SMILES C(=O)(CCS(=O)(=O)C(F)(F)F)N1CC(NC(c2ccc(O)cc2)=O)CC(C)(C)C1 N1(C(C2(C)CC2(Cl)Cl)=O)CCC(CNC(=O)CC2C=CCCC2)CC1 C1(C(=O)NCC(C(C)C)(C)NC(C2OCCC2C(F)(F)F)=O)CC(=O)C12CCC2 C(=O)(CCCN(C)CC(C)(C)C)N(C1CC(NC(C(C2CCOC2)OC)=O)C1)C c1(C(=O)NCCC(C)NC(CCc2cnc(C)o2)=O)ccncc1OC(C)C c1(C(=O)NCC2C(CNC(c3c(OC)cc(C)cn3)=O)C2)sccc1S(N)(=O)=O CC(O)CCCCCC(=O)N1CCC(C)(CCNC(=O)C=Cc2ccccn2)C1 C1(CSC(c2ccc(F)cc2F)C)CCC(F)(F)C(=O)N1 c1(C(=O)NC2CC(NC(C(C)NC(CC)=O)=O)C(O)C2)cc2oc(C)cc2[nH]1 C(=O)(C(CC)(CC)C(C)C)N1CCC(N(C(C2OC3CCC2C3)=O)CC)CC1 N1(C(CCn2ccc(C)n2)=O)CC2(CCC2CNC(=O)CSc2nnnn2C)C1 N1(C(C)C)CCC(C(=O)NCC(O)CCNC(=O)C(C)(C)O)CC1 C#CC1CCC(C(=O)NC2CCC(NC(C3CC4CC3CC4O)=O)C2)CC1 C12(C(=O)NCC(CCCC)O)COCC1CN(C(C1OC3CCC1C3)=O)C2 c1(C(=O)NCCCC(C)(C)NC(=O)Cn2cc(C#N)cn2)ccn2ccnc2n1 c1(C(=O)OC)ncncc1C(N1CCC1C(=O)NC1(CC)CCCC1)=O c1(NC2(CC(=O)O)CC2)ccc(Br)c2c1CCCC2 C1(O)(C(=O)NCC2(C)CCN(C(C)=O)C2)CCCN(C(c2occc2Cl)=O)C1 C(=O)(N=c1[nH]nc(-c2ccc3c(c2)OCO3)s1)Nc1c(CC(C)C)cccc1 N1(Cc2cn(C(C)C)nn2)C(C)CN(C(=O)C(F)C2CCCC2)CC1C Cc1cc(F)ccc1C(C)NC(C1CC(c2nc(=O)o[nH]2)C1)=O C1(CNC(N(C2(NC(=O)CCc3csnn3)CC2)C)=O)CCCO1 N1(C(CCCOCC)=O)CC2(NC(c3cc[nH]c3)=O)CCC1CC2 N1(C(C2CCCN(C(C3CCOC3)=O)CC2)=O)CCn2c(Br)nnc2C1 C1(C(=O)OC)CCCC(CC(C)C)N1CCCc1nc[nH]n1 C1(C(=O)NC2(C(=O)OC)CC2)CCN(C(=O)Cc2cc(C)on2)CC1 C1(COCC(=O)N(CC(CN(C(COC)=O)C)O)C)CCCCO1 c1(SCCC)ccc(C(N2CCC(NC(c3ccoc3)=O)C2)=O)cc1 CCC(C)(CN=c1nc(N(CCC(O)C(C)(C)C)C)c2ncccc2[nH]1)C(N)=O N1(C(c2ccncc2Cl)C)CC(C)(Cc2ccc(Cl)cc2)CC1=O C1(C(C)(C)CNC(=O)CCn2ccnc2)CCCN1C(=O)CC(O)C1CCCC1 C1(C(=O)NCc2c(C(C)C)ocn2)CN(C(=O)C(C)c2ccco2)CCO1 O(C=CC(=O)N(CCNC(=O)CN1CC(C)C1)CCOC)CC Cc1ccc(NCC(=O)NCCCN(C(C2(c3cncs3)CC2)=O)C2CC2)cc1 C1(C#C)(C(=O)NC(C#C)C(C)C)CCN(C(C2CC3(CCC3O)C2)=O)C1 c1(C(=O)NC2C(NC(c3scc(C)c3Cl)=O)C2)c(F)ccc(F)c1O C(=O)(C1=CCC(C)CC1)N1CCC(F)(CNC(C(C)C)=O)C1 N1(C(C2C(=C)CC2)=O)CCC(CCOC)(NC(c2ncc(OC)cc2F)=O)CC1 C(CC(O)C(=O)NCCCCCC1CC1)NC(c1scc(C)c1)=O c1(SCC(=O)N(C2CCN(C(C(CC)O)=O)CC2)CCO)ccc(C#N)cc1 c1(C(C)NC(c2nnnn2Cc2cccs2)CCC)cc(CC)no1 N1(C(CNC(C)=O)=O)CCC(OC(CCCOC(C)C)=O)C1C(F)(F)F O=C(CC(C(F)(F)F)NC(c1cnsc1)=O)NCCN1C(=O)CNC1=O C1(COC(c2ccc(Cl)c(Cl)c2)=O)CN(C(c2cccc(Cl)n2)=O)C(=O)CO1 CCC(C(=O)N1CC2CCC(C(N3CCN(CC(N)=O)CC3)=O)(C2)C1)C(F)(F)F c1(C(=O)NC2(CNc3ncc(C)cc3[N+](=O)[O-])COC2)oc2c(C)cccc2c1C c1(C(=O)NC2CCN(Cc3[nH]c(=N)sc3)C2)ccc([N+](=O)[O-])cc1F C12CCC3CN(CC3C1)C2.C1(C(=O)NC(c2nc(C3CC3)no2)C)CCC(C)(C)C1 C1(C(C(N2CC(CN(C(CCOC)=O)C)C2)=O)O)CCCCC1 CCCCCC(O)CC(=O)NC1CC(C)N(C(=O)Cc2ccc(F)cn2)C1 c1(C(=O)NC2CCN(C(CCSC)=O)CC2O)ccc2nc(C)c(=O)n(C)c2c1 c1(OC)ccc(C)cc1C(N1CCC(O)C1C(=O)Nc1ncc(O)cc1Cl)=O c1(CC)nonc1C(=O)NCC1(F)CC(NC(c2ccn(C(C)C)n2)=O)C1 N1(C(CCNC(c2nccs2)=O)=O)CCC2(CCCN(C(=O)OCC(F)(F)F)C2)C1 C#Cc1cc(C(=O)NC(CNC(=O)C(C)(C)n2cnnn2)(CC)CC)cc(F)c1 C(=O)(C(O)CC(C)C)N1CCC(CCC(=O)NCC(COC)(C)CO)CC1 Cn1cnc2cccc(C(=O)NCC(C3CC3)Nc3cncc(Cl)n3)c12 C#CC(C)N(C)N1CCN(CCN(S(C)(=O)=O)C)CC1 CCC(COC)C(=O)NCC(c1ccccc1OC)NC(c1sncc1C)=O c1(C(CC)C)cc(C(=O)N(CCCCCNC(c2nsnc2O)=O)CC)on1 C1(C(N(CC(CN(C(=O)CCC2CC2)C)O)C)=O)CC12CCSCC2 c1(C(=O)NC2CC(NC(c3cc(Cl)cc(Cl)c3O)=O)C2)cc2cccnc2[nH]1 C1(NC(=O)CNC(C(c2ccccn2)N(C2CC(=O)C2)C)=O)CC(F)(F)C1 C1(CNC(C(C)OCC)=O)CCC(C)(C)CN1C(=O)CCCc1ccccn1 C1(C(N2C(C)CC(CNC(=O)C(N)=O)CC2)=O)CN(C)C(=O)CCO1 N1(C(C(COC)C)=O)CCN(C(c2cn(C)nc2Cl)=O)C2CS(=O)(=O)CC12 CC1=NC(C)(C(=O)N(C)CC2CCCCN2C(C2CC(O)C2)=O)N1C N1(C(C2CCC(=O)NC2)=O)CCC2C(C1)CN2C(c1cn[nH]c1)=O N1(C(c2cc(CC)[nH]n2)=O)CC2CCN(C(c3noc(CC)c3C)=O)C2C1 C1(C#N)(CCSC)CCN(C(=O)C(=O)Nc2cc(OC(F)(F)F)ccc2F)CC1 C(=O)(CCCCC(C)C)N1C2CC(CNC(CC3(COC)CCCC3)=O)C1CC2 N1(C(C(CCC)C)=O)CC(C)(C)CC1C(=O)NC1(CC(=O)OC(C)C)CC1 C(C(=O)N1CC(NC(C2CC(C)(C)C2)=O)C(C(F)(F)F)C1)(C(C)C)OCC(C)C CC1(C)C(NC(=O)CC2CCCOC2)CCN1C(=O)C1=CSCS1 c1(C(=O)NC(CNC(C(CC)N2CCCC2=O)=O)C)cc(NC(C)=O)cnc1O c1(-c2ccc(CN3C(CN)CCCCC3)o2)c[nH]c2ccccc12 C=CC1CN(C(=O)C2=CCSC2)CC1NC(=O)CC1CSCCS1 C(C)(CCCCNC(c1cncc(N)n1)=O)NC(CN1CCC(OC)C1)=O C1(C(N2CCC(CC=C)(NC(c3nnc(C(C)C)s3)=O)C2)=O)CCCCN1N=O C12(CNC(C3C(CNC(c4c(C(C)C)ocn4)=O)C3)=O)COC(C1)C(O)C2 C1(N(CCC)C(C2CCC2c2ccccc2)=O)Cc2ccccc2C1 c1(C(=O)OC2CCC(=O)NC2=O)cccc(S(=O)(=O)N2CCC(O)CC2)c1 N1(C(Cc2cn(C)nn2)=O)CCN(C(c2ccc(OCCO)cc2)=O)C(CO)C1 c1(C(N2CC(C)C(C)(CNC(c3ccc(F)o3)=O)C2)=O)cc2cccn2c(O)n1 CC(CC(F)F)C(=O)NCC1(O)CCCN(C(C2(CCN(C)C)CC2)=O)C1 C=CCC(CC(=O)N1CC(N2CC(O)C2)C1)NC(c1cn(CC)cn1)=O C1(CC(=O)NCCOCCCN(C)C(c2ccco2)=O)CC2CC1C2 c1(CCC)sc(C(N2CC(CNC(C3(C)CCCC3)=O)CC2C)=O)cc1CC O=C(C1=CCC2CCC1N2C(c1cn(C2CC2)nn1)=O)NC1C(O)C2CCOC12 c1(CN(C2(C)CCCCC2C(=O)O)C)cnc2sc(Br)cn12 C1(OC(C)C)CCN(C(C2CC(C)N2C(=O)COc2cccnc2)=O)C1 c1(C(=O)NC(C(=O)NC(CC#C)C(N)=O)COCC)c[nH]c2nccc-2c1 N1(C(c2c(-c3n(C)ncc3)n[nH]c2)=O)CCOC(C)(C)C1CO C(c1csc2ccccc12)=CC(=O)NCC(CNC(C1(OC)CCCCC1)=O)C C#CCCCCCC(=O)NCC1(O)CCN(C(=O)Cc2cn3c(n2)CCCC3)C1 c1(CN(CCN)CC)ccc2nonc2c1 N1(C(C2(C#N)C(C)C2)=O)CCN(CC(CC(C2CC(C)(C)CO2)=O)=O)CC1 c1(C(N2CC3(C(NC(C(C)N(C(C)=O)C)=O)CC3)C2)=O)cn(C)c2ccccc12 C(=O)(C1SCCc2sccc21)NCC(CO)NC(CCCC)=O C1(NC(c2c(C)nc(C)[nH]2)=O)CCCC(NC(=O)CN2CCCNC2=O)CC1 c1(OC)ncc(Cl)cc1NC(C1(F)CCN(C(C2(c3cccs3)CC2)=O)C1)=O C1(CC(=O)NC2(CN(C(CCN(C(C)=O)C)=O)C)CC2)CCC(C2CC2)O1 c1(C(=O)NCC2N(C(C3OCCC(=O)C3)=O)CCC2)cc[nH]c2nccc1-2 c1(CC(N2CC(O)(CN(C(CSCC(=O)OC)=O)C)C2)=O)cccc(C)c1 c1(C(=O)NC(C)CN(C(=O)C(C)OCC(C)C)C)cnn(C(F)F)c1 C1(C(N(CC(C)C)CC(=O)NCC2(CO)CC3CC3C2)=O)CCCCOCC1 N1(C(C(COC)O)=O)CC(=O)NCC1C(=O)N(C)Cc1ccncc1C C(=O)(CC1=CCCCC1)N1CCC(C(=O)NC(c2nccs2)CC)C1 C(CCCCCNC(C1(C)CC1(F)Cl)=O)NC(CN(C)C(c1ccccc1)=O)=O N1(S(CC)(=O)=O)CCCC1C(N1CC=CC1CNC(=O)Cn1cc(C)cn1)=O Cn1cc(Cl)c(C(=O)NCC(CO)NC(c2cccn2C)=O)n1 C(C)(C)(CC(=O)N1CC(CNC(=O)CCc2nc(C)cs2)(OC)C1)OC Cc1[nH]c2ccccc2c1CCC(N1CC2CN(C(=O)C3=NOCC3)CCC12)=O N1(C(CCOCC#C)=O)CC(CNC(=O)CC2CC(F)(F)C2)N2CCC1C2 C1(C)(CNC(C2C(C)=C2)=O)CCCN1C(C1CC(C)OC1C)=O c1(-c2n(CCCC)nc(CSC)n2)nn(-c2ccccc2)cc1[N+](=O)[O-] C#CCC(C)C(=O)NC(C)CNC(=O)COc1ccc(C(C)C)cc1 N1(C(c2c(C)oc(Cl)n2)=O)CCC2(C)CN(C(=O)CCC3CC3(C)C)CC12 N1(C(CC2C(C)CCN(C(C3(CC(C)=O)CC3)=O)C2)=O)CC2(CNC(=O)C2)C1 C1(NC(c2cc(CC)no2)=O)CCOCC1NC(c1cc(C)n(C(C)(C)C)n1)=O C1(CC=C)(NC(C2CCOCC2)=O)CCN(C(C2CC(=O)N(CC)C2)=O)C1 C(=O)(CCCCC(=O)N1CC2(CCC(NC(C3CCCC3)=O)C2)C1)OC N1(C(CC2N(C(C3(C)CC4(CC4)C3)=O)C3C2CCC3)=O)CCC2CCC(C2)C1 c1(N2CCCC(N3C(=O)NCC3)C2)nc(=NCCC(F)F)[nH]c2c1CCCCC2 c1(C(=O)NC2CC(C(=O)NCc3ccc(Cl)nc3)C2)ccccc1C1CC1 N1(C(C=CC2N(C)CCC2)=O)CCCC(C)(C)C1CNC(c1cccc(N)n1)=O C1(CC)CN(C(=O)C(C)n2ccnc2)CCN1C(=O)CCNC(=O)C=CCl c1(C(=O)NCC2CCN2C(C2CC3C=CC2C3)=O)cc(F)ccc1Br C1(C(N2CC(CC)N(C(=O)CSC)CC2)=O)Cc2ccncc2C1 c1(OC)ccc(C)cc1C(=O)NC1CN(C(=O)C(F)(F)C(C)O)CCC1CO C1(CC)(CNC(C2CC2(C)C)=O)CN(C(=O)CNC(=O)C(c2cnn(C)c2)O)C1 N1(C(CC(C=C)(C)C)=O)CCC2(CNC(c3coc(SC)c3)=O)CCCCC12 C=CCCC(C)(C)C(=O)N1CCCC(N(C)C(c2ccc(C(F)(F)F)cc2)=O)C1 Cn1cc(C(=O)OCCc2ccccn2)c(C2CCCO2)n1 S(=O)(=O)(c1nc2c(s1)CCCC2)NC(c1ccc(N(C)C)cn1)=O Cc1cc2cccnc2nc1C(=O)NC1CCC(NC(=O)Cn2cnnc2)CC1 C1(OCC)COCCC1CC(N1CC=CC(NC(=O)CCC(C)SC)C1)=O C(C(=O)NC1(C)CC(NC(C2(C(=O)N(C)C(C)C)CC2)=O)C1)(C(C)C)NC(C)=O c1(C2CCN(C(C(C(C)C)F)=O)CC2)nnc2n1CCN(C(=O)C=CC1CC1)C2 c1(C(=O)NC2CC3(C2)CC3C(=O)NCC2CC3(CCC3)C2)c(F)cccc1F c1(C(N2CC(C=C)C(NC(c3cnc(C)[nH]3)=O)C2)=O)sc2ccccc2c1Cl C1(NC(C2(CNC(C(C)OCC3CC3)=O)CC23CCC3)=O)C=CC(C)(C)CC1 C(=O)(C(C)(C)C1=CCN(C(c2cccnc2S)=O)C1)N1C(C)C(C)(C)CC1 CC(C)C(CCN(C(=O)C(C)(C)c1ncco1)C)NC(=O)CO C(=O)(C(C(C)C1CCCC1)N(C)Cc1ccccc1Br)NCCCCCC Cc1cc(C)c(C(=O)NCC(O)CN(C(=O)C(c2cccnc2)O)C)s1 C1(C(=O)NCC(CC(C)C)NC(c2c(C)nccc2)=O)CC2CCCCN2C1 c1(C(=O)NC2CCN(C(C(CC(C)C)N(C)C)=O)C2)cccc2c1OCC2(C)C c1(C(=O)NC(CNC(C2CC(CC(F)(F)F)C2)=O)C2CCC2)ccc(Cl)[nH]1 CC1(C)CCOC1C(=O)NCC1(NC(=O)C2=CCSC2)CC1 c1(C(=O)NCCOCCCN(C(c2ccc(CC)cc2)=O)C)cccn(C)c1=O c1(C(N2CCN(C(C3CC(OCC)C3)=O)CC2)=O)ccc(Cl)nc1Cl Cc1cnc2c(cnn2CC(N2CCCC([Si](C)(C)C)C2)=O)c1 c1(C(N2CC(NC(C3CCSC3)=O)CC3(C2)CC3)=O)cc2cc(Cl)cnc2o1 c1(OC)cc(C)nc(NC(C2CC(NCc3cccn3C)C2)=O)n1 N(C(=NCCC(C)C)NCC1CCC2(COC2)O1)CC(c1ccc(Cl)cc1)CC Cc1n[nH]c(C)c1CCC(N1CCC(C(C)NC(=O)Cc2ccc(F)cn2)C1)=O c1(C(=O)NCC2(F)CCN(C(C(C(C)C)C#N)=O)C2)ccsc1S(N)(=O)=O C1(N(C(=O)C(=O)NC(C)C)CC)CCCN(C(=O)C(c2cn(C)nc2C)C)CC1 Cc1cc(C(=O)N(CC(C)CNC(=O)C(O)C(F)(F)F)C)cc(C)c1F CN(C)N=Nc1ccccc1C(N1CCOCC(C(=O)O)C1)=O C1(c2cccc(OC)c2)CN(C(=O)COCCF)CCN1C(C1(C)C=CCC1)=O c1(C(N2C(CNC(CNS(CC)(=O)=O)=O)C=CC2)=O)cc(SC)ccc1O C1(N(C)C(c2cc(Cl)no2)=O)CCCN(C(c2cnc(O)nc2O)=O)CC1 c1(C(N(C2CN(C(C3CCC4(CC4)C3)=O)C2)C)=O)c(Br)ccc2n[nH]cc12 c1(C(N(CC(C)N(C)C(C2CC(F)C(=O)N2)=O)C)=O)ncc2c(F)cccn12 C1(CC(=O)NCCN(c2nccc(-n3ccnc3)n2)CCC)CCC2CC2C1 C1(C(=O)NCCNC(Cc2ccn(C(C)C)n2)=O)COCCN1CC(F)(F)F N1(C(C2CC(CNC(C3COCC(C)O3)=O)OC2)=O)CCC(F)(F)C(O)C1 c1(CCC)ncc(C(N2CC(O)(CNC(c3coc(C)c3)=O)C2)=O)s1 C1(C(=O)NCC(CN(C(=O)Cn2nnnc2-c2ccccc2)C)O)OCC1(C)C CC(C)CC(C)CC(=O)NCCC1(O)CN(C(=O)C(C(C)C)SC(F)(F)F)C1 c1(C(=O)NC23C(NC(C(C4CC4)SC)=O)CC(CC2)C3)ccn2ccnc2n1 n1(CC(=O)N(CC(C)NC(=O)COCC2CCOC2)CC)[nH]cnc1=N N1(C(c2c(OC)n(C)nc2)=O)CCC2CCCC(C1)N2C(C1CSCCS1)=O N1(C(CC2C(C)C2)=O)CC2CCC(C1)C2NC(c1cc(Br)cc(Br)c1)=O C=C=CC(C)C(=O)N1CC(F)CC1C(F)(F)F C12(CNC(C3N(C(C4C(C)C4C)=O)CCOC3)=O)CCN(CC1)CC2 C12(CNC(C=CC)=O)CC1CN(C(=O)OC(C)(C)C)C2.c12ocnc1NC(=O)C2 Cc1cc(=NCC(C(C)C)N2CCC(C)CC2)[nH]c(N2CC(C)C(F)(F)C2)n1 C1(NC(C2(CC)C=CCC2)=O)CC2CC(NC(=O)CC(=O)NCC(F)(F)F)C1C2 C(=O)(C(C)(F)C(C)(C)F)NC1CC(F)(CNC(c2nc(C)nn2C)=O)C1 c1(CNCC2(C(N3C(C)C(=O)N(C)CC3)=O)CC2)cc(F)c(F)c(Cl)c1F C1(C(F)(F)F)(C(=O)OCC)CCN(C(=O)NCc2cnc(CC)s2)CC1 C1(C(=O)OC)(CNCC(C)(C)CCO)CCCCCC1 c1(CC)csc(CNC(C2(C3CCCN3C(C3(O)CCOC3)=O)CC2)=O)n1 CCCC(C)(CC)C(=O)NC(C)CC1CCN(C(=O)CC2CCNC2=O)CC1 C1(C(=O)NCC=C)CC(F)(F)CN1Cc1ccc(C2CC2)cc1 N1(C(C(=O)NC(CN(C(c2ccn(CCCC)n2)=O)C)C)CC)C(=O)CCC1=O C1(CC(=O)N(CCCNC(c2[nH]ccc2C2CC2)=O)CC)CCC(C)(C)CO1 C1(NC(N(C(C(C)C)CO)C(C)C)=O)COc2cccc(Br)c2C1 c1(C(=O)NCC2(C)CCC(NC(=O)CC3CCC3)C2)cc(Cl)ncc1O c1(OCCCC(=O)NCCNC(CSCCCC)=O)ccc(C)cc1Br N1(C(C2CN(CCC)C(=O)C2)=O)CCC2(CCC2NC(=O)CN(C)CCO)CC1 N1(C(C2CCC(N=[N+]=[N-])C2)=O)CCC(C2CCN(C(C3CC=CCO3)=O)C2)CC1 C1(CN(C(=O)COC)CC)CCCCN1C(=O)C(C)n1cccc1 N1(C(C(CCCC)(C)F)=O)Cc2n[nH]cc2C1C(=O)N1CCC(O)CC1 N1(C(C(c2cc(C)oc2C)C)=O)CC2CC1CN2C(c1ncoc1C(F)(F)F)=O N1(C(CC2N(C(CC(C)C3CCCO3)=O)C3C2CCC3)=O)CCOCC(C)(C)C1 c1(OC)nc(=NCC2CN(C(c3nc(O)sc3C)=O)CCCO2)[nH]c2[nH]cnc12 c1(CC(=O)NCCN(C(=O)C2=CCOCC2)C2CC2)cc2ccccc2o1 N1(C(c2c(CC)nc[nH]2)=O)CC(NC(C2CC3OC2C2CC32)=O)C2CCCC12 C(C1CCC(C)CC1)=C(C)C(N1CC(O)(C(C)NC(c2ncoc2C)=O)C1)=O CC1CC2CN(C(C3CSCCN3C(c3cnc(O)o3)=O)=O)CCN2C1 c1(-c2scc(NCC(C3CCCC3)N)n2)cccc(F)c1 c1(OCC(=O)NCC(C)NC(CCCN(CCOC)CC)=O)c(F)cccc1F c1(C(=O)NC(CCCCNC(C(CC)N(C)C)=O)C)nn(C)c(C)c1Br CCCCCC(=O)NCC(N1CC(CNC(=O)COCCF)C(O)C1)=O n1(CC)nccc1C=CC(=O)NC(C1(O)CN(C(C2CC(C)OC2C)=O)C1)C c1(C(N(C2CCN(C(c3nncs3)=O)C2)CC)=O)cc(F)cc2cnccc12 C1(C(=O)NCC2N(C(c3n(CC)c(O)nc3)=O)CCOC2)CC1C1CCOCC1 CC1C2CN(C(=O)C(C)(C3CCCO3)C3CC3)CC12.C1(CC2CC2)CCC1 N1(C(C(C)(C)OC)=O)C2CCC1C(C(N1CCC13CN(C)C3)=O)C2 C1(C(N2CCC(F)(CNC(CC3(OCC)CC3)=O)C2)=O)C2CCC(F)(F)C12 c1(C(N2C(C)C(NC(C3CCC34CCC4)=O)CCC2)=O)nn(C)c2c1COCC2 C(C(CO)C(F)(F)F)NC(c1c(CNC(C2CC(SC)C2)=O)cco1)=O C(=O)(C1=NOC2(CCC2)C1)N1CCC(NC(C(CCCC)O)=O)C1C Cc1cc(C(=O)N(C)CC2CCCCN2C(=O)CN2C(=O)CCC2=O)cc(N)c1 CC1CCN(C(c2cccnc2)=O)CC1NC(C1CNC(=O)N1)=O N1(C(Cn2ncc(C)c2)=O)CCC(NC(C2CC3CCC3C2)=O)CC(C)(C)C1 C1(CC)(NC(C23CSCC2C3)=O)CCN(C(=O)C(C(C)C)c2ccn(C)n2)CC1 C1(C#N)(CC(N2CCC(C)(CNC(=O)OC(C)(C)C)C2)=O)CC2CC2C1 N1(c2ccnc(OC)n2)CC2CCCN(C(c3cc(Cl)ccc3F)=O)C2C1 C=CCC(C(=O)NC1COC(C)(C)C1)NC(C1CC(=O)C1)=O c1(C(=O)NCC(C2(O)CN(C(CSCC)=O)C2)(C)C)cscc1C#N N1(C(c2ccc(C)cn2)=O)CCC2(C1)CN(c1ccc(C3CCCC3)cn1)C2 CCC(CCOC)C(=O)NCCOCC(=O)NCc1cc(C)sc1C c1(C(N2CCC(C(C(=O)NCCCOC(C)C)(C)C)C2)=O)cccc2cc[nH]c12 C(C#CC(=O)NC(C)CCN(C(=O)CC1(COC)CC1)C)(OCC)OCC C1(NC(C=CC(C)C)=O)CC2(C1)CN(C(C1CCC(F)(F)CO1)=O)C2 CN1CCOCC1C(=O)N(C)CCOCCC(=O)Nc1ccc(N(C)C)nc1 C(CC1CCC1)(C(=O)N1CC(O)(CCNC(=O)CCc2cc[nH]n2)C1)NC(C)=O CC(CCl)CS(=O)(=O)NC1CCCC2OCCC12 c1(N2CCCC(CCNC(C(C)(C)CF)=O)CC2)nccn2nnnc12 Cc1ccccc1-n1ncc(C(=O)NCC2(CNC(C3CC3F)=O)CCCC2)n1 c1(C(=O)NC(C(C)NC(COCC=C)=O)CO)ccc(C(=O)OC(C)(C)C)cn1 C(CO)(C(=O)NCC(C)(C1CC1)NC(=O)Cn1nnnc1-c1ccsc1)N(C)C c1(N(C(C(C)C)=O)C)ccc(C(=O)NC(CNC(=O)C2=CCOC2)C2CC2)cc1 c1(OC)ccc(C(N2CCC(O)C(NC(=O)COCC3CCOC3)C2)=O)cc1Br N(C1CCCc2ccccc21)N1CCN(C(=O)NC2CC(CC)OCC2)CC1 c1(CN2CC(C(N(C(C)(C)C)C(C)=O)=O)OCC2)cc(C#N)n(C)c1 C(CS(=O)(=O)CC)NC(c1n(CC(=C)C)nnn1)(C)CCC Cc1cncc(C(=O)NC2CCCN(C(=O)Cc3ccnn3C3CCC3)C2C)c1Cl n1(C(C)C(=O)NCC2CCC2NC(C2(C)CC2)=O)ccc(C(F)(F)F)n1 CC(CC(=O)NCc1ncccc1NC(C1CCCC1(C)CO)=O)C(C)(C)C N1(C(=O)OCCOC(F)F)CCC(O)C(N(C(=O)C2=CCCS2)C(C)(C)C)C1 Cc1ncc(Br)cc1C(=O)NC1CC1CNC(=O)C=C1CCC1 c1(COC(C23C(CN(Cc4ccc(COC(C)=O)o4)C2)C3)=O)cc(Br)ncc1Cl c1(C(=O)Nc2nnc(C(C)(C)C)s2)nc2ccc(-c3cnc(O)nc3O)cc2s1 c1(OC)cccc2c1OCC2NC(=O)C(C)(c1ccccc1)N(C)C CC12CN(C1)N2CCC1CCCCN1.c1(CCCC2CCOCC2)cccnc1 N1(C(CC(C=C)C)=O)CC2(CC2)CC1C(=O)NCCc1ccncc1C N1(C(C2OCCC(NC(CCCN(C(C)C)C)=O)C2)=O)CC2(CCOC(=O)N2)C1 Cc1ccc2oc(C(N3CCCC(CCNC(=O)C=CC(N)=O)C3)=O)cc2c1 c1(C(N(CCCNC(C(CC)COC)=O)C)=O)cc2cc(Br)cn2c(O)n1 c1(C(N2C(C(=O)Nc3c(CC)cccn3)CC3CC32)=O)cccc(CO)c1F C1(C)(C(=O)NCCN(C(=O)Cc2ccsc2)C(C)C)CCCO1 CC(C)C(C)C(=O)NC1CCC(CCNC(C2(CO)CCOCC2)=O)C1 C(=O)(C(C#N)C(C)(C)C)C1C2(c3c(C)nsc3C)N(CCSC3CC3)CCC(C1)C2 Cc1cc(C(=O)NC(C)(CNC(C2CC(C)(C)CN2C)=O)C2CC2)nc(O)n1 CCS(=O)(=O)CCNC(C1CCC(CNC(=O)C(CO)NC(N)=O)O1)=O C1(NC(=NCC)NCCNC(=O)OC)CC2CC(OC)C2C1 CCC(CC(C)C)C(=O)N1CCC(NC(=O)CC2CSC2)CC1C c1(CN(C)C)cn(C2COCC2NC(=O)C(N)COC(C)(C)C)nn1 C1(C(=O)NCC2(CN(C(c3c(COC)cco3)=O)C)CC2)CC(=O)N(C)C1 N1(C(C(CCCC)NC(=O)CN(C)CCC)=O)CCOC(C2(C)N=N2)C1 c1(OC)ccc(C(=O)N(CC)CC2CCCN2C(c2cc(Cl)cnn2)=O)c(F)n1 N1(C(c2cc(C)oc2)=O)CC(NC(c2ccccc2C(C)(C)C)=O)CC1C C(N=c1cc(C(F)(F)F)nc[nH]1)C1CCC(CNC(C2CCC(C)CC2)=O)CC1 N1(C(c2cc(=N)[nH][nH]2)=O)CC2C=CC1C(C(=O)NCC1CC3(CCC3)C1)C2 C(=O)(CC(C)(C)NC(=O)CSc1ccc(CN)cc1)NC C1(NC(=O)CNC(C2CCCC2F)=O)CCn2ncnc2C1 CN1CCC(O)C2(CCCN(C(=O)CC3CN(Cc4cccc(Cl)c4Cl)C3)C2)C1 C1(C(C)(C)CNC(=O)C2=CCSC2)CCCN(c2nccs2)C1.N12CC(F)(C1)C2 c1(C(=O)NCCCNC(COCC=C)=O)cc(F)cc(C)c1N c1(C(=O)NCC2C(NC(C(CCC)N(C)C)=O)C2)cc(C)c(CC)nc1O c1(N(C)C)cccc(C(N2CCCC2CCNC(C2CCNC2=O)=O)=O)c1 C(C(CC(=O)OC)C(F)(F)F)NC(c1n(CC=C)nnn1)CCCC N1(C(CCc2ccc(C)s2)=O)C(C(=O)NC2CCCC2C)C2CC(F)C1C2 c1(CN(C(C2CCN2C(=O)CC2CCOC2)=O)CC)occc1C.OCC S(=O)(=O)(c1ccc(Br)cc1Cl)Sc1ncnc(-c2ccc(C)cc2)c1N.c12nnc-1[nH]2 C(=O)(CC(CN(C)C)C(F)F)N(C1CN(C(CCOCCCOC)=O)CC1O)C CCC(C)C(C(=O)N1CC(COC)(OC)C1)NC(=O)CN(CC)CC N1(C(C(CC)Cc2ccccc2)=O)CC2CC(C1)N(C(=O)CSCC(=O)OC)C2 C(Cn1ccnn1)(C(=O)N1CCCCO1)NC(C1CN(C)C(=O)C1)=O C(CCCCC(=O)NC(C)(CNC(c1c(C)c[nH]c1CC(N)=O)=O)CO)SC c1(C(N)=O)ccnc(N2CCC(CNC(C3(CO)CCCCO3)=O)C2)c1[N+](=O)[O-] CCCC(C(=O)NC1(C(=O)OC)CC1C)NC(N)=O.c12ccsc1C(=O)NC2 c1(C(=O)NC2(CO)CN(C(c3occ(C(N)=O)c3)=O)C2)csc2c1CCCC2 CCCCCC(C)CC(=O)N1CCCC1C(C)(C)C(=O)NNCCC.CC CCC(C)(C)CC(=O)NC1CCN(c2cc(C3CC3)ncn2)CC1O Cc1cccc2c(CC(=O)NC3CCC(NC(=O)C(C)(C)C(F)F)C3)c[nH]c12 c1(C(N2C(C)(CNC(C#C)=O)CCC2)=O)cccc(CC(=O)OC)c1Br C12(NC(c3cncc(C(N)=O)c3)=O)CCN(C(C3CCSCC3)=O)CC1C2 C1(CN(C(c2ccc(C#N)s2)=O)CC)CCN(C(C2CCC(F)C2)=O)CC1 C1(C(N2CC(NC(C)=O)C2)=O)(CC)CCN(C(C2CC=CCC2)=O)C1 C(=O)(CC(C)C)NCCN(CCC(=O)OCCCOCCC(=O)NC)C1CC1 Cc1nn(CC(=O)NCC2CCN(C(c3ncncc3Cl)=O)C2)c(=O)n1C N1(C(C(n2ncc(C)c2)C)=O)CCC(NC(c2ccoc2)=O)C1C C#Cc1cccc(C(C(=O)NCC)N(C2CCCCCC2)CC(C)C)n1 Cc1c(C(N2CCC(NC(=O)C=Cc3nnc(C(C)C)o3)CC2)=O)ccn1C C#CC1(N(C)C)CN(C(C2(C(C)NC(C3C=C(C)CS3)=O)CC2)=O)C1 c1(C(=O)NC2CN(C(C(CC)C)=O)CC2CC)nnc2ccccc2n1 C1(C(N2CC(CS(N)(=O)=O)C2)C)CCOC1=O c1(C(N2CCN(C(C3CCCO3)=O)CC2CO)=O)ccc(F)c(F)c1F Cc1ccc(C(=O)NCC2(CNC(C3CCN(c4ncccn4)C3)=O)CC2)nc1 CCCC(C(=O)N1CCCC(Nc2cc(C(C)=O)ncn2)CC1)C(C)C c1(C(C(N)=O)N(CC(Cc2ccccc2)OC)C(C)C)ccc(Cl)cc1 CC1(c2cn(-c3ncc(O)cc3F)nn2)CCCN(C(=O)C(F)(F)C(F)F)C1 Nc1c(C(=O)NC(CNC(=O)C=CCN2CCCC2)CO)cccc1Br c1(CNC(=O)NC(c2cc(Br)ccc2OC)CC)cc2ccccc2s1 N1(C(C(CO)NC(N)=O)=O)CC2CC(NC(C3(O)CCSC3)=O)C2C1 S(=O)(=O)(c1ccc2c(c1)CCC2)Nc1ncc(C(=O)OC)cc1I C(CN=c1cc(NCc2nnc(C)o2)nc(C(C)C)[nH]1)NC(=O)NCC c1(CNC2CCC(C)S(=O)(=O)C2)ncnc2c1CCC2 C1(NC(C(c2ccn(C)n2)C)=O)CCN(C(=O)C(C2CCCCC2)C)C(C)C1 CC1CC(C(N2CCC(CF)(NC(c3ccnc(N(C)C)n3)=O)C2)=O)CC(=O)N1 c1(C(=O)NC2C(NC(c3c(C)onc3)=O)COCC2)ccc(C(C)C)nc1O C(=O)(C(C)CS(C)(=O)=O)N1C(CNC(c2ncc(C)c(C)c2)=O)CC1 N1(c2nc(C)nc(C#N)c2)CCCC1C1CCCCN1C(C1CCCN(C)C1)=O c1(NC2CC3N(C)C(CC3)C2)ccc(S(=O)(=O)N(C2(C)CCOC2)C)cn1 O=C1CC(C(=O)NCCCCNC(=O)C(F)C(F)(F)F)CC(=O)N1 c1(C(=O)NCC(C)CNC(=O)Cc2cc(C(F)(F)F)n[nH]2)ncn2c1CCCC2 N1(C(C(C)OCC=C)=O)CC(C)(C(=O)N(CC(F)F)C)CC1(C)C Cc1[nH]c2ccccc2c1C(=O)N(C)CCNC(c1cncc(Cl)c1Cl)=O C1(NC(C=CC(C)C)=O)CC(CNC(C2CC2c2ccc(F)cc2)=O)C1(C)C C1(NC(C2C(C)N(C)CC2)=O)CC(F)CN(C(C2(F)CC=CC2)=O)C1 N1(C(CC2N(C(C3C4CC(=O)CC43)=O)CCC2)=O)CC2(CCC(=O)O2)C1 N1(C(Cc2cc(OC)c(F)cc2)=O)CC2CN(C(=O)COCC(C)(C)C)CC2C1 c1(C(N2CC(C)OC(CCNC(=O)Cc3cnc[nH]3)C2)=O)n[nH]c2c1CSCC2 c1(C(=O)NCC(CC)NC(=O)C(C)(F)C(C)(C)F)cc(OC)c(OC)cc1C Fc1cccc2nc(N3CCCC3)[nH]c(=NC3CCOCC3)c12.c1ccccn1 c1(C(=O)NC(CNC(c2c(=N)[nH]cnc2)=O)CO)ccc2c(c1)CCCC(=O)N2 N1(C(C=C(C)C)=O)CCOCC1CN(C(=O)Cc1ccc(C2CCC2)cc1)C c1(C(N(C2CN(C(=O)Cc3nnc(O)s3)CC2F)C)=O)ccc(F)c(C(F)F)c1 CC(C)C(F)(CNC(c1cncn(C)c1=O)=O)C(=O)N1CCC2(CCSC2)C1 c1(OC)ncc(Br)c(NC(C)(C)CN(C)C(C2CCCC(O)C2)=O)n1 C(CC(C(=O)NCCN(C(=O)Cn1nnc(C2CC2)n1)C)NC(N)=O)N(C)C CC1(CCO)CCN1C(c1n[nH]cc1CNC(=O)Cn1ncnn1)=O c1(C(=O)NCC2CC(COC)CN2C(=O)COC(C)=O)cc(=O)n(C)cn1 c1(C(N2CC(CNC(c3cc[nH]n3)=O)C3C2C3)=O)cc2ccc(Cl)c(F)c2o1 c1(NC(C2N(c3c(F)cnc(OC)n3)CC(F)C2)=O)ccc(O)c2ncccc12 c1(C(=O)NC(C)CN(C(=O)C(C)C(C)O)C)ccc([N+](=O)[O-])[nH]1 c1(OCC(=O)OC(C)C(=O)Nc2ccc(N)cc2)c(Cl)cccc1Cl N1(C(CSCCC)=O)CC2CCC1C2NC(c1cc(C(=O)OC)on1)=O N1(C(=O)CCCCC(F)F)CCC2(CCN(C(=O)CC3CC(F)(F)C3)C2)C1 C1(C(C)NC(c2coc(CNC(=O)CC3CCC4CC34)n2)=O)CC(O)C(O)C1 c1(NC(C2C(NC(C(CC)NC(N)=O)=O)CCO2)=O)cnc(F)nc1 Cc1c(C(=O)NCCOCCNC(=O)CC23COCC(C2)C3)cccc1C#N.C1(O)CC1 C#Cc1ccc(C(=O)NCC2(F)CC(NC(c3ccncc3OC)=O)C2)nc1 N1(C(C2CCCC(F)(F)C2)C)CC2C3CCC(C3)C2(C)C1 C12(C(=O)NC3CC(NC(=O)CSc4ccncc4)C3)CC3CCC(CC(C3)C1)C2 C1(C(=O)NCC(N(C(=O)CCN2CCC(O)CC2)C)C2CC2)OC2CCC1CC2 N1(C(=O)OC)CCCC(NC(C2C3CC2N(C(=O)CC2CCCCC2O)C3)=O)C1 C1(C(=O)NC2(CNC(c3c(C)c(N)ccc3)=O)CCCC2)CCCCC(C)(C)C1 C(=O)(C1CC=Cc2ccccc21)NCC(CC)NC(=O)C(F)(F)CN(C)C CCCC(C)(C)CC(=O)N1CCC=CC1C(=O)NC(C12CCC(CO1)C2)C CCCC(CC)CC(=O)NCc1cc(C2CCN(C(C3(SC)CC3)=O)CC2)no1 CC1(C)CCN(C(c2c(N)cccc2F)=O)CC1NC(=O)C=C1CCCC1 CC1CCC(NC(c2cnn3ccsc23)=O)CN1C(=O)CC12CC(C1)C2 c1(OC(CC)CNC(C2(C)CCSCC2)=O)cccc(C)c1 c1(C(=O)NC(CC)CC(=O)NC2COC(C)(C)C2)ccc(O)nc1C C(=O)(C1CCOc2ccccc21)NCC1C(NC(CCCN=[N+]=[N-])=O)CCCC1 C(CN(C)C(C1CN(CC(C)C)C1)=O)(CO)(CO)NC(COCCC=C)=O CCCCC(=O)NCC1(O)CC(C(N2CCOCC2)=O)C1 c1(C(=O)NCC2(F)CCCN(C(COC)=O)C2)cc2c(Cl)cc(F)cc2[nH]1 C1(NC(C(C)N(C(C(C)NC(=O)C2CC2)=O)C2CC2)=O)CCC(=O)NC1C C1(CC(C)C)COCCN1C(C1CC(CCNC(=O)C(=O)C(C)C)C1)=O CCC(C)(C(=O)Nc1ccc(C(N2CCC(C(C)OC)CC2)=O)nc1)OC C(C(=O)NC(c1cnc[nH]1)C)(C(C)(C)C)NC(c1c(C)cc(F)s1)=O N1(C(c2c(OC)ccs2)=O)CCCC2CN(C(c3cnc(C)n3C)=O)CC12 N1(C(C(C2CCCC2)SC)=O)CCC(CNC(=O)C=CC2CC2)C(CO)C1 O=C1CCN(C(c2cn(-c3cccc(CNc4ccccc4)c3)nn2)=O)CC1 N1(C(CCN(C(=O)CC(C)(C)CCC)CC#C)=O)CC2(CCC2)CC1C c1(C(=O)NCC2(NC(C(C(C)C)c3ccc(Cl)cc3)=O)CC2)ccccc1C#N C(=O)(CC(C)CN(C)C)NCCC1N(C(C(C2CCOC2)OC)=O)CCC1 Cc1ncc(CC(=O)N(CCN(C)C(C2(C3CC3)CC2)=O)C(C)C)o1 c1(OC)ncc(C(N2CC(O)(CCNC(c3ccns3)=O)C2)=O)cn1 C(=O)(CCCC(C)(C)CC)NC(CCCC)CNC(c1cc(Br)no1)=O C1(NC(c2cnc(C)n2C)=O)CCC(C)N(C(c2cc(C(N)=O)cc(F)c2)=O)C1 N1(C(C2C(C)CCS2)=O)C2CCC1CN(C(C1(c3ccsc3)CC1)=O)C2 C(=O)(CC1OCc2cc(Cl)ccc21)N1CCCC(CC)(NC(c2cnsc2)=O)C1 c1(C(N(CCCNC(C(C=CC)O)=O)Cc2cccnc2)=O)ccncc1O N1(C(C(C)OCCOCC)=O)C(C(=O)NC2(C(O)CO)CC2)CCC1C1CC1 C1(NC(Cc2ccc(C)[nH]2)=O)CCCN(C(c2cn(C(C)C)nc2C2CC2)=O)CC1 N1(C(C(C=C)(C)CCOC)=O)CCCC2(CCCN2C(=O)Cc2coc(C)n2)C1 c1(C(N2CC(O)(C(C)NC(C3CN(C)C(=O)N3)=O)C2)=O)ccc2cn(C)nc2c1 c1(C(=O)NC2C(C)CCN(C(c3c(C)ccnc3O)=O)C2)cccc2ccnn12 n1(CC(N2CC(CCC=C)(C(=O)NCCC3CCCOC3)C2)=O)nc(C)nc1C C1(COC)CN(C(c2ccc(Cl)nc2N)=O)CCN1C(C1CNC(=O)N1)=O CC(C)C(F)(F)CC(=O)N1CC2CCC1C2NC(=O)C=CCN1CCCC1 N1(C(C2(CC#C)CCOC2)=O)CCC(CNC(=O)Cn2ccnn2)C(F)(F)CC1 C1(NC(CCCN(C(=O)OCC)C)=O)CC2CCC(C1)N2C(=O)CCCC(C)C CCC(C)CC(=O)NCCOC1CCN(C(=O)C(C)CC2CCCCC2)CC1 n1(C(C)CNC(=O)C(C)n2ccnc2)cc(CC2CCOCC2)nn1 CC(C)C(C)CC(=O)N1CCC(NC(=O)CCC(=O)c2ccc[nH]2)CC1C C1(C(=O)NCC(C)CO)CCCCN1C(=O)CN(C)C=O.c1(N)ccccc1 CN1CCN(C(c2coc(C#N)c2)=O)C(CNC(c2n[nH]cc2Br)=O)C1 c1(C(N2CCC(NC(c3nc(C)c(C)s3)=O)CC2)=O)cnc2n1CCS2 C1(CNC(C2(CC)CC2)=O)C(C2CC2)CCN1C(c1cc(Cl)ns1)=O CC(C)CC(=O)C(=O)N(C1CCN(C(=O)C(C)C2CCCO2)CC1)C N1(C(C(C)SCC)=O)CC(C(=O)N(C)CCN(C)CCO)C(C)(C)C1 c1(C(N2CCOC(CCO)C2)C(=O)NCCC)ccc2ccc(Br)cc2c1 C(S(=O)(=O)C(F)F)C1N(C(C2(n3cc(CN)nn3)CC2)=O)CC1.N#CCCCN n1(CCCC)ncc(NC(=O)C(C2CCN(C(=O)CC3CCC3)CC2)C)c1CC N1(C(C2C(C)N(C(=O)COCCCN(C)C)CC2)=O)CCC2(CC(N(C)C)C2)C1 C(C)(CSC)(C(=O)NCCSC)NC(c1n(CC)ccc1)=O CC(CCCc1ccccc1)C(=O)N1CC(NC(C2CC=CC2)=O)C(C(F)F)C1 C=C=CCC(=O)N1CCC(C(F)C(=O)N(C)CC2(O)CCC2)C1 c1(C(=O)NC2CN(C(C3C(C=C)OCC3)=O)C(C)C2)ccc(C2CC2)cc1C C1(CNC(C(C(C)C)OC)=O)CN(C(=O)CN(C)Cc2ccccc2)C(C)(C)C1 CCC(C)(C#N)C(=O)NC(CNC(c1cc(O)cc(F)c1)=O)C(C)(C)C N1(C(C2(CC)COC2)=O)CCC2(CC1)CN(C(=O)CC1CCCN1CC)CCO2 c1(C(N2CCCC(CNC(C3C(C)CC(C)O3)=O)C2)=O)cnn2c1C(=O)NCC2 CCCCCC(O)CC(=O)NCCN1CCN(C(C2(C)CC2C(F)(F)F)=O)CC1 CC(=O)CC(C)C(=O)NC1CC2CC1CN2C(=O)CSc1ccccn1 C(c1cn(C)nn1)=CC(=O)NCC1(NC(Cc2c(C)ocn2)=O)CC1 C1(C(C)NCCCC(=O)NCc2cscn2)CCCN(C(c2ccco2)=O)C1 N#CC1CCCC(C(=O)NCCCCCCNC(=O)Cc2ccc(CO)cc2)C1 C12(C(N3CC(NC(CN4CCC(C)C4)=O)C3)=O)CC3CC(C)(C1)CC(C)(C3)C2 C(CC(F)F)(C(=O)NCCCCCC1CC1)NC(c1c[nH]c(=N)o1)=O C1(C)(CNC(C2(C(=O)NC)CC2)=O)CCN(C(=O)C#CC(=O)N(C)C)CC1 C1(n2cc(OC(C3CCCOC3)OC)nn2)CN(C(c2cn(C)nn2)=O)CC1C c1(C(N2CC(n3cc(C(=O)N(C)C)nn3)C2)C)nnc2ccccn12 S(=O)(=O)(c1c(Br)cc(F)c(Cl)c1F)SCC(CC)N(CC(=O)O)C c1(OC)cccc2c1OCC(C(=O)N1CC=CC(NC(=O)C(F)C(F)(F)F)C1)=C2 N1(C(c2n[nH]c(C)c2C)=O)CCC(C2CC2)C1CNC(C1CCC(C)CC1)=O C1(NC(CC2(C)CC2)=O)CCCC2CN(C(=O)C=Cc3ccc(Cl)cc3)CC12 O=C1CCC(CNC(=O)CN2CCC(n3ccnc3)C2)C1 C(=O)(C1CCCc2nn[nH]c21)NC1CC(NC(c2c(CC)nns2)=O)C1 c1(C(=O)NCC(CC)NC(c2nn(C)cc2Cl)=O)c(Cl)n[nH]c1C1CC1 c1(C(=O)Nc2cccc(C)c2Cl)[nH]c2ccccc2c1-c1ccc(C#N)c(O)c1 C1(C(=O)NCCOCC(=O)NC)C(C)OCCN1C(C1CC2(C1)CC21CC1)=O C(=O)(C(=O)C(C)(C)CC)N1CC(CCC=C)(C(=O)NC2CCCN(C)C2)C1 N1(C(CCC)C(=O)NCc2cccc3ccccc23)Cc2ccccc2CCC1C N1(C(c2n(CCC)nc(C)c2)=O)CCC2(CCCN2C(c2cccc(=O)o2)=O)C1 c1(COC)nccc(=NCCC(C)NC(=O)C(C(C)C)NS(C)(=O)=O)[nH]1 C1(C(C(=O)NCCCCNC(=O)C(C)c2ccco2)OCC)CC(F)(F)C1 C1(C(N(CCN(C(c2c[nH]nc2C(C)(C)C)=O)CC)CC)=O)CNC(=O)N1 N1(CC(N2CCCC(C)C2CNC(c2occc2Cl)=O)=O)CCc2ccccc21 c1(C(N2C(C)C(C)CCC2)=O)cc2oc(Br)cc2[nH]1 c1(CC(=O)NCC(C)NC(=O)C(c2cccc(F)c2)O)c[nH]c2cnc(Cl)cc12 c1(OCC(=O)OC)cccc(C(=O)NC2(OC)CCN(C(=O)CCOC(C)C)C2)c1 CCCC(C(=O)NC(C(=O)NCCC1CCOC1(C)C)C(C)CC)C(C)C C1(O)(C(=O)NCCF)CCN(C(c2ccc(-c3ccccc3)cc2)=O)C1 c1(CCC)sc(C(N2CCOC(CNC(=O)CCc3cccs3)C2)=O)cc1CC c1(C(C(N2CC(CNC(C(C)CO)=O)C2)=O)C)cccc(Br)c1 c1(C(N2C(C(=O)NCc3ccccc3F)CC(=O)C2)=O)cnn2c1OCC2 CC(C)CC(CNC(C1(c2cc[nH]n2)CCC1)=O)NC(C1CC(F)C1)=O C(=O)(C(F)(F)C1=CCOCC1)N1CCC(NC(C(CCC)OC)=O)C(CC)C1 C(C(C(C)C)C(C)C)OC(C1C(C(=O)OC)C1)=O C12(C(=O)NCC3(CNC(=O)Cn4cc(Cl)cn4)CCC3)CCCCC1OCC2 CCCC(O)CC(=O)NCC1CCCCCN1C(c1cnn(C(C)C)c1N)=O c1(C(N2CC(NC(c3c(C)cnnc3)=O)C(O)C2)=O)ccc2c(c1)NC(=O)C2 C1(CC)(NC(c2c[nH]c(=NC)s2)=O)CCN(C(=O)CC(C)COC)CC1 C(C1OCCc2sc(F)cc21)NC(=NCC)NCC1CCN1CC N1(C(C(CO)N(C)C)=O)CC(CNC(C2CC(=O)CCO2)=O)C(C)(C)C1 CC(C)C(C(=O)NCc1nnnn1C)C(C)NC(=O)C(=O)C(C)(C)C Cc1cc(C)c(S(=O)(=O)Nc2ncc(CCNc3ncco3)s2)c(C)c1 C1(C(=O)NC(CN(CCCC)C)C)(NC(c2ccns2)=O)CCCCC1 c1(C(=O)NC(C2CC(NC(C(C)OCCCC)=O)C2)C)cccc2c1OCC2 N1(Cc2ccnc(SC)n2)CCCC2(CCCN(C(c3ccncn3)=O)C2)C1 N1(C(C(CC(C)C)C)=O)CCCCC12CC(NC(c1cncn1C)=O)C2 c1(C(N2CC(CC)C(NC(c3scnc3C)=O)CC2)=O)cc2cnn(C)c2s1 C(=O)(CCCn1cncn1)N(CCC(C)NC(C1(NC(C)=O)CCC1)=O)CC Cc1ccc(Cl)c(C(=O)N(C2CCCCN(C(=O)C#CC3(C)CC3)C2)C)c1 N1(C(C(c2cccc(C)n2)(F)F)=O)CCCCC(CNC(=O)CCC(C)C)CC1 C1(NC(=O)NCCCNC)CN(C(c2ccc(OC)nc2)=O)CC1C(F)F N1(C(Cc2cc(C)nn2C)=O)CC2CCC1C1CN(C(=O)C=CBr)CC21 N1(C(CC(=O)OCC)=O)CCCCC(C(=O)Nc2cc(Cl)ccc2OCC)C1 C(c1ccc(F)cc1)=CC(=O)NCCCC(C)NC(c1ccn(C(C)(C)C)c1)=O c1(C(=O)OCC)cn(C)[nH]c1=NC(=O)N1CCC(c2nc(=O)o[nH]2)CC1 C1(C(N(CCCN(C)C(c2csc(C(F)F)n2)=O)C)=O)CCCCS1 c1(C(N2CC(CCCCNC(C(C=CC)O)=O)C2)=O)cc2n(c1)CCCNC2=O C=CCC(C(=O)OCC)NC(=O)C(O)C1CCC1.C(C)(C)(C)O N1(C(C=CC(C)C)=O)CCC2(NC(c3cc(Cl)c(Br)[nH]3)=O)CC2C1 c1(NC(C(N2CC(Br)=C(C)CC2)=O)=O)cnc2c(c1)C(=O)NCC2.C1(=O)CO1 c1(C(N(CC(C)(C)C)CCOC)=O)ccc(Cl)c2c1OCCO2 C1(NC(C=CCN(C)CC)=O)CCCC12CCN(C(=O)C(C)C(F)F)CC2 c1(OC)ccc(C(c2nnnn2C2CCC2)NC23CC(F)(C2)C3)cn1 C1(C(=O)NCCC(F)(F)F)CCC2CCC1N2C(c1ccsn1)=O C1(NC(c2snnc2C2CC2)=O)COCCN(C(C23CCCCC2C3)=O)C1 C1(NC(N(Cc2cn(C(C)C(=O)O)nn2)O)=O)CC2CC3CC(C2)CC1C3 c1(N2C(C(=O)Nc3ccc(C)nc3I)C=CC2)nc(C)c2cc(Br)ccc2n1 Cc1ccc(C(N2CCC2CC(=O)Nc2c[nH]ccc2=O)=O)nc1 C(=O)(CC1COc2ccccc21)NCCC1(NC(c2c(C)cnn2C)=O)CCC1 C=C(C)C(CC(=O)NC1CCCC(NC(=O)C=C2CCCCC2(C)C)C1)OCC C(=O)(C1OCCc2ccccc21)NCCC(C)NC(C1CC2CC1C1CC21)=O C(=O)(C(C)CCOC)NC(C(CO)NC(c1c(CC)ncs1)=O)C c1(C(N2CCCC(NC(C3(C)CCC34CCC4)=O)C2)=O)ncc2ccccn12 C1(C(=O)N(C)CC2CCOC2)(CC)CCCN(C(=O)CC2CCC2C)C1 C(=O)(C(C(C)(F)F)c1ccccc1)N1C(C(C)C)C(NC(=O)CCC(N)=O)CC1 C1(C(N2CC(C(C(=O)O)OC)C2)=O)CCC(=O)N(C)C1 C#CC1CC2CCC1N(C(c1cc(-c3ccco3)on1)C(=O)NC(C)(C)CC)C2 N1(C(c2ccc(C#C)cc2)=O)CC2CCN(C(=O)CCCn3cc(C)cn3)C2C1 NC1c2ccccc2CC12CCN(Cc1cc(Cl)cc(Br)c1)CC2 C=Cn1nccc1C(=O)NCC(F)CNC(=O)C=Cc1ccc(Br)s1 C1(C)(COC)CCCN(C(=O)CC(C)(C)N(C)C(c2ncc(F)cc2N)=O)C1 c1(OC)cc(C(=O)NC2CCN(C(C34CCC3CC4)=O)CC2C)c(F)c(Cl)c1 N1(C(CC2ON=C(CC)C2)=O)CCC2(CC2C(=O)Nc2cccc(Cl)c2O)C1 c1(C(=O)NCC(C2CCN(C(C(CCCC)O)=O)CC2)C)cc2cccn2cn1 C(=O)(CC(CNC=O)CC(C)C)N1CC(CNC(C)=O)(Oc2ccc(Cl)cc2)C1 CC(C)C(O)C(C)C(=O)N1CCCC(C)(C)C1C(=O)NCC(Cl)=CCl N1(C(C(Cc2ccoc2)NC(CC2COCC(C)O2)=O)=O)CCC(F)(CO)CC1 CC(CCC(C)(C)C)C(=O)NCC1CCN1C(c1ccc2c(c1O)CCC2)=O C1(CNC(Cc2cn(C)nc2)=O)CCN(C(c2ccnc(CO)n2)=O)CC1(F)F N1(C(=O)CCCN2CCOC2=O)CC(C2CN(C(=O)CC3COCC3O)C2)C1 c1(CC(=O)NCCN(C(c2csc(Cl)c2)=O)C2CC2)coc2ccccc12 CCC(CC)C(=O)NC1CC1NC(c1nc(C)n(-c2nc[nH]n2)n1)=O c1(C(=O)NC2CCCN(C(=O)Cn3ccnn3)CC2)cc(Cl)cc2c1CCC2 C1(NC(=O)CC2COCC2O)CCOCC1NC(c1cscc1C1CC1)=O CC1=C(C(=O)N2CCC(C(=O)NC3CCN(C)CC3C)CC2)SCCO1 CC(C)C(C)C(CNC(c1cnnn1C1CC1)=O)NC(c1cn2c(n1)SCC2)=O CCN=c1ccc(C(N2CC(NC(=O)C=Cc3nccs3)CC(C)C2)=O)c[nH]1 C(=O)(CCCC(=O)N1CCCC1CN(C(=O)CN1CCS(=O)CC1)CC)NCC c1(CC)ccc(F)c(C(=O)NC2CC(CCNC(=O)CC=C(C)C)C2)c1F c1(OC)cc(O)ncc1C(=O)NC1CCC(C)N(C(c2ccnc(O)c2F)=O)C1 N1(C(c2ccc(C)nn2)=O)CCOCC(C(N2CCC(O)CC2C)=O)C1 CC1(C#N)CCN(C(C2(CNCc3ccccc3)CCCOC2)=O)C1 c1(CC(=O)NCC(CNC(c2ccc(OC)c(O)c2)=O)C)ccn2cncc2c1 N1(C(c2cc(C(C)C)on2)=O)CCC2(C1)CN(C(c1cnncc1O)=O)CCO2 C1(NC(c2c[nH]c(=N)s2)=O)CCCOC1C1CCN(C(=O)COCCCF)CC1 N1(c2c(C)cncn2)CC2CC(NC(=O)C(C)C3CCOC3)CC1C2 c1(CC(=O)N(CCC)CCNC(C2CC2(C)C(C)C)=O)ccc(OC)cn1 C1(OC)CCC1C(=O)NCC1CC1NC(=O)CNC(c1ccco1)=O n1(CC)ncc(C(N2CCCC(CN(C(=O)C(c3cncnc3)C)C)C2)=O)c1Cl CC1CCC(CC(=O)NCC2(CNC(c3cnc(C4CCC4)s3)=O)CCCC2)O1 CC(C)(C)CC(O)C(=O)NC(C)(C)CC=CC(N1CCCC(C)(O)CC1)=O CCC(CC)C(C(=O)NC1CC(F)CN(Cc2conc2C)C1)N1CCOCC1 C1(C(=O)NC2CC(CNC(C(CCSC)N(C)C)=O)C2)CCc2nncn2CC1 c1(OC)cc(O)ncc1C(N1CCC(CF)(NC(C2CN(CC)CCO2)=O)C1)=O C=CCC(CC)C(=O)NCCOC1CCN(C(=O)Cc2cc(C)sc2C)C1 c1(OCC)cc(C(N2CC(NC(=O)Cn3c(C)csc3=O)C(O)C2)=O)ccn1 c1(C(=O)NCC2CN(C(CC(C)C)=O)CC23CC3)occ2c1CCOC2 CCC(CCCC(=O)N(CC(C)(F)F)C)NC(c1cc(CO)n(C)n1)=O CC1(C)OC(C)(C)C1C(=O)NC1CC1NC(c1cnoc1-c1ccoc1)=O c1(SCC)ccc(Cl)cc1C(=O)NCCCNC(c1cc(C#N)no1)=O C1(CC(=O)NC(C)CCNC(c2cnn(-c3ccccc3)n2)=O)CC(C2CC2)C1 C1(F)(C(=O)NCC(C)(C2CC2)NC(c2csc(=N)[nH]2)=O)CCC(F)(F)CC1 C1(C)(C(=O)Nc2cccc(NC(C#CC(C)(C)C)=O)c2)CCCNS1(=O)=O C1(C(C)NC(=O)CCN2CCOC2=O)CCCN(C(c2cnoc2C(C)C)=O)C1 Cc1ccc(Br)c(CC(=O)OCC2CCC(=O)NC2)c1 C(=O)(CC(=O)N1CCCC1C(C)(C)NC(C1CNC(=O)N1)=O)OC c1(C(=O)NCCCCCNC(CSC(C)C)=O)ccc(C2CCCO2)cc1 C(=O)(CCCC(C)(C)C#N)NC1(C(N(CCCCC=C)C)=O)CC1C c1(C(=O)NCC(CC)NC(C2CCCC23CC3)=O)cc2cc(C)ccc2nc1C CCC(O)(CC)CCNC(C1CCCN(C(C2(O)CCCCCC2)=O)CC1)=O C1(C(N(CC(CN(C(CCNC(=O)OCC)=O)C)O)C)=O)CCCC(C)CC1 c1(OC)ccc([N+](=O)[O-])cc1C(=O)OCCN(S(C)(=O)=O)C C1(NC(C2CCCCC2(F)F)=O)CC2CCC(C1)N2S(=O)(=O)c1cccs1 N1(C(c2c(N)nccn2)=O)CCN(C(=O)CN2C(=O)CCC2=O)C(C2CCC2)C1 N1(c2c(C)c(O)ncn2)CCC2CCC(C1)N2C(C(C)(C)C)=O C12(C(=O)NC3CN(Cc4n(C)cnc4)CC3(C)C)CC3CC(CC(C3)C1)C2 C1(NC(CCSCCCC)=O)CC1C1CCCN(C(C2(CC)CCCC2)=O)C1 c1(C(CNC(CC2(C#N)CC2)=O)NC(C2CC2(F)F)=O)cc(F)cc(Cl)c1 S(=O)(=O)(c1ccc(F)cc1Cl)NC1CCC(NC(c2ccc(C)c(Br)c2)=O)C1 c1(C(=O)NCC(C)CN(C(=O)C(C)C#N)C)cccc2scnc12 Cc1c(CC(=O)NOCCCCC(=O)NC2CCC2)cnn1C C(=O)(CCN1C(=O)CCc2ccccc21)NCC(C)NC(C1CCCCC1)=O Cc1ncc2ccccc2c1C(=O)NC1CC(C)CN(C(C2(C#N)CCC2)=O)C1 Cc1ccc(C)c2c(C)c(C(=O)NC3CCCC(C)C3)oc12 c1(CN2CCCC(C(N(C)CC3(OC)CC3)=O)C2)ccc(O)c(OC(F)(F)F)c1 c1(C(=O)NCC2C(NC(CN(CCCCCC)C)=O)C2)c(Cl)ccc(F)c1C N1(C(C(C#C)(C)C)=O)CC2(C1)OC1(C)CC2(NC(c2ccn3ncnc3c2)=O)C1 c1(C(=O)NC(C)(CNC(=O)CCc2cnc(O)[nH]2)CO)cnc2[nH]cnc2c1 Cc1cc(C(=O)N(C)CC2(CNC(C3CC4CC4C3)=O)CC2)c2c(c1)CCO2 C#CCC(CC)NC(=O)C(C1(O)CN(C(=O)C(C)n2ccnn2)C1)F c1(C(=O)NC(CCNC(C(CC)F)=O)C(C)C)ccc2nc(N(C)C)sc2c1 C(=O)(CC(C)C(=O)NCCCCC(N1CC(=O)NCC1C(N)=O)=O)OC Cc1cn(CC(=O)NC2CCC2NC(C2CCc3nncn3C2)=O)c(=O)nc1O C(=O)(CC(C)(O)C(F)(F)F)N1CCC(N(C(c2cnc(C(C)(C)C)o2)=O)CC)C1 CC1CCC(C2CCC2)CN1C(=O)C(=O)Nc1ccc(S(C)=O)cc1 C1(CNC(C(C)C2CC2)=O)CCN(C(=O)C=Cc2cccc(F)c2)C12CCC2 C1(CNC(C2CCN(C(C)C)CC2)=O)CC2(CCO1)CC(F)(F)C2 N1(C(CC(=C)C)=O)CCC(c2ccccc2)C(NC(C2(CO)CCCO2)=O)C1 N1(C(C(CNC(=O)CC2CCC=CCC2)N(C)C)=O)CCC(C)(C2CC2)C1 c1(OC)cccc2c1OCC(C(=O)NCCCCCNC(=O)CC(C)OC)C2 C1(CC#C)CCNCC1.c1(OCCN(C=O)C)ccccc1C(C)C c1(C(N2C(CNC(c3c(C)nc[nH]3)=O)CC2)=O)cnn(CC(C)C)c1C N1(C(C2CCC(CC)C2)=O)CCN(CCCNC(c2cccc(CF)c2)=O)CC1 CCS(=O)c1ccccc1C(=O)NCC1CC(F)CN1C(=O)CN1CC2CC2C1 c1(C(N2CCCC(F)(CNC(C(CC)OC)=O)C2)=O)cc2cc(F)ccc2cn1 C1(C)(C(=O)NCC(CC=C)NC(C2CC(O)(CC#C)C2)=O)CCC(=O)N(C)C1 C(CCCCCNC(=O)COC1CCCCC1C)N(C(c1c(C)occ1)=O)C c1(C(=O)NCC2N(C(c3c(C)nc(C)[nH]3)=O)CCCC2)cc(Cl)n[nH]c1=N CC(Cc1cccs1)N=c1[nH]c(=N)[nH]c(=NC2CCC(S(C)(=O)=O)CC2)[nH]1 C1(CNS(CC(=O)OC)(=O)=O)CN(C(C2(c3cccs3)CC2)=O)CC1(C)C N1(C(C(C(C)O)C)=O)CC2CC(NC(c3cc4n(n3)CCO4)=O)C2C1 CC#CCCC(=O)N(CC(=O)N(C)CC1CCCS1)C(C)C Cc1[nH]c2c(C(N3CC4C(C3)N4c3ncnc4ccccc34)=O)cccc2c1C N1(C(C(C)OCCOCC)=O)CC2(CC(NC(c3coc(C)n3)=O)C2)C1 CC(O)CC(C)(C)CNC(c1ccc(CNC(C2COCC2C(N)=O)=O)s1)=O C1(O)(CNC(CN(CC)CC)=O)CCN(C(=O)Cn2cccc(N)c2=O)CC1 C(=O)(CCS(C)=O)NCC(C(C)C)NC(c1n(CC)ncn1)=O Cc1coc(C(=O)NC(C)CCN(C(=O)CSCc2ccccn2)C)c1C N1(C(CN(C)C)=O)CC2OCCN(C(c3cc4cccc(F)c4o3)=O)C2C1 Cc1cc(C(N2CC(NC(c3cnnn3C3CC3)=O)CC(C)C2)=O)c(F)cc1Cl c1(NC(C2(CNC(C(C(COC)C)C)=O)CC(C)(C)C2)=O)cncc([N+](=O)[O-])c1 c1(OC)ccccc1NC(C1CN(C(=O)C(F)F)CCO1)=O N1(C(c2cc(C)nc(O)c2)=O)CC2(CCN(C(c3ccoc3Br)=O)CC2)C1 N1(C(CCNC(=O)CO)=O)CC=CC1C(=O)NCC1(F)CCC1 C12(NC(CCCCOC)=O)CCN(C(=O)C(=Cc3cscn3)F)CC1C2 c1(C(=O)NC2C(C(=O)NCC3(OCC)CC3)CCC2)cc(COC)nn1C N1(C(c2nc(CN3CCOCC3)cs2)=O)CCC(c2cccc(F)c2)CC1 CC1=NOC2(C1)CC(C(=O)NC1CCN(C(C3CCC(=O)O3)=O)C1C)C2 C1(NC(c2cnc(C#N)s2)=O)CS(=O)(=O)CC1NC(=O)C(F)(F)C1CCCC1 c1(COC)nc(NCc2ccoc2C)cc(N(C)CCc2nccs2)n1 c1(CCC(=O)N(CC(C)NC(C2(C)CC2C(F)(F)F)=O)C)cc(F)ccc1F C(CC(C)(CC)NC(C1CC12CCCC2)=O)NC(COCCC)=O C1(F)(CNC(=O)CC2(c3ccon3)CC2)CC(CNC(=O)Cn2cnnn2)C1 C#Cc1cc(C(=O)N(C2CCN(C(=O)C=COCC)C2)C)ccc1C Cc1ccc(Cl)cc1C(=O)NC1CCCC1CN(C)C(c1sccc1C(C)C)=O C(C(CC(=O)NCC1C=CCN1C(c1cc[nH]n1)=O)C(F)(F)F)N(C)C C(=O)(C(C)(COC)CC)NC(CNC(c1nc(COCC)sc1)=O)C(C)C C12CCC(CC1)NC2=O.c1(NC(C2(CC(C)=O)CC2)=O)cncnc1O C1(NC(c2cnns2)=O)CC(F)CN(C(C2CCS(=O)(=O)N2)=O)C1 C1(C(N2C(CNC(=O)CC(=O)NC3CC3)C=CC2)=O)CC(=O)N(C2CCCC2)C1 C(=O)(CS(=O)(=O)C1CC1)N1CC(CNC(c2ccn(CCF)n2)=O)C2(C1)CC2 C1(NC(CN(C)C(C2CC(=O)OC2(C)C)=O)=O)CCC(=O)NC1=O C1(C(=O)NC(CNC(COCC#C)=O)CC)CCC2(CC1)OCCO2 CS(=O)(=O)C1CCCCN(C(=NCC2CC2)NCc2ccn(CCF)n2)C1 c1(N2CC(CC)(CC)OCC2)nc(N2CC3CC(C2)N(C)C3)c2ncn(C)c2n1 N1(C(=O)CC2CCCN2C(c2cc(CO)[nH]n2)=O)CCC(O)C1C(C)(C)C C1(N(C(=O)CCCC)CCNS(=O)(=O)N(C)C)CCCN(C(=O)NC(C)=O)C1 C1(N(C(CSCCOC)=O)CCO)CCN(C(C2(C)CC=CC2)=O)C1 N12CCCc3cc(ccc31)C2.C(=O)(CCCC(F)(F)CO)N(CC)CC c1(C2(C(=O)NC(C3CN(C(=O)CC4CC4)CCO3)C)CC2)c(Cl)cccc1Cl C1(C)(C(=O)NC(C)CN(C(=O)CNC(=O)OC(C)(C)C)C)CCC(=O)C1 c1(OC)ccc(C(=O)NC2(CO)CN(C(=O)C=C(Cl)Cl)C2)cc1Cl C1(CC)C(C(N2CCC=CC2COC)=O)CCN1C(=O)C=C(C)COC c1(C(C)(C)C)cccc(C(=O)NC2CCC(NC(C3C4(CC4)C34CC4)=O)CC2)c1 c1(C(=O)NC2CC(C(=O)NC(C)C(N)=O)C2)ccccc1Cl C=C(CNC(c1cnoc1-c1cccs1)=O)CCNC(C1(CC)CCOC1)=O c1(COC2CCN(C)CC2)cnn2c1CN(C(=O)C(Cl)=CCl)CC2 C1(C(N(C(C)CCNC(=O)CCC(=O)c2ccncc2)C)=O)CCCCC1(C)C CCC(C)C(CC(=O)N1CCC12CC(O)C2)NC(=O)CC1CCCO1 c1(OC)c(C)ccc(NC(c2csc(N3CCCCC3)n2)=O)c1C N1(C(Cc2cccc(OC)c2)=O)CCOCC(NC(C2(C)CCC(=O)C2)=O)C1 C1(NC(CCSCCC)=O)CCC(C)N(C(=O)CCOCC(F)(F)C(F)F)C1 C(=O)(C(CO)C(F)(F)F)N1C(C2(NC(CC3(OC)CCC3)=O)CC2)CCCC1 N1(C(c2c(C)c[nH]c2)=O)CCS(=O)(=O)C(CCNC(=O)CCOC2CC2)C1 Cc1cc(C(=O)NCC2(F)CCCN(C(c3cnc[nH]c3=N)=O)C2)nc(O)n1 Cc1c(F)ccc(C(=O)NC2CC(CC(=O)Nc3cc(Br)cnc3O)C2)c1F c1(OC)cccc(C(N2CC3CC(NC(c4cc(O)cc(F)c4)=O)C2C3)=O)c1N C(=O)(CC(O)CC(C)C)N1CCC(C(=O)NC(c2nn[nH]n2)CC)(CC)C1 C1(C(=O)OCC)NC(=O)N(c2cccc(NC(=O)C(=O)N(C)CCOC)c2)C1=O C(=O)(C1CCCc2nn[nH]c21)NCCOCCNC(c1cnn2ccn(C)c21)=O C1(O)(C(C)NC(=O)CCN2CCCC2)CCN(C(=O)CSc2ccccc2O)C1 N1(C(c2ccc(=N)[nH]n2)=O)CCC(NC(=O)COCC2CCOCC2)C(F)C1 C(=O)(C(CC(C)(C)C)NC(=O)C(C)NC(=O)C1CC1)N1CC(N(OC)C)C1 C1(N(C(N2CC(c3c(C)nccn3)C2)=O)CC2CC2)CC2CC(N(C)C)C1C2 Cc1ccc2c(C(=O)NCC3CC4CCC3N4C(C3CC3(C)Br)=O)coc2c1 CC(CC(=O)NCCC1CN(C(c2n[nH]c3c2CC(C)CC3)=O)C1)CC(F)(F)F C(C(C)(C)CC(=O)NCCN1CCNC(=O)C1)NC(COCC=C)=O N1(C(C2CCCN(C)C2)=O)CCC2(CCCN(C(=O)CCCCBr)C2)C1 C1(NC(=O)Cc2nc3c([nH]2)CCCC3)CCN(C(c2cnco2)=O)CCC1CO C(C(N=[N+]=[N-])C(=O)NCC1CC(NC(C2CNC(=O)O2)=O)C1)OCC c1(C(N2CC(CNC(c3cccc(C#C)c3F)=O)C2)=O)c(F)c(F)cc(F)c1F CC(=O)C(C)(C)CC(=O)NC(C1CCCCC1)C(=O)NCC=CC1CC1 c1(NC(C2(N(C)C(c3ccccc3F)=O)CC2)=O)ccc2c(c1)OCC2 Nc1cc(C(=O)NC2CCN(C(C3(C4CC4)CCC3)=O)C2)cc(Cl)n1 Cc1cc(C(=O)NCC2(C3CC3)CC2)ccc1C#N.C12CCCC1NC2=O C(C(CC(=O)N1CCCCC1CNC(=O)CC(C)(C)C#N)C(F)F)N(C)C1CC1 C(C(=O)NC(C)(CNC(=O)C(C)=C1CC1)C1CC1)(C(C)C)SCC Cc1nc2ccccc2nc1NC(C1C=CC(NCc2cccs2)C1)=O N1(C(c2ncc(C)cc2C)=O)CCCC2(CCCN2C(=O)CC2CCC2(C)C)C1 n1(CC(=O)NCCN(C(=O)CC23CCCC2C3)C(C)C)c(O)nnc1O [N-]=[N+]=NC1CCCCC1CC1CCN(C(N2CC(CCC(=O)CCO)C2)=O)CC1 N1(C(C=CC(=O)OCC)=O)CCCC(C(=O)NC2C=C(C)CCC2)C1CC Cc1cnn(C(C)C(=O)N2CC(CNC(=O)C(F)(F)c3cscn3)C2)c1 N1(C(c2n(C)cc(C#N)c2)=O)CCC(C2(NC(=O)CC=C(Cl)Cl)CC2)C1 C12(NC(c3ccn(CCCC)n3)=O)CCCC1(F)CN(C(=O)C(C)CN(C)C)C2 c1(OCCC(=O)NCCCC2CN(C(=O)CCF)CCO2)ccc(F)cc1F c1(OC)cc(C(=O)NCC2CC(O)CN2C(=O)CC2CCCO2)c(C)cc1O c1(NC(C2CC(O)CN2S(=O)(=O)CC2CC2)=O)cc(Cl)c(Br)c(Cl)c1 c1(N2CCC(CCOC)(NC(=O)CNC(N)=O)CC2)ncnc(C)c1C#N CCC1=NOC(CC(=O)NC(C)(C)C(C)NC(c2ccncc2OC)=O)C1 CCCC(CC)C(=O)NC1(CNC(c2sc(Cl)cc2Cl)=O)CCCCC1 N1(C(CCCC(C)O)=O)CCCCC(C2CN(C(=O)CC3CC3(Cl)Cl)C2)C1 Cc1cc(F)c(CC(=O)Nc2cccc(NC(=O)C3=CCCS3)c2)cc1F c1(C(=O)NCC2C(C)CCN(C(=O)CNC(=O)C3CC3)C2)cn2ccncc2n1 C=CCC(C)(C(=O)NCC(C1CC1)NC(=O)CCC(C)OC)N(C)C N1(C(c2cc(OCC)n[nH]2)=O)CC(=O)CCC1C(N1CCCCC1CF)=O c1(COC(CC2(CC=C)CC2)=O)c(CC(C)C)n(C)c2c(C)cccc12 C1(NC(CN2CCC(C)CC2)=O)CCC12CCN(C(C1CCS(=O)CC1)=O)CC2 CCCCC(O)C(=O)Nc1ccc(C(C)NC(c2csc(CC)n2)=O)cc1 C(c1cncn1C)=CC(=O)N(C(C)C(N1CCC(N2CCCC2)C1)=O)C1CC1 CCCCCC(F)C(=O)NCc1cc(C(=O)NCC2(C(=O)OC)CC2)n[nH]1 n1(C(C)C)ncc(Br)c1C(=O)NC1CC(F)(CNC(=O)CC2CC23CC3)C1 C1(C(=O)NCCC(C)(O)C2CC2)C2CN(C(=O)CC3CCOC3=O)CC12 O=C(N=c1ccc(C2CCOC2)n[nH]1)NC1CCCC(N2CCOCC2)C1 c1(C(=O)NC2COCCN(c3ncnc(CC)c3F)C2)ccc2nsnc2c1 Cc1cc(C(N2CC(NC(c3c(Cl)cnn3C)=O)C(CC(C)(C)C)C2)=O)sc1C c1(NC2CCCN(C(C(c3n(C)ncc3)O)=O)C2)ccc(C#N)cc1[N+](=O)[O-] Cn1cc(C(=O)NCC23CC2CN(C(=O)COc2ccc(Cl)cc2)C3)ncc1=O N1(C(CCNC(=O)OCC)=O)CCC2(CNC(c3cnn[nH]3)=O)CCCCC12 c1(OCCCOC)ccccc1-c1nc(-c2ccc(OC)nc2)no1 C(=O)(CCCC(C)(C)C)N(CC(=O)NC1(CC2CCC2)CC1)C CCCC(C)(C)C(=O)N1CCN(CC(=O)Nc2cc(C(F)(F)F)cc(Cl)c2)CC1 c1(NC(C2COCC2C(=O)O)=O)ccc(NC(C2CCCO2)=O)cc1 c1(C(C)=O)ccccc1C(N1CCC(NC(C2(C)C=CCCC2)=O)C1)=O Cn1nc(C(=O)NC2CCCCC2CNC(=O)COC2CC2)c2c1CCCC2O C1(C(=O)NC2C=CCC(C(=O)NCc3n(C)cnn3)C2)CC2CC(=O)C1O2 C1(NC(CCOCC#C)=O)CCOCC1C(=O)NCCc1ccccc1C Cc1nc2cccc(C(N3CC(C(F)Cn4cc(C5CCCO5)nn4)C3)=O)n2n1 C1(F)(CNC(C(C)NC(CC)=O)=O)CCN(C(c2ccccc2C(=O)OC)=O)C1 c1(C(=O)NCC2C(NC(CC3C(C)C3)=O)CCCC2)cnc2ccccn12 c1(CC(N2CC(O)CC(NC(C3(N(C)C)CC3)=O)C2)=O)ccc2cccnc2c1 CC1CC(=O)NC1C(N1CCC(NC(c2cc(-c3ccn(C)n3)on2)=O)CC1)=O c1(C(N2C(C=CCC(=O)NCCSC)CCC2)=O)ccc2[nH]ccc2c1 N1(C(C(C)CC2CC2)=O)CCC2CN(C(=O)C=Cc3cnc[nH]3)CC2CC1 c1(C(N(CCCNC(c2cccnc2)=O)C2CC2)=O)cc2c(s1)CCCCCC2 c1(C(c2nnnn2C2COC2)NCC(CC(=O)NC)C)cc([N+](=O)[O-])cc(C)n1 C(=O)(CC(C)C(F)(F)F)N1CCC(CC#C)(C(=O)N(C)CCCC(=O)OC)C1 N1(C(c2cc(C)n(C)c2)=O)CCCC(C)(CNC(=O)CSc2n[nH]c(O)n2)C1 c1(C(N2CC(C)CC(NC(c3c(C)nc(O)cc3)=O)C2)=O)cnc2c(c1)COC2 Cc1cc(C)c(C(=O)NC2CC3CCC2N(C(c2snc(O)c2Cl)=O)C3)cc1N N1(C(C(CC=C)C)=O)CCCC(CO)(CNC(C2(CCCC)CCC2)=O)C1 C1(CC)CC(C(N2CC(NC(c3cccnc3CC)=O)CC(C)C2)=O)CC(=O)N1 O=C1Cc2ccc(NC(C3C=CC(Nc4ncc5[nH]ncc5n4)C3)=O)cc2N1 C1(NC(=O)C(O)C2CC2)CCCCN(C(c2scnc2Br)=O)C1 N1(C(c2cc(C)sc2C)C(=O)NCC2CCCO2)CCOC(C)C1C N1(CC(=O)NC(C2CCN(C(C(COC)C)=O)C2)(C)C)CCN(C)CC1 O=C1CCC(S(=O)(=O)N2CCC(O)CC2C(N2C3CCC2CC(O)C3)=O)CC1 N1(C(C(C(C)C)c2cnc(C)s2)=O)CCCC(NC(=O)COCC2CC2)CC1 O=C1CC(CNC(=O)C(Cc2cn[nH]c2)NC(=O)CN2CCOCC2)CN1 c1(CC)cc(C(=O)N(CC(O)CN(C)C(c2cncnc2)=O)C)cc(Cl)c1 Cn1nc2c(c1C(=O)NC1CC3CN(C(c4ccns4)=O)CC13)CCCC2 C1(OC(c2ccc(Cn3ccnc3)cc2)=O)CCC2(CCOC2)C1 c1(C(c2n(C(C)(C)C)nnn2)NCCC2(CS(C)(=O)=O)CC2)ccc(Cl)c(F)c1 C1(C(N2CCC(NC(C(C)(C)OCC)=O)C(F)C2)=O)CC(c2cnn(C)c2)=NO1 C1(C(=O)NC(CNC(c2cccc(OC)n2)=O)CO)Cc2ccccc2C(=O)O1 C(=O)(C1=CC2(CCN(C(=O)C(N3CCNC3=O)C)C2)C1)NCCCOC(C)C C1(CC#C)CN(C(=O)CN(C(C(N2CCOCC2)C2C3CCCC23)=O)CC)CCO1 N1(C(c2n(CC)nnc2C)=O)CCCN(C(=O)CP(C)(C)=O)CC1C C1(C(=O)NC(C(C)NC(=O)CCCNC(C2CCC2)=O)CO)CCC(C)(C)O1 CC(C(O)C(=O)N(C(C)CCNC(=O)CCOCC(F)F)C)c1ccccc1F C1(CC(NOCCC)=O)CC(NC(=O)C(O)C2CC2)C1(C)C N1(C(C2CC(C(C)C)C2)=O)CCN(C(C2CN(C(N)=O)C2)=O)C(C(C)(C)C)C1 C1(C(=O)NCCSCC(=O)NC(C2CCCCO2)(C)C)CC(=O)NC1=O C(=O)(CC1CS(=O)(=O)c2ccccc21)N1CCC(NC(CNS(N)(=O)=O)=O)C(O)C1 S(=O)(=O)(c1ccc(N(C)CCOC(C)(C)C)c(Cl)c1)NCC1C(C)COCC1 CCC(Cc1cccc(C)c1)C(=O)NC1CC1NC(c1ccc(SC)cc1)=O C1(C(=O)NCC(C2CCCC2)NC(C2(CC(C)C)COC2)=O)COCCN1CC.CC=C N1(C(c2c(CC)non2)=O)CCC(F)(CNC(c2cnc(O)o2)=O)C1 C1(CC(=O)NCC2(NC(c3c(C)[nH]cc3)=O)CCOC2)CCCC12CC2 Cc1nc(C)n(CC2CCCCN2C(=O)CSc2ncccc2C)n1 C1(c2cccnc2)(C(N(CCCNC(C2C3COCC23)=O)CCO)=O)CC(F)(F)C1 C1(NC(C(COC)OC)=O)CCC2(CC1)CN(C(c1ccccc1C)=O)CCO2 N1(C(COCCC#C)=O)CCC(C(=O)NC(C)CCCC)(COC)C1 c1(C(N2CCCC(NC(C(C)(C(C)C)NC(C)=O)=O)C2)=O)c(F)ccc(Cl)c1N c1(OC)ncc(C(=O)NC2CCCC2CNC(c2cnccc2C)=O)cc1Cl C1(C(=O)Nc2cccc(C(C)C)c2)(OC)CCN(C(=O)C=Cc2ccncn2)C1 N1(C(C2C(C)CCOC2)=O)CCC(C)(C(N2CCC2CF)=O)CC1 N1(C(C2CC(=C)C2)=O)CCCC1(C(=O)N(CCS(C)(=O)=O)C)CC Cc1ocnc1C(c1nnnn1Cc1cccs1)NCCc1ccc(Cl)s1 c1(C(N2CC(NC(Cn3c(C(C)C)nnn3)=O)C(O)C2)=O)cn2cc(Cl)cnc2n1 n1(CCC)ccc(=NC(=O)C2(CCNC(C3CC=CC3)=O)CCC2)[nH]1 C1(C(=O)NCC2CC(CF)C2)C=CCN(C(c2ncc[nH]2)=O)C1 C1(NC(N2CCCC(NC(=O)CCc3ncccn3)C2)=O)CCCC12OCCO2 C#CC1CN(C(=O)C(O)C=C)CCN1C(=O)COC1CCCC1 c1(OC)cc(C(=O)NC2CC(C)N(C(=O)CCn3cncn3)C2)cnc1C C1(NC(CCC=CC)=O)CN(C(c2cccc3c2CCOC3)=O)C2(CCOC2)C1 C1(NC(COCCCCC)=O)CCCCC1CNC(=O)C=CS(C)=O C(=O)(C1=C(Cl)CCC(C)C1)N1C(CCNC(CNS(CC)(=O)=O)=O)CCC1 N1(C(C2OCCN(C)C2)=O)CC(NC(=O)Cc2cccc(O)c2F)CC12CCC2 C1(C(=O)Nc2c(C)cccc2)CC2(CC2)CN1C(=O)CC1CCCOC1 Cc1n[nH]c(C)c1C(=O)NCC(C)CC(=O)NC1(C)CC(C)(C)C1 c1(C(=O)NCCCCN(CCCNC(C2(C)CCCO2)=O)C)cn(C)c(C(F)F)n1 C(=O)(CCC(=O)NN(C)C)NC1CC2(C(C(N(C(C(C)SC)C)C)=O)C2)C1 C1(CNC(C2CCS(=O)(=O)C2)=O)CCC2(CCC2)CN1C(=O)COCCF C1(CC)CCCN(C(=O)C(C)OCCC(C)C)C1C(=O)NCc1ccncc1Cl c1(C(C(=O)NC(C(C)NC(c2c(CCC)nns2)=O)C)(F)F)ccc(F)cc1 Cc1coc2ccc(C(N3CC(NC(=O)C(O)CC(N)=O)CC3CO)=O)cc12 C(=O)(CC(O)C(C)C)N(CCC(=O)N(C1COCC1OC)C)CC N1(C(C2CC(C(C)C)C2)=O)C(C(=O)NC(C)C(=O)N(C)C)CC1C C1(C(=O)NC2CN(C)C2)C2CC1N(C(c1cccnc1Br)=O)C2 c1(C(=O)NCCNC(C2CCN(C3CC3)C2)=O)ccc(OC2CC2)cn1 C1(CC(=O)NCCCCN(C(c2c(C(C)C)nn(C)c2)=O)C)CCC2(CCC2)O1 N1(C(c2ccc(=N)[nH]n2)=O)CCN(C(=O)CNC(C2CCC2)=O)C2CCCCC12 C1(N(C(C2CC(C)(C)C2)=O)CC)CCCN(C(=O)COC(C)(C)C(F)(F)F)CC1 CCC(C)(C)CCCC(=O)N1CCC(=CCNC(C2CC2F)=O)CC1 Cc1c(O)ccc(C(=O)Oc2ccc(NC(c3cccs3)=O)cc2)c1C C1(CNC(C(c2cccc(Cl)c2)OC)=O)CC2CC2N1C(=O)C(C)(F)F C#Cc1ccc(Cl)c(C(=O)NCc2cc(F)ccc2N2CCCC2)c1 Cc1ccc(C)c(CNC(c2n[nH]cc2NC(c2ccccc2CC#N)=O)=O)c1 C1(c2cccc(CC)c2)NC(=O)N(CC(C)C)C(C(C)=O)=C1C(=O)OCC C1C(N(C)C)C(=O)NC(CC)C(=O)N1.C(C(=O)OC)SCSCC Cc1cccc(C(N2CCCCC2C(=O)NC(C)(CO)C(F)(F)F)=O)c1F S(=O)(=O)(c1ccc(C(=O)NC23CC(C2)N(C(=O)CC(C)COC)C3)cc1)NC C1(C(N2CCN(CCNC(C3(OC)CCC3)=O)CC2)=O)CC(C2CCC2)C1 c1(C(N(CCCNC(C2CC23CCCC3)=O)C)=O)cccc(N)c1C(F)F C1(CCNC(C(CC)OCC)=O)CSCCN1C(c1ccnc(OCCO)c1)=O N1(C(C(C2CCN(C(C(C(=O)OC)(C)F)=O)CC2)C)=O)CC2CC(C1)C2(C)C N1(C(C)=O)CCC(NC(=O)Cc2ccccc2-c2ccccc2CO)C(F)C1 CC(C)CCC(F)C(=O)N1CCC(C(=O)NCC2CC3C=CC2O3)C12CC2 C1(NC(C2(COCC)CC2)=O)CCC(N(C(=O)C(C)n2ccnn2)C)CC1 N1(C(CC=CC)=O)CC(NC(C2CC(=O)N(CCOC)C2)=O)C(O)C1 C(c1ccc(SC)cc1)=CC(=O)NC1CN(C(C2CC(OCC)C2)=O)C2C1C2 c1(C(C)=O)ccc(CC(N2CCN(C(=O)Cc3cnc(C)[nH]3)CC2)=O)cc1 c1(C(=O)NC2CCC(N(C)C(c3ccc(=O)oc3)=O)C2)cc2ncccc2o1 CCN=C(NCCC1CCC1)N1CCCC(OCCOC)C1.N(CCOC)C1CC1 c1(C(=O)OC)cc(Cl)ncc1CNCC1CCCOC1c1cnn(C)c1 c1(C(=O)NCCN(C(C=CC(=O)NC2CC2)=O)C2CC2)cc(F)cc2nc[nH]c12 c1(CC)cnsc1C(N1CC=CC1C(=O)NC(c1snnc1C)C)=O c1(CONC(Cc2cc(OC)c(Br)cc2)=O)cc(OC)c(OC)c(I)c1 C1(NC(C(c2ccsc2)NC(C)=O)=O)CC(O)(C(F)(F)F)C1 Cn1nnc2cc(C(=O)NCC3(C)CN(Cc4cc(Cl)cnc4F)C3)ccc12 C1(NC(c2cc(Cl)c[nH]2)=O)CS(=O)(=O)CC1NC(c1cc(C2CCCC2)no1)=O Cc1ccc(COC(N2CCOC(OC(C)C)C2)=O)cc1F Cc1ccc(C(=O)NCC2CN(C(c3cccnn3)=O)CC2C(F)(F)F)c(C)n1 CCC(C)(CNC(=O)C=C(C)COC)C(=O)NCc1nc(C2CC2)n[nH]1 c1(C(=O)NCC(C)(C2CC2)NC(C2C(OC)CCC2)=O)c(C)cc(C)oc1=O N1(C(CCNC(=O)C=CCl)=O)CC2CC(C1)N(C(C1CCOC1C(F)(F)F)=O)C2 N1(C(c2nc(CC)oc2)=O)CCC(F)C(NC(c2ccccc2C2CC2)=O)C1 N1(C(CN(C(C2CN(C(C)C)C2)=O)CC2CC2)=O)CCCC(F)(F)C1 N1(C(C(F)=C(C)C)=O)CCC2(CCCCC2NC(c2cc(C(N)=O)[nH]n2)=O)C1 c1(C(N2CCC(C(C)NC(c3cc(C)cc(C)c3)=O)C2)=O)cscc1S(C)(=O)=O C(=O)(C(C)CC(C)C)N(CC(CNC(C=Cc1cc(C)no1)=O)(C)C)C C1(CS(=O)(=O)NCC(c2ccc(F)cc2F)(C)O)CC2C(C1)C2(F)F C1(CNC(c2cccc(C)c2F)=O)CN(C(c2cnc(O)n2C)=O)C2(CCC2)C1 c1(C(=O)NC2(CCNC(CCCC(C)=O)=O)CCC2)cc2c(s1)CCSC2 CCC(C)(C)C(=O)NC(CN(C)C(c1c[nH]c(=N)s1)=O)Cc1ccccc1 C1(C(=O)NCCOCCOCCNC(c2c(C)scn2)=O)CN=C2N=CNN2C1 c1(C(=O)NCC2CN(C(CC(C)F)=O)C3(C2)CCC3)cc2ccccc2cc1F C=CCCCC(C)(C)C(=O)NCC1C(O)C(O)CN1C(=O)CN(C)C(C)C c1(C(N2CC(CC(C)NC(c3cnnc(O)c3)=O)C2)=O)cc2c(O)cccc2[nH]1 C(=O)(CCCC(F)(F)CO)N1CCC(C(C)NC(c2nn(C)cc2Cl)=O)C1 C(CC(C)(C)C)(c1n(CC=C)nnn1)(C1CC1)NCc1c(C)ccnc1C c1(C(=O)NC2CCN(C(C3C4COCC34)=O)CC2F)ccc(F)c(Cl)c1F Cc1ccc(C(F)C(=O)N(C2CCN(C(c3ccncc3F)=O)C2)C)cc1 c1(C(N(CCN(C(COCC)=O)C)C)=O)ccc(N2CCN(C)CC2)c(F)c1 N1(C(C(c2c(NC(C)=O)cccc2)(F)F)=O)CCC(O)(CNC(=O)C(C)C)CC1 c1(C(=O)NC2C(CNC(C3(CC)CC3)=O)CCC2)cc(N)cnc1Cl c1(C(=O)NC2(C(=O)NC(CCCC)CCCC)CCC2)cccn2cncc12 C(=O)(CC(F)(F)C(F)(F)F)N1CC2C(CNC(c3c(SC)nccn3)=O)C2C1 c1(OC)cnccc1C(=O)NCCC1CC(NC(=O)CC(C)n2ccc(C)n2)C1 N1(C(C(CCOC)(C)C)=O)CCCC2(CC(NC(C3(F)CCOCC3)=O)C2)C1 c1(C(=O)OC)ccc(F)c(S(=O)(=O)NC2CCCN(C(=O)Cn3cccn3)C2)c1 C1(C2CCN(C(c3n[nH]cc3C(F)(F)F)=O)C2)(NC(c2ccc(Cl)cc2)=O)CC1 C12(CNC(C(CC)(C)C#N)=O)CCCC(CN1C(c1ccc3nc[nH]c3c1)=O)C2 c1(NC)cc(C(=O)NC2(CCCCNC(=O)C=CC(F)(F)F)CC2)[nH]n1 CC1CC(NC(=O)CSc2nncs2)CN1c1cc(-n2ccnc2)ncn1 N1(C(C2(CC)CCCO2)=O)CCOC(C2CN(C(c3csc(=N)[nH]3)=O)C2)C1 N1(C(C(CNC(c2ccc(C)s2)=O)C)=O)CCc2ccncc21 n1(C(C)C)cc(C(=O)NCC(C2CC2)NC(=O)CCCCN(C)C)c(Br)n1 Cc1ccc2c(C(N3CCC(C(C)NC(c4occc4F)=O)CC3)=O)csc2c1 c1(C(N2CC(NC(C(C)n3cccc3)=O)(CO)C2)=O)cc2c(cn1)CCCC2 C#Cc1cccc(NC(=O)CC(=O)NCCCNC(=O)C(C)(C)c2cnsc2)c1 Cc1c(C(=O)NCC2CC2NC(C2(C(F)F)CC2)=O)noc1-c1ccccc1 c1(CC(=O)NC(CNC(COCc2onc(C)n2)=O)(C)C2CC2)cc(Cl)n(C)n1 C(=O)(CCN(OC)C(=O)C(C)C(O)C(C)C)NCC1C(CCC)CCC1 c1(C(N2CCC=C(CNC(c3ncn(CC)n3)=O)C2)=O)cc(O)c(F)cc1N C(=O)(C1=CC2CCC(C1)C2)NCC(C(=O)NCC1(O)CCC(C)(C)C1)N(C)C c1(-c2ccc(CNC(C3CCOC3c3nc[nH]n3)=O)s2)ccc(Cl)cc1 c1(CC)cnn(C)c1C(=O)NC(C)CCNC(=O)C(c1ccccc1)OC c1(C(N(CC)CC2CCN(C(C3(CO)CC3)=O)CC2)=O)cc2sc(Cl)cc2s1 c1(C(=O)NCC(C)CNC(C2CC2Br)=O)cn2ccccc2n1 c1(CC)ncnc(CC)c1C(=O)NC(C)CCN(C(=O)CC(C)c1ccco1)C CC1(C)CCN(C(C2CCS(=O)(=O)C2)=O)C1CNC(=O)CC(=O)Nc1nccs1 c1(CNC(=NC)NCCCCl)cccc(CNC(=O)OC(C)(C)C)c1 c1(C(N(C2CN(C(c3c(C)nns3)=O)C2)C)=O)cncc2ccccc12 c1(CCN(C)CCO)cn(CC(=O)N(C)CCN2CCOC2=O)nn1 O=C(C#CC1CC1)NC(C(=O)NCCCF)C1(O)CCC1 N1(C(C(C)SCC)=O)CCC(C)(C)C1CNC(c1c[nH]nc1-c1ccncc1)=O c1(C(C)OC(c2cc(COC)no2)=O)ccc(F)cc1 c1(C(=O)NCC(C)NC(C23CC(C(F)F)(CO2)C3)=O)c(Cl)cncc1Cl C1(CNC(c2ccc(C)cn2)=O)CCN(C(C2C=CCC2)=O)C1(C)C c1(OCn2ncc(NC(c3onc(C)n3)c3nnnn3C)c2)ncccc1Br C1(NC(C(C)O)=O)CCC2CN(C(=O)C=CCN3CCCC3)CC2C1 c1(C(=O)NC)cccc(C(N2CC(NC(=O)CC3CCN(C)C3)C(C)C2)=O)c1 C1(CC=C)(NC(=O)C(C2CC2)OCC)CCN(c2ncc(Br)c(C)n2)CC1 N1(CC(c2cccc(SC)c2)NCC(C)C)CCCC(C)(C#N)C1 N1(c2sc(C(=O)OC)c(Cl)n2)CCN(C(=O)CCn2cnnn2)C(C)C1 N1(C(c2c(NC(c3c(C)nccc3)=O)cnc(F)c2)=O)CCc2n[nH]c(C)c2C1 C(=O)(C1=CCCCC1)NCC(C1CCCC1)NC(=O)CC1CCC12CCC2 c1(OC)ncc(Cl)cc1C(=O)N(C(C)CN(C(=O)Cc1ccco1)C)C C1(CC(C)NC(C2(OCC)CCC2)=O)CCN(C(=O)CC2C=CCC2)CC1 N1(C(C2ON=C(C(=O)OC)C2)=O)CCCC2CN(C(C3CC(C(C)C)C3)=O)CC12 C1(NC(CCCCOCC)=O)CN(C(=O)C(C)n2cncn2)CC(F)(F)C1 C(CC(=O)NCC12CCC(CC1)C2)(C(F)(F)F)NC(C(CSC)O)=O N1(C(c2[nH]cc(C)c2)=O)CCC(C)C(CC(=O)NCC(=O)NCC(F)F)C1 N1(C(c2c(COC)noc2)=O)CC(C)CCC1CNC(=O)C(F)(F)C1CCCC1 CC1(C)OC(C(=O)NCC(C)(F)CNC(=O)Cc2csc(Cl)n2)C(C)(C)O1 C1(C)(CNC(CCc2onc(CC)n2)=O)CCCN(C(c2c(C)nsc2C)=O)C1 Nc1ccc(F)cc1CNC(c1coc(C(F)F)n1)=O N1(C(=O)CC2CC=CC2)CC2(C1)CN(C(C1CC13CCOC3)=O)CCO2 N1(C(COCCOCC#C)=O)CCC2OCCN(C(c3ccsc3C#N)=O)C2C1 C1(NC(=O)CCCc2cn(-c3ncc(F)cn3)nn2)CC2CC(C1)C(=O)N2 N1(C(c2cnc(C(C)C)s2)=O)CC(CNC(C2CC(=O)N(C)C2)=O)C(C)(C)C1 C1(C(=O)NCc2nc(CNC(c3cc(C4CC4)on3)=O)sc2)CCCC(F)C1 c1(C(N(C)CC2CCCCN2C(c2ccc(F)cn2)=O)=O)c2c(nn1C)CCC2 c1(OC)c(C(=O)NCC(C)(C)NC(=O)C(C)CC(C)C)oc2ccccc12 C1(CNC(=O)NC(c2c(F)cccc2I)CO)CCc2c(O)cccc2C1 c1(SC)ccccc1C(C)NC(=O)NC1CCN(c2ccc(Br)cc2)C1 N1(C(CN(C(C)C)C(c2ccncn2)=O)=O)CCC2(C1)CC2(F)F S(=O)(=O)(CCC(=O)NCc1ccccc1)NC1C(CN(C2CCCC2)C)OCC1 c1(C(=O)NCCCN(C(c2ccnnc2O)=O)CC)cncc(OC)n1 N1(C(C)=O)CCC2(CC1)CN(C(C)=O)C2.C(=O)(C(C)CC=Cc1ccccc1)OC