=O)NC(n2nccc2Cc2ccc(C)o2)C2CC2)ccc(F)nc1C c1(C(N2C3CN(C(C(CC)C(C)O)=O)CC2CC3)=O)cc(F)cc2c1NCCC2 N1(C(CSc2cn(C)nc2)=O)CC2CC(NC(=O)Cc3ccc(O)cn3)CC2C1 C#CC1CCC(NC(C2CCC(CNC(=O)C(C)(F)c3ccon3)CC2)=O)C1 N(C1CCCn2ccnc21)c1c(C)c(NCc2nc(-c3ccco3)n[nH]2)ncn1 c1(CC(=O)NC2C(NC(C3(C)C(C)CCC3)=O)COCC2)coc2ccccc12 C(CC)(C(=O)NCC(O)CN(C(=O)CC1CCSCC1)C)=CC CC(CC(F)(F)F)C(=O)NCC1CCCCC1NC(=O)Cc1cnns1 C(c1cscn1)=CC(=O)NC1CCC(CNC(=O)CNC(c2ccoc2)=O)C1 Cc1c(C(=O)NCCC2(NC(C3CCCN3C3CC3)=O)CCC2)nnn1C C1(CNC(C=CCOC)=O)CN(C)CCN1C(C1CCC(C)(O)CC1)=O c1(OC)ccccc1CC(C)(C)C(=O)NCC1CC1NC(=O)C1=COCC1 C#Cc1ccc(CC(N2CC(CN(C)C(C3(N(C)C)CC3)=O)C(C)(C)C2)=O)cc1 c1(OC(C)C#N)ccc(C(=O)NCc2cc(Cl)ccc2N2CCC(O)C2)cc1F N1(C(CC2CC(=O)OC2)=O)CCC2CCN(C(c3cc4n(c3)CCCC4)=O)CC12 N1(C(CCSC)=O)CC2CC1CCC2NC(C1CSCC(=O)N1)=O c1(OC)ncc(C(=O)Nc2nc(CN3CCCC3=O)cs2)cn1 c1(C(=O)OC(C(=O)NC(c2ccccc2)CCC)C)ncn(C)c1C CCC(C)C(O)C(C)C(=O)NC1CC1NC(=O)CC(C)c1cnn(C)c1 C#CCC(CC(=O)NC(C1CCCC1)CO)NC(=O)COCCC C1(NC(C2(CC#C)CC2)=O)CN(C(C2CCCC2c2nc(S)n[nH]2)=O)CC2CC12 CC(C)CCC(=O)NC(C(C)NC(=O)CCOC1CCOCC1)C(C)C N1(C(C2C(CC)CC2)=O)CC2CCN(C(c3ccc(=O)n(CCF)n3)=O)CC2C1 C1(NC(CC2N(C(C)C)CCC2)=O)CN(C(c2ncoc2C(F)(F)F)=O)CC1F CN=c1[nH]cc(C(=O)NCC2CCC2NC(C2C3COCC23)=O)s1 O=C1Cc2c(C(N3CC4CC(NC(c5cccs5)=O)C4C3)=O)ccnc2N1 C12CCN(C1C)N2CC#CC.C1(NC(=O)NCC(=O)OC)CCCC1 N1(C(=O)C(=Cc2cscn2)F)CCC(C2CCCC23OCCO3)C1 C1(CC)CN(C)C(=O)CN1C(=O)C(F)C(C)CNC(C1CCN(C)C1)=O N1(C(C(=O)NCC2N(CC(=O)NCCCOC)CCC2)C)CCN(C)CC1 N1(c2nc(N3CC(C#N)OCC3)c3c(n2)CCS3)CCOC2(CCSC2)CC1 c1(C(=O)NC2C3CN(Cc4c(C)nn(C)c4Cl)CC32)cc(F)c(F)c(F)c1F c1(C(N2C3CC(NC(CSCC#C)=O)C3CC2)=O)cc(C)c(Br)c(C)c1 N1(C(c2cc(C(C)C)on2)=O)CCC2(CC(NC(=O)C(F)=C3CCCC3)CO2)C1 C(=O)(CCCCNC(=O)CC1(CC)CCC1)NCC=C=C S(=O)(=O)(c1ccc(Cl)s1)N1CCC(NC(C2C(C)(C)C2)=O)CC1 C1(NC(C2=C(C)CCCC2)=O)CCCCC12CCCN(C(c1cc(O)cs1)=O)C2 c1(C(=O)OC(C)C)cc(C)n(CC(=O)OC(C)(C)C)c1C.C(CC1C(=O)O1)SC c1(C(N(C2CCN(C(=O)CC3C=CCCC3)CC2)C)=O)csc(=NC2CC2)[nH]1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCOCC(C)(CNC(=O)C2=CCCSC2)C1 C1(CNC(C(CC=C)CC)=O)CC2CCC(C1)N2C(C1CN2CCCN1CC2)=O Cc1c(C(=O)NCC2CCCN2C(=O)C2=CC(C)C2)cnn1C(C)C CC1=C(C(=O)NCc2ccc(CNC(C3CCCC3CN(C)C)=O)cc2)CCC1 c1(N(C(C)C)C)cc(Br)ccc1S(=O)(=O)NCC(C)C1(C(=O)O)CC1 N1(C(c2cccc(C3CC3)c2)=O)CCCN(C(=O)C(c2ccccc2F)O)CC1 C1(C(=O)NCC=CCNC(Cc2cn(C)nc2C(F)(F)F)=O)CC1C1(C)COC1 C(=O)(C(C)(C)C(C)C)N1CCC(C(C(C)C)NC(=O)Cc2ccc(Cl)cn2)CC1 c1(C(=O)NC2CCCCC2CNC(C23CCC(CO2)C3)=O)cc(O)nc(O)n1 C1(COCC#C)CCCN1C(=O)CC1(NC(=O)C=CC(C)(C)SC)CCC1 Cc1cc[nH]c1C(=O)NC(c1cccnc1)C(=O)NCCC1(CO)CC1 C(=O)(C(C)(O)CC(C)C)NC1C(NC(Cc2c(C)nn(C)c2C)=O)COCC1 N1(C(c2ccc(F)c(Br)c2)=O)CC2(CCC(NCc3ccc(I)o3)C2)C1 c1(NC(C2CCN(C(C3CC(C)OC(C)C3)=O)C2)C)ncc2ncn(C)c2n1 C(C(C)C)(C(C)(C)O)NC(CC1(OC)CN(C(C2(CCN(C)C)CC2)=O)C1)=O C1(C(=O)NC(CNC(C(C(C)C)NC(C)=O)=O)(C)C)CN2CCCN1CC2 N1(C(C2C(C)(C)NC(=O)C2)=O)CC2(COC(CNC(C3(O)CCSCC3)=O)C2)C1 c1(CNC(=O)NC2CCOC(C)(C)OC2)cc2cc(Br)ccc2cn1 c1(C(=O)NC2(CCNC(C3CCCCS3(=O)=O)=O)CC2)ccc2c(c1)CNC2=O N1(C(c2ccc(C)c(CO)c2)=O)CCC(C2CN(C(c3ncccc3F)=O)C2)C1 C(CCN=c1[nH]cnc2ccsc12)N(C(C(C(C)(C)C)NC(N)=O)=O)CCO C#CC1CCCC(C(=O)NCC2CCCCN(C(C3(CO)COC3)=O)C2)C1 C1(CC(N2CCC(CC)C2)=O)C2CCCC2N1C(=O)Cc1ncccc1C C1(CC(=O)NCC(C)NC(c2cccnc2SC(F)F)=O)CC2CCC(C1)C2 CC1CCCC1CC(N1CC(O)(CNC(C2CC2(C)C(F)F)=O)C1)=O Cc1coc(C)c1C=CC(=O)Nc1cccc(CNC(=O)C(=O)N(C)C)c1 N1(C(c2ccc(C)cn2)=O)CC2CCCC2C1C(N1CC2C(C1)C2(C)C)=O C(=O)(C1CCOc2c(F)cccc21)N(CCCNC(c1cc(F)n(C)n1)=O)CC c1(C(N2CCC(N(C(C(C=C)c3ccccc3)=O)C)C2)=O)ccc(CC)cn1 c1(C(=O)NC2CC(CO)N(C(C3CSC3)=O)C2)cnc2[nH]nc(O)c2c1 c1(C(=O)NCCCC(C)NC(c2cccn2C)=O)noc2ncccc12 c1(C(C)=O)ccc(OCCC(=O)NCC2CCC2NC(c2ncoc2C)=O)cc1 C(=O)(C(C)CC(F)(F)F)NCC1C2CN(C(Cc3cc(OC)c(Cl)cc3)=O)C1C2 C1(n2cc(CNC(C(C)O)=O)nn2)CN(C(=O)CC2CSC2)CC1S(C)(=O)=O C1(NC(=O)CN2CC3CC3C2)CC(N=c2[nH]nc(-c3ccccc3)s2)C1 N1(C(C(=O)NC(C)C)C)Cc2cc(Br)ccc2CC1C C1(NC(CCNC(=O)CO)=O)CN(C(=O)CC2CCCC23CC3)C2CCCCC12 C(=O)(C(F)C(F)(F)C(F)(F)F)N(CCOCCNC(C(C)OCC#C)=O)C c1(CN2C(C(=O)NCC(=O)NCC(F)(F)F)CC(OC)C2)ccc(F)c(Cl)c1F c1(OC)c(C(=O)NC2CC(NC(c3cncnc3C)=O)C2)cccc1Br N1(C(CCS(=O)(=O)NC)=O)CC(NC(c2nnc(S)n2C)=O)C2(CCOCC2)C1 c1(OC)ccc(S(=O)(=O)N2CC(C)CC2C(=O)Nc2ccccc2CC#N)cn1 c1(C(=O)NCC(C2CCC2)NC(C(C=CC)O)=O)ccc(C2CCC2)nc1 Cc1cccc(C(N2CCC(NC(=O)CCc3cnc[nH]3)CC2C2CC2)=O)c1N CCC(C)CCCCC(=O)NC(C)CCC(=O)NCCN(CCCF)C c1(OC)ccc(Cl)c(C(=O)NCC2CC2NC(c2cnn(C)c2C(C)C)=O)n1 C1(NC2(c3n(Cc4occc4)nnn3)CC3(CC3)C2)CC2(C1)CC(O)C2 c1(C(=O)NC2(C)CCCN(C(C3(C)CC(F)(F)C3)=O)C2)ncc2c(F)cccn12 C1(C(=O)NC(C#C)CC)C(O)CCN1C(=O)C(O)CN1CCCC1 c1(C(=O)NC2CC3(CC(NC(CC(C)OC)=O)C3)C2)cc2c(nc1O)CCSC2 C(CC(C)C(=O)NC1CC1NC(=O)Cn1nc(C(F)F)cc1C(F)F)=CC C1(NC(C(COC)N(C)C)=O)CC(O)CN(C(c2cc(NC3CC3)ncc2Cl)=O)C1 Cc1cccc(C(=O)NCC2N(C(=O)C3=C(Cl)CCC3)CCC2(C)C)c1F N1(C(C)C)C(=O)COCC1C(=O)NCCN(C(=O)CSC)Cc1ccc(Cl)nc1 C1(COC)CCN(C(=O)C=CC(C)NC(=O)CN2CSCC2=O)C1(C)C N1(C(CN2C(C)CCC2)=O)CCC(C(=O)NC2CCCNC2=O)C(C)(C)C1 CC1CCC(CNCC2(N)CC(O)C2)C1 N1(C(c2c(COC)cco2)=O)Cc2n[nH]cc2C1C(=O)NCCC1CC1C1CC1 N1(C(c2ncc(CC)[nH]2)=O)CCN(C(C2CC2c2ccc(Br)cc2)=O)CC12CC2 N1(C(C2C(C3C(C)C3)C2)=O)CCC(C2CCCN(C(=O)C=CC3CCCC3)C2)C1 Cc1ccc(CCC(N2CCN(C(c3cc(Cl)cnn3)=O)C3CC23)=O)c(C)c1 C1(OC)(CNC(c2ccnc(CO)c2)=O)CCN(C(C2(C)CCC(C)C2)=O)C1 C1(C(=O)NC(C2CCCCC2)CNC(C(C=C)C)=O)CCS(=O)CC1 c1(NC(=O)NC(CC)C(=O)NC(c2cccnc2)C(C)C)ccccc1C N1(C(C=C(C)C(C)(C)C)=O)CC(CNC(=O)C(C)OCC2CC2)C(O)C1 c1(NC(C2N(S(c3cnc(N(C)C)s3)(=O)=O)CCC2)=O)ccc2cnccc2c1 c1(C(N(C(CNC(COCCC)=O)C2CC2)C)=O)n[nH]c2cc(C)ccc12 c1(C(N2CCC(OCCNC(C=COCC)=O)C2)=O)ccc2ccc(C)cc2n1 c1(C(C)=O)ccc2cc(NC(CN(C(=O)NC(C)(C)C)CCN)=O)ccc2c1 C(C)(C)(CCC(=O)NC1CCC2CC12)NC(CN(C)CC)=O C1(C(=O)NCC(C)NC(CN(C(=O)OC)C)=O)COCCO1 N1(C(C(C)NC=O)=O)CC(C)(C(=O)NCCN2CCC3CC23)CC1(C)C C(c1ccc(F)c(Cl)c1)=CC(=O)NC1C(NC(c2c(C)ccc(Cl)c2)=O)CC1 CCCCCC(CC)C(=O)NC1CC12CC(NC(C13COC(CF)(C1)C3)=O)C2 N1(C(Cc2cc(C)sc2C)=O)CCC(CO)C(NC(=O)CC(C)C(F)F)C1 C1(C)(CNC(CCCNC(C)=O)=O)CCN(C(C2OCCC2(C)C)=O)C1 Cc1cc([N+](=O)[O-])c(C)cc1C(N1CCCC(OC(=O)C2=NNC(=O)CC2)C1)=O C#CCC(C)(CNC(C1N(C(C2C=CCCC2)=O)CCC1(C)C)=O)CO C=CCC(C)(C)C(=O)NCC1CCN(C(=O)COc2ccccc2O)C1(C)C C1(NC(c2c(C)[nH]cc2)=O)CC2(C1)CC(C(N1CCC13CCCC3)=O)C2 CC(C)(CNC(C1CC2(C1)CC21CC1)=O)CC(=O)NCC(O)CCO c1(C(COC(=O)CCc2nc[nH]n2)NC(=O)OC(C)(C)C)ccccc1 c1(OC)ccc(CNC(=O)CN2CCN(C(=O)Cn3ccccc3=O)CC2)c(C)c1 N1(C(Cc2nc(C)oc2)=O)CCC2CC12C(=O)NCc1cn(C)cn1 c1(C(N2CCN(C(CN3C(=O)CSC3)=O)C3C2C3)=O)cc2n(c(=O)c1)CCS2 c1(C(=O)NC2CCN(C(c3c(C)[nH]nc3Cl)=O)CC2O)coc(S(N)(=O)=O)c1 C(=O)(C(C)(C)COCc1ccccc1)NCCC(C)NC(=O)CC12CCCC1C2 c1(OC)cccc(=NC(=O)CCC2CCCN2C(C2CN(C)C2)=O)[nH]1 c1(C(N2C(C)(CNC(CSc3c(C)cccc3)=O)CCC2)=O)ccc(Cl)c(O)c1 CCC(C)C(=O)C(=O)NCC(C1CC1)NC(=O)CCc1ccccc1O c1(C(C)(C)C)cnc(C(N2CC(CNC(=O)CCC3CCCO3)C3CC23)=O)cn1 C1(CC(=O)N(CCC#C)CC)CN(C(=O)CC2CCC(C)(C)C2)C(C)(C)C1 C1(C(=O)NCCC(C)SC)(CC)CCCN1C(C1COCOC1)=O N1(C(CSCC#C)=O)CCC2(CCC(NC(=O)C3=CCCC3)C2)CC1 C1(C(=O)NC2CCC(CNC(=O)CSC3CC3)C2)CCCCCCC1 c1(C(N2CCN(C(c3cc(Cl)ccc3Cl)=O)C3(CC3)C2)=O)ccc2cncn2c1 N1(C(CSCCC)=O)CCC2(CC(C(N3CCCC3C(=O)OCC)=O)C2)C1 C#Cc1ccc(Cl)c(C(=O)NCCCN(C(c2csnc2OC)=O)CC)c1 C12(CNC(c3c[nH]c(C)c(Cl)c3=O)=O)CCC(CC1)N(C(C1CC1C(N)=O)=O)C2 N1(C(CCC=C=C)=O)CC(NC(=O)CC2=CCCC2)CCC1C CC(=O)CCCC(=O)N1CCC(C(=O)NCC(C)CC2CCCC2)C1 N1(C(C(C)(C)CC(F)F)=O)CC2(CCCCN(C(=O)CCc3ncc[nH]3)C2)C1 C1(NC(c2cc(CCC)on2)=O)CC(O)CN(C(=O)CCc2cncc(C)c2)C1 COn1cnc(C)c1C(=O)NCCC1(O)CCN(C(=O)C(c2csc(C)n2)=O)C1 C1(C(=O)NC(C2(O)CCN(C(C=C(C)C(C)C)=O)C2)C)CC2(C1)NC(=O)NC2=O c1(C(=O)NCC2(NC(c3c(C)cno3)=O)CCCCC2C)nccc2n[nH]cc12 N1(C(C(CC#CC)NC(c2noc(C3CC3)c2C)=O)=O)CCOCC(C)(O)C1 C1(CCC)CN(C(C2CCC(C#N)CC2)=O)CCN1C(C1CC(=C2CC2)C1)=O c1(OC(CC(C(F)(F)F)SC)=O)cc(OC(F)F)c(F)cc1[N+](=O)[O-] CC1CC(NC(=O)Cn2ccnn2)CCN1C(c1csc(-c2ccncc2)n1)=O c1(OC)cccc(C(C(=O)N2CC(C(C)(C)O)(CNC(=O)C(C)C)C2)C(C)C)c1 CCC(CC)(CC)C(=O)N1CC2CC(NC(C3CCCCN3C(N)=O)=O)CC1C2 C1(CNC(Cc2c(C)nc(C3CC3)s2)=O)CCN(C(c2csc(O)n2)=O)C12CC2 C1(NC(c2c(C(C)C)n[nH]c2)=O)CC(NC(=O)CCC2CCCC(=O)N2)CC1O C1(CC)CN(C(c2cnc(Cl)c(C)c2)=O)CCN1C(=O)NCCCl c1(SCCC(=O)NCC(CN(C(C(C)OCC#C)=O)C)O)nc2ccccc2s1 c1(C(N2CC3C(NC(Cn4c(C)cc(C)n4)=O)C3C2)=O)ccc(Cl)cc1N(C)C c1(OC)cc(C(=O)N(C)CCOCCNC(=O)C(C)C2CCCO2)ccc1OC c1(NC(C2(C)CCN(CCN)CC2)=O)c[nH]c2cccc(F)c12 c1(C(N2CC(O)CC2C)C(=O)NCC)cccc2c1COC2=O FCCCN=C(NCCc1ccccc1F)NCCN1CCCCCCC1 S(=O)(=O)(c1ccc2c(c1)CCO2)Nc1ccccc1.C1(OC)CN2CC1C2=O C(=O)(CCCCNC(C1CCOC1CNC(=O)CCCC1CC1C)=O)NC C(=O)(C(O)CC(C)(C)C)NC1CC2C(NC(c3c(C)cco3)=O)C2C1 c1(COC)nc(=NCC(C2CC2)NC(=O)Cc2cc(F)c(F)cc2F)s[nH]1 N1(C(C(CC)N2CCCC2=O)=O)CC2CCCC(C1)N2C(c1cc(C)sn1)=O N1(C(CN2C(C)CCCC2)=O)CC(=O)NCC1C(=O)N(C)CC1(O)CN(C)C1 C=C(C)CCC(=O)NC1C=CCN(C(c2cc(C(F)F)ncn2)=O)C1 C1(CNC(N2CCC(NC(=O)OC(C)(C)C)C2(C)C)=O)CN(C)CCN(C)C1 CC(C)(CC#N)C(=O)N1CCN(C(=O)COc2ccc(Cl)cc2)C(CF)C1 N1(CC(=O)OC)CCN(C(=O)Cn2cc(C(F)(F)F)nn2)CC1.C(CC(=O)N)S N1(C(C#CC)=O)CCOC2(CCCN(C(c3cc(Br)cc4[nH]ccc34)=O)C2)C1 c1(C(=O)Nc2ccc(C)c(N(C)C)c2)coc2c1CN(C(=O)CC1CC1)C2 Cc1ccc(CN(CC(n2cnnc2)=O)N(CCCO)C)cc1.C1(C=O)CCCO1 c1(OCC)ccc(CC(=O)NC2CC2CNC(c2cncn2C)=O)cc1OC c1(CC(=O)NCC(C(C)C)NC(CC(C)OC)=O)cnc2c(C)cccn12 C1(C(=O)NC2(CC(N3CC(C(=O)NCC)C3)=O)CCCCC2)CC(=O)NC1(C)C n1(CCC(=O)OCCOC23CC4CC(CC(C4)O2)C3)ccc2cc(Cl)ccc12 N1(C(C=Cc2cnc(OC)nc2)=O)CCNc2ncc(C)cc21 C=CCCC(C(=O)N1CCCCC1CC(N)=O)NC(C1OC2CCC1C2)=O c1(CN2CCC(C)(C(=O)NCc3ccc(OCCBr)cc3)C2)cn2ccccc2n1 c1(NC)cc(C(=O)NCCCN(C)C(C2CCC(OC)C2)=O)cc(Cl)n1 CC(C(=O)NCC1CC(C)N(C(c2csc3c2CCCC3)=O)C1)C(C)S(C)(=O)=O Cc1cccc(CCC(=O)NC(C)CCCCNC(=O)CC2CC(C)(C)CO2)c1 c1(C(N2C(CNC(c3c[nH]c(=NCC=C)s3)=O)CC2)=O)cc2c(cn1)CCCC2 C(=O)(CCCCCN=[N+]=[N-])NC(CSCC)C(=O)NC(c1ccccc1)C c1(C2(C(N(CCN(C(C(C)OCCC#C)=O)C)C)=O)CC2)ccc(Br)o1 C#Cc1cccc(C(=O)NC2CCCN(C(C3CCC(=C)CC3)=O)C2)c1Cl C1(F)(CNC(C(C)NC(N)=O)=O)CCN(C(=O)Cc2cccc(Cl)c2Cl)CC1 c1(CN2CC(NC(=O)CNC(=O)C3CC3)C(F)C2)ccc(O)c(Br)c1 Cc1nnc(O)c(C(N2CC(CNC(c3ccn(CC#N)n3)=O)C2)=O)c1C c1(C(N(CCC(C(C)C)NC(C2CCN(C)C2C)=O)C)=O)ccn2c1CSCC2 C1(OCC)CC2(C1)CC2NC(=O)C(CCF)NC(=O)CC1(C)CC1 C(C(=O)N(CCNC(=O)C=CC(C)=O)C1CC1)OCC CN1CC(CC(N2CCCCC2C2(NC(=O)CS(C)(=O)=O)CC2)=O)C(O)C1 C1(C(C)C)CN(C(C2(F)CCC2)=O)CCCN1C(=O)Cc1coc2ccccc12 N1(C(CCCC)=O)CCCC2(NC(c3cn(CCO)c(=O)nc3O)=O)CCCC12 C1(NC(c2scc(CNC(C3C(CCC)CCC3)=O)c2)=O)CN(C)C(=O)C12CC2 c1(C(N2C(CNC(COC)=O)CCC2)=O)ccc(-c2ccccc2C)cn1 n1(C2(CNC(=O)NC(C(=O)OC)C)CC2)cc(Cl)cn1 c1(OC)ccc(NC(=O)Cc2ccc(N(C)C(=O)N(C)C)cc2)cc1Cl C(CN=c1cc(NCN2CCCCC(O)C2=O)nc(C)[nH]1)(C1CCCC1)OCC S(=O)(=O)(c1ccc(-c2nnc(C)o2)cc1Cl)NC(c1ccnc(C)n1)C C(CCC(C)C)(C(=O)N1CC(CO)C(O)C1)NC(COCC(=C)C)=O CC1=C(C(=O)NCC2CCN2C(C2CCC(C(C)(C)C)CC2)=O)S(=O)(=O)CCO1 N1(C(=O)OC(C)(C)C)CCC2(CC(NC(=O)Nc3cc(Br)ncc3Cl)C2)C1 CCCN(OC)C(=O)C1C(NC(=O)C(c2ccc(C)o2)C)C1(C)C N1(C(c2c(SC)c(F)ccc2)=O)CCN(C(c2nnc(O)nc2O)=O)C2CCC12 c1(C(N2CC(C)C(CNC(c3ccc[nH]3)=O)CC2)=O)cccc(N=S(C)(C)=O)c1 Cc1nc2ccccc2cc1C(N1CCN(C(C2SCCCS2)=O)CC(O)C1)=O c1(C(NOCCCOC)=O)ccnc(CNC(c2cc[nH]n2)=O)c1 N1(CC(=O)NC)CCN(C(=O)NCCCc2nc(C(C)(C)C)no2)CC1 C1(C(=O)NCC2(CC(=O)OC)CC2)CN(C(=O)CCS(C)(=O)=O)CC12CC2 c1(OC)cc(-c2ccc(Cn3nnnc3N3CNC(=O)CC3C)cc2C)ccc1C N1(CC(N2CC(CNC(C3CC(CC)OCC3)=O)(OC)C2)=O)OC(C)(C)CC1=O c1(CC=C)ccc(CS(=O)(=O)NOCC#N)cc1 C(CN=C(NCCSC)NC1CC1C)NCCCC C1(NC(C)CCN(C)C(=O)OC(C)(C)C)CCOC1CC(N)=O C#CC1CCC(CNC(C2(CO)CCN(C(C3CCOC3C(C)C)=O)C2)=O)CC1 c1(NC(C(=O)NC(CCC)CCc2ccccc2)=O)ccc(Cl)c(C(F)(F)F)c1 N1(c2snc(COCC)n2)CCN(C(=O)C(C(C)C)NC(C)=O)CC(O)C1 N1(C(c2c(C)ccnc2Cl)=O)CC=C(CCNC(c2cccnc2C)=O)CC1 C1(N(C(=O)COC(C)CC)CCC)CCN(C(=O)CCCSC(C)(C)C)C1 c1(CCC(N2C(CNC(C=C)=O)C(C)CCC2)=O)ccc2ocnc2c1 C(c1ccccc1)=C(CC)C(=O)NC1(C)CN(C(=O)Cc2nncn2C(C)C)C1 CCCCC(CNC(=O)CCOC(C)=O)NC(C12CC(C#N)(C1)C2)=O C1(C(=O)NC2C(NC(CC3(OCC)CCC3)=O)C2)CN2CCC1(C)CC2 C1(NC(C(CCC2CC2)NC(=O)Cc2ccsc2)=O)CC2CCC(C1)S2 C1(NC(C2C(C)CC2)=O)CC2(C1)CC(C(N1C3CSCC1C3)=O)C2 C(=O)(C(F)CC(C)(C)NC(=O)CN(C)CCOC)NC(c1ccccn1)CC N1(C(c2cc(CCC)on2)=O)CC2(C(N3CC(O)CCC3C)=O)CCC1CC2 C1(NC(C(C)N(CC(C)CNC(C23CC(C)C2C3)=O)C)=O)CCCCCC1 N1(C(CC2CCC(=O)NC2)=O)CC2CCC(NC(=O)C3=C(Cl)CCCC3)(C2)C1 C(CCC(C)(C)C(=O)NCc1cnc(F)c(C)c1)NC(C(CSC)C)=O Cc1sc(CNCCN2C(=O)CNC2=O)c(Br)c1C N1(C(C2N(CC)CCC2)=O)CC(NC(=O)CCc2cccnc2Cl)CC(C)(C)C1 C=CCC(CC=C)C(=O)NC1CCN(C(=O)C(C)CCCOC)CC1C c1(C(=O)NC(CC(N2CCN(CC)C(C)C2)=O)(C)C)cc2ncccc2[nH]1 Cn1cc2ccc(NC(C3CC3NC(c3cc4cccn4cn3)=O)=O)cc2n1 c1(CC)[nH]nc(Cl)c1C(=O)NCC1CCC(NC(=O)CC2CN(C)C2)C1 c1(CC(C)NCC(=O)Nc2cc(Br)ccc2N)ccccc1[N+](=O)[O-] Cc1sc(C(=O)N(C2CCCCC2N(C(=O)C(c2cncnc2)C)C)C)nc1O Cc1nc(C(N2CCCCC2CCCNC(C2(C)CC(C#N)C2)=O)=O)cn1C N1(C(C23CC(C(=O)Nc4nccc5cc[nH]c45)(C2)C3)=O)CC2CCCC2C12CC2 C1(NC(CC(C)N(C(c2c(C)oc(CO)c2)=O)C)=O)CN2CCC1(C)CC2 n1(CC(=O)NC2CC(NC(C3(C(F)F)CCCO3)=O)C2)nc2ccccn2c1=O N1(C(Cc2ccn(C)n2)=O)CC2CC1CC2CNC(C1C2COCC12)=O C(=O)(C(C#N)C(C)(C)C)NC12CN(C(c3ccc(CCN(C)C)cc3)=O)C(C1)C2 C1(NC(N2CC3(CCN(C)CC3)C2)=O)CCCN1NC(=O)C1=CC(C)(C)C1 CC1(CNC(=O)CN2CCCNC2=O)CCC(NC(C2CC(CC3CC3)C2)=O)C1 C1(C(=O)NCC23COC(CO)(C2)C3)CCC2CCCCC2C1 c1(OCC(=O)N(CCCCCNC(C2CC2C#N)=O)C)cccc2cccnc12 C#Cc1cccc(CC(N2CCN(C(=O)CCCC(C)C)CC2CC)=O)c1 c1(CN2CC(NC(C(=O)OCC)=O)C(F)C2)cc(I)ccc1OC CC1OC(C)(C)OC1(C)C(=O)N(CCCNC(c1cn(C)nc1C(F)F)=O)CCO C(=O)(C(C)(O)CC(F)F)OCCOCCNC(C(C)NS(C)(=O)=O)=O N1(C(C2C(NC(C=CC3(C)COC3)=O)CCC2)=O)CCC2CCC(O)C1C2 N1(C(C(c2ccccc2)OC(C)C)=O)CC(O)CC1C(N1CCC(N(C)C)C1)=O N1(Cc2ccc(N(C)C)nc2)CCCC(O)(CNC(c2cccnc2Br)=O)C1 C(=O)(C(CC(C)C)NC(=O)NCC(C)C)N1C(CNC(C2(CC)COC2)=O)CC1 c1(C(=O)NC2CN(C(c3scc(C)c3C)=O)C(C)C2)cc[nH]c(=N)c1[N+](=O)[O-] C1(NC(C2C(C)(C)CCCC2)=O)CC1C1CCCN(C(C2CC3CCC2C3)=O)C1 Cc1ccc(N(C)C(c2ccc(CNC(C3CC4(C3)CC4(F)F)=O)s2)=O)cc1C C1(NC(C(C)(O)C2CCC2)=O)COC2C(NC(c3cccc(=O)o3)=O)COC12 C(=O)(C(C)(C)C(C)NC(c1cc(=O)cc[nH]1)=O)NCC1(OC)CCC1 n1(CC(=O)NC(C)C(C)NC(=O)CCC(C)(C)C#N)ccc2ccccc2c1=O C1(CCCNC(COCCC#C)=O)CCN(C(=O)COCC2(C#C)CC2)CC1 N1(C(CCN(C(C(C(C)C)SCC)=O)C2CC2)=O)CCCC2COCC12 c1(C(=O)NCCC(C)NC(Cn2ccc(C)cc2=O)=O)cc2cc(F)ccc2[nH]1 C1(c2nc(CCSC)nn2-c2c(C)noc2C)CC12CCOc1ccccc12 c1(C(=O)NCCC(=C)CNC(=O)CN2CC3CC3C2)ccccc1S(C)=O C1(C(N2CC(OC)C2)=O)C=CCN1C(=O)CCc1ccc[nH]1 c1(C(N(C(c2cccnc2)CC)C)=O)nccc2c(C)cccc12 N1(Cc2cnc(OC)nc2)CCC2(CC2C(=O)NCc2cc(Cl)nc(Cl)c2)C1 C(=O)(CCCC(C)(C)C#N)NCC1N(C(c2c(C)n(C)nn2)=O)CCC1 N1(C(C(C)=C(C)C)=O)CCOC2(CCC(NC(=O)CC(C)(C)O)CC2)C1 c1(CC(=O)NC2(N(C(C(C=CCCC)O)=O)C)CC2)cccc(OC)c1F N1(C(CCC(=C)C)=O)CC2(CCCC(CNC(=O)CC3CCN(C)C3)O2)C1 CC1CCN(C(C2(n3cccc3)CCCC2)=O)CC1NC(C1CCCO1)=O C1(C(N)=O)CCCC1NC(=O)Cc1csc(NC=O)n1 c1(C(=O)NCC(C)CN(C(=O)C(F)(F)c2cncs2)C)ccc2oc(O)nc2c1 C(C)(CCN=c1[nH]c(=NC(C)Cc2nccn2C)c2cc(F)cc(F)c2[nH]1)SC C1(NC(CCC=CC)=O)CCCC12CCN(C(c1ccc(N)c(SC)c1)=O)C2 C1(CNC(c2cc(CC)[nH]n2)=O)CCN(C(=O)Cc2ccc(F)cc2)CC1(F)F C1(N(C(C(C)=CC2CC2)=O)CCO)CCCN(C(=O)C(c2cccc(C)c2)O)C1 Cc1cccc(-c2nccnc2OCC(=O)NCC2CN(C)CCO2)c1 c1(NC(C2C3CN(Cc4ccc(C(=O)O)cn4)C2C3)=O)cc(Cl)cc(Cl)c1F N1(C(c2ccc(C(C)C)s2)C(=O)NCC=C)CCN(CC(=O)NC)CC1 C1(CCC)(NC(C2CC(C)(C)CO2)=O)CCCN(C(=O)Cc2nc(=N)[nH][nH]2)C1 N1(C(CCSCCC)=O)CCN(C(c2c[nH]ccc2=O)=O)CC(CO)C1 N1(C(CC(CCC)C)=O)CCC=C(C(=O)N2CC(OC)C(CO)C2)C1 Cc1ccc2c(C(N3CCN(C(=O)CSC4CC4)C(C4CC4)C3)=O)c[nH]c2c1 CCCC(C(=O)N=S(C)(=O)c1cn[nH]c1)NS(C)(=O)=O C1(CNC(CCN(C(CCC)C)C)=O)COCC1NC(c1nnsc1C)=O N1(C(C=CC=CCC)=O)CCCC1(CNC(=O)CC1CCOC1C)CC CC(CC(=O)NCC1CN(C(C2C3CC4C(C3=O)C24)=O)C(C)(C)C1)C(C)(C)C c1(C(N(C)CC2(O)CCN(C(C3C(CC)C3)=O)C2)=O)cnc2c(cnn2C)c1 CC1CN(C(=O)CCF)C(C)CN1C(=O)CN(C)S(N)(=O)=O c1(C(=O)NCC2CCN(C(CC3C(C)OCC3)=O)C2)sc(=N)[nH]c1C1CC1 N1(C(C2C(CCC)CN(C(C3CCCO3)=O)C2)=O)CC2(CCCCCC2)C1 C1(C)(CC)CN(C(C2CC23CC(NC(C2C(C)C2C)=O)C3)=O)CCO1 C1(NC(C2CCC(C)C2)=O)CCN(C(=O)C(C)N(C)C(C)=O)C12CC2 C(=O)(CCCC(F)F)N1CC(C(C)NC(=O)CSc2cnn(C)c2)OCC1 C1(C(=O)NCCCC(CCC)NC(=O)CC=C(C)C)CCN(S(=O)(=O)NC)CC1 c1(CC(=O)NCC2C(C)(C)CN(C(=O)CC3CC3)C2)ncn2c1COCC2 CCC(C)(C)C(O)C(=O)N(C)CCC1CCCCN1C(c1ccc(C(C)=O)[nH]1)=O N(C1CCc2ccccc21)C(C(CCCNC(C(CO)OC)=O)O)=O C1(CNC(C=C(CC)CC)=O)CN(C(c2ccc(F)cc2C)=O)CCC1(C)C n1(CC)cnc2nc(=NCc3ccc(C#N)o3)[nH]c(NCCCC3CCOC3)c12 c1(NC2CCC(NC(C3(NC)CCCCC3)=O)C2)cccc(NC(C)=O)c1 c1(OC)ccc2[nH]c(C(N3CCOCC3CNC(=O)CC3C=CCC3)=O)cc2c1 c1(OC)c(C(=O)NC23CC2CN(C(C2CCOC2)=O)C3)cnc2ccccc12 CC1OC2(C)CC1(C(=O)NCC1CC(NC(C3CCS(=O)(=O)CC3)=O)C1)C2 CC1C=C(C(=O)NCC2CCCN2C(=O)CCCn2ccccc2=O)CC1 c1(C(=O)NC2C(NC(C3(F)CCCN(C)C3)=O)CCC2)cc(N)cc(O)c1F C1(C(=O)NCc2cc(C)c(C)o2)CCN(C(C2(C)CCCCO2)=O)CC1C C1(C)(NC(C(c2csc(-c3ccccc3)c2)C)=O)CCCN(C(=O)NC2CC2)C1 C1(N(C(=O)Cc2cnn(C)c2)CC)CCCN(C(=O)Cc2cc(C)on2)CC1 N1(c2nc(SC)nc(Cl)c2)CCN(C(=O)C2=COCCO2)CCC1C CC1CC2(CCO1)CC2C(N1CC(NC(=O)C(C2CCC2)C2CCC2)C1)=O c1(NC(COC2CC(NC(C3(C(=O)NC)CCC3)=O)C2)=O)cccc(Cl)c1 N1(C(C(C)(C)OCC)=O)CCC(CNC(C2CC2C(C)(F)F)=O)C(CC)C1 C#CCC(O)C(=O)N1CC2CC2(CNC(=O)CNC(=O)C(C)(C)C)C1 CCC(CNC(C1(C)CC1C(F)(F)F)=O)N=c1ccc(C(F)(F)F)n[nH]1 C1(CCNC(CN(C)CCO)=O)CC(F)(F)CN1C(c1csc(C2CC2)n1)=O c1(OC)cc(C=CC(=O)NC(Cn2cc(-c3cn[nH]c3)nn2)CC(C)C)ccc1O C1(CC(=O)NC2CCCC2NC(=O)COC2CCOC2)CCC2(CC1)CCC2O c1(C(N(C2CCOCC2)C(C)C)=O)ccc2c(c1)CC(=O)NC2 c1(C(=O)NCC23C(CN(C(C4(C)CC(C)C4)=O)C2)C3)cc2c(ccn2C)s1 C(=O)(C(C)(C)C(C)(C)C)N1C(CNC(C2CC(OC)C(OC)C2)=O)CC2CC21 C1(C(N(CC(CC)NC(c2ccccc2O)=O)CC)=O)C(F)(F)C12CCC2 c1(C(=O)NC23CCC(n4cc(CC(C)O)nn4)(CC2)C3)cc2cc(F)ccc2s1 c1(C(=O)NC2C(CNC(c3cccc(CN(C)C)c3O)=O)C2)c(F)ccc(F)c1Cl C1(CC(=O)NCc2c(C(N3CC(COC)C3)=O)nco2)C=NN(C)C1=O C(=O)(C#CC1CCCCC1)N1CCC(C(C)NC(CC(COC)(C)O)=O)CC1 C1(CNC(=O)CCc2ncc(-c3ccccc3)o2)NCC12CCOCC2 CN1C(=O)CCC1C(=O)NC(C)(C)CN1CCN(C(C2(F)CCCOC2)=O)CC1 C1(NC(=O)OCC2(NC(=O)OC(C)(C)C)CC2)CCP(C)(=O)CC1 c1(C(N(CCC)CCNC(=O)CCC2CCC(C)O2)=O)cc(C)[nH]c1C CCN(CC(=O)NCC1CC1)N1CCCCC(C)(F)C1 C1(CNC(C=CC(CC)C)=O)CN(C(=O)CC(F)(F)CC)CC12CCC2 CC1CCCc2nc(S(=O)(=O)N3CCC(CN(C)S(=O)(=O)N(C)C)CC3)cn21 c1(C(N2CC(NC(CS(CC)(=O)=O)=O)C(O)C2)=O)coc2cc(F)cc(F)c12 CCC(C)C(O)CC(=O)NN(C(=O)CCc1ccc(OC2(CO)CC2)cc1)C c1(CCC(=O)NCC(C)NC(CC2(C=C)CC2)=O)ccc(C(F)F)cc1 c1(CC(=O)NCC(CC=C)NC(C2(n3cnnn3)CC2)=O)ccc(C)c(Br)c1 c1(C(=O)NC2CC(NC(C3CCCS3)=O)C2)ccc([N+](=O)[O-])cc1F c1(CN(c2ccccc2)C(CNC(C)(C)CC(N)=O)=O)ccc2c(c1)OCO2 C#CC(C(C)C)NC(=O)Cn1cc(CNC(c2cc(C(N)=O)c[nH]2)=O)nn1 C12(C(N3CCC(CC)C3)=O)C(NC(C3OCCCC3(C)C)=O)C3CC1C2C3 c1(C(=O)NCC(CCNC(C2CC23CC3)=O)OC)cc(C(C)=O)cnn1 C1(NC(Cc2c(C)n[nH]c2C)=O)CN(C(C2CSC2)=O)C2(CCC2)C1 c1(C(N2CC(CC(C)NC(C(F)OC)=O)C2)=O)nc[nH]c1C(F)(F)F C1(NC(c2ccoc2C(F)(F)F)=O)CCN(C(c2cccc(F)c2Cl)=O)CC1O Cc1cccc(C)c1OCC(=O)N(C(C)CNC(C1CCC(=O)CC1C)=O)C N1(C(C(CC)O)=O)C(CC(=O)Nc2ccc(N(C)C)c(F)c2)C2CCCC12 C=CCC(Cc1ccccc1)C(=O)N1CC(NC(=O)C=CC2CCCC2)C(O)C1 Cc1c(NCCc2ccc(F)c(Br)c2)nc[nH]c1=NCC1CC(C)(C)OC1(C)C c1(CCC)c(C(=O)NC(C2CCOC2)CNC(=O)C=CCOCC)nnn1CC c1(CC)ccc(CC(=O)N(C(C)CNC(C2CCCN(S(C)(=O)=O)C2)=O)C)cc1 C1(COC)(NC(c2cc(C)co2)=O)CN(C(=O)C(C)SC)C1 c1(N(CCCN(C(C(CC)C(C)O)=O)C)C)nc2cc(Cl)cc(Cl)c2o1 Cc1cc2c(C(=O)NC3COCC3CNC(C3(C)CCNC3=O)=O)nccn2n1 C12CCN(CC1)C2=O.n1(CC)cc(C(=O)NC2(C)CC2C)nn1 O=C(C1=Cc2ccccc2OC=C1)NC12CC(C1)N(C(c1cnsn1)=O)C2 C(C(CCC)C(=O)N(C)Cc1cc(CC)no1)NC(C1(CC=C)CCCCC1)=O N1(C(c2c(C)nccn2)=O)CCCC2(CCN(C(c3c(O)cccc3F)=O)C2)C1 CN1CCN(C(=O)Cc2ccc(C#N)cn2)C(c2cn(Cc3ccno3)nn2)C1 C(=O)(C1=CCSC1)N1C2CCC1C2.c1(C(N(C)C(C)=O)=O)ccn(C2CCCC2)n1 C(CCC(O)CO)NC(CCN(CC=C)C(C1CCC2(CC2)C1)=O)=O CCCC(C(=O)NCCC1CCN(C(C2CSCCS2)=O)CC1)OCC CCC(C)CC(C)CNC1(c2ccccc2Br)CCC1 c1(OC)ncnc(OC)c1NC(C1(C#N)CCN(C(=O)CCc2ccco2)C1)=O c1(C(N2C(CNC(C=Cc3n(CC)ccn3)=O)CC2)=O)ccc2nc(S)[nH]c2c1 CC1C(NC(c2cc(Cl)ccn2)=O)CCCN1C(c1ncc(Cl)nc1Cl)=O CC1CCC(F)(C(=O)NC2CC(NC(=O)COc3ccc(Cl)c(Cl)c3)C2)CC1 C1(C(=O)NC(C2CN(C(C3CCC(CO)CC3)=O)CCO2)C)CCCCCC1 C1(NC(C=C(C)C(C)C)=O)CCCCN(C(C2COC(C)C2)=O)C1 C1(C(=O)NC2CC3CC(NC(c4cc(C)nnc4)=O)C2C3)CCc2nnnn2C1 CC(C)CC(C(=O)N(C)C(c1cnn(C)c1)C)ONC(=O)C1(F)CCC1 c1(CC(C(=O)OCC)NC(c2ncoc2CC(C)C)=O)ccc([N+](=O)[O-])cc1 N1(C(C2C(C)OCC2)=O)C2CCCC1CN(C(c1cc(Cl)cc3c1CCC3)=O)C2 N1(C(C2C3(CCN(Cc4c(OC)cccc4Br)C3)C2)=O)C2CCC1CN(C)C2 c1(C(N2CCC(N(C(=O)CSc3nccn3C)C)C2)=O)nnn(C)c1N CC1=C(C(=O)N2CCC(C)C(NC(c3cnc(C)cn3)=O)C2)CCCO1 C1(N(C(C2CCC(NC(CC(C)(C)SC)=O)CC2)=O)C)CCOC(C)(C)C1 C(C(C)(C)CC(=O)N(CC(C)O)CCNC(c1cnccc1C)=O)OC(C)=O N1(C(CSC(C)(C)C)=O)C2CCC1C(CNC(=O)CC(F)(F)Cl)C2 C1(N(C(C(C=CC)O)=O)C)CN(C(c2cn3ccsc3n2)=O)CC1(C)C CC1CCCn2cc(C(=O)NC3CCCC3CNC(=O)CCOCC3CC3)nc21 CCCC(CCCO)C(=O)NCC1(C)CCN(C(C23CCCN(CCC2)C3)=O)C1 CCCCC(CC)CC(=O)N1CC(C)C(C)(CNC(C2(CC)CCOCC2)=O)C1 c1(C(=O)NC2CN(C(CCCC)=O)CC(O)CC2)cc(S(=O)(=O)CC)cnc1O N1(C(=O)NCCCOC)CCC(C)(NC(C2CC(OC)C2)=O)C1 C=C=C(C)CC(=O)N1CCCC(N(C(=O)C(c2ccnn2C)C)C)C1 c1(OC)ccc(F)c(CNCCC(N)=O)c1Cl C1(NC(CCC(=C)C)=O)CC(F)CN(C(C2(CCC)CCNC2=O)=O)C1 CC1CN(C(c2cc(C(F)(F)F)cc(F)c2)=O)CCC1NC(=O)CCC(F)(F)F n1(C(C)C)nc(C2CC2)cc1C(=O)SC1(O)CC(C(=O)OC(C)(C)C)C1 C1(C(=O)NC2C(NC(c3ccc(C(C)=O)o3)=O)C2)CCCN1N=O C(CC(C)(C)C(=O)NCC(C)(CC(C)C)NC(=O)CC1CCCN1C(C)C)OC C=CCC(CC)C(=O)NC(C)(CNC(=O)Cc1ccn(CC)n1)C1CC1 N1(C(CCOCC#C)=O)CCN(C(=O)C(CC)n2cccn2)C(CC(=O)OC)C1 CCC(C)(C(=O)N(C)CC1CCCCN1C(=O)COCc1ccc(Cl)cc1)OC N(C1CCCc2c(I)n[nH]c21)CC1N(S(C)(=O)=O)CC1 C12(C(=O)NCC(=C)CCNC(c3ccc(CN(C)C)o3)=O)CCC(CC1)C2 c1(CNC(C2(OC)CCOC2)=O)ncc(C(=O)NCC2CCC2(F)F)cn1 c1(OC)ccc(I)c(NC(=O)Nc2ccc(CCO)c(F)c2)c1 N1(C(C(=O)Nc2cccc(-c3ncco3)c2)=O)CC2C3CCC(C3)C2C1 c1(OC)ccccc1C(CNC(=O)Cc1cnoc1)NC(c1nc(OC)c(C)s1)=O Cc1ccc2[nH]c(C(=O)NC3COC(c4ccccc4)C3)c(Cl)c2c1 C(=O)(C(CNC(=O)C(C(C)C)OCC)C(C)(C)C)NC(CCCC)CO C1(NC(C(CC)O)=O)CCS(=O)(=O)C12CN(C(c1cnn3c1OCCCC3)=O)C2 C1(C(N(C2CN(C(c3ccc(Cc4nccs4)cc3)=O)C2)C)=O)CCC(C)CC1 c1(CNC(CC(C)(F)F)c2nnnn2C2(C)CC2)cc(Cl)nc(Cl)c1 N1(C(c2cc(C)c(C)o2)=O)CCC2(COC(CNC(C3CC3C)=O)C2)C1 Cc1ccc(C=CC(=O)NCCCNC(=O)CC2CCC2)c(C)c1 c1(N(CC)CC)cc(Cl)ccc1C(=O)NC1CCC(NC(=O)C2CC2)CC1 C12(C(N3CCC(O)(C(C)NC(=O)CCC=CBr)C3)=O)CCC(CC1)OC2 C#CC1CN(C(=O)COC(F)(F)F)CCN1C(=O)C(F)=CCC CC1(C)CC(CCNC(=O)CCN(C(C2SCCS2)=O)C2CC2)CO1 c1(COC)cccc(C(=O)NC2CC(CNC(C3(CC)CC(=O)C3)=O)C2)n1 c1(OC)ccc2c(c1)CC(C)CC2Nc1nccc(N(C(C)CS(N)(=O)=O)C)n1 N1(C(CCC(=O)NCC)=O)CCN(C(C2CC2(C)CC)=O)C(C(C)(C)C)C1 C1(C(=O)NCCCC)CCN(C(=O)CCc2ncc(C)[nH]2)C(C)C1 c1(CNC(C2C(CNC(Cn3ccc(C)c3)=O)CCO2)=O)ncccc1C CCCCC(C)C(=O)NC1CCC1CNC(=O)C(c1cnn(CC(=O)OC)c1)=O CCC(C)C(CNC(C1(C)CCCN1C(=O)C(CC1CCC1)OC)=O)CO C1(N(C(CC2(C=C)CC2)=O)C)CN(C(=O)C(F)C2CCC2)CCC1C C(C)(C)(CC(=O)NCC1(C)CC(NC(=O)CC2CCOC2=O)C1)SC C1(CCCNC(CCN(C)CC)=O)CCCCN1C(c1nccn1C)=O CC1N(C(C2CC(F)CCN2C(=O)CN(C2CCC2)C)=O)CCC1(C)C CCC(CC)CCC(=O)NCC1(CN(C)C(c2cc(O)n(C)n2)=O)CC1 N1(C(c2ccc(CC)o2)=O)CCCCCC(NC(C2(C#N)CC(C)C2)=O)C1 N1(C(C(N2CCC(C)C2)=O)=O)CC2CCC(CNC(=O)CC3CSC3)(C2)C1 N12CCCC1C(=O)NC(C)CNC(=O)C2.c1(CO)cscc1C(F)F c1(CCC(=O)NCC(CNC(CCSC)=O)F)cnc2n1CCOC2 c1(C(=O)Nc2scc(-c3ccc(SC)s3)n2)ccc2c(c1)C(=O)CCC2 n1(CC(N2CC(NC(Cc3c(C)non3)=O)C(C)C2)=O)ccc2c(C)cccc12 Cc1nc(=N)[nH]cc1C(=O)NCc1cn(C2CCN(C(C3CC3Cl)=O)CC2)nn1 C1(CC(=O)NCC(CNC(=O)CC2CS(=O)(=O)C2)CO)CCCCCC1 CC1(C)CN(C(c2coc(CO)c2)=O)CC1CNC(=O)CC1CCCCCCC1 C1(OC)CCCN(C(C2CCN(C(=O)Cc3ccc(F)cc3)C(C)C2)=O)CC1 Cc1nc(CCC(=O)NCCN(C(C2CCCN(C(N)=O)C2)=O)C(C)C)oc1C c12cc(n[nH]1)C(=O)NC2.C1(COC)OCCC1C(=O)NOCC(C)(C)C Cc1cncc2cc(C(=O)NC(CNC(c3cnc(C(C)C)[nH]3)=O)C(C)C)sc12 c1(C(N2CC(C)C(NC(=O)COC(F)F)C2)=O)c(OCOC)ccc(F)c1N CN1CCC(CNC(=O)C(C)(C)C2(N)CCC2)C1 C1(CC)CN(C(=O)COC2CCN(C)CC2)CCN1C(=O)COCC1CCOC1 C=CC(CC)CC(=O)NCC(O)C(=O)NCCN1CC2CC2C1 CC(C(=O)NCC1(NC(c2n[nH]c3ccc(O)cc23)=O)CC1)C(C)S(C)(=O)=O N1(C(C=CC)=O)CCCC(C(C)NC(=O)C(COc2ccccc2)OC)C1 c1(C(=O)NC2CCC(C(=O)NC(C3CCOCC3)C)C2)cc(Br)ccc1O c1(CNC(=O)CCN(C)C(C)C)cccnc1.C12(CC1)C(=O)NC2.CC(C)C1CC1 C1CC2(CCCN(c3nnc(C)o3)C2)C1.c12ccc(cc1)SCC(=O)N2C.CO CC1=C(C(=O)NC2CC(NC(c3cc4ccc(F)cc4o3)=O)C2)CCS1(=O)=O C1(NC(c2c(C)cc(N)cc2)=O)C(C)CN(C(=O)CCN(S(C)(=O)=O)C)CC1C c1(C2(C(=O)NCC#CCNC(C3C(C)OCC3)=O)CCC2)ccc(Br)cc1 Cc1oc(C(=O)NCCC2CCCN(C(=O)CC3CCCCC3O)C2)cc1CO Cc1cnn(C)c1C(=O)NC1CNCCC1C C1(NC(c2cc(CC)on2)=O)CCN(C(c2cocc2C)=O)CC1C(C)C N1(C(C=CC=CC)=O)CC(n2cc(C(C)(C)C(N)=O)nn2)C(C)C1.