Cc1[nH]nc2ccc(C(N3CCCC(F)(CNC(=O)CSC(C)C)C3)=O)c(Cl)c12 c1(C(C)=O)c(NC(=O)CC2CN(C(C3CC3C)=O)C2)cccc1F CC1CCN(C(C2CCCN2C)=O)CC1CNC(c1cnc(C2CCOC2)s1)=O N1(C(C=CC2(C)CCOCC2)=O)CCC2CN(C(=O)CC3CC(=O)NC3=O)CC12 c1(C(N2CCC(NC(CCN(C)CC)=O)CC2C2CC2)=O)cc(C)c(C)nc1C CCC(CNC(c1cc(COC(C)(C)C)on1)=O)(CC)NC(=O)C(C)N(C)C O=C(C#CC1CCOC1)NCC1CCCCN(C(c2cc3cnccc3[nH]2)=O)C1 c1(NCC(C)CO)ccc(S(=O)(=O)NCc2cc(Cl)n(C)n2)cc1C#N CC1CC(c2ccsc2)CN1CNCc1ccc(Cc2ccccc2)cc1 C1(NC(C(CN(C)C)c2ccccc2)=O)(CO)CCCN(C(=O)CSC(F)F)C1 c1(OCC(=O)NCC2CC(F)(CNC(C(C)C)=O)C2)cc(F)ccc1F CCC(C(=O)NCC#CC(N1CCC(C2CCC2)C1)=O)C(C)(C)CC C(=O)(C#CC(=O)N(C)C)NCC1CCN(C(C(CC)F)=O)C1 c1(C(=O)NCCNC(C(CC)n2nccc2C)=O)ccnc(OC(F)F)c1 c1(CCC(=O)NC2CC(NC(CCC3CCCN(C)C3)=O)C2)c(O)cccc1F C#Cc1ccc(C)c(NC(=O)C(C)(C2CC2)N(C)C(c2cnc(O)n2CC)=O)c1 c1(C(=O)NCC2CC(NC(C3OCCCO3)=O)C2)ccc(-c2ccccn2)o1 CCC(N=c1nc2sccc2c(NC2CCNC(=O)CC2)[nH]1)C(C)C N1(C(C(C2CCCN(C(C3CC(=O)CC(=O)N3)=O)C2)C)=O)CCCN(C)CC1C N1(C(CN2CC(C)(OC)C2)=O)CCC2CCN(C(=O)CCC(C)N(C)C)C2C1 C(C)(CCN(C(=O)C(C)n1cnnn1)C)NC(COCC)=O C1(C)(CNC(C2(COC)COC2)=O)CCN(C(c2cc(Br)nn2C)=O)C1 N1(C(c2c(C(C)C)occ2)=O)CCC(CNC(=O)Cc2nnc(O)s2)C(C)C1 CC(=O)CCCC(=O)NCC1CN(C(=O)CCOCC2CC2)CC1C CCCCCC(CC)C(=O)N1CCC(CC(C)NC(c2csc(C)c2N)=O)CC1 Cc1ccc(C(N2CC(CN(C(=O)C=CCO)C)C2)=O)cc1Br N1(C(CC2(OC)CC2)=O)CCC2(CCC2)C(NC(=O)CN2CC(=O)NC2=O)C1 c1(C(=O)OC)cc2c(s1)C1(CCN(CC3CCCCCCC3)CC1)OCC2 c1(C(N2CC(CC=C)(NC(=O)COC3CCOC3)C2)=O)ncnc2sccc12 N1(C(CC(C)(C)OC)=O)CCCC12CCCN(C(C1(CC3CCC3)CC1)=O)C2 Cc1cc(C(N2CCC(N(C)C(c3ocnc3C)=O)C2)=O)c(C(F)(F)F)o1 CC(CO)C(=O)NCC1CC1C(N1CC(CO)C1)=O c1(OC)ccc(C=CC(=O)N(C)CC2CCCN(C(c3csnc3Cl)=O)C2)cc1 c1(C(N2CCC(NC(c3ccc(C)s3)=O)CC2)=O)cnc2[nH]ccc2n1 c1(C(=O)NCc2scc(CNC(c3c(CC)nn[nH]3)=O)n2)cc(Cl)ccc1C C(CC1CCC1)(C(=O)N1CCC(Cn2ccnn2)C1)NC(=O)C=CC(F)F CC1(NCCC2CCOCC2)CCOC12CC2(F)F C(C)(CC1CCC1)(C(=O)NC(C)C(C)NC(c1csc(C2CC2)n1)=O)OC c1(CC(=O)NC(CC2CN(C(COCCOC(C)(C)C)=O)C2)C)ccc(F)cc1 N1(C(c2cncc(C(=O)OC)c2)=O)CC=C(CCNC(C2CNC(=O)N2)=O)CC1 c1(C(=O)NCC(C)NC(c2ccc[n+]([O-])c2)=O)c[nH]c2nccc(Br)c12 CCCCC(CNC(=O)C=Cc1cccn1C)NC(=O)C(CN(C)C)N(C)C N1(C2CCC(=O)NCC2)CCc2ncnc(O)c2C1 c1(C(N(C2CCCN(C(c3ccccc3C(N)=O)=O)C2)CC)=O)cc[nH]c(=N)c1 c1(C(N2CCCC(NC(CCC#CC)=O)C2C)=O)oc2ccccc2c1COC C(=O)(C(C)(C)C(F)F)N1CC=CC(C(=O)NC(COC)C(C)C)C1 C1(CNC(C=CCN(C)C)=O)CCC2(CN(C(c3noc4ccccc34)=O)C2)O1 c1(C(=O)NC2CC(CNC(=O)C(F)=CCCF)C2)csc2cncn12 c1(OC)cc(CN2CCC(C)(CNC(=O)CN3CCCCC3)CC2)ccc1Cl c1(C(=O)NCC2(CO)CCN(C(C3C(C#C)C3)=O)CC2)cc(Cl)cc(C#C)c1 N1(C(C(CC)Cc2cnc[nH]2)=O)CCCN(C(C2CCCSC2)=O)CC1 c1(NC(=O)Nc2ccc(OCC(F)(F)F)cc2)cccc(F)c1F C1(C(=O)NCCN(CCC)C(C2CCCN2N=O)=O)CCc2cc(C)ccc2O1 Cc1c(C(N2CCC(F)(CNC(C3(CCO)CC3)=O)C2)=O)ccc2ccccc12 C1(C(=O)N)CCN(C(=O)CC2C=CCC2)C1.N=C(O)OCCC1CCC1 CCCCC(=O)C(=O)NCC=CCC(=O)N(C)CC1(CO)CCC1 Cc1[nH]nc(C(=O)NC(C(N2CCC2(C)CCO)=O)C2CCCC2)c1Cl Cc1cccc(OCC(=O)NC2CCC(NC(C3CCCC3C(F)F)=O)CC2)c1 CC1(C)C(c2ccccc2)CN1C(=O)Cc1nc(C2CC2)cs1 CC(c1ccsc1)=CC(=O)NC1COCCC1NC(=O)C(n1cc(C)cn1)C C1(C(C(=O)N(CC(CC)NC(C2(COC(C)C)CC2)=O)C)O)CCOCC1 C1(CC(N2CC(NC(C(C(C)C)(C)C)=O)C2)=O)Oc2ccccc2NC1=O C1(C(=O)OC)(C(N2CC(CO)(NC(=O)C(C(C)C)N(C)C)C2)=O)CC2(CCC2)C1 c1(N(C)C)ccc(C(=O)Nc2nc(CC(=O)Nc3cnc(Cl)cn3)cs2)cc1F Cc1cc(C(N2CCC(C(=O)NCC3CC34CC4(F)F)C23CC3)=O)cnc1C C1(C(=O)NC2CCSC23CN(C(C2CC2CF)=O)C3)CC(c2cccnc2)=NO1 N1(C(Cc2cnc(C)[nH]2)=O)CCOC(CCCNC(=O)CN(C)C(C)C)C1 CC(c1ccccc1)=CC(=O)NCC1CCC(C)CN1C(=O)CSCC(F)(F)F CC(C(=O)N(CC(C)(C)NC(=O)CC1CCCC(C#N)C1)C)C(C)(C)C C#CCC(C)C(=O)NCC=CCNC(c1ccc(Cn2ccnc2)cc1)=O c1(N(CCCNC(C2CCCN2C2CCCC2)=O)CC)ccncc1C#N c1(C(N2CC(NC(C(CC)n3cccn3)=O)(CO)C2)=O)cc(F)ccc1N c1(OC)ccc(C(=O)NC2CCCCC2NC(=O)C(C)OCCC(C)C)nc1 C1(CC(=O)NCCC(=O)N(CC)CC)CN(C(c2ccon2)=O)C(C)(C)C1 c1(C(N2CCC3(C(C(=O)NCC4C(C)(C)COC4)C3)C2)=O)ccn2ccnc2c1 C(=O)(C1=CCOCC1)N1C2(C(N3CCC(NC(=O)NC)C3)=O)CC2CC1 C=CCC(C(=O)N1CC(CNC(c2sc(C)cc2C)=O)C(C)(C)C1)C(C)C CCC(CCC(=O)NC1(COC)CCN(C(=O)C2=C(C)CC2)C1)OCC c1(N(C2CN(C(C3CCOCC3)=O)C2)C)nc(-c2ccsc2)ns1 N1(C(c2c(-c3cnn(C)c(=O)c3)cccn2)=O)CCC(O)C(F)(F)C1 Cn1c(O)nc2cc(C(=O)NC(CO)C3(C)CC3)ccc12 c1(OC)nc(C)ncc1C(=O)NC(CNC(c1cc(C)cc(Cl)c1)=O)C1CCC1 C1(C(=O)NCC(C)(C)NC(C(c2ccc(F)c(Cl)c2)C)=O)CCc2ncnn2C1 C1(C(=O)NCc2nccc(C)c2)CC12CCN(C(=O)Nc1ccccc1)C2 c1(OCCOC)cc(C)ccc1CNC(=O)NCC1CC(F)C(=O)N1 N1(C(c2c(C)coc2C(C)(C)C)=O)CCC(C)C(NC(C2C3(CC3)C23CC3)=O)C1 C(=O)(CC(C)(C)c1cccc(Br)c1)NC(C(CO)NC(C(F)=CC)=O)C C(C(=O)NC1CN(C(c2cc(Cl)n(C)n2)=O)CC1C)(C(C)C)(C(C)C)NC(C)=O N1(C(CC(C)SC)=O)CCCC12CCN(C(C1CCc3nnc(C)n3C1)=O)CC2 C1(C(=O)NC(CCSC)C)CCOC1CNC(=O)Cc1coc(C)n1 C1(NC(c2c(C)c[nH]n2)=O)CN(C(=O)C2=CCSC2)CC12CCOCC2 CC(=O)CCCC(=O)NC(CNC(=O)COc1cccnc1)C(C)C C1(NC(c2c(C)n(C3CCC3)nc2)=O)CCC(C)N(C(c2ncccc2N)=O)C1 S(=O)(=O)(c1ccc(Br)cc1N1CC2CCCN2C(C(C)C)C1)N(CC(C)C#N)C C12(C(=O)NCCC(C)N(C(c3cnn(C(C)C)n3)=O)C)CCC(CC1)C(C)(C)O2 c1(NC(N2C(C(=O)Nc3ncc(C)cc3O)CC2)=O)ncc([N+](=O)[O-])cc1Br C1(CNC(C=CCCC)=O)CCCN1C(=O)C(C)c1cncs1 CC(F)(F)CCCC(=O)NC(C)(CNC(C1C2COCC12)=O)C1CC1 c1(C(N2CC(N(C(c3cnc(C)s3)=O)C)C(F)C2)=O)cnn2ccncc12 c1(C(C)NC(=O)NCC(C=C)(F)F)cccnc1F C1(C(N(C2CC(C#N)C2)CC(=O)N(C)CC2CC(F)C2)=O)CCNC1=O c1(C(=O)NNc2cccc(Cl)n2)ccc2c(c1)CNCCN2 C1(NC(C2C(C)(C)CO2)=O)CCN(C(c2cnc3[nH]cncc2-3)=O)C12CCC2 c1(C(=O)NCC2(F)CC(NC(COC)=O)C2)cncc(-c2ccoc2)c1 c1(-c2n(C(CC)C)nc(-c3cccc(Br)c3)n2)cc2c(O)ncnc2cn1 CC(=O)CCN=C(NCC#Cc1ccccc1Cl)NCc1noc(C(C)(C)C)n1 N1(C(c2n(C)cnc2)=O)CCCC(CNC(=O)CCCc2ccc(Br)cn2)C1 Cn1ccc2ccnc(C(N3CCC3CNC(C3CC4CCC(C3)S4)=O)=O)c12 CC(CC(=O)NC12CCC(CC1)N(C(=O)C(C)(C)CC(F)F)C2)CC(F)(F)F C(=O)(CCCCCCC(=O)OC)NC1CCCC(NC(C(C(=C)C)(C)C)=O)CC1 N1(C(C(C)NC(C2CCCC2)=O)=O)CC=CC(NC(C2(S(N)(=O)=O)CC2)=O)C1 N1(C(c2cnc(C3CC3)nc2)C(=O)NCC)CCCC2(C)CCCC12 C1(C(=O)NCc2ncc(CC)s2)(NC(=O)CCC2CCC2)CCCC1C CC(CCCC(=O)NC1(C)CCCN(C(c2ccc[nH]2)=O)C1)c1ccccc1 c1(C(=O)OC)ccc(COC(C23CCCC(CO2)C3)=O)c(F)c1 c1(CC)cc(C(=O)NCC2C(CC)CCN2C(C2C=CCC2)=O)oc1CC C1(NC(C(Br)=C(C)C)=O)CC2CCC(C1C)N2C(c1ccc(CO)cc1)=O C(=O)(C(CNC(=O)CCc1nccn1C)N(C)C)N(CCOCC)C c1(C(=O)NCC2(O)CCCN(C(CNC(=O)OC)=O)C2)cc2cc(Cl)ncc2[nH]1 c1(C(N(CC(CC)(C)Cl)c2ccccc2)=O)cc(C(F)(F)F)cn1C CCCCCCC(CC)C(=O)N1CC2CC1CCC2NC(=O)COC(F)(F)F c1(C(=O)NC(C(N2CC(C)CC(OC)C2)=O)C(C)CC)cccc2[nH]ncc12 N1(C2CN(CC(=O)NC(=O)NC3C4CCCC34)C2)CCN(CC(F)(F)F)CC1 CCCC(O)CC(=O)NC(C)CNC(c1cn(-c2cccc(F)c2)nc1C)=O c1(C(N(CCCNC(c2ccnc(-c3cc[nH]n3)c2)=O)C)=O)ccc(F)cc1N N(C1CCSc2ccc(Br)cc21)C(C(=O)N(c1ccc(Br)cc1)CCOC)=O C(=O)(C(F)C(F)(F)C(F)(F)F)NC(C1CN(C(Cn2nc(C)n(C)c2=O)=O)C1)C C1(F)(C(=O)NCC(CN(C(c2c(C(C)C)[nH]cc2)=O)C)C)CCN(C)CC1 CCCCC(C(=O)NCCC(C(C)C)NC(=O)C=CCCC(C)C)ON=C(C)C S(=O)(=O)(C(C(F)(F)F)OC)NC(=O)OCc1cn(CCC=C)nn1 C1(C2CN(C(=O)CCCNC(c3ccsc3)=O)C2)(NC(CN(C(C)C)C)=O)CC1 C#Cc1cccc(C(=O)N(CC(=O)NCC2CC2Cl)C(C)C)c1C CC1Cc2sc(C(=O)NNC(=O)c3cccc(O)n3)cc2C(C)C1 CC1=CC(C(=O)N(C(C)C(=O)NC(c2nc(=O)o[nH]2)C)C)SC1 c1(C(c2n(CC=C)nnn2)NCC(F)C2CCC2)cncc(C=C)c1 c1(CC)ccc(C(=O)N(C)CC2(C(=O)NCC3(O)CCCCC3)CC2)cc1 Cc1cc(NC(C(C)NC(C2(C)CC3(CC3)C2)=O)C(C)C)nc(C(F)(F)F)n1 C(=O)(C(F)(F)C(F)F)N1CCC(N(c2cnc[nH]2)C(=O)COC(F)F)C1 S(=O)(=O)(c1cccc(=NC(C)c2ccccc2Br)[nH]1)NCc1cc(OC)no1 c1(C(=O)NCC(CC)NC(C2(COC)CC=CCC2)=O)cnc2cccnn12 Cc1ccc(F)cc1C(N1CCC(O)(C(=O)NC(C2CCOC2)C)C1)=O C1(C(=O)NCC(CC)(CC)NC(=O)CCCN(C)N=O)CCC2(CCCO2)CC1 C1(CNC(c2nc(-c3ccc(C)cc3)sc2)=O)C(C)CCCN1C(=O)C=C1CC1 C1(C(CNC(=O)CCC(F)(F)F)=O)CC(N=c2cc(Cl)nc(C(F)(F)F)[nH]2)C1 C1(CC)CN(C(=O)C(C)(C)CN(C(=O)C(CN(C)C)N(C)C)CC)C(C)CO1 CC(C)C(C)(C)C(=O)NC(CNC(=O)C(C)OCC1CC1)CO c1(NCC)cncc(C(=O)NC(C2CN(C(C3CCC(C(N)=O)O3)=O)C2)C)c1 C(=O)(C(C)(C)CF)N(CCCCCNC(C1C(C)(C(C)C)C1)=O)C c1(C(=O)NC2C(CNC(c3ccc(C4CC4)s3)=O)C2)cccc2nc(S)oc12 C(=O)(C(C)(C)C(=O)N(CC(C)N(C)C(c1cc(SC)oc1C)=O)C)NC C1(NC(COc2cccc(C#C)c2)=O)CC2CN(C(C3(C)CC3)=O)CC2C1 c1(CNC(CCC2(NC(CC(C)n3cccc3)=O)CCCC2)=O)cccc(F)c1 C1(C(N(CCCNC(=O)C(C)(O)C(C)C)CC)=O)CCCCC12CCC2 c1(C(=O)NCCC=C(C)C)ccc(C2CC2)o1 C1(CC(=O)NCCC2N(C(c3c(COC)scc3)=O)CCC2)CCCCC1F C(CN=c1cncc[nH]1)NC(=O)NCC1CCCC1F C1(NC(c2cnccc2Cl)=O)CN(C(=O)CCCCC2CC2)C2(CCCCC2)C1 CC1c2cc(Cl)c(Cl)cc2CCN1C(c1cncc(C(N)=O)c1)=O C(=O)(C(F)CC(CC)CC)NCCC1CCC(NC(C(C)OCC)=O)C1 C1(N(C)C(=O)Nc2cccc(C(F)C(F)(F)F)c2F)CC(C)(C)OC(C)(C)C1 C=CC(C)(O)CC(=O)NC(C(=O)NCC1(O)CCCCCC1)C(C)O C1(NC(c2cc(C)nc(C)c2)=O)CCC12CCN(C(c1cc(C)oc1C)=O)CC2 Cc1c(Cl)ccc2[nH]c(C(=O)NCC(F)CNC(c3c[nH]c(=N)o3)=O)cc12 c1(NC(C2(COC)CN(C(=O)Cc3ccc(C)cc3)C2)=O)nccc2occc12 C1(C(C)C)CN(C(c2cncnc2)=O)CCN1C(=O)Cc1cccc(Br)c1 Cc1cccnc1CC(=O)NC(C)C(CO)NC(c1cc(C(C)(C)C)c[nH]1)=O c1(-c2c(C)cccc2)nc(=NC2CN(C(C3CCCOC3)=O)CC(C)(C)C2)s[nH]1 c1(C(C)C(N2CCC(N(C(=O)C=CCOC(C)(C)C)C)C2)=O)cccc(F)c1 C(=O)(C(C)C(C)NC(=O)C(CCC1CC1)NC(C1CC12CC2)=O)OC Cc1cccc2[nH]c(C(N3CC(O)CC3C(=O)NCCc3nn[nH]n3)=O)cc12 c1(C(N2CC(CSC)C2)=O)ccc(CNC(=O)C(=O)C(C)C)nc1 C#CCC(CC#C)C(=O)NC1CC2CCC1CN2C(C12CCCC1C2(F)F)=O N1(C(c2ncc(C)nc2)=O)CC2CC(NC(c3cncc(Cl)c3Cl)=O)CC2C1 Cc1c(NC(=O)CC2CCCC2NC(=O)CNC=O)cnn1CCO CCC(C(=O)NC1(CNC(c2n[nH]c(C)c2Cl)=O)CCCC1)C(C)(F)F CN(C1CCCC1C(F)(F)F)N(CCOC(C)(C)C)C1CC1 N1(C(CCCCN(C(C)=O)C)=O)CCN(C(C2CCCC(O)C2)=O)CC12CC2 C1(CNC(C2OCC(C)(C)C2)=O)CCN(C(c2cnsc2)=O)C12CCC2 c1(N(C(C)C(=O)OCC)CC)ccc(C(C)(C)C#N)cc1 C1(NC(C(CC)C)=O)(CNC(c2cc(OC)ncc2F)=O)Cc2ccccc2C1 c1(C(=O)NC(CC)CNC(=O)C(CC)C(F)(F)F)cnc(P(C)(C)=O)cn1 c1(C(=O)NCC(C)N(C(c2csc(C(C)OC)n2)=O)CC)ccnnc1O c1(C(=O)NCC2(F)CN(C(c3ccc(Cl)nc3O)=O)C2)c[nH]c2ccc(F)cc12 N1(C(CN(C(C)CN)C)=O)CCC(CO)CC1.c1(C2C(C=O)C2)cccs1 c1(CN(C(=O)C=CSc2ccccc2)C)ccc(CCNC(=O)C(=O)NC)cc1 Cc1cc(CC(=O)NCCC(O)CNC(c2cccn2-c2ccccc2)=O)n[nH]1 CCC(CC(=O)NCC1CC2(CC(NC(=O)C(O)CC(C)C)C2)C1)C(F)F CCC(CC)C(=O)NCC1(F)CCN(C(=O)CC2CC(OC)C2)C1 C#Cc1cccc(CCC(=O)NCC2(CC(N3CC4CC4C3)=O)CCC2)c1 c1(OC)ccc(F)c(C(=O)NCC(F)CNC(C2CCSCC2)=O)c1F c1(C(N2C(CNC(CC(C)c3cccnc3)=O)C=CC2)=O)ccn2ccnc2c1 Cc1ncc2ccc(C(=O)NC3CC4CC(NC(c5ccncn5)=O)CC34)cn12 CC1(C)CCCC1CNC(C1OCCC1NC(=O)C(O)c1ccco1)=O C(CC(C)CC)(C(=O)NCc1nnn(C)n1)NC(C=CC)=O O=C(CCCC(F)(F)CO)NCCC1CCCN(C(=O)CC2CCCC2)C1 c1(C(=O)NCC23C(CN(C(Cc4cnc(C)s4)=O)C2)C3)cnc2[nH]cc(C)c2c1 C1(C)(CNC(C=COCC)=O)CCN(C(=O)CC2CC(F)(F)C2)C1 C1(NC(c2ccc(C(F)F)c(Cl)c2)=O)CN(C(=O)C#CC2CC2)CC2(CCC2)C1 C1(CC)CN(C(C2CCCSC2C)=O)CC1C(=O)NCC(C)(C)C(N)=O C(=O)(C(C)(C)C(=O)NC1CCN(C(=O)C(NC(C)=O)=Cc2cccs2)C1)NC N1(CC(N2CCN(C3CCN(Cc4ccc(F)cn4)C3)CC2)=O)C(=O)CNC1=O c1(C(=O)NC2C(F)CCN(C(c3cn(CC=C)nn3)=O)C2)cscc1S(C)(=O)=O C1(C(=O)NCCc2cn(CC)nn2)C=CCN(C(=O)CCn2ccnn2)C1 c1(C(=O)NC(CC)CCOC)cccnc1CNC(=O)CC1CC2CC2C1 c1(C(N2CC(Cn3cc(C(C(C)(C)C)O)nn3)C2)=O)ncc(Cl)cc1F C(C(CC(=O)NC1CCCNC1=O)C1CCC1)NC(c1cc(C2CC2)on1)=O N1(C2CCN(C(CC3(C)CCC3)=O)C2)CCC(NC(C2CC2(Cl)Cl)=O)CC1 c1(C2C(=O)OCCCN2CC)ccn(CC2CC(SC(C)C)C2)n1.C(C)(=O)OC n1(CCC)nc(C)c(C(=O)NCC2(F)CC(NC(=O)Cn3cnc(=N)[nH]3)C2)c1C c1(C(NNC(N2CCCS2(=O)=O)=O)=O)cc2c(s1)-c1ccccc1OC2 C1(NC(C(COC)(F)F)=O)CCN(C(c2c(F)cncc2Br)=O)CC1C N1(C(C=CCN(C)CC)=O)CCC2CC2(NC(=O)CCCCCF)CC1 N1(C(C(C)N(C(C)=O)C)=O)C2CC=C(C(=O)N(CCCN=[N+]=[N-])C)C1CC2 C=CC1(CC(N2CC(O)CC2CNC(=O)CC2CC=CCC2)=O)CCCCC1 C1(NC(Cc2n(C)nnc2)=O)CC2CC1CN2C(c1ccc(OCCF)cn1)=O C(CO)(C(=O)NCCC1CCCOC1)NC(c1nsnc1O)=O c1(C(=O)NC2C(C(=O)NCc3c(OC)cccc3)C2)cccc(Cl)c1OC c1(CN2CC3C(NC(=O)Cc4cc(F)ccc4F)C3C2)ccc(Br)c2nsnc12 c1(OC)cc(C(N2CC(NC(=O)Cc3cc(C)no3)CC2C)=O)cc(C)c1 c1(C(=O)NCC2C3CC2N(C(=O)CCCc2ccncc2)C3)cc(F)cnc1O C=CCC(CNC(C1(C)CC(=C)C1)=O)NC(=O)Cc1[nH]cnc1C C(Cc1cn[nH]c1)(C(=O)NCC(F)F)NC(CCOCCOC)=O c1(C(=O)NC(CC)(CNC(c2ccnc(OC)n2)=O)CC)cc(Cl)c(C)cn1 C1(NC(=O)NC2(c3ccc(Cl)c(Br)c3)CC2)CCc2nn[nH]c2C1 c1(CC)cnn(C)c1C(C(=O)NC(C)C(=O)OCC)N(C(C)CCC)C1CC1 C1(c2nnnn2C(C)(C)CC)(NCC(=C)Br)CCC(P(C)(C)=O)C1 c1(C(N(CCC(C)NC(CS(CC)=O)=O)C)=O)nc2ccccn2c1F CC1CN(C(=O)CCc2cnn[nH]2)CC(C)N(C(=O)CC23CCC(CC2)CC3)C1 c1(CC)c(C(=O)NCC23CC(NC(=O)C(C)C(F)F)(C2)C3)[nH]c2ccccc12 c1(OC)nc(C(=O)NC(C2CCCCN2C(=O)C=Cc2nnn(C)n2)C)sc1C N1(C(c2nn(CC)c(O)c2)=O)CC2CCCC(C1)N(C(c1ccns1)=O)C2 C(CC(O)C(F)(F)F)NC(CNC(CN(C(CNC(C(C)C)=O)=O)C)=O)=O CCC(C)CC(C)C(=O)N1C2CC1CN(C(=O)CC1(C)CCOC1)C2 C(=O)(C1=NNC(C(F)(F)F)C1)NC1CC(CNC(c2c(C)coc2)=O)C(O)C1 N1(C(C(C(C)C)O)=O)CCOCC(C)(CNC(c2ccc(C(C)(C)C)cn2)=O)C1 C1(C(N2CC(OCCC(=O)N(C3(CN(C)C)CC3)C)C2)=O)C(C(N)=O)C1(C)C C1(NC(CC)=O)CN(C(c2ccc(C)c(C)n2)=O)C2(CCCOC2)C1 c1(C(N2CCC(O)(C(C)NC(c3ccnn3C)=O)CC2)=O)ccc(F)c(Cl)c1N CC(CCC(C)(C)C)C(=O)NCC1CCCCN1C(c1cnoc1)=O Cc1cnc(C(=O)NCC(CO)NC(c2csc(C)c2C)=O)cc1Br N1(C(C(F)=C(C)C)=O)CCN(C(=O)CCC(N)=O)C(CF)C1 C12(C(=O)NC3CC(CNC(C(C)NC(C4CCCC4)=O)=O)C3)CCC(C)(CO1)C2 c1(C(N(CCCCCCNC(C2COCCO2)=O)C)=O)cncc(C(C)(C)C)c1 C1(C(N2CCC(NC(c3c(CC)con3)=O)(CF)C2)=O)CCC(C2CC2)CC1 Cc1cc(C(=O)NCC2CCCN2C(=O)COCCF)c(C(F)(F)F)o1 C1(NC(c2c(CC)occ2)=O)COC2(CNC(=O)C(O)c3cnc[nH]3)CC1C2 C(C1CCC(NC(c2ccnc(Cl)c2)=O)C1)=CC(=O)O CC1(CNC(c2cc(=O)cc[nH]2)=O)CCN(C(=O)CNC(=O)CC(F)(F)F)C1 C12(CNC(C(C)SCC)=O)CC(NC(c3cnc(CC)[nH]3)=O)(C1)C(C)(C)O2 c1(CCC(=O)NCC2CCC(NC(COCC=C)=O)CC2)ccc(C(F)F)cc1 C1(NC(c2ccc(OC)cc2)Cc2cccc(OC)c2)CCC2(CNC2)OC1 C12(CNC(CCCNS(C)(=O)=O)=O)COC(CNC(=O)C(F)=C3CCC3)(C1)C2 Cc1cc(C(=O)NC2CCCC2CNC(C2CCCC23CC3)=O)nc(O)c1 Cc1c(CC(N2CC=CC(NC(c3cnns3)=O)C2)=O)ncn1C Cc1cc(F)ccc1CC(=O)NC1CC(C)(NC(c2ccc(Br)cc2C)=O)C1 c1(C(N2C(C)(C)C(NC(=O)CSCCC#N)CC2)=O)ccc(F)c(F)c1F CC1CC(NC(c2ccc(F)o2)=O)CCN1C(C1CC2CC2CC1C)=O c1(C(=O)NCCC2CCCN(C(=O)C=Cc3cc[nH]n3)C2)cc(O)nc(O)c1 C(=O)(C(O)C(C)(C)C)N1CC(C(N(C2(CN3CCOCC3)CC2)C)=O)C1 CCCC(C)CC(=O)N1CCCC(N(C)C(c2c[nH]nc2OC)=O)C1 Cc1ccc(C(=O)NOCC(=O)NCC2(O)CCC(C)(C)C2)nc1O C1(NC(c2cncc(N)n2)=O)CCCCN(C(c2cncc(C(F)(F)F)n2)=O)C1 O=C(C1=CCCCO1)NCc1csc(CNC(c2cccc(Cl)c2O)=O)n1 c1(CC(=O)NCCN(C(C2CC2C2CCC2)=O)CC)cccc(OC)c1Cl N1(C(CCCNC(C2CC(C)(C)C2)=O)=O)CCCN(C2CC2)CC1 c1(C(=O)NC(CC)CN(C(=O)CCc2ccn(C)n2)C)cncc(OC(C)C)c1 c1(CNC(=O)NC(C)CCC(F)(F)F)cnc2ccccn12 O=C(C1OCCn2ccnc21)NC12CC1CN(C(=O)CCn1ccnc1)C2 C1(C(=O)NC(c2csnn2)C)CC2(CCN(C(=O)CN3CCOC3=O)C2)C1 N1(C(COC)=O)CCC2C(C(=O)N(C(C)C(C)C)C3CC3)C2C1 c1(OCC(N2C3C(NC(COCC(C)(C)C)=O)C(C3)C2)=O)ccccc1[N+](=O)[O-] CC1CCC(CNC(=O)C=CC(C)(C)C)CN1C(=O)Cc1nnc(O)s1 C1(CNC(C(CCN(C)C)O)=O)(NC(=O)Cc2ccc(Cl)s2)CCCCC1C n1(CC(=O)NCC(CC)NC(C2Cc3nccnc3C2)=O)c(C)cc(O)cc1=O C(=O)(C(O)C1=CCCCC1)NC1CC(NC(C2CCC2(F)F)=O)C(O)C1 c1(COCC)nc(N2CCC(C(C)NC(=O)C(C)CCN(C)C)CC2)cc(Cl)n1 c1(OC)cccc(Cn2nnnc2C(c2csc(-c3ccsc3)n2)NC2CC2)c1 C(=O)(C(CCC1OCCO1)NC(c1ccncc1C(F)(F)F)=O)OC C1(NC(C(C)SCC)=O)CCC2(CCN(C(=O)C(CC)(CC)CO)C2)C1 C1(C(N(CCN(C(=O)C(F)(F)C2CCOCC2)C(C)C)C)=O)CC2CCCC12 c1(OCC)ccc(C(=O)NCC2(N(C(=O)C=CCO)C3CC3)CCOC2)cc1 N1(C(Cc2c(C)cc(Cl)nc2)=O)CC2CCN(C(=O)CSc3nncn3C)CC12 C(CC(C)C)(CC(C)C)NC(CCC(C)NC(c1c(OC)nn(C)c1)=O)=O N1(C(c2c(CC)cnn2C)C(=O)NCC2CCCO2)CCN(C)CC1CC(C)C c1(OC)ccc(CCC(N2CCC(C)(CC(=O)Nc3cc(O)ccn3)C2)=O)cn1 c1(OC)cncc(CNC(C2CCN(C(=O)C=Cc3cncn3C)C2)=O)c1 CCCCCCC(C)CC(=O)N1CCCCC(NC(=O)C(C2CCCO2)OC)C1 N1(C(CC=C=C)=O)CCC2(CC(NC(=O)C(C)CN(C)C)C2)C1 c1(SC)ccc(N)cc1C(=O)N(C)CC1(O)CCN(C(=O)C2CC2)CC1 c1(C(=O)OC)cc(CO)ccc1NC(N1CC(C(F)(F)F)CC1C)=O c1(C(=O)NC2(CCCC(=O)N3CC(C(CC)C)C3)CCC2)cc(O)ncn1 CC1CCN(C(C2CCC=CC2NC(=O)Cc2cnoc2)=O)CC1O c1(CN(C(C)CS(C)=O)C)nc2cc(Cl)ccc2n1C C(=O)(NN1CCCC1C(=O)NC1(C)CS(=O)(=O)C1)c1cc(C)c(C)o1 Cc1cc(N)c(C)nc1C(N1CC=CC(NC(=O)COC2CCOC2)C1)=O c1(C(C)C)c(C(=O)NCC2CC3CC3N2C(=O)CO)cnc2ncnn12 C1(C(N(CCCC#C)C)=O)(NC(c2[nH]cc(C)c2C)=O)CCC(C)(C)C1 C#Cc1ccc(F)c(C(=O)NCC2CCN2C(=O)C(F)C2CCCC2)c1 C=Cn1nccc1C(=O)NCC1(C(=O)NCC2CC2c2ccoc2)CC12CCC2 S(=O)(=O)(c1cccc(C(C)C)c1)Nc1c(C)ccc(C(=O)OC)c1 C12(NC(C34CC(COC)(OC3)C4)=O)CCC(CC1NC(=O)Cn1cc(C)cn1)C2 Cc1ccc(C(N2CC(NC(=O)CC34CCC(CC3)C4)CC(C)C2)=O)c(F)c1C c1(Cn2c(C(c3nnnn3C(C)C)NCc3c(C)ncs3)ccc2)cccc(F)c1 C(=O)(C(CCC(C)C)NC(c1ccc(C)n1C)=O)NCCC=C=C N1(CC2C3CN(C(=O)NCc4cn(C)nc4)CC32)C(=O)CCCC1=O c1(C(N(C2CCCN(C(=O)CS(=O)(=O)C3CC3)C2)C)=O)ccc2oncc2c1 CC(c1ccccc1)=CC(=O)N(C)CC1CCCN1C(=O)CCc1cnc(O)[nH]1 C1(NC(C2CCS(=O)CC2)=O)C=CCCC1C(=O)NC1CCC(O)CC1 Cn1cc(C(N2C(CNC(C3CCCC3O)=O)CC3CC23)=O)c2cccnc12 C1(NC(C(c2ccc(C)cc2)O)=O)CN(C(c2cnc(C)cn2)=O)C2(CCC2)C1 N1(C(c2c(Cl)cn(CC)n2)=O)CC2CC(NC(c3ncccc3OC)=O)CC2C1 C(=O)(CC(C)CCCCCC)N1CC(CCC)N(C(c2ccn(CF)n2)=O)CC1 c1(C(=O)NC(CNC(CC(C(C)C)OCC)=O)C)ccc(=O)n2c1CCCCC2 C12(C(=O)NCC3C4CN(C(C=CSC)=O)CC43)CCCN(CCC1)C2 CCC(Cc1ccccc1)C(=O)N1CC(NC(c2cc(=O)cc[nH]2)=O)C(F)C1 c1(C(CC)NC(C2(N(C)C)CNC2)=O)cc(F)ccc1F N1(C(C(=O)NCCCC)=O)CCC2CCN(C=O)CC2C1.c1(C(CN)=O)cnc[nH]1 C1(NC(C(CC)CN(C)C)=O)CC2CC1CN(C(C1(CCO)CC1)=O)C2 C1(CNC(C(N2CCCCC2=O)C)=O)CN(C(C2COCCO2)=O)CCC1C c1(OC)nc(N2CCC(C)(NC(=O)CC3CC(F)(F)C3)CC2)cc(C)n1 c1(C(N2C(C(=O)Nc3occ(C)n3)CSCC2)=O)ccc(Br)cc1C(F)(F)F C(=O)(CC(C)(C)c1cccc(Br)c1)N(CCCNC(C1C(C)C1C)=O)C C1(CC(=O)NCCOC2CCOC2)CCCN1C(C1CC1Cl)=O N#Cc1ncc(C(=O)NCCN(C2CCCCCC2)C(c2ccoc2Cl)=O)s1 CC1(NC(c2ncsc2Br)=O)CCN(C(=O)Cn2cnc(C#N)n2)C1 c1(NC(C2C(c3c(C)cccc3)C2)=O)nc2ccc(Br)c(C)n2n1 CC1CN(C(=O)C=Cc2ccc[nH]2)CCN1C(C1CC(=C2CCC2)C1)=O CCCCC(CC)CC(CC)(c1nnnn1C)Nc1cc(Cl)c(O)c(Cl)c1 N=c1ccc(C(=O)NCC2CCC2NC(C2CCC2(F)F)=O)c[nH]1 c1(N(CC(=O)N(C(=O)C(C)C(C)(C)C)C(C)C)C)nc2ccccc2s1.CC C1(NC(COc2cn(C)nc2)=O)CCC(C)(CNC(=O)C2=CCCCO2)CC1 c1(C(=O)NC2CC(NC(=O)CC3(CO)CCCC3)C2)ccc2ccncc2c1 c1(CN2C(C(=O)Nc3c(C(N)=O)ccs3)C=CC2)cnc2[nH]ccc2c1 C1(NC(c2c(CCC)nns2)=O)CCN(C(c2ccnnc2S)=O)CCC1CO C1(C(N2CC3C(NC(=O)C(O)C4CCCC4)(C3)C2)=O)CC2(CCCCC2)C1 C1(C(N2CC3(CN(C(CCCOCC=C)=O)C3)C2)=O)CC2COCCN2C1 c1(OC)ccncc1C(=O)NC1CC1NC(=O)CC(C)c1cccnc1 N1(C(COC2(C)CCCC2)=O)CC2(NC(=O)CCc3cncc(F)c3)CC1C2 N1(C(CC(C)F)=O)CCC2(CC1)CN(C(=O)Cc1cccc(C(F)(F)F)c1)C2 c1(CCC=C)n[nH]c(=NC(=O)c2cn(C)nc2OCC(F)(F)F)s1 c1(C(=O)NC(CNC(CC(C)CF)=O)(C)C2CCC2)cccc2ncccc12 C(=O)(CCCC(F)F)N(C)CC1CCN(C(C(C)O)=O)C1 C(CC(=O)N1CC(O)CCO1)C1N(C(Cc2cnc(C)s2)=O)CCCC1 c1(C(N2CCC(NC(C(C)C(C)(C)C)=O)C(C)(C)C2)=O)nn2cccnc2c1Cl c1(CC)ccc(OCC(=O)NC2(CNC(=O)CCNC(N)=O)CCCCC2)cc1 C1(C(N2CCC(CC)C2)=O)(CC)CCN(C(c2csc(CO)n2)=O)C1 N1(C(c2nc(C)[nH]n2)=O)CCCC12CCN(C(C1CC(C(C)(C)C)=NO1)=O)C2 c1(-c2c(C(=O)NCC3CN(C(CCC)=O)C(C)C3)cccn2)ccc(F)c(F)c1 c1(C(C(N2CCC(CNC(c3ccnnc3)=O)C2)=O)(F)F)cccc(Cl)c1Cl C12(NC(=O)NCc3c(N4CCCC(C(N)=O)C4)nccc3)CCC(CC1)CO2 CC(C)CC(C(=O)NCC1CC12CC2)ONC(=O)C(C)N1CCCCC1 CN=c1[nH]c(=NCC2(COC)CC2)[nH]c(=NC2c3ccc(F)cc3OC2C)[nH]1 c1(C(N2C(C)CCC(NC(CC(=O)NC)=O)C2)=O)cccc2c(C)c(C)[nH]c12 c1(CC)cc(NC(=O)CC(C)CNC(c2ncoc2C2CC2)=O)cc(C)c1 C1(CC(=O)NCC2(C)N(C(COC)=O)CCC2)CC(c2ccccc2)=NO1 C1(c2nnnn2C2(C)CC2)(NC2(COC)COC2)CCCC(C(=O)OC)C1 Cc1cc(C)n(CC(N2CC(C(C)NC(c3cnn(CC(C)C)c3C)=O)C2)=O)n1 CCC(CC(=O)N1CCCCC1c1cn(Cc2[nH]nnc2C)nn1)C(C)C N1(C(=O)Cc2ccc(Br)s2)CCC2(CCCN(Cc3c(Cl)cc(Cl)cc3Cl)C2)C1 c1(OC)cc(OC)cc(CN2CC3CC3(C(N3CCCCC3CCCO)=O)C2)c1 c1(OC)cc(CNC(C2C=CCN2C(=O)CCC2CCCC2)=O)ccc1F Cc1cccc(OC(C)C(C)NCc2ncc(C3OCCO3)s2)c1 C1(CNC(C2(C)CC2)=O)CC(CNC(c2cnoc2C2CCOCC2)=O)CO1 C(C1=NOC(C)C1)OC(C1(C(CC)=O)CC1)=O.C1C(F)C(=O)N1 c1(C(=O)NCC2CC2NC(C2CCOCC2)=O)cccc(F)c1F c1(OCC(N2CCC(O)C2c2ccc(Br)cc2)=O)cc(Cl)nc(Cl)c1 c1(CC)oc(C(N2CCC(CNC(C3CCC(=O)N3)=O)C2)=O)cc1C(=O)OC N1(C(C=C(COC)C)=O)CCOC2(C1)CN(C(c1cncc3c[nH]nc13)=O)C2 S(=O)(=O)(c1ccc(N2CCN(C=O)CC2)c(Cl)c1)NCc1c(C)cc(Br)cc1C c1(SC)ncc(C(N2CC3CC(NC(=O)CCc4ccsc4)C2C3)=O)c(O)n1 c1(C(=O)NCCN(C)C(c2cccc(F)c2)=O)ccccc1OC(C)(C)C C(=O)(CC(F)(F)C(F)(F)F)N1CCC(CCNC(C=Cc2c(C)cncc2)=O)C1 c1(NC(CC(C)OCC)=O)cccc(C(=O)N(C)CCN(CC2CC2)CC)c1 Cc1ccc(-n2nc(COc3ccc(C(C)(C)C)cc3)nc2-c2ccc[nH]2)cc1Cl N1(C(CCCC=C)=O)CCC2(NC(=O)CC3C=CCC3)CCCCCC12.CC=O N1(OC(=O)CC2COC3(CCCC3)O2)CC2(CC(NC(C)(C)C)c3nccn32)C1 N1(C(C(CC)NC(C)=O)=O)CC2CCC1CN2c1nccc(SC)n1 C1(C(=O)O)(CNCCc2ccc(C)nc2)CCCCCCC1 Cc1cnc(C(=O)NCC(C)CNC(=O)C(C(C)(C)C)n2ccnn2)cc1C#N C1(NC(CCC(=C)Br)=O)CC2(C1)CC(NC(=O)C(C)NC(=O)C(C)(C)C)C2 c1(CN(C(C2CCCN(C(=O)C(F)(F)COC)C2)=O)CC)ccc(O)cc1 c1(C(=O)NCCC2CCCN(C(c3sc(Cl)nc3Cl)=O)C2)cc(Br)c(O)c(Br)c1 C1(C(=O)NC(C2(CNC(=O)C(c3ccc(F)cc3)(F)F)CC2)C)CCS(=O)(=O)C1 N1(C(c2nccc(CC)c2)=O)CCC2C(CCCN2C(=O)CC2CNC(=O)C2)C1 N1(C(CC2C(CC)C2)=O)CCC(CC(=O)NCCC(C)C(C)(C)C)C1(C)C CC(CC(=O)N1CC(O)(CNC(=O)C=CCN2CCC2)C1)c1cnn(C)c1 c1(C2C(C(=O)NCC(c3cccc(Cl)c3)CO)CNC2)ncc2c(n1)CCC2 C1(N(C(=O)OC)C)CCCN(Cc2ccccc2)C1=O.c12nc(n[nH]1)NC2=O N1(C(CCNS(C)(=O)=O)=O)CCCC(C2CCCCN2C(=O)Cn2ccnn2)C1 c1(N2CCC(C)C2)nc(N(C)Cc2cc(Br)cn2C)c2c(n1)CSC2 c1(OC)ccc(CN2CCSCC2C(=O)NCC2CNC(=O)CO2)c(Cl)c1OC Cc1nc(CN2CCC(C)(NC(=O)C(C(C)C)N(C)C)CC2)ccc1C(C)O C1(C)(CNC(C2(COC)CCCO2)=O)CN(C(c2cc(Cl)cn2C)=O)CC1C N1(C(Cc2c(SC)cccc2)=O)CC(NC(c2cc(O)nc(Cl)c2)=O)CC(F)C1 CCC(C)CCCC(=O)NC(Cc1ccc(Cl)cc1Cl)C(=O)NCCOC(C)C c1(C(N(C(C)CNC(c2c(Cl)cccc2Cl)=O)C)=O)cc(F)cc2ccncc12 C(=O)(CC(C(F)(F)F)c1nccn1C)NC(CC)CNC(=O)CCOCC(C)C C1(C(N2CC(NC(C3=C(C)OCC3)=O)C(O)CC2)=O)CCOCC12CCCCC2 Cc1ncccc1CN1CCOCC1C(=O)Nc1cc(-c2cccc(Br)c2)no1 C1(NC(C(COC)C)=O)CN(C(C2(Cc3ccc(F)cc3)CCC2)=O)CC1O N1(C(C2CCN(C(=O)CC(O)C3CCCC3)C2)=O)CCc2c(F)cccc21 Cc1cc(C(=O)OCCCC2CC2C#N)c(Sc2ccccc2)s1 C(=O)(C(C)C(CC)CC)N1CC(NC(c2cc(CC)nc(O)c2)=O)C2(C1)CC2 N1(C(C2CCCN2C(c2cc(Br)no2)=O)=O)CCC(OCC2CCOC2)CC1 c1(CC)ccc(CC(C)C(N2CC3C(CNC(=O)CC4CSC4)C3C2)=O)cc1 C1(NC(=O)CCOCC(F)(F)F)CN(C(C2CCCNS2(=O)=O)=O)CC1C1CC1 c1(CN(C(c2c(F)ccc(C)c2)=O)C)cnn2c1CN(C(C1CC1(F)F)=O)CC2 N1(C(C2CCCN(Cc3onc(CCCC)n3)CC2)=O)CCOC2COCCC12 C1(NC(C=C(C)C(F)F)=O)CCCC12CCN(c1nccnc1C#N)CC2 N1(C(CCC(C)NC(CC2(CSC)CC2)=O)=O)CCn2c(cnc2C)C1 N1(C(C(CC)C)=O)CC(OC)CC1CNC(C1(Cl)CC1C(C)=O)=O CC(C)C(C(=O)NC1CCC(CCN)C1)NS(=O)(=O)C1CC1 C(=O)(CCCCC(=O)N1CC2(COC(CNC(=O)CSCC(N)=O)C2)C1)NC N1(C(C2CC(C#N)(O)C2)=O)CCc2ccccc2C1CNC(C1CC=CCC1)=O N1(C(C(=O)NC2CCC(C(=O)O)CC2)=O)CCC2NCCCC2C1 C(C1CCCCCC1)=CC(=O)NCC(C)(C)CNC(=O)COCCF c1(CC)ccnc(C(N2CCOCC2CNC(=O)CCN(C)CC)=O)c1 C1(C(=O)NC(C#C)CCC)CCN(C(=O)C2=CCCCC2)CC1C N1(C(C(C)OCCC#C)=O)CCN(C(=O)C(C)(C)CF)CC1C1CCCC1 C1(C(=O)NCC(CNC(C(CCC)OCC)=O)CO)Cc2cscc2C1 N1(C(CCC#C)=O)CCCN(C(c2c(F)cccc2F)=O)CCC1 C(CC(CC)C(=O)N(C)CC1(NC(c2oc(C3CC3)nc2C)=O)CC1)=CC C1(CC(=O)NCC(=C)Cl)(OC)CC2NCCC12 c1(C(=O)Nc2cnncc2Br)[nH]c2ccccc2c1-c1cn[nH]c1 C1(=O)CCCCCOC2(CCOCC2)N1.C(CCOC)SCCN(CC)CC N1(C(C2C(C)(C)C2(C)C)=O)C(C(=O)NC(C2CCOC2)CO)CCC12CC2 C1(NC(C=CCC(C)(C)NC(c2c[nH]nc2Cl)=O)=O)CC2CC1CC21CC1 Cc1c(C(=O)NCC2CC2NC(=O)C2=COCCO2)nc2sccn12 C1(NC(c2scc(C)c2)=O)CCCCC1C(=O)NCCC1CCCCC1O C(C(=O)NC(C)(C)CCNC(=O)CC1CCCN1C)(C(F)(F)F)OC(C)=O C1(NC(CCN(C)C)=O)(CNC(c2coc(C3CC3)n2)=O)CCC(F)(F)CC1 N1(C(C(=Cc2ccccc2)OC)=O)CCN(C(C2CCNC2=O)=O)CC1CO C1(O)(CNC(C2CC(C)(C(=O)OC)C2)=O)CCN(C(c2cn(CCO)nn2)=O)C1 N1(C(c2ccc(OC(C)C)cc2)=O)CC2CC(NC(=O)CCCN=[N+]=[N-])C1C2 C1(c2n(C)cnc2)CN(C(C2CCCO2)=O)CC1NC(c1ccc(C2CC2)s1)=O Cc1ncnc(C)c1OCC(=O)N(C)CC1(NC(c2ccoc2C)=O)CC1 c1(C(=O)NCCN(C(C2CCCC2)=O)CC)ccoc1C(F)(F)F N1(C(CNC(CCC)=O)=O)CC2(CCC2)CC1C(=O)NC(c1ccc(C)nc1)C c1(C(=O)NC(C2CCCC2)CNC(CN(CCC#C)C)=O)c(N)sc2c1CCC2 C1(NC(C(C)SC)=O)CN(C(=O)CCc2ccc(F)cc2F)CC12CCC2 c1(NC2C(OC)CCOC2)nc(N(CC(C)(C)C)C)nc2c1cnn2C c1(OC)cc(F)c(C(c2nnnn2-c2ccc(Cl)cc2F)NCC(N)=O)cc1Br Cn1cc(C(=O)N(C2CCCC2)CCNC(C2C3CC3C3CC23)=O)c(O)nc1=O C1(NC(C(C)(C)CO)=O)CN(C(=O)CCn2cncn2)CC2CCCC12 C(CSC)(C(=O)N1CC(C(C(=O)N(C)Cc2cc(C)cs2)OC)C1)OC C1(CC)CCOC2(CCN(C(=O)CCC(=O)N(CC)CC)CC2)C1.C1(C)C(=O)N1 c1(C(N2C(C(C)NC(c3nc(C(C)OC)sc3)=O)CCC2)=O)cc(C)c(F)cn1 c1(CNC(CCSC)=O)cccc(C(=O)NCC2CN(C)CCO2)n1 c1(CN2CCC(F)(CNC(c3c(C)cc(Br)cn3)=O)CC2)ccc2n[nH]cc2c1 C(=O)(C(=O)N1CC(OCCC(=O)N(CCN(C)C)CC)C1)NCC.C(C(F)F)N c1(OC)c(Br)ccc(CNC2CCC(C(=O)Nc3ccc(C#N)c(Cl)c3)C2)c1F C1(NC(CCC(=C)Cl)=O)CCCC12CN(C(=O)C(C)OC)C2 C1(CNC(c2cnc[nH]2)=O)C2CCC(C2)N1C(=O)C=CC1CCCCC1 C1(C(=O)NCCCOCCNC(CC2CC(OC)C2)=O)CCCC2CC12 O=[N+]([O-])c1cc[n+]([O-])cc1NCc1cnc(C(F)(F)F)c(F)c1 CN1C(=O)CSC1=CC(=O)NCC1CC2(C1)CN(C(C13CSCC1C3)=O)C2 CC(C)S(=O)(=O)CC(=O)N1CC(NC(=O)CCS(=O)(=O)N(C)C)CC(C)C1 C1(C(=O)NCCN(C(C(CC)NC(N)=O)=O)CCOC)CCCC1(C)C c1(C(N2CC(N(C(C3C(=C)C3C(=O)OC)=O)C)C2)=O)ccc(F)c(C(F)(F)F)c1 C1(C)(C(N2CCC(N(CCC)C(c3ncoc3COC)=O)C2)=O)CCC(=O)N1 c1(-c2cc(C(=O)O)cc(OCC(=O)N(C)C)c2)ccc(C(F)(F)F)c([N+](=O)[O-])c1 N1(CC(C)NCCc2ccccc2C(=O)O)C(=O)c2ccccc2C1=O C1(NC(=O)CCCNC(c2ccsc2)=O)CN(C(=O)Cn2cccc2)C2CC12 C1(C(N(C2CCCN(C(C=CCCC)=O)C2)CC)=O)Cc2ccc(F)cc2C1 C1(C(=O)NCC2CC(NC(c3cc(F)cc(F)c3)=O)C2)CNc2ccnn2C1 c1(C(=O)NC2CC(F)(CNC(C(C)NC(=O)NC)=O)C2)nn(C)cc1[N+](=O)[O-] C1(C(=O)OC)CC(C)CN(C(c2cccc(-c3ccc(C(=O)O)cc3)c2)=O)C1 N1(C(c2ccn(C(C)C)n2)=O)CCC(C2CCCN(C(=O)C=CC(N)=O)C2)CC1 CCC(O)CC(=O)NC1(C(N2CCN(C(=O)CC)CC2)=O)CCSC1 C1(CC)CN(C(c2cccc(N)c2O)=O)CCN1C(=O)CC(C)c1cccnc1 N1(CC(N2C(CNC(C(CC=CC)C)=O)CCCC2)=O)CCCC2(CC2)S1(=O)=O c1(OC2(C(=O)NC(CC)CNC(C3CC(C)=NO3)=O)CC2)cccc(F)c1 C[Si]1(C)CCC(c2ccccc2)(CNCc2cccc3occc23)CC1 C12(Nc3cc(CC)ncn3)CCCC1CN(C(C1(F)CC3(CCC3)C1)=O)C2 CCC(C(=O)N1CCCCC1C(N1CCCC(O)CC1)=O)C(C)(C)CC N1(C(c2c(CNC(CC3(N(C)C)CC3)=O)cco2)=O)CC(C)(CO)CC1(C)C N1(C(C2(C=C)CCOCC2)=O)CCN(C(=O)C(CC2CCCC2)CC)CCC1C c12ccc(cc1C#N)S(=O)(=O)NCCN2.CC1COCCN1C(=O)OC(C)(C)C c1(C(N2C(CN(C(CC(CC)SC)=O)C)CCC2)=O)ccc(S(=O)(=O)NC)o1 CCC(C)(C)C(O)C(=O)NC(CCF)C(=O)N(CCCN(C(C)C)C(C)C)C c1(NC(C)=O)ccc(C(=O)NC2CCC(C)N(C(=O)C(=O)NC(C)C)C2)c(Cl)c1 c1(C(=O)NC2C(CNC(C(C)OCC)=O)CC2)cnnc(C2CC2)c1 CCC(C(=O)N1CCC(N(C)C(c2[nH]c(C)nc2C)=O)CC1)C(C)O C#CCCCC(C)C(=O)NC(CN(C)Cc1ccccc1)C(=O)NCC(C)C#N Cc1cc(N(C)CCN(C(c2cn(C3CCOCC3)nn2)=O)C(C)C)nc(Cl)n1 C1(C(N2CCC(CC(C)NC(C3CC(=O)N(C)C3)=O)CC2)=O)C(F)(F)C12CCC2 c1(C(c2noc(-c3sc(Cc4cccc(F)c4)nc3Cl)n2)C)cccc(OC)c1 Cn1nc(C(F)(F)F)c(CN2CCC3(CC3C(N3CCC(C)(C#N)C3)=O)C2)c1Cl C(=O)(CCC(CC)OC)N(C(C(=O)NC(CCCC)CC)C)CCC c1(C(N2CC(NC(C3(CCC)CCC3)=O)C(C)CC2)=O)oc2ccccc2c1Cl C12(NC(CCOC)=O)CCCCCC1N(C(=O)CCc1ncccc1C)CC2 N1(C(C(=O)NCCC)C2CC2(C)Br)CCC(C2CC2)C1 N1(C(CCC(C)NC(CN(C(=O)OCC)C)=O)=O)CC2(CC(C)CO2)C1 C(=O)(C(C)(CC)C(=O)N(C)CCN(C(=O)C1=NOC(C)(C)C1)C)OCC c1(OC)cccc(OC)c1C(N1CC(C(C)NC(=O)C=C(C)C(C)C)C1)=O C(C(=O)NCC1CN(C(=O)Cc2ccn(C(C)C)n2)CC1O)(C(C)(C)C)OC Cc1cc(C(=O)N(C2CCCN(C(=O)CCN3CCNC(=O)C3)C2)CC)n(C)n1 C1(CNC(NCC(C)(C)C)=NCC2CCCSCC2)CC2(C1)C(F)(F)C21CC1 C1(C)(CC)C=C(C(=O)N2CCC(O)(CCNC(=O)CCC(F)F)CC2)C1 c1(COC)ncc(C(=O)NC2CCCC2CNC(=O)CCc2ccn(C)n2)s1 N1(C(C2(c3cc(OC)ncc3)CCC2)=O)CCN(C(C)=O)C(C2CCC2)C1 N1(C(C#CC(C)C)=O)CCC(O)(CN(C(=O)COCC2CCCC2)C)CC1 c1(OC)ccnc(OC)c1C(=O)NC1CC2CC1N(C(=O)C=C(C)Cl)C2 C(=O)(CC(O)C(Cl)(Cl)Cl)NC(CC)CN(C(=O)C=Cc1ccc(C)nc1)C C12(NC(C3N=C(C)SC3)=O)CCCN(C(c3ccncc3OC(C)C)=O)CC1C2 C1(C#N)(CNC(C(Cn2ccnn2)NC(C(C)SC(C)C)=O)=O)CCCCC1 C(=O)(C(C)C(O)C(C)C)NC1CCCC(CN(C(c2cc(C)ncc2C)=O)C)C1 c1(C(=O)NCc2cc(OC)nn2C)ccc2c(n1)CN(C(C1CCO1)=O)CC2 c1(COC)ccc(Cl)c(F)c1Cl.N12CC(CC(F)C1)C(=O)Nc1ncc(cn1)C2 N1(C(CNC(C)=O)=O)CCC(C(C)NC(C2CCCN2C(C)=O)=O)C1 c1(C(=O)NCCC(=O)NC(C)(C)C=CC(=O)NCCC2CC2)ccc(O)cc1 C(C(CC(=O)N1CC=CC(O)C1)C1CCC1)NC(C(CC)OC1CC1)=O N1(C(c2ccc(C#C)nc2)=O)CC(NC(=O)CCC(=O)NC2CC2)CC(C)(C)C1 C1(N(C(c2ccccn2)C)CC2CCC3(CC3)C2)CCN(S(C)(=O)=O)CC1 N1(C(Cc2nc(CC)sc2)=O)CCC(NC(c2n[nH]cc2Cl)=O)C1(C)C c1(CC(=O)NC(C)CCNC(C2CC2(Cl)Cl)=O)cccc2ccccc12 C(=O)(C1=CC2(CN(C(c3cn(CCO)nn3)=O)C2)OC1)N1C(CO)CCC(C)C1 c1(NCCNC(C(CC(C)C)NC(C)=O)=O)ncnc2c1nnn2C1CC1 CCC(C(=O)N(C1CCN(C(=O)CC2(N(C)C)CC2)CC1)CC)C(F)(F)F n1(CCC(C)C)cc(C(N2CC(O)(CNC(=O)COCc3nc[nH]n3)C2)=O)nn1 CN1N=C(CC(=O)NC2CC3CC(NC(C4CCC(C)(C)OC4)=O)CC23)CC1=O C1(C(N(C)Cc2cn[nH]c2)=O)COCCN(C(=O)C2=CCCOC2)C1 c1(C(N2CC(OC)(CNC(=O)Cn3nc(C)cc3C)C2)=O)cnc2c(c1)CCC2 Cc1cc(C(=O)NC(c2ccccc2)CC2(O)CCCCC2)nc(S(C)(=O)=O)n1 c1(N(C)C(C2CNCCC2(F)F)C2CC3(CCC3)C2)ncnc2c(Br)c[nH]c12 C1(C)(CC)C=C(C(=O)NCCN(CCCN(C)C)C(c2[nH]c(C)nc2C)=O)C1 CC(C)CC(CNC(c1ccoc1)=O)NC(=O)C(C)OC1COC1 Cc1nn(CO)c(C)c1Br.c1(CN(C)C(c2ccc(C(=O)O)cc2)=O)cccc(CN)c1 c1(CNC(c2cscn2)=O)cccc(C(=O)NC2CCC(F)CC2)n1 c1(C(=O)NCCOC(CNC(C(C)=C(C)C)=O)(C)C)csc(C)c1C n1(CC)nccc1C=CC(N1CCOCC1CNC(C1CC1CCOC)=O)=O CC1(C#CC(=O)NC2CN(C(=O)C(O)c3cnc[nH]3)C2)CCCO1 C(=O)(C1=CC2CCC(C1)C2)NCCC1CC(NC(CSc2n(C)ccn2)=O)C1 C1(C(N(C)CC2CCN(C(CCCC#C)=O)C2)=O)CCC2(CCOCC2)O1 c1(C(=O)NC2CC3(CN(C(CC(=O)NCC)=O)C3)OC2)cnc2snc(C)c2c1 C(C(O)CC(=O)N(CCCN(C)C(C1CC(c2cccc(Cl)c2)C1)=O)C)N(C)C C=Cc1cncc(C(=O)NCC2CN(C(c3conc3CC)=O)CC2C)c1 C1(NC(C(CSC)OC)=O)C2CCN(C(c3cc(OC)cc(OC)n3)=O)CC12 CC1(C(=O)NCC2C=CCC2)C=CCN1C(c1cc(C#N)c[nH]1)=O N1(C(c2c(C)csn2)=O)CC(C(=O)NCC(c2ccncc2)C)C2(CC2)C1 CCC(CC(=O)NC(Cc1cn(-c2ccccc2)nn1)C(=O)OC)C1CCC1 C(c1ccc(Br)cc1)=CC(=O)NCC(C)(C)CCNC(=O)C1=CCC1 CCC(C)(C)C(=O)Nc1ccsc1C(N1CCCC1COC)=O CC1C2CCC(C2)C1C(=O)NCCCN(C(=O)C=Cc1ccc[nH]1)C CC1CCC(Cl)=C(C(=O)NC2C=CCN(C(=O)CC3CC(=O)C3)C2)C1 Cc1nc(C#N)c(NCCC(=O)NC(C)CNC(=O)C(C(C)C)c2ccco2)o1 c1(OC)cc(C(=O)NC2COCCC2NC(=O)CCC(C)(F)F)ccc1C#N N1(C(C(C)N(C(C)=O)C)=O)CC2(COC(CNC(C34CCCN3CCC4)=O)C2)C1 C(=O)(C1=CCOCC1)NCC1C(NC(CC2C(C)C2)=O)CCC1 c1(OC)ncc(C(=O)NCC(C2CCCN2C(C2CC2CN(C)C)=O)(C)C)s1 c1(C(=O)NC2CCN(C(CC(C)C3CCCCC3)=O)C2)cc(F)c(F)cc1Cl C1(CNC(C2C(CCC)C2)=O)(NC(c2cccc(NCC)c2)=O)CCCCC1 N1(C(c2ccc(CC)cc2F)=O)CCCN(C(C2CC2C(F)F)=O)CCC1 n1(CC)cc(NC(=O)CC2CCCN2C(=O)Cc2n[nH]c(C)n2)c(C)n1 N1(C(c2cnc(C)nc2C)=O)CC2CCCC(NC(=O)C=Cc3ccco3)C2C1 CON(CC1CCCCC1)C(=O)C1(CNC(c2cn(C)c(C)n2)=O)CCCO1 c1(C(N2C(C(=O)NCC3(CCOC)CC3)CSC2)=O)cn(C)c(=O)n1C c1(C(=O)NCC(CC=C)NC(C2CC(C(=O)OC)C2)=O)cc(C)ccc1Br c1(COC(c2cccc3occc23)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 c1(C(=O)NCC2N(C(c3scc(C)c3)=O)CCC2C)ccc2ccccc2c1 n1(CC(=O)NC2C(NC(c3c(C)oc(Cl)n3)=O)CCC2)ccc(=O)n(C)c1=O C1(O)(CNC(C2(O)CCCC2)=O)CC2CCC(C1)N2C(C1(CO)CC1)=O c1(C(=O)N(C2CCCC2)CCNC(C2CCOC2)=O)ocnc1C1CC1 C1(CC(N2CCC(CCNC(c3cscn3)=O)C2)=O)Cn2ccnc2NC1=O CCCC(O)CC(=O)NCC1CC(O)CN1C(c1cc(Cl)cnn1)=O C(=O)(CC1=NNC(=O)C1)NC(CC)CN(C(=O)CCn1c(C)csc1=O)C N1(C(C2(CC)CC2)=O)CCC(CO)(CNC(=O)C(C)(O)Cn2ccccc2=O)C1 C(=O)(C1=NOCC1)NC1(CC=C)CN(C(C2CC23CC(OCC)C3)=O)C1 Cn1cc(CC(N2CC3CC2C3NC(c2cocn2)=O)=O)c2ccccc12 N1(C(c2ccc(C)o2)=O)CC2(CCCC2NC(=O)COCC(=O)NCC(N)=O)C1 C12(CNC(Cc3cccc(COC)c3)=O)CCC1CN(C(C1(C#N)CC1)=O)C2 C1(OC)CCC2(C(=O)N(C3CCCCC3N(C)C(C3C4COCC34)=O)C)CC12 C1(C(C(=O)OC)O)CCN(C(=O)Nc2cccc(-n3cncn3)c2)CC1 C(CNC(c1ncoc1C(C)C)=O)(C(C)(C)C)NC(C1C(CC(C)C)C1)=O Cc1cc2nc(Cl)[nH]c(=NCC(C3CC3)NC(c3cnc(Cl)cn3)=O)c2s1 O=S(=O)(c1cccnc1NCCc1cc(Cl)ccc1F)NC(CO)CCF n1(CC(N2CCC(SC)CC2)=O)ccc2ccc(-c3ccc(F)cc3C#N)cc12 c1(NC(=O)CC2CCC2)ccc(CO)cc1O.C12(CO)CCCN(C1)C2=O N1(C(C2ON=C(C)C2)=O)CCCC(C)(NC(c2cc(Cl)c(Cl)s2)=O)C1 N1(C(c2n(C)cc(C(N)=O)c2)=O)CC(NC(=O)CCC(C)(C)C)C2(CCC2)C1 c1(C(=O)NC(CNC(c2cccc(N)c2)=O)CO)cc(F)cc(F)c1 C1(C(=O)NC2(C)CC(NC(CC(=C)C)=O)C2)CN(C)CCO1 C1(C(=O)NC(C2(O)CN(C(=O)Cc3cnc[nH]3)C2)C)CCC2(CCC2)C1 C1(N(C(=O)Cc2cc[nH]n2)CC)CCCN(C(c2ocnc2C2CC2)=O)C1 c1(C(C)(C)C)ccc(SCC(N2CC3CC2C3NC(C2(F)CCOC2)=O)=O)cc1 O=C(CCCCCn1cc(CC2C3CCCCCC23)nn1)N1CC2(CCOC2)C1 CC1CCN(C(C2C3CCC23)=O)CC1N(C(=O)CCC(N)=O)C c1(C(N2CCOCC2(C)C2CC2)C(=O)NC(CC)C)ncc(Br)cc1C C=CC(C)(CC)C(=O)N1CC(CNC(=O)COCC2CC2)C(SC)C1 C1(NC(c2n(CCC)ccc2)=O)CCN(C(C2C=C2C)=O)C12CCCC2 N1(C(CC(CC=C)NC(C2CC(=O)NC(C)C2)=O)=O)CCC2(CC1)CN(C)C2 Cc1ccc(Cl)c(N)c1C(N1CC2OCC(NC(=O)CCc3cccs3)C2C1)=O N1(C(Cc2cn(C)nn2)=O)CCCC(CNC(C2(C#N)CCC2)=O)C1 c1(CC)nc2ccccc2cc1NC(=O)C(N1CCC2CCCCC2C1)=O Cc1ccc(S(=O)(=O)N(CC(N2CC3(CC(NC(=O)C(C)O)CO3)C2)=O)C)cc1 N1(C(c2cc(OC)no2)=O)CCC(CC(C)NC(C23CSCC2C3)=O)CC1 C1(F)(CNC(C2C(CC)C2)=O)CN(C(C2CCN2S(C)(=O)=O)=O)C1 c1(NC(C2C3CN(Cc4ccc(-c5ccc(F)cn5)s4)CC23)=O)cccc(Cl)c1 C(C(C)(O)C(C)(C)C)NC(C1(C#C)CN(C(=O)C2=NOC(C)C2)C1)=O C1(C(N2CCCC(C)(O)C2)C(=O)NC(C(=O)OC)C)CC2C(C1)C2(F)F Cc1cccc2c1CC(C(=O)Nc1cc(F)cc(F)c1CO)N2 C1(CNC(C2(C)CCCCO2)=O)CCN(C(c2nnc(O)cc2O)=O)CC1(F)F C1(NC(C2C(C)(C)C2)=O)CN(Cc2ncccc2F)CC1F C#Cc1cccc(CNC(=O)NC(CN2CCCC2)CC)c1F N1(C(CSC(C)C)=O)CCC2(CCN(C(C3CCc4n[nH]cc4C3)=O)CC2)C1 C1(N(C(c2ccc(CC)[nH]2)=O)C)CCCN(C(=O)C(C)Cc2ccccc2)C1 CC(C)CC(C(=O)NC1CN2CCCC1C2)ONC(=O)C(O)C1CCCC1 Cc1ncc(CC(=O)NC2(CNC(C3COC(=O)N3)=O)CC2)[nH]1 c1(C(=O)NC2(CC(=O)NCC(CC(=O)NC)C)CCC2)cncc(F)c1C C1(NC(C(CC)OC)=O)C2CC3CN(C(C4(CC)CC(OC)C4)=O)C1C3C2 c1(C(N(C2CN(C(C=CC=CC)=O)C2)C)=O)c[nH]c2ccc(OC)cc2c1=O c1(C(N2CCC(C(C(=O)NC(C(=O)NC)C)C)CC2)=O)cc([N+](=O)[O-])ccc1C N1(C(c2cc(C(C)C)on2)=O)CCC(CNC(=O)Cn2cc(CO)nn2)C12CC2 N1(C(C2OCCC(C)C2)=O)CC2(CC2)CC1C(=O)NC1CC1CN(C)C c1(C(=O)O)cc(Cl)c(O)c(S(=O)(=O)N2CC3CC2CN3c2ccncn2)c1 C(=O)(CCN(C(=O)CNC(N)=O)CC1CC1)NCCCCC C1(O)(CNC(c2cc(C)n(C)c2)=O)CCCN(C(c2ccc(C(F)(F)F)s2)=O)C1 c1(-c2cn(CCCCNC(=O)COC3CCS(=O)(=O)C3)nn2)ccc(Cl)c(F)c1F CCCCCC(F)C(=O)NCC(=O)NCC(=O)NCc1cnn(C(C)C)c1 CC(CN=C(NC1CCC1)N(C)Cc1ccc2c(c1)OCO2)C(C)(C)C c1(C(=O)NCCC2(NC(c3ncc[nH]c3=O)=O)CCC2)cc2n(n1)CC(F)C2 Cc1cc(C(=O)NC(Cn2ccnn2)C(=O)N2CC3CC3C2)cnn1 S(=O)(=O)(c1ccn(C)n1)N1C(C)CN(C(=O)CO)CC1 C1(C(=O)NCC2C(C)CN(C(=O)C=CBr)C2)C2C3CC4C1C1C2CC3C41 C(=O)(C(O)(CN(C)C)C(F)(F)F)N1CC(CNC(c2c(OC)scc2)=O)C1 N1(C(C=C(C)Cl)=O)CCC2CN(C(=O)CCn3cncn3)CCC2C1 C(c1ccncc1)=CC(=O)NC1(CC=C)CN(C(=O)C(C2CCOC2)OCC)C1 C1(NC(C(C)OCC#C)=O)CCN(C(c2cc(F)c(Cl)cc2F)=O)CC1(C)C N1(C(c2nc(C)c(Br)cc2)=O)CCC2CN(C(c3[nH]nnc3C)=O)CC2C1 C(CC(C)CC)(C(=O)NC(c1nccc(O)n1)C)NC(C1CC(CCC)C1)=O N1(C(c2n(CC)nc(C)c2)=O)CC(C(=O)NCc2ccnc(C#N)c2)CC1(C)C C1(C(=O)NC(CC)C(N)=O)CN(C(c2ccc(O)cc2)=O)CC1F C#CC1CN(C(c2nccn2C)=O)CCN1C(c1csc(C(C)=O)n1)=O Cc1c(C(N2CCOC(c3cccc(F)c3)C2)=O)[nH]c2ccccc12 C(=O)(C(C)(C)C(C)C)NCC(C1CC1)NC(C1CN(CC(C)C)C(=O)C1)=O C1(C(=O)NC(C)C=CC(=O)NCC(=O)N(C)O)CCCC(=O)CC1 CC(C(C)(C)NC(c1cnn(CCO)c1)=O)NC(=O)CCOC1CCOC1 C1(NC(=O)C2=CCCCC2)CCN(C(=O)C2=CCOC2)CC(O)C1 c1(C2(C(=O)NC3CCN(C(COCCC#C)=O)C3)CC2)ccc(F)cc1O CCCC(C)(CC)C(=O)NC(CN(C(=O)C(=O)NCCNC(C)=O)C)CC Cc1ccncc1C(=O)N(C)CC1CCN(C(=O)Cc2cncc(F)c2)C1 c1(CC=CCOCCNC(CCOCCOCC)=O)ccncc1 N1(C(C(C)n2ccnc2)=O)CCC2C(CCCN2C(c2cc[nH]c(=N)c2N)=O)C1 C1(C)(CC)CC(C(=O)NCC(C2CCCN2C(=O)CSC(F)(F)F)(C)C)C1 C(=O)(C(=O)CCC(C)C)N1CCC(C(C)NC(c2c(C)nn(CCO)c2)=O)C1 n1(CC)nc(CCCN2CCCCC2)nc1C1CC1F c1(C(N(CCOCCN(C(CC)=O)C)C)=O)cccn(C(C)(C)C)c1=O N1(C(C(c2cncnc2)C)=O)CCC(C)(C)C1C(=O)NC1CC2CCCCC12 C1(NC(C(CC=C)NC(=O)CC2CCOC2=O)=O)CCCCCC1C(N)=O C1(C(=O)NCCCN(C(C(C(C)C)C)=O)C2CC2)CCN(C)S1(=O)=O C1(C(=O)Nc2cn(CC)nn2)CCN(Cc2c(Br)cncc2Br)CC1O Cc1ccc(O)c(C(N2CCC(CNC(=O)CC(C)C3CC3)C2(C)C)=O)c1 C1(NC(c2c(CC)c[nH]c2)=O)CC2CCC(C1)N2C(C1CCC(=O)N1C)=O C1(C(N2CCC(C)(NC(C3CCC(C)(C)C3)=O)C2)=O)(COC)CCCCC1 C#Cc1cc(C(=O)NC2CCC2NC(C2CCCCN2CCCC)=O)cc(F)c1 Cn1c(=O)ccn(CC(=O)NC2C=CCN(C(C3CCNC3=O)=O)C2)c1=O C1(CN(C)C(C2(N(C)C)CC2)=O)CCN(C(=O)NC(C2(C)CC2(F)Cl)=O)CC1 C(=O)(CCCCCNC(c1cnn(C)c1)=O)NC(CC(=O)NC)C N1(C(COC)=O)CCC1CNC(C1CC1C)=O c1(CC)c(C(=O)N(C(CNC(=O)CC(C)C(=O)OC)C2CC2)C)cccc1C CC(C(=O)N(CC(C)CNC(=O)COCC1CCOC1)C)OCCN(C)C C1(CC(N2CCC(Cc3ccsc3)C2)=O)CCCCN1C(=O)CSCC(F)F c1(C(C(=O)NCCN(CCC)C(C2CC2C#N)=O)(C)C)c(F)cccc1F N1(C(C2C(=C)C2)=O)CCCCC(C2CN(C(=O)C(O)C(C)CC)C2)C1 c1(C(=O)NCCCCC=C)ccc2c(c1)CN(C(=O)C=CCC)CC2 c1(OC)cccc(C(C)CC(=O)N(CC(C)CNC(c2ncccc2F)=O)C)c1 C1(CC(=O)NCCC(C)NC(c2cn3c(n2)SCC3)=O)CC2C=CC1CC2 C(=O)(C1CCCc2ccnn21)NC1C(NC(C(C(C(C)C)O)C)=O)CCCC1 C1(C(=O)NCC(CCOC)NC(=O)C=CCN2CCOCC2)CC2(CCCO2)C1 C1(C(=O)NCCC(C)NC(C(CC)NC(C)=O)=O)CCC2(CC2)C1 N(C1CCCc2ccc(Cl)cc21)Cc1c(O)cccc1O S(=O)(=O)(c1cc(C(=O)O)co1)N1CCN(C(=O)C(O)CC(F)F)CC1 C1(NC(C(C2(O)CCCCC2)NC(=O)CCCF)=O)CCN(C2CC2)C1=O CCCC(O)C(=O)NC1CN(C(=O)CN2CCC(O)CC2)CC1CC c1(NC(CN(C(C2CCC(C(C)C)CC2)=O)C)(C)C)ncc([N+](=O)[O-])cc1Cl CC1(NC(c2ccnc(-c3ccco3)c2)=O)CC2CCC1CC2=O C1(C2CCC2)(C(=O)NC(CCCNC(c2n(CCOC)ncc2)=O)C)CC1 N1(C(C(C)N(C(c2cnc(CC)o2)=O)C2CC2)=O)CC2C(C)C2C1 CN=c1nc(C(=O)NCCCCNC(c2cncn2C)=O)cc(C)[nH]1 C1(CNC(C(CSC)OC)=O)(CNC(C2(C(C)C)CCOCC2)=O)CC12CCC2 c1(NCc2ccc(OC)c(N)c2)cc(=NCC2(SC)CCC2)[nH]cn1 N1(C(C(CC)(C)OCc2ccccc2)=O)CC(S(=O)(=O)N(C)C)C1 c1(C(=O)NC2CCN(C(CC(C)OC)=O)C2C(C)C)ccc(Br)c(F)c1C C#CCCCC(C)C(=O)NC(COC)C(=O)Nc1cccc(OC)c1C c1(C(N2CC(C(C)NC(C3(C(F)(F)F)CCC3)=O)C2)=O)nn(C(F)F)cc1Cl C1(Nc2cnc3cc(C)nn3c2)C2Cc3cc(F)ccc3C12 C(=O)(C(C)(C)C(N)=O)N(C)CCN1CCN(C(=O)Cc2ccccc2F)CC1 c1(C(N(CC(CC)NC(=O)C(C)=CC(C)(C)C)CC)=O)cnc(O)nc1O N1(C(C2(SC)CC2)=O)CCC2CN(C(=O)C(C)OCC3CCCO3)C2C1 CCC(C(C)C)C(C(=O)Nc1cccc(OC)c1)N1CCSC(C)C1 C(CC(C(C)C)NC(=O)CC1CC(C2CC2)C1)N(C(C(C)SC(C)C)=O)C C1(O)(CN(C)C(c2ccc(SC(F)(F)F)s2)=O)CCN(C(C2(C3CC3)CC2)=O)C1 Cc1[nH]c(=N)ccc1C=CC(N1CCC1CNC(c1cc2c([nH]1)CCCC2)=O)=O N1(C(C(C(=O)OCC)(C)C)=O)CC2(CCCC(CNC(=O)CC3(C)CCC3)O2)C1 C=C=CC1CCN(CC(=O)Nc2sc3c(c2C(N)=O)CCC3)CC1 CCCCC(F)C(=O)NCCCC(O)C(=O)NCC1CC2(CCC2)CO1 C(C(C)C(C)C(=O)NC1COCCN(C(=O)Cc2c(C)noc2Cl)C1)OC c1(OCc2scc(C(=O)NC(C)CCCNC(=O)C(N)=O)n2)cccc(F)c1 c1(C(N2C(CNC(C(CCC)C)=O)C=CC2)=O)ccc([N+](=O)[O-])c(N(C)C)c1 S(=O)(=O)(c1cnccc1N1CCCC2(CCCC2)C1)NC(C)CCN(C)C Cc1ccc(-c2ncc[nH]2)cc1C(=O)NCc1cc(C(N)=O)co1 Cc1cc2c[nH]nc2c(C(=O)NCC(C)CNC(C2C(C)C2C)=O)c1N N1(C(C2CC(=O)NCC2)=O)CC2CC(NC(C3CCC4(C3)CC4(F)F)=O)C(C2)C1 C1(C)(C(=O)NCC2N(C(C3N(C(C)C)C(=O)CC3)=O)CCCC2)CCN(C)CC1 c1(CNC(C2(CO)COC2)=O)nc2c(s1)CCN(C(C1CC3C=CC1C3)=O)C2 Cc1cncc(C(N2CC=CC2(C)C(=O)NCC[Si](C)(C)C)=O)n1 N1(C(=O)Cc2ccc(-c3nn[nH]n3)cc2)CC2CCCC(C1)N2C1CC1 N1(C(CCCC(C)C)=O)CC(NC(C2CCCS2(=O)=O)=O)C(N=[N+]=[N-])C1 N1(C(c2[nH]cc(CC)c2)=O)CC2C(CN(C)C(c3cnoc3C3CCC3)=O)C2C1 CC1CCC(C(=O)NC(C2CCCCC2)CNC(c2cc(C(N)=O)c[nH]2)=O)O1 N(C1c2ccccc2CC1NC(=O)COc1ccccc1)C(CCS(C)(=O)=O)=O c1(C(=O)NCC(Cn2cc(-c3cccc(O)c3)nn2)OC)cc(Cl)c(Cl)cn1 N1(C(CCCC)C(N)=O)CCC(C2CC(=O)N(C(c3n[nH]c(C)c3F)=O)C2)CC1 CCC(C)(CNC(C)=O)C(=O)NCC(c1csc(COC)n1)N(C)C C1(NC(c2c(C)ccs2)=O)CN(C(=O)Cc2ccc3nc[nH]c3c2)CC1C1CC1 c1(C(=O)NCC(CN(C)C(c2cnc(O)o2)=O)O)ccc(CC2CCC2)cc1 C1(CC(N2CC(C)C(CCNC(=O)C(N)=O)C2)=O)CCOC(C)(C)C1 C12(CC(=O)NC3C(C)CN(C(C4CCC(=O)N4)=O)C3)CC3CC(C1)CC(O)(C3)C2 O(N(C)C(=O)CN=C(NCC1CC1)N1CCC(C(C)C)C1)CC c1(C(N2CCC(CN(C(C(CCC)OC)=O)C)C2)=O)nnc(O)c(Br)c1O CCC(CO)C(=O)NC(Cc1ccccc1)CCNC(=O)CCn1ccnn1 C(C(CN=c1[nH]cc([N+](=O)[O-])c(=N)[nH]1)C(F)(F)F)NC(C=Cc1n(C)cnc1)=O C1(C(=O)NCCNC(C2C(C)C2)=O)CCCN(C(=O)CC2COC(=O)N2)C1 C12(C(=O)NCC=C(C(=O)NCCC(C)OC)C)CC(C#N)(C1)C2 NS(=O)(=O)c1ccc(C(=O)NC2CCN(C(c3cnc4[nH]ncc4c3)=O)C2)cc1Cl c1(OC)cc(N)c(C(=O)NCC2CCCCN2C(C2CC3C=CC2C3)=O)cc1F c1(NC(c2cccc(CNC(C(CN(C)C)N(C)C)=O)c2)=O)cccc(F)c1O c1(C(N2CC3(F)C(NC(C=CC)=O)(CCC3)C2)=O)ccc2c(c1)C(=O)N(C)C2=O C(=O)(C1CCc2nccn21)NC1(COC)CCCN(C(C(CC)(CC)CO)=O)C1 C1(NC(=NCC)NC(c2ccc(F)cc2)C2CCC2)CC1C1CCCC1 C(=O)(CC(F)(F)C(F)(F)F)N1CCC(NC(c2ccnn2C2CCC2)=O)C(F)C1 C#Cc1ccccc1CC(N1CCC(C)(C)C1CNC(=O)CCC=C)=O c1(C(=O)NCC(c2ccccc2)NC(CC=CC)=O)nn[nH]c1Cl c1(OC)cc(C(=O)NCCC2CN(C(c3cc(CN(C)C)n(C)n3)=O)C2)ncn1 C1(NC(CC2N(C)CC=CC2)=O)CCCCCC1NC(c1ccc(Cl)cc1)=O c1(C(=O)NCC(C2CCCC2)NC(c2c(C)ocn2)=O)c(F)ccc2c1OCC2 CC1(C)CCCN(C(c2ccc(C#N)cc2)=O)C1C(=O)NCCC12CCCC1C2 Cc1cc(C(N2CC3CC2CN3C(c2cn3ccnc3s2)=O)=O)cnc1C Cc1nc(C(=O)N(CC(C)NC(=O)C(C)(O)C2CC2)C)sc1C c1(C(=O)NC2CN(C(c3cccc(NC)n3)=O)CC2O)ccc(C)c([N+](=O)[O-])c1 c1(C(=O)NC(C)C(C)(C)C(=O)N(CCN=[N+]=[N-])C)cc2cccnc2[nH]1 C1(CC)CCN(C(c2cnn(C)c2)=O)C(C(=O)NCC2(CO)CC=CC2)C1 N1(C(c2c(Br)ncn2C)C(=O)Nc2c(C)c(Cl)ccc2)CCC2(CCCO2)C1 C1(CN(C(CCN(C(=O)Cn2nc(C)oc2=O)CC=C)=O)C)CCCC1(C)C c1(C(=O)NCCN(C(CN(C(C)=O)C)=O)CC2CC2)cscc1C#N Cc1nn(C)cc1C(COc1cccc(F)c1)NCc1cn(C2CCCC2)nn1 C1(C(=O)NC2CC(CNC(CCc3ccc(NC)cc3)=O)C2)CC(=O)NC(=O)N1 Cc1cc(C(=O)NCCC(C)NC(=O)C2=CCOCC2)cnc1OC(F)F c1(CNC(c2n[nH]c(C)c2O)=O)cnn2c1CN(CCS(C)(=O)=O)CC2 c1(CC)cc2c(NC3CCCCC3CNC(=O)CCOC(C)=O)nc(C)nc2s1 C1(CNC(CC2CCN(C)C2=O)=O)CCC12CN(C(c1ccc(F)cc1Cl)=O)C2 CC1(C)CC(C(N2CCCC(C(N)=O)CC2)=O)CCN1C(=O)Cn1cc(Cl)cn1 C1(C(N2CC(C)CC(NC(CCOCCOC)=O)C2)=O)CCCN2CCCC12 C#CCC(C(=O)OC)NC(=O)C(Cc1ccco1)NC(c1cc(CCO)on1)=O c1(N)ccc2[nH]ccc2c1.N1(C(c2c(C(=O)O)cco2)=O)CC2(C1)CC2(F)Br c1(C(=O)NC2CC(CNC(C(C)OC)=O)CC2O)cc(C)c(C)c(C)c1 c1(C(=O)NCCn2cc(C(C)(C)S(C)(=O)=O)nn2)sc2c(Br)cccc2c1N C1(NC(c2ccc(C#N)o2)=O)CN(C(c2coc(Br)c2)=O)CC2CC12 C12(NC(CCCc3onc(CC)n3)=O)CCN(C(c3c[nH]nc3C)=O)CC1C2 c1(C(N2CC(OC)C(NC(c3ccc(=N)[nH]n3)=O)C2)=O)c(F)cc(Cl)cc1Cl C12(C(N3CC(C)N(C)CC3)=O)C3C4C1C1C2C3C41C(=O)NCc1cnn(C)c1 c1(N2CCC(NC(C3C(OC)CCCC3)=O)C(F)C2)ncc2c(ncn2C)n1 O=C(N=c1ccc2nnc(C(F)(F)F)n2[nH]1)c1ccc(Cl)o1 C1(C(=O)NCC(C(CC)C)CO)CC2(CCN1C(C1COCCC1C)=O)CC2 C(C(CNC(c1nnsc1C)=O)S(C)(=O)=O)NC(C=CCOCCOC)=O N1(C(c2c(C)cccn2)=O)CC2(C1)CN(C(c1cc(Br)cn1C)=O)CCO2 C(=O)(N=c1cc(C)n(-c2nnc(C(C)C)o2)[nH]1)C1(c2ncc(C)o2)CCCC1 C12(C(=O)NC3C4CN(C(C5CC6CC(=O)C5C6)=O)C3C4)CCCC1CS(=O)(=O)C2 C1(NC(c2nc(C#C)sc2)=O)CC2CC1N(C(=O)CCC(=C)C)C2 c1(C(=O)NC(C(C)C)CCNC(=O)CCCn2cncn2)cc2c(s1)CCOC2 C1(NCCn2cc(CNC(CCC(C)OCC)=O)nn2)CCN(C(C)=O)CC1O C1(C(=O)NCc2cccc(OC)n2)N(C(=O)CC2(C)CC2)CCCC1(C)C c1(C(N(CC(C)CNC(=O)CCN2C(=O)CCC2=O)C)=O)c(N)sc2c1CCC2 C(=O)(C1OC(=O)c2ccccc21)NCC1CC(NC(c2ccncc2)=O)C(O)C1 C1(O)(CC(=O)NCC2C(C)CCN2C(c2cc(C(N)=O)[nH]n2)=O)COC(C)(C)C1 N1(C(C(C(C)(C)C)OC)=O)CCN(C(c2csc(C)c2C)=O)CC(C)C1 N1(C(=O)NC2CC23CC3(F)F)CCC(C2CCOCC2)C1 CC1(C)COC(C)(C(=O)NC2CCC(CNC(=O)CC(F)(F)Cl)CC2)CO1 C(C)(C(CC(=O)N1CCSCC1)NC(C1(C)CC1C)=O)OC C(Cc1cnc[nH]1)(C(=O)N(CCC(=O)N)OC)C(C(CCCC#C)C)=O C1(NC(c2c(C(N)=O)cccc2)=O)CCCCN(C(c2nnc(O)nc2O)=O)C1 C#CC1(C(=O)NC(CO)CCC=C)CCN(C(c2nc(=N)cc[nH]2)=O)C1 c1(C(N2CC(OCCNC(CC3CCN(C)C3)=O)C2)=O)ccn2[nH]c(=N)nc2c1 c1(C(N2CCC(CNC(C(C)=C(CC)C)=O)CC2)=O)cc2c(s1)CCC(CC)C2 c1(CNC(=NC)NCc2cc(C3CC3)nn2C(C)C)ccc2c(c1)C(=O)OC2 N1(c2n(CCCOC)c(-c3ncnn3C)nn2)CCOC(C)(C(F)(F)F)C1 C(=O)(CS(=O)(=O)c1ccccc1Cl)NCC1N(C(C(CC)F)=O)CC(O)C1O c1(C(=O)NCC2CC(NC(c3n(C(C)C)nnc3)=O)C2)cc(Cl)ccc1F c1(C(=O)NCC(=C)CCNC(C2COC(C)C2)=O)cc(Cl)cc(Cl)c1Cl N1(C(Cc2cnc(C)o2)=O)CCC(NC(c2c(C)nc(C)n2O)=O)CC1C C(=O)(N=c1cc(C(F)(F)F)[nH][nH]1)c1cccc(NC(c2ccc(C)c(C)n2)=O)n1 N1(C(C2C(C)(C)CC2)=O)CCC(C)(CNC(=O)C(O)C2CCCC2)C1 CN1CCN(C(c2ccsc2C#N)=O)CC1C(=O)NCC(O)C1CCC1 C1(OC)CC2(CCC(C(N3CCN(CCC4CC4)CC3)=O)CC2)C1.S(C)(=O)(=O)N C1(C(N2C(C(=O)OC)CC2)=O)CCCN(c2cc(O)ncn2)C1.Cc1nscc1C=O C(C(C)CCCO)NC(CC1N(C(C2CC(C(C)C)C2)=O)CCC1)=O c1(C(N2CC(CN(C)C(C3CCCSC3)=O)C2)=O)nc(=O)cc(N)[nH]1 c1(OC)ccc(C)c(C(=O)N(CCNC(c2ccc([N+](=O)[O-])s2)=O)CC2CC2)c1 c1(C(=O)NC(C2(O)CN(C(c3nc(C(C)OC)sc3)=O)C2)C)ccccc1Cl C1(C(=O)NC2(C)CCN(C(C3CN(C)C(=O)CC3)=O)CC2)CS(=O)(=O)CC12CC2 S(=O)(=O)(c1ccc(Cl)c2ccccc12)N1CCCC(O)(CC(N)=O)C1 CC1(NC(=O)C(O)CC2CC2)CCCN(C(c2cnc(N(C)C)cn2)=O)C1 N1(C(C2(CC)CCC2)=O)CCOC(C(=O)NCCc2ncccc2F)C1 N1(CCC)CCCCC1C(=O)NCCC(CSc1ncc[nH]1)NC(=O)CSCC N1(C(c2c(O)nccc2)=O)C2CCCC1CC(N=c1ccnc(C(F)(F)F)[nH]1)C2 N1(CC(C(CC)C)OC)CCC(NC(=O)OC(C)(C)C)C(C)(C)C1 Cc1ccc(C=CC(=O)N(CCCNC(C2CC3C=CC2C3)=O)C(C)C)s1 c1(NC(CC2N(C(CN(CC)CC)=O)CC2)=O)ccc(F)cc1F c1(-c2nc(C(CCC)C)nn2C2CSC2)cc2ccc(Br)cc2s1 CCC(CC(F)F)C(=O)NC(c1ccccc1)CNC(=O)Cc1cncnc1 Cn1nc(CNC(C2C=CCC2)=O)c2c1CCN(C(C1(C#N)CCC1)=O)C2 C1(CNS(CC2(N(C)C)CC2)(=O)=O)CCC2(CCC2)O1 c1(C(=O)Nc2cccc(C(=O)Nc3c(C)cc(CC)s3)c2)cc(Cl)c(Cl)nc1Cl C1(NC(c2n[nH]c3c2CCCC3)=O)CC2CC(C1)N(C(=O)CCC1CCCO1)C2 CC1CCCC(C(=O)NC(C2CN(C(c3cccc(F)c3)=O)C2)C)CC1 CC1CN(C(c2nccnc2Cl)=O)CCC1CNC(c1c(Cl)cnn1C)=O C1(NC(c2nc(CCC)oc2)=O)CC2CCC(C1F)N2C(C1CC(C)(O)C1)=O CC(C)CC(C(=O)NC(CSC)C(=O)NCc1ccn(C2CC2)n1)C(C)C c1(C(=O)NC2CN(C(C(C(C)C)(C)O)=O)CC2(C)C)noc2c1CC(C)(C)CC2 N1(C(c2cnn[nH]2)=O)CC2C(NC(=O)C(F)(F)c3nccs3)C2C1 c1(NC(C(N2CCC(CCCC)C2)=O)=O)ccc(F)cc1OC c1(-n2cc(NC3(C(=O)OC)CCN(C(=O)C(F)(F)CO)C3)nn2)c(F)cccc1F n1(CC(=O)NCCCNC(=O)CC2CCCCC2F)c(=O)cnc2ccccc12 C12(CC(=O)NC(C(=O)OC)(C)C3CC3)CCC1CN(C(C1CC(C)(C)C1)=O)C2 Cc1ccsc1C1CCC1CNC(=S)NC1CCOC1 N1(C(C2C(C(=O)OC)CCC2)=O)CCOCC1c1cn(CCn2cccn2)nn1 N1(C(CN(C)CCO)=O)CCC2CN(C(=O)C(C)(O)CCc3ccccc3)CC12 c1(C(=O)NC(C(C(C)C)C)CNC(c2cnsc2)=O)ccc2c(c1)NS(=O)(=O)C2 c1(OC)ccc(CN(C2CS(=O)(=O)CC2O)Cc2nc(C(C)C)no2)cc1Br CCC(C)(CNC(=O)C(C)c1ccsc1)C(=O)N(CCC(=O)NC)C N1(C(CC(C(F)F)NC(c2c(OC)csc2)=O)=O)CCc2cccnc2C1 CCCCC(CCCC)C(=O)NC1CCN(C(=O)Cc2cc(C3CC3)no2)C1 n1(C(C)C)cccc1C(=O)NCC(C)N(C(=O)CC1CC12CC2)C C(CCCC(=O)N(C)CC=CC(=O)N(c1ccc(C)cc1)C(C)C)(OC)OC c1(OCC)cccnc1C(=O)NCC1CCCN(C(C2(O)CCOC2)=O)C1 c1(OCC(=O)NC(CNC(C(C)=C2CCCC2)=O)CC(C)C)c(F)cccc1F CCCCCC(O)CC(=O)NC(C)C(C)(C)C(=O)N1CC2(CCC2O)C1 N1(C(c2cccc(N)c2Br)=O)CCC2(CCN(C(c3ccccn3)=O)CC2)C1 c1(C(=O)NC(C(=O)NC2CCC(OC)C2)CCF)cc2cccnn2c1 N1(C(c2cc(C)nc(Cl)c2)=O)CCCC2(CCN(C(c3cnc(Br)s3)=O)C2)C1 C1(C(=O)NCCNC(=O)OC)CN(C(c2ccc(C#N)cn2)=O)CCN1C C1(C(=O)NCC2CC(C)N(C(C3CC=CC3)=O)C2)CCS(=O)(=O)C(C)C1 C(=O)(C1Cc2c(Cl)cccc21)NCC1C(C)CN(C(=O)CCOCC2CC2)CC1 C1(CNC(C(C)OCC=C)=O)CCC2CN(C(=O)C(C#N)CC)CC12 c1(C(N(CC#CC)C)=O)ccc(CNC(=O)C(C)c2cccs2)cn1 CC(CC(=O)NC(C(N1CCC(CCCO)CC1)=O)c1ccoc1)CC(C)(C)C O=C1NCC2(CCN(C(=O)CN(C(=O)Cc3ccns3)CC3CC3)C2)N1 C(C(C)CC(=O)N1CCC(Nc2ncccc2C2CCCCC2)CC1)OC c1(SCC)ccccc1C(N1CCOC(CN(C(=O)CCC(C)C)C)C1)=O C1(NC(CNC(CCC)=O)=O)CCCC(NC(=O)CCCN2C(=O)CCC2=O)C1 c1(C(N2CCC(N(C(C(CN(C)C)N(C)C)=O)C)C2)=O)cc(F)c2[nH]nnc2c1 C1(CNC(c2cccc(C(C)C)n2)=O)CN(C(C2CC(F)(F)CS2)=O)C(C)(C)C1 n1(CC)ncc2c1CC(C(N1CCC(CN(C(=O)CSC)C)C1)=O)CC2 c1(OC)ccc(C(=O)NC(CNC(c2coc3c2CSC3)=O)C2CCC2)cc1O c1(C(=O)NCCC2CCN(C(=O)C=CBr)CC2)cc2c(=O)[nH]ccn2n1 C1(N(C(CC)=O)C)CCCN(C(=O)C=Cc2ccc(I)o2)CC1 CCC(C)(COC)C(=O)N1CCCC(CO)(CNC(=O)C(O)CC2CCCC2)C1 c1(NC(C)=O)ccc(C(N2CCN(C(=O)CC3CCCC(=O)N3)CC2C)=O)cc1F C(C)(CCC(=O)NC(C1CCCC1)CNC(C1(CC)CCNC1=O)=O)OCC c1(NCC(CC)(C)CO)cc(C)c(Br)cn1 C1(N(CC(c2ccccc2Cl)(C)C)C)CCCN(C(=O)OC(C)(C)C)C1 c1(C(=O)NC(CNC(C(C)=C2CCC2)=O)C(C)C(C)C)nn(C)cc1[N+](=O)[O-] c1(C(N2CCN(C(CC=C)=O)C(CCOC)C2)=O)cccc2c1OC(C)(C)C2 c1(-c2nc(C(c3c(F)ccc(C)c3)C(C)C)on2)cc2c(s1)CCCC2 c1(C(=O)NC2C(NC(C(=O)NC(C)C)=O)CC2)cocc1Br c1(OC(c2ccc(C(C)C)cc2)C)ccnc(O)c1C=O C1(CNC(c2ccsc2C(F)F)=O)CC2(CCN(c3nnc(O)s3)C2)CO1 Cc1cc(Br)c(C(=O)NCC2C3CN(C(c4coc(C#N)c4)=O)CC23)s1 CC(C)CS(=O)(=O)CC(=O)NCC1CSCC(CO)C1 C1(NC(c2ccc(C)cc2F)=O)CCN(C(C2CC(=O)N2)=O)CCC1CO C(=O)(C(C)C(C)(F)F)N(C1CCN(C(CCn2c(C)ccc2C)=O)CC1)C C(C(C)C(F)C(=O)N(C)CC1OCCC1(C)C)NC(C(CC)C#N)=O C=Cn1nncc1C(=O)NC1(C2CCCN2C(=O)C(C)OCCOCC)CC1 C(N=c1nc2sccc2c(N2CCCCC(c3ccccc3)C2)[nH]1)C1(Br)C(F)(F)C1 N1(CC2(NC(Cc3nnc(C)o3)=O)CC2)CCN(C(=O)C(C)(Cl)Cl)CC1 Cc1ccc(C(N2CCOC(c3nnn(C)n3)C2)C(=O)NC2CC2)cc1Cl Cn1ncc2c(NCc3cn4c(n3)COCC4)[nH]c(=NCCC3CCOC3)nc12 C(CC(O)C(F)F)NC(COC(CNC(c1c(C)noc1)=O)(C)C)=O c1(OC)ccc(S(=O)(=O)N2CC(C)CC2C(=O)N=c2cc(Cl)n(C)[nH]2)cc1Br c12ccccc1S2.N1(C(=O)NC(C)(C)C)CCN(CC)CC1.C12CN(C1)C2 S(=O)(=O)(c1cc(C(N2CC(NC(=O)CC(C)(C)C#N)C(C)C2)=O)n(C)c1)NC Cc1ncc(C(N2CCCC2CCNC(=O)CC(O)C(C)C)=O)cc1N n1(CC)ncc(C)c1C(N1CCCC(C(N2CCOC3CC23)=O)C1)=O C12(C(=O)NCC3(CNC4CC(C(=O)C5CC5)C4)CC3)CCC(CO)(CC1)CO2 C1(NC(CC=CCCCCC)=O)CCCC(NC(=O)COCc2scnc2C)C1 C(N=c1nc(OC)c(F)c(C)[nH]1)C1C2CN(C(c3c(CC)cncc3)=O)CC21 C1(NC(C(CCNC(c2c(=N)[nH][nH]c2)=O)O)=O)C2C3CCC(C3)C12 N1(C(c2c(CC)noc2)=O)CCCC(C(=O)NCC(C(C)CC)OC)C1 N1(C(Cn2cnc(=N)[nH]2)=O)CCCCCC1Cc1cccs1 c1(CC(N2CCC(C(=O)NCCC(C)F)CC2)=O)cnc(C)c(C)n1 Cc1nn(Cc2ccc(CCCN3CCCC3c3cnn(C)c3)cc2)c(C)c1Br c1(-c2cn(CCCC(=O)N3CC(OC)C3)nn2)ccc2c(c1)Cc1ccccc1-2 c1(OCCNC(c2n(CC)nnc2)c2nnnn2C2CC2)cc(F)ccc1C CC(C)C1=CCC(NC(c2occc2CNC(C2(C)CC3CC3C2)=O)=O)CC1 c1(NC(C2CCN2C(c2cnccc2Cl)=O)=O)cccc(Br)c1Cl C1(C(N2CC(NC(CC(=O)NCC)=O)C(C)CC2)=O)CCC(C2CCC2)CC1 c1(OC)ccc(F)c(F)c1CN1CCC(CC(=O)NC(C)CC#N)CC1 C1(CNC(C=C(C)CNC(c2ccc(F)s2)=O)=O)CCCCS1 c1(C(N2C(C(C)NC(c3cnc(OCC)s3)=O)CCCC2)=O)ccc(F)cc1C N1(C(C2(C)CCC2)=O)CCN(CCNC(c2ncccc2Br)=O)CC1 CC#CC1CCN(C(C2CCC(CNC(=O)C3=CCCC3C)C2)=O)C1 c1(CNC(N2C(C)(C)CC(CO)C2)=O)c(Cl)oc2ccccc12 C(=O)(NNc1cc(I)ccn1)NC(CC(=O)O)CC1CC1 C(=O)(C1=COCCO1)N1C(C2CCN(C(CN(C(COC)=O)C)=O)CC2)CCC1 c1(OC)ccc(Cl)cc1C(F)(F)C(=O)NC(c1c(C)nn(C)c1C)C N1(C(N2CC(C3CCCO3)C2)=O)CCN(C(=O)C(=O)NCCC(F)F)CC1 N1(C(C(C)(C)c2ccno2)=O)CC(NC(C2(CCO)CC2)=O)C(N=[N+]=[N-])C1 C=CCC(CC(=O)N(C1CN(C(C)C)C1)C)NC(=O)C(C)COC c1(C(N2CCN(C(C(CCC)C)=O)CC2CCO)=O)cnc2ncnn2c1N CC(C)(C)C(CNC(=O)CCN1CCCCC1)NC(C12CCCC1(C(N)=O)C2)=O C(CC(F)CN=[N+]=[N-])NC(C(C)(CO)NC(CC1ON=C(C)C1)=O)=O c1(C(=O)NC2(COC)CCN(C(C(CCC)OCC)=O)C2)cccc2c1COC2 c1(OC)cc(C)c(C(N2CC3CC2CN(C(C2(C)CC2Br)=O)C3)=O)cc1OC c1(CNC(=O)NC(C(C)NC2N(S(CC)(=O)=O)CCC2)=O)ccccc1Cl N1(C(c2c(C)nns2)=O)CCC(C)(CC(=O)NCCNC(=O)CO)C1 C1(C(=O)NCC#C)CC12CCN(Cc1ncc(Cl)cc1Cl)CC2 C1(CNC(CC(CC)C)=O)CC2CN(C(c3ccc(C)nc3)=O)CC12 c1(C(N2C(C#N)CC(F)(F)C2)=O)csc2c1CCN(Cc1ccc(Br)cc1Br)C2 C1(C(=O)NC2(C(N(CC)Cc3cnn(C)c3)=O)CCCC2)CC2(CCO1)CC2 c1(C(N2C3C(C(=O)Nc4ncc(C)c(Cl)n4)C(C3)C2)=O)ccc2c(c1)NC(=O)C2 N1(C(c2cccc(C)c2)=O)C2C=CCC1CC2.C1(=O)CCC(C)N1C C(CCCCCC(=O)NC1CCCCC1O)NC(CCC(C)(C)OC)=O C1(CNC(C2(OCC)CCC2)=O)CCN(C(c2coc(C(N)=O)c2)=O)C12CCC2 Cc1cccc(NC(=O)C(C2CCCO2)NC(=O)C(Cl)Cl)c1C C(CCCC(=O)NCCC(C)(C)CNC(=O)Cc1cscc1Br)OC C(C)(C)(C(=O)NCCN(C)C(C1(O)CC(c2ccccc2)C1)=O)OC(C)C C1(C(=O)NCC2C(C(=O)OC)CCC2)CCCCC1CNC(=O)CCCN(C)C c1(C(N2CCC(NC(CCC(=O)NC)=O)CC2C2CC2)=O)ccc([N+](=O)[O-])cn1 C1(NC(c2cncc(F)c2)=O)CCCCN(C(C2CCC23CCC3)=O)C1 C12(CNC(C=CCC)=O)CCC(CC1)N(C(=O)C(C)(Cl)Cl)C2 c1(CN(C(CN(CCC)C)=O)C)ccccc1CNC(=O)C=CCOCCO CC1CCN(C(=O)CC2CCSCC2)C1CNC(c1nccc(C(F)(F)F)n1)=O c1(NC)ncnc(SCc2noc(CNC(c3ccc4c(c3)CC4)=O)n2)c1F C(c1c(C)noc1C)=CC(=O)NCC(CCOC)NC(c1cc(C(N)=O)c[nH]1)=O C1(C(N(CCCN(C)C(c2ccc(C(N)=O)cc2)=O)C)=O)CC2CCCCC2O1 CCC(CC(=O)N1CCCCC1C1CCN(CC2CCS(=O)(=O)C2)C1)C(C)(C)C C(=O)(C(CC(C)C)C(N)=O)N1CC2(CC(NC(c3c(C)c[nH]c3)=O)C2)C1 Cc1ccc(F)c(C(=O)NCCC2C(C)CCCN2C(=O)COCCCF)c1Cl CCCCCCCCOCC(=O)NCC1(O)CCN(C(C2(F)CC=CC2)=O)C1 c1(C(=O)Nc2cc(C(F)(F)F)c(Cl)cc2Cl)c[nH]c(=O)c2ccnn12 c1(C(C2CCC2)NC(C(C)N(CC(=O)NCC(C)C)C)=O)ccccc1 c1(C(N2C(CNC(c3c(C4(C)COC4)noc3)=O)CCC2)=O)cncc(O)c1 c1(OC)c(C(N2CCC(O)C(NC(c3csc(C(C)C)n3)=O)C2)=O)c(C)nn1C N1(C(C(C2CC2)OCC)=O)CCOCC(C)(CNC(c2nc(C)sc2C)=O)C1 c1(C(C(=O)NC(CC)C)N(CC(C)C(C)C)CC)cc(Br)cs1 C1(Nc2c(C)[nH]nc2-c2ccccn2)CC2(CCCC2)C1 c1(C(=O)NC(COC)CNC(=O)CC2CC=CCC2)cc([N+](=O)[O-])no1 Cc1cn2c(C(=O)NC(C)(C)CNC(C3CS(=O)(=O)CCO3)=O)c(Cl)nc2s1 CC1CCCc2nc(C(=O)OCCC3(CNC(=O)OC(C)(C)C)CC3)cn21 C1(CC(=O)NCC(C(CC)C)C)CC(C)(C)CN1C(=O)C(CC)C(=O)OC Cc1[nH]nc(C(C)C)c1C(=O)NC(C)C(CO)NC(C1CCCS1)=O C1(N(C(C)Cc2ccccc2)C(c2cc(C)no2)=O)C2CCC1CNC2 Cc1nnccc1C(=O)NC1COCCC1NC(c1cc[nH]c1C1CCCC1)=O CCC(C)(CNC(=O)CCOC1COC1)C(=O)N(C1CCC1C)C Cc1ccnc(O)c1C(=O)NCC1CCCCC1NC(c1csc(C2CC2)n1)=O CC1(NC(C2CCN(c3cc(-c4cn(C5CC5)nn4)ccn3)CC2)=O)CCNC1=O C(=O)(CCC(=O)NC1CC(CNC(c2coc(Cl)n2)=O)C1)NCCC C(CN=C(NCC1(CS(C)(=O)=O)CCC1)NC1CCNC(=O)C1)OCC N1(C(CN(C)C2CC2)=O)CCC(CNC(=O)COCC2CCCO2)C12CC2 C12(C(=O)NCC3(CNC(C4CCC(OC)C4)=O)CCCCC3)CCC(CC1F)C2 C(=O)(C1CCCc2ccnn21)N(CCN(C(CC(C)P(C)(C)=O)=O)C)C(C)C n1(CC)nnnc1NC(C1CN(C(=O)C=CC2CC2)C1)=O c1(N(CCNC(C=CCC)=O)CC2CC2)cc(C2CC2)ncn1 c1(C(=O)NCCN(C(C(C)C)=O)CC(C)O)ccc(-c2ccccc2)o1 C(C(C(=O)NC1CC(F)(F)C1)C(C)C)NC(COCC=C)=O Cc1scc(C(=O)NC(C)CNC(=O)C(c2ccc(Cl)cc2)C)c1N CCC(CN(C)C(C1CC(NC(N)=O)C1)=O)N(C)C.C12(CC1)C(=O)N2 c1(C2C(C(=O)NCCCN(C(=O)CC(C)F)C(C)C)C2)c(F)cccc1F CCCC(CC)C(C(=O)NC1CCC(F)(F)CC1)N(C)Cc1ccc(F)cc1C CC1(NC(C2CC2)C2CC2)CCOC1C1CC1.c1(C)cccnc1 c1(C(=O)NCC2CC(F)(CNC(=O)Cc3ccoc3)C2)cc2cccnn2c1 c1(C(C(=O)NCC(F)F)N(CCCn2ccnc2)CC)ncc(C(C)(C)C)o1 c1(C(=O)NCCC(CNC(CC(C)SC)=O)O)ccc(C2CC2)c(Cl)c1 C1(CNC(C2CC(C#C)(O)C2)=O)CC2CCCC2N1C(c1ccn(C)c(=O)c1)=O c1(C(=O)C2CC2)cc(Cl)cnn1.C12CC(C1)C(=O)NC1CC(C1)C(=O)NC2C c1(CCC(=O)N(C)CC2CCSCC2)nc2ccccc2[nH]1 Cc1ccc(OCCC(N2CCOCC2c2ccccc2Br)=O)cc1 C1(C(N2C(CNC(c3nc(C)n(C)c3)=O)C=CC2)=O)CC(O)c2ccccc2O1 O=C(CCCCC(F)(F)F)NC1(CO)CN(C(C2(C3CCCO3)CCC2)=O)C1 C12(C(=O)NC3C(NC(CN(C)C(N)=O)=O)COC3)CCN(CC1)CC2 n1(CC)nc(C(=O)NCC(C2CC2)NC(=O)C(=O)NC2CC2)cc1C c1(C(=O)N(CCC2CC2)CC2CC2)cccc(C2CC2)c1 CC1CC(C(=O)NCC2CCCN(C(C3(Nc4ccc(Cl)cc4)CC3)=O)C2)=NO1 Cn1ncc(C(N2CC(NC(=O)C=Cc3cc[nH]n3)C(O)C2)=O)c1N c1(C(=O)NCC2(NC(c3ccc(-n4ccnc4)cc3)=O)CCC2)cncc(O)c1 N1(C(C=C)=O)CCCC1(C)CNC(c1cc(C(F)(F)F)nn1CC)=O C1(CNC(=O)Cn2ncnn2)CCCN1C(=O)Cc1nncs1 N1(C(C(CC)F)=O)CC2C3CCC(C(NC(=O)Cn4cc([N+](=O)[O-])cn4)C3)C2C1 c1(NCCC2(C)CC2(Cl)Cl)cc(S(=O)(=O)N(CCCCO)CC2CC2)ccc1C#N N1(C(CN(C(=O)C=Cc2ccoc2)CC#C)=O)CCC(c2ncco2)C1 C(CCN=C(NCCc1cccc(C(F)(F)F)n1)N1CCC(SC)C1)OCC C1(C)(NC(=O)CC2(N)CCCCC2)CCCCC1C(=O)NCC1C(C)(C)OCC1 CC1(C)CC1(C)C(=O)N(C1CC1)C.C1(OC2CC=CC2)CN(C(=O)CO)C1 CCCCCC(O)C(=O)N(C(C)C(=O)NC(C1CCCCC1)=O)CCCN(C)C c1(C(N2CCCCC(NC(=O)C(F)CC3CC3)C2)=O)cc(O)nc2c1CCCN2 CC(C)(F)C(C)(F)C(=O)N1CC(NC(c2cc(N)cnc2Cl)=O)C(C)(C)C1 Cc1cccc(C(N2CCC(NC(c3c(Br)cncc3Br)=O)C(O)C2)=O)c1I C1(O)(CNC(c2nn(C)nc2Br)=O)CSCC1(C)C CC1(F)CCC(C(N2CC(C3(NC(C4CCCC(O)C4)=O)CC3)C2)=O)CC1 c1(C(=O)NC(c2nnnn2CCNC2CC2)C2CCOC2)cc(CO)ccn1 c1(C(=O)NC2(CNC(C3CCC(C(=O)OC)C3)=O)CC2)[nH]c2cc(C)ccc2c1C c1(NC2C3N(C(c4ccc(C)cn4)=O)CC(CC3)C2)nc(C)c([N+](=O)[O-])cc1Cl C1(C(N2C(C(=O)OC)CC2C)=O)CC2CC2N1C(c1ccc(C)cn1)=O CCCCCCC(CNC(=O)NCC1CC=C1C)CC CCS(=O)CC(=O)N(C1CCCC1)CCNC(c1ccc(Cl)cc1)=O CCC(CC(=O)N(CCCCO)C)NC(C1CCC(F)CC1)=O N1(C(C2CCC=CO2)=O)CCCC(O)(Cn2cc(-c3cccnn3)nn2)CC1 N1(C(C(C)OCCCC)=O)CCC(C(C)(C)C(=O)N(C)Cc2ncc(C)o2)C1 N1(C(CC2CN(C(C(n3c(C)ccn3)C)=O)CC2C)=O)CC2C=CC1CC2 C1(CC(=O)NC2CCN(C(CCCC=C)=O)CC2)SC2=NCCN2C1=O CC1=NOC(C)(C(=O)NCC(O)CNC(c2ccn(C(C)C)n2)=O)C1 C(=O)(C1Cc2ccccc21)N1CC2C(CNC(C3(F)C(C)(C)C3(C)C)=O)(CC2)C1 C(=O)(CCCCC(N)=O)NCC(CNC(c1ccc(OC)c(Br)c1)=O)(C)O n1(CC)nncc1C(=O)NC1COCC1NC(=O)COC1CCOC1 Cc1sc(Cl)nc1C(=O)NC1CC1NC(=O)CC(O)c1cnc(Cl)s1 N1(C(c2cnc(CC)[nH]2)=O)CC2CCN(C(=O)CC(c3ccccc3F)C)C2C1 Cc1cn(C)nc1C(=O)NCCC1CCN(C(c2ccccc2CO)=O)CC1 C1(C)(C(=O)OC)CCN(C(=O)CC2CCCCO2)C1.n1(CC(=O)OCC)cc(C)nn1 c1(N(C(c2ncn(CCNC)n2)=O)C)c(Cl)cncc1[N+](=O)[O-].CCO C(C(C)(C)C#CC(=O)NC(C)Cc1ccccn1)NC(c1cc(COC)on1)=O C1(F)(CNC(C(CC)(C)CO)=O)CCCN(C(c2cc(Cl)ccc2N)=O)CC1 N1(C(c2cnc(C)s2)=O)CC=C(C(=O)NC2(C(F)F)CCC2)C1 c1(C(=O)NC(CC(C)NC(CSCCCC)=O)C)cc(C)c(C)c2ncccc12 C1(C(N2CCN(CCNC(C3C(C)C3C)=O)CC2)=O)CC2(C1)CC(C)(C)C2 c1(C(=O)NC2CCC(F)(CNC(C(COC)C)=O)C2)cnc2c(ccn2C)c1 c1(C(C)(C)C)ocnc1C(=O)NC(CNC(C12COCC1C2)=O)C1CC1 N(C(=NCCNC(c1sccc1C(F)F)=O)NC1CCCCC1C)CC(=C)C CC(C)C(C)CCNC(C1CCC(C2CC2)N1C(=O)C=Cc1ccn(C)c1)=O N1(C(C2CCC(OC)CC2)=O)CCCC2C1CCN2c1nc(SC)ncc1Br Clc1cccnc1CNC(c1ccccc1)CC1COCCO1 CC1=C(C(=O)N2CCSCC2C(=O)NCC(N2CCOCC2)=O)CCO1 CCC(C)(C)C(=O)NC1(C(=O)N(CC(O)CN(C)C)C)CSC1 Cc1cnc(C(N2CCN(C(c3cccnc3C)=O)C(C3CC3)C2)=O)c(F)c1 C1(CC(=O)NCCN2CC(c3cn(C(C(=O)OC)C)nn3)C2)CC2CCC1CC2 N1(C(c2n(C)c(=O)ccc2)=O)CCOC2(C1)CN(C(c1ccc(F)cc1Cl)=O)C2 C1(C(N2C3(CNC(CCN(S(C)(=O)=O)C)=O)CC(C2)C3)=O)CCC2(CCC2)O1 c1(NC)cnncc1C(=O)NC(C)CCNC(c1sc(CO)nc1C)=O c1(C(C(=O)NCCCOC)N(C(C)CC#N)C)ccc(OC)c2oc(C)cc12 c1(NC(C2CN(C(c3cc(Br)cnc3Cl)=O)CCC2O)=O)ccc(Br)c(Cl)c1Cl c1(CCC)nc(C)c(C(=O)NCC2CC3CC3N2C(=O)C=CC2CCCO2)s1 c1(C(N2CCN(C(C3C(=C)CC3)=O)CC2CCO)=O)ccc2c(c1)B(O)OC2 c1(OC)cc(OC)c(C(N2CCOC(C(C)NC(=O)CCCN(C)C)C2)=O)cn1 c1(C(N2CCC(C3CCCN3C(C3CCCS3)=O)C2)=O)cc2c(Cl)nccc2o1 c1(C(=O)NCCCNC(C(C(=O)OCC)OC)=O)cncc(Cl)c1C C1(NCc2cc(C(=O)OCC)cn2C)CCC2(CC1)CNCCO2 C1(C(N(C2CCN(C(C3CN(S(C)(=O)=O)C3)=O)CC2)CC)=O)C2CCC1CC2 Cc1cc(C(N2CCCC(C(=O)NCc3cccc(F)c3Cl)CC2)=O)ccc1O CC1C(C=CC(=O)NCC2CN(C(c3c[nH]c(=N)s3)=O)CC2N(C)C)C1(Cl)Cl Cc1cnccc1C(=O)NC1CCC(N(C(=O)C(C(C)O)NC(N)=O)C)CC1 c1(C(=O)NCc2c(CNC(CCC#C)=O)cccc2)cnc(OC(C)C)c(Cl)c1 C12(C(N3CC(CCNC(c4cc5cscc5s4)=O)OCC3)=O)CCCN(CC1)C2 C1(C(=O)NC(CN(C(c2cc3sccc3[nH]2)=O)CC)C)CCc2[nH]nc(O)c2C1 c1(OC)ccc(C(=O)NC(CCN(C(=O)CCCC(F)F)C)C(C)(C)C)c(C)c1 CCS(=O)(=O)C=CC(=O)NC(C1(O)CCN(C(=O)Cc2sc(O)nc2O)C1)C C(=O)(C1CCCn2cc(C)nc21)NC1(COC)CN(C(=O)CC2CSC2)C1 c1(C(N2CC(C3CN(C(c4cc(Br)cs4)=O)C3)OCC2)=O)ccc(F)c(Cl)c1 C1(C#N)(C(N2CCCC(O)(CNC(CCC(C)OC)=O)C2)=O)CCN(C)CC1 c1(C(=O)NC2C(CNC(=O)Cc3cccc(Cl)c3)CC2)ccc(Cl)c(F)c1 Nc1c(Cl)c(C(=O)NCC2CCC2NC(=O)C=Cc2ccco2)cc(F)c1Cl c1(C(N2C(CNC(C3CC3CF)=O)CCCC2)=O)ccc(F)cc1OC(F)F C1(OCC=C)CCN(C(=O)C(C2CC2)NC(c2cc(C(C)C)on2)=O)C1 C1(NC(c2n(COC)ncc2)=O)CC2CCC1(CNC(=O)CCc1nccs1)C2 c1(C(=O)NC(C)CNC(=O)CCSc2ccccc2Cl)cc(O)cc(O)n1 S(=O)(=O)(c1[nH]c(=NC(Cc2ccncc2)CO)ccc1Br)NCC1(C)CC1 C1(Oc2ccccc2)CCN(C(N2CCC(C)C(O)C2)=O)CCC1C(=O)O c1(C(N2CC(C)C(NC(=O)CC3CCC(C)(C)C3)C2)=O)cccn2c(O)nnc12 N1(C(C(C=C)(C)CC)=O)CCC(C2(O)CC(NC(=O)C(C)=C3CC3)C2)CC1 C1(C(=O)NC(C(C)NC(c2[nH]cc(CC)c2)=O)(C)C)CCc2n[nH]c(C)c2C1 C1(COC)CN(C(C23CC2CNC3=O)=O)CCN1C(c1cncc(C)n1)=O C(=O)(C(C(C)(C)O)NC(C1CC1F)=O)NCc1nnn(C)n1 C(CCNC(C1C2CCCC12)=O)(C(=O)N1CCC(C(C)(C)O)CC1)OC N1(C(C=CCCC)=O)CCN2C(=O)C(NC(C3CCN(C4CC4)CC3)=O)CC2C1 CC1(C)C(NC(=O)C(=O)NCC2CC3C=CC2CC3)CS1(=O)=O Cc1cc(S)nc(N2CCCCC2)n1.C1(C#N)(C(=O)O)CN(Cc2ccccc2)C1 C1(C(=O)NCC2(C(C)NC(c3c(C)nccc3)=O)CC2)CC2CS(=O)(=O)CC2C1 N1(C(C=CC(C)C)=O)CCN(C(c2cc(Cl)cn2C)=O)CC(CO)C1 c1(C(=O)NC2C=CC(CNC(C3CC=CCC3)=O)C2)cc(F)cnc1O C(=O)(C1OCCc2ccccc21)N1CC(CN(C(COC(CC)C)=O)C)C1 c1(C(=O)NC2CCN(C(CC=C=C)=O)C2C(C)(C)C)nn(C)c(=O)cc1C C(C1CCNc2ccccc21)NC(C12CC(C(=O)OC)C(C1)C2)=O N1(C(CC2CCCC(NC(C3C(C)CC3)=O)C2)=O)CCC2(CSC2)C1 C1(N(C(c2ccc(C)c(N(C)C)c2)=O)C)CCN(C)C12CCCNC2 CN=c1cc(C(=O)NC2CCC(CCNC(=O)CCC3CCCCC3)C2)cc[nH]1 C12(C(=O)NC3(C#C)CCCOC3)CCC(CC1)N(C(C1(OC)CCSC1)=O)C2 CC(C)(C)C(CNC(=O)C=Cc1cnc[nH]1)NC(=O)CSCc1cscn1 C12(CNC(C(CC)SC)=O)CCC(CC1)N2CC(=O)Cn1cc(C(=O)OC)nn1 N1(C(C2C(C(C)C)CCO2)=O)CC2(C1)CN(C(c1ncccc1N(C)C)=O)C2 N1(C(Cc2c(OC)cccc2)=O)CCC(NC(C2CN(S(C)(=O)=O)C2)=O)C(F)C1 C1(SC)CCCC(OC(C2(n3nnnc3N(C)Cc3ncccc3Br)CC2)=O)C1 N1(C(C(CCOCC)NC(c2cnsc2)=O)=O)CC(C(N)=O)CCC1C C(CCCC(=O)NC1(CC(=O)NCc2cccnn2)CC1)(OC)OC N1(CCC)CC(C)CCC1C.n12cnnc1C(=O)NCC2=O.C(C(C)C)SCC C1(NC(c2c(CNC(=O)CC3CCOC3)cco2)=O)CCCC2(CC2)C1 n1(CC(N2CCC(NC(C3C(C(=O)OC)CCC3)=O)C2)=O)ccccc1=O c1(CC(=O)NC(c2ccc(C(=O)O)o2)CO)cc(F)cc(Cl)c1 C1(NC(C=CCCCC#C)=O)CCN(C(=O)CCc2c(C)c[nH]c2C)CC1 c1(CC(=O)NC2C(CNC(CCSC)=O)CC2)ccc(OC(C)C)cc1 C1(NCc2ncc(Cl)cn2)CC2C=CCC(C1)C2 n1(CCC(=O)NC2(CCNC(=O)CSc3cn[nH]c3)CC2)ncc2ccccc12 c1(-c2nc(-c3c(OC)ccc(C)n3)n(C3CCOC3)n2)ccc2nc[nH]c2c1 C12(C(=O)NCC(CNC(C3COC3)=O)OC)CCC(C1)S(=O)(=O)CC2 C12(C(=O)NCc3c(C(=O)NC4C(C)COCC4)n(C)nn3)CCCN(CC1)C2 N1(C(C2(N(C)C)CCC2)=O)CC2CC(C1)N(C(=O)CCC(=O)OC(C)(C)C)C2 C1(C)(C(=O)NCC23C(CN(C(c4c(C)nncc4)=O)C2)C3)CCN(C)CC1 Cc1ccnc2c(C(N3CCC3CNC(C3Cc4nccn4C3)=O)=O)cnn12 c1(C(N2CCC(C(C)NC(c3cscc3C(F)F)=O)C2)=O)ccc([N+](=O)[O-])s1 NS(=O)(=O)CCCCCCC(=O)NC1CCN(C(=O)CCCC#N)CC1 C1(C(c2n(C(C(=O)OC)C)nnn2)NCCCSC(F)(F)F)CC2(C1)OCCO2 C1(NC(=O)COCC2CCOCC2)CCN(C(=O)CN2CCCC2)CC1CO N1(c2c(C#N)cncn2)CCc2sc(C(=O)Nc3cc(Br)c(F)cc3Br)cc2C1 c1(C(=O)NCC2CCCN(C(C3C=CCC3)=O)C2)c(Cl)ccc2ncccc12 N1(CCCOCC)CCC2(CC1)CN(C(=O)CCNC(N)=O)CC(C)O2 C1(C(=O)NC2CCCC(NC(c3c(OC)c[nH]n3)=O)C2)CCCCC(F)(F)C1 c1(C(c2nnnn2CCCC2CC2)NCCCCC=C)nn(C)c(Cl)c1Br CCC(C)CCC(=O)NC1(CO)CCCN(C(c2ncc[nH]c2=O)=O)C1 C1(CC=C)(NC(=O)CC2(CN(C)C)CCC2)CN(C(=O)CC2CC2(C)C)C1 C(=O)(C(O)CCCNC(c1cncc(C)n1)=O)NC(CC(C)(C)OC)C C(=O)(C(CC)C(C)C)NC1(CC=C)CCN(C(c2cnc(Cl)[nH]2)=O)C1 N1(C(c2c(CC)n(CC(C)C)nc2)=O)CC(NC(C2CC(O)C2)=O)C(C)(C)C1 c1(C(N)=O)ccc([N+](=O)[O-])cc1NC(=O)CCc1nc[nH]n1 CCCCCCC(C)C(=O)N(C1(CC(N2CCC3(CCC3)C2)=O)CC1)C Cc1ccn(CC(=O)NCCN(C(=O)CC2(C)CCS(=O)(=O)N2)C)c(=O)c1 C(=O)(C1=CNC2=NCCC2=C1)NCC(CCNC(c1c(SC)cnn1C)=O)(C)C c1(CC(N2CCC(N(C(CC(C)(C)OC)=O)C)C2)=O)cc(Br)ccc1C c1(C(N2CCC(CS(=O)(=O)NC)C2)C(=O)NC(CC)(C)C)cc(C)co1 C=C(C)CCCC(=O)NC1CCCC1NC(=O)Cn1nc(C)n(C)c1=O CC(C)(C)C(CNC(C1(c2ccccc2)CCOC1)=O)NC(C1(CCO)CC1)=O C1(NC(CCCCNC(C)=O)=O)COC2(C1)CN(CCOc1ccccc1C)C2 c1(NCCOC)cccc(CSc2cccc(NC(=O)OC(C)(C)C)c2)c1 CN1C2CCC1CC(C(N1CC(NC(=O)COCC3CCCC3)C(C)(C)C1)=O)C2 C1(NC(Cc2cc(C)sc2C)=O)CCN(C(C2(CO)CCC2)=O)CC1F C1(C(=O)Nc2c(C)scc2)CN(C(=O)CNC(N)=O)CC1C C=CCC(C)(CC)C(=O)NC1CCCC1NC(=O)CCC(C)(F)F Cc1ccccc1C(C)CC(=O)NCC1(NC(c2cnc(CO)s2)=O)CC1 C(CCC(=O)NCCN(C(=O)CNC(=O)CC1CCCCC1)C1CC1)OCCC C1(NC(c2c(C)n(C)cc2)=O)CC=C(C(=O)NC2COCCN(C)C2)C1 N1(C(C=NOC)=O)CC2CC1CC2NC(=O)Cn1nc(C(F)(F)F)cc1C C1(NC(C(C)OC)=O)CC2CC(NC(c3noc(C4CC4)c3C)=O)CC12 c1(C(=O)NC2COCCN(C(c3nncc(C)c3)=O)C2)cccc2oc(O)nc12 C1(CNC(=O)CO)CN(C(c2cnn3ccsc23)=O)C2(CCOCC2)C1 C1(C(=O)OC)CCC(N=c2[nH]nc(CO)cc2Br)CC1 c1(CC)c(C(=O)Nc2cnn(CC(N)=O)c2)ccn1C.C12(CC1)CC=CC(=O)N2 C1(CNC(c2c(C)cno2)=O)CC2CCC1N2C(c1cccc(C)c1O)=O C1(NC(c2cc(CC)no2)=O)CN(C(=O)C(C)(OC)SC)CC1c1cnn(C)c1 c1(N2CC3CCC(O)C3C2)nc2ccccc2nc1N1CCC(F)C2(CCC2)C1 C1(C(=O)NCC#CCNC(=O)CCCc2ccsc2)CN2CCN1CC2 c1(C(N(CCCNC(=O)C#CC2CC2)CC)=O)ccc(F)c(C)c1C#N c1(OC)cc(CN2CCC(C)(C(=O)NCc3cccc(F)n3)C2)c(Br)cn1 O=C(C1CCCc2ccccc21)NC1CC(NCc2cn3cc(F)ccc3n2)C1 N1(C(C=CC)=O)CCC(C(N)=O)(CNC(=O)CCC2CCC(C(N)=O)O2)C1 N1(C(C(=Cc2ccc(F)cc2)C)=O)CCC2CCN(C(C(C)(C)C(F)(F)F)=O)C2C1 c1(OCC)cnc(C(N2CC=CC(NC(C3(C4CC4)CC3)=O)C2)=O)c(Cl)c1 N1(C(C(CCC)N(C)C)=O)CC2CCC2(NC(=O)C=CCOCCOC)C1 C1(C(c2c(C(=O)NCC3CC3CNC3CC3)cn(CC)n2)=O)CC(C2CC2)=NO1 CCCCCCC(C)C(=O)N1CC2(CC(CC(=O)NC3CCCCCC3C)C2)C1 C1(C(=O)NC2(C(N(C)CC3(C)CCCO3)=O)CC2(C)C)C2CCCC(=O)C12 c1(-n2c(-c3[nH]cc4c3CCC4)nc(C(C3CC3)OCC)n2)ccc(C)c(Cl)c1N c1(C(=O)NC(CC)CNC(c2cnnc(O)c2)=O)ccc2oc(O)nc2n1 C1(NC(C(c2scc(C)n2)C)=O)CCCC(NC(c2ccnc(C(N)=O)c2)=O)C1 C(=O)(C(C)N=c1[nH]c2ccccc2s1)NC1CN(C(CC2C(CC)C2)=O)C1 N1(C(CC=C)=O)CCCCC1C1CCCN1C(c1cc(OC)ccc1N)=O c1(C(=O)NCCCN(C(C(C=C)O)=O)CC)cn(CCOC)c(C)cc1=O C=Cc1cncc(C(=O)N(CCC(C)N(C)C(C)=O)C)c1.C12CCCN(C1)C2=O C(=O)(CN1C(=O)Cc2ccccc21)NCC1(C)N(C(CN=S(C)(C)=O)=O)CCC1 C1(C(=O)NCC2(N(C)C)CC2)CC(NC(=O)C(F)C2CCOC2)C1 c1(SC)ncc(N)c(C(=O)NCC(C)(C)CNC(C2CCCN2C2CC2)=O)n1 c1(C(=O)NCC(CC)NC(C2(C(F)F)CC2)=O)sc2ccccc2c1CS(C)=O c1(-c2nc(C)sc2)cccc(C(=O)N(CC(C)NC(C2CCCN(C)C2)=O)C)c1 C12(CNCC(c3ccc(F)cc3)CO)CC1CCC2(F)F N1(C(C2CC2C(F)F)=O)CCC2C(C1)CN2C(=O)CC(C1CC1)C1CC1 c1(C(N2CCC(C(=O)NCCCCC#C)C(O)C2)=O)ccc(O)c([N+](=O)[O-])c1 c1(CNC(=O)CC2CN(C)CC2O)cccc(SC(C)(C)C(=O)N(C)OCC)c1 N1(C(CC(C)=C(C)C)=O)CCOC(CNC(=O)C(C)(F)c2ccon2)C1 CN1CC=C(C(=O)NC(C2CN(C(c3cccc(N(C)C)n3)=O)CCO2)C)C1 c1(C(N2C(C3CCN(C(C(C)OCC#C)=O)C3)CCC2)=O)nnn(C)c1CC C1(CNC(C2C3(CC(NC(C4C5CCCOC45)=O)C3)C2)=O)CC2(C1)CC(O)C2 C(CC(C)(C)C(=O)NCc1nn(C)cc1CO)NC(C1CC(OC)(OC)C1)=O C(=O)(C1=NN2CCCN=C2N1)NCC1CCC(NC(c2cc(C)cc(C)c2)=O)C1 C1(CC)(CC)CCN(C(=NCC2CCCC23CCOCC3)NC2CCCC2)C1 c1(C(=O)NCC(C)NC(c2c(C)n(C)nc2Cl)=O)cc2cc(Cl)sc2[nH]1 C(C(CNC(=O)CC(C)N(C)C(c1nnccc1C)=O)C(C)C)OC O=C(NNc1ccc2ccccc2n1)NCCC1CC2CCC1C2 c1(OCC)cccc(C(=O)NC2(C)CC(NC(C3CN(C)CC3C)=O)C2)c1N C(C(C)(C)CC(=O)N1CCCC(F)C1)NC(C(c1ccn(C)n1)(C)C)=O C1(CC(=O)NCC(C)NC(CC)(C)C)CC2(CC2)CN1C(=O)C(C(C)(C)C)OC N1(C(C2CCCN(C(C=CC(C)C)=O)C2C)=O)CCN2CC(F)CC2C1 N1(C(Cn2nc(C)c(Cl)c2)=O)CCC(NC(C2CC(F)(F)C2)=O)C12CC2 C1(C(N2C(C)(C(N3CCC(OC)C3)=O)CC2)=O)C2CCC(C2)C1C Nc1cnc(Cl)cc1C(N1CC(CNC(c2ccc(F)cc2Cl)=O)C(F)(F)C1)=O C12(C(NOCC(=C)Cl)=O)CCC(CC1NC(C1(C#N)CCOC1)=O)C2 C=CC(O)C(=O)N1CC(=C(F)CNC(C2CCCN2C(=O)OC(C)(C)C)=O)C1 c1(CC)noc(C)c1CNC(=O)CN(C1CC(C#N)C1)C(C1C2CCC(F)C12)=O n1(CC)ncc(C(N2CCC2(C2CCOCC2)C)C(=O)NCCC#N)n1 c1(C(=O)NCC(C)(C)OCCNC(C(C)OCCC#C)=O)ccccc1Cl c1(C(=O)NCC(CNC(C2C(CCCC)C2)=O)OC)cccc(C2OCCO2)c1 c1(C(=O)NCCC(C)N(C(C=C(C)C)=O)C)cc(C(F)(F)F)nn1C c1(C(N2CCCC(N(S(=O)(=O)CCCCl)C)C2)=O)c(Cl)cccc1[N+](=O)[O-] CCCC(C)(O)CC(=O)N1CCC(NC(c2ccnn2CC(F)(F)F)=O)C(O)C1 Cc1cnccc1C(=O)N(C)CC1CCCN(C(c2ncccc2N(C)C)=O)C1 Cc1c(CC(N2CCCC(Nc3cncc(Cl)n3)C2)=O)cnn1C c1(-c2c(C(=O)NC)nccc2)ccc(S(=O)(=O)N2CCC23CCCCC3)cc1 CC1CC2CN(C(=O)C(O)C3CC3)CC2N1C(C12CCC(CC1)C2(C)C)=O C1(C(=O)NCC(N(OC)C)=O)CCC2CCC1N2C(=O)CN1CCCNC1=O C1(n2cc(CC3(n4cncn4)CC3)nn2)CCCN(C2CCC2)CC1 CC(C)C(F)(CNC(=O)C(N)=O)C(=O)NCC1(n2ccnn2)CC1 c1(NC(c2ccc(C)cc2)C)ncnc(NC(C2CSC2)C2CCC2)c1C c1(CC)sc(C(=O)NCC2CC2CNC(=O)CCc2cccnc2F)cc1C CC(C)C(C)C(CNC(c1cccc(F)c1)=O)NC(c1coc(Cl)c1)=O c1(C(=O)NC2CCCC(CNC(=O)C=C3CC3)C2)cc(F)cc2cc[nH]c12 Cc1nc(C#N)ccc1NC(C1C2CCC(C2)N1C(c1sccc1Cl)=O)=O Cc1cc(C(=O)NC2CN(C(=O)COC3CC=CC3)CC2(C)C)cc([N+](=O)[O-])c1 c1(CC)cc(C(=O)NCC2CCCCC2NC(C2C=C(C)CS2)=O)n(C)n1 c1(C(C)C)cc(C(=O)NC2CC3CC2N(C(C2(F)CC2)=O)C3)c2ccccc2n1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1C2C(NC(=O)CSc3cn[nH]c3)CC(C2)C1 c1(C(=O)NCC(C(C)(C)C)NC(c2cc(C)sc2)=O)cc2c(C)cc(Cl)cc2[nH]1 C(=O)(C1=NN(CC)C(=O)CC1)N1C2CC(NC(CNC(CCC)=O)=O)CC1CC2 C12(CNC(c3cc(C(C)C)ncn3)=O)CCC1C1(CC2)OCCO1 N1(C(C)=O)CCCCC1CC(=O)NC(C)(C)CCNC(C1CC(CF)C1)=O C1(N(C(c2ccc(CC)[nH]2)=O)C)CCCN(C(=O)C(C)(C)C2CCCO2)CC1 c1(-c2cc(C)cc(C)c2)ccc2c(c1)CCN(C(=O)CNC(N)=O)C2 C#CCCCCCC(=O)N1CCC2(NC(c3cnn(CCN(C)C)c3)=O)CC2C1 N1(C(Cn2c(C)cc(C)n2)=O)CCC(CO)C(NC(c2cnc(S)n2C)=O)C1 N1(C(C2C(CC)CCO2)=O)CCc2c(OC)c(O)cc(C(=O)O)c2C1 C12(NC(C(CC#C)O)=O)CCC(CC1)N(C(c1cc(O)ncc1Br)=O)C2 c1(C(N2CC3C(CNC(c4cccc(C)n4)=O)(C3)C2)=O)oc2ccccc2c1C Cc1nn(C)c(Cl)c1C(N1CCC12CN(C(c1ccnc(CC(C)C)n1)=O)C2)=O C(CCCC(OC)OC)(C=O)N(C(C)C(=O)OC(C)(C)C)C.CN Cc1cnn2ccc(C(=O)N(CC(C)NC(=O)C(C)(C)c3cnn(C)c3)C)nc12 N1(C(C(C)Nc2nccs2)=O)CCC2(C1)CN(C(c1ccc(F)cn1)=O)C2 C(CCCN=c1[nH]c(=NCC23COCCN2CCOC3)c2ccccc2[nH]1)OC C1(OC)CC(NC(c2cnns2)=O)C12CCN(C(c1c(C)[nH][nH]c1=N)=O)CC2 C(CCCCC(=O)NCC1CCN(C(=O)CCS(C)=O)C1)=CC C1(N(C)C(C2CCCCC2)=O)CC2CCC(C1)N2C(=O)C(=O)Cc1ccccc1 c1(C(=O)NCC(CC)NC(=O)CSC(C)C)cc(=O)c2ccc(O)cc2o1 c1(C(NOCCOCC#C)=O)coc2c1CN(C(=O)CN1CCCC1C)C2 c1(C(=O)NCCCCN(C(=O)CCCC2(C)N=N2)C)cnn2ccncc12 N1(C(c2cc(C)c(C)s2)C(=O)NCC=C)CCNC(=O)CC12CCOCC2 C12(C(CNC(=O)COc3ccccc3)NC(C3CCCO3)=O)CCC(CC1)C2 c1(C(C(=O)NCc2nnn(C)n2)N(CCC(N)=O)CC)cc(Cl)ncc1Br N1(C(c2c(CC)onc2)=O)CCC(C2(O)CCN(C(=O)C(C)(C)C)CC2)CC1 CCC(C(=O)NCC1CC2(C1)CN(C(=O)CC(C)=C(C)C)C2)C(C)O C(=O)(CCCC(=O)NC1CCC(N(C(=O)Cn2nnc(C(C)C)n2)C)C1)OCC C1(N(C)Cc2ccc(-c3c(C)n[nH]c3)cc2F)CCNC2(CCC2)C1 c1(NC(N2CCC(c3scc(C)n3)C2)=O)cc(F)c(N2CCOCC2)c(F)c1 N1(C(CN2C(C)CC2)=O)CC2C(CNC(=O)C=Cc3ccc(C(N)=O)o3)C2C1 Cc1nc2cc(C(=O)NC3CCN(C(c4ncsc4C)=O)C(C)C3)cnc2[nH]1 CCS(=O)(=O)C=CC(=O)NCCCCC1CN(c2ncc(C#N)cc2F)C1 c1(OC)ccnc(-c2nc(C(N3CCN(CCNC4CC4)CC3)=O)cs2)n1 n1(CCOCC)nnnc1C(c1cnc(C)s1)NC(CC)CC c1(C(N2CCC(C(C)NC(COCC)=O)C2)=O)cc(NC)ccc1Cl N1(C(c2nc(C(C)=O)sc2)=O)CCC(CCCNC(C2(F)CCOC2C)=O)CC1 c1(C(N(C2CN(C(C3(C)CC3F)=O)C2)C)=O)cc2oc(Br)cc2[nH]1 c1(N2CCC(CCOC)(NC(c3cnc(O)n3C)=O)C2)nc2cccnc2s1 c1(CNC(c2ccsn2)C)nnnn1C1CC1 Cc1nc2c(C(=O)NCC3=CCN(C(=O)CCS(C)=O)CC3)ccnc2[nH]1 CC(C)C(O)C(=O)N1CC(O)(C(F)C(=O)NCC2CCCN(C)C2)C1 Cc1cc(C(N2CCCC3C2CCCN3C(=O)C=CCO)=O)c(N)c([N+](=O)[O-])c1 C(CCCCC(=O)NC1C2CC1N(C(=O)Cc1cnc(C)s1)C2)NC(C)=O C(=O)(C(F)Cc1ccccc1)NC1C(NC(=O)CN2CCC2)C1 N1(C(c2c(C)nsc2Br)=O)CCC2(C1)CN(C(=O)CSCCC#N)C2 c1(OCC)cc(N2CCCC(C(C)NC(=O)C(F)n3cccn3)C2)ncn1 C1(CCNC(C(CCOC)C)=O)CCCN(C(c2ncn(C(C)C)n2)=O)CC1 c1(CC)onc(C(N2CCCC(N(C(=O)C(CC)NC(N)=O)C)C2)=O)c1C C(=O)(C#CC1CCCCC1)N1CC(NC(CCCCCCC)=O)C2(C1)CCC2 N1(C(c2c(C)nc(C)o2)=O)CCC(C(=O)NCC2CCN(C(N)=O)C2)CC1(C)C C1(NC(CNS(CC)(=O)=O)=O)CC(C)CN(C(c2ccnc(C)c2)=O)C1 N1(C(CCN(C)CCO)=O)CC2(C1)C(NC(C1CC3CC3C1)=O)CCS2(=O)=O c1(C(=O)NC(CC)(C)CNC(=O)CSc2cccs2)cnccc1Cl N1(C(C2CC2(Cl)Cl)=O)CC2CCN(C(=O)CCCOc3ccccc3F)C2C1 c1(C(CC(=O)O)C(=O)OC(C)(C)C)ccnc(-c2ccc(-c3ccco3)cn2)c1 N1(C(c2nccc(OC)c2)=O)CCCN(C(C2CC=CCC2)=O)CC1CO c1(OCC(=O)N(CCCCCNC(=O)CNS(C)(=O)=O)C)cccc(F)n1 C1(CN(C(C2CS(=O)(=O)C2)=O)CC)CCN(C(=O)CC2CCCCC2)CC1 C1(CCCC)CN(C(C23CC(F)(C2)C3)=O)CCN1C(=O)CCC1CC(F)(F)C1 N1(C(C(c2n(C)cnc2)O)=O)CC(O)CC1CNC(=O)Cc1cccc(F)c1 N1(CCCOCC)CCC(C(C)NC(=O)C(C2CCCC2)OC)CC1 c1(OCC)cccc(C(=O)NC2CC(O)CN(C(=O)CCCF)C2)c1N c1(C(=O)NC2C(CNC(c3c(Br)cn(CC)n3)=O)C2)cccc2[nH]ncc12 N1(c2cc(NCC(C)(C)CCO)nc(C)n2)CCN2CCCC2C1 c1(C(N2CCC(C(=O)NC3C(CN(C)C)CCC3)CC2)=O)ccc(N)c(F)n1 C1(C(C)C)CN(C(c2cnn(C)c2)=O)CCCN1C(c1cnc(O)c(F)c1)=O C1(NC(C2OCCN(C(C)C)C2)=O)CCN(C(C2CC3(CCC3)C2)=O)CC1O c1(C(N2CC(c3c(C)ccs3)(O)C2)=O)ccnc(C(F)(F)F)c1[N+](=O)[O-] C1(NC(C(C(C)C)C)=O)CN(C(C2(c3ccccc3F)CCC2)=O)CC1(C)C C1(OC)CN(C(C2(S(N)(=O)=O)CC2)=O)CC1NC(c1coc(C)n1)=O c1(C(=O)NCC(=C)CCNC(C2(C)CCOC2)=O)cc(Br)cc(Cl)c1F C1(NC(c2cncc(OC)c2)=O)CC1C1CCN(C(C2(CC(F)F)CC2)=O)CC1 C(=O)(C(C(=O)NC1(C(=O)NC(c2ncc[nH]2)C)CCN(C)C1)OC)OCC C1(CNC(C(C(C)(C)C)OC)=O)CC2CCC(C1)N2C(=O)C(C)(C)SC N1(C(c2cccc(CC)c2)=O)CCC(CNC(=O)Cn2ccccc2=O)C(C)C1 CCC(CC(=O)N1CCN(C(c2nccc(C)n2)=O)CC1CCO)CC(F)(F)F C12(NC(C(c3ccccc3F)C)=O)CCCC1N(C(=O)CCC(N)=O)CC2 N1(C(C)=O)CCc2c(NC(c3cc(-n4nnnc4C)cc(F)c3)=O)cccc2C1 N1(C(C(CC(=C)C)NC(c2nnn(CC)c2C)=O)=O)CCC(O)C(C)(O)C1 c1(C(N2CC3N(C(C=C(CC)C)=O)C(CC3)CC2)=O)cc(C)cc([N+](=O)[O-])c1N C(=O)(C(CO)N(C)C)NCCN(C(=O)COCC1CCCOC1)CCC c1(OCC)cc(Cl)ccc1C(=O)NC1(CCNC(=O)Cc2ccon2)CC1 c1(N2CC(C)NC(C)C2)ccc(S(=O)(=O)N2CCC3(CC(F)C3)C2)cc1 C1(CNC(C23CC(CCC)(C2)C3)=O)(COC)CCN(C(=O)CC)CC1 Cc1ccc(-n2nc(C(=O)N(C3CCC4(CC3)CC4)C)c(C)n2)c(C)c1 CCCCCC(O)CC(=O)N1CC(CC(F)C(N2CCOC(CC)CC2)=O)C1 CCC(C)CCCCC(=O)NC(CC(=O)N(CCO)C(C)C)C(C)OC c1(CC)cc(OC)cc(C(=O)NCC2CN(C(=O)C(C)(COC)CC)CCO2)c1 c1(C(=O)NC(C)CCCNC(c2ccoc2)=O)ccnc2ccccc12 C1(C(=O)NC2C(C)(C(F)F)C2)(NC(c2ccc(CCF)cc2)=O)CC(F)(F)C1 c1(-c2onc(-c3cc(C)cc(C)c3)n2)cnn2c1CCCC2 Cc1ccc(C(N2CC(NC(=O)C(C)(C)c3cnc[nH]3)CC(C)C2)=O)c(O)c1C Cc1nc(=NCCC2CCC(NC(c3nc(F)ccc3Cl)=O)C2)[nH]cc1Br C1(C(C(=O)NCC2(NC(c3ccc(Cl)[nH]3)=O)CCC2)=O)CCCCC1 N1(C(C=C(C)Cl)=O)CC(NC(=O)C(c2ccc(C(F)(F)F)cc2)F)CC1(C)C c1(CC(=O)N(C)CC2N(C(C(CC)=CC)=O)CCOC2)cccc(C)c1Cl C1(NC(c2cc(C(C)=O)[nH]n2)=O)CC(C)CN(C(C2CC3CCC(C2)S3)=O)C1 c1(COC)cc(C(=O)NC(C)(C)CN(C(=O)CCCn2cccn2)C)no1 c1(CCC(=O)N(CC(C)NC(=O)CC2CCC(C)CO2)C)ccc(Br)cc1 C(=O)(C(C)(C)C1=CCS(=O)(=O)CC1)N1CC(N(C(CC(CC)C(F)F)=O)C)C1 c1(C(=O)NCCN(C(C2CCC(=O)O2)=O)CC)c(C(F)(F)F)nn2ccccc12 c1(C(=O)NCC(c2ccccc2)NC(C=C(C)C2CC2)=O)ccnnc1S CC1CN(C(=O)C2CC2)CCCN1C(=O)C=Cc1ccc(Cl)cc1F N1(C(C(=O)Nc2ncc[nH]2)=O)CCC2(CCN(C(c3ccc4c(c3)CC4)=O)C2)C1 N1(C(c2cnn(-c3ccc(Br)cc3)n2)=O)CC2CCCC(C1)C2(F)F C1(CNC(c2c(C)csc2)=O)CCN(C(c2[nH]ccc(=O)c2C)=O)CC1O c1(C(N2CCN(C(C=C(C)C(C)C)=O)C3C2C3)=O)cnc2c(c1)CCCO2 N1(C(C2C(C(=O)OC)C2)=O)CC(C2CCCN(C(=O)C(C)N(C)C)C2)C1 C(N=c1nn[nH]n1C)C1(F)CC(NC(C(C)C2CC2)=O)C1 N1(C(c2c(C)c(=O)cc[nH]2)=O)CCC(C)(C)CC1C(=O)NC12CC(F)(C1)C2 N1(C(C=CCC)=O)CCN(C(c2cc(C)[nH]n2)=O)CC1c1ncc[nH]1 c1(CC(=O)NCC(C(C)C)NC(CC(CC)SC)=O)ccc2occc2c1 N1(C(C(C=C)C)=O)CC2CC(C(=O)NC(C(C)C)C3CCC3)C(C2)C1 c1(C(=O)NCC(CO)NC(C2(OCC)CCCC2)=O)cccc2c1NCC2 CN1C(=O)CCCC1C(=O)NCC1CN(C(c2ccc(CO)nc2)=O)CC1(C)C N1(CCC)CC(C(=O)NCCOCC(C)(C)NC(c2sccc2C)=O)CC1=O C1(C(=O)NCC2C(NC(c3cc(C4CC4)[nH]n3)=O)CC2)COc2ccccc2O1 c1(C(=O)NC(CNC(C2(C)C(C)C2)=O)C)cc(C(F)(F)F)ncc1N c1(C(N2CC(NC(C3(OC)CCCOC3)=O)C2)=O)ccc(C)c(F)c1N C(=O)(CCC(=O)NC1CC(N(C)C(C2COCCN2CC2CCC2)=O)C1)OC C(=O)(C1=CCS(=O)(=O)C1)NCC(CNC(Cc1ccn(C(C)C)n1)=O)(C)O C(CC)(C(=O)NC(C)C(CO)NC(c1ccc(C2CC2)s1)=O)=CC C(=O)(C(O)C(F)(F)F)N1CCN(CC(=O)NCC(C)(C)O)CC1 C1(CCNC(c2cc(C3CC3)ncn2)=O)CSCCN1C(=O)CC1C=CCC1 c1(N2CC(OC)C(F)C2)nc2c(c(=NCC3(C4CCCO4)CCC3)[nH]1)CCC2 CC(C)C(C(=O)NC(CCF)C(=O)N(C1CC2CCC1O2)C)C1CCC1 Cc1cc(C(=O)NC2CCN(C(=O)Cc3ccc(Cl)cc3)C2)c2c(n1)CCCC2 c1(CC)ncc(Br)cc1NC(C1CN(C(c2ccc(O)cn2)=O)C1)=O c1(C(N2CC(NC(c3ccnc(OC)n3)=O)CC2(C)C)=O)cc(F)c(F)c(F)c1 c1(NC2(c3n(CCCSC)nnn3)CCCSCC2)ccc2[nH]ccc2c1 C(CC(=O)NC(C)(CNC(C1(O)CCOCC1)=O)CC(C)C)(C(N)=O)NC(C)=O c1(C(=O)NCC2CCCCC2NC(=O)CCc2cncs2)cnc2ccoc2c1 N1(C(c2cc(SC)oc2C)=O)CCC(C)(NC(=O)CC2C(=O)ON=C2C)CC1 CC1CCCCC1CC(=O)NCC1CN(C(=O)CCc2ccccc2F)CCO1 C(CC(C)c1ccccc1)(C(=O)Sc1ccc(F)cc1)N1C(CC)CC(C)C1 c1(C(=O)NC2C(NC(c3cn(C)nn3)=O)CC2)cccc2c1CCCC2=O c1(C(N2CCC(O)C(C)C2)C(=O)NC(CC)C)sc(S(N)(=O)=O)c(OC)c1OC C1(NC(Cc2nc(C(C)C)sc2)=O)CC2(C1)CN(C(=O)C(F)CC1CCOC1)C2 C(CC(=O)N1CC(C)CC(O)C1)(C(F)(F)F)NC(C1C(C)CCOC1)=O CC(CN(C(c1cccc(C(F)(F)F)c1)C(=O)NCCC#N)C)C(F)(F)F C=C=CC(C)C(=O)N1CCN(C(=O)Cn2cnc(-c3nc(C)no3)c2)CC1 N1(C(C2(C#C)CC2)=O)CCC(O)(C2(NC(c3coc(S(N)(=O)=O)c3)=O)CC2)CC1 CCC(CC)(C(=O)N(C)CCOCCNC(C1CC2CCCC2C1)=O)OC c1(C(N2C(CNC(c3cccnc3)=O)COCC2)=O)nccn2cnnc12 Cc1cccc(C)c1C(N1CSCC1C(c1ccccc1)=O)=O.NCS CCC(F)C(=O)NCC(C)(C1CCC1)NC(=O)C(C)(C)C1CCCCC1 CCC(CCC(=O)NC1CC(=O)N(C)C1)NC(c1cc(C)sc1N)=O c1(CNC(=O)CN(C(=O)Cc2ccsn2)C2CC2)ccc(O)c(F)c1 N1(C(CCC(C)C)C)CCC2(CC1)CC2(C)C(N1CCNC(=O)C1C(C)C)=O N1(C(CC(C)F)=O)CC2CC1CCN2C(=O)CSS(C)(=O)=O c1(C(N2CC(N(C)C(c3cnc(Cl)s3)=O)C(C)(C)C2)=O)ccc(S(N)(=O)=O)o1 C(C)(C)(C(=O)NCC1(F)CN(C(=O)CC2(C)CCCO2)C1)OC(C)=O C(=O)(CCCCCC(=O)NCCCC(C)NC(C1CCS1(=O)=O)=O)OCC c1(CC(=O)NCCNC(C2C(c3c(C)nn[nH]3)C2(C)C)=O)c[nH]c2cnccc12 N1(C(=O)C#CC2CC2)CC(CO)C2(CCN(C(C3CCC=CCC3)=O)CC2)C1 N1(C(C(C#C)(C)C)=O)CCC2CCN(C(c3c(SC)cccc3F)=O)CC2C1 Cc1ccn(CC(=O)NCC2(O)CN(C(=O)Cc3ccccn3)C2)c(=O)c1 C12(NC(C(CCC#C)O)=O)CC(C)(C1)OC21CN(C(=O)C(CC)SC)C1 OC1CCN(C(=NCCCOc2ccc3c(c2)CCC3)NCc2ccco2)C1 Cc1ccc(CC(=O)OCCSC2CCCC2)cc1C.c12ccc(cc1)c(=O)[nH]2 C(C1COCc2ccccc21)NC(=NCC=C)NCC1CCS(=O)(=O)C1 c1(C(=O)NCC(CCNC(c2ccc(CO)o2)=O)O)cc2ccncc2s1 N1(C(C2(SC)CCC2)=O)CCC2(CC(NC(c3ccnc(C(C)C)n3)=O)CO2)C1 C(=O)(C(C)(F)C(=O)NC1CCC(C(=O)NCc2cnsc2)C1)OC c1(C(N(CCCN(C(=O)Cc2c[nH]nc2O)C)C)=O)nn(CC(F)(F)F)cc1Cl N1(C(C=CCC)=O)CCC2(COCC(CNC(=O)CCC3CC(F)(F)C3)O2)C1 C(=O)(C(CCC(C)C)NC(=O)CC(C)C(C)C)NCc1c(C)ncs1 C1(C(=O)NC2(CNC(=O)C(C)Cn3ccnc3)CC(OC)C2)CCCCCCC1 c1(OCC(=O)NC2C(NC(C3CC(C)(C(=O)OC)C3)=O)COC2)ccccc1C c1(CC)nc(C)c(CC(N2CC(C)N(C(=O)COC3CC3)CC2C)=O)c(C)n1 N1(C(COCCOCC#C)=O)CCC(C)(CNC(C2CC3CC2CC3O)=O)CC1 C(CC(C)C(F)F)NC(C1CCC(CNC(c2c(C)snn2)=O)C1)=O c1(C(=O)NCCCC2(NC(CC=C)=O)CC2)nnn(C2CC2)c1C(F)F C(C(C)(C(=O)NCC(O)(CO)CO)NC(=O)Cn1cnnc1)SC N1(C(c2c(CCNC(C(C)=CC3CC3)=O)n[nH]c2)=O)CCC(CC2CC2)CC1 c1(C(N2CCOCC(NC(C3(C)CS(=O)(=O)C3)=O)C2)=O)cc2c(s1)CCC2=O C(=O)(C(C)(C)C(=O)N(C)C)NCC(CCC)NC(c1cnn(C(C)C)c1F)=O n1(CC(=O)NC(C2N(C(c3c(OC)csc3)=O)CCCC2)C)ncc(C)cc1=O Fc1c(CCCNC(=O)CCn2cc(I)cn2)cccc1Cl C1(C)(CNC(CN(C(=O)OCC)C)=O)CCN(C(=O)C=C2CCSCC2)C1 CCCCCCC(=O)NC(c1ccc(F)cc1)CNC(=O)C(C)(C)OC(C)C C1(CC(N2CC(NC(c3n(CC)ncc3)=O)C2)=O)CCCC2(CC2)C1 c1(OC)c(NC(c2cccc(I)c2)c2ccc(F)cc2)nnn1-c1ccccc1 N1(C(C(C)O)=O)CC2CN(C(=O)CCn3ccnn3)C2C1 c1(C(C(=O)NC(C)CC)N(C2CC(OCC)C2(C)C)C)ccc([N+](=O)[O-])c(Cl)c1 C1(CNC(C2(CCCC)CC2)=O)CCCCC1NC(C1(SC)CC1)=O c1(CC(=O)NC(C(=O)OC)Cc2cn(C(C)C(=O)O)nn2)cncc(C(C)C)c1 c1(C(N(C(CC)C(N2CC3(C2)CC3(F)F)=O)C)=O)ccc2nccn2c1 c1(CC(=O)NC(C2(CNC(C(CC=CC)C)=O)CC2)C)ccc(C(C)=O)c(C)c1 c1(C(N(CC(C)NC(C2(O)CCSC2)=O)C)=O)ncc2[nH]ncc2n1 c1(C(=O)NCC(CC)(C)NC(c2csc(C)c2)=O)cn2c(n1)C(C)CCC2 C1(CNC(C2C(OCC)C2)=O)CCCN(C(=O)CN(C2CCSC2)C)CC1 c1(C(=O)NCCCCC(C)NC(c2nc(OC)c(C)s2)=O)cc(N)c(O)c(F)c1 c1(CCC(=O)N(C2CCN(CC3CCNC3=O)CC2F)C)nc2ccccc2s1 C(=O)(C(C)CCCC(C)C)N1CCC(C(=O)NC(CC#C)CO)C1(C)C C(CO)(C(=O)NC(CC1CCCC1)C(=O)NCCOC(F)F)OC N12CCC3(CCCN3C(=O)C=CC1=O)C2.c1(C(=O)NC2CC2)cccc(=O)o1 O=C1CN(CCc2cc(Cc3ccccc3)on2)C(=O)N1Cc1ccccc1 c1(CCCOC(c2n(CC)ncc2)=O)ccnnc1C CCC(C)CCC(=O)N1CC2CC(NC(c3cnn(C)c3CC(C)C)=O)C1C2 c1(C(=O)NC2C(CNC(C=Cc3ccc(C)s3)=O)CC2)cnc2[nH]cnc2c1 c1(C(C(N2CC(CCNC(CCCCOC)=O)C(C)C2)=O)=O)ccc(F)c(Cl)c1 c1(C(=O)NCC(C)NC(C2CCCN2C(=O)OC(C)(C)C)=O)cncn(C)c1=O C1(Cn2cc(CNCc3n(C)nc(C(F)(F)F)c3)nn2)CCCC(F)(F)CC1 C1(C)(C(=O)OC)CC(OC)CN1C(=O)CCc1ccncc1 C12(C(=O)NCCNC(CCC3(C#N)CCC3)=O)CCCC(=O)N1CCC2 c1(C(=O)OC2COCCN(C(=O)OC(C)(C)C)C2)cc(N)c(Br)c(F)c1 n1(CCC(=O)NC2CN(C(C3COC3)=O)CC2O)sc2ccccc2c1=O C1(C(N2C3(CNC(c4cc(C(F)(F)F)no4)=O)CC(C2)C3)=O)CCCNS1(=O)=O CC1CN(C(c2ccc(CN(C)C)[nH]2)=O)CCC1NC(=O)C(O)C1CCC1 C1(C(=O)Nc2ncc(C#N)s2)CN(Cc2cccc(-c3ccco3)n2)CCC1O c1(C(=O)NCCOC2CN(C(C3(CC)COC3)=O)C2)cc2ccccc2n1C Cc1ccc(NC(=O)C(C2CCN(C(c3cnnc(Cl)c3)=O)CC2)C)c(C)n1 C=C(F)C1(CC(=O)NC2(CNC(=O)CC3CCCC3(C)C)CC(F)(F)C2)CCC1 c1(OC)cccc(-n2c(SCC3CC(F)C(=O)N3)nnc2-c2ccco2)c1 CC1CC(=O)NCC1C(=O)NCCCCCNC(c1cscc1C(N)=O)=O C1(C(N(C2CCN(C)C2)C)=O)CC(C)(C)CN1C(c1ccc(C(F)F)o1)=O N1(C(c2c(CCC)[nH]cc2)=O)C(C(=O)NCC(C(C)(C)C)OC)CC2CC12 CCC(C)CC(=O)NCC(CC(=O)NCc1cccnc1O)OC c1(OC)cc(CN(c2cc(NCc3ncc(Br)s3)ncn2)C)ccn1 c1(OC)ccc2cc(COC(=O)C(C(C)C)N3CCCS3(=O)=O)c(Cl)nc2c1 C1(C(=O)NCCN2CCNC2=O)CC12CCN(C(=O)CC1CCCCC1)C2 C1(CNC(c2c(C)nccn2)=O)CCC(C)(C)CN1C(C1C(C)C1(F)F)=O CC1(C)Cc2cc(Br)ccc2C1NC1C(C)(C)C1(C)C N1(C(C(=O)NC(COC)C(F)(F)F)=O)CC2(CCSCC2)C1 Cc1cc(C)c(NC(C2CCCCC2NC(=O)CC(C)Oc2ccccc2)=O)cn1 N1(C(C2N(CC)CCOC2)=O)CC2(CCC2NC(=O)CSc2cnn(C)c2)C1 c1(CNC(c2cnc(C)s2)=O)ncc(C(=O)NC2CC3CCC2C3)cn1 Cc1cc(C(=O)NC2CC2NC(=O)CC23CCCC2C3)no1 Cc1cc(NC(c2ncoc2C2CC2)=O)c(F)cc1F C=C1CCN(C(=O)CCNC(C)=O)C(C(=O)NCCC(F)(F)CC)C1 c1(CNCC2CC(C)SCC2)cnc2sc(Br)cn12 c1(C(=O)NC(c2ccc(OCC)cc2)(C)C)ccc2c(c1)c(C#N)cn2C Cc1ncc(N)cc1C(=O)NCC(O)CN(C)C(c1csc(Br)n1)=O CCCCC(F)C(=O)NC(C)C=CC(=O)N(CCC(C)(C)C)C C1(C(C)NC(C(C)N(CC)CC)=O)CCCN1C(=O)Cn1ccc(C(=O)OC)n1 C(=O)(CCN=c1ccc(C)c[nH]1)NC(C1(NC(=O)C(C)SC(F)(F)F)CC1)CC N1(Cc2ccc(NC(C)=O)cc2)CCCCC(SC)C1 S(=O)(=O)(CCc1ccccc1)N(C(C1C=CCC1)=O)C1CC1 Cn1cnn(CC(=O)NCCCC2CN(C(C3CNC(=O)N3)=O)CCO2)c1=O c1(C(=O)NC2CN(C(c3scc(C(N)=O)c3)=O)C(CO)C2)cc(O)nc(O)n1 N1(C(C(C(C)C)CNC(C23CC2CNC3=O)=O)=O)CCC2CC1C(=O)O2 CC1CCOCCN1N1CCCC(Oc2ccc(F)cc2)C1 C12(NC(C3CC3NC(c3nc(N(C)C)oc3)=O)=O)CCC(CN)(CC1)C2 C1(C(=O)NC(c2cnc[nH]2)C)C(C)CCN1C(C1CNC(=O)N1)=O C1(C(=O)Nc2cc(O)nc(C(F)F)n2)CC12CCN(Cc1cccnc1O)CC2 C(C(=O)N1OC2C=CC1CC2)NC(=O)Cc1ccc(F)c(F)c1 C1(CNCC(=O)NC2CC(OCC(c3ccccc3)C)C2)CCC2(CCC2)O1 c1(C(CNC(CC2CC(=O)C2)=O)NC(=O)CCF)cccc(Cl)c1 Cc1ccc(Cl)cc1C(=O)NC(C)CN(C)C(C1CC1(C)C)=O N1(C(c2ccc(OC)o2)=O)CC(C(=O)NC2CC23CCOCC3)C2(CCC2)C1 C(=O)(CC(C(C)C)C(C)C)NCC(CNC(C(CC(C)C)OC)=O)C c1(C(=O)NC2(C)CCN(C(CC3N(CC)CCC3)=O)C2)ccc(N)c(SC)c1 c1(Cc2cn(NCC(N3CCOCC3)CO)nn2)cnn2c1CCC2 c1(C(=O)OC)ncnc(SC)c1OCCOCCNC(=O)NCCCOC C(CC(C)C)(C(=O)NCCc1ccoc1)NC(C(CC)OCC)=O N1(C(=O)OC(C)(C)C)CC2ON=C(CNC(C3CN(S(N)(=O)=O)C3)=O)C2C1 CC1(C)CCC(C)(C(=O)NC2CCN(C(=O)CN3CCOC3=O)CC2(C)C)CC1 CC1CC2(CCN(C(=O)CCCN3CCCC3)CC2)CN1C(C12CCC1C2)=O C1(C(=O)Nc2cccc(NC(c3n(CCC)ccc3)=O)c2)CC12CC(C)(C)C2 Cc1cc2[nH]c(C(=O)NCC3CC(C)(C)CN3C(=O)CSCC#N)cc2o1 C(CN=c1[nH]c(=NCC(C2CCCO2)OC)c2sccc2[nH]1)c1n[nH]c(=N)o1 c1(C(N(CC2N(C(C3C(=C)C3C(=O)OC)=O)CCC2)CC)=O)cc(Cl)cn1C N1(C(C(C)SCCCC)=O)CCC(CNC(=O)CCn2ccnn2)(COC)C1 Cc1nc(=NCC(CC(C)C)NC(=O)CCC2CC2(Cl)Cl)s[nH]1 CC1CC(F)(F)CN1C(=O)C(=O)NCC(c1cc(F)cc(Cl)c1)N CCC(C)C(O)C(=O)N1CCCC1CN(C(=O)C(c1ccc(C)s1)C)C1CC1 c1(C(=O)NCC2CN(C(C(C)(C)OC)=O)CC2C)cc2cnccc2cc1F CC1CN(N2CCCCC2c2cncnc2)CCC1(F)F c1(C(N2CCCOC(CC)C2)C(=O)NCCCSCC)cc(F)c(F)c(F)c1F Cc1cc(CN(C)C)nc(NC(C2CC(F)C2)=O)n1 Cc1nc(C(C)C)ccc1C(=O)NCCC12CCC1CN(C(c1ccns1)=O)C2 c1(C(=O)NC(C2N(C(C(C)c3ncco3)=O)CCC2)C)ccc(Cl)cn1 CN1CCN(C(=O)CC2(C)OCCO2)C(C(=O)NCCC2CCC(C)(C)O2)C1 C=C(Br)CCC(=O)NCc1cn(C2CN(C(=O)CC3(n4ccnc4)CC3)C2)nn1 Cn1cc(CC(N2CCC2CNC(c2cncnc2O)=O)=O)c(Cl)n1 N1(C(CC(CN(C)C)O)=O)CC2CCC(Nc3nc(C#N)ncc3Cl)C2C1 C1(NC(C(C)(C)OC(C)=O)=O)COCCC1NC(c1cnc(C(F)(F)F)nc1)=O N1(C(C)C)CC2CCC1CN2N1C(C(=O)N(C)C)CCC1CO N1(C(C=CC(CC)=CC)=O)CCC2CCN(C(c3ccc(C)nn3)=O)CC12 c1(C(N2CC(NC(C(CC)(C)C)=O)C(F)C2)=O)ccc(NC(C)=O)cc1O c1(NS(CC)(=O)=O)cccc(F)c1C(=O)Nc1cc(OC(F)(F)F)cc(Br)c1 C1(C(=O)NCCC(CCNC(c2n(CC)cnn2)=O)C)CCCC(C)(C)CC1 c1(OC)cccc(C2CC(C)CN2C(N2CC3(CCC3)C2)=O)c1 c1(C(N2CCN(C(CC(C=C)C)=O)CC2C)=O)cc(C)c(C)cc1C c1(OC)cc(C(=O)NC23CCN(C(=O)Cc4cnoc4)CC2C3)ccc1OC C1(CNC(N2C(C)CN(CC(C)(C)O)CC2)=O)CC2CCC1N(C)C2 Cc1nc(C)n(CC(=O)NCC2CC2CC(=O)NCc2cnco2)n1 C12(C(=O)NC3C(CNC(C4=C(C)CCC4)=O)CCCC3)CC3CC(CC(C3)C1)C2 C1(C(N2CC3C(CNC(c4cc(Cl)ccn4)=O)(C3)C2)=O)CC2CCC(C1)C2 C1(C(=O)NC2CC(NC(c3c(C(=O)OC)c[nH]c3)=O)C2)COCCN1C(C)=O N1(CCCNC(=O)N(Cc2ccoc2)CC2CC2)CCCCC1 C=C(Cl)CC(C(=O)N(CCCN1CCCC1)C(C)C)NC(=O)CSCC(N)=O C1(C(N(C)CCN(C)C(C2CC(NS(C)(=O)=O)C2)=O)=O)CC(C2CC2)=NO1 C1(CC(=O)NC2CC(CNC(C(C)CN(C)C)=O)C2)OCCCC1(C)C C1(C(=O)NC(c2ccc(O)cc2)C)C(O)CCN1C(c1ccc(F)cc1)=O c1(NCC(C2CCC2)OCC)ncccc1S(=O)(=O)NCC1COCC1O N1(C(c2c(CC#N)ccs2)=O)CCC2(CCC2)C(NC(=O)C=CC2CCCO2)C1 CC(C)C(=O)C(=O)NC1CCOCC1C(=O)NC(C1CCCC1)C CON=C(C(=O)NCC1CCN(C(=O)CC(C)(C)O)C(C)C1)c1ccco1 N1(CC=C)C(=S)NC(c2cc(C)c(F)cc2Br)C(C(=O)N(C)C)=C1C C=C=C(C)CC(=O)NC1COCC1C(=O)NCCCC(=C)C c1(CCC(=O)NCCNC(C=CC(=O)NC2CC2)=O)c[nH]c2ccccc12 c1(C(=O)NCCCOc2nnc(C)s2)ccc(C(F)C(F)(F)F)cc1 n1(CCCOC)nc(-c2cccc(OC(C)C)c2)nc1C1CC1CF N1(C(Cc2c(C)nc(O)nc2C)=O)CC(C)CN(C(C2CCOCC2)=O)CC1C c1(C(C(=O)NC2COC2)N(C)Cc2c(C)noc2C)ccc(S(N)(=O)=O)s1 C(CC(C(C)(C)C)NC(C1CCC1)=O)N(C(=O)C(c1ccc(O)cc1)(C)C)C C1(C(=O)NCc2nc(CNC(C(C)n3ccnn3)=O)sc2)CC(=O)NC(=O)C1 C1(NC(c2cccc(OC)c2O)=O)CC2CC(NC(C3(Cl)CC3)=O)CC2C1 O=C(NNc1ccnc(Cl)c1)Nc1cnn(C(F)(F)F)c1 C1(C(=O)OC)CN(C(c2onc(C)c2I)=O)CC2(CCC2)O1 N1(C(C(=O)NCSc2ccccc2)C2(CCCCC)CC2)CCC2CCCC2C1 C1(NC(C(CCOCC)NC(=O)CC2CCC(=O)CC2)=O)CCOCC1(C)C C(C(N=[N+]=[N-])C(=O)N1CCC(C(=O)NOCC2CCOC2)(CC)CC1)OCC C(CC(=O)NCC(O)CNC(=O)CCCOc1ccc(C)cc1)(C(F)(F)F)OC C(CN=c1ccnc(N2CCC(n3ccnc3)C2)[nH]1)OC1CCN(C(COC)=O)C1 CN1CCCC1(C)C(=O)NCC1CCN(C(c2ccnn2-c2ccncc2)=O)C1 C1(C(=O)NCC(CNC(=O)CCC2CCOC2)F)CCN(c2ccncn2)CC1 C(=O)(C1=CC2(CCOC2)C1)NCC(CCCC)NC(CCCC#C)=O C1(C(N(C)Cc2nnc(CC)o2)=O)CCCN1NC(=O)COCCC(C)C n1(CC(C)C)ccc(CNC(c2nnnn2C2CCCC2)C2CCSCC2)n1 CCC(C)(C)C(C)CC(=O)NCC1CC(C)(C)CN1C(=O)CCc1ccco1 C(CC(=O)NCC1(CCCF)CC1)N(C(=O)CO)CC C1(C(N(CCCN(C)C)CCNC(c2c(CC)cco2)=O)=O)CCCCS1(=O)=O CC(C)(C)C(C(=O)NCc1cc[nH]n1)NC(c1cn[nH]c1)=O C1(C(CNC(C)CCC2CCCO2)(C)C)CCN(C(=O)OC(C)(C)C)CC1 C1(NC(c2ccc(SC)o2)=O)CCCCC1C(=O)NCCCSC(F)F c1(OCCC)ccc(CCC(=O)NCC(C(C)C)NC(C2CN(C)C2)=O)cc1 c1(CNC(c2cnc(CS(C)(=O)=O)s2)=O)ccc(Cl)cc1Br C1(CNC(CC2C(C)CCO2)=O)CN(C(=O)COc2cccnc2)CCC1(F)F c1(C(=O)NC(C(C)C)CNC(C2CC(N(C)C)C2)=O)c(F)c(F)c(F)c(F)c1F c1(C(N2CCC(NC(c3ccc(C)cc3Br)=O)C2)=O)cc(F)c(C)cc1N C1(CNC(C2N(C)C(=O)CC2)=O)CCN(C(=O)C=Cc2ccsc2)CCC1(F)F N1(C(CC=CC=C)=O)CCCC(N(C(=O)CCOCC(C)(C)C)C)CC1 Cc1nn(C)cc1CNC(C1CC(O)CN1C(=O)Cc1cnn(C)c1)=O Cn1nccc1C(O)CNC(C1CCC1NC(C1CCC1C#N)=O)=O C12(NC(c3c(C)sc(Cl)n3)=O)CCCN(C(=O)CCC3CCC(C)O3)CC1C2 C(CC(C(=O)N(C1(C)CC1)C)NC(C1CCS1(=O)=O)=O)OC c1(NC)ccc(C(=O)NC2CCC2NC(=O)C(c2c(C)cccc2C)O)cc1F C12(CNC(CC(C)(C)OC)=O)CN(C(=O)C=C3CCOCC3)CC1(C(F)(F)F)C2 Cc1cc[nH]c1C(=O)NCC1CCC(NC(=O)CSc2n[nH]c(O)n2)C1 N1(C(c2c(CC)nccc2)=O)CC2CCC2(NC(=O)C(C)Oc2cccnc2)C1 C1(C2CCC2)(CNC(=O)C(N2CCC(N3CC=CC3)C2)=O)CCNCC1 N1(C(C(C)OCC(F)(F)F)=O)CCOC(CNC(=O)Cc2ccn(C(F)F)n2)C1 c1(C(=O)NCC2(C#N)CCOCC2)ccc2c(n1)CN(C(C1C=CCC1)=O)CC2 C1(C(N2CCC(NC(C(C(CC)C)OC)=O)C2(C)C)=O)CCn2ccnc2C1 N1(C(c2ncn(C(C)(C)C)n2)=O)CC(C2CN(C(c3coc(C4CC4)n3)=O)C2)C1 c1(CCC(N2CC(CCNC(C3CC(C)(CC)C3)=O)C2)=O)nc2ncccn2n1 S(=O)(=O)(c1ccc2c(c1)C(=O)NC2=O)Nc1ncc(C)[nH]1 c1(C(N2CC3(CC(NC(c4cnc(C)c(N)c4)=O)C3)C2)=O)cccc2c1OCC2 C(c1cnc(O)nc1O)=CC(N1CCC(NC(CC2N(C)C(=O)CC2)=O)C1)=O C(C(C)(C(C)C)NC(c1cnn(C)n1)=O)NC(C(Cc1ccccc1)OC)=O c1(NC(c2nnnn2Cc2ccco2)CCOC)nc2ccccn2c1C C1(C(=O)NCC(CCNC(C=CC)=O)O)N(C(=O)OC(C)(C)C)CCC12CC2 C=C(C)CC(C(=O)NCC(c1ccco1)O)NC(c1sccc1C)=O C12(CNC(c3[nH]cc(C(C)=O)c3)=O)CCCN(C(c3cccc(C)c3F)=O)C1C2 C1(C(N2CC3(CN(C(C4C(C)(Br)C4)=O)C3)C2)=O)Cc2ccccc2N1 CCC(CNC(c1ccc(C(C)(C)O)cc1)c1nnnn1C1CCCC1)CCO C1(C(=O)NCC(CN(C)C)O)COCCN(C(c2ccc(C#N)cn2)=O)C1 C1(NC(=O)CCn2ccnn2)CCC2(CC1)CN(C(c1cnco1)=O)CCO2 c1(C(=O)NCCCCNC(CC2(OC)CC2)=O)cc([N+](=O)[O-])ccc1C N1(C(=O)Nc2c(O)ccc(N)c2)CCCN2CCCC12 c1(C(N2CC(NC(C)=O)C(C)C2)=O)ccc(Oc2ccncc2)c(Cl)c1 C1(CC)CN(C(C2CCC2(C)C)=O)CCC1NC(=O)CCCn1cncn1 c1(NC(C(c2ccccc2)NC(c2ccc(C)[nH]2)=O)C)cc(O)ncn1 CC1CN2CCN1C(C(=O)NCC#CCNC(C1CCOC(=O)N1)=O)C2 N1(C(c2cc(C)oc2C)=O)C2CCCC1CC(NC(c1ccnc(C)c1N)=O)C2 c1(C(=O)NCC2(C)CCC(NC(COCCOC)=O)C2)nc(C)ncc1Br N12CCCC(C)(CC1)C2.Cc1nc(C(C)C)oc1CCNC(=O)OC(C)(C)C c1(CC)ccc(NC(=O)CC2CN(c3ncnc(OC)c3OC)C2)cc1[N+](=O)[O-] c1(C(=O)NC(C(C)NC(c2cc(C(C)C)no2)=O)CO)ccc2oc(=N)[nH]c2c1 c1(C(=O)NC2CCCC(N(C)C(c3ccc(F)s3)=O)C2)csc2ncnc(O)c12 N1(C(c2cccc(OCC)c2O)=O)CCC2CC2(NC(=O)C(N)=O)CC1 C(C)(C)(CC(F)(F)CC)NC(C(NC)OC)=O C1(C(N2C(CN(C)C(c3ccc(N(C)C)cn3)=O)CCC2)=O)COC2CCCCC12 N1(C(c2n[nH]c(C)c2C)=O)CC(C)CCC1CNC(=O)Cc1c(C)ncnc1C N(C(=NCCc1nc2c(s1)CCCC2)N1CCCC2(CCOC2)C1)C(COC)C C(C(=O)Nc1ccc(-n2cnnn2)cc1)(C(C)C)OCC(C)C c1(C(N(C(C)(CN(C)C)NC(=O)OC(C)(C)C)C)=O)ccc(C(F)(F)F)c(Cl)c1 C1(NC(C2C(c3n(C)ncc3)C2)=O)Cc2nc3ccccc3n2C1 c1(CC)cncc(C(=O)NCCC(C(=O)NC2(CO)CCSC2)OC)c1 Cc1cccc(C)c1C1(C(=O)NC(C)C(CO)NC(=O)C(C)S(C)(=O)=O)CC1 c1(N2CCC(c3c(OC)cccn3)C2)nc(N2CCC(C#N)C2)c2sccc2n1 C1(c2cn(CCCC(=O)OCC)nn2)COCCC1NC(=O)C(C)COC c1(OC)cc(OC)cc(C(=O)NC(C)CN(C)C(c2c(C)ccnc2Cl)=O)c1 Cc1cccc2[nH]cc(C(=O)NC3(C)CN(C(=O)CCc4n[nH]c(=N)s4)C3)c12 c1(C(=O)NC(C(=O)NCCN2CCCCC2)C2CC2)ccc(O)cc1 c1(C(N2C(CNC(c3cc4n(n3)CC(F)C4)=O)CC2)=O)cc2nc[nH]c2cc1F C1(OC)CC2CCC(C1)N2C(c1coc(C(C)NC(c2ccc(C)o2)=O)n1)=O O(NC(=O)CC1(c2c(NC(=O)OC(C)(C)C)c[nH]c2)CC1)CC(C)C C(=O)(C#CC1CCCO1)N1C2CC(NC(COCCCC(C)C)=O)C(C2)C1 CCC(CC)(CCNC(=O)C(SC)SC)NC(=O)CCSc1ccccn1 N1(CC(=O)NCC(=C)CCNC(=O)C(C)(C)F)CCC(OCC(F)F)CC1 C(=O)(C(C)CC1CCCCC1)NC(C)CNC(C1(C(c2ccccc2)=O)CC1)=O c1(C(N2CCC(C)(NC(C(CC(C)(C)C)O)=O)C2)=O)cc2ccccc2nc1O c1(OC)cnc(C(=O)NC(C)(C)CCNC(C2(CO)CC2(F)F)=O)nc1 N1(CCCc2n(C)ncn2)CCC(c2ccccc2)(C(=O)O)CC1 CC1CN(C(C2CC3(C2)CC(F)C3)=O)CCC1NC(C1Cc2cscc2C1)=O C1(CC(N2C(CC(=O)NC)CC2)=O)CN(C(c2csc(Cl)c2)=O)CC12CC2 C(C1(O)CCc2cc(F)ccc21)NC(N1CC(C)(C)C(C(N)=O)CC1)=O Cc1cc(C(=O)NC(C)CNC(c2cncnc2)=O)c2c(O)n[nH]c2n1 c1(C(c2nnnn2CC)NCC2(CCSCC)CC2)cc(C)on1.C1CC1 CCC(C)(CC)C(=O)N1CCN(C2COCC2NC(=O)CCNC(=O)CO)CC1 N1(Cc2ccc(CCN(CC)CC)cc2)CCOCC12CCC2 C#CCC(C)C(=O)NC1CCCC1CNC(c1occc1-c1cnn(C)c1)=O C#CC1(O)CN(C(=O)CC2(NC(=O)Cc3cncs3)CCC2)C1 N1(C(C2=CCN(C(C3CC(C)OC3)=O)C2)=O)CCCC[Si](C)(C)C1 CCCCC(C(=O)NCC12CC1CN(C(=O)C(CO)N(C)C)C2)N(C)C Cn1ccc2cc(CNC(C(C)(C)C)c3nnnn3CC3CCCO3)ccc12 c1(CC)nc(C)ncc1C(=O)NC1CCCC(NC(=O)CC(C)(C)C#N)CC1 CN1CCN(C(C2CN(Cc3cc(Cl)cc(Cl)c3)CCC2O)=O)C(CO)C1 N1(C(C=CCN(C(C(C)C2CCOC2)=O)C)=O)CCOCC12CC2 C1(C(=O)NC(Cc2cc(C)[nH]n2)C)C2CCN(C(C3(CO)CC3)=O)CC12 c1(C(N2CCCC(O)(CN(C(CS(CC)=O)=O)C)C2)=O)cc(Br)c(C)nc1O C(=O)(C(COOC(C)(C)C)CC(C)C)NCC1(C(=O)OCC)CCOC1 C1(NC(c2c(CC)noc2)=O)CCN(C(=O)C(F)(F)c2cnn(C)c2)CC1O C1(CNC(C(C)(C)n2cccn2)=O)CN(C(=O)CCC2OCCO2)C2(CCC2)C1 CN1N=C(CC(=O)NC2CC3COCC(C2)N3C(=O)CSC(F)(F)F)CC1=O C12(C(N3C(CNC(=O)CSc4ccncc4)CC(OC)C3)=O)CCCC1C2(F)F c1(C(=O)NC2CC(CNC(C=CCOCCOC)=O)C2)c[nH]c2nc(F)ccc12 N1(C(=O)CC2CCCN(C(c3ccc(O)cn3)=O)C2)CCC2(CCCO2)CC1 N1(C(c2ncn(C)c2)=O)CC(NC(c2c(Br)ccnc2Cl)=O)C(F)(F)C1 C(CC(C)C)(C(=O)NC1CCN(C(=O)C(C)CC(N)=O)CC1C)NC(C)=O C(=O)(C1=CCCSC1)NC1CC(CNC(c2ccc(=N)[nH]c2)=O)C1 N1(C(C2C(OC)CC2)=O)C(C(N2CCC(O)C2)=O)C2CC(O)C1C2 CC1=NN(C)C(=O)C1CC(=O)NC(C)CCN(C)C(c1cc(Cl)cs1)=O N1(C(C(CSC)C)=O)CC(NC(=O)CCc2ccn(C)c2)C(n2ccnn2)C1 C1(CC)CN(C(=O)C(O)C2CC2)CCN1C(c1ccc(C(C)(F)F)cn1)=O c1(C(N2C(C(=O)OC)C(C)CC2)C(=O)NCCOC(C)=O)ccc(F)c(C)c1F C1(NC(c2c(C)n[nH]c2)=O)CC2(C1)CC2NC(=O)CC1COCCO1 N1(C(CCC=C)=O)CC(=O)N(C)CC1C(=O)Nc1csc(Br)n1.c12cn(nn1)C2 C1(C)(CNC(c2c(C)n(C)nn2)=O)COCCN(C(=O)C2=NOC(C)C2)C1 C1(C(N2CC3C(CNC(=O)CCc4ccoc4)(C3)C2)=O)CCC(F)(F)CC1 c1(C(=O)NC23CCC(CC2NC(C2CCCS2(=O)=O)=O)C3)ccc(CC)cc1F C(=O)(CC(CC(C)C)NC(=O)Cc1sccc1C)Nc1c(C)ccc(C)c1 C(CC(C)CC)(C(=O)N1CCn2cnnc2C1)NC(c1cncc(C#C)c1)=O c1(C(C(=O)NC(CNC(C(C=C)O)=O)C(C)C)(F)F)ccc(F)cn1 C(=O)(C1=NN(C)C(=O)CC1)NCC(C(=O)N(CC#CC)C(C)C)CC(C)C c1(C)nc2cc(C)cc(C)c2[nH]1.C1(C)C2(CC2)C12CC2.CN=C1NN2CCC(N1)C2 O=C1CCC(C(=O)N2CC3CC3(C(=O)Nc3nccc(C(F)F)c3F)C2)=NN1 CN1CCN(C(c2cccc(N3CCCC3)n2)=O)CC1CNC(C1CCCS1)=O c1(-c2cn(CC3(NC(Cn4c(C)nc(C)n4)=O)CC3)nn2)ncc(Cl)cc1Cl C1(NC(C2(C)CCC(F)(F)CC2)=O)Cc2ccccc2C1NC(C1CCC1)=O C(CCSC)(C(=O)N(CC(C)SC)C)NC(c1cn(CCC)nn1)=O c1(CCC)ccccc1C(=O)NCC1CCN(C(C2C3CCCC23)=O)C1 N1(C(C2N(C(c3cc(C)sc3N)=O)CCCCCC2)=O)CCC(C2=NOCC2)C1 C(N=c1[nH]c(Cl)ncc1C(=O)OC)C1CN(C(COCC)=O)CC1(C)C CC(C)C(CNC(=O)Cc1ccc2c(c1)CC2)C(=O)NCc1ccncc1 N1(CC)CC(NC(=NC)NCC2(C)CCCO2)CC1=O CCC(C)C(O)C(C)C(=O)N1CCC(NC(c2c[nH]nc2C2CC2)=O)CC1C C(C)(CCC(=O)N1CCCC1(C)CNC(=O)CCc1cnco1)OCC C1(C(N2CC(NC(C3C(C=C)C3)=O)CC2(C)C)=O)CCC(=C(F)F)CC1 CN1CCc2nc(O)c(C(=O)NCC(O)CCNC(C3CC3C(N)=O)=O)cc2C1 C(=O)(CC(C)C(F)(F)F)N1CCC(C)C1C(=O)NC12CCC(CC1)CC2 C1(C(N(C(C(N2CC(O)(C(C)C)C2)=O)C2CC2)C)=O)CC2(CC2)CN1C N1(C(CC(C)c2cnn(C)c2)=O)CCN(C(=O)Cc2cnoc2)C(CCO)C1 C1(NC(c2nc(CC)oc2)=O)CCCC(N=c2[nH]nc(-c3ccon3)s2)C1 c1(C(=O)NC2C(CC)CN(C(c3n[nH]c(C)n3)=O)CC2)cnc2c(c1)COC2 C(=O)(C(CCCC(=O)OC(C)(C)C)N(c1ccc(Cl)nc1)C)NC(C)C C#CCC(C(=O)N(C1CCN(C(C2(C3CC3)CC2)=O)CC1)CC(C)C)C1CC1 c1(C(=O)OC)cc2c(s1)CN(C(=O)C(C1CCCCCC1)C)CC2 C1(C(N2CC(CNC(Cc3c(C)n(C)cn3)=O)OCC2)=O)CC2CSCC(C1)C2 N1(C(c2[nH]nnc2C2CC2)=O)CCC(N(CCO)C(c2snc(O)c2Cl)=O)CC1 C1(NC(c2c(C)csc2Cl)=O)CN(C(=O)C(F)C(F)(F)F)CC1(C)C c1(C(=O)NCCOCCNC(C(CC#C)CC#C)=O)ccc2[nH]ccc2c1F C(=O)(C(F)(CNC(C1(O)CCC1)=O)C(C)C)NC1C(C(C)O)CCC1 C1(CNC(Cc2cccc(OCCC)c2)=O)CN(C(C2CSC2)=O)CCC1C C=CC(CCC)CC(=O)NC1(C)CCCC1NC(c1cc(Cl)cs1)=O CC1N(C(=O)CCC2CCCN2C(C2CC3CCCC3C2)=O)CCC1(C)C C1(CCCNC(C(CC)N(CC)CC)=O)CCCN(C(c2ccc(C)o2)=O)C1 C(=O)(CC(C)(O)c1ccccc1)NCCOC1CN(C(C(CC)OC)=O)C1.C(C)(=O)N CON(C)C1CCN(C(C2CCS(=O)(=O)C2C)=O)CC1 Cc1nc(C(=O)N(C2CCC(NC(=O)C(C)(C)n3ccnn3)C2)C)c(C)o1 Cc1cn2c(n1)CCC(n1cc(CNC(C3CNC(=O)CC3C)=O)nn1)C2 C1(C(=O)NC(CN(C(C(C)=C(C)C)=O)C)C)(CF)CC1(F)F C1(NC(c2cc(Cl)ccn2)=O)COC2(CNC(C3(C(F)(F)F)CCC3)=O)CC1C2 c1(NC(C)=O)ccc(C(N2CC(Nc3nccc(C(F)F)n3)C(O)C2)=O)c(Cl)c1 Cn1ccc2cnc(NC(c3ncc(-c4ccc5cnn(C)c5c4)cn3)=O)nc12 CCC1=NOC(C(=O)NC(CO)C(=O)NCCc2ccon2)C1 c1(C(=O)NCC2N(C(C3(C)CC4CC4C3)=O)CCCC2)cnc2[nH]nnc2c1 c1(CC)cc(C(=O)N(CC(C)(C)CNC(=O)CC2(C)CC(F)(F)C2)C)n(C)n1 S(=O)(=O)(c1cccc(=NCC(C)(C)CC2CC2)[nH]1)NC1(C=C)CC1 N1(C(Cn2c(C)ncc2)=O)CCC2(CCCN(C(=O)CC3CCCOCC3)C2)C1 c1(OC)ccc(CN2CCCC(C(=O)NC3CCC(F)(F)C3)CC2)c(Br)c1 c1(CN2CCC(CC(=O)CCn3c(C)ncc3)C2)nc(-c2nccs2)nn1C C1(C(N(CCCN(C)C(C2(c3ccccc3)CC2)=O)C)=O)CCC12CCOCC2 c1(C(N(C2CCN(C(C3CCOC3=O)=O)C2)CC)=O)cc2n(n1)CC1(CC1)C2 C=CCCC(C(=O)N1CC(N(C)C)C(C)(C)C1)NC(C1CC2(CSC2)C1)=O N1(C(c2c(=N)[nH][nH]c2)=O)CCC(F)CC1C(=O)NCC1CC2CCCC2C1 C1(NC(COC)=O)CN(C(c2cccc(C#N)c2)=O)Cc2ccnn2C1 C1(C(=O)OC)(CC)CCCN1C(C)=O.C12CCCN1NC2=O C1(CNC(CCCN(CCCC)CCCC)=O)CC(NC(=O)C(C)O)C(O)C1 CCCCCCOC(C)C(=O)NCC1CCCN1C(=O)Cc1cnn(C(C)C)c1 C1(CCC)(NC(c2cc(CN(C)C)on2)=O)CCN(C(=O)CC(C)C)CC1 C1(CNC(c2cc(C)oc2)=O)CC(F)(F)CN1C(c1coc(C)n1)=O N1(C(CC2(OC)CC2)=O)CC(F)(F)CC1CNC(c1cnc(-c2cccs2)s1)=O C1(OC)CC(N(C)C(c2ccccc2F)c2nn[nH]n2)C12CCC2 N1(C(C(C2CN(C(=O)CCCn3ccnn3)C2)OC)=O)CC2CCC(C1)C2C#N c1(C(N2CCN(C(CS(C)(=O)=O)=O)C3C2C3)=O)cc(Br)cc2cn[nH]c12 C1(C(C)C)(C(=O)NCCCOCCO)CCN(C(=O)Cc2ccccn2)C1 N1(C(C2C(C(C)C)(CC)C2)=O)CCC(NC(C2(CO)CCCCO2)=O)C1C1CC1 C1(CCC(=O)NCC=C(Cl)Cl)CCN(C(=O)C(C2(O)CCCC2)F)C1 CC(C)C(O)C(F)(F)C(=O)N1CCC(=CCNC(C2CCC(=O)N(C)C2)=O)CC1 N1(C(C(n2ccc(C)n2)C)=O)CC(NC(c2cc(C)sn2)=O)C(n2ccnn2)C1 C1(OC)CC(N=c2[nH]c(=NC(C)c3cccc(Cl)n3)[nH]c3ncn(C)c23)C1 C1(CCO)(CNC(c2n(CC=C)nnn2)c2csc(Br)n2)CCCCC1 c1(C(C(=O)NCCN(C(c2ccccc2OC)=O)CC)O)ccc(Cl)cc1 C1(C#N)(N)CC2CC2C1.C1(OC2CN(C(C)=O)C2)CCN(C(C2CCCSS2)=O)CC1 C12(C(=O)NCCCCCN(C(CC(=O)NCC#C)=O)C)CCC(CC)(C1)OC2 c1(C(N(C2CCN(C(Cc3c(OC)nccc3)=O)C2)C)=O)cccc(F)c1Cl C(C)(CO)(C(C)(C)O)NC(C=CC(C)NC(c1nc(C)oc1C)=O)=O c1(C(=O)NCCCCCN(C)C(c2cnc(C(C)(C)C)o2)=O)cc(N)cc(O)c1 c1(CC(N2CC3CC(CNC(COCCOC)=O)C3C2)=O)c(C)nc(O)nc1C c1(C(=O)OC)ccc(S(=O)(=O)NC2CCCCN(Cc3nccs3)C2)n1C C(=O)(C1=NOC(C)C1)N(CC(C)NC(=O)CS(C)(=O)=O)CC c1(OC)ccc(CCC(=O)NCC(C)NC(c2cscc2SC)=O)cc1 c1(CC)nonc1C(=O)N(CC(C)(C)CNC(c1cnc(C2CC2)o1)=O)CC N12CC(CC1C(C)C)C1(CC1)NC2=O.c1(CC)cc(CC(=O)OC(C)(C)C)on1 Cc1cc2cc(NC(c3ccc(OC4COC4)cc3)=O)ccc2[nH]1 C(=O)(C1CCCc2ncnn21)N1CC2(CN(C(c3ccn4nccc4c3)=O)C2)C1 CC(C)CCC(=O)NCCC1CCN(C(C2(CC(F)F)CCOCC2)=O)C1 CC1C2CCC(C2)C1C(=O)NC1CC2(C1)CC2NC(=O)CC1CCC(C)(C)C1 C(CCCC(C)(C)C(=O)NNC(=O)CCCC1CCC1)NC(c1c(C)occ1)=O CC1(C)C(SCCOC(C2CCN(S(=O)(=O)c3ccccc3)CC2)=O)CCS1(=O)=O c1(C(N2CCC(C(C)NC(c3nc(C)oc3)=O)CC2)=O)cc2c(cc1Br)OCO2 C(=O)(C1=C(Cl)CCCC1)N(CCC(=O)NCC1CC(O)C1(C)C)C C(=O)(C1=CC2C=CC1C2)NCC1CCN(C(CCc2c(C)cccn2)=O)C1(C)C c1(C(C(N2CC(NC(CCCC(=C)C)=O)C3C2C3)=O)=O)ccc(F)c(F)c1F C1(NC(C2(OC)CC2)=O)CCC(C)(C)CC1CNC(=O)CN1CSCCSC1 N1(C(c2cncc(C)n2)=O)CCN(C(c2ccc(C(C)(C)C)nc2)=O)C2CC12 C1(CNC(=O)NC(COCCCC)C)CCC(C(=O)OC(C)(C)C)CC1 CN1CCOC(C)C1.C1(C=O)C2CC1N(C(C13CC(CN1C1CC1)C3)=O)C2 CN1CCC(C(=O)NC2(C)CCN(C(C3(C)CC3(F)F)=O)CC2)S1(=O)=O N1(C(C=C2CCC(C)C2)=O)CCC2CN(C(=O)C=CSc3nc[nH]n3)C2C1 CCC(C)(C)C(C)CC(=O)N1CCCCC(NC(=O)CNC(=O)NC(C)C)C1 C12(NC(C=CC)=O)CC3CC(C1)CC(NC(=O)C(C)CSc1ccccc1)(C3)C2 c1(C(=O)NCCCc2cn(C3(C(N)=O)CC3)nn2)ccc(C2CC2(F)F)cc1 C12(C(=O)NCC3CCC(NC(c4c(C)cnn4C)=O)C3)CCC(N=[N+]=[N-])(CC1)C2 C(CNC(=O)Cc1ccc(OC)cc1C)(C(C)C(C)C)NC(CS(=O)(=O)NC)=O C=CCC(CNC(=O)C(C)(C)C(O)C(C)C)C(=O)NOCC(N)=O Cc1ccc(F)cc1C(=O)NC1(C)CC(NC(=O)CN2CCCCS2(=O)=O)C1 c1(CCC(=O)NCC#CCNC(CC(C)SC)=O)ccc(O)c(Cl)c1 N1(C(c2cnc(C)n2C)=O)CC(NC(=O)CSCCN(C)C)C(F)(F)C1 CC1OC(=O)NC1C(=O)NCC12CC1CN(C(=O)CN(C)C(=O)C1CC1)C2 CC1CC(C(=O)NCC2CCCC2NC(c2ccc(C(F)F)cn2)=O)CCC1=O C#Cc1ccc(C(=O)NC(C)(C)CNC(=O)C(c2ccccc2Cl)C)nc1 C(=O)(CCC(=O)C(C)(C)C)N1CCCC(C(=O)Nc2c(C)ccc(OC)c2)C1 c1(C(=O)NC2CCC(CNC(=O)C=Cc3cc[nH]c3)C2)cnnc(O)c1 N1(C(c2csc(C(C)(C)C)c2)C(=O)NCC)CCC(C2(C)OCCO2)CC1 C1(NC(c2cn(CC)nc2C)=O)CCCC12CN(C(c1sccc1COC)=O)C2 CC1CCCN(C(C2C3CCC2CC3)=O)C1CNC(=O)CN(C1CCC1)C C1(CNC(c2ccc(NC(C(C)C)=O)s2)=O)CC2CCC1N2C(=O)CCCF N1(C(CC2CCC(C)(C)CO2)=O)CC2(CC(NC(C3(O)CCOCC3)=O)CO2)C1 c1(C(N(CCN(C(=O)CCC2CCC(=O)N2)C)C)=O)nc2ccccc2s1 C1(CNC(CNC(CCCCC)=O)=O)CC2(CCC2)CN1C(=O)COC N1(C(C2(C)CC2Br)=O)CCC2(COC(CNC(c3c(F)cccc3F)=O)C2)C1 C1(CN(c2cc(N3CC(C)OC(C)C3)ncn2)C2CC2)CC(F)(F)C12CCC2 c1(NC(C(C)OC(c2c(C)n[nH]c2)=O)=O)ncccc1C(F)(F)F c1(-c2nc(C(CCC)C)nn2CC(C)C2CC2)ccc(F)c2occc12 C1(NC(=O)Cc2ccncc2)CCC2(CC1)CCN(C(=O)CC1CC1)CC2 c1(CCC(=O)Nc2cccc(NC(=O)C(F)C3CC3)c2)ccc(SC2CC2)cc1 c1(C(N2CCC(NC(C3CC4(C3)CC4(F)F)=O)C(F)C2)=O)cc[nH]c2nccc1-2 C1(NC(C(C(C)(C)O)F)=O)(CNC(c2ccc(F)cc2N)=O)CC2CCC1CC2 C(=O)(C1=CC(O)CCC1)N1CCC(C(C)(C)NC(CNC(=O)OC(C)(C)C)=O)C1 C(=O)(C(CC=CC)NC(c1c[nH]c(=NC)o1)=O)NCCOCCC#C CCC(O)C(C)C(=O)NC1CC2(C1)CC(NC(=O)C(O)COC)C2 C1(C(=O)NCc2ccc(CC)cc2)COCCN(C(c2cnc(C)s2)=O)C1 c1(CC)nc(C(C)NC(=O)CCOCCCNC(c2ccccn2)=O)n[nH]1 C1(CC)CCCCC1C(=O)NC(C)(CNC(=O)CCOCC(C)C)CC CCCC(C(=O)N(CC(CC)NC(=O)C(C)c1cccs1)CC)NC(N)=O N1(C(=O)C2=CCCC2)CCC2OCCN(C(C3CC4CCC(C3)S4)=O)C2C1 Cc1nc(C)n(CC(=O)NC(c2nc(C(=O)NCC3CCC(C)C3)co2)C)n1 C1(CC)CC(NC(=O)C=CC(C)NC(=O)C(C2CCC2)SCC)C1 C(=O)(C#CC1CCCCC1)N1CCC(=CCNC(=O)Cc2csc(Cl)c2)CC1 C(CCCCO)(C(=O)N1CCCC(F)C1)NC(C(=O)NC(C)C)=O c1(OCC(=C)C)ccccc1C(=O)NC1CC(NC(c2n[nH]cc2Cl)=O)C1 