[SH](=O)C(=O)C C1(CC(=O)NC(CNC(C2C(C(C)=O)C2(C)C)=O)(C)C)CCCCC1(C)C c1(C(=O)NC2CN(C(COC)=O)CC(C)C2)ccc(P(C)(C)=O)s1 C1(C(N(CC(=O)NCCN2CCNC2=O)CCOC)=O)CCN(C)C1=O c1(CC)cn2c(C(=O)NCC3CN(C(c4cc(Br)c[nH]4)=O)CCO3)cccc2n1 n1(CC)nc(C)c(C(N2CCOC(CNC(c3sc(C)c(C)c3C)=O)C2)=O)c1C c1(OC)ccc(C)cc1C(=O)NCC1(O)CC(CNC(=O)C(C)C#N)C1 c1(C(=O)NC2CC(NC(C3(C#N)CCCC3)=O)CC2O)c(F)ccc2n[nH]cc12 c1(C(=O)NC(CNC(C(C)NC(C)=O)=O)(C)C2CC2)ccc(C#N)c(O)c1 N1(C(C(CC2CCOCC2)NC(C2C(C)CCO2)=O)=O)CCC(CO)C(C)(C)C1 N1(C(Cc2ccc(C)o2)=O)CC(NC(=O)CC2(C)CC2)C(c2ccccc2)C1 N1(CC(=O)NCC23CC2CN(C(c2ccc(C(N)=O)s2)=O)C3)C(=O)CNC1=O c1(C(=O)NCC2CN(C(c3c(C)cco3)=O)C2)cc2n(n1)CCCCC2=O C1(CC(=O)N(C)CC2COCCN2)CC2(C1)CC(F)(F)C2 CC(c1cccs1)=CC(=O)NCC(N1CCN(C(=O)CC2CCC(O)C2)CC1)=O C#Cc1cccc(C(=O)NC2CCC(C(=O)NCc3ccc[nH]3)CC2)c1 c1(C(=O)NC2CCCCC2NC(c2coc(O)n2)=O)cnc2c(c1)NCC2 c1(C(=O)NC(C(C)NC(Cc2c(C)nsc2)=O)CO)c(C)nn(CCO)c1C C(C1CCCO1)=CC(N1CC(CNC(=O)CSC2CC2)C1)=O c1(CC)ccc(NC(C2CCN(C(=O)OC(C)(C)C)CC2)CO)nc1 CC1COCCC1N(C)C(C1(C2CCCN2C(c2c[nH]ccc2=O)=O)CC1)=O N1(C(c2c(N)nccn2)=O)C2CCC1CC(CNC(=O)CC1CCCCC1O)C2 C(=O)(CCCC(C)(C)C)NCCN(C(c1cc(C(N)=O)[nH]n1)=O)CC N1(CC(=O)NCCCN(C(=O)COCC2CCCO2)C)C(=O)CNC1=O c1(OC)ccc(C(=O)NC2CC(CNC(=O)Cc3cnccn3)C(O)C2)cc1F c1(CCNC(CC2N(C(C(COC)O)=O)CC2)=O)ccccc1C C1(C(C(=O)N(CC2(CNC(C3C(C)CN(C)C3)=O)CC2)C2CC2)O)CCS(=O)(=O)CC1 C(C)(C(=O)NC1CN(C(c2cc(C3CCC3)on2)=O)C1)(C(C)C)OC C12(NC(CC=C=C)=O)CC1CN(C(=O)C(c1ccc(Cl)cc1)C1CC1)C2 CC1CCN(C(C2CC3(CC3)C2)=O)C1CNC(=O)CCF C1(C(N(CC(C)O)CCNC(=O)CSCc2cccs2)=O)CN2CCN1C(C)C2 C(=O)(C1=CCN(C)C1)NCc1occ(C(N(CC(C)CO)C)=O)n1 N1(C(COCC)=O)CCC(C)(C)C(NC(=O)CC(C)(C)c2cccs2)C1 c1(-c2ccc(CCCC)s2)ccn2nc(C(=O)Nc3sccc3C(C)=O)cc2c1 C(=O)(C(C)(F)C(=O)NC1CN(C(c2ccc(N(C)C)cc2F)=O)C(C)(C)C1)OC O=C(C1CCCc2nccn21)NCCc1cn(-c2cc[nH]c(=N)c2)nn1 n1(CC(=O)NC(CNC(CC(C)C(F)F)=O)CO)nnc2ccccc12 N1(C(C2CCC(C)N2C(c2ccn(C(C)C)n2)=O)=O)CCNC(=O)CC1C CC1C2CN(C(=O)C(O)CNC(C3CC4(CC4)C3)=O)CC12 c1(C(=O)NCCOCCC)conc1CNC(c1ocnc1C)=O C(=O)(C1Cc2ccc(Cl)cc21)NCC1C(NC(c2nc(Cl)cs2)=O)CC1 c1(CC(C)C(=O)NCC2CCN2Cc2nnn(C)n2)ccc(F)cc1 N(C1CCc2ccc(Br)cc21)C(c1scnc1-c1cnc(CSC)cn1)=O N1(C(C(F)OC)=O)CCC(C)(CNC(C2(CO)CCCC2)=O)C1 C(=O)(C1=NN(CC)C(=O)CC1)NC1CN(C(CNC(CC)=O)=O)CC12CCC2 CC1(C)CC(C(=O)N2CCCC(C(N3CC(NC(=O)C4CC4)C3)=O)CC2)=NO1 c1(CC(=O)NCC(CNC(C2C(CC)OCC2)=O)O)cccc(C(F)F)c1 C(CC)(C(=O)N1CC(O)(C(F)C(=O)NCC2(C)CSC2)C1)OCC C(=O)(C(CC(C)CC)NC(c1cc(C)sn1)=O)N1CCC(CCC#C)CC1 CC1CC(CNC(=O)Cc2cnnn2C)CN(C(c2cc3scnc3[nH]2)=O)C1 Cc1cnoc1C(=O)NCC1C=CC(NC(C2(C)CCCO2)=O)C1 C1(NC(N2CCCC(C(C)(F)F)C2)=O)COC2CCCCC12 C1(C(CC)NC(=O)CC2CCCN2C(c2cscc2Cl)=O)CCCN1C(C)=O c1(C(N2CCC(N(C(=O)COC(F)(F)F)CCC)CC2)=O)ccc(=O)n(C)n1 c1(C(=O)NC(CC(C)NC(c2c(SC)cccc2)=O)C)noc(C)c1[N+](=O)[O-] c1(COC(=O)CN2CCC(O)(c3cccc(Br)c3)C2)cc2cc(Cl)ccc2s1 CC1CC(=O)NCC1C(=O)NCCOCCCN(C)C(c1ncc(N)cc1Cl)=O N=c1[nH]c(=NCc2ccsc2)[nH]c(=NC2CC3C(C2)C3(F)F)[nH]1 CC1(C)CCC(CNC(c2cnc(O)s2)=O)N(C(=O)CSCC(F)(F)F)C1 N1(C(C(C)OC(C)=O)=O)CCC(C(O)CNC(C2CC3(CC3)C2)=O)CC1 C1(C(=O)NCC2CCC(NC(CSC(C)C)=O)C2)COC(C)(C)CO1 c1(C(N(C(C)CCNC(=O)Cn2nccn2)C)=O)csc(Cl)c1Cl Cc1cc(N)cnc1C(=O)NCC(O)CN(C(=O)C(C(C)(C)C)NS(C)(=O)=O)C C1(CNC(c2ccc(F)cc2Cl)=O)CCN(c2nnc(C3CC3)s2)CCC1(F)F C(=O)(CCCCN(C)C)NC1(CC=C)CN(C(=O)CC2(n3cncn3)CC2)C1 CC(CC(=O)N1CCC(CNC(c2ccc(-c3ccsc3)cc2)=O)C1)C(C)(C)C C1(C(=O)NC2(C)CC(NC(C(CCCC)C)=O)C2)CCc2nncn2C1 O=C(CC1OCCc2ccsc21)NC1(CF)CCNC1 c1(CC(=O)NC2(CNC(C(CC=C)C(C)C)=O)CCC2)ccc([N+](=O)[O-])c(N)c1 C1(C(N2CC(NC(C34CCC(N)(CC3)C4)=O)C3CC23)=O)CCc2nc[nH]c2C1 CC1CCc2n[nH]cc2C1C(=O)NCC1(C)CCCC(F)(F)C1 Cc1c(C(N2CCC(C)C2CNC(=O)Cc2csc(Cl)n2)=O)cccc1N c1(CC(=O)N(CCCNC(=O)CC2CC(F)C2)C)cn2ccccc2n1 C1(CNC(c2[nH]cc(CC(C)C)c2)=O)CCCN(C(C2CCC(C)CC2)=O)CC1 C(=O)(CCCCC(C)C)NC(CCC(=O)NCC(=O)N(CC)CC)CC N1(C(C(C)CO)=O)CCCN(C(c2ccc(SC(F)(F)F)cc2)=O)CCC1 C1(C(=O)NCCCOC2CCC2)CC2(CCN1C(c1ccccc1)=O)CC2 c12ncnc(c1F)NC1CCC(C1)NC2=O.c1(CC)ccc(N(C)C)cc1 c1(OC)nc(C)ccc1C(=O)NCC(CNC(=O)C(F)(F)C(O)C1CC1)CO C1(CNC(C2(C(C)C)COC2)=O)C2CN(C(c3scnc3C(F)(F)F)=O)CC12 C(c1ccc(Cl)s1)=CC(=O)NC1(CCCNC(C(C2CCOCC2)OC)=O)CC1 C=C1Cn2c(C(=O)NCCC(C)NC(C3OCCOC3C(F)(F)F)=O)nnc2S1 N(C)(S(N)(=O)=O)CC(=O)NC1CC(N(C(=O)CCC2CCCCC2)C)C1 N1(C(C(C2CC2)OC)=O)CC(CC(=O)NCCCc2cc[nH]n2)C2(CC2)C1 C1(NC(C(C(C)NC(C2CC2NC(N)=O)=O)C)=O)CC(C)N(C)CC1C N1(C(C2N(C)C(=O)NC2)=O)CCCC(C)(C)C1CNC(c1ccoc1C1CC1)=O c1(C(C(=O)NCSc2ccccc2)N(C(C=C)C)C)ccnc(OCC)n1 C(=O)(CCS(N)(=O)=O)NC(CN(C(c1cc(OC)cc(Cl)c1)=O)CC)C C=CC(C)(CC)C(=O)N1CCC(N(C(=O)COC2CCCCC2C)CCO)CC1 N1(C(=O)C(F)F)CCC2CC12C(=O)NCc1ccc(F)cc1 CCCCC(O)C(C)C(=O)NCC1CC(C(=O)Nc2ccc(C)c(C#N)c2)=NO1 C1(C(N(CC)CC2(C#N)CCC2)=O)CCCCN1C(=O)CC1(O)CCC1 C1(C(=O)NCCCCNC(C2OCCC2c2ccccc2)=O)(COC)CC1(F)F C1(NC(c2cc(C(C)=O)cn2C)=O)CC(F)CN(C(=O)CC(C)(C)C)C1 C1(NC(=O)C(c2ccccc2)C2CC2)CCCC1C(=O)NCCc1ccsc1 C1(CCNC(C(C)(C)CO)c2n(C3(C)CC3)nnn2)CCCCCC1 C1(C(C)(C)C)(CNC(C(CC)NC(N)=O)=O)CCN(C(=O)CCCC2CC2)C1 c1(OC)ccc(Cl)cc1CC(=O)NCCC1CCCN(C(=O)COC)C1 N1(C(c2ccc(C(C)=O)s2)=O)CCCC(C2CC2NC(c2cnc(CN)[nH]2)=O)C1 C(C(C)C(=O)NC(C(F)(F)F)C1CC1)NC(C(C)NC(=O)C1CC1)=O CC(C)C#CC(=O)N1CC=CC1CNC(=O)C(c1ccccc1)C CC1CCc2[nH]c(=NC(CN3CCc4ccccc4C3)CCO)c(C#N)cc2C1 c1(OC)cc(C(N2CC3CN(C(c4cc(F)cc(I)c4)=O)C3C2)=O)cc(C)c1 c1(C(N(C(C)CNC(=O)CCN2CCOCC2)CC)=O)nccc(N)c1Cl CCC(CC)CCCC(=O)N(CCC(C)(C)NC(=O)C=CS(C)=O)C c1(C(N2C(CC)(CC)CC(NC(=O)C=CC(F)F)C2)=O)cnn2cccnc12 N1(CC(=O)NCCc2c(CNC(=O)CCC3CC3)nco2)CSCCSC1 Cc1ccn2ncc(C(=O)NC3CCCN(C(C4CCOC4(C)C)=O)CC3)c2n1 C=CC1(C(=O)NCCC(CCC)C2CC2)CCN(C(=O)C(C)C(=O)OC)CC1 C1(C(=O)NC2CCC(CNC(c3c(CC)occ3)=O)C2)CCN(CCO)C(=O)C1 C1(NC(C2C(C)C2)=O)CCN(C)C12CCCN(C(c1ccoc1)=O)C2 CN1CC(C)(C(N2CC3CC(NC(c4ccc([N+](=O)[O-])o4)=O)C2C3)=O)CC1=O c1(C(N(C2CCN(C(=O)CC=C(C)C)C2)CCC)=O)ccc2c(c1)CCN2C c1(CC)ncc(Cl)c(C(N2CCC(CCOC)(NC(c3cnc(O)s3)=O)C2)=O)n1 Cc1cc(C(N2CC3CCC(C2)N3C(C2CCCOC2)=O)=O)nc2ccccc12 N1(C(C2NC(=O)OCC2)=O)CC2CCCN(C(c3cc(Cl)c(Cl)s3)=O)C2C1 c1(C(C)OC)nc(-c2nn(C)cc2Cl)n(C2CCC(C)(C)C2)n1 c1(C(=O)NCCC)c(C)[nH]c(C(=O)NCC(C)CN(C(=O)C2=CCC2)C)c1CC C1(CN(C(C(C)(C)C2CCOC2)=O)C(c2cccs2)=O)CCCC12CCC2 C#Cc1ccnc(C(=O)NCC23CC(C2)C(NC(=O)CCNC(C)=O)CO3)c1 N1(C(C=Cc2n(CC)ncc2)=O)CC(C)OC2(CCCOC2)C1 C1(CNC(C(C)Cc2ccnn2C)=O)CC(NC(=O)Cc2cncnc2)CC1O C1(CNC(=O)CCC2CCC2)CC(O)CN1C(=O)CCn1cnnn1 N1(C(C2C(C)N(C(=O)CN3CC4CC4C3)CCC2)=O)CCC2CCN(C)CC12 Cc1nc(N(C(=O)C(C)(C)CCl)CC(=O)NC(=O)CO)sc1I C1(OC)CC2CCC(C1)N2C(=O)CN(C)C(C1CCOCC1)=O C12(C(=O)NC(Cc3cc[nH]n3)C(=O)NC3CCCC(F)C3)C(=O)C3CC1C2C3 C(C1CCOCC1)=CC(=O)NCCNC(C1C(Cl)(Cl)C12CC2)=O C1(NC(C2(O)CCCCC2)=O)CCOCC1C(N1CCC(CO)C1)=O N1(C(C(C(C)C)SC)=O)CC(NC(c2csc(C(C)=O)n2)=O)C2(CCOCC2)C1 C=C(CNC(=O)CC1CN(C(C2C3CCC(F)C23)=O)CC12CC2)c1ccccc1 Cc1cccc2c(C(=O)NCC3CC3NC(=O)C=Cc3ccsc3)coc12 C=CCCC(C)(C)C(=O)N(CC(C)NC(=O)CCC1C(=O)NN=C1C)CC N1(C(c2cc(OC)ncc2)=O)CCC(CO)(CNC(C2C3CCCC23)=O)CC1 c1(C(=O)NC2C(CNC(c3cc(C)sn3)=O)C2)csc(S(C)(=O)=O)c1 C(CCN(C(=O)C(C(C)C)NS(C)(=O)=O)C)(C(C)(C)C)NC(C=CSC)=O C1(NC(CCNC(C)=O)=O)CCCOC12CCN(C(C1CCC(C)O1)=O)CC2 C1(OCC(=O)N(C2CCC2)C)CCN(C(=O)CN(C2CC2)Cc2ccccc2)C1 C1(NC(C2C(CCOC)C2)=O)CCN(C(=O)Cc2ccc(F)cn2)CC12CCC2 CCCC(C(=O)NCC(C)N(C)C(c1cc(OC)no1)=O)N(C)C Cc1ccc(Cl)c(OCC(N2CCOC(C)(CNC(c3scnc3C)=O)C2)=O)c1 C12(CCNC(=O)CC3CCOC3)CCC(CC1)N(C(C1CCCCC1O)=O)C2 c1(C(N(CCNC(C2C(C)(C(=O)OCC)C2)=O)C)=O)sc(CC(C)C)nc1C Cc1ccc(CCC(N2CC(NC(c3nc(O)sc3C)=O)C(C)C2)=O)cc1 C1(NC(CCC#CC)=O)CC(CNC(=O)Cc2nc[nH]n2)C12CCC2 c1(C(=O)NC(CC)CNC(c2ccc(C(C)F)cc2)=O)noc2cc(F)ccc12 N1(CCCC=CC)CCCC(c2cccc(OC)c2)C1 CCC(C(=O)N1CCCC1CN(CC)Cc1csc(Br)n1)NC(C)=O Cn1cnc2[nH]c(=NCC3CC=CC3)nc(N3CCCC(C)(F)C3)c12 CN1CCN(C)CC(C(=O)NC2CCCCC2NC(c2cnc(=N)[nH]c2)=O)C1 CCC(CO)CN=C(NCc1snnc1C)NCC1CCOC1 c1(C(=O)NC)c[nH]c2ncc(-c3ccc(C(=O)N(C)C)cc3F)cc12 N1(C(C2CCN(CC(C)C)C2)=O)CCN(C(c2ccc(N)c(N)n2)=O)C(CF)C1 CC(C)C(CCNC(=O)CSCc1csc(=N)[nH]1)NC(C1CC2CC2C1)=O c1(C(N2C(CN(C(=O)COC(F)F)C)CCC2)=O)cccc2c1OCC(=O)N2 N1(C(C(C)OCCOC)=O)CCC2CCC(NC(c3ncc(Cl)s3)=O)C1C2 c1(CCC(=O)NC2CC(C(C(=O)NC)F)C2)cncnc1 C(c1ccc(C(=O)OC)cc1)=C(CN1CC(C=C)C1)C C1(NC(CNC(C(C)(C)C)=O)=O)CCCCN(C(=O)COC2CCOC2)C1 c1(CC(=O)NCC(C)NC(CC2(COC)CC2)=O)ccc(OC)cn1 N1(C(C2CN(CCOC)C(=O)C2)=O)CCC(C)C(NC(=O)C(C)n2cncn2)C1 c1(OC)oc(C)nc1C(=O)NCC1CCCC1NC(C1CC=CCO1)=O C#CCCCCC(=O)NC(Cc1ccccc1Br)C(=O)N(C)CC1(O)CCC1 C12(C(N(CCCN(C(=O)COCc3cccc(Cl)c3)C)C)=O)CCC(CC1)C2 C1(NC(CCC2(C#N)CC2)=O)CCCC(F)C1 C1(C(N(CCN(C(C(c2ccccc2)OCC)=O)C(C)C)C)=O)COC(C)C1 N(C1COc2cc(F)cc(F)c21)N1CC(C2OCC2(F)F)C1.C1(NC=O)CCCC1 c1(CC(=O)NC2CC(NC(C(CC=C)C)=O)C2)c(C)cc(C#N)cc1C N1(C(C(CC#C)C)=O)CC(C)(C)CCC1CNC(=O)COCCOCCO CC(C)(O)C(C)(C)C(=O)N1CCCC(C(N2CC(O)C2)=O)C1 c1(C(=O)NC2CC(NC(C3C(C=C)OCCC3)=O)C2)cc(Br)cc(C)c1F CC1(NC(c2ccsc2)=O)CCN(C(=O)CC2CCCO2)CC1 C1(CCNC(c2cnnn2-c2ccccc2)=O)COCCN1C(C1CC1(F)F)=O c1(C(=O)NC2C(NC(c3c(C(C)C)con3)=O)CCCC2)nsc2ccccc12 N1(C(C2(COC)CCCC2)=O)CCC(F)(CNC(C2(N3CCOCC3)CC2)=O)C1 C1(C(=O)OCC)C2COC(C(=O)NCC(C)(O)CNC(c3ccncc3)=O)CC12 C1(NC(C2CC(C(=O)OC)C2)=O)C2CN(C(=O)CC(c3c(C)noc3C)C)CC12 C1(NC(=O)NCC2CCN(C)C2)CCc2ncc(Br)n2C1 c1(C(=O)NC(C(=O)NC2CC2O)C2CCCC2)c[nH]c2nccc-2c1 N1(C(C2CCC(CNC(C(C)(F)c3ccon3)=O)CC2)=O)CC2(CCNC2=O)C1 CCC(C)(O)CCNC(C1CCOCC1NC(c1cccnc1C)=O)=O S(=O)(=O)(c1cc(C(=O)NCC(C)N(C(=O)CCCCN(C)C)C)ccc1F)NC N1(C(c2nc(CC)sc2)=O)CCC2(N(CC)CC)CCCC12.C(C1CCC1)=CC=O c1(CC(=O)NC2CC(NC(CCCCC#N)=O)C2)c(F)c(F)c(F)c(F)c1F Cc1nn(C(C)(C)C)cc1C(=O)NC1CCCC1CNC(c1ccncc1N)=O C1(C)(C(N2CC3C(CN(C(C(COC)OC)=O)C)C3C2)=O)CC(=O)N(C)C1 c1(C(N2CC(C)(C(=O)OC)C2)=O)cc(F)ccc1CC(N1CCC1CO)=O CCCC(O)CC(=O)NCC1(NC(c2cc(OC)cnc2F)=O)CCCC1 C(=O)(C(O)CC(F)(F)F)NCC12OCC(C(=O)Nc3c(F)cccc3F)(C1)C2 c1(OCC)ccc(C(=O)NC2CC(C)N(C(=O)CCCN=[N+]=[N-])C2)cc1[N+](=O)[O-] c1(C(=O)NCCCCNC(C(CC)N(C)C)=O)cnn(-c2ccccc2F)c1C N1(C(C2N(Cc3c(C)noc3C)CCOC2)=O)CCC2(CCOCC2)C1 c1(C(N2CCC(NC(c3ccc(SC)o3)=O)C2C)=O)ncc(N)cc1Cl n1(CC(=O)NC(C)C(C)NC(=O)CC2CSCCS2)nnc2ccccc12 c1(C(N(CCOC)CCNC(=O)C(F)(F)C2(O)CCC2)=O)ncc(C#N)cc1Cl Cc1csc(C(=O)NC(C2CCCN2C(=O)CCc2ncc[nH]2)C)c1Cl CC(C)CC(F)C(=O)N1CC(CNC(c2nc(=O)n(C)[nH]2)=O)C1 c1(C(=O)NCC(N(C(CC(CC)C(C)C)=O)C)C2CC2)nc2ncc(C)cn2n1 c1(-c2ccc(NC(c3cc(Cl)nc(Cl)c3)=O)nc2)cnn2ccccc12 c1(CCCC)cc(N2CC3CC2CN3C(C2CC23CC(O)C3)=O)n2ncnc2n1 C12(CNC(C=CC=CC)=O)CC1CN(C(c1nccnc1C(F)(F)F)=O)C2 S(=O)(=O)(c1ccc(C)cc1)N1C(=O)C(CC)N(C(=O)COC2CCNCC2)CC1 C(C1Cc2ccccc21)NC(C(CNC(c1c(C)ccc(C)n1)=O)C)=O Cn1cc2c(n1)CC(C(N1CCC(NC(=O)C=Cc3cn[nH]c3)C13CC3)=O)CC2 C1(C(N2CCC(NC(CCCCC)=O)C(C)C2)=O)CCS(=O)(=O)C1(C)C c1(C(=O)NCCCNC(C2C(C(=O)OC)CCCC2)=O)csc2ccccc12 N1(C(C(C)SCC)=O)CCC(C)N(C(c2cccc(OC(F)(F)F)c2)=O)CC1 CC1(C)CN(C(C2CNCC(F)C2)=O)CCN1C(=O)CCn1ccccc1=O c1(C(N2CC(CNC(C(CC)(C)F)=O)OCC2)=O)cc2c(C#N)c(F)ccc2[nH]1 C#CC1CCC(CNC(=O)CCC2CCCCN2C(=O)C=CCCC)CC1 N1(C(CCC(CC)OC)=O)CCCN(C(=O)CN(c2ccc(Cl)cn2)C)CC1C C(=O)(C1=COCCC1)NC1(C)CC(C(=O)NCC(C)(C)N2CCCC2)C1 C12(CNC(c3c(OC)cccn3)=O)CCC1CCN2C(=O)CCCNC(N)=O N1(C(CC(=O)NCCC)=O)CC(c2cccc(C(F)(F)F)c2)OCC1(C)C Cc1cc(Br)c(C(N2CCCCC2CF)C(=O)Nc2ccccc2)s1 c1(SC(C(=O)NC(CC)CNC(c2[nH]c(C)nc2C)=O)C)nc2ccccc2s1 N1(C(C(C)=CC)=O)CC2CCN(C(c3sc(Br)cc3F)=O)C2C1 c1(C(=O)NC2CC(N(C(=O)CN3CCCC3=O)C)C2)c[nH]c(=O)c2ccnn12 CC(CN=C(NCC1OCCO1)NC1CCCC1)Oc1ccccc1Br CC1CCN(C(c2nccnc2N)=O)CC1CC(=O)NOCc1ccccc1F C(CC(=O)SCCCC)N(C(=O)NCCN(C)C(=O)OC)CC C(=O)(C1CCCc2scnc21)N1CCC(NC(C2CCOCC2)=O)C12CCC2 CCCC(C(O)C(=O)N1CCC(C#N)CC1)NC(=O)CC1CCSC1 C1(CNC(CN(CCOC)C)=O)CN(C(c2cnc(Cl)cc2C)=O)CCC1(C)C c1(CCCNC(=O)C(F)F)ncc(Br)cn1 CN=c1[nH]cc(C(=O)NCC(C)(C2CC2)NC(=O)CCn2cncn2)o1 C1(SCn2cc(C(C)OC)nn2)C(C2CC2)CCN1C(C1CC2C=CC1CC2)=O N1(C(C(n2cc(-c3c(Cl)ccc(OC)c3)nn2)C)=O)CCC(O)C(C)(C)C1 C(CC(C)CC)(C(=O)N1CC(O)CC(O)C1)N(C(CC(CC)OC(C)=O)=O)C N1(C(c2c(CCCCCC)cccc2)=O)CC(CC(=O)OCC)OCC12CC2 Cc1cncc(C(=O)N(C2CCCCC2)CCNC(=O)CC2CC2(Cl)Cl)c1Cl N1(C(CNC(c2ccccc2)C)=O)CC2(N)CC1C2 N1(C(C=CCOC)=O)CC(F)(F)CC1C(N1CC(c2ccccn2)C1)=O c1(-c2nc(CCN(CC(F)(F)F)C)n(-c3ccc(Br)cc3)n2)cc(F)cc(F)c1 N1(C(COCC#C)=O)CC(NC(=O)Cc2ccc(Cl)cc2)CC(C)C1 C1(C(=O)NCC(CO)NC(C2CSC2)=O)Cc2ccccc2S1(=O)=O C(=O)(C1=NOC2COCC12)NCCC(C(=O)NC1C(C)(C)CCC1)O Cc1cc(C)c(C(N2CC(C(C)NC(c3ccc(NC(C)C)cc3)=O)C2)=O)cn1 c1(SC)cccc(CC(N2CC3CC3(CNC(=O)Cc3cc[nH]n3)C2)=O)c1 Cc1cc(C2(C(=O)N(c3cnccn3)CC(=O)NC3CCNC3=O)CC2)on1 c1(NC(C2CC(NCc3ccc(Br)nc3Br)C2)=O)cc(Cl)c(Cl)c(Cl)c1 N1(S(CC(C)C)(=O)=O)CC2CCC1CN(C(c1c(F)ccc(Cl)c1F)=O)C2 C(=O)(C(C)(C)NC(=O)CC(C1CC1)SC)N1CC(NC(=O)OCC)C1 CC(C)C(F)C(=O)NC1CN(CC2CC2NC(c2ccccc2N(C)C)=O)C1 N1(C(c2cccc(Cl)c2Cl)=O)CCCN(C(C23CCN(CC2)C3)=O)CC1CO N1(C(C2CC(CC)NC(=O)C2)=O)CC2CCC(C1)N2C(C1NC(=O)OC1C)=O c1(C(=O)NC2CCC(C(=O)Nc3cnc(Cl)c(Cl)c3)OC2)ccc2c(c1)CCC2 N1(C(COC(C)C)=O)CCCC1C(C)NC(=O)Cn1ccnc1C(C)C c1(CC)c(C(=O)NCC2(NC(C3CC3C)=O)CCC2)sc2ccccc12 C#CCCCCCC(C(=O)NCC)N1CCOCC1CC1CCCO1 c1(C(N2C(CNC(CC(=C)C)=O)CC2)=O)ccc(-c2cccc(OC)c2)nc1O C1(C(=O)NC2CN(C(c3c(C)cn(C)c3)=O)C2)CC2CCCCN2C1 C(C(CC1CC1)C(=O)NCCc1ccns1)NC(c1cc(C)sn1)=O C(N(C)N1CCCC1C)c1ccc(C(C2CCCN2C)=O)cn1.CO C(CCCN(C(=O)CC1CC1CNC(=O)C(C)OC(C)=O)C)OC Cc1ccncc1CC(N1CC(C)(NC(=O)Cn2nccn2)C1)=O C1(NC(c2ccccc2[N+](=O)[O-])=O)CCC2CCN(C(c3sccc3F)=O)C12 C1(CNC(C2N(S(C)(=O)=O)CC2)=O)CCCCN1C(c1cnc(C2CC2)s1)=O O=C1CCCC(C(=O)NC2CC(CNC(c3c[nH]nc3C3CC3)=O)CC2O)O1 C(=O)(C1CS(=O)(=O)c2ccccc21)N(CCNC(C(CSC)O)=O)CC1CC1 CC1CCn2ncc(C(=O)NCC(C)(C3CC3)NC(C3(C4CC4)CCC3)=O)c2C1 N1(C(CCCc2scc(C)n2)=O)CCC(C)(CNC(=O)CN2CC3CC3C2)CC1 C1(C(N(C)CCN(C)C2CC2)=O)(NC(=O)CC2CC2(C)C)CCCCC1 c1(C(=O)NCC2CN(C(CCN(CC)CC)=O)C3C2C3)cc(F)cc([N+](=O)[O-])c1 C1(NC(C2(NC(c3cccs3)=O)CCC2)=O)CC2CC2C1 C(=O)(C(Cc1ccsc1)NC=O)NCCNC(CNC(=O)OCC)=O C12(C(=O)NCCCN(C(=O)C(C)CC3CCCCC3)C(C)C)CCCC(C1)OC2 c1(CC(=O)NCC2N(C(C(n3c(C)ncc3)C)=O)CC=C2)cncc(Br)c1 C1(C(N2C(CN(C(c3c(C)nsc3N)=O)C)CCC2)=O)CCCCCC1(F)F c1(C(=O)NC2CCCC(NC(CC3(C)CCCO3)=O)C2)cn2cnnc2cn1 CC1CCCC(C(=O)NCC(F)(F)Cn2cc(-c3cnccc3C(=O)O)nn2)C1 c1(C(N(CCNC(=O)Cc2ncoc2C)CC)=O)cn(C2CCOC2)nn1 c1(C(N2CCCC(NC(c3ccc(Cl)c(Cl)c3)=O)CC2)=O)c(F)cc(O)cc1F C1(C(N(C(CC(=O)NCc2nc(C)c(C)s2)C)C)=O)CC2(CCC2O)C1 C1(C(=O)NC2CN(C(C3(C(=O)OC)CC3C)=O)C2)CSCC(=O)N1 C12(C(=O)NCC(C)CNC(c3ccccc3C3(C#N)CC3)=O)CC=CC(C1)OC2 c1(C(NNC(=O)NCC)=O)cc(O)ccc1Br C1(CNC(c2c(SC)cccn2)=O)C2CCC(C2)N1C(c1cc(Cl)ncc1O)=O c1(C(=O)NCC2N(C(C(CC=CC)C)=O)CC(C)(C)C2)cncc([N+](=O)[O-])c1 N1(C(CCC(=O)NCCC)=O)CCOC(C)C1C(=O)Nc1ccc(SC)nc1 c1(C(N(CCOC)C)=O)cc2c(C)cc(OC)cc2o1 N1(C(c2ccn3c(O)nnc3c2)=O)CCC2(CC1)CCN(c1cc(Cl)ncn1)C2 c1(CCC(c2n(CCOCC)nnn2)NC(C2CCCC2)C2CC2)ccccc1C c1(CN2CCC(C)(NC(CC(C)C)=O)CC2)cc(Br)c(F)cc1[N+](=O)[O-] C1(CC)CCN(C(=O)C=C2CCOCC2)C1CNC(=O)C(C)n1cncn1 N1(C(C=C2CCC(C)CC2)=O)CCC2(CC(NC(C3OCC4CCCC34)=O)C2)C1 c12ccc(F)cc1N2.CC1(NC(=O)CN2CCCC2=O)CCN(NC(=O)NC=O)C1 CC1ON=C(C(=O)NCC2(NC(=O)CSc3ccc(Cl)cc3)CCC2)C1C c1(C(=O)NCC2N(C(C(C)O)=O)CCC(C)C2)coc2cc(O)ccc12 C1(C(N2CCCC(C(C)C(=O)N(C)C(C)C3CC3)C2)=O)(OC)CCOCC1 N1(C(CC(C=C)C)=O)CCC2CN(C(c3[nH]nnc3COC)=O)CCC12 C1(C(=O)NC2CCCC(C#C)C2)CCCN1NC(=O)C1CCN(C)C1 C1(C(=O)OCc2nnc(C3CCCCC3)o2)OCCOC12CCC2 N1(C(=O)NCC2C(C)(C)C3CCC2C3)CCC(=O)Nc2cc(F)ccc21 N1(C(c2cc(C(=O)OCC)no2)=O)CCC2CCN(C(c3csc(Cl)n3)=O)C2C1 Cc1c(C(=O)NCCC2CCN(C(C3CC(C)CCO3)=O)C2)nn(C)c1Br C1(O)(CCNC(c2c(SC)ccs2)=O)CCN(C(c2cscc2C(N)=O)=O)CC1 C#Cc1cnn(C)c1C(=O)NC1CCOCC1NC(=O)C(C)Oc1ccccc1 N1(C(C2ON=C(C)C2)=O)C2CCC1CN(C(c1cccn1C)=O)C2 c1(OC)cnc(C(N2CCCC2(C)CNC(=O)C(c2ccn(C)n2)C)=O)cn1 C1(OC)CC2(CCC(C(=O)NCC3C4CN(C(=O)CC5(O)CCC5)CC34)CC2)C1 C1(CC)CCCCC1NC(c1n[nH]cc1CNC(c1sncc1C)=O)=O C1(C(=O)NCC2(NC(c3c(F)ccc(OC)c3)=O)CC2)CCC2C(C1)C2(F)F C1(NC(C(=O)NCC)=O)COC2C(NC(c3cnn4c3CCC4)=O)COC12 c1(C(N2CCCC(CN(C(c3c(CC)cco3)=O)C)C2)=O)cc(C)c(F)cc1O C(=O)(C(CC(=C)C)OC)NC(CC=C)C(=O)NCC1(OC)CC1 C#Cc1ccc(F)c(CNC(=O)N(CCCCC(C)c2ccccc2)CC)c1 Cc1cnc(NC(C2CCCN(Cc3cnc(Cl)cc3Cl)C2)=O)c(C)c1 c1(CC(=O)NC2C(NC(CC(=O)NC3CC3)=O)CC2)ccnc(F)c1F C12(CCC1)C(=O)OC2.C(=O)(C(C)O)NC C(=O)(CC(C)(C)CC)N(CC(CC)NC(c1cc(Br)cn1C(C)C)=O)CC c1(C(=O)NC2C(NC(C3(N(C)C)CCCC3)=O)CCC2)cccc2oncc12 CCC(F)(F)C(C)(C)C(=O)N1CC(C(C)NC(=O)COCCc2ccccc2)C1 N1(C(COCc2ccc(C)cc2)=O)CC2(CCN(C(c3cn(C)c(C)n3)=O)C2)C1 C1(NC(C2C(OC)CC2)=O)CCC(CNC(=O)C=Cc2cc(OC)ns2)CC1 C1(C(=O)NCC(C(C)C)(C)NC(=O)C=C2CCSCC2)CN2CCN1C(C)C2 C1(NC(=O)CCSc2ccccc2)CCCCN(C(=O)CC2(CO)CC2)C1 c1(NCC(=O)NCC(CNC(C(C=C)(C)C)=O)OC)ccc([N+](=O)[O-])c(SC)c1 CC1CCCC=C1C(=O)NC(c1cnn(C)c1)C(=O)N1CC(N2CCC2)C1 c1(CCC)ncc(C(=O)NCCC2(CNC(c3nnsc3C)=O)CC2)s1 C#CC1CC2(CC(C(=O)N(C3CCN(C(=O)CN(C)CCO)CC3)CC)C2)C1 C1(NC(C(CC#C)O)=O)CN(C(=O)Cn2cc(C)cn2)CC12CCC2 N1(C(CCC(C)(C)C)=O)CCN(C(=O)CCc2nc3cccnc3[nH]2)CC(O)C1 C(=O)(C1=NOCC1)NCC1(C)CC(NC(c2[nH]ccc2-c2ccccc2)=O)C1 c1(NCCC(=O)NC2C(CN(C(COCCCOC)=O)CC)C2)ccccc1 C1(CNC(c2nc(C)[nH]n2)=O)CCN(C(=O)C(C)OCC(F)(F)F)C12CCC2 N1(C(CCCc2c(C)ccs2)=O)CC(NC(C2COCCO2)=O)CC(C)(C)C1 O=C(N=c1ccnc(N2CCCCC2)[nH]1)c1cc(COc2ccc(Br)cc2)c[nH]1 C(=O)(C(CC(C)(C)C)NC(=O)CC1CCN(C)C1=O)NCCC=C=C N(C1CCC(Nc2ncncc2Cl)c2ccccc21)C(c1c(CC)csc1)=O c1(NC(C(CN(C)C)O)=O)cccc(CNC(=O)Cc2nc(C3CC3)cs2)c1 CC1(NC(=O)CC2CCCOCC2)CCN(C(c2ccoc2)=O)C1 C=CCCCC(C(=O)NCC(C)C)NC(C)=O Cc1cc2sc(C(=O)NCC3CN(C(c4cnc(O)o4)=O)C3)cc2s1 N1(C(C2(COCC)CC2)=O)CCC2CCN(C(C3CC(=O)N(C(C)C)C3)=O)CC12 C(=O)(CCCC(=O)NCC1(C)CCN(C(=O)Cc2ccc(C)c(Cl)c2)C1)NCC N1(C(C2(CC#C)CCCCC2)=O)CC2CCCN(C(=O)CCc3nncs3)C2C1 C1(C(=O)O)CCC(C(=O)O)N(C(c2ccccc2NCC2CC2)=O)C1 c1(CC(C(=O)NCC2CC(NC(c3cnc(C)[nH]3)=O)C2)C)cccc(Cl)c1 C1(NC(CCSCCC)=O)CCC(NC(C2(CC3CC3)CC2)=O)CC1 CC(=O)C(C)CC(C)C(=O)N1CCCC1CN(C(=O)C=Cc1cccnc1)C c1(OC)noc(C)c1C(=O)NCC(CNC(C1CNC(=O)N1)=O)OC O=[N+]([O-])c1cccc(N2CCN(Cc3sc(I)cc3Cl)CC2)c1 C1(OC)CN(C(C2(F)CC(NC(=O)OC(C)(C)C)C2)=O)CC1OC(=O)C1CC1 C1(NC(CCNS(CC)(=O)=O)=O)CCCN(C(=O)CCc2cnccn2)CC1 c1(CC)ccc(C(N2CCC(C)(CC(N3CC(F)CC3CO)=O)C2)=O)nc1 C(CNC(=O)Cc1nccn1C)(CC(=O)NOCCC1CC1)OC C(CCCCC(=O)NC1CCCCC1CO)N(C(C1CCC(CC)O1)=O)C c1(CC)cccc(C(=O)NCC2C(C)CCN2C(C2CCC(O)CC2)=O)n1 C1(C)(CC=C)CN(C(C2COCC2NC(=O)CN(c2ccncc2)C)=O)C1 C1(NC(C2(CC=C)CC2)=O)CCN(C(=O)C(c2ccc(C)cc2)C)C1C1CC1 CCCCC(CC(=O)NCCc1ncccn1)NC(=O)C(C)c1ccsc1 N1(C(Cc2n(C)ncc2Cl)=O)CCC2(CCCN2C(C2CC(N(C)C)C2)=O)C1 C1(NC(CCN(C)CC)=O)CCC2CCN(C(c3nccc(OC)c3F)=O)C1C2 CC(C1=Cc2ccccc2OC1)NC(=NCCF)NC1C(F)(F)C12CCOCC2 N1(C(CC(CC)O)=O)CC2(C1)CN(C(c1cncc(O)c1)=O)C2 C1(C(F)(F)F)(C(N2CCN(Cc3c(OC)cccc3)CC2)=O)CC2CCC1C2 C(=O)(C(CC)CC(C)C)NCCC(C)(C)NC(c1c(CC)ocn1)=O C1(C(=O)NC2CC(NC(=O)CS(=O)(=O)N3CCOCC3)C2)CCC2(CCC2)C1 N1(S(=O)(=O)CCn2cccn2)CC2(CCC2)C1C1CCCO1 CCC(CC(=O)NCC1(C#N)CCC1)NC(C1CC(N(C)C)C1)=O C1(C)(C(=O)NCC2(O)CN(C(c3c(C)onc3)=O)C2)CC2CCC(C1)S2 N1(C(C2C(CNC(C(CC)OC)=O)C2)=O)CC(F)(F)C1C1CC1 C1(CNC(=O)Cc2ccc(CO)cc2)CC2CCC(C1)N2C(=O)Cn1ncnn1 Cc1ccc(C)c(C(=O)NCC(C)(O)CNC(=O)C(C)N2CCCC2)c1N CCC(COC)C(=O)N(CCN(C(C1CCN(C(C)=O)C1)=O)C(C)C)C1CC1 c1(C(N2C3CCN(C(C(CC)(C)OC)=O)C(C3)C2)=O)ccc(Cl)c2ncccc12 C#Cc1ccnc(C(=O)NC(C2CCN(C(=O)Cc3ccc(C)cc3Cl)C2)C)c1 N1(C(C=CC(=O)OCC)=O)CCC(C(=O)N(C(C)C(C)CC)C2CC2)CC1 C1(CNC(C(c2ccc(S(=O)(=O)N(C)C)cc2)C)=O)CCCN1S(=O)(=O)N(C)C C(CCCC(C)NC(=O)C(C)N(C)C)NC(CCCC)=O.C1(=O)CC(C)CN1 C1(NC(c2n(CC=C)ccn2)=O)CCN(C(C2CCC(N(C)C)CC2)=O)C(C)C1 C12(NC(CC(C)(C)SC)=O)CCC(CC1)N(C(=O)COCC(C)C)C2 Cc1c(-c2cc(C(=O)N(CC(O)CN(c3ccncn3)C)C)no2)cnn1C CCC(C)C(O)C(=O)N1CC(O)(C(C)NC(=O)Cc2c[nH]ccc2=O)C1 C1(C(N(C)CC2COCCO2)=O)CCOCCN1C(=O)CN1CCOCC1=O C(=O)(C1Cc2ccccc21)N1CCCC(NC(c2c(C)nc(O)s2)=O)CC1 N1(C(C2C(CC(C)C)C2)=O)CCC2(CC2NC(=O)CC2CC(F)(F)C2)C1 CCC(C(=O)NCC=C1CCN(C(c2ccc(C)c(F)n2)=O)CC1)C(C)C c1(C(=O)NCC2(F)CC(NC(C(COC)(C)C)=O)C2)ccc(C)cc1Cl C1(CCC=C)(C(=O)NCC(C)(C)C)CN(C(C2CCC3CC23)=O)C1 C(=O)(C1=NOC2COCC12)NC(C)(CO)C(N1Cc2cncnc2C1)=O c1(NC(=O)Cn2cc(CNc3ccc(C(=O)O)cc3)nn2)cccc([N+](=O)[O-])c1 N1(C(COC(=O)Cc2ccc3ncsc3c2)=O)CCCc2ccccc21 c1(COC)onc(C(=O)NC(C)(CNC(=O)COCC2CCC2)C2CCC2)c1C C=CC1(C2(C(N3CC4CC3CN4C(=O)CCCOCCC=C)=O)CCC2)CCC1 C(=O)(C(C)(C)C(C)NC(c1occ2c1CCC2)=O)N1CCC(CCOC)C1 c1(N(C)CC2(OC)CCSCC2)ccc(S(=O)(=O)NC(c2cnccn2)C)cn1 CCCC(O)CC(=O)NC1CCCC(NC(c2cccc(C)n2)=O)C1 c1(C(N2CCN(C(C3CCCS3)=O)CC2CF)=O)ccc2c(n1)CCC2 c1(C(=O)NCc2sc(C(C)=O)c(C)n2)ccccc1S(=O)CC(O)CC C1(NC(C2CCC(=O)NC2)=O)CCC2CC1CN2C(=O)Cc1cc(F)ccc1F C(=O)(CC(C)CC)N1CCC(C(=O)NC(CCC)C2CC2)C1 C1(NC)CCC12CCN(C(=O)COCC(N1CCCC1)C)CC2 c1(N(C)Cc2ccc(Cl)s2)nc(=NCC(C)Oc2ccccc2)[nH]c2ncn(C)c12 C12(NC(C(C(C)(C)C)NC(c3cc(C)oc3)=O)=O)CCC(CC1)C2(C)C c1(C(N2CCN(CCN(C(CCCC)=O)C)CC2)=O)[nH]c2c(c1C)C(=O)CCC2 c1(OCC)cccc(CCC(=O)NC(C)CCN(C(=O)C2=COCC2)C)c1 N1(CCCCNC(c2cnc(C)s2)=O)CCCN(C(C2(C)CC(C)(C)C2)=O)CC1 C1(NC(C2CC=C(C)CC2)=O)CN(C(c2ccc([N+](=O)[O-])cn2)=O)CCC1(C)C N1(C(C(CC#C)O)=O)CCN(C(=O)CSS(C)(=O)=O)C(c2cccc(OC)c2)C1 C1(CC(=O)NC(c2ncc[nH]2)C)CCN(C(=O)C(C)CC2CC2)C1 c1(CC(=O)N(CCOC)CCNC(c2ccc(C(C)C)s2)=O)sccc1Cl C1(CC(=O)NCCN(C2CCCC2)C(C=CCOC)=O)CC2(CC2)C1 c1(-c2c(C(N(C3CN(C(=O)C#CC(=O)N(C)C)C3)C)=O)nco2)ccccc1F CN1CC(CNC(=O)CC2CCC(NC(=O)CN3CCC(=O)CC3)C2)CC1=O O=C(CC1C(=O)Nc2ccccc21)NCC(F)CNC(c1ccsc1)=O c1(C(=O)NC(C2CCN(C(C(C)C)=O)C2)(C)C)cccc2cccc(O)c12 N1(C(c2ccc3nccnc3c2)=O)CCC2(CCCN(C(C3CCO3)=O)C2)C1 N1(c2ncc(C(=O)OCC)cn2)CC2(CCN(C(c3cccc(F)c3Br)=O)C2)C1 C(=O)(CS(=O)(=O)CCO)N(CCC(C)NC(C1(CC)CCCC1O)=O)C c1(-c2c(C)cc(OC(C)C)nc2)c[nH]c2cc(NCc3nccn3C)ccc12 N1(C(C(C)=CC2CC2)=O)CCC(NC(C2OCCC2C(F)(F)F)=O)C(O)C1 c1(C(N2C(CNC(c3c(COC)cc[nH]3)=O)CC(OC)C2)=O)cn(C)c(C)cc1=O N1(C(c2c(CNC(C34CC(C(C)C)(C3)C4)=O)nnn2C)=O)CC2CC(C)C2C1 CCCCC(O)C(C)C(=O)NC1(C)CN(C(c2ccc(CC)nc2C)=O)C1 N1(C(CCCOCC=C)=O)CC2CCCC2C1C(N1CCCOC(C(C)C)C1)=O C1(COC)CCC(NC(c2cnc(C)s2)C(=O)NCC2CCOCC2)CC1 Cc1[nH]c(C#N)cc1C(=O)NCC1CCCN(C(C2CCOC2C)=O)C1 N1(S(CC(=O)OCC)(=O)=O)Cc2[nH]nc(-c3ccc(C(C)C)cc3F)c2C1 N1(C(CN(CC(C)(C)C)C)=O)CCN(C(c2cc3[nH]ccc3s2)=O)C(C(F)F)C1 N1(C(CCC=C(C)C)=O)CCN(C(c2ccnn2CC2CCC2)=O)C(C)CC1C CCCCC(O)C(C)C(=O)N1CC(C(N2CCCC2CC)=O)(CC)C1 c1(CC(N2CCN(C(CSCC)=O)C(CCCC)C2)=O)cccc(S(C)(=O)=O)c1 C1(C(NOC(c2ccncc2)C)=O)N(C(=O)CSC2CC2)CC12CCCC2 C1(C(N2CCC(N(CCC)C(C3CC(OC)(OC)C3)=O)C2)=O)NC(=O)NC1=O N1(C(CCN(CCC)C)=O)CCN(C(c2ccoc2C)=O)C2(CC2)C1 Cn1nc(C(N2CCC(CNC(=O)CC(C)(C)O)C2)=O)c(Cl)c1Cl C(C(C)(O)CC(=O)NCC1CC2(CC(NC(=O)C(C)SC(C)C)C2)C1)OC c1(C(=O)OC2CCSCC2)cccc(CN(C(=O)COC(=O)NC(CC)C)C)c1 c1(C(=O)OC)cc(F)c(C)c(S(=O)(=O)N2CCOC3CCN(C)CC23)c1 n1(CC)cc(C(N2CC(CCNC(=O)C=CC(C)(C)SC)C2)=O)c2ccccc12 C12(SC)CN(C1)C(=O)C1(C)CCN1C2.C12(C(=O)OC(C)(C)C)COCC1C2 N1(C(CC2N(C(c3cc(C)sn3)=O)CC(C)(C)C2)=O)CCC(O)CC(C)C1 CCCCCC(C(=O)N1CCCC1CCCNC(C1CCC(F)(F)C1)=O)C(C)C c1(C(N2CCCC2CC(=O)OC)C(=O)NCCOCC)cn(C)nc1C CC1CC(CNC(=O)C2=CCOCC2)CCN1C(C1CCC1c1nncn1C)=O c1(OCOC)ccc(F)cc1-c1cnc(F)c(C(=O)NCc2ccccn2)c1 C(CC1=CCOCC1)NC(C(CC1CN(C(c2c(C)scn2)=O)C1)F)=O C(=O)(C(C)S(=O)(=O)C(C)C)NC1C2CC(CNC(C=CC)=O)(C2)OC1 C1(O)(CNC(c2cncc(N(C)C)c2)=O)CCCN(C(C2CCCNC2=O)=O)C1 c1(C(N2CCC(NC(c3cn(CC)nn3)=O)C2)=O)cccc[n+]1[O-] N1(C(CC(C(=C)C)C)=O)CCC2(CCC2NC(c2ncc(F)cn2)=O)CC1 C(=O)(N=c1[nH]c(Cl)ncc1C)C1(C)CCN(C(c2cnc(C)[nH]2)=O)CC1 c1(N2CC(C)CC(C)C2)ncc(S(=O)(=O)NC2(CO)CC=CC2)cc1Cl N1(C(C=C(C)C(C)C)=O)CCOC2(CCN(C(=O)C=Cc3cc[nH]c3)CC2)C1 c1(C(N(C2CCOC2)CC)=O)ccc(C(C)C)c(Cl)c1 N1(C(CC(c2ccns2)C2CCC2)=O)CCN(C(F)F)CC1.c1(CC(=O)O)ccoc1 c1(N2CCOCC2)ccc(Cl)cc1C(=O)NC1C(OC)CNC1 c1(NC2CCC(NC(=O)Cn3nccn3)C2)ncc2[nH]cc(I)c2n1 C=Cc1cc(C(=O)NCC2CCCCCN2C(=O)Cc2cccn2C)cc(F)c1 n1(C(C)C)ccc(C(=O)NCC2CC2NC(C2CCC(=O)N2C2CC2)=O)cc1=O c1(C(=O)NCC2N(C(c3[nH]cc(CC)c3)=O)CCCC2)n[nH]c2ccc(C)cc12 N(C1CCC(NC(=O)COC(F)(F)F)c2ccccc21)C(c1c(C)nccc1)=O S(=O)(=O)(CCCOc1ccc(C(F)(F)F)cc1)NC(C)C(C)(C)c1ccccc1 CCC(C)C(O)C(C)C(=O)NCC1(C)CCCN1C(=O)CN1CCCNC1=O c1(-n2cc(CCC(=O)NC3(C(=O)O)CC(C(=O)OC)C3)nn2)cccc(Br)c1 C1(C(N2CC(O)(C(=O)OC)C2)=O)CCN(C(=O)CC2CCCC23CC3)C1(C)C N1(C(C2C(CCOC)C2)=O)CCCC1(C)CNC(=O)CCCn1cc(C)cn1 Cn1nnc(CN2CC(c3cn(CC(=O)OC)nn3)(C(=O)O)C2)c1C(F)(F)F.C(F)F c1(C(=O)NCC2C(NC(C(C)n3cncn3)=O)COC2)ccc2c(c1)OCC2 Cn1nccc1C(O)C(=O)NCC1COCC1NC(c1cccs1)=O c1(C(=O)NC(CCCNC(CC(=C)C)=O)C)cc(S(N)(=O)=O)c(C)s1 c1(COC)ccc(C(=O)NC2CCCC2NC(=O)CCOC2CCCC2)s1 c1(C(N(C2CCN(C(=O)CCCC)CC2)CCCC)=O)ccc(F)c(OC)c1 N1(C(C(CCOC)NC(=O)CSC(C)C)=O)CCCC(C)(OC)CC1 c1(C(=O)OCC(=O)N(C(C)(C)C)CCC#N)ccn(C2CC2(F)F)n1 C1(COC)CN(C(=O)C(n2cc(C)cn2)C)CCN1C(c1cscc1C)=O C=CCCCC(C(=O)Nc1ccc(Cl)c(C)c1)NC(C1CC(CC2CC2)C1)=O Cn1ccc(CC(=O)NC2(CNC(=O)CCSCc3ccccn3)CC2)n1 CC(C)(C)C1=NOC(C)(C(=O)NC(c2ccccc2)CNC(=O)CC2CCC2)C1 c1(NC(CC2CCCN(C(C(C)(C)Br)=O)C2)=O)nc2cc(Cl)ccc2s1 C1(NC(CCC(CC)C)=O)COC2CN(C(=O)CCc3ccnc(C)n3)CC12 C1(C(N(CCC(N)=O)C(c2ccccc2)C)=O)COCCN(CC(F)(F)F)C1 CCCCCC(O)CC(=O)N(C)CCNC(c1cccc(C(F)F)n1)=O c1(C(=O)NC(C2(C(=O)NC(C3CCCO3)CO)CC2)C)cccc(C#N)c1 C(CCC(C)(c1nnnn1C(C)CC)NCC(C)Cc1ccccc1Cl)OCC C1(NC(c2cn(C)nn2)=O)CN(C(C2CCC2(C)C)=O)CCC12CCC2 CC(C)C(CNC(c1cccc(C2CC2)c1)=O)C(=O)N1CCC(F)(C#N)C1 C1(C(=O)NCCCOCCNC(c2snc(C)c2N)=O)CC(=O)NC(=O)N1 c1(OC)ccc(C(N2CC(NC(=O)NC(C)(C)C)C3(CC3)C2)=O)c(C)n1 c1(C(N2CCN(CCNC(CS(CC)(=O)=O)=O)CC2)=O)cnn2cccc(C)c12 c1(OC)cc(C(=O)N(CCNC(=O)C(C)NC(C)=O)C(C)C)cc2cnn(C)c12 C1(NC(C)=O)COC2(CCN(C(=O)C(C)O)CC2)C1.c1(S)ccccc1 C1(OC)CC2(C1)CC(C(N1CCC1CNC(C1(F)CCOC1)=O)=O)C2 CN1CCCC1(C)C(=O)OCC1C(c2ccccc2)CC1 N1(C(C(COC(C)C)NC(=O)CN2CCC(=O)CC2)=O)CCC12CC(C)(CO)C2 C1(CC(=O)NCC2C(NC(c3n(CCC)ccc3)=O)CC2)CC2(CCC2)CCO1 c1(C(N(CCCNC(C23CC(C)(C2)C3)=O)CC)=O)ccc2c(c1)C(=O)CCC2 C1(C(F)(F)F)(CNC(c2nnnn2CCCF)(CC)C2CCC2)CC(F)(F)C1 Nc1ncc(NC(C2CCN(C(=O)CC3CC3)C2)=O)cc1CC1CC1.C1CC1 C1(CC(=O)NC2CCC(SC)CC2)CC2(C1)CN(C(C1C3CCC(C3)C1C)=O)C2 C12CCCCN1CC(=O)O2.N1(C(=O)OC)CCNC(=O)C1 C=CCC(CNC(C1(C2CCCN2C(=O)C(C)C)CCC1)=O)CC(C)C C#Cc1cccc(C(N2CCCCCC2CNC(=O)CCC(C)(C)C)=O)c1Cl C1(CCCCNC(Cc2c(C)n[nH]c2)=O)CCCN(C(c2csc(=N)[nH]2)=O)C1 N1(C(CC2C(=O)NC(=N)S2)=O)CCCN(C(c2cccc(C(F)F)c2)=O)CC1 C1(CC)CN(C)CCCN1C(C1(C2CC2)CN(C(=O)C(C(C)C)SC)C1)=O c1(NC(C2C(C)N(C(c3cc(O)ncn3)=O)CC2)=O)ccc2c(c1)CCC2 c1(C(=O)NCCCN(C(C23CC(CC)(OC2)C3)=O)C)ccc(Cl)c(O)c1 C(=O)(CC1=CCCCC1)NC(C)CN(C(=O)C(c1cccnc1)O)C c1(C(=O)NCCC2N(C(c3c(C)noc3)=O)CCC2)cc(P(C)(C)=O)ccn1 C1(NC(C2N(CC)CCC2)=O)CC(OC)CN(C(c2ccc(C(F)(F)F)o2)=O)C1 N1(C(C(C)N(C(=O)C(C)(C)c2ccno2)CCN(C)C)=O)CCc2sccc2C1 C1(CNC(CCC)=O)CC2CCCCC2N1C(=O)COc1ccc(Cl)cc1F n1(CC)cc([N+](=O)[O-])c(C(N2CC3(CC(NC(C4CC4(C)C(F)F)=O)C3)C2)=O)n1 CC1(NC(=O)CCC2CC=CCC2)CC(CNC(=O)CCc2cnoc2)C1 c1(N2CCC(N(OC)C)CC2)nc(=NCCC(F)(F)C(C)C)[nH]c2cc[nH]c12 N1(C(CC(=O)NC)=O)CCC(C)C(CNC(c2n[nH]c(C3CC3)n2)=O)C1 CC1(C)CCCN(C(=O)Cc2ccc(F)cc2)C1C(N1CCC2(CC(F)C2)C1)=O C1(C(C)(C)C)(CNC(c2cc(Cl)n[nH]2)=O)CCN(C(=O)CSCC2CCCO2)C1 CC(CC(N)=O)C(=O)NC1CC1NC(C1(Cc2cccc(Br)c2)CC1)=O c1(SC(C)C(=O)O)ccccc1C(=O)NCc1cc(-c2cccc(F)c2)on1 O=C(C(C(C1CCC1)C1CCC1)N(CC)CC1CCC(F)(F)C1)NC1CCCC1 O=C1CC(C(N2CCCC2CC2CCCCCC2)=O)CN1C1CCC1.[nH]1ccnn1 CC1C(NC(=O)CC2(N3CCCC3)CC2)CCCN1C(=O)Cc1ccnc(F)c1 C(CC1=CCN(C(c2ccc(C(N)=O)o2)=O)CC1)NC(C(CC=CCC)C)=O C(=O)(NNc1cccc(OC)c1)c1cc(C(C)NCCOC)on1 N1(C(CCC(=C)Br)=O)CC(C2CN(C(=O)CC(C)(C)F)C2)C1 C1(CC)C(C(=O)Nc2cnn(C)c2C(N)=O)CCN1C(C1CC(C)=NO1)=O C(=O)(C(C)CC(=O)N(C1CCN(C(C2CCC(=O)N2CC)=O)CC1)CC)OCC CCCS(=O)(=O)CC(=O)N(CC)CC1CCCN1C(=O)CC1CC=CC1 c1(CC)nc2ccccn2c1C(=O)NCCN(C)C(C1(C)CCC(C)C1(C)C)=O n1(CCC(N2CC(NC(CC3N(C(C)C)CCC3)=O)(CO)C2)=O)cccnc1=O c1(CC)nnc2cc(NCC(C3CC3)NC(=O)CC3CCCCO3)ncn12 C1(NC(c2ccc(CC)cc2)=O)CC2CC(C1)CN(C(C1(C)C=CCC1)=O)C2 N1(C(c2[nH]c(=NC)sc2)=O)CCN(C(=O)CCCCCF)C(C)C1C C1(O)(C(C)NC(c2cnco2)=O)CCN(C(c2c(Br)noc2C2CC2)=O)C1 Cc1cc2sc(C(=O)NCC3CC34CCN(C(=O)CC3CCCC3)CC4)cc2s1 CC1(NC(c2ccc(C(F)(F)F)s2)=O)CC(NC(=O)CC2CCC(O)C2)C1 C=CCC(CC)C(=O)NCCCCCCNC(C1CC1c1c(C)cccc1C)=O N1(C(CN(CCC)C)=O)CC=CC1(C)C(=O)NCCc1csnn1 c1(C(=O)NC2C(NC(=O)CC3CCCO3)CC(F)(F)C2)[nH]cc2c1CCS2(=O)=O c1(C(=O)NCC2CCN2C(C23CCC(CC2)CC3)=O)ccnc2ccnn12 C(=O)(C(C)(C)CCS(C)(=O)=O)NCCC1N(C(CN(CC)CC)=O)CCC1 C1(O)(CNC(C2C(CCC)C2)=O)CCN(C(=O)C(c2cc(Br)co2)=O)C1 c1(CC)oc2cc1CCCCC1N(C(CN3CC4(CC(F)C4C)C3=O)CC1)C2=O C1(N(C(Cc2c(OC)nccc2)=O)CC(F)F)COC2(CCNCC2)C1 C(=O)(CCCC(C)(C)C(=O)OC)N1CCC(CCNC(C(CC)C(F)(F)F)=O)C1 N1(C(CNC(CNC(C)=O)=O)=O)CC2(C)CC1(C(=O)NC(c1nccn1C)C)C2 c1(NCc2n(C)ncc2Br)ccc(S(=O)(=O)N2CCC(C(N)=O)CC2)c(Cl)c1 Cc1cc(C(N2CC(O)(C(C)NC(=O)C(O)CCc3ccccc3)C2)=O)c(C)s1 c1(C(=O)NC2(CNC(C3C(CC)OCCC3)=O)CCCC2)cc(NC)nc(Cl)c1 C12CCC(C)N(C1)Cc1ccccc1CC(=O)N2.c1(CC)nccn1CC N1(C(C(CC)F)=O)CC(CO)C2(C1)CN(C(c1ccc(C(F)(F)F)[nH]1)=O)C2 c1(C(=O)NC2(C)CN(C(C3C(COC)C3)=O)C2)cccc(C2COC2)c1 C(=O)(CCCCC(C)(C)C)N1CCC(C)C(CC(=O)NCCCCCF)C1 CCC(CNC(=O)CN1CCCNC1=O)(CC)C(=O)NC(c1nnc(C)s1)C C1(CNC(C(F)=CC)=O)CC(NC(c2cn(C3CC3)cn2)=O)C12CCC2 c1(C(=O)NCC2(C)CC(NC(C(C)N(C)C)=O)C2)csc2c(F)cccc12 Cc1ccc(C(=O)C(=O)N(C)CC2CN(C(=O)CSc3ncccc3F)C2)cc1 C(=O)(C1=CCCCO1)NCC1CC(CNC(c2c(C)cns2)=O)C1 CC(C)C(CC(=O)N1CCC(F)(CNC(C2CC(C)C2)=O)C1)C(C)C CS(=O)(=O)c1cc(C(N2CC=CC2Cn2cc(CCCCCO)nn2)=O)co1 C1(C2CN(C(=O)Cc3ccsc3)C2)CN(C(C2CCN(C3CC3)CC2)=O)CCO1 C(=O)(C(C(C)(C)C)NC(=O)N(CC(C)(C)O)CCSc1cccc(F)c1)OCC C1(C(=O)NCCC(C(C)C)NC(C2CN3CCC2CC3)=O)SC2C=CC1CC2 C1(CNC(C2CC(C)(O)C2)=O)CCCCC1NC(C1C=CCS1)=O c1(C(N2CCC(NC(CNC(=O)NC)=O)(CF)C2)=O)c(C)nn(C)c1C(F)(F)Cl C=C(C)CC(=O)N1CC(CNC(c2ccc(C(C)C)s2)=O)(COC)C1 N1(C(c2c(C)nc[nH]2)=O)CC(NC(C2CCCC(C)(C)CC2)=O)C2CCCC2C1 c1(C(=O)NC(CNC(CSCCN(C)C)=O)(C)C2CC2)cc2ccsc2n1C C(=O)(C(C(C)(C)O)NC(=O)CCc1cc(C)[nH]n1)NCc1ncc(C)nc1 Cc1noc(C)c1CC(=O)N(CC(C)(C)CNC(c1cccc(CCO)c1)=O)C c1(C(N(C2CCCN(C(C)=O)C2)CC)=O)ccc(OCC2CCCO2)cc1F c1(C(=O)NC2(CC=C)CCN(C(c3cscn3)=O)C2)ccc(C)c(F)c1F c1(C(=O)NC(C(C)NC(c2c(C#C)c[nH]n2)=O)C(C)C)cc(Cl)c(F)cc1O C1(C(N2CCN(C(=O)CN3CCCCS3(=O)=O)C3C2C3)=O)CCC2(CCC2)CC1 C1(NC(=O)Cc2ncc(Cl)s2)CCC(NC(C2(Cl)CC2(F)F)=O)CC1 C1(NC(C(=O)NCCNC(c2ccc(Cl)cc2)COC)=O)CCCC(N)C1 c1(NCC2(C)CCN(C(C3CC(N=[N+]=[N-])C3)=O)CC2)cc(=O)n(C)c(=O)n1C CCCCC(C)(F)C(=O)N1CCC(CO)(CNC(C2(C(F)F)CC(O)C2)=O)CC1 C#CCC(C(=O)NC1CC(C)OC1=O)NC(c1ccnn1CCC)=O N1(C(C(N2CCOCC2=O)C)=O)CC2(COC(CNC(=O)C(N)=O)C2)C1 CC(CC(=O)N=S(C)(=O)c1cnn2c1CN(C(=O)CC1CC1)CC2)c1ccco1 c1(C(=O)NCC(CN(C(=O)Cc2cncnc2)C(C)C)O)cc(C(F)(F)F)no1 c1(OC)cc(C(N2CC(CNC(C3CC3F)=O)CC23CCC3)=O)cc(OC)c1C C(=O)(CCC(C)(C)F)NC(C(C)C)CNC(C1CCS(=O)(=O)N1)=O N1(C(C(CNC(C)=O)(C)C)=O)CC2CC(NC(C3(C(F)F)CCCO3)=O)CC1C2 N1(C(C(c2ccc(CC)s2)=O)=O)CCC(C)C(NC(=O)C(n2cc(Cl)cn2)C)C1 Cc1cncc(F)c1C(=O)NCc1ncoc1CCNC(=O)CC1CC=CC1 CC1CN(C(C2(CO)CCOC2)=O)CCN1C(c1cnc(C(C)(C)C)[nH]1)=O c1(C(=O)NC2CCN(C(C(CC)O)=O)C2(C)C)sc2cccc(F)c2c1C C1(C)(C(N(C)CC2CCCN(C(=O)CC3CC(OC)C3)C2)=O)CC2CCC(C1)S2 C1(C)(CNC(C2(C)CCN(C)C2)=O)COCCN(C(=O)C2=NOCC2)C1 c1(OC)ccc(CN(C)C(=O)NCC2(Br)CC2)c2ccccc12 N1(C(c2cc(C)on2)=O)CCC(C(C)C(=O)NCC(N2CCCC2)=O)CC1 c1(OC)cc(C)c(C(=O)NC2COCC2CNC(C2CS(=O)(=O)C2)=O)c(C)c1 N1(C(C2(C#N)CC2)=O)CCC2(CCC2NC(c2ccc(Br)o2)=O)CC1 C(C(C)CCO)NCC(=O)NC(C)C(=O)OC1CC(N(C)C)C1 c1(C(N2C(CNC(C3=C(C)OCCS3)=O)CC(O)C2)=O)cc2c(s1)CC(C)(C)C2 c12cc(ccn1)C(C)(C)S2.C(=O)(CC(C)C)NC1C(NC(C)=O)C1 C1(C(=O)NCC2(C)C(C)CN(C(=O)CCNC(N)=O)C2)Cc2cc(F)ccc2O1 c1(OCC(N2CCC(C(c3cn(C)nc3)=O)C2)=O)cccc(CO)c1 Cc1cnnc(C(=O)NCC2(CCNC(=O)CC3SC(=N)NC3=O)CC2)c1 C12(NC(C(CCOC)(C)C)=O)CC(CO)(C1)OC21CCN(C(=O)CSC)CC1 C1(O)(C(C(N2CC(N(C(C=CC(C)C)=O)CCO)C2)=O)F)CCCC1 C(CN=c1cccc(S(=O)(=O)NCC(C)(C)n2cccn2)[nH]1)(C1CC1)OC C1(NC(CC2(CNC(C(C)C3CC3)=O)CC2)=O)CC2CCCCN2C1 c1(C(=O)NC2C3(CCN(C(C4(C(C)=O)CC4)=O)CC3)C2)cnn2c1OCCCC2 C(CCS(N)(=O)=O)(C(=O)NCCCC1CCC1)NC(=O)OC(C)(C)C CCCC(C(=O)NC1CC(C(F)C(=O)N(C)Cc2ncnn2C)C1)C(C)C N1(CC(=O)NCC(CN(C(C=Cc2n(CC)ccn2)=O)C)O)CCS(=O)(=O)CC1 C(=O)(CCCCCOC(C)(C)C)Nc1cc(COC)ncc1 CC(CN=c1[nH]c(=NC(C)CCCO)[nH]c2c1CSC2)c1ccccn1 CC1=C(C)CC(C(=O)NCC2(F)CC(CNC(=O)CN=S(C)(C)=O)C2)CC1 C1(C(N2CC(O)(CNC(c3cc(CO)[nH]n3)=O)C2)=O)CCCOCC1 C(C1CN(C(C2(CC)CCCC2)=O)CC1C(N1CCOC(C)(C(C)C)C1)=O)=CC c1(OC)cc(Cl)ccc1C(N1CC(c2cccc(C)c2)(O)C1)C(=O)NC1CCCCC1 c1(C(=O)NCC2(C(=O)Nc3cncc(C#N)c3)CC(=C)C2)cccc(C)c1C#N C1(C)(NC(c2cn(CCOC)nc2)c2nnnn2CC(F)F)CC=CCC1 c1(C2C(C(=O)NCCN(C(c3cc(F)cs3)=O)CC)C2)ccccc1C c1(N2CCCC(C=C)C2)nc(=NC(C)Cc2nccn2C)[nH]c2ccsc12 C(=O)(CCCN=c1nccc[nH]1)N1C(C)CN(C(c2cc3sccc3[nH]2)=O)CC1 c1(C(N2CCC(C(=O)NCc3n(C)ccn3)C2)=O)ccc(Br)cc1O c1(C(=O)NCC2CC(F)CN2C(C2C=CCCC2)=O)coc(=O)c2ccccc12 c1(NC(C(C)NC(C#CC(C)C)=O)C(C)C)ncnc2cnccc12 C(C(C)(C)S(C)(=O)=O)NC(CCc1ccc(C(=O)NC2(C)CC2)[nH]1)=O CN1CC(=O)Nc2ccc(C(N3CCC(C)(C)C(CO)C3)=O)nc21 CCC(F)(F)C(=O)NC1CN(C(c2nocc2C)=O)CC1c1ccc(F)cc1 C1(CC)(NC(C2OCCC2NC(=O)CCC(C)OC)=O)CC(C)(C)C1 c1(C(N2CCC(=O)NCC2)=O)nccc2cc[nH]c12.c12cn(nn1)CCC2 C1(CNC(C2N(C(C)=O)CCC2)=O)CCN(C(=O)C2=C(Cl)CC2)CC1 C(CCN(C(=O)Cc1cncnc1)C)(C(C)(C)C)NC(C(CC)OCC)=O C1(=CCNC(=O)COC(F)F)CCN(C(C2CCS2(=O)=O)=O)CC1 C(=O)(C(C)(C)C(C)(C)C)NCC1CCCC(NC(c2c(Cl)cn(C)n2)=O)C1 c1(N(C)Cc2nncs2)ncnc(NC(c2cccc(C)c2)C2CC2)c1C C1(C)(C(=O)NC2CCC(CNC(CCC=C(C)C)=O)CC2)CCCNS1(=O)=O c1(C(N=c2cnn(C)[nH]2)=O)cc2cc(C3=CCC(C)(C)CC3)ccc2o1 c1(NC(C(C)N(C)Cc2ccccc2)=O)ccccc1CCN.c1(CC)cccnc1 C#CC1(C(F)(F)F)C(=O)N1.O(NC(=O)OC(C)(C)C)CCCSC C(=O)(C(CO)C(F)(F)F)N(C(CN(C(CCOCCOCC)=O)C)C)C c1(CC)ncccc1C(N1CCC(NC(=O)C(=O)N(C)C)C1c1ccccc1)=O C(=O)(C(C)C(F)(F)C(F)F)N1C(CN(C(c2ccc(O)cc2F)=O)CC)CCC1 CC(CC(=O)NCC1CN(C(C2CCC(=O)O2)=O)CCC1C)CC(F)(F)F c1(CC(=O)NC2C(NC(c3n[nH]c(C)c3O)=O)CCCC2)ccc2ncsc2c1 C(C)(CNC(c1ncoc1C)=O)(C(C)C)NC(CSCC(=O)OC)=O C1(CC)C(NC(=O)CC(C)(C)C)CCCN1C(=O)CC1CCCC1(F)F C1(CNC(C#C)C(C)C)CC2(CC(NC(=O)OC(C)(C)C)CCS2=O)C1 c1(CC(=O)NC2C(OC)CN(C(c3csc(C)c3)=O)C2)cnn(C)c1 c1(SCC(=O)OC)cccc(COC(=O)C2=CC(C)C2)c1 C1(NC(CN(C(COC)=O)C)=O)CCCCN(C(C2(C)CCNC2=O)=O)CC1 c1(CCC(=O)NCC(F)CNC(C2(F)CCCOC2)=O)cc2ccccc2o1 N1(C(Cc2ccc(OC)cc2F)=O)CCCC1C1CCCN1C(C1CN(C)C1)=O c1(C(N2C(CN=c3[nH]nc(C)s3)CCC2)=O)ccc2c(c1)nc(C)n2C C(=O)(C(F)CC(C)(C)NC(C1CCC(=O)C1)=O)N(C)CC1CCCCO1 N1(C(c2c(COC)cc[nH]2)=O)CCC(F)(CNC(C2(NC(N)=O)CC2)=O)CC1 CN1CC(C)(NC(C2CCC=CC2NC(c2cnc(Cl)s2)=O)=O)CCC1=O c1(C(N2CC(NC(c3c(C)nn(C)c3C)=O)C(O)C2)=O)ccnc2cc[nH]c12 N1(C(c2c(C)ocn2)=O)CCCC(NC(C2CCCN2C2CC2)=O)C1C C1(C(=O)NCC2C(C)(C)N(c3nnc(C(F)(F)F)s3)CC2)CCCC2(CCC2)O1 C1(C(=O)NC(CCSCC)C)(NC(=O)C=CCO)CC(CO)C1 Cc1c[nH]c2ncnc(N3CCCC(C(=O)Nc4cc(Br)ccc4I)CC3)c12 C1(NC(C2CC(OC)C2)=O)CCN(C(c2cc(-c3csc(C)n3)cn2C)=O)C1C C(=O)(C(O)C(C)(C)C)N(C(C)CNC(c1ccn(C(C)(C)C)c1)=O)C CCCCC(CNC(C1CCC2(CC2)C1)=O)NC(=O)C(C)(C)C1CCCC1 C1(C(=O)NCC2(C)N(C(CN3CC(C)(C)C3)=O)CCC2)CCCCCCC1 C1(COC)(NC(c2cc(OC)nn2C)=O)CCN(C(C2CCCC2CF)=O)C1 c1(C(N(CC2N(C)CCC2)CC2CCCO2)=O)cnc(Cl)c(Cl)c1 C1(NC(C2COC2)=O)CC2CCCC(C1)N2C(=O)CC1CCCCCO1 C1(C(=O)NCCN(C)C(c2cn(C)nn2)=O)COC2COCC2O1 C(=O)(CCC(N)=O)NCCCC1(CNC(CCc2cc(C)[nH]n2)=O)CCCC1 c1(C(=O)NC(CNC(CCOC(C)C)=O)C)cccn2[nH]c(=N)nc12 C1(O)(C(C)NC(=O)CN(C2CCSC2)C)CCN(C(c2cc(Cl)ns2)=O)C1 c1(OC)ccc(F)cc1C(=O)NC1(CCNC(=O)C(C)S(N)(=O)=O)CCC1 N1(C(C2CCN(C(C(C)CC(N)=O)=O)C2(C)C)=O)CCCOC(C)(C)C1 c1(C(=O)NC(C(C)NC(=O)C=CC=C(Cl)Cl)(C)C)ccnc2ccnn12 c1(C(=O)NCC2C(CNC(=O)C3=NOCC3)C2)cc(=O)n2ccccc2n1 N1(CC(C)C)CC(C(=O)N(C2CCN(CC(=O)N(c3nccs3)C)C2)C)CC1=O C(=O)(CCCCC(C)(C)OC)N1CCN(C(CN(CC)CC)=O)C(CC(F)F)C1 N1(C(c2c(OC)ccc(OC)c2)=O)CCOC2(CCCN(c3ccncn3)C2)C1 N1(C(CN(C)C(N)=O)=O)C2CCC1(CNC(=O)Cc1ccccc1Cl)CC2 Cc1c(C(=O)NC2COCCC2NC(=O)CC2CCOC2(C)C)sc2cncn12 C#Cc1ccc(NC(=O)C(C(C)OC)NC(=O)C=CCCC(C)C)cn1 c1(NC(C(CNC(c2cnns2)=O)N(C)C)=O)cnc(O)c(F)c1 CCC(CC)(CCNC(=O)C1=NOC(C)C1)NC(C1CCC(=O)C1)=O C12(NC(C3CC(OC)C3)=O)CCC(CC1)N(C(C1CCC1c1ccccc1)=O)C2 C1(OC)CN(C(c2cc(O)no2)=O)CC1NC(c1ccc(I)cc1)=O n1(C(C)C(=O)NCC(c2cccs2)(C)C)cc(CC2(N(C)C)CCC2)nn1 N=c1[nH]c2ccc(C(=O)NCC3CC(F)CN3C(C3CCCNC3=O)=O)cc2s1 Cc1cc(C(N2CCOC(CCNC(=O)CCCc3cc[nH]n3)C2)=O)ncc1F N1(C(CC2CC(NC(c3[nH]cc(C)c3)=O)C2(C)C)=O)CCn2ncc(O)c2C1 C(=O)(C=C1SCC(=O)N1C)N1CCC(COC)(NC(c2ccc(Cl)cc2)=O)C1 C12(NC(=O)C3=CCC3)CCCC1CN(C(C1(CC3CC3)CCC1)=O)C2 N1(C(C2(NC(CN(C3CCC3)C)=O)CC(F)C2)=O)CCC2CCCC2C1 N1(C(c2cccc(C(N)=O)c2N)=O)CC2CCC(CC2)C1 C1(NC(C(c2c(C)noc2C)CC)=O)CCC(C)N(C(=O)CCc2cncs2)C1 c1(C(N(C(C)CN(C)C(c2ccc(C#N)cn2)=O)C)=O)cnn2ncccc12 C1(C(=O)NCC(C)C)CC2CCCCC2N1Cc1cccc(-c2ccccc2)c1 C1(NC(C(C(C)CN)F)=O)CC2CC(C1)CN(Cc1ccccc1)C2 CCCS(=O)(=O)C(C)C(=O)NC(CN(C(c1n[nH]cc1CC)=O)CC)CC c1(C(C(=O)NCCN(C(=O)CC23COC(CF)(C2)C3)CC)O)ccc(Cl)cc1 c1(NC(C2CCN2C(=O)C=Cc2ccc(C(F)(F)F)s2)=O)cccc(C2CC2)c1 C1(N(C(C2CN(c3nncs3)C2)=O)NC(CCc2cnc(C)s2)=O)CCC(C(F)F)CC1.N C=CC1COCC1NC(=O)CCC1CC(NC(=O)Cn2ccc(C)cc2=O)C1 C12(Nc3cc(NC(c4ccoc4)COCC)nc(C)n3)CC3CC(C1)C(C)CC3C2 c1(N2C(C(=O)Nc3ccc(C#N)cc3I)CC2)ncnc2ncc(Br)cc12 Cc1sncc1C(=O)NC1COCC1C(N1CC(n2ccnn2)C1)=O c1(Cn2c(-c3snc(C)c3N)nc(COC(C)C)n2)cc2n(n1)CCCC2 N1(C(c2c(OC)nccc2)=O)CCCC2CN(C(C3CCCN(C(C)=O)C3)=O)CC12 c1(C(N(CCCCCNC(c2n(CC=C)ccc2)=O)C)=O)cccnc1C(F)F N1(C(C2CC(C)(C)C2)=O)CCN(C(C2CCN2C2CCCC2)=O)CC(O)C1 c1(C(N2CCC(C(CNC(C(CC)(C)CO)=O)O)CC2)=O)cc(C)c(C)cc1C c1(C(N2CCCC(C)(C)C2C(N)=O)=O)ccc2c(c1)SCC(=O)N2 N1(C(C(C)SC(C)C)=O)CCC(CNC(=O)CCn2ccnn2)C(F)(F)C1 C1(C(=O)NCC(C(C)C)OC)CCCCN(C(=O)COCCC(C)C)C1 c1(OC)cncc(CCC(=O)NC2CCCC2(C)CNC(C2C3CCC23)=O)c1 CC(C)C(O)CC(=O)N1CCC(CN(C)C(c2ccccn2)=O)C1 C(=O)(C(C)(C)C(C)O)NC(CCN(C(c1c(C)csc1)=O)C)C c1(C(=O)NC(C2N(C(CCCCOC)=O)CCCC2)C)ccc2nsnc2c1 c1(CC(=O)NC2C(NC(CCC#C)=O)C2)sc(SCC)nc1C c1(NC(=O)NC(C2CC2n2ccnn2)C2CC2)csc2ccc(Cl)cc12 c1(C(=O)NCCC)nc(=NC(=O)N2CC(=O)NC(c3ccccc3)C2)s[nH]1 C(=O)(C1=CCCCO1)N1CC(CNC(c2cc(C)nn2CC(F)(F)F)=O)C(C)C1 n1(CC(N2CCC(CNC(CC3CC(=C)C3)=O)C2)=O)cc(-c2ccccc2)cn1 CC1(C)C2CC(C(N3CCC(O)C(NC(c4ccc([N+](=O)[O-])[nH]4)=O)C3)=O)CC12 CC1CN(C(=O)NCc2cccn(C)c2=O)CCC1O N1(CC(=O)NCC#CCNC(C(COC)O)=O)CCN(C2CC2)C1=O C12(CC(=O)NCC(=C3CN(c4ncn(C)c(=O)c4)C3)F)CCCCC1C2(F)F c1(C(C)C)nnc(C=CC(=O)NC2CCN(C(=O)C(F)(F)C3CC3)CC2)o1 c1(CC(=O)NCCOC(CNC(C(CC)=CC)=O)(C)C)cccc2[nH]ncc12 CC1CCc2nc(C(=O)NCCC(C)N(C)C(c3ccsc3)=O)ccc2C1 C(=O)(C(O)C1=CCCCC1)NC1(C2CN(C(CC(COC)COC)=O)C2)CC1 CC(CC(=O)NCC1CC2CCC1O2)C(C)(C)NC(=O)C(F)=CC1CC1 CN1CCC(C)(C(=O)NCC2CCN(C(=O)C=Cc3ccccn3)CC2)CC1 C(C(O)C(=O)N=c1ccn(C(C)(C)C)[nH]1)NC(c1nn(CC)c(C)c1)=O C1(NC(CCCOCCC)=O)CN(C(C2C3CCC23)=O)C2(CCCCC2)C1 c1(C(N(C2CCCN(C(C3C(COC)C3)=O)CC2)C)=O)cccn2ccnc12 CC1(C)COCCC1C(=O)NCC12COC(CNC(=O)C=Cc3cncs3)(C1)C2 C1(C(=O)NC2(c3ccc(Cl)cc3)CC2)CCN(C(c2ncsc2Br)=O)CC1(F)F C1(c2nc(C)on2)CCN(C(c2ccc(-c3ccccc3)cc2)C)CC1 C1(CNC(C(C)CF)=O)CC2(CO1)CN(C(c1ccc3ccnn3c1)=O)C2 N1(C(C(=O)NCC23COCCN2C(=O)OC3)=O)CC2CC(O)CC(C2)C1 c1(NCC2(N(C)C)CCC2)cc(S(=O)(=O)NCC2CC23CC3(F)F)ccc1C#N C(=O)(CS(=O)(=O)C1CCCC1)NC1CCC(CNC(C2(C(C)C)CCC2)=O)C1 O=C(CC(C(F)F)n1cccn1)NC1C=CCN(C(c2cnn(CCO)c2)=O)C1 c1(CCCC)cn(CCN(C(=O)CNS(=O)(=O)NC)CC)nn1 C1(F)(CNC(CN(c2ccccc2)C)=O)CCCN(C(=O)C(C)(C)CF)C1 CC1(F)CCN(C(C2CCC(C3CC3)N2C(c2cc(C(N)=O)c[nH]2)=O)=O)C1 c1(C(=O)NCC2(OC)CN(C(c3cnncc3O)=O)C2)cc(S(N)(=O)=O)c(C)s1 c1(C(C)(F)F)ccc(C(=O)NCCOCCCNC(C2CCCN2C=O)=O)cn1 c1(CNC(N2CCOCC2CC2CC2)=O)ccc(CN2C(=O)CNC2=O)cc1 C1(NC(CSC)=O)CCC2CCN(C(c3ccc(Cl)nc3)=O)C1C2 C#Cc1cc(C(=O)NCC(C)N(C(c2cn(C)nc2O)=O)CC)cc(Br)c1 CN=c1[nH]c(=NCC2CCCCC2)[nH]c(=NCc2cccc(Br)c2C)[nH]1 Cc1nc(CNC(=O)CC2CCCO2)oc1C(=O)NCCC(F)F c1(SC)ccc(NC(=O)Nc2ccc(NC(C3(O)CCCC3)=O)cn2)cc1 C(=O)(C(CNC(=O)C(C1CC1)SC)OC)N(CCC(=O)NC)C Cc1nc(CNC(=O)C(=O)N(C)CCSc2ccncc2)n[nH]1 n1(CC(=O)N(CC(C)(C)NC(C(C)C2CC2)=O)C)ncc(O)nc1=O C1(CCC(=O)OCC)CCCN(N2CC=C(C(=O)N(C)C)CC2)C1 c1(C2C(CNC(CCNC(C(C)c3cc[nH]n3)=O)=O)C2)cn(C)cn1 C(N=c1[nH]c(=N)[nH]c(=NC2CCCN(C)CC2)[nH]1)c1nc(C)sc1C c1(C(c2n(CCCSC)nnn2)NCC(C)CCCO)cc2ccsc2n1C C(=O)(C1=CC2(CCNCC2)C1)NC(C(=O)OC)Cc1cncc(Cl)c1 c1(C(C(=O)NC2CC2)N(CC(C)N(C(C)=O)C)C)ccnc(Br)c1 C1(C(=O)NCCCCN(C)C(c2nc(C3CC3)cs2)=O)CCOCC1(C)C C#CCCCCCCCC(=O)N(CCNC(=O)CC(O)CCCC)C1CC1 CC1=C(C)CC(C)(NC(C2CCN(C(c3cc(C#N)cs3)=O)CCO2)=O)CC1 c1(C(=O)NC2C3(CCN(S(CC)(=O)=O)CC3)C2)cc(O)c(OC)cc1[N+](=O)[O-] N1(C(C=C(C)c2cccs2)=O)CCC2CN(C(=O)C=Cc3ccc(C)o3)CC2C1 CCCCC(O)C(=O)N1CCCC(C)(CNC(=O)COc2c(C)occc2=O)C1 N1(Cc2cc(C)nn2C)CC(NC(c2cccc(C(F)(F)F)c2Br)=O)C2(CC2)C1 C1(OCC)CCN(C(c2cc(CNC(=O)CN(C)C(C)=O)[nH]n2)=O)CC1C CC1CCN(C(=O)CC2(n3cccn3)CC2)CCN1C(=O)C(CO)C(F)(F)F c1(C(=O)NC(CC=C)CNC(c2ccc(C)n2C)=O)cc2cccnn2n1 C1(C(=O)NCc2nnc(CC)o2)CCCN(C(c2cnn(C)c2OC)=O)C1 Cc1ccc(CCC(=O)NCCCCN(C(=O)C(O)C2CCCC2)C)c(C)c1 Cc1n[nH]c(C)c1CC(=O)NC1CCCCC1CNC(=O)CCc1nc(=N)[nH][nH]1 c1(C(=O)NCC2C(NC(c3c(C)oc(C#N)c3)=O)CCC2)cnc2c(c1)NCC2 C(CCC(C)CC(=O)N1CCC(N(C)C(c2ncn(C)c2C)=O)C1)=C(C)C C1(C(=O)C(C)C(C)(C)C)(CCC)CCCN(C(=O)CCc2ccc[nH]2)C1 C1CCC(=O)NCC(CNC(=O)C(C)N(C)C)OC12CC2.n1(CC)cnnn1.CS c1(CC(=O)CN(C(=O)C=CSCCc2ccco2)Cc2ccco2)ccc(Cl)nc1 c1(C(=O)NCCCNCC2(OCC3CCCC3)CC2)cc(Cl)cc2cccnc12 O=S(=O)(CCC(F)(F)C(F)(F)F)N1CCCC1c1ccnc(Cl)c1 O=C1NCCCCC1C(N1CCCC(CO)(NC(=O)C2=COCCO2)C1)=O Cc1cnc(C(=O)N(C2CCCN(C(c3ccnc(S)c3)=O)C2)CCO)cn1 C(=O)(C(F)C(C)(F)F)NC(C(=O)NC1(C)CCOC1)CO c1(C(=O)NCC(C(C)(C)C)NC(C2CC(OC)C2)=O)cncc(P(C)(C)=O)c1 c1(N2CC(F)CC(NC(=O)C(c3ccccc3)=O)C2)ncnc2n[nH]c(I)c12 C12C3CCC4C(C3)C14N2.c1(OCC)ccc(C2CCCC2N(C)C)cc1 Cc1ccc2c(c1)CN(CC(c1ccc3c(c1)OCCO3)C)CC2 C1(NC(C(COC)(C)OC)=O)CCC2(CC1)CN(C(C1(C)CC=CC1)=O)CCO2 c1(CN2C(C)(C(=O)Nc3ccc(C)nc3CO)CC2)ccc2sccc2c1 C(N=c1[nH]c2c(F)cc(Cl)cc2s1)C1CCCN(C(C2CN(CC)C(=O)C2)=O)C1 c1(C(=O)NCC2(C(N)=O)CN(C(CC(CC)SC)=O)C2)cccc(S(C)=O)c1 c1(CN2C(C(=O)NCC(C)(C)CO)C=CC2)ncc(-c2ccccc2)cc1F CCCCC(C)(F)C(=O)N1CCN(C(c2ccc(=O)n(C)n2)=O)C(C2CC2)C1 N1(C(COCCOC)=O)CCCC(CC(N2CCC(OC)C2(C)C)=O)CC1 c1(C(=O)NCC2N(C(C(C)n3cncn3)=O)CC2)cccnc1OC1CCCC1 c1(C(N(CCOCCCN(C(C2ON=C(C)C2)=O)C)C)=O)cccc(C2CC2)n1 CCCC(C)(O)CC(=O)N1CC2CC(NC(C3CCCO3)=O)C2C1 C1(C2CN(C(=O)COC3CCC(C)CC3)C2)(NC(CCSC)=O)CC1 C#Cc1cnn(C)c1C(=O)NC1CN(C(c2ccccc2COC)=O)CC1C n1(CC(=O)NCC2CN(c3snc(C)n3)CC(C)(C)O2)c(=O)oc2ccccc12 c1(C(=O)NCCCNC(c2c(N(C)C)ccnc2)=O)cc(O)nc(Cl)c1 S(=O)(=O)(c1ccc(F)c(NC(C)=O)c1)NCC(c1ccnn1C)OC C1(NC(CCC#CC)=O)C(C)CN(C(=O)CCCc2ccc(Cl)c(Cl)c2)CC1C CC(=O)CC(C)(C)C(=O)NCC1CCCC1NC(=O)CCc1ncc(C)[nH]1 N1(C(C(CC)CC)=O)C2CCC1CC(CNC(c1cc(C(C)(C)C)ccn1)=O)C2 C1(C(=O)NC(C2CCC2)C)(NC(=O)CC2(O)CCOC2)CC(O)C1 CCC(CC(=O)NCC1CCCCC1NC(c1ccc(COC)[nH]1)=O)OC N1(C(C(CCCC)O)=O)CCn2ncc(CNC(c3nc(C4CC4)cs3)=O)c2C1 c1(CC)ccc2nc(NC(N3CCC(C)C(CSC)C3)=O)sc2c1 Cc1nc(C)c(C(=O)NC2CC(C(=O)NC3CC=CCC3C)C2)o1 Cc1nc(Cl)ccc1CC(=O)NC1(CNC(c2ccc(Cl)nn2)=O)CCC1 CC(C)C(C)(CNC(=O)CCn1ccccc1=O)NC(c1occc1Br)=O C1(OC)CC2N(C1)C2=O.c1(C(C(=O)NC2(CC(=O)OC)CC2)C)ccn(C)c1 Cc1cccc(NCCCNC(=O)NCc2cccc(-n3cncn3)c2)c1 C1(C(=O)O)CCC2(C1)CN(Cc1cccc(-c3sccc3[N+](=O)[O-])c1)C2 C1(SC)CCCC1n1cc(CN(C(=O)CSc2ccco2)C)nn1 C1(Nc2ccc(C(C)=O)cn2)COCCN(C(c2cn3c(n2)CCC3)=O)C1 C1(C(N2CCOCC(NC(C(=C(C)C3CC3)F)=O)C2)=O)CC2(CO1)CC(F)(F)C2 c1(C(N2CCCC(NC(C)=O)CCC2)=O)ccc2c(c1)C=CS2(=O)=O C#CC1CCN(C(=O)CC(COC)NC(c2cccn2C(C)C)=O)CC1 c1(CC(C(=O)OC)NC2CCCC(C)(C)C2)c[nH]c2ccc(F)cc12 C1(C(=O)NC(C(CO)NC(C2(CCOC)CCC2)=O)C)CCC(C2CCC2)CC1 C1(CCOC(c2cccc(NC(C)C)c2C(=O)O)=O)Sc2ccccc2NC1=O Cc1ncn(O)c1C(=O)NC1CC1CNC(C1CC(C(F)(F)F)C1)=O Cn1cnc(CC(O)C(=O)N(C2CCCC2)CCN(C2CCC2)C)c1 C1(CNC(C(C)Cc2ccc(F)cc2)=O)CC2(C1)CN(C(c1ccsn1)=O)C2 CC1CN(C(=O)Cc2cnccc2Cl)CCCN1C(C12CC1CCC2(F)F)=O C1(C(N(CC(=O)NCc2ccc(CO)cn2)CC)=O)CCOC(C)C1 c1(N2CCCC3(CO)C2C3)nc(N2CCN(C3CC3)CC2)nc2c1ncn2C C1(N=[N+]=[N-])(CNC(c2n(CC#C)ccc2)=O)CCN(C(=O)OC(C)(C)C)C1 C(CCCC(F)(F)F)NC(C=CCN(C(c1c(OC)n(C)nc1)=O)C)=O Cc1cncc(C(=O)NC2(C)CN(C(=O)CCCc3n[nH]c(=N)s3)C2)c1C c1(C(=O)NC(CC=C)CNC(C2(CC(F)F)CC2)=O)cccc(CSC)c1 c1(C(N2C(CNC(c3nnn4c3COCC4)=O)CC2)=O)ccc([N+](=O)[O-])cc1O c1(C(N(CC(=O)NCC(C)(C)Sc2nccn2C)CCC)=O)ccc(F)cc1C Cc1n[nH]c(C)c1CN(C)C(C1(CN)CC(O)C1C)=O N1(C(CSCC(C)C)=O)CCCN(C(=O)Cc2cn3ccccc3n2)CCC1 N1(C(C2CCC(C)S2)=O)CCC(O)(CNC(c2cnc(Cl)s2)=O)CC1 N#Cc1nccnc1N1CCOCC(CNC(=O)C(F)(F)c2cccnc2)C1 N1(CCC(=O)NCC=CCNC(C(c2c(C)noc2C)CC)=O)CCCCC1=O c1(OC)cc([N+](=O)[O-])ccc1CN1CCC(N2CCCOCC2)C1 N1(Cc2ccc(C(=O)NC(COC)C)cc2)CCC2CCCC12 C1(NC(=O)CC2CCCC2)CN(c2nc(Cl)ncc2Br)CC2(CC2)C1 CCCS(=O)(=O)CC(=O)N1CCC(NC(c2n[nH]c3c2COC3)=O)C1 c1(C(=O)NCC(CC)NC(c2ccc(CC)o2)=O)cc2c(cn1)OCCO2 C1(CNC(C=C(C)Cl)=O)CC2CCC1N(C(=O)C1=CC3CCCC13)C2 C1(C(=O)Nc2cnc(C(N)=O)nc2)CC2(CC2)CN1C(=O)C=Cc1ccsc1 C1(NC(C=CSC)=O)CCN(C(c2nnn(C(C)C)c2C)=O)CC1C c1(CN2CC(N(C(=O)COc3ccccc3)C)C(F)C2)ccc(Cl)cc1I N1(C(C(C=C)O)=O)CCN(C(c2cccnc2SC)=O)CC1CO CCC(O)C(C)C(=O)N1CCN(C(=O)C=Cc2ccco2)CC1 C(c1cccnc1)=C(C)C(N1CCC(CO)(CNC(C2CN(C(N)=O)C2)=O)C1)=O C1(NC(C2N(C(c3n(CCC)ccc3)=O)CC(C)(C)C2)=O)CC(C)(C)OC1(C)C N1(C(C2CC(C#C)(O)C2)=O)CCC2(CCCN(C(c3nccs3)=O)C2)C1 N1(C(C(COC)O)=O)CC(C2(NC(C3C(C)C3(F)F)=O)CC2)C1 C(=O)(C(C)C(=O)N1CCC(F)(C(=O)NCc2cc(C)c(C)s2)C1)OC c1(OC)cc(CO)ccc1C(=O)N(C1C2CN(C(=O)CCC=CC(C)C)CC12)C N1(C(CCN2CCN(CC)CC2)=O)CC(NC(C2(C)CC(F)(F)C2)=O)CC(O)C1 C(=O)(C(c1ccc(Cl)cc1)=Cc1ccc(C)cc1)NC(CCP(OCC)(C)=O)C C1(C2CC2C(=O)OC)(NC(=O)CCc2ccsc2Br)CCCC1 c1(CC)cc(C(=O)N(CC(C)NC(C2CC(OC)(OC)C2)=O)CC)n(C)c1 c1(Nc2cn(CC(P(OCC)(=O)OCC)O)nn2)ccc(S(=N)(=O)C(F)F)cc1 C(C(C)(O)CC(=O)N1CC(OC)CC1CNC(c1sncc1C)=O)OC N1(C(C)=O)CCc2ccccc2C1CC(=O)N(C1CN(C(=O)C(C)(F)F)C1)C N1(C(C(c2cccnc2)C)=O)CCC(C2(NC(c3ccc(Cl)cc3F)=O)CC2)C1 C1(C(=O)OC)CC(=O)NN(C(=O)c2cc3cnc(Cl)cc3s2)C1 C1(C(=O)NC2CN(C(c3cnoc3-c3cccs3)=O)CC2O)CCCNS1(=O)=O c1(C(=O)NCC2C(NC(c3cnccn3)=O)C2)cc(C(F)F)ncn1 N1(C(C(CC)C)=O)CC2CN(C(C3CCCS3)=O)CC12 O=C1CCCC(C(=O)NCC2(O)CN(C(C3COCCO3)=O)C2)O1 C1(CC(=O)NCCN(C(=O)CCCF)C2CCCC2)CCCCC12CC2 c1(OC)cc(=O)n(C)cc1C(N1CC(NC(C2(C3CC3)CCC2)=O)CC1(C)C)=O C1(COC)(CNC(=O)C(F)C2CCC2)CCCN1C(=O)Cn1ncn(C)c1=O