C(C1CN(C(c2snnc2C)=O)CC1C(N1CCCC1CC1CCC1)=O)=CC C1(NC(CCCCC#C)=O)CCCCCN(C(c2cnc(CCCC)s2)=O)C1 c1(C(=O)Nc2scc(C(=O)NCC3CCOC3)n2)ccc(I)c(Cl)c1 C1(C(N(C(C)CO)CC)=O)COC2(CCN(C(c3ccno3)=O)CC2)C1 C12(C(N3C(C(C)O)CC3)=O)CCC(CN(C(C3(C)CCCC3(F)F)=O)C1)C2 C(c1nnn(C)n1)=CC(=O)N(CCCCN(C(=O)CCCN1CCCC1)C)C Cc1cc(C)c(CNC(C2C=CCN(C(=O)C(=O)C3CCCC3)C2)=O)s1 C1(C(=O)NC2CCN(C(C)=O)C2)CC(F)(F)CN1C(=O)COC(C)C N1(C(C(CCCC)O)=O)CCC2CN(C(=O)C(O)CC)CC2CC1 N1(C(=O)NCC(C)OCC=C)CCC2(CCNC2=O)C1 C(=O)(C(C)(CC)CCCCCC)N1CCC(NC(C2(CC=C)CCCCC2)=O)C1 C1(C(=O)NC(CCCOC)(C)C)CC(C)CN(C(c2sccc2C)=O)C1 C1(NC(c2ccnc(Cl)c2Cl)c2n(CC)nnn2)CC2CC(OC)C2C1 c1(CCNC(C(C)C2CCCO2)=O)ccc(CNC(=O)Cn2ccnn2)cc1 C(C(C)C(C)C(=O)NCCC(C)N(C(=O)C(C)NC(=O)CC(C)(C)C)CC)OCC Nc1ccc(C(=O)NCC2CCN(C(=O)Cc3cccnc3F)C2)nc1 O(NC(=O)C(C)CNC(C1(F)CCOCC1)=O)CCC C12(C(=O)NCCC3(CNC(c4n(C)ccc4)=O)CC3)CCCCN1CCC2 C1(C(=O)NCC(C)(C)OCCNC(C2(CC)CC2)=O)CCCCN1C C1(c2nnnn2CCc2cccc(F)c2)(NC(C2COC2)C)CN(C)CC1C Cc1cc(C(N2CCCCC2C(C)NC(=O)CCSC(F)(F)F)=O)ccn1 c1(C(N2C(CNC(C(COC(C)=O)C)=O)CC(F)C2)=O)cc(C)c(C(F)F)cn1 C(C(NC(=O)NCCOCC1CC1)OC1CCC1)OC C1(CNC(CN(C(c2c(CC)ccs2)=O)C2CC2)=O)CC2CCC(C1)C2 C1(CC(N2CCC(CC(N)=O)C2)=O)C2CCCC2N1C(c1cccc(F)c1)=O c1(C(C(N2CC(C(C)NC(=O)CCC3CCCN3C)C2)=O)O)ccc(F)cc1 C1(CC)(CC)C(OC)CC1N(C(=O)CC1(OC)CCOCC1)C N1(C(C2(C#N)CC2)=O)CCC2(CCC2NC(c2ccc3ncccc3n2)=O)CC1 CCCCCCC(C(=O)N1CCC2C(C(=O)OC)CC12)NC(=O)CC1(COC)CC1 c1(CNC(C2CC(O)CN2Cc2ccncc2Cl)=O)cnc2cc[nH]c2c1 N1(C(c2ccc(C(=O)OC)o2)=O)CCC(C(=O)NCC2(SC)CCOCC2)CC1 C(=O)(C(CNC(=O)Cc1ccccc1C)C(C)C)NCC(C#C)C(C)C N1(C(c2ccncc2F)C(=O)Nc2c(C)cccc2)CC2CC2C2CC12 c1(C(=O)NCC2(F)CC(NC(c3c(C)ccs3)=O)C2)cnc2nccn2c1 CCCC(C)(O)C(=O)N1CCC(CN(C(=O)CCOCC)C)C1 C1(C(=O)NC2(CC(=O)NC3CC(C4CC4)C3)CCC2)CCCC1C1CC1 CCCCN=C(NCC(C1(O)CCCOC1)(C)C)NCC1CC1c1ccccc1 C1(C(C(=O)NCCC(C)NC(c2cc(C)nn2C2CC2)=O)C)CCC(C)(C)CC1 C1(C)(C(=O)NCC2(COC)CN(C(C3CC(CC)OCC3)=O)C2)CCC(=O)NC1 C1(NC(C2(C)C=CCC2)=O)CN(C(C2(F)CCCC2)=O)CC2(CCOCC2)C1 CCCC(C)(CCC)C(=O)NC1CN(C(C2CC2CC(C)C)=O)CC1CC1CC1 C1(C(=O)NC(COCC)C(C)C)CCN(C(c2ncsc2C)=O)C12CCC2 Cc1cc(NC(C2CCCS2(=O)=O)=O)ccc1NC(=O)CCN1CCC(F)C1 N1(C(C(CCCC)C)=O)CC2CCCC(C1)N2C(C1CCn2cnnc2C1)=O C1(CCC=C)(C(=O)NC(C2CCOC2)CC)CN(C(=O)C(C)=C(C)CC)C1 C1(NC(C2COCCO2)=O)CN(C(=O)CC2COCCO2)CC12CCCC2 c1(N2CCC3(CC2)CCN3)cc(C)c(C(N)=O)cn1.C(C)(C)(C)OC(=O)NSCC Cc1cccc(OCC(=O)NCCCC(C)NC(c2ccn(C(F)F)n2)=O)c1C C(=O)(C1CCCc2scnc21)NC1(C)CN(C(c2cc(C)c(N)cc2Cl)=O)C1 Cc1nn(C)c(Cl)c1C(=O)NC1CC(O)CN(C(C2CC3CCCCC23)=O)C1 c1(CC(N2CCCC(Cn3cc(C4(C)CCCC4)nn3)C2)=O)cc(F)cc(F)c1 C1(OC)CN(C(=O)CCC(C)C)CC1NC(c1ccc(C(F)(F)F)cn1)=O C(CC(C)C)(C(=O)NCC1(NC(C2CCCC(C)(C)C2)=O)CCOCC1)OC N1(C(c2occ(C(N)=O)c2)=O)CCCC(NC(C23CSCC2C3(F)F)=O)CC1 C1(NC(c2cc(OC)nn2C)=O)C(C)(C)CN(C(=O)CP(C)(C)=O)CC1(C)C S(=O)(=O)(CC(=O)NC1CCCN(C(=O)Cc2ccc(OC)nc2)C1)NC C(CC(=O)N1CCC(NC(c2cc(F)cc(F)c2)=O)C1(C)C)(C(C)C)OCC N1(CC#CCOCC)C(=O)c2ccccc2C1=O.C1(C(F)(F)F)CN1 N1(C(COCCCC)=O)CCCC(C)C1CNC(c1cnc(O)n1C)=O CC(C)S(=O)(=O)C(C)C(=O)NC1CCC1NC(c1cc(S(N)(=O)=O)ccn1)=O C(=O)(CCCCCC(C)O)NC(CC(C)C)CNC(c1ccc(C(N)=O)o1)=O C1(C(N(CCCCC)C)=O)C2CC1N(C(=O)C(CC)OCC)C2 N1(C(C(c2ccoc2)NC(c2ccc(C)[nH]2)=O)=O)CC(C)OC2(CCC2)C1 c1(CNC(C(CC)=CC)=O)cc(O)nc(CNC(=O)C(F)CC2CC2)n1 CC1CCCCC1CC(=O)NCCCN(C)Cc1csc(Br)c1 C(=O)(C(F)(F)C(F)F)N1CC(CN(C)C(C2(N3CCOCC3)CCCCC2)=O)C1 S(=O)(=O)(c1c(C)cccc1Cl)N(CC=C)C1CC1 C1(CNC(CNS(CCCC)(=O)=O)=O)CN(C)CCN1C(c1cccnc1Cl)=O c1(C(N2C3CC(CC(NC(C4CCC4)=O)C3)C2)=O)cc2c(F)cccc2s1 c1(C(N(CC(C)NC(CNC(C(CC)C)=O)=O)C)=O)cccc(OC(C)C)c1F c1(C(=O)NCC2(CF)CC2)csnc1-c1ccccc1 Cc1cc(C(N2CCCC2CN(C(=O)CSc2cnn(C)c2)C)=O)on1 C(=O)(C(C(C)C)N1CCCC1=O)NCC(CNC(C(C)C)=O)F C#CCCCCC(=O)NCC(C)(C1CCC1)NC(=O)Cc1ccc(F)c(C)c1 C1(CCOC)(NC(=O)CCCF)CCN(C(c2cnn(CC3CC3)c2)=O)C1 c1(C(=O)NC2(C)CN(C(c3c(C)n[nH]c3)=O)C2)ccc2c(n1)CCC(C)C2 N1(C(C(c2ccc(OC)cc2)CC)=O)CCCN(CC(=O)NC2CC2)CC1 Cc1cocc1C(=O)NC1CC(CCNC(=O)CSCc2cccs2)C1 Cc1cccc(CC(=O)NCC(C2CC2)NC(c2conc2C)=O)c1Br Cc1cnc(C(=O)NCc2ccc(CNC(C3CC(N(C)C)C3)=O)cc2)cc1C c1(N(C)Cc2cc(Cl)cc(Cl)c2)nc(N2Cc3ncsc3C2)nc2c1CSC2 C#CCCCCCC(=O)N(C1CN(C(C2CC2c2cc(F)cc(C#N)c2)=O)C1)C Cc1noc(C)c1C(C)C(=O)NC1CN(C(c2conc2C2CCC2)=O)CC1C Nc1cncnc1C(=O)NCC1CCCC1C(=O)NC1CC(CO)C2CC12 Cc1ccnc(NC(C2CC(F)CN(C(=O)Cc3cc(Br)cc(Br)c3)C2)=O)c1Br CCC(C(=O)N(C)CC1(CNC(c2c[nH]nc2C)=O)CC1)C(F)(F)F Cc1cc(F)cc(Cl)c1NCC1CN(C(=O)OC(C)(C)C)C(C)(C)C1 C(=O)(C(C)C(=O)OC)NC1CCC(SCc2onc(CCC)n2)CC1 C1(CC)CCCN(CC(=O)NC2C3CN(C(=O)C(C)CCOC)CC23)C1 Cc1ccnc(C)c1CNC(=O)CC1CCCCN1C(=O)CCP(C)(C)=O C(=O)(C(C)(C)C)NCC1CN(C(CN(C)C(c2ccns2)=O)=O)C1 C12(C(=O)NCC3(O)CN(C(C4CC5(C(C(=O)OC)C5)C4)=O)C3)CCCN(CC1)C2 N1(C(C(CC=C)(C)O)=O)CCC2(CC1)CC(NC(=O)C(C)C(O)CCCC)C2 c1(OC)cccc(C(C)C(=O)N(CCCNC(=O)C(C)N2CC(C)C2)C)c1 c1(C(N(CCCNC(C2Cc3nncn3C2)=O)CC)=O)cc2sccc2n1C C(=O)(C(F)(F)Cc1ccccc1)NCC1N(C(C(c2nc(C)sc2)=O)=O)CC1 c1(OC)ccc(CC(=O)NCC2C=CCN2C(=O)CN2CC(C)C2)c(Cl)c1 C1(CC(=O)NCCNC(c2cncc(Br)c2)=O)Cc2ccccc2NC1=O c1(CC(=O)NC23CCCC2N(C(=O)C(F)C2CC2)CC3)cccc2c1OCCO2 c1(C2CCCN(C(c3cn(C4CCNC4)nn3)=O)C2)cc(F)ccc1F C1(NC(c2ccc(Cl)o2)=O)CN(C(C2CCC2)=O)CCC12CCC2 N1(C2CCCN(C(C3C(=C)C3)=O)C2)CCN(C(=O)COCC(=O)OC)CC1=O C1(NC(CSCC=C)=O)CCN(C(C2CC23CC(C)(C)C3)=O)CC1O c1(C(=O)NCCCCCN(C(=O)C=CC2CCCO2)C)ccc([N+](=O)[O-])cc1O c1(CC)cc(C(=O)NC(C2CN(C(=O)CCc3cnn[nH]3)CCO2)C)cc(O)n1 c1(C(=O)NCCN(CC)CC)c(Cl)cc(OC)cc1Cl c1(N(c2ccnc(C)n2)CCO)cccc(NC(=O)C(C2CCCCCC2)O)c1C C1(c2cn(CC3N(C(c4ncn(CCOC)n4)=O)CCC3)nn2)COCCOC1 C1(C(=O)NC2CC(C)(NC(=O)CCCc3cnccn3)C2)(OC)CCSC1 C#CC1(C(=O)NC2CC(F)(CNC(c3nccnc3C)=O)C2)CCOCC1 C12(C(N(CC(C)(C)C)C)=O)CC(CCO1)N(C(c1sccc1Cl)=O)C2 CC(CNC(=O)C=Cc1cnccn1)CC(=O)N1CCC1 C1(C(=O)NCC(C)(Cn2cccn2)NC(C2(CO)CCCC2)=O)CC12CC(O)C2 N1(C(C(CCN(C)C)O)=O)CC(C(N2CC3(CCC(=O)N3)C2)=O)CC12CCC2 C(N=c1[nH]c(=NCC(C)OC(F)F)[nH]c2c1COC2)c1c2ccn(CC)c2ccc1 C(=O)(C(C)N(OC)C(=O)C1CCC(NC(=O)C2Cc3ccccc32)CC1)OC C1(C(=O)OCC)(C(=O)N(CCNC(C2CC(Cl)(Cl)C2)=O)CC2CC2)CC12CC2 c1(C(=O)NCC(CC=C)NC(c2c(Cl)n[nH]c2CC)=O)cnc(C(F)(F)F)cn1 N1(C(c2cccc(C#C)c2Cl)=O)CCC2CN(C(C3CCCS3(=O)=O)=O)CCC12 c1(OC)ccc(C(C)NC(C2CC(F)(F)C2(C)C)=O)c(F)c1 N1(C(C2(OC)CCC2)=O)CCC12CN(C(c1cccc(C)c1N)=O)C2 c1(C(=O)NC2CN(C(c3cc(Br)ncc3F)=O)CC2O)cc(F)c(Br)cc1F N1(C(C(C)SCC)=O)CCC(C)(NC(=O)Cc2cnn(Cc3ccccc3)c2)C1 CCCCC(C(=O)NCC1CCCC(=O)N1)NC(=O)Cc1cc(C)nn1C C12(C(N3CCC(C(=O)NC(COC)COC)CC3)=O)CCC(CC1)C(C)(C)O2 C1(C(=O)NCCCC#C)CCCN(C(C2CCN(C)C(=O)C2)=O)C1C C(=O)(C1CCCc2nncn21)N1CCCC(N(C(=O)C2=COCCO2)CC)C1.C1CC1 CC1(CNC(=O)CC2CCNC2=O)CCCN(C(C2CC(C#N)C2)=O)C1 c1(CNC(c2cnc(CC3CC3)n2C)c2n(CCC)nnn2)ccccc1SC C(=O)(C(CC)C(=O)NC1(C)CCN(C(c2ccn(C(F)(F)F)n2)=O)C1)OCC CCCCC(CC(=O)N1CC(C(=O)N(C)C)C1)NC(=O)CCc1cnccn1 CCC(CC(=O)NC(C1CCCCC1)CNC(c1ccc(COC)o1)=O)SC N1(c2nnc(C(N)=O)s2)CCC(C2CC2)C1CNC(C1(C)CCC(=O)N1)=O C(=O)(C1=CCC2(COC2)OC1)N1CC(O)CCC(NC(=O)C=CC2CCCC2)C1 CC1CCC(CNC(=O)C(N2CCCCCCC2)c2ccccc2)C(C)C1 N1(C(c2cn(CC=C)nc2)=O)CC(CNC(c2cc(C(F)(F)F)ns2)=O)C(C)C1 CC(C(=O)OC(C)(C)C)C(=O)NCCC(C)N(C(=O)CCCn1ccnn1)C CC(C(=O)NCC(C1CCCC1)NC(c1ccc(-n2cnnn2)cn1)=O)C(F)F C1(CNC(C(C(C)C)n2ccc(C)c2)=O)CN(C(c2cc(F)c[nH]2)=O)CC12CC2 c1(C(=O)NC(CC)(C)CNC(c2cc(COC)on2)=O)ccc2c(c1)CCCC2 C1(C(N(CCCCCNC(c2ccc(C#C)cn2)=O)C)=O)CCC2(CCC2)OC1 c1(SC)cc(C)ccc1C(=O)NCC1(O)CCN(C(C2C3(CC3)C23CC3)=O)CC1 C1(C(=O)NCC(C2CC(C)(C)C2)O)CCCN(C(C2CC23CCC3)=O)C1 N1(C(C(C)Oc2ccc(Cl)cc2)=O)CCC2(CC2NC(C2CCCO2)=O)C1 Cc1c(NC(=O)CC2CC(C)N(C(=O)COCC(F)(F)F)C2)cccc1F C1(F)(NC(C(C)OCCOCC)=O)CCN(C(=O)Cc2cnn(C)c2C(F)F)C1 Cc1cc(C(=O)NCC2CC2NC(=O)CN2CCS(=O)CC2)nc(N(C)C)n1 c1(NC(c2n(C)ncc2CNC(=O)CN2CC(C)(C)C2)=O)cnc2[nH]cnc2c1 CCCCC(C)CCC(=O)N(C(C(N1CCC2(CCC(OC)C2)C1)=O)C1CC1)C c1(NC(C2CC3CC3N2C(c2ccccc2C(F)F)=O)=O)ccc(CO)cc1O c1(C(N2CCN(CC)CC2)C(=O)NC)cccc(OC)c1Br.N12CCCC(C1)C2 c1(C(=O)NC(C)CNC(=O)Cc2cnn(C)c2)ccc2nc(O)[nH]c2n1 C1(NC(c2cc(C(C)(C)C)no2)=O)CN(C(=O)CC2NC(=O)NC2=O)CCC1(F)F CC(C)(C)CC(=O)NCC(c1cccc(Cl)c1)NC(=O)CN1CSCCSC1 N1(C(COCC(=O)NC)=O)CCC(C)C(NC(c2cc(Cl)cs2)=O)C1C N1(CC)CC(C(=O)NCC2CCCN2C(C2CC=C(C)CC2)=O)CC1=O c1(NC(=O)NC(C)CCNC(=O)Cc2csc(C3CC3)n2)cc(O)c(F)cc1N N1(C(Cc2cccc(OC)c2)=O)CC(NC(=O)C(F)C2CC2)CC12CCC2 C1(C(N2C(C)CC(NC(C(C(C)C)N(C)C)=O)C2)=O)CC2(CCCCC2)C1 CCCC(F)C(=O)N1CCSCC1CCNC(c1ncsc1CC)=O Fc1ccc2ncnc(N3CCCC(n4ccnn4)CC3)c2c1 CCC(C#N)C(=O)N(C1CN(C(c2snc(Cl)c2Cl)=O)C1)C c1(C(=O)NCc2ncc(OC)nc2)c(C)ccc(C)c1O N1(c2ccc(C#N)nc2)CCC(C2CC2)(CNC(c2ccc3sncc3c2)=O)C1 N1(C(C(C)SCC(C)C)=O)CCC(c2ccccc2)(NC(=O)C(C)O)CC1 CCC(C)C(CN(C)C)NC(=O)C(C)N(C(C1(C)CC(=O)C1)=O)C1CC1 Cc1cc(NC(c2ccc(C3(Cn4cccc4)CC3)cc2)=O)ncc1Cl C1(CCC)CCCN(C(C2(C)CCN(C(c3nn(C)cc3Cl)=O)C2)=O)C1 N1(C(COCCOCCOC)=O)CC2CCC1C2NC(c1nn(C)cc1N)=O c1(OC(C(=O)NCCC(c2cccc(OC)c2)C)C)ccc(C#N)cc1 N1(C(C2CCC=CO2)C(=O)NC)CCc2oc(-c3ccccc3)cc2C1 c1(OC)c(N2CCC(CNC(=O)Cc3coc(C(F)F)n3)C(C)C2)ncnc1Cl c1(C(=O)NCCC(C)N(C(C(COC)OC)=O)C)cc(F)c(Br)c(F)c1N c1(C(=O)NC2(C)CCN(C(C34CC(F)(C3)C4)=O)C2)cccc(Br)c1Cl c1(NC(CNC(C(C2CCCCC2)OC)=O)C)cnc(C#N)c(C#N)n1 C1(C(C)C)(C(N2CC(O)(CCNC(c3ccns3)=O)C2)=O)CNC(=O)C1 C1(C(N2C3(C#C)CC(C2)C3)=O)CN(C(c2cc(C)c(O)nn2)=O)CCC1(C)C C1(NC(C2(CCN(C)C)CCCC2)=O)CCCC(CNC(=O)Cn2ncnn2)C1 CCCC(C)C(=O)NC1CCN(C(c2ccccc2COC)=O)C1C c1(C(=O)NC2CCC(NC(=O)CCc3cncs3)CC2)cc2ccncc2o1 N(C1c2ccccc2OC1C)C(=O)NCCC(CC)CO c1(C(C)(C)C)ccnc2c(C(=O)Nc3cc(Cl)cc(F)c3O)cnn12 C1(C(CC)O)COCCN1C(=O)C(O)C1CC1 N1(C(C2(CC)CN(C(CCSCC)=O)C2)=O)CCCC(C)(C)C1C C1(O)(C(N2CCCC(CNC(=O)C(F)(F)C3CCCCC3)C2)=O)CCCCC1 C1(C(=O)NCC(C)CC(C)O)(CNC(c2c(CC)nco2)=O)CCCCC1 CON(CCC(=O)N(c1cncc(F)c1)CC)C(=O)CS.c1(CN2CCCC2)cccs1 C12(C(=O)NC(C(=O)OCC)CC)CC1CN(C(C1CC13CCCC3)=O)C2 C1(NC(Cn2ncc(CC)c2)=O)CN(C(=O)CCC(=O)c2ccccn2)CC1O c1(C(=O)NC(CNC(=O)COc2cccnc2)CO)cn(C(F)F)nc1C(F)F Cc1c(C)c(C)c(C(N2CCCC(C)(CNC(=O)C(N)=O)C2)=O)c(C)c1C C(C)(CCC(=O)NCC(CC(C)C)NC(=O)C(O)Cc1ccccc1)OCC C1(CNC(c2ccccc2)=O)CCCN1C(c1csc(C(F)F)n1)=O C(=O)(C1=NN(CC)C(=O)CC1)NC1C(NC(C(CC)=CC)=O)CCOC1 CC(CC(=O)N1C2CCC1CN(C(c1cnn(C)c1Cl)=O)C2)CC(F)(F)F C1(C(N(CCCNC(CCCC(=C)C)=O)CCO)=O)CCC2CCCCN12 C1(NC(c2c(C(C)NC(=O)CN3CCNC(=O)C3)noc2)=O)CCC12CCCC2 C#CCC(O)C(=O)N(CC(C)C(=O)NC(CC)CCO)C c1(C(=O)NCC(C2CCOC2)NC(C=C(CCC)C)=O)c[nH]nc1C(C)C c1(SCCC(=O)N(C2CCC(NC(=O)Cc3nccn3C)C2)C)ccccn1 C(CC(=O)NC1CC(F)CN(C(=O)C=C2CCCCC2)C1)(C(F)(F)F)OC C1(CC=C)(NC(=O)CC(C)(C)O)CCN(C(=O)COC2CCOC2)CC1 CC(C)CC(CC(=O)NC1CCCC1O)NC(=O)CC(O)C(C)C CC(O)C(C)C(=O)NCCCC(C)(C)NC(=O)CCNC(c1ccccc1)=O N1(Cc2ccc(C#C)s2)CCC2(CC1)CC2C(=O)Nc1cccc(I)c1 C12(CNC(C3(COC)CCCCC3)=O)CCC(CC1)N2C(=O)Cn1cc(C)cn1 c1(C(C)C(=O)NCC(=C2CN(C(=O)C(F)(F)C3CC3)C2)F)ccc(F)cc1F C1(CNC(c2ccc(OC)cc2)=O)CCN(C(=O)C=Cc2cc[nH]c2)CC1(F)F C(=O)(C(F)(F)C(C(C)C)NC(C1CCCCC1CC(F)(F)F)=O)OC C=CC(CC)CC(=O)N1CC(CNC(=O)CC(=O)NCC(F)(F)F)C(C)C1 N1(C(c2c(C)csc2)=O)CCC(C(=O)NCc2cnnn2C)C(C)(C)C1 N1(C(c2nc(CC)[nH]n2)C)CCC2CCC(C1)N2C(c1cc2n(n1)CCCC2)=O C1(C(N(CC(N2CCC(C#C)C2)=O)CCOC)=O)CCCCCN1C CC1(C(=O)NC2CC(NC(=O)CCCNC(=O)C3CC3)C2)COc2ccccc2O1 C1(C(=O)NC(c2n(C)cnn2)CO)CCN(C(C2CC(O)C(F)C2)=O)C1(C)C C(=O)(CC(C(F)(F)F)NC(c1c[nH]c(=NC)o1)=O)N(CC(C)OC)CC CC1(NC(c2cc(C(N)=O)co2)=O)CCN(C(c2cnc(C(C)(F)F)s2)=O)CC1 c1(C(=O)OC)c(NC(=O)C(=O)Nc2cccc(NC(=O)N(C)C)c2)ncn1C c1(NC(C2CCCCN(C(C(C)OCC#C)=O)C2)=O)c(C)cccc1[N+](=O)[O-] C1(NC(C=C(C)c2ccsc2)=O)CCOC12CCN(C(=O)CN1CC(C)C1)CC2 CCC(O)C(C)C(=O)NC1(CNC(c2c(C)coc2CC(N)=O)=O)CCCC1 C1(C(=O)NC(C2(O)CCN(c3snc(CC)n3)CC2)C)Cc2ccccc2O1 N1(C(C2(COC)CC2)=O)CC(NC(c2cnn(C(C)C)c2N)=O)C(SC)C1 c1(C(=O)OCC(=O)NCC(=O)NC)ccc(F)cc1Br c1(CC)cc(C(N2CCCC2CNC(=O)C(C)(C)CNC(C)=O)=O)ccc1OC C1(CC)CN(C(C2(C(F)(F)F)CC2)=O)CCC1CNC(=O)Cc1ncc[nH]c1=O c1(C2(C(=O)NC3C(CNC(CN(C(C)=O)C)=O)C3)CCC2)c(F)cccc1F N1(C(CN(C)CC)=O)CCCC(N(C(=O)Cc2ccc(F)c(C)c2)CC)CC1 c1(C(N2CCCC(C(N3CCCC(CC)C3)=O)C2)=O)cc(C)c(O)nn1 c1(NC(=O)NCC2COC(=O)O2)ccc(F)cc1C(F)(F)F C(CCCCCC(=O)NC1CC12CCC(NC(C1(C)C=CCCC1)=O)CC2)SC n1(CC(=O)NC(C(C)NC(C=CSC)=O)C)c2ccccc2c(=O)c2ccccc12 N1(C(COCc2nnc(C)s2)=O)CC(NC(C2CC(C)CC(C)C2)=O)C(C2CC2)C1 N1(C(c2nc(OCC)sn2)=O)CCN(C(c2cc3occc3s2)=O)CC1C C1(CSCc2nc(-c3ccccc3)no2)CCN(Cc2n(C)nnn2)CC1 Cc1nc2cccc(C(=O)NCCCNC(C3CCCSC3C)=O)c2[nH]1 C(CCCCS(=O)(=O)CC)n1cc(C2OCCN(C(C(CC(=C)C)C)=O)C2)nn1 C1(CNC(C2CC(CC)(CC)C2)=O)(NC(=O)CC2(C)CC2)CCCCC1C c1(CCCC(=O)N(C(C)CNC(=O)CCCNC(C)=O)CC)ccc(C#N)cc1 c1(NC(C2(F)CN(C(C3CC3(F)Cl)=O)C2)=O)ccc2nn[nH]c2c1 C1(CNC(C(C)CF)=O)C2CN(C(=O)Cc3sccc3Br)CC12 C1(C)(CC)CC(NC(C2(CCCC)CCCC2)=O)CN1C(c1ccc(C)o1)=O c1(C(=O)NCC#CCNC(CNC(C(CC)C)=O)=O)cnc(Cl)n1C C1(CCNC(CCC=C)=O)CN(C(=O)CCCn2ccnc2C)CCS1(=O)=O c12ccc(cc1)CS(=O)(=O)N2.n1(CCCCC)cc(-c2noc(C(F)F)n2)nn1 c1(C(CNC(=O)C(F)=CCCF)NC(c2ccc(CO)s2)=O)ccccc1 C1(CCC)(NC(c2cc[nH]c(=N)n2)=O)CCN(C(c2ns[nH]c2=O)=O)CC1 n1(CC)ncc(C(=O)N(C2CCN(C(c3cnc(Cl)s3)=O)C2)C)c1C1CC1 C1(NC(c2[nH]cc(C)c2)=O)CC1C1CCN(C(c2ccncc2O)=O)CC1 CCC(C)C(=O)C(=O)NC(CCC1CC1)C(=O)N(C)Cc1nc(C)cs1 N1(C(c2n(C)cc(Cl)c2)=O)CCCN(C(=O)C(C#N)CC2CC2)CC1 N1(CC(N2CC(C(C(=O)NC34CCC(CC3)C4)OC)C2)=O)C(C)CCC1C c1(C(=O)NC(CC)(C)CNC(=O)COCC(C)C)ccc(OC(F)(F)F)cn1 C(CCCCC(=O)NC1CC1C(=O)NC1CC1c1cccnc1)NC(C)=O c1(C2N(CC(C3(CNC(C)=O)CCCC3)=O)CCOC2)cccc(F)c1F C1(C(N2CCC(O)(CCNC(C3CCCCS3)=O)CC2)=O)CCCCC12CCC2 c1(C(=O)OC)cccnc1-c1cn(C(C)C(=O)NCCC2CCCC2(C)C)nn1 C(=O)(CC1OCc2ccccc21)N1CC=C(CNC(C2CCCC2(F)F)=O)CC1 C1(C(C)NC(c2n(CC)ncc2)=O)CN(C(=O)CCn2c(C)ccc2C)CCO1 C(=O)(C(C)CC(=O)N1C(CNC(c2ccc(F)cc2F)=O)CC2CC12)OC c1(C(=O)NC(CC)CNC(=O)C(C)c2ncco2)cc(C)ccc1[N+](=O)[O-] C1(CNC(C(C(C)C)NC(N)=O)=O)CN(C(c2coc(C3CC3)n2)=O)C(C)(C)C1 C1(O)(CNC(=O)CC(F)F)CCN(C(c2ncc(Cl)cc2Cl)=O)CC1 Cc1cc(C(=O)N(C)CC2(CNC(c3nc(C4CC4)cs3)=O)CC2)n(C(F)F)n1 C#CC1(C(=O)NCc2cc(C(=O)NCC(C)(O)C(F)F)n(C)n2)CC(=O)C1 C1(NC(c2cc(CCC)nn2C)=O)(CO)CCCN(C(c2ccc(C)nn2)=O)C1 CC(C)C(O)CC(=O)NC1CN(C(=O)CN2CCCCCC2)CC1C N1(C(CCC(C)OCC)=O)CCC(C)CC1C(=O)NCC=Cc1ccccc1 CCC(CC)C(C(=O)N1CCCC1CNC(=O)C(=Cc1ccccc1Cl)C)OC c1(C(=O)NC2(CC=C)CN(C(C3CC3c3ccc(Cl)s3)=O)C2)ccc(F)cc1Cl C1(CNC(C(C)(C)C2CCCCO2)=O)NCCC1C1CC1 C1(CC(=O)N(CC(C)NC(C(C)C(C)(C)C)=O)C)CCCCCC1(F)F c1(OC)cccc(CCC(=O)NCCN(C(=O)CCOCC(C)C)C2CC2)c1F c1(C(N(CCCNC(=O)C(F)(F)CN(C)C)CC)=O)ccc(NC)cc1Cl c1(C(=O)NC2CC(NCc3c(Cl)ncc(C)c3)C2)cnc2cccc(Cl)c2c1 C1(C(=O)NCc2cc(C(N(CCCO)CC)=O)on2)CC2CCCC2C1 c1(C2CCN(C(C(N3CCC(O)(C(C)(C)C)C3)=O)=O)C2)cccc([N+](=O)[O-])c1 CC1CCCC(Cn2cc(-c3ccccc3)cn2)C1 c1(CC(=O)N(CC(C)(C)CNC(=O)C(C)=C(C)C)CC)cccc(C#N)c1OC C(=O)(CC(CC)N(C)C(c1ccsc1C#N)=O)N(CCCO)CC#C C=CCC(CC(C)C)C(=O)NC1(C(=O)NC(CC)C(C)(F)F)CC1 C(C(CC)(CC)CC)NC(c1ccc(CC)nc1)=O c1(-c2ccc(C(=O)OCC)nc2)c(Cl)ccc(NC(=O)CCCCCSC)c1F C(=O)(C(C)C(C)(F)F)NC(CC)CNC(=O)Cn1cc(Cl)c(C(F)(F)F)n1 C(c1ccccc1C#N)=CC(N1CCCC(N2CCN(C(CC)=O)CC2C)C1)=O C(=O)(C1CCCc2cncn21)NC1CN(C(C(F)=CCC)=O)C2C1CCC2 c1(SCC(C2CC2)OC)cc(CO)cc(F)c1 C12(CNC(C=Cc3nc(C)sc3)=O)CCCC1N(C(C1CC3C=CC1O3)=O)CC2 N1(C(CCOCC)=O)CCCCC1C1(CNC(c2nsnc2O)=O)CCOCC1 C1(CC=C)(NC(=O)C(C)COC)CCCN(C(=O)CN2CCC(=O)NC2=O)C1 c1(OC)cncnc1C(=O)NCC(CC1CC1)C(=O)N1CC2(CC2)C1 N1(C(C2N(C(CC3C(C)OCC3)=O)CCOCC2)=O)CCCC(N=[N+]=[N-])C1 c1(OC)ccc2cc(C(=O)NC(C)(C)CN(C(=O)C(F)(F)C(C)O)C)ccc2n1 C1(NC(c2cncc(F)c2Cl)=O)CCN(C(C2CCCC2(F)F)=O)C12CC2 c1(NC(C(CSC)(C)NC(=O)CC2CC(F)(F)C2)=O)cc(C)cnc1C C#CCCN=C(NCc1ccc(CN2CCCC2)cc1)NC(c1ccccn1)C C=C(C)CCCC(=O)NC(C1CCCCC1)CNC(c1cncc(O)c1)=O N1(C(c2occ3c2CCC3)=O)CCC2(NC(C3(NC(N)=O)CC3)=O)CCCCCC12 N1(C(c2c(OC)cccc2F)C(=O)NCCSC)CCCOCC1(C)C C(=O)(C=C1SCC(=O)N1C)NCC1(O)CN(C(C2CCN(CC)CC2)=O)C1 Cc1cccc(C)c1NC(=O)C(c1ccoc1)NC(=O)CN(C)C(N)=O N1(C(CC(C)(C)NC(N)=O)=O)CCC2(CCCN2C(=O)COC2CCOCC2)C1 c1(C(N(C2CC(NC(=O)CCc3csc(Br)c3)C2)C)=O)cnccn1 N1(C(C=C(CC)CC)=O)CC2CCCC(CNC(=O)C=CC(C)C)C2C1 Nc1ccc(Br)c(C(=O)NCC2(F)CC(NC(c3cnsc3)=O)C2)c1 N1(C(CC(=O)NC)=O)CCc2ccccc2CC1.C(C)(C)(C)OC(=O)C1CC1 C1(CNC(C(COC)N(C)C)=O)CN(C(=O)C(C)(C)CSC)CCO1 Fc1c(Cc2cn(-c3ccc(N4CCCC4)cc3)nn2)ccnc1Br Cc1cnc2n1CC(C(=O)NCC(C1CCC1)NC(=O)C(F)(F)C(F)(F)F)CC2 CC1(C)CC(NC(=O)C=CC2CCOCC2)CN1C(c1cc(CO)ccn1)=O c1(C(N(C)CC2CCCN2c2ccnc(C3CC3)n2)=O)nnc(O)nc1O Cc1nc(C2CC2)ccc1C(=O)N(CCNC(C1CC(=O)N1)=O)C1CC1 Cc1cc(C(=O)NC2CC(F)CN(C(C3CC3C)=O)C2)n2ncnc2n1 c1(C(C(=O)NCc2cccs2)N(C2COCC2(C)C)C)cnc2ccnn2c1 Cc1cc(C)n2nc(C(N3CCCC3C3(O)CN(C(=O)CN(C)C)C3)=O)cc2n1 c1(C(N(CC(C)(C)NC(C=CCOC)=O)C)=O)cc(CCO)on1 C(=O)(C1=C(Cl)CCCC1)N1CCN(C)CC1C(=O)NC1CNC(=O)C1 n1(CCC)ncnc1CN(C)CCN(C)C(=O)NC1CCN(C)C1 C#Cc1cc(C(=O)NC2C(=O)OC2)cc(F)c1.c1(OC(C)C)ccc(C)cc1F c1(N(C)C)ncc(C(=O)NCCCC(C)NC(c2ccncn2)=O)cc1Cl c1(C(C(=O)N(CC(=O)N(C)C)C)NC(C(C)C)=O)cccc(C(F)(F)F)c1 N1(C(C2C(=C)C2C(=O)OC)=O)CCOC(C)C1C(N1CC(F)(F)CC1C)=O C1(C(=O)NC(c2csnn2)C)CCC2CCC1N2C(c1ccncc1)=O C1(C(N2C(Cn3cc(-c4nc(C)sc4)nn3)CC2)=O)CCC2CC2CC1 C1(N(C(c2cnc(Cl)[nH]2)=O)CC)CCCN(C(=O)Cc2c(Cl)cnn2C)C1 c1(C(=O)NC2(CCOC)CCN(C(=O)C(C)CO)C2)cncc2ncn(C)c12 n1(C2CC(C(N(CC=C)Cc3cccs3)=O)C2)cc(C(=O)OCC(=O)OC)nn1 CS(C)(=O)=NCCNC(c1ncc(-c2cccc(Cl)c2)s1)=O N1(Cc2c(OC)nccc2)CC2CCC(NC(c3cnncc3O)=O)CC2C1 C(=O)(C(C)C(C)S(C)(=O)=O)N1CCC(n2cc(-c3cccc(C)c3)nn2)CC1 CN(OCc1ccccc1)C(=O)C(CCOCCO)NC(C1CCOC1)=O C1(NC(C2C(CC)C2)=O)CN(C(c2ccc3ncnn3c2)=O)CC(C)(C)C1 Cc1nn(C)c(C)c1C(=O)C(=O)NCC(CO)NC(=O)C(O)CC1CCCCC1 c1(C(CNC(C2(C)CCN(C)C2)=O)NC(C2(C(N)=O)CC2)=O)cc(F)cc(Cl)c1 Cc1cc(O)c(C(=O)NC2CCCC(CNC(=O)Cc3cnc[nH]3)C2)nn1 C1(CCNC(C(C=CCCC)O)=O)CCCN(C(C2CCCCS2(=O)=O)=O)CC1 Cc1ccc2ncnc(N3CCC(CNC(C4CCc5ccccc5O4)=O)C3)c2c1 CN1CCCCC1C(=O)NC1COCC1NC(c1cnc(O)o1)=O C(=O)(C(C(C)(C)C)NS(C)(=O)=O)NCC(C)NC(c1cccc(NC(N)=O)c1)=O CC(C)C#CC(=O)NC(Cc1cn[nH]c1)C(=O)NC(c1cccnc1)C c1(C(N(CC(C)NC(=O)CC2CC=CCC2)C)=O)cc(C(N)=O)[nH]n1 N1(C)CC2OCCN(C(C)(C)C)C2C1.Cc1c(C(N2CC(C(=O)O)C2)=O)cncc1Br C#CC1(C(=O)NCC(O)CC(=O)NCC(c2ccccn2)C)CCCCC1 C1(CNC(C(C)C(F)F)=O)CN(C(c2cccc(Br)c2Cl)=O)CC12CC2 C(=O)(CC1=CCN(C(=O)C(C)(C)OC(C)C)CC1)N(CC)CC1CCC1 N1(C(C2(CCC=C)CC2)=O)CCC(OCC(N2CC(O)(c3cnn[nH]3)C2)=O)C1 CCCCC(O)C(=O)NC1CCCC1NC(C1CCC(CC)CC1)=O N1(C(c2ccc(Cl)nc2)=O)CC2CCC(C1)C2NC.C(CCCCN1CCCC1)O N1(C(C(C(C)C)(C)O)=O)CCN(C(c2ccc(C#N)[nH]2)=O)CC12CCC2 C1(CC(N2CC(c3c(C)con3)C2)=O)CC2(CC2)CN1C(=O)C=Cc1cncn1C CC1COC2(CCCC2)CN1C(=O)Cn1cc(CCC2CCOC2)nn1 CCC(C)(CC)C(=O)NC(C)CCNC(c1cccn1Cc1cccs1)=O Cc1cc(=NC(=O)C(=O)N2CC(O)(C(C)NC(=O)CC(C)C3CCCC3)C2)[nH]o1 c1(N(CCCC)C(=O)NCC2CCOC(c3ccncc3)C2)ccc(Br)cc1 CC(C)(CCC(=O)NC1(CF)CCN(C(c2ccc(Cl)nc2N)=O)C1)[N+](=O)[O-] C(=O)(C1CCCc2sc(C)nc21)NC1C2C(NC(C(F)=CC)=O)CC(CC2)C1 c1(OC)ccc(-c2cccc(OC)c2F)c(CN2CCC(O)(CN(C)C)C2)c1 c1(C(N2C3(CN(C(CC(=O)NCC)=O)C3)CC2)=O)ccc(S(C)=O)cc1 CCCC(C(=O)NC1CCCC(CNC(=O)CCC2(C)CC2)C1)S(N)(=O)=O c1(C(=O)NC(c2nccs2)Cc2ccccc2)coc2c(F)c(Cl)ccc12 C(CC(C)(C)C)(C(=O)NCC1(CNC(C2CCOC2)=O)CC1)OC Cc1nc2cncc(C(N3CC=CC3CNC(=O)COCC3CCCC3)=O)c2[nH]1 c1(C(=O)NC2C(NC(C(C)(C)OC)=O)CC2)ccn2ccnc2c1 CC1CN(C(=O)C(C(C)O)NC(c2cc(Cl)cn2C)=O)CC1F N1(CCCCN(C(=O)Cc2ccoc2)CC2CC2)CCCCC1 C1(C)(CNC(C2CC(OC)C2)=O)COCCN(C(=O)CC2(O)CCCCC2)C1 C(c1ccc(Cl)nc1)=CC(=O)NCCNC(c1ccn(-c2ccncc2)n1)=O c1(NC(CNC(CC2CCCC(C)(C)O2)=O)=O)ccc2c(c1)OCO2 C12(NC(C3C(C)(C)COC3)=O)CCCC(NC(c3cnccc3Cl)=O)(C1)C2 N1(CCC2CCC2)CCOCC1.c12ccc(s1)NC(=O)C1C(C1)NC2=O C=C(C)C(C)(C)C(=O)N(CCC(=O)NCC1CC1c1ccoc1)C(C)C S(=O)(=O)(c1cccnc1)NCCC(=O)NC(c1ccc(F)cc1F)(C(=O)OC)C C(=O)(C1=CC2(CCN(C(c3c(F)cccc3F)=O)C2)C1)N(CC(C)C)C N1(C(C(CC)(C)F)=O)CCC(CNC(=O)CC2(CO)CC2)C(F)(F)CC1 c1(N(CC(Cl)Cl)C)[nH]c(=NCc2ccccc2C2CCC2)nc2scnc12 C1(CCOC)(NC(=O)Cn2ncccc2=O)CCN(C(c2ccnn2C)=O)CC1 CC1(C2CCCN(C(C3CCCN(C(=O)COCCF)CC3)=O)C2)CC1 Cc1ccc2c(c1)CC(C(=O)NC1CCC(CNC(=O)C3=COCC3)C1)S2(=O)=O C1(CNC(C(CC)OCC)=O)C(C2CC2)CCN1C(=O)CC1(COC)CC1 C=C(C)CC(C(=O)NC(C)C(C)C(=O)OC)NC(c1cccc(C)n1)=O C(C(C)(C(=O)NCCCOC(F)(F)F)NC(=O)C(C)N=[N+]=[N-])SC c1(C(N(CC(C)NC(C2CCC(O)C2)=O)C)=O)cc2c(F)cc(Br)cc2[nH]1 Cc1cc(N(CCCNC(=O)CC2CCCC2(F)F)CC2CC2)nc(C(C)C)n1 N1(C(C(C)(C)c2ccns2)=O)CCC(F)(F)C(CNC(C2CC3CC3C2)=O)C1 CC1CC=C(C(=O)N2CCC(C(=O)NCCC3OCCC3C)C(O)C2)CC1 N1(C(c2c(C)nc(C)s2)=O)CCN(C(=O)COCCCF)CC(C)C1 C(=O)(C(C(C)CC(C)(C)C)N(c1ccccc1)CCCSCC)NCCCSC c1(OC)cc2c(c(OC)c1OC)CN(C(CC(C)CO)C(=O)NCC1CCC1)CC2 c1(C(N2CCC(CNC(C34CCC(C3)C4)=O)C23CC3)=O)cc2ncccc2o1 Cc1ccc2c(CC(N3CC(NC(=O)CC4(O)CCOC4)C3)=O)coc2c1 c1(C(N2CC(CCC)C(C(N3CC(O)C(O)C3)=O)C2)=O)c[nH]c(C)cc1=O C1(NC(CNC(CCC)=O)=O)CC(F)CN(C(C2(C(=O)OC)CCCCC2)=O)C1 c1(C(N2CCC(F)(CNC(C(C=CC)O)=O)CC2)=O)c(OC)ncc(Cl)c1C CN1CCN(C)C2(CCN(C(C(=O)NC3CC3)C3=CCCCCC3)CC2)C1 C1(C)(CC(=O)NCC(CNC(CC2(N(C)C)COC2)=O)CO)CCCCC1 c1(C(N(CCNC(CCSCCC)=O)C)=O)coc2cc(OC)ccc12 N1(CC(=O)NCc2onc(CCC)n2)CCN(C(=O)CCc2cc(Cl)no2)CC1 C1(CNC(C2(CC#C)CCCO2)=O)CCCCN(C(=O)C=Cc2ccn(C)c2)C1 N1(C(C(c2ccccc2)C)=O)CC(F)CC1CN(C(=O)C=CSc1nc[nH]n1)C C1(C(N2C(CC)CCCC2)=O)CCN(C(=O)c2cc[n+]([O-])cc2)O1 CC1CC2(CCN(CC3(O)CCOC=C3N=C3CCC3)CC2)CN1C(=O)C1CC1 c1(CNC(C2C(NC(c3cc(C)sn3)=O)CCO2)=O)ccc(C2CC2)cc1 c1(CNC(C(c2ccn(C)c2)C)=O)ccc(C(=O)N(CCCC(O)CO)C)nc1 c1(NC(CC2N(C(C=NOC)=O)CCC2)=O)cn(CC)nc1C#N c1(C(=O)NCC2CCCN2C(C2(F)CCS(=O)(=O)C2)=O)cc(O)nc(C2CC2)n1 N1(C(CCC(=O)N(C(C)C)C)=O)CC(NC(=O)C(C)C2CCC2)CC2(CCC2)C1 c1(C(=O)OC)cnc(O)c2c1CCCN2C(=O)CCc1ncco1 N1(C(CCCNC(C)=O)=O)CCC2CCN(C(=O)C3CC3)C2C1 c1(C(N2CCN(C(C3CCN(CC#C)CC3)=O)C(C)C2)=O)ccc(Cl)c(C)c1O C(=O)(CCCCCN(C)C)N(CCN(C(C(CC#C)O)=O)C)C c1(C(N2CC(NC(c3cc(CC)cc(Cl)c3)=O)C2)=O)c(C)ccc2nsnc12 Cc1cnc2c(C(=O)NC(C)CC3CN(C(C4CCC(C)(C)C4)=O)C3)cccn12 c1(C(=O)NC2CCC(CCNC(c3c(Cl)cn(C)n3)=O)C2)nc2cnccc2s1 C1(CC)CN(C(=O)CN(CC(=O)NC(C)C)C)CCN1C(=O)C1=CC(C)CC1 N1(C(=O)CC2CCCOCC2)CCN(C(c2cnc3n2CCS3)=O)C(CF)C1 C1(CCC)(NC(=O)C(C)CC(C)C)CCCN(C(=O)C=Cc2ccc(SC)s2)C1 c1(C(N2CCCC(CCN)C2)=O)sc(C(=O)O)c2c1CCCC2 N1(C(C=C(C)C(=O)O)=O)CCC2C(CCN2Cc2ccc(Cl)cc2)C1 C1(C(NOCC)=O)CC(NC(C2CCN2C)=O)C1(C)C c1(CNC(C23CC(NC(=O)CCc4ccsc4)(C2)C3)=O)c(F)cncc1F N1(C(C(C(C)C)OCC)=O)CCC2CN(C(=O)COCCF)CC12 C1(CCC(=O)N(C2COCC2O)C)CCN(C(=O)CCC2(C#N)CCC2)C1 c1(CNC(C(CC)C)=O)ccc2c(c1)CCCC2NC(C12CC(C)(C1)OC2C)=O n1(CC)c(C)c(C(=O)NC2CN(C(=O)CC3CC3)C3CC23)c2cc(OC)ccc12 C1(NC(=O)C=CBr)CCC12CN(C(c1ccn(-c3cccc(F)c3)n1)=O)C2 Nc1cc(F)c(O)cc1C(=O)NC1CCC(CCNC(=O)CC(=O)NC2CC2)C1 C12(CNC(CN(CCOC)C)=O)CCCC1N(C(=O)COCC(F)F)CCC2 CCC(CC(C)O)NC(N1CC(Oc2ccccc2C(N)=O)C1)=O C1(C(=O)NC2C3(CC(NC(C4CN(C(C)C)C4)=O)C3)C2)CC(=O)NC(=O)N1 CCC(CC)(CO)C(=O)NCC(C)(C)OCC(=O)NC(CO)C(=O)OCC(C)C CCCC(CNC(=O)C(C)c1ccco1)NC(c1cnc(C)[nH]1)=O c1(NS(c2c(C(N)=O)c(F)ccc2)(=O)=O)ccc2c(S(N)(=O)=O)cccc2c1 C1(NC(C2(OCC)CCC2)=O)CCC(C)N(C(=O)CCOCC(C)C)C1 c1(CC(=O)NCC(C)N(C)C(c2cccn2C)=O)ccnn1-c1ccccc1 N1(C(C(C)NC(CC)=O)=O)CCC(N(CC(C)C)C(C2(F)CC=CC2)=O)CC1 C1(CNC(c2ncn(CC)n2)=O)CC(O)C(O)CC1C(=O)NCCN1CC=CC1 C1(C(=O)OC)CCCCCCN1C(c1cnccc1OC)=O C1(C(=O)Nc2c(C)cccc2)CCN(C(=O)C2CCNC(=O)C2)O1 C1(C(C)NC(c2c(CC)scc2)=O)CCN(C(=O)CCOC)CC1 C(=O)(C(CC(C)C)n1ccnc1)NC(CC)CNC(=O)C=CC(c1cccnc1)=O C(=O)(CC(O)CC(C)(C)C)N1CCC(CN(C(c2cc(C)n(C(C)C)n2)=O)C)C1 c1(C(N2CC(CNC(c3ccc(CCC)s3)=O)C(C)C2)=O)ccc(OC)cc1C C1(N(C(CSCCOC)=O)C)CN(C(c2cn(C(F)(F)CO)nn2)=O)CC1F C1(NC(C(C)(C)c2nccs2)=O)CCCC2CN(C(=O)Cc3ccsc3)CC12 C1(C(=O)NCCCN(C(c2c(OC)nsc2)=O)C)CCC(=O)N(C2CC2)C1 N1(C(C(=O)NCCCSCC)C2CC2COC)CCC(C#N)(CCC(C)C)CC1 Cc1cc(Cl)c(C(=O)NC2CC2CNC(c2ccc(Br)cc2)=O)cn1 c1(C(=O)NC(C2N(C(CCOCCOC)=O)CCC2)C)sc(C)cc1OC c12ccccc1OCC(C)NC(=O)C1CN(CC1CC)C(=O)N2.O(C(F)F)CC C(=O)(C(CN(C)C)NC(C1CC1C(C)(C)C)=O)NC(c1nc[nH]n1)CC C12(CNC(C3C(CC)CCN3C(C3CCOC3(C)C)=O)=O)CCCN(CC1)C2 N1(C(CCC2CC(C)C2)=O)CCC2CCN(C(=O)C=CC(F)F)CC12 c1(C(N2CC(CC=C)(NC(c3csc(C)n3)=O)C2)=O)csc2ccccc12 Cc1cc(C(=O)Nc2cc(C(F)(F)F)cc(Br)c2O)c2c(C3CC3)noc2n1 C(=O)(C1=CCCC(C)(C)C1)N1C(CC)CN(C(=O)CCOC2CC2)CC1 C1(NC(CC2OCC(C)(C)C2)=O)CCN(c2nnc(CO)s2)C12CCC2 N1(C(c2ncn(CC)c2)=O)CCC(CNC(C2CCCN2C)=O)C(O)C1 C1(O)(CNC(=O)CCN2CCCCC2)CCCN(C(=O)CCc2cnc[nH]2)C1 C1(NC(CC2ON=C(C)C2)=O)C2CC3C1C3C2C(=O)NCCN1CCCCC1=O C1(NC(C(CC)NC(C)=O)=O)C2CC1CN(C(c1cc(C)nc(C)n1)=O)C2 C(=O)(CC1=CCN(C)CC1)NCC(C(=O)NC(CC)(C)CN(C)C)C Cc1n[nH]c(C)c1CC(C)C(=O)NCC1(NC(=O)CC23CCC(CC2)C3)CC1 N1(C(c2n(CC#C)ccc2)=O)CC(C(N2CC(N(C)OC)C2)=O)CC1(C)C C1(NC(=O)C(F)CC2CN(C(=O)CCC(F)(F)F)C2)CCC=CCCC1 C1(C(=O)NC(C(=O)NCc2cncnc2)Cc2ccco2)CC2C=CC1O2 CCCC(C)CC(=O)NC(Cc1ccco1)C(=O)N(C)CC CC1CC(NC(c2csc3nccn23)=O)CCN1C(c1cc(N)c(Cl)cn1)=O CC(C)(C(=O)NCCOC1CCN(C(c2c[nH]c(=N)s2)=O)C1)N1CCCC1 c1(C(=O)NCC2C(C(=O)NCC(CC3CC3)OC)CCC2)cncn1C c1(NC(C=CCC)=O)cccc(Cl)c1NC1CC(=O)N(c2ccc(Cl)c(F)c2)C1 c1(C(=O)NC(C2N(C(C(C)=C(CC)C)=O)CCCC2)C)noc2c1CCCCC2 C1(C(=O)NCc2cn(C3CN(C(C(C=CC)O)=O)C3)nn2)CCC(SCC)CC1 c1(C(=O)Nc2nccc(CC)c2)cc(C)nc2ccnn12 c1(C(N2C(C(C)(C)NC(C(F)=CC)=O)CCC2)=O)cc(F)c(F)cc1O C1(C(=O)NC2CC3CC(C2)C3)C(CC)CCN1C(=O)C(=O)N(C)C N1(C(CCCC#C)=O)CC2(CNC(C3CCCS(=O)(=O)C3)=O)CC(F)(C1)C2 C1(CNS(C)(=O)=O)CCCCN1C(=O)N(CCc1ccccc1F)CCO C(=O)(C(C)C(O)C(C)C)N(CC(=O)NCCc1cc(CC)no1)C(C)C C1(NC(c2c(C)sc(Cl)n2)=O)COCCN(C(C2CC3CCC2CC3)=O)C1 c1(C(N2C(CCNC(C(C)C(C)(C)C)=O)COCC2)=O)ncn2c1CCCC2 C(CNC(=O)CC1(NC(C2CC2CC(C)C)=O)CC1)(C(C)(C)C)OC C(=O)(CCCCCC(=O)NCC(C)N(C(=O)C(C)n1ccnc1)CC)OCC CCCC(C(=O)NC(C(=O)NCCN(C)CCOC)C(C)OC)OC CCCCC(CC)C(=O)N1CCC(CNC(=O)C=Cc2nccs2)C1(C)C N1(C(CN(CC)CC)=O)CC2CCCC(NC(c3ccncc3F)=O)C2C1 CCC(CO)(C(=O)NCC1COCCN(C(c2sc(C)nc2C(C)C)=O)C1)OC c1(OC)ncc(C(N2CCC(NC(=O)CNC3CC3)C(C)C2)=O)cc1Cl C1(OCCC(C)c2cn[nH]c2)(NC(CNC(CNC(=O)OC)=O)=O)CCC1 N1(C(CCC2C(C)(C)C2)=O)C(CNC(C2COC(=O)N2)=O)CC2CCCC12 N1(C(CCS(=O)(=O)N(C)C)=O)CC(NC(c2cncc(N)c2)=O)CC2(CC2)C1 N1(C(C=CC)=O)CCN(C(c2cc(C)c(C#N)cn2)=O)CC12CCC2 C1(CC)C(C(=O)N(C)Cc2cccnc2)CCN1C(=O)C(O)C1CCC1 C1(NC(CC2(C)CC2(Cl)Cl)=O)CC(Nc2ncccn2)C12CCC2 N1(CC)CC2CN(C3COC3)CC2C1.CC(C)C(C(=O)O)NC(c1ccccc1)=O CC(O)C(C)(C)C(=O)N1CCC(N(C(=O)CC2(CS(C)(=O)=O)CC2)C)CC1 c1(C(N(CCNC(C(C=C)O)=O)CC2CC2)=O)nnn(Cc2cc(C)on2)c1C c1(OC)c(C(=O)NCCN(C(C2CCOCC2C)=O)C(C)C)cc(F)cc1F c1(C(N(CCCNC(Cc2nc(C)oc2)=O)C2CC2)=O)snc(O)c1Cl Cc1cc(F)cnc1C(=O)NCCc1cn(CC2(CC(=O)O)CC2)nn1 c1(CC)ccc(C)cc1NNC(=O)c1ccc(Cl)c(C)c1Cl C(C(=O)N1CCC(=CCNC(=O)C(CC)OC)CC1)(C(C)C)NC(=O)OCC C(=O)(C1CCC(=O)c2ccccc21)NCC1N(C(C2(C)CSC2)=O)C2CCC1C2 C1(CNC(CCSCCCC)=O)CCC(NC(c2ccccc2)=O)CC1 N1(C(C23CN(C(CCN(C)CCO)=O)C(C2)CO3)=O)CC2(COC(C)(C)C2)C1 c1(C(=O)NC(C2CN(C(c3cc(C)no3)=O)C2)C)c(O)cc(F)cc1F c1(C(=O)OC)cc(Cl)ccc1CNC1CN2CCC1(C(F)(F)F)C2 N1(C(C(n2c(C)ccn2)C)=O)CC2(CC2)CC1CNC(c1cc(Cl)cs1)=O Cc1cc(Br)cc(C)c1COc1ccccc1C(=O)NC1CCCCC(F)(F)C1 N1(C(C2CC(CC)C2)=O)CCCC(C)C1CCNC(c1cnc(O)cc1OC)=O C1(F)(C(N(C2CCCC2)CC=C)=O)CCN(C(=O)Cc2cc(C)[nH]n2)CC1 C#CCCC(O)C(=O)NCC1CCC1NC(c1cccc(C(F)(F)F)c1)=O n1(Cc2ccccc2)nc(C2CCOC2)nc1C.C1(Cn2cnnn2)CCCCO1 c1(CC)cc(C(=O)NCCNC(C2CC(CCO)C2)=O)c(Br)s1 c1(NC(CCC2CCCN(C(Cc3c(C)ocn3)=O)C2)=O)ccc(O)c(CO)c1 C1(C(=O)Nc2nc3cccc(C(=O)OC)c3o2)CCCC2(CCOC2)O1 CCCCC(CNC(C1(C(F)F)CC(F)(F)C1)=O)NC(c1cc(F)c[nH]1)=O c1(SC)ncc(N)c(C(N2CC3C(NC(C4(C)CC4)=O)C3C2)=O)n1 c1(N2CCC(NC(c3cccc(=O)o3)=O)C(F)C2)ncnc2[nH]ccc12 C1(C(=O)NC2CCC(NC(c3n(CC)ccc3)=O)C2)CCCS1(=O)=O N1(C(c2ccc(C)o2)=O)CCCCC1C1(NC(c2cnn(C(C)C)c2)=O)CC1 CCCCCCC(=O)NC1CN(C(C2C=CCCC2)=O)CCC1C C(=O)(C1CCCc2c[nH]nc21)N1CCC(C(C)Nc2snc(C)c2C#N)C1 N1(CCC=CCC)CCC2(CC1)CC2C(=O)NC1(C(=O)OC)CC1 N1(C(c2cncc(OC)n2)=O)CC2CCCC1(CNC(=O)C(C)(O)C(C)C)C2 C1(C(C)NC(=O)Cc2cc(CN(C)C)no2)CCCN(C(c2ccncn2)=O)C1 Cc1cnc(Cl)c(C(=O)NCC2(O)CCCN(C(=O)CNC=O)C2)c1 Cc1nc(C2CCC2)oc1C(=O)NC(C1CCCN1C(c1ccc(CO)s1)=O)C C1(C(C)C)CN(C(=O)C(C)c2cc[nH]n2)CCN1C(=O)C1=CCCC1 c1(N(C)Cc2cc3ccccc3o2)ccc(S(=O)(=O)NC2CCC(F)C2)cc1Cl C1(C(=O)NC(C)C(N2CCC(N3CCCC3)C2)=O)(CO)CCCO1 Cc1ccc(C(N2CC3(CNC(=O)Cc4csc(Cl)c4)CC2CO3)=O)nc1F c1(N2CC3(C(C(=O)Nc4c(OC)nn(C)c4)C3)C2)ncnc2ccccc12 Cn1cnc2cc(C(=O)NCCCOCCCNC(c3ccsn3)=O)ccc12 C1(CNC(=O)CCc2nccn2C)CCN(CC2N(C)CC(O)C2)C1(C)C C1(CNC(c2n[nH]c(C)c2Cl)=O)CC2(CC2)CN1C(=O)CCc1nc(O)n[nH]1 C1(CC)CN(C(=O)CC2NC(=O)NC2=O)CCN1Cc1sncc1Br c1(OC)ccc(C(N2CC(NC(CC(N)=O)c3cn(CCO)nn3)C2)=O)cn1 c1(OCC(=O)N(C2CN(C(CCSCC)=O)CC2F)C)ccc(Cl)cc1F C(=O)(C1c2ccccc2C2CC1C2)NC1(CN(C(=O)C(C2CC2)N(C)C)C)CC1 c1(C(N2CCC(NC(C3CC(CF)C3)=O)C2)=O)ccc2[nH]c(=O)c(=O)[nH]c2c1 C1(CCNC(C2(CNC(C(C)OCCOC)=O)CC2)=O)CC(=O)N(C)C1 c1(C(N)=O)ccc(S(=O)(=O)N2CC(NCc3cnc(Cl)cc3Cl)C(C#N)C2)cc1 CCCC(CC(=O)NC(C)CF)NC(c1cnc[nH]c1=N)=O N1(C(C(C)O)=O)CCC(CF)(NC(=O)CCCCN(C)C(=O)OC(C)(C)C)C1 N1(C(CCC(=O)NC)=O)CCC2(CC1)COC(CNC(=O)C(C)(C)C)C2 Nc1ccc(F)c(C(N2CCC3C(NC(c4cnsc4)=O)C3CC2)=O)c1F c1(CN2CCC(C(C(N)=O)F)CC2)cc2c(cc1O)CCCC2 N1(C(c2c(CC)cns2)=O)CC2CC(C1)CN(C(c1conc1C(C)C)=O)C2 C(CCCCC(=O)N(CC(O)CN(C)C(c1cn2ccsc2n1)=O)C)=CCCC Cc1ccc2nc(C)c(C(=O)NOCCNC(=O)OCCC(C)(C)C)n2c1 CCCS(=O)(=O)CC(=O)NCC1(NC(=O)Cc2ccnn2CC)CCCCC1C CCCCCC(F)C(=O)N1CCC(NC(=O)C=CC(=O)N(C)C)C1C1CC1 C(C(C)C(=O)NC(C1(O)CN(C(=O)C=C2CCC2)C1)C)OC c1(C(C)NCC2CC2)ccc(F)c(C(=O)Nc2c[nH]nc2-c2ccco2)c1 c1(C(=O)NC)ccc(C=CC(=O)NCCN(C(=O)C(C)(C)O)CC2CC2)cc1 C1(C(=O)NCCOCCCNC(CC(C)(C)O)=O)Cc2c[nH]cc2S1(=O)=O CCCC(C)CC(=O)NOCC(N1CC(c2cc(OC)ncn2)C1)=O C1(C(N(CCN(C(c2nc(C)oc2)=O)C(C)C)C)=O)CCOCC12CCCC2 C1(C(=O)NCC(O)C2CC2)CCC(CNC(c2n[nH]c(O)n2)=O)O1 C1(N(C(CCc2ccc(C)cc2)=O)C)CCN(C(C2CCCOC2)=O)CC12CC2 CCC(CNC(=O)C(C)NC(c1ccc(CO)s1)=O)C(C)(F)F N1(C(c2nn(CC)nc2C)=O)CCC(C2CCN(C(=O)CC(C)O)C2)C1 C1(OC)CN(C(c2ccc(C(N)=O)cc2)=O)CC12CCOCC2 N1(C(C2CC(C)=C(C)CC2)=O)CC2CCC1CN(C(=O)CSC(F)(F)F)C2 N1(C(C2(C(=O)OCC)CC2)=O)CCC(O)(CNC(c2cc(Cl)c(C)cn2)=O)CC1 c1(CC)cc(C(N2CCC(C)C2CNC(C2CCOC2)=O)=O)c2c(c1)CCO2 c1(C(CNC(COCC=C)=O)NC(c2cc(CC)[nH]n2)=O)cccc(Cl)c1 N1(C(C(C)(C)CNC(c2ccncc2Cl)=O)=O)CC2(C)CC1CCO2 c1(C(N(CCN(C(C2C(CC)C2)=O)C)C(C)C)=O)cnc2cc[nH]c2c1 CC(C)CC(=O)C(=O)N1CCC(C(N2CCOC(C3CC3)CC2)=O)C1 N1(C(c2ccc(OCC)nc2)=O)CCN(C(=O)C(C)c2cc[nH]n2)CC(O)C1 Cn1cc(NC(C2CCCN2C(=O)CC(F)(F)F)=O)c(O)n1 CC(O)CC(=O)OCC1(c2ccccc2)CCO1 c1(OCC)cnc(C(N2CCCC(N(C(=O)CC3CCCC3(F)F)C)C2)=O)cn1 O=C(C1=CC2CCC=CCCC12)NCC1CC(O)CN1C(=O)C=Cc1nccs1 C(=O)(CCN=c1[nH]ccs1)NC1CN(C(C(c2c(C)n[nH]c2C)C)=O)CC2C1C2 c1(N)cc(C2CC2)cc(SS)c1.C(C(C)C)CN(C1CC1)N N1(C(C=CCOC)=O)CCC2CC1CN(C(=O)C1=CCCOC1)C2 c1(C(=O)NCC(CNC(c2scc(C)c2)=O)F)snc(Cl)c1Cl C1(C)(CNC(c2n(CC)nnn2)c2csc(C(C)(C)C)c2)CC2(CCC2)C1 C=C(Br)CCC(=O)N1CC(NC(=O)CCN2CCCCC2=O)C(SC)C1 N#CC1(C(=O)NC(CNC(=O)CSCc2cccc(Cl)c2)CO)CCCO1 c1(OC)nsc(OC)c1C(=O)NC1CCC(NC(=O)C(C)(C)N2CCCC2)CC1 C(=O)(C(C)(C)C(=O)NCC1COCC1NC(=O)C1=CCCCO1)N(C)C C(=O)(C#CC1(C)COC1)NC(C(=O)NCC(C#C)CC)C1(C)CC1 c1(NC(C(C(C)OC)NC(c2ccsc2C)=O)=O)ccc(C)nc1O N1(C(C2(NC(c3ncc[nH]3)=O)C(C)(C)C2)=O)CCC2CC12C(=O)O C1(C(C)NC(c2cnc(C)[nH]2)=O)CCCCN1C(c1nnsc1C)=O c1(C(=O)NC2C(C)CN(C(c3cccc(CF)c3)=O)C2)ccc2nnn(O)c2c1 CC1c2cc(Cl)cc(Cl)c2CCN1C(=O)NC1CCOC1c1ccnc(Cl)c1 c1(OC)ccc2c(c1)C(C(=O)N1CCN(C(C)C)C(=O)C1)CC2 c1(CC)cc(C#N)ccc1NC(c1nc(NC(C2(Br)CC2)=O)cn1C)=O C1(O)(CC(=O)NCC2CC3CCC2N3C(C2CC2C2CCC2)=O)CCCCCC1 C(N=c1[nH]c(=NC2CC3CCC(C2)S3)[nH]c2c1SCC2)c1cccn2c1ncc2 c1(CC(=O)NC(CC=C)CNC(c2ncncc2Br)=O)cc(F)ccc1F CC1COC2(C1)CN(C(=O)CC1C3CCCC3N1C(=O)C(C)S(N)(=O)=O)C2 N1(C(C2(NC(c3c(C)scn3)=O)CC(F)(F)C2)=O)CCC(C2CC2)CC1 CC1Cc2ccccc2N(C(=O)NCc2ccnn2-c2ccccc2)C1C c1(C(N(CCCNC(COCCC)=O)C(C)C)=O)cnc2ccccc2c1OC C1(CNC(C(C)SC(C)C)=O)CCC2(CN(C(=O)CN3CC(C)(C)C3)C2)O1 c1(NC(CC)=O)cccc(C(=O)NC2CN(C(=O)CCNC(N)=O)C3CC23)c1 C1(C(=O)NCC2(CN(C(CC(C)C)=O)C)CC2)CC(=O)N(c2ccccc2F)C1 Cc1ncccc1C(=O)NC(CNC(=O)Cc1cc(C(C)C)nn1C)C(C)(C)C N1(C(CC2CC(C)(C)OC2)=O)C2CCC1C1CC1(NC(=O)CNC(N)=O)C2 C1(NC(=O)C(O)Cc2cnc[nH]2)CCC(NC(=O)CCCC2CCCCC2)CC1 N1(C(C(c2ccc(C)o2)C)=O)CCC2OCCN(C(c3nc(C)sc3C)=O)C2C1 C1(C(=O)NCC(C(C)O)C)CCC(C)(C)N(C(C2CC2(C)C)=O)C1 Cc1ccc([N+](=O)[O-])cc1C(=O)NC(Cn1cc(CC(C)(C)C)nn1)CC(C)C C1(NC(c2c(C(C)C)cccc2)=O)CCCCN(Cc2nc(=O)n(C)[nH]2)C1 c1(C(N(C)CC2CCCN(C(C(=O)NC)=O)C2)=O)cc2ccc(Cl)nc2s1 CN(C)NC(=O)CCC(=O)NC1CN(C(C2C(F)(F)C23CC3)=O)C1 c1(OCCC)ccc(C(F)(F)F)cc1C(=O)OCC(=O)C(F)F c1(C(=O)NC2CC(NC(=O)CC3CCC(O)C3)C2)ncc([N+](=O)[O-])cc1Br C(=O)(CC(C)CC(C)(C)C)NC1CC(NC(C2CC(C)(OC)C2)=O)C1 Cc1cc(C(=O)NCC2CCC2NC(c2nc(Cl)ccc2N)=O)cc(C)c1Cl C(C(CCNC(C1CCCN1C(=O)CCN1CCOCC1)=O)OC)OC C(N=c1[nH]c(=NCc2cnsc2)c2c(F)cccc2[nH]1)C12C(F)(F)C1CCCC2 CS(=O)(=O)CCCC(=O)N1CCN(C(=O)C=Cc2ccc(F)nc2)C(CCO)C1 c1(N2Cc3n(cc(C)n3)CC2)nc(=NCC2CC=CC2)[nH]c2c1CCCCCC2 CC#CCCC(=O)N(CC(C)CNC(c1ccccc1CC(=O)OC)=O)C N1(C(C2OCCC(C)C2)=O)CC2(CCCN(C(=O)C(C)(C)CN(C)C)C2)C1 N1(C(C(C)NC(COC)=O)=O)CCN(C(c2cn(Cc3ccco3)nn2)C)CC1 c1(C(=O)NCc2cc(Br)cs2)cc(F)ncc1NCc1ccc(Cl)cc1 C(=O)(CCCC(C)(F)F)N(CC(O)CN(C(=O)Cc1n[nH]c(=N)s1)C)C C#Cc1ccc(OC)c(C(=O)N(CC(O)CN(C(=O)C(C2CC2)OCC)C)C)c1 c1(C(N2CCC(C)(c3nc(C(=O)OC)[nH]n3)C2)=O)cc2cn[nH]c2cc1OC C1(Cc2cn(CCCNC(C(C)n3cccn3)=O)nn2)CN(C(N)=O)CCO1 c1(SC)cc(C)c(C(=O)NC2CC(F)(CNC(=O)C(C)C3CCCC3)C2)s1 c1(C(N2CCC(C(=O)NCCCCC#C)(CO)C2)=O)nccc(C)c1N C1(NC(C(OC)OC)=O)CC2(C1)CN(C(c1cc(F)ccc1C(F)F)=O)C2 Cc1ccc(C(=O)NC(c2cn(C(C)C)nc2CCC2(F)CC(C(=O)O)C2)=O)nn1 N1(C(C2CCN(C(c3cnns3)=O)C23CC3)=O)CCc2ccccc2C1 c1(NC(c2n(CC)ccn2)C)cc(NCc2nc(=N)[nH][nH]2)ncn1 n1(C(C)C)cc(Br)cc1C(=O)N(CC(=O)O)Cc1noc(-c2ccccc2)n1 N1(C(C(c2ccc(C)o2)C)=O)CCN(C)CC1CNC(c1nscc1C)=O C(=O)(CS(=O)(=O)C(C)C)NCc1c(C2CCN(C(C(CC)(C)O)=O)C2)n[nH]c1 N1(C(c2c(CC)nn(C)c2)=O)CCCCC(NC(C2CC(=C3CCC3)C2)=O)C1 N1(C(c2ncc(C#C)cc2C)=O)CCOC2(C1)CN(C(=O)C(CC)SC)C2 N1(C(C=CC(=O)OCC)=O)C2CCC1CC(F)(CNC(=O)C(C1CC1)N(C)C)C2 C1(CNC(C2CC(C(F)(F)F)(OC)C2)=O)CCN(C(=O)C=C(C)C(F)F)CC1C C(CN=c1[nH]c(N2CCNC(=O)CC2)nc2c1CSC2)(c1cccc(C)c1)OC C12(C(=O)NC3CCN(C(C4C(C)(C)C4(F)F)=O)CC3)CC=CCN1CCC2 c1(NC2CCC(CNC(=O)C=Cc3ccncn3)CC2)c(Cl)cc([N+](=O)[O-])cc1Cl C(=O)(C(C)(C)C(N)=O)NC(CC)CN(C(=O)CCc1ncccc1C)C C(=O)(C(CCC1CC1)NC(=O)C(C1CCOCC1)C)NCc1ccc(CC)s1 C12(NC(CNS(CC)(=O)=O)=O)CCCCC1CN(C(=O)Cc1ccc(Cl)nc1)C2 c1(N2CC3C(C(=O)Nc4c(C)cc(Br)nc4)C3C2)[nH]cnc2nc(Br)cc1-2 c1(C(=O)Nc2cccc(OCCC=C)c2)cccc(Cl)c1-n1cncn1 CC1(C)CC(C(N2CCCC2CC(N)=O)=O)CN1C(=O)CC1CCCCC1 C1(C(CNCC(CN(CCCC)CC)(C)C)O)CCC(C)CC1 C1(CNC(C(C2CN(C(=O)C(N)=O)C2)OC)=O)CCC(O)C1 n1(CC)nc(Cc2cc(Cl)cc(Cl)c2F)c2ccccc2c1=O c1(CC)ncnc(N2CC3(CC3)CC2CNC(=O)CCCc2ccsc2)c1F c1(CC)[nH]ccc1C(N1CC(C(C)(C)O)(CN(C(=O)Cc2cnc(C)[nH]2)CC)C1)=O N1(C(C(C(C)C)OCC)=O)CCC2(CC1)CCN(C(c1cnc(C)[nH]1)=O)CC2C C12CCCC(CC1)NC2=O.c1(C(=O)NCCNCC2CC2)cncn1C1CC1 c1(CC(=O)NC2CC3(NC(=O)CC=C(Cl)Cl)COC2C3)n[nH]c2c1CCCC2 Nc1c(Cl)ccc(Br)c1C(=O)NC1(CNC(C2CCC2)=O)CCCCCC1 C1(CC#C)(C(=O)NCC2C3CN(C(c4nonc4N)=O)CC23)CCCCC1 c1(C(N2CCC(NC(C3(C(=O)NC)CCC3)=O)C2)=O)ncccc1Br Cc1cc(Br)cc(C)c1C(=O)OCC(C1C=CC=CC=C1)=O C1(CNC(=O)CC2CCSC2)CN(C(C2(c3ccno3)CC2)=O)CCC1(F)F C1(CC(=O)NCCCC=C)CCCCN1C(=O)Cn1cc(C)cn1 C1(NC(=O)CC2(NC(c3cc(Cl)n[nH]3)=O)CCC2)CCC(F)(F)CC1 c1(C(=O)NCC2C(NC(CCC3N(C)CCC3)=O)CCCC2)ccc(C#N)cn1 c1(C(N2CC(C(=O)NCC3CCN(C(C)C)C3)(COC)C2)=O)cc(O)n(CC)n1 C1(CNC(CCC#C)=O)C2CCCC1N(C(C1CNC(=O)O1)=O)C2 c1(OC)cc(C(N2CCN(C(=O)C(C)(C)C3(C)CC3(F)F)CC2C)=O)nc(C)c1 Cc1cccc([N+](=O)[O-])c1C(=O)NC1CC2CC(C1)N(C(C1(CF)CC1)=O)C2 N1(C(CCCNC(C)=O)=O)CCCC2CN(C(C3CC=C(C(C)C)CC3)=O)CC12 c1(C(N(C(C)CN(C)C(C2(C)CC=CCC2)=O)C)=O)ccc2c(O)n[nH]c2c1 N1(C(c2cnc(OC)nc2C)=O)CCC2C(C1)NC(=O)CCN2C(=O)C(C)SC C(=O)(CCCCC(=O)N(C(C)C(N1CCC(C)(O)CC1C)=O)C)OC CC(C)(C)C(O)C(=O)N1CCCC(CCC(=O)NCC2(C)CCC(O)CC2)C1 c1(C(C)NC(N2CC(C(F)F)C2)=O)nc(C2(OC(C)(C)C)CC2)no1 c1(C(=O)NC2CCOC2C(F)(F)F)cn(-c2cccnc2)nn1 c1(NC2CCC(CC)C2)ncc(C)cc1S(=O)(=O)NCc1cnsc1 N1(C(C2CCC(C)N2C(c2cc(I)cnc2Cl)=O)=O)CCNC2(CCC2)C1 c1(C(=O)NC2(C)CN(C(c3cc(CC)ncn3)=O)C2)cn(C)c2ncccc12 C1(C(=O)NCCCCN(C(C(C)N2CCC2)=O)C)CC12CCC1(CC1)CC2 c1(SCC(C(=O)NCCSC)N2CCCC2NC(C)=O)ccc(F)cc1 N12CCCC(C1)NC2=O.C1(O)(COCC)CCN(CCCC2C3CCCCC23)C1 c1(C(C)NC(CNC(=O)NC(c2scc(CC)n2)CC)=O)ccc(Br)cc1 C=CCCC(C)(C)C(=O)N(CC(C)NC(=O)C(c1ccccc1F)C)C C1(C(=O)NC(C)C(C)NC(C23CC(c4ccccc4)(C2)C3)=O)CCCN1C=O CC1CCCC1NC(c1n[nH]cc1CNC(=O)CCOC1CCCC1)=O C1(C(N2CCC(CCNC(C34CCC(CC3F)C4)=O)C2)=O)CC2(C1)CC2(F)F CC1CC(C(=O)NCC2(C(=O)NC3(CF)CC3)CC2)=NO1 Cc1ccc(CCC(=O)NCC2(NC(=O)C(C)n3ccnc3)CC2)cc1C C1(CNC(C2(C)CCC2)=O)CN(C(=O)CCCc2ccccc2)CCC12CCC2 Nc1c(F)ccc(F)c1C(N1CCC2CC2(NC(c2cnc(O)s2)=O)CC1)=O CC(O)CCCCCC(=O)NCCC1CCCN(C(c2ccc(O)nc2)=O)C1 C12(CNC(CCOCCNC(c3ccn(C)n3)=O)=O)CCC(CC1)CC2 c1(CNC(C2C(NCc3cc(C)oc3C)C2)=O)ccc(Cl)c(Cl)c1 N1(C(=O)Cn2cnnc2O)CCN(C(=O)C2=CCCC2)C(C2CC2)C1 C=CC(C)(C)C(=O)NC(C)CCNC(=O)CC1CCC(C2CC2)O1 C12(CNC(C3CCCN(C(C(CC)C)=O)C3)=O)CCC(CC1)CN2C(C)=O N1(C(C(CSC)C)=O)CCCC2(CCN(C(c3cc([N+](=O)[O-])c[nH]3)=O)CC2)C1 N1(C(c2ccncc2)C(=O)NC)CCN(CC(C)O)CC1 C(C(COC)CC(=O)NCCC1(C)CCN(C(C2CC(C3CC3)=NO2)=O)C1)OC c1(NC(C2(O)CCN(Cc3c(F)ccc(C)c3)C2)=O)ccc(S(N)(=O)=O)cc1 C(N=c1[nH]c(Cl)ncc1F)C1CC(NC(C2CCC(CC)O2)=O)C1 C=CC(C)CC(=O)NCc1cccc(C(=O)N(C)CC2(OCC)CCC2)n1 C1(NC(c2cc(C3CCCC3)no2)=O)CCN(C(=O)Cc2ccsc2)C1 N1(C(C(C)SC(C)C)=O)CCC(NC(=O)C(C)(C)c2ccccn2)C(C)(C)C1 N1(C(C(=O)NCCC2CC(C)(C)C2)=O)CCCSCC1C1CCC1 c1(OC)c(C(=O)NCC(C2CC2)N(C(=O)CCC2CC2C)C)cnn1C c1(NC(C2C3(CN(c4nnc(C)s4)C3)C2)=O)ccc([N+](=O)[O-])cc1S(C)(=O)=O CC1CC(NC(C2(CCF)CC2)=O)CCN1C(=O)CCN1CCCS1(=O)=O CC1=NNC(=O)C1CC(=O)NCc1cn(CC(=O)N(C)CCn2cncn2)nn1 c1(CCC(=O)N(C)CCN(C(=O)CC=CC(C)(C)C)C)cncc(O)c1 C(=O)(C(CC(F)F)NC(=O)CCC(C)(C)F)NCCCN(OC)C C(=O)(CC(C)C(=O)N1CCN(C(=O)C=Cc2scnc2C)CC1C(C)(C)C)OC c1(CC)noc(CC)c1CC(=O)NCC1C2CN(C(=O)CN3CCOC3=O)CC12 N1(C(C2(NC(CC3CC(SC)C3)=O)CC(F)(F)C2)=O)CCCC(C=C)C1 C=CC1OCCC1C(=O)NCCC1(NC(=O)C(n2nccc2C)C)CCC1 N1(C(CC2COCC(C)O2)=O)CC(C2CC2)(C(=O)NCC2CCN(C)C2)C1 CC1CC(NC(C2C=CCC2)=O)CCN1CC(O)CC1OCCCO1 C#CC1(O)CCCN(C(=O)CNCC2CC(OC)(OC)C2)C1 C1(CCC)CN(C(c2nc(C)oc2C)=O)CCN1C(=O)C1=CCCC1C c1(C(=O)NC2C3CN(C(CC(CC)O)=O)CC32)cccc2c1CCCO2 c1(NC(C)CCS(C)(=O)=O)ncnc2c1cnn2CCC#N C(=O)(CCCC(=O)NCC1C(OC)CCN1C(C1CC2C(C1)C2(C)C)=O)OC C(CCCCCNC(c1cscc1Cl)=O)NC(=O)CC1CC1C1CCCC1 CCC(C(C)C)C(C(=O)NCCCOC)N(C(CC(C)C)C(N)=O)C CC1(C(=O)NCC2COCCN2C(=O)Cc2nc([N+](=O)[O-])n[nH]2)CCC(=O)NC1 C1(C(c2ccccc2)C)C(=O)NCCN1C(c1ccc(-c2cnn[nH]2)cc1)=O C1(C(=O)NC(CC#C)CO)CN(C(C2(Cl)CC2(F)F)=O)CCO1 c1(C(N2CCC(C)SCC2)=O)cc(O)nc2c1CN(C(=O)CCCF)CC2 N1(C(c2n(C)cnc2)=O)CC(CNC(=O)C(O)CC(F)F)CC12CCC2 N1(C(Cc2ccc(C#C)cc2)=O)C2CCC1C(C)C(NC(C1(CCO)CC1)=O)C2 C1(CNC(C(=C)CC)=O)CCCCCCCCC1 Cc1ncc2n1CCN(C(=O)CC1CCN(C(C3CNC(=O)C3)=O)C1)C2 CCCC(CCCNC(c1cc(Cl)n(C)n1)=O)NC(=O)C1=CCOC1 c1(CC)ccc(O)c(C(=O)NCCC2(CNC(C3CCCC4CC34)=O)CC2)c1 C1(C)(COC)CC(NC(c2csc(Cl)n2)=O)CN1C(c1cn(C)nc1OC)=O N1(C(C=CCN(C)C(C2CC3C(C2)C3(F)F)=O)=O)CC(S(N)(=O)=O)C1 Cc1ccc(C(=O)NCCCNC(=O)C(O)C2CCC2)o1 C12(C(N3C(C)CC(CC(=O)NCCOCCN(C)C)C3)=O)CCCN1CCC2 c1(C(N(C2CC(NC(c3c(O)cccc3F)=O)C2)C)=O)ccc([N+](=O)[O-])s1 Cc1cc(NC2(CNC(c3ncn4ccccc34)=O)CCC2)n2ncc(C)c2n1 C=CCC(CC=C)NC(=O)C(CO)NC(=O)C(C)OCC C1(NC(C(C(C)C)F)=O)CN(C(c2ncc(C(F)(F)F)s2)=O)CC1(C)C N1(C(c2c(C)coc2)=O)CCC(CO)(CNC(=O)C(O)C2CCCC2)C1 c1(COC)n[nH]c(C(C(=O)NC2CCC2)N(C)CCC2CCC2)n1 O=S(=O)(c1ccc(Br)cc1)N1CCCCC1CN1CCC(Cl)=C(Cl)C1 c1(N(C(c2cc(F)ccn2)C(=O)NCCC2(C)CC2)C)cc(Br)cc([N+](=O)[O-])c1 N1(C(CC2N(C(CC(C)CN(C)C)=O)CCOC2)=O)CCC2(CC1)CC2C#N C(=O)(CS(=O)(=O)CC(=O)NC1CCCN(C(=O)C(C)CC(C)C)CC1)OC Cc1ncc(N)cc1C(=O)NCC(C)(O)CNC(=O)CC(C)n1cccn1 Cc1nc2ccc(C(=O)NC(C)CNC(C3CCC(C)CC3)=O)cc2[nH]1 N1(C(C2CC(C)(C)OC2)=O)CCCC(C2(NC(=O)C#CC3CCCCO3)CC2)C1 C(C)(N=c1[nH]c(=NCC2COc3cscc3O2)[nH]c2c1COC2)c1c(C)ncs1 Cc1cc(C(=O)NCC2CCCC(NC(c3ocnc3C3CC3)=O)C2)cc(O)c1 c1(C(N(C(CNC(c2c(SC)csc2)=O)C)C)=O)cnn2ccc(C)cc12 C(=O)(CS(=O)(=O)C12CC(C1)C2)NCC(CNC(CC(CC(C)C)C)=O)C CCCC(C(=O)N(CCC(=O)NC1(C2CCCCC2)CC1)OC)N(C)C C1(CC(=O)NCC(=C)CCNC(=O)Cn2ccccc2=O)C(=O)N(C)N=C1C C1(C)(NC(CC(CC)OC)=O)CCC(NC(=O)COCC2(F)CC2)CC1 C1(N(C)C)CCC(C(=O)NCC(CNC(=O)C(c2cccc(Cl)c2)O)CO)CC1 c1(C(=O)NC23C(CN(C(C4N(S(C)(=O)=O)CC4)=O)C2)C3)cc(N)ccc1Cl c1(C(N(C2CCC(NC(=O)C3=CCC3)CC2)CC)=O)ccc2c(c1)NC(=O)C2=O c1(C(=O)NCCSCc2cn(CC3COCCO3)nn2)[nH]nc2ncnc(O)c12 N1(C(c2n(CC)nc(C)c2)=O)CC2CCCCC2(NC(=O)C(C)n2ccnc2)C1 C(C(C)(C(F)(F)F)c1ccccc1)NC1CCN(C(=O)NC(C)C)CC1 C1(CC=C)(NC(=O)CN(C(=O)C(C2CCCCC2)O)CCOC)CCOC1 c1(CNC(c2c(CCNC(C3CC(N(C)C)C3)=O)n[nH]c2)=O)ncc[nH]c1=O C1(COC)CCCCC1C(=O)N(CC(O)CN(CC(O)Cc1cccc(F)c1)C)C CC1(CNC(=O)CC2CCC(=O)N2)CCCN(C(C23CCC(C2)C3)=O)C1 C=C(C)CCCC(=O)N1CC2(CC2)CC1C(N1CC(C)CC(O)C1)=O Cc1ncc(C(=O)NCC(C)CN(C)C(C2(CCN(C)C)CC2)=O)o1 C(=O)(CC(C)(O)C(F)(F)F)NC1C2CCN(C(c3cccc(C)c3N)=O)C2C1 C1(C(=O)NC(CC)C(N)=O)CC(C)CCN1C(=O)CC1OCCO1 C1(C(=O)NC2CN(C(C3=C(C)CCC3)=O)CC2O)COc2ccccc2O1 c1(NC(c2ccc(CNC(C(CC=C)CC)=O)o2)=O)cc(C)c(F)cc1C N1(C(C=NOC)=O)CCN(C(=O)C(C)CO)CCC1C N1(C(CCCCNC(N)=O)=O)CC2ON=C(CNC(c3coc(Cl)n3)=O)C2C1 C1(NC(C2C(C)(C)C2C#N)=O)CC(C(N2CCC3(CC2)N=N3)=O)C12CCC2 c1(C(=O)NC2C(NC(=O)Cc3ccccc3)COC2)c(F)ccc(F)c1Br Cc1nn(C)c2sc(C(N3CCC(NC(=O)C(C)C(F)(F)F)C3)=O)cc12 N1(C(C2(C#C)CCOCC2)=O)CCN(N2CC3CCC3(CO)C2)CC1 C(C1=CCCN(C(C2C3CC4C(C3)C24)=O)C1)NC(CCOCCN(C)C)=O C1(NC(C2ON=C(C)C2)=O)C2CC3CN(C(=O)CCP(C)(C)=O)C1C3C2 n1(CCC)nc(C)cc1C(=O)NC1CC(NC(=O)C(C)C(C)O)C(O)C1 c1(-c2cn(CCN(C(=O)C=CC3CCCO3)CC)nn2)ccc(Br)cc1OC c1(OCCC(=O)NC2CN(C(C3(C=C)CC3)=O)C3C2C3)cc(F)cc(F)c1 N1(C(C2(C(=O)OC)CC2)=O)CCC2(CC1)CC(NC(=O)CC1CCOC1)CO2 CC1CN(C(=O)CN2CCCC2C)CC1NC(C1CC1C#N)=O CC1CN(C(c2sccc2CC#N)=O)CCN1C(=O)CCCC(=O)NC1CC1 N1(C(=O)Cc2csc(Br)c2)CCN(C(=O)CC2(O)CCCOC2)CC(O)C1 c1(C(=O)NC2C3CN(Cc4cc(C)c(Cl)c(C)c4)CC32)oc2ccccc2c1C N1(C(=O)OC(C)(C)C)CC2OCCN(C(C3CN(CC(F)(F)F)C3)=O)C2C1 C1(OC)(CNC(=O)C=CSCc2ccco2)CCN(C(C2CC2C#N)=O)C1 S(=O)(=O)(CCC(=O)NCCOCCN(C(=O)Cc1ccn(CC(C)C)n1)C)NC Cc1n[nH]cc1CC(=O)NC1(C(=O)NCCC2CCC3CC23)CC1(C)C C(C)(C)(CCC(=O)NC1CN(C(=O)C(F)(F)c2cccnc2)CC12CC2)N(C)C C12CCC(CC1)CN(CC(O)CO)C2=O.C1(C=O)CC1CC(C)C.CO C1(NC(=O)CSc2ccccc2)CCN(C(C2(O)CCSC2)=O)CCC1(F)F c1(CCC)ccc(-n2nc(CCCOc3ccccc3)nc2C2CCCO2)cc1 C1(C(=O)NC2CC(CN(C)C)C2)CN(C(c2cocc2C(N)=O)=O)CCO1 c1(C(N2CC(C)C(NC(C3CCC(C)=C(C)C3)=O)C2)=O)cnc(O)c(Cl)c1 CN1CCCC(C(=O)NC(C2CCCCC2)CNC(C2CCCC2O)=O)C1 N1(C(C(c2ccc(OC)cc2)OC)=O)CC2CC(NC(=O)CSC(F)(F)F)C(C2)C1 Cn1cc(S(=O)(=O)NC(c2ccccc2)Cc2nn[nH]n2)cc1C(N)=O N1(C(C2(CC)CCC2)=O)CCC2(CCC(NC(=O)CN(CC(=O)NC(C)C)C)C2)C1 C(=O)(C(N=[N+]=[N-])C(C)C)NC1(C(=O)NCCCn2c(C)nnc2)CCOCC1 Cc1[nH]nc2c1CN(C(=O)CC1CN(C(c3cccc(Br)c3CBr)=O)C1)CC2 c1(NC(=O)C(=O)N(C(c2ccc(Br)cc2)CC)CCC)ccc(OCC)cc1 C1(CCOC)(NC(c2ccc(CC)nc2)=O)CCN(C(C2(C)CCOC2)=O)CC1 c1(N2CCC(NC(C3CC3F)=O)(CF)C2)nc(C(F)F)nc2ccccc12 c1(NCC(CCOC)NC(=O)OC(C)(C)C)c(C)nn2c1CCCC2C Cc1c(O)c(=O)ccn1CC(=O)NCCOCCN(C)C(C1CC=CCC1)=O CC1CN(C(=O)CCOC2COC2)CC1CC(=O)NCC1CC(F)(CO)C1 Cc1ccc(C(=O)NCCC2(C)CCN(C(=O)C(C)C(F)(F)F)C2)n(C)c1=O c1(CC(=O)NC(CNC(c2n(C)cnc2)=O)CO)coc2cc(F)ccc12 N1(C(C2C(NC(c3c(C)nccc3)=O)CCCCC2)=O)CC(C)c2ncccc21 CC(C)C(C(=O)N(C(C)CNC(=O)CCCn1ccnn1)C)NS(N)(=O)=O N(C(=NCC#Cc1ccccc1)NC(c1ccc(SC)cc1)C)CCC(=O)NC C1(NC(c2cn3c(Cl)cccc3n2)=O)CC(N=c2nc[nH]c3[nH]c(Br)cc23)C1 CC1CN(C(=O)C(C)(C)N=[N+]=[N-])CC(C(=O)N(C2CCCN(C)C2)C)O1 N1(C(Cc2cccc(C)c2F)=O)CC2CCN(C(c3ncccc3Cl)=O)C2C1 N1(C(C(C)OCC(C)C)=O)CC2(CC(NC(C3CCCC34CC4)=O)C2)C1 c1(C(=O)NC2CC(F)(CNC(c3sccc3Cl)=O)C2)cc(Br)ccn1 c1(C(=O)NC(CNC(c2sc(C)c(Br)n2)=O)C)cc(C(C)C)cnc1O N1(C(c2ncn(C(C)C)n2)=O)CC2(C(=O)NCC3CCCC(C)(C)C3)CC1CO2 c1(C(C)C)cc(C(=O)NCC(O)CNC(=O)C(F)(F)CC2CCCO2)nn1C C(CNC(=O)Cn1cc(Cl)cn1)(CCC)NC(C(C)=C(CC)C)=O c1(OC)ccc(CN(CC(CC2CCCC2)CN)C)cc1OC(F)F c1(C(N2CCC(C(C)NC(COCC=C)=O)C2)=O)cccnc1N(C)C N1(C(C2C(=C)C2)=O)CC(NC(c2cc(-c3ccc(Cl)cc3)[nH]n2)=O)CC(C)(C)C1 N1(C(C(CCSC)O)=O)CC(CNC(=O)CCC(=O)N(C)C)CC12CCOCC2 CCCC(CC)CCC(=O)N1CCC(NC(C2(CNC(C)=O)CCC2)=O)C1 N1(CC)CCN(CCC(=O)NC2(CNC(c3cccc(COC)c3)=O)CC2)CC1 c1(C(=O)NC2CC(F)(CNC(COCC#C)=O)C2)cc(C(N)=O)ccc1C C#Cc1ccc(C(=O)NC(C)CN(C(=O)CCOc2c(F)cccc2Cl)C)nc1 c1(NC(CCOC)C2CCC2)ccc(F)cc1OCCCSC Cc1cc(=NC(=O)C2CCN(C(=O)C(C)S(C)(=O)=O)CC2C)[nH]n1C c1(CNC(=O)CC2C=CCC2)ccccc1CNC(c1cnccn1)=O C1(CNC(=O)C=CC2CC2)CC2CCC(C1)N2C(=O)Cc1ccccc1O C1(C(=O)NCC(C)N(C)C(c2[nH]cc3c2CCCC3)=O)CC2OC(C)(C)OC2C1 Cc1nc(C)c(C(=O)NCC2COCC2NC(C2CCCN(C)C2)=O)o1 N1(C(c2cn(CCCC)nc2C)=O)CCC(NC(c2cc[nH]c2)=O)C(CC)C1 C(=O)(C(F)(CNC(=O)C(C)CC(N)=O)C(C)C)NC(c1nc[nH]n1)CC c1(C(N2CCN(C(C(COC)C)=O)CC2CCO)=O)ccc2ncccc2c1Cl c1(C(=O)NC2C(NC(c3c(C)c(O)ccc3)=O)CC2)nc(C)n2ccccc12 CCC(C(=O)NC1(CCCNC(=O)Cc2cc[nH]n2)CC1)C1CCOCC1 c1(C(C(N2C(CNC(c3c(C)c[nH]n3)=O)CCCC2)=O)=O)cc(F)c(F)cc1F C1(C(=O)Nc2c(C)noc2C2CC2)CC(C)(C)CCN1C(=O)C=CCl.N1CCCC1 N(C1CCc2cccc3cccc1c23)C(=O)NCC1CCC(O)C1 c1(NC(c2c(C)c(Cl)ccc2)=O)nc2ccc(O)nc2s1 C1(C(=O)NC2C(NC(c3n(C=C)ncc3)=O)CCCC2)CC2(C1)CC(C(=O)OC)C2 C(CCN=C(NCCc1cnc(C)s1)N1CCOC(C2CCCO2)C1)OCC Cc1nn(C)c(C)c1C(=O)NCC1C(C(=O)NC2(C3CC3)CC2)C1 C1(NC(=O)Cc2ncccn2)CN(C(C2CCCS2)=O)CC12COC2 C1(C)(C(N2CC3C(NC(C(=Cc4ccco4)C)=O)(C3)C2)=O)CCCCC1(F)F C#Cc1cc(C(=O)NC(C2(O)CCN(C(=O)COc3ccsn3)C2)C)cc(F)c1 Cc1ccc(C(N2CCN(C(c3ns[nH]c3=O)=O)CC2C(C)C)=O)c(O)c1C C(=O)(C1CCc2ccccc21)NC1CCCN(C(C2CN(C)C(=O)C2)=O)CCC1 S(=O)(=O)(c1cccc(F)c1)Nc1c(CNC(=O)OC(C)(C)C)nc2n1CCCC2 c1(C(=O)NC2C(CNC(C3C(OC(C)(C)C)C3)=O)CCC2)c(F)cc(Cl)cc1F N1(C(C=CC(C)(C)NC(c2n[nH]cc2Cl)=O)=O)CCCNC(=O)CC1 C(=O)(C1=NOC(C)(C)C1)NCCC1(NC(CC2CCCC(C)C2)=O)CCC1 N1(c2snc(CCC)n2)CCC(NC(=O)CC(=O)NC)C(C)(C)C1 n1(C(CC)C)nc(C(N2CCC(CNC(c3c[nH]cc3C3CC3)=O)C2)=O)cc1C N1(C(C(C2CCCC2)OC)=O)CC(NC(c2coc(C)c2)=O)C2(CCC2)C1 c1(C(N2CC3CC2CN3C(C2CC(F)(CO)C2)=O)=O)ccc2ncnn2c1 c1(CNC(=NC)NCC(n2cccn2)C)cc(C2CC2)[nH]c(=N)n1 C(N=c1cc(Cl)nc[nH]1)C1C(NC(C(c2cccnc2)C)=O)CCC1 C1(n2cc(-c3c(OCCOC)cccc3)nn2)CON(C(=O)c2cncnc2C)C1 c1(OC)cccc(C(=O)NC2CN(C(=O)CC3CC(C)=NO3)CC2O)c1C c1(C(N2CCN(C(=O)Cc3cncs3)CC2C2CCC2)=O)cc2ccncc2o1 C1(C(=O)NC2C(NC(CC(CC)c3ccccc3)=O)COC2)CCS(=O)(=O)CC1 N1(c2c(C)c(NCc3ccnc(Cl)c3)ncn2)CC2CCC1CN2CCO Cn1cc(C(N2CC(NC(=O)Cc3ccccc3CO)C2)=O)c(O)nc1=O c1(C(=O)NC2C(SC)CN(C(C3CC34CCC4)=O)C2)ccc(Cl)c2ccccc12 S(=O)(=O)(c1cc(C)c(F)c(C)c1)NC1(CC(=O)OCC)CCOC1 Cc1csc(C(C(F)(F)F)NC(=O)CCC2CC(C(=O)O)C2)n1 c1(C(c2n(CCCC)nnn2)NCC2C=CCOC2)ccc(Cl)cc1OC C1(N(C(=O)C(Cl)=CCl)C)CCCCN(C(C2(CO)CC2(F)F)=O)C1 C(=O)(CC1=NNC(=O)C1)N1CC(NC(CCCOCC)=O)C(F)CC1 CCCCC(CNC(=O)Cc1c[nH]nc1C)NC(C1CCC(=O)N1C1CC1)=O C(=O)(CC(C)CN(C)C)NCC(CCOC)NC(c1cnc[nH]c1=N)=O C1(F)(C(=O)NCCc2cnc(C)[nH]2)CCN(C(c2sncc2C)=O)CC1 C1(C(N(CCNC(=O)C(C)(C)C#N)CC)=O)CC(c2cccc(F)c2)=NO1 c1(CC)ccc(CC(=O)NC(C)C(C)NC(c2csc(C(=O)OC)c2)=O)cc1 N1(C(CCNC(CCC)=O)=O)CCC(NC(=O)Cc2nc(C)no2)C(CO)CC1 C1(C(F)F)(CNC(c2cc(C)[nH]n2)=O)CCN(C(=O)Cc2ccccn2)C1 C1(C(=O)NC(C2CN(C(C3CCC(NC(CC)=O)C3)=O)C2)C)C2(CC2)C12CC2 C(=O)(C(C)C(O)CCCC)N1C(C(=O)NC(CC#C)CCOC)CCC12CC2 CC1CCNC(=O)C1NC(c1cc(CNC(c2cc(Cl)ns2)=O)ccn1)=O N1(C(c2cccc(OC)c2O)=O)CCCC2(CC(NC(c3sccc3Cl)=O)C2)C1 c1(C(c2nnnn2C2COC2)Nc2ncn(C)n2)c(Br)ccc2c1OCO2 c1(C(N(CC(C)(C)NC(C(COCC)C)=O)C)=O)cc2c(C)cc(Cl)cc2[nH]1 C(=O)(CCN1C(=O)COc2ccccc21)N1C(CC(C)C)CC1 C1(COC)CC(O)CN1C(c1cc(CNC(C2CCC(=O)NC2)=O)no1)=O CCC(C)CC(=O)C(=O)NC(C(N1CCCCC(C)(F)C1)=O)C1(O)CCC1 C(=O)(CC(CC(C)C)NC(=O)Cc1cccnc1C)NCC(CCC)C C1(C(N(CCCO)CC)=O)CC12CCN(C(=O)CNC(c1ccccn1)=O)C2 Cc1coc2c(C(=O)NCC(C)CNC(c3cnn(CCF)c3)=O)cccc12 C#CC1CC2CCC1N(C(=O)CC1CC1CNC(=O)Cc1cc(C)[nH]n1)C2 