C(=O)(CCCC(=O)NCC(CCO)C(F)F)NC c1(C(=O)NCC(C(C)C)NC(C(CC)(C)OC)=O)c(F)cccc1F C(C(C)(C)C(=O)N(CCC(C(C)C)NC(C1CC(O)CN1C(C)=O)=O)C)OC c1(C(N2C(CNC(C(F)OC)=O)CC2)=O)cc2c(s1)CCCCCC2 CC1CC(NC(=O)CCC2(C)CN(C(C3CCOCC3)=O)C2)c2nccn21 c1(NC)ccc(C(=O)NCC2(CNC(C3CCNC(=O)C3)=O)CC2)nc1 CCC(F)(F)C(C)(C)C(=O)NC1CC2CN(C(=O)COCCOC)CC12 C(=O)(C1CNC(=O)c2ccccc21)NCC1(C(C)NC(c2cnccn2)=O)CC1 N1(C(Cc2cc(C)on2)=O)CCCC(C(N2CCC(n3cncn3)C2)=O)C1 N1(C(CSCC)=O)CC(F)CC1CC(=O)NC1CCN(CCN(C)C)C1 C1(C(N2CCCC(N(C(Cc3c(C)nc[nH]3)=O)C)C2)=O)CC(C)(C)CN1C C1(C(=O)NCC2N(C(c3scc(C(N)=O)c3)=O)CC2)C2CCCCC12 N1(Cc2c(OC)cccc2)CC2CC(C1)C2Cc1ccc(C(N)=O)cc1 CCC(COC)(CC)C(=O)NCC1CCCC1C(=O)N(C)Cc1cn[nH]c1 CC(C(C)(C)C(=O)N1CCCC1)NC(c1nnsc1N)=O N1(C(C2CN(C(C(CCCCC)F)=O)CC(C)O2)=O)CCc2ccncc2C1 n1(CC)cc(C(=O)C(=O)NC(C)CNC(=O)C(C)N2CC(C)C2)cn1 C1(C(N(CCCNC(CCC#CC)=O)C(C)C)=O)CC(=O)c2ccccc2C1 C(c1ccc(Cl)nc1)=CC(N1CCN(C(=O)C2=CCCO2)C(CCO)C1)=O C1(NC(=O)Cc2nnc(O)s2)CN(C(C23CC(F)(C2)C3)=O)CC12CC2 c12ncc(C)cc1S(=O)(=O)NC1CC(C)(C)C1N1CCN2CC1.CCC=O n1(CC(=O)NC2C=CCN(C(c3cncc(C)c3Cl)=O)C2)cc2ccccc2n1 C(C1CCCN1C(=O)COCC(C)C)=CC(=O)NCc1n(CC)cnn1 c1(C(=O)NCC(C)CN(C)C(C2CC2c2ccsc2)=O)cc(Cl)n[nH]1 N1(C(C(CC=C)N(C)C)=O)CC(C2CN(C(c3cccc4sncc34)=O)C2)C1 c1(CNC(CCOCC#C)=O)cc2n(n1)CCN(C(=O)Cc1scnc1C)C2 c1(NCCOCCCN(C(=O)CCC2(C)CC2)C)[nH]c(=O)n(C)c(=O)c1C#N Cc1ccc(CC(N2CC(CF)(NC(=O)C(C)c3ccsc3)C2)=O)c(Cl)c1 c1(OC)ccnc(C(N2CCC(O)(C(C=C)C3CC3)C2)=O)c1O.C1(=O)CCN1 C(=O)(C(C)(C)C(=O)NCCCC1(NC(=O)Cc2ccc(F)c(C)c2)CC1)OCC N1(C(C(=O)NCCCC)CC2CCCCO2)CCN(c2cccc(F)n2)CC1 Cc1ccc(C(=O)NCC2CC2NC(=O)CN(C)S(N)(=O)=O)cn1 c1(C(=O)NC2CCC(NC(C(C)(CO)OC)=O)C2)cc2sc(C)cc2s1 c1(CNC(c2n(CC)nnn2)CCc2cn(C)nn2)cccc2c1CCC2 c1(CC)nc(C)cc(=NC(C)CCNC(c2c(C)ccnc2OC)=O)[nH]1 c1(CNCCN2CCCC2)ccc(-c2nnnn2C2CC2)cc1 CCC(CC(=O)NC1CC(F)CN(C(c2ccncc2OC)=O)C1)C(C)(C)C c1(C(N2CCC(CC=C)(C(N3CCC(CSC)C3)=O)C2)=O)cncc(C#N)c1 C#Cc1cc(F)ccc1CN1CCOC(CNC(=O)Cc2cncnc2)C1 C1(C(=O)OC)CC2(CCOCC2)CN1C(C1CCC12CCCO2)=O CC1=C(C(=O)N(C)CC=CC(N2CC(C)CC2CO)=O)CC1 c1(OC)cc(C(=O)NC2CCNC2(C)C)nn1C N1(C(C(C)OC2CCOC2)=O)CC2CCC(C1)C2NC(C1CC(F)C1)=O N1(C(c2occ(C(C)C)c2)=O)CCC2CCC12CNC(c1ccc(=O)n(C)c1)=O c1(C(N2CCC(CC(=O)NC(CC)CO)C2)=O)cc2sccn2c1 Nc1ccc(Cl)c(C(=O)NC2CC(NC(C3(CF)CCOCC3)=O)C23CCC3)c1 c1(Cn2cc(-c3cnc(C)nc3)nn2)cc(O)cc([N+](=O)[O-])c1 C1(C)(C(=O)NCCCC(=O)NCC(C(=O)OC)C)CC2(CCC2)C1 C12(C(=O)NCC(CO)NC(C3(S(N)(=O)=O)CCC3)=O)CC3CC(C(=O)N1)C2C3 C(CCC(=O)NCc1nc(CNC(=O)CC2CCC(O)C2)cs1)OC(C)=O Cc1ncc(F)c(NC(C2CC3(C2)CN(C(=O)CCCCCBr)C3)=O)n1 C(=O)(CCC(=O)NCC(CO)NC(=O)C(C(C)C)c1cccc(OC)c1)NCC C1(CNC(c2cc(OC)cc(F)c2)=O)CC2(CCN(C(=O)CCC3CC3)CC2)C1 C(C1=CCN(C(c2cnc(N)c(Br)c2)=O)CC1)NC(CC1N(C)CCCC1)=O c1(C(=O)OC)cc(OC)ccc1NC(c1nc(-c2cnn(CCO)c2)sc1C)=O N1(C(C(C)=CC)=O)CC(NC(=O)C(C(C)C)n2cc(C)cn2)C(C(F)F)C1 N1(CC(=O)NCc2cn(-c3ccc(OC)cc3)nn2)CCOc2ccccc21 C(=O)(C#CC1CCOC1)N1CC(C)(n2cc(CCC3CCCOC3)nn2)C1 Cc1cccc(C(=O)N(C2CCN(Cc3ccc(O)c(O)c3)C2)C)c1I Cc1onc(-c2ccsc2)c1C(=O)NCC1CC1NC(=O)CC1CCCN(C)C1 N1(C(CC(C(C)OC)NC(=O)CC2(O)CCOC2)=O)CCC2(CCC2)CC1 CC1CC(N=c2ccc3nnnn3[nH]2)CN1C(=O)CCCCCn1cnnn1 Cc1ccn(CC(=O)NC2COCC2CNC(=O)C(C)(C)C(N)=O)c(=O)c1 C(N=c1nc2sccc2c(N2CCc3c(cnn(C)c3=O)C2)[nH]1)c1nc(C)sc1 C1(NC(c2c(CC)c[nH]c2)=O)CC12CCN(C(C1COCCN1C)=O)CC2 C1(C(=O)NC2N(S(C)(=O)=O)CCC2)CCCN(C(c2cccc(F)c2F)=O)CC1 c1(CN=C(NC2(C)CCC2)NC2CCS(=O)(=O)C2)ccc(O)c(Cl)c1 C1(NC(C(C(C)NC(=O)C2=CCCCC2)(C)C)=O)CCCOC12CCC2 CC(C(=O)OCC=C(C)C)N(C(=O)CNC(c1ccoc1)=O)C(c1cocn1)=O N1(C(c2scc(C)c2Cl)=O)CC(F)(F)CC1CNC(C1Cc2nccn2C1)=O c1(C(=O)OCC)nnc(SC)nc1N1CC(NC(C2C=CC(=O)NC2)=O)C(F)C1 C=C(C)CC(C(=O)NC1CCCN(C(c2scc(Cl)c2Cl)=O)C1)NC(C)=O c1(CC)noc(C(=O)NCC2CCCC2NC(=O)C(CC)N(CC)CC)c1C C(=O)(CC1OCCc2ccsc21)N(CCCNC(c1c(CC)occ1)=O)C(C)C c1(C(=O)NCC(F)CNC(C2CC3CC3C2)=O)cnc2ccccc2c1 c1(CC)ccc(C=CC(=O)N(C)CCN(C(C23CC(C)C2C3)=O)C(C)C)o1 c1(OCC)ccccc1C.c12cn(nn1)C(C)C(=O)N2C(C)CC1CNC1 C#CC1(C)CCCN(C(C2C(O)CCN2C(c2cc(C(C)C)[nH]n2)=O)=O)C1 C1(C(=O)NCCCCn2cc(-c3cccc(F)c3Cl)nn2)CCn2cnnc2C1 C1(NC(Cc2cc(C)sc2)=O)CS(=O)(=O)CC1NC(=O)C(C)(C)C1CCCC1 N1(C(C2(C(=O)OC)CC2)=O)CCCCC(N(CC(F)(F)F)S(C)(=O)=O)C1=O C1(C(=O)NC2CN(C(CCSC)=O)CC2C)CCc2ccc(F)cc2O1 CC1(C)C(C)(C)C1(F)C(N1CCC(CF)(NC(=O)CCN2CCCS2(=O)=O)C1)=O Cn1c(=O)ccn(CC(N2CCCC(NC(=O)C=CC3CC3)C(F)C2)=O)c1=O N1(C(CC(C)(C)O)=O)C2CCC1C(C(=O)NCc1ccccc1OC(F)F)C2 C1(NC(C(C)Cc2cccc(Br)c2)=O)CCCN(C(=O)CCCF)C1C Cc1ccc2occ(C(=O)NC3CCN(C(c4cnn(C)c4Cl)=O)C34CC4)c2c1 CC1COC(C)(CNC(=O)CCOC2CN(C(=O)Cc3ccoc3)C2)CO1 c1(CNC(CC2C(NC(C3(C)CC3)=O)CCC2)=O)nc(C#N)cs1 N(C1CCCc2ccc(OC)cc21)C(C1(CC)CCCCCC1)=O C(=O)(CCC(F)(F)C(F)(F)F)N1CC(CCNC(c2c(CC)nc[nH]2)=O)OCC1 c1(SCCC(=O)NCCC(C)NC(C2(CO)CCOCC2)=O)ccc(Cl)cc1 c1(CC)cccc(-n2cc(C(CCC)NC(=O)C=CCc3csnc3Cl)nn2)c1 Cc1ccc(CNC(=O)C(C2CCCO2)NC(=O)CCc2cncn2C)nc1C C=CCCC(C(=O)OC)NC(=O)C(CCC)NC(=O)CC1COCCO1 C(=O)(C1=CC2(CN(C(=O)C(C)(O)C(F)(F)F)C2)OC1)NC(CC)(C)C(F)(F)F c1(COC)nc(NCC(C2CCCC2)NC(c2cc(C)oc2C)=O)cc(O)n1 C1(CN(C(=O)CCN2CCC(F)C2)C)CCN(C(c2scnc2Cl)=O)C1 c1(C(N(CCNC(C(c2ccc(C)cc2)C)=O)C)=O)cccc2cnnc(O)c12 N1(C(c2c(C(C)C)scn2)=O)CCC(CC(C)NC(=O)C(C)(C)CN(C)C)CC1 N1(C(c2c(C)ncs2)=O)CCC2(CC1)CC2CNC(C1(F)CC1(Cl)Cl)=O C(=O)(C1CCCc2ccnn21)N1CC(Nc2ccccc2)CC(C)C1 N1(CC(=O)OCCCC)CCC(S(=O)(=O)N(C)C)C1 C(=O)(C1SCc2cccnc21)NCC(C)(CO)NC(=O)CN1CCOCC1=O CP(C)(=O)c1ccc(C(N2CCOCC2CCNC(C2CC(CC3CC3)C2)=O)=O)o1 CN1CCCC1(C)C(=O)N(CC(CO)(CO)NC(=O)COC1(C)CCCC1)C N1(C(c2n(C)cnc2)=O)CCC2(CC2C(N2CCCN(CCO)CC2)=O)C1 c1(C(=O)NC23CCC(C(=O)OCC)(CC2)C(CN)O3)c(C)[nH]c2c(OC)cccc12 Cc1cc(C(=O)NC2CC2CNC(=O)CCCC2OCCO2)c(O)nn1 C1(C)(NC(c2n(C(CC)(C)C)nnn2)(CC)C2CC2)C(C)(C)C1(C)C n1(CC(=O)NCC(CNC(C2(CC)CCC2)=O)F)ccc(=O)c2ccccc12 C=CC1CCCCN1C(C1CCOCCN1C(=O)C(C)N=[N+]=[N-])=O C1(CNC(c2cc(C)c(N)cn2)=O)CC2CCC1N(C(=O)COC1CCOC1)C2 C1(NC(CCC)=O)CCC12CCN(C(c1cnn(C(C)C)c1C(F)(F)F)=O)CC2 Cc1nocc1CC(N1CC(O)(CNC(C2CC2[N+](=O)[O-])=O)C1)=O c1(NC(=NC)NCCC(C(F)(F)F)OC)cnc2c(Cl)cnn2c1 c1(C(N2C(CNC(=O)CC3CCCC3)CCC2)=O)cc(-n2cccc2)ccn1 N1(C(C(n2cc(C3(C)CCCC3)nn2)C)=O)CCC(Cc2ccccc2)C(F)(F)C1 CC1(CNC(c2csc(C(F)(F)F)n2)=O)CCCN1C(=O)C1=CCOC1 C1(C(N2CCC(CN(c3ncncc3Cl)C)CC2)=O)CCc2nnn(C)c2C1 C1(NC(c2cc(C3CC3)[nH]n2)=O)CC2CCC(C1)N2C(=O)CCCC1CCCO1 N1(C(C2CCCC2)=O)CC2(CCN2C(C2CCC2C(F)F)=O)C1 Cc1ccc(F)c(C(=O)NC2CCC(CNC(=O)CC3(C#N)CC3)C2)c1F CN(CCCC(=O)NCC1C2CN(C(C3CCCC3C3CC3)=O)CC12)N=O N1(CC(COCCCCC)O)CCc2cc(OC)cc(C(=O)OC)c2C1 Cn1nc(C(c2nnnn2C)NCC2CC(=C3CCC3)C2)c(Br)n1 C1(C(CNC(=O)N(CCN(C)C)C2CC2)OC2CCCC2)(OCC)CCSCC1 C(CC(=O)N(C)CCOCC1(NC(c2ncc[nH]2)=O)CC1)NC(COC)=O C1(C(=O)NCCC2(O)CCN(C(C3CCSC3)=O)CC2)CN2CCCC2CO1 C(=O)(C1CCSc2ccccc21)NCCOCCCN(C(C=CCC)=O)C C=CC(C)(O)CC(=O)NC1CN(C(C2(n3cccn3)CC2)=O)CC1CC1CC1 C=C(Br)CC(=O)N(C(c1ccccc1)CNC(C1CC1CC)=O)C CCCC(C)CCCC(=O)N1CCC2(CC1)CC(NC(C1CN(C)CCO1)=O)C2 N1(C(C2(OC)CC(C)(C)C2)=O)CCC(NC(=O)Cc2ccns2)CC(O)C1 S(=O)(=O)(c1cccc(C(=O)N(C2CCCC2)C)c1)N(C(C)C)CCC1CCCO1 c1(OC)ccc(Br)cc1C(C(=O)NCC1CC1)N(C1CC1)CC1COC(C)(C)O1 n1(C(COC)C)cc(C(=O)NCC(CO)NC(c2cn(C)cc2C)=O)c(C)n1 Cn1ccc(C(=O)NC2COCC2CC(N2CCC(CO)CC2)=O)cc1=O C1(NC(CCC#C)=O)CC2CC1CC2C(N1CCCOC(CC)C1)=O C12(CNC(c3cc(COC)on3)=O)CCC(C1)N(C(C1(C)CCCNC1=O)=O)C2 Cc1cccc2[nH]cc(C(=O)NC(C)(C)CNC(=O)C(O)C(C)C)c12 N1(C(C(=Cc2ccccn2)C)=O)CC2CC(NC(=O)C=Cc3ccc[nH]3)CC1C2 C1(CNC(CC(CC)(F)F)=O)COC(C)(C)CN1C(c1cnnc(C2CC2)c1)=O N1(C(c2nccc(CC)c2)=O)CC(NC(C2CC(=C3CC3)C2)=O)CC2(CCC2)C1 c1(C(N(C(CNC(C(C(C)C)NC(C)=O)=O)C)C2CC2)=O)cc(C)cc(C)c1N c1(C(N(CC(C)NC(c2coc(C#N)c2)=O)CC)=O)cnc2c(c1)c(C)nn2C c1(C(=O)NCC(CCOC)NC(CC(=C)Br)=O)ccc(OC)cc1 N1(C(C2(COC)CCOCC2)=O)CC2CCC1C(NC(c1c(C)ncn1C)=O)C2 c1(SC)cn(C)nc1C(=O)NC1CC(CNC(C2CCOC2(C)C)=O)C(O)C1 C1(C(=O)NCC2CC(NC(C3N(CC)CCCC3)=O)C2)CC2(CCCC2)C1 N1(C(C=C(COC)C)=O)CC2(CCC2)CC1CNC(c1ccn(C)n1)=O c1(N2CCCN(C)CC2)nc(N2CCC(S(=O)(=O)N(C)C)CC2)c2sccc2n1 C1(CCC=C)(C(N2CC3CC3C2)=O)CN(C(=O)CSCCC(C)C)C1 C1(C(N2CCC(C)(NC(c3cc(CC)[nH]n3)=O)C2)=O)CCc2nnnn2C1 C=CCCC(C(=O)NCn1cnnc1CC)NC(=O)C(C)NC(=O)NC C(C1c2ccsc2CCN1C(C1(F)CCCCC1)=O)NC(c1cc(C)ncn1)=O C1(NC(CSCC#C)=O)CCCC(N(C)C(c2nnn(C)c2CCC)=O)C1 CCC(CC)(C(=O)NCCN(C(=O)COCC(F)F)CC1CC1)OC N1(C(C(CC)N(C)C(c2ccc(CO)cn2)=O)=O)CCC(OC)CC1 c1(-n2c(CC3CCC4(CC4)C3)nc(-c3c(C)n[nH]c3)n2)cc(F)c(F)c(F)c1 c1(CCC(=O)NCCC(CCNC(c2n(CC)ncc2)=O)C)cc(C)cc(C)c1 c1(N(CCOC)Cc2nc(O)c(C)s2)cc(=NCc2ccccc2)[nH]c(Cl)n1 C(=O)(CCCCCS(N)(=O)=O)NCC(C(C)C)(C)NC(c1cnc2n1CCC2)=O C1(CC#C)(C(=O)NC(C)C(C)(C)CN(C)C)CCN(C(c2c[nH]ccc2=O)=O)C1 c1(C(=O)NCC(CC)(C)NC(C2CCCO2)=O)cc(C)n(-c2cnn(C)c2)c1C CC(C)(F)CCC(=O)NCC1(C)CCCN(C(C2(F)CCCC2)=O)C1 C1(NC(C2(C)CC(=C)C2)=O)CCC(C(=O)NCCC2CCCO2)CC1 N1(C(c2cc(CC)on2)=O)CCN(C(=O)CC(O)CN(C)C)CCC1C c1(CC(=O)N(CCCNC(C(C)SCC)=O)CCO)ccc2oc(C)nc2c1 N(C1CN(C(=O)C=CCF)CCc2ccccc21)C(C(C1CCCC1)OC)=O N1(C(c2cnc(C)[nH]2)=O)CCOC(CCNC(=O)C(CO)NC(=O)C(F)(F)F)C1 N1(c2onc(-c3c(C)ccnc3)n2)CCCC(CO)C1C CCCCC(F)C(=O)N1CCC(C)(C)C1CC(=O)NCCC1=CCOCC1 C(C(=O)NCC(C)CN(C)C(C1CCSC1)=O)(C1CC1)OC C(=O)(CCC(=O)C(C)(C)C)N1CCC(C)C(NC(C2CC2(F)F)=O)C1 c1(CC)cc(C(=O)NC2CC(F)(CNC(=O)CC(C)OC)C2)cc(F)c1 CC(C)(C)C(C(=O)NC1CN(C(=O)CSC(F)(F)F)CC1F)n1ccnn1 Cc1nccc(C(=O)NC2(C)CC(NC(=O)CCCn3ccccc3=O)C2)c1N N1(CC(=O)NC2CCC(CNC(c3ccsn3)=O)C2)CCn2ccnc2C1 Cc1cc(S(C)(=O)=O)cc(C(N2CCCC2c2cn[nH]c2)=O)c1C c1(C(N(CCCOCCNC(CC(C=C)C)=O)C)=O)cccc2c1OC(C)C2 c1(C(CNC(CNC(C(CC)C)=O)=O)NC(=O)Cn2cncn2)cc(F)cc(Cl)c1 c1(C(N(CC)CC2CCCN2C(=O)C(CO)N(C)C)=O)cccc2c1OC(C)C2 N1(C(c2c(CC)csc2)=O)CCN(C(C2(F)CC3(CCC3)C2)=O)CC1CO C1(NC(C2N(C)CC(C)(C)C2)=O)CC12CCN(C(c1ccn3ccsc13)=O)CC2 c1(C(N2CCN(C(c3ccc(C(C)=O)[nH]3)=O)C3C2C3)=O)cc([N+](=O)[O-])ccc1Cl C1(OC)CC(CNC(c2n[nH]cc2C)=O)N(C(c2c[nH]nc2C)=O)C1 C(=O)(CC(C)(C)C(F)F)NC(CC(=O)NC1C(C)CN(C)C1)C(F)F S(=O)(=O)(c1cc2oc(=O)[nH]c2cc1F)N1CC(C)CC(C(=O)OC)C1 N1(C(C(C)Cc2cnc[nH]2)=O)CC(O)CC1CNC(c1ccnnc1O)=O c1(CNC(C2CC23CCOCC3)=O)cccc2nn[nH]c12 N1(C(CC=CC(C)(C)C)=O)CCC(N(C(=O)Cn2cnc(=N)[nH]2)CCO)CC1 c1(C(=O)NC2CN(C(CN(C3CC3)CC)=O)C(CSC)C2)ccn2ccnc2n1 Cc1cc(C(N2CC(NC(=O)C(C)(C)CC3CC3)CC2CO)=O)nc(O)c1 N1(C(C2CC(=C)C2)=O)CCCC(C)(NC(C2CCCCN2S(C)(=O)=O)=O)C1 C=CC(CCC)CC(=O)NCCCOCCNC(c1cc(F)c(Cl)cc1Cl)=O C1(NC(c2ccon2)=O)CC2CC(NC(C3CCC3c3ccc(F)cc3)=O)C1C2 N1(C(C(C)CC(N)=O)=O)CC2CCC1(CNC(=O)CNC(C1CC1C)=O)CC2 c1(C(N2CC3(C(NC(CCSC)=O)CC3)C2)=O)cc(F)c(F)c(C#N)c1 C1(NC(C2CSC2)=O)C(CN=c2[nH]ncs2)CCC12CCC2 C1(CNC(C(C)C)=O)CN(C(=O)Cc2ccc(F)cc2)CCC1C c1(C(=O)NC(C2OCCN(C(CNC(=O)OC)=O)C2)C)cc(=O)c(OC)c[nH]1 C1(NC(c2ccc(OC(C)C)nc2)=O)COC2(C1)CN(C(c1c[nH]cc1Br)=O)C2 C1(CC)CCC(C(N2CCC(OCCNC(=O)CN3CCNC3=O)CC2)=O)CC1 CCC(CC)CCCC(=O)N1CC(O)(CNC(=O)CCNS(C)(=O)=O)C1 Cc1c(F)ccc(Cl)c1C(=O)NC1CC(C)N(c2ncnc3[nH]cnc23)C1 CCC(=O)CCC(=O)NC(C)(CSCOC)C(=O)N(CC(O)CN(C)C)C c1(C(=O)NC2CC(NC(C(C(=O)NCC)(C)C)=O)C2)cc(O)c(OC)c(C#N)c1 N1(C(C2CCCN2CC(F)(F)F)=O)CCC(c2ccc(Br)cn2)CC1 c1(C(C(=O)N(C2CCN(C(C3CC34CCOC4)=O)C2)CC)C)ccc(C#N)cc1 c1(C(=O)NC2C(CNC(c3cc(C)nc(O)n3)=O)C2)ccc2oc(C)nc2c1 C(C(C)(C(=O)NC1CC(C(C)O)C1)NC(C1C2CC(=O)CC12)=O)SC c1(OCC=C)ccc([N+](=O)[O-])c(C(N2CC(CNC(=O)C(C)(C)C)C(C)C2)=O)c1 c1(C(N2CCC(O)(CNC(C3(COCC)CC3)=O)C2)=O)ccc2nn[nH]c2c1O c1(CC(=O)NC2(CCNC(C3C(OCC)C3)=O)CCC2)ccccc1C(C)C N1(C(CCC2(C)CN(C(=O)C3=CCSC3)C2)=O)CCOCC1C1CC1 C(=O)(C(F)C(C)CNC(c1ccncc1)=O)N1CCC(CCC#C)CC1 C1(NC(C(C=C)(C)CC)=O)CC2(CCN(C(=O)CCOC(C)C)CC2)C1 c1(SCC)cccc(CC(=O)NCC2CC2NC(c2cccc(CO)n2)=O)c1 Cc1cc(C(=O)NC2CC(CNC(=O)C(F)(F)CO)C(O)C2)c2ccccc2n1 c1(C(=O)NCC2(C)CCC(NC(C(CC)OCC)=O)CC2)cc(C)c(F)cc1O c1(OCC)ccc(CCC(C)NC(c2cnc(-c3ccccc3C)s2)=O)cc1 C1(N(C(=O)C=CC(F)(F)F)CCC)CCN(C(=O)CCCN2CCCC2)C1 c1(OCC(=O)NC2C(NC(C3(C)CC(F)(F)C3)=O)CCOC2)ccc(F)cc1Cl CC1CCC(O)C(NC(C2C(NC(=O)CNc3ncccn3)C2(C)C)=O)C1 N1(C(c2cc(C)ncc2C)=O)CCN(C(C2(F)C(C)(C)C2(C)C)=O)CC(C)(C)C1 CC1(NC(=O)CC2CCCC2)CCCN(C(=O)CCS(C)(=O)=O)C1 C1(CNC(C(CCC2CC2)NC(=O)CC2CSC2)=O)CC2(CCO1)CC2 c1(C(=O)NCC(C2CC2)NC(CN(C2CC2)CC)=O)c(C2CCCC2)noc1C C1(NC(C2C=CCN2)=O)CC2CCC(C1)N2C(c1cc(C2CC2)on1)=O N1(C(C(CC)(F)F)=O)CC2CN(C(c3cn(C)nc3C(C)C)=O)CC2C1 c1(C(=O)NCCCN(C(c2cnc(NCC)s2)=O)CC)cc(SC)ccc1O N1(C(c2cc(COC)on2)=O)C2CCC1CN(C(=O)CSc1n[nH]c(C)n1)CC2 C1(NC(c2c(CCC)cccc2)=O)CN(C(=O)CCCN=[N+]=[N-])CC(C)(C)C1 c1(SC)c(C(=O)NCC2C3CN(C(c4cccc(C)c4N)=O)CC23)cccc1F C1(C(=O)NC2(C3CCCN3C(C3CC=CCO3)=O)CC2)CCCCCCC1 Cc1nc(C)c(C(=O)NCC#CCNC(c2ccc(C(C)(C)C)nc2)=O)o1 C(=O)(CC(O)C(C)(C)C)NCC1CCCN(C(c2c(Br)cn(C)n2)=O)CC1 c1(C(N2CC(CC(CNC(C3C(=C)CC3)=O)(C)C)C2)=O)ccc(CCC)cc1 Cc1[nH]nc2c1CC(C(=O)NCCN(CC1C(CCC(=O)OC)C1)CC1CC1)CC2 c1(CC(=O)NCC2(C(=O)OC)CC2)ccc(F)cn1.C12CCC(C1)CNC2=O c1(C(=O)NC2CCN(C(c3cccc(OC)c3O)=O)C2)cc([N+](=O)[O-])ccc1C C(=O)(CC(O)CC(C)(C)C)NC(CCCC)CNC(c1c(C)ccc(F)c1N)=O C1(CNC(C2C(C(C)(F)F)C2)=O)CCCN(C(=O)CCSC2CCCC2)C1 Cn1cc(C2=NOC(C(=O)NC3CN4CCC3(C)CC4)C2)cn1 C(CCCCCNC(C1CCN(C2COC2)C1)=O)N(C)C(C1(C)CCCN1C)=O C(C(O)(CNC(=O)CCCCN(C)C(C1(C(=O)N(C)C)CC1)=O)CO)OC C1(CNC(c2cn(C(C)C)nn2)=O)(CO)CCN(C(c2ccnc(O)c2)=O)CC1 c1(CCC(=O)NC(C(C)NC(CCCSC)=O)(C)C)ccc(Br)cc1 N1(C(CCn2c(C)ccc2C)=O)CCN(C(c2sccc2C#N)=O)C2CC12 C(=O)(C1=CCCCC1)N1CC(OCCNC(c2cc(-c3cn(C)nc3)[nH]n2)=O)C1 C1(C(=O)NCC2C(NC(C=CC(CC)=CC)=O)CC2)COc2ccc(O)cc2O1 c1(C(N2C(CCNC(CC(C)C(F)F)=O)CSCC2)=O)ccn2ccccc12 C#CC1CC2CCC1N(C(C1(CC)CCCN1C(c1cc(O)nc(C)n1)=O)=O)C2 c1(OCC(=O)NCC2CC(C)N(C(c3nncs3)=O)C2)cc(Cl)ccc1Cl S(=O)(=O)(c1cccc(C(=O)NC2CC3CCC2N(C)C3)c1)NCCOC N1(C(c2c(C)noc2C2CC2)=O)CCC(NC(=O)CCC2CCCCC2)C(F)C1 C1(CC=C)(C(=O)OC)CCN(C(=O)NCC(c2nccn2C)CC)C1 c1(OCC)ccc2cc(C(N3CCCOC(c4ccccc4)C3)=O)[nH]c2c1 N1(c2cc(OCC)nc(C(C)C)n2)CC2C(C(=O)O)(C1)c1ccccc1S2(=O)=O N1(C(=O)CSc2ccccn2)CC2COCC2(CO)C1.C(=O)(CSC)O CCC(CC)(CC)C(=O)N1CC2(C1)CN(C(c1ccc(Br)o1)=O)C2 c1(OCCC(=O)NCCCCCNC(=O)C(F)C2CCOC2)cccnc1 C1(CNC(C2C(CC)C2)=O)CN(C(c2cc(N)c(C)cc2Cl)=O)CCC1(F)F N1(C(C2C(C(C)C)C2)=O)CC(C2(NC(C3COCCN3CC(F)(F)F)=O)CC2)C1 c1(C(CC)NC2CC(CN)C2)ccc(F)cc1 C(C(F)(F)CCC(=O)N1CC2OCCOC2C1)n1cc(C(COC)(C)O)nn1 CP(C)(=O)CCC(=O)N1CCC(C(=O)NCC(F)C2CCC2)(CO)C1 C1(CC(=O)NCc2c(CC)nco2)(NC(C2CC23CCCC3)=O)CC(C)(C)C1 N1(CC)CC(C(=O)NC2(CCNC(C3CC3CF)=O)CCCC2)CCC1=O Cc1cc(CC(=O)NC(C2CCCC2)CNC(=O)CC(=O)OCC(C)(C)C)n[nH]1 c1(C(N2CCN(C(C(CC=C)N(C)C)=O)CC2C)=O)cn(C)c(=O)nc1O c1(CCC(C)OC(c2ncsc2Br)=O)ccccc1 C1(CC)CC(C(=O)N(C)Cc2ccoc2)CCN1C(=O)CCCC1CCCO1 N1(C(CN(C)C(=O)C2CC2)=O)CCC2C(C1)CN2C(=O)Cc1csc(NC(N)=O)n1 N1(C(c2c(C(C)C)con2)=O)Cc2nccn2CC(NC(=O)Cc2cscn2)C1 CN1N=C(C(=O)N2CCN(C(c3ccoc3C3CC3)=O)CC(O)C2)CCC1=O CC(C)(O)C(O)CNC(C1CC=CCC1NC(c1scnc1Cl)=O)=O c1(NCC(C(=O)NC)C)nc(N2CC3CCC3C2)nc2c1cnn2C(C)C c1(C(N2CCC(O)(CCNC(C(C)(C)C(F)F)=O)CC2)=O)ccccc1[N+](=O)[O-] CCC(CCCC(=O)NCC(c1ccsc1)C)NC(c1csnn1)=O c1(-c2c(C(=O)OCC(CCC(=O)OCC)C)cccn2)c(F)cccc1F CC(F)(F)CC(=O)N1CCCCC1CCC(N1CC(CO)(CO)C1)=O C(=O)(C(CNC(=O)Cc1csc(C)n1)CC(C)C)NCCC1(COC)CC1 c1(CC)cc(C(N2C(C(=O)NC(CC)C(N)=O)CC2C)=O)c(C)o1 C(=O)(C1=CCC2(COC2)OC1)NCCCCCCN(C)C(C1CC2CCC2C1)=O N1(C(C2C(=C)C2C(=O)OC)=O)CCC(C)C1C(=O)NCCCCCSC(C)C C(N=c1nc(N2CCc3nn(C)c(N)c3C2)c2cnn(C)c2[nH]1)C1CC(SC)C1 N1(C(c2c(C)nncc2)=O)CCCCCC1C(=O)NC(C)CF CC1CC(NC(=O)C(=O)Nc2cnc3n2CCOC3)CC(C)S1(=O)=O N1(C(c2ccc(C#C)cn2)=O)CC2(CCN(CC(=O)Nc3cnccn3)C2)C1 N1(C(c2cc(C)on2)=O)CC(F)(F)CC1CCNC(=O)CCCNC(N)=O CC1CC(NC(=O)CCOC2CN(C(=O)Cn3cnnc3O)C2)CS1 c1(C(=O)NC(CNC(C(c2ccc(C)s2)C)=O)C2CC2)cnc(O)c(Cl)c1 N1(C(CC=CCC)=O)CCN(C(c2ccncc2Br)=O)C(c2cn[nH]c2)C1 Cc1cc(C(=O)NC(c2ccccc2)CNC(c2ccnnc2)=O)cc(C)c1N c1(C(=O)NCCOCC(C2CC2)OCC)cc(C)ccc1OC c1(N2CC(CN(C)C(C3(F)CCC3)=O)OCC2)nc(Cl)ncc1Br C=CC1CN(C(=O)C(C(C)C)c2cnc(C)s2)CC1NC(=O)CCC N1(C(C(F)=CCC)=O)C(C(=O)NCc2conc2C2CC2)CCC12CC2 c1(C(=O)NC(c2cccc(F)c2)C)ncccc1NC(c1ncccn1)=O c1(C(N2CCC(NC(CSCCOC)=O)C2)=O)ccc(-c2ccccn2)c(F)c1 c1(SCC(=O)NCC(C2CC2)NC(c2c(CC)sc(=N)[nH]2)=O)ccc(C)c(C)c1 CC1C=C(C(=O)NC2(C)CCN(C(c3c[nH]ccc3=N)=O)C2)CC1 C1(C(=O)NC2C(CNC(c3cc(Br)co3)=O)CCC2)CC2C=CC1C21CC1 N1(C(Cn2ccc(C)n2)=O)CCCN(C(=O)C=C2CCC(C)CC2)CC1C O=C(N=c1ccn(C2CCC2)[nH]1)C1c2c[nH]nc2CN1C(=O)C#CC1CC1 CCCC(F)C(=O)NC1CC(C(N2CC3CC3(CO)C2)=O)C1(C)C C1(C(=O)NCC2(C(=O)NCC(C)(C)OC)CC2)CCCCC(=O)N1 C(=O)(C(C)CC(=O)Nc1cccc(NC(c2ccc(Br)c(C)n2)=O)c1)OC N1(C(c2ccc(C(C)=O)[nH]2)=O)CCN(C(c2cnn(C3CC3)c2)=O)CC1CF C123COCC1CN(C2)C3=O.CC(C)CCN1CC(NC2CC(N(C)C)C2)C1 c1(C(=O)NCC(C2N(C(C3C(OC)CC3)=O)CCC2)(C)C)snc(Cl)c1Cl N1(C(C(C)C)=O)CC2CC2(C(=O)NCC2CCN(C(=O)C(C)C)C2)C1 C(C(CC(=O)NC1CC(F)(CNC(=O)C=CCO)C1)C(F)(F)F)N(C)C c1(C(N2CC(N(C)Cc3ncccc3F)C2)=O)ccc2[nH]nc(Br)c2c1 n1(CC(=O)NCC(N(C(C=CCOCCOC)=O)C)C2CC2)ccc(CO)n1.C1CC1 CCC(c1ccc(C)cc1)=CC(=O)NCC(C1CC1)NC(c1sc(O)nc1C)=O N1(C(CCC(CC)NC(=O)C(F)C(F)(F)F)=O)CC(=O)NCC12CC2 C1(CCNC(C=COCC)=O)CSCCN1N(c1ncncc1F)CC.C(C)=O c1(OC)nccc(=NC(=O)C2CCCC2NC(=O)CCc2ccc(C)c(C)c2)[nH]1 c1(COC)nc(NCc2cccnc2N)cc(N2CCSCC(C)C2)n1 N1(CC(=O)NC(CCCC)CNC(c2cc(Cl)n(C)n2)=O)C(=O)NC(C)(C)C1=O N1(C(c2cc(C)n(C)n2)=O)CCC2CC2(NC(c2ccc3ncsc3c2)=O)CC1 C(=O)(CCN=C(NCCc1ccccc1F)NCC(C1CC1)SC)NC c1(C(=O)NCC(CCCC)NC(=O)CN2CC=CC2)[nH]c2ccccc2c1OC CC1CC(CNC(C2CCC(C)(C)C2)=O)CN(C(=O)CCC(N)=O)C1 C=C1CC(C(=O)N(CC(=O)NCC(C2CCCO2)O)C2CC2)(COC)C1 N1(Cc2ncc(COC)s2)CC(C)CSc2ccccc21 O=C(CCCC1CCOCC1)NCC1CN(C(=O)CN2CSCC2=O)C1 c1(-n2ncc(NC(N(C3CCOC3)CC)=O)c2)ccc(Br)cc1 C1(O)(C(=O)OC(C)(C)C)CC2(CCN(N(CCC(C)c3cn[nH]c3)C)C2)C1.C=O C1(C(=O)NCC(C)(C)NC(c2nnc(O)cc2O)=O)CCC(=O)N(C2CC2)C1 c1(C(=O)NC(C(C)OC)CC(=O)NC2C3CCCOC23)cccc2ccnn12 CC(C)(Cc1cn(CC2(O)CCN(C(=O)Cc3ccns3)C2)nn1)C(=O)O N1(C(C(=Cc2cccnc2)C)=O)CCC(CN(C)C(C2CCCS2(=O)=O)=O)CC1 c1(C(=O)NC2C(C)N(C(=O)CSC3CC3)CCC2)cc2cc(Cl)sc2[nH]1 C1(NC(c2n(C(C)C)ccn2)=O)CCC2(CC1)CN(C(C1CCCCC1C)=O)C2 c1(CCC(=O)NC(CNC(C(C2CC(F)(F)C2)OC)=O)C)ccc(N(C)C)cc1 N1(C(C2C(CC)C2)=O)CCCC2CN(C(=O)CCCN(C)C)CC12 c1(C(N2CCOC(C)C2)C(=O)Nc2c(C)cccc2)ncc(Cl)cc1F CCC(CC(=O)NCC1C2CC2CN1C(=O)COCC(F)(F)F)NC1CCCC1 C(=O)(C1=NOC(C)C1C)NC(C(C)C)CCN(C)C(C1CC=CCC1C)=O C(CCC(N)=O)(C(=O)N(C)Cc1ncnn1C)n1cc(C(C)N(C)C)nn1 C1(F)(C(N(CCCN(C(c2ccc(CC)[nH]2)=O)C)C)=O)CC12CCCCC2 Cc1c(C2CCOCC2)n[nH]c1C(=O)NCC=CCNC(C1(CN(C)C)CC1)=O C12(C(N3CC(C4N(C(c5ccc(COC)s5)=O)CCC4)(O)C3)=O)CCC(CO1)C2 c1(CC(=O)NC2(CNC(=O)C(F)(F)C(F)F)CC2)ccc(O)c(Cl)c1 C1(NC(C2CC(OC)C2)=O)CCCC1CNC(=O)C=CI C(=O)(CC(C(F)F)NC(=O)CCCCOC)NC(C#C)CC c1(OC)ccc(C)c(C(N2CCCOC(CNC(=O)C(C)n3ccnc3)C2)=O)c1 CC1CN(C(=O)C(c2cccc(Cl)c2)(F)F)CC1NC(=O)C(C)(C)C c1(NCC2(OC)CN(C(C3C(COC)C3)=O)C2)ncc(C#N)c2ccsc12 C1(C(C)C)OCCC1C(=O)N(CCC(=O)NCC(O)C1CC1)C Cc1cc(C#N)cc(C)c1C(=O)NCC(C)CNC(=O)C(F)C1CCOC1 CC(C(=O)N(CCCCNC(C1CCCN1C(=O)CC(C)(C)C)=O)C)P(C)(C)=O Cc1cc(NCC2(C)CCCN2C(C2(c3ccncc3)CCC2)=O)nc(C)n1 CC(CC(=O)NCC(C)(CO)NC(C1(Cc2cccc(Cl)c2)CC1)=O)C(F)F C1(C(=O)NCc2nc(N(C(C=C)=O)C)sc2)CCCN(c2nncs2)C1 c1(C(N2CC(CN(C)C(C3(CC4CC4)CC3)=O)OCC2)=O)ccn2c1CCC2 CC1(C)CCN(C(C2CCCC2)=O)C1CC(=O)Nc1cccc(O)c1F c1(OCC(=O)NCC(C)N(C(Cn2c(C)ncc2)=O)C)ccc(F)nc1 C12(C(N3CCCC(CC=C)(NC(c4ccc(F)s4)=O)C3)=O)CCC(C)(CC1)CO2 c1(C(C(=O)NCC(C)CN2CCCC2)NC(=O)C=CCN2CCCC2)ccccc1 Cn1nccc1CCC(=O)NC1(CCCCNC(=O)C(F)n2ccnc2)CC1 Cc1ccc2c(CC(=O)ON3CCC(C(=O)OC(C)(C)C)C3C(C)C)c[nH]c2c1 c1(C(N2C(C3(NC(C(C)C(C)(C)C)=O)CC3)CCC2)=O)cncc(N=[N+]=[N-])c1 n1(CC(=O)Nc2cccc(NC(=O)CO)c2)ncc2cc(Br)cnc12 N1(C(CCNC(C(CC)OCC)=O)=O)CC(C)CCCC1C N1(C(C(c2ccc(F)cc2)C)=O)CC(CNC(=O)CSc2nncs2)CC(C)C1 C(C)(C1CCCCC1)=CC(=O)N(CCCNC(C(CC1CC1)OC)=O)CCO c1(OCCOC)ccc(Cl)cc1C(=O)NCC(O)CNC(=O)Cc1cc(C)ns1 N1(C(c2c(C(N)=O)coc2)=O)CC2(C(=O)NC3CCCC(O)C3)CC1CO2 C1(NC(=O)NCCOCCCOC)Cc2cc(OC)ccc2O1 C(=O)(C1=NC2=NCCCN12)N1C(CNC(C(C(C)C)OCC)=O)CCC1 C(=O)(C(N)CCO)NC(c1ccc(Cl)cc1)CC(=O)OCC C#CCC(CC(F)F)NC(=O)C(C1(O)CCCCC1)NC(=O)C(=O)C1CCCC1 CCCCC(C)(C)NC(=O)C(C)NC(=O)CCCSC C1(CCC)CN(C(c2occc2C(C)C)=O)CCN1C(=O)C(CSC)NC(C)=O C1(C2CCCN(C(=O)Cc3cccnc3)C2)(NC(=O)CCCF)CC1 C1(F)(C(N(CCC(C)O)C)=O)CCCN(C(C2CC23CCCC3)=O)C1 N1(C(C(C2CCC2)OC)=O)C2CCC1CC(O)(CNC(c1c[nH]nc1C)=O)C2 c1(C(N2C3C(NC(c4n(C(C)C)ccc4)=O)CC(C3)C2)=O)nccc2n[nH]cc12 c1(COC)cc(C(=O)NCC2(F)CC(NC(=O)C(C)Cc3ccncc3)C2)on1 C1(NC(C2N(CCC)CCC2)=O)CC2CCC1CN(C(C1CC(OC)C1)=O)C2 c1(OC)ccc(-n2nc(-c3ccc(Cl)s3)nc2Cc2cn(C(C)C)nn2)cn1 n1(CC(N2C(CNC(C(C)NC(CC)=O)=O)C(C)CC2)=O)ncc(C#N)c1N N1(C(=O)CC2CC(F)(F)C2)CCCC(N(C(C2CCCS2)=O)CC2CC2)C1 c1(C(=O)NC(CC)CNC(c2cc(Cl)c[nH]2)=O)ccc(C(F)F)cc1 N1(C(CCNC(COC)=O)=O)CC=CCC1NC(=O)OC(C)C(=O)N(C)C C(=O)(C1CCCc2nn[nH]c21)NCCOC1CN(C(c2c(C)cncc2)=O)C1 CCC(C)C(CCN=c1cc[nH]cc1S(=O)(=O)NCCC#N)SC C1(NC(C2CN(C(C(COC)COC)=O)CC2(F)F)=O)CCCCC1N=[N+]=[N-] CC(C)S(=O)(=O)C(C)C(=O)NCCN(C(c1cnc2ncccn12)=O)C(C)C c1(-c2ccc(C(=O)NC(CC)C(=O)OC)nn2)ccc(S(=O)(=O)F)cc1 C1(CNC(CSc2ccc(CC(C)C)cc2)=O)CN(C(=O)CCC#N)CCCO1 C1(C(=O)NC2CCN(C(C(C=C)CC)=O)CC2C(N)=O)CCc2ncnn2C1 c1(NC(C2(CC)COC2)=O)cccc(CNC(=O)COC2CCCOC2)c1 c1(C(=O)NC(C(C)NC(c2cc(Cl)cnc2O)=O)C)[nH]c2ccccc2c1C#N c1(SCCC)ccccc1.C1(C)C=CCN1 N1(C(C=CC)=O)CCCC2(CC(NC(=O)C=Cc3ccccc3F)CO2)C1 C(C(=O)NC(CC)CCO)(C(C)C)NC(c1ccc(CC)s1)=O N1(C(c2cnn(-c3ccccn3)c2)C(=O)NCCCC)CCC(O)(C(F)F)CC1 c1(C(N(CC(CC)NC(=O)CC2CC(C)(C)CO2)C)=O)ccc2c(c1)CC2 c12ccc(cc1C#N)S(=O)(=O)NCCC(C(C)C)N2C.N(C)(CC=C(C)C)CC S(=O)(=O)(c1ccc([N+](=O)[O-])c(Cl)c1)N1CC2CN(C(CCC(C)=O)=O)C2C1 c1(CCC)cc(C(=O)NCC2COC(CNC(c3c(C)cnn3C)=O)C2)n(C)n1 Cc1cc2c(NC(C3CCCN3C(=O)CCc3ccccc3F)=O)ncnc2[nH]1 c1(C(N2CC3C(C2)N3C(C2(F)CCOCC2)=O)=O)ccc(F)cc1Br C(=O)(CC(C)(C)CNC(C12CCC(CO)(CC1)C2)=O)N1CC(CC)C1 C1(NC(CN(C(C2CCN(CC)C2)=O)CC2CC2)=O)CCCCCCC1 N1(C(C=CC)=O)CCCC(C2CCN(C(c3c(Br)n[nH]c3C)=O)C2)C1 c1(C(=O)NC2CN(C(CC(C)CF)=O)CC2F)ccc2cncn2c1 C=C(C)CCCC(=O)N1CCCCC1CCCNC(C1CCS(=O)(=O)N1C)=O N1(CCNC(CNC(C)=O)=O)CCN(C(C2(CO)CCCCC2)=O)CC1 C1(CNC(CCc2nnc(C)o2)=O)N(C(C2C3CCCC23)=O)CCCC1(C)C CC1(C)CC=C(C(=O)NC(CN=[N+]=[N-])C(=O)NCCC2CCCC2)CC1 c1(OC)ccc(CN2CCC(O)(c3ccc(C(F)(F)F)cc3)CC2)cc1I N1(C(c2cc(C(C)(C)C)no2)=O)CCC2(CCCN(C(=O)CNC(N)=O)C2)C1 c1(CC)ncnc(CC)c1C(N1CC(CCNC(=O)CC2CCCO2)C1)=O N1(C(C2(C)CCSCC2)=O)CCC2CC2(C(=O)NC2CC3(CCCC3)C2)CC1 N1(c2ncc(OC)c(C)n2)CCc2n[nH]c(C=CC(=O)N(C)C)c2C1 C12(CNC(=O)Nc3ccc(OCCF)cc3)CCCC1C2(F)F C1(OC)CCCCN(CC(=O)NCC(C)(CC(C)C)NC(C2CC=CC2)=O)C1=O C(C(C)C(C)C(=O)NC1CCC(CNC(c2cccc(=O)n2O)=O)C1)OC CC1(O)CCC(CC(N2CC(NC(=O)C(O)C(C)(C)C)C3(CC3)C2)=O)CC1 c1(C(N2C3CN(Cc4c(C)nc[nH]4)CC32)=O)c(Br)cc([N+](=O)[O-])cc1[N+](=O)[O-] c1(C(=O)NC2C(C)CCN(C(C(C(C)C)O)=O)C2)cnn2ccn(C)c12 CCC(C)C(O)C(C)C(=O)NCC1CC(C)CN(C(c2c(C)cccc2O)=O)C1 Cc1scc(C(=O)NC2C=CC(CNC(C3CC(n4ccnc4)C3)=O)C2)c1N c1(C(=O)NC(C)(CNC(=O)C(O)C2CCCC2)CO)ccnc2ccc(O)cc12 N1(C(C(COC)OC)=O)CCN(CCNC(=O)C(C)(C)CN2CCOCC2)CC1 CC(C)CC(C)CC(=O)NC1CCC(N(C)C(c2ccc3ncccn23)=O)CC1 c1(NC(N2CCCC2)CC)nc(=NC)[nH]c(=NCc2ccc(N)cc2Cl)[nH]1 N#Cc1cc(C(=O)NC2C3CCC2N(C(C2CCCN2C=O)=O)C3)ccc1F CC(CC(=O)NC1CC2CCCC2C1)C(C)(C)NC(=O)CCC(C)(C)N(C)C c12ccc3nc([nH]c3c1)S2.CC1(C)CN(c2ccccc2)CC1c1cccnc1 N1(C(C23CCC(OC)C2C3)=O)CC2(CO)CC1(C(=O)NC1CCCCCC1O)C2 C1(C(C)(C)NC(c2cc(C)oc2)=O)CCN(C(c2cnsn2)=O)CC1 C(=O)(C1CCCc2c[nH]nc21)N1C(C)(C)C(NC(=O)CCCCO)CC1 c1(C(=O)OCC(=O)N(C)Cc2nccs2)cc(C2CCC2)nn1C.O CCC(C)(C)C(=O)C(=O)NC1CCN(C(c2ccn(C3CC3(F)F)n2)=O)C(C)C1 C1(C(=O)NC2(C)CC(NC(c3cc(Cl)ccc3F)=O)C2)CC2(CO1)CC(F)(F)C2 Cc1cc(C(=O)NC2CN(C(C3C4C(=O)OCC34Br)=O)C2)cnc1O n1(CC)c(CCNC(C2CCCCC2C(=O)O)=O)nnc1O c1(C(=O)NC(CNC(CCc2cccc(OC)c2F)=O)C)cc(Cl)c(O)cc1C c1(C(=O)NCCCC2CCCN2c2nnc(CO)s2)c(C(F)(F)F)cccc1F c1(OC)ccc2c(C(N3CCN(C(c4ccc(SC)o4)=O)CC3)=O)cnn2c1 C1(CN(CC(C)C)CC)CCN(C(=O)Nc2ccsc2OC)CC1 C1(CNC(C2(SC)CN(C(C34C(=O)C5CC3C4C5)=O)C2)=O)Cc2nccn2C1 CC(C)CC(C)CC(=O)N1CCN(C(=O)CCSC2CCCC2)C(CF)C1 c1(C(=O)OC)ccc2sc(N(CC(C3CCOC3)O)C(C)=O)nc2c1 N1(C(C(CC(F)F)N(C(C2(C(CC)=O)CC2)=O)C)=O)CCC(C2(C)CC2)CC1 N1(C(CC(=C=C)C)=O)CCC2(CC1)CC2(CO)CNC(C1CC1c1ccsc1)=O Cc1cc(C(=O)NCCN(C(C2CC(F)(CO)C2)=O)CC2CC2)ccc1F c1(C(N2CCCC(NC(c3ccc(C(C)C)o3)=O)C2C)=O)ccc2cc[nH]c2n1 c1(C(N2CC(C)(NC(COCc3cccc(C)c3)=O)C2)=O)ccc(O)c(Cl)c1 C1(C(=O)NC2CCN(C(CC)=O)C2)CCC(NC(=O)CCCN(C)C)CC1 N1(C(c2c(C)nc(C)o2)=O)CCN(C(C2CC2C(F)(F)F)=O)C(CCO)C1 c1(OCC)cc(CO)ccc1NC(c1ccc(=O)n(SCc2cccnc2)n1)=O c1(C(N(C2CCN(C(C3(C)CCNC3=O)=O)C2)CCO)=O)ccc(P(C)(C)=O)o1 C1(NC(c2c(C)sc(Cl)n2)=O)CC1C1CCCN(C(=O)CN2CCOCC2)C1 N1(C(c2cc(C)n(C(C)C)n2)=O)CCC(NC(c2cc(C3CC3)sn2)=O)C(C)C1 C1(NC(C2C(OC)CC2)=O)CN(C(=O)Cc2cc(Br)cs2)CCC12CCC2 CC(C)CC(CNC(=O)C=CC1CCCN1C)C(=O)NCC1(CO)CCCCC1 c1(NC(=O)CC2(O)CCN(Cc3cccc(Br)n3)CC2)[nH]nc2ncccc12 CC(C)(CS(C)(=O)=O)C(=O)N1C2CCC1CC(CNC(=O)CCc1ccoc1)C2 C1(NC(C=Cc2n(C)ncc2)=O)CN(C(c2sccc2Cl)=O)C2CCCC12 c1(CNC(C2(c3ccn(C)n3)CCOCC2)=O)cc(-n2nnnc2O)cc(F)c1 c1(NC2(C)CC(C)C2)cc(-n2nnnc2C2CC2)cc(F)c1 c1(C(N(C2CN(C(C3CCCOC3)=O)CC2(C)C)C)=O)c(F)ccc2c1OCO2 c1(OCC(=O)NCCN(C(C)C)C2CC2)ccc2ccccc2c1Br C(CCCCCCO)NC(CCC1N(C(CN(C(=O)OC)C)=O)CCC1)=O N1(C(C(C)Cc2ccccn2)=O)CCCC(CN(C)C(c2nocc2Cl)=O)C1 c1(C2C(C(N3CC(CNC(C(n4cnc(C#N)n4)C)=O)C3)=O)C2)cccc(Br)c1 C1(CC(=O)NC2(C#C)CCOC2)CN(C(=O)Cn2nnnc2C)CCC1C c1(C(=O)NC(C2CN(C(C3CC(S(C)(=O)=O)C3)=O)C2)C)cc2cc(F)ccc2[nH]1 CC1CN(C(C2CCS(=O)(=O)C2)=O)CCN1Cc1ccnc(Cl)c1 Cc1c(Cl)cnn1CC(=O)NC(C1CCCN1C(=O)CC1(OC)CCOCC1)C CC1(C)CCN(C(=O)CP(C)(C)=O)C1CC(N1CC(C2(C)CC2)C1)=O c1(N(C2CCC(C)(C)C2)C(=O)CC2C(OCC)CC2O)ccc(C)c(C)c1 C1(C)(c2nnco2)CC(F)(F)CN1C(=O)CCCCCF.Cc1nc(C2CC2)n[nH]1 CC1CN(C(=O)CC(C)(C)C#N)CCC1CNC(=O)CCC1CC(F)(F)C1 N1(C(C)C(=O)NCCC(O)CNC(c2cccnc2)=O)CCN(C)CC1 c1(CCNC(C(Cn2ccc(C)n2)C)=O)ccc(CNC(c2cnco2)=O)cc1 C12(CNC(CC(COC)(C)O)=O)CN(C(=O)Cc3coc(C)n3)CC1CCO2 c1(C(N2CCN(C(C(C)CC(N)=O)=O)C(CCO)C2)=O)cccc2c1nnn2C C1(C(=O)Nc2ncc(C)nc2)CC12CCN(C(c1ncccc1Br)=O)C2 N1(C(c2c(C)nc[nH]2)=O)CCC(NC(=O)C(O)Cc2cnc[nH]2)C12CC2 C(=O)(CCS(=O)(=O)CC(C)C)N1CC(C)CC(NC(c2cn(CCC)nc2)=O)C1 C(CC(C)C)(C(=O)NC(C(C)OC)=O)ONC(C1CCCN(C(C)=O)C1)=O N1(C(C(CSC)C)=O)CCN(C(c2ccc(=O)n(C)n2)=O)C(C2CC2)C1 c1(OC)ccc(C(=O)NC2C3CCC2N(C(C2CC(N(C)C)C2)=O)C3)c(C)c1 O=C1NC(=O)c2c(C(=O)NC3CCN(C(C4CC(F)C4)=O)C34CC4)cccc21 C1(C(=O)NCCOC2CCN(C(C3C(OCC)C3C)=O)C2)CCN(C)C(=O)C1 c1(-c2nc(CCC(C)C)nn2-c2cccnn2)cc2c(Cl)c(Cl)ccc2[nH]1 CC1CC2(CO1)CN(C(=O)CCCCNC(C1OC3CCC1C3)=O)C2 C1(NC(c2cncc(C)c2)=O)CN(C(c2cc(C)n(C)c2)=O)CCC1F C1(CNC(C2(CCC)CC2)=O)CC2(CC2)CN1C(=O)C(c1ccc(Cl)s1)=O N1(CC(=O)N(C2CC2)Cc2ccccc2)CCCC1C1CCCC1 C1(NC(C(CC(C)C)(C)C)=O)CC2(CCCN(C(c3nncn3C)=O)C2)C1 C(=O)(CCCC(C)(F)F)NC1C2N(C(C(CCSC)O)=O)C(CC2)C1 Cc1ccc(C(=O)NC2C=CC(CNC(C3CC(C(F)F)C3)=O)C2)n1C c1(NC(=O)CCn2cncn2)ccc2c(c1)CN(C(c1ccc(F)c(Br)c1)=O)C2 C1(C(=O)NC(CC)C(N)=O)CCN(C(=O)C(O)CC2CCCC2)CCO1 C1(NC(C2CCCCC2(F)F)=O)CC(C(F)(F)F)CN(Cc2cncc(O)c2)C1 c1(C(=O)NC2(CC=C)CN(C(=O)C(C)C#N)C2)ccc(C(C)C)cc1 C(=O)(CCC(C)(C)NCc1ccc(F)cn1)N1C(CC=C)(C(=O)OCC)CCC1 Cc1ccc(C(N2CCC(CO)(NC(c3cc(C#N)[nH]c3C)=O)C2)=O)c(F)c1 c1(C(N2CC(NC(C34CC(C)C3C4)=O)C(CO)CC2)=O)cn2c(n1)C(C)CCC2 Cc1nn2cc[nH]c(=O)c2c1C(=O)N(CC(O)CNC(=O)CN1CC=CC1)C C1(CN2CC3(CC(NC(c4ncn(CC)n4)=O)C3)C2)COc2ccccc2O1 N1(CCOC(C2CCCN(C3COC3)C2)=O)C(=O)NC(C)(c2ccc(Br)cc2)C1=O c1(CC(=O)NCCN(C(=O)C(C(C)(C)C)N(C)C)CCC)ccccc1S(C)=O N1(C(c2c(C#C)cn(C)n2)=O)CCC2CC(C1)CN(C(c1ncsc1CC)=O)C2 N1(CC)CCCC(C(=O)NCC(F)CNC(c2ccc(OC(F)(F)F)cn2)=O)C1 C(CCCCCC(=O)N1CCC(O)C12CCCC2)N(C)C(=O)C1CC1 c1(C(=O)NC2CN(C(C3(C)CCCNS3(=O)=O)=O)C2)cc2ccc(O)nc2s1 c1(CC)cc(NC(C2CC3CC3N2C(C2CCCS2)=O)=O)cc(F)c1 c1(OC)ccc2[nH]c(CN3CC(F)CC3C(=O)Nc3cc(C)cc(Cl)c3)cc2c1 C#Cc1cccc(CC(=O)NCC2CCN(C(C3CCS3(=O)=O)=O)CC2C)c1 C(=O)(CS(=O)(=O)NC1CC1)N(c1c[nH]nc1-c1cccnc1)C(C1CCCCC1)=O Cc1cc(CC2CCCN2S(=O)(=O)C(C)C(=O)OC(C)(C)C)ccc1F c1(CC(=O)NCC2OCCCN(C(CCC(C)(C)F)=O)C2)ccc2ccoc2c1 N1(C(CC(C(C)C)O)=O)CC2CCCC(C1)N2C(=O)C=Cc1ccc(F)cc1F N1(c2nnc(COCC)n2CC(F)(F)COC)CC2CS(=O)(=O)CC2C1 c1(C(N2C(CNC(Cn3c(C)cc(C)n3)=O)CCC2)=O)csc2c(Cl)cccc12 CC(C)(C#N)CC(=O)N1CCCC1C(=O)NC1(c2ncccn2)CC1 c1(NC(C(=O)NC(c2cc(F)ccc2F)CC)=O)ccnc(OC)c1F N1(C(CC(C(C)C)OCC)=O)CC2CN(C(c3ccnc(F)c3N)=O)CCC12 CCC(C)(C)CC(=O)N1C2CCC(C2)C1CNC(=O)COC1(C)CCOCC1 Cc1cc(CN2CC3CC3(NC(c3nc(C)c(C)nc3C)=O)C2)cc(C)c1Cl CCC(C)C(O)C(=O)NCCCN(CCCCNC(=O)C(C)CN(C)C)C CC(CCNC(=O)CCc1ccccn1)CCNC(=O)C(C1CCCCCC1)O N1(C(C=CC=CC)=O)CCC12CCCN(C(=O)C(c1ccccc1)OC)C2 C1(C(=O)NCCCOC2CCN(C(C3CC34CCOC4)=O)CC2)CC2(CSC2)C1 C1(COC)(CO)CCCN1CCN1CC(C)C(C)C1 C(=O)(C(O)C(C)(C)C)N1CC(SC)C(NC(=O)CCOc2ccccc2)C1 C(=O)(C1=Cc2ccccc2C1)NCCCCNC(C(c1c(C)cccc1)C)=O C1(CC)CN(C(=O)C=CSCc2ccco2)CCC1Nc1cc(C)nc(C)n1 c1(C(N(C2CN(C(C3CCSC3)=O)CC23CC3)C)=O)ccc2c(c1)CC(C)(C)C2 C1(CC)CCN(C(=O)C(=O)OC)C1CN1CCOCC1C(C)C c1(NCC2N(CC)CCC2)nc[nH]c(=NCC2(OCCO)CCCCC2)c1C CN1CC=CCC1CC(=O)NC1(CNC(=O)Cc2cncn2C2CC2)CCOC1 N1(C(C=CC)=O)CCC(C2CC2)C1CNC(c1nc(C2CCOCC2)oc1C)=O N1(C(Cn2cc(C(C)O)nn2)=O)CC(NC(c2ccnc(C3CC3)n2)=O)CC1C CN1CCc2cc(C(=O)NCCC3(NC(=O)C4CC4)CCCC3)ccc21 C(=O)(CC1CCOc2ccccc21)NCC(C)(CO)NC(=O)CCc1cn[nH]c1 c1(C(=O)NCC(O)CNC(C2CCC(C(F)F)CC2)=O)cc2ccc(Cl)cc2[nH]1 n1(CCC(N2CCN(C(CS(CC)=O)=O)CC2CCO)=O)ncc2ccccc12 c1(N(C)Cc2c(C)nn(C)c2)ncnc(N2CCN(Cc3ccco3)CC2)c1C C1(C(=O)NC2(CN(C(C(C3CCOCC3)OC)=O)C)CCC2)CCC(F)CC1 C1(C(=O)NC(CCN(C(C(C)NC(C)=O)=O)C)C)CC2CS(=O)(=O)CC2C1 CCCCC(C)C(=O)NCCOCCNC(c1cnc(C(C)(C)C)nc1)=O C1(NC(CCC(=O)NC)=O)CC2CC1CN(C(=O)CC1CC(OC)C1)C2 c1(C(=O)NCC23CC(NC(=O)C=Cc4cn[nH]c4)(C2)C3)cccnc1S C(C(CNC(=O)CC1(O)CCC1)C(F)(F)F)NC(CCc1cnc(C)s1)=O C1(C(=O)NCC(C)OC)CC(C)(C)CCN1C(=O)Cc1scnc1C N1(C(COC(C)C)=O)CC2CCCN2c2ccccc21 CN1CCCC(C(=O)NCC(O)CC(=O)NOC(C)(C)C)C1.c12cc(n[nH]1)C2 CON(CCC(=O)NCC(C)C(C)(F)F)C(=O)C1(C(C)(C)O)CC1 C(=O)(CCCC(C)NC(C1CC(=O)C1)=O)Nc1c(C(C)C)nsc1 c1(CC)nnsc1C(=O)N(C1CCN(C(c2ccc(C3CCCCC3)o2)=O)C1)C n1(CC)ncc(C(N2CC(NC(=O)CC3CCSCC3)CC2C)=O)c1Cl c1(C(=O)NC2C=CCN(C(c3c(C#N)nc[nH]3)=O)C2)cccc2nncn12 c1(C(=O)NCCCCNC(C2C3CC4C(C3)C24)=O)cc2ncccn2n1 c1(C(=O)NC2CC(C)CN(C(C3CC(F)(F)C3)=O)C2)nn(C)c2ccccc12 Cc1cc(NC(C2CCC(NC(=O)C=Cc3ccccc3)CO2)=O)nc(Cl)c1 c1(C(=O)NCCN2CCN(C(C3C(C)(C(F)F)C3)=O)CC2)ccnc(Cl)c1Cl C1(C)(CC)CC(NC(C2CC(F)(CO)C2)=O)CN1C(=O)C(C)=C1CC1 C1(C)(COC)CC(NC(=O)Cn2cncn2)CN1C(=O)C=CCc1cnc(C)[nH]1 c1(CCC)ccc(CNC(C)COCc2ccccc2)s1 C(=O)(C(C)(C)C1CCCN1C(C1CCC1C#N)=O)NC(c1nc(=O)o[nH]1)C c1(C(N(CCOCCN(C(C(F)=CCC)=O)C)C)=O)cn2cc(C)c(C)cc2n1 C1(C(N(C(C=C)C)CC2CC2)=O)CC(NC(=O)COCC2CCC2)C1 N1(C(c2nccc(C)c2F)=O)C(C)CC2CN(C(C3C4CC(=O)CC34)=O)CC12 CC1CN(C(=O)CC(F)(F)C(F)F)CCCN1C(c1cnc(NC2CC2)s1)=O Cc1cc(C(=O)NCCN(C(=O)CC2CCCCCC2)C(C)C)ncc1C(N)=O c1(C(=O)NCC2C(C)(C)CN(C(c3ccnnc3S)=O)C2)cccc2[nH]ncc12 N1(C(C)C)CCc2onc(C(N3CCC3CNC(C3(C)CSC3)=O)=O)c2C1 CCCC(C(=O)N(CC(O)CN(C(=O)CNc1nccs1)C)C)S(N)(=O)=O c1(C(N2CC(CNC(c3n(C(C)C)ccn3)=O)C3C2C3)=O)cccc2nsnc12 C1(F)(CNC(c2c(=O)ccn(C)c2)=O)COCCN(C(=O)C2=NNC(=O)C2)C1 C(=O)(C(C)(C1CCC1)NC(=O)C=CCOC)N(CCCC)CCO C(C1c2ccccc2CCN1C(C1CC1C)=O)NC(CSSC)=O C(=O)(C(C)CC(=O)N1CCN(C(=O)COc2cn[nH]c2)C(C2CCC2)C1)OC N1(C(C(CC2CCCC2)NC(CC(C)N(C)C)=O)=O)CCS(=O)(=O)CC1 O=C(CCCC(F)(F)F)NCc1ccc(CNC(c2csc3sccc23)=O)cc1 c1(C(=O)NCCNC(c2nc(C)sc2)=O)ccccc1-c1nc[nH]n1 c1(NC(CC2CCCN(C(CCC)=O)C2)=O)cccc(O)c1Br C1(C(C)(C)C)CC(CNC(C2CC=CC2)=O)CN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 C1(C2CCN(C(C3CCO3)=O)C2)(NC(C2CN3CCN2CC3)=O)CC1 c1(C(=O)NCC2C(NC(Cc3c(Cl)cn(C)n3)=O)CCC2)ccc(S(C)(=O)=O)[nH]1 CCCCCCCCCC(=O)Nc1cnc(NCc2c(Cl)ccnc2Cl)c(O)c1 CC(CN(C)C)CC(=O)N1CC2CC2(CNC(=O)CCc2ccc(N)cc2)C1 C#Cc1cnn(CC(=O)NC(C)C(C)NC(c2ccc(CCC)cc2)=O)c1 O=C(NNc1ccc(Cl)nc1)NCC1CC1CO c1(C(CC2CCCC2)NCCC(C)C)nnnn1C1CCCC1 N1(C(CCCCOC)=O)CC2OCCN(C(c3ccc(=N)[nH]c3)=O)C2C1 c1(C(N2CC(C)(OCC(=O)N(CC(O)COC)CC)C2)=O)c(C)n[nH]c1C C1(NC(C(CNC(C)=O)(C)C)=O)COC2(C1)CN(C(=O)CC1(C)CC1(Cl)Cl)C2 C1(n2cc(C(C)(C)NC(c3[nH]ccc3C3CC3)=O)nn2)CC2CC1N(C(N)=O)C2 C1(F)(C(=O)NCCCCCN(C(c2cccc(SC)c2)=O)C)CC12CCCCC2 N1(C(c2c(O)ncc(CC)c2)=O)CC2CCCC(NC(C3CC3C)=O)(C2)C1 N1(C(CCOC2CN(C(C(=Cc3ccco3)C)=O)C2)=O)CCC2(CCSC2)C1 c1(NC(C(F)(F)C2(CC(c3ccccc3Cl)O)CCC2)=O)nc2ccccc2o1 c1(NC(C(=O)NC(c2ccc(OCC)cn2)C)=O)cnc2ccnn2c1 C1(C(=O)NCC2CCCCC2NC(=O)C(C)(C)c2ccns2)(CC)CCOCC1 c1(CC(=O)NC2CN(C(C(C)(O)CC(F)F)=O)C2)csc2ccc(Cl)cc12 N1(C(c2ccnc(F)c2)C(=O)NCCOCC)CCOc2ccc(F)cc21 C1(C(=O)NCC2(O)CCN(C(CCc3cc(C)on3)=O)C2)CCS(=O)(=O)C1(C)C c1(OC)ccccc1C(C)C(=O)NCC(C)(F)CNC(=O)C(C)(C)OC(C)C C1(NC(=O)CSc2cccc(Cl)c2)CC2CC1N(C(c1cccc(CO)n1)=O)C2 N1(C(C2CCCOC2)=O)C2CCC1C(CNC(c1cccnc1SC(F)F)=O)C2 c1(-c2cn(CC3CN(C(=O)Nc4cn(C)nc4)OC3)nn2)ccc2[nH]ccc2c1 N1(C(c2c(C)cc(CC)o2)=O)CC2CCC2(CNC(c2cncc(C)n2)=O)C1 CCC(CC)CC(F)C(=O)NCCCC(C)(C)C(=O)NCc1ccc(C)nc1O Cc1ccc2cc1NC(=O)C(C)CC(C1CC1)OC2=O.S(C)(=O)(=O)OC NC(=O)CCCC(=O)NC1(c2cncc(F)c2)CCC1 C12CCCCN(C1)C2=O.c1(CC)ncc(NC(c2cncc(C)c2)=O)cn1 C(CNC(=O)CSc1cn[nH]c1)(CC(C)C)NC(C(CC)SC)=O Cc1cccc(Br)c1C(C(=O)NC1CCSC1)NC(C1CCCCS1)=O CC1c2cc(Br)ccc2NCN1C(=O)C(n1cc(-c2ccc(CO)cn2)nn1)C1CC1 N1(C(c2ccc(N)c(Cl)c2)=O)CC(NC(=O)C=C2CC2)CC12CCCC2 c1(OC)cccc(CCC(=O)NCC2CCN(C(=O)CC3CCCC(C)O3)C2)c1 c1(C(=O)NCC(c2ccccc2)N(C)C(C2(C#N)CC2)=O)cnn2cccc(Cl)c12 C(=O)(NNc1cccc(C(C)(C)C)n1)NC(C)(C)COc1ccccc1C(N)=O CCCC(C)(O)CC(=O)NCc1cncc(C(N2CCC(C(=O)NC)C2)=O)c1 N1(C(CN(C(C)C)C)=O)CC(NC(C2OCCC2Cn2ccnc2)=O)C(O)C1 c1(CC)cc(C(=O)NCC2COC(CNC(c3ccc(OC)s3)=O)C2)on1 c1(C(=O)NCC(N2C(CNC(CCC)=O)COCC2)=O)c(NC)sc2c1CCC2 N1(C(C(C)(C)F)=O)CCC(NC(C2CCC(C3CC3)CC2)=O)C2(CCC2)C1 C(=O)(C1CCc2c[nH]nc21)NC1CCC(C)(NC(CCC=CC)=O)CC1 C(C)(CNC(=O)Cc1ccc(C(N)=O)cc1)(C(C)C)NC(C(C)OCC(C)C)=O N1(C(C)=O)CCC(CN(C)C(c2cc(C(N)=O)c[nH]2)=O)C1 C(=O)(CC(C=C)CCC)N1CCC(N(CC#C)C(c2ccc(CC)cc2N)=O)C1 CCCCCCC(=O)NC(C)(CSC)C(=O)NCCC1(COC)CCC1 CC1(C)COC(=O)C1NC(=O)NCCNc1cncc(Cl)n1 C=CCC(F)(F)C(=O)NCC1CC1NC(c1nc(Br)sc1C1CC1)=O C=Cn1ncc(C(=O)NCC(C)(C)OCC(=O)NCc2cccnc2C)c1N c1(CC(C(=O)NC(CCOC)CO)NC(C2CCOC(C)C2)=O)ccccc1Br CC(C)(C)C1=NOC(C(N2CC(CNC(=O)CCCCC3CC3)C(O)C2)=O)C1 Cc1c[nH]c(C(=O)NCC(C2CCCC2)NC(=O)CC2CN(C)C2)c1 C(C)(C)(CC(F)C(=O)N1CCc2nc[nH]c2C1)NC(CC1CCCC(C)C1)=O c1(CNCC2(C(=O)Nc3cc(=O)cco3)CC2)cccc([N+](=O)[O-])c1 C1(C(N(CCC(=O)OCC)C)=O)CN(C(C2CC2F)=O)CC12CC2 c1(NC(c2c(OC)n[nH]c2)=O)ccc(NC(c2cnc(O)n2C)=O)c(C)c1 c1(C(C(=O)NCSc2ccccc2)N(c2cc(C)on2)C)ccnc(Cl)c1Cl c1(CC(=O)NC2CC(NC(CC=CC(C)(C)C)=O)C2)cnc2cccnn12 CC(CC(=O)N1CC(CCCCNC(c2cc(N(C)C)ccc2O)=O)C1)C(F)F c1(OC)cc(C(=O)NC2CCCC2NC(c2ccc(F)cc2O)=O)cc(Cl)c1 C1(NC(C(CN(C)C)O)=O)CCOC12CCN(C(c1snc(O)c1Cl)=O)CC2 N1(C(=O)NC(c2ncc(C)o2)C)CCC(N(C2CCOCC2)C(C)C)CC1 c1(C(=O)NC(c2ccccc2Br)(C(=O)N(CCC#C)C)C)ccn2ccnc2c1 c1(NC(=O)NC(C)(Cc2cccc(Br)c2)CO)ccc2ccccc2c1 C1(C2CCCCO2)(C(=O)NCC(C(C)C)NC(=O)CS(C)(=O)=O)CCOCC1 Cc1cc(NC(C2(CCNC(c3cccnn3)=O)CC2)=O)c(O)cc1F c1(NC(C2(N=[N+]=[N-])CCN(C(=O)C=CCF)C2)=O)ccc2ccncc2c1 Cc1ccc(Br)c(C(=O)NC2CCC23CN(C(=O)C(O)C2CC2)C3)c1 Cc1cc(C(=O)NCC(C)NC(c2coc(Cl)n2)=O)ccc1-n1cnnn1 C1(COC)(CO)CCN(C(C)(C)C)C1.c1(C=O)ccnn1CCn1cc(CO)nn1 c1(C(=O)NC2CN(C(Cc3nc(C)[nH]n3)=O)CC2C)ncc(C2CC2)cc1F CC(C)(O)C(F)(F)C(=O)N1CCC(N(C(=O)CNC(N)=O)Cc2ccsc2)CC1 C1(CC(=O)NCCC2CCN(C(C=CC(C)(C)C)=O)C2)CCS(=O)(=O)C1 Cc1nc(C(=O)NCC(C2CC2)NC(=O)Cc2c[nH]nc2O)nn1-c1nc[nH]n1 c1(C(=O)NC2(C(N(C(C(=O)Nc3cn(C)nn3)C3CC3)C)=O)CC2)ccccc1 CC(CC(C)SC1CCC2(CCCCC2)O1)CC(C)(C)C C(=O)(CC(C)P(C)(C)=O)NCCOC1CCN(C(c2nccc(C)n2)=O)C1 c1(NCCC2(C)CC2(Cl)Cl)nc(N2CCOC(C(N)=O)C2)nc2scnc12 c1(CCC(=O)NC2CCN(C(CSCC)=O)C2)cccnc1Cl c1(C(=O)NC2CCC(NC(C(C)OCCCC)=O)CC2)ccc(N)c(N)c1 N1(C(c2cc(COC)[nH]n2)=O)CC2CCC1CC2NC(=O)C(C1CCCCC1)O C1(NC(c2nc(C)oc2)=O)C(C)CN(C(c2ccc(Cl)s2)=O)CC1C CCC(C)(C(=O)NCC1CCN(C(c2ccc(OC)nn2)=O)C1)C(N)=O C(C(CC)(CC)C(=O)N1CCCC(C(C)(C)O)C1)NC(CC(CC)SC)=O C1(CC=C)(NC(C2CC23CCC3)=O)CCN(C(=O)CCn2cnccc2=O)C1 N1(C(c2ccc(OC)cn2)=O)CCC(NC(c2[nH]nnc2C2CC2)=O)C(F)C1 C1(NC(C2CC(C)(CC)C2)=O)CCN(C(C2CC(=O)NC(=O)N2)=O)CC12CCC2 C(=O)(C1=CCCOCC1)N(C1C2CN(C(C(COC)C)=O)CC21)C CN1CC(F)CC1C(N1CCC(C)(C(N2CC(c3ccncn3)C2)=O)C1)=O c1(CC(N2CCC(OCCN)CC2)=O)cc(Cl)ccc1I O=C(C1=CCCN(C(c2cnsn2)=O)C1)NCc1cnccn1 N1(c2n(CCC#C)c(COC(C)(C)C)nn2)CC(C)OC(C)(C(F)F)C1 c1(C(=O)NC2CC(CNC(c3n(C(C)C)ccc3)=O)C2)ccc(N)cc1[N+](=O)[O-] C(C)(CCC(=O)N1CCCCC1CNC(C1(SC)CC1)=O)SC c1(CC(C)C)cc(C(N2CC(N(C(=O)CC3C=CCC3)C)C(O)C2)=O)cc(O)n1 C1(C(=O)NC(C2CCOC2)C)(OC)CCN(Cc2nc(CC(C)C)no2)CC1 C(=O)(C1=C(C)OCC1)N(C1CCN(C(=O)CC2COCC2O)CC1)CC#C N#CC1=C(C(=O)NCCOC2CN(C(C3CN(C4CCC4)C3)=O)C2)CCC1 Cc1cc(N2CC3CCC3(CCN)C2)n2ncc(Br)c2n1 c1(C(=O)NC(C)C(N2CCCCC2C)=O)cc([N+](=O)[O-])c[nH]1 C1(C(=O)NCC(CC(C)C)NC(=O)C=CC2CCOCC2)(OC)CCCCCC1 C(CN=c1[nH]cnc2c(Br)cccc12)(C(C)(C)C)NC(c1ccc(CCC)[nH]1)=O c1(CC(=O)NC(CN(C(=O)CC2CCSCC2)CC)C)c(C)nn(CC)c1C CCCCC(=O)NCCN(CCOCCO)C(C12CC(O)C1C2)=O c1(N2C(C3(NC(c4ccc(C#C)cc4)=O)CC3)CCC2)ncc([N+](=O)[O-])cc1F C(=O)(CC(F)(F)C(F)(F)F)NCC(c1ccc(F)cc1)NC(c1c(CC)noc1)=O C(=O)(CCS(=O)(=O)N(C)C)NCCC(C)CCNC(=O)Cc1ccc(F)cc1 c1(-c2cn(CC3CN(C(c4c(CC)ccs4)=O)C3)nn2)cccnc1C c1(C(=O)NC2CC(N(C(C3(CC)CCC(O)CC3)=O)C)C2)cc2cc(Cl)sc2[nH]1 c1(CC(=O)N(C(C)CCNC(=O)CC2CCCC2(F)F)C)ccc2c(c1)COC2 N1(C(C=C(C)C)=O)CCN(C(c2ccc(Cl)cc2)=O)CC1c1cn[nH]c1 c1(CC(CC)C)nc(-c2cccc(SC)c2)n(-c2cccc(C(=O)O)n2)n1 C1(C(N(C(c2cn(-c3ccc(C(=O)O)cc3)nn2)C)C)=O)CCC(=O)N1C C12(CNC(C3(CC=C)CC3)=O)CCC(CC1)N(C(C1(CN(C)C)CCCC1)=O)C2 C(C1=CCCCC1)(c1n(C(CC)C)nnn1)NCC(=C1CCOCC1)F Cc1ccccc1C(C)NC(C1(CNC(=O)C#CC2CC2)CCC1)=O c1(CNC(C(N2CCNC2=O)C)=O)ccc(C(=O)NCCC(=O)NC2CC2)o1 CCCC(CCC)N=c1nc(N2CCN(C)C(C)(C)C2)c2c([nH]1)c(C)nn2C c1(NC(C2SCCN(Cc3ccc(C)cn3)C2)=O)c(Br)ccc2ncccc12 N1(C(c2ccc(CC)[nH]2)=O)CCC(NC(=O)CC2CCCCO2)C2(CCC2)C1 N1(C(C(C)(C)N(C)C)=O)CCN(C(c2ccccc2)=O)CC1 c1(NC(C23CC(NC(=O)CCc4ccc[nH]4)(C2)C3)=O)ccccc1C(=O)NCC C(CC(C)C(=O)NCCN1CCN(C(C2CCC(N(C)C)CC2)=O)CC1)OC C#CC1(C(N2CC(CO)(OC)C2)=O)CCN(C(=O)CC2CCC(=O)C2C)CC1 C1(OCC)CCN(C(=O)Cn2nc(C)cc2C)CCO1.C12CCCN(C1)C2=O C1(c2n(CCSC)nnn2)(NCCC2CCC2)CCC2(CC1C)OCCO2 N1(C(C2N(C)CCOC2)=O)CC2(CNC(c3ccn(C)c3)=O)CC1CO2 n1(CCCC)cc(CN(CCN)CC)nn1 c1(C(=O)NCCNC(CC2CC(C(C)(C)C)C2)=O)nn(C(C)(C)C)cc1Br Cc1cc(C#N)ccc1C(N1CCC2(NC(c3ccc[n+]([O-])c3)=O)CC2C1)=O CCC(CC(=O)N(C)CC1CCCC1(C)C)N(C(=O)C(SC)SC)C c1(C(=O)NCC2N(C(C)=O)CCC2)oc(CNC(C2CC23CCC3)=O)nc1C N1(C(CC23CC(C)(OC2)C3)=O)CC(NC(=O)CC2CCC2)CC12CCCCC2 Cc1cc(=NCC2CCN(C(c3c(N(C)C)cccc3F)=O)C2)c(C#N)c[nH]1 N1(C(CC2CCN(C(C3=NNC(=O)C3)=O)C2)=O)Cc2ccccc2C1 CONC(=O)C(=O)N1CCC(C(=O)NC2CCCC2CF)C1C N1(C(CCC#N)=O)C2CCC1C(CNC(=O)C(O)Cc1cnc[nH]1)C2 N1(C(C(c2ccc(C)s2)C)=O)CC(NC(c2ccc(=O)oc2)=O)CC(C)(C)C1 CCS(=O)(=O)CC(=O)N1CCC(C(=O)Nc2c(C)ncn2C)C1 C(=O)(C(CC)CCCC)NC(CCCC)CNC(c1cc(=O)n(C)o1)=O c1(CC)ccc2cc(C(=O)NC3(C)CN(C(C4CCCN4C4CC4)=O)C3)[nH]c2c1 N1(C(C(C=C)(C)O)=O)CCC2(CCC(NC(=O)C(O)c3ccsc3)CC2)CC1 c1(C(N2CC3C(N(C)C(c4cc(O)cs4)=O)C3C2)=O)cnc2c(c1)COCC2 C1(NC(C(C)=C2CC2)=O)C(C)(C)C(NC(=O)CCc2ncc(C(C)(C)C)o2)C1(C)C N1(C(c2n(C)ncc2Cl)=O)CCN(C(C2(C)CCOC2)=O)CC12CC2 N1(CC(COCC(C)C)O)CCC(C)C(NC(N)=O)C1.C1(=O)CCCCN1 N1(C(C2(C)CCCCC2)=O)CCCC(C2CCN(C(c3ncccc3N)=O)C2)C1 N1(C(C2(C)CC(=C)C2)=O)CC2CC(NC(c3cn4cc(C)nc4s3)=O)CC1C2 N1(C(c2c(Cl)ccc(SC)c2)=O)CCCC12CCN(C(=O)C(C1CC1)N(C)C)C2 N1(C(c2ccn(CCC)n2)=O)CC(NC(=O)C(N2CCN(C)CC2)C)C2(CC2)C1 N1(C(Cc2ccc(C#C)cc2)=O)CC2CCN(C(=O)CC3COC(C)(C)C3)C2C1 C1(CC(N2CCC(N(C(c3n[nH]c(CO)n3)C)C)C2)=O)CCC(C)CC1 C1(C(=O)OC)CC2N(C1)C2=O.C(C(C)C1CCC1)OC(C)=O C1(NC(c2n(CCCOC)nnn2)c2occc2Br)COC2(CCCC2)C1 C1(C(=O)NC(CC)C2CCC2)C2CC1N(C(c1ccn(CC)c1C)=O)C2 N1(C(C(CC)OCC)=O)CCC2(CC1)CC2NC(c1ccc(CC(N)=O)cc1)=O C12CCCCCN1C2=O.C1(O)(CC(=O)NC2CC(NC(=O)NC3CC3)C2)CCC1 N1(C(c2nc(N(C)C)oc2)=O)CC2(CCCC2)C1C(N1CC(CNC(N)=O)C1)=O C12(C(N(CC(CN(C(=O)C(C)(C)C)C)O)C)=O)CCCCC1OCC2 C1(NC(C(C2CC2)NC(C)=O)=O)CCN(C(=O)Cc2ccn(C)n2)C1C Cc1ccc(C(=O)NC(C)C(C)NC(c2cnn(C3CC3)c2C)=O)nc1C N12CCCCC(C1)CNCC2=O.c1(O)ncccc1F.Cc1noc(COC)n1 N12CC3(COC(C3)CNC1=O)C2.CC1CCC(C)(Nc2ccncn2)CC1 CC(C)(C[Si](C)(C)C)C(=O)Nc1ccc(N2CCNCC2)nc1 C1(CC)CN(C(c2c[nH]cc2-c2ccc(C)s2)=O)CCN1C(=O)CCN(C)CC Cc1ccc(F)c(C(=O)NC2CC(CNC(=O)C(C)C)C2)c1F c1(C(=O)NCC2C(NC(C(C=CC)O)=O)CC2)cn(CCCC)nc1C C(=O)(CCC(CF)CF)NCC(C1CCCN(C(c2c(CC)nn[nH]2)=O)C1)(C)O c1(C(=O)NC2C(CNC(CCC(=O)NC)=O)CCC2)c(C)nn(C)c1C1CC1 N1(C(C(F)OC)=O)CCC(CNC(=O)C(C)Oc2ccc(Cl)cc2)C(F)(F)CC1 C1(C(N(CCCNC(=O)Cc2ccnc(C(N)=O)c2)CC)=O)CCCC(C)(C)C1 CC(COc1ccccc1)C(=O)N(C1CCN(C(=O)C(C)(C)c2cccs2)C1)C N1(C(CNS(N(C)C)(=O)=O)=O)CC(NC(=O)CNS(N)(=O)=O)C2CCCC2C1 CC1CC(NC(=O)CCn2ccccc2=O)CCN1C(C1CC12CCOCC2)=O c1(C(=O)NC23CN(C(CSCCCC)=O)C(C2)C3)oc2c(OC)cccc2c1C CN1CCN(C(=O)C(F)C2CCC2)CC1C(=O)NCCOCC(N)=O c1(C(=O)NC(C2CCCN2C(c2ccncc2)=O)(C)C)csc(-c2ccoc2)n1 C(=O)(C1=CCOCC1)NC(C)CCN(C(=O)C(C1CCOCC1)C)C C(=O)(C1CCCc2sccc21)N1C2(CCN(C(=O)C=CC=C(Cl)Cl)C2)CCC1 c1(C(n2c(CNC(C)=O)nc(-c3ccccc3Cl)n2)C)ccc(Cl)cc1 C1(CC=C)(C(=O)NC(C)(C)CNC(c2cnn(CCN(C)C)c2)=O)CCOC1 Cc1ccc(S(N)(=O)=O)cc1C(=O)N(C)CCN(C)C(c1csnc1C)=O c1(C(N2CCSC(C)(C)C2)C(=O)NCCCOC)cc(OC)cc(C(F)(F)F)c1 N1(C(C2CC(OC)CN2C(c2nocc2C)=O)=O)CCC12CCN(C)C2 C#CC12CCC(C(=O)NCC(O)CN(C)C(C3C4CCCOC34)=O)(CC1)CC2 C(=O)(CCC1CC(OC)C1)NCC1C(NC(C=CCC)=O)C1 c1(C(=O)NC2CN(Cc3cnn(-c4ccccc4)c3)CC2F)cc(F)cnc1Cl C=CC(C)(CCOC)C(=O)N1CC(F)(CNC(=O)Cc2cc(C)ns2)C1 N1(C(COCC)=O)CCCC(C(=O)NC(c2csc(-c3ccc(C)cc3)n2)C)C1 C(=O)(C(CC)CCCCC)N(C1CCC(NC(C(CC=C)(C)CC)=O)CC1)C Cc1ccc(C=CCC(=O)NC(C)CNC(c2cc(C(N)=O)cc(F)c2)=O)cc1 Cc1nc(CC(=O)NC2CCC(NC(=O)C(N3CCNC3=O)C)C2)cs1 Cn1nnc2ccc(C(=O)NC(Cc3nc[nH]n3)C(=O)O)cc12 c1(C(=O)NCC2(CCC)CCC2)cccc(S(=O)(=O)Nc2ccsc2C(F)F)c1 c1(C(N(CCOC)CCNC(C2(C)CC(F)C2)=O)=O)c(C)cc(C)cc1N C#CCCCCCCCOC(c1cnnc(-c2ccccc2CC(=O)OC)c1)=O N1(C(CC(C=C)(C)C)=O)CCN(C(=O)CC2CCC(=O)C2C)C2(CC2)C1 N1(C(C=CC)=O)CCN(C(=O)CCc2ccc(O)cc2)CC1C(F)(F)F C12(C(N(C)CC3CCN(C(COCCC=C)=O)C3)=O)CCC(C(F)F)(CC1)CC2 C1(NC(C2(CCCC)CC2)=O)COC2(CCN(C(C3(CF)CCC3)=O)C2)C1 CCCC(CCC)=CC(N1CCC(O)C1C(N1CCC1CC(C)C)=O)=O N1(C(CNC(C)=O)=O)C2CCCC1CN(C(C13CC(CCC(F)(F)F)(C1)C3)=O)C2 c1(CC(=O)NCC23C(CN(C(CCCSC(C)(C)C)=O)C2)C3)c[nH]c(=N)nc1O C1(NC(CNS(NC)(=O)=O)=O)CCN(C(c2cncnc2C)=O)C(C)C1 Cc1cc(F)sc1C(N1CC2CC1C2NC(C1(CC(F)F)CCC1)=O)=O CC(=O)C(C)CC(C)C(=O)NCCn1cnc(C(N2CCn3nccc3C2)=O)c1 C=CC(CC)CC(=O)NCC1(NC(=O)CC2OCCO2)CCCCCC1 C1(CCNC(C2C(=O)NCC2)=O)CSCCN1C(c1c[nH]ccc1=O)=O C1(O)(CNC(C(C)OCC(C)C)=O)CCCN(C(=O)CCC(N)=O)CC1 C(Cc1ccco1)(C(=O)NC(C)CC1CCCCC1)NC(CN(C)CC)=O C1(NC(c2nnc(C)s2)=O)CN(C(=O)C=Cc2ccco2)CCC1C C(C)(C(O)C(=O)NC(C1CN(C(=O)Cn2cc(-c3ccccc3)nn2)C1)CC)OC N1(C(CN(C)C(N)=O)=O)CCCC(NC(=O)CCc2ccc(N)cn2)CC1 c1(C(=O)NCC2(NC(C3CCCC(F)(F)C3)=O)CCC2)cccc2c1COC2 c1(C(N(CC(C)(C)NC(c2ccc(F)cn2)=O)C)=O)ccc([N+](=O)[O-])n1C Cc1[nH]nc(C(N2CCOC(CNC(=O)C(C)(Cl)Cl)C2)=O)c1F C1(CC)(NC(c2ncoc2CNC(=O)Cc2ccc(F)cc2)=O)CC(C)(C)C1 c1(C(N2CCCN(CC(O)CO)CC2)C(=O)NC)cnc2c(C#N)cnn2c1 C(=O)(C(F)C(C)(C)O)N1CCC(CN(C(c2cc(CC)c(C)s2)=O)C)CC1 CC(C)(O)C(F)C(=O)NCCN(C1CCCCC1)C(=O)CCNS(C)(=O)=O Cc1c(F)ccc(N)c1C(=O)NCCN(C(=O)C(c1cccc(Cl)c1)O)C CCCC(CC(=O)N1CCC1C1CCC1)NC(c1ncccc1Cl)=O Cc1c(Cl)ccc(C(N2CC(NC(c3ncccc3C3CC3)=O)CC2C)=O)c1O c12cccc(C)c1OCCOC2=O.c1(CCC(=O)OC)ccnn1C C1(C(=O)NCCN(C(C)C)C(c2cc(C(F)F)no2)=O)COCC1C(N)=O c1(CCCC(=O)NC2CCOC(c3ccc(F)cc3)C2)ccc(F)cc1 CC1(C)CCC(C(N2CCCCC2CS(C)(=O)=O)C(=O)NC2CC(F)(F)C2)CC1 N1(C(C(CC#C)C)=O)CCCC12CCCN(C(c1ccc([N+](=O)[O-])o1)=O)C2 Cc1cc(N2CCC(C)(NC(=O)C(=O)N(C)C)CC2)n2nc(C(F)(F)F)nc2n1 c1(C(N2C(CN(C(=O)CCCNC(N)=O)C)CCC2)=O)cccnc1NC(N)=O Cc1cc(C)n(CC(=O)N(CC(C)NC(c2[nH]ccc2C)=O)C)n1 c1(C(=O)NC2CCCC(NC(Cc3n(C)cnc3)=O)C2)cccc2c1CC(=O)N2 CCCS(=O)(=O)CC(=O)NCc1ccc(C(C)NC(=O)CNC(C)=O)cc1 c1(OC)cc(-c2csc(NC(C3CCN(C(C)=O)CC3)=O)c2)cc(C)c1 N1(C(c2cc(=NC)[nH]cc2)=O)CC2CCC(C1CO)N2C(=O)Cc1nonc1C Cc1ncsc1C=CC(N1CCC(NC(C2(C)CCN(C)C2)=O)C1)=O c1(C(N2CCC(NC(C3C(C)(C)CC3)=O)C2)=O)cc2ccc(F)cc2s1 c1(C(=O)OC)ccc(OC)c(NC(=O)NCC2CC(O)C2)c1 C1(C(=O)NC2(C3CCCN3C(=O)C(F)(F)c3ccccc3)CC2)(OC)CCOC1 [N-]=[N+]=NC1(C(=O)NCC2CCOC2=O)CCN(C(c2ccc(F)c(O)c2)=O)C1 C(=O)(C1=CCCC1(C)C)N1CCC(O)(CN(C(c2c(C)snc2)=O)C)C1 N1(C(C(N)=O)=O)CC2CCCC(CNC(=O)CN3CCCNC3=O)C2C1 N1(C(c2ccc(C)nn2)=O)CCC2CCCC12CNC(c1coc(C(F)F)n1)=O c1(OC)cc(C(=O)NCCN(C(=O)C=CBr)C2CCCC2)cc(Cl)n1 c1(C(=O)NC(C2(O)CCN(C(C=CC)=O)C2)C)cn2cc(C)nc2s1 N1(CC(=O)O)CCN(CCNCc2cnn(CC(O)CO)c2)CC1 c1(C(=O)NC2(C)CCN(C(=O)C=C3CCSCC3)C2)cc2c(Cl)cncc2s1 C(CCC(=O)NN1C(=O)NC(C)(C)C1=O)c1c(-c2ccc(S(C)=O)cc2)csc1 c1(C(N2C(CNC(C(C)CC(N)=O)=O)C=CC2)=O)ccc2cc(F)ccc2n1 c1(-c2n(C3C(C)OCC3)nc(CCO)n2)cc2scc(Cl)c2[nH]1 C(=O)(C#CC1CCC2(CC1)OCCO2)NCC1CC(O)(CNC(CC=C)=O)C1 N1(C(C(CC)SC)=O)CCC(C)(CNC(c2cn(CCN(C)C)nn2)=O)CC1 Cc1cc(F)c(CC(N2CC(CNC(=O)CC3COC(=O)C3)C2)=O)cc1F c1(CN=C(NCC(c2cn(CC)nc2)O)NCC(F)F)cc(F)ccc1C c1(CC)cc(C(N2CCCC(C)(NC(=O)C3=NOCC3)C2)=O)cc(N)c1 c1(C(=O)NCC(CNC(c2ccsc2Cl)=O)CO)n[nH]c2c1CSCC2 C1(CC(N2C(C=O)CCC2)=O)CCOC1(C)C.CC(C)(C(=O)N1CCSCC1)N CCCCCCCCC(F)C(=O)NC12CCC1CN(C(=O)CCNC(=O)NC)C2 C(c1nc2ccccc2s1)=CC(N1CC2(CCN(C(CC(CC)CC)=O)C2)C1)=O CCC(CC)C1C(=O)N1.C1(C(=O)NCC(CSC)OC)CC(F)(F)C1 C(CNC(=O)COc1cnn(C)c1)(C(C)(C)C)NC(C(C)C1CC1)=O c1(C(N(C(C)CN(C(=O)CCn2ccnn2)C)C)=O)cccc(C(C)(F)F)c1 c1(C(N2CC(C3(NC(CC4(C=C)CC4)=O)CC3)C2)=O)cc2ncc(C)cn2n1 CCC(CC)(CC)C(=O)N1CC2C(CNC(c3ccc(CSC(F)F)o3)=O)C2C1 Cc1ccc2c(=NCCCc3nc(C)cs3)[nH]c(=NCC(=O)N3CC=CC3)[nH]c2c1 CCC(CC(F)F)C(=O)NC1CC(CNC(=O)CCNC(=O)CO)C1(C)C C(=O)(C1=CC2(CCN(C(=O)CSCC(F)F)C2)C1)N1CCC(C2(C)CC2)C1 c1(OC)ccc(F)cc1C(F)(F)C(=O)NC(C1CN(C(C2CC3CC3C2)=O)C1)C C=C(C)C(CC(=O)NCCC1COCCN1C(c1cscn1)=O)OCC CC1(C)CN(C(=O)Cc2nccs2)CC1C(N1CC(C2(C)CC2)C1)=O N#Cc1cc(F)c(NC(C2C3C(CN2Cc2ncccc2Br)C3(C)C)=O)cc1F c1(C(N2CC(C(C)NC(C(C(CC)C)OC)=O)C2)=O)ccc2nc[nH]c2c1 C1(O)(CCC)CN(C(=O)C(C)(C)NC(=O)CCCSC)C1 C1(C(N2CC(NC(C(CC=CC)C)=O)C2)=O)CC2(COC(=O)N2)C1 c1(C(N2CCN(C(CCCC(OC)OC)=O)C(C)C2C)=O)ccc2c(c1)CC(C)O2 c1(C(N(CCNC(=O)C(C)OCC(F)(F)F)CC)=O)ccc(O)nc1Cl c1(CCC(=O)NCCCNC(C2N(CC)CC2)=O)csc(Cc2ccccc2)n1 CN1C(=O)CC(NC(=O)CCOCCNC(C2CCC2)=O)C1=O.C1(C)(C)CO1 CC(C)CC(C)(CNC(c1ccccn1)=O)NC(c1cnc2n1CCC2)=O N1(C(CCCNC(C2C(C)(C)OC(=O)C2)=O)=O)CC(=O)N2CCCC2C1 N1(C(COc2ccc(NC(=O)OC(C)(C)C)c(Cl)c2)=O)CC(O)C(O)C1CO CCC(C(=O)NN(C)C(C1CCCC1CCOC1CC(O)C1)=O)N(C)C N1(C(c2nccs2)=O)CCCC(N(C2CCC2)C2CC2)C1 Cc1[nH]c2ncccc2c1C(=O)NC1CN(C(=O)C=C2CCC2)CC1C N1(C(c2c(CC)nn(C)c2)=O)CCN(C(C2CCN(C)C2C)=O)CC(C)C1 C12(CNC(COC(C)(C)C(F)(F)F)=O)CCCC1CCN2C(c1cnc[nH]1)=O N1(C(C2(CCOC)CC2)=O)CC(CNC(c2ncoc2C2CC2)=O)C(O)C1 N1(C(C2(NC(N)=O)CC2)=O)CC2CC(NC(C3CC4(CCCO4)C3)=O)CC1C2 CCC(=O)CCC(=O)NC(c1cnn(C)c1)C(=O)NC(C)C(=O)N(C)C Cc1cc(C(N2CCCC(CCC(NC[Si](C)(C)C)=O)C2)=O)cc(C)n1 N1(C(C2CC(C(F)F)C2)=O)CCCC(C2CCN(c3ncns3)CC2)C1 c1(C(=O)NC2CN(C(C(C)=C(CC)C)=O)CC(O)C2)ccnc2[nH]ncc12 