C1(NC(=O)C=CC=C(Cl)Cl)CC2CC(C1)N(c1cc(C3CCCC3)ncn1)C2 c1(C(C2CC2)NC2C(C(C)C(=O)OC(C)(C)C)CCC2)ccc(F)c(Cl)c1 C(=O)(CCCCCCCCCO)NCC(C)N(C(C1(C)COC(=O)C1)=O)CC C(C(C)(C)CCC#N)(c1nnnn1CC(F)F)N(CCN(CC)CC)CC N1(C(C(CC#C)O)=O)CCN(C(c2ccc(Cl)c(OC)c2F)=O)C2COCC12 c1(C(N2CC(NC(C(C(C)(C)O)F)=O)CC23CCC3)=O)cc2c(Cl)cccc2s1 C(=O)(C(F)(CC)C(=O)OC)NC(CC)CNC(C1OCCC1(C)C)=O c1(C(C)=O)cncc(C(=O)NCC2(CNC(c3sc(N(C)C)nc3Cl)=O)CC2)c1 C(C(=O)NC(C)C(C)F)(C(C)(C)O)NC(c1cnc(C)s1)=O N1(C(CC(CC)(C)C)=O)CCC2C(C1)CN2C(=O)CCc1cc(C)nn1C C1(CCC)CCC(C(=O)NCC=CCNC(=O)C(n2nccc2C)C)CC1 C(=O)(C1=CSCCO1)NCC1N(C(c2cc(C3(C)CC3)on2)=O)CC1 C(N=c1[nH]cnc2ccsc12)C1(F)CCN(C(C2CC23CC3)=O)CC1 c1(C(=O)NC2CCC(NC(C(C)SCCCC)=O)C2)oc2cc(Cl)ccc2c1C CC1(C(N2CCC(C(F)(F)CO)C2)=O)CC(c2ccccc2)=NO1 Cc1cc(N2CCC(CC(C)NC(c3sccc3N(C)C)=O)CC2)nc(C)n1 c1(-n2ccc(C)c2)ccc(C(N2CC(NC(C3(C)CC(C)=NO3)=O)C2)=O)cc1 N1(C(C2C3CCCC23)=O)CCCN(C(c2ccoc2C2CC2)=O)C(CO)C1 C1(C(=O)NCc2cc(C)no2)CC(F)CN(C(=O)Cn2ccc(C)n2)C1 N1(C(C2N(C(CC(C)C(F)(F)F)=O)CCCC2)=O)CCOC2(CCCC2)C1 c1(OC)cccc(C(N2CC3CCC(C2)N3C(=O)CP(C)(C)=O)=O)c1[N+](=O)[O-] c1(OC)cccc(C(=O)NCC(C(C)C(C)C)NC(c2c[nH]nc2OC)=O)c1F c1(C(N2CCC(O)(C(C)NC(COCC#C)=O)C2)=O)cc(CC)nnc1C C=C(Cl)CCC(=O)NC1CCOCC1C(=O)NCCn1ccnc1CC c1(CC)ccc(F)cc1C(N1CC(OC)CC1CNC(c1nocc1C)=O)=O CON1CC(C(N2CCN(CC(N3CCOC(CF)C3)=O)CC2)=O)CC1=O c1(SC)ccc(CCC(=O)N(C(C)(C)CO)CC2(C)CC2(Cl)Cl)cc1 C1(C#N)(C(=O)NCCN(C)C(c2cn(CC(F)(F)F)cn2)=O)CCCO1 C(=O)(C1=CC(O)C(NC(=O)C2=NOC(C)C2)C1)NC(c1nc(C)[nH]n1)CO c1(C(N(C)Cc2cnc(-c3cccnc3C#N)cn2)=O)cccc2ccccc12 c1(C(=O)NC2C(CNC(c3c(C)coc3)=O)COC2)sc2ccc(C)cc2c1C Cc1ccc(NC(=O)CN2CCC(C(C)NC(=O)CCSC(F)(F)F)CC2)cc1 C=CC1CN(C(=O)CCCF)CC1NC(C1CC(CC)=NO1)=O C1(NC(C(C)=C(C)C)=O)CN(C(=O)CCC(F)F)CC1C1CC1 C(=O)(C(C)(C)C(O)C(C)C)NC1(C)CN(C(c2c(OCC=C)cccn2)=O)C1 N1(C(c2[nH]cc(COC)c2)=O)CCC2(CCCN(C(=O)CN3CCC3C)C2)C1 C(=O)(CCCCCC(C)O)NC1(C2CN(C(c3c(NC)cncc3)=O)C2)CC1 C(C(N=c1[nH]nc(C2CC2)o1)C1CC1)NC(C(=O)Nc1ccc(C)c(C)c1)=O c1(OC)ncc(CN2CCCC2CCC(=O)NCc2cccnc2)cc1Cl C1(NC(c2c(SC)scc2)=O)C=CCN(C(=O)CCOC(C)CC(C)C)C1 C1(CNC(C2COc3ccccc3O2)=O)CC(N=c2c(Cl)c[nH]cc2[N+](=O)[O-])C1 n1(CC(=O)NCC2(COC)CN(C(=O)C=CC3CCC3)C2)ccccc1=O CCC(C)(C)CC(=O)NCC12CCC(CC1)N2c1nc(C(C)C)ns1 C(N=c1ccc(Br)c(S(=O)(=O)N2CCCC(C)(C)C2)[nH]1)C1CCCN(C(C)=O)C1 N1(C(CC2(C(=C)F)CCC2)=O)CC2(CCC2NC(=O)C(Br)=C(C)C)C1 C1(C(N2CC(CNC(c3c(=N)[nH]cnc3)=O)OCC2)=O)CCC12CCOCC2 C=CCC(C)(C)CC(=O)NCC1CCC(CNC(c2cc(F)ccc2F)=O)CC1 N1(C(C(C(=O)OC)OC)=O)CC2CC(C(N3CCN(C)C(=O)C3C)=O)C(C2)C1 c1(C(N2C(C(=O)Nc3cccc(C)c3O)CCCC2)=O)cc(Cl)c(Cl)c(Cl)c1 C1(OC)CC(C(=O)NC(CNC(C2CN(CC(F)(F)F)C2)=O)CO)CC1OC Cn1nc2ccccc2c1CN=c1ccnc(NCCN2CCCOCC2)[nH]1 C(=O)(C1=NOC(CN)C1)N(C(CNC(=O)Cc1cccc(F)c1Cl)C1CC1)C N1(C(c2ccc(OC)nn2)=O)CCC2CN(Cc3ccccc3C)CC12 CCC(CC)CCCC(=O)NCCCC(C)NC(=O)CC1(O)CCCOC1 N1(CCCNC(C(C)c2ccsc2)=O)CCC(NC(=O)CCc2cnccn2)C1 c1(C(=O)NCCCCCNC(C2CC3CCCC3C2)=O)ccc2ncccc2n1 c1(CC)ccc(C(=O)NC(CSC)C(=O)N(C(C)C(C)C)C2CC2)[nH]1 N1(C(C2(C=C)CCCCC2)=O)CCC2CCCN(C(=O)COCC(F)(F)F)C2C1 C(=O)(CC(=O)N1CCC(C(F)C(=O)NCCNC(N)=O)C1)OC N1(C(C(C)OCCCC)=O)CCCCCCC1C(=O)NCc1csc(C2CC2)n1 C1(C)(CNC(c2ccc(OC)cc2)=O)COCCN(C(=O)CC(O)C(C)C)C1 C1(C)(CNC(c2nccc(C)c2)=O)CCN(C(c2coc(Br)n2)=O)CC1 CC1(C)CCCC(CC(N2CC(NC(=O)CNC(N)=O)C(F)C2)=O)O1 c1(C(N2C(CNC(=O)COc3ccsn3)CC(OC)C2)=O)cnc2ncccn12 N1(C(CCc2n[nH]c(=N)s2)=O)CCCC(Oc2ccccn2)C1 N1(Cc2onc(CCOC)n2)CCC2CCC(C1)N2C(c1ccoc1Cl)=O N1(C(CN(C(=O)C(CC)C(F)(F)F)CCC)=O)CC(C)CCCC1C Cc1ccc2ncccc2c1C(=O)NC1CCC1CNC(=O)CCC(C)C#N CN1CCN(C(=O)C(O)C(F)(F)F)CC1CNC(c1scnc1Cl)=O c1(C(C)C)ccc(C(=O)NCC2COC(CNC(c3cn[nH]c3)=O)C2)o1 c1(CC(=O)NCC2CC(OC)CN2C(=O)C2=CCCS2)ccc(F)c(Cl)c1 c1(C(=O)NCC(CC)(C)NC(C2CC3C=CC2C3)=O)n[nH]c2nccc(Cl)c12 Cc1cc2c(C(=O)N(CCCN(C)C(c3ccnc(F)c3N)=O)C)cccc2o1 CCC(C)(CCNC(C1CC2(CC2)CO1)=O)NC(=O)CCC1CCC1 N1(C(c2cc(C)c(C)o2)=O)CC2CCC1CN(C(c1c(C(C)C)cnn1C)=O)C2 c1(SCc2ccc(-c3n(C(CC)(C)C(=O)O)ccn3)cc2)ccc(C)c(N)c1 N1(C(c2ccc(C(C)C)s2)=O)CC2CCC1C(NC(C1(Br)CC1)=O)C2 C1(C(=O)NC2(C)C(C)CCC2)CCCN1NC(=O)C1Cc2ccccc21 Cc1c(F)ccc(C(=O)NCC2CC(O)CN2C(c2ccc(Cl)c(N)c2)=O)c1F C1(OC)CN(C(=O)CC(F)(F)CC)C(C)(CNC(c2cc[n+]([O-])cc2)=O)C1 N1(C(CC(=C)C)=O)CC(CNC(c2noc(C3CC3)c2C)=O)OC2(CCC2)C1 c1(C(c2nnnn2CCCC2CC2)NCC(C)(C)SC)n[nH]c(C)c1C N1(c2ncc(CC)cn2)CCN(C(=O)CC=C(C)C)CC1C(F)(F)F c1(CNC(C2(F)CN(C(CC(C)C)=O)C2)=O)cc2ccc(C#N)cc2[nH]1 n1(CC(N2CCN(C(=O)Cn3nccn3)C(CCO)C2)=O)ccc2ccccc12 c1(C(=O)NCC2N(C(CCCC#C)=O)CC(OC)C2)c(C)ccc2ncccc12 N1(C(=O)OC(C)(C)C)CCOCC(F)(CNC(=O)Cc2nc([N+](=O)[O-])n[nH]2)C1 C(=O)(CS(=O)CCC(F)(F)F)N1CC(CC(C)NC(CSCC)=O)C1 N1(C(C2C(OCC)C2)=O)CCOC(C)(CNC(c2cnc(C)cc2C)=O)C1 c1(CNC(C(C)CC2CCC2)=O)ccccc1CNC(=O)C(C)OC1CCCC1 N1(C(COCCCC#C)=O)CCCC(N(C(=O)C(N2CCCCCC2)C)CC)C1 Cc1nc(C(C)C)oc1C(=O)NC(c1cccnc1)CNC(=O)CC(C)C C(=O)(C(C)(C)Cc1nn[nH]n1)N(C(C1(C)CC1)C)C N1(C(C2N(C(C)=O)CCC2)=O)CCN(CCNC(C2(CC(F)F)CCC2)=O)CC1 Cc1cc(C(c2nc(-c3ccn(C)n3)nn2C2CCC2)C)ccc1Br C(=O)(C#CC1(C)CC1)NCCCN(C(=O)C(C1CCC(C(C)(C)C)CC1)O)C CC1C2CC(C2NC(=O)C=Cc2cncs2)N1C(=O)CCC(C)(F)F N1(C(C=C(CCC)C)=O)CCC(NC(c2cc(C)ccc2OC(F)F)=O)C(O)C1 C1(C(N2CC(F)(CNC(C3CC=C(C)CC3)=O)C2)=O)Cc2ccncc2N1 N1(C(Cc2cccc(SC)c2)=O)CCC2(CC2NC(c2csnn2)=O)C1 n1(CC(=O)NC2C3CN(C(c4c(N)cccc4F)=O)CC32)ccc2ccccc12 C(=O)(C(F)(F)C(F)(F)F)N1CCCC(C(=O)Nc2cc(O)ncn2)CC1 N1(C(c2nccc(C)n2)=O)CCN(C(c2nc(Br)cnc2N)=O)C(C)C1 C(=O)(C1CCCc2ccccc21)NC1C(C)N(C(=O)CC2COC(=O)C2)CC1 c1(C(=O)NC2CN(C(C3C(C)CCO3)=O)CC23CCC3)cc(Cl)ccc1[N+](=O)[O-] CC1(C)CC(C)(CO)CN1C(c1cc(CNC(C2C(C#N)C2(C)C)=O)cs1)=O N(C1CCCn2nccc21)C(C(=O)N(C)Cc1c(OC)nc(C)cc1)=O Cc1cn2c(n1)CCC(C(N1CCCN(C(c3cnc(C4CC4)s3)=O)CC1)=O)C2 C1(OC)CC2CCC1(C(=O)NCC1CCCN1C(=O)C(O)C1CCCC1)C2 c1(C(=O)NC2C(C(=O)OC)CC2)ccc([N+](=O)[O-])[nH]1 c1(CNC(COCC)=O)ccc2c(c1)CCN(C(=O)C(COC)NC(C)=O)C2 C1(C)(C(=O)NCC2(CC(=O)OC)CC2)CCCN(C(=O)C(C)C(F)F)C1 C(CC(C(=O)N(C1CCCCCC1)CCNC(=O)CP(C)(C)=O)NC=O)SC n1(CC(=O)NCCCOCCN(C(c2c(C)[nH]cn2)=O)C)cc(C#N)cn1 CC(C)C(O)C(F)(F)C(=O)N1CCC(NC(=O)CC2CCC2)C(O)C1 N1(C(C(CC#C)O)=O)CCC2CN(C(=O)CCc3nc(C)cs3)CCC12 Cn1nccc1C(=O)NC(c1ccccc1)CNC(=O)CC1CCC1(F)F N1(C(CC2(OCC)CCC2)=O)CCC(CCNC(=O)COCC)CC1C C1(CNC(COCC(=O)NC)=O)CN(C(C2CCC2C#N)=O)C2CCN1C2 C(=O)(CCC(=O)NC(C)CNC(=O)CN1CCS(=O)CC1)OC O=C(C1=CCCCCC1)NCCC1CCCN(C(C2CC=CCC2)=O)C1 CCCCCS(=O)(=O)CC(=O)NC1CCN(C(c2cc3cc(F)ccc3[nH]2)=O)C1 N1(C(C2(SC)CC2)=O)CC(C)(C)C(NC(C2CCC(C)(F)CC2)=O)C(C)(C)C1 C(=O)(C1CCc2ccccc21)NC1CC2N(C(Cc3nnc(C)o3)=O)C(CC2)C1 N1(C(C(CC)(C)CNC(c2cscn2)=O)=O)CCCC(O)(C2CC2)C1 c1(SC)c(CCNCC(C)(C)NC(=O)C=Cc2cocn2)cccc1C c1(NC(C)CC2CC2)ncccc1S(=O)(=O)N1CCN(C(=O)OC(C)(C)C)CC1 c1(CN(C(C2C(CC)CCCC2)C(=O)NC2CCOC2)CC)ccc(C)c(C)c1 Nc1c(Cl)ccc(F)c1C(=O)NC1CC(CNC(c2ccn3c2CSCC3)=O)C1 N1(C(Cn2c(C)cc(C)n2)=O)CCCC(NC(C2CC3CC2C3)=O)C1C c1(NCC2N(C)S(=O)(=O)CC2)nc(N2CCCCC(C)(C)C2)nc2scnc12 C=CCCC(CO)NC(C1CCN(C(=O)CN(C)CCC)C1)=O CC(C)C(O)C(C)(C)C(=O)N1CCOC(CNC(c2ccc(C(F)(F)F)s2)=O)C1 C(=O)(CCCS(C)(=O)=O)N1C(CNC(c2cn(C)c(Br)c2)=O)CC2CC21 N1(C(C(=O)N2CC(N3CCOC3=O)C2)=O)CCCCC1OC(=O)CCc1cscn1 c1(C(=O)NC2CC(NC(c3c(C)ccc(C)c3)=O)C2)ccc(F)c2cnccc12 c1(C(C(=O)NCCC2CCCN(C(C(C)(C)CO)=O)C2)O)cc(F)cc(F)c1 c1(SC)ccc([N+](=O)[O-])cc1C(=O)NC1CCCCCC1NC(C1CC(F)C1)=O C1(CNC(C(C)c2cc[nH]n2)=O)CN(C(c2cc(C3CC3)ncn2)=O)CC1(F)F C=C1CCN(C(=O)CCN(C(c2cnn(C(F)F)c2)=O)CC)C1 c1(OCOC(C(=O)OC)C(C)C)ccccc1C(N1CC(OCC)C1)=O N1(C(C(C)(F)F)=O)CC2CC3CC2C1C3NC(c1noc2cc(F)ccc12)=O Cc1ccc(Cl)cc1C(N1CCCCC(NC(c2c(C)[nH]c(C)c2C)=O)C1)=O N1(C(=O)C(F)CC2CCOC2)CCC(F)(C(N(C(C)C(=O)NC)CCC)=O)C1 C1(CNC(C(CC2CCC2)NC(C(N2CCOCC2)C)=O)=O)CC2(CC2)C(=O)O1 CC1CN(C(=O)CC(C)(C)CNC(C23CCC(CO)(CC2)C3)=O)CCC1N(C)C CCC(C)CCN=c1[nH]c(N2CCC(C)(C(F)(F)F)CC2)nc2c1COC2 C12(NC(CNC(CCC)=O)=O)CCOC(CNC(=O)C=Cc3sccc3C)(C1)C2 c1(CCCC)ccc(C(=O)N(C)CCNC(C2COCC(C)O2)=O)cc1 N1(CC)Cc2c(C(F)(F)F)cccc2C(C(=O)OC)C1.C12CC1(C)COC2=O c1(C(C(=O)NC2(C(NOCC(C)C)=O)CC2)C)ccn(C)c1 C123CCCC1N(CC2)C3=O.c1(NC(CNC=O)=O)cccc(Cn2cccn2)c1 c1(C(=O)NCC(C(C)C)(C)NC(=O)CC(C)n2cccn2)cnc2c(c1)NCC2 c1(CC(=O)NC(CCN(C(C2(CC#C)CCCC2)=O)C)C)c(F)cccc1Cl c1(C(=O)NCC2OCC3(CN(C(C)=O)C3)C2)ccc2cc(N(C)C)ccc2c1 c1(C(N(C(C)CCNC(c2ncccc2C(F)F)=O)C)=O)cnc2[nH]ncc2c1 c1(C(N2CC3C(NC(c4ccc(CC)s4)=O)(C3)C2)=O)ccc(S(N)(=O)=O)o1 C=CCCCC(C)(C)C(=O)NC1CC2(C1)CN(C(=O)C(N1CCCCCC1)C)C2 c1(SC)c(C(=O)NCCCN(C)C(c2cn(CCO)nn2)=O)cccc1F c1(CC)cc(C(N2CC(C(C(=O)NC(c3nncn3C)C)OC)C2)=O)no1 c1(Cc2ccc(C(N3CCN(CC(=O)O)CC3)=O)cc2)cc(O)nc(O)n1 CCC(C)C(CNC(=O)CCC(C)(C)NC(c1cnn(C)c1OC)=O)CO C1(C(N2CCN(C(C=C(C)C)=O)C(C3CCC3)C2)=O)CC(C)CC(C)(C)C1 c1(-c2n(CCC)ncc2)ccc(-c2nccn2CCC2NC(=O)NC2=O)nc1C C1(C(N(CC#C)CC)=O)CC(F)CN1C(=O)C(CO)OC c1(CC(=O)N(CCNC(c2[nH]cc(C(C)=O)c2)=O)C2CC2)cc(C)nn1C1CCC1 C(C(=O)N(C1CN(C)C1)C)(C(C)C)NC(c1cc(C)no1)=O C1(NC(C(C(C)C)SCC)=O)CCCC2CN(C(=O)C=Cc3cccnc3)CC12 c1(NC2CN(C(=O)CCc3nc(O)n[nH]3)CC23CCC3)ncc2c(n1)CCOC2 N1(C(COCC=C)=O)CCC(CO)C(NC(=O)CNC(=O)C(CC)CC)C1 C1(CC(=O)NC2(CF)CCN(C(c3cc(SC)n(C)n3)=O)C2)CCC(C)(C)CC1 c1(CNC(=O)NC2(C34CC(NC(C(CC)C)=O)(C3)C4)CC2)cc(C)ccc1C c1(C(=O)NCC(CCCC)NC(C2CC2C)=O)coc(=O)c2ccccc12 C(C(C)(CC)NC(c1ccn(CC)n1)=O)NC(CCN(CCCCC)C(C)C)=O c1(OC)coc(C(=O)NC(C)CNC(c2cc(C)cnc2C(F)(F)F)=O)cc1=O C#Cc1cccc(NC(=O)CC2(CNC(c3ncccc3F)=O)CC2)c1 Cc1cc(Cl)ccc1OC(C(=O)NCC1(n2cnc(C(N)=O)n2)CC1)C C1(NC(C2N(CCC)CCCC2)=O)CC1C1CCCN(C(=O)CCC2CC2)C1 CCCC(CCCNC(C1CC12CC(O)C2)=O)NC(=O)CCOC(C)=O C1(N(C(C(=O)NCCSC)C2CC2(Br)Br)CC=C)CCCCC1 c1(C(=O)OC)ccnc(CCNC(C2CCN(C3CCCCC3)C2)=O)n1 Cc1cccc2c(C(=O)NCCC3CN(C(c4cnn5c4CCC5)=O)C3)c[nH]c12 CC1(C)CN(C(C2CC23CC(NC(=O)CCc2nncs2)C3)=O)CCO1 C1(C(=O)NCCC(CNC(CC=CC=C)=O)O)CCC(C(C)(C)O)CC1 c1(CC(=O)NC(CN(C(CCOCCOC)=O)CCO)C)ccc(Br)s1 c1(C(=O)NCCC2CCN(C)C2=O)cc2cccnc2nc1O C1(NC(Cc2c(C)scc2)=O)CN(C(=O)C(C)OC2CCOC2)C2CCCC12 Cc1cnc(NCCc2cnco2)c(S(=O)(=O)NCC(N2CCCC2)C)c1 C(c1ccc(Cl)c(Cl)c1)=CC(=O)NCC(C)(C)CNC(c1ccccc1)=O c1(C(CNC(C=CC(C)C)=O)NC(c2cn(C(C)(C)C)nn2)=O)cccc(Cl)c1 C(C)(N=c1[nH]c2c(c(=NC(C)C3CCCC3)[nH]1)CSC2)c1cccc(C)n1 CC1=NOC(C(=O)NCCC2CN(C(c3coc(C(F)F)n3)=O)C2)C1C C1(CNC(C2CN(C)C2)=O)COCC2(CCN(C(c3cccnc3S)=O)CC2)O1 C(=O)(NNC(=O)C(F)(F)c1cccc(O)c1)c1c(N)c[nH]n1 N1(C(C(C=C)(C)O)=O)CCCC(NC(=O)Cc2c(C)nc(CC)nc2C)CCC1 c1(NC(=O)NC(Cc2cnc[nH]2)CO)cccc(NC(C2CCC(F)C2)=O)c1 N1(C(CCC(C)OC)=O)CC(F)(F)CC1CNC(C1(C)CCNC(=O)C1)=O c1(C(=O)NCCC2COCCN2C(C23CSCC2C3)=O)nccc2c[nH]nc12 c1(CC)ccc(C(=O)NC2(CF)CCN(C(c3sc(F)cc3Cl)=O)C2)cc1F N1(CC(=O)N(CC(=O)NCC2C=CCN2C)CC)CCCCC1C C1(NC(c2cnccc2Cl)=O)CN(C(C23CCCC2(C(N)=O)C3)=O)CC12CCC2 C1(NC(C(c2cn(C)nc2)(F)F)=O)CCCN(C(c2cscc2F)=O)C1 C1(C(=O)NCCN(C(c2cccc(C)c2C)=O)CC)CCc2ncccc2C1 C(CN=c1cc(C)c(S(=O)(=O)NCC2CCN2C)c[nH]1)=CCCC CCCCC(C(=O)NC1C2CN(Cc3ccc(OC)cc3O)CC12)NC(N)=O n1(CCOC)cccc(C(=O)NC(C)CNC(=O)C(C2CCCC2)OC)c1=O C(CC(O)CC(=O)NCC1CCC(NC(c2scnc2Cl)=O)C1)SC N1(C(CC2CCC(=O)NC2=O)=O)CCCCC(NC(=O)COCCF)CC1 CC1CN(C(=O)CS(=O)(=O)CCO)CCCN1C(=O)C=C1CC1 C1(C)(CNC(C(N2C(CC)CCC2)=O)=O)CCCN1C(=O)CC(C)(C)C C(=O)(C(C(C)(C)C)NC(N)=O)N1CCCC(N(C(=O)CSC(F)(F)F)C)C1 c1(CC)c(C(=O)N(C)CC2CCCCN2C(=O)Cc2cnsc2)cnn1C C1(C(=O)NCC(CNC(c2c(C)c[nH]n2)=O)F)CCCN(c2ncccn2)C1 N1(C(C(C=C)C)=O)CCN(C2CN(C(c3conc3COC)=O)C2)CC1 c1(C(=O)NC2C(NC(CCCC)=O)CCCCC2)cc(S(=O)(=O)N(C)C)c[nH]1 CC(C)CC(CNC(C1CC1(C)C(F)F)=O)NC(c1cc(Cl)no1)=O Cc1ccc(C(C)CC(N2CCC(O)(CNC(c3ccc(Cl)o3)=O)C2)=O)cc1 C(C)(CCC(=O)NCCN(C1CCCCC1)C(C1(C#N)CC=CC1)=O)SC c1(C(=O)NC2C(NC(Cc3cc(C)ns3)=O)COC2)cccc2nccn12 C1(C(N2C(C3(O)CN(C(c4cnn[nH]4)=O)C3)CCC2)=O)CCc2nnc(O)n2C1 CCC1C(=O)Nc2ccc(C(=O)NC3CC[Si](C)(C)C3)cc21 c1(C(=O)NCC2(C(C)(C)C)CCN(C(CC(CC)OC)=O)C2)c(C)oc(C)c1C c1(CC(=O)NC23C(n4cc(CN(C)C)nn4)CC(CC2)C3)ccc2ccoc2c1 c1(C(C)C)ccc(F)cc1C(=O)NC1CC2CCC1N2C(c1cc[nH]c(=N)c1)=O CC(C)CC(C)C(=O)NCC(C)=CC(=O)N(CC(C)(C)O)C n1(CC)cc(C(=O)N(CC(C)NC(c2coc(C(C)C)n2)=O)CC)c(C)n1 c1(CCC)ccccc1S(=O)(=O)N1CC23CCCC2(CO)C13 c1(C(=O)NC2C3CCN(C(c4cccc(OC)c4C)=O)C32)nccc2cc[nH]c12 c1(C(=O)NCC(CN(C)C(C2(Br)CC2(C)C)=O)O)ccc2c(c1)COCO2 Cn1cc(C=CC(=O)NC2CCC(F)(CNC(=O)Cc3cncs3)C2)nn1 c1(C(=O)NCCC23C(CN(C(CC(=O)OC)=O)C2)CC3)cnc2n1C(C)CCC2 c1(C(=O)NCC(CO)NC(CCn2ncc(C)c2)=O)c(Br)sc(C)c1C C1(C(=O)NCCNC(CC23CC(C)(OC2)C3)=O)CC1C1CC(F)(F)C1 C(=O)(CCCN=c1nccc[nH]1)NCC1OCCN(C(c2c(C)nncc2)=O)C1 CC1CN(C(=O)CC2CCN2C(=O)CCC(=O)N(C)C)CCN1CCO c1(SCCCS(=O)(=O)N(C)CC)cc(Cl)nc(Cl)c1 C#CCC(C(=O)N1CCC(OCC=C)C1)NC(=O)Cc1csnc1C N1(C(Cn2cc(C(C)=O)nn2)=O)CCN(C(C2CC2c2cc[nH]n2)=O)CC1C CP(C)(=O)c1ccc(C(=O)NCC2CC(CNC(=O)C(F)=CC3CC3)CO2)nc1 N1(C(CNC(CN(C)C)=O)=O)CCOC(C(=O)N(CC(C)(O)C2CC2)C)CC1 N1(C(C2CC(OCC)C2)=O)CCCCC(NC(c2sccc2SC)=O)C1 CC1CN(C(C2(Cl)CC2)=O)CCC1NC(=O)C=Cc1cn[nH]c1 C#CCCCCC(=O)NCC1(F)CCN(C(=O)C(F)OC)C1 c1(C(=O)NC2CC(CC(=O)N(CCCOC)C)C2(C)C)cc[nH]c2nccc1-2 c1(C(N2CCCC2CNC2CCC2)C)ccccc1F N1(C(C(COCC)C)=O)CCC(O)C(NC(=O)C(C)(C)CSC)C1 c1(C(N2C(C(=O)NC(c3nc(C)on3)C)CCCC2)=O)coc2ccccc12 c1(NC(C2C3CC2N(Cc2ccc(N4CCOCC4)cc2Br)C3)=O)cnc(O)nc1O C(=O)(C(C)(C(C)C)OC)NCCCC(C)(C)NC(c1cccc(SCC)c1)=O c1(OC)cccc(Cl)c1CC(N1CCN(c2cc(F)ncn2)C(CCO)C1)=O C1(NC(CCC)=O)CC2CC1N(C(c1nn(-c3ccsc3)nc1C)=O)C2 C12(NC(=O)C=CCN3CCCCC3)CCCN(C(=O)CCC3CCOC3)CC1C2 c1(C(=O)NCCC2(OC)CN(C(C3CN(C)CCO3)=O)C2)ccnc2ccsc12 N1(C(C(CCCC)C)=O)CC2CCN(C(c3cn(C)c4ncccc34)=O)C(C2)C1 N1(c2n(CCC#C)c(COc3ccccc3Br)nn2)CC=CCC2(CCCC2)C1 n1(CC(=O)NC(C)C(C)NC(=O)CNC=O)cc(CO)nn1 CC(C)C(C)(CNC1CC2CCC1C2)NC(=O)Cn1nc(C2CC2)cc1C1CC1 C1(NC(c2nc(C(N)=O)sc2)=O)(CNC(c2cncc(F)c2)=O)CC2CCC1C2 C=C1COc2c(C(=O)NCC(C3CCCC3)NC(c3sccc3C)=O)cnn2C1 C1(C(=O)OCC)CCc2nc(NC(C3(C)CC(COC)C3)=O)sc2C1 CC1CC=C(C(=O)NCC(Cc2ccccc2)NC(C2CCOC(C)C2)=O)CC1 Cc1ccccc1C(C(C)(C)C)NC(c1ccccc1OC1CCNCC1)=O c1(CC)ncc(C(=O)NCC(C2CC2)N(CC(C)(C)CC2CCOCC2)C)[nH]1 C(=O)(C(C)(C)C(=O)NC(CCN(C)C(C1Cc2nccn2C1)=O)C(C)C)OC CCCCC(CNC(c1cn(C(C)C)nn1)=O)NC(=O)C(c1nncn1C)OC CCCC(C)(O)CC(=O)NC1CC2(C1)CC(C(N1CCOC(C#N)C1)=O)C2 N1(C(C(=O)NC(C)C)=O)CCn2nnc(C(=O)NC(C)CCO)c2C1 C(=O)(C(C)(O)CCC)N1CC(CCC)C(NC(c2c(C)nsc2C)=O)C1 c1(C(=O)NC23CC(CC(=O)NC4C(OC)C(O)C4)(C2)C3)cnn(C)c1C#N C1(C)(CNC(CCCC)=O)CCN(C(=O)C(N2CCC(O)CC2)C)C1 C1(NC(C(C=C)C)=O)CC2CC(C1)CN(C(=O)CCc1cccc(C)c1)C2 Cc1ccc(C)c(C(=O)NC2CCC(NC(c3[nH]c(C)cc3C)=O)CC2)n1 CC1CCN(C(c2nc(C3CC3)cs2)=O)CC1NC(c1ccc(C(C)(C)C)[nH]1)=O c1(C(=O)NC2C(NC(C(C(CC)C)O)=O)CCCC2)cc(F)cc(Cl)c1O Cc1nn(C)c(=O)c(C(N2CC3(C2)C(NC(=O)C(N)=O)CCS3(=O)=O)=O)c1C N1(C(COCCOC)=O)CCCC(C)(CNC(=O)CC(C)SC)C1 CC(C)CC(C(=O)NC(CNC(c1ccn2ccnc2n1)=O)C(C)(C)C)C(C)C C1(NC(c2c(CC)n(C)nc2)=O)CC2CC(NC(=O)C(F)(F)C(O)C3CC3)C1C2 N1(C(CC2CN(C(C)=O)C2)=O)CCCC(C(C)C(=O)NCCC(C)F)C1 CC(C)C(O)CC(=O)NC(C)(C(=O)NCC1(S(C)=O)CC1)C1CCC1 c1(C(CNC(c2conc2-c2ccccc2)=O)C(F)F)c[nH]c2ccccc12 C12C3CN(CC13)C(=O)C=CC2=O.C1(C(=O)NC2CCCC2)CC=CCO1 C12(CNC(CNC(C)=O)=O)CCC(CC1)N(C(C1C=CCC1)=O)C2 C1(NC(COC(CC)C)=O)CC2CCC1(C(=O)NCC(=O)N(C)C)C2 Cc1cnc2n1C(C(=O)N(CC(O)CN(C(=O)CSCC(N)=O)C)C)CCC2 c1(C(=O)NCC2(O)CN(C(C3CC34CCOCC4)=O)C2)c[nH]c2ncccc12 C(C(CC=C)C(=O)NCC(=O)NC(N)=O)NC(CCCOCC=C)=O c1(NC(C2C(NC(=O)Nc3ccc(Cl)cc3Cl)C2)=O)ncc([N+](=O)[O-])cc1O C12(NC(C(C)NS(CC)(=O)=O)=O)CCCN(C(c3cc(O)ccc3F)=O)CC1C2 C(CCN=c1nc(C(=O)N(C)C)cc(SC)[nH]1)N(C(C(C(CC)CC)C)=O)C C1(C(N(CC)CC)=O)CCN2CCOCC12.c1(CCC=O)ccc(C2CCCC2)o1 Nc1ccc(C(N2CCCCC(CNC(C3CC4CCC(C3)O4)=O)C2)=O)c(F)c1 C(=O)(C(C)(C)CNC(c1ccn(C)c1C)=O)NCCCOC C=CCC(C(=O)N1CCC(C(N2CCC(OC3C4CCCC34)C2)=O)CC1)OCC C1(C(=O)NC2CC(CCNC(c3cc(CSC)c(C)o3)=O)C2)(CC)CCNC1=O C(=O)(C1=NOC2(CCN(Cc3ccccc3O)C2)C1)OC.CCC(C)C1C(=O)N1 c1(C(N(CC(=O)NCCN(CCCC)C)CCC)=O)sccc1Cl C=CCC(CNC(=O)CCCF)C(=O)NC(C)CN(CCCC)C c1(C(=O)OC)ccc(C)c(S(=O)(=O)NCCNC(C2CC(C(=O)O)C2(C)C)=O)c1 C#CCC(CC(=O)NC(c1cnsc1)C)NC(=O)C(C)=C(C)CC N1(C(C(CC=CC)NC(c2cc(C)c(C)cn2)=O)=O)C2CCC1CC(F)C2 C1(CNC(CN(C2CCC2)C)=O)CC(C)(C)CN1C(C1CS(=O)(=O)C1)=O C1(NC(C=C(C)c2ccco2)=O)COC2(CCN(C(C3CCCCC3O)=O)C2)C1 Cc1ccc2n[nH]cc2c1C(=O)NC(CNC(=O)CC1CCCC1(F)F)CO N1(C(C(=O)NC2C(COC)C2)=O)CCCc2sccc2C1 N1(c2nccc(SC)n2)CCCC(CCNC(=O)C(C)SC(F)(F)F)CC1 C1(NC(c2cc(C)[nH]c2C)=O)CCCCCN(C(C2CCCCCC2)=O)C1 Cc1cc(OCC(=O)NC2CCC(NC(c3ccnc(S)c3)=O)CC2)ccc1F N1(CC)CCCN(C(C2(CNC(=O)CC(O)C(C)C)CCCO2)=O)CC1 C1(NC(c2ccsc2)=O)COC2C(NC(C3CC4CCC3CC4)=O)COC12 c1(C(=O)NC(C)CCN(C(=O)CC2(C(F)(F)F)CC2)C)ccsc1Cl c1(CN(C(CN(C(c2cnccn2)=O)CC)=O)C)cnnn1C CC1CCCC1(C(=O)N(C1(CCO)CC1)C)NC(=O)CN(C)C(N)=O C1(O)(CCNC(c2cc(CF)on2)=O)CCCN(C(C2COCCC2(F)F)=O)C1 c1(C(N2C(Cn3cc(C(C)(C)O)nn3)CC(O)C2)=O)csc2c(F)cccc12 N1(C(C2(C)CCCN(C(C(=C)F)=O)C2)=O)CCC2(C=Cc3ccccc32)CC1 C=C(C)c1cccc(NC(=O)NC23CCCC(C2)N(C(C)=O)C3)c1 S(=O)(=O)(c1cn(C)nc1C)Nc1ccc(C(=O)Nc2c(C)ccc(Br)c2)nc1 C(=O)(CC(F)(F)F)N(C1CC(F)(CNC(C(C)OCC#C)=O)C1)CC(F)(F)F C1(C(=O)NC(C2CN(C(CN(C(C)=O)C)=O)C2)CO)CCCCC1 C#CCCCCCC(C(=O)NC1CCOCC1)N1CC2CCC1C(O)C2O N1(C(c2cn(CC(=O)OC)nn2)=O)CC=CC(NC(=O)Cc2ccc(F)cc2)C1 c1(NC(c2cc(O)ccc2O)=O)c(-c2cccnc2OC(F)F)ccc2c1OCO2 c1(CN(CCC)C(=O)NC2CC(C(=O)OC)C2(C)C)ccc(Cl)cc1Cl C1(C(N2CCC(CCNC(CC(C)(C)F)=O)CC2)=O)Cc2nncn2C1 C#CCC(CC(=O)NC1CCCC1(C)N(C)C)NC(=O)C(C)NC(C)=O C1(CC)CN(C(c2cccc(Br)c2)=O)CCN1C(c1cc(C)cc(Cl)c1)=O C1(C(=O)NC2(C(=O)NC3C=CCCC3)C(C)C2)(CF)CC(=O)C1 Cc1cc(F)c(C(N2CCC(NCc3cn4ccsc4n3)C(C)C2)=O)c(F)c1 Cc1ccc2sc(C(=O)NC(CNC(c3c(C)ncn3O)=O)C3CC3)c(C)c2c1 c1(CNC(C)C(=O)NCC2CCCO2)cccc(C(=O)OC(C)(C)C)c1 CCC(CCC(=O)N1CCC(C(=O)NCC(C)C(=O)OC)(CC)CC1)OC C1(CNC(CCNS(CC)(=O)=O)=O)COCC1NC(=O)Cc1ccsc1C C1(CCCC)(C(=O)NCC2CCCN2C(=O)CC2CCOC2C)CCCC1 N1(C(COCC)=O)C2CCC1CC(CNC(=O)CC1(C)CCOC1)C2 c1(C(N)=O)cc(F)ncc1C(=O)NCCNC(C1CCCC1)=O.C12(CCl)CC(N)(C1)C2 O=S1(=O)CCCN1c1ccc(-n2cc(C3CCCCC3)nn2)cc1 C1(CC)(NC(c2cn(C)c(=O)cn2)=O)CCN(C(=O)CSc2nccn2C)CC1 C(=O)(CCCCCSC)N(C(C)C(O)C(=O)NCC1CC2C=CC1C2)CC CC(CCNC(=O)NCC=C1CCSCC1)C(C)(C)C c1(C(=O)NCC(=O)NCC(C)N(C(=O)CCOCC(F)F)C)ccncc1 CCC(C)CC(C)C(=O)N1CCC(NC(C23CC2COC3(C)C)=O)C1(C)C C1(NC(=O)C=CCOCC(F)(F)F)CCCCN(C(C2(n3cc(Cl)cn3)CC2)=O)C1 C(C(=O)N(CC1CC1)OC)C1CCN(C(c2ccc(CC)s2)=O)CC1 N1(C(CN2CCC(C)C2)=O)CCC(O)CC1C(=O)NCC1(O)CCCCCC1 CCCCC(CC)CC(CNC(=O)NCCOCC)CC.C1CCOC1 O=C1CN(C(=O)C2=C(F)CSC2)c2ccccc2N1.N1CCc2ncccc2C1=O C1(C(N2C(C3(NC(C4C(=O)NCC4)=O)CC3)CCC2)=O)Cc2cccnc2C1 CN1N=C(C(=O)N2CCC(C(=O)NCCn3ncnn3)C2C2CC2)CCC1=O c1(NC(C)=O)cccc(C(C)NC2CCOC(c3ccccn3)C2)c1 c1(OCC)ccc(Br)cc1CNC1CCC(NC(C(=O)OC(C)(C)C)=O)C1 N1(C(C2(CC)COC2)=O)CCC(C)(NC(c2cnc(C)nc2)=O)CC1 C1(C(NOCC(C(C)(C)C)O)=O)CCC2CCC1N2C(=O)Cc1ccc(O)nc1 C=CC1CC(N=c2nc3[nH]c(SC)ncnc-3n2)C1 C1(N(C)C(c2csc(CO)n2)=O)C2CN(C(=O)COCCc3ccccc3)CC12 c1(CNC(C2(NC(C(COC)N(C)C)=O)CC2C)=O)ccncc1Cl C1(CC(=O)NCC2C(NC(=O)COCC3CCOC3)C2)C=CS(=O)(=O)C1 N1(C(C2C(C)C2)=O)CCC(F)C(NC(c2ccc(CCF)cc2)=O)C1 C1(C(N2CCC(C(CNC(=O)CCCC3CC3)O)CC2)=O)CCC2(CCC2)O1 N1(C(CCOC)=O)CC(F)(F)CC1(C)CNC(=O)CCNC(N)=O CC1(C)CC(C(N2CC(F)CC2CC(=O)Nc2cnc(F)nc2)=O)CCO1 c1(C(N2CC3C(C2)N3C(=O)C=Cc2cccs2)=O)cccc([N+](=O)[O-])c1O CC1COCCN(C(=O)C=CCC2(NC(C3CC(=O)CS3)=O)CCC2)C1 Cc1cc(Cl)c(C(=O)NCC(CC(C)C)NC(C2CCN2S(C)(=O)=O)=O)s1 C(=O)(C(C)(C)CCS(C)(=O)=O)NC12C(CN(C(CCC=CC(C)C)=O)C1)CCC2 c1(C(N(C)CC2CN(C(C3(F)CCOC3)=O)CCO2)=O)ccc2nn[nH]c2n1 N1(C(C2NC(=O)OCC2)=O)CC(NC(c2cc3ccncc3[nH]2)=O)CCC(O)C1 CCCCC(O)CNC(=O)C(Cc1cc[nH]n1)NC(c1coc(CC)n1)=O CCC(C)(C(=O)N1CC2CCC(C1)N2C(c1nccc2occc12)=O)C(F)F N1(C(C=CCCCCC)=O)Cc2[nH][nH]c(=NC(=O)c3cnnc(O)c3)c2C1 C12(C(=O)NCC(C)CN(C(=O)C(c3ccc(C#N)cc3)O)C)CCC(C)(CO1)C2 c1(C(=O)NCC2C(NC(C3CC(C)(C)OCC3)=O)COC2)cc(F)cc(N)c1F N1(C(c2cc(OC)ncc2)=O)CC2CCC(C1)C(NC(C1CC13CCCC3)=O)C2 C(=O)(C(Cc1ccccc1)C(F)(F)F)NCC(C)N(C(C(C)OC)=O)C c1(C(=O)NCCC2CC(NC(c3nc(COC)oc3)=O)C2)cccc(Br)c1 c1(C(=O)OC)cc(Br)c(C)cc1F.C1(C(=O)OCC)CN2CC1NC2=O C(=O)(C1CCc2nnc(C)n21)NC1CC(NC(CC(C(=O)OC)(C)O)=O)C1 Cc1cc(C(N2CCCC2C(=O)NCC(F)F)C(=O)NC(C)(C)C)ccn1 C=C(C)CCCC(=O)N(CC(C)NC(=O)C=Cc1ccc(Br)o1)C CC(CNC(=O)CC1CCCC12CC2)C(F)C(=O)NC1C2CCCOC12 Cc1cn2c(n1)C(C(=O)N(C)CC1CCCN(C(c3ccnnc3)=O)C1)CCC2 N1(C(c2c(NC)cccc2)=O)CC2CC1CN2CCc1ccns1 C12(C(=O)NCCC(C)CCNC(C3CCC(F)(F)C3)=O)CCC(CC1)C2(C)C n1(CC(N2CC3C(CNC(c4cnn(C)n4)=O)(C3)C2)=O)ccc(O)nc1=O c1(N(C(CCNC(CCc2ccc(C)s2)=O)C)C)ccc([N+](=O)[O-])cc1 Cc1ccc(Br)c(-n2cc(CONC(c3cc(Cl)cnn3)=O)nn2)c1 N1(C(CCc2scc(C)n2)=O)CCCC(NC(C2CN(C3COC3)C2)=O)C1 C#CC1CN(C(=O)C(C)C(C)O)CCN1C(=O)Cc1cc(F)ccc1Cl C(N=c1[nH]c(Cl)nc2ccc(Cl)nc12)C1C(NC(=O)Cc2cc[nH]n2)CCCC1 C(CN=c1[nH]c2c(c(=NCc3csc(Cl)c3)[nH]1)SCC2)(S(C)(=O)=O)OC c1(C(N2CCC(N(C(=O)CCN(C)CC)CC)CC2)=O)cnc2n1CCC(C)C2 N1(C(C(c2scc(C)n2)(F)F)=O)CCC2C(NC(c3conc3C)=O)C2CC1 N(C(=NCC1CCC1)NCC1CC1(F)F)CC1(C#C)CCC1 C(=O)(C1=NOCC1)NCCc1cc(C(N(C(C)C2CC2)CC)=O)no1 c1(C(=O)NC(C)CN(C)C(c2nccc(Cl)c2F)=O)ccn2c1CS(=O)(=O)CC2 N1(C(C2CCN(C(c3c(C)nn(C)c3C)=O)CC2)=O)CCc2cccc(C)c21 C1(C(N2C3(C(=O)NCCC(C=C)C)CC(C2)C3)=O)CC2CCCC2C1 C(=O)(C(F)CC(C)(C)NC(=O)CC1CSC1)NC(CC)C(C)CN(C)C N1(C(C(C)OCCOC)=O)CCN(CCCCCNC(C2(COC)CC2)=O)CC1 C(C(O)C(F)(F)F)N(C)C(=O)NCc1nc(-c2cc(Br)cs2)cs1 C1(C(=O)NCc2cc(COC)on2)CCC(O)CN1C(c1ccccc1F)=O CCC(CC)C(C)C(=O)N1CC(NC(=O)CSc2nncn2C)CC1(C)C c1(CCC)nc(C(=O)NC2COCC2NC(=O)C(C)CN(C)C)co1 C1(C(=O)NCC2CC(NC(C(C)(C)c3ccccc3)=O)C2)Cc2ccccc2S1 C1(N(C)Cc2ccccc2)CCCN(C(=O)C(N)CC2CCOCC2)C1 CCCC(F)(F)C(=O)NCC#CC(N1CCC(C#N)C1)=O CC(=O)CC(C)(C)C(=O)N1CC2C(CNC(=O)CSCC(F)(F)F)C2C1 c1(C(N(CCCCO)C)=O)cccc(CNC(=O)CC2(O)CCOC2)c1 C1(C(=O)NC2CC(CCNC(=O)CCc3cc(C)[nH]n3)C2)(CC)CC(F)(F)C1 O=C(CCS(=O)(=O)c1ccc(Cl)cc1)NCC1(F)CC(N)C1 c1(C(N(CC(CNC(CCCN(C(C)=O)C)=O)O)C)=O)ccc2oc(S)nc2c1 CCCCCC(CC)C(=O)N1CC(C(=O)Nc2ccc(Cl)c(F)c2)CC(C)(C)C1 c1(C(=O)NC(CC=C)CNC(c2cncc(OC)c2)=O)c(F)c(F)cc(F)c1F Cc1c(CC(=O)NCC(C)CNC(=O)CCc2ccc(O)nc2)cnn1C CCCC(C(=O)NCC1(C(N)=O)CN(C(=O)Cc2cc(Cl)n(C)n2)C1)N(C)C CC(C)CC(=O)C(=O)NC(c1ccc(SC(F)F)cc1)C CCCC(C)(O)CC(=O)NC1(C(=O)Nc2cc(C)ccc2C)CCN(C)C1 c1(C(N2C(C(CCC)C)CCC2)=O)cc(Br)c(I)s1 c1(C(=O)NC(CC(C)C)CNC(=O)C=C2CCCCC2)ccc(N)cc1Cl N1(C(C2C(OC)CN(C(c3cc(C)nc(C)c3)=O)C2)=O)CCC(C)(C2CC2)C1 c1(C(=O)NC2CC3CN(C(CC4CCCC(=O)N4)=O)C2C3)cc2ccccn2c1 CC(C)(CCC(=O)NCC1CCCCC(=O)N1)NC(=O)CC1CCCC12CC2 C1(C(=O)NCCC2N(C(Cc3n(C)ccn3)=O)CCCC2)CCn2cncc2C1 Cc1cc(F)cnc1C(N1CCCC(C(=O)NCC2CCOCC2)C1C)=O c1(C(=O)NC(CC)C(O)C(=O)OC)c2c(nn1C)CCC2 c1(CC)ccc(NNC(=O)C2CC3(CCCC3)CN2C(=O)OC(C)(C)C)cc1 c1(C(C)C)nscc1NC(=O)NCC1CCC1C(=O)OC(C)(C)C c1(C(N2CCC(NC(C3(CC=C)CCOC3)=O)C2)=O)ccc(C)nc1C N1(C(C(COC)(C)O)=O)C2CCC(C2)C1CNC(=O)Cc1ccc(OC)cc1 N1(C(c2n(CCC)ncc2)=O)CCC2(C1)CN(C(=O)C(C)CSC)C2 C1(C(=O)NCC2(CNC(c3ccc(C4CC4)o3)=O)CC2(F)F)CCC2(CC1)CC2 Cc1nn(C)c(CNc2cccc(SCc3ccccc3)c2)c1Cl c1(C(N2C(CNC(CCc3n(C)cnc3)=O)CCC2)=O)c(F)ccc2[nH]ccc12 C1(CC(N2CC(OCCNC(C(C)Cn3ccnc3)=O)C2)=O)COCC1(C)C c1(CNC(=O)Nc2cccnc2)ocnc1C(=O)NC1CCC(NCCO)C1 C1(NC(c2cnnc(O)c2)=O)CN(C(=O)CSCc2ncc[nH]2)CCC1F C(=O)(C(C)(C)O)NC1CC(CC(=O)N(CCC(N)=O)CC)C1 CC1CC(NC(c2scnc2C(C)(C)C)=O)CN(C(=O)C2=CCCSC2)C1 c1(C(=O)NCCOC2CCN(C(C(C=C)(C)C)=O)C2)ccc2c(c1)CC(=O)N2 C1(C(N2CC(OCCN(C(=O)COCC(F)F)C)C2)=O)CCC(F)C1 C1(O)(CC)CCCN(C(C(=O)NCCCF)C(C2CCC2)OC)C1 C(=O)(C1=NNC(=O)CC1)N1CC(C)C(CNC(C2CCCC3(CCC3)C2)=O)C1 C1(CNC(COCC(=C)C)=O)CC2CCC1N2C(=O)CC1CCN(C)C1 c1(CC)nc2sc(C)cn2c1C(=O)NC1CC2CCC1(CNC(=O)COC)C2 C=CCC(CC(=O)NC1CN(C)C1)N(C(=O)CCCCNC(=O)OC(C)(C)C)C C12(C(=O)NCCO)COCC1C2(F)F.C12CC1C(=O)N(CC)CCNC2=O C(=O)(C1=NOC(CNC(c2occc2C(C)C)=O)C1)N1CC(C)(OCC)C1 N1(C(C(C(=O)OCC)F)=O)C2CCC1CC(C(=O)NCc1ccc(F)cc1F)C2 c1(C(=O)NC(c2ccc(Cl)c(Cl)c2)CC(=O)OC)ccc(C)cc1C N1(c2cc(SC)ncn2)CCCC(O)(C(=O)Nc2ccc(Br)cc2)C1 C(=O)(C(O)CC[S+](C)C)N1CC(CN(C)C(c2cccc3ccoc23)=O)OCC1 N1(C(CCC(N)=O)=O)CC2CCN(C(=O)CCc3ccnc(Cl)c3)CC12.CCC#N c1(C(=O)NCC2(NC(CCC#CC)=O)CC2)cc2c(C)ccc(Br)c2[nH]1 c1(C(=O)NC2CC(C(C)O)C2)cccc2nn(C)cc12 C1(CNC(C2C(CCC)C2)=O)CCN(C(c2cc(C)[nH]n2)=O)CC1(F)F C1(NC(c2ccn(C(C)(C)C)n2)=O)CN(C(=O)Cn2ccnn2)CC1n1ccnn1 c1(CC(N2C(CNC(C3N(CC)CC3)=O)CC3CC32)=O)cccc2ccsc12 c1(C(N2CC(C)(NC(C(c3ccnn3C)C)=O)C2)=O)cnc2ccccn2c1=O N1(C(C(CN(C(c2cc(CC)no2)=O)C)C)=O)CCc2nn[nH]c2C1 c1(C(=O)Nc2cc(C(=O)OC)sc2)cc(O)nc2[nH]c(=N)ccc12 C1(CC(N2CC(NC(c3cnc(CC)[nH]3)=O)C(F)C2)=O)CCC2(CCC2)O1 N1(C(c2cnn(CCF)c2)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)C2CCC12 C=CC(CC)CC(=O)N1CCOC(CN(C(=O)C(F)(F)CC2CC2)C)C1 C1(C(=O)NCC(C2CCC2)NC(C2(COC)CCCO2)=O)CN2CCCN1CC2 C(C)(C)(CC(=O)NCC(C)(C)NC(=O)C(CC#N)c1ccccc1)N(C)C C(=O)(CC(C)CNC(=O)C(C)(C)OC)N1C(C)(CCC)CC1 c1(SCC(=O)NCC2CN(C(CC=CC=C)=O)C3C2C3)ccc(F)c(F)c1 Cc1ccnc(O)c1C(=O)NCC(C)(CO)NC(c1cccc(Cl)c1)=O C1(C(C)=O)CC(CC(=O)NCC2CC(=C3CCC3)C2)C1(C)C N1(C(CC=CCC)=O)CCN(C(=O)C(=O)NCCNC(C)=O)CCC1C C(=O)(C(C)(C)C(F)(F)F)N1CC(C)(C)C(CNC(=O)C(F)=C2CCC2)C1 CN1CCN(C(C2CCC2C(N)=O)=O)CC1CNC(c1scnc1C(F)F)=O N1(C(C#CC(C)NC(=O)CNC(=O)C(F)(F)F)=O)CC(C(=O)O)C2(CCC2)C1 C1(C(=O)OC)CC2CN(C(=O)NC(c3ccc(C(C)C)cc3)C)CC2C1 C(=O)(C(CC(F)F)C1CCC1)NCC1CCC(CNC(CC2CN(C)C2)=O)CC1 C1(CC(=O)NCCCCCN(C(c2cc(COC)sc2)=O)C)CCCNC(=O)C1 C(c1ccc(Cl)cc1F)=CC(N1CCC(NC(C2CCC(=C)CC2)=O)C(F)C1)=O C1(C(=O)Nc2c(CC)noc2)CN(C(=O)C(CC)NC(C)=O)CCO1 c1(NCC(CCC)OCC)ccc(S(=O)(=O)NC2CCCC(F)(F)C2)cc1F c1(C(N2CCCN(CCNC(C3CCSC3)=O)CC2)=O)cccc2c1CCC2=O N1(C(CC2(C=C)CCC2)=O)CCC(NC(c2cc(C)oc2CC)=O)C(O)C1 c1(CNC(C(n2ccc(C)n2)C)=O)ncccc1C(=O)NOCC1CCCN1C N1(C(CC2CC(CC)OCC2)=O)CC2(CCN(C(=O)C=C(C)c3cccs3)C2)C1 c1(C(N(C2CC3CN(C(C(CCC)N(C)C)=O)C2C3)C)=O)cnn2c1OCCC2 C1(C#C)(C(=O)NC(C2CCCC2)C#C)CCN(C(=O)C(CC(C)(C)C)OC)CC1 C1(C(=O)NC2C=CCN(C(C(n3c(C)ccn3)C)=O)C2)SC2C=CC1CC2 N1(C(C(CC)C)=O)CC2CC3CC2C1C3NC(c1cc2nc(=O)ccn2[nH]1)=O N1(C(CCn2c(C)nc(C)n2)=O)CCCCC(NC(=O)CN2CCCC2=O)CC1 c1(CCCC)ccc(C(N2CC3CC2(CNC(C2CC4CCC2O4)=O)C3)=O)cc1 C(N=c1[nH]cnc(Cl)c1F)N(CCCN(C(C1(C(N(C)C)=O)CC1)=O)C)C N1(C(CN2CCC(OC)C2)=O)CCC(=CCNC(=O)Cn2cnc(C#N)n2)CC1 C1(C(=O)NC2(CF)CCN(C(C3CCCSC3)=O)C2)CCC(F)(F)CC1 C12(C(=O)NCC(CNC(C3(COC)CCC3)=O)(C)C)CCCCC1C2(F)F O=C1CC(CC(=O)NC2CN(C(=O)Nc3ccccc3)C2)CCCN1 c1(CCC)ccc(C(=O)NC(C)CCCNC(=O)CC(C)C(C)C)cc1[N+](=O)[O-] C1(C)(C(=O)NCC2C(C)(C)C2C(=O)NCCCCOC2CC2)CCCC1O C12(NC(C(C)=CC)=O)CCC(CNC(c3cc(C)n(CC)n3)=O)(CC1)OC2 C1(CNC(C2C(OC)CCC2)=O)CCC(C(N2CCSC(C)C2)=O)CC1 c1(C(N(CCNC(C2(C)C(C)(C)C2)=O)C2CC2)=O)ccc(F)cc1 Cc1cc(C(N2CC(NC(c3cccn3C(C)C)=O)C(O)C2)=O)cc(C(F)F)c1 C1(NC(Cc2c(C(C)C)con2)=O)CN(C(C2(C)C=CCCC2)=O)CC12CC2 N1(C(C)C)CCCC(C(=O)NCC2CC(NC(=O)C(C)(O)C3CCC3)C2)C1 Cc1cc(F)ccc1-n1cc(O)c(C(=O)NC2CCn3nccc3C2)n1 c1(C(=O)NC2C(NC(=O)CN3C(=O)CNC3=O)CC2)c(F)cccc1F Cc1cnccc1C(=O)NCCCC1CCCN1C(=O)C(C)Cc1cnn(C)c1 c1(CC)noc(C(=O)NCCNC(C2CCN(c3ccc(C)cc3)C2=O)=O)c1C CC1CN(C(=O)C2=C(Cl)CC2)CCN1C(=O)C(F)(F)C1CC1 c1(C(=O)NC2(C)CC(NC(C3CC(C(=O)OC)C3)=O)C2)snc2ccccc12 c1(C(N2C(C)CC(NC(c3ccoc3)=O)C2)=O)cc2c(nn1)CCCC2 Cc1nc(C)c(C(=O)NC2(CCO)CCOC2)o1.C12CC1C(=O)NC2 C1(C(=O)NC2C3CN(C(C(c4ccccc4)OC)=O)C2C3)CC2CCC1CC2 C1(CC)C(NC(=O)C(CSC)OC)CCCN1C(C1CSCC(=O)N1)=O N1(C(C(n2ncc(C)c2)C)=O)CCC(NC(C2CC3CCCC23)=O)CC1C c1(CC)cnn(CNC(C2(c3cccnc3)CC2)=O)c1.C1(=O)COCCN1 C(CC(C(=O)NCCn1cnccc1=O)OC)NC(CSCCCC)=O c1(C(=O)NC(C)CCCNC(C2(Cl)CC23CCC3)=O)cnc2ccoc2c1 Cc1cc(C(=O)NC2CCCC(C(=O)NC3CC4(CCCC4)C3)CC2)cc(C)c1 Cc1ccn2cc(C(=O)NC(C3CCN(C(=O)C(F)CC4CCC4)C3)C)nc2c1 Cc1cc(P(C)(C)=O)oc1C(=O)NC(C1CCN(C(C2(F)CC=CC2)=O)C1)C n1(CC)[nH]c(=NC(=O)c2cc(C)n(C3CCC(C)CC3)c2C)cc1C1CC1 c1(N2CCC(F)(n3cc(Cc4c(C)noc4)nn3)C2)ncc2c(n1)NC(=O)C2 c1(CC)ncccc1C(=O)N(CC(=O)Nc1ccc(OC)cc1)CCN(C)C C1(O)(C(C)NC(=O)Cn2ccc(C3CC3)n2)CCN(C(C2CC(F)C2)=O)C1 [N-]=[N+]=NC1CC(C(N2CCC(F)(CO)C2)=O)N(C(=O)C2=CC3C=CC2C3)C1 Cc1cn2cc(C(=O)N(C)CC3CCCCN3C(=O)C(C)n3ccnc3)sc2n1 C1(C(=O)NCC=CCNC(C(C2CCC(C)(C)CC2)C)=O)CC(C(C)(C)C)=NO1 C(C)(C(F)(F)C(F)(F)F)NC(C(C)Oc1ccc(Cl)cc1)=O Cc1cnc(N2CC=CC(OC)C2)c(S(=O)(=O)N2CC3CCOC3C2)c1 N1(C(c2nccc(OC)c2)=O)CCC2CCCC(C1)N2C(C1CCS(=O)CC1)=O c1(C(=O)NC2COCCN(C(=O)CC3CCC3)C2)ccc2c(c1)S(=O)(=O)NC=N2 C1(N(C(c2c(SC)ccs2)=O)C)CCCN(C(=O)C(C2CC(F)(F)C2)O)C1 Cc1nc2ccc(C(N3CC4CC(C3)N4C(=O)CCC(C)CN(C)C)=O)cc2[nH]1 C(CC(C)C(=O)NCC(CC(C)C)NC(c1c(Cl)n[nH]c1C)=O)OC C=CCC(CCC=C)NC(=O)CN(C(=O)C(C=C)CC)C(C)C C1(C(=O)NCC2(C)N=C(C)SC2)CC2(C1)CN(C(c1ncncc1N)=O)C2 C1(C)(C(N(CCCCCC=C)C)=O)CCCN(C(=O)C(C(C)C)NC(C)=O)C1 Cc1nn(C)c(Br)c1C(N1CCCC1Cc1ccccc1)=O CS(=O)(=O)c1ccc(-c2cc(CNCCCCCCCCCCO)ccn2)cc1 Cc1coc(C)c1CNC(C1(NC(=O)C(F)OC(F)(F)F)CC(O)C1)=O CC1(C)CCCCC1C(N1CC(C2CC2C(N2CC(C(F)(F)F)C2)=O)C1)=O N1(C(C(CCOCCO)NC(Cc2c(C)n[nH]c2)=O)=O)CCOC(C)(C)CC1 N1(C(=O)Nc2cn(CCOC)nc2)CCC2(CC1)CC2(C#N)CO c1(CC)cc(C)ccc1C(=O)NC(CNC(=O)C=CCN1CCOCC1)(CC)CC C(CNC(C1CCC1CNC(=O)CC1OCCC1C)=O)(C(F)(F)F)OC N1(C(c2scc(C(C)=O)c2)=O)CC2CCC(CNC(=O)C(F)(F)CO)C2C1 c1(C(=O)NCCOC(CNC(c2ccn(C)c2)=O)(C)C)cncc(P(C)(C)=O)c1 C12(OC)CCC(C(=O)NC(C)CN(C(=O)CCNC(c3ccco3)=O)C)(CC1)C2 c1(C(=O)NCC(CC=C)NC(=O)C(C)CCOC)ccc(Cc2nc[nH]n2)cc1 C1(O)(C(=O)NC2C(NC(C(C)(C)SC)=O)CCOC2)CCc2ccccc2C1 c1(C(=O)NCC#CCNC(C(C)C(F)F)=O)cc(N)c2ncccc2c1 C1(CCNC(C=CC(CC)C)=O)(N(C(=O)Cc2ccccc2)CC)CCCC1 C=C(C)C1OCCC1CN1CC(CC(=O)NCc2ccc(F)c(C)c2)C2(C1)CC2 Cc1cc(C(c2nnnn2C2CCOCC2)N(CCCN(C)C)C)cc(C)c1 C1(OC)CCC2(C(=O)NCC(C)CN(C)C(c3csnn3)=O)CC12 C1(C(=O)NCCN(C(C)C)C2CC2)CN(C(c2ccc(C3CC3)s2)=O)CCO1 C1(NC(Cc2c(C)con2)=O)CCN(C(c2nnsc2C)=O)C(C)C1 c1(C(=O)NC2CCCN(C(CCCN=[N+]=[N-])=O)C2)n[nH]c2ccc(Cl)cc12 N1(C(C(CC=CC)NC(C(CC[N+](=O)[O-])CC)=O)=O)Cc2nncn2C(C)C1 S(=O)(=O)(c1ccc(NCC(O)C2(Cl)CC2)c(Cl)c1)NC1C2(CC(OC)C2)C1 C(=O)(C1=CCCCC1P(C)(C)=O)N1C(CCNC(c2[nH]cc(CC)c2)=O)CCC1 CC1CC(NC(c2cccc(=O)n2C)=O)CCN1C(c1cc(F)c[nH]1)=O N1(C(CSCCC=C)=O)CCC(CO)(NC(c2oc(C3CC3)nc2C(F)F)=O)C1 C1(C(=O)NCc2c(C3CN(C(c4c(C)nco4)=O)C3)ocn2)CC(O)CN1C c1(CC(=O)NC2CCCC(NC(C3(C)CC(C)(C)C3)=O)C2)cc(O)nc(O)n1 Cc1nn2ncccc2c1C(N1CC2CCC(C1)N2C(=O)CN1CCC(C)C1)=O C1(NC(c2n(CC)ncc2Cl)=O)CN(C(=O)COc2ccc(O)cc2)CCC1C C1(NC(COCc2nnc(C)s2)=O)CC(C)N(C(=O)Cc2nccn2C)C1 N1(C(C=C2CCC(C)C2)=O)CCC2(CCCN(C(c3cnc[nH]c3=N)=O)C2)C1 O=C1CN(CC(=O)NCC2CCCC2)CCN1.C12(O)CCN(C1)C(=O)CNC2=O Cc1cccc(Cl)c1CC(=O)Nc1cccc(NC(=O)C(C)CN(C)C)c1 c1(C(N(C2CC(NC(=O)Cn3cnnc3O)C2)C)=O)c(OC(F)F)cccc1Br C(=O)(C(F)C(F)(F)F)N(C(C(=O)N(C1CN(C)C1)C)C1CC1)C c1(CC(=O)NC2CCC(CCNC(C3(N4CCOCC4)CC3)=O)C2)ccccc1 C1(NC(C2CCC(=O)N2)=O)CC2CN(C(=O)CCc3nc[nH]n3)CC12 N12CC(CC1=O)NC(=O)CCC(C)N2.c1(C(=O)OCC)ccoc1C1CC1 C1(C(=O)NCCCNC(CCN(c2ccncc2)C)=O)COC2(CCC2)CO1 c1(CN2C(COC(COc3cccc(OC)c3)=O)CC2)ccc(C)cc1Cl c1(OC)ccc(CC(=O)NC(C2CCN(C(C3CC(=C(F)F)C3)=O)C2)C)c(Cl)c1 C1(C(=O)NCC(CC)(CC)Nc2ncc(C#C)cn2)CCC2(CCC2)CC1 C(=O)(C(Cc1cnc[nH]1)NC(C1(NC(=O)CCNC(C)=O)CCCC1)=O)OCC c1(OCCC)ccc(Cl)cc1C(=O)NCC1CCN(C(=O)C=C2CCC2)C1(C)C n1(CC(=O)Nc2c(C)nc[nH]2)ccc(=NC(=O)c2cc(F)ccc2Cl)nc1O c1(C(N2CC(C)(NC(Cc3ncc(CC)[nH]3)=O)C2)=O)ccc2ncsc2c1 c1(C(C(=O)NCC2(C(N)=O)CN(C(C3C(C)OCC3)=O)C2)(C)C)ccc(N)cc1 c1(CC(C(=O)N(CCSC)CC)NC(=O)CNC(=O)C2CC2)ccc(Cl)cc1Cl C1(C(N2CCC(NC(CC)=O)C2)=O)CC2(CCN1C(=O)C#CC1CCC1)CC2 C1(N(C(C=C(C)Cl)=O)Cc2ccccc2)CCCN(C(=O)CC2CC2(Cl)Cl)C1 Cn1cc2c(n1)CCC(C(=O)NCCOCCCNC(c1cncc(Br)c1)=O)C2 N1(C(c2c(C)cccc2Cl)=O)CCC2(CC1)CC2(C)C(=O)N(CCC#N)C CON(CCC(=O)N1CCOC(C)(C)C1C)C(=O)c1ncnc(O)c1F c1(NCC(=O)NC2CCN(C(C34CC(OC)C3C4)=O)C23CC3)ccccc1[N+](=O)[O-] c1(OC(=O)CN2CCN(Cc3c(C)cc(Br)cc3)CC2)cc(Cl)c(Cl)cc1Cl C1(NC(C2C(OC)(OC)CC2)=O)CC2CCC1(C(N1CCC(C3(C)N=N3)C1)=O)C2 N1(C(=O)CC2CCN(C(c3ccn(C4CCCC4)n3)=O)C2)CCC(F)CC1 O=C1Cc2c(C(=O)NCC3C=CCN3C(C3COC(=O)O3)=O)cccc2N1 C(=O)(C(F)(F)C1CC1)NC(CNC(=O)C(c1ccccn1)O)C1CC1 CCC(CC(C)C)C(=O)N1CCC2C(C1)CN2C(c1cncc(C)c1)=O c1(CNC(CC(C)(C)O)=O)ccc(CNC(C2CC(=O)OC2(C)C)=O)cc1F c1(C(N(CC(C)N(C(CCNC(COC)=O)=O)C)C)=O)nccc(Cl)c1O C1(CNC(COC(CC)C)=O)CCC(CNC(=O)C(c2ccc(Cl)cc2)O)CC1 C1(C(=O)NC2(CO)CC(O)C2)CC2(CCN(C(C3OC4CCC3C4)=O)C2)C1 Cc1nc2c(s1)C(N(C)C(CCC(O)C(=O)OC(C)(C)C)=O)CCC2 Cn1ncc2nc[nH]c(=NC3CCCN(CC4(c5ccccc5)CC4(C)C)C3)c12 C(=O)(C(CC)C(C)(F)F)NCC1(F)CCN(C(c2c(CCC)nco2)=O)C1 c1(CC(=O)NC2CC(CNC(=O)CN3CCC(O)CC3)C2)cn2ccccc2n1 CCCC(CC)CC(=O)N(C1CN(C(=O)COC2CCC(F)(F)CC2)C1)C C1(N(c2cn[nH]c2)C(C2CCCO2)=O)CCCC12CCNCC2 c1(C(=O)NC2CN(C(C3(OC)CCS(=O)(=O)C3)=O)C2)cc2nn[nH]c2cc1F c1(C(=O)NC2CCC(CNC(C3CC4(CSC4)C3)=O)C2)cccc2cnnn12 C(CC(C)C)(C(=O)NCC(C)N(C)C(C1CC(F)(F)C1)=O)NC(=O)OC C=C1CC(N=c2[nH]c(=NC(CCC)CCO)[nH]c3cccc(F)c23)C1 C1(NC(=O)CN2CC3CC3C2)C=CCN(C(=O)CC2(c3ccccc3)CC2)C1 N1(C(C(CC)n2cccn2)=O)CCC(C(O)CNC(C2CCC23CCC3)=O)CC1 C1(SCCNC(C(CC2CCCCC2)OC)=O)CCCOC1(C)C c1(C(=O)NC(CNC(CC2CC(OC)C2)=O)C)ccc(CO)cc1 C1(C(N(CCCC(F)(F)F)C)=O)CC(F)CCN1C(=O)CCCCCF C1(CC(=O)N(CCOC(C)(C)CNC(=O)CCOC2CC2)C)CC(F)(F)C1 C1(CCNC(C=CCC)=O)CN(C(c2cc(N)ccc2Cl)=O)CCS1(=O)=O c1(NC(=O)NCc2ncc(C(C)(C)C)o2)ccc(-c2cn[nH]c2)cn1 Cc1cc(=NC(C)c2nncs2)[nH]c(=NCc2cnc(C(F)(F)F)s2)[nH]1 CC1CCC(CC(=O)NCC2COCCN2C(c2cc(CN(C)C)c[nH]2)=O)CC1 c1(NC(C2C3(CN(C(C(C)O)=O)C3)C2)=O)ccc(N(C)C)c(C(F)(F)F)c1 Cc1cc(F)cc(C(N2CCC(CNC(=O)CCCc3nccs3)C2)=O)c1C N1(C(C2CC(=C)C2)=O)CCC(F)C(NC(=O)C(C)(CC)CC)C1 S(=O)(=O)(c1ccc(F)cc1)NCC(F)(F)F.N12CCCN(CC1)CCCC2=O c1(CCC(=O)NCC2C=CCN2C(C2CCC(=O)N2)=O)ccc(F)cc1Br C(=O)(C1=C(c2ccccc2)CCCC1)NCCNC(c1csc(C)c1C1CC1)=O c1(C(=O)NC(CC)CNC(=O)CSc2nncs2)coc2c(C)cccc12 C1(F)(C(N(CCN(C(C(C)CSCc2cccnc2)=O)C)C)=O)CC2(CCC2)C1 CC1CCn2ncc(C(=O)NCC3CC(F)CN3C(=O)C#CC3CCCO3)c2C1 c1(C(=O)NCc2nc(N(CCOC)C(C)=O)sc2)ccc(O)c([N+](=O)[O-])c1 c1(C(=O)NCCOCC(N2CC(OCC)C(OC)C2)=O)ccc2[nH]ccc2c1F N1(C(c2cc(-n3ccnc3)no2)=O)CCOCC1c1cn(CC2CCCO2)nn1 N1(C(C(C)C(C)O)=O)CCC(F)(F)C(CNC(=O)CC2CCCCN2C)C1 CCC(CC)(CCNC(=O)C1=CC(C)(C)C1)NC(=O)CC1CCCC1C c1(C(=O)NC2C(C)CN(C(c3ccc(Cl)c(F)c3)=O)C2)ccc2c(c1)NC(=O)C2 c1(C(N2CCC(C)(NC(C3C(C(C)O)C3)=O)C2)=O)ccc(Cl)c(C#N)n1 S(=O)(=O)(CCC(=O)NCC1C(C)CCCN1C(=O)C(C1CCC(=O)N1)C)NC Cc1ncc2ccc(C(=O)NC3CCN(C(C4CCC(N(C)C)C4)=O)CC3)cn12 C(c1ccco1)=CC(N1CSCC1C(N1CCC1CO)=O)=O Cc1cc(C(N2CCC(CNC(C34CCC3C4)=O)CC2)=O)cn(C)c1=O c1(CC)c[nH]cc1C(N1CC(N(C)C(c2cc(C(C)C)[nH]n2)=O)C1)=O N1(C(c2c(CC)c[nH]n2)=O)CCN(C(C2CCC2)=O)CC1c1cnn(C)c1 C1(C#N)(C(N(C(C)CNC(=O)C=Cc2ccc(Br)s2)CC)=O)CCOC1 CC(C)C(C)CC(=O)NCc1ccc(C(=O)NC2CC(=O)N(C3CC3)C2)cc1 N1(C(C)C(=O)Oc2ccccc2)CC(COC(c2cnccn2)=O)OCC1=O c1(CC)cncc(CNC(=O)OC(C)(C)C)c1.C(C)(CC)(C(=O)ON)NCN N1(C(CCCOCC)=O)CCC2CCN(C(C3CCOC4(CCCC4)C3)=O)CC12 c1(CN2CCC(CNC(c3nn(C)c(O)c3)=O)C2)ccc(F)c(S(C)(=O)=O)c1 C1(OC)CN(C(=O)CC2(C)CCN(C(C3(CO)CC3)=O)C2)CC1F c1(CC(N2CC(NC(C3C(C)(C(F)F)C3)=O)C2)=O)cc(C(F)(F)F)co1 C(C(C(=O)N(CC(=O)N(CC(C)(O)CO)CC)C(C)C)NC(N)=O)OC c1(-c2n(CC=C)nc(-c3cc(N(C)C)ccc3Cl)n2)cnc2ncn(C)c2n1 S(=O)(=O)(c1cccc(CNC(=O)C(=O)Nc2ccc(C#N)nc2Br)c1)NC C1(C(=O)NC(C(N2CC(C(C)OC)C2)=O)C2CCCO2)CC(C)(C)CCO1 c1(OC)ccncc1-c1nc(-c2ccsc2)nn1CCc1ccccc1 c1(C(N(C2CCCN(C(=O)C(C)(C)C3CCCO3)C2)CC)=O)cn(C)nc1O c1(CNC(=NCCF)NC2CCN(CC3CC3)C2)cccc2c1OCC2 C(=O)(C1=CCC(NC(=O)CCc2ccn(C)n2)C1)NC1(C)CC(C(=O)OC)C1 c12ncc(Br)nc1C(=O)N2.c1(C(N(CCCC)CCO)=O)ccc(OC)nc1 S(=O)(=O)(c1ccc(NCc2ccccc2Br)c(F)c1)N(C)Cc1ccn(CC)n1 C1(C(=O)NC2CCN(C(C(C(C)OC)N(C)C)=O)CC2)C2CCC(F)(F)C12 N1(C(CN(C)Cc2cnccn2)=O)CCN(C(C2(CC(C)=O)CCCC2)=O)CC1 Cc1cccc(F)c1C(=O)NCC1CC(C)N(C(=O)Cn2cc(N)cn2)C1 CCCS(=O)(=O)NC(C)C(=O)NCC1(C(C)NC(c2csc(=N)[nH]2)=O)CC1 N(C(=NCCC1CCOC1)NCc1ccc(C)cc1C)CC(C1CC1)OC C(=O)(C1=C(C)S(=O)(=O)CC1)N1CC(CNC(c2ccc(CC)cn2)=O)CC1(C)C c1(C(=O)NC(CC)CNC(c2cn(CC(N)=O)nn2)=O)cc(O)nc(C2CC2)n1 C1(C(=O)NC(c2cn(-c3ccc(C)cc3C)nn2)CC(N)=O)CN(C)C(=O)CCO1 C1(C)(C(=O)NC)CCCN(C(=O)C)C1.Cc1ccc(C(=O)O)cn1.N12CCCC1C2 c1(CCCC)ccc(CN2CC(NC(c3cn(C(C)C)nn3)=O)C(C(=O)O)C2)cc1 c1(CN(C)C(=O)NCc2ccccc2)cccc(OC2CC2OC(C)C)c1 C(=O)(C(CC(C)C)NC(=O)NCC1CC(OC(F)(F)F)C1)NCC(=C)C C(=O)(C(C)(C)C(O)C(C)C)NCC1C(NC(Cn2nc(C)c(Cl)c2C)=O)CC1 Cc1cc(C(=O)NC(C2CCOC2)CNC(c2ccnnc2O)=O)cc(C)c1F N1(C(C(C)c2ccco2)=O)CC(C)(NC(=O)C(F)Cc2ccccc2)C1 c1(NC(=O)NC(CC#CC)C)ccc(Oc2ccccc2COC)nn1 c1(C(=O)OCC)ccc(NCC(C)CNC(=O)Cc2ccoc2)nc1 [N-]=[N+]=NCCCCNC(c1csc(CNC(=O)C(O)C2CC2)c1)=O N1(C(c2ccn(CC)c2C)=O)CCCC(C2CC2NC(c2ccc(F)s2)=O)C1 c1(N2CC3(C(NC(C4N(C)C(=O)CC4)=O)CCS3)C2)nc(Cl)nc2ccccc12 C1(C(=O)OC)CCC2(CCOCC2)N(C(=O)Cn2cc(-c3cn(C)cn3)nn2)C1 c1(C(N2C(CNC(c3[nH]cc(CC)c3)=O)CCC2)=O)nccc(C(F)(F)F)n1 N1(C(NNC(C)C(C)(C)C)=O)CC2OCCN(Cc3ccccc3)C2C1 N1(c2ncc(C#N)cc2F)CC2CCCC(NC(=O)C=CCO)C2C1 CC1(C(=O)NC(CNC(c2ncc(F)cc2N)=O)C2CC2)CCCCC1(F)F C1(CNC(c2c(F)ccc(C)c2)=O)CN(C(C23CC(C#N)(C2)C3)=O)C2(CCC2)C1 C12(C(N3CC(NC(C(C)c4cc[nH]n4)=O)C3)=O)CC1COC21CCC1 N1(S(CC2CCN(C(C3CCCCC3)=O)C2)(=O)=O)CCC2(CC1)C(O)CC2O C1(NC(c2c(OC)n[nH]c2)=O)CN(C(C2CSCCS2)=O)C(C)(C)C1 N1(C(CCCNC(=O)OC)=O)CCCCC1C(=O)N(CC(C)CO)C n1(CC)c(CN2CCC(C3CCOC3)C2)nc2cc(Cl)ccc12 N1(C(C2C(CCOC)C2)=O)CCC(C)(C(=O)NC(c2ccsc2)C)C1 c1(C(N(C2CCCN(C(C3C(C)C3C)=O)C2)CC)=O)ccncc1Br c1(C(=O)NCCC2CCC(NC(c3cc(Cl)cs3)=O)C2)cc(F)c(O)c(F)c1 CC1CN(C(C2(NC(=O)Cc3nc(=N)[nH][nH]3)CCC(C)(C)C2)=O)CC2(CCC2)O1 C(=O)(C(C)(C)C(=O)OC)NC(CN(C(CCCC=C)=O)CC)C c1(C(=O)OCC(N2C(C(C(=O)OC)(C)C)CCC2)=O)ccc2c(c1)OCO2 S(=O)(=O)(c1ccccc1C1(C)N=N1)N(C(C)C)CC1CC1 c1(C(=O)NCC2CN(C(c3ccnc(CC4CC4)c3)=O)C2)cncc2[nH]ccc12 C1(OCCNC(=O)Cc2cscn2)CCN(C(c2cnc(-c3ccsc3)s2)=O)C1 CC1(C)C(C)(C(N2CCOC(CNC(=O)CC3CCC(O)C3)C2)=O)C1(C)C C1(NC(C2C(C)C2C)=O)CN(C(c2cc(F)c(Cl)cc2Cl)=O)Cc2nccn2C1 CCCC(CC)CCC(=O)NC1(CN(C)C(c2ncoc2COC)=O)CC1 CC(C)C(F)(CNC(C1CCC(C)C1)=O)C(=O)O N1(CC)CC(F)C(F)C1.c12cc([nH]n1)C(=O)NC1CC(C1)CC(=O)N2 C1(NC(=O)NCC(=O)NC(CNC(C2(CO)CCCC2)=O)CO)CCCCC1 C(=O)(C1Cc2ccccc21)N1CC(=O)NCC1C(=O)NCc1ccnc(O)c1 N1(C(COCCC)=O)CCN(CC(C)(C)NC(C2CC2C)=O)CC1 c1(C(=O)NCC(C)CNC(c2coc(C3CCC3)n2)=O)ncccc1Cl CC1(CNC(c2cc(C3CCC3)on2)=O)CCCN1C(c1sccc1F)=O N1(C(C2C(CC)C2)=O)CCCC1CN(C(=O)C(c1cnn(C)c1)C)C c1(C(CNC(N(C)Cc2ccn(C)c2)=O)(C)O)cccc(Cl)c1 N1(C(C2CCN(C(CC)=O)C2)=O)CCC(O)(CNC(c2nc(C)sc2C)=O)CC1 c1(-c2nc(-c3csc(C)c3C)on2)ccc(Br)cc1O c1(C(N2CCCC(N(C(CC3(C=C)CC3)=O)C)C2)=O)cc(C)nc2c1cnn2C CC1COc2ccc(C(=O)NC3CC4C3CCN4C(=O)C=Cc3ccco3)cc21 C1(O)(CNC(C(C)=CC2CC2)=O)CCCN(C(c2ccc(O)nn2)=O)CC1 c1(OC)cnc(C(=O)NCCC2(O)CCN(C(C3CC3F)=O)C2)nc1 c1(C(N2CC(CNC(C=CCOCCOC)=O)C2)=O)csc(CCP(C)(C)=O)n1 C(=O)(C1=NOC2(CCN(C(c3cnc(OC)cn3)=O)CC2)C1)NCCCSC c1(C(N2C(CNC(c3ccc[n+]([O-])c3)=O)CC2)=O)cccc(Cl)c1O n1(CC)c(C(=O)NCc2csc(C(N3CCCC3C(C)O)=O)c2)cnc1O c1(C(=O)NCCC(C)NC(=O)Cc2cnccn2)cc(C2(C)CC2)on1 c1(SC)cc(C(N2CCC(N(C(=O)CC(C)C3CC3)C)C2)=O)cc(Cl)c1 Cc1nsc2ncc(C(=O)NC(C)(C)CN(C)C(C3(C)CCCC3O)=O)cc12 c1(CCC(=O)NCC2(CN(C(C(C=CC)O)=O)C3CC3)CC2)ccc(=N)[nH]c1 Cc1cc(-c2cn(CC3CCN(C(C4C5C(=O)OCC45Br)=O)C3)nn2)ccc1F Cc1ccc(CC(N2CCC(C)CC2CNC(=O)CC2COCCO2)=O)cc1C C(C(C)(C)CCO)NC(c1cccc(Cl)c1)c1n(CCC(=O)OCC)nnn1 N1(C(CC(COC)C)=O)CC2(CCN2C(c2nccc(OC)c2O)=O)C1 N1(C(C(c2cn(C)nn2)NC(C(CC=C)C)=O)=O)CC2(CCOC2)C1 C(=O)(C1=C(C)CCOC1)NCC(CCNC(C1CC(C)=C(C)CC1)=O)O N1(C(c2cnc(C)[nH]2)=O)CCC(O)C(C(=O)NC(c2ccccc2C)C)C1 N1(CCCCCCC)Cc2ccccc2CC1CNC(=O)C(C)OCCC(C)C c1(C(C)=O)cc(NC(C2CC3CC3N2Cc2cn(C)cn2)=O)ccc1F c1(NC(N2CC(CO)CC(C(C)(C)C)C2)=O)cc(Cl)nc2ccccc12 CCC(C)(O)C(=O)N(C1CCN(C(c2sc(NC(=O)C3CC3)cc2C)=O)CC1)C C#CCC(CC(=O)NC(COC)C1(C)CC1)NC(=O)CC1(N(C)C)CCC1 N1(C(c2c(C)n[nH]c2)=O)CCC(NC(C2(N(C)C)CCCOC2)=O)C(F)C1 C(c1c(C)cc(C)cc1C)=CC(=O)NCC1CN(C(CC(C)SC)=O)C1 c1(C(C)C)ccc(OCCC(=O)NCC2CCN2C(C2C(C)(C)C2(F)F)=O)cc1 c1(CCCSCC(=O)NC(c2ccccc2)CNC(C2CC2CF)=O)ccccc1 c1(C(C(=O)OC)N(CC(=O)OC)CCNC2CCOCC2)cc(F)cc([N+](=O)[O-])c1 CCCC(CCC)=CC(=O)NC1(C(=O)NCC2(N(C)C)CCC2)CCOCC1 N1(C(C(CC#C)C2CC2)=O)CCN(C(=O)CC(O)C(C)C)C2(CCC2)C1 Cc1nc(C(=O)C(=O)NC(C2CCOC2)CNC(c2ccsc2Cl)=O)cs1 C1(C(N(CC(CNC(C(C)OCC)=O)C)C)=O)Cc2cc(C)ccc2S1 C(=O)(CC(O)CNC(=O)CCCOC(C)(C)C)NC1CC(C)(C(=O)OCC)C1 Cc1cc(CCC(=O)NC2CC2NC(=O)CCc2ncc(F)cn2)cc(C)n1 CC1=CCSC1C(=O)NCC(CO)NC(=O)CCn1ccnc1 CCCCCC(CC)C(=O)NC1CC1NC(c1cn(C)c(C)cc1=O)=O Cc1cccc(CN2CCCCC2C2CC2)c1.C1CCC=CC(=O)N1C C(=O)(C1CCCc2nc[nH]c21)N(CCC(C(C)(C)C)NC(c1cncs1)=O)C C1(NC(C(C2CC2)OC)=O)Cc2ccccc2C1N=c1[nH]nc(C)s1 C1(COC)CCN(S(=O)(=O)NC2CCCN(Cc3ccccc3)C2)C1 c1(CC(=O)N(CCCC(=O)O)C)ccccc1O C(=O)(CC(CC(C)C)NC(c1c(C)ccnc1O)=O)NC(C=C)C1CC1 N1(C(CC2N(C(c3ccc(C)c(O)c3)=O)CCCC2)=O)CCCN(C=O)CC1 C(C)(CC1CCC1)(C(=O)N(CCNC(=O)CCCCO)C1CC1)OC C#Cc1ccc(C(=O)NC23CCN(C(=O)Cc4nocc4C)CC2C3)nc1 c1(C(=O)NCC(CNC(C(C)(C)OCC)=O)(C)O)cnn(CCC(C)C)c1C c1(CC2CC(OCC3CCCC(=O)N3)C2)ccc2c(c1)OCO2 c1(NC(=O)CC2CCCN2C(C2CC(O)C2)=O)nc(Br)ccc1O c1(C(=O)NCC2OCCC(NC(c3cc(C)ns3)=O)C2)cc(S(N)(=O)=O)co1 c1(CC)cc(C(N2CCCOC(CNC(C3SCCS3)=O)C2)=O)c2c(c1)CCO2 Cc1c(CC(=O)NC(=O)Cn2cc(CC3CC3CO)nn2)cnn1C c1(C(C)=O)cccc2ccc(NC(c3ccccc3)CC3CC3)nc12 C1(C(N2CCC(NC(Cc3n[nH]c(=NC)s3)=O)C2)=O)CCS(=O)(=O)C12CCC2 CC1=CCC(NC(=O)NCCC2CCN(C(=O)Cc3ccccc3)C2)CC1 c1(NCCc2cccc(OC)c2)ccc(S(=O)(=O)NC2CCS(=O)C2)c(Br)c1 CC1(C2CCC(=O)N(CCNS(=O)(=O)CC3CCC4(CCCC4)O3)C2)CC1 C1(C)(NC(CC(C)SC)=O)CCN(C(C2(F)CCOC2C)=O)CC1 C(CCF)(C(=O)NOCC(C)O)NC(CC(CC)SC)=O c1(C(N(C2CCN(C(C(C(C)(C)C)N(C)C)=O)C2)CCO)=O)cc(Cl)c(F)cc1F C(=O)(C1=CC2CCCCCCC12)NCC12N(c3snc(C(C)C)n3)C(CC1)CC2 C1(C(N2CC3C(CNC(c4cnn(CC(F)F)n4)=O)(C3)C2)=O)CC12CCSCC2 c1(C(N(C(C)C(=O)NCCCn2ccnc2C)CCC)=O)ncn2ccccc12 c1(OC)ccc(F)cc1S(=O)(=O)N1CCN(Cc2ccc(Cl)c(O)c2)C(CO)C1 c1(CNC(COCC)=O)ccccc1CNC(=O)CSCCOC C1(C(=O)NCC(C)N(C(c2cc(CC)oc2C)=O)C)CC(=O)OC1(C)C c1(C(=O)NC(C2CCN(C(=O)CCC#N)C2)C)cccc(NC(N)=O)c1 C(C(C)(C)C(=O)NCCCN(CCO)C(c1ccoc1Cl)=O)N(C)C c1(C(=O)NC(CC)CN(C)C(c2cncc(C)n2)=O)cnc(N(C)C)c(Cl)c1 c1(C(C(=O)NC2COC2)N(C(C(=O)OC)C)C)ccoc1C C1(NC(C=C(C)C)=O)CC2CCC(C1C)N2C(C1CCCCCC1)=O N1(C(C(N2CCC(O)CC2)C)=O)CC2(CCCC2NC(=O)CCC(C)(C)C)C1 Cc1cn2cc(C(N3CC4CCC3C(CNC(=O)C(C)(C)C(F)F)C4)=O)nc2s1 c1(N2CC(C)OC(C3CC3)C2)nccc(=NCc2cnc(O)nc2O)[nH]1 C(CCCCNC(=O)C(F)(F)c1ccccc1)CCC(=O)O.c12cn(nn1)CC2 CC1(C)CN(C(=O)Cn2[nH]cnc2=N)CCC1NC(c1[nH]nc2ncccc12)=O c1(C(=O)NCCC2CC(NC(Cc3c(C)n[nH]c3)=O)CC2O)ccc(N)c(F)c1 Cc1cnc2nccc(C(=O)NC3CC(C)N(C(=O)Cc4sccc4C)C3)c2c1 n1(CC#C)cccc1C(=O)NC(C1CCCCC1)CNC(c1cscc1Cl)=O CCC(Cc1cccc(Br)c1)C(=O)NC(C)CC1CN(C(C2(C)CC2)=O)C1 C1(CCC2(C(CC)(C)C)N=N2)CCCN1C(C1CC(F)(F)C1)=O C=CC1CCN(C(C2CN(C(=O)C(CO)OC)CC2CCC)=O)C1 C1(C)(NC(C(CCC)C)=O)CCCN(C(C2CCN(C(=O)OC)CC2)=O)C1 C1(CNC(C2C(C)CC2)=O)CC2(CO1)CN(C(C1CC(n3cnnc3)C1)=O)C2 CCC(C)C(=O)NCC(=O)NC(CNC(=O)COC1CC=CC1)Cc1ccccc1 c1(CSCC)cccnc1C(=O)NC1CN(C(=O)CSC2CCCCO2)C1 C12(CCNC(c3cc(CC)c(CC)o3)=O)CCC(C1)N(C(=O)C(=O)N(C)C)C2 C1(C(N2CC(NC(CC(=O)NCc3c(Cl)cncc3Cl)=O)C2)=O)CC2C(C1)C2(F)F CC(C(F)(F)F)NC(=O)C(c1ccoc1)NC(C1CC12CC2)=O CCCC(CCC)CC(=O)NC(C)(C)CNC(=O)C(C)(C)COCC N1(C(C2(C(C)C)COC2)=O)CCC2(CCCN2C(=O)CCc2cncc(O)c2)C1 Cc1c(CNCc2ccccc2Nc2nnccc2C(F)F)[nH]c2ccccc12 N1(C(C(C=C=C)C)=O)CC23CCCC2(C1)CN(C(=O)CC1CNC(=O)C1)C3 c1(CC(C)C)ncccc1C(=O)NC(CNC(c1cncc(NC)c1)=O)C1CC1 N1(C(CCC)=O)Cc2ccccc2CC1CNC(c1nnn(C)c1C(F)(F)F)=O c1(OC)cc(C(N2CCC(SCC(c3cccc(Cl)c3)=O)C2)=O)n(C)c1 N1(C(CCC)=O)CCC2CCN(C(=O)C(CCSC)NC(N)=O)C2C1 N1(C(c2ccn(C(C)C)n2)=O)CCCC(C)(CNC(=O)C(C)(C)CF)C1 CCCCC(C)(F)C(=O)N1Cc2[nH]nc(C(=O)NCC3(O)CC(CO)C3)c2C1 N1(C(CCC(C)(C)C)=O)CCC(NC(=O)CC2CCOC(C)(C)C2)C(C)(C)C1 C1(COC)(NC(C2CC3CC3C2)=O)CCCN(C(=O)CCn2ccc(C)n2)C1 CC1CCSC1C(=O)NCCNC(=O)CN(C(C(=O)CCc1ccccc1)=O)C(C)C C(=O)(CC(C(F)F)N1CCCCC1)NCC(CO)NC(CCC(=C)Cl)=O C=CCC(C)(C)C(=O)N1CCC(C(=O)N(CCCC)CCCO)C(C)C1 N1(C(C2C(C=C)CC2)=O)CC(NC(c2ncc(C)cc2OC)=O)C(S(C)(=O)=O)C1 c1(SC)cccc(C(C)NC(c2cc(C3CCC3)n[nH]2)c2nnnn2C)c1 C12(CC)CCN(C1)C(=O)C1C(COC1)C(=O)N2.C1(C(=O)OC)(SC)CCC1 Cc1ccc(CC(=O)NC23CC(C2)N(C(=O)CNC(=O)CCCCO)C3)c(F)c1 c1(C(=O)NC(CCCNC(C2CCC(C)C2)=O)(C)C)cc2ncccc2[nH]1 C(CC(=O)NCc1cc(CC)cc(C)c1)(CC(C)C)NC(C1(C(CC)=O)CC1)=O c1(CC(=O)OCc2cccc3c2CCCC3)ccc(Cl)c2cccnc12 C1(NC(C2CC(C)(NC(c3c(COC)nn[nH]3)=O)C2)=O)CCCCC1CO C1(NC(C(COC(C)C)NC(C)=O)=O)CN(C(=O)C(F)(F)CO)CC1C Cc1ncc(NC(C2CCN(C(=O)CCc3ccccn3)C2(C)C)=O)c(C)c1C CN=c1[nH]c(C(N2CCCC(CNC(C3ON=C(C)C3C)=O)C2)=O)cs1 c1(C(C)C)ncc(CN(CS(C)(=O)=O)C(=O)OC(C)(C)C)o1 N1(C(c2nc(CC)sc2)=O)CCCN(C(=O)CCCC(C)(F)F)CC1C N1(C(C2CN(c3n(CCC4(C)CC4)nnn3)C2)=O)CCN(c2cc(Cl)ncn2)CC1 CCCCCCC(C)C(=O)N(CCC(=O)NCCc1ccccc1)C1CC1 C1(NC(C(C)n2cnnn2)=O)(CNC(=O)C(C)C(F)(F)F)CCC(C)(C)CC1 c1(C(n2nnc(C3(OC(C)(C)C)CCOC3)n2)C(=O)O)ccc(Cl)cc1 CN1CC=C(CC(=O)N2CC3CCC(C(=O)NCC4(NC(N)=O)CC4)(C3)C2)CC1 c1(CC(N)=O)ccc(C(=O)NCC(O)CCNC(=O)CNc2ccccc2)cc1 C(=O)(C(C(C)(C)C)OC(C)(C)C)NC1CN(CC(=O)NCC(C)C)CC1C C(=O)(C1=CCC(C)(C)CC1)N1CC(C(C(=O)NCCn2ncnn2)OC)C1 c1(C(CC)OC(C(C2CCOCC2)OCC)=O)ccccc1 N1(C(COCC(=C)C)=O)CC(CCNC(=O)CCCC2CCC2)OC(C)C1 c1(CC(=O)NC2CN(C(c3c(CC)cccc3)=O)C2)cc2c(cc1Br)OCO2 n1(CC)ccc2ccc(NC(=O)C(n3cc(CC4CCCCN4C)nn3)C)cc12 N1(CCC(C)NCC23CCC(C(=O)OCC)(C2)CO3)C(=O)c2ccccc2C1=O C1(C(=O)NCC(C2CCN(C(=O)CSC(F)F)CC2)F)CC2(CCC2)C1 c1(C(N(CCOC)CCNC(C2C3CCC2CC3)=O)=O)cccc(C)c1Br N1(C(CN(C)C(=O)C2CC2)=O)CCC2(C1)CN(C(C1CCCC3CC13)=O)C2 c1(NC(C2C(C(=O)Nc3n(C)nc(C)c3Br)C2)=O)ccc(C#N)c(Cl)c1 c1(OC)ccccc1NC(c1ccc(-n2cccn2)nc1)c1nnnn1C N1(C(C2C(C)=CCS2)=O)CCCCC1c1ccc(F)cc1 N1(C(CNS(CCOCC)(=O)=O)=O)CCN(C(=O)C(C2CC2)OC)CC1C(C)C C1(C)(C(=O)NCC(C)N(C(c2cc(COC)on2)=O)C)CCNC1=O C12(C(=O)NCC3(O)CC(CNC(C4CS(=O)(=O)C4)=O)C3)CCC(CC1)CO2 C(=O)(C(CC(C)C)C(N)=O)NC1C(CNC(c2cc(C)c(O)nn2)=O)CC1 CC1CC(C(=O)NC2COC(C)(C)C2)CCN1C(C1CC2(C1)CC(O)C2)=O c1(C(N2CC(C)C(NC(=O)CN3CCCCC3)CC2)=O)c[nH]c2ccc(Cl)cc12 CC1(C)CC(O)(CC(N2CCC(F)(CNC(=O)C=Cc3ncco3)CC2)=O)CO1 N1(C(C2C=CC=CC=C2)=O)CC2CCN(C(C3CC(C(F)(F)F)C3)=O)C2C1 Cc1cc(C(=O)N(C)CCN(C(c2c[nH]nc2C)=O)C(C)C)ccc1Cl c1(C(=O)NCC(CC=C)NC(c2cccc(C(C)C)n2)=O)c(C)ccc(C)c1O N1(C(c2c(C)oc(C#N)c2)=O)CC2CN(C(=O)C=Cc3cncc(F)c3)CC2C1 C(=O)(C=CS(F)(F)(F)(F)F)NC(C)(C)CCNC(C12CC=CC(C1)OC2)=O N1(C(c2sc(C)c(O)n2)=O)CCN(C(=O)CN=S(C)(C)=O)CC1CS(C)(=O)=O Brc1ccccc1C1(NCc2noc(Cc3ccco3)n2)CC1 C1(C(N2CC(CCC)C(CO)C2)=O)CCN(C(=O)Cc2ccon2)O1 c1(CC)ccc(OC)cc1C(N1CC(NC(=O)CN=S(C)(C)=O)CCC1C)=O C1(NC(CC2(OCC)CCC2)=O)CCN(C(=O)C(C)OC)CC1F N1(c2snc(C(C)C)n2)CC2(COC(CNC(c3cnc(Cl)s3)=O)C2)C1 n1(CC)ncc(C(N2CC(NC(=O)Cn3cnnn3)C(SC)C2)=O)c1C1CC1 N1(C(CCCCCC)=O)CCOC2(C1)CN(C(C1(F)CCCC1)=O)C2 C(C)(C(CC)CC)NC(c1ccc(CNC(c2ccc(CC)s2)=O)o1)=O N1(C(C(=O)NCCC)c2cocn2)CC2C3CCC(C3)C2C1 CC(CNC(=O)CCc1cnn[nH]1)C(=O)NCc1nc(C2CC2)n[nH]1 C1(NC(c2cncs2)=O)CN(C(=O)Cc2cnsc2)CC1C1CC1 c1(CCC(=O)N(CCNC(C2CCCCN2C)=O)CC)cccc(F)c1Cl N1(C(CN(C2CCC2)C)=O)CC2(CC(NC(C3(C)COCCO3)=O)C2)C1 C1(NC(CC2CN(C)C2)=O)CN(C(C2(C)CNC(=O)N2)=O)CC1CO CC1CCCCCC1NC(C1OCCC1NC(C1CCCC1O)=O)=O Cc1ccc(F)c(N)c1C(N1CCN(CCNC(C2CCC2)=O)CC1)=O N#Cc1ccc(C(=O)NCC2(F)CCN(C(c3ccc(Cl)cn3)=O)CC2)cc1Cl CCC(CCC(=O)Nc1cnccc1CO)NC(=O)C=Cc1cc[nH]n1 N1(C(C2CCC(SC)C2)=O)CCC(CNC(c2c(Cl)n[nH]c2C)=O)CC1 C(=O)(C(C#N)C(C)(C)C)N1CCC(CC#C)(C(=O)NCC2(OC)CN(C)C2)C1 c1(OC)ccc(N=c2scc(CC3CCCO3)n2-c2cccc(SC)c2)cc1 C(=O)(C(F)CC(C)(C)C)N1C(CNC(C2C(CC)C2)=O)COCC1 C=CC(C)(O)C(=O)NCC1CC(F)CN1C(=O)COC(C)=O c1(C(=O)NCC(C2CCCC2)NC(C2=NOC(C)C2)=O)cc([N+](=O)[O-])cnc1O C1(CC(C(=O)NCCCF)N(CC(CC)CC)C)CCC(F)(F)CC1 C1(O)(C(=O)NC2CCCN(C(c3c(C)n(C)cn3)=O)C2)CCOC1(C)C C1(NC(=O)CCCC2CCCCC2)CN(C(C2CC(O)C2)=O)CCC1C(F)(F)F c1(NC(C2CC(CC(=O)NCC(F)CO)C2)=O)ccc2cccnc2n1 C(=O)(C#CCNC(=O)CN(C)C)NC(C#C)(C)C1CC1 c1(C(C)(C)C)ccc(NC(C2CCCN2CCCOCc2ccccc2)=O)cc1 C1(NC(CNC(C)=O)=O)CCN(C(c2ccc3cn(C)nc3c2)=O)CC(C)(C)C1 C1(=CC(=O)NCC(CNC(c2c(C)nsc2Br)=O)C)CCCCC1(C)C CC(C)C(CNC(=O)C=Cc1ccncn1)C(=O)N1CC2CC2C2CC12 c1(NC(C2C=CC(NC(c3cccc4ncsc34)=O)C2)=O)cccn2ncnc12 C(=O)(C1Cc2c(Cl)cccc21)N1CC2N(C3CCN(CC=C)C3=O)C(CCC2)C1 N1(C(c2c[nH]c(=NC)s2)=O)CC2(CO)CC1(C(=O)NCC(O)C(C)C)C2 c1(C(=O)NC2(CC=C)CCN(C(COCCCC#C)=O)C2)cnc(F)cc1C O(NC(=O)C(C)CNC(C1(OCC)CCC1)=O)CCCCC N1(C(C=C(C)c2ccco2)=O)CCC2CCN(C(c3oc(C)cc3C)=O)CC2C1 c1(C(C(=O)NC(C)C(C)NC(=O)C(F)(F)C(C)(C)O)(C)C)c[nH]c2ccccc12 CC1(C)CC(=O)OC1CNC(=O)C=CCNC(c1cccc(F)c1O)=O c1(OC)ccccc1CCNC(c1cncc(-c2ccncc2)n1)=O C1(C(C(=O)NCCC2(CNC(COC)=O)CC2)F)CCOCC1 N1(C(C(n2cc(CCN(C(C)(C)C)C)nn2)C)=O)CCCN(S(N)(=O)=O)CC1 Nc1sc2c(c1C(=O)NCC1CC1CNC(c1ccc(=O)oc1)=O)CCC2 C=C(C)C(C)(C)C(=O)NCC1CN(C(=O)C(C2CCC2)OCC)CC1C C1(NC(C(C)Oc2cccc(F)c2)=O)CC(N=c2[nH]c(Cl)ncc2C(F)(F)F)C1 C(=O)(C(=O)CCC(C)(C)C)NCCN(C(=O)C=Cc1ccncc1)CC N1(C(c2cccc(C)c2N)=O)CC2CC1CCC2NC(=O)CC(C)C n1(CC)nc(C(=O)NC23CC(NC(=O)C(CCN(C)C)N(C)C)(C2)C3)c(C)n1 CCC(CC)C(=O)N1CC(CCNC(c2ccc(-c3ccccc3)o2)=O)C1 c1(OC)cc(C)ccc1C(N1CC(F)(C(=O)NCC2COCCO2)C1)=O N1(C(C(CC)CC)=O)CC2CCC(N(C)C(c3ncc4[nH]ncc4n3)=O)C2C1 Cn1ccc2ccc(C(=O)Nc3ccc(NC(c4cc(O)no4)=O)cc3F)cc12 c1(C(N2CC(NC(C(CC)(C)CC)=O)C(N=[N+]=[N-])C2)=O)ccc(F)c2c1CCC2 C1(NC(C(CSC)O)=O)C2CN(C(=O)CCOCC(C)C)CC12 C1(O)(C(C)NC(C)=O)CCN(C(c2cccnc2-c2ccncc2)=O)C1 C1(C(=O)NCCC2(O)CN(C(C3CCCN3C(C)C)=O)C2)(CC)CCCC1 N1(C(C(C)OCCC#C)=O)CCC2(C1)CN(C(=O)Cc1sc(C3CC3)nc1C)C2 Cc1nc(-n2nc(C3CCCO3)nc2-c2cc(N3CCCCC3)on2)n(C)n1 N1(C(CC=CC=C)=O)CCC2CCCN(C(c3nc4ncc(C)cn4n3)=O)C2C1 N1(C(c2ccc(OC)c(O)c2)=O)CCCC2C1CCCN2C(C12CSC(C1)C2)=O C(=O)(CC(C(C)OC)NC(c1ccc(O)cc1F)=O)N(CC=C)C c1(C(N2CCC(C(C)NC(c3ocnc3C3CC3)=O)C2)=O)cccc2ncnn12 c1(C(=O)NC2CN(Cc3c(F)cccc3F)CC2F)ccc2c(c1)C(=O)CC2 N1(C(C2C(COC)C2)=O)CCN(CC(C)(C)NC(c2cncc(CO)c2)=O)CC1 CCCC(O)CC(=O)NC(C)(CNC(c1cn(CC)nn1)=O)CC(C)C C1(NC(CC2(CN(C)C)CCC2)=O)(CF)CN(C(C2CC2CC(C)(C)C)=O)C1 C1(C(C)C)CC(c2nnnn2CC2CC2)(NCc2cccnc2Br)CS1 C1(NC(CCOCCC)=O)CC2CC(NC(=O)CCC(C)SC)C2C1 c1(OCC(=O)N(C(C)CCNC(=O)C(n2cc(Br)cn2)C)C)ccc(O)cc1 c1(C(=O)NC23CCC(C(=O)NCC4(O)CCCC4)(CC2)C3)c(F)cccc1Cl C(=O)(CC(C(F)F)NCC1NCCC1C1CC1)OCC N1(C(C2(CC#C)CC2)=O)CCCCCC(NC(=O)C(CC=C)NC(C)=O)C1 Cc1noc(C)c1C=CC(=O)NCC(C(C)C)NC(=O)CC1(C#N)CC1 C(CC(=O)N(C1CC1)CC1CSCCS1)(C(F)(F)F)NC(C)=O C1(CCC)(NC(C2CCS(=O)(=O)C2)=O)CCCN(C(c2cc(C3CC3)cs2)=O)C1 CC(CN(C)C(C1CC2(CC2)C1)=O)C(=O)NC(C)C(C)(C)O CCS(=O)CC(=O)N(C)CC1(O)CN(C(=O)COc2cccc(OC)c2)C1 C(=O)(C(=O)Nc1ncc[nH]1)N(CCCNC)C N1(C(CC2N(C(C(C)(C)n3cccn3)=O)C3C2CCC3)=O)CC2COC(=O)C2C1 CC1(C)CCN(CC(=O)NC(C)(C)CCCCNC(C2CCNC(=O)C2)=O)CC1 Cc1ccc2[nH]c(C(=O)NCCNC(c3ncnc(O)c3F)=O)c(Cl)c2c1 c1(OC)ccnc(O)c1C(=O)NC1CC2(C1)CN(C(=O)C(CC1CC1)OC)C2 c1(-c2ccc(CCCC)nc2)cccn2ncc(C(=O)NCCC(C)C)c12 n1(CC)nnc(C)c1C(=O)NCC1C(C)CCN1C(c1ccc(C)cn1)=O C(=O)(CC(F)(F)C(C)C)NCC(C(C)C)(C)NC(c1cncc2c1CCC2)=O C1(CC)CCOCC1(c1nnnn1C1CCCCC1)NC1CCC(CO)CC1 N1(C(CCN(C(CC(CC)C2CC2)=O)CCO)=O)CCC(O)C(C)C1 c1(OC)ccc(C)cc1C(=O)NC1CCN(C(=O)CC2CCCC(C)C2)C(C)C1 N1(C(C2N(C=O)CCC2)=O)CCN(C(=O)Cc2cccc(F)c2O)C(C2CC2)C1 C=CCCCCC(=O)N(CC(C)NC(C1CC2(CC(OC)C2)C1)=O)C C(C)(CCC(=O)Nc1cnn(C)c1C)NC1C(CC)N(NC(=O)OC(C)(C)C)C1 c1(C(N2CCC(OCCNC(C3CCC(C)C3)=O)C2)=O)cccnc1S C1(CC=C)(C(=O)NCc2cnc(F)cn2)CNCCO1 CCC(CC(=O)NCCCCc1ncc[nH]1)NC(C1CCCSC1)=O C(=O)(CC1CC(=O)Nc2ccccc21)N(C(C)C)CCNC(C1CC=CCC1)=O N1(C(CC(C(CC)C)NC(=O)C(CCOC)OC)=O)CCC2C(=O)NCC2C1 N1(CC(Cc2ccccc2)OC)CC2CCCN(C(C3COCCO3)=O)C2C1 C12(C(N3CCCC(NC(=O)Cn4nnc(C5CC5)n4)C3)=O)COCC(C1)OC2 C1(C(=O)NC(CCCNC(c2cncc(OC)c2)=O)(C)C)CCCC2(CC2)C1 N1(C(CCC)=O)CCC2C(NC(c3ccc(C4(C)CC4)cc3)=O)C12 C=CCC(C(=O)N1CC(CNC(c2scc(C)c2OC)=O)C1)C(C)C c1(CCC)nc(-c2cncc(F)c2)nn1-c1cccc(Cl)c1 n1(COC)nccc1C(N1CCCC1CC(=O)NC1CC(F)C1)=O C1(CNC(CCSCC)=O)CC(C)N(C(=O)C=Cc2cn[nH]c2)C1 C(=O)(C(CCC1CCC1)NC(C1CC2(CC2)CO1)=O)NCC1CCC(C)C1 N1(C(C=CC(=O)OCCCC)=O)CCC(CNC(=O)Cc2cnn(C)c2)C1(C)C N1(C(C(C)OCC=C)=O)CCN(C(c2cc(NC(C)=O)ccc2Cl)=O)C(C#N)C1 N1(C(Cc2ccc(OC)nc2)=O)CC2CCCC1C2NC(=O)CN(C)S(N)(=O)=O c1(OCC)ccc(CN2CC(NC(C3CCCC3C)=O)C(F)C2)cc1Br Cc1nc2ccnn2c(C)c1C(N1CCN(C(=O)CC(C)CF)CC1C)=O N1(C(CC2CCN(C(C)C)CC2)=O)CCCC(O)(c2nn[nH]n2)C1 Cc1cc(Cl)c(C(=O)NCCCC(C)NC(=O)CSC(F)F)s1 C(=O)(C1=NOC2(CCC2)C1)N1CCC(C=C)(C(N2CCOC3CCCC23)=O)C1 C1(C(=O)NCC(CNC(C(C)C2CCC2)=O)F)CCn2c(O)nnc2C1 C(=O)(C(C)C(C)NC(C1CC(OC2CC2)C1)=O)NCCSC(C)C C(CCCC(=O)OC)OC.c12nc(co1)C(=O)NOCC(=O)N(C)CCO2 c1(C(=O)NC(C)CN(C(=O)C(F)(Cl)c2ccccc2)C)ccnc2ccsc12 C1(C(N(C2CC(F)(F)C2)C)=O)CCCCN(C(=O)Cn2cccn2)C1 C1(CNC(CCC(C)=O)=O)CCN(C(=O)C(C)CCOc2ccccc2)CC1C CC1(C)CCC(CNC(=O)CSC(F)F)(NC(=O)CC2COC3CC2C3)CC1 c1(C(C(=O)NCC(C)C)N(C(c2ccc(C)cc2)C)C)cn2ccc(Br)cc2n1 N1(C(CC(C(F)(F)F)OC)=O)CC2CC(NC(c3cnsn3)=O)CC(C2)C1 c1(OC)cccc(CCC(=O)NC(CNC(c2ccc(SC)o2)=O)CO)c1F C1(CCC)CN(C(=O)CCc2cccs2)CCN1C(=O)COCC1CCOC1 c1(OC)ccc(C(=O)NC(C)CCNC(c2c(C(C)C)cccc2F)=O)c(F)c1 c1(OC)ccc(C(C)C(=O)NCC(C)(C2CC2)NC(=O)Cc2cn[nH]c2)c(C)c1 N1(Cc2cn(CCNC3(C)CCN(C(CCC(C)C)=O)C3)nn2)CCSC(C)(C)C1 N1(C(C2(COC)CC2(F)F)=O)CCN(C(c2csc(C(=O)OC)n2)=O)C(CF)C1 C1(c2n(CCCSCC)nnn2)(NCCC2CC23CCC3)CSCCSC1 C(=O)(C#CC1CC1)NCC(CNC(c1oc(Br)cc1C)=O)OC Cc1[nH]nc(C(=O)NC(C)C(C)NC(=O)Cc2ccccc2O)c1C c1(OCC)cccc(CC(=O)NCCC(C)NC(=O)CCc2ccoc2)n1 c1(C(N2CCC(F)(CNC(c3csc(F)c3)=O)C2)=O)cnc2c(n1)CCCC2 C(=O)(CCCCSC)N1CC(C(=O)NOCC(C)(C)C)(CC)C1 c1(C(N2CC(NC(Cn3c(C)cc(C)n3)=O)C(F)C2)=O)c(Cl)cccc1Cl Cc1nc(C)c(CC(=O)NC2(CNC(=O)CC3CCC(=O)N3)CC(F)(F)C2)s1 N1(C(C(=O)NCC(F)F)=O)CCCC2(CNC(=O)C3=CCCS3)CCCC12 N1(C(CN(C(C)C)C)=O)CC2CCOCC2(NC(=O)C=CC2CCC2)C1 c1(CCC(=O)NCCC(C)N(C(CCCCOC)=O)C)nc2ccccc2[nH]1 N1(C(C2CC(C)(C)CC(O)C2)=O)Cc2ccnc(Cl)c2C1 C1(OC)CN(C(C2CCCC(C)C2)=O)CCC1NC(c1ccncc1Cl)=O C(=O)(N=c1nc(Cl)nc2[nH][nH]cc1-2)C1C(C(=O)Nc2cccc(C)n2)C1 c1(C(=O)NCC2(C)CCN(C(C3(C)CCC(=O)C3)=O)C2)cc2n(c1)CCCC2 CCC(O)C(C)C(=O)N1CCC(NC(=O)CNc2ccc(C#N)cc2)C(C)C1 C1(C(=O)NCC(CN(C(COCC)=O)C)(C)C)C2CCCCCCC12 N1(C(CC(COC)C)=O)CCC(NC(=O)Cn2nccn2)C(OC)C1 c1(NCC)cccnc1C(N1CCC(C)(NC(c2ncc(Cl)n2C)=O)C1)=O Nc1c(C(N2CCN(C(c3cc(Cl)no3)=O)C3CC23)=O)cccc1F C(C(=O)NOCc1cccnc1)(C1CCCC1)NC(C(CC)N(CC(C)C)C(C)=O)=O C1(NC(CS(=O)(=O)NCC)=O)COCCN(C(=O)C(N2CCCCC2=O)C)C1 c1(C(N(C)CC2C3CN(C(C=C(COC)C)=O)CC32)=O)c(C)[nH]c2ncccc12 C1(CC(=O)NC2CN(C(=O)Cn3nccn3)CC2F)CC2(CCCC2)CO1 c1(C(=O)NCCCN(C(=O)CCC(C)OC)CC)ccc2c(C)noc2n1 c1(CC(N2CC(CC(=O)NCc3c(C)cccn3)C2)=O)c(F)cccc1F Cc1cc(C)c(C(=O)NCC2(NC(c3cc(Cl)ncc3N)=O)CCCC2)c(C)n1 C(=O)(C(C)(C)CNCC1(O)CC(C(N2CCC(C(F)C(=O)NC)C2)=O)C1)NC C1(C)(C(=O)NC2CCC(NC(c3ncn(C)n3)=O)C2)CC2(CC2)C1 C1(C2CCC2)(C(=O)NCC=CCNC(C2(CCOC)CCC2)=O)CC1(F)F C(=O)(NNc1ncc(F)cn1)c1c(NC(=O)OC(C)(C)C)cccc1 C1(NC(=O)Cn2cnnc2)CCCCCC1NC(c1ccc(OC(F)F)cn1)=O C(CC(C(=O)NCC1CCC(=O)NC1)NC(=O)C(C(C)OC)N(C)C)=CC C(=O)(C(F)(F)C(F)(F)F)NC1CCCC(NC(c2ccncc2F)=O)CC1 Cn1ccc(=O)c(C(N2CCN(C3CCN(C(=O)Cc4cc[nH]n4)C3)CC2)=O)c1 C1(C(=O)NCC(C)CNC(c2nnc(C(F)(F)F)s2)=O)CCCC(C)CC1 CCCCCC(C)(C)C(=O)N(C)CCNC(c1c(C)sc(C)c1C#N)=O N1(C(C2CC(C)C2)=O)C2CCC1CN(C(c1ccnc(N3CCCC3)n1)=O)CC2 c1(C(=O)NCCN(C(=O)C(C2CCCC2)OCC)CCC)cccs1 c1(C(=O)NC(C)CCNC(C2CC3(C2)CC3(F)F)=O)ccc2n[nH]cc2c1Cl C(CCCCN(C)CCNC(=O)CCc1nncs1)OC c1(C(=O)NCc2scc(C(=O)NCC3N(CC)CC3)c2)ccc(C)c(O)n1 c1(NC(C2(CO)CCN(C(C3CC(OCC)C3)=O)C2)=O)nc(OC)ccc1C CN1CCc2ccc(C(=O)NC3CC3CNC(c3cc4cnccc4o3)=O)cc21 c1(C(C(=O)NC2CCN(C(Cc3ncc(C)s3)=O)C2)O)ccc(F)cc1 N1(C(c2ccn(C)n2)=O)CCOC2CN(C(c3ccc4nc[nH]c4n3)=O)CC12 c1(C(=O)NCC=CCNC(C2(CCC=C)CC2)=O)cnn(CC2CCOCC2)c1 C1(C(=O)NCC2CCCCN2C(c2ccc(CN(C)C)o2)=O)CCCCC12CC2 N1(C(CN2C(C)CCC2)=O)CCC(C2(O)CN(C(C3CC3(C)C)=O)C2)CC1 c1(CNCC2(NC(CS(C)(=O)=O)=O)COC2)cc(Br)ccc1[N+](=O)[O-] C(=O)(CC(C)CC(C)(C)C)N1CC(NC(c2nc(CC)sc2N)=O)C(C(F)F)C1 c1(NCCC=CC=C)ccc(S(=O)(=O)N2CCC(C3CCCCO3)C2)cc1F C1(NC(C2(C(=O)OCC)CCC2)=O)CCCN(C(=O)CN2CC3CC3C2)CC1 N1(C(C2CCN(C(C(=Cc3ccco3)C)=O)C2)=O)CCc2ncncc2C1 C1(C(N(CC)CC2CCCN2C(c2cocc2C)=O)=O)CCCN(C(=O)OC)C1 C12(OC)CCC(c3nc(-c4cc(C)n(-c5cccc(F)c5)n4)no3)(CC1)CC2 C1(NC(c2c(CC)n[nH]c2)=O)CC(F)CN(C(c2ccc(C)s2)=O)C1 N1(C(C(C)CC2CCC2)=O)CC(CNC(c2ccccc2CC#N)=O)C(C)(C)C1 CC(C#N)C(=O)N(CC(C)C(=O)NCc1nnn(C)n1)C C1(CNC(CCCOC(C)=O)=O)CN(C(=O)CCCCC(F)F)C2(CCC2)C1 c1(C(c2n(CCC(=O)OC)nnn2)NCCc2ccco2)ccnc(C2CC2)n1 CC1(N2CCCC2)CCC(NC(=O)CCSc2cccc(Br)c2)CC1 C1(C(N2CCC(OCC#C)C2)=O)CNC(=O)CN1C(=O)C(CC)CC Cc1csc(Cl)c1C(=O)NCC(O)CCNC(=O)C(C)C1CCCC1 c1(-c2onc(CC3(O)CC(C(=O)OC)C3)n2)nc2cc(Br)ccc2[nH]1 N1(C(c2cc(C)nc(O)c2)=O)C2CCC1CC(NC(c1cn(C)nc1O)=O)C2 N1(C(c2c(C)cc(F)s2)=O)CC2CCC(C1)N2C(c1cscc1C#N)=O c1ccc(-n2cccn2)cc1.C(CCC(=O)NCC(=O)NC(C)C1CC1)SC CCC(CNC(c1cnc(C(C)C)[nH]1)=O)(CC)NC(=O)C(C)N1CCC1 C1(C(N(CC(C)CNC(=O)CN(CC(C)(C)C)C)C)=O)CCS(=O)(=O)C(C)C1 Cc1cnc(C(=O)NC(CCC2CCC2)C(=O)Nc2cnc(F)cc2C)c(F)c1 c1(C(N2CCCC(CNC(C(CNC(C)=O)(C)C)=O)C2)=O)ccc2sccc2c1 C1(O)(CNC(C2C(C(N)=O)C2)=O)CCN(C(c2c(Cl)cccc2Cl)=O)CC1 C#CCC(O)C(=O)NCCCN1CCC(C(=O)Nc2ccc(C(N)=O)nc2)C1 C1(NC(CC(C)CNC(C2CC(=O)N(C)C2)=O)=O)CC2(C1)CN(C)C2 Cc1oc2ccccc2c1CNC(NC(=O)OC(C)(C)C)=S CCS(=O)CC(=O)N1CC(C)(CCC(=O)NC2CCOCC2F)C1 C(=O)(C1=CCN(C(C2COCCN2C)=O)C1)NCCC(C)N(C)C C(=O)(C(CNC(=O)C(c1cccnc1)O)CC(C)C)NC1CCN(CC)CC1C N(C1c2ccccc2CC1NC(=O)Cc1ccc(CO)cc1)C(C(CC#C)C)=O N1(C(c2c(C)nn(C)c2)=O)CCCC(C2CN(c3ccnc(C(C)(C)C)n3)C2)C1 c1(C(N(CCOCCNC(CC(CC)(C)C)=O)C)=O)cc2ccncc2s1 Cc1nc(CC(=O)NC2(C)CC(NC(c3csc(C4CCCN4C)n3)=O)C2)n[nH]1 C1(N(C(c2c(CC)cco2)=O)C)CCCN(C(=O)CCc2nccs2)CC1 C1(NC(Cn2cc(C3(C)CC3)nn2)=O)CCOC12CCCCC2 c1(C(N2CCC(O)(C(=O)Nc3n(C)nnc3)C2)=O)coc2ccccc12 CC1(C)CCCN(C(=O)CN2CCCC2)C1C(=O)NC1CCn2cnnc2C1 c1(CCC(=O)NC(CCNC(C(C(C)C)SCC)=O)C)cnc(C)nc1O C=CCC(C)(C)CC(=O)N(C)CC1CCCN1C(C1(C)CC=C(C)CC1)=O N1(C(C(=O)NCC2CCN(C(c3c(COC)noc3)=O)C2)C)C(=O)CCC1=O S(=O)(=O)(c1cnccc1N1CCC(F)(CF)C1)N(CCN(CC)CC)CC c1(C(=O)N(Cc2ccncc2)Cc2ccsc2)csc(-c2ccco2)n1 c1(CC)ccoc1C(=O)NC(CC1CCCC1)C(=O)NCC=CCl C(=O)(C1=CCCO1)N1CC(C)(OCC(N2C(C#C)CC2)=O)C1 C1(CC(N)=O)(NC(CCCSC)=O)CCN(C(C2C3CS(=O)(=O)CC23)=O)CC1 c1(CN(CCCN(C(C2C(C)C2C)=O)C)C)nnnn1CC(F)F C1(CNC(c2c(CC)c[nH]n2)=O)CC(C)(C)CN1C(=O)CCC1CCCCC1 C(=O)(CC(CN)C(F)(F)F)Nc1c(C)c(-c2ccccn2)ccc1 N1(C(C(C(C)O)(C)C)=O)CCC(C(=O)NCCC(F)(F)F)C(C)(C)C1 CC1OC2(C(=O)NCC3CCC4(CN(C(C5CCCO5)=O)C4)O3)CCC1CC2 c1(OC)ncccc1CC(=O)NCC1CCN(C(c2n[nH]c(C)c2C)=O)CC1 CCCCC(C)C(=O)N1CCC(CCC(=O)Nc2cn(C)nc2OCC)C1 n1(C(C)C)ncc(C(=O)NCCCNC(c2nn[nH]c2C(F)(F)F)=O)c1F c1(C(c2nnnn2CCCF)NC(CCSC)C)ccn(CCF)n1 Cc1c(C(=O)N(C2CCCC(NC(=O)CN3CCC(F)CC3)C2)C)c[nH]c1C#N Cc1c(C(N2CCOC(c3cccc(Br)c3)C2)=O)nnn1CCN CCCCC(CNC(c1cccnc1)=O)NC(=O)C(c1cccc(OC)c1)C C(C(C)(C)CC(F)F)NC(C(c1n(C)ncc1)NC(C1CCCS1)=O)=O N1(C(C2C(C)CC2)=O)CCC2(CC2)CC1C(=O)NCc1ccnc(CO)c1 N1(C(c2ccn(CCCC)n2)=O)CCN(C(c2cnc(O)n2CC)=O)C(C)C1C C(=O)(C#CC(C)(C)CNC(C1CCC(F)C1)=O)N1CC(C)N(C2CC2)CC1 Cc1sc(C)c2sc(C(=O)NC3CN(C(C45CCC(CO4)C5)=O)C3)cc12 N1(C(CCn2ncn(C)c2=O)=O)CC(NC(c2sc(C#N)cc2Cl)=O)C(C)(C)C1 n1(CC)ncc(NCc2nocc2C(C)(C)C)c1CC C(=O)(CC(C=C)CCC)N1CC2C(NC(CSc3ccc(OC)cc3)=O)C2C1 N1(C2CN(N3CCC(C)C3)C2)CCN(C(C23CCC(C2)C3)=O)CC1.C(=O)C=CC=O c1(C(N2CCN(Cc3cc(C)c(O)cc3C)C3C2C3)=O)c[nH]c2ncc(Br)cc12 C1(NC(CCn2ncc(C)c2)=O)C2CC(NC(C3(F)CCOC3C)=O)CC12 c1(C(=O)NC2CC3CN(C(COCCC)=O)C(C2)C3)ccc2c(c1)C(=O)NCC2 CCC(C)CC(=O)N(C1CCCN(C(=O)Cc2cnn(CC)c2)C1)C C1=NC(NCCSC)=C(C(=O)NS(C)(=O)=O)OCC1 c1(C(=O)NC2CC(n3cc(-c4c(C(=O)OC)n[nH]c4)nn3)C2)c(C)cccc1Cl C1(C(N2C(CNC(C3(C(=O)OCC)CCC3)=O)CCC2)=O)C(Cl)(Cl)C12CC2 N1(C(c2c(C)cc(C)c(Br)c2)=O)C(C)Cc2cc(F)ccc2C1C C1(CNC(=O)NCc2nc(C)c(C)o2)CC1C1CCCC1 C1(NC(C=C(C)C)=O)CS(=O)(=O)C12CCN(C(C1C(C#N)C1(C)C)=O)CC2 C1(C(=O)NCCOCCC)CSCCN1C(c1cc(C(C)=O)[nH]n1)=O CC1(C)COCCC1NC(=O)C=CC1CCCN1C(=O)CCN1CCCCC1 C(=O)(C1CCCc2cccnc21)NC1CC2(CN(C(C(C(C)C)OC)=O)C2)OC1 c1(C(=O)NCC(C2CC2)NC(C2CC(CC)(CC)C2)=O)ccc2c(n1)OCCO2 C1(C(N2C(CC(=O)NC)CC2)=O)CCN(C(=O)C(CC)CC=CC)CC1C N1(C(C(CC)OCC)=O)CCC=C(C(=O)NCCCCC(C)C)C1 C(=O)(C(C)C(C)NC(c1cnnc(C)c1)=O)NCc1occ(C)n1 N1(C(C2CC2(Cl)Cl)=O)CCC(n2cc(CNC(C34CC(F)(C3)C4)=O)nn2)CC1 c1(CN(C)C(c2ncc(C(F)F)s2)=O)cnn2c1CN(C(=O)CCC(N)=O)CC2 C(=O)(C1CCCn2cc(C)nc21)NC(CC)CNC(C1(O)CCCCCC1)=O N1(C(CCSCC(=O)OC)=O)CC(NC(=O)C(C)(C)c2ccncc2)CC1C c1(C(=O)NC2CN(C(CC(CC)SC)=O)CC2C)cnc(Cl)cc1N N1(C(c2ccc(C)nc2)=O)CCN(C(=O)CCc2cn(C)nn2)CC1CC(F)F c1(N2CCC(CC=C)C2)nc(NC(c2ccc(Cl)cc2)C(C)C)nc2c1CCC2 c1(SCC(=O)NCCCCc2cn(CCC(=O)NC)nn2)ccccc1OC c1(OC)ccc(C(=O)NC2(CCNC(=O)C3=NOC(C)C3C)CC2)c(F)c1Cl CC(C)C(CO)C(=O)NC(Cc1ccccc1)CCNC(=O)C(C)C1CCC1 N1(CC)CC(C(=O)NC2(CNC(=O)CC3COC(=O)C3)CCCCC2)CCC1=O C1(C(C(C2CCC(N(C)Cc3c(OC)cccc3)CC2)=O)C)CCC2(CCC2)O1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CNC(c1ccc(NC(=O)OC)cc1)=O)CO CC1=C(C(=O)N2CCN(C(=O)CCCOc3ccccc3)C3CCC23)CCCC1 C12(CNC(c3nnc(C)s3)=O)CCCC1CCN2C(=O)Cn1ccc([N+](=O)[O-])n1 N1(C(Cc2c(C)ncnc2C)=O)CCC2(CC1)CC(NC(C1C=CCCC1)=O)C2 O=C(C1=NN(c2ccc(Cl)cc2)C(=O)CC1)N1CC2OCCOC2C1 C1(NC(C(n2cc(C3(O)CCOC3)nn2)C)=O)CCOC12CCC2 c1(O)ccc([N+](=O)[O-])cc1C.C1(C(CNC)CC)CCCC1 c1(C(=O)NC2CCC(CNC(C34CC(C)(C3)C4)=O)C2)ccc(S(C)(=O)=O)cc1Cl Cc1nc(CC(=O)NCC2CCC(NC(c3csc(C)n3)=O)C2)cs1 N(C(=NCCCN1CCOCC1)NC1CC(OC(F)F)C1)CC1N(C)CCC1 c1(C(N(C(C)C(C)NC(=O)CSn2cncn2)C)=O)c[nH]nc1C(F)(F)F N1(C(C2ON=C(C)C2)=O)CCC(NC(c2cc3n(n2)CCO3)=O)C(F)C1 C1(NC(c2cc(CCC)on2)=O)CCN(Cc2cc(F)cc(Br)c2)C(C)C1 S(=O)(=O)(c1cccc2c1NCCC2)N1C(C)C(C)N(C)CC1 C1(C(=O)NC2CC(CCNC(c3c(SC)cn(C)n3)=O)C2)CC2(C1)CS(=O)(=O)C2 n1(CCC(=O)N(CCC(=O)OC)C2CC2)cncc1-c1ccccc1 CC(CN(C)C)CC(=O)NCC1(NC(c2cncnc2)=O)CCOC1 Cc1cccc(N(C(c2cc(Br)ccn2)C(=O)NCCCC2CC2)C)c1 C(=O)(CCCC(C)(C)NC(=O)CCc1cncs1)NCC1(CC)CCOC1 C1(CNC(c2c(C)nccc2)=O)CCC2CN(C(C3COCOC3)=O)CC12 n1(C2CN(CC(=O)N(C(c3cccs3)=O)CC)C2)ncc([N+](=O)[O-])n1 CC1(O)CCCN(C(c2cc(C3CNC3)[nH]n2)=O)CC1 C1(C(=O)NCc2ncc(Br)s2)CN(Cc2ccncc2O)CCC1O C(=O)(CC(CC)C(C)C)NCCCCC(C)NC(c1ccc(OCC)nc1)=O N1(c2n(Cc3ccccc3)c(C3CCCCO3)nn2)CCCC(O)CC1 C1(CCOC)CN(C(c2cc(C(C)(C)C)n[nH]2)=O)CCN1C(=O)C(O)CC(N)=O c1(C(C)(C)C)nccc(=NCC(O)CNC(=O)Cc2ccc(S(C)(=O)=O)cc2)[nH]1 C12(NC(c3cc(SC)oc3)=O)CCCC1N(C(C1CCc3nccn3C1)=O)CC2 C1(OC)CC(C(N2CCC(N(C(=O)Cc3ccns3)C)C2)=O)N(S(C)(=O)=O)C1 c1(OC)coc(C(=O)NCC2CC2CNC(=O)CCc2ccccc2O)cc1=O C(C)(C(=O)N=c1ccn(C(C)(C)C)[nH]1)N(CCC)C(C1CCCC(C2CC2)C1)=O c1(C(C(=O)NCCC)N(CCCN2CCCC2)C)cccc(C#N)n1 c1(OC)ccc(C(N2CCOCC(CNC(c3sccc3C)=O)C2)=O)c(OC)c1 C1(C(=O)NC(CCC)C)CCCN(C(c2cnn(C)c2N)=O)C1C N1(C(c2ncccn2)=O)CC(C(N2CCn3cnnc3C2)=O)CC2OCCC12 CC(C)C(C(C)NC(C1(O)CC1)=O)NC(c1csc(-c2cccs2)n1)=O C12(S(=O)(=O)N1)CC2C.C12(C(CN(c3nncs3)OC)O)CC(CO1)C2 CC1CC(CC(=O)NCc2cnccc2Cl)CN1C(C1(C)CC(C#N)C1)=O N1(C(C2N(C(C(SC)SC)=O)C(C)C2)=O)CC(C)(C#N)C1 Cc1cnc(N2CCC2)[nH]c1=N.C1C2CC3COC1C3C2 N1(C(CCC#C)=O)CCCC2(C1)C(NC(=O)CCC1CCCCC1)CCN2C c1(N2CCN(C(c3c(C)nc(C)[nH]3)=O)CC2C)ncnc2cnn(C)c12 C(C(C)(C)CNC(=O)CC(C)C1CC1)N(C(C1CC(CC2CC2)C1)=O)CC N1(C(C(CCC)CCC)=O)CCC(C2CCCN(C(c3cncn3C)=O)C2)CC1 C1(C(=O)NCCCNC(CCSCCC)=O)CCCN1C1CCCC1 c1(OC)cc(Cl)c(C)cc1C(=O)NCC1CC1NC(=O)CC1(O)CCC1 CN1CCN(CC(=O)NCCC2CN(C(C3(C(F)F)CCCO3)=O)CCO2)CC1 C1(NC(c2cnc(CC(C)C)s2)=O)CN(C(c2nccn2C)=O)C2CC12 c1(-c2cc(F)cc(CCCl)c2)cccc2c1oc1ccccc21 C(CC(C)C(=O)N(CC(C)NC(c1cccn1Cc1ccccn1)=O)C)OC C=CC1(C(=O)NC2CCC(NC(=O)COCCc3cccs3)CC2)CCCCC1 CC1C2CCC(C2)C1C(=O)NCc1nc(C(=O)N(c2ccccc2)C)co1 N1(C(C)=O)CCC(C2CN(C(C3CC3C(N3CC(C(=O)OCC)C3)=O)=O)C2)CC1 N1(C(CCC=CC)=O)CCC2(CCN(C(=O)COC(F)F)CC2)C(C)C1 c1(CC)ncoc1C(=O)N(CC(=O)N(CC(O)CO)CCO)C c1(SC)cc(C(=O)NCC2CC2CNC(=O)CCc2ccncn2)oc1C C(c1cc2ccccc2o1)=CC(=O)NC1CCCCN(C(=O)C2=COCC2)CC1 C1(C(=O)Nc2cccc(NC(C3C(COC)C3)=O)c2)CCC2(CCCCC2)C1 c1(C(=O)NC2CCC(Cn3cc(C(C)(C)OC(C)=O)nn3)C2)ccc(Cl)cc1Br c1(CC)nc(=N)[nH]cc1C(=O)NC(CCNC(c1cc(Cl)cnn1)=O)C(C)C C(=O)(CC(C)CC(C)(C)C)NCC1(CNC(C#CC(C)C)=O)CCCC1 CCC(C)CC(=O)C(=O)N(CCC(=O)NCC1CCC2(CCC2)O1)CC1CC1 C1(C(=O)NCC(C)N(C(c2cc[nH]c(=N)n2)=O)CC)CCC2CC1CO2 c1(NC(C(C)C)=O)ccc(Cl)c(C(=O)NC2C=CCN(C(C3CC3(F)F)=O)C2)c1 CC(C)(CNC(=O)C(CCC1CC1)NC(=O)CC1OCCCO1)C(F)F CC1CN(C(c2cn(C)nn2)=O)CCC1C(=O)NCCc1nccc(O)n1 C=CCC(C(=O)NCC(C(C)C)NC(C1CCCC1CC)=O)N(C)C C(C1CCN(C(C2(F)CC=CC2)=O)CC1)=CC(=O)NC1CC=CC1 c1(C(N2CCC=C(C(=O)NCc3cc(Br)ccn3)C2)=O)ccc2ccccc2c1 N1(C(=O)NCCc2nc(-c3ncccn3)no2)CC2C=C(Br)C2C1 c1(OCC)c(C(=O)NCC2CCCC(NC(=O)COC3CCCC3)C2)csc1C C1(C(=O)NCC)CCCCCC1NC(C1CC1C(C)(F)F)=O CC(CC(=O)N(C(C)CCNC(c1[nH]ccc1C1CC1)=O)C)c1ccco1 CCC(C(=O)OC)C(=O)N(C(C)(C)CC(=O)N(C1CC1(C)C)C)C Cc1c(N)ccc(C(=O)NC2CCCC2NC(C2CCS2(=O)=O)=O)c1C C1(NC(C=C(COC)C)=O)CC(F)CN(C(C2CC(=O)N(C3CC3)C2)=O)C1 C1(NC(CC(N2CCCCC2=O)C)=O)CN(C(=O)Cn2cnnc2)CC1N=[N+]=[N-] c1(CC(C(C)C)C)ccc(NC(=O)C(=O)NC2(c3ncc(F)cn3)CC2)cc1 CC(C)CC(C(=O)NC1CCCC1NC(=O)CC1CCCC1O)n1ccnc1 c1(C(=O)OC)ccc(CNC(C2CCN2Cc2ccc(SC)o2)=O)cc1 C1(C(=O)OCC)CCCN(C(=O)CC2(C)CCN2C(c2cn(C)nn2)=O)C1 CCC(CC(F)(F)F)C(=O)NC12CC(CNC(c3cnn4c3N(C)CC4)=O)(C1)C2 Cc1ccc(C(N2CCC=C(CNC(=O)CC(C)(C)C3CC3)C2)=O)c([N+](=O)[O-])c1 C(=O)(CC(F)(F)C(C)C)N(C1CCCN(C(c2cc(C3CC3)cs2)=O)CC1)CC Cc1cc(C(F)F)nn1CC(=O)N(C)CC1(CNC(C2(C)CCC(=O)C2)=O)CC1 c1(-c2cncc(C)c2)cccc2c1CN(C(c1ccc(Br)cc1I)=O)CC2 N1(C(C2ON=C(C(C)C)C2)=O)CCCC2CN(C(C3CCCS3)=O)CCC12 C1(NC(CCCC(C)=O)=O)CCN(C(=O)C=Cc2ccc(SC)cc2)CC1(C)C C1(C(N(C)CC2CCCCN2S(C)(=O)=O)=O)COC(C)(C)O1 c1(NC(=O)CCc2cc(Br)ccc2F)cc2ccccc2nn1 c1(C(=O)NCCCC(C)(C)NC(c2cncc(C)n2)=O)cc(C)c(C)c(C)c1 c1(C(N)=O)ccnc(NCc2cc(Br)cnc2Br)c1F c1(C(C(=O)NCC(CO)NC(C=CCCC)=O)C)ccc2ccccc2c1 N1(C(CCCOC(C)C)=O)CCC(NC(=O)C(C)CC2CC2)CC(C)(C)C1 C1(C)(C(N(C2CC3CCC2CC3)C)=O)CC12CCN(C(c1ccccc1)=O)CC2 C1(N(C(C(C2CCC2)OC)=O)Cc2ccccc2)CCN(CC2CCOC2)CC1 C12(CNC(C(C(C)C)OC)=O)CC(C1)C(NC(c1c(C)ncn1C)=O)CO2 N1(C(CC2N(C(C)C)CCC2)=O)CCCCC(CNC(c2cn(C)[nH]c2=N)=O)C1 c1(C(N2CC(CCCCNC(C(C=C)(F)F)=O)C2)=O)ccc([N+](=O)[O-])c(C#N)c1 c1(C(N2CCC(C(C)NC(CC(C)SC)=O)CC2)=O)ncc(F)c2ccccc12 C(C1=Cc2ccccc2OC1)=CC(=O)N(C1CN(C(CSC(C)C)=O)CC1O)C C(=O)(C#Cc1ccccc1)NCc1cccc(C(N2C(C(N)=O)CC(O)C2)=O)c1 C1(NC(c2cc(C)no2)=O)CC2CN(C(=O)Cc3c(F)cccc3Cl)CC2C1 CC1CN(C(c2c(Cl)cnn2C)=O)CCC1CNC(=O)CN(S(C)(=O)=O)C N1(C(C2(CCNC(C(CC)CC)=O)CCCC2)=O)CCN2CC(C)CC2C1 N1(C(c2cc(OCC)n[nH]2)=O)CC2(CC(CNC(=O)C(C)C3(O)CCC3)C2)C1 C(C(CNC(c1cnsn1)=O)C(F)(F)F)NC(c1ccc(-c2cccs2)s1)=O c1(C(=O)NC2C(CO)CCN(C(c3c(C)nco3)=O)C2)ccc2oncc2c1 CC(F)(F)CCC(=O)NC1CCCC1NC(c1cnsn1)=O S(=O)(=O)(c1c[nH]c2ccc([N+](=O)[O-])cc12)NCC(=O)Nc1c(C)scc1 c1(C(=O)NC(CC(C)NC(c2cnnc(O)c2)=O)C)ccnc(CO)c1 CC(C)C(O)C(F)(F)C(=O)NCC1(C)CCCN(C(c2cc(C(F)F)no2)=O)C1 n1(CC(C)C2CC2)nc(-c2ccoc2)nc1-c1ccc(-c2ccccc2F)n1C C(=O)(C(CO)C(C)(C)C)N(C)CC1CCCCN1C(c1cnc(O)o1)=O CCCC(C)(O)CC(=O)N(C)CC=CC(N1CCOCC(C)C1)=O c1(NC(C(CCC)C)C)ccc(S(=O)(=O)NCC2(C)CC2)c(Cl)c1 c1(NC)ccc(C(F)F)cc1C(=O)NCC1CCCN(C(C2CC2Br)=O)C1 C(=O)(C(COC)C(C)(C)C)NCC1CC(NC(C2C(CCC)CCC2)=O)C1 c1(OC)cccc(C(=O)NCCC2CCCCN2C(=O)CNc2ccccc2)c1 c1(CC(N2CCCCC2)C)nccc(=NCCOC2CCSCC2)[nH]1 C1(CC(=O)N(C2CCN(C(=O)Cc3csc(Br)c3)C2)C)CCC(O)C1 c1(C(=O)NCC(CNC(CC(C)N2CCCC2=O)=O)C)ccc2sccc2c1 C(=O)(C(C)CC#C)NC1(NC(=O)CC2CCCC23CC3)CC1.C#CCN C1(COC)(NC(c2cc(OC)ns2)=O)CCCN(C(c2ccc(C)n2C)=O)C1 C(CC(C)(C)C(=O)N1CC2(NC(=O)C(C)OC3CCCCC3)CC1C2)SC N1(C(c2cc(SC)c(F)cc2)=O)CCC2(CC1)CC2NC(=O)C=Cc1cn[nH]c1 c1(N(C(C)=O)C)ccccc1C(N1CCC(CNC(c2scnc2Cl)=O)C1)=O N1(C(=O)C(N2CCCC(c3cc(O)cc(Br)c3)C2)=O)CCC(=C(F)F)CC1 Cc1cc(CN=C(NC2CC2C)N(C)CC2c3ccccc3C2)ccc1O c1(C(=O)NC2CC(O)(CNC(c3c(C)cc(F)s3)=O)C2)cn2cccc(C)c2n1 N1(C(CCOCCOC)=O)CC(NC(C2CCC(=O)O2)=O)C2(CCC2)C1 CC1=NOC(=O)C1CC(=O)NCC1(O)CC(NC(C2(O)COC2)=O)C1 C1(CNC(C(COC(C)C)(C)C)=O)CCN(C(C2CC2C(N)=O)=O)C12CC2 S(=O)(=O)(C1(CSc2cccc(Cn3cncn3)c2)CC1)NC C12(C(N(C)CC3CCN(C(c4cccs4)=O)C3)=O)CCC(C)(C1)OC2 N1(C(C2C(CNC(C=C(CC)CC)=O)OCC2)=O)CCOCC1CCO CC(CC(C)NC(c1ncoc1C1CCC1)=O)NC(=O)CCc1cnoc1 N1(C(c2cc(C(C)=O)[nH]n2)=O)CCC2(CC1)CC2NC(=O)CC1CCC1 n1(CC(N2CCOCC2)=O)cnc([N+](=O)[O-])n1.[nH]1cc(CC)nn1 c1(CC)noc2ncc(C(N3CCN(C(=O)CS(=O)(=O)NC)C4CC34)=O)cc12 C1(NC(Cc2c(C)occ2)=O)CCCN(C(=O)Cn2cccnc2=O)CCC1 N1(C(C(CCOC)NC(=O)Cn2nccn2)=O)CCOC(C)CC1 c1(C(N2CCCC(C(N(CC(=O)NC)C)=O)C2)=O)cc2c(C)cc(OC)cc2[nH]1 CC1CN(C(c2sc(Br)cc2F)=O)CCN1C(=O)Cc1ccc(F)cn1 c1(OC)ccc2c(=NC(C)C3CC4(CCC4)C3)[nH]c(=NCc3cccs3)[nH]c2c1 c1(C(=O)NC2C(CNC(c3ccnnc3)=O)C2)csc2nccn12 c1(C(N2CC(NC(C3C(CC)CCO3)=O)C(C)C2)=O)c(N)cc(Cl)cc1F C(C)(C)(CCCCC(=O)NC1CN(C(C2(COC)CC2)=O)CC2(CCC2)C1)OC c1(NC(C(Cc2ccc(C)cc2)OC)=O)nc2cnc(Cl)cc2s1 C(CN=c1[nH]c2c(c(=NCC3COCC(C)O3)[nH]1)CCC2)c1nc(C)oc1C Cn1c(C(=O)NCC2CN(C(C3CS(=O)(=O)C3)=O)CCO2)cnc1Cl c1(OC)cc2[nH]c(C(N3CCCCC3CCN(C)C)=O)nc2cc1S(N)(=O)=O CC1CCN(C(=O)CC2CC(F)(F)C2)CC1CC(N1CCCN(CCO)CC1)=O c1(C(=O)NC(C(=O)N(CC=C)CC=C)c2ccoc2)ccnnc1O c1(C(=O)NC(C)(CNC(=O)Cc2c[nH]ccc2=O)C2CC2)ccc2snnc2c1 C1(C)(C(=O)NCCCN(C(C)C)CC)CCCN(C(=O)COC2CC=CC2)C1 c1(OC)ccc2c(=NCC3CC3Cl)[nH]c(=NCC3(CO)CC3)[nH]c2c1 Cc1cc(C(=O)NCCCOCCNC(c2coc(Br)n2)=O)nnc1C CC(=O)CCCC(=O)N1CCCC(CNC(=O)C(O)Cc2[nH]cnc2C)C1 C12(NC(C(=O)N(CCNC(C)=O)F)C)CC(CO)(C1)OC2(C)C.S(C)(=O)(=O)N N1(C(C(CCC)NC(N)=O)=O)CCN(C(C2CN(C)C(=O)N2)=O)CC1CO c1(C(N2C(C)(C(=O)NC(C3(CO)CC3)C)CCC2)=O)ccc2cncn2c1 c1(C(=O)NC2CC(O)CN(C(=O)Cn3cnccc3=O)C2)cccc2cc[nH]c12 CC(N=c1ccc(C#N)n[nH]1)C1CCCN(C(=O)CC(c2ccccc2F)C)C1 N1(C(c2cc(C)c(F)nc2)=O)CCC(C2CC2)C1CNC(c1c(C)noc1C)=O c1(N(c2ccccc2)C(=O)CCC2CCCO2)ccc(C(=O)CF)cc1 C1(CC(=O)N(CCC)CCNC(c2cc(C(F)(F)F)no2)=O)CN(C)CC1O c1(OC)cc(C)c(CN2CC(C(=O)Nc3nc(Br)c(Br)cc3Br)C2)cc1OC c1(C(=O)NCC2(C)C(C)CN(C(c3cc(C)sn3)=O)C2)cc(Cl)c(N)c(Cl)c1 c1(OCC)nccc(C)c1C(N1CCC(NC(c2csnc2Cl)=O)C(O)C1)=O C1(C(=O)Oc2c(Cl)cc(OC)cc2Cl)CC2(C1)C(C(=O)OC)C21CCC1 C1(C(N(C)Cc2ccc(C)s2)=O)CCCN(C(C2(C)CC3(CCC3)C2)=O)CC1 N1(C(c2ccn(C)n2)=O)CCN(Cc2cnco2)CC1Cc1ccccc1 CCCN=C(NCC1CCCSC1)NCC(C)(C)Oc1ccccc1 c1(C(=O)NC2(C)CCN(C(=O)C(Cl)=CCl)C2)cc2c(Cl)cncc2s1 CC1(C(=O)NCC2CCCC2NC(=O)CN(c2ccc(Cl)cn2)C)CCC(=O)N1 N1(C(CC=C(C)C)=O)CCC2CN(C(c3cc(S(C)(=O)=O)cs3)=O)CC2C1 N1(C(c2c(CC)scc2)=O)CCN2CCOCC2(CNC(=O)CC2CC23CC3)C1 c1(CNC(COCC(=O)OC)=O)cn(C2c3ccccc3CCC2C)nn1 N1(C(CC(=C=C)C)=O)CCC(O)(C2(NC(c3cn(C4CC4)cn3)=O)CC2)CC1 C(c1ccncc1)=CC(=O)N(C1CCC(NC(c2cncn2C(F)(F)F)=O)C1)C c1(C(N2CC(C)OC(C)C2)C)ccc(S(=O)(=O)N2CCCN(C)CC2C)cc1 C(=O)(C(F)(F)CC(C)C)NCCC1CCC(NC(C(C)=C2CCCC2)=O)C1 C#CCCC(O)CCNC(=O)C(C)(C)CNC(C1CC=CCC1)=O C1(NC(c2cccc(C3CCC3)c2)c2n(CCOC)nnn2)COCCC1(F)F C1(CCC)(NC(C2CCOC2)=O)CCN(C(=O)COC(C)CC)CC1 Cc1n[nH]cc1CC(N1CCC(N(C(C2CCOC2C2CC2)=O)CC2CC2)C1)=O C1(C#N)(CNC(C(CCSC)NC(=O)CC2COCC(C)O2)=O)CC(C)(C)C1 C1(C(=O)NC2CC(F)(CNC(c3ccc(OC)s3)=O)C2)COCCC1(F)F N1(C(C2C(=C)CC2)=O)CCC(CO)C(NC(=O)COCC(c2ccccc2)=O)C1 C(=O)(CCCCCO)NC(C)CNC(=O)CCN1CCCCC1 Cc1cc(C(C(=O)NCC2CCOC2)N(CC#N)C2CC2)c2c(c1)CCC2 c1(CC(=O)NCCNC(C(c2ccc(OC)cn2)(F)F)=O)ccc(OC)c(O)c1 n1(CC)ccc(C(N2CCOC(CCNC(c3ccc(Cl)[nH]3)=O)C2)=O)c1C c1(C(=O)OCC)cn(C)nc1C(=O)NC1CCN(C(C2CCCC2(C)C)=O)C1 c1(C(=O)NCC2(CNC(C3C(CN(C)C)C3)=O)CC2)cc(Cl)no1 N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCC(O)(CNC(C23CCC(CC2)O3)=O)C1 CC(C(C(=O)NC1CCOCC1)N(C1CC(=O)NC1=O)C1CC1)C(C)(C)C N1(C(c2c(C)nsc2)=O)CCC(O)(CN(C)C(c2cc(C(C)(C)C)n[nH]2)=O)C1 c1(OC)cc(N)ccc1C(=O)NCC1(CO)CCN(C(C2C=CCS2)=O)C1 Cc1nn(C)c(C)c1C(=O)NC1CC(NC(c2nscc2Br)=O)C1 CC(C(=O)NC1CCCCC1CNC(c1cc2c(s1)CCC2)=O)C(C)(C)C C12(NC(=O)CC34CCC(CC3)C4)CCOCC1CN(C(=O)C(F)(F)C(F)(F)F)C2 Cc1cc(F)cnc1C(=O)NC12COC(C1)C(NC(=O)CC(C)n1cccc1)C2 c1(C(=O)NC23CC(NC(c4ccn(C(F)F)n4)=O)(C2)C3)cc([N+](=O)[O-])ccc1O CC1=NC(C(=O)NCCCOCCNC(c2ocnc2C(F)F)=O)CS1 c1(CC)cnc(O)c(C(=O)NC2CCN(C(=O)CNS(C)(=O)=O)C2C)c1 N1(C(=O)Nc2ccc(N3C(=O)CCC3=O)cc2)CCCC2CCCN2CC1 N1(C(CC(=O)OCC)=O)CC(C)CN(C(C2(CF)CCC2)=O)CC1C C1(C(N2C(C(=O)NC3CCC(O)C3)CC3CC32)=O)CCc2ccccc2C1 N1(Cc2c(C#C)cc(F)cc2)CCC2CN(C(=O)Cc3ccccc3)CC2C1 c1(COC)cncc(C(=O)NC2CCCC2NC(=O)CCCc2cc[nH]n2)c1 C=C(C)CC(C(=O)NCc1noc(C(C)C)n1)NC(=O)Cc1cc[nH]c1 N1(C(C(c2n(C)ccc2)=O)=O)CC2CC2(C(N2CCOCC2CN(C)C)=O)C1 C(=O)(C1CCCc2nn[nH]c21)NC1C(NC(c2cc(C)nc(NC3CC3)c2)=O)C1 c1(OC)nccc(C(=O)NC2CC(NC(c3ccnc(OC)c3F)=O)C2)c1F C1(N(C(C(CSC)C)=O)C)CCCN(C(c2csc(-c3nc[nH]n3)n2)=O)C1 N1(C(C(=O)NCCOC)c2ccsn2)CC(C)C12CCOCC2 N1(C(CCCC2C(C)C2)=O)CCC(C)(CCNC(=O)Cn2nnc(C3CC3)n2)C1 c1(C(N2CCC(CN(C)C(C3CCC(=O)N3C)=O)C2)=O)ccnc2[nH]c(O)nc12 C(CCC[Si](C)(C)C)N(C)C(c1ccc(Br)cc1CC#N)=O Cc1cccn2cc(CC(=O)NCC(C(C)C)NC(C3CC(=O)C3)=O)nc12 N1(C(=O)Cc2ccc(Cl)cc2)CCC2(CCCN2C(=O)COC2CCCC2)C1 N1(C(CC)=O)CCc2c(CNC(c3cc(Cl)c(C)cn3)=O)cccc2C1 C(CC(O)C(=O)N1CCC(C(N2CCC(COC(C)=O)C2)=O)(CO)C1)SC C1(CC(=O)NCC2CC(NC(=O)CCSC3CCCC3)C2)(OC)CCC1 c1(C(N(C2CCN(C(C3(CCCC)CC3)=O)C2)C)=O)ccc(Cl)cc1C c1(C(=O)NCCCC2(NC(c3n(CC#C)ccc3)=O)CC2)cc(C)c(C)nn1 c1(C(=O)NC2C(NC(c3cccc(C(=O)NC)c3)=O)CC2)cnc2occc2c1 N1(C(CCSC)=O)CC2CC1CN(C(C1OCCC1C(C)C)=O)C2 c1(C(=O)NCC2(CNC(C(CO)OC)=O)CC2)[nH]c(C)nc1C CC1OC2(CNC(c3ccns3)=O)CC1(NC(=O)CCn1ccnn1)C2 c1(C(=O)OCCSCC2(OCC)CCOC2)cc([N+](=O)[O-])ccc1N1CCCC1 C(=O)(CC1=NNC(=O)C1)N1C(CCCC)CN(C(C2(C)CCCS2(=O)=O)=O)CC1 C1(NC(=O)CN2CCCNS2(=O)=O)CCC2(CC1)CC2NC(c1cnns1)=O C(CCN=C(NCCC1CCN(C(C)C)CC1)N1CC(C)N(C)C(C)C1)SC c1(C(N(CC(N2CC(CNc3ccccn3)C2)=O)C)=O)cccnc1S C(=O)(CCC(C)(F)F)N(C1CCN(C(CC(C)O)=O)CC1)Cc1ccccn1 N1(C(CS(C)(=O)=O)=O)CC2CC(O)C1C2NC(=O)CNC(C1CCC1)=O C(=O)(CCC(C)NC(c1cn(C2CC2)nn1)=O)N(CC)CC1CCC1 N1(C(C2(F)CCN(C(CC(CC)C)=O)C2)=O)CCC(CO)C(C)(C)C1 c1(CC)ccc(C(=O)Nc2ccccc2COCC(F)(F)F)cc1C#N c1(C(=O)NC(COC)C(N)=O)cc(Cl)cc(Cl)c1F CCCCC(C)C(=O)N(C1CC2CCC(C1)N2)C(C)(C)C(N)=O C1(NC(c2n(C)ccn2)=O)CCN(C2CCN(C(=O)CC3CC3(C)C)C2)CC1 CC(C)CC(CNC(=O)CN1CC=CC1)C(=O)NCCNC1(C2CC2)CC1 C1(CNC(C2(C#C)CN(C(=O)C(C)n3cccn3)C2)=O)OCC2CCC1C2 C12(CNC(CCCCC=CC)=O)CCC(CC1)N(C(=O)C(C)OC)C2 c1(N(C2CCCC2(F)F)CC2(n3cc(C(C)(C)C(=O)O)nn3)CC2)ccc(Cl)c(N)c1 C1(C(=O)Nc2c(C)cc(Oc3ccccc3)cc2)CN2CC3CC2(CO1)C3 C1(OCCOC(c2[nH]cc(C#N)c2)=O)CCS(=O)(=O)CC1 N1(C(C2CNC(=O)N2)=O)CCC(CO)(CNC(c2cnc(Cl)s2)=O)C1 c1(C(=O)NCC(Cc2cccc(C)c2)CO)cc(Br)c(C)c([N+](=O)[O-])c1 C1(NC(c2cc(CNC(c3cccc(C)c3)=O)nn2C)=O)C(C)CCCC1C C1(NCc2scc(OC)c2)CCN(C(=O)CC(C)(C)c2cccs2)CC1C c1(C(N2C(CCNC(c3c(CC)cc[nH]3)=O)CCC2)=O)cnc2ncccc2c1 C1(NC(=NCCCOCC)NCC2(S(C)(=O)=O)CCC2)CC(C2CCCCC2)C1 c1(C(=O)NCCOC2CCN(C(c3c(C)snn3)=O)C2)ccc2c(c1)NCCC2 N1(C(c2n(C)nc(Br)c2)=O)CCC2(CC1)CC(NC(=O)C1=CCCOC1)CO2 N1(C(c2n(C)cnc2)=O)CCC2C(CCN2Cc2nc(Br)cs2)C1 c1(CNC(C2(CNC(CCC3C(C)C3)=O)CC(F)(F)C2)=O)cnc2ccccn12 CCCC(C)(CC)C(=O)N1CCC(=O)C(NC(C)=O)C1 N#Cc1ncc(C(=O)NC2CN(C(c3cncc(-n4ccnn4)c3)=O)C2)s1 N1(C(C2C=CC(NC(CCOC)=O)C2)=O)CC2COC(=O)C2C1 C1(CC(=O)NCCOCC(C)C)C2CCC(C2)N1C(C1CC2C=CC1C2)=O c1(OC)ccc(C(=O)Nc2ccc(C(C)(C)CO)c(Cl)c2)cc1Br N1(C(CCNC(=O)OC)=O)CC2CCC2(CCNC(c2c(C)nn(C)c2C)=O)C1 C1(COC(CC2(N(C)C)CCCCC2)=O)CC2CCCCC2N1 N1(C(c2n[nH]c(C)c2O)=O)CCN(C(=O)C(C)CCN(C)C)CC(O)C1 c1(C(=O)NC2CN(C(c3n(CC)ccn3)=O)C(C)CC2)cnn2cnnc2c1 Cc1cccc(C(CNC(c2ccccc2O)=O)N(C)Cc2ncc(Cl)n2C)c1 Cc1cc(NCC2(C)CCN(C(=O)C(C)C(C)(C)C)CC2)c(F)cc1[N+](=O)[O-] C(=O)(C(C)C1=CCCC1)NC1CC2CN(C(c3n(CC(C)C)ncc3)=O)C1C2 c1(C(=O)NC(C)CC(C)NC2CCOCC2)cncc(NC(=O)OC(C)(C)C)c1 C1(C)(C(=O)NCCC(CCNC(c2c(COC)cco2)=O)C)CCC(C)=C(C)C1 CCCCC(C)CCC(=O)NCC1OCCC1C(=O)NC(C)C(=O)OCC c1(NC(CN(C2CN(Cc3ccc(O)cc3)C2)C)=O)ccc(OC(C)(C)C)cc1 c1(Nc2c(C(=O)NCc3c(C)noc3C)cccc2)ccc(S(N)(=O)=O)cc1 CC(C)(O)CC(=O)N1CCN(C2CCCN(C(c3ccc[nH]3)=O)C2)CC1 N1(C(C(N2CCC(O)CC2)C)=O)CCCC(NC(c2cc(F)ccc2N)=O)CC1 C1(NC(COC(C)C)=O)CC2CN(C(c3cc(C4CC4)[nH]n3)=O)CC12 Nc1ncc(C(=O)NCC2CC(NC(=O)Cc3ccc(Cl)s3)C2)cc1CO N(C1c2ccccc2CC1NC(c1cscc1F)=O)C(C(COCC)(C)C)=O C1(C(N2CCC(NC(C(CCC)NC(N)=O)=O)CC2)=O)CC2(CCOCC2)CO1 C(=O)(CC(C(F)F)NC(=O)C(C)=C(C)C)NC(C=C)C N1(C(C=CCC)=O)CC(C(F)(F)F)OCC1CNC(c1occc1CC)=O Cc1[nH]cc(C(=O)NC2CC3CCC2N3C(C2CC=CC2)=O)c(=O)c1Cl CN1CC2CCN(C(c3ccoc3CNC(c3sccc3Cl)=O)=O)C2C1 C1(NC(c2cc(Cl)c[nH]2)=O)CN(C(=O)C(F)(F)c2ccncc2)CC12CC2 Cc1ccn(CC(=O)NC(C)C(C)NC(c2cccs2)=O)n1 c1(C(CC)NC(=O)C(C2CCCO2)NC(=O)COCC(F)(F)F)ccccc1 CCC(CC(=O)NC12CC1CN(C(=O)CCc1ccc(F)nc1)C2)CC(C)C Cc1cc(O)c(C(=O)NC(c2ccccc2)CNC(=O)CCc2cn[nH]c2)nn1 C(CCC(C)(C)C(=O)NCC1CC(C(=O)NCC2CCCC2)=NO1)OC N1(C(CC(=C)C)=O)CC2(CCN(C(c3cnn(CC(F)(F)F)c3N)=O)CC2)C1 c1(C(C)=O)ccc(C(=O)NCC(C2CC2)NC(=O)CCn2ccc(=N)[nH]2)nc1 c1(C(N(CC)CC2CCCN2C(C2(C)CCCN2C)=O)=O)ccn(C)c(=O)c1 C1(C(=O)NCc2cc(C(=O)NCC(C)F)no2)COCC1(C)C N1(C(c2c(C)c(Cl)ccn2)C(=O)NC2CCC2)CCc2ccsc2C1 C1(C(N(CCCCn2ccnc2)C)=O)(NC(=O)CC2CC3CC3C2)CCN(C)C1 N(C1CCCc2ccc(Br)cc21)(CC(C)NC(C1(C2CCCCO2)CC1)=O)CCC N1(C(C(N2CCC(c3c(OC)cccc3)CC2)=O)=O)CCCC2(CNC(=O)C2)C1 c1(CC(N2CC3C(CN(C(C(C)NC(CC)=O)=O)C)C3C2)=O)cccc(F)c1O CCC(C)(CNC(=O)C(Cc1cnc[nH]1)NC(c1ccc(=N)[nH]n1)=O)C(N)=O N1(C(C=C(C)c2cccs2)=O)CCC(C)C(NC(C2CCCS(=O)(=O)C2)=O)C1C C1(C(CC(=O)OC)C(=O)OC)CCCN(C(=O)C(=O)N(CC(C)C)C)C1 C1(C(=O)NC2(CN(C(C(C=C)O)=O)C)CC2)CCc2nncn2CC1 C1(NC(C(C2CC(F)(F)C2)OC)=O)C=CCN(C(c2ccc(CO)nc2)=O)C1 N1(C(c2cc(OC)n[nH]2)=O)CCC2C1CCCN2C(C1CCS1(=O)=O)=O CCC(COC)C(=O)NC(C(=O)NCC(O)C1CC1)C1(C)CC1 C1(NC(C(F)OC)=O)CC2CCC1C(NC(c1csc(S(C)(=O)=O)c1)=O)C2 n1(CC(N2CC(C)(CCC(N3C(CCC)CCCC3)=O)C2)=O)ccc(O)nc1=O N1(C(CCC2(NC(CC3(C)C(C)(C)C3)=O)CCCC2)=O)CCC(O)C(CO)C1 C(c1ccccc1)=CC(C(=O)NC1CC(C)(NC(c2cc(C)on2)=O)C1)C c1(C(N(C)Cc2ccccc2CNC(C2CCSC2)=O)=O)ccc2occc2n1 c1(OC)cc(F)ccc1C(C)NC(c1nnnn1CCCC1CC1)c1ccon1 C=C(C)C1OCCC1C(=O)NCCOCCNC(c1ncoc1-c1ccon1)=O CN1CC(C(N2CCC(C)(NC(c3ccc(F)c(N)c3F)=O)C2)=O)OCCC1=O c1(C(N2CCC(C)(CNC(c3ccc(C(C)C)cc3)=O)C2)=O)cc2sccc2s1 N1(C(C2ON=C(CC)C2)=O)CC2CCCC1(CNC(=O)Cn1ncccc1=O)C2 C1(OCC)(CNC(C2CCC3CCC23)c2nnnn2C2CCC2)CCCOC1 CCCCCC(=O)NCC(=O)NC(c1ccccc1)CNC(c1ccsc1SC)=O C(=O)(CCCC(F)(F)CO)N1CC(NC(C(c2cccc(C)c2F)O)=O)C(O)C1 C(CC(O)C(=O)NCC1(F)CC(NC(c2cc(C(F)(F)F)ncn2)=O)C1)N(C)C c1(OC)cc(NC(C2CC3(C2)CN(C(=O)CCN2CCOCC2)C3)=O)c(F)cn1 c1(C(=O)NCC(C)(CO)NC(C2COCCC2(F)F)=O)ccn2ncccc12 C(=O)(CCC(=O)NC1(CNC(C2CC3C=CC2C3)=O)CCCCC1)OC Cc1ccc(Cl)c(S(=O)(=O)c2csc(N3CCSCC3)n2)c1 c1(C(=O)NC2CN(C(c3cc(Cl)ncc3F)=O)CC23CC3)cc(Br)cc(Br)c1O Nc1c(F)cc(F)c(F)c1C(=O)NCCCNC(C1(C2CCC2)CC1(F)F)=O CC1CCC(CNC(c2ccc(O)cc2)=O)N(C(=O)Cn2cc(Cl)cn2)C1 Cc1cnc2cc(C(=O)NC(CNC(=O)C(C(C)C)N(C)C)C(C)C)ccn12 c1(CNC2(CNC(c3ccc(Cl)cc3)=O)CC2)ccc(F)cc1C1CC1 c1(C(C(=O)N(CC(C)CNC(=O)CC2(O)CC2)C(C)=O)C)ccc(Cl)c(Cl)c1 Cc1cc([N+](=O)[O-])cnc1NCCCN(c1ccc2nc(OC(C)C)sc2c1)C C1(CNC(c2n(CC)ccn2)=O)CCC2(CN(C(=O)CC3CCCCN3C)C2)O1 C1(NC(CS(=O)(=O)CC)=O)CCN(C(c2cc(C)[nH]c(=NC)n2)=O)CCC1CO c1(NCc2cccc3c2NC(=O)C3)ccc(S(=O)(=O)C(F)(F)F)cc1 C1(CNC(CC(CC)C)=O)CCN(C(c2ccnc(C)c2)=O)C1(C)C c1(NC(CN(C(CCCC)=O)C)C)ccc([N+](=O)[O-])cc1Cl CN(CCCC(=O)N1CC(CCNC(=O)CCc2cccnc2Cl)C1)N=O CCCCCCCCC(C)C(=O)NCC1CN(C(c2cncnc2C)=O)C1 c1(C(=O)NC(c2cccnc2)C(=O)N(CC)Cc2ccccn2)ccnnc1O C(=O)(C(C)(C)C1CCCCO1)N1CC(CN(C(C=C(C)C(C)C)=O)C)C1 c1(CC(=O)NC2(CC=C)CCCN(C(C(CC#C)O)=O)C2)nc(F)c(F)cc1F Cc1cc(N)c(C(=O)NC(CNC(c2cc(C)c(C)s2)=O)C(C)C)c(F)c1 n1(CC)cc(Cl)c(C(c2nnnn2C2(C)CC2)NC(c2ccccc2F)C)n1 c1(C(N(CCNC(C2(C)CC2(F)Cl)=O)C2CC2)=O)ccc(F)c2[nH]ccc12 c1(C(=O)NCC(CN(C(C2CCCN(CCC)C2)=O)CC)(C)C)cccc(F)c1O O=S(=O)(c1ccc(Cl)cc1Cl)N(c1nc2ccccc2o1)C1CC1 c1(C(N2C(CCCNC(C3CN4CCN3CC4)=O)CCC2)=O)cc(F)ccc1F S(=O)(=O)(c1[nH]c(=NCC23CCC(CC2)C3)ccc1Br)NC(C(C)C)CCO CCCCC(C)C(=O)NCC(O)CCNC(c1cccc(C(=O)NCCC)c1)=O C1(C(N2CCC=C(CNC(C3CC(=O)NC3)=O)C2)=O)CCC([N+](=O)[O-])CC1 Cc1ccc(CC(=O)NCC2(C(=O)Nc3ccc(OC(F)F)nc3)CC2)c(C)c1 N1(C(c2c(CC)nccn2)=O)CC2CC1CN2C(c1cc(C)n(C(F)F)n1)=O c1(OC)cc(C)c(Cl)cc1C(=O)N(CC(C)(C)NC(=O)Cc1ccsc1C)C CC(=NOC(C)(C)C1(c2ccccc2)CC1)C(=O)N(CC(C)C(=O)N(C)C)C C=C1Cn2c(C(N3CCC(CF)(NC(=O)C=CC4CCOCC4)C3)=O)nnc2S1 C(=O)(CC(C(F)F)C(C)(C)C)NC1CN(C(CC2OCC(C)(C)OC2)=O)C1 c1(CC(=O)N(C2CCCN(C(CC(C)(O)C3CC3)=O)C2)CCF)ccc(Cl)cc1F c1(NC(N2CCN(C(C(C)C)=O)CC2)=O)ccc(S(C)(=O)=O)cc1C(F)(F)F C1(NC(C2(CC(=O)OC)CC2)=O)CN(C(c2c[nH]ccc2=N)=O)CC12CCC2 CCCC(C)CC(=O)NCCOCCCNC(c1cc(C)cnn1)=O C1(CNC(C(CC)SC)=O)CC(C)(C)CN1C(=O)CCc1nnc(S)n1C c1(CN(C(C(=O)OC)C)C)ccc(SCc2sc(C3CCCCC3)nc2C)cc1 C#CC1(C(=O)NC2CCC(O)CC2)CCN(C(=O)CC2CC=CC2)C1 c1(NC(c2cncc(-c3ccc(OC)cc3F)n2)=O)cc(Cl)c(Br)cc1F Cc1ccc(C(=O)N2CC(n3cc(C4CC45CC5)nn3)CO2)c(Cl)c1 C(CC(C(=O)NCC(C1CCCCC1)O)NC(=O)C1CC1)=CC O=C(C1CCCc2scnc21)NC1CN(C(C2CCC3CC23)=O)C1 C(=O)(C(C)(O)CC)NCC(CC)NC(=O)C=Cc1ccc(C(F)F)o1 C1(CNC(c2ccc(C)c(C)n2)=O)C2CCCC1N(c1ncc(I)cn1)C2 c1(CNC(CCN(CCC)C)=O)cnn(C)c1C(=O)NCCC(C)CO c1(C(=O)NCC2(F)CC(NC(CC(C)OC)=O)C2)cc(SC(F)(F)F)oc1C c1(C(N(C2CN(C(c3ccc(C4CCCO4)[nH]3)=O)C2)C)=O)cc(N)cc(O)n1 c1(NC(C(C(C)C)C)CNC(C2CCOCC2)=O)nc2c(cc1C#N)CCCC2 C1(CNC(c2c(C)nn(C)c2)=O)N(C(=O)CSc2nncn2C2CC2)CCC1(C)C CCCCCS(=O)(=O)CC(=O)N1CCCC(N(C(c2ccc[nH]2)=O)CC)CC1 C1(NC(C(CC)N(C)C)=O)CC(F)CN(C(=O)CCc2cn(C)cn2)C1 S(=O)(=O)(c1cnn(CC(F)(F)F)c1)NC(C(=O)NC)CC(C)C C1(CNC(C(C)=CC)=O)CCCN(C(=O)CC2COCC2O)CC1 N1(C(CC=C=C)=O)CCN(C(c2ccc(Br)c(C)c2N)=O)C(C)C1C C1(C(=O)NCC2CCN2C(c2cnco2)=O)COCC1C(F)F N1(C(C2CCC(CC)CC2)=O)CCOC(C(=O)NCC(F)(F)CO)CC1 CC(C)(C)CCCCC(=O)N(CC(C)O)CCNC(C1(C)CC2CC2C1)=O C(=O)(C1CCc2c[nH]nc21)NCCC1(C(=O)NC(C)Cc2ccco2)CC1 C(=O)(CCS(=O)(=O)c1ccc(Cl)cc1)NCC(C)N(C(CC=C)=O)C C1(C)(C(=O)NCC2C(CC(=O)NC3(CN(C)C)CC3)C2)CC(O)CN1C c1(CC(=O)NC2CN(C(CC(=O)OC)=O)C2)cn2c(n1)CCCC2 C1(CNC(C(N2CCCCC2=O)C)=O)C2CCC(C2)N1C(=O)C(C)n1ccnc1 c1(C(=O)OCC2(c3ccc(OCC)cc3)CC2)nc(F)ccc1Cl C1(C(=O)Nc2cccc(-c3n(CC)cnn3)c2)CC2C=CC1CCC2 c1(C(=O)NC(c2nccs2)CC)cn2c(n1)CCN(C1CCS(=O)(=O)CC1)CC2 N1(Cc2c(OC)cccc2)C2CCC1CC(N(C)C[Si](C)(C)C)C2 Cc1cn(C)nc1C(N1CCC1C(=O)NCc1nnc(O)o1)=O C12(C(N3CCC(N(C(C(CC=C)C(C)C)=O)C)C3)=O)C3CCC(CC13)C2(F)F N1(C(c2c(NC(CC)=O)cccc2)=O)CCCC(N=c2[nH]nc(O)s2)CC1 C1(NC(c2nnc(CC)s2)=O)CCCN(C(c2ccnc(C(F)(F)F)c2)=O)C1C Cc1cc(C(=O)NCCC(C)NC(C2CC2(Cl)Cl)=O)cs1 N1(C(CCc2cc(C)no2)=O)CCN(C(=O)CC2COCCOC2)C(C(F)F)C1 CCC(CC)N(CCC(=O)NC(C1CCCC1)CNC(C)=O)C C12(NC(=O)NCCCC(=O)OCC)CCC1CN(C(C1(C)CC3CC3C1)=O)C2 Cc1nc(Cl)ccc1NC(C1CC1C(=O)Nc1csc(-c2ccccc2)c1)=O c1(C(N2CCC(C)(C(N3CCC(C#N)C3)=O)C2)=O)cccc2[nH]ccc12 C1(CNC(C(CC)OC)=O)COCCN1C(=O)CC1CCC=CCC1 C(=O)(C(CNC(=O)CN=[N+]=[N-])C(C)(C)C)NCC1(C)ON=C(C)C1 c1(C(=O)NC(CNC(C=C(CC)CC)=O)CO)cn2ccc(OC)cc2n1 N1(CC(n2cc(C(=C)C)nn2)NC(C)C)CC(C)(C)C(O)C(C)(C)C1 C1(C(=O)OCCC(C(=O)Nc2c(COCC)cccc2)OC)CCCC(C)(C)C1 N1(C(c2cc(C(=O)OC)n(C)c2)C(=O)NC(CC)(C)C)CC2CC1CS2=O N1(C(c2[nH]nc(OC)c2Cl)=O)CC2(CC(NC(=O)COC3(C)CCC3)CO2)C1 CC(C)CC(C(=O)N1CC(NC(C2CC23CCCCC3)=O)C2(CC2)C1)NC(N)=O c1(NC(c2n(C)nnn2)c2cnn(-c3cncc(Br)c3)c2)cc(Cl)cc2c1OCC2 C1(NC(c2cn3c(n2)CCCC3)=O)CC2CCC1CN2C(=O)CC1CC1(Cl)Cl C1(CNC(C2(CC#C)CCCO2)=O)C(C)CCN1C(=O)Cc1ccc(F)cn1 Nc1ccc(C(N2CCN(C(c3ncc(Br)cn3)=O)CC2CF)=O)nc1N Cc1cnc2[nH]cc(CN3CCC(C(=O)OC(=O)CNC(C)C)C(F)C3)c2c1 c1(C(=O)NC)ccc2c(c1)CN(C(=O)C(=O)N(C)CC1CC1)C2 N1(C(c2c(C)cco2)=O)CCC2(COCCN2C(c2cccc(F)n2)=O)C1 c1(CC)c(C(N2CCOC(CCNC(c3[nH]cnc3C#N)=O)C2)=O)cnn1CC c1(CC(=O)NC2CC3(CN(C(CNS(NC)(=O)=O)=O)C3)C2)cn2c(C)csc2n1 c1(C(=O)NCCc2c(C(N(CCC3CC3)CC)=O)c[nH]n2)[nH]ccc(=O)c1C Cc1ccc(C(N2CC(C)(NC(c3ccc(Cl)c(C)c3Cl)=O)C2)=O)c(F)c1F CC1(C)CCC(C(N2CC(NC(C3CCC3)=O)C(C(F)F)C2)=O)CO1 c1(CNC(=O)Cc2ncc(-c3ccccc3)o2)ccc(OC(F)(F)F)cc1 C1(CC(=O)N(C2(C(=O)NC3CCC4(CC4)C3)CC2)C)CC2CCC1O2 C1(NC(=O)NCCc2ncc(CC)s2)CCN(c2cc(C)nn2C)C1=O N1(C(c2n[nH]c(C)c2O)=O)CC(N(C)C(C2CCNC(=O)C2)=O)C2(CC2)C1 c1(C2C(C(N(CCNC(CCC=CC)=O)C)=O)C2)ccccc1Br O(NC(=O)C(Cc1cn[nH]c1)NC(C1CC(=O)NC(C)C1)=O)CCCC#C N1(C(c2cc(C)nn2C)=O)CCN(C(c2ccc(=O)n(CC(C)O)c2)=O)C2CC12 S(=O)(=O)(c1ccc(F)c(C(N2CCC(CO)(NC(=O)C3CC3)CC2)=O)c1F)NC C(C)(CC#CC)NC(CCN(CC=C)C(C1CCNC1=O)=O)=O c1(NC(C2(O)CN(C(Cc3cn(CC)nc3)=O)C2)C)ncc(C)c(SC)n1 c1(NC(CCC(CC)NC(C2(C#C)CC(=O)C2)=O)=O)ccc2c(c1)OCC2 c1(C(N(C2CN(C(CCCOCCOC)=O)C2)C)=O)ccc(CC2CCC2)cc1 c1(C(=O)NC2CCCN(C(C(C)=C3CC3)=O)C2)cccc2[nH]c(=N)oc12 C(=O)(C(C(C)CC)N(C)C(c1ccc(C)s1)=O)NCCCCCC#C c1(C(=O)NC(CN(C(CCOCC#C)=O)C)(C)C)cc2c(CC)cccc2[nH]1 C1(NC(c2cccc(OC)c2)=O)CC(F)CN(C(C2CC(O)C2)=O)C1 C(CC(F)F)(C(=O)NCc1nn(C)cc1C)N(C(C(C)=C1CC1)=O)C CC1(CNC(=O)C2CC2)CC(F)(F)CN1C(=O)C(=O)Nc1ccc(Cl)cc1 C(=O)(C1=NOC(c2ccccc2)C1)NCCNC(C=C(CC)C)=O N1(C(C2=NOC(CNC(=O)CCC3CCCOC3)C2)=O)CC2(CNC(=O)OC2)C1 Cc1cc(NC(C23CCC2C3)=O)ccc1NC(c1cc2n(n1)CCC2)=O C1(CCC)C(=O)NCCN1C(C1(NC(=O)CC(C)(C)CC)CC1)=O c1(C(N2CC(C(=O)NCc3cc(Cl)ccc3Cl)OCC2)=O)c(F)ccc(Cl)c1Cl C1(C(=O)NCCCCCCNC(c2c(C)cccc2F)=O)CC2COCCN2C1 C1(CCC(C)(C)NC(=O)C(F)F)CCCCN1C(=O)C=CC1CCCC1 c1(OC)ccc2occ(C(=O)NCC3(C)CCN(C(=O)CCNC(C)=O)C3)c2c1 N1(C(C2N(C)CCN(C)C2)=O)CCC=C(C(=O)N2CC(O)CC2(C)CO)C1 c1(OCCC(=O)NCCCNC(c2c(N)nccn2)=O)ccc(F)cc1Cl N1(C(c2[nH]c(=NCC)sc2)=O)CCCC2(CC(NC(=O)CP(C)(C)=O)CO2)C1 Cc1cc(N(C(C)(C)CNC(c2nnn(C(C)(C)C)n2)=O)C)nc(CO)n1 C12(C(=O)NCC3N(C(COCC(=O)NC)=O)CC3)CCCCC(F)(C1)C2 C1(C(=O)NCCCC)CC12CN(Cc1ccc(C(=O)OC)nc1)C2 C(C(C)(CO)NC(=O)COCCOC)NC(C1(C(=O)NC)CC1C)=O C=C(C)CCCC(=O)N(C)CC1(CNC(C2CN(S(N)(=O)=O)C2)=O)CC1 N1(C(c2c(CC)occ2)=O)CC(O)(C2CCN(C(=O)CC3CCCC3O)CC2)C1 N1(C(CC(C)SC)=O)CC2(C=C(C(=O)N3CC4(CC(F)C4)C3)CO2)C1 C(C(=O)NCCC(C)NC(c1ccnc(N2CCCC2)n1)=O)(C(C)C)OC C1(C(N2CC(N(C(=O)CCC3OCCO3)C)C2)=O)CS(=O)(=O)CC(=O)N1 C1(C(N2C(C)(COC)CCC2)=O)CC(NC(C2CC(O)C2)=O)C12CCC2 CC(C)(O)C#CC(=O)NC1(CCC(=O)NC2(N3CCCC3=O)CC2)CCC1 Cc1nc(NC(C2C3CC2N(Cc2nc(C)n(C)n2)C3)=O)ccc1Br CC1CCN(C(=O)CN(C)C(c2cncn(C)c2=O)=O)C(C)C1 C1(CNC(COCc2cc(C)on2)=O)C(C)CCN1C(c1ccc(C#N)s1)=O C(CC)(CCC(=O)N1CCCC1C1CCOC1)NC(C(CC)=CC)=O c1(NC(C2CN(NC(=O)OCC)C2)C)ccc(CS(=O)(=O)Cc2ccc(F)cc2)cc1 C1(C(=O)NC(C2CCCCC2)C(=O)NCC2(SC)CCC2)CC(O)C(F)C1 C1(C2(O)CCC2)(C(=O)NCC(C)(O)CNC(c2cc(C3CCC3)no2)=O)CC1 N1(S(CC(=O)OCC)(=O)=O)CCC2(CCCN2C(c2ccc(I)cc2F)=O)C1 C1(NC(c2cnn(C)c2Cl)=O)CN(C(c2cc3c([nH]2)CCC3)=O)C2CCCCC12 N1(C(C2(OC)CCOC2)=O)CCC(C=CC(=O)NC2C(=O)OCC2CO)CC1 CC1(C)CCn2cc(C(=O)NC3CN(C(C45CC(F)(C4)C5)=O)CCC3F)nc2C1 c1(C(=O)NC(C2CCN(C(=O)CCOCC(F)(F)F)C2)C)ccn(C)c(=O)c1 N1(C(c2cc(C)c(I)cc2)=O)CCC2(C)C(C1)C2(Cl)Cl c1(N2CCC(NC(C3CC(C)SCC3)=O)C2)cc(Cl)nc(CS(C)(=O)=O)n1 C1(C(=O)NC2CC(CNC(CSCC(N)=O)=O)C2)C2COCC12 c1(C(=O)NC(CN(C(c2nnc(C)s2)=O)CC)C)ccc(C)nc1N C1(NC(CC=CC=C)=O)C=CC(C(N2CCC(C(CC)CC)C2)=O)C1 c1(NC(=O)CC2CN(C(C3CC3F)=O)C2)cccnc1I N1(CC)OCC(NC(=O)C(c2cn(C)nn2)NC(=O)CC(C)COC)C1=O Cc1cnncc1C(N1CC=CC1C(=O)NCC(C)(C)N(C)C)=O C1(CNC(C(C#C)(C)C)=O)COCCN(C(c2cccnc2OCC)=O)C1 CC1(C)CC(c2ccccc2)N(C(=O)C(c2cc(F)cc(F)c2)F)C1 c1(CN2CC(CNC(c3ncn(C)c3)=O)C2)nccc(OCC(F)(F)F)n1 C1(NC(C2(CC)CCCC2O)=O)CCN(C(=O)CCN2CCOCC2)CC1OC c1(C(N(CC(C)N(C)C(c2ccc(Cl)cc2)=O)C)=O)ccc(Cl)nc1N CC(C(=O)NC1CCC1C(=O)NCC(F)Cl)=C1CC1 [N-]=[N+]=NC1CCC(C(N2CCCCC2C(=O)NCc2cc(O)ccc2F)=O)C1 C1(NC(C2COCC(C)(C)O2)=O)CC2CCC(C1F)N2C(c1coc(CO)c1)=O C1(CC=C)(NC(=O)CC(C)C2CC2)CCN(C(C2(C)CC(C)(C)C2)=O)C1 N1(C(CNC(=O)OC(C)(C)C)=O)CCC(NC(=O)C#CC2CC2)C1C1CC1 N1(C(CCNC(COC)=O)=O)CCC2CCCC(C1)N2C(=O)CCC(F)(F)F C1(C(=O)NC(CNC(c2scc(C)c2)=O)C2CCC2)CC(C)CC(=O)N1 c1(CC)[nH]nc(C(=O)NCCCCNC(=O)CC2C(C)(C)C2(C)C)c1Br N1(C(C2(F)C(C)C2)=O)CC2OCC(NC(c3ccsc3-n3cnnn3)=O)C2C1 N1(C(C=CC)=O)CCN(C)CC1CNC(c1cncc(C#N)c1)=O C1(N(C)C)CCCN(CCC(=O)N(CCNC(=O)Cc2cncn2C)C2CC2)C1 CC(C)CC(CNC(=O)CCc1ccccn1)C(=O)NCCN1CCCCC1 N1(C(CCNC(c2nc3c(s2)CCCC3)=O)=O)CCC(C2(O)CC2)C1 C1(C(N2CCC(C)(CCCC)C2)=O)(NC(C(C)OCCC=C)=O)CCC(C)(C)C1 C(=O)(CCCCCN(C)C)NCCC(C)NC(c1n[nH]c(=N)[nH]1)=O CC(C)C(CCC(=O)NC1(CO)CCCCC1)NC(C12CCC(CC1)C2)=O C1(CCC)CN(C(C2CCCCC2F)=O)CC1C(=O)NCCN(C)C(=O)C1CC1 c1(C(N2CCC(C)(NC(CCOCC#C)=O)C2)=O)cc2c(s1)CCC(C)C2 CCCCCCCCC(C)C(=O)NCC1CC(NC(=O)C(O)CCn2cncn2)C1 c1(CCC(=O)NC(C(C)NC(=O)CSc2ccccn2)(C)C)cc(F)ccc1F C1(C(=O)NC(C)C(C)NC(c2cncc(N)c2)=O)(OC)CCCCCCC1 C1(CNC(c2ccc(CC)nc2)=O)COC(C)(C)CN1C(=O)C=C(C)C(C)(C)C c1(OC)ccc(Br)nc1NC(c1nc(-c2cnn(CCF)c2)cs1)=O C1(CNC(C(C)(C)c2sccc2Cl)=O)(NC(c2ccccn2)=O)CCOCC1 CC(C)CS(=O)(=O)CC(=O)NC1C=CCN(C(c2ccnc(C(C)(C)C)n2)=O)C1 C1(C(C)C)CN(C(=O)C(C)C2(O)CCC2)CCN1C(C1CC1(F)F)=O C(=O)(C(S(C)(=O)=O)C1CC1)NC1C(C)CN(C(c2csc(C(C)(C)C)n2)=O)C1 c1(NC(C2OCCN(Cc3ccc(C)cc3F)C2)=O)cccc2nc(O)oc12 S(=O)(=O)(c1cc2sc(=NC(CCO)C3CCC3)[nH]c2cc1Cl)N(CCCCC)C N1(C(C(CCC)(C)C)=O)CCC(NC(C2(C)CCCS2(=O)=O)=O)CC(O)C1 c1(C(=O)OC(C)C(=O)NCc2ccc(F)cc2)cc(S(C)(=O)=O)cs1 N1(C(c2ccc(N(CCC)CC)cc2)=O)CC(NC(=O)CC(C)COC)C(C)(C)C1 c1(OCC(=O)O)ccc(CCNC2CCC(CN)C2)cc1.c1(C=O)ccc(Cl)cn1 c1(OC)c(C)ccc(C(=O)N(C(C)CCNC(=O)C(C(C)C)NC=O)C)c1F c1(OC)ccc(-c2nc(CCN3CCCCC3)nn2CC(C)C)nc1OC N1(C(C2CC2CCC)=O)CCN(C(=O)COCc2ccccc2)C2(CC2)C1 c1(C(=O)NCC(C)(CO)NC(C(CSC)C)=O)ncnc2cc[nH]c12 c1(CC(=O)N(CCNC(C2CC(CC)C2)=O)C)ccc(OC)c(OC)c1Cl c1(C(=O)NC2CN(C(C(C)=CC)=O)CC2F)cc(OC)c(OCC)c(Br)c1 c1(C(=O)NCC(C)NC(c2ncc(Cl)n2C)=O)c(C#N)cnn1C C1(NC(C2CC(F)(F)C2)=O)CC2CCC1N(C(=O)C(c1ccc(F)cn1)(F)F)C2 c1(OC)c(C)cc(CNC(=O)CNc2ccccc2I)cc1C C1(C(=O)NCC(CC)NC(=O)C(C)Cc2ccccc2F)CCCC(C)(C)C1 C1(NC(C(CNC(C2(CC(C)C)CC2)=O)O)=O)CCN2CCC1C2 c1(C(C)C)cc(F)ccc1NC(=O)C(=O)NCc1nccn1-c1ccccc1 C(C)(C)(CC(=O)NCCCC1(NC(C2CC(C)OC2=O)=O)CC1)SC c1(CC(=O)N(CC(CNC(C(C)=C(CC)C)=O)O)C)ccc2nn[nH]c2c1 c1(C(N(CCNC(=O)C(C)Cn2ccc(C)n2)CC)=O)ccc(O)c(Cl)c1 c1(CN2CCC(OCCCCc3cnccc3)C2)cc(C2CCCC2)on1 CC1CN(C(c2cc(O)cc(O)n2)=O)CCC1NC(c1ccc(C(N)=O)nc1)=O c1(N(C)CC2CCN(C(C(C(C)O)(F)F)=O)C2)nc(Cl)nc2c1COCC2 C1(CNC(=O)CC(F)(F)F)CN(C(=O)COC2CCCOC2)CCCO1 Cc1cc(O)cc(=O)n1C(C)C(=O)NCCC1CN(C(C2(CF)CC2)=O)CCO1 C(=O)(CCCCN1CCOCC1)NC(CC(C)NC(C1C2CCC(=O)C12)=O)C c1(OCC)ncccc1CC(=O)NCCNC(C1CC(=O)N(CC(F)(F)F)C1)=O CN1CCOC(C(=O)NC2CCN(C(c3cnns3)=O)C23CC3)C1=O Cc1ccc(C2OCCCC2C(=O)OCCCCCOc2ccccc2)cc1 c1(C(=O)NCC2CCN(C(c3cc(C)ncn3)=O)C2)cc2ccccc2o1 N1(C(c2c(C)coc2)=O)CC2CCN(C(C3CCC(=O)N3)=O)CCC2C1 c1(CC)cccc(CC)c1C(=O)N(C)CC1CN(C(c2cncc(O)c2)=O)C1 CCC(CC)CC(=O)NCc1nc(CNC(=O)Cc2ccc(O)c(C)c2)cs1 CCCC(C)(C)CC(=O)NCC(CC(F)(F)F)NC(c1cnn(C2CC2)c1C)=O C=CCC(CC)C(=O)N(CCC)CCNC(c1ccc(=O)n(CCCC)c1)=O C1(CNC(C2(OCC)CCOC2)=O)CC2CCC1N2C(c1cnc(C(C)C)o1)=O CC(C)C(CCN(C)C(c1occc1C1CC1)=O)NC(=O)C=C1CC1 C1(CC(=O)NC(CNC(=O)CCC2CCC2)C2CCC2)CCCO1 C(=O)(CC(C(F)F)C(C)(C)C)NC1C2CN(c3snc(C)c3C#N)CC21 C1(CNC(C2(OC)CCC2)=O)CN(C(C2CCC3(CC3)C2)=O)C2CCCCC12 C1(C(=O)NC(C(C)C)C(C)C)CN(C(c2cccc(CO)c2)=O)CCN1C N1(C(C(c2cncnc2)C)=O)CCC2CC12C(=O)NCCC(C)C(F)F C(C)(CCC(=O)NC1CCS(=O)(=O)C1)NC(C=C(CCC)C)=O N1(C(C(C)(O)C2CCC2)=O)CCCCC(CNC(c2ncsc2Br)=O)C1 C12(C(=O)NCc3c(C(=O)NC(CCC(=C)C)C)nco3)CCCC1CCC2 CC(CC(=O)NCCC1(C)CCN(c2nnn(C)n2)C1)CC(C)(C)C C=CCC(C)(C(=O)N1CCOCC(N2CCOCC2)C1)NC(=O)OC(C)(C)C Cc1nonc1CC(=O)NCc1cn(CCNC(=O)CN2CCCC2C)nn1 C=CCC(C)C(=O)NCc1cc(C(=O)NC(C2(OC)CCC2)C)n[nH]1 C1(C(=O)NCC(F)Br)(CNC(CCNC(N)=O)=O)CCOC1 N1(Cc2ccc(CC(=O)OC)[nH]2)CCNC(=O)C1C C1(NC(C2CCCC2O)=O)CC2(C1)CC(NC(C1CC1(F)F)=O)C2 C#CC1(C(N2CCC(c3nc[nH]n3)C2)=O)CCN(C(c2cnc(OC)nc2)=O)C1 C1(C)(C(=O)NCCC(C)CCNC(=O)CCCn2ccnc2)CCCC(F)(F)C1 c1(C(N2CC(NC(C(C)(C)C)=O)C(O)C2)=O)nc2c(s1)CCC2 c1(NC(C2N(Cc3c(C)noc3C)CCC2)=O)ncc(Br)nc1CO CC(C(C)(C)CN(C)C)NC(=O)CC1(NC(=O)Cc2cccnc2)CC1 N1(C(C(C(CC)CC)C)=O)CCCCCC(N=c2[nH]n3cc(C)nc3s2)C1 c12ccccc1N(C(=O)C(C)Cn1cccn1)C21CC1.C(=O)(CNC(=N)N)OC c1(C(=O)NC(CC)CC)conc1C(C)NC(=O)COc1ccsc1 c1(CCCC=C)ccc(C(N2CC(CNC(c3nccn3C)=O)C3CC23)=O)cc1 Cc1c(C(N2CCCC2C(N2CCSCC2)=O)=O)cccc1O CC(CC(N)=O)C(=O)N(C)CC1CCN(C(=O)Cc2cc(F)ccc2O)C1 C1(NC(C2(C#C)CN(C(c3ncn4ccccc34)=O)C2)=O)CCc2n[nH]cc2C1 N1(C(C=C(C)C(C)C)=O)CC=CCC1C(=O)NC(CO)C(C)(C)C C12(C(N3CC4(N(C(CNC(N)=O)=O)CC4)C3)=O)CCCCC1OCC2 c1(OC)ccc(Cl)cc1C(N1CC2CC(NC(C3CC(=O)NC(C)C3)=O)C1C2)=O c1(NC2CCN(C(N(CC(=O)N(c3ccccc3)C)C)=O)C2)ccc(Cl)s1 C(C)(CS(C)(=O)=O)N(CCC)C(=O)NCc1csc(CC)n1 n1(CCOC)ccc(=NC(=O)CC2CCC(NC(=O)CCCn3ccnc3)C2)[nH]1 C(c1cccc([N+](=O)[O-])c1)=CC(=O)N(C)CC1CN(C(C(F)OC)=O)CC12CC2 CC1(C)CC(CO)CN(C(=O)C(C2(C)CC2)NC(c2ccc(C#N)cn2)=O)C1 C1(NC(C2C(C)OC(C)C2)=O)Cc2ccccc2C1NC(c1cc(Cl)n(C)n1)=O C1(COCC(=O)N(C2CC(NC(C3CCC(O)C3)=O)C2)C)CCOCC1 Cc1cc(Cl)c(C(=O)NCC(C)CNC(=O)CN(C)Cc2ccccc2)cc1N c1(OC)c(C(N2CCC(n3cccc3)C2)C(=O)NCCCF)ccc(Br)c1F c1(C(N(CC(C)N(C(CCOCC)=O)C)C)=O)cn(C(F)F)cn1 c1(CNC(CCOCC#C)=O)ccc(CCNC(c2ccoc2C(C)C)=O)cc1 N1(C(c2ccc(COC)s2)=O)CC2CCCC2(CNC(C2CC23CCC3)=O)C1 C(CNC(c1c[nH]nc1-c1ccco1)=O)(N=c1nc[nH]s1)c1c(OC)cccc1 C(=O)(C(C(C)C)c1ccc(F)cc1)Nc1c(C(=O)NC)ccs1 CCCC(C(=O)NCC12CC1CN(C(=O)C=Cc1cccnc1)C2)OCC c1(COC)cccnc1C(=O)NC(CNC(C1(C)CCCC1O)=O)CC(C)C N1(C(c2ccc(=N)[nH]c2)=O)CC2(NC(c3cc(-c4ccns4)on3)=O)CCC1C2 n1(CC(=O)N(C)CC2N(C(CCC=C=C)=O)CCOC2)cc2ccccc2n1 C1(CC)CN(C(c2coc(C(F)F)n2)=O)CCC1NC(c1nc(=O)n(C)[nH]1)=O C1(C)(NC(CN(C(C(C(=O)OCC)OC)=O)CC)=O)CCC(C)=C(C)C1 C1(CNC(c2c(C)c(N)ccc2)=O)(NC(=O)C=C2CCC2)CCC(F)(F)CC1 C(=O)(CCCCCN(C)C)N(C(C)C(=O)NCC(F)(CC)CC)CC CC(C#N)CCC(=O)N1CCCN(C(C2(C)C=CCCC2)=O)CC1 C1(NC(C2CC(CC)(CC)C2)=O)CCCC(C(=O)NCCOC2CC2)C1 c1(C(N2CCc3ccc(Br)cc3C2)C(=O)NC)ccc2c(c1)OCC(=O)N2 C(=O)(C(C(C)(C)C)NC(c1n[nH]c(CC)c1C)=O)NC(C1CCCC1)C#C Cc1cc(N)c(C(N2CC(C3(NC(=O)C(C)OCCN(C)C)CC3)C2)=O)nc1C Cc1nc(N(C)CC2CCCN(C(=O)C(C)C3CCC3)C2)nc2ccccc12 c1(C(N2C(C(=O)Nc3c(C(C)C)ccnc3)CC(F)C2)=O)csc2ccccc12 N1(C(C2C(C(=O)OC)C2)=O)CCN(C(=O)C(C)(C)SC)CC1C(C)C C(=O)(C1=CCCC1)N(C1CN(C(=O)CCc2cccnc2)CC1F)C CCC(CC)CCC(=O)NCCOC1CCN(C(c2cnccc2Cl)=O)C1 CC1Cc2c[nH]nc2C(C(=O)NC2(CCNC(c3c(Cl)nn(C)c3Cl)=O)CC2)C1 c1(C(=O)NC2CC(CNC(C3CCSC3)=O)C2)cn2cc[nH]c(=O)c2n1 C1(C(=O)NCC2OCCCN(C(c3nc(C)n(C)n3)=O)C2)CCC(N=[N+]=[N-])CC1 C1(NC(C2(CC)CCN(C(c3cncc(C#C)c3)=O)C2)=O)CC1C1CCCCC1 C1(NC(Cc2c(C)nn(C)c2)=O)CCN(C(=O)Cc2ccno2)C12CC2 c1(C(N(C2CCN(C(=O)CO)CC2)CCOC)=O)ccc2cc(C)ccc2n1 n1(CC)c(CNC(=O)C(C)N(C(=O)CCC2(C)CCC(=O)N2)C2CC2)cnc1C c1(COC(c2c(C)[nH]nc2C(F)(F)Cl)=O)cccc(Cl)c1O c1(OC)cc(C(=O)N(CC(C(=O)OC)C2CCC2)C)cc(F)c1OC C1(NC(CC)=O)CN(C(C2CCN(S(=O)(=O)C(F)F)C2)=O)CC2(CC2)C1 CC1(C(N2CCOC(CNC(c3cc(N)cc(O)c3)=O)C2)=O)CCCC(F)(F)C1 C=CCC(C(=O)NC1CN(C(=O)CC23CCC(CC2)OC3)C(C)(C)C1)C(C)C C=Cc1cnn(C)c1C(=O)NCC1CCC(C)CN1C(=O)CC1CC(C)(C)C1 N1(C(C(CSC)OC)=O)CCC2C(C(=O)NCCCn3cnnc3)C2C1 C(CCNC(=O)OC(C)C)(C(C)C)Oc1ccc(COCC)cc1 CC(C)CC(F)C(=O)N1CCCCC1C1CCN(C(c2n[nH]cc2F)=O)CC1 C1(NC(=O)CCCn2cccn2)CC1C1CCCN(c2ccncc2[N+](=O)[O-])C1 C1(C(N2CCC(CCC(C)C)C2)=O)CCN(C2CCCCC2)CC1 CCC(CNC(=O)NC1C2CC3C(C2)C13C(=O)OC(C)C)(CC)C(N)=O C1(NC(c2cnco2)=O)CN(C(C23CCCC2C3(F)F)=O)C2CCCC12 C(=O)(CC(C)(F)F)NC1CC(CC(=O)NCC2N(C(C)=O)CCC2)C1 C1(NC(CNC(CNC(Cc2cc(C)sc2)=O)=O)=O)CC2C=CC1C2 C1(CCNC(c2cc(=O)cc[nH]2)=O)COCCN1C(=O)C=Cc1cnc[nH]1 Cc1ncsc1C(=O)NCCC(C)NC(c1ncoc1-c1cccs1)=O Cc1cn2cc(C(=O)N(CC(C)(C)CNC(=O)Cn3ncnn3)C)nc2s1 C1(NC(CCCOCC)=O)COC2CN(C(=O)Cc3ccc(C)nc3)CC12 c1(C(=O)NC(CC)CN(C(=O)C(O)CC(C)C)C)cc2c(s1)CCCCC2 Cc1c(F)c(CN2CC3OCCC3(C(=O)O)C2)cc(Br)c1F C#CC1CC2CCC1N(C(c1cnn(CCNC(C3CCCOC3)=O)c1)=O)C2 C1(OC)CC(NC(=O)CCC(=O)N(C)C)CN(C(c2cn(CCF)nn2)=O)C1 N1(C(c2cn(C)nc2)=O)CC2CC1CC2NC(c1cccn(C2CCC2)c1=O)=O CC(C)(C)C(C(=O)NCCc1sccc1Cl)n1cc(-c2ccccc2)nn1 Fc1ccc(C2CCCC(NCc3ccc(-c4ccsc4)nc3)C2)cc1 N1(C(C)=O)CC2CC1CN2C(=O)C(C(C)O)NC(=O)CC(C)C(F)F C(=O)(CCCCC(N)=O)NCC(c1ccccc1F)NC(CN(C)C(=O)C1CC1)=O c1(C(=O)NC(C2(O)CCN(C(C3(CC4CCC4)CC3)=O)C2)C)cc2ccsc2s1 N1(CCC(N2CCC(N(C(=O)CCc3ccc(C)s3)CC)C2)=O)CCOCC1=O C1(CCC)(NC(c2ccsn2)=O)CCN(C(c2ccc(O)c(Cl)n2)=O)CC1 C12(NC(CCCCCN(C(C(C(C)(C)C)OC)=O)C)=O)CCC(CC1)C2(C)C