N1(C(C(CC=C)CC)=O)CC2CCCC2(CNC(=O)CNS(=O)(=O)NCC)C1 C1(CNC(C(c2cccs2)SC)=O)CC2(CO1)CN(C(C1C3COCC13)=O)C2 c1(C(=O)NC2CCC(CNC(c3cnns3)=O)CC2)cc(O)ccc1Cl CCCCC(CC(=O)N(CCC(=O)OC)OC)NC(=O)C=NOC c1(C(=O)NCCOC2CN(C(Cc3n(C)ncc3)=O)C2)ccn2c(O)nnc2c1 C(CC(O)CC(=O)Nc1cccc(F)c1C(N)=O)SC C1(CNC(C(C)Cn2cccn2)=O)CCCN(C(=O)CSc2nccn2C)CC1 N1(C(c2c(Br)cc(C)s2)=O)CCC(C)N(C(=O)Cc2ccsn2)CC1 Nc1cc(Cl)ncc1C(N1CCCC(CO)(NC(C2CC23CCOCC3)=O)C1)=O C(=O)(C(C)(F)CCCC)N1CCC(CC(N2C(CCC#C)CCC2)=O)CC1 N1(C(C(C(C)C)C(C)C)=O)CCC2(CCN(C(=O)CSCCC(F)(F)F)CC2)C1 Cc1cc(F)cc(Br)c1NC(=O)C(=O)NC1CC2(CCCC2)C1 c1(CC(N2CC(COC)(NC(c3cc(O)no3)=O)C2)=O)nccc(C)n1 N1(C(C2(C=C)CC2)=O)CC2CCCC(NC(c3ccnc(NC(C)=O)c3)=O)(C2)C1 C1(CNC(c2n(CC)nnc2)=O)C2CCCC1N(C(=O)CC(C)C)C2 CCS(=O)(=O)c1ccc(CN=C(NCc2cccs2)NCC2CNC(=O)O2)cc1 c1(C(N2CC(CNC(C(C3CC3)OCC)=O)C2)=O)c(C(F)(F)F)cccc1Br C(=O)(CCCC(=O)N(CCC(C(C)(C)C)NC(=O)C(F)C1CCC1)C)OC N1(C(C(C)=CC)=O)CCC2(CCN(C(=O)C(C)CS(C)=O)CC2)C1 C1(OC(=O)C(=O)NC2CS(=O)(=O)CC2C(F)(F)F)CCS(=O)(=O)CC1 CCC(CC(C)C)C(=O)NCC(C)N(C(=O)C(Cl)=CCl)CC c1(C(=O)NCCN(C)C(C2CC3CCC(C2)S3)=O)cccc2cc(F)ccc12 N1(C(C(CC#C)(C)NC(=O)CN2CC3CCC2C3)=O)CCN2C(=O)CCC2C1 C(=O)(C(O)CNC(C1CCC1CNC(c1cnc(C)s1)=O)=O)NC CC1(C)CCCCC1C(N1CC(NC(=O)C(c2ccccc2)n2cccc2)C1)=O CC1(CC(=O)NC2CC(NC(C3(c4ccccc4Cl)CC3)=O)C2)CC(F)(F)C1 N1(C(CNC(CN(C)C)=O)=O)CCCC(CO)(NC(C2CN(C)C(=O)N2)=O)C1 C(CCCC(=O)NCC1OCCC1(C)C)N(C(=O)CSC(F)(F)F)C N#CC1(C2CCCC2)CCN(C(c2cnc3c(c2)COCC3)=O)CC1 N1(C(c2cnn(C3CCC3)n2)=O)CC2CN(C(C34CCCN3CCC4)=O)CC2C1 c1(C(N2CC(NC(c3cc(C)nn3CC(F)F)=O)C3C2C3)=O)ccc([N+](=O)[O-])[nH]1 c1(C(=O)NCC(CO)NC(CCC(CCCC)C)=O)cc2ccncc2c(O)n1 Cc1c(C(=O)NCCOCCNC(=O)Cn2cnnn2)cnn1C(C)C N1(C(CC2CN(C(CC(COC)COC)=O)CC2C)=O)CCC(F)(F)CC1C c1(C(N2CCN(C(C(C)=CC3CC3)=O)C(C)C2C)=O)cc2nccn2c(O)n1 N1(Cc2nnc3n2CC(C(=O)OC)CC3)CCCn2[nH]c(=N)cc2C1 N1(C(C(Br)=C(C)C)=O)CCCC(NC(=O)Cc2cc(F)ccc2C)CC1 N1(C(c2c(CC)noc2)=O)CCC2(CCN(C(=O)C(C)(CC)CO)CC2)C(C)C1 C(CN=c1[nH]c(=NCC2CCC=CO2)[nH]c2c1COC2)n1cc(Br)nn1 C12(CC)CN(C(C3(CC)CCCC3)=O)C(CNC(=O)CC3CCCOCC3)(C1)C2 c1(C(N2CCC(C3N(C(c4c[nH]c(=N)s4)=O)CCC3)C2)=O)cc2ccsc2s1 Cc1nc(C)c(C(N2CCC(NC(=O)CCc3cncc(F)c3)C2)=O)[nH]1 c1(C(=O)NCC#CCNC(c2c(=N)cc[nH]c2)=O)cc2c(o1)CCCC2 c1(OC)ccc(CN2CC3CC2CN3C(=O)NC2CCC(C)CC2)c(OCC)c1 c1(C(=O)NCCN(C(CN(CCC)C)=O)CC2CC2)c(CC)nn(C)c1Cl C12=NC(=NCCCOCCN1C)NC1=C2CSC1.C(C)(COC1CC1)SC C12(CC)CN(C(c3cccc(N)c3)=O)C(CNC(c3ccc(=O)oc3)=O)(C1)C2 C1(CCCNC(CCn2ncc(C)c2)=O)CN(C(c2nccc(C)n2)=O)CCO1 N1(C(C(CCSC)O)=O)CCC2(C1)CN(C(=O)CCS(N)(=O)=O)C2 Cn1cnc2c(NC3CC3)[nH]c(=NC(CC3CC3)c3nc(C(F)(F)F)cs3)nc12 c1(C(=O)NCC(CC)(C)NC(C2CN(C)C(=O)N2)=O)cc2ccc(F)cc2cn1 C#Cc1nc(C(=O)NCC2(CNC(C3CC(N(C)C)C3)=O)CCCC2)cs1 CC1=C(C(=O)N2CC3CN(C(c4c(C)cc(C)oc4=O)=O)CC3C2)COCC1 C(=O)(C(C)(C)CC(C)C)NC1(CNC(c2nc(C)oc2C)=O)CCCCC1C CCCC(C)(O)CC(=O)N1CCC(COC)(NC(=O)C(F)=CC2CC2)C1 C1(C(C)NC(=O)CSc2nncs2)CCN(C(C2(C(F)(F)F)CC2)=O)C1 C(=O)(C1Cc2ccccc21)NCC(CCC)C(=O)NCc1ncnn1CC C(=O)(CCC(F)(F)F)NC(C(C)NC(c1[nH]ccc1COc1ccccc1)=O)C C(CN=C(NCC12COCC1C2)NC(C)C)c1scc(COC)n1 C(=O)(C(C)C1OCCc2sccc21)Nc1cccc(NC(C(F)=CCC)=O)c1 CC(C)CC(CNC(=O)CC1(C)OCCO1)C(=O)NCC(O)C(C)O c1(C(N2CC(C(C)NC(CNC(=O)NC)=O)C2)=O)cc(C)c2ncccc2c1 c1(C2C(C)C2)ccc(C=CC(=O)NC2CC(c3nn[nH]n3)C2)o1 Cc1ccc(CC(=O)NCCC2CCN(C(c3cc(C)c(C)[nH]3)=O)C2)c(F)c1F O=C(C1=NOC2(CCOC2)C1)NCC1(F)CN(C(=O)C=Cc2ccccn2)C1 C(=O)(CC1=CCOCC1)NC(C)C(C)(C)C(=O)NCCc1ccc(O)nc1 C1(CNC(C2(CC)CC2(F)F)=O)CC2(CCN(C(C3CC34CCCC4)=O)C2)CO1 c1(C(=O)NCCC(C)(C)NC(C2C(F)(C(=O)OCC)C2)=O)cc2ccccc2[nH]1 C(c1ccc(Cl)c(Cl)c1)=CC(N1CCN(C(C2C(c3n(C)ncc3)C2)=O)CC1)=O c1(OC)cccc(C(C)C(=O)NCC2(C)CCCC2NC(=O)C=C(C)Cl)c1 C(C)(C(C(=O)NCCOC1CCN(C(c2occc2Br)=O)C1)N(C)C)OC C1(CC=C)(NC(=O)CC(C)(C)O)CCN(C(C2(SC)CC2)=O)CC1 N1(CC)CCCC1C(=O)NCCSCC(=O)Nc1csnc1OC c1(OCC2CN(CCC(N3CC(OCC)C3)=O)C2)ccccc1CC1CC1(F)F c1(C(=O)NC2CC(CNC(c3c(Cl)cc(C)s3)=O)C2)ccnc2[nH]ncc12 Cn1nc(Br)c2c(NC3CN(C(=O)CCC4CC4(F)F)CCC3CO)ncnc12 CC1(C)OC(=O)NC1C(N1CCC(Cc2ccc(Br)cc2)C1)=O C(N=c1[nH]nc(O)s1)C1CCC(NC(CCC(C)SC)=O)C1 C(C(C)(C)C(=O)NC(C1CSCCO1)(C)C)OCC CC1CC(CC(=O)NCCCCC(CO)NC(=O)CP(C)(C)=O)CCC1C C1(C(=O)NN(CCCCNC(C=CC(C)(C)SC)=O)C2CC2)CC(O)(C(F)(F)F)C1 c1(C(C)NC(=O)CC2OCCOC2(C)C)cc(F)c(Br)cc1F C=CC1CN(C(=O)OC(C)(C)C)CCC1CC(=O)OCc1cnc2c[nH]nc2c1 c1(OCC)ccc(C(=O)NC(C)C(C)NC(C2CC(O)(C#C)C2)=O)cc1O C(=O)(C(C)C(O)C(C)CC)N(C)CC1N(C(CCC(CC)CC)=O)CCC1 c1(CNC(CN(C)C2CC2)=O)nc(CN2CCOCC2)cs1.C12(CCC1)C(=O)N2 c1(SC)cc(C)c(C(=O)NCC2CCCC2NC(=O)CCN2CCNC(=O)C2)o1 N1(C(c2c(OC)nn(C)c2Br)=O)CCCC2(C1)NC(=O)NC2=O Cc1cncc(C)c1C(N1CCC(NC(=O)C(F)C(C)(F)F)C(F)C1)=O Cn1nc2ccccc2c1CNC(=O)Nc1cn(CC2CCCOC2)nn1 C1(NC(=O)Cc2cn[nH]c2)CCC12CCN(C(=O)CCc1cncc(F)c1)CC2 c1(CNC(C2CC(CNC(=O)CC3CC(F)(F)C3)C2)=O)cc(F)c(F)c(F)c1 CC(CCCC(=O)NCCCN(CCCNC(=O)CCF)C)c1ccon1 c1(C(=O)NCCNC(c2occc2C2CC2)=O)cccnc1C(F)(F)F C1(CNC(C2C(CC)OCC2)=O)CCN(C(=O)C(C)(C)CSC)CC1C1CC1 C1(N(C(COCC)=O)C)CN(C(=O)CNC(c2cccc(F)c2)=O)CC1(C)C Cc1ccccc1C(=O)NC1CCCCC1C(N1CCC1(C)C)=O CCC(CCCC(=O)NCC1(Cl)CC1(F)F)NC(C1CCCC(C)(C)C1)=O C1(N=[N+]=[N-])(C(=O)NCc2n(C(C)C)cnn2)CCN(C(=O)C=CC(C)(C)C)C1 C1(C(=O)NC(CC2(O)CCC2)CO)CCC(Nc2ccccc2Br)CC1 c1(CC(=O)N(CCNC(C2CCCC(OC)C2)=O)C)coc2ccccc12 N1(C(c2c(F)cncc2Br)=O)CCC2(CCN(C(c3cc4ncsc4[nH]3)=O)C2)C1 N1(C(C(=O)Nc2ccccc2)c2ccsn2)CCC2(C1)OCc1ccccc12 N1(CC#C)CCC(C(=O)NCCC2CN(C(c3cnc(OCC)cn3)=O)C2)CC1 CC1CCCNC1C(=O)NCC1(C)CCN(C(c2cccs2)=O)C1 C1(CNC(c2c(Cl)cccc2Cl)=O)C(C2CC2)CCN1c1ncc([N+](=O)[O-])cn1 CC1(C)CC(C(=O)N2CC3CC(C(=O)NCCCN4CCC4)(C3)C2)=NO1 N1(C(C2CCCN(CC)C2)=O)CCCC2(CC(NC(=O)C#CC(=O)N(C)C)C2)C1 N1(CC)CCOCC1C(=O)N(CCCNC(C1(n2ccnn2)CC1)=O)C CCCC(C(=O)NC1CCC1NC(c1csc(C)c1CC)=O)S(N)(=O)=O N1(C(=O)CC2CCSC2)CCN(C(=O)C(c2cccnc2)O)C2(CC2)C1 CN1CC(O)CCC1C(N1CCOCC1CCNC(C1SCCS1)=O)=O C12(NC(c3ccc(Cl)c(O)c3)=O)CCN(C(=O)CSc3ccncc3)CC1C2 C1(C(=O)NC(C=C)COC)CN(C(c2ccc(C(C)=O)[nH]2)=O)CCC1(C)C C1(NC(c2cc(C)nnc2)=O)Cc2ccccc2C1NC(=O)Cc1ccc(C)o1 C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NCC(=C)CCNC(C12CC(C)C1C2)=O N1(c2nc(C#N)cc(C)n2)CCCC2C1CCN2C(c1cc(Br)c(O)cc1O)=O O=C1CCC(C(=O)NCC2CCCN2C(=O)CC2(CO)CC2)N1 C=CCC(C(=O)NCc1cnn(C)c1N)NC(=O)C(C)COCC Cc1c(N)ccc(C(N2CC(CNC(c3cc(C#N)c[nH]3)=O)CC2C)=O)c1Cl Cc1cc(C(=O)NC2CN(C(c3cc(C)c(C)[nH]3)=O)CC2C)n(C2CC2)n1 C1(C(=O)NCC2(O)CN(C(CN(C)C(N)=O)=O)C2)CC2CC(C1)CS(=O)(=O)C2 n1(CC=C)nnnc1C(C1(C)COC1)NCCCC1CCC1 N1(C(C(C)NC(CC)(C)C)=O)CCCCC1CNC(c1ocnc1C)=O C1(CNC(COCCOC)=O)CN(C(=O)CCc2ccc(C)c(C)c2)C(C)(C)C1 Cc1ccc(C)c(C(=O)OCC2CCC(C)(C)C2)c1N C(=O)(CC(F)(F)C(F)F)NCC1CCC(NC(C2C(C)(C)OCCO2)=O)CC1 c1(CC(=O)NC(CNC(C(CCC(C)C)O)=O)C)ccc2cnccc2c1 C1(NC(Cc2c(C)n[nH]c2C)=O)CCN(C(c2c(C)noc2C)=O)CCC1(F)F C(=O)(C(CO)S)NCCCOCCOCC.C1(CC(=O)N(C)C)(SC)CC1 N1(C(C(CC)(C)C)=O)CCN(C(C2CC(F)C2)=O)C(c2cccnc2)C1 c1(C(N(C)CCNC(C2(C)CC(F)C2)=O)=O)cc(CO)n(C)n1 C1(NC(C(C2CCCC2)NC(C)=O)=O)CN(C(=O)CCc2ccncc2)CC1C C1(OC)CCC12CC(C(=O)NCC1N(C(c3cnsc3)=O)CCC1(C)C)C2 C1(CC(C)C)C(=O)N2CCC(C23CC3)C(=O)NO1.CCCCSCC(=O)OC C(=O)(C1=NNC(=O)CC1)NC1C2(CN(C(c3c(C)nc(C)s3)=O)C2)CC1 C1(NC(c2ccc(CC3CC3)s2)=O)COCCN(C(c2csnn2)=O)C1 C1(NC(C2(OC)CCCCC2)=O)CCN(C(C2CC2(Cl)Cl)=O)CC(O)C1 c1(C(=O)NCC(CC=C)NC(=O)C(C)NS(C)(=O)=O)ncc(F)cc1F N1(C(c2cnc(CC)s2)=O)CC(NC(=O)CC23COC(CF)(C2)C3)CC(C)C1 c1(OC)ccc(N(CCC(F)(F)F)Cc2nnc(C3CCCO3)o2)cc1 c1(C(=O)NC(C)Cn2cc(C3(O)CCOC3)nn2)ccc(OC(F)F)cn1 c1(-c2nnc(SCC(=O)NC(CNC(C(CC)OC)=O)C)o2)ccc(OC)cc1 c1(CC(=O)NCC2C3CN(C(=O)CCCCCF)CC23)nsc2ccccc12 C12(C(=O)NCC3CCCCN(C(=O)CCCN4CCC4)C3)CC1Cc1c[nH]nc12 c1(C(=O)NC2(CC=C)CN(c3cc(CC)ncn3)C2)c[nH]c2cccnc12 C(C)(C)(CC(C)(C)C)NC(c1cc(Cl)cc(Cl)c1)COC c1(C(C=CC(=O)NCCC(C)NC(CCc2cc(C)on2)=O)=O)ccc(Cl)cc1 N1(CC#C)CCN(C(c2cnnn2CC)C(=O)NCC)CC1=O c1(-c2cn(CCCCC(=O)NC3CCC(COC)C3)nn2)ccccc1SC C=C(F)C1(CC(=O)NCCC2CSCCN2C(=O)CC2(C(F)(F)F)CC2)CCC1 Cn1ncc(C(N2CCC(OCCNC(c3ccnnc3)=O)C2)=O)c1C1CC1 Cc1coc(C(=O)NCC(O)CNC(c2n[nH]c(C)c2F)=O)c1C CC1=C(C(=O)NCC2(NC(=O)CCc3ccc(C)cc3C)CC2(F)F)CCO1 C1(C(=O)NC(C)C(=O)OC(C)(C)C)CN(Cc2cc(Br)co2)CCC1O c1(COC)ccc(C(N2CC(O)(C(C)NC(=O)CCNC(=O)OC)C2)=O)cc1F C1(OCC)CC2CN(C(=O)C(CC3CCC3)NC(=O)Cn3cccn3)CC12 CC(CC(C)(C)C)C(=O)N1CCC(CCn2cc(-c3cncs3)nn2)CC1 Cc1ccc(CNC2CCN(C(c3ccc(C(F)(F)F)cn3)=O)CC2F)c(Br)n1 C12(C(=O)OC)CC1CN(C(C1CCC(NC(=O)CC3CC=CCC3)C1)=O)C2 c1(CCC)ccc(C(C)NC(=O)NCCCCCCO)cc1 C1(C(N(CC(CN(C(=O)CC2(CO)CC2)C)O)C)=O)CN2CCN1CC2 C(=O)(C1=CCCCCC1)NC1C(NC(C2(CC)CCCCO2)=O)CCOC1 CC1CCC(C(N2CCCC2CCNC(=O)CC2COC(=O)C2)=O)CC1 C(=O)(C(=O)CC(C)C)NCc1oc(C(=O)NC(CSC)(C)CO)c(C)c1 Cc1cc([N+](=O)[O-])cnc1C(=O)NC1CN(C(C2CCCO2)=O)CC1O c1(C(N2CC(CC(C)NC(c3c(C)cc(C)s3)=O)C2)=O)cncc(S(N)(=O)=O)c1 C(CC(C(C)(C)C)NC(C1CCCN1C)=O)N(C(C1(CC=C)CCOCC1)=O)C c1(CC)nc[nH]c1C(=O)NCC(COC)NC(=O)CCn1ccnc1 N1(C(C2C(C(C)C)C2)=O)CCC(O)(CCNC(=O)CN2CCCCC2)CC1 C12(C(=O)NC(C)CCCCNC(=O)COCC3CCCOC3)CCC(CC1)OC2 N1(C(C(CCC)OC)=O)CC2CCN(C(c3cc(F)c(C)cc3F)=O)CC12 N1(C(c2n(C)ncn2)=O)CCC(C2CC2)C1CNC(=O)CCC(C)(F)F c1(NC(N2CC(CNC(c3ccc(SC)cc3)=O)C2)=O)cccc(F)c1F CC1CCN(C(=O)CCC2OCCO2)CC1NC(C1(F)CCCCC1)=O CC1(C)CCN(C(=O)C(F)CC(C)(C)NC(C2CCSC2)=O)CC1CO C(=O)(C(O)CCNC(C1(C)CCCS1)=O)NCC1(C(C)C)CCCC1 c1(N2CCC(C(C)NC(c3c[nH]c(C(N)=O)c3)=O)C2)ncnc2scnc12 Cn1cc(C(=O)NCC2CC(O)CN2C(C2SCCCS2)=O)c2ccncc12 C1(C(=O)Nc2cc(C)cnc2C)(COC)CCCN(C(C23C(=O)C4CC2C3C4)=O)C1 C1(CNC(c2c(CC)ocn2)=O)CCCN(C(C2CC23CCCCC3)=O)CC1 C=CC(C)(C)CC(=O)NCC1C(C)CCCN1C(c1cc(C(C)(C)C)n[nH]1)=O Cc1nnccc1C(=O)NC1CC2C(NC(=O)CN3CC(=O)NC3=O)C2C1 CC1=NOC2(C1)CC(C(=O)NCC1COCCN1C(=O)CCn1cc(C)cn1)C2 C(=O)(CS(=O)C(F)(F)F)NC1CN(C(c2ccc(OC)c(N)c2)=O)CC1C Cc1c(C(=O)NCC2CCCN2C(C2(C(F)F)CCCO2)=O)oc2ccccc12 c1(CN)nnn(C)c1C(=O)NC(CNC(CN(c1ccccc1)C(C)=O)=O)(C)C c1(C(=O)NCC2C3CN(C(C(CC)SC)=O)CC32)cncc2nnn(C)c12 C(CC1=CCOCC1)NC(=O)Nc1c(OCCCN(C)C)cccn1 C(=O)(C(O)CCC(C)C)NCc1c(CNC(Cc2c(C)noc2C)=O)cccn1 N1(C(c2c(C)scc2)=O)CCN(C(=O)C(C)Oc2ccccc2)CC1CCO CC1CCSCCN1C(C1CC(C)(C)CN1C(=O)CCC1CCCC1)=O C1(CCNC(C2(SC)CC2)=O)CN(C(=O)C(=Cc2ccccc2)OC)CC(C)O1 C(=O)(C1=CC(O)CCC1)N1CCC(O)(C(C)NC(c2n(C(C)C)ncc2)=O)CC1 N1(C(=O)NC(CC2C(=O)NC(=O)N2)=O)CC2(Nc3cnnc(O)c3Cl)CC1CO2 CC1CCC(CNC(C2CS(=O)(=O)C2)=O)N(C(=O)CCc2cccc(F)c2F)C1 c1(C(N2CC(CCO)(NC(C(C)C(F)(F)F)=O)C2)=O)cccc2nc(CO)[nH]c12 C1(C(=O)NCC23CC(NC(CCCSC)=O)(C2)C(C)O3)Cc2cccc(F)c2O1 C(C)(C(=O)NNC(=O)Cc1ccc(Cl)c(Cl)c1)c1onc(C)n1 c1(C(=O)NC(C2CN(C(CCOCCCOC)=O)C2)C)ccc(C)c(O)n1 c1(C(N2CC3C(C(=O)Nc4ccc(OC)cc4F)C3C2)=O)c(Br)cc(Br)cc1Br C1(NC(C(C)=CC)=O)CN(C(=O)CCCc2cnccn2)C(C)(COC)C1 c1(SCc2scc(-c3ccc(F)cc3)n2)nc(C2CC2)ncc1Cl C(=O)(C1=CCS(=O)(=O)C1)N1CC(CCn2cc(CN(C)CCO)nn2)C1 C1(C(N(CC)CC2CCOC2)=O)N(C(c2cocn2)=O)CC12CCCC2 Cc1ccc(Br)cc1C(=O)N(C1CCN(C(c2nonc2N)=O)C1)CCO C(N=c1nc2c(cnn2C(C)C)c(NCC2CC(F)(F)C(=O)N2)[nH]1)C1C(CC)C1 c1(SCC(=O)N(C(CNC(c2cc(CO)[nH]n2)=O)C2CC2)C)ccc(F)cc1 C12(CNC(C3C(C)C3)=O)COC(CNC(=O)CCC3CCCCC3)(C1)C2 N1(C(C2CC2C2CCCO2)=O)CCC(NC(=O)C(F)(F)COCC(F)F)CC1 N1(c2ccc(NC(C(C)(C)n3ccc(C4CC4)n3)=O)cc2)CCS(=O)(=O)CC1 c1(CC(N2C(CCCNC(C(CC)(C)CO)=O)CCC2)=O)ccc2nonc2c1 C1(C(N2CC(CC(=O)OC)C2)=O)CCCC1CNC(C1(C)COC1)=O C1(CS(=O)(=O)NC(c2c(C)nco2)=O)C(C)(C)C1(C)C C1(C)(CNC(C(=O)NCCOC)=O)CCN(C(c2noc(C3CC3)c2C)=O)C1 N1(C(CCN(C(c2n(C(C)C)ccn2)=O)C)=O)CCCC2CN(C)CC12 C1(NC(C2(CC)COC2)=O)CN(C(C2CC(=O)NC(=O)C2)=O)CC2(CC2)C1 c1(C(=O)NCCC(C)NC(=O)C(C)(F)C(F)(F)F)cc2c(s1)CCC2=O C1(C(C)C)CN(CC(C2CCCN(C3CCOCC3)C2)=O)CC(=O)N1 N1(C(CCC#CC)=O)C2CCCC1CC(NC(c1ncc(Br)cc1C)=O)C2 Cn1cnc2c1CCCC2C(=O)NC1CC2CN(C(c3n[nH]cc3Cl)=O)CC2C1 Cc1nc(C(N2CCC(NC(c3cnc(N(C)C)cn3)=O)C2)=O)cn1C CC#CCC(C(=O)NCC1(C)CNC(=O)O1)NC(=O)CCC1CCCO1 c1(C(N2C(C(=O)NCCNC(C=C)=O)C=CC2)=O)c(Cl)cnn1C C1(COC)CC(CNC(c2ncccc2O)=O)N(C(c2cnn(C(C)C)n2)=O)C1 n1(CCC(=O)NC2(CC=C)CN(C(C3CC(F)C3)=O)C2)cc([N+](=O)[O-])nc1C C(=O)(C(F)(F)CC1CC1)NC1CC(Cn2cc(CC(COC)O)nn2)C1 C1(C(N(CCC#C)C)=O)CCN(C(=O)C2CN(C)CCO2)O1 c1(CC)cc(-c2cnc(C(=O)NCC(c3cccc(O)c3)O)cc2C)ccc1F C=CCCCC(=O)N(C1CCCN(C(c2cc(C(C)CC)no2)=O)C1)CC C1(N(C(C(CC(C)C)O)=O)C)CC2CCC(C1)N2C(c1ccnn1C(C)(C)C)=O C(C1CCCN1C(C1C2(CC2)C12CC2)=O)=CC(=O)NCC(C)(C)C1CCC1 n1(C(C)C)cc(C(=O)NCC2CC2NC(=O)C=CC(C)(C)C)c(Br)n1 Nc1ccc2c(c1)CCN(C(=O)NCc1ccsn1)C2 c1(N2CCC(C(=O)NC(c3ccccc3OC)CC)C2)ncnc2cnccc12 n1(CC)c(C)cc(C(=O)NCC(=O)Nc2ccc(OC)cc2)c1C CC(O)C(C)(C)C(=O)N(C1CCN(C(C2CCCC23CCC3)=O)CC1)C C1(C)(COC)CC(NC(C2CN(CC(C)C)C2)=O)CN1C(c1csc(C)c1C)=O C1(C(=O)NCC2(O)CN(C(c3cc(CC(C)C)[nH]n3)=O)C2)CCSC(C)C1 CCC(C)C(O)CC(=O)N1CC(C(=O)NC2(CO)CCC(C)(C)C2)C(F)(F)C1 c1(OC)cc(F)ccc1CNc1cc(NCC2CCC(O)C2)nc(C)n1 S(=O)(=O)(c1ccccc1Cl)NC(C1CCCN(c2cccc(OC)n2)C1)=O c1(OC)ccc(CN(C)C(N2CCC2C2CCOC2)=O)cc1F c1(NCC)ccc(C(=O)NCCNC(C23CCC(CC2)O3)=O)cc1[N+](=O)[O-] c1(C(=O)NC2CCN(C(c3c(Cl)ccc(C)c3)=O)CC2C)ncnc2ccsc12 C(=O)(C1=Cc2ccccc2OC1)NC1C(F)CCN(C(C(C=C=C)C)=O)C1 CCC(CCC(=O)NCC1(C)CCCN(C(=O)Cc2ccncc2Cl)C1)OC C(=O)(C(C)(C)C(=O)NCCNC(=O)C(c1c(F)cccc1F)(C)C)N(C)C C=CCCN=C(NCC12CC(CO1)C2)NC1CCCC(O)C1 c1(C(=O)NC2CN(C(c3cnc(CC)nc3C)=O)C(C)C2)cc(C#N)ccc1F C1(CC(=O)NCC(CO)NC(c2ccn(CCOC)n2)=O)CCCCN1C C(C)(C)(C(=O)NCCCOCCN(C)C(=O)NC1CC1(F)Cl)OCC c1(C(=O)NCC2C(C(F)(F)F)CCN(C(COC)=O)C2)ccc(S(N)(=O)=O)cn1 Cc1coc(NC(=O)C(N2CCN(CC3CCC3)CC2)=O)c1C#N C1(NC(=O)CCC2CCCO2)CCN(C(c2coc3c2COC3)=O)CCC1(F)F Cc1nc(C)c(CC(=O)NCC(O)CN(C)C(c2oc(CO)cc2C)=O)c(O)n1 c1(NC(C(=O)NCC(C)N(CCC)Cc2ccnc(CC)c2)=O)ccc(F)cc1 C(=O)(C(O)C(F)(F)F)NCC(=O)N(C)Cc1cccc(O)c1 Cc1cc(CCN(C)C)cc(F)c1F.C12CCCN(N(C)C1)C2 N1(C(c2cn(CC)nc2)=O)CCOCC(F)(CNC(=O)C(C)OCC2CC2)C1 CC(C)(C)C(O)CC(=O)NC1C2CN(C(=O)CCc3cccnc3)CC12 C1(CNC(=NCCC)NCCN2CCCOCC2)Cc2ccccc2C1 N1(C(c2c(C)n3c(s2)cnc3)=O)CCC2(CCCCC2NC(c2ccno2)=O)C1 c1(OCC(=O)NCC(CNC(c2cnn(C)n2)=O)CO)cccc(F)c1 c1(C(=O)NC(c2ccc(F)cc2Cl)CC(=O)OCC)ncn2ccc(C)cc12 Cc1ccn(C)c1C(=O)NCCC(O)C(=O)N(C(C)CCC(C)C)C Cc1cn(C)nc1C(=O)NC(CNC(=O)Cc1cc(Br)cs1)CO N1(C(CCCOC)=O)CCCC2C1CCCN2C(c1cc(C(C)C)no1)=O N1(C(CN2C(=O)OCC2)=O)CC2CCC1CN2C(c1cc2ccnc-2[nH]n1)=O CC1CN(C(c2ncccc2F)=O)CC1NC(=O)CCC1(O)CCC1 CCC(C)CCCC(=O)N1CCCCCC1C(N1CC2(C)CC1CCO2)=O c1(CC(N2CC(NC(c3ccco3)=O)C3C2C3)=O)ccc2[nH]ccc2c1 Cc1cc(CN2CC=CC2C(N2CCSC(C(C)C)C2)=O)cc(C)c1O N1(S(CC)(=O)=O)CCCC1C(=O)NC(C)(C)CNC(=O)CC1CSCCS1 C1(CNCC(C=C)O)CCCCN1C(=O)OC(C)(C)C N1(C(C2N(Cc3scc(C)c3)CCC2)=O)CCN2CCCC2C1 C(=O)(C1Cc2ccccc21)NC1CCC(N(C(=O)CCc2nc[nH]n2)C)CC1 C(c1cccnc1C)=CC(=O)NC1C(OC)CN(C(C2(CO)CCC2)=O)C1 CC1CCCc2c(C(=O)NCCCOCCCNC(C3CC3C3CC3)=O)cnn21 c1(CN2C(C(=O)NCc3ncon3)CC3CC32)ccnc(F)c1Cl c1(CCC(N2CC(O)(CN(C(=O)CC3CCCN3C)C)C2)=O)ccccc1O N1(Cc2n(CC)ncn2)CCC(CNC(=O)CNC(=O)C2CC2)CC1 c1(OC)cnc(Cl)cc1C(=O)N(C1CCC(NC(=O)C2=CCCC2C)CC1)C CCCCC(C(=O)N1CC(NC(C2(Cl)CC2(F)F)=O)C1)N(C)C C1(C(=O)NC(CC=C)CO)C2CCC(C2)N1c1cc(C(C)C)nc(C)n1 N1(C(=O)OC(C)(C)C)CC(C(=O)OCCc2ccccc2Cl)C2CCCC12 C1(CNC(=O)Cc2cscn2)CC2(CO1)CN(C(=O)Cc1sccc1Cl)C2 C(=O)(CCCC(C)(C)NC(c1csc(C#N)c1)=O)NC1CN(C(C)C)C(=O)C1 S(=O)(=O)(CC(=O)N1CCC(NC(=O)CC2CC=CCN2C)C1C(C)(C)C)N(C)C Cc1ccc(C)c(C(=O)NCCC2CN(C(C3CCC(O)CC3)=O)CCO2)n1 N1(C(C(CC=C)(F)F)=O)CC2CCCC(NC(=O)CCN3CCCC3=O)C2C1 c1(NC(n2cc(C3CCN3)nn2)=O)cccc(CO)c1 Cc1cncc(C(N2CCC(C)(NC(C3CC34CCSCC4)=O)C2)=O)c1C C(=O)(CCC(CNC(=O)NC(C1CN(C)CCN1C)C)C(F)(F)F)OC c1(C(=O)OC)c(OC)ccc(NC(=O)CCCOCCCl)c1Br.C(N)(=O)NS C1(CC(=O)NCC(C2OCCOC2(C)C)(C)C)CC(O)CN(C(N)=O)C1 C1(C(N(CCCC)CCO)=O)CCN(c2nnc(CC)o2)C1 C1(C(=O)NC2CCC(CNC(CCC(N)=O)=O)CC2)Cc2ccncc2C1 C1(C(F)(F)F)(OC)CCN(C(c2ccn(CCCF)n2)C(=O)NC2(C)CC2)C1 N1(c2cccc(CN(CC)Cc3c(C)cccc3C)c2)CCN2CCOCC2C1 c1(CNC2C(C(=O)Nc3cc(OC)c(Cl)nc3)C2)ncc2ccccn12 C1(C(=O)OC2(C3CCOC3)CC2)COc2cc(Cl)ccc2C1 CCCC(C(=O)NCC(C(C)(C)C)NC(=O)C(c1ccnn1C)C)OCC C1(CNC(C2(OC)CC2)=O)CC(OC)CN1C(c1ccc(-c2ccncc2)o1)=O c1(C(N2CC(NC(C(CC=C)CC(C)C)=O)C2)=O)cc(F)c(Cl)c([N+](=O)[O-])c1 c1(CC(N2C(C)CCC(NC(=O)CN(C)C)C2)=O)cc2cc(Br)ccc2o1 c1(C(=O)NC2(C(=O)NC(C)C3CC3)CSC2)ncn(C(C)C)n1 N#CCCC(=O)NC1CCC1CNC(=O)CCC1CCOC1 C1(NC(c2cnc(C(C)C)[nH]2)=O)CS(=O)(=O)CC1NC(c1cccn1C1CC1)=O c1(C(N2CC3CC(NC(c4c(C)onc4)=O)C3C2)=O)ccc(F)c2ccncc12 C(C)(CN=c1[nH]c(C(C)(C)C)nc(=N)[nH]1)(C1CC1)NC(C1=CCC(C)CC1)=O CC(C(F)(F)F)NC(=O)COC(C)(C)CNC(C1COCC1C(N)=O)=O N1(CC)CCCCC1CNC(CC1OCCN(C(C2COCCOC2)=O)C1)=O Cc1ccc2[nH]cc(CN3CCCCCC3C(C)C)c2c1 C12(C(=O)NCC3(COC)CN(C(=O)Cc4cc(C)n(C)n4)C3)CCC(C1)OC2 S(=O)(=O)(c1ccc(NCCCOC2CCOC2)c(Br)c1)NC(CC)C(C)(C)C CC1CCN(C(=O)CCc2cc[nH]n2)CC1CNC(=O)CC1OCCCO1 c1(C(N2CCC(N(C(COC)=O)C)C2)=O)cc(C(N)=O)ccn1 N1(C(=O)Cc2cc(F)cc(F)c2F)CCC2(CC1)CCN2C(C1CCCS1)=O CC(C)C(C(=O)N1CCC(C2N(C(c3cc[nH]n3)=O)CC2(C)C)CC1)N(C)C N1(C(c2c(C)coc2)=O)CC2CC1CCC2NC(=O)CCN(c1ccncc1)C c1(CCCC)cn(CCCC(=O)NCC2CCNC2)nn1 c1(CNC(C(=O)Nc2scc(C)n2)C)cnc2cnccn12 C1(C)(C(=O)Nc2ccc(C)nc2)Cc2ccc(C)cc2C(=O)O1 N1(C(c2cccc3c[nH]nc23)=O)CCCC2(CCCN2C(c2ccc(Cl)s2)=O)C1 c1(C(N2CC(N3CCN(S(CC=C)(=O)=O)CC3)C2)=O)cccc(C)c1O c1(C(N2CCC(NC(C(COC)C)=O)C(C)C2)=O)cc([N+](=O)[O-])cnc1N C(=O)(C(CNC(=O)CC(O)CN(C)C)C(C)(C)C)NCCCC(C)OC N1(C(CCC2CCN(C)C2)=O)C2CCC1CC(N(C(=O)C#CC1CC1)C)C2 c1(N(C(C)=O)C)ccccc1C(N1CC(F)CC1CNC(=O)CCC(C)N(C)C)=O Cn1nc(C(=O)NC2CCCC(CNC(=O)CCCNC(N)=O)C2)cc1F CC(C)C(C(=O)N(C)C)NC(C1CC(C(=O)OCC2CC2CO)C1)=O c1(C(=O)NC2CCN(C(CC=C)=O)C2)nn(C)c2ccc(F)cc12 n1(CC)ncc(Br)c1CS(=O)C(C)c1csc(=N)[nH]1 c1(OC)ccnc(C(=O)NCCC2CCCN(C(C3(C(N)=O)CCC3)=O)C2)c1 C1(N(C(=O)C=CC2CCC2)CC#C)CCN(C(C2CC2c2ccccc2)=O)C1 c12cc(ccc1F)CN=C(NCC(C)(O)C1CC1)NC2.C(F)(F)F.C(=O)(COC)NC c1(C(N2CC(CC=C)(NC(c3ccc(CCC)s3)=O)C2)=O)cc(OC)nc(Cl)c1 C#Cc1ccccc1C(=O)Nc1cccnc1C(=O)Nc1cnc(Cl)c(Br)c1 CC(C(=O)NNC(=O)NCc1nc(C(F)(F)F)cs1)NS(=O)(=O)c1cccnc1 C1(C(=O)NC2C(C)C2)CCN(C(=O)COc2ccn(C)n2)O1 c1(C(C(=O)NCC(CC)NC(=O)C(O)C2CC2)C)ccc(C)o1 CC1CC(C(=O)NCCN(C(=O)CCNC(c2cccc(Cl)c2)=O)C)C1(C)C C(=O)(C(C)(F)C(=O)N(CC(C)NC(=O)CCc1ccccc1F)C)OCC Cc1ccc(-c2cc(C(=O)NCCCNC(=O)CC3(C)CC3F)on2)cc1 C(=O)(CC(C)(C)C(C)(F)F)NC1C(CNC(C(CCC)C(C)C)=O)C1 C1(OC)CC(NC(=O)C2CC2)CN(OC(c2cnc(N3CCC(C)CC3)s2)=O)C1 N1(C(C(C=C=C)C)=O)CCN(C(c2cc(C)nn2CCC)=O)C(c2ncc[nH]2)C1 N1(C(C=Cc2ccc(C)s2)=O)CCC2C1CCCN2C(C1(C2CC2)CC1)=O c1(C(N2CCC(CCNC(CNC=O)=O)C2)=O)nc[nH]c2ncnc1-2 C1(C(N(CC(C)N)C)=O)CCNC12CCCC2 c1(C(=O)OCC2C3CCCCC23)cc(Cl)cc2cc[nH]c12 c1(CNC(C2(CO)CCN(C(C3CN(C)C3)=O)C2)=O)c(F)cncc1F Cc1ccn2ncc(C(=O)NC3CC(NC(=O)Cc4sccc4Cl)C3)c2c1 C1(OC(C)C(=O)N(CC(C)N(C(=O)Cc2cncs2)C)C)CCCCC1 c1(C(=O)NCC(CC)NC(=O)C(C)CC2CC2)cc(F)c(O)c(Br)c1 C(CC(=O)NC(C)C=CC(=O)N(C)CC)(CC)OCC1CC1.C12CC(C1)C2 N1(C(c2c(C)cccc2)=O)CC(NC(=O)CCCn2cccc2)CC1(C)C N1(CC(N2CC(C)OCC2)=O)CC(NC(C2CC2C)=O)C(C)(C)C1 C1(n2cc(CC(OC)OC)nn2)C=CCC(C(=O)NCC(C)(C)C(C)O)C1 N1(C(C=COCC)=O)CCCCC1CCN(C(=O)C=CCCc1ccccc1)C C1(N(CCCC)C(=O)CC2CCCCC2)CCN(C(=O)COC2CC2)CC1 C1(O)(C(N(C(c2cn(CCCC(=O)OC)nn2)C)C)=O)CCCC(C)(C)C1 c1(OC)cc(C(N2CC3CC(C2)C3NC(c2nnc(O)nc2O)=O)=O)c(Cl)cn1 C1(NC(c2cn(C)nn2)=O)C=CCN(C(=O)CCc2ccc(C(N)=O)cc2)C1 C1(CNC(CN(C)S(N)(=O)=O)=O)CCN(C(c2cc(C#N)cs2)=O)C12CC2 c1(C(N2CC3CCCN(C(C4C(=C)CC4)=O)C3C2)=O)ccc2c(c1)C(=O)C(=O)N2 c1(C(=O)NC23CN(C(C(C(C=C)C)C)=O)C(C2)C3)ccc(C)c([N+](=O)[O-])c1 N1(c2cc(CC)ncn2)CCC(NC(c2n[nH]c(COC)c2I)=O)CC1C C12=NC=CC(=NCCCC(=O)N1)N2.C(CCCNC(c1ccco1)=O)OCC c1(OC)ccc(CC(CNC(=O)NOC2CCC2)CO)cc1O N1(C(c2csc(C)c2N)=O)CC2C3CCC(C2C1)N(C(=O)CSCCN(C)C)C3 C1(C(=O)NCC2(OC)CCN(C(=O)C(O)P(C)(C)=O)CC2)OCCOC12CCC2 Cc1cccc(CC(=O)NCCC(C)(C)NC(C2CCCC(C)(C)O2)=O)c1C C1(NC(c2c(C)c[nH]n2)=O)CC(N=c2nc[nH]s2)C1(C)C CC(CS(C)(=O)=O)C(=O)NC1CCC(NC(=O)Cc2cnn(C)c2C(F)F)C1 Cc1ncsc1C(=O)NCCCC(=O)NC(C1CCN(C(=O)CN(C)C)C1)(C)C c1(C(=O)NCCCN(C(C2(CC3CC3)CCC2)=O)CC)cocc1C(N)=O C(=O)(C(C)(C)C(C)O)N1CC(NC(c2c(C)sc(-c3ccco3)n2)=O)C1 C1(C(=O)NCC2CCN2C(=O)CSCc2ccc(Cl)cc2)CC2CC1CC2(F)F C(CCCCC(=O)NC(CC1CCOCC1)C(=O)NC(C)CCOC)OCC C1(NC(C#CC2(C)CC2)=O)CC2CCC1CC2O N1(C(C=CC)=O)CCCN(C(c2c(F)cc(Cl)cc2F)=O)CC1CO c1(C(N2CCC(O)(C(C)NC(c3c(C)nc(CO)s3)=O)C2)=O)cc(C#N)[nH]c1C c1(CNC(=O)NCC2(COC)CCCCO2)ccn2c(C)ncc2c1 C(c1ccc(C(F)F)o1)=CC(=O)NC(CNC(C(CC)OCC)=O)CC C(C(O)CC(=O)N(CC(C)(CC)OC)C)NC(c1c(CCC)n[nH]c1)=O C1(C(N(CCCNC(CNC(N)=O)=O)CCO)=O)CCCCN1S(N)(=O)=O c1(CC)cccc(C(N2CCOCC2CCO)=O)c1O N1(C(C2CCC(CC)O2)=O)CCC2(C1)CN(C(=O)CC(CC)Sc1ccccc1)C2 C1(CNC(c2ccc(F)c(Cl)c2)=O)CCN(C(=O)CC2(O)CCOC2)C12CCC2 c1(OCC)ccc(C(=O)NCCC2(O)CCCN(C(=O)C(Cl)=CCl)C2)cc1OC C1(NC(c2cnc(C(F)(F)F)c(Cl)c2)=O)CCNCC12CCC2 C1(NC(=O)CCC2CCCCC2)CC2CC1N(C(=O)CN1CCCNS1(=O)=O)C2 O=S(=O)(c1ccc(NCCC2(C3=CCOCC3)CC2)c(F)c1)NC1CCSC1 Cc1ncccc1CC(=O)NC(C)C(C)(C)NC(c1sc(F)cc1C)=O C1(CNC(c2cc(C)ns2)=O)CCCCN1C(=O)C(F)(F)C1(O)CCCC1 CCCCCC(O)C(=O)NC(CC)CCCC(=O)N(C)Cc1occc1C C1(C(=O)NC2CC(CC(=O)NCCc3ncc[nH]3)C2)CCC=CCCC1 C(C(CC)CC(C)C)NC(C(Cc1ccccc1Br)NC(C=CC)=O)=O N1(c2c(C)c(NCCN(CC(F)(F)F)C)ncn2)CCc2[nH]ccc2C1 c1(C(=O)NCC2C(NC(CN3C(C)CC3)=O)C2)cccc2c1oc1ccccc21 Cc1noc2ncnc(N3CCCC(CNC(=O)CSc4nncn4C)CC3)c12 c1(C(=O)NCCNC(C(C)Oc2c(Cl)ccc(C)c2)=O)nc2sccn2c1C c1(OC)cccc(C(N2CCC(CC(=O)NCCCN3CCOCC3)C2)=O)c1F c1(CC)ccc(C(=O)NCCC2C(C)CCCN2C(c2n[nH]cc2C)=O)cc1Cl CCC(CC)C(C(=O)N1CC(CNC(c2c(C)nsc2C)=O)OC(C)(C)C1)OC C1(C(=O)NC(CCN(C(C2CC(OC)C2)=O)C)C)CC=CCC1C c1(CNC(N2CC3(CC(C(=O)O)C3)C2)=O)cccc2c1oc1ccccc21 C1(CC(=O)NC2C(SC)CC2O)CN(C(C2(CC(=O)OC)CC2)=O)CC1C n1(CCCC(=O)NCC2CCC(NC(C(C)N(C)C)=O)C2)c(O)nnc1O C(C)(C)(CC(=O)N1CC2CC1C2CNC(c1ccc(Br)o1)=O)OC C1(N(CC#C)C(C2(CC)CCOC2)=O)CCN(C(C2CC(CN(C)C)C2)=O)CC1 N1(C(Cc2c(C)cnn2C)=O)CC=C(C(=O)NC(C)CS(C)(=O)=O)CC1 c12ccc(cc1)C(C)N(C(=O)OC)C2=O.c1(C(c2ccco2)SC)ccco1 C1(CN=C(NCC(C)C)NCC(C2CCCC2)C)COc2ccccc2O1 Cn1nc2c(c1C(N1CC3C(NC(=O)CNC(=O)C4CC4)C3C1)=O)COCC2 CC(C)C(CCN(C)C(C1CSCCS1)=O)N=c1[nH]c(Cl)ncc1Cl Cc1cc(C(=O)NCC(C)(C)CN(C)C(c2cc[nH]n2)=O)ncc1S(N)(=O)=O c1(NC(CCC2(NC(c3ncn(C(C)C)n3)=O)CCC2)=O)cn(C)nc1C#N Cc1c(C(=O)N(c2nc(CN(C)C)c(C(F)(F)F)s2)C2CCCCC2)nnn1C C1(CNC(=O)Cc2ncncc2Cl)CCC(F)(CNC(C2(F)CCOC2)=O)CC1 c1(C(N2CC(C3CN(C(CCC(=O)OC)=O)C3)C2)=O)cc([N+](=O)[O-])cc(C)c1Cl N1(C(C(=O)NCC(C)C)C2CCC2)CC(CO)CC1(C)C c1(NC(C2N(Cc3ccn(C)n3)C3C(C2)C3)=O)cc(O)ccc1[N+](=O)[O-] c1(C(N(CCNC(c2cc(CO)[nH]n2)=O)CC)=O)nccc2ccn(C)c12 N1(CC(N2CC(CNC(C=COCC)=O)OCCC2)=O)C(=O)NC(C)(CC)C1=O c1(C(=O)NCC2(NC(c3ccn(C)c3)=O)CC(OC)C2)cc(F)cc(F)c1 N1(C(Cc2c(C)n[nH]c2C)=O)CC2CCCCC2(CN=c2[nH]nc(C(F)F)s2)C1 N1(C(CC2(C=C)CC2)=O)CCN(C(=O)C(F)F)CC2CCCCC12 N1(c2cc(NC(C=C)C)nc(COC)n2)CCC2(CCC2)S(=O)(=O)CC1 C(C(=O)N1CC(=O)NC(C)C1)(C(C)(C)C)NC(c1c(OC)scc1)=O c1(C(=O)OC)cnc(CNCC2CCCC2C(=O)NC2(NC(C)=O)CC2)cc1C CC1CC(C(=O)NC(C)CN(C)C(c2cc3[nH]ccc3s2)=O)CCN1C N1(C(CC)=O)CCC(C2CCCN2C(=O)NCCSCCO)CC1 C1(F)(CNC(c2nc(CS(C)(=O)=O)oc2)=O)CCN(C(C2COC(=O)N2)=O)C1 C1(CNC(C(CC)n2ccnc2)=O)CCN(C(c2cn(CCO)nn2)=O)CC1C C(CC(C)(C)S(C)(=O)=O)NC(CCN(C)C)(C)c1nnnn1CCC1CC1 c1(C(N2CC(CC)N(C(=O)CCNC(N)=O)CC2)=O)cc(C)c2[nH]cnc2c1 CS(=O)(=O)C1CCN(C(c2ccc(CCC(=O)NCCN3CCCC3)[nH]2)=O)CC1 C1(OCCn2cc(-c3c(C)ccs3)nn2)CCN(C(=O)Cc2cn[nH]c2)CC1 C1(C(N(CCCN(C(C=CC(=O)OC)=O)C)C)=O)CC1(C)C(C)C c1(SC)ccc2cc(C(N3CC(NC(=O)CCn4ccnn4)C4CC34)=O)[nH]c2c1 CC1CC(N=c2[nH]n(C)c(C3CCCC3)c2[N+](=O)[O-])CN1C(C1C=CCCC1)=O c1(OCC)ccc(Br)cc1CNC(=O)NCc1ccc(F)cc1 S(=O)(=O)(c1[nH]c(=NC(C)CCF)ccc1Br)NCC(N1CCCCC1)C c1(C(=O)N(C2(C)CC(F)C2)C2CC2)ccc(Br)cc1 Cc1nc(C(=O)NCC2CCN(C(c3scnc3C(F)(F)F)=O)C2)nn1C c1(C(=O)OCC)cc(NCc2nc(C(C)(C)C)no2)cc(Br)c1C Cc1sncc1C(=O)NC(CO)C(C)NC(C1CC1C(N)=O)=O C1(C(=O)NC2(C)CN(C(CCc3ccn(C)c3)=O)C2)CCn2cnnc2C1 C12(CC)CC1CN(C(C1C(O)CCN1C(c1cc(Cl)ns1)=O)=O)C2 Cn1ncc2c1CCC(C(N1CC3CC(NC(C4(CO)CCCC4)=O)C1C3)=O)C2 C1(CNC(c2cccc(C)c2)=O)C(C2CC2)CCN1C(=O)Cc1ccnn1C CC1(C)OCCC1C(N1CCC2CC12C(=O)NCCC1CC=CCC1)=O CCCCC(O)CC(=O)NCCC1(CNC(=O)C(C)Cc2cccc(F)c2)CC1 N1(C(c2c(SC)ccs2)=O)CCCC2C1CCCN2C(C1CN(C2CCC2)C1)=O c1(SC)cc2[nH]ccc2cc1-c1cccc(F)c1C Cc1nsc(C)c1C(=O)NCC(C1CCC1)NC(c1cc(C(C)(F)F)n[nH]1)=O Cc1ccc(CCC(=O)N(CCNC(C2CCCN2CC(C)C)=O)C2CC2)s1 C=CCC(CC)C(=O)NC1(CO)CCN(C(c2cnc(CO)nc2C)=O)C1 C=Cn1nncc1C(=O)N(C(C)C(N1CCCC1C(=O)NC(C)C)=O)C C#CC1(O)CCN(C(C2(CNC(C3CN(C)C(=O)N3)=O)CC(=C)C2)=O)C1 Cc1nc(CC(C)C)c(C(=O)NCC(C)CN(C)C(C2(C)CC2)=O)s1 c1(N(C2CCCN(C(=O)C(c3ccc(F)cc3)F)C2)C)ncccc1[N+](=O)[O-] C1(C(=O)NC(CNC(C(C)=CC2CC2)=O)C)CNc2ccnn2C1 N1(C(C(CSC)C)=O)CCN(C(c2c(Cl)nsc2Cl)=O)CC1C1CCC1 N1(C(C(CC(C)C)OC)=O)CC2CCCC(C1)N2C(=O)Cn1c(C)c(C)sc1=O C(=O)(C(F)C(F)(F)C(F)(F)F)NC1C(NC(CCOC(C)=O)=O)CC1 N1(c2nccc(C)n2)CCC(O)CC1C(=O)Nc1cnc(F)c(Cl)c1 Cc1cc(CNC(=O)C(CCC2CC2)NC(c2nocc2C)=O)cc(C)n1 C1(CCC)(NC(C2CCC2OC)=O)CCCN(C(c2cccc(=S)n2O)=O)C1 C12(CNC(=O)CCCc3ccccn3)CCC(CC1)N2C(C1CCCCC1F)=O c1(OC)cccc(F)c1C(N1CCN(C(=O)COCc2ncc(C)o2)C(C)C1)=O c1(C(=O)NCC(CNC(C(C(C)C)SCC)=O)O)ccc(O)cc1[N+](=O)[O-] N1(C(Cc2ncc(C)s2)=O)CC2CCN(C(=O)CC34CCC(CC3)C4)CCC2C1 N1(C(C2CCN(C(CC)=O)C2)=O)CC(C)(C)CC1CNC(=O)CCC1(C)CC1 N1(C(CCNC(=O)C=CCl)=O)CC(NC(=O)CNS(=O)(=O)C2CC2)CC(O)C1 c1(NC(C2N(Cc3ccc(CC)cc3)CC=C2)=O)cnc(C#N)c(C)n1 C12(C(=O)NCC3CCCCC3NC(=O)CCN3CCCC3=O)CCC(CC1)CO2 N1(C(c2cccn(CC#C)c2=O)C(=O)NCCCC)CCC2(CC1)CNC(=O)C2 c1(C(=O)NCC2N(C(C(N3CCCCC3=O)C)=O)CCCC2)[nH]cc2c1CCC2 c1(C(=O)NCC2N(C(CSCC(C)C)=O)CC=C2)ccc(F)cc1F C(=O)(CCC(F)(F)F)NCCC(C)N(C)C(c1ccc(CO)nc1)=O C(=O)(C1=NOC(C(N2CC3CC2C3CNC(=O)CC2CC2(C)C)=O)C1)OC C(C(C(=O)N1CC(c2cc(O)no2)C1)C(C)(C)C)NC(C1N(CC)CCC1)=O C1(C(N(C)CC2CCCN2C(c2ccsc2C#N)=O)=O)CSc2ccccc2O1 C12(C(N(C(C)CNC(=O)C(=O)N=S(C)(C)=O)C)=O)CCC(N=[N+]=[N-])(CC1)C2 C1(C2(O)CCN(C(=O)C(C)(F)CCCC)CC2)(NC(CCC(=C)C)=O)CC1 C1(N(C)C)CCCN(C(=O)CC2(C)CCN(C(C3(CO)CCCCO3)=O)C2)CC1 C1(OCC)CCCC1NC(=O)C(C1CCC1)NC(=O)CC1CCOC1C C1(C(=O)NC2CC3N(CC(=O)N(CC)CC)C(CC3)C2)COc2ccccc2O1 N(C1COCc2ccccc21)C(C1CCC(NCc2cc(I)ccc2F)C1)=O c1(OC)ccc(CCC(=O)NC2CCC2NC(c2ccc(C)nc2)=O)cc1Cl c1(CC)ccc(C(=O)NC(C)(C)CNC(=O)CCC2CC2(Cl)Cl)c(C)n1 C(CC)(C(=O)NC1CC(CNC(=O)C(C)CC2CCCC2)C1)=CCCC c1(CN(CCCN2CCCC2=O)C)cc(Cl)ccc1Oc1ccccc1 C12(C(=O)NC(C3CCN(C(C4(C)CC(C)C4)=O)C3)C)CC3CC(C1)CC(C)(C3)C2 c1(OOC(CC(C)(C)N(c2ncc(C)s2)C(C)=O)=O)cccc(CC2CCN2)c1 CCC(CCCC(=O)N1CCC(N(C)C)C1C)NC(C1CC12CCCC2)=O c1(C(=O)NCC2CCN(Cc3cccc(OCOC)c3)C2)ccc2c(c1)CCO2 C1(C(=O)NCC2(C(=O)NCCC#C)CCC2)CC2CC(=O)C1O2 C=CC(C)(O)CC(=O)N1CCCC1C1CCN(C(C2CCCN(C)C2)=O)C1 C1(C(=O)NCCC(C)CCO)CCN(C(c2cccc(=O)n2C)=O)CC1O C1(CCCC)(C(=O)NC2(CCCNC(C3CC(C(N)=O)C3)=O)CC2)CCCCC1 CCCC(C(=O)NC1CC1)NC(=O)CCN=[N+]=[N-] N1(C(C2(CC#C)CC=CCC2)=O)CCCC(NC(c2ccc(N)c(F)c2)=O)CC1 C(=O)(C(CC(N)=O)NC(=O)CN1CCCC1C)NC1(CCC)CCOC1 CC1(C)CC(CC(=O)NCC2CN(C(=O)CSCC(F)(F)F)CC2O)CCO1 CC(C)CCCCCN(C(=O)CNS(=O)(=O)c1cccs1)C(C)C Cc1nc(NCCCCCCC2CC2)cc(=NCC2(CS(C)(=O)=O)CCC2)[nH]1 C(=O)(C(C)(C)C(F)(F)F)NC1CCCC(NC(C(CC)(C)F)=O)C1 c1(C(N2CCC(C)(CNC(c3ncn(C(C)(C)C)c3)=O)C2)=O)cc2n(n1)CCC2 C(=O)(C1=CCCC1(C)C)N(CC(CNC(C(C(C)C)O)=O)O)C N1(C(CCN(CCCCC)C)=O)CCCC(CC)(NC(=O)C=C2CCC2)C1 c1(C(=O)NCC(CC)(CC)NC(C2ON=C(CC)C2)=O)cc(C#N)cn1C N1(C(C2CCCC(=O)C2)=O)CCC(NC(c2ccc(C(F)F)cn2)=O)CC(O)C1 c1(C(=O)NC2(C)CN(C(C(N3CCNC3=O)C)=O)C2)ccnc(C2CC2)n1 C1(C)(C(N(C(CC#C)C)C)=O)CC(NC(=O)C(C)CC2CCCC2)C1 c1(C(=O)NCC2N(C(c3cc(C)on3)=O)CCCC2C)nccc2ncccc12 C1(C(=O)NCCC2(O)CN(C(C3Cc4nncn4C3)=O)C2)CCC12CCOCC2 c1(CCC(=O)NCC=CCNC(C(C)=C(C)C)=O)nnc(S)n1C N(C(=NCC(C)C)NCc1cnc(C)o1)CC(c1ccc(OC)cc1)O N1(CCc2c(C)nn(C)c2)CCC(=O)N(CC2(C(F)(F)F)CC2)C1=O c1(NCCC2CC(OC)C2)ccc(S(=O)(=O)NC2CC2C2CCOCC2)c(Br)c1 C1(NC(c2cc[nH]c2)=O)CCN(C(=O)C=C2CC2)CC1F c1(COC(CNCC(Cc2cn(C)nc2)C(F)(F)F)=O)ccc(S(=O)CC#N)cc1 C1(CNC(C2(F)C(C)C2)=O)CCCN1C(c1cc(CN)cs1)=O.C(C)(C)(C)OC=O N1(C(C(c2n(C)ccn2)(F)F)=O)CCC(C)(CNC(=O)Cn2nccc2N)CC1 C1(C(=O)OCC)CN(C(C)C(=O)Nc2nnc(C(C)(C)C)s2)CCC1(F)F N1(C(C(CNC(CC(C=C)CC)=O)CCC)=O)CCC2CN(C)CC2C1 CC(C)C(C)CC(=O)NCC1(O)CCCN(C(=O)Cn2ncn(C)c2=O)C1 N=c1[nH]cc(C(N2CCC2c2ccccc2)=O)o1 C1(NC(C2CN(C(C)C)C2)=O)CC2(CCCCN2C(=O)CCc2nncs2)C1 c1(CC(=O)NC2C(CNC(C(C)S(N)(=O)=O)=O)C2)ccc2c(c1)COCC2 N1(C(=O)NC2CCC(CC)CC2)CCN(C(c2cccc(F)c2F)=O)C(C)C1 O=C1CCN(CC2CSCCS2)C(=O)N1CCc1ccnn1C1CCC1 C(=O)(C(O)C1=CCCCC1)NCCC1N(C(C(C2CCCCC2)C)=O)CCCC1 C12(NC(C(C)NC(N)=O)=O)CCCC1N(C(c1cccc(F)c1N)=O)CCC2 c1(CC(N2CCCC(n3cc(CC(COC)O)nn3)C2)=O)cc(F)cc(Br)c1 C1(C(=O)NCc2n(C(C)C)ncn2)CCCC2NCCC12 c1(OC)ccc(CNC(=O)C(c2csc(C#N)c2)N2CCCC2C2(C)CC2)cc1 C1(C(N2CC(C)(CC=O)C2)=O)CC(C)CN(N2CC(C(CC)CC)C2)C1.C(C)(C)(C)C N1(C(C2(CC)COC2)=O)CCCC2(CC(NC(=O)C(C)(C)c3cnsc3)C2)C1 C1(NC(C(C)(C)S(C)(=O)=O)=O)CC2CCC1CN(C(C1CC1C1CCCC1)=O)C2 c1(C(N2CC(C)CC(NC(CCC(C)=O)=O)C2)=O)cc(S(N)(=O)=O)ccc1C c1(OC)cccc(C(=O)NCC(C2CCN(C(C3(F)CC3C)=O)CC2)C)c1Cl c1(N2CCN(C(C3C4CCCCCCC34)C)CC2C)nc2c(C)cccc2o1 C(C)(CCCC(=O)NCCC1CC1)NC(Cc1cc(C)[nH]n1)=O C1(F)(C(N2CC(C=C)C2)=O)CCN(C(c2ncsc2C)=O)C1 C(=O)(CC(C)C(=O)N1CCC(C=CC(=O)Nc2cc(OC)cc(O)c2)CC1)OC Cc1noc(CCC(=O)NCC(O)CCNC(C2CNC(=O)C2)=O)n1 C1(C(N(CC#C)CCOC)=O)CCC(C2CC2)N1C(=O)Cn1ccnn1 N1(C(CC2CC(=C)C2)=O)CC(NC(c2cnc(C)nc2)=O)CC(O)C1 N1(C(C=C(C)C(F)F)=O)CCC(NC(c2ccc(CS(C)(=O)=O)o2)=O)C(C)(C)C1 C1(CNC(COCc2cccc(C)c2)=O)C(O)C(O)CN1C(=O)C(C)C(C)C C1(NC(c2sc(C)c(Br)c2)=O)CC2CC1N(C(C1CCC(=O)C1)=O)C2 c1(C(N(CC(C)NC(C2(CC=C)CC2)=O)C)=O)cc(SC)oc1C CCC(CC(=O)N(C)CC1C2CN(C(=O)CSC(C)(C)C)CC12)C(C)C c1(C(N2C(CNC(CCC(=C)Br)=O)CC3CC32)=O)cn2c(n1)CCCC2 C1(c2cn(N3CC4C(Sc5ncc(C)nc5)C4C3)nn2)CCCCC1C1CC1 C1(CNC2CC(=O)N(CC(F)(F)F)C2)CCCS(=O)(=O)N1 C1(NC(C2(NC(C3(CO)CCOC3)=O)CC2)=O)CC(C2CC2)C1 c1(OC)ccc(CN2CCCC(CNC(=O)CC3CCC(C)C3)C2)c(OC)c1 C(=O)(C#CC1(C)CCCO1)NC12C(CN(C(CCCOCC=C)=O)C1)CCC2 n1(CC)cc(C(N2CC3CC3(CNC(C3CCNC3=O)=O)C2)=O)c(C(F)(F)F)n1 C(=O)(C(CCCC(C)(F)F)NC(=O)NC(C)C)Nc1c(C)n(-c2ccccc2)nc1 N1(C(C(CCC)O)=O)CCC(C)(C)C1CNC(=O)C=Cc1ccc(C2CC2C)o1 C(=O)(CC(CC)C(C)C)NC(=O)NCC(CN(C(C(COCCC)(C)C)=O)C)(C)C C1(NC(C(CC)=CC)=O)CCC2(CC1)CC2NC(=O)C(=O)NCC N1(C(CC(CCCC)CC)=O)CC2CCN(C(=O)C(CC)CCOC)CCC2C1 c1(C(N2CCC(C)(CNC(=O)CC3COCCOC3)C2)=O)cccn2nccc12 c1(CC)nc(C)oc1C(=O)NCc1occc1C(=O)NCCS(C)(=N)=O N1(C(CC(CC)CN(C)C)=O)CC2CCN(C(=O)C3=CCCCC3)CC12 C(=O)(C1CCNc2cc(F)ccc21)NC(C1CN(C(C2CC(C)(F)C2)=O)C1)C Cc1cccc(C(CNC(c2ncoc2C)=O)NC(=O)CCc2cnn[nH]2)c1 C1(NC(C(C)Cc2ccccc2Cl)=O)CN(C(=O)Cc2cccnc2)C(C)(C)C1 c1(C(=O)NC2CN(C(C3(C)CCN(C)C3)=O)CC2F)ccc2nnn(C)c2n1 N1(C(C2(OCC)CCCCC2)=O)CCCCC2(CCN(C(=O)C(C)C(C)O)C2)C1 N1(C(C)C)CCCC(CC(=O)NC2CCC(NC(=O)C(CO)NC(N)=O)CC2)C1 C1(C(N2CCC(N(C(=O)COCC3CCCO3)CCC)C2)=O)NC(=O)OC1(C)C C1(NC(CCCCCCSC)=O)CCCC2CN(C(=O)C3=C(C)OCC3)CC12 c1(C(=O)NCC(C(C)C)NC(C2(C)CCCO2)=O)cc[n+]([O-])cc1 Cn1ncc2c(O)c(C(=O)NCC#CCNC(=O)Cc3csc(Br)n3)cnc12 c1(N(C(C2C=CC(NC(c3nc(CC)oc3)=O)C2)=O)C)ccc(C)cc1C N1(C(CC(C)SC)=O)CCOCCC1C(=O)NCCOCC(N)=O CC12CCN(C(C3CCCCC3(F)F)=O)C1CN(C(C1CCCN1C1CC1)=O)C2 c1(CC(=O)NC2C=CCN(C(C3(F)CCCOC3)=O)C2)cc(Cl)ccc1[N+](=O)[O-] C1(COC)CN(C(c2coc(C3CC3)n2)=O)CCN1C(C1CC1F)=O.c1nncs1 N(C(=NCCCc1nnc(C)n1C)NC(C)COC)C(CC)C(F)F C1(CC(=O)NCCC=CC)CN(C(c2ccns2)=O)C(C)(C)C1 C1(C(N2CCCC(OC)C2)=O)C2CCCC1CN(C(c1cc(Cl)nc(Cl)c1)=O)C2 C(=O)(CCC(C)(C)C)NCc1ccc(C(N2CCCC(OC)C2)=O)o1 c1(C(N2CCC(CNC(=O)C=C3CCC3)C2)=O)n[nH]c(C(F)(F)F)c1Cl c1(SCC(=O)NC(CN(C(=O)Cn2ccnn2)C)(C)C)n[nH]c(O)n1 c1(OCCOC)ccc(F)cc1C(=O)N(CC(C)CNC(=O)C=CC1CCC1)C C(CCCCCN=c1ccc(S(C)(=O)=O)c[nH]1)NC(C(CC)OC1CCCC1)=O c1(C(N2CCC(C)C(CNC(=O)CCc3cnn[nH]3)C2)=O)cnc(O)n(C)c1=O C#Cc1cc(F)c(C(=O)NC(CNC(C23CCN(CC2)C3)=O)C(C)C)c(F)c1 N1(C(C(CC)N(C)C)=O)CC2(COC(CNC(=O)C(F)=CC3CC3)C2)C1 C(=O)(CN1C(=O)CCc2ccccc21)N1CCC(NC(C(CC=C)C)=O)CC1C c1(C(=O)NC(C)C(CO)NC(=O)CC2CC=CCC2)cc(O)nc2c1CCCC2 CC1=C(C)CC(C(=O)NCC(CC(C)C)NC(c2cc(C)c(O)nn2)=O)CC1 c1(OC)cccc(C(=O)NCCN(C(=O)C(C)(C)CSC)CC2CC2)c1 C(=O)(C1=CCCCCC1)NC1CCN(C(Cc2c(OC)ccc(F)c2)=O)CC1O N1(C(C(C2CCN(C(CSCC)=O)CC2)C)=O)CCC2CN(C)CCC12 c1(C(C(C)NCC(=O)C(C)=O)N)ccccc1.C(C)(C)OC.C1(=O)CC2(CC2)N1 C1(C(C)NC(C2CCC2)=O)CCN(C(=O)C=C(Cl)Cl)C1 C1(NC(=O)CC2(C(F)(F)F)CCC2)CC(O)CN(C(c2ccon2)=O)C1 N1(C(C2(CO)CCC2)=O)CC(C(N(C2(C(=O)OC(C)(C)C)CC2)C)=O)C2(CC2)C1 N1(C(CSCC=C)=O)CC(NC(c2sccc2OCC)=O)CC1(C)CC CC(C)C(C(=O)NCC1(CCNC(C2CC(Cl)(Cl)C2)=O)CC1)n1cncn1 c1(CN2CCC(C(=O)Nc3c(C)[nH]nc3Cl)C2)c(Br)cc(Br)c(O)c1Br C1(CC)(CC)CCN(C(=NCc2ccc3c(c2)ncn3C)NC)C1.CS(C)(=O)=O c1(CC)nc(C)c(CNC(=O)CC2CCCN(C(c3nc(C)oc3C)=O)C2)o1 CCCCCCCNC(c1ccc(Br)s1)c1nnnn1C1CC1 N1(C(CC2CC(OC)C2)=O)C2CC1CN(C(c1ccc(C)c(C)n1)=O)C2 N1(C(C=NOC)=O)CCCC(C)C1CNC(=O)Cn1nc(C(F)F)cc1C C1(NC(C2(COCC)CC2)=O)CN(C(=O)CC2CS(=O)(=O)C2)CC1S(C)(=O)=O c1(Cn2cc(-c3c(N)cc(F)cn3)nn2)cc(F)cc(Br)c1Cl CC1CC2CN(C(c3cccs3)=O)CC2N1C(c1ccc(=N)[nH]n1)=O c1(C(=O)NCC2CCC(NC(C3CC3(F)F)=O)C2)c(Cl)csc1Cl N1(C(COCC=C)=O)CCCC2C(CCCN2C(=O)CN(S(C)(=O)=O)C)C1 c1(C(N2C(CNC(c3[nH]cnc3C)=O)CC(OC)C2)=O)cccc2[nH]ncc12 C=CC(CCC)CC(=O)NC(CCCC)CC(=O)NCC(CC)CCCC CC(C)C(C)CC(=O)N(C1CCC(NC(=O)COC2CCOC2=O)CC1)C N1(C(C2N(C)CCC2)=O)CCCCCC1CNC(C1OC2CCC1CC2)=O N1(C(c2csc(C(F)(F)F)n2)=O)C2CN(Cc3cnc(Cl)nc3)CC12 CN1CCC(NC(c2cccnn2)=O)C12CCCN(C(=O)C1=C(Cl)CCOC1)C2 C1(CCNC(CC(C)NC(=O)C2CC2)=O)CSCCN1C(c1cscc1F)=O N1(C(CN(C(C)=O)C)=O)CCC(C)(CCNC(C2(COC)CCOC2)=O)C1 CC1(NC(C2CC2F)=O)CCN(C(c2ccc(C(F)(F)F)o2)=O)C1 C1(n2ncc(C)c2)CCN(C(c2cc(C(=O)O)n(-c3cccc(F)c3)n2)=O)CC1 N1(C(C(C)=O)=O)CCOCC2(COCCN2C(=O)C#CC2CCOCC2)C1 c1(CNC(CC(C)=O)C)nn(C)c2c1COCC2 C1(CNC(C(=O)NC(C)C)=O)(CO)CCN(C(C2CC23CCCC3)=O)CC1 CC(CC(=O)N1CC(CNC(c2cccnc2-n2cncn2)=O)C1)C(F)F N1(C(c2c(C)cncc2F)=O)C2CCC1CC(NC(=O)CCc1cn[nH]c1)C2 c1(C(=O)NCC(C(C)(C)C)NC(C2CC(C)(F)C2)=O)c[nH]c2ccc(Cl)cc12 CC1(O)CCN(C(=O)CSc2cccs2)CC1O C1(NC(N(C)Cc2nc(O)n[nH]2)=O)CC(C)CC(C)C1 C1(C#N)(C(=O)NC2CC(CC(=O)NCc3ccn(C)n3)C2)CCCC1 C(N=c1[nH]c2cc(Cl)cc(Cl)c2o1)C1N(C(C2CC23CC(O)C3)=O)CCC1 C(=O)(CCCC(=O)N(C)C)NC1CC(F)(CNC(c2c(C)nncc2)=O)C1 n1(CC)nc(C(C)C)cc1C(=O)NCC(CC)(CC)NC(=O)CCc1ccco1 c1(C(=O)Nc2nc3ccccc3o2)cccc2c(I)n[nH]c12 CCC(C)(C)C(=O)C(=O)N1CC=CC(NC(c2csc3nnsc23)=O)C1 N1(c2nccc(SC)n2)CCN(C(C23CC2COC3(C)C)=O)CCC1C N1(C(C2N(C)C(=O)CC2)=O)CC2CCC(NC(C3CC4(CCCC4)C3)=O)(C2)C1 C1(C(N2CCC(C)(NC(=O)CNc3ccccc3Cl)C2)=O)CCc2nncn2C1 c1(C(N(C(C)CCNC(c2ccoc2Cl)=O)C)=O)cccc(C2CC2(F)F)c1 C(CC)(C(=O)NC(CN(C)C)C(=O)NC(COC(C)=O)CO)=CCCC C1(C)(C(N2CC3C(CC(=O)N(c4ccc(OC)cc4)C)C3C2)=O)CCCN(C)C1 C(=O)(C(C)C1=CCCC1)OC.c12c(sc(C)c1-c1ccccc1)NC(=O)COC2=O c1(C(=O)NCC2(C)CN(C(=O)C=CC3CC3)CCO2)nnc(O)c(Br)c1O C1(NC(CSC(C)C)=O)CCN(C(c2cccc(N(C)C)c2)=O)C(C)C1 C1(Cc2cn(CC(=O)OCC)nn2)COCCN1C(c1csc(C2CC2)n1)=O c1(C(=O)NC(CNC(c2c(C)oc(Cl)n2)=O)C)cnc2n1CCC(C)C2 c1(OC)ccccc1-c1ncccc1CN1CCOCC1CC(C)C CS(=O)(=O)c1cc(N2CCCC2CNC(=O)CCc2ccc(Cl)s2)ncn1 N1(C(c2nc(C(C)=O)sc2)=O)CCOC(CNC(c2cnn(C)c2C2CC2)=O)C1 O=C1NCC2(CCN(C(=O)C(=O)Nc3ccc4sccc4c3)CC2)C1O c1(CN(C)C(c2cc(CNC(c3coc(CO)c3)=O)[nH]n2)=O)nncn1C N1(C(C(CCC(C)C)O)=O)CC2(CCC2)CCC1CNC(=O)CC1CC1 CC(CCCCN=c1ncc(F)c[nH]1)NC(=O)CCOCC1CCCO1 C(=O)(CC(C)C(=O)O)Nc1cnc(N(C)C)n1C Cc1cc(F)sc1C(=O)N(C(C)CN(C)C(c1csc(-c2cnccn2)n1)=O)C C(=O)(CCCC(F)(F)F)N1C(CNC(c2nccc3cc[nH]c23)=O)CC(F)C1 O=C(CC(C(F)(F)F)NC(C1CC1Cl)=O)NCC(O)C1CCC1 c1(C(=O)NCCC2(O)CCCN(C(=O)CCCF)C2)ccc2c(c1O)CCCC2 c1(CC)nc(C)c(CC(=O)NCCCCCNC(C2(C)CCCC2O)=O)c(C)n1 C=C(C)CC(C(=O)NCCCN(CC)CC)NC(=O)Cc1cncc(C)c1 C1(OC)CC(NC(C2CC3C=CC2O3)=O)CN(C(C2CC(C#N)(OC)C2)=O)C1 C1(C(=O)NC2CCCN(C(c3cccc(Cl)c3F)=O)C2)CC2CCCCN2C1 C1(C(N(CC(C)NC(C2(OCC)CCC2)=O)CC)=O)CC(=O)N(CSC)C1 C1(C(N2C(CNC(c3c(C)cns3)=O)CC2)=O)CCC(O)CN1C C1(CC(=O)NCC2(COC)CC2)CN(C(c2cc(OC)n[nH]2)=O)C(C)(C)C1 c1(OC)ccc(C(=O)NC(C2CCCN2C(c2ncncc2Cl)=O)(C)C)cn1 CC(C)(C)C1=NOC(Cn2cc(CN3CC4CCC3C(O)C4)nn2)C1 c1(C(=O)NCC(CC(=O)N(CCNC(C)=O)C)C2CC2)ccnc(O)c1F C1(F)(CNC(c2c(C)ccnn2)=O)CCC(CNC(C2CCNC(=O)C2)=O)CC1 N(C(=NCCSC)NC1CCOc2ccc(F)cc21)CC(C)N(CC)CC C12(C(=O)NC(C34CC(CO3)C4)C)CCC1CN(C(c1ccc[nH]1)=O)C2 N1(C(=O)NC(C(=O)Nc2c(OC)cc(C)cc2)C)CCCc2cccc(Br)c21 CCC(CCC(=O)NC1CC2CC1CC2C(=O)NCC(C1CCCC1)OC)OC c1(OC)ccc(Br)cc1NC(=O)C(N1CCOC(CCN(C)C)C1)=O Cc1nc[nH]c1CC(=O)NC(C1CCN(C(c2cnsn2)=O)C1)C N1(C(CCC2CCN(C)CC2)=O)CCN(C(=O)COCC2CCOC2)C2CCC12 C=C(CNC(=O)C(CC(C)C)N(C)C(C1CCCC(=O)N1)=O)C1CCOCC1 c1(-c2cc(C(=O)Nc3cnc4ccccn34)ncc2)cccc(C2=CCOC2)c1 C1(NC(C(F)=C(C)C)=O)C2COCC1CN(C(c1cccc(C#CCO)c1)=O)C2 CC1(C)CC(CC(=O)NCC(C)(C)N(C)C)N(C(=O)CCn2cccn2)C1 c1(OC)cc(C(=O)NC(CNC(=O)CCC2(C)CCC(=O)N2)C2CC2)c(Cl)cn1 C1(C(N2CCC(C(=O)NC3CC(N(CC)CC)C3)CC2)=O)Cc2ccccc2C1 Cc1ccc(O)c(C(=O)NC(C)(CNC(=O)CC2SC(=N)NC2=O)C2CCC2)n1 CC(C)(CCCNC(c1cccs1)=O)C(=O)N1CC2(CNC(=O)C2)C1 N1(C(CCOc2cc(C)cc(C)c2)=O)CCCC12CCCN(C(=O)CCF)C2 c1(-c2nc(CC(C)(C3CCC3)OC)n(CC(F)(F)F)n2)ccc2ccccc2c1 CN1CC(O)CCC1C(=O)NC1(C2CN(C(=O)CN3CC4CCC3C4)C2)CC1 c1(C(N(CC)CC2CCCN2C(c2csnn2)=O)=O)ccc(C)nn1 C(=O)(C(O)(C(C)C)C(F)(F)F)N1C2CCN(C(CCC)=O)CC2CC1.C1COCC1 C(=O)(C1CCCc2ccnn21)N1C(C)CCC(NC(=O)C2=NNC(=O)CC2)C1 CC1(C(=O)NC23CCCC2C3)CCN(C(=O)CC2CCC(=O)N2)CC1 c1(C(=O)NCC(CNC(C2(COC)COC2)=O)C)nc2cc(F)ccc2s1 Cc1cc(C(=O)NC(C)CC(C)NC(=O)COCC(C)(C)C)cc(Cl)n1 C1(C#N)(C(=O)NCC2(O)CC(C(=O)NCCC(C)CCO)C2)CCCOC1 c1(C(N2CC3C(CNC(C(CO)NC(N)=O)=O)(C3)C2)=O)ccc(C(F)F)nc1O C(C(C(=O)NC(C)CCC(=C)C)C(C)C)NC(C(CC=C)NC(C)=O)=O C1(CC=C)(C(=O)NCCn2ncnn2)CN(C(=O)COCc2ccnn2C)C1 C1(C(=O)NCC2(NC(c3cc(N)c(O)cc3)=O)CCC2)CCCCC12CCC2 Cn1ncc(COC(C)(C)C)c1S(=O)(=O)NOCC1CCO1 c1(NC2C3(CC(NC(CN(C(COC)=O)C)=O)C3)C2)ccnc(S(C)(=O)=O)n1 C1(NC(C2CN(C)C2)=O)CC(NC(c2c(O)cccc2Cl)=O)C12CCC2 Cc1cc(C(N2CC3(CNC(C4CC(C)C4)=O)CCC2C3)=O)nc(O)c1 C(CC(=O)NCCOC1CCCC1)(C(C)OC1CC1)NC(C=C(COC)C)=O C(=O)(C1=CC(O)C(NC(C2(O)CCOC2)=O)C1)Nc1cc(C)cc(C)c1 c1(NC(c2[nH]c(=NCc3ccc(OC)cc3)sc2)=O)c(C)ccc2ncccc12 c1(N(C)CC)ccc2[nH]cc(NC)c2c1.C1(C)(CN2C(=O)NCC2)COC1 c1(CC)ccc(C(=O)NCc2occc2C(=O)NCC(F)Cl)nc1 Nc1cnc(Cl)cc1C(N1CCC1CNC(=O)CC(O)C1CC1)=O C1(C(=O)OC2CN(C(=O)CNC3CC3)C2)CN(Cc2cccnc2)CCC1(F)F C(C)(CO)(C(=O)N(CCCCCNC(=O)C(C)N1CCC1)C)OC c1(C(C)C(N2CCC(NC(C3CCC(=O)C3)=O)CC2)=O)ccc(S(N)(=O)=O)cc1 C1(C(C)OC)(OCC)CCOCC1.c12cccc(c1)C(=O)NCC2 c1(C(=O)NC2(C)CN(C(C3(C=C)CCCCC3)=O)C2)cc(C)c(Cl)c([N+](=O)[O-])c1 N1(C(C(CCC)OC)=O)CCN(C(c2cc(Br)cnc2CC)=O)C(CC)C1 c1(NC(C2CCCN(C(=O)C=Cc3cccs3)C2)C)cc(-n2ccnc2)ncn1 N1(C(=O)NCC(C)Oc2cccc(C)c2)CC2COC(C1)C2O CCC(CC(=O)NC(c1ccc(OC)cc1)CNC(C1CNC(=O)C1)=O)SC C(=O)(C(C)(C)CF)N(CC(CN(C(=O)CCc1c[nH]c(=N)[nH]1)C)O)C C(=O)(CC(C)(C)C(C)(F)F)N1CC(C)N(C(c2nonc2N)=O)CC1 N1(C(C=NOC)=O)CC2(C1)SCCC2NC(c1ncc(C)cc1OC)=O Cc1sc(Br)c(C(=O)NC(C)CCCNC(C2(O)CCOC2)=O)c1C N1(CCC)CCCCC1C.C1(COC)CC(c2nnnn2CCC2(C)CC2)(N)C1 N1(C(C(=O)C=Cc2cccs2)=O)CCC(NC(c2cc(C3CC3)on2)=O)C(F)C1 N1(C(=O)NCC2CCC(CCC)C2)CC(C(=O)OC)C2CCCC12 C1(C(=O)NC(C=C)CO)C=CCCN1C(c1cc(=O)cc[nH]1)=O c1(OC)c(C(c2nnnn2C)NC2C3CCCCCC23)cc(Cl)cc1Cl N1(C(c2c(C)ncs2)=O)CCCC1(C)CNC(c1ccc(SC(F)F)cc1)=O C(=O)(CCCCC(N)=O)NCCCC(C)NC(=O)C(C)NC(c1ccoc1)=O N1(C(C(CCCC)F)=O)CC2(C=C(C(=O)NCc3oc(CC)nc3C)CO2)C1 N1(C(C(C(C)C)=O)=O)CCOCC(C(=O)NC(C)C(N)=O)C1 N1(C(C(C)OCC=C)=O)CCC(C(C)(C)NC(=O)C(F)=CC2CC2)C1 C1(C)(NC(c2c(OC)cnnc2)=O)CCCCC1C(=O)NCC1CCCC(C)C1 Cc1c(C(=O)NCc2nc(CNC(C3(C)CC3C)=O)cs2)cccc1C#N C(=O)(C(C)C(O)C(C)CC)N1CC=C(C(=O)NC(CC=C)CC(F)F)C1 c1(C(C)=O)ccc(CC(N2CCC(O)(c3cn(C4(C)CC4)nn3)C2)=O)cc1 c1(C(N2CC(CC(C)(C)C)N(C(=O)CSC(F)F)CC2)=O)ccn2cnnc2c1 C1(CC#C)(C(=O)NC(CO)C(N)=O)CCN(C(=O)CSC(F)F)C1 c1(C(=O)OC)ccccc1C(=O)NCCCN(C(=O)Cc1cncs1)C Cc1nn(C)c(C(=O)Nc2csc(-c3cnn(CCC#N)c3)c2)c1F N1(C(C(C)C(F)F)=O)CC(NC(c2cc(C3CC3)nc(O)c2)=O)C(C2CC2)C1 N1(C(CC2CC(=C)C2)=O)CCCC(C2CN(C(c3cnc(C)cn3)=O)C2)C1 Cc1c(N2CCC(CCC(C)CO)CC2)ncnc1NC1CNC(=O)C1 n1(CC(=O)NCC2CCN(C(c3nn(C)nc3Br)=O)C2)cnc([N+](=O)[O-])n1 C=CC(CCC)CC(=O)NCC1(C)CN(C(c2c[nH]nc2CCC)=O)CCO1 CCCCCC=CC=CCC(=O)N1CC(NC(=O)C(C)Cc2cccnc2)C1 N(C(=NCC(C)C)NCC1(S(C)=O)CCC1)CC(CC)(CC)CO C(=O)(CC(C)(C)C#N)NCC(c1ccc(-c2cccc(C(C(=O)OC)C)c2)cc1)=O C1(NC(C=C(COC)C)=O)CCCCC1CNC(=O)CCC1(C)CC1(F)F c1(C(=O)OCC)ccc(C(=O)CN2CCN(C(=O)Cc3cc(C)no3)CC2)cc1 Cc1nnccc1C(N1C(C(=O)NCc2ccc(O)nc2)CC1C)=O C1(C(=O)NCC(CC(=O)N(C2CCCC2C#N)C)OC)CN2CCN1CC2 C1(NC(c2nnc(O)cc2O)=O)CCN(C(=O)C(F)=CC2CC2)C12CCC2 c1(C(=O)NCCC(CNC(CS(CC)=O)=O)O)nc(-c2ccccc2)ncc1Cl c1(C(N(C(=O)NCC2C(CC)OCC2)C)C)c(C)nn(C)c1C c1(C(=O)NC2C(NC(c3cnc(C)o3)=O)C2)ccc(OCCO)cc1 c1(OC)ccc(C2CC2)cc1-c1csc(C)c1 Cc1cc(C(N2CCCCC2c2cn(-c3cccc(C)n3)nn2)=O)cc(Cl)c1 c1(C(=O)NC2(CNC(Cc3n[nH]c(=N)s3)=O)CC2)ccn2ccnc2n1 Cn1nnc2cc(C(N3CCN(C(c4ccn(CC(F)F)n4)=O)C4CC34)=O)sc12 c1(NC2CN(C(C#C)=O)CC2O)ncc(C)c(C)n1 c1(C(CNC(C23CCCC2C3)=O)NC(c2csnn2)=O)ccc(F)cc1F C(=O)(CC(C)CC(C)C)NCC(C)(C)CNC(C1C(C=C)C1)=O c1(CCONC(Cc2cc(COC)on2)=O)ccc(OC)cc1.c1(S)ccccc1 C1(NC(C(CC)C2CCC(=O)N2)=O)CCCC1(C)NC(c1ccncc1)=O C1(CCC)(NC(c2ccnc(C3CC3)n2)=O)CCN(C(c2nn[nH]c2Cl)=O)CC1 CC(CO)(C(=O)NCC1CCCCO1)NC(C1CC(F)C(=O)N1)=O c1(C(CNC(CC(CC)C)=O)NC(c2[nH]cnc2C)=O)ccc(F)cc1F C1(C(N2CC(C(C(=O)N(CC(C)C)CC)O)C2)=O)CCC(O)C1 c1(C(C)C)cc(CC(=O)N(C(C)CCNC(c2ocnc2C2CCC2)=O)C)on1 c1(C(CNC(=O)CSCCC(C)C)NC(CCCC)=O)ccc(F)cc1 CCCCCC(C)(C)C(=O)NCC(O)CNC(=O)C(C)(O)CC(C)(C)C N1(C(c2nc(C(C)C)oc2)=O)CCCC2(CNC(=O)CCc3cnccn3)CC12 c1(CC(N2CCC(CN(C)C(c3cc(F)cs3)=O)C2)=O)cnc2cccnn12 N1(C(C2(CC)CC2)=O)CC2CC(C(N3CCN(C)C(C)(C)C3)=O)C(C2)C1 C#CCCC(=O)N(C(CNC(C1CCC1CF)=O)Cc1ccccc1)C C1(C(N2CC(F)(CNC(C3(COC)C=CCC3)=O)C2)=O)Cc2nccn2C1 C#CCCC(O)C(=O)N1CCN(CC(C)NC(=O)CCc2cn[nH]c2)CC1 C(=O)(C1=C(C)CCOC1)N1CC(CNC(C2(C#C)CC2)=O)C(F)(CO)C1 N1(C(C2CC2C(=O)NCC(=O)NC2CC=CC2)C)C2CCC1CC(CO)C2 Cc1ccc(C(=O)NC2(C)CCN(C(=O)CC3CC4C=CC3C4)C2)c(O)c1 C12(C(=O)NC(C3CCCN3C(C3CCCCS3)=O)C)CCC(CC1)C2(C)C c1(-c2cn(-c3c(Br)cccc3Br)nn2)ccc(C2=CCC(C#N)CC2)cc1.CO C=CCC(CNC(=O)CCc1ccn(C)n1)NC(c1ccn(C2CC2)n1)=O N1(C(C=C(C)c2ccco2)=O)CCC2CCN(C(=O)CC(=O)N(C)C)C2C1 C1(CNC(CC(CC)SC)=O)CN(C(=O)CCc2ccon2)CCC1(C)C c1(C(=O)NC2C(C)CN(C(c3csc(S)n3)=O)CC2)c[nH]c2cccnc12 c1(C(c2nnnn2C)NC2C(C(C)C)CCC2)cccc2c1COCC2 CC1CCOC1CC(=O)NC(C)(C)CN(C)C(c1cnn(CC(F)F)n1)=O C1(NC(C(C)(C)C2CCCN2C(C2CCC(C3CC3)C2)=O)=O)CCCN(O)C1=O Cc1ccccc1C=CC(N1CCC1CNC(c1cnc2n1CCS2)=O)=O C=CCN=C(NCCc1ccccc1)NCCN1CCCC1 c1(C(N2CCCC(CCNC(c3cc(C)sc3)=O)C2)=O)cc2c(cn1)CCCC2 c1(NC(C2C(NCc3cnc(N(C)C)nc3)C2)=O)nccc(Br)c1Cl c1(OC)cc(C(N2CCC(O)(CCNC(C3CC(C)(C)C3)=O)CC2)=O)ccc1C C(=O)(CC(C)(C)C(F)F)C(=O)CCC(=O)C1CCCN1.CC1CNCCS1 Cc1[nH]c(=N)sc1CCSC1N(C(c2ccc(C3CC3)cc2)=O)CC1 Cc1c(F)cc(C(=O)NC(C)CCNC(C2CC=CCC2)=O)c(F)c1N C(=O)(C(CC)C(F)(F)F)NCCC(=C)CNC(=O)CCCN(C)C(=O)OC c1(CC(=O)NCC2C(CNC(c3n(C)ncc3Cl)=O)C2)cccc(C#N)c1 c1(C(=O)NC2C=CC(C(N)=O)C2)n[nH]c2c1CN(C(=O)Cc1ncccc1F)C2 Cn1cc(Cl)cc1C(=O)NC1CN(C(C2CCN(c3ccncc3)CC2)=O)C1 N1(C(c2c(OC)csc2)=O)CC2(CCCC2)C1C(N1CCC(C(C)(C)O)C1)=O C(=O)(CCCCC(=O)N1CCCC1C(C)NC(c1ccncc1F)=O)OC C1(C(C)(C)CNC(c2ccc(CO)o2)=O)CCCCN1C(=O)C=C1CCC1 c1(CCC(=O)NC(CNC(c2c(SC)ccs2)=O)(C)C2CC2)ccnc(Cl)c1 c1(CC)ccc(C(=O)N(C)CCN(C(=O)C(F)(F)c2cnn(C)c2)C)c(O)c1 c1(OC)ccc2c(=NCCC(N)=O)[nH]c(=NCc3cc4cnccc4o3)[nH]c2c1 C12(CNC(C(C)(C)C3CC3)=O)CN(C(c3csnc3Cl)=O)CC1CCO2 c1(C(=O)NC(C2CCN(C(C(CC)=CC)=O)C2)C)sc(OC)nc1C C1(C(=O)NC(C2CCN(c3ccncn3)CC2)C)CCN(C(=O)c2cnsn2)O1 C1(C(N(C(CCNC(C(C)C)=O)C)C)=O)CC2CC(F)(F)CC(C1)C2(F)F N1(C(C(C)NC(=O)Cn2cnnn2)=O)CCC(C)(C)C(NC(c2cc[nH]n2)=O)C1 CC1CN(C(=O)CN(C2CCC2)C(C2CC(=O)CC(=O)N2)=O)CC(=O)N1C CCCCC(CC)C(=O)NC1CCC(CCNC(c2c(C)ccn2C)=O)C1 CC(C)(C)C(O)CCC(=O)NCC1CCCCN(C(c2ccc(C(N)=O)[nH]2)=O)C1 N1(C(c2c(C(C)C)c[nH]c2)=O)C2CCC1CC(C(=O)NCC(C)C#N)C2 C1(C#N)(C(N2CC(CC(C)NC(c3ccn(C)c3)=O)C2)=O)CCCC1 c1(CCC)cc(C(=O)NC(C)(C)CNC(=O)C(c2ccccc2Br)O)ccn1 c1(NC(C2N(C(CCN(C)CC)=O)CCSC2)=O)cc(OC)c(OC)cc1C C=CCCC(C)(C)C(=O)N1CCN(C(=O)C(=O)C2CCOC2)C(CC)C1 C1(O)(CN(C(COCC(=O)NC)=O)C)CCN(C(=O)C=CC(=O)N(C)C)CC1 N1(C(=O)NC2CC2C(C)(C)C)CC2CC1(c1cn(-c3cccc(Cl)n3)nn1)CO2 c1(C(=O)NCC2(F)CC(NC(c3cc(C)ns3)=O)C2)cn(C)nc1C(F)F c1(C(=O)NCCN(C(=O)CC2(O)CC2)CC)cc(S(N)(=O)=O)ccc1F N1(C(=O)C2CC2)CC(C2CCN(C(C3CCCC(C4CC4)O3)=O)CC2)C1 CC(C)(C)CCCCC(=O)N1CCC1C(=O)NC1CC(n2ccnc2)C1 N1(C(C(c2ccc(F)cc2)(C)F)=O)CCOC(CCNC(c2cnc[nH]2)=O)C1 N1(C(CNC(C2C(C)C2)=O)=O)CCC2(C1)CN(C(c1c[nH]ccc1=N)=O)C2 C(c1ccc(Br)s1)=C(C(=O)NC(CCNC(CC(=C)Br)=O)C)C C1(NC(C2OC(C)(C)OC2(C)C)=O)CN(C(=O)Cc2csnn2)C2(CCCC2)C1 C1(CC(=O)N(CC(C)(C)CNC(C2CCCC2)=O)CC)CCCS(=O)(=O)C1 c1(CNC(C2C(NC(c3c(COC)cc[nH]3)=O)CCCC2)=O)cc(C)cc(F)c1 CN1C(=O)Cc2ccc(C(=O)NCC(CNC(C3CC34CCC4)=O)CO)cc21 N1(C(C(CCCOC)C)=O)CC(NC(c2cc3sc(C)nc3[nH]2)=O)C2(CCC2)C1 C1(C(N(CC(C)C)CC(=O)NCC2=NOC(C)C2)=O)CCC(C)(O)CC1 CC1CN(C(=O)CCCC(N)=O)C(C)CN1C(c1cc(-c2ccccn2)no1)=O Cc1ncc(C=CC(=O)NC2CC(N(C)C(C3CCCCS3(=O)=O)=O)C2)c(O)n1 C(=O)(CC1=CCCCC1)N(C)C.C1C(N(C(=O)C(CN(C)C)N(C)C)C)C(=O)N1C N1(CCN(C(C)=O)C(c2cccc(Cl)c2)=O)CCCCC1OC(CC)=O CCCCC(F)C(=O)NCC(C)(CO)NC(c1cncc(C2CC2)c1)=O N1(C(C2N(C(C#CC3(C)COC3)=O)C3CCC2C3)=O)CCC2(CNC(=O)C2)C1 S(=O)(=O)(c1ccn(C)n1)N1C2CN(Cc3cccc(C=C)c3)CC1C2 c1(C(=O)OC)ccc(C=CC(N2CCC(F)C(NC(C)=O)C2)=O)cc1F C1(OCC)COc2ccccc2O1.n12nc(C)c(c1C)CC(C)C(=O)OC2 c1(SCC(=O)NC2C3(NC(C4C(C)(C)C4)=O)CCC(C2)C3)nnc2ccccn12 c1(NCC(CC)CCO)ccc(S(=O)(=O)N(C)CCc2ccc(Cl)cc2)cc1F c1(C(=O)NCCCC(CCC)NC(C2CCS(=O)(=O)C2)=O)c(F)ccc(F)c1F CCCCCC(C)(CC)C(=O)N1CCC(O)(CNC(=O)CCNC(C)=O)C1 c1(C(N(C(C)CN(C)C(C2CC(CF)C2)=O)C)=O)ccn(C2CCCC2)n1 N1(C(CCC=C)=O)CCCC2(CCC(NC(c3cncc(C(C)(C)C)c3)=O)C2)C1 C1(CC(=O)NCC2CCN2C(=O)C(O)C2CCC2)CCn2cncc2C1 N1(c2ccnc(C(C)C)n2)CC(NC(c2cc(=O)cc(Cl)[nH]2)=O)C2CCCCC12 C1(NC(C(C(C)C)N(C)C)=O)CC2(CCCN(C(C3(C)CCCOC3)=O)C2)C1 c1(C(=O)NCCC(CNC(C=CCOC)=O)O)c(F)cc(F)cc1F C(=O)(CCCCCS(N)(=O)=O)N1CC(N(C(C(C)S(N)(=O)=O)=O)C)C1 Cc1cnc(CC(=O)N(C2CCN(C(=O)CCNS(C)(=O)=O)C2)C)[nH]1 N1(C(CCC)=O)CC(C)(NC(C2CC2CN(C)C)=O)C1 C(=O)(C(F)CC)N(CCCNC(=O)CC1(OCC)CCC1)CCC c1(C(=O)NC(CCCNC(CC=CC)=O)C)cc2ccsc2n1C C1(CCC)CCCN1C(=O)CCN(CCCO)C(=O)Cc1ccc[nH]1 c1(N2CCN(C)CC2CNC(c2ccc[n+]([O-])c2)=O)ncnc2c1CCO2 N1(C(C#CC2(C)CC2)=O)C2CCC1CC(NC(c1cc(C(F)(F)F)no1)=O)C2 c1(C(=O)NCC(C(C)(C)C)NC(c2c(C)con2)=O)cc(Cl)c2n[nH]cc2c1 c1(NCCNC(C2C(CCC#C)N(C(=O)OC(C)(C)C)C2)=O)ccc(F)c(F)c1 C(CN(C(=O)CCC(C)OCC)C)(CO)(CO)NC(COCC=C)=O N1(C(CN(C(C)=O)C)=O)CCC2(CCOCC2)C(NC(=O)C(C)C(F)(F)F)C1 c1(C(N2C(C)CC(NC(C3CC(C#C)(O)C3)=O)C2)=O)cnc(OC)c(Cl)c1 C1(NC(CC(C)c2ccncc2)=O)CN(C(c2csc3nccn23)=O)CC12CC2 N1(C(CC2(NC(C)=O)CC2)=O)CCOC2CN(C(C34CC5CC(CC3C5)C4)=O)CC12 CC1CN(C(c2ccc(CNC(c3cccs3)=O)s2)=O)CC(C)(C)C1 C1(N(C(C2C(C(C)NC(=O)CCCN3CCCC3)C2)=O)C)CCCC1C#N CCC(CC)(CC)C(=O)N1CC(C(N2CCC(C)(COC)C2)=O)CCC1(C)C C1(CC)(NC(=O)C(O)CC(C)C)CCCN(C(=O)C=Cc2ccc(C(F)F)o2)C1 N1(C(c2c(SC)cccc2)=O)CC(NC(c2nn(C)cc2SC)=O)CCC1C C(=O)(CCCCN1CCOCC1)NCC(CCOC)NC(=O)C1=CCOC1 C1(NC(c2scc(C)c2)=O)CN(C(C2CC2Cc2ccccc2)=O)CC2(CC2)C1 Cc1cn2cc(C(=O)N(C(C)CNC(c3cc[nH]c3)=O)C)sc2n1 