N1(C(CC2(C)CCC2)=O)CCCCC(C2CN(C(=O)CC3COCCO3)C2)C1 C(=O)(CCC(F)(F)F)N1CC(SC)C(NC(=O)C(C)OCC2CCCO2)C1 N1(C(c2ccn(CC)n2)=O)CC2CCC(C1CO)N2OC.C12(CC)CCN1C2=O C1(C(N(C)CC)=O)CC(NC2CCN(C(=O)CNC(N)=O)C2)CCO1 C1(CNC(c2n(CCOC)ncc2)=O)C2CC2CN1C(c1cc(C)nn1C)=O C1(NC(c2nnc(C)s2)=O)CCN(C(=O)C(CO)N(C)C)CCC1(F)F Cc1ccnc2sc(C(=O)NC(CNC(=O)C(F)n3cccn3)C3CC3)c(C)c12 c1(SCC(c2cc(C)n(C3CCS(=O)(=O)C3)c2C)=O)cc2ccccc2n1C C(C(CC(C)C)C(=O)NCC1CCCCC1(C)C)NC(CCSCC)=O c1(C(=O)OCC)noc2c1CN(C(=O)NC1CCCC13CCCO3)CC2 C12(C(=O)NCC3(C(C)C)CC3)CC(C)(CN1C(c1cc(C(F)F)[nH]n1)=O)C2 Cc1nn(C)c(Cl)c1C(=O)NC1CCCC1CNC(=O)C(N1C(=O)CCC1=O)C N1(C(c2c(CC)onc2)=O)CC(C)N(C(C2C3CCC2CC3)=O)CC1C N1(C(c2cc(Cl)ncn2)=O)CCC2(CCC(C(N3CCC3)=O)C2)CC1 N1(C(CCC=C)=O)CCCC1(CNC(=O)COC1CCCOC1)COC O=C(CC(C(F)F)NC(c1ccccc1F)=O)NCCCC1CCCCO1 Fc1ccc(CNC(=NCCN2CCCC2)NCC2CCC23CCC3)c(F)c1Cl C(C)(C)(C(=O)NC1CCN(C(C2CC2C(C)C)=O)C1)NC(=O)OC N1(C(c2cccc(CNC(C3CC=C(C)CC3)=O)n2)=O)C2C=CCC1CCC2 N#Cc1nccc2cc(OCc3ccc(Cl)c(Cl)c3)ccc12 C(=O)(C1=CCC(NC(=O)CC2CCCOC2)C1)NCCOCC CCCCC(=O)C(=O)NCc1nnn(C)c1C(=O)NC1CCOC1C C(=O)(CCCC(C)(C)C)NC(CNC(C(C)Cc1ccncc1)=O)CC(F)(F)F C=CCC(CC(C)C)C(=O)N1CCC(CNC(=O)C(CC)(CC)CC)C12CC2 N1(C(Cn2cnc(C#N)n2)=O)CCOC2(CCN(C(c3csnc3Cl)=O)CC2)C1 c1(OC)cccc(Br)c1C(N1CCN(C(=O)Cc2ccc(O)cn2)C(CO)C1)=O n1(CC(=O)NCC(CNC(C(C)=C(CC)C)=O)(C)O)ccc(Br)cc1=O C(C(C)(C)CC(=O)NCC1(C)CCN(C(c2conc2C2CCCO2)=O)C1)OC C1(CCC(=O)NCCCCC#C)CCCCN(C(=O)C(CC(C)C)N(C)C)C1 C1(C(N(C2CCN(C(=O)C(C3CC3)SC)C2)CCC)=O)CC2CCC(C1)N2C N1(C(CCOCC#C)=O)CCC(=CCNC(=O)C(F)=CCC)CC1 CCCCC(C(=O)NCC(C1CCCC1)NC(=O)C(F)(F)CC)NC(N)=O C1(C)(C(N2CC(NC(CC3C=NN(C)C3=O)=O)C3(C2)CC3)=O)CCS(=O)(=O)CC1 C1(CNC(CCCOCCC)=O)CCN(C(C2(O)CCOC2)=O)CC1(F)F C1(NC(=NCC(=C)C)NCc2cncc(OCCO)n2)CCc2ccccc2C1 C1(NC(CNC(=O)OC)=O)CCCCC1N=c1[nH]ccnc1F C(=O)(C1CCCc2scnc21)NCC1CN(C(c2nc(OC)c(F)cn2)=O)C1 N1(C(C(CC)N(CC)CC)=O)CCC2(CC1)CC2C(N1CCCC1c1ccon1)=O C1(C(=O)NC(C(=O)NC2CN(CC)CC2C)Cn2ccnn2)CC(C)(C)CCO1 C1(C(=O)NCC2C(C)CN(C(C3(C)CC4CCC3C4)=O)C2)Cc2ccccc2C1 c1(C(N(CC(CC)NC(=O)C#CC2(C)CC2)C)=O)cccc(Br)c1Cl C1(CC=C)(NC(=O)CCOCC)CCCN(C(C2(C(=O)N(C)C)CC2)=O)C1 C(=O)(C(C#N)C(C)(C)C)N1CCCC(C)(C(=O)NCC2CC(F)(F)C2)C1 N1(C(C=CC)=O)CC(F)(F)CC1C(=O)NC(C)C N1(C(CCNC(C2(OC)CCC(C)C2)=O)=O)CC2C3CCC(C3)C2C1 C(C(C)(O)CNC(C1CC1(c1ccccc1)C)=O)N(C(=O)NC)C1CC1.C1C(=O)N1 C(=O)(C(CNC(C1COCCC1C)=O)C(C)(C)C)NCc1cncc(CC)c1 c1(C(N2CC(C(=O)NC(CCOC)(C)C)C(O)CC2)=O)cnn2cccnc12 c1(SC)cc(C(=O)NCC(C)N(C)C(c2ccc(CCC#N)cc2)=O)oc1C Cc1cc(C(N2CCCC2(C)CNC(=O)Cn2ncnn2)=O)cc2ccoc12 C1(NC(c2ncc(CC)cn2)=O)CC1C1CCN(C(=O)CC(C)(C)C)CC1 O=C(C1=C(Cl)CCC1)NC1CCC(CNC(c2cc[nH]c2)=O)C1 N1(C(CC2(C)CCC2)=O)CCN(C(=O)CCC2CC2)C(CC(F)F)C1 c1(C(=O)NCC(CCNC(C=CCCC)=O)O)cc(CCC)c(C)s1 CC(N=[N+]=[N-])C(=O)N(C)CC1CCCCN1C(=O)CCCC1CC1 CCC(O)C(C)C(=O)NCC1(C(N)=O)CN(C(=O)C2=CCCS2)C1 C1(C(=O)OC)CC(N(C)C)CN(C(=O)C(=O)N(CCCCCCCC)C)C1 Cc1cc(CC(=O)NC(Cc2cn[nH]c2)C(=O)NC2CC(OC(F)F)C2)nn1C N1(CCCC(=O)NC(CNC(C2C(CC)C2)=O)(CC)CC)CCc2ccccc21 C1(C(N2C(CC(C)C)COCC2)=O)CCC(C)(C)N(C(C2(C)C=CCCC2)=O)C1 C1(O)(CNC(C(C)OCC=C)=O)CCN(C(=O)CNc2ccc(C(N)=O)cc2)C1 C1(NC(c2cc(C)c(C)s2)=O)CCCN(C(=O)CCCc2ccccn2)CC1F c1(OC)cc2ccccc2cc1C(=O)NCCN(C(C1CCNC1=O)=O)C1CC1 O=C(C1COc2ccccc21)NC1CN(C(c2cc3c(s2)CCCC3)=O)CC1F C(=O)(C(C)C(C)NC(c1oc(CNC(C2CC(=O)C2)=O)nc1C)=O)OC Cc1cc[nH]c(=N)c1C(=O)NC1CC(NC(=O)CS(C)(=O)=O)C12CCC2 C(c1ccc(Cl)s1)=CC(=O)NCC(C1CC1)NC(Cn1c(=N)scc1)=O c1(CNC(C2CCS(=O)CC2)c2n(C3(C)CC3)nnn2)ccnc(F)c1F C1(NC(C(C)c2ccco2)=O)Cc2ccccc2C1NC(=O)CCc1nc[nH]n1 c1(NCCNC(=O)NC2CC(=O)N(CC3CC3)C2)ccc(Cl)cc1 C1(CNC(c2cnc3nccn3c2)=O)CN(C(c2ccco2)=O)C2COCC2O1 C(CC(=O)N1CC(OC(F)F)C1)N(C(=O)C(C)N(C)C)CC#C N1(C(CCc2nc(C)sc2)=O)CCCC(NC(c2coc(C(F)F)c2)=O)C(F)C1 C1(NC(C2C3CC4C(C3)C24)=O)CC2CC(C1)N(C(c1ccn3nncc3c1)=O)C2 c1(OC)cc(F)c(F)cc1C(N1CCN(C)CC1CNC(C)=O)=O N1(C(C2=C(C)CCC2)=O)CC2CC(NC(=O)COc3cc(Cl)ccc3Cl)CC1C2 C1(NC(CN2CC(C)C2)=O)CC(C)CN(C(C2(F)C(C)(C)C2(C)C)=O)C1 C(=O)(C(F)CCC(C)(C)C)N1C(C(=O)NC(CCC(=C)C)C)CCC1C(C)C C(CO)(C(C)(C)CO)NC(C1(C(C)NC(=O)CC2CNC(=O)O2)CC1)=O c1(C(N)=O)cc([N+](=O)[O-])cnc1N1CCCCC(NC(=O)C(C)n2ccnc2)C1 C1(NC(CCN(C)CCO)=O)COC2(C1)CN(C(c1ccns1)=O)C2 C=CC1(C(=O)NC2CC(NC(C3(C)CC4CC4C3)=O)C(O)C2)CCOCC1 CCC(C(=O)N1CC(CNC(=O)CCN2CCCC2=O)C2(CCC2)C1)C(F)(F)F C=CC(C)(CCOC)C(=O)NC1CCN(C(c2cn3ccc(CO)cc3n2)=O)C1 C1(CN(C)C)CCC(C(N2CCC(Nc3ccccc3)C2)=O)O1 CC1=NN(C)C(=O)C1CC(N1CCC(NC(C2COCCOC2)=O)C12CC2)=O C1(C(c2cccc(SC)c2)N2CCC(OCC)C2)(NC(C)(C)C)CCOCC1 CCCC(CCCNC(=O)CCn1cnnn1)Nc1nnc(COC)s1 C(=O)(N=c1ccn(-c2ccc(F)cn2)[nH]1)C1CC2(CC(C(=O)OC)C2)C1 c1(C(N2CC(C(C(=O)NCC3CCC3CO)OC)C2)=O)csc(Cl)n1 N1(C(c2c(C(C)C)ncs2)=O)CCC(CNC(C2(O)COC2)=O)C(C)C1 C(=O)(C(C)CCNC(=O)OC(C)(C)C)N.C(C(O)CCC)NC(CNC(C)=O)=O C1(CNC(=O)CSc2nc[nH]n2)CCCCN1C(=O)Cc1ccco1 N1(C(C(C=CC)O)=O)CC(O)CC1(C)C(=O)NOCc1ccccc1 Cc1cc(OC(C)C)ccc1C(=O)NCC12CC1CN(C(=O)CC1CC=CC1)C2 CC1(C)OC(=O)NC1C(N1CC(NC(=O)C(=O)NC2(OC(F)F)CCC2)C1)=O C(CCC(=O)NC(C1CCN(C(C2CCOC2=O)=O)C1)(C)C)=CC c1(CNC(C(CC)C#N)=O)ccc2c(c1)CCC2NC(c1cc(COC)cs1)=O CC1OC2CCC1(NC(C1CC(NC(c3cccc(=O)n3C)=O)C1)=O)C2 Nc1cccc(C(N2C3CCC2C(NC(=O)C(c2ccccc2Cl)O)C3)=O)c1O N1(C(C(C)OCC)=O)CCCC1(C)CCCN(C)C(C1(C)CCC1)=O C(=O)(C(CO)C(C)(C)C)NC1C(NC(C2CCN(S(CCC)(=O)=O)CC2)=O)C1 C(N=c1nc2ncn(C)c2c(NCC(Cc2ccccc2)C(C)C)[nH]1)C1C(C)C1 c1(CNC(C2(C(N(C)C)=O)CC2)=O)cc(C(=O)NCCN2CC=CC2)no1 C(N=c1[nH]c(=NC2CCCCC2C#N)c2ccccc2[nH]1)c1c(CC)c[nH]n1 c1(C(=O)NC(CC(C)C)CNC(=O)C(C2CCCCC2)=O)cccc2cnnn12 c1(C(=O)NCC(C)(CO)NC(CC2(OC)CCC2)=O)nc(C)[nH]c1C(F)(F)F C(C#Cc1cn(CC2CC(F)(F)C2)nn1)NC(CC1C(C)CCCC1)=O c1(C(C)(C)C)ncc2c(n1)CCN(C(c1c(F)cc(Br)cc1Cl)=O)C2 N1(C(Cn2ccc(C)n2)=O)CCC(F)(CNC(=O)CN(C2CCSC2)C)C1 N1(C(C(C)C2CC2)=O)CC(S(=O)(=O)N2CCN(C(=O)Cc3n[nH]c(=N)s3)CC2)C1 c1(C(N2CC(CCC)C2)=O)ccc(CNC(C2(N(CC)CC)CCC2)=O)cn1 C1(CNC(C(C)(C2CCC2)NC(CCSC)=O)=O)C2CCCCCC12 CN1CCCC(O)(CC(=O)NCC(C)(C2CC2)NC(c2ccnc(CO)c2)=O)C1 c1(C(=O)NC2(CCNC(C(C(C)(C)C)NC(N)=O)=O)CC2)cc2c(s1)CCC2=O Cc1ccc2c(C(=O)NCC3CCCCC3NC(=O)CS(C)(=O)=O)coc2c1 N1(C(c2c(C)ncs2)=O)CC(CNC(=O)CCCCN(C)C(C)C)CCC1C Cc1cc(C(=O)NC2CCCC23CN(C(C2CCN(C)C2=O)=O)C3)c(O)nc1C Cc1ccc2snc(C(=O)NCCC(O)CNC(=O)CCc3nc[nH]n3)c2c1 C1(C(=O)NCCN(C(C2CC(N(C)CC)C2)=O)C)CCCCC1N=[N+]=[N-] c1(CC(=O)NCC2(NC(C(CC)OCC)=O)CCC2)nc(C)sc1Cl c1(C(=O)NC(C2CCCCC2)CNC(C2CC(n3cnnc3)C2)=O)ccccn1 N1(C(c2cc(COC)on2)=O)CCCCC(NC(C2OCCCC2(C)C)=O)C1 C1(NC(=O)Cc2ccccc2)CCN(C(=O)CCO)CCC1CO C12CN(CCO1)C2=O.c1(C2(N(C(COCCCN(C)C)=O)C)CC2)cc[nH]n1 N1(C(C(CCSC)O)=O)CCc2[nH]nc(CNC(=O)C(C)SC)c2C1 c1(C(=O)NC2C(NC(C=Cc3n(CC)ccn3)=O)C2)ncc(Cl)cc1Cl N1(C(C2CCC(C(N)=O)C2)=O)CCCN(C(c2sccc2Cl)=O)CC1CN(C)C C(=O)(C(=O)CC(C)C)N1CCC(OCCNC(CC2(CC)CCOCC2)=O)C1 N1(C(C2CC(C)N2C(c2ccc3n[nH]cc3c2)=O)=O)CC(C)(CO)CC1(C)C CC1CN(C(=O)Cc2nc(C3CC3)nn2C)CC(CCNC(=O)C=CCO)O1 C1(CNC(c2c(C(C)(C)C)ncs2)=O)C2CN(C(c3cc(Br)n[nH]3)=O)CC12 c1(N(CC(=O)NC2(COC)CN(C(C(COC)O)=O)C2)C)ccccc1[N+](=O)[O-] c1(C(C(=O)NCCCC2(NC(CN(CC)CC)=O)CC2)CO)ccc(Cl)cc1 CN1CCCCC(CNC(=O)C(Cn2ccnn2)NC(=O)C2=CCSC2)C1 Cc1cc(CCC(=O)NC23CC(CNC(C4CC45CC5(F)F)=O)(C2)C3)cc(C)n1 C(=O)(C(C)(C)CC(=O)OC)N1CCN(C(CN(S(CC)(=O)=O)C)=O)C(C(C)C)C1 N1(C(c2c(C)con2)=O)CC(NC(c2cc(Br)c(C)o2)=O)CC(O)C1 CCCCCC(=O)NCC(N1CC(NC(=O)C(C)CN2CCOCC2)C(C)C1)=O C1(C(=O)NC(CCC)CO)COCCN(C(c2cnc(Br)s2)=O)C1 C=CCC(C(=O)NC1COCC1NC(=O)CCc1ccc(Cl)cc1F)C(C)C c1(OC)ccnc(C(=O)NCCC(C(C)C)NC(c2cccc(N)n2)=O)c1OC Cc1cnc[nH]c1=NCCC1CCCN(C(=O)C(O)C(C)C)C1 N1(C(C(CC(C)C)NC(C)=O)=O)CC2CC(C1)N(c1ncc3ccnc-3[nH]1)C2 C1(CC)CCN(C(C2CCSCC2)=O)C1C(=O)Nc1ccccc1O C(=O)(C(C)(C)CC(=O)N1CCCC(NC(C2CCN2S(C)(=O)=O)=O)C1)OC N1(C(c2cncnc2)=O)CCCC2(CCCN(C(c3ccnc(Br)c3Cl)=O)C2)C1 C1(C2(O)CCCOC2)(CNC(c2n(C)nc(C3CCC3)c2)=O)CC1 N1(C(C23CC=CC(C2)OC3)=O)CCC(N=c2cnc(F)c[nH]2)(CO)CC1 C1(C(=O)NCC2(COC)CCC2)CCN(C(=O)C2(C)CC2(C)C)O1 c1(C(N2C(C(N3CCC(C(=O)OC)C3)=O)CC3CC32)=O)cc(Br)c(O)c(Br)c1 c1(C(=O)NC2CCN(C(CCCSC)=O)C2)cc2cc(C#N)ncc2[nH]1 C(=O)(CC(F)(F)C(F)F)N1C(CNC(C2CC2C(F)(F)F)=O)CC1 n1(CC(=O)NCC(C)CN(C(=O)C(c2cncnc2)C)C)cc(S(C)(=O)=O)cn1 C1(C(N2CC(CC(C(=O)N(CCCC(C)O)C)F)C2)=O)NC(=O)OC1(C)C Cc1cc2c(N3CCC(Oc4ccc(C(F)(F)F)cc4)CC3)ncc(I)n2n1 N1(C(CNC(=O)OCC)=O)CC(NC(c2csc(C(C)(F)F)n2)=O)C2(CCC2)C1 C1(C(=O)NC2(C)N=N2)CCCC1CN(C(C1(C)CSC1)=O)C1CC1.COC C1(NC(CCOC(C)C)=O)CCCN(C(=O)CCC2NC(=O)NC2=O)C1 C12(C(=O)OCC)CCN(C)CC1CN(C(=O)Nc1ccn3nccc3c1)C2 C1(CC(=O)NC(C2CCN(C(C(C)NC(CC)=O)=O)C2)(C)C)C(=O)ON=C1C CC(CC(N)=O)C(=O)N1CCN(C(=O)CC2CC(C3CC3)C2)C(C2CCCC2)C1 CC(CS(C)(=O)=O)C(=O)NCc1cccc(NC(=O)CCC2CCCN2C)c1 C1(c2cn(C(C)C(=O)N3CCCC3)nn2)(N(C)C)CCN(C(=O)C(F)F)CC1 N1(C(C(C)(C(F)(F)F)OC)=O)CCC2(COCCO2)C1 N1(C(C2(C)C(C)OCC2)=O)CCCC(NC(=O)CSc2ccncc2)CCC1 C1(NC(CC(=O)OCC)=O)COC2(CO)CC1C2.C12CCCN(C1)C2=O C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NC(C1CN(C(CC(C)(C)SC)=O)C1)C CC(CCOc1ccccc1)C(=O)NC1CC(NC(c2ncn(C)n2)=O)CC1O N1(C(CN(CCOC)C)=O)CCCC(C(N2CCC(C)(C)C2C)=O)CC1 C=CC1CN(C(=O)CC(CNC(C2CCC2COC)=O)OC)CC1O c1(OCCCCC)ccn(CC)n1.C1(C(N2CC(O)C2)=O)CC(C)(F)C1 c1(-n2cc(COC)nn2)ccc(NC(c2ccc(Br)cc2)(C)C(=O)O)cc1F C1(NC(CC(=O)NCC#C)=O)CC2CC1N(C(C1(N(C)C)CCOCC1)=O)C2 Cc1cc(C(=O)NC2CC3(C2)CC3C(N2CCOC(C)(C3CC3)C2)=O)cc(C)n1 N1(C(C(C)N2CCC2)=O)CCCC(O)(CNC(C2(C)CC=CC2)=O)C1 c1(C(=O)NC(C)C(CO)NC(c2ccc(Cl)o2)=O)ccccc1Br CC1CCN(C(C2(n3ccnn3)CC2)=O)CC1NC(c1ccc(Br)s1)=O c1(C(=O)NC(C)CCCNC(=O)C=Cc2cc[nH]n2)cccc(-n2cccn2)c1 N1(C(Cc2n(C)c(S)nn2)=O)CCC2CCCC(C1)N2C(C1CCOCC1)=O c1(CC(=O)NCCNC(c2cn(C3CC3)nn2)=O)cccnc1OC(F)F C1(C)(CC(=O)NCCCC(C)NC(=O)CCn2cc(Cl)cn2)CC(F)(F)C1 Cn1cc(Br)c(C(N2C3CCC2CC(NC(=O)CCC#N)C3)=O)cc1=O N1(C(CNC(C)=O)=O)CCN(C(=O)C=CC2CCOC2)C(c2ccncc2)C1 C(=O)(C(C)c1ccsn1)N(CCCNC(C1(C(F)(F)F)CC1)=O)CC C1(CNC(C=CC)=O)CN(C(=O)COCn2ncnn2)CCC1(C)C.c1(C)nc[nH]n1 C1(NC(C2CC(C(F)F)(OC)C2)=O)CN(C(C2CC(C)(O)C2)=O)CC1O c1(C(N2C(CNC(c3nn(CC)c(C)c3)=O)CC(O)C2)=O)nc(C)n(C)c1C c1(C2(C(C)NC(c3cncc(F)c3)C)CCC2)ccc(Cl)cc1 N1(C(c2c(C)cn(C)n2)=O)CCCC2C1CCN2C(C1CN2CCN1C(C)C2)=O C1(C(=O)NC(CNC(=O)NC)C2CC2)CCCCC1Nc1ccccc1 C1(C(N2CCC(CC)(CC)C2)=O)CN(C(c2cc(C#N)cs2)=O)C(C)(C)C1 c1(C(=O)ON2CCC3(C(CC)C3)CC2)cnc(O)c2ccsc12 C1(NC(C(F)=CCC)=O)CCCC1NC(c1oncc1CC)=O C(=O)(CC(COC)COC)N(C1CCN(C(=O)CCC2CC(C)C2)CC1)CC O=C1CC(C(=O)N(CCCN=[N+]=[N-])CCO)N(C(=O)CCN2CCOC2=O)C1 C=C1CCC(C(=O)NCCC(C)(C)CNC(=O)C(C(C)C)OC)CC1 c1(C(=O)NCC2=CCN(C(C(C=CC)O)=O)CC2)cccc2c1ncn2C N1(C(C=Cc2c(C)ccnc2)=O)CCC(NC(=O)Cc2cn[nH]c2)CC(C)(C)C1 C(C1c2ccccc2CN1C(C1CCCOC1)=O)NC(c1ccnnc1)=O C(=O)(CCCC(C)(C)C)NC1(CCC)CCCN(C(c2c(C)cccc2F)=O)C1 C(=O)(C(C)C(F)(F)F)N(C1CCN(C(c2nc(CC)oc2)=O)CC1)CC C1(NC(c2ccncc2C(F)(F)F)=O)CCCCC1NC(C1CC1C(F)(F)F)=O c1(C(N(C2C3CN(C(C(CC)C(C)C)=O)CC32)C)=O)c[nH]c2cccc(F)c12 N1(C(CCC(c2ccc(CC)cc2)=O)=O)c2ccccc2N(C)CCC1C N1(C(c2ccc(CC)cc2)=O)CC(NC(=O)CCn2cc(C)cn2)CC(C)C1 c1(OC)ccc(CC(C)C(N2CCC(O)(CNC(=O)C(C)=CC3CC3)C2)=O)cc1 N1(c2ccnc(COC)n2)CCC(C2CC2)(CNC(c2cnc(SC)s2)=O)C1 c1(C(=O)NOC2(F)CC=CCC2)ccccc1-c1noc(-c2ccccc2)n1 c1(-c2cccc(C(N(c3ccccn3)CCCC)=O)c2)nnc2n1CCC2 c1(OC)ncc(Cl)cc1C(C(=O)NC1CCCC1)N(CCC#N)C c12oc3ccccc3c1C2.c1(C(C)(C)C)ccccc1C(N1CCCC1CO)=O C(=O)(C1CN(N(CC2CC2)CCN(C)C)c2ccccc21)NCC C1(CNC(C(C2CC2)OC)=O)C2CN(C(=O)Cc3ccc(F)cn3)CC12 C1(CNC(c2c(C(C)C)nns2)=O)COCCN(C(c2nncn2C2CC2)=O)C1 C1(C(=O)N(CCCOCc2ccco2)CCOC)CSC(Cc2ccco2)C(=O)N1 c1(C(N2CC3(C(CNC(C)=O)CC3)C2)=O)ccc2c(c1)nc(O)n2CC1CC1 C(=O)(C(C(C)O)N(C)C)N1C(CC(=O)NC(c2nc(C)[nH]n2)C)CCC1 C1(CC)CN(C(c2cc(C3CC3)n(C)n2)=O)CCC1NC(=O)C(F)(F)C1CC1 Cc1cc(Br)c(C(=O)NCC2CN(C(=O)C3=CCSC3)C3CC23)s1 C1(CCOC)CC(N=c2cc(NCCc3ccccc3C)nc(C(C)C)[nH]2)C1 Cc1ccn(C(C)(C)C(=O)N(CC(O)CN(C)C(c2c[nH]cc2C)=O)C)n1 c1(CNC(=O)NCCC(N2CCS(=O)(=O)CC2)=O)nc2cc(O)ccc2[nH]1 c1(OC)cc(NC2CC(NC(=O)Cn3nc(C)oc3=O)C23CCC3)nc(OC)n1 C12(NC(C3CCCC3)=O)CC(CNC(c3cnc(C4CCCO4)s3)=O)(C1)C2 c1(C(=O)NCC2(O)CC(NC(C(C)NC(=O)NC)=O)C2)c(Cl)c([N+](=O)[O-])nn1C c1(NC(CCC2(C)N(C(CC3N(C)CCC3)=O)CCC2)=O)cccc2cncn12 CCC(C(=O)N1CC(F)(CNC(=O)C(C)CSc2ccc(F)cc2)C1)C(C)C Cc1cc(C)c([N+](=O)[O-])c(C)c1C(N1CC(NC(=O)C(O)C2CCC2)C(C)C1)=O N1(C(C(C=C)(C)C)=O)CCC2C(NC(c3ccccc3OCCC)=O)C2CC1 N1(C(C(CCC)NC(C)=O)=O)CCC(NC(=O)C(C)=C(C)CC)C(C)C1 C(c1ccncc1)=CC(=O)NCCC(C)NC(c1c(C(C)C)noc1)=O n1(CC(=O)N(CCOCCNC(C2CCC(C)C2)=O)C)ncc2ccccc12 c1(CC(N2C(CCNC(CN3CC(C)(C)C3)=O)COCC2)=O)ccc(F)cc1F C(=O)(Nn1cnn(C)c1=S)C1(C)CN(C(C(C=C=C)C)=O)C1 c1(C(=O)NCc2ccc(C#N)cc2)cc2n(c1)CC(N)CCC2 C(C)(C(C(C)C)NC(=O)CCc1cccc(O)c1)NC(CCOCCC)=O N1(C(c2c(Cl)cn(C(C)(C)C)n2)=O)CC(NC(C2CCCC2)=O)C(S(C)(=O)=O)C1 C1(NC(C(C)SC)=O)CCCC1(C)NC(=O)CN(CC(C)(C)C)C N1(C(C(c2cccs2)NC(c2nnnn2C)COC)=O)CCC(=C(F)F)CC1 c1(N2CC(NC(COc3c(CC)cccc3)=O)C(C)CC2)cc(C)ncc1C#N N1(C(Cc2ccc(C)cc2)=O)CC2CC1CCC2NC(=O)CC1CC2CC2C1 CC(C)C(C)(O)C(=O)NC1CN(C(c2cc(C#N)cs2)=O)CC1n1ccnn1 c1(C(N2CC(F)(c3ccccn3)C2)=O)sc(F)cc1Cl N1(C(Cn2c(C(C)C)nnn2)=O)CCC2CC2(NC(c2cn(C)cn2)=O)CC1 c1(CNC(c2c(CCNC(C3C(C)(C)C3)=O)n[nH]c2)=O)ccc(F)nc1F C1(C(=O)OC)C2CCCC2CN1C(c1coc2c1CNC2)=O C(C(CO)(CO)NC(=O)COCC1CCCO1)N(C(=O)COC(F)F)C CCC(COC)C(=O)NC1CCC1NC(=O)Cc1sc(S)nc1C CCCCC(CC(=O)N(C1CC2C=CC1C2)CC)NC(=O)CCc1ncccn1 n1(CC(N)=O)cc(NC(C2CCN2C(=O)CC2CC2)=O)cn1 CN1CCC(CC(N2CCC(C)(NC(c3cn(CC(N)=O)nn3)=O)C2)=O)C1=O c1(C(=O)NC(CCOC)C)ccccc1NC(c1cccc(C)c1)=O N1(C(CC2C(NC(CC(C)CN(C)C)=O)CCC2)=O)CCC2(CC1)CSC2 C1(C(=O)NC2CC(C)(NC(C(C(C)C)n3ccnc3)=O)C2)CN2CCCC2CO1 C(=O)(CC(O)CC(C)(C)C)NCCC1(O)CCN(C(C(CCC#C)O)=O)CC1 CC1CN(C(C23CC(F)(C2)C3)=O)CC1CCNC(C1CCCC1(F)F)=O c1(C(=O)NCC(CNC(C(c2cccnc2)C)=O)C)ccc2c(c1)N(C)CCO2 C1(c2ccc(F)cc2)(C(=O)NCCCNC(=O)CN2CC3CC3C2)CCCCC1 C1(C#N)(CC)CCN(C(C2C=CCCN2C(C2CC3CC3C2)=O)=O)CC1 N1(C(CCCN(C)C(C2CCCN2C2CC2)=O)=O)CCN(CC(N)=O)CC1 C1(CSC)COCCC1c1ccccc1.C1(N2c3cc(sn3)C2=O)CCCC1(F)F C1(NC(C(CC)NC(C)=O)=O)CC2C1CCN2C(c1ccco1)=O N1(C(C(CN(C(C2C(=C)C2)=O)C)(C)C)=O)CC2CC(C)C2C1 N1(CC)CC(NC(=O)CCC2CC(NC(=O)Cc3cc[nH]c3)C2)CCC1=O c1(C(=O)NC2(CC=C)CCN(C(=O)CC(F)F)C2)nc(C)[nH]c2nccc1-2 N1(C(C2C(C)(C)C2)=O)CCCC(C)(NC(c2ccc[nH]2)=O)C1 C(C(CC(C)C)C(=O)NCC(C(C)(C)C)NC(C1CC(=O)C12CCC2)=O)OC c1(C(N2CCC(C(=O)NCc3cc(C)cc(F)c3)C2)=O)cc(F)c(Cl)cc1C C1(C(=O)N(C(C)C=CC(=O)NC(c2cscn2)CO)CC)(OCC)CCOC1 C=CCCCCCC(=O)NC1CC(F)(F)CC1NC(=O)C(C)CSC c1(C(=O)NCCCCC(C)NC(C2CC(C)OC2C)=O)nnc2ccccc2n1 C=CC(C)(CC)C(=O)N1CCC(C)(CCNC(c2coc(C(C)C)n2)=O)C1 N1(C(C(CC)n2cncn2)=O)CCCN(C(c2cc(C)c(C)nc2C)=O)C(C)C1 c1(C(N2CCC(C)(CNC(C(CC)C#N)=O)C2)=O)cc(Br)cc2scnc12 C1(CCCC)C(=O)N(C)CCN1C(=O)NC1CCOC12CCOC2 C1(C(=O)NC(CC)CSC)(C(C)C)CCN(C(=O)C=Cc2ccoc2)C1 c1(CCNC(C=Cc2ccc(OCCCC)cc2)=O)ccc2c(c1)CCN2 CC1(C)CCC(C(=O)NCC(=O)NCC(=O)NCCC(Cl)Cl)CO1 N1(C(C(CC(CC)CC)F)=O)Cc2n[nH]cc2C1C(=O)N1CCCC1CC(N)=O CCC(C)C(O)C(C)C(=O)N1CCCC1CCC(=O)NC1(C)CSC1 c1(C(C)NC(c2csc(Cl)c2Cl)=O)ccc2c(c1)CCCO2 c1(C(N2CCCC(NC)C2)C(=O)NCC=C)cc(C)cc(Br)c1.c12nc(n[nH]1)C2 Nc1ccc2nccnc2c1C(=O)NCCC1CCN(C(C2(O)CC2)=O)CC1 C1(CN(c2c(C)cc(Br)cc2)CCO)CN(C(=O)OC(C)(C)C)CC(C)(C)O1 C(=O)(C(CC)C(F)(F)F)NC1(CC=C)CCN(C(c2ccnn2C(C)(C)C)=O)C1 c1(C(=O)NCCC2(NC(CCc3n(C)ccc3)=O)CCC2)cnn(C)c1C(F)F C(=O)(CC(O)(C(F)(F)F)c1ccc(C)o1)NCC(C(C)(C)C)NC(COCC)=O c1(C(=O)NCCOCCN(C(c2c(CC)con2)=O)C)cc(Br)ccc1C C(=O)(CCCCCC#N)N1CC(C)OC(CCNC(=O)C(C)(C)C2CCC2)C1 Cc1ccc(CCN2CC3C(CC(=O)O)C3C2)cc1[N+](=O)[O-] CC1=C(C)CC(C)(NC(=O)C(CO)NC(=O)CCc2ccccn2)CC1 Cc1[nH]c2ncnc(NCc3nncn3-c3ccccc3)c2c1C C=C1CCN(C(c2c[nH]nc2OC)=O)C(C(=O)NCC(C)C(F)F)C1 C(C(C)(CC(C)C)NC(=O)CCc1cncn1C)NC(COCCCC(C)C)=O C1(NC(c2cc(SC)oc2C)=O)CCN(C(c2ccn(C(C)(C)C)c2)=O)C(C)C1 C(=O)(CCCCCS(N)(=O)=O)N1C2CN(C(c3c(C)nc[nH]3)=O)C(C2)CC1 C(C(=O)N1CCOC(CCCNC(c2ccsn2)=O)C1)(C(C)C)n1ccc(C)c1 CCCS(=O)(=O)CC(=O)N1CC(F)CC1CNC(C1CC1C1CCC1)=O C1(N(C(CC(=O)OCC)=O)CC)CCCN(C(C2CC(c3ccccc3)C2)=O)C1 c1(CNc2nc(COC)nc(N3CCCC(C)(OC)C3)c2)cc(C#N)ccc1Br N1(C(C2N(C)C(=O)NC2)=O)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC1CCO CC1CN(C(C2(C)CSC2)=O)CCC1NC(c1cc(OCC(F)F)ccn1)=O N1(C(c2c(COC)cco2)=O)CCC(NC(C2(C)COC2)=O)C(C)C1 N1(C(Cn2c(C)ccc2C)=O)C2CCC1CN(C(c1cnn(C)c1CO)=O)CC2 N1(C(C(c2cn(C)nc2)=O)=O)CC2(C1)CN(C(C1CCCCC1F)=O)C2 C1(C(=O)NCC(O)CCOC)(CC)CN(C(=O)CCc2ccoc2)C1 n1(CC(=O)NCC2CN(C(C3C(C)COCC3)=O)C2)cnc2ccccc2c1=O c1(OC(C)C(N2CCC(C)(NC(=O)CC3(C)CCC3)C2)=O)ccc(F)cc1Cl C1(C(=O)NC2C=CCN(C(C3(CO)CCOCC3)=O)C2)CC2CCCCC12 c1(NC(C2(C)N(C(c3c(Cl)ncc(OC)c3)=O)CC2)=O)ncc([N+](=O)[O-])cc1I c1(C(N2CCC(O)(CNC(=O)C3=CCCCC3)C2)=O)cc(Cl)cc2ccccc12 C1(n2cc(-c3nc(C(C)(C)C)sc3)nn2)CN(C(C2(C)COCCO2)=O)CC1O CCCC(C(=O)N(C)CCOCC)NC(=O)CC1CCCN1C CC1(CNC(c2cc(C3CCCCC3)[nH]n2)=O)CCN(C(C2CCCCO2)=O)C1 c1(C(=O)NCC(C2CCCC2)NC(C(C)NS(C)(=O)=O)=O)ccc(F)cc1OC N1(C(C2N(C(=O)NC)CCC2)=O)CC2(CC(NC(=O)CCC(C)C)CO2)C1 c1(C(N2CCN(C(CCC(C)OC)=O)C(CF)C2)=O)ccc(Cl)c(C)c1Cl c1(N(C)CC2CCCN(C(C(COC)O)=O)C2)nc(C(F)F)nc(=N)[nH]1 c1(C(=O)NCCC(CNC(C2CCC(C)(C)OC2)=O)O)cc2cccnc2[nH]1 C(CNC(c1cc(F)ccc1OC)=O)(C(C)C(C)C)NC(c1ccn(CC)n1)=O C1(CC)C(NC(=O)CSC(F)(F)F)CCN1C(C1CC(C)N(C)C1)=O c1(C(=O)NC2CCC(CNC(C3CCC(CC)O3)=O)C2)cc2cc[nH]c(=O)c2s1 N1(C(c2c(C)cno2)=O)CCC(NCC2CCCCC2C)C(C)C1 c1(NC(C(CC)OC)=O)ccc2c(C(=O)NC3CCCCC3)ncn2c1 C(=O)(C#CC1(C)CC1)N(CCCCCNC(=O)COCC1CCC1)C c1(CCCC(=O)NCC(C)NC(=O)Cc2ccnn2C)ccc(Br)cn1 c1(N2CCC(OCCNC(C3CCCOC3)=O)C2)nccc(-n2ccnc2)n1 N1(C(c2n(C)c(O)nc2)=O)CC2CC(NC(c3csc(C(C)(F)F)n3)=O)CC1C2 N1(C(c2cc(C)nn2C)=O)CCN(C(c2cc(CO)oc2C)=O)C(CO)C1 N1(C(Cc2ccc(SC)cc2)=O)CCN(C(=O)C(F)=CC2CC2)C(C)C1 C1(C)(C(=O)NCCN(C(c2cnc(C3CCOC3)s2)=O)CC)CC(C(C)C)=NO1 N1(C(CC(=O)OC)=O)C(C)CC2CN(C(=O)CCc3cnc(C4CC4)o3)CC12 N1(C(C(C)(C)C(F)F)=O)CCC2(CCC(NC(=O)C3=CCOC3)CC2)CC1 C(CN=c1[nH]c(N2CCOCC(C)(F)C2)nc2c1CSC2)c1c(C)cccc1 CC1(C)C(CC(=O)NC2CCC(NC(=O)CNC(=O)Cn3cncn3)C2)C1(C)C C1(CNC(c2n(CC)ncc2)=O)CCCC(C)CC1.n12cc(cn1)C(=O)NCC2 CC(C)(C)C(C)(C)C(=O)NC1CN(C(=O)CCc2ccco2)CC1O C1(CC(=O)N(C)CC2CCCOC2)C2CCCC2N1C(=O)C(C)(C)CF c1(CN(C(CCC2(C)CC2)=O)CCNC(C2CC2Cl)=O)cccc(Cl)c1 CC(CCC(=O)NCC(C1CCC1)NC(c1ccncc1C1CC1)=O)S(C)(=O)=O c1(CN(C(C(C)N(C(c2c(CC)con2)=O)CCO)=O)C)cccnc1O Cc1cc(C#N)sc1C(N1CCC(N(C)C(C2CCC(C)(C)OC2)=O)C1)=O N1(C(C(=C)F)=O)CCOCC1CC(N1CCOC(C(N)=O)C1)=O Cc1cccc(C=CC(N2CCC2CNC(=O)CN2CCC(CO)CC2)=O)c1 CCC(C)C(O)C(=O)NCCC1CCCN1C(=O)CC1CCN(C(=O)OC)CC1 C(=O)(C1CCCn2ccnc21)N1C(CNC(CC(CCC)C)=O)CCC1 c1(C(c2nnnn2C(C)C)NC(COC)COC)cnn(C)c1C(C)C N1(C(C(C)C2CCOC2)=O)CCCCCCC1c1ccccc1.C12CC(C1)C2 c1(C(=O)NC(CCNC(CC2CCCN(C(C)C)C2)=O)C)occ2c1CCOC2 CCC(C(C)(F)F)NC(=O)CC1CCCC1NC(c1cc(OC)nn1C)=O N1(C(C)=O)CCC(CC(=O)O)C(NCc2ccnc(SC3CCCC3)c2)C1 N#CCCCCC(=O)N1CC(NC(c2cccc(C3CC3)n2)=O)C1 c1(C(=O)NCC2(NC(c3ccc(O)cc3O)=O)COC2)n[nH]c2cccc(F)c12 C=CC1(CC(=O)NC2CCCC(NC(=O)Cc3ccc(C)cc3)C2)CCCCC1 C=C=C(C)CC(=O)NC(C)CN(C(=O)CCCc1ccc(Cl)cc1)C Cc1cc(S(=O)(=O)N(C2CCC(F)(F)C2)C(C)C)c(C)cc1-c1sccc1C C=CCCCCCC(=O)N(CC(O)CN(C)C(C1(F)CC2(CCC2)C1)=O)C c1(C(=O)OCC)ccc(NCc2n[nH]c(C)c2C)cc1O c1(C(N2CC(O)CC(NC(c3scnc3Cl)=O)C2)=O)ccc2ccsc2c1 c1(C(=O)NC2CCC(CNC(CCCS(N)(=O)=O)=O)C2)cnc2ccccc2c1 c1(-c2cn(C3CCC(C(N(C)CC4(OC)CCCC4)=O)C3)nn2)cnccc1Cl c1(CC)cnn(CNC(=O)C(C)(C)C2CCN(C(=O)CCOC3CCCC3)C2)c1 C12(CNC(C3=NOC(C)C3)=O)CCCC1N(C(=O)CC1(C)CC1)CCC2 c1(CC(=O)NCC(CN(C(c2cnn(CCC)c2C)=O)C)O)noc(C)c1C#N c1(C(=O)NC2C(C)CN2C(=O)CC(C)F)ccc(N(C)C)c(F)c1 C1(NC(c2ccc([N+](=O)[O-])s2)=O)CN(C(=O)CC(F)F)C2(CCOC2)C1 C1(N(C(C=Cc2occ(C(=O)OC)c2)=O)C)CCCN(C(=O)C(C)C(C)O)CC1 N1(c2[nH]c(=NCCn3c(C)nnc3)[nH]c(=N)n2)CC(C)(C)C12CCOCC2 C#Cc1ccc(C(=O)NCCCN(C(C2CC3(C2)CC3(F)F)=O)CC)nc1 N1(C(CCc2n(C)c(S)nn2)=O)CC2CCCCC2(CNC(=O)C(N)=O)C1 C1(NC(C(CCC)=CCC)=O)CN(C(c2cnn(C)c2)=O)C2(CCOCC2)C1 C1(c2cn(C3CCCC(C(C)(C)C)CC3)nn2)CCC2(CC1)OCCO2 c1(CN2C(C(N3CCC(N(CC)CC)CC3)=O)CCC2C)cc(C)c(F)c(F)c1 c1(CC(N2CCCC(CNC(C(CC)=CC)=O)C2)=O)ccc2cnccc2c1 N1(C(c2c(C)oc(Br)c2)=O)CC2CC(NC(c3ncncc3Cl)=O)CC2C1 C=C(CNC(=O)C(C)CNC(=O)CCCCC=CC)c1ccccc1 c1(C(N(CC(CNC(C(C)OCCC=C)=O)(C)C)C)=O)cccn(C)c1=O c1(C(N(C2CN(C(CNC(C(CC)C)=O)=O)C2)C)=O)cnc2c(c1)NC(=O)CS2 C(=O)(C1CC(C)Nc2ccccc21)NCCCNC(c1c(C(C)=O)cccc1)=O Cc1cc(=NC(=O)C(=O)NCCOC2CN(C(=O)C(C#N)N)C2)[nH]o1.C1(CO)CC1 C(=O)(CC(C)C(C)C)N(C(CN(C(c1c(C(=O)OC)nccn1)=O)C)C)C C1(CN=[N+]=[N-])COCCN1C(c1ccc(CNC(c2ccc(O)cn2)=O)cc1)=O c1(C(N2CC3C(NC(=O)CCCCc4cnn[nH]4)(C3)C2)=O)nc[nH]c2ncnc1-2 N1(C(Cc2ccc(C)s2)=O)CCC(NC(C2C3CNC(=O)C23)=O)C(O)C1 Cc1ccc(CC(N2C(C(=O)NCC3CC(n4cnnc4)C3)CC3CC23)=O)cc1O C(C(C)(C(=O)N1CCC(C(N)=O)C1)NC(=O)COCC1CC1)SC CC1CN(C(=O)NCCCC2CCOC2=O)c2ccc(Br)cc2O1 CC(CCC(=O)NC1CCCC(C(=O)Nc2cccc(C(C)F)c2)C1)N(C)C c1(OCC#C)ccc(C(=O)NCCN(C(C2CC2Cl)=O)CC)cc1CC c1(C(=O)NCCC(C)N(C(=O)C2=CCCOCC2)C)cc2sccc2n1C c1(OC)cc(C(=O)NC(C)C(CO)NC(c2ccc(=N)[nH]c2Cl)=O)ccc1Cl c1(CN2CC(NC(c3c(C(F)(F)F)cccc3Cl)=O)C(F)C2)c(O)cccc1O Cc1ccc(S(N)(=O)=O)cc1CN1CCCCC1C1CCNC1 C(C(CNC(c1cnc2n1CCOC2)=O)C(F)(F)C(=O)O)OC C(=O)(C1CN(C(=O)N(C)CC2COC2)Cc2n[nH]cc21)OC O=S(=O)(c1ccc(NCC2(CO)CCOCC2)c(F)c1)N1CCCC(F)CC1 C1(c2nnnn2C)(NCc2nnn(CC)n2)CCCN(C2CCCC2)C1 CC(C)CC(C)(CNC(=O)NC1COCC1CNC(=O)OC(C)(C)C)CC c1(NC)cc(C(N2CC(OC)CC(NC(=O)CC3CCOCC3)C2)=O)cc(Cl)n1 Cc1ccc(C(N2CC(N3CCN(C(C4(O)CCSCC4)=O)CC3)C2)=O)nc1C C(CCCCC(=O)N(C)CC1CCCN1C(C1CC2CC1CO2)=O)SC c1(C(C)SCCNC(=O)NCC(C#C)O)ccc2ccccc2c1 N1(C(C(C)C)=O)CCC(C)(C)C(CNC(=O)CC(C)c2cnn(C)c2)C1 C1(CNC(Cc2cnc(C)[nH]2)=O)CC2(CO1)CN(C(=O)Cn1ccnn1)C2 C1(CC(=O)NC(c2cn(Cc3ccc(Cl)cc3)nn2)CCC)CC2C=CC1C2 C(CC(C)CCNC(c1c[nH]cc1C(=O)Nc1ccccc1)=O)NC(C(C)C)=O Cc1cc(CNC(C2SCCS2)=O)oc1C(=O)N(CC(C)C)CCO C(=O)(CCCCCOC)N(C1CCN(C(=O)COCC)CC1)CC#C N1(C(C2N(CCC)CCCC2)=O)CC(NC(c2ccn(CC)n2)=O)C(C2CC2)C1 N1(C(C2(C)CCCC2)=O)CCCC(C(=O)NCCN2CCNC2=O)C1 c1(CCC(=O)NC(CCNC(C(CCSC)OC)=O)(C)C)ccc(F)cc1Cl c1(OC)cc(CN(C)C(C2CC2c2ccc(C(C)(C)C)cc2)=O)ccc1C c1(C(=O)NCC2(C)CCN(C(CCC#C)=O)C2)cc(S(N)(=O)=O)c(C)cc1C Cc1cc(C(=O)NC(C)(CNC(=O)CC2CC3C=CC2CC3)CO)cc(N)c1 N1(C(CSC)=O)CCCC2(CNC(C3CCC(C(N)=O)CC3)=O)CCCC12 C(C(=O)N=S(=O)(c1ccccc1F)C(F)(F)F)c1cccc(OC)c1 N1(C(=O)NCCc2cccc(Br)c2F)CCC2CS(=O)(=O)CC2C1 C(=O)(C1=CCCN(C(C2C3CCC(F)C23)=O)C1)NC(C)C(C)n1cncn1 c1(OC)nc(C(=O)NCC2(C)CCC(NC(c3cc(Br)no3)=O)C2)ncc1F CCC(CC(=O)NC1CON(CC)C1=O)NC(=O)Cc1ccccc1 C(=O)(C(C)(C)CC(C)(C)C)N1C2C(NC(c3cncc(OCC)c3)=O)C(C2)C1 c1(NC(c2c(C)nc(-c3ccco3)cc2)=O)ccc2cnn(C(F)F)c2c1 c1(CC(N2CCCC2CC(N2CCCC2C(F)(F)F)=O)=O)ccnc(F)c1 c1(CC(=O)N(C2CCCN(C(C(C)OCCC#C)=O)C2)C)ncc(F)cc1F c1(C(c2nnnn2C)(C)Nc2ccc3ncoc3c2)cccc2cncn12 N1(c2nc(C(C)C)nc(N3CCC(c4ccco4)CC3)c2)CC2CC(O)CC2C1 C1(C(N2CCCC(Cc3ccc(F)cc3)C2)=O)CCn2cnnc2C1 C12(OCC)CCC(C(N3CCCC(CN(C)C(c4nnsc4C)=O)C3)=O)(CC1)C2 N1(C(c2c(OC)cncc2)=O)CCC2CCCC12C(=O)NC(c1nnc(C)s1)C N1(C(COC(C)=O)=O)CCC2(CC1)CC2(CO)CNC(c1ccc2c(c1)CC2)=O C(=O)(C1CNc2ccccc21)N1CCC(NC(C2C(C)CC(C)O2)=O)C1(C)C CCCCCC(O)C(=O)N1CCN(C(c2ccn(CC)n2)=O)CC1CCCC c1(C(N2CCC(OC)(CNC(C3CCCC3O)=O)C2)=O)cc(F)ccc1F c1(C(=O)NCCCCCN(C(=O)C(F)C2CCOC2)C)nccc2ncccc12 C1(NC(C(=O)N(CCC(=O)OC)CCCO)=O)CC2CCCCCC2C1 c1(C(=O)NC(CC2CN(C(C(CC)CCOC)=O)C2)C)c(F)cc(Cl)cc1F C1(CC(=O)N(C)CCOCCNC(c2cc(C3CC3)on2)=O)CCC(=O)NC1=O C1(C(=O)NC2CC(NC(c3c(N(C)C)nccc3)=O)C2)C2CC3CC(C2)CC1C3 c1(C(N2CC(NC(C3CC34CC4)=O)CC23CCC3)=O)cncc2cc(Cl)ccc12 c1(C(=O)NCC(Cn2cc(COC)nn2)(F)F)cc2sc(C)cc2s1 c1(C(N2CC(CC(C)NC(c3cc(CN(C)C)on3)=O)C2)=O)nc(Cl)cs1 C1(NC(C=CC=CC)=O)CCC(F)(CNC(=O)CN2CCCCC2=O)C1 C=CC(C)(CC)NC(C1(F)CC(C(=O)O)C1)=O C(c1ccccc1)(C(F)(F)F)=CC(=O)NCC1CC(NC(C2CC2(F)Cl)=O)C1 C1(CNC(C(COC)C)=O)CC(NC(c2cc(N3CCCC3)ncn2)=O)C(O)C1 C#CCCCCC(=O)N1CCC(C(C)C(=O)NC2CC3CCC2C3)CC1 CC1CCN(C(c2cnc(Cl)n2C)=O)C1C(=O)N(CC(O)CO)C N1(C(=O)CCc2ccncc2)CC(F)CC1CNC(C12CCCCC1C2)=O C1(CC(=O)NCC(CNC(=O)CCCOCc2ccccc2)OC)C=CCCC1 CC1=CCN(c2ccccc2NC(=O)C(=O)NC(c2cn(C)nn2)C)CC1 C1(O)(CNC(CCN(CC#C)C(C2C[SH](CCC)C2)=O)=O)CCCC1 Cc1cc(C(=O)NCC2CCCN2C(=O)C(F)F)n(C2CCC2)n1 N1(C(=O)CN2CCOCC2)CC2CCC1CN2C(c1cc(Cl)ncc1Cl)=O C(=O)(CCCC(=O)NC1CCOC1C(=O)NCc1ncc[nH]1)N(C)C Cc1ncccc1C(N1CCC(C)C1C(=O)NC(CCO)C(C)C)=O c1(CNC(c2cnn[nH]2)=O)ccc(N2CCC(O)C2)cc1 c1(CC#N)ccc(C(N2CCN(CC3COC(c4ccccc4)C3)CC2)=O)cc1 N1(CC)C2CCC1CC(NC1(C(=O)Nc3sc(C)cc3Cl)CCC1)C2 c1(NC(Cc2c(C)occ2)=O)cccc(NC(=O)C(c2cccc(Br)c2)C)c1 C(=O)(CCC(CF)CF)NC1CCCC(C(N2CC(C)C(C(N)=O)C2)=O)CC1 N1(C(CC2(C)CCN2C(c2cc3ccccc3[nH]2)=O)=O)CCC12CCCSC2 S(CS(C)(=O)=O)CC(=O)N(CC(=O)N(C)C)CCOC c1(C(=O)NCCN(C(C(COCC)(C)C)=O)C2CC2)cnc2cc[nH]c2c1 C(c1ccc(C)nc1)=CC(=O)NC(CC=C)CNC(c1ccc(C2CC2)nc1)=O c1(N2C3C(NC(C=CCCC)=O)(CCC3)CC2)c(F)cc(C#N)cc1[N+](=O)[O-] Cc1nc(NCCSc2ccccc2)cc(=NCCN2CCCC2)[nH]1 C1(NC(C(c2cccc(C)c2)F)=O)CC2CC1N(C(c1[nH]nnc1C)=O)C2 Cc1cc(Cl)ccc1CC(=O)NCC1(CNC(C2CNC(=O)C2)=O)CC1 c1(NC(CC)(C)C)cc(C)c([N+](=O)[O-])cc1CNC(C1CCC(C(F)(F)F)O1)=O C(=O)(C1=CCC(F)(F)CC1)N1CCC(OC)(CNC(C2(C)CCCS2)=O)C1 n1(CC)nc(C)cc1C(=O)NC1(CC(=O)NC2CCCC2(C)CO)CCC1 c1(OC)cc(C(=O)NC23CC(C2)N(C(=O)CC(C)c2ccco2)C3)c(F)cc1N C=CCCCCCCCC(=O)NCC(CC=C)NC(=O)CC12CC(C1)C2 c1(C(N2CC(NC(C(CC)NC)=O)C(C)C2)=O)ccc(N2CCOCC2)c(Br)c1 N1(C(c2c3n(nc2)CC(C)CO3)=O)CCOC2(CCN(Cc3ccco3)CC2)C1 CCC(C)(CO)C(=O)NCC(C)CN(C)C(c1cnc(=N)[nH]c1)=O c1(C(N2CC=C(CNC(c3c(C)nsc3)=O)CC2)=O)cccc2cc[nH]c12 C1(C(=O)NCc2cc(C)c(F)cc2)CCN(C(=O)C(O)CCC(C)C)C(C)(C)C1 C1(CC)CN(C(c2cnc(CC(C)C)s2)=O)CCN1C(c1cncn(C)c1=O)=O C#Cc1ccc(C(=O)NC(C2CCCN2C(C23CCC(C)(C2)OC3)=O)C)cc1 N1(C(C(C)OCCOC)=O)C2CC1CN(C(c1ccc(O)cc1OC)=O)C2 c1(COC)ccc(C=CC(=O)NC2(NC(=O)C(C3CCCCC3)OC)CC2)cc1 Cc1cc(C(=O)NCCc2n[nH]cc2C(=O)NC2(C)CC2C)no1 CCCC(CCCNC(C1CCc2cc(Br)ccc2C1)=O)N=c1nc(CC)[nH]s1 c1(C(N2CCC(c3cccc(Cl)c3)C2)=O)cc2cccc(O)c2[nH]1 C(C(CC(F)(F)F)NC(=O)C(C1CCCCC1)F)NC(c1cncc(O)c1)=O CCCCCCC(=O)N1CCCCC(N(C)C(c2cnc(OCC)cn2)=O)C1 N1(C(c2c(C)nco2)=O)CCN(C(C2CCC(=O)N2C)=O)C(CC(F)(F)F)C1 c1(C(=O)NCC2(C)CCCN(C(C3(C)C=CCC3)=O)C2)ccc2c(c1)CCOC2 C1(C(N(C)Cc2cccc(CNC(C3CC(F)C3)=O)c2)=O)CC2C(C1)C2(F)F CC1CCCCC1(CNC(C1CC2(C1)CC(O)C2)=O)NC(=O)COC(F)(F)F C(=O)(CS(=O)(=O)C(C)C)N1CC(CC)C(NC(=O)C=Cc2ccccn2)C1 C1(C)(CCNC(C(COC)N(C)C)=O)CCN(C(c2c[nH]nc2F)=O)C1 C(=O)(C1CCc2nccn21)NC(C(=O)NC(c1ccc(C)cc1)C)c1cccs1 c12n[nH]c3c1CN(CC3)C2.C1(C)(NC(CSC(C)(C)C)=O)COC(C)(C)OC1 C1(NC(c2cn(CC=C)nn2)=O)(CC)CCN(C(=O)C(C)NC(C)(C)C)CC1 C(=O)(C1=CC(O)C(NC(C2(CCOC)CC2)=O)C1)N1CC(O)(CC=C)C1 c1(SC)ccc(Cl)c(C(N2CCC(CNC(=O)C(CO)NC(=O)C(C)C)C2)=O)c1 N1(C(CCOCC(C)C)=O)CC2CC1C2NC(C1CC(CC(C)(C)C)C1)=O Cc1cc(NC(=O)CC2C3CN(C(c4c[nH]c(=N)c(C)c4)=O)CC23)c(C)cc1F c1(C(N(C(C)C)C)=O)ccc2c(c1)C1CN(C(=O)C(C)(C)F)CC1NC2=O C1(NC(c2c(OCC)cccc2)=O)CN(C(=O)C=C(CC)CC)CCC1CO C1(C(=O)NCC2(COC)CN(C(=O)C=CC3CCCO3)C2)CC(=O)NC(=O)N1 CN1CCC(NCCC2COCCN2)CC1c1ccc(Br)cc1 C1(CN(CCNC(c2csc(C(C)(C)C)n2)C)CC)CC2CCC1C2 N1(C(=O)NCc2nccc(OC)c2)CC2CCCCN2CC1C c1(NC)cnc(C(=O)NCC(O)CN(C(=O)C=Cc2ccc(C(N)=O)o2)C)cn1 C(=O)(C1=COCCO1)N1CC(CNC(c2c(C)nc(CCCC)s2)=O)C(O)C1 Cc1n[nH]c(C)c1CC(N1CC(NC(c2cc(Br)ccn2)=O)C(O)C1)=O O(NC(=O)C(CNC(c1scnc1C)=O)N(C)C)C(COCC)C c1(OC)cc(Cl)c(Cl)cc1C(=O)N(C(C)CCNC(C1CCCC(=O)O1)=O)C N1(C(C2N(C(C3CC(=O)C3)=O)CCC2)=O)CCCC2(CCNC2=O)C1 c1(C(N2CC3C(CNC(c4ncn(C)n4)=O)(C3)C2)=O)cc2cccc(F)c2o1 N1(C(C2C(C)C2)=O)CC2(CC(NC(c3cc(-c4cn(C)nn4)on3)=O)CO2)C1 c1(C(N(C)CCNC(=O)C=Cc2ccccn2)=O)ccc(Cl)c2c1OCCO2 c1(C(=O)NC2CCN(C(Cc3c(C)n[nH]c3)=O)CC2C)cc2c(nn1)CCC2 CCCC(C)CC(=O)N1CC2(CC2)CC1CNC(=O)CCn1ccnc1 c1(C(=O)Nc2ccc(C)nc2I)cc(-c2ccccc2F)cc2cc[nH]c12 N1(C(C2(C(C)C)CC2)=O)CCCC(N(C)C(c2cnn(C)c2Br)=O)C1 C1(CNC(CCCCNC(C)=O)=O)CN(C(c2cnc(NC)cn2)=O)CC1(C)C c1(-c2cc(N(C3CCOCC3)CC(COC)C)no2)ccc(F)cc1F N1(C(CCCOCC)=O)CCC2(C1)CN(C(c1nccc3occc13)=O)C2 C1(CNC(c2c(C)cc(F)s2)=O)CC(NC(=O)Cc2cc[nH]n2)C12CCC2 c1(C(=O)NC2C(NC(C(CC)N(C)C)=O)CCCC2)ccc(OC)cc1C CC1(C)C(NC(c2cc(Cl)no2)=O)CC1CNC(c1ccccc1SCCO)=O N1(C(c2ccc(C)cc2O)=O)CCC2CCC(NC(=O)CCC3CCCO3)C1C2 Cc1nc2ccnn2c(C)c1C(=O)NCC(Cc1ccccc1)CO C1(c2n(CCCOC)nnn2)(NCC(c2ccc(F)c(F)c2)C)CCCN(C)C1 C1(NC(c2c(C)nc(C(C)C)s2)=O)CC(F)CN(C(=O)CCN2CCCC2=O)C1 C(CCCCC(=O)N1CC(OCCC(N2CCOC(C3CCC3)C2)=O)C1)OCC c1(C(=O)NCCN(C(=O)CCc2cccc(Cl)c2)CCC)cc(C)cnc1F N1(C(c2ccc(F)c(C(F)(F)F)c2)=O)CCC(C2CCN(C(C3CCC3)=O)C2)C1 C1(CC(=O)NCCOCCNC(Cc2cn(CC)nn2)=O)CCCC(=O)C1 C1(C(=O)NC(C(=O)OC)C(C)C)CC(C)CN(C(C2CS(=O)(=O)C2)=O)C1 c1(C(C(=O)NCc2nnn(C)n2)N(CCOCC=C)C)ccc2c(n1)OCCO2 C12(NC(c3[nH]cc(CC(C)C)c3)=O)CCCC1N(CCc1ccc(Cl)cc1)CC2 N1(C(CCC)=O)CCCC(N(C(=O)C(F)=CC2CC2)CC2(COC)CC2)C1 C1(NC(C2C(OC)CCC2)=O)C2CCCC1N(C(=O)CC(C)(C)NC(C)=O)C2 C1(CNC(=O)NC2CCC(N3CCCC3)CC2)CCCC2C1C2(F)F CC1(C)CCC(C(=O)NC2CCSCC2)(NC(=O)Cc2cc(C3CC3)no2)C1 CC1Cc2c[nH]nc2CC1NC(=O)COC(c1ccc(C(N)=O)cc1[N+](=O)[O-])=O C1(C)(CNC(c2ccnc(C)n2)=O)CCCN(C(=O)CCC2CCCCN2C)C1 N1(C(C(COC)(C)C)=O)CCC2CN(C(=O)Cc3cn[nH]c3)CC2C1 c1(N(CC(CN(C(=O)CN(C2CCSC2)C)C)O)C)nnc(C(F)F)s1 CC1(C)CN(C(C23CCC(CN(C(c4ccns4)=O)C2)C3)=O)CCCO1 CCC(CC(=O)N1CC2(CCN(C(C3CCC3(C)C)=O)C2)C1)C(F)F N1(C(C=C(C)C(C)(C)C)=O)CCC2C(NC(c3ccc(N(C)C)nc3)=O)CC12 C1(OC)CC(C(=O)NCC2(CNC(=O)C(F)C3CCCC3)CCC2)C1 N1(C(c2cnc(CC)nc2O)=O)C2CCCC1CN(C(C1CCCOC1)=O)C2 c1(C(N2CCC(CCCCNC(CCCOCC)=O)CC2)=O)cc(O)nc(O)n1 c1(CC(=O)NC2CN(C(CN(C3CC3)CC)=O)CC(O)C2)n[nH]c2c1CCCC2 O(NC(=O)CCOC(C)C)CC(=O)NCC(F)OC C1(C(=O)NCCC2CCN(C)CC2)(NC(C(CC)=CC)=O)CCCC1C N1(C(C2CCC(C)O2)=O)CCCC2(C1)CN(C(=O)CCN1CCOC1=O)C2 C1(CC)(NC(=O)CC2CCOCC2(C)C)CCCN(C(=O)Cc2c[nH]nc2O)C1 C=CC(C)(C)CCNC(=O)CC1CC(C)N(C(c2cnc(Cl)s2)=O)C1 C1(NC(c2cc(C)nc(Cl)c2)=O)CCN(C(C2CCSCC2)=O)C12CCCC2 C#Cc1ccc(OC)c(C(N2CCC(C)C(NC(=O)Cn3ccc(C)n3)C2)=O)c1 CC(C)CCCCCC(=O)N1CCC1C(=O)NCc1conc1C(C)C C#CCCC(O)C(=O)N1CCCCC1CN(C)C(c1c(C)nn(CC)c1C)=O c1(C(N2CCC(C3N(C(c4c(C)cncc4)=O)CCC3)C2)=O)ccc(Br)cc1F C1(C(N(CCCNC(CCCCCC)=O)CC)=O)CCc2c[nH]nc2C1 c1(NC(=O)NC(CC)COCC(=O)N(C)C)ncc(C)s1 N1(C(C(CC(C)C)C)=O)CC(C(=O)N(C2CCOCC2)C2CC2)C2(CCC2)C1 N1(CC(=C)Cl)CC2(CN(C(c3cc(OC)n(C)n3)=O)CCO2)C1 C1(N(CC(=O)NCC(C)C)CCN(C)C)CCN(c2ccccc2Cl)C1=O C1(C(=O)NC2(CC=C)CCN(C(=O)CNS(=O)(=O)N(C)C)C2)COC(C)(C)CO1 c1(CC)ccc(C(N2C3CCC2CN(C(=O)C(C)NC(N)=O)C3)=O)cc1C#N N1(C(c2nc(CC)sc2)=O)CCC(C)(C)C1CC(=O)NCC1=NOC(C)C1 CC1(CNC(=O)COCCN(C)C)CCCN1C(=O)Cn1nccn1 c1(C(N2CCN(S(Cc3nc(C)sc3)(=O)=O)CC2)=O)ccc(OC(C)C)c(Br)c1 Cc1nc(C(=O)NCC2(C)CCN(C(c3ccn(C)c(=O)c3)=O)C2)cc(O)n1 c1(N2CCCC(NC(C(CCSC)O)=O)C2C)cc(C#N)nc(C)n1 N1(C(CC2CCN(Cc3ncc(C)cc3F)CC2)=O)CCc2cc(F)ccc2C1 C1(CNC(c2cnn(C(C)C)n2)=O)CCC(NC(=O)CCCC2CCCO2)CC1 N1(C(c2c(C)coc2C)=O)CCC(NC(=O)CCOCC(C)C)C(O)C1 CC1CN(C(=O)C=Cc2cc[nH]n2)CCC1NC(=O)C(c1ccccc1)C c1(N(C(C(=O)NC(C)CNC(=O)CC2CC2C2CC2)C)C)nccn2cnnc12 C1(C(C(=O)NCCCNC(=O)CCC2CCOC2)OC)CCCCC1 N1(C(c2cc(F)cc(F)c2)=O)CC2CCCCC2(CNC(C2CC(O)C2)=O)C1 c1(-c2cc(C)c(=N)[nH]c2)cccc2c(C(=O)NCc3noc(C(C)C)n3)[nH]nc12 N1(C(CC2CCN(C)CC2)=O)CCN(C(=O)Cc2c(O)ncnc2O)C(CF)C1 c1(C(C=O)N(C2CCC(F)(F)CC2)CCCC(C)O)nc(F)ccc1F.CO c1(C(N2C3C(NC(=O)C(F)CC4CCOC4)C(C3)C2)=O)ccnc2[nH]ncc12 Cc1nn(C)c(S(=O)(=O)NC(c2ccccc2)(C)Cc2ccccc2)c1C(F)F Cc1cc(OCC(=O)NC2C=CC(CNC(C3C=CCCC3)=O)C2)ccc1Cl c1(C(C)=O)ncc(CCC(=O)NCCN(c2ccccc2)C(=O)CSS(C)(=O)=O)o1 c1(C(=O)NCCC2OCCN(C(C(CCC)O)=O)C2)ccc2c(c1)OCC(=O)N2 C1(C#N)(C(=O)NC(C2CC2NC(c2cc(F)ccc2F)=O)C)CC12CCCC2 CC(CC(=O)NC(C)C(C)OCCCN(CC(N)=O)C)n1cccn1 c1(OC(c2ccc(C(N3CCSC(C(=O)C)C3)=O)cc2)=O)cc(Cl)cc(Br)n1 N1(C(=O)CCC2CC2)CC(C(N2CCOCC2)=O)C2CC12.C12(CCCC1)C(=O)N2 c1(CN2CCCC(O)(c3onc(CC)n3)C2)ccc(OC)c(S(N)(=O)=O)c1 C1(NC(C(CC)(C)CO)=O)CN(C(c2ccc(F)c(Cl)c2)=O)C2(CCOCC2)C1 O=S(=O)(c1ccc(Nc2ccnc3ncnn23)cc1)NCc1cccc(F)c1 C1(CN(C)C(C2(C)CC2(F)F)=O)CCCN(C(=O)C=CI)C1 Cc1cc(C#N)sc1C(=O)NC1CCCCC1NC(C1CC12CCCC2)=O c1(NCCN(C(CC)C)C)nccc(=NCCCCCNC(C)=O)[nH]1 C(=O)(CC(C)CC(C)C)NC(C(=O)NCc1nnc(CC)o1)CN(C)C c1(C(N2CCN(C(c3cnc(=N)[nH]c3)=O)C3C2CC3)=O)cc(F)cc2nc[nH]c12 c1(OC)cccc2c1OCCC2NCc1cc(S(=O)(=O)N(C)C)ccc1Cl c1(C(C)NC(C2(N(C(=O)CC3CCOC3)C)CC2)=O)cncnc1 c1(OC)ccc2c(C)c(C(=O)NCC3CCC(NC(=O)CC(C)F)C3)[nH]c2c1 c1(C2(OC)COC2)cccc(C(=O)N(C)CCNC(=O)CC2CC3COCC23)c1 Cc1cccc(C)c1C(=O)NC(C)Cn1cc(-c2cc(F)cc(Cl)c2)nn1 C=C(C)CC(Cc1ccccc1)NCC1(CC)CNC(=O)N1 N1(C(C2N(C(=O)OCC)CC2)=O)C(C)CC2CN(C(=O)C(O)COC(C)=O)CC12 C(c1cocn1)=CC(=O)NCC(COC)NC(=O)C(C)C#N C(CCCCN=[N+]=[N-])NC(C1(CO)CCN(C(CC(C)CN(C)C)=O)C1)=O C1(O)(CNC(C2C(C)(C)CO2)=O)CCCN(C(=O)CSc2n[nH]c(O)n2)C1 c1(C(=O)NC(C2CCN(C(C3CCOCC3)=O)C2)C)cc2cccnc2[nH]1 S1(=O)(=O)c2ccc(c(Br)c2)NCC(C(C)(C)C)N1.N1(CCOC)CCCOCC1 c1(C(=O)NC2(CCC)CC2)coc(CNC(=O)CC(C2CC2)C2CC2)c1 C1(C(=O)NCC(n2ccnc2)C)COCCN(C(=O)CC2CCC(=O)NC2)C1 CCCC(C)(C)CC(=O)N1CCC(CNC(C2CC3CC3C2)=O)(OC)C1 Cc1cc(C)c(C(=O)NCCCCCN(C)C(C2CN3CCC2C3)=O)cn1 c1(CC)ccc(C(=O)NCC2CCC(NC(=O)CNC(=O)CC(C)(C)C)C2)cc1 C1(CNC(c2n(CC)ncn2)=O)C2CN(C(=O)C(Cc3ccccc3)CC)CC12 N1(C(C2(F)CN(C(c3nccc(CC)c3)=O)C2)=O)CC(C#N)C2(CCC2)C1 Cc1nc(C2CC2)ncc1C(=O)NC(C)CNC(c1cnn(C(C)(C)C)c1)=O C1(C(=O)OC)CCCC(C(=O)NCC2CC(NC(c3ncccc3NC)=O)C2)C1 C1(C(=O)NC2CC2)CCN(N2CCC(CO)(CO)CC2)CC1 N1(C(C2CC(C)(O)C2)=O)CCC2(NC(=O)Cn3nnc(C4CC4)n3)CCCCCC12 N1(C(Cc2c(C)non2)=O)CC2(CCN(C(=O)CC3CCS(=O)(=O)C3)C2)C1 c1(C(N(CC(O)CNC(C2CCCC23CC3)=O)C)=O)cc2nccc(Cl)c2s1 c1(C(=O)NCC(CNC(C2(C)N(C(C)=O)CCC2)=O)(C)O)ccc2nnnn2c1 C1(NC(C2CC(N3CC(F)C3)C2)=O)CCN(Cc2cnn(-c3ccccc3)c2)C1 C1(CNC(C2N(S(CCCC)(=O)=O)CCC2)=O)CCCS(=O)(=O)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1C(CN(C(C2C=C(C)CS2)=O)C)COCC1 c1(C(=O)N(CCNC(C23CCC2C3)=O)CC2CC2)cccc(C2CC2(F)F)c1 c1(OC)cc(F)cc(S(=O)(=O)NCC2C=CCCCC2)c1 C1(=O)C(C(C)(C)C)n2cc(nn2)CN1.CC1(CC2CC=CCN2)CNC(=O)O1 c1(C(=O)NC2(CC=C)CN(C(c3cc(C)co3)=O)C2)cccnc1S C1(NC(COc2cc(C)on2)=O)CC2CCC1(NC(c1cc(F)cc(Cl)c1)=O)C2 C(=O)(CS(=O)(=O)CC(=O)NC1CN(CC)C(O)NC1c1noc(C)n1)OCC N1(C(C(CC)OC)=O)CCC(F)CC1C(=O)NC(C)(C)COC(C)C c1(CC)ccc(C(=O)NC2CC23CC(NC(=O)C(C)(C)CN(C)C)C3)nc1 C1(c2nnnn2CC2CCCO2)(Nc2cc(CC)nn2C)CC2(COC(C)C2)C1 N1(C(C2CCC(C)(C)CC2)=O)Cc2nccn2CC(NC(=O)C=C2CCCC2)C1 c1(C(=O)NC(C(=O)NCC2(CC)CCCO2)c2ccoc2)cc2n(n1)CCO2 CCC(C)(C(=O)NC1CN(C(=O)Cc2ccnc(Br)c2)C1)OC c1(C(=O)NC2CCC(CNC(c3cc(C)n(C)n3)=O)C2)ccc2ocnc2c1 C1(OC)CC(NC(=O)CN2CCCS2(=O)=O)C12CCN(C(c1cn[nH]c1)=O)CC2 c1(OC)ccc(F)c(CN2CCN(C(c3ccccn3)C)CC2)c1OC N1(C(CCCOCC)=O)CC(NC(C2CC2c2ccc(Cl)cc2)=O)C(O)C1 N1(C(c2c(N)ccc(C)c2)=O)CCC2CC(NC(C3CC34CC4)=O)CCC2C1 C1(CC)CCCCC1C(=O)NC(c1ccnn1C)C(=O)N(C)CCOCCO c1(C(=O)NCC(CNC(C2CNC(=O)N2)=O)OC)ccc(Cl)c(F)c1 C1(O)(CCNC(C2CC(OCC)C2)=O)CCN(C(C2OCCC2C)=O)CC1 C1(C(=O)NCC23CC(NC(C4CC(=O)N4)=O)(C2)C3)C2C3CCC(C3)C12 N1(C(CN(C2CCSC2)C)=O)CCC(CO)(CNC(=O)C(C)(Cl)Cl)CC1 N1(C(c2c(CC)cc(F)cc2)=O)CC(NC(=O)C(C)(C)C)CC(C)(C)C1 N1(C(c2c(C)nccn2)=O)CC(C)(C)OCC1CNC(C1CSCCS1)=O c1(OC)ccnc(C(=O)NCC2CCCC2NC(C2(C)CCCO2)=O)c1 C1(N(C(C2(C)CNC(=O)N2)=O)CC)CCCN(C(=O)CCOC(C)C)CC1 C1(CC)(CC)CC(C(=O)NCCC2CC(NC(=O)C(C)C3CCC3)C2)C1 c1(SC)ccc(C2CC2C(=O)NCCC2CCCCCC2)cn1 N1(C(CN2CCC(C)C2)=O)CCN(C(CNC(C2(CCO)CC2)=O)C(F)F)CC1 C1(C)(C(N(CCC#C)C)=O)CCN(C(=O)C=CC2(C)COC2)C1 C1(C(N(CC(N2CC(N(CCC)CC)C2)=O)C(C)C)=O)CC2CCCC2C1 c1(C(=O)NCC(C)N(C(c2cnc(COC)s2)=O)C)c(C)csc1Cl C=CCCCCC(=O)NCCC1(NC(=O)CC2(O)CCOC2)CCC1 CC1CN(C(c2ncc(Br)cn2)=O)CCCN1C(c1cnc(O)s1)=O C1(N(c2ccc(C(=O)OCC)s2)C(c2ccc(Cl)o2)=O)CCNCCC1C C(=O)(CCCC(C)(F)F)NC(CNC(C(COC)C)=O)C1CCC1 C1(CC(=O)NCC(NOCC)=O)CN(C(c2cc(C)[nH]n2)=O)C(C)(C)C1 c1(OC)ccc2c(C(=O)N(C3CCN(C(C4(C)CC4(F)Cl)=O)CC3)C)n[nH]c2c1 C1(NC(CCCCC#C)=O)CCCC12CCN(C(c1cnc(CC)s1)=O)CC2 C=C(Cl)CC(C(=O)NCC1C(C)C1C)NC(=O)CNC(=O)NC C1(CC)CC(CC(N2CCC2CNC(c2cscn2)=O)=O)CCO1 C1(CC)CN(C(=O)C(=O)NCCCn2ccc(C(F)(F)F)n2)C(CC2CC2)CO1 c1(-n2cc(CN3CC(COCCOC)CC3(C)C)nn2)ccc(S(N)(=O)=O)cc1Cl c1(C(=O)NCC(C)N(C(C(CC)NC(C)=O)=O)CC)cc(F)c(F)cc1O N1(C(C=CC(=O)OCC)=O)CCCC(NC(C2(CO)CCC2)=O)C1C C1(CC)CCCC(NC(C2(CC)CN(C(c3n[nH]cc3CC)=O)C2)=O)CC1 C1(NC(CCN(C)CC)=O)CCC(O)CN(C(C2(C)CCN(C)C2)=O)C1 C1(CNC(=NCC)NCC(=O)NC2CCCCC2)CCC2(CCCCC2)O1 Cc1sc(C(=O)NCCCC(C)NC(=O)C2=COCCC2)cc1S(N)(=O)=O C(=O)(C(=O)CC(C)C)NCC1(C(=O)NCC2C3COCC23)CC(=C)C1 c1(OC)ccc2nc(C(=O)NCC3CC(OC)CN3C(c3cnco3)=O)cn2n1 C1(NC(C2(C)CCSCC2)=O)CN(C(=O)Cc2cn[nH]c2)CC2(CCOCC2)C1 c1(OC)cc(NC(c2cn(C(C)C)cn2)=O)ccc1-n1cccc1 C1(C(N2CC(CC(C)NC(c3c(C)nns3)=O)C2)=O)CCc2nnnn2CC1 C1(CC)CCC(C(=O)NCC2C=CC(NC(=O)CSc3ccccn3)C2)O1 C1(NC(CC2(C=C)CCCCC2)=O)CC1C1CCN(C(C2(O)CCSC2)=O)CC1 C1(NC(c2nn(C(CC)C)c(C)c2)=O)(CO)CCCN(C(=O)C(C)(CC)CC)C1 N1(C(CCCCOC)=O)CC2CCC1C(NC(c1ncccc1Cl)=O)C2 c1(OC)ccc2[nH]c3c(c2c1)CCCC3C(=O)N1CCc2cccc(OC)c2C1 C1(CNC(C2CC3CCC2O3)=O)CN(C(c2c[nH]nc2C2CCC2)=O)CCCO1 N1(C(c2ccc(CC)c(N)c2)=O)CCCC2CN(C(=O)C(C)N3CCC3)CC12 C1(C(=O)NCC(C#C)OC)C2CC2CN1C(=O)CCc1ccccc1 c1(C(=O)NCCCC(C)NC(C2C(F)(C(=O)OC)C2)=O)cc(C(F)(F)F)cn1C c1(CC(=O)NC(CCCCNC(c2ccc(OC)s2)=O)C)cccc(F)c1Cl N(C(=NCCCC1CCOC1)N1CCC(N2CCC2)C1)CC(c1ccccc1)F C(c1ccncc1)=CC(=O)NCC1(F)CC(NC(c2ccoc2C(F)(F)F)=O)C1 C1(NC(c2[nH]c(=NC)sc2)=O)CC2CC(NC(=O)C(F)C(C)C)CC2C1 c1(C(=O)NC2CCC(CNC(CCC)=O)CC2)cc2scnc2[nH]1 c1(CC(=O)NC2CC(O)CN(C(c3ccccc3F)=O)C2)ccc(Cl)c(Cl)c1 Cc1ncc(CCC(=O)NC(CNC(c2ccsc2Cl)=O)C2CCC2)s1 CC1(C)CN(CC(=O)NCC(=O)NC2(CCCN3CCCC3)CCC2)C1 C(C(C)C(C)(C)C)N(C(C(CC)N(C)C(c1ccc(COC)o1)=O)=O)C c1(C(=O)NC(C(C)NC(c2cn(CCC)nc2)=O)C)ccc(OC(C)C)cc1 N1(CC)CCN(CC(=O)NCC2(OC)CN(C(=O)C=C(Cl)Cl)C2)C(=O)C1=O N1(C(C2(CSC)CC2)=O)CCC(C2CCN(C(c3c(C)ncn3C)=O)CC2)CC1 c1(C(=O)NCCCNC(C(c2ccc(Cl)cc2)OC)=O)cccc(Cl)c1N CC1CC=C(C(=O)NCC(=O)N(CC(C)C(F)(F)F)C)CC1 C1(CNC(c2cccc(SCC)c2)=O)CC2CCCC2N1C(C1CC(CC)=NO1)=O C#CC1(C(N2CC3CCCC2C3)=O)CCN(C(C2CN3CCC2C3)=O)CC1 C(=O)(CCC(=O)N(CCCCCCNC(=O)C(F)(F)C1CCCCC1)C)NC C1(NC(CCc2cnc(C)o2)=O)CN(C(C2(C#N)CC2)=O)Cc2nccn2C1 c1(C(=O)OC)ccnnc1NCCNC(CNC(C1(C(F)(F)F)CCC1)=O)=O C12CN(C3CC13)C2=O.C1(NC(C=C(C)C)=O)CCC(NC(=O)OC(C)(C)C)CC1 C(=O)(C#CC1(CC)COC1)NC(CC)CN(C(=O)Cc1nncn1C)CC C(=O)(C(C)S(N)(=O)=O)NC(c1cn(C)nn1)C(=O)NCC(NOC)=O C1(CNC(c2c(C)cn(C)n2)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)C12CC2 C12(CNC(c3n(CCC)ccc3)=O)CC1CN(C(=O)Cc1cc(COC)on1)C2 CC1C(=O)CC1C(=O)N(C)CC1CCN(C(=O)CCOC2CCCC2)C1 O=C(CCS(=O)(=O)C(F)(F)F)NC1CCC(CCNC(=O)Cn2cccn2)C1 c1(C(=O)NCCN(CCOC)C(c2cnn[nH]2)=O)ccc(Cl)cn1 C(C(CNC(C1(C)CCCCO1)=O)C(F)(F)F)NC(CC(=O)OCCC(C)C)=O C12(CNC(c3cc(C)no3)=O)CCCC1N(C(=O)CN1CC3C=CC1C3)CCC2 c1(C(=O)NCC2CC(C)N(C(c3cnn(C)c3Cl)=O)C2)n[nH]c2ccc(Cl)cc12 C1(C(=O)NC(C2CCCO2)(C)C)CC2CCCC2N1C(=O)CC1NC(=O)NC1=O Cc1sc(C(=O)NC2CC(NC(=O)C(C)Cn3ccnc3)CC2O)nc1O C1(C(=O)NC2C(CNC(C3(F)CC3)=O)CC2)CCC2(CCCC2)CC1 c1(C(=O)NC(CNC(c2nc(C)sc2)=O)C(C)C(C)C)cc(Cl)cc2c1CCC2 O=C1CNc2ncc(C(=O)Nc3csnc3OC(F)F)cc2N1 C1(NC(CC2C(CNC(C3CC(C)(C)C3)=O)C2)=O)CCC2CCCC1O2 c1(C(=O)NCC2(NC(=O)CCN3CCCCC3)CCC2)ccnc2nccnc12 N1(C(C(c2c(C)cc(F)cc2)O)=O)C2CCC1CN(C(c1cccc(=O)o1)=O)C2 C=CCC(C(=O)NC(C1CCCN1C(c1cnc(O)n1C)=O)(C)C)C(C)C C(CCCC(=O)N1CC(F)(F)CC1C(=O)NCCc1cn(C)nn1)(OC)OC C1(C(=O)OC)CC2(CCC(CNC3CCCC3N3CCCC3)O2)C1 C=CC(C)CCNC(=O)C(C)N(C(=O)CC1(CC)CCC1)C1CC1 CC1CN(C(c2cc(F)ccc2O)=O)CCN1C(=O)CC1CC=CC1 C1(CNC(C=CC=CCC)=O)C2CN(C(c3cnn(C)c3C)=O)CC12 n1(C(C)C)cc(-c2cn(C(C)CNC(C3CCC3C#N)=O)nn2)cn1 c1(C(N2C(C(=O)Nc3c(OC)ccc(C)n3)CC(O)C2)=O)ccc(Br)c(F)c1F N1(C(CC2CCN(C(c3c(C#C)c[nH]n3)=O)C2)=O)CCC(C)C(O)C1 Cc1nc(N2CC(C(C)NC(=O)CCC3CCC(C)O3)C2)cc(C#N)n1 CC(CO)OCC=C.C1(=O)C=CC(=O)NCCN1C.C(C)(C)(C)OCC1CC1 c1(CNC(C(=O)NC(c2nnnn2C)C)=O)cn(C2CCC2)nn1 C1(NC(=O)C2=CCCC2)CN(C(c2ccn3ccnc3c2)=O)CC1C1CC1 O=C1CC(c2cn(CC(c3ccc(Cl)cc3O)N3CCOCC3)nn2)NC(=O)N1 C1(NC(Cc2c(C)noc2C)=O)CC(O)CN(C(c2ccnc(N(C)C)c2)=O)C1 C(CCCC(=O)NCCCN(C(=O)C=C1CCOCC1)CCO)OCCC=C C(CCC(c1ccccc1)NCCCOC(F)F)NC(=O)NC1CCCC1 Nc1cc(C(=O)NC2CC(NC(C3COC4(CCC4)C3)=O)C2)c(Cl)c(F)c1F N1(C(c2cc(C)ncn2)=O)CC(C2CCCN(C(=O)CCC3CCC(=O)N3)C2)C1 N1(C(CC(=O)N(C)C)=O)CCCN(C(c2cccc3c2CCO3)=O)C(CO)C1 CC(C)CC(F)C(=O)N(C1CCN(C(C2CCCC2)=O)CC1)C C1(C(N2CCN(C(c3c(OC)ccnc3)=O)CC2CO)=O)CCc2cncn2C1 c1(-c2cn(CCN(C(c3cc(CC)sc3)=O)C)nn2)c(C)nsc1N c1(C(N2CCC3(C(C(=O)Nc4c(Cl)ccnc4Br)C3)C2)=O)cc(Br)c(O)cc1O c1(OC)cnc(C(=O)NCC2CCN2C(=O)CSc2ccccc2O)c(F)c1 C1(NC(C(C)SCC)=O)CC2(C1)CC2NC(c1coc(C(F)F)n1)=O C1(C(=O)NC2C(NC(c3nc(COC)oc3)=O)CCC2)CC(O)CN1C C1(O)(C(C)NC(CSCCCC)=O)CN(C(C2CCCC2c2ccccc2)=O)C1 c1(C(=O)NC(C(=O)NC(C(=O)OCC)C)CC2CC2)nccnc1C C1(CC)C(NC(C)=O)CCN1C(C1(COC)CCCO1)=O N1(C(c2ncc(C)c(Br)c2)=O)CCOC2(CCCN(C(=O)CCCCBr)C2)C1 C1(CC)CN(C(=O)CCOCC(F)(F)C(F)F)CCC1N(CC)CC c1(OCC)ccccc1C(=O)NC(c1cn[nH]c1)C.C12(CC1)C(=O)N2 C1(CC)CN(C(=O)C(F)(F)CO)CCC1CNC(C1CC1C1CCCO1)=O C1(CNC(C2CN(S(CC)(=O)=O)C2)=O)CN(C(=O)CCCSC)CCCO1 C(=O)(C(C)(C)C)CNC(=O)OC(C)(C)C.C1C(=O)NC2CC2C(=O)N1CCC N1(S(CC(C)C)(=O)=O)CC2CC1CN2Cc1c(Cl)cncc1Cl C(=O)(C1=CCS(=O)(=O)C1)NC1(C2CN(C(c3cc(C)ns3)=O)C2)CC1 C1(C)(C(=O)NC2CC(CNC(C3CCN(C)CC3)=O)CC2O)CCCCC1(F)F N1(C(C(c2ccc(C)o2)C)=O)CCOCC(CNC(c2ncoc2C)=O)C1 N1(C(C2(OC)CCCC2)=O)CCC2(CC1)CN(C(C1CC1C)=O)C2C(C)C CC1(C)CCCC(O)(C(=O)NCC2CCC(NC(C3(CO)CCCC3)=O)CC2)C1 C1(N2CCC(NC(C3(N(C)C)CCC3)=O)C2)CCN(C(=O)CSC(F)F)CC1 C1(CC)C(NC(=O)CC(O)CN(C)C)CCCN1C(C1CCOCO1)=O C1(NC(CC2CCN(C(CCCCCC)=O)C2)=O)C2CCC(C2)C1(C)C c1(CC(=O)NC2CC(CNC(C34CC(OC)C3C4)=O)C2)c[nH]c2cccc(Cl)c12 Cc1c(CN2CCCC(CCNC(C3CCC(=O)N3)=O)C2)cnn1C c1(C(=O)NCCN(C2CCCCCC2)C(C2C(C)CCS2)=O)cccc2nsnc12 C12(NC(C3(CN(C)C)CC3)=O)CCCC1CN(C(c1cnc(C(F)F)[nH]1)=O)C2 c1(C(N(CC(CNC(C2CCCC(OC)C2)=O)C)C)=O)cnc2[nH]cnc2c1 C1(OC)CC(CO)(NC(=O)CCF)C1.C12C=CCN1C2=O.C(C)(C)(C)OC(=O)NC C12(C(=O)NC(C#C)(CC)CC)COCC1CN(C(=O)C(CCC)CCC)C2 C1(CC)CCN(C(C2CN3CCC2CC3)=O)C(C(N2CCC(C)(CCO)C2)=O)C1 Cn1cc(CC(O)C(=O)N2CC(CNC(c3ccsc3Br)=O)C2)cn1 C1(=CC(=O)N(C)CCN(C)C(c2cn(CCCF)nn2)=O)CCN(C)CC1 C(=O)(C(C)(O)C(C)(O)C(=O)N1CC2C=CC2C1)OC C1(NC(CCc2ccn(C)c2)=O)CC2(C1)CC(NC(=O)CC1C=CCC1)C2 C1(NC(c2n(C)c(S)nn2)=O)CCC2(CCN(C(C3CC3(C)C(F)F)=O)C2)C1 Cc1cc([N+](=O)[O-])cc(C(=O)N(C2CCN(C(=O)C(C)C(C)C)C2)C)n1 c1(CNCC2(CC)CCCO2)cc2c(s1)CCC(C)(C)C2 N1(CC(N2CCN(C(C(CC)(C)C#N)=O)CC2)=O)CC(=O)Nc2ccccc21 CC1(C)CN(C(C23CSCC2C3)=O)CC1NC(c1cc(N)ccn1)=O Cc1c[nH]c(=NCCCC2CCN(C(=O)CC3C(=O)N(C)N=C3C)C2)nc1O CC1CCC(CC(=O)NCC(C2CC2)N(C(=O)Cn2nnc(=N)[nH]2)C)C1 c1(C(=O)NCCC2CCN(C(C3N(C)C(=O)CC3)=O)C2)nc2c(s1)COCC2 N1(C(C2OCC(C)C2)=O)CCC2(CCN(C(=O)COCC3CC3)CC2)C1 C(=O)(CC(C(C)C)NC(=O)CCCCOC)N(C(c1cn(C)nn1)C)CC c1(C2C(C(=O)NCC(CCNC(CCCN(C(C)C)C)=O)O)C2)ccccc1Cl C=C1CC2(C1)CC(C(N1CCC1CNC(c1c(C)nn(C)c1C(F)(F)F)=O)=O)C2 C1(NC(C2CCc3nnnn3C2)=O)CC2(C1)CC2N=c1[nH]nc(CO)s1 C1(C(N2CCC(NC(=O)Cn3cnnn3)(CF)C2)=O)Cc2cc(F)ccc2O1 C(CN=c1cc(C)nc(NCC2CN(C)CCN2C)[nH]1)OCC(=C)C N1(C(CC(C)OC)=O)CC(NC(C2(NC(=O)OC(C)(C)C)CCC2)=O)C2(CC2)C1 c1(NC(CC(C)C)=O)ccccc1C(=O)NCC1CCCN1C(C1CC(O)C1)=O C(C)(CC(=O)N1CCC(N(C(=O)C(F)n2cccn2)C)CC1)(C1CCC1)N(C)C S(=O)(=O)(c1cccc(Cl)c1)NCCC(=O)NC(CN(C(=O)CCOC)CC)C c1(NC(C2(OC)CCOCC2)=O)[nH]c(=NCCNCCC#N)nc2c1ncn2C C1(C(=O)NC2(C3N(C(C4CNC(=O)N4)=O)CCC3)CC2)CCC2(CCC2)CC1 c1(C(N2CCCC(NC(C(CC)(C)C#N)=O)CC2)=O)[nH]c2ccc(C)cc2c1C N1(C(C2(F)C(C)C2)=O)CCCCC(CNC(=O)Cc2ccc(F)cc2F)C1 C#Cc1ccc(C(N2CCCC2CNC(c2occc2C(C)C)=O)=O)c(OC)c1 Cc1cc(C(N2CCC(NC(C3(F)CC3)=O)C(O)C2)=O)c(C)n1C1CCCCC1 c1(C(=O)NC(C)CCN(C)C(C2CC(=C3CC3)C2)=O)cc2cc(Cl)ncc2[nH]1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(CC(C)NC(C(c1cc(C)c(Cl)nc1)(F)F)=O)C C1(C(=O)NC(c2ccc(-c3ccc(F)c(F)c3)s2)C)CCCN(C(=O)C(N)=O)CC1 Cc1ccc(C(=O)NCCC2CCN(C(=O)C(C)n3cccn3)CC2)cc1O N#CCCCC(=O)NC1CC1CN(N1CCOCC1)C(c1cnn(C2CCC2)c1)=O C1(C(=O)Nc2cccc(CNC(=O)CC3CCOC3)c2)CC2CCC(C1)S2 N1(CC)C(=O)CCC1C(=O)NC1(CCCNC(=O)C=Cc2cccnc2)CC1 Cc1cn(C)nc1CNC(=O)C(C)C(C)NC(c1ccc(C(N)=O)o1)=O N1(C(C2CC=CCO2)=O)CCC2C(CCCN2C(=O)CCOc2cccnc2)C1 C(C)(C)(C(=O)NCc1ccccc1)NC(=O)NCC.C12CCCN1CNC(=O)C2 Cc1cc(N)cc(C(=O)NC(c2cn(-c3ccc(CO)cc3)nn2)(C)C)c1F C(=O)(C1=CNS(=O)(=O)N=C1C)NC1CN(C(C2N(CCC)CCCC2)=O)CC1C c1(C(=O)NCC(CN(C(=O)C(CO)c2ccccc2)C)O)cnc(C#N)s1 c1(C(=O)NC(CC(C)C)CNC(C2CN(C(N)=O)C2)=O)ccc2sncc2c1 C(CCCCC(=O)N1CC=CC(C(=O)NC2CN(C)C(C)(C)C2)C1)OC c1(C(=O)NCCCN(C(C(C2CCCOC2)OC)=O)C2CC2)c[nH]nc1Cl C(CC(C)CC)(C(=O)N(CC(C)(C)OC)C)NC(C(CCC)OC)=O C1(O)(CC(N2CCOC(CNC(C3CC4C=CC3C4)=O)C2)=O)CCCCCC1 Cc1cc(-c2cn(CCOCCOCCOCC(N)=O)nn2)cc(F)c1 c1(CCC)cc(C(=O)NC2CC23CC(NC(C2CC2F)=O)C3)cc(O)n1 C1(NC(CN2CCN(C)C(=O)C2)=O)CCCC2CN(C(=O)C(=O)NCCF)CC12 C(=O)(C(C)C(C)C(C)(C)C)NC1CC(CNC(c2ccc(C(=O)OC)nc2)=O)C1 Cc1ccc(CCCC(N2CC(C)CCC2CNC(=O)CNC(N)=O)=O)cc1C C1(CC#C)(C(=O)NCC(=O)NCC(=O)N(CC)CC2CCC2)CC1 Cc1noc(CCC(=O)NCC=CC(=O)NCCc2ncc(C)o2)n1 C1(NC(c2c(CC)c[nH]c2)=O)(COC)CCCN(C(=O)C(c2cnn(C)c2)C)C1 C(CCCCC(=O)N(CCCNC(=O)C(C)c1ccco1)C(C)C)NC(=O)OC c1(OC)ccc(C(=O)NC2CC(C(=O)NC3(C4CCCCO4)CC3)C2)o1 C1(C(=O)OCC)CCC(NC(=O)C(c2ccsc2Cl)N2CCOCC2)C1 C(N=c1[nH]c(=NCCCOC2CCOC2)[nH]c2cc[nH]c12)C1(C)CC(C)(C)C1 N1(C(C(C)Cc2ccc(Cl)cc2)=O)CC2CC(C1)CN(C(=O)C1=CCC1)C2 C1(OCC)CN(C(=O)C(c2ccccc2)O)CC1NC(=O)CN1CCC1C c1(OCC)cc2c(cc1F)N(CNc1cccc(OC(F)F)c1)CC2 C1(C(=O)NCC(C(C)(C)C)NC(CSCC=C)=O)CC(C(C)(C)C)=NO1 C12(NC(CC(C)(C)C3CC3)=O)CCCC1CN(C(=O)C(C)(C)S(C)(=O)=O)C2 Cc1cc(Cl)c(C(=O)NCC(C2CCC2)NC(=O)C(C)(C)N2CCOCC2)cn1 CCCCCCC(CC)C(=O)NC(C)CC(C)NC(=O)C(C(C)C)SC C1(C(C)CNC(=O)NC(C)C(=O)NC2CCC2)CCCCC1 N1(C(C2CCC(C)(C)C2)=O)CCC2CN(C(=O)CC(C)(C)C(F)F)CC2C1 c1(C(=O)NCC2(NC(C(CO)N(C)C)=O)CCC2)cccc2nonc12 C1(CN(C(c2[nH]cc(C)c2)=O)C)CCCC(NC(c2sccc2C#N)=O)C1 N1(C(C(C(CC)C)O)=O)CCC(C2(NC(=O)CCNS(=O)(=O)CC)CCC2)CC1 N1(c2nc(C(C)C)cc(C)n2)CCC2(CCN(C(=O)CCc3ccon3)C2)C1 c1(OC(C)C)cc(CNC(=O)NCC2CC2(F)Cl)ccn1 C(c1ccc([N+](=O)[O-])s1)=CC(=O)N(C1CCN(C(=O)CC2(O)CC2)CC1)CCO c1(-c2ccc(OC)cc2)n[nH]c(=NC(=O)N(C)Cc2nnc(C)o2)s1 N1(C(C2CC(=O)NCC2)=O)CCC2(CC(C(=O)N3Cc4ccncc4C3)=NO2)C1 C123CCN(CCC1C2)C3=O.N1(OC(C)=O)CCCN(C(=O)Cn2cnnc2O)CC1 n1(CCN(C)C)nccc1C(=O)NCC1(O)CN(C(c2cc(Br)no2)=O)C1 C1(CNC(c2ccc(C3CC3)cc2)=O)CC(O)CN1C(c1ncc(Br)cn1)=O C(=O)(C(C)(C)C1=CCSCC1)NCCCN(C(=O)COCC1CCOC1)CC c1(C(=O)NCC2(O)CN(C(C(CCC(C)C)O)=O)C2)cnc2c(c1)NCC(=O)N2 C(N=c1[nH]c2c(c(=NCCCS(C)=O)[nH]1)CSC2)C1(OC)CCC(C)(C)CC1 Cc1cccnc1-c1cn(C2CN(C(C3(N4CCCC4)CCC3)=O)C2)nn1 C12(CNC(=O)C=C3CCC3)CCC(CC1)N(C(=O)C(F)C1CCCC1)C2 CC1CN(C(=O)C(CC(N)=O)N(C)C(=O)OC(C)(C)C)Cc2ccccc21 C(=O)(C1=CC2C=CC(C1)C2)NCC(COC)NC(=O)CC(C)(C)CCOC Cc1ccc(Cl)c(C(=O)NC(C)CC(C)NC(=O)CCOC(C)C)c1 C1(O)(CNC(C2(CCC)CC2)=O)CCCN(C(=O)CCOCCF)C1 c1(C(=O)NCC(CN(C(CC=C=C)=O)C)O)nc2c(Br)cncc2[nH]1 N1(C(Cn2c(CCC)ncc2)=O)CC2C(CNC(c3conc3C3CC3)=O)C2C1 C(=O)(CC(C)(O)C(F)(F)F)N1C2CCC(CNC(CCC=C)=O)(C2)C1 O(N(C(=O)C1CC(CCNC(=O)CC(O)CN(C)C)C1)C(C)C)CC N1(C(c2cc(Br)nn2C)C(=O)NC)c2ccccc2CC1Cc1ccccc1 Cc1oc([N+](=O)[O-])cc1C(=O)NCC12CC(NC(c3ccc(N)cc3Cl)=O)(C1)C2 Cc1nn(CC(C)C)c(Cl)c1C(=O)NC(C)C(CO)NC(=O)CC(=O)OC(C)(C)C C12(C(=O)NCCOC(C)(C)CNC(c3ccc(N)cn3)=O)CCN(C1)S(=O)(=O)C2 Cc1ccc2c(C(=O)NCC(C)(C)NC(=O)C3=NOC(C)C3)ccnc2c1 c1(NC(N(c2ccc(Cl)cc2)C)=O)nc2c(F)cccc2n1C N1(C(C23CC(C)C2C3)=O)CC(NC(=O)CN(C2CCCC2)C)CC(C)C1 c1(CNc2c(F)ccc(Br)n2)cc2cc(Br)ccc2s1 N1(C(C(C)c2ccsc2)=O)CC(C(C2CC2)NC(=O)Cc2cccs2)C(O)C1 CCCCC(CC)CCC(=O)NCC1CC(C)N(C(=O)CSC(C)C)C1 CC(C)CC(=O)NC(C1CN(C(=O)CCN2CCC2)C1)C N1(C(C2C(C)(C)CO2)=O)CC2CCC1CN2C(=O)CCC(=O)N1CCOCC1 c1(CC)cc(C(=O)NCCC2CC(NC(=O)C(C)(C)C3CCOCC3)C2)ncn1 C(=O)(CC(C)(C)C(=O)NCc1cn(C2CN(C(=O)C=CCO)C2)nn1)OCC c1(OS(CC2CC(C)OC(C)C2)(=O)=O)ccc(N=NC(N)=O)cc1 