CN1CC(=O)N(CC(N2CCN(C(c3cnc(Cl)[nH]3)=O)C(C(F)F)C2)=O)C1=O C=C1CC2CCCC(C1)N2C(C1C2CC1N(C(=O)CNC(C1CC1C)=O)C2)=O CC1COCC(C(=O)NC2CCC2CNC(c2cn(C)nn2)=O)O1 Cc1ccc(C(C)C)cc1C(=O)NCCCNC(C1CC(C)CCO1)=O c1(NS(=O)(=O)CCCCl)cccc2c1CN(Cc1ccncc1Br)C2 C(CCC(O)C(=O)NCC1(C)CCCCO1)NC(c1c(CC)n(C)cc1)=O C1(C(=O)NCC2CC(NC(CCc3nc(C)sc3)=O)C2)CCC(=O)C(C)C1(C)C c1(NCCC(C)NC(=O)C(C)C2CCC2)nc(Cl)nc2[nH]c(O)nc12 N1(C(=O)CNC2C(CNC(=O)COC3CC=CC3)C2)CCOCC1 N1(C(CC(=O)NCC#C)=O)CCCC(C)C1CNC(=O)COCc1cc(C)on1 C1(NC(CCN2CCC(CN(C)Cc3ccccc3)CC2)=O)CCCCC1(C)C N1(C(CCOCCOC)=O)CCN(C)CC1CNC(c1n[nH]cc1C)=O c1(C(N(C2CN(C(C(CC=C)CC(C)C)=O)C2)C)=O)ccc2c(=N)[nH]cnc2c1 CN1CCN(C(C2CCC3(CCC3)O2)=O)C(C(=O)NCc2ccnc(Cl)c2)C1 N1(CC(=O)NC(C2N(C(Cc3c(C)scc3)=O)CCC2)C)CCS(=O)CC1 O=C(C(F)C(F)(F)F)Nc1ccc(-c2cn(CCC3CCCC3(F)F)nn2)cc1 C(C(C(=O)N1CCC(CNC(c2cn(C(C)C)nn2)=O)CC1C)C(F)(F)F)OC c1(C(N(CCCNC(C(C)=C(C)C)=O)C)=O)ccc(C(F)F)nc1O c1(C(N2C3(C(N(C(C#C)C)C)=O)CC3CC2)=O)cncc2[nH]ccc12 c1(C(=O)NC(CNC(C2C(C(=O)OC)C2)=O)C(C)(C)C)nccc(N)c1Cl N1(C(C(CC)n2ccc(C3CC3)n2)=O)CCc2[nH]nc(I)c2C1 C1(=O)C(CC(C)C)NC(=O)C(CSC)(C)N1.N1(C(C)=O)CCC(N(C)C)CC1 c1(C(N(CCCCO)C)=O)cn(CCNC(c2coc(C(F)F)c2)=O)cn1 N1(C(C(C(C)C)C)=O)CCn2c(CNC(=O)CC3NC(=O)NC3=O)nnc2C1 CC(O)CCCc1cn(CC(F)(F)CNC(c2ccco2)=O)nn1 CC1CCN(C(=O)CC2(c3ccccc3)CCC2)CCN1C(=O)COCCF Cc1cc(O)ncc1C(=O)N(C(C)C(=O)NCC1(C)CCCC1O)C C(C(CC(F)(F)F)NC(C1CCS(=O)(=O)N1)=O)NC(c1c(C)n[nH]c1C)=O c1(C(=O)NCC2(C)CCCN(C(COC(C)=O)=O)C2)cn2ccncc2n1 C1(C(=O)Nc2n(C)nc(Br)c2)CC(F)(F)CN1C(=O)CCc1ccc(F)c(Br)c1 c1(NCc2cc(OC)no2)nc2ccc(F)cc2n1Cc1cc[nH]n1 C1(c2ccc(C)o2)CSCCN1N1CC(C(N2CCOCC2)C2CC2)C1 c1(CC(N2CC(Cn3cc(-c4cncnc4)nn3)C2)=O)cncc(Br)c1 C1(C(=O)NCc2cn(CC(=O)NCCN3CC=CC3)nn2)CC2(C1)CC(O)C2 CCC1=C(C(=O)NCc2cccc(C(=O)NCC(C)C)c2)SCCO1 c1(OC)ccc(CNC(=O)C(c2ccc(N(C)C)nc2)N2CCOCC2C)cc1 C1(O)(CNC(c2nc(C)[nH]n2)=O)CCN(C(c2nocc2Cl)=O)CC1 N1(CC)CCCN(C(=O)C(C2CCC2)NC(C2CC2C(C)(C)C)=O)CC1 CCC(CCC(=O)N1CC(CO)CC1CO)NC(=O)CC1(C)OCCO1 C(c1ccc(Cl)nc1)=CC(=O)N(CC(O)CN(C)C(c1cc(Cl)ccn1)=O)C N1(C(C2OCCN(C(C=CCOCCOC)=O)C2)=O)CC2(C1)CC(C)(O)C2 c1(C(=O)NC(CNC(CNC(=O)NC)=O)(C)CC(C)C)ccc2c(c1)CCC=C2 C(=O)(CS(=O)(=O)C1CC1)NC12CC(NC(c3c(C)nc(C(C)C)cc3)=O)(C1)C2 CCC(C)C(C(=O)N(CC(c1nn[nH]n1)C)C)NC(=O)C(CN(C)C)CC C(=O)(C1=C(C)S(=O)(=O)CC1)N1C(CC)CN(C(c2cnn(CCO)c2)=O)CC1 N1(C(C(C)CC2CCC2)=O)CCOCC(NC(=O)Cn2cccnc2=O)C1 c1(C(=O)NCC2CCN(C(c3c(C)cc(C(F)(F)F)s3)=O)C2)cccn(C)c1=O C1(NC(N2CCCC(C(=O)Nc3ccon3)C2)=O)CC2CCC(C1)N2C1CC1 c1(CN(CC(=O)NCC)CC(=O)NC)ccncc1 C12CCCC1NC(=O)NC2.C1(CN(C)CCCCl)CCCN1 c1(CC)cc(CC(=O)N(C)CCN(C(=O)C(C)NC(C2CCC2)=O)C)no1 N(C1CCCn2nccc21)C(C(CC(C)C)ONC(c1nc[nH]n1)=O)=O C#CCC(O)C(=O)N(C)CC1(O)CN(C(c2ccc(C(=O)N(C)C)cc2)=O)C1 n1(CC(N2CCC(O)(C(C)NC(=O)C(N)=O)C2)=O)c(=O)c(=O)[nH]c2ccccc12 N1(C(C(CC)CO)=O)CCN(C(c2nnn(CC3CCCC3)c2C)=O)CC1C C1(C(F)(F)F)(C(N2CC(NC(C3(SC)CCC3)=O)C(C)C2)=O)CC2C=CC1CC2 C1(C)(C(N(C(C(C)C)CO)C)=O)CCN(C(=O)Cc2ccc(O)nc2)C1 C=CC1(CC(N2CCSCC2CO)=O)CN(C(c2ccc(OC)o2)=O)C1 c1(C(=O)NC(C2N(C(CCCOCC)=O)CCC2)C)c(C)cnc(OC)c1Cl CCC(CC(=O)NC1(CC(=O)OC)CC1)N(C)C(c1sc(C)cc1C)=O c1(CN2C(C)CC(NC(=O)Cn3ncnn3)CC2)cn2c(n1)CCCC2 Cc1ccc2c(c1)CC(C(=O)NC(C)CNC(=O)CCc1cccc(F)c1)S2 C=C(C)CCC(=O)N1CCC(NC(c2ccnc(OCCO)c2)=O)C1 C(=O)(C1=CCSC1)NC(C1CCCCC1)C(=O)NCCCC1CC(C)C1 CCCCCCC(C)(C)C(=O)N(C)CC1CC(F)CN1C(C1CC1(C)C)=O C1(C(=O)NCC#C)N(C(c2ccc(O)cc2)=O)CCCC1(C)C CCCCCC(=O)NC1CC(NC(=O)C(C)NC(=O)NC2CCCC2)C1 C=C1CCC(C(=O)NC2CCN(C(c3ncoc3CCC(F)(F)F)=O)C2)CC1 c1(N(c2nc(CN3CCCC(C(O)C(F)F)C3)cs2)CC)ccc(F)cc1 CC1(C)CCCC(NC(C2(O)CCN(C(=O)COCc3nccs3)C2)=O)C1 n1(CC(=O)NC2CCC(NC(C3(SC)CCC3)=O)CC2)cnc([N+](=O)[O-])n1 C(=O)(C1=CNC2=NCCC2=C1)NC(CCCNC(C1CN(C(C)C)C(=O)C1)=O)C C1(CNC(c2c(OC)nn(C)c2)=O)CN(C(=O)C=C2CCN(C)CC2)CCCO1 c1(OC)cc(OC)c(C(C)(C)C)cc1CN1CCCC1(C)c1ccccc1 C(=O)(C1=CCC(NC(c2cccs2)=O)C1)C1CC1.C1(C)CCNC(=O)CSN1CC C=CC(C)(O)CC(=O)N1CCCCCC1C(=O)NCc1nccc(OC)n1 N#Cc1ccc(N)c(C(=O)NC2CCC(CCNC(c3ccc(F)cn3)=O)C2)c1 C(C)(C(=O)NOCC(=O)N(C)C)NC(C(CC)C)c1ccccc1 Cc1oc(CO)cc1C(N1CCC(N(C(=O)CC2(O)CCOC2)CC2CC2)C1)=O c1(C(N2CC(C)C(NC(C3CC(=O)N(C)C3)=O)C2)=O)ccc2c(c1)CCC=C2 N1(C(=O)Cc2csc(Cl)n2)CC2OCCN(C(c3ccc4c(c3)NCC4)=O)C2C1 C(=O)(CCC(=O)N1CCCC1(C)CNC(=O)Cc1nc(C)c(C)s1)N(CC)CC C1(CN(C(=O)C(F)=CCCF)C)COCCN1Cc1ccc(Cl)cc1 O(NC(=O)CC1C(NC(C2CS(=O)(=O)C2)=O)CC1O)C1CC(OC)C1 C1(C(=O)NCC(C(C)(C)C)NC(C=C(C)c2ccco2)=O)CCS(=O)(=O)C(C)C1 C1(CC=C)CCCC1N=c1[nH]c(=NC)[nH]c(=NCCCn2ccnc2)[nH]1 CC(C1OCCc2ccccc21)N(C)Cc1c(C(F)(F)F)nc2c(Br)cccn12 N1(C(c2ccnn2C2CC2)=O)CC2CCN(C(c3cccnn3)=O)CC2C1 c1(CC)noc(C(N2CCCCC2CN(C(=O)C(C)N(C)C(=O)OC)C)=O)c1C N1(C(CS(CC)(=O)=O)=O)CC=C(CCNC(c2csc(C3CCCO3)n2)=O)CC1 Cc1ccc(-n2nc(C)c(CC(=O)NC3CC3(c3ccccc3Br)C)c2C)cc1Cl C(C(C)(C)CC(=O)NCCC1(O)CN(C(=O)CNC(=O)CCNC(C)=O)C1)OC c1(CNc2cn(C3CN(C(c4nc(N(C)C)sc4)=O)C3)nc2)ccc(C#N)cc1 N1(C(CC#N)=O)CC2(CCC2)CC1C(=O)Nc1ccc(NS(C)(=O)=O)cc1 C1(CNC(=O)Nc2c(C)n[nH]c2)(CO)CC2CCC1CC2 N1(C(CC(C=C)CC)=O)CC(C)CN(C(=O)C(c2ccc(C)o2)C)C(C)C1 N1(C(C(C)=C(C)C)=O)CCCC(C2CC2NC(c2ccccc2CN(C)C)=O)C1 c1(C(C(=O)NC2C(C)N(C(C3CC4C=CC3O4)=O)CC2)(F)F)cccc(F)c1Cl c1(OC)cc(CC(=O)NCC(O)CCNC(=O)Cc2cnccc2OC)ccn1 C(=O)(C1CCCn2cnnc21)NC1C2CC(CNC(=O)CCC3CC3)(C2)OC1 Cn1cc(C(=O)NC2CCCC2NC(c2cnsn2)=O)nn1 C1(NC(C(COC)O)=O)CCN(C(c2ccc(-c3nnc(C)o3)cc2)=O)C(C)C1 CC(C)C(C(F)(F)F)NC(c1ccccc1Nc1cccc(C(F)(F)F)c1)=O c1(C(=O)NCC2N(C(Cc3ccn(C)n3)=O)CC(F)C2)cc(Cl)c(F)cc1N n1(C(COC)COC)nc(-c2ccc(N3CCCCC3)nc2)nc1C1CCCO1 C(C(C)(O)C(=O)N1CCCCC1C(=O)N(C)Cc1ncc[nH]1)OC CC1(C)CC(CCNC(C23CC(NC(c4ccc(=N)[nH]c4)=O)(C2)C3)=O)CO1 C1(NC(=O)CN2C(=O)CCC2=O)CCCCCC1NC(=O)C(O)Cc1cnc[nH]1 c1(C(N2C(COC)CN(C(C3CCSC3)=O)CC2)=O)cc(F)cc2cccnc12 CCC(C)C(C(=O)NCC1(C(=O)Nc2cc(C)sc2C)CC2(CC2)C1)N(C)C C1(OC(CC)=O)CCN(C(c2[nH]ccc2CNC(c2ccc(F)s2)=O)=O)C1 Cn1ncc2c1CC(C(=O)N=c1ccc(C(F)(F)F)n[nH]1)CN2 C(CC(C(C)(C)C)NC(c1ccnn1C(F)F)=O)N(C(CSCC=C)=O)C c1(CC)cc(CC(=O)NC(C)CNC(=O)CC(c2c(C)noc2C)C)n(C)n1 c1(CC(=O)NC2(CCNC(=O)C=CC3CCCCC3)CC2)ccc2nc[nH]c2c1 c1(C(N2CCCCC(N(C(C3CCN(C)C3)=O)C)C2)=O)cccc2nc(Cl)cn12 CCCC(CC(C)C)C(=O)N1CCCC(CC(=O)N(C2(COC)CC2)C)CC1 C(CCC(=O)NCC1C=CCN1C(c1c[nH]c(=N)o1)=O)N(C)C c1(C(C)C)cc(OC)ncn1.c12noc(n1)CCC(=O)OCCO2.N1(CC)CCCCC1 CC1C(NC(=O)CNS(C)(=O)=O)CCCN1C(c1ccc(C(F)(F)F)c(F)c1)=O N1(C(CCC(=O)N(C)C)=O)CCCCC(C2CN(C(=O)CC3CCCCO3)C2)C1 CC1CCN(C(C2CCCCN(C)C2=O)=O)CCN1c1ncnc(=N)[nH]1 C1(c2ccc(F)cc2)(C(=O)NCCN(C(=O)Cc2ccoc2)CC)CCOCC1 N1(C(c2ccc(C)c(C)n2)=O)CCOC2CCN(C(C3CCN(C)C3=O)=O)CC12 C(=O)(C(CO)C(F)(F)F)N1CCC(n2cc(-c3cccc(N)c3)nn2)C1 C1(C(=O)NC(C(=O)OCC)COC(C)C)CC(N)CC(C)(C)O1 N1(C(C(=O)N(c2ccccc2Cl)CCOC)=O)CCNCC1CSc1ccsc1 Oc1nc2ccc(CNC(c3[nH]nnc3-c3ccccc3)=O)cc2[nH]1 C1(CC(=O)NCCc2n(C)ncn2)CC(NC(c2cccc[n+]2[O-])=O)C1(C)C O=C(CCC(F)F)NCCN(C(c1cnc(N2CCOCC2)s1)=O)C1CC1 N1(CCC)CCC(NC(c2ncoc2CNC(=O)CCc2ccnn2C)=O)C1 C#Cc1cnn(C)c1C(=O)NC1CCC(C)N(C(c2cccnc2O)=O)C1 CCCCC(O)C(=O)N1CCC(N(C(=O)C(C2CC2)C2CC2)C)CC1 Cc1cc(C(=O)NCCC2(C)CCN(C(C3(C)CC3C)=O)C2)c(C)n1C CCCCCCCCCCCC(O)C(=O)N(CCC(=O)O)CCC c1(CN(C(c2c(O)ccc(C(N)=O)c2)=O)C2CC2)ccc(F)c(F)c1F c1(C(=O)NCC(C)(CO)NC(Cn2nc(C)oc2=O)=O)cc2c(Cl)cncc2s1 CC1CC(CNC(c2ccc(Cl)nc2N)=O)CCN1C(=O)C=Cc1ccco1 CC1CC2CCC(C(=O)NC3C4CC3N(C(=O)CSC3CCCCO3)C4)CN2C1 C1(NC(c2c(C)cc(CNC(=O)CN3CCNC(=O)C3)o2)=O)CCOC(C)(C)C1 C1(CNC(C2CC(C)C2)=O)(NC(c2ccc(N3CCCC3)nc2)=O)CCCCC1 CC1(C)CCN(C(c2ccc(CO)cn2)=O)CC1CNC(C1CCC12CCC2)=O C12(C(=O)NCC3C(NC(CC4(C(F)(F)F)C(C)C4)=O)CCC3)CC(C)(CCO1)C2 N1(C(CC(CCC)O)=O)CCC2(CCN(C(=O)CC(C)(F)F)C2)C1 C1(C(=O)NCC2(O)CN(C(C3N(CC)CCC3)=O)C2)(N(C)C)CCCOC1 c1(OC)ccc(Br)c(CNCC2(C)CCCN2C(=O)NC(=O)OC(C)(C)C)c1 c1(CC(=O)NCC(CCOC)NC(=O)C(C(C)(C)C)OC)c(C)ncnc1C c1(CC)noc(C)c1CN(C)CC1CN(C(c2cnoc2C(C)C)=O)CCO1 C1(COC(C)C)CN(C(=O)CN2CCOCC2=O)CCO1 C=CCCN=C(NCC(CCCC)N(C)C)N1CCCC2(CCS(=O)(=O)C2)C1 c1(CNC(C(CCCCC)O)=O)nn(C)c2c1CN(C(C1CN(C(C)=O)C1)=O)CC2 c1(Cc2n(-c3cc(O)ncc3)nc(CCO)n2)n[nH]c2c1CCCC2 N1(C(c2n(COC)ncc2)=O)CCCN(C(=O)COCC2CCCC2)CC1C O=C(C1CCCn2cnnc21)NC1(CNC(C23CCCCC2C3)=O)CC1 N1(C(C(CNC(C(CC=C)C(C)C)=O)CC=C)=O)CCCC2(C)CCCC12 C1(OC)CCC(C(F)(F)F)N(C)C1.c12ccc(cc1)C(=O)c1cn-2nn1 N1(C(c2cc(C(=O)OCC)c(C)[nH]2)=O)CCN(C(c2ncc(Cl)s2)=O)CC(O)C1 c1(OC)nc(Cl)c(C(=O)NCC2CCC2NC(=O)C(c2cccc(OC)c2)C)s1 c1(C(N(CCCCN(C(C(COC)O)=O)C)C)=O)ccc2c(c1)CCC(C)N2 C1(NC(=O)CC(F)(F)Cl)CN(C(=O)CCOC2CCC2)CC12CC2 c1(C(=O)NC2CCN(C(C(COC)C)=O)C2(C)C)cnn2ccnc(C)c12 c1(CN2CCC(O)(C(=O)NC(c3cccnc3)CC)C2)cc(Cl)cnc1Br N1(C(c2nccnc2C)C(=O)NCCCOC)CC(=O)N(C)CC1C(=O)OC C1(CNC(C23CC(C)C2C3)=O)CCCC(NC(=O)Cc2ccon2)C1 CN1CC(C)(NC(C2(C(=O)NC(=O)CN3CCCCC3)CCCC2)=O)CCC1=O c1(C(N2CC(CCNC(C(CC)(C)C#N)=O)C2)=O)cccc2c(Cl)c(Cl)sc12 C=CCCCCCCCCC(=O)NCC1CCCN1C(C1(C)CC1(F)F)=O CCC(O)(CC)CCNC(=O)C(C)(C)C1CCN(C(c2csc(C)c2C)=O)C1 C1(NC(c2sc(CC)c(C)c2)=O)CC2(CCN(C(C3CCC(=O)N3C)=O)C2)C1 Cc1cc(Br)ccc1CCNCCC(N1CCN(C(=O)OC(C)C)CC1)=O c1(N(CC(O)CO)C(c2c(OC)nc(C)nc2)=O)cccc2ncccc12 Cc1ccc(-n2nc(C3CCC3)nc2CC2CCCC(O)C2)cc1 Cc1cc(=NC(C)COc2ccccc2)[nH]c(N2CCSC(C)(C)CC2)n1 C(=O)(C(CS(C)(=O)=O)NC(C1CCCCNC1=O)=O)OC c1(NC(C)=O)ccc(C(=O)C(N2CCC(N(C(=O)C(C)O)CCO)CC2)=O)cc1 c1(C(=O)NC2CCN(c3cccnc3)CC2)cc(C(F)(F)F)cnc1O N1(C(C(C)CO)=O)CCN(C(=O)C(F)(F)Cc2ccccc2)CC(C)(C)C1 c1(C(N(CC(CC)NC(=O)C(F)C2CCC2)CC)=O)cnc(C(C)(C)C)nc1C C1(C)(C(=O)NCCCCNC(C(=Cc2cccs2)C)=O)CCOCC1 n1(CC)cc(Cl)c(C(=O)NCCC2(NC(C3CC=CCO3)=O)CCC2)n1 c1(C2(NC(C(C)(C3CCOCC3)OC(C)C)=O)CC2)cccc(O)c1 C1(C(N2CC3CN(C(C=C(CCC)C)=O)C3CC2)=O)Cc2c(C)cccc2O1 c1(C(N2C(CNC(c3nnsc3SC)=O)CCC2)=O)ccc(-n2ccnc2)cc1 Cc1c(CCC(=O)NC2CC2CN(C)C)cnn1C.C12(CC1)C(C)NC2=O N1(C(c2ncc(N)nc2)=O)CC(NC(c2ccn3c2CCCC3)=O)C(C2CC2)C1 c1(C(=O)NC2CN(C(C3C(C=C)C3)=O)CC2C)ccc(Br)c(C)c1 C(CC(CC)C(=O)N1CCC(C)(NC(c2cnc(C)n2C)=O)C1)=CC c1(C(=O)NCC(C2CCC2)NC(C2CSCCS2)=O)cccc(F)c1O c1(C(=O)NC(C)CCCNC(=O)C(C)(C)OCC(F)(F)F)cnn(C)c1N C1(C(NOCC(C(C)C)O)=O)CCN(C(c2ccncc2Cl)=O)CCO1 C1(CNC(C2CCC(O)(Cc3n(C)cnn3)CC2)=O)CCn2ccnc2C1 C12CC(C1)NC(=O)COCC(=O)OCCCNC2=O.C(C)(C)(C)NC(C)=O.CS c1(C(N2CCCC(N(C(CCC#CC)=O)CC)C2)=O)ccc(=NCCOC)[nH]c1 C1(NC(=O)CCCCN2CCCC2)CN(C(C23CCC2C3)=O)CCC12CCC2 CC1CCCCC1C(=O)NCC1(CNC(=O)CC#N)CC=CC1 N1(c2nccc(C(C)C)n2)CCCC2C1CCN2Cc1ccnn1C(C)C N(C1CC2(CCC2)Oc2ccc(F)cc21)S(=O)(=O)CCc1ccccn1 C12(C(N3CCC(CCNC(C(C)=C4CC4)=O)CC3)=O)CC3CC(C1)CC(F)(C3)C2 CC(CCC(C)(C)C)C(=O)NCC1C(CNC(C2CC3(CCO2)CC3)=O)C1(F)F N1(C(C2C(C)(CC)C2)=O)CCC(NC(c2cnc(C3CCC3)cc2C)=O)C(F)C1 c1(NC(c2ccc(P(C)(C)=O)o2)=O)ccc2oc(Cl)cc2c1 CC1(C)CCN(C(=O)CCc2nc(=N)[nH][nH]2)C1CC(=O)NCC1CCCCC1 c1(C(N(CCN(C(=O)Cc2nnc(O)s2)C)C)=O)ccc(-c2nnc(S)o2)cc1 C1(CNC(c2cc(C)oc2)=O)CCN(C(c2cc(C3CC3)[nH]n2)=O)CC1(F)F c1(C(N(CCCNC(=O)C(C)(C)C)CC)=O)c(OCC2CC2)cccc1Cl CC1(C)C2CN(C(C34CC3CCN4C(=O)CC3CCCSC3)=O)CC12 C(=O)(C(F)C(C)C(F)(F)F)NCCCCNC(c1ccc(CC)cc1OC)=O c1(N(C(=O)CCCc2ccncc2)CCC)cc(F)c(Br)c(F)c1 S(=O)(=O)(c1nnn(C)n1)NC(c1ccc(F)cc1)c1nc(C)on1 C1(NC(c2nccc(COC)c2)=O)CN(C(=O)C(C)N(C)C)C2(CCOCC2)C1 C1(CC(=O)NCC(N2CCN(C(=O)C=CC3CC3)CC2)C)CC(=O)NC(=O)C1 c1(N2C(CNC(CC(C)C(F)(F)F)=O)CCC2)ccc2c(n1)CCCC2=O C1(CNC(C2CCS2(=O)=O)=O)CN(C(=O)Cc2occc2C2CC2)CC12CC2 C1(CCCC)CN(C(=O)C(CCC)OC)CCN1C(=O)C1=CSCCO1 c1(CC)ncc(C(=O)NCC#CCNC(=O)Cc2nc(C)sc2Cl)c(C)n1 C1(C(=O)NC2C(NC(c3cccnc3SC(F)F)=O)COC2)CC(C2CCC2)C1 c1(CN(C(=O)NC2C(OC)(OC)CC2)C)ccncc1Cn1ccnc1 c1(C(N2CCC(C)C(NC(=O)Cc3cncs3)C2)=O)cc2n(n1)CCCCO2 C(=O)(C1OCCc2cc(O)ccc21)NC1(CNC(C(C)C(C)(F)F)=O)CC1 C=C1CC(C(=O)NC(C)COCC2CC2)(CNC(=O)C(C)OC2CCCC2)C1 C(CC(C(=O)NCC1CC(C)(O)C1)NC(=O)CC1CCN(C)C1=O)OC c1(OCC)cc(-c2cn(C3CC(C(=O)NCCOC(=N)O)C3)nn2)ccn1 c1(NC(C)=O)cccc(C(=O)NC(C)CC(C)NC(=O)C(C(C)O)N(C)C)n1 Cn1cnc2c1CCN(C(=O)CC(C)(F)F)C21CCN(CCOCC(F)(F)F)C1 CC(C)C(C(C)NC(=O)Cn1cnnn1)NC(c1cc(C#N)no1)=O C1(C(N2CCCC(CO)(NC(C3CC4CC4C3)=O)C2)=O)(OC)CCS(=O)(=O)C1 N1(c2cc(NCCCCCCO)nc(COC)n2)Cc2c[nH]nc2C(C)C1 CCC(C(=O)NC1CC1CNC(c1cnn(-c2ccc(Cl)cc2)c1)=O)C(F)(F)F N1(C(C2C(C)(C)C2)=O)CCC(NC(c2c[nH]ccc2=N)=O)C2(CCC2)C1 N1(CCC(=O)NC(C)C(N2CC(CO)(CO)C2)=O)CCOCC1 N1(C(CCCCCC#C)=O)CC2OCCN(C(=O)C(C)OCC3CC3)C2C1 CC(C)(C#N)CCC(=O)N1CCC12CN(C(c1ccc(CO)nc1)=O)C2 C12(C(N3C(C)C(O)CC3)=O)CCCC1CCN2C(=O)C(Cl)Cl N1(C(C2CCC(CCC)CC2)=O)CC2CC(NC(=O)CN3CCOCC3)C(C2)C1 O=C(CCCc1cncs1)NCCOC1CN(C(c2cccs2)=O)C1 CCCCCCC(C(=O)NC(CNC(=O)C=Cc1ncc(C)[nH]1)CC)NC(C)=O C1(C2CCCCC2)(NC(C2N(C(CC3OCC(C)(C)C3)=O)CC=C2)=O)CC1 CCC(C)CCCC(=O)N1CCC2CC2(C(=O)N(c2cccc(C)c2)C)CC1 C(CC(C)C)(C(=O)N1CC2CC2(CNC(c2cc(C)ccc2C)=O)C1)NC(C)=O c1(C(N2CC(NC(C(c3c(OC)cccc3)C)=O)C2)=O)cc(F)cc(N)c1N c1(C(C(=O)NC2C(CNC(=O)Cc3nnc(O)s3)C2)O)ccc(F)cc1 c1(CC)ncnc(N2CCC(C(=O)NC(c3ccc(Br)cc3)C(F)(F)F)C2)c1F C(=O)(C(CC(C)C)NC(c1nonc1C)=O)N(CC(CC)CC)CC C#Cc1cnc(C(=O)NCC2CCCC2NC(C2NC(=O)OC2C)=O)c(C)c1 CCC(C(=O)OC)C(=O)NCc1ncccc1C(=O)NC1(CC)CC1 N1(C(C2(CC#C)CCCO2)=O)CCN(C(=O)CCCOCC)C(c2cn[nH]c2)C1 C(=O)(CCCCCCNC(=O)C(C(C)C)SC)NCC(CC#C)(C)CO C1(C(=O)Nc2cc(C(N)=O)[nH]n2)CC(F)CN(C(=O)CC2COCCO2)C1 c1(C(=O)NC(CC=C)CNC(=O)CCC2CCC(=O)NC2)csc([N+](=O)[O-])c1 N1(C(C2(OC)CCCC2)=O)CC(CCNC(c2ccc(Br)cc2)=O)C(C)C1 C(=O)(C(C)(C)CS(C)(=O)=O)N1CCC(N(C(C=CC)=O)CCO)CC1 C(=O)(CC(O)CC(C)(C)C)NCC(CCNC(c1cc(C)n(C(F)F)n1)=O)OC c1(C(C)C(=O)NCC2CCN2C(=O)COCc2nc[nH]n2)c(F)cccc1F N1(C(c2nn(C)c(=O)cc2)=O)CCC2(NC(=O)CN3CC=CC3)CCCCC12 n1(CC(N2CC3C(CNC(C(C)O)=O)(CC3)C2)=O)ccc2ccc(F)cc12 Cc1cc2cc(-c3nc(C)nn3-c3cccc(C#N)c3)[nH]c2cc1Cl C1(NC(CCCCC)=O)CCN(C(=O)Cc2cc(C(F)(F)F)n(C)n2)CC1CO c1(CS(=O)(=O)NCc2n(C)nnc2)ccc(F)nc1 Cc1cnc(Cl)c(S(=O)(=O)NC2CCc3ccccc3C2)c1 C1(CNC(CN(C(=O)Cc2cnsc2)CC)=O)CN2CCC1CC2 C1(C(C)CNC(=O)OCc2ccccc2)CCN(C(C2(N(C)C)CCCC2)=O)CC1 C1(NC(C2CCC(OCC)C2)=O)CCN(C(=O)Cn2cc([N+](=O)[O-])cn2)C(C)C1 O=C(CS(=O)(=O)NCc1cscn1)Nc1c[nH]nc1NC(c1cccs1)=O C1(NC(CN(CCC)C(C2CCCCS2)=O)=O)CCOC(C)(C)C1 c1(C(=O)NC(CC=C)CNC(C2CCC2C(=O)OC)=O)cc(C)c(Cl)cc1F CCC(CC)C(C(=O)N(C1CC(C(N2CCC3CC23C)=O)C1)C)OC Cc1ccc(C)n1CC(=O)NC(CCC1CC1)C(=O)NCCCc1cncnc1 c1(C(C(=O)NC2CCC2)N(CCF)CC)ccc(-c2ccco2)cc1 c1(C(=O)NCC(C)CNC(c2nc[nH]c2C(C)(C)C)=O)ocnc1C1CC1 c1(C(C)C(=O)N2CC(Cc3ccccc3)C2)ccc(Br)cn1 C1(CNC(c2cc(C3C(C)C3)on2)=O)CC(C)N(c2nnc(CC(=O)OC)s2)C1 C1(NC(C(OC)OC)=O)CCN(C(c2cccc(N)c2F)=O)C1(C)C C1(C(N2CC(C(C(=O)NC(CCOCC)C)O)C2)=O)CCSCC1 c1(C(N(CCC2N(C(C(CCC)C)=O)CCCC2)C)=O)cc(OC)nc(OC)c1 CC1=C(C(=O)N2CC(NC(C3CC34CCCC4)=O)C(CC(C)(C)C)C2)CCO1 C(=O)(C1=C(Cl)CCOC1)NCCCCCCN(C(C1C2(CC(OCC)C2)C1)=O)C C1(N(C(=O)CSCc2ncc[nH]2)C)CN(C(=O)C=CC(=O)N2CCC2)CC1O c1(CC)cccc(C(=O)NC(CNC(c2ccco2)=O)C2CC2)n1 n1(CC(=O)NCC2CN(C(C(=O)NCC)=O)CC23CC3)cnc2c1CCCC2 c1(C(=O)NC(C(=O)NC(C=C)(C)C)Cn2cccn2)ccc(F)c(O)c1 c1(C(=O)NC(C(C)NC(=O)C(C)(C)C2CCCC2)C)cnn2cc[nH]c(=O)c12 C1(C(=O)NC2CCCN(C(c3c(CC)occ3C)=O)C2)CCc2nncn2CC1 N1(CC(=O)NCCN(C(=O)CCOCC(F)F)CCC)C(=O)NC(C)(CC)C1=O Cc1ccc(C(CNC(C2CCC(F)(F)C2)=O)NC(=O)Cn2cnnc2O)cc1 N1(C(c2c(OC)noc2C2CC2)=O)C2CCCC1CC(NC(=O)CCC1CC1)C2 C1(C)(NC(c2n(CC)cc(Br)c2)=O)CCCN(C(C2COC(=O)C2)=O)C1 c1(C(=O)NCCN(C(c2ccc(CCC)[nH]2)=O)CCOC)cc(C)c(C)nc1O C1(C(=O)NC(C)CCNC(c2c(C(C)(C)C)nsc2N)=O)CN2CCN1C(C)C2 c1(C(C(=O)N(C(CCNC(C2(CC#C)CC2)=O)C)C)O)cncn1C CCCCC(C(=O)NCC(C1CC1)N(C(=O)Cn1nc(C)cc1C)C)C(C)C N1(C(CN(CC)CC)=O)CCN(C(=O)C(OC)OC)CC1CC(F)F C1(CC)C(=O)NCCN1C(=O)C(N1CCCC(c2cc(C)ccc2C)C1)=O N1(C(CC2(OCC)CCC2)=O)CCOCC1CCNC(=O)CN1CCCNC1=O c1(SC)nc(C(N2CC3(CC3)CC2CNC(c2ccc[nH]2)=O)=O)c2ccccn12 C(=O)(CC(C)(C)CC)NCC(c1ccc(F)cc1F)NC(C=CCC)=O c1(C(=O)OC)cc(C(=O)NCC#CCNC(C2(Cc3ccccc3)CC2)=O)[nH]n1 C1(NC(C(C)C)=O)CCN(C(=O)C(C)Cc2cnn(C)c2)C12CC2 Cc1[nH]nc(C(=O)NCCC2CCCN2C(=O)Cc2ccsc2Cl)c1Cl c1(C(=O)NC2CCC(CNC(=O)C(O)C3CCC3)C2)csc2nnsc12 C1(C(N2C(C(C)NC(c3ccnn3C3CC3)=O)CCC2)=O)CC(=O)NC(C)C1 CC(C)CC(C)(C)C(=O)N1CCC1Cn1cc(-c2cncc(F)c2)nn1 C1(C(=O)NC)C=CC(NC(=O)CC2CCC(C)O2)C1 C1(C(=O)OC(C)(C)C)(C(=O)OCc2cnc(C(C)(C)C)o2)CCCCO1 N1(C(=O)CN2CCCOC2=O)CC2CC(C1)CN(C(=O)C(O)CC1CC1)C2 N1(C(C(C)(C)SC)=O)CC2C(C(=O)NCCc3ccc(O)cn3)C2C1 CC(C)(CC(=O)NCC1CCC(NC(C2(C)CC2C(F)(F)F)=O)CC1)C(F)F C1(C)(NC(C(C)C2CCC2)=O)CCCC1NC(=O)COc1ccsc1 C1(NC(C2CCC(C)(C)OC2)=O)CN(C(=O)CC2CC(F)(F)C2)CCC12CCC2 C(C(C(=O)NCC=CCCNc1ncc[nH]1)NC(=O)C1CC1)OC C(CCC(C)(C)C(=O)NCC1(CO)CC2CC2C1)NC(CCC1CC(OC)C1)=O CC(C)(CCCO)C(=O)N1CCC(N2CCN(C(=O)CCCNC(N)=O)CC2)CC1 c1(C(N(CC(CNC(C2(CC)CCCO2)=O)(C)C)C)=O)nn(C)cc1Cl Cc1nc(CC(C)C)c(C(=O)NCCCCC(C)NC(=O)C(C)N(C)C)s1 C(CCC(C(=O)N1CCOC(C)(C)C1)NC(=O)Cn1nc(C)cc1C)OC C(C)(C(C(=O)N=c1cc(C)n(CCO)[nH]1)NC(c1ccoc1Cl)=O)OC C1(O)(C(C)NC(c2ccccn2)=O)CCN(C(c2cccnc2C2CC2)=O)CC1 C(C(CC(=O)NOCC1CCOC1)C1CCC1)NC(C1(F)CCOC1)=O N1(C(CNC(CCC)=O)=O)CCCC(CNC(c2coc(C(F)F)c2)=O)C1 N1(C(CC(CC)SC)=O)CCC(C(C)C)CC1CNC(=O)C(Br)=C(C)C N1(C(C2CCCC23CC3)=O)CC2CCCC2(NC(C2(F)CCCCC2)=O)C1 c1(C(N2CC(O)(CNC(Cc3ccc(C)c(C)c3)=O)C2)=O)ccc2nncn2c1 C1(CNC(c2c(CC)[nH]c(=N)s2)=O)(NC(=O)CC2CCOC2)CCCCC1C C1(c2cc(C(=O)OCC)on2)CCN(N(C)C2CCCC2C(C)(C)C)CC1 C1(NC(C2(CC=C)CCCCC2)=O)CCC(C)(CNC(c2cccnc2)=O)CC1 c1(C(N2C(C)CC(NC(CN(C(C)=O)C)=O)C2)=O)ccc2c(c1)OC(C)(C)O2 N1(C(C(CC)C#N)=O)CCN(C(=O)Cc2ccc(Br)cc2C)C2CCCC12 N1(C(c2cc(C)sn2)=O)CC=CC(NC(=O)C(N2CCOCC2)C2CC2)C1 CCCC(C#N)C(=O)N1CCCC(n2cc(-c3cnc(C(C)C)o3)nn2)C1 c1(N(CC(C)NC(=O)Cc2cc(F)ccc2F)C)c([N+](=O)[O-])cnn1C CCC(C)(C)C(=O)NCC1CCC(NC(=O)C(c2cccnc2)O)C1 N1(C(c2c(C)c(O)ccc2)=O)CCC2C(C1)CN2C(=O)Cc1ncn2c1COCC2 N1(CC(=O)N(C)CC2CN(C(CCn3c(C)ncc3)=O)C2)CC2C=CC1C2 N1(C(c2c(C(C)(C)C)con2)=O)CC2CC(C1)N2C(C1CC2CCC2C1)=O CC(C)CC(C)(CNC(=O)C(F)(F)C(F)F)NC(C1CC(C)N(C)C1)=O CCCC(CCC)C(=O)N1CCC(C)C1C(=O)NOC1CCOC1=O.CC=O C1(C2CN(C(C3CCNC(=O)C3)=O)C2)(NC(C(C)Cn2ccnc2)=O)CC1 c1(C(=O)NC2CCN(C(C3(C(N)=O)CC3)=O)C2)ccc(F)c(C(F)(F)F)c1 n1(C(C)C)cncc1C(=O)NCC(C1CC1)NC(=O)CC1(c2ccon2)CC1 CS(=O)S(=O)CCN=c1[nH]c(N2CCC(Cc3ccncc3)C2)nc2ccsc12 c1(SC)ccc(C)c(C(=O)NCCC(C)(C)NC(=O)Cn2cccc(O)c2=O)c1 CCCCCCC(CC)C(=O)NCC(C)NC(c1ccc(-n2cccc2)cc1)=O C1(CC(=O)NCC2C(NC(=O)CN3CCCC3=O)CCC2)(CO)CCOCC1 N1(C(CC(CC)c2ccccc2)=O)CCC2(CCCN2C(=O)CC=C(C)C)C1 c1(-c2cn(CC(C)C)nc2)ccc2c(c1NCc1cnn(C)c1Cl)OCO2 CC1CCOC1CCNC(=O)C(=O)NC1(CCO)CC1 c1(CN(C)CCC2CC2)cc2c(cc1[N+](=O)[O-])OCCCO2 c1(C(=O)NC(C)CN(C(=O)CCc2cccc(O)n2)C)cc2c(s1)CCSC2 Cc1cc(F)ccc1C(=O)NCC1CCN(C(=O)CC(C)(C)N(C)C)C(C)C1 c1(C(=O)NCC(C)N(C(CN(CC)CC)=O)C)cc(OC)cc2c1OCC2 N1(c2ccc(CC(=O)OCC)cn2)CCC2(NC(C3CC3F)=O)CCCC12 c1(CCC)nc(C(=O)N(CCCNC(=O)C(F)(F)c2nccs2)CC)cs1 N1(C(C(CC(C)C)O)=O)CCC2(CCC2)C(CNC(=O)C#CC(C)(C)C)C1 C12(CNC(c3nn(CC)nc3C)=O)CC(NC(=O)C=C(Cl)Cl)(C1)C(C)(C)O2 c12cc(C)c(cc1OC)o2.n1(CCCNC2C(C(F)(F)F)(CC)C2)cc(Br)cn1 C(=O)(CCCC(=O)NC(C)C(C)(C)C(=O)NC1CCC(C(C)C)CC1)OCC CCC(CNC(=O)C(O)CNC(=O)C(=Cc1ccco1)C)C(C)(F)F C(c1cccc(Cl)c1)=C(C)C(=O)NCCCCCNC(C1CC(C(C)(C)C)C1)=O C(=O)(C(O)C1=CCCCC1)NC1(CCC(N2CC(C)(CO)C2)=O)CCCC1 c1(C(=O)NCCSC(F)F)ccc2c(c1)OCCO2 CCC(C)(C)C(=O)C(=O)N1CCCC(C)(NC(C2C3CCCCCCC23)=O)C1 C1(C(=O)NC2C(CNC(C(C)N(C)C)=O)COC2)C2CCCCC12 C(=O)(C(C)CC(F)(F)F)NC(C)CC(N1CC(F)C(F)C1)=O C1(C(=O)NC2C(OC)C(O)C2)CCCCCN1C(c1ncncc1N)=O C(=O)(CC(F)(F)Br)N(CCCNC(=O)C=C1CCOCC1)CC c1(OC)nc(C(=O)NC(CNC(c2cn(C(C)C)cn2)=O)C2CC2)sc1C C1(CNC(c2n(CC)ccc2)=O)CN(C(=O)C(C)CC2CCC2)CCN1C C(=O)(CC(C)(O)COC)NC1(CCCC(=O)NCC(CC)CO)CCC1 CC(C)P(=O)(CC(=O)NC(C)Cc1ccccc1Br)C(C)C c1(C(C)=O)ccncc1NC(c1ccnc(-c2ccc(Br)cc2)n1)=O c1(N2CCC(CC(N3C(C)COCC3)=O)C2)cnc(C#N)nc1 c1(NC(CC)C(O)C(C)C)ncccc1S(=O)(=O)NCc1nc(C(N)=O)co1 C#Cc1ccc(C(N2CCCOC(CCNC(=O)CN(C)C3CC3)C2)=O)nc1 c1(C(=O)NC2(CNC(C(c3ccccc3F)C)=O)CCOC2)ccc(=O)oc1 C1(C(N(CCOCC#C)C)=O)CC2CN(C(=O)C#CC3CCCC3)CC2C1 Cc1ccc(CN2CC(NC(c3cccc(Br)c3)=O)CC(F)(F)C2)cc1[N+](=O)[O-] c1(NC(=O)C(c2nc(CCO)cs2)N2CCC(CF)C2)ccc2c(c1)OCCO2 Cc1cc(C(=O)NCC2(O)CC(NC(C3(CCO)CC3)=O)C2)ccc1[N+](=O)[O-] CC1CCN(C(C2CCC3CC2CO3)=O)CCN1C(c1csnn1)=O Cn1nnc2ccc(C(=O)NC3CN(C(c4cc[nH]n4)=O)CCC34CCC4)cc12 N1(CC(=O)N(CCNC(CC2C(OC)CC2)=O)C)C(=O)NC2(CCOCC2)C1=O C1(NC(C(CC)C)=O)CCN(C(C2CC(C)C2)=O)CCC1CO C(C)(CO)(C(=O)NC1CCCC(CC(=O)N(C)Cc2ncccn2)C1)OC N1(C(c2cnc(C)n2C)=O)CCC(C2CC2)C1Cn1cc(C2(O)CCOC2)nn1 CCCC(C)(CC)NC(C1(CF)CCN(C(C2CCCOCC2)=O)C1)=O c1(-n2c(C)cc(C)n2)ccc(C(N2CC(Cc3cc(O)n[nH]3)C2)=O)cc1F C1(C(N(C2CCN(C(C3C(C)OCCC3)=O)C2)C)=O)C2CCC3(COC(=O)C13)O2 N1(C(c2cc(CC)n(C)n2)=O)CCCC1C1CCCCN1C(c1cnn(C)c1)=O C1(OC)CCCCN(CC(=O)NCC(C(C)C)NC(=O)C(OC)OC)C1=O C1(NC(C(c2cccc(Cl)c2)C)=O)CC12CCN(C(C1CCCC(=O)O1)=O)CC2 c1(C(=O)NC(CC)CO)ccc(Nc2ncc(CCSC)s2)cc1 C12(C(N3CC(CNC(c4c(C)noc4)=O)C(C)CC3)=O)CCC(O)(CC1)CC2 N1(C(CCN(CCCCOC)C)=O)CCC(NC(C2CCOC2(C)C)=O)C(O)C1 C(=O)(C1CCCc2nc[nH]c21)NCCCN(C(c1cc(C#C)cc(F)c1)=O)C c1(C(N2CCC(N(C(C3CCCNS3(=O)=O)=O)CC)C2)=O)ccc(N)c(F)c1F N1(C(CN(CC(CNC(COCC(=O)N(C)C2CC2)=O)O)C)=O)CCOCC1 O=CN=c1nc2cccc(Cl)n2[nH]1.c1(C(N2CCCC2)CC)c(F)cccc1F c1(C(N2C(CNC(C(CC(C)C)OC)=O)CC2)=O)c(C)nc2ncnn2c1C C(=O)(CCCCNC(C1CN(Cc2cc(C)ccn2)CCS1)=O)OC c1(C(=O)NCCC2CCN(C(C(CC)(C)C(N)=O)=O)C2)cccc2nc(C)sc12 Cc1cc(C(N2CCOC(CCCNC(C3CCCCS3)=O)C2)=O)cc(N)c1 c1(CC(=O)NC2CCC(CNC(C3(C)CSC3)=O)C2)cncc(O)c1 C(=O)(C1CCCc2nnn(C)c21)NCC1(NC(CCN(C(C)=O)C)=O)CCOC1 N1(C(CCCOCC)=O)CCN(C(C2CC(F)C(=O)N2)=O)C(c2nccn2C)C1 CC1(C)CN(C(=O)C=CC2CCOCC2)CC1NC(C1(c2ccccc2)CC1)=O c1(C(N2CC(C)N(C)C(C)C2)=O)cc2cc(-c3ccoc3)ccc2s1 C1(CC)CN(C(c2ccsc2-n2nc(C)nc2C)=O)CCC1NC(=O)C(C)(F)F c1(C(=O)NC2(CNC(C(C)(C)CO)=O)CCCCC2)ccc2c(c1)COC2 C1(C(=O)NCC2(C)C(C)CN(C(C34CC(CO3)C4)=O)C2)COc2ccccc2O1 C1(C)(CNC(c2cc(C)c(C)o2)=O)CCN(C(C2SCCC2C)=O)CC1 CCCC(C)(C)CC(=O)NCc1cc(C)c(C(N2CCC(C)(F)C2)=O)o1 Cc1nc(C(N2CCN(C(c3cnn4cccnc34)=O)CC2C)=O)cn(C)c1=O CC12CSCC1CN(C(=O)CNC(C1CN3CCN1CC3)=O)C2 c1(CC(=O)N(CC(C)NC(C2C(OCC)C2)=O)CC)ccc(-n2cnnn2)cc1 C1(NC(C(C)CF)=O)CC2CCC1C(NC(c1cc(F)cc(Cl)c1O)=O)C2 N12CC(CC3OCCC13)C2=O.c1(CC)cccc(OCCS(=O)(=O)N2CCC2)c1 C(=O)(CC(C)(O)COC)N(C1CCN(C(=O)Cn2ncc(Cl)c2C)C1)CC Cc1cccn2nc(C(N3CC(CNC(=O)C(C)n4cccc4)CC3C)=O)cc12 O=C(N=c1ccn(CCC(F)(F)F)[nH]1)N1CCCC(Nc2ccc(Cl)cc2)C1 C1(C(=O)NCC2CCN(C(COC)=O)C23CC3)COc2c(OC)cccc2C1 c1(C(N(c2ccc(C)c(Br)c2)C)=O)cnc(C)c(Cl)c1Cl C1(n2cc(CC(Cc3ccccc3)NC)nn2)CCCN(c2nccs2)C1 C1(CNC(=O)Cc2ccc(F)cc2Cl)CCN(C(=O)CC=C(Cl)Cl)CC1(F)F c1(C(N(C(C)CNC(=O)Cc2nocc2C)CC)=O)ncoc1Br C1(C(N2CC(CCC)C(CO)C2)=O)CNC(=O)CN1C(C1CCS(=O)CC1)=O c1(CCOC(C)=O)cn(CC(C)NC(=O)CC2CCCC2C)nn1 C(=O)(C1CCc2cccc(F)c21)NCCCCCCNC(c1n(C=C)nnc1)=O C1(C(=O)NCCC2CCN(C(Cn3c(=N)nc[nH]3)=O)C2)CC12CCC(F)(F)CC2 C(C(C)C(F)C(=O)Nc1ncccc1C#N)NC(C(C)NC(CC)=O)=O C1(F)(C(N2CCCC(C(C)C)C2)=O)CCCN(C(=O)CC2CC3(CC3)C2)C1 C#CC1(C(N2CCC(C(F)F)CC2)=O)CCN(C(c2ncn3c2CCC3)=O)C1 c1(C(N2CC3(C(NC(c4nnn(C)n4)=O)CCC3)C2)=O)cc([N+](=O)[O-])cnc1N N1(C(c2cn(CCC=C)nn2)=O)CCCC(C2(NC(=O)C(C)CN(C)C)CC2)C1 c1(OCC)ccc(CC(=O)NCC2CCCC(NC(C3C4COCC34)=O)C2)nc1 Cc1cccc(C(N2CCC3C(NC(C4CCOC4C)=O)C3C2)=O)c1O c1(-n2c(C(C)CN(C)C)nc(-c3ccccn3)n2)cccc2cnccc12 C1(C(N2CCC3(CC(NC(CC4(C)CC4)=O)C3)C2)=O)CC12CCOc1ccccc12 O=C1CC(C(=O)NCC2CC2NC(=O)C2=CCSC2)c2ccc(F)cc2N1 CC(CN=c1[nH]ccnc1F)(C1CC1)N(C(C1(C(c2cnn[nH]2)=O)CCC1)=O)CC CC1CN(C(c2nnn(C)c2C(F)(F)F)=O)CC1NC(c1cc(C(F)F)[nH]n1)=O N1(C(Cc2ccc(C(C)=O)s2)=O)CC(C)(C)C(NC(=O)C(C)CO)C(C)(C)C1 c1(C(N2CCC(C(C(=O)NCC(CC)C#N)C)C2)=O)cc(C)c(C)o1 c1(C(=O)OC(C)(C)C)ccnc(C(N2CCC2CNC(=O)C(Cl)=CCl)=O)c1