C1(NC(c2c(C)nc(C)s2)=O)CCCCCC1C(=O)N(C1CC(O)C1N)CCOC C=CCCC(F)(F)C(=O)N1CC(CNC(=O)C(c2ccn(C)n2)C)(OCC)C1 c1(C(N2CC3CC(NC(c4nc(Cl)ccc4Cl)=O)C3C2)=O)cccc2ncoc12 c1(CC(N2C(CCCNC(c3cc(C)ncc3)=O)CCC2)=O)ccc(O)c(Cl)c1 c1(C(=O)NCC2C(NC(c3c(OC)nsc3)=O)CCCC2)csc([N+](=O)[O-])c1 N1(C(c2c(CC)c(C)ccc2)=O)CC(NC(=O)CC(C)SC)C(C2CC2)C1 CC12CC(C(=O)NCC3CCC(NC(c4cc(O)ncn4)=O)C3)(C1)C1(CCC1)O2 c1(CNC(=O)N(C2CC2)Cc2ccccc2)cc2ccccc2s1 Cc1ncc(CCC(N2CCOCC(NC(C3CCC(=O)O3)=O)C2)=O)c(O)n1 c1(C(=O)NCc2nnc(CN(C)CCO)o2)cccc2c1nnn2C N1(C(C(C)OCC)=O)CCC(C(=O)NOc2ccc(CC)cc2)C12CC2 c1(N(CC(=O)N(CCCNC(=O)Cc2ccnn2C)CC)C)ccc(Cl)cc1 C1(NC(Cc2nnc(C)o2)=O)COC2(CCCN(C(c3cccnc3O)=O)C2)C1 N1(C(CCC=C=C)=O)CC2(C1)CN(C(=O)CCC(=O)NCCOCC)CC2CO c1(C(=O)NC(C(C)NC(=O)CC2CCOC2=O)CO)cc(Cl)cn1C N1(C(CN(C(C)C)C(C2COCCC2C)=O)=O)CCN(C2CC2)CC1 c1(OC)ccc(CC2(OC)CCC2)cc1NC1(c2ccccc2)CC2(CNC2)C1 C(=O)(CCCCNC(C)=O)N1CC(C(N)=O)(CNC(c2ccc(CC)o2)=O)C1 CC(CC(=O)N(C)CCN1CCOCC1)C(C)(C)NC(C1CC1C(C)(F)F)=O c1(C(=O)NC(C2CCCCN2C(=O)C2=CCC2)C)cn(C)c2ncccc12.CCCCl CC(C)CC(C)(O)C(=O)Nc1cccc(NC(C2CC(=O)N(O)C2)=O)c1 c1(C(=O)NCC(CNC(c2nccnc2C)=O)OC)ccc(C(C)C)c(C)c1 c1(NC(C2N(C(c3c(C)ocn3)=O)CCC2)=O)ccccc1C(C)(C)C C1(NC(c2ccc(C)nn2)=O)CCC(C)N(C(C2CCC(C)(C)O2)=O)C1 C(C(C(C)C(C)C)NC(c1cc(O)nn1C)=O)NC(COCCC=C)=O C=C1CCC(C(=O)NC2CC(NC(=O)Cc3ccc(NC(N)=O)cc3)C2)CC1 C(=O)(C(CNC(c1cc2occc2[nH]1)=O)CCC)NC(C=C)C c1(NC(N(C)Cc2ccnn2C)=O)coc(C2CCCN2c2ccncn2)n1 CS(=O)(=O)c1ccccc1C(=O)NCCNC(=O)CC1CCC2CC1C2(C)C c1(OC)cc(C)c(C(N2CCC(O)C(NC(=O)CC(C)NC(N)=O)C2)=O)c(F)c1 C(C(C)(C)CC(F)F)NC(C1CN(C(c2ncn(CC)n2)=O)CC1F)=O CCCCCC(F)C(=O)NCC(C)CNC(C1(CC(C)C)CC1)=O Cc1nc2cnn(C)c2cc1C(N1CCC(N(C)C(c2cscn2)=O)C(C)C1)=O N1(C(=O)CC2CC3CCC2O3)CCN(C(=O)Cc2nc[nH]n2)C(C2CC2)C1 C(=O)(C(C)C(C)C)NC(C(=O)NC(C)Cc1ccnn1C)Cc1cn[nH]c1 C(N=c1[nH]c2c(c(=NCc3ncc(C)[nH]3)[nH]1)COC2)c1c(CCC)nns1 C1(CNC(C(C=C)(C)C)=O)CC2(CCC2)CN1C(C1CCC(=O)NC1)=O Cc1c(Cl)c(C(=O)NCC(C)(CO)NC(c2csc(C(C)=O)c2)=O)nn1C N1(C(CC=CCNC(C2(C)CCC(=O)NC2)=O)=O)CC2CCC(O)C2C1 c1(C(=O)NCC2(NC(Cc3ccc(C)o3)=O)CCC2)cnc2n1CC(C)CC2 c1(NC(C2C(NC(CC(C(=O)OC)(C)C)=O)C2)=O)cc(C)c2cc[nH]c2c1 C(=O)(C1CCCc2c[nH]nc21)N1C2CC(NC(c3cc(C)sn3)=O)C(CC2)C1 C1(NC(=O)C=Cc2ccncn2)CC(O)CN(C(c2cnccc2Cl)=O)C1 Cc1cccc(Br)c1C(C(=O)NCCCCS(C)=O)NC(=O)C1=CCOCC1 N1(C(C(CC)C)=O)CCN(C2CCN(C(=O)Cc3c[nH]nc3O)CC2)CC1 N1(C(CCCCC)=O)CC2CCCC(C1)N2C(=O)CSCc1csc(=N)[nH]1 N1(C(C(CC)OCC)=O)CC2CC(C)C(C1)N2C(=O)C(C1(O)CCCC1)F c1(CC)cccc(C(=O)N(CC(O)CNC(=O)C(F)n2cccn2)C)n1 CC1(NC(c2ccc(Cl)c(O)c2)=O)CCN(C(=O)C=Cc2ccc(Cl)s2)CC1 C1(C(=O)NC(CC(=O)NC)C)CCN(C(c2cccc(CO)c2)=O)C12CCC2 C1(C(=O)NC23CC(NC(=O)C(F)F)(C2)C3)CCC2C1C2(F)F Cc1ccc(-c2csc(NC(=O)C(C)Sc3ccccc3)n2)cc1 Cc1ncccc1C(N1CCCC(CCC(=O)NC(C(C)C)c2nc[nH]n2)C1)=O c1(OC)ccc(N(CC(=O)NCC(CC2CC2)CO)C)cc1 N1(C(C2C(=C)C2)=O)CCC2CCC(C1)N2C(=O)C=C1CCCCC1(C)C c1(NC(CCN(CC=C)C(c2cncc(OC)n2)=O)=O)ccc(C)cc1C C1(N(C(C(C)S(N)(=O)=O)=O)C)CCN(C(c2cc(C3CC3)ccn2)=O)CC12CC2 C#CC1(C(=O)N(C)CC2CCCS2)CCN(C(=O)CC2CCC(C)(C)O2)C1 c1(NC(C)=O)c(C(=O)N(CCCNC(=O)Cc2cnc(C)[nH]2)C)cccc1C c1(C(N2C(CC)CN(C(=O)C(C)(C)SC)CC2)=O)cccc2c1CNC2=O C1(CN(C(COC(C2CC(=C)C2)=O)=O)Cc2ccccc2)CC(C)CO1 N(C1CCc2c(Br)ccc(Cl)c21)CC1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1 N1(C(c2c(CC)occ2)=O)CCCC(NC(C2CCN(c3ccncc3)C2)=O)C1 c1(CCn2c(-c3ccc(C#C)c(Cl)c3)nc(C)n2)nc2nc(C)c(C)c(C)n2n1 c1(CC(=O)NCC(N2CCCCC2)C)ccnn1C C1(NC(C2(C(N(C)C)=O)CC2)=O)CCN(C(C2CC3CCC2C3)=O)CC1(C)C c1(C(N2CCC(OC)(CNC(=O)CSC)CC2)=O)sc2[nH]cnc(=O)c2c1C N1(C(=O)C=Cc2cn3c(n2)CCCC3)CCc2nc[nH]c2C1c1ccccc1 C1(C(N2C(C(C)NC(=O)CCc3ccccn3)CCC2)=O)COC(C)(C)CO1 c1(CC)cc(C)ccc1NC(c1c[nH]nc1CCNC(C1(C)CC1)=O)=O N1(C(C(CCC)N(C)C)=O)CCCC(CNC(c2c(C)n[nH]c2C)=O)CC1 N1(C(c2c(C)nsc2)=O)CC(CNC(=O)C=Cc2cnc[nH]2)CC12CCC2 CC1CN(C(=O)C(C)(C)C2CCCO2)CCN1C(C1(C(N2CCOCC2)=O)CC1)=O C(=O)(C(C)(C)CC(F)(F)F)N1C(CO)CC(NC(c2cc(C)n(C(C)C)n2)=O)C1 C1(N(C(C(C)=C2CC2)=O)C)CCC(NC(=O)Cc2cc(C)cs2)C1 CS(=O)(=O)c1ccc(Cl)c(C(=O)NCCC2CN(C(C3CC3F)=O)CCO2)c1 c1(OCCN(C)C)cc(Br)ccc1CNC(=O)Nc1cn(C2CC2)nn1 c1(OCCn2c(C(C3CC3)NC3(CC)CC3)nnn2)ccncc1 C1(CNCC2(COC(C(COC)O)=O)CC2C(F)(F)F)CCC(NC)CC1.C(F)(F)F C1(C)(OC)CC(NC(=O)CCNC(=O)CC2CCCCO2)C1(C)C c1(CC)ncsc1C(=O)N(C)CCOCCC(=O)NCCn1cncn1 N1(C(CCCC)=O)CC(OC)C(NC(=O)CSCc2cccc(F)c2)C1 C1(NC(c2c(C)nsc2)=O)CC(C2CCN(C(=O)Cc3cccc(Cl)c3)C2)C1 n1(CCC=C)cc(C(=O)NCCC2(O)CN(C(c3cnc(C4CC4)o3)=O)C2)nn1 CCCC(CCC)CC(=O)NCC(CO)NC(C1CCC1C(=O)OC)=O CC1CCCCN1NC(=O)C1(c2ccccc2Cl)CCC1 C1(C(=O)NC(C)Cc2ccsc2)CCCCCN1C(=O)COC(F)F Cc1cncc(NC(C2(CNC(C3(C)CCSCC3)=O)CC2)=O)c1 C(C)(C)(CC(F)C(=O)N(C1CCN(C)C1)C)NC(c1c(CC)cncc1)=O C12(CNC(=O)C(c3cccs3)NC(C3CC4CC4C3)=O)CCC(CC1)C2 C(=O)(C#CC1CCCO1)NC1CCN(C(c2ccnc(C)c2C)=O)CC1 C=CCC(C)(CNC(C1CC(O)CN1C(=O)CCOCCCOC)=O)CO C1(NC(c2cc(C)nc(O)c2)=O)CCSC12CN(c1ncnc(C(C)(C)C)n1)C2 CCCC(CC)CC(=O)NC1(C)CCN(C(c2ccc(CNC(C)=O)cc2)=O)C1 c1(C(N(CCCCNC(C(CCSC)OC)=O)C)=O)cnn2c1NCC(C)C2 C(=O)(CC(C)(C)C(F)F)N1CCN(CC(=O)NCC(C)(C)F)CC1 C1(C)(CNC(=O)Nc2sc(C(=O)OC)c(C)n2)CCC(C)C1(C)C C1(N2C(C#C)CCC2)C(=O)NN2CC(CC1C)C2.C1(C(=O)OC)CCOCC1 CCCCCC(O)C(=O)N1CCCC(CCNC(c2c(C3CC3)cnn2C)=O)C1 CCC(CC)CC(=O)N(CCSC)CC.C12CCN(CC1O)C2=O N1(C(CNS(N)(=O)=O)=O)CCC2CC2(NC(c2cc(Cl)ccc2Cl)=O)CC1 C#CCCC(=O)NCCCCNC(=O)C(C)(C)NC(=O)Nc1ccccc1 c1(CC)cc(C(=O)NCC(C)(CO)NC(c2sc(C3CC3)nc2C)=O)cc(O)n1 C(=O)(CCCCCNC(=O)COC1CCOC1)NCC1(C)CC=CCC1 N1(C(c2[nH]c(=N)sc2)=O)CCCC(NC(=O)C(O)Cc2cnc[nH]2)CC1 C1(CNC(C(C=C)(C)O)=O)CN(C(c2ncoc2CC)=O)C2(CCC2)C1 c1(CC(=O)NC(C(N2CCC(COCC)C2)=O)(C)C2CCC2)ccc(F)cc1 C12(C(=O)NC(CNC(CNC(CCNC(C)=O)=O)=O)C3CC3)CC(C1)C(C)(C)O2 C#CCC(C)C(=O)NC1CC1CNC(=O)CSCC(=O)N(c1ccncc1)C C1(C(N(C(C)C(=O)NCC2SCCS2)C)=O)CCCN1C=O c1(C(N2CC(COC)(CNC(=O)CCC(C)N(C)C)C2)=O)cnc(Cl)c(N)c1 C1(NC(CCc2c(C)n(C)nc2)=O)CC2(C1)CN(C(C1(C)CCC(C)CC1)=O)C2 N#Cc1ccccc1N1CCCC(NC(=O)NC2CSC(C(F)(F)F)C2)C1 Cc1cc(NC(C23COC(Cc4ncc(OC(C)C)cn4)(C2)C3)=O)oc1Br C1(=CC(=O)NCCSCC(=O)NCCC2CCSC2)CCOCC1 C1(NC(C(C)CC2CC2)=O)CC12CCN(C(c1ccc(C3CC3)o1)=O)C2 c1(CC(N2CC3(C(NC(C(C)C)=O)CCS3)C2)=O)ccc(Cl)cc1[N+](=O)[O-] C1(CNC(c2cscc2F)=O)CCCCN1C(c1conc1C(F)(F)F)=O c1(CC(=O)NC23C(CN(C(c4c(C)ccs4)=O)C2)C3)ccc2n[nH]cc2c1 N1(C(c2n(C)cnc2)=O)CC2(CCCN(C(C3CC3c3ccccc3Cl)=O)C2)C1 N1(C(c2ncn(C)c2)=O)CC2COCC2(C(=O)NC2CCCC(C(N)=O)C2)C1 N1(C(Cc2nc(CC)sc2)=O)CCC(NC(c2cc(C)n(C)n2)=O)C1(C)C c1(C(=O)NCCC2(CNC(C3CCC(CC)C3)=O)CC2)cnc(OC)c(C)n1 C1(CNC(=O)COCCO)CCCN(C(=O)CN2CC3CC3C2)C1 c1(OC(C(=O)N(CC(C)NC(c2cncc(O)c2)=O)CC)C)cc(Cl)cc(Cl)c1 C(CC(C)C(=O)NC(CCOCCO)C(=O)NCc1ncnn1C)=CC N1(C(CCc2n(C)cnn2)=O)C(CC(=O)NCCn2cnccc2=O)C2CCCC12 Cc1ccncc1C(=O)NCCC1CC(C(=O)NCc2cnccn2)C1 CC(C)CCC(O)C(=O)N1C2CCC1CC(NC(C1(C)CCCC1)=O)C2 c1(Cn2cc(C(C)NC(C3CCC(SCC)CC3)=O)nn2)ccc2c(c1)CCO2 C1(C2CCCN(C(=O)C(C)(C)N(C)C)C2)(NC(c2n(C)c(S)nc2)=O)CC1 c1(C(N2CCC(CNC(C3(O)CC(C)(C)C3)=O)C2)=O)ncc(Cl)cc1Cl CC(CS(C)(=O)=O)C(=O)N1CCC(CCNC(c2cncc(C(N)=O)c2)=O)CC1 N1(C(C2C(C)CCS2)=O)CCN(C(c2ccc3[nH]ccc3n2)=O)CC12CC2 c1(C(C(=O)NCCCF)N(CCCC)C)ccc(OCCOC)cc1 C12(C(N(CC)CC3CCCN3C(=O)CSC(C)C)=O)CCCC1C2(F)F C(=O)(C(C)C(O)CC(C)C)N1C2CC(NC(c3cc(CC)ncc3)=O)(C2)C1 c1(CC(=O)NC2(C)CN(C(=O)CCC(F)(F)F)C2)cc(C(F)(F)F)cc(F)c1 C12(C(N3C(C(=O)NC)CC3)=O)CCCC1CCN2C(=O)C(n1cc(C)cn1)C N1(C(=O)Cc2cccc(F)c2F)CC2CCN(C(C3(C4CC4)CC3)=O)CC12 N1(C(c2c(C)oc(Br)c2)=O)CCC(O)(CNC(=O)C=C2CCC(C)C2)CC1 C1(O)(C(=O)NC2C(NC(C(=O)NCC)=O)CCC2)CCCC(C)(C)C1 C1(C(N2CC(=C(CNC(C(CC)N(C)C)=O)F)C2)=O)NC(=O)CC1C C(C(C(=O)N(C1CC=CC1)C)NC(=O)CC1CC=CC1)OC(C)C C1(NC(c2cnc(OC)nc2)=O)CCN(C(c2ncc(C)cc2OC)=O)CC1C C=CCCCCCC(=O)NN1CCCC1C(=O)NCC1C(C)(C)C1(F)F C1(C2=CCOCC2)(CNC(N2CCCC(C(=O)OCC)C2)=O)CC1 N1(C(C(Cc2ccc(Cl)cc2Cl)NC(C2CC2Cl)=O)=O)CC(O)C2(CCCC2)C1 c1(C(=O)Nc2ncc(Cl)cc2I)csc2c1CCN(c1nccc(C(F)F)n1)C2 CC1(CNC(C2CCN(C3COC3)C2)=O)CN(C(c2cnc(O)s2)=O)CCO1 C(CC(C(=O)N1CCOCC1CCC)NC(C1C=CC=CC=C1)=O)=CC N1(C(c2c(C)con2)=O)CCN(C(c2cc(Br)cnc2O)=O)C2CC12 C(=O)(C(F)C(=O)N(C(C)C(=O)NC1C=CC(C(=O)OCC)C1)C)OCC c1(N2CCC(OC)(OC)C2)ccc(S(=O)(=O)NCc2ccn(C(F)F)n2)cc1Cl C(=O)(C1=CCC(C)(C)CC1)N1CCC(C)C(NC(=O)CCc2cnccn2)C1C C1(C(N2C(C)(C(=O)OC)CC2)=O)CCCC(NC(=O)CCc2cnco2)CC1 C#CC1(OC)CCN(CCCNC2CC2c2cc(Br)ccc2F)CC1 C1(C(C)C)CN(C(C2CC2C)=O)CCN1C(c1cc(Cl)no1)=O N1(C(CC(CC)C(C)C)=O)CCC2CC(CNC(=O)C3=COCCO3)CCC2C1 Cn1ncc2c1CN(C(c1csc(NC(c3ccc(O)cc3)=O)n1)=O)CC2 C1(C(N2CCC(C3N(C(=O)OC(C)(C)C)CCCC3)CC2)=O)C2CC(F)(F)CC12 C(=O)(C(C)(C)c1cnsc1)N(CC(O)CNC(=O)C1CC1)C N1(C(c2nc(C#C)sc2)=O)CCCC2(C1)CN(C(=O)CC1(OCC)CC1)CCO2 N1(C(C2CC(C#C)(O)C2)=O)CCC(CCNC(C2(COC)CC2)=O)C(F)(F)CC1 C1(NC(=O)Cc2cc(Cl)ccc2O)CC12CCN(C(C1(Cl)CC1(F)F)=O)CC2 C1(NC(CCC#C)=O)CCCCCC1NC(=O)COc1ccc(F)cc1Br Cc1c(C(=O)NCCC(C)NC(=O)CC(F)(F)F)ccc2c1CCC2 c1(C(=O)OC)cc(NC(=O)C(=O)NC2CC(CS(C)(=O)=O)C2)ccc1F C(N=c1nc2c(ncn2C)c(NC(C)Cn2ccnc2)[nH]1)c1cc(C)ns1 CN1CCOC(CNC(C2OCCC2NC(c2cnn[nH]2)=O)=O)C1 CCCCCCCC(=O)N(CCNC(c1cc(C)ncn1)=O)CC1CC1 CCC(C(=O)NC(C(=O)N1CCC1CN=[N+]=[N-])c1ccco1)C(C)C CCCCC(CCC)NC(C1(NC(c2cn(C3CC3)nn2)=O)CCN(C)C1)=O C(=O)(C(C)(C)CCCF)N1CC(C(NOC)=O)C(CNC)C1 C(CC(C(C)(C)C)NC(=O)Cc1ccc(Cl)cc1)N(C)C(C1CCNC1=O)=O c1(CNC(C(CO)NC(=O)OC(C)(C)C)=O)sc([N+](=O)[O-])cc1Cl CC(C)(C)CCCC(=O)NCC(CNC(C1C(C)(C)OC1(C)C)=O)CO N1(C(C(CC)O)=O)CC2CCOC2(CNC(c2c(C(F)(F)F)cccc2F)=O)C1 c1(NC(COC(C)(C)CNC(=O)CN2CCCC2=O)=O)ccc(CCO)cc1 C1(NC(C2CCC(CCC)CC2)=O)CCN(C(c2ncccc2F)=O)CC1F C1(NC(C2CC(=C)C2)=O)CN(C(=O)Cc2nc(C3CC3)cs2)CC12CCC2 CC1(C)COCC1CNC(=O)Cn1cc(CCc2ccc(C(F)(F)F)cc2)nn1 C(C)(C1=NOC2COCC12)NC(N(c1ccc(Cl)nc1)CCNC(C)=O)=O C(=O)(C(CC)(CC)CC)N1CC(CCC)C(NC(=O)CN(C(=O)C(C)C)C)C1 n1(CCC)ncc(C(=O)N(CCNC(=O)C(=O)NC2CC2)CC)c1Cl C1(NC(C2CC(C)(O)C2)=O)CC(CNC(c2cc(F)n[nH]2)=O)C12CCC2 C1(NC(COCCOC)=O)CC2CCC1CN2C(=O)CCc1cccc(O)n1 C#CCCCC(=O)NCC(C1CC1)NC(=O)Cc1conc1C C1(NC(C2CC(C)N(C)C2)=O)CC2CCC1CN(C(C1(C)CCCN1C)=O)C2 c1(C(=O)NCC(C(C)C)C(=O)NC2CCC=CCCC2)cccc2cncn12 c1(C(=O)NC(C(C)NC(=O)Cc2cc(Br)cs2)C)ccc(Cl)cc1N C12(NC(C3CC(C)(C)C3)=O)CC(C1)N(C(=O)C(=O)NCc1ccc(F)cc1)C2 S(=O)(=O)(c1cnccc1N1CCC(O)CC1)NCC1CCN(CCC)C1 C1(NC(C(C)OCC)=O)CCCN(C(c2ccc(C3CC3)o2)=O)C1CC C1(NC(C2(OC)CCSC2)=O)CN(C(C2SCC=C2C)=O)CC1(C)C n1(CC)cnc2c(NC(C)=O)[nH]c(=NCCNC(C)(C)COC)nc12 c1(C(N2CCC(COC)(NC(c3csc(C(F)F)n3)=O)C2)=O)cc(C)cnc1C CC(C1CCCc2ccccc21)NC(C1CC1CF)=O c1(C(CC(=O)Nc2c(C)ncn2C)O)nc2ccccc2[nH]1 N1(C(CNC(=O)OC)=O)CC(OC)C(C(=O)NC(CN2CCC2)CO)C1 C1(C(=O)NC(CNC(c2scc(C)c2)=O)C2CCC2)Cc2c(C)cccc2O1 C(C)(C(C(=O)NCc1nccnc1C)NC(=O)CC1CC2CCC1O2)OC N1(C(c2[nH]cc(CC(C)C)c2)=O)CC(C)N(C(=O)C=Cc2ccco2)CC1C C1(CNC(C(CC)CC)=O)CN(C(=O)CCCN(C)C(C)C)CC(C)(C)O1 N1(C(CCC2(C)CC2)=O)CC2CCC2(CNC(=O)CCCCNC(N)=O)C1 C1(NC(C2C(c3c(Cl)ccc(OC)c3)C2)=O)Cc2cccnc2NC1=O C(C1CCCN1C)=CC(=O)NC(C1CN(C(c2coc(C(F)F)c2)=O)CCO1)C Cc1cc(C(F)(F)F)nc(NC2(CNC(=O)C(C)C3CCCO3)CCC2)n1 c1(C(=O)OC)ccc(Br)c(C(=O)NCCCCc2cccc(Cl)n2)c1 C1(NC(C2(C)CC(C)C2)=O)CC2(C1)CC(CNC(=O)Cc1cncn1C)C2 Cc1oc(COc2ccc(C(n3cc(CN)nn3)C)cc2)cc1Br Cc1ccc(C(=O)N(C)Cc2cn(Cc3ccc(Cl)cn3)nn2)c2c1NCCC2 CC(F)(F)CCCC(=O)NCCN1CCN(C(=O)C(C)(C)C2(O)CCC2)CC1 c1(C(=O)NCC2(O)CCCN(C(CCCC(C)=O)=O)C2)c(Cl)nc2sc(C)cn12 c1(C(=O)NC(C2CN(C(C3(C)CC3F)=O)C2)C)nccc2cc[nH]c12 CC1C(NC(C2CCCC3(CC3)C2)=O)C(C)CCN1C(=O)Cc1cn(C)nn1 C1(NC(C(C)NC(N)=O)=O)CCC12CN(C(=O)CN1CCN(C)C(=O)C1)C2 N1(C(=O)CC2CCCCN2C(c2cnn[nH]2)=O)Cc2ccc(O)cc2C1 C(c1ccc(F)cc1F)=CC(N1CC2C(NC(C3N(C)CCOC3)=O)(C2)C1)=O CCC(C)C(O)CC(=O)NC(C)C=CC(=O)N(CC(F)(F)CC)C C1(C)(CNC(=NCCC)NCCCOC(C)CC)CCC(F)(F)CC1 c1(OC)cc(F)c(C(=O)NC2CCC(NC(=O)CC34COCC(C3)C4)C2)c(F)c1 n1(C(C(=O)NCCNC(CC2C(C)(C)OCC2)=O)(C)C)cc([N+](=O)[O-])cn1 c1(C(N(C2CCCO2)CC)=O)cc(-c2cc(OC)ccc2OC)ccc1F C1(NC(c2cncc(CC)c2)=O)CCN(C(c2coc(Cl)n2)=O)CC12CCC2 O=C1NCC2(CN(C(=O)CCN(CCO)C(c3cc[n+]([O-])cc3)=O)C2)N1 c1(CC(N2CC(O)CC(NC(c3cc(C)c(C)s3)=O)C2)=O)ccccc1[N+](=O)[O-] c1(NC(=O)NCc2c(C)ccs2)cc([N+](=O)[O-])ccc1F C1(C(=O)NCc2ccncn2)CCC(C2CC2)N1C(c1ccnc(O)c1)=O c1(C(=O)NC(CNC(CC(CC)C)=O)(C)CO)cc(C)cc2c1OCC2 Cc1ccnc2nc(C(=O)NC(C)C(C3CCCCC3)NC(=O)C(N)=O)nn12 C1(CNC(=O)C(Cl)=CCl)CCN(C(c2cnc(-c3cccnc3)s2)=O)C12CCC2 C1(C(N2C(C)(C)CC(c3ccccc3)C2)c2ccccc2)CNc2ccnn2C1 C(=O)(CCCCC(C)=O)NC1CN(C(C)=O)CC1(F)F N1(C(C2(CCC)CCC2)=O)CCC2(C=C(C(=O)N3CC(CCOC)C3)C2)C1 n1(CC(N2C3CN(C(C4=NNC(=O)CC4)=O)C(C3)C2)=O)ncc(=O)c2ccccc12 c1(C(N2C(CNC(=O)OC3CCC3)CCC2)=O)cnc(O)c2ccccc12 C(=O)(C1CCCc2ccccc21)N1CC(NC(c2nn[nH]c2Cl)=O)CC2(C1)CC2 CC1C(C(=O)NCCCn2nccn2)CCCN1C(=O)C(C)n1ccnn1 c1(CCC)cccc(CC(=O)NC2(CO)CN(C(=O)COCCN(C)C)C2)c1 c1(C(C)=O)ccc(C(=O)NC(C)C(C)NC(=O)CC2CC(N(C)C)C2)cc1F CC1CN(C(C2CCCCN2N=O)=O)CCCN1C(C1CCN(C)CC1)=O c1(CC(=O)N(CC(CNC(C(C=CCCC)O)=O)C)C)cccnc1C c1(CC(=O)NCC2(O)CC(NC(c3ccnc(O)c3)=O)C2)nc2c([nH]1)CCCC2 Cc1cc(=NC(=O)C(C2CCCO2)NC(C2SCCS2)=O)[nH]n1C(C)C CC1C(C(=O)NCC2(CN(C)C(c3cnn(C(C)(C)C)c3)=O)CC2)CCN1C c1(C(=O)NC2C(OC)CN(C(=O)CSC(C)C)C2)nccn2nccc12 c1(C(=O)OCC)[nH]c2ccc(Oc3cn(C)nc3C)cc2c1C c1(CCN(CC(=O)NC(=O)NCCc2ccsc2)CCC)ncc(OC)cn1 c1(C(=O)NCC2N(C(C(C)N3CCC3)=O)CCCC2C)ccnc2nccnc12 c1(OC)c(C(N2CC3CC3(NC(=O)Cn3ccc(C4CC4)n3)C2)=O)csc1Cl N1(C(=O)CNC(C2CCCO2)=O)CCN(C(C2(c3ccccc3)CCC2)=O)CC1 c1(C(=O)NCC2C3CN(C(C(CC4CC4)OC)=O)CC32)ccc(Cl)cc1F C(CCC(=O)N(C(C)C(=O)N(C)CCc1ncccn1)C)OC(C)C C1(NC(c2c(CC)nc[nH]2)=O)CCN(C(=O)CCOCCOC(C)(C)C)CC1C Cc1cc(C)c(C(=O)NC2CC(NC(C3CCC(C(F)F)CC3)=O)C2)cn1 n1(CC(N2C(CCCNC(C3CC(=C)C3)=O)CCC2)=O)nc(C2CC2)n(C)c1=O C1(C(N2C(CC(=O)NC(c3ccncc3)C)CCC2)=O)CCCN1C=O C1(NC(CC(C)(C)OC)=O)C(C)(C)C(NC(=O)C(CCO)N(C)C)C1(C)C N1(C(CC2CN(C)C2)=O)CCC2CCCN(C(c3cnsn3)=O)C2C1 Cc1ccc2c(c1)CC(C(=O)NC1CN(C(=O)C(C)(C)CN(C)C)CC13CC3)S2 C(=O)(CCS(=O)(=O)C(F)(F)F)NCC(CCCC)NC(C1CC1(C)C(F)F)=O CCC(C)C(O)C(=O)NC1CC2CC1N(C(c1cnc(C)s1)=O)C2 C1(CC)C(NC(=O)C(C)CC(N)=O)CCCN1C(=O)CC1CC(C)(C)CO1 C(CCCOC)(C(=O)N1CCOCC(O)C1)NC(C(COCC)C)=O C1(OC2CN(C(CNS(C)(=O)=O)=O)C2)CCN(C(c2cccnc2)=O)CC1 c1(C(=O)NCCOCCNC(C(C2CCOCC2)C)=O)cncc2nnn(C)c12 c1(C(=O)NC2(C)CC(NC(C3CCC(C)(CC)O3)=O)C2)cc([N+](=O)[O-])cn1C c1(C(=O)NC(CNC(C(CC)OC)=O)C2CCC2)ccc2ncncc2c1 C1(C(=O)NCC=CCNC(CN(S(CC)(=O)=O)C)=O)CC(=O)N(OC)C1 N1(CC2CC(C)C2)CCC2(CCCN(C(c3cnn(CC4CC4)c3)=O)C2)C1 N1(C(c2n(C)c(Cl)nc2)=O)CCC2(CCCN(C(C34CCCC3OCC4)=O)C2)C1 C=C(C)C(CC(=O)NC(C1(CNC(=O)C(=O)N(C)C)CCCC1)C)OCC C=CCCCC(C(=O)NCc1c[nH]nc1C1CC1)NC(C1CC(C2CC2)=NO1)=O c1(C(N2CC(C(C)NC(=O)CC3CC=CCC3)OCC2)=O)ccc2ncsc2c1 C(C(=O)NCC(C)C(C)O)(C(C)(C)O)NC(c1c(C)oc(CO)c1)=O c1(C(=O)NC2CC(C)N(C(c3cnsn3)=O)C2)cc(=O)cc(Cl)[nH]1 CC(C)C(CCC(=O)NCc1nnn(C)n1)NC(=O)C(C)(C)CCC#N C1(CNC(=O)CSC2CCSC2=O)CCC2(CCN(C(C3(CCF)CC3)=O)C2)C1 C1(c2nnc(-c3cc(C#N)c[nH]3)o2)(C2CCCO2)CCN(C(=O)CSSC)CC1.CO c1(CCC(=O)N(CCCNC(CC=C)=O)CC)cccc(C(=O)OC)c1 C1(CC=C)(C(=O)NC2CN(C(=O)Cn3nccn3)CC2C(F)F)CCOCC1 N1(C(CC2C(C)CCC2)=O)CC2CCCN(C(C34CCOC(C)(C3)C4)=O)C2C1 c1(COC)nc(C)c(C(=O)NCC2CN(CCC(C)OCc3ccccc3)C2)s1 C12(C(N3CC(NC(C4=C(C)CCC4)=O)C(CO)CC3)=O)CC3CC(CC(C3)C1)C2 CC(C)CC(O)C(=O)NCC1CC(CNC(=O)Cc2cccc(C(C)C)c2)C1 C12CCN(CCC1CO)C2=O.CC1(C(=O)NC2(C3CCCO3)CC2)CCOCC1 C1(C(=O)C(=O)O)C2CCN(C(C3CN(C(C)(CO)C4CC4)C3)=O)CC12 N1(C(CC=CC)=O)CCC(NC(c2ccc(NC(=O)NC(C)C)cc2)=O)CC1C c1(OC(C(=O)N(CC(CC)NC(=O)CCC#N)C)C)ccccc1F c1(C(=O)NC2(CO)CN(C(C(CC)O)=O)C2)ccc(Br)c(OC)c1 c1(N(C2CCN(C(C3C4CCCC34)=O)C2)C)ccc([N+](=O)[O-])c(C#N)c1 C(=O)(C1=NNC(C(F)(F)F)C1)NC(CC=C)CNC(C1(OCC)CCSCC1)=O c1(C(=O)NC23CC(CNC(c4ccoc4)=O)(C2)C3)cc2c(F)cc(F)cc2o1 n1(CC)nc(C(=O)NC2CC2NC(=O)COCC2CCC2)cc1C(F)(F)F C1(CNC(c2c(C)nns2)=O)CN(C(=O)CCCN(C)C)CC1O C(=O)(CCC(C)(C)NC(C1C(C)(C)C1(C)C)=O)NC(c1ccccc1)C C#CC1(C(=O)N(C)Cc2ccc(F)cc2)CCN(C(=O)C(C)Cn2cccn2)C1 c1(C(=O)NC2(C)CC(NC(C3(c4ccccc4)CC3)=O)C2)ccc(C2CC2)c(F)c1 N1(C(C2C(C3C(C)C3)C2)=O)CC2CC1CN(C(=O)CN(C)C(c1cccs1)=O)C2 C1(CC)COCCN(C(=O)CC2CN(C(c3ccc(C(C)=O)[nH]3)=O)CCO2)C1 N1(C(c2cn(CC3CCCO3)nn2)C(=O)NC=O)CCCS(=O)(=O)CC1 N1(C(c2ncn(CC)n2)=O)CC(C)C(NC(c2cnn(C(C)C)c2N)=O)C(C)C1 CN1C(=O)C(c2nnc(-c3ccn(C)n3)o2)Cc2ccccc21 c1(COC)nc(NC(=O)C(C)Oc2ccccc2)n[nH]1 C(=O)(CCS(=O)(=O)c1ccccc1)N1C(CNC(C(C(C)C)F)=O)CCCCC1 CC(C)CC(CN(C)C)N=c1[nH]c(=NC(C)c2nc(=N)[nH][nH]2)[nH]c2cc[nH]c12 c1(CC(=O)NC2CC3CN(C(COCC(=O)OC)=O)C2C3)ccc2nonc2c1 c1(NC(C2CC3(CN(C(c4n(C)ncc4Br)=O)C3)C2)=O)ccc2ncccc2c1 C12(C(=O)NCC3N(C(C4CCOC4)=O)CCC3)COCC1CS(=O)(=O)C2 CCCCC(C)CCC(=O)N1CC=CC1(C)C(N1CCCC1)=O C=CC(C)C(C)C(=O)NC1(CC)CCN(C(c2csc(C)c2Br)=O)CC1 N1(C(CC2(C)N(C(CC(C)C(F)F)=O)CC2)=O)CCC(F)(F)C(O)C1 N1(Cc2scc(C)c2)CCC(NC(c2ccc(Br)s2)=O)C(F)C1 C1(CNC(c2ncoc2CO)=O)CN(C(C2CCCC(O)C2)=O)CC1C(F)(F)F N1(C(C2CN(C)C2)=O)CC(O)CC1C(N1CCC(F)(C(N)=O)C1)=O C(C(=O)NOC1CC1)OCCN(C(C(C)C1CCCC1)=O)C c1(C(=O)OC)cc(CNC2CN(C(c3ccccc3)C(=O)OC)CC2F)n(C)c1 c1(NCC2(F)CC(NC(C(C)=C3CC3)=O)C2)ncnc2cccc(C)c12 n1(CC)c(=O)oc2cc(S(=O)(=O)NCc3ccc4c(c3F)OCCO4)ccc12 Cc1noc(C)c1C(N(C(CC(CCBr)CN)=O)CC1CCCO1)=O C1(NC(C(C)OCCC(C)C)=O)CC2CCC1CN2C(=O)C(C)CC(F)(F)F N1(C(=O)Nc2ccccc2OC)CCCC(NC(C(C)OCC2(CN)CC2)=O)C1 Cc1nc(Cl)ccc1CC(=O)NC1COCC1NC(=O)C(C)O c1(NC(C(CNC(CC2C(C)(C)CCO2)=O)CC2CC2)=O)cccc2c1CCC2 CN(C)S(=O)(=O)N(C)CC(=O)NC1CC(C)(NC(=O)CC2(O)COC(C)(C)C2)C1 C1(CCOC)CN(C(=O)C=C=C(C)C)CCN1C(=O)C(C1CCOCC1)F Brc1ccc(C=CCCCN2CCN(C3CCCC3)CC2)cc1 c1(C(C)C(N2CC3CC2C3NC(=O)CCc2cnccn2)=O)ccc(Cl)c(Cl)c1 C1(CNC(C2C(C)OCCC2)=O)CN(C(=O)CC(Cl)Cl)CC12CCC2 c1(N2CCC(N(C(=O)C=CS(C)(=O)=O)CCC)C2)cncc(C#N)n1 C=CCC(CNC(=O)CCCN(C)C)C(=O)N1CC=CC1(C)COC N1(C(C2(COC)CC=CC2)=O)CCCC(N(C)C(C2(C3CCCO3)CC2)=O)CC1 c1(C(N2CCC(CC)C2CNC(C2CCCCC2O)=O)=O)cccc(F)c1C c1(C(=O)NC2(CNC(c3ccn(C)c3)=O)CCCC2)cn2ccsc2n1 C1(NC(CCC(=O)NC)=O)COCCN(C(C2CC(C)=NO2)=O)C1 C1(C(=O)NCCN(C(C2(C(=O)OC(C)(C)C)CCC2)=O)CC)CC2COCC2C1 c1(C(=O)NC2CC3(C(NC(c4c(N)nccn4)=O)C3)C2)cc(F)cc(F)c1 c1(C(N2C(C3(NC(C(CC#C)(C)C)=O)CC3)CCCC2)=O)cc(F)c(C)cc1F CC(CC(C)(F)F)C(=O)NCC1(C)CCN(C(=O)CCc2cnc(O)[nH]2)CC1 C1(NC(C=C(CCN(C)C)Cl)=O)(CO)CCN(C(=O)C(O)CC2CCCC2)C1 C12(C(N(CCCNC(C3(C)C(CC)CCC3)=O)C)=O)CCOC(C)(C1)C2 CN1CCCCC12CCN(C(c1cc(Br)c3ccccc3c1)=O)CC2 c1(C(=O)NCCN(CCCCCC)C(C2CCCOC2)=O)ccc(OC)nc1F c1(OC)nccnc1C(=O)NCC(C)CC(=O)NCC12CCC(CC1)O2 C1(CNC(c2c(C)nn(C(C)C)c2)=O)CCN(C(=O)CC2CC(F)C2)C1(C)C C(=O)(CCCCCO)NC1CCC(CNC(CCNC(COC)=O)=O)C1 c1(N2CCCC(CC)CC2)nc2cc[nH]c2c(=NCc2c(F)cc(F)cc2F)[nH]1 N#Cc1ccc(C(N2CC3CC2CN3C(c2cc(Br)c(O)cc2F)=O)=O)c(Br)c1 c1(OC(C)C)ccc(C(=O)NCCCCNC(=O)CCc2ccc(O)nc2)cc1 N1(C(Cc2ccn(C)n2)=O)CCC(C2CCCN(C(=O)C(C)(C)C)CC2)CC1 c1(C(N2CCC(F)(CNC(CCC=C(C)C)=O)C2)=O)cc(F)cc2cccnc12 CS(=O)(=O)C1CCCN(C(c2cc(=NCc3ccccc3)cc[nH]2)=O)C1 N1(C(c2cnc(C3CC3)s2)C(=O)NC2CC2)CCOc2cc([N+](=O)[O-])ccc2C1 C1(F)(C(N(C)C)=O)CCN(C(c2cccc(-c3cccc(CO)c3)c2)=O)C1 c1(C(N(CCCNC(=O)COC2CCOC2)C)=O)sc2ccccc2c1Cl CCC(CN(C)C)C(=O)NC1(C(=O)NCC(C)NC(N)=O)CCCCC1 C(=O)(CC(O)C(Cl)(Cl)Cl)NC1C2CCN(C(C(c3cn(C)nc3)=O)=O)C21 N1(C(C(C(C)OC)NC(c2cnn(C3CC3)c2)=O)=O)CCCC(CCF)C1 CCCCC(CC)C(=O)NCC1(C)CCN(C(=O)C(C)(C)C2CCOCC2)C1 N1(CC)CCOCC1C(=O)NCCC(O)C(=O)NCCn1cnccc1=O c1(C(=O)NCCCCCN(C(C(COC)(C)OC)=O)C)cnc2nc(C)oc2c1 c1(-c2c(OC)cccc2)nc(=NC2CC(NC(=O)C3=CC4(CCOC4)C3)C2)s[nH]1 C1(COC)(NC(=O)C(O)C2CCCC2)CCN(C(C2(S(N)(=O)=O)CCC2)=O)CC1 c1(CC)nccnc1C(=O)NCC(c1ccccc1)NC(=O)C(F)CC N1(C(C2OCCN(C)C2)=O)CCC2CN(C(c3cnn(C4CCC4)c3)=O)CC2C1 Cc1cccc(N2CCC(OC(=O)CC3CC(C)OC3C)C2=O)c1 N1(CC(C)C)CCC(CC2CCCCC2)C1.C12CC(C1)CNC2=O C1(CN=[N+]=[N-])CCCN(C(C2CCCCN2C(=O)C=CC2CCCC2)=O)C1 CN1CC(C(=O)N(C)CCNC(c2cccn2C)=O)NC1=O CON(CCCO)C(=O)C1(NC(=O)COCC(C)(C)C)CC1(C)C c1(C(N2C(C)(C(=O)OC)CC2)=O)[nH]c(C)c(C(=O)NCCCn2ccnc2)c1C N1(C(c2c(CC)con2)=O)CCC(C)N(C(c2conc2C)=O)CC1 Cc1cncc(C(=O)NCC2CC(NC(=O)Cn3ncn(C)c3=O)C2(C)C)c1C N1(C(Cn2c(C)cc(C)n2)=O)CCCC12CCN(C(C1CCCN1C(C)C)=O)C2 C1(NC(CC2(C)CC2)=O)CC2COCC(C1)C2NC(=O)CCCOC1CCCC1 Cc1ccc(C)c(C(N2CC3(NC(C4CCCOC4)=O)CCC2C3)=O)c1O N1(C(C=CC=CC)=O)CC(C(=O)Nc2ccc(C(F)(F)F)nc2)CC(F)C1 c1(C(=O)NC2CCC2CNC(=O)C(O)c2ccsc2)ccccc1N1CCCC1 N1(C(C(CCCC=C)NC(=O)C(C)CC(=O)OC)=O)CCc2oc(C)nc2C1 Cn1cc(C(=O)NCC(CNC(c2cccn2C2CCCC2)=O)CO)nn1 c1(C(=O)NCC(Cc2ccccc2)CO)ccc2cccc([N+](=O)[O-])c2n1 N1(C(COCCC=C)=O)CCCC(N(C(=O)CN(C(=O)COC)C)CC)C1 C(=O)(CCCCCC#N)N.C1(Cn2cc(COCC)nn2)(CO)CCOCC1 C1(C(=O)NCCCCSC)N(C(C2CCC(F)(F)C2)=O)CCC1(C)C CC1(C)CC(Nc2ccc([N+](=O)[O-])cc2)CN(C(c2ccc3scnc3c2)=O)C1 N1(C(c2cn(CC=C)nn2)=O)CCOC(C(=O)Nc2ccsc2SC)CC1 N1(C(c2n(C)c3c(c2)occ3)=O)CC(CO)C2(C1)CN(C(C1C=CCCC1)=O)C2 C(=O)(CCC(=O)N1CCC(C(C)NC(=O)Cn2cnnn2)C1)Nc1nnc(C)s1 c1(CNC(C23CC(NC(C45COCC4C5)=O)(C2)C3)=O)ccc(F)cc1OC(F)F c1(C(=O)NCC(CC)NC(C2(C#N)CC3CC3C2)=O)c(F)ccc(C)c1F c1(CCCC(c2n(CC)nnn2)NC23CC=CC(C2)OC3)c(F)cccc1F c1(NC(=O)OCC)nnc(S(=O)(=O)N2CCN(C(c3nc(C)c(C)o3)=O)CC2)s1 CCC(CC)C(C(=O)N1CC(NC(c2nc(O)c(C)s2)=O)C(C)(C)C1)OC c1(SC(CC)C(=O)OCCCCc2ccccn2)cccc(Br)c1 c1(C(N(CC(CC)NC(c2ccc(Br)o2)=O)C)=O)ccc(-c2nc[nH]n2)cc1 C(C(C(C)(C)C)NC(C1NC(=O)CC1C)=O)NC(C1C(C)(C(C)C)C1)=O CCCCC(CC)CCCN(C)C(=O)NC(c1cccs1)CN1CCOCC1 N1(C(C2CCCN(CC(C)=CC)C2)=O)CCCN(Cc2ccc(F)nc2F)CC1 c1(CC)ccc(C(N2CC(NC(=O)Cc3nc[nH]n3)C2)=O)cc1Br c1(C(N2C(C(=O)NCCc3n(C)cnc3)C=CC2)=O)cccc(CO)c1 N1(C(CC(C)(C)OC)=O)CCOCC(C)(CNC(c2cncc(C)n2)=O)C1 c1(C(N2CC3C(CNC(C4C(C)C4C)=O)(C3)C2)=O)occ2c1CCC2 c1(C(N2CC(NC(=O)CCc3nc(O)n[nH]3)C2)=O)cc2c(o1)CCCNC2=O c1(C(=O)NCCOCCNC(CC(=O)NCC#C)=O)ccc(C(F)F)cc1 N1(C(=O)Nc2ccc(OCCC)cc2C)CCC(CO)C(F)(F)C1 c1(NC(c2nnnn2C)C2(CSC)CCC2)cccc(-c2ncco2)c1 c1(C2(C(=O)NCC(C)N(C(=O)COC3CC3)C)CCCC2)ccc([N+](=O)[O-])cc1 C1(C(=O)NCC(C)CNC(c2cnc(S)[nH]2)=O)CC2(C1)CC(O)C2 C1(CC(=O)N(C)CC2CCCN(C(=O)C(C)(F)F)C2)CC2CCC(C1)C2 C(CC(=O)NN1CCCC1C(=O)NCC1CCN(CCF)C1)OC(C)(C)C C(=O)(C(CC(C)C)NC(=O)CC(C)N(C)C(c1cc(F)n(C)n1)=O)NC c1(C(=O)NC(C)CCCCNC(c2cc(Br)no2)=O)cccn2cnnc12 C(=O)(CC(CC)CCC)NCC(CNC(c1cnc(CCCC)s1)=O)C N1(C(C(C2CC2)OCC)=O)CCCN(C(=O)C(C)C(C)C)CCNC1 CCC(C(=O)NCc1cn(C2CCN(C(C3(C4CC4)CC3)=O)C2)nn1)C(C)C c1(C(=O)NCC2C(NC(c3cc(OC)nn3C)=O)COC2)cnc2n1CCS2 CCC(CC)C(C(=O)NC(C1CCCN1C(c1sccc1C#N)=O)(C)C)OC N1(C(N2C(C)C(N3CCOCC3)CC2)=O)CCC(S(=O)(=O)c2ccccc2)C1 C1(CC)CCCCC1C(N1CCC(C(C)(C)C)(CNC(=O)C(C)CSC)C1)=O C(CC(CNC(C1C=C(C)CS1)=O)NC(=O)CNS(C)(=O)=O)OC N1(C(c2ccc(N)cc2Sc2c(Br)cnc(C)n2)=O)CCC2COCC2C1 N1(C(C2=CC(C)(C)C2)=O)CCC2(CC1)CC2NC(=O)Cc1cnc2cccnn12 C1(F)(CNC(CCSCC(C)C)=O)CCCN(C(C2CC(C)(C)CO2)=O)C1 CCCCCCCC(=O)N(C)CC1CCCCN1C(C1CC(=O)CCO1)=O c1(OCC)ccc2c(c1)CC(C(=O)NCC#CCNC(=O)C(C)(CC)OC)CO2 C1(C(=O)NCC(c2ccccc2)(C)C)CCC(Cn2ccnc2)C1 c1(C(=O)NC2(CNC(c3cc(CC)[nH]n3)=O)CCCCC2)ccc2nn[nH]c2c1 c1(C(C(=O)NC)N(C(CC(=O)OCC)C2CCCCC2)C)ccc2ncsc2c1 C(=O)(C#CC1CCCOC1)N1C(CNC(C2(CCCC)CC2)=O)COCC1 N1(C(CCc2n(C)ccc2)=O)CC(O)CCC1C(=O)NCC1OC(=O)CC1(C)C N1(C(C(COC)O)=O)CCn2ncc(CNC(c3cc(Cl)ccc3Cl)=O)c2C1 C1(NC(c2ccc(-n3cccc3)cc2)=O)CCCC(NC(C23CCC2CC3)=O)C1 CC1(C)CC1(C#N)CNC(C1(n2cc(Br)nn2)CC1)=O C1(C(N2CCC(F)(CNC(CP(C)(C)=O)=O)C2)=O)CCCCC12OCCO2 c1(CCC)cc(C(=O)NC(C2CCCN2C(C2C=CCCC2)=O)C)n(C)n1 O=C1NC(C(=O)NCC#CCNC(c2sccc2-n2cccc2)=O)CO1 CCC(CCO)C(C)NC(=O)NC1C2CCOC2C1(C)C O=C(C#CC1CCCC1)NC1COC2(C1)CN(C(=O)COc1cccc(Cl)c1)C2 N1(C(C2C(C)CCCC2)=O)CCC(C)C(CNC(C2CCC3CC3C2)=O)C1 c1(CN2C(C(N3C(C)(C(=O)OC)CCC3)=O)CC(O)C2)cccc(Br)c1O c1(C(N(CCNC(C2CC(C)(F)C2)=O)CC)=O)ccc(NC)c(F)c1 c1(OC)ccc(Br)c(CN2CC(CNC(=O)CCc3ccccc3)C2)c1F c1(NC(CN(C(CCNC(=O)OCC)=O)CC2CC2)=O)cnc(C)cn1 O=C(CC1CCOc2ccccc21)OCC1(c2ccccc2)CC1(F)F C1(CC)CCC(C(=O)NC(C)C=CC(=O)NCC2(C3CC3)CC2)O1 CN1C2CCCC1CN(C(c1cnc(C3CCC3)[nH]1)C(=O)NC1CC1)CC2 CC1=CCN(C(C2(NC(=O)CC3CCCC3C)CC(F)(F)C2)=O)CC1 C1(C(N(C(C)CC(c2ccc(Cl)cc2)=O)C)=O)CCOC(C)(C)C1 c1(C(=O)NCCC(=C)CNC(c2ccc(C)n2C)=O)c(Cl)cc(C#N)cc1Cl N1(C(=O)Cc2cnsc2)CC2=C(C1)CN(C(=O)Cc1ccc(Cl)cc1F)C2 N1(C(c2cn(CC=C)nn2)=O)CCC(NC(c2sccc2F)=O)C12CC2 c1(C(=O)NCC(N2CCN(C(C3C(C)CCC3)=O)CC2)=O)cnc(Cl)cc1N c1(NCC(S(=O)(=O)NC)C)ncccc1S(=O)(=O)N(C)Cc1csc(C2CC2)n1 C1(CC)CCCN(C(C2CC(C)(C)CO2)=O)C1C(=O)N(C1COCC1O)C N1(C(COCC)=O)CCN(C(c2cccc(C(F)F)n2)=O)CC1c1nccn1C C(=O)(C1CCCc2c1ncn2C)N1CC(CNC(CCOC)=O)CC12CCC2 c1(CNC(C2C(C)C2)=O)cnc(O)c(F)c1.C12CC(F)(C1)CNC2=O.C1(=O)CCN1 O=C1NC2(CCN(C(=O)NCCCNC(=O)C3CC3)CC2)CO1.C12CCCCN1C2=O c1(OC)ccc2[nH]c(=O)c(C(=O)NCCc3cc(C)sc3C)cc2c1 c1(NC2CC(F)(CNC(=O)Cn3ccc([N+](=O)[O-])n3)C2)ncnc2c1CCO2 C1(CNC(c2ccc(C)nc2O)=O)CCC2(CN(C(=O)C(C)(C)C(C)(F)F)C2)O1 C1(C(=O)NC(C2CC(NC(=O)CC3CC3)C2)C)C=CCC1.c1nc[nH]n1 n1(CC)cnc(C(=O)NCC2C=CC(NC(=O)CC=CC(C)(C)C)C2)c1 CC(CCCNC(=O)CCN(C)CCO)NC(=O)CC1CCSC1 N(C1CCOc2c(Cl)cc(Cl)cc21)C(C(=O)Nc1cccc(Br)c1)=O N1(C(C(CC)C(C)C)=O)CCC2(CC1)CC(NC(C1CCCCS1)=O)C2 C1(C#N)(C(=O)NC(C(C)NC(Cc2c(C)cnn2C)=O)C(C)C)CCOCC1 c1(CC)ccc(C(=O)NC2CC(NC(c3nc(C)ncc3Br)=O)C2)c(OC)c1 O=C(C(Cc1cn(CCCO)nn1)CC(F)F)NC1(c2ccsc2)COC1 Cc1cc([N+](=O)[O-])nn1C(C)C(=O)N(CC(=O)O)C1CCC1 N1(C(c2c(CC)c[nH]n2)=O)CCOCC(NC(c2oc(C3CCC3)nc2C)=O)C1 C(=O)(C(C)C(C)NC(=O)CCOC)N(CC=C)C c1(C(=O)NCC(CCC)NC(=O)CC2OCCC2(C)C)cc(C(C)C)nn1C C1(OC)(CNC(=O)C(C)SC(C)C)CN(C(C2CCN2S(C)(=O)=O)=O)C1 C(=O)(C(O)(C(F)(F)F)C1CC1)N1CCN(C(C(CC)c2cccnc2)=O)CC1 C1(NC(COCC=C)=O)CC(NC(=O)C(C)Cc2ccnn2C)CC1O c1(C(CC)=O)ccc(C(=O)NCC(C)(C)NC(=O)C(c2cncc(F)c2)C)cc1 c1(C(N(C)CC2N(C(CCCC)=O)CCC2)=O)c(F)ccc(C)c1Cl N1(C(C(CC(=C)Cl)NC(C2CCC(C)CC2)=O)=O)CCC2(CCC(O)C2)C1 C1(NC(c2c(CNC(C(C)CC(F)F)=O)nccc2)=O)CC12CCCCCC2 N1(C(C2(OC)CCOCC2)=O)CCOCC(CNC(C2CC(C(C)C)=NO2)=O)C1 Cc1nc(C)c(CNC(C2CCCC2CNC(=O)CC2CCOC2C)=O)[nH]1 c1(SC)ccc(Br)cc1C(=O)NCC1C=CCN1C(c1cccnc1)=O Cc1nc(O)ccc1C(N1CCC(C)CC1C(=O)Nc1c[nH]ccc1=O)=O c1(N2CC(c3scc(C)n3)OCC2)nc(=NC(C)CCO)[nH]c2c1ncn2CCO Cc1cc(C(=O)NC2(C3CCN(C(=O)C(C)N(C)C)C3)CC2)c(Cl)cc1Cl C(N=C(NCC1CC1)NC1CCN(Cc2ccccc2)CC1)C1C(C)C1 CCC(C)CCCCC(=O)N1CCCC(Cc2cn(Cc3cnns3)nn2)C1 CCC(CCOC)C(=O)N1CCC(C(N2Cc3cccc(Br)c3C2)=O)O1 c1(CNC(C2CCN(C(=O)Cc3cncnc3O)C2)=O)ccc(Cl)cn1 N1(C(c2cn(C)c(O)n2)=O)CCN(C(=O)Cc2cnc(C3CC3)[nH]2)C2CC12 CC1CN(C(c2cccc(Cn3cc(COCCO)nn3)c2)=O)CC(C)(C)C1 N1(C(C2(NC(c3cc(CSCC)on3)=O)CC(F)(F)C2)=O)CCCC(C)(C)C1C C1(C(=O)NCCC)CN(C(C2CC3(CC3)CO2)=O)C2(CCC2)C1 c1(C(=O)NCCOC(C)(C)C)cnc2c(c1)CCN(Cc1cnc[nH]1)C2 c1(CC)ncccc1C(=O)NCCOCC(=O)NC1(CCCC)CC1 c1(C(N2C3CC(CNC(c4c[nH]c(=O)o4)=O)C(C3)C2)=O)n[nH]c2ccc(F)cc12 N1(C(CN2CCN(CC)CC2)=O)CCN(C(c2cc(OC)cc(F)c2)=O)C(C)C1 c1(C(=O)NCC(C2CCCCC2)NC(=O)CCF)sccc1Cl N1(C(c2c(CC)nc(C)[nH]2)=O)CC(NC(=O)CN2CCCCC2=O)C2CCCC12 Cc1nccn1C(C)C(=O)N(C)CCNC(=O)Cc1nccn1C C(=O)(C(CNC(=O)CCc1cn[nH]c1)N(C)C)NC(C1CCOCC1)C#C NS(=O)(=O)C1(C(=O)NC2CCCN(C(=O)CCCCc3cnc[nH]3)CC2)CCC1 c1(C(=O)NC2CC(NC(c3nc(C(C)(C)C)oc3)=O)C2)ncc(Br)cc1N Cc1cc(C)n2nc(COC(c3csc(Cl)c3)=O)nc2n1 c1(C(=O)NC2CCCN(c3nccnc3Cl)C2)n[nH]c2cccnc12 c1(C(=O)NC2CC(CNC(=O)CC3CC3(Cl)Cl)C2)cccc2c1CCO2 N1(C(c2c(CC)cc[nH]2)=O)CCCCCCC1C(=O)NC1COCC1OC C1(=O)CCCCCC(c2nn[nH]n2)N1.C(C1CCCc2n[nH]cc21)c1n(C)nnn1 N1(C(CNC(=O)NC)=O)CC2CC(Nc3ncc(Cl)cn3)CC1C2 C#Cc1ccnc(C(=O)NCCC(O)CNC(=O)C(C(C)(C)C)SC)c1 Cc1cc(CNC(C2C=CCS2)=O)oc1C(N1CCC(c2ccco2)C1)=O C12(C(N(CCNC(c3csc(COC)n3)=O)CC)=O)CCCC(C1)OC2 C1(CNC(c2cc(C)on2)=O)CN(C(c2ccc(S(N)(=O)=O)o2)=O)CCC1(C)C CCCC(C)(O)C(=O)N1CCC(C)(CNC(c2cc(F)ccc2C(C)C)=O)C1 C=Cc1cc(C(=O)N(C2CCCCN(C(=O)C3=CCCCC3C)C2)C)cc(F)c1 CC(C)CC(C(=O)C(=O)CC1CC2(CC2)C1)N.C1(C(N(CCN)C)=O)CC1C CC(C)C(O)CC(=O)NC(C)CC(=O)NC(c1ncccn1)(C)C C1(OC)C(C)OCCN1C(=O)CCCC1(c2cn(-c3cccc(Cl)n3)nn2)CC1 C12(CNC(=O)CSCC3CCCCO3)CCC(CC1)N2C(C1CC1F)=O CCC(C)(F)C(=O)N1CCC(NC(=O)Cn2cc(-c3ccccc3)nn2)C1 C1(CC(C)NC(CC(=C)C)=O)CC2CCC(C1)N2C(=O)CSc1ccc(C)cc1 Cc1[nH]c2cccnc2c1CNC1CCN(CCC(C)C)CC1 N1(C(C=Cc2c(C)nccc2)=O)CCC2(CC1)CN(C(C1CC3(CCC3)C1)=O)C2 N12CC(F)(F)CC1NC2=O.c1(NCc2c(OCC)cncc2)ncc(Br)nc1CO C(=O)(CCCCCN(C(=O)CC1(OCC)CC1)C)N1C(CCC)CCC1 Cc1cc(CCNC(=O)C(C)CNC(c2scnc2Cl)=O)n[nH]1 C1(NC(C2C(CN(C)C)C2)=O)COCCC1NC(c1ccc(F)cc1)=O C12(C(=O)NC(C)(CNC(c3cnn[nH]3)=O)C3CCC3)CC(CC(F)(F)F)(C1)C2 c1(C(=O)Nc2ccc(-c3cccc(O)c3)cn2)c[nH]c2cc(Cl)ccc12 c1(OC)ccc2c(c1)CCC(C(=O)NCCOCCNC(C1CCCC1O)=O)C2 c1(NCc2c(CNC(=O)Nc3ccc(Br)cc3)[nH]nn2)ccc(C(F)(F)F)cc1Cl c1(CNC(CC(CC)CN(C)C)=O)cc2n(n1)CCN(C(=O)COCCOC)C2 C=CC(C)C(=O)N(C(C)CC(=O)NCC(CSC)OC)C C1(C)(C(=O)NCC(CNC(=O)C(c2cnccc2C)(C)C)OC)CC2CC2C1 N12c3ccccc3CC1OC2=O.N1(C(C)(C)C)CCC(O)C(Cn2ccnn2)C1 C(C(C)(C)CNC(c1cnc(-c2ccoc2)s1)=O)N(C(C(=O)NC(C)C)=O)C C(CC(C)(C)C(=O)NCC(CO)NC(c1cccc(-c2nc(=O)o[nH]2)c1)=O)OC N1(C(c2n(CC)ccn2)=O)CC(=O)N2CCCC2C1 C12(CNC(c3c(C)cnn3C)=O)CCC(CC1)N(C(=O)C(CN(C)C)N(C)C)C2 N(C1COc2cc(Cl)ccc21)C(=O)CSCc1ccccc1Cl S(=O)(=O)(c1ccc(CN)s1)N1CC(C(N(CC)Cc2noc(C)n2)=O)C(O)CC1 C(=O)(N(C)OC(F)F)C1CC(NC)C1.c1(CC2CC(CC=O)C2)ccccc1 CC1CC(CNC(C2(C(F)F)CCCO2)=O)CCN1C(c1ccc(Cl)nc1N)=O N1(C(c2c(CC=C)cccc2)=O)CCC(F)CC1C(=O)NCCCP(C)(C)=O C1(C(N(C)CC2(O)CN(C(CNS(NC)(=O)=O)=O)C2)=O)CCCC1(F)F N1(C(C=CC=CCC)=O)CC2(CCCC2NC(C2Cc3nnc(C)n3C2)=O)C1 C1(CC=C)(NC(=O)C=CC2CC2)CN(C(c2cnccn2)=O)C1 c1(C(=O)NC(c2cc(Cl)ccc2Cl)C)ccc(-c2ccncc2)nc1O N1(C(CN(C(=O)C(C)CC#N)CC)=O)CCCOC(C(C)C)C1 c1(C(=O)NCCCC(CCO)C(=O)O)cccc2cc(F)ccc12 C(=O)(C(C)CC(C)C(C)=O)NC(COCC)C(=O)NCc1coc(C)c1 c1(C(N(CC(C)NC(=O)C(O)Cc2ccccc2)C)=O)cccc2c1NCCC2 C1(NC(c2[nH]cc(CC)c2)=O)CCN(C(=O)Cc2ccccc2O)C1(C)C c1(CC)cc(Cl)c(NC(C2CCNC(C(=O)NC)C2)=O)cc1Cl C1(NC(CCc2c(C)nn(C)c2)=O)CN(C(=O)CC2CNC(=O)C2)CC1(C)C N1(C(CN(C2CCOC2)C)=O)C2CCC1CC(NCc1ccccc1S(C)=O)C2 C1(N(CCC)C(C2CC3CC(C2)C3)=O)CCN(C(=O)C(C)SC(C)C)O1 C(=O)(C(F)C(F)(F)F)N1C(CNC(C(C=C)C)=O)CCC1 C(=O)(C(COC)CC(C)C)N1CCC(O)(CCNC(CC(C=C)(C)C)=O)C1 N1(C(c2cc(OC)cc(Cl)c2)=O)CCC(F)(F)C(COC(=O)CC(C)(C)C)C1 Nc1cc(C(N2CC(CNC(c3ccccc3Br)=O)C3CC23)=O)cnc1N O=C(C1=CCCOCC1)NC1CC(NC(c2ccc3c[nH]nc3c2)=O)C12CCC2 c1(C(=O)OC)nc(C)oc1NCC1C(CNC(c2cc(CCCCC)[nH]n2)=O)C1 N1(C(C2(O)CCC(C)CC2)=O)CCCC(C2CC2NC(C2CC2(C)Br)=O)C1 Cc1nnc2c(C(=O)NC3COCC3NC(C3CCOC(C)(C)C3)=O)cccn12 c1(CNC2CN(C(COc3ccc(C)cc3)=O)CC2F)ccc([N+](=O)[O-])cc1F c1(C(N(CC(C(C)C)C(C)C)CCC)=O)c(Cn2cc(CN)nn2)nn2c1CCC2 Cc1ccccc1C(C)CC(=O)NC(C)(C)CN(C(=O)CC1CCCO1)C N1(C(COCCC=C)=O)CCOC2CCN(C(c3cccc(=O)o3)=O)CC12 c1(OCCNC(c2nc(-c3cn(C(C)C)nc3)sc2)=O)c(F)cccc1F Cc1cn2c(CC(N3CCOC(C(=O)NC4(c5cnn[nH]5)CC4)C3)=O)csc2n1 C(=O)(C(C)(C)CNC(Cc1ccccc1)C(=O)Nc1cc(C)sc1C)OC C(CO)(C(C)(C)CO)NC(C(CSC)(C)NC(c1cncnc1C)=O)=O CCC(CC)CCCC(=O)NCCNC(C1(c2ccncc2F)CCC1)=O N1(C(C2CCC(=C)CC2)=O)CCC(NC(=O)C(C)(C)c2ccc(Cl)s2)C(CC)C1 c1(C(=O)NC(CC)CNC(=O)CCC#N)ccc(C2CCC(=O)N2)cc1 CC(C)C(O)C(F)(F)C(=O)NCC1CCCN1C(=O)CCCC(F)F CCCCS(=O)(=O)CC(=O)NC1CC12CC(NC(=O)CNC(=O)NC)C2 C1(NC(C(c2cnn(C)c2)NC(CCN(C)CC)=O)=O)CC=C(C)CC1 C(=O)(CCCCCc1nn[nH]n1)NC1CCN(CCOC)C1 c1(C(=O)NC2CC(C)(CNC(c3nscc3Br)=O)C2)coc(C#N)c1 c1(C(=O)O)ccc2c(c1)N(C(c1ccc(Cn3cc(Br)cn3)o1)=O)CCOC2 CC1CCC(CC(N2CC(CC(F)C(=O)NC(C3CC(F)(F)C3)C)C2)=O)OC1 c1(C(=O)NCCN(CCC)C(C2(C)CCC(C)(C)CC2)=O)cnc2ncccn12 CC1CN(C(=O)CCc2cscn2)CC1CNC(c1cccc(C2CC2)c1)=O CC(CC(=O)OCC1(Oc2ccccc2)CC1)CC(F)(F)F c1(N2CCCC(CC#N)C2)nc(=N)[nH]c(=NC2CC2c2ccsc2)[nH]1 c1(CCNC(C2(CC)CC2)=O)cncc(C(=O)NCC2=NOC(C)C2)c1 C1(NC(c2n(C)ncc2Br)=O)CN(C(c2ccnn2CC#N)=O)C(C)(C)C1 C1(NC(C(c2c(C)cccc2)C2CCNCC2)=O)CCC2(CC1)CNC(=O)C2 N1(C(C2N(C)C(=O)OC2)=O)CCC(C)(C)C1CC(=O)NCC1CC12CCCCC2 N1(C(CN2CCC(C(N)=O)CC2)=O)CCC(NC(C2CC2C2CC2)=O)C(C)(C)C1 C1(C(=O)NCC2(CN(C)C(c3csc(C(C)(C)C)n3)=O)CC2)CC(C2CC2)C1 c1(-c2cccc(OC)c2C)ccc2cc(C(N3CCC(C)C3)=O)cn2c1 C1(C(N2CC3C(CNC(c4[nH]cc(CC)c4)=O)(C3)C2)=O)CS(=O)(=O)CCO1 C1(NC(CSCC#C)=O)CN(C(=O)CCSc2ccccn2)C2CCCC12 c1(CC)ccc2ccccc2c1CNC(=O)Cc1ccc(O)cn1 N1(Cc2ccc(C)o2)CCC2(CC2C(=O)O)C1 CCCC(O)(CCC)CC(=O)NC1(C)CCN(C(c2conc2COC)=O)C1 Cc1nc(O)ccc1C(N1CCCC(N(C)C(C2CC3(CCC3O)C2)=O)C1)=O C1(C(=O)NC(CCNC(c2c(SC)csc2)=O)(C)C)CC2(C1)CC2(F)F C1(NC(C2C3CCCCC23)=O)CCN(C(c2c[nH]c(=O)cn2)=O)C12CCC2 c1(OC)c(NC(=O)C(C(C)(C)O)NC(c2sc(O)nc2C)=O)cccc1F n1(CC)cnc2c(NCc3cnc(C)o3)[nH]c(=NCCCc3ccco3)nc12 O(P(C)(=O)CNC(C1CC(C)CN1C(=O)CCC1CCOC1)=O)CC N1(C(CCC(C)C)=O)Cc2ccccc2C(NC(C2CCC=CCCC2)=O)C1 N1(c2cc(NCCCOCCOC)nc(C)n2)CCc2ncnc(C)c2C1 n1(C(C)C)nncc1C(=O)NCC1CCN(C(=O)C=CC2CCCC2)C1 C(=O)(CC(O)CC(C)(C)C)NCc1c(C(N2CC(OC(CC)=O)C2)=O)[nH]cc1 C1(C(=O)Nc2c(CC)cccc2)CCN(C(=O)CCCCCNC(C)=O)C(C)C1 N1(C(C2N(CCC)CCC2)=O)C2CCC1C(CNC(c1ccncc1F)=O)C2 CCC(C)(C)C(O)C(=O)NCc1cc[nH]c1C(=O)N(C)CC12CCC(CC1)C2 CC(CN=C(NCc1ncccc1F)NCC1CC1)Oc1ccc(CO)cc1 CC1CNCCN(C(=O)NC2(CO)CCC(C)(C)C2)C1 N1(C(C2CC(OC)C2)=O)CCCCC1CN(C(=O)CCCOC)C C(CC(C)C(=O)N(C1(C(N2CCSCC2C2CC2)=O)CC1)C)=CCC c1(CNC(C(CCC)CC2CCCC2)=O)cc(F)c(C(=O)O)c(F)c1 C(CNC(C1CCN(C(=O)C(C)C)CC1)=O)(C(C)C(C)C)NC(CCOCC)=O c1(C(=O)NC(CNC(COC)=O)C(C)C)ccc(O)cc1F C(=O)(CCCCCN(C(=O)C=CC1CCOCC1)C)NC(C=C)C(F)(F)F c1(C(N2C(CNC(C=CC(=O)OCCCC)=O)CCC2)=O)cccc(C#N)c1 S(=O)(=O)(c1cccc(Cl)c1F)N1CC(OC)C(NC(C2CCCCO2)=O)CC1 N1(CC)CCC(NC(C2CCN(C(=O)CCc3nc(C)no3)CC2)=O)C1=O C1(NC(CNC(=O)CN(C2CCCC2)CC2C=CCC2)=O)CCCC1CCCO Cc1c(CC(=O)NC(C)C(C)NC(c2ncn(C)n2)=O)ncn1C N1(C(c2c(C)scn2)=O)CCCCC(CNC(c2ccc(=N)[nH]n2)=O)C1 n12cc(nn1)NC(=O)C2.C1(C(CC(N)=O)NC(CC2CN(C)C2)=O)CCCCC1 C(=O)(C1=C(C#N)CCC1)N(CCCNC(c1cc(C)n(C)c1)=O)CC c1(CC=C(C)C)cccc(OCCOC(=O)Nc2[nH]cnc2C)c1 CCC(CC)C(F)C(=O)N(C1(CC(=O)N(C2COCC2(C)C)C)CC1)C N1(c2c(C#N)ccc(N3CCCC3)n2)CCc2cc(F)ccc2C1 CC(CC(=O)N(C)CC1(CNC(=O)COC2CCC2)CC1)P(C)(C)=O CN1CC2CCC(C1)N2C(c1c(O)ccc(F)c1F)C(=O)OC1CCCCC1 C1(CC)(NC(c2ccoc2C)=O)CCN(C(c2cccc(N)c2N)=O)CC1 N1(C(c2cc(C)ns2)=O)CC(NC(c2ccc3scnc3c2)=O)CC12CCOC2 N1(C(C(CC=C)CNC(C2CC2OC(C)=O)=O)=O)CCC(C)(O)C(O)C1 C12(NC(CC(C(C)C)OCC)=O)CC3CCC(C1C2)N3C(c1ccc(Cl)s1)=O Cc1ccc(N(C)C(C2CCN(C(c3cnc(O)o3)=O)C23CC3)=O)cc1F C12(C(N3C(Cn4cc(CCN(CC)CC)nn4)C=CC3)=O)CCC(C)(CC1)OC2 N12CCOC(C1)C(=O)N1CC3C(C3C1)CC2=O.C12(CC)CC(C1)C2 c1(C(=O)NC(C(=O)NCCOCCC)Cn2cccn2)cncnc1C C1(NC(C23N(C(c4cccc(C)c4O)=O)CC(C2)C3)=O)CCN2CCCC2C1 N1(C(COCC)=O)CC2CCC1C(NC(c1ccc(NC(C)C)cc1Cl)=O)C2 C(N=c1[nH]cnc(Cl)c1C#N)C1CCCC(NC(CC2N(C)C(=O)CC2)=O)C1 CP(C)(=O)c1cccc(NC(=O)C(=O)NC2CC3CCC2CC3)c1 N1(C(C(C)CC(F)(F)F)=O)CCC2CN(C(c3cc(O)cc(O)n3)=O)CC2C1 c1(C(=O)NC(C)CN(C(=O)CC2COCCO2)C)cc(Cl)c(F)c(Cl)c1 C1(C(=O)NC2CC3N(C(CC(=O)OC)=O)C(CC3)C2)CC(F)(F)CCC1(C)C N1(C2(NC(=O)CO)CC(NC(C3N(N=O)CCCC3)=O)C2)CCCCCCC1=O N1(C(C(c2ccc(OC)cc2)=O)=O)CCC(O)C(NC(=O)CCCC(N)=O)C1 N1(c2cccc(C)n2)CCCC(C(=O)NCc2cc3c[nH]nc3s2)CC1 Cc1nc(-c2ccccc2)sc1C(=O)NC(C)CNC(=O)COc1cnn(C)c1 c1(C(=O)NCCC(C)N(C(COCC=C)=O)C)cnc(OCC)c(C)c1 CC(CC(=O)N1CC(CNC(c2ccc(C3CC3)nc2O)=O)CC1C)C(F)(F)F C(=O)(C(C(C)(C)C)O)N1CCC(NCCC)C1.c1(C(=O)OC)ccccc1SCC c1(NC(CNC(C2C(CCC)CCC2)=O)=O)cn(CC)nc1C#N C(=O)(CCCCCOC)N1C(CN(C(C23CCN(CC2)CC3)=O)CC)CCC1 C1(NC(c2c(C)nn(C)c2Cl)=O)CC2(CCCN(C(=O)C(O)C3CCC3)C2)C1 c1(SCC)ccccc1C(N1CC2C(N(C(=O)C(C(C)C)OCC)C)C2C1)=O C1(O)(C(C(=O)NCCC(O)C2CCC2)NC(C2CCS2(=O)=O)=O)CCCCC1 c1(C(=O)NCc2cccc(CNC(c3ccc(F)nc3)=O)c2)cc(O)ccc1Cl Cc1ccc(OCC(=O)NCC23CCC(C2)N(C(C2OCCO2)=O)C3)cc1C C(=O)(C(CC(C)C)NC(=O)C=CCC(C)(C)SC)N1C(CC)CCCC1 N1(C(C2C(C)(C)C2(C)C)C(=O)NCCSC)CCCC(CCO)CC1 c1(C(=O)NCCOCCNC(C(C(C)C)n2cnnn2)=O)cnc2[nH]c(O)nc2c1 N1(C(COC)=O)CCC(C2(O)CCN(C(=O)CC3COC4(CCC4)CO3)C2)CC1 N1(C(CC(C)SC)=O)CC2(C1)CN(C(c1ccn3c(C)cnc3c1)=O)CC2CO C1(OCCOC)COCCC1NC(=O)N(C1CCCN(C(C)C)C1)C C1(NC(C=Cc2ccc(C3C(C)C3)o2)=O)CCN(C(=O)CO)CC1(C)C C(CC(C)(C)CC(=O)NC1CN(C(C2CC(OC)C2)=O)CC12CC2)OC C1(COC)(NC(C2CC3CC3C2)=O)CCN(C(=O)C(C)CF)CC1 C1(CC(N2C(COC)COCC2)=O)CCCN(C(C2SCCS2)=O)CC1 N1(C(CCCCC)=O)CCN(C(c2c(C)nsc2NCCC)=O)CC1CCC Cc1nn(Cc2sccc2Br)c2sc(C(=O)N(C)Cc3ccccc3)cc12 c1(C(=O)OC)ccc(C(=O)NC(C)CCCNC(c2cc(Br)no2)=O)[nH]1 Cc1nsc2ncc(C(=O)NC(C)C(C)NC(=O)C(C)(C)CC(F)(F)F)cc12 C1(NC(C2(COC)CC2)=O)CCCN(C(c2cnn(CCO)c2N)=O)CC1 CCC(C)C(CC(=O)NCC1CCC2(CC2)C1)NC(c1csc(C)n1)=O N1(C(COCCC=C)=O)CC2CC(C(N3CCCC(CC(C)C)C3)=O)(C2)C1 C(=O)(C(F)CC(C)(C)C)N(C)CC1N(C(c2cncc(C)n2)=O)CCCC1 c1(C(=O)NCCNC(c2c(CCC)nsc2N)=O)ccc2scnc2c1 C(=O)(CCC(C)(C)C#N)N1C(C)CN(C(C2(C)CC=CCO2)=O)CC1 N1(C(c2c(C)onc2)=O)CC2(CCCC(CNC(C3CC(=O)NC3(C)C)=O)O2)C1 c1(CCN2CCC(CNC(c3ncsc3Br)=O)C2)cccc(F)c1 N1(C(c2c(OC)ccnc2)=O)CCC(NC(=O)CN(C)S(N)(=O)=O)C(F)C1 C1(c2cn(CC)nc2)CN(C(N2CCC(c3n[nH]cc3CN)C2)=O)CCO1 C(c1ccc([N+](=O)[O-])cc1)=CC(C1(F)C(C(=O)OC)C1)=O.C(=O)OC NS(=O)(=O)CCCC(=O)NC1CCCC1NC(=O)CCN1CCC(O)CC1 C1(C)(C(=O)NC(C)CCNC(=O)C(C)O)CCCCC1 c1(C(N(CC(=O)N(C)CC2CCCC2(C)C)CC2CC2)=O)cc(O)ncc1F c1(OC)ccc(C(=O)NCCC(O)CNC(c2nocc2Cl)=O)nn1 C(=O)(C#CC1CC1)N(CC)CC1CCCN1C(C1CCC(c2cc[nH]n2)O1)=O N1(C(C(CC)n2ccnc2)=O)CCN(C(C2CCC(=O)N2)=O)C(COC)C1 C#CCC(CC(F)F)C(=O)NCCC1(O)CCN(C(=O)C(OC)OC)CC1 N(C(=NCc1ncc(Br)s1)N1CCC(OC)C1)C(C=C)C Cc1csc2ncnc(N3CCC(O)CC3C(=O)Nc3ccccc3)c12 O=C1CCOC(C(=O)OCc2ccc(C(F)(F)F)cc2)C1 c1(C(=O)OC)cccc(Cl)c1S(=O)(=O)NC1CN(C(=O)CNC(N)=O)CC1(F)F Cc1cccc(Cl)c1C(=O)NC1CN(C(C23CC(C)(CO2)C3)=O)CCC1C c1(C(C)(C)C)ncsc1C(=O)NCCCNC(=O)CC12CC(C1)C2 c1(C(=O)NC2CCN(C(c3cnc(Cl)nc3)=O)CC2F)c(O)cc(O)cc1O CCCCC(C)(F)C(=O)NCCCC(C)NC(=O)Cc1nc(C)sc1C N1(C(c2ncn(C(C)(C)C)n2)=O)CCC2(CC(NC(C3CC34CCC4)=O)C2)C1 c1(NS(CCOC(=O)C2CC2)(=O)=O)ccc(F)c(N2CCC(=O)NC2=O)c1 c1(CC)cc(CC(N2CC(C(N3CC=C(C)C3)=O)(COC)C2)=O)on1 n1(CC(N2C(CNC(C3C(C)C3(F)F)=O)CCC2)=O)nnc2ccccc2c1=O c1(C(=O)NC(CNC(C(C)=C(C)C)=O)C)cnc(N(C)C)cn1 N1(C(C=C(C)Cl)=O)CC2C3CCC(C2C1)N(C(c1cc(C#N)cs1)=O)C3 NC(=O)CCCCC(=O)N1CCCC(NC(C2CC(n3ccnn3)C2)=O)C1 C(=O)(C(CCC1CC1)NC(=O)CCC=CC(C)C)NC(CC)CSC N1(C(COCC(C)(C)C)=O)CC2CC(NC(=O)CC3CNC(=O)C3)CC(C2)C1 c1(CN(C(=O)C(C)CN(C(=O)CN2CCNC2=O)C)CC)ccncc1 c1(CCC(=O)N(C)CC2(NC(C3CC(CC)OCC3)=O)CC2)cccc(F)c1Cl Cc1cnccc1C(C)C(=O)NC(C)CNC(=O)CCC1CCC1 CCC1=C(C(=O)NC(C)C(c2ccccc2)NC(=O)CN(C)C(C)C)CCCO1 c1(C(N2CC(C(=O)Nc3csc(Cl)c3)(SC)C2)=O)cc[nH]c(=N)n1 Cc1c(C(N2CCN(C(=O)CC3CCN(C(C)C)CC3)C3CC23)=O)cccc1F C1(C(CNC(C2CC=CC2)=O)NC(c2ccn(C3CC3)n2)=O)CCCCCC1 N1(C(CNC(=O)OCC=C)=O)CCC2CCN(C(c3c[nH]cc3Br)=O)CC2C1 CN1CC(O)CC1(C)C(N1CC(C)(NC(c2cc(C(C)(C)C)c[nH]2)=O)C1)=O N1(C(c2c(C)c[nH]n2)=O)C2CCC1CC(NC(c1ccc(CN(C)C)cc1)=O)C2 c1(CC)nn(C)cc1C(=O)NCC(O)CNC(=O)COc1ccccc1O C1(C(N(CCC(C)NC(=O)CCC2CNC(=O)N2)C)=O)CN2CCCN1CC2 c1(NC)nc(C(N2CCC(C)C(CNC(=O)CC3(OC)CC3)C2)=O)cc(O)n1 N1(C(CCOCCOC)=O)CCC(C(=O)NC2(CCOC)CCC2)C1 C1(CCCC)CN(C(=O)CSC(F)F)CCN1C(=O)CCCCSC c1(CC(=O)NC2CC3CC2N(c2ccncn2)C3)ccc(F)c(F)c1 C=CCCCCCC(=O)NC(C)(C(=O)N(C)Cc1ccn(C)n1)C1CCC1 c1(OC)ccc2ncccc2c1C(N1CCCC(CCNC(=O)CC(C)O)C1)=O C1(NC(=O)C=Cc2cn[nH]c2)CCCCCN(C(C2CC(F)C2)=O)C1 C12CC(C1(C)C)CC(=O)N2.C1(NC(=O)OCC)CN(C(=O)CCn2ccnn2)C1 c1(C(N(C(CNC(CC2(OC)CCCC2)=O)C)C)=O)ccccc1CC#N c1(NC2CC(=O)NCC2)ccc(S(=O)(=O)NCc2nc(Cl)cs2)cc1F c1(C(=O)NC2(CSC)CCC2)conc1CNC(=O)C(N1CCOC1=O)C c1(C(=O)NCC2N(C(c3c(C)cco3)=O)CCCC2)c(F)ccc([N+](=O)[O-])c1C c1(-c2cn(CCN(C)C)nc2)ccc(C(=O)Nc2cc(C(F)F)no2)c2[nH]ccc12 c1(OC)cc(C(N2CC(CC(C)NC(C3CCC3)=O)C2)=O)cc(N)c1N c1(C(N2CC3C(CNC(C(C)OCCC#C)=O)(C3)C2)=O)c(CC)nn(C)c1CC C(c1cnn(C)c1)=C(C(=O)NC1C(CNC(C(C)=C2CCC2)=O)C1)C C(=O)(C1=NN(CCO)C(=O)CC1)NC1C(C)CN(C(=O)CC2OCCC2C)C1 c1(C(=O)NCC2(CNC(C3(C)CC3(F)F)=O)CCCC2)cc2cnccc2[nH]1 C1(C(=O)NC(CC(C)C)c2ccccc2)CC12CN(Cc1cncn1C)C2 C1(NC(=O)CCOC2CN(C(c3cn(CC#C)nc3)=O)C2)CC1C1CCCC1 N1(C(c2ncn(CC)c2)=O)CC(NC(c2ccc(Br)cc2)=O)CC1(C)CC c1(C(N(C)CC2OCCN(C(CSCCOC)=O)C2)=O)ccc2nc(S)oc2c1 C1(CCNC(C2CC2c2ccsc2)=O)CN(C(=O)C=Cc2ccsc2)CCCO1 Cc1cnc(NC2CCCOC2C2CCN(C(=O)C3CC3)CC2)nc1S(C)(=O)=O C1(O)(CN(C(C(C)NC(C2CCCC2)=O)=O)C)CN(C(C2CC(F)(F)C2)=O)C1 O=C(C1=CCC(F)(F)CC1)NC1(CNC(C2CCS2(=O)=O)=O)CC1 C1(C(=O)NCC2(C(C)NC(c3nc(C(C)C)oc3)=O)CC2)OCC2CCCC12 c1(C(=O)OC)cc(C(=O)NC2(CNC(c3cocc3C)=O)CCC2)c(C)s1 N1(C(C(C)S(C)(=O)=O)=O)CC=C(CC(=O)NC2CCCN(C)CC2)CC1 CC1(C)CN(C(=O)C(=O)NCC2(F)CC3(CNC3)C2)CC2(CC3CCC2C3)O1 C1(CNC(C(=O)N(C)CC2N(CC)CCC2)=O)CCC(N(C)C)CC1 C1(CC(C)NC(=O)CC2(CNC(C3CCCS3)=O)CC2)CCOC1 C1(C(=O)NCC2(C(=O)NC3(C)CCSC3)CCCC2)Cc2nccn2C1 CC(C)(C)C(CNC(C1CCOC(=O)CC1)=O)C(=O)NCC1(CO)CCCC1 c1(C(=O)NCC=CCNC(c2ccc(NCC)o2)=O)ccc(CC)cc1Br C1(CCOC)(C(=O)NCC2(CCNC(=O)C=CC(=O)N(C)C)CC2)CCC1 C1(C)(C(N(C)CCOCCNC(c2[nH]nnc2C2CC2)=O)=O)COC(=O)C1 N1(CC(=O)N(CC(CCC)C)Cc2ccccc2)CCC(F)(F)C(C#N)C1 Cc1c(C(N2CC(F)(CNC(C3CCOC3)=O)C2)=O)sc2cc(F)ccc12 C1(NC(C(C(C)C)NC(=O)Cc2cn[nH]c2)=O)CCC2(CC1)N=N2 C1(CC(=O)NC(CNC(c2ncc(C)cc2C)=O)CO)CC(C)(C)OC(C)(C)C1 C1(C(=O)NC2CN(C(c3cc(C)cc(F)c3)=O)C(C)C2)Cc2ccccc2N1 CC(C)(C(=O)NCC(O)CNC(C1CCCN(S(=O)(=O)C(F)F)C1)=O)C(N)=O N1(c2n(CCC=C)c(-c3coc(C#N)c3)nn2)CCc2ccc(COC)cc2C1 C(=O)(C1=CCC2CCC1N2C(=O)C(C)CC(C)C(C)=O)Nc1c(CC)noc1 C1(CNC(C(CO)NC(C2C(C)(C(F)F)C2)=O)=O)NC(=O)CC1(C)C Cn1ccc2ccnc(C(=O)NC3(C)CC(NC(c4cnc[nH]4)=O)C3)c12 c1(OC)ccc(C)cc1CC(=O)NC1CC(O)CN(C(c2csc(C)c2)=O)C1 C(=O)(C(CCCCNC)N(C(CCC)C(=O)NC)C)NCCC C1(C(=O)NCC(CNC(c2n(CCCC)ncc2)=O)CO)CN(C(C)C)CCO1 c1(NC(CN(CCCCCC)C(C=CCC)=O)=O)cc(C)c(C)nn1 N(C1CCc2cccnc21)C(C(Cc1ccoc1)NC(CC(C=C)CCC)=O)=O Cc1cccc(F)c1C(N1CCC(NC(C2CCC2(F)F)=O)CC1)=O C1(C(N2C(CCC#C)CCC2)=O)C=CCCN1C(=O)C(C)=CC(C)(C)C c1(C(=O)NCCCOCCNC(CC(C)CF)=O)c([N+](=O)[O-])cnn1CC(F)F c1(C(=O)NCCOC2CCN(C(C3(O)CC(O)C3)=O)C2)cc(F)c(F)cc1F N1(c2nc(SC)nc(C)c2)CC(C2CCCN(C(c3cc(O)ncn3)=O)C2)C1 Cn1nc(C(=O)NCC=CCNC(C2CCCCN2CC(F)F)=O)c(Br)n1 C(=O)(CC(C)F)N(C1CCN(C(=O)CCSC)C1)CC N1(C(C(CC)N(C)C)=O)CC(NC(C2CC(C(C)C)=NO2)=O)C(C)(C)C1 C1(C2CCC2)(C(N(C)CC2CCN(C(c3cncs3)=O)C2)=O)CC1(F)F C(=O)(C(CC)CC(C)C)NCC(CNC(COCCCC)=O)OC c1(OC)cc(C(N2CC(c3nncs3)C2)=O)cnc1C(F)(F)F c1(CC(=O)NC(C(C)(C)C)CNC(c2cc(C3CC3)no2)=O)cc(O)nnc1O N1(C(C(C)SC)=O)CCC2(CCN(C(=O)CN3CCCC3)C2)C1 CCC(CC)CCCC(=O)NCC1(C(=O)NC(C)C(=O)N(CC)CC)CCCO1 c1(C(=O)NC(C(C)C)CNC(=O)Cc2csc(NC=O)n2)cnc2[nH]cnc2c1 C1(NC(C(CC)C#N)=O)CC2(CCCCN2C(=O)C(c2ccccc2)F)C1 C1(NC(C(C)C)=O)CCN(CCNC(=O)C(c2ccnn2C2CCCC2)C)CC1 C1(NC(c2ccncc2-n2cccn2)=O)CC2CC1N(C(C1CC1F)=O)C2 C1(CNC(C(C)OCC=C)=O)CC2CCC1N2C(C1(O)CN2CCC1CC2)=O c1(N2CCC(NC(c3c(C)noc3C3CC3)=O)C2)ncccc1S(C)(=O)=O N1(C(C(C)OCCOCC)=O)CCCC(O)(CN(C(=O)C2=NOC(CC)C2)C)C1 N#Cc1ccc2cc(C(N3CCN(C(c4csnn4)=O)C4CCC34)=O)ccc2c1 C1(C(N2CCC(CCNc3c(C#N)c(Cl)ns3)CC2)=O)Cc2cccnc2C1 c1(C(N2C(C(N3CCCCC3)=O)CC(O)C2)=O)ccc([N+](=O)[O-])cc1Cl N1(C(C(COC)(C)C)=O)CC2(CCCN(C(=O)CS(=O)(=O)CC(=O)OC)C2)C1 Cc1cccnc1C=CC(N1CCC2CCC12CNC(=O)CCCC(C)C)=O Cc1ccc(CN(C(=O)C(CCN(C)C)NC(C2CC(O)C2)=O)C)nc1 N1(C(c2cc(C)c(Br)s2)=O)CC(NC(c2n[nH]c(C)c2F)=O)CC(F)C1 C12(CNC(c3scc(C)c3C)=O)CCC(C1)N(C(=O)C(C1CCC1)C1CCC1)C2 C=CC1(C(=O)NC2CCN(C(=O)C(=O)CCc3ccccc3)C(C)C2)CCOCC1 C1(C(N2CCN(C(c3cnn(C)n3)=O)C(CO)C2)=O)CCCCCC1(F)F C1(C)(NC(c2nc(C(C)C)sc2)=O)CCN(CCO)CC1 Cc1cc(C)c(C(=O)NCC2CCC(C)(C)CN2C(c2oncc2C)=O)c(=O)o1 c1(C(=O)NC(CNC(C(CC)C)=O)(C)CC)ccc2c(c1)CCO2 c1(NC(C2N(C(CCC=C)=O)CCSC2)=O)ccc(C(=O)OC)c(C#N)c1 C1(SCC(=O)NC2C(NC(c3c(CC)c[nH]n3)=O)CCC2)CCS(=O)(=O)C1 N1(CC(=O)N(CCC(=O)N(C)Cc2cccs2)CC)CCCNC1=O CCCC(CN=Cc1cc[nH]n1)C(=O)N(CC(C)C(=O)OC)C c1(N(C(C2(C)CN(Cc3sc(Br)nc3Br)C2)=O)CCO)c(Cl)cc(C#N)cc1Cl C=CC1(C(N2CCC(CNC(C3(C)CCCC3O)=O)CC2)=O)CCOCC1 CCCCC(CC)CC(=O)NCc1ccc(C(C)NC(c2ccncn2)=O)cc1 c1(NC(c2c(NC(C(C(C)C)O)=O)nccc2)=O)ccc2c(c1)n(C)c(=O)n2C c1(CC)ccc(O)c(C(=O)NCCCCC(C)NC(c2ocnc2C)=O)c1 N1(C(CSCC=C)=O)CC(NC(=O)CN=S(C)(C)=O)CC12CCCOC2 c1(C(N2CC(N(C(C3CCC(OC)C3)=O)C)C2)=O)nc(C)c(C)[nH]c1=O CCN=C(NCc1nc(Cc2ccccc2F)no1)NC(c1ccc(F)cc1)C c1(C(=O)NCC(C(C)C)NC(=O)CCCS(C)(=O)=O)nnc(O)c2c1CCCC2 C1(C)(C(=O)NCC2C(N(C)C)CN(C(COCC)=O)C2)CC2(CCC2)C1 Cc1ccc(O)c(CNC(=O)C(CO)NC(c2ccc(C(C)C)o2)=O)n1 n1(CC(=O)NC(C)CC(C)NC(c2cc(C(N)=O)co2)=O)ccc(=O)n(C)c1=O C1(OC)CN(C(C2CC2C2(C)COC2)=O)CCC1NC(C1CCC1(F)F)=O c1(CNC(C(=O)NC2(COC)CCNC2)=O)cncc2c1CCC2 C(CN=c1[nH]nc(C(F)F)s1)C1N(C(CC(=C)C)=O)CCCC1C CC(C)C1=NOC(C(N2CCC(CF)(NC(=O)CCCc3cccnc3)C2)=O)C1 C(=O)(C#CC1CCCOC1)NCC1N(C(c2cccc(CC)c2F)=O)C2C(C1)C2 N#Cc1ncc(CC2CC2)nc1N1CCC(C(N)=O)CC1 C1(NC(C2CC(=C)C2)=O)CN(C(c2cn(CC(F)F)nc2C)=O)CCC1C C1(NC(c2c(C)[nH]c(C(C)(C)C)c2)=O)CC12CCN(C(=O)CO)CC2 Cc1[nH]nc(C(=O)NCC2CC2NC(=O)CCC(=O)c2cccc(Cl)c2)c1O c1(OC)ccc(C(C)=CC(N2CCCC(NC(=O)COC3CC=CC3)C2)=O)cc1 CCCCC(CC(=O)NC1(CO)CCCOC1)NC(=O)CC1CCCC(C)O1 N1(C(c2c(-c3c(C)cc(F)nc3)cncn2)=O)CCc2c(F)ccc(F)c2C1 c1(C(=O)NC2CCN(S(C)(=O)=O)C2)cc(OC(F)F)ccn1 C1(CNC(=O)Cc2cc[nH]c2)COCCN1C(=O)CC1CC=CC1 Cc1cc(CO)oc1C(=O)NC(CNC(=O)C(O)CCc1ccccc1)CO C=CCC(C(=O)N(C)CC1(C#N)CCC1)NC(=O)CCN1CCOCC1 CC1(C)Cc2cccc(C(N3CC4CC4(NC(C4CNC(=O)C4)=O)C3)=O)c2C1 c1(CCNC(c2sccc2Br)=O)ccc(-n2cc(CCCO)nn2)cc1 C1(C(=O)Nc2c(-n3cc(C4CC(=O)C4)nn3)cccn2)CC2C(C1)C2(F)F C#Cc1ccc(OC(=O)C(CC(C)C)OC(=O)C(OC)OC)cc1 C(CC(C(C)(C)C)NC(=O)C1=CC(C)(C)C1)N(C(C(CC)n1cncn1)=O)C c1(C(N2CCC(C(C)NC(CN(C(COC)=O)C)=O)C2)=O)ncc(Cl)nc1Cl Cc1cn2nc(N3CCN(C(c4ccnn4C)=O)CCC3C)sc2n1 N1(C(c2cc(C)oc2)=O)C2CCCC1CC(NC(=O)Cc1c[nH]c(=N)nc1O)C2 C1(NC(c2ncn(CCNC(CC(C)C#N)=O)c2)=O)CC2CCC(C1)N2C C(=O)(C(C)CCCc1ccccc1)NCC(CC(C)C)NC(c1cnsc1)=O N1(C(CNS(C)(=O)=O)=O)CC2CC1CC2NC(c1cc(Cl)ccc1O)=O C(=O)(C(C)N=c1cc[nH]cc1)N1CCC(NC(C(C=C)CC)=O)C12CC2 CC1(C)C(CO)CCN1C(c1ccnc(CNC(c2cc(O)cc(=O)o2)=O)c1)=O n1(CC(=O)NC2C(CNC(c3c(CCC)n[nH]c3)=O)C2)nc(C)n(C)c1=O N1(C(C(Cc2ccccc2Br)NC(CC(CC)OC)=O)=O)CCC(C)(F)CC1 c1(CNC(=O)NC2C(=C)CC2)ccccc1C1CCCC1 CN1CC(CNC(=O)COCCNC(=O)CCCC2CCCO2)CC1=O C1(C(=O)NC(C2CSC2)C)CCOCCN1C(=O)Cc1nc(=N)[nH][nH]1 Nc1c(C(N2CCC=C(CNC(=O)CC3CC=CCC3)C2)=O)cnc2ccnn12 c1(C(=O)NC2(CCNC(C(CCSC)O)=O)CC2)cc2c(nc1N)CCCC2 Cc1cccc2nc(NC(c3ccc4c(c3)CC4)C3CC3)sc12 C(=O)(C(F)(CNC(c1ccn(COC)n1)=O)C(C)C)NC(C1CCOCC1)CC c1(C(=O)NCC2C(NC(CCCC=C)=O)C2)ccc(C(F)(F)F)c(O)c1 C1(CCCC)CN(C(=O)C(C2CCC2)OC)CCN1C(C1CC1C(F)F)=O c1(CC(=O)NC(C(C)NC(CCOCCC)=O)C)cccc(OC(F)F)c1 C1(C(=O)NCC2C(C)CCCN2C(c2cnc(Cl)cn2)=O)CCc2nncn2C1 N1(C(c2cc(F)ccc2F)C(=O)NCCCSCC)CCC2(CC1)CNC(=O)C2 N1(C(c2nccc(C)c2)=O)CCCC(O)(CN(C(=O)CCC(C)(F)F)C)C1 c1(C(=O)NCCCN(C(CC2CCC(C)O2)=O)C)cc2c(=O)[nH]ccn2n1 c1(CNC(CN(CCOC)C)=O)ccc(C(=O)NC2CCN(CCF)C2)s1 c1(C(=O)NCCC(C)NC(C2CC3C=CC2CC3)=O)c(F)ccc(O)c1F c1(C(=O)NCCC2OCCN(C(C(CC)(F)F)=O)C2)c(N)cccc1[N+](=O)[O-] c1(C(N2CC(N(C(Cc3c(C)nsc3)=O)C)C2)=O)[nH]c2ccccc2c1Cl C#CCCCCC(=O)NC(C1CCCCC1)C(=O)NCC1CC(C)=NO1 c1(CCC(=O)NCCC(C)N(C)C(c2cc(C(F)F)n(C)n2)=O)cncc(F)c1 c1(C(=O)OCC2C(C)(C)C(=O)C2)ccc(F)c(F)c1F C#CC1CN(C(C2CC(O)C(F)C2)=O)CCN1C(=O)CCCSC(C)(C)C c1(C(C(=O)NC)N(CC(C)C)Cc2ccc(C)o2)ccc(F)c(I)c1 N1(C(c2c(C(=O)OC)con2)=O)CC(NC(C2CCN2S(C)(=O)=O)=O)C(C)(C)C1 N(C1CC2(CCCC2)Oc2ccc(F)cc21)C(=O)C=Cc1c(Cl)nc2sccn12 N1(C(CC(C)=C(C)C)=O)CC2CC(C(=O)NCC(C)(CC)C(N)=O)C(C2)C1 Cc1cc(Cl)cnc1C(N1CC(C)CC1C(N1CCS(=O)CC1)=O)=O c1(C(=O)NC2CCN(C(C)C(=O)N(C3CCCCC3)C)C2)nc(C#N)cs1 CCC(C(=O)N1CCCC1CC(=O)NCc1ocnc1C)C(F)(F)F C(=O)(CC1C(=O)Nc2cc(Cl)ccc21)NCC1C(NC(CN(C)CC)=O)CC1 N1(C(CCC(C)OC)=O)CC(NC(c2cn(C)c(O)n2)=O)CC12CCCC2 CCCCC(C(=O)N(C)C)NC(=O)C(C)(C)CNC(=O)C=CCO C1(NC(COCCCC#C)=O)CCCC(CNC(C2CC(OC(C)(C)C)C2)=O)C1 N1(C(CCOC(C)=O)=O)CC(O)CC1C(=O)NCc1conc1C c1(C(N(CCN(C(=O)CCN2CCCCC2=O)CC)CC)=O)nn(C)c(N)c1C n1(CC(C)(C)C)nc(-c2ccc(F)cc2)nc1CC1COC(C)(C)C1 C(=O)(C1=CCCOCC1)N1CC=CC(C(=O)NCc2nc(C3CC3)n[nH]2)C1 c1(C(C(C)C)NC(C(=O)NCC(C)NC)=O)ccc(Br)c(F)c1 CCC(CCCC(=O)N(OC)C1CCOCC1)NC(=O)CC1COC(=O)C1 C1(CNC(C=C(C)Cl)=O)CCN(c2ncnc(Cl)c2[N+](=O)[O-])CCC1(F)F c1(CN2CCC(NC(=O)C(c3ccccc3)C3CC3)CC2)cc(Cl)nc(Cl)c1 C1(C(N2CC(N(C(=O)CCc3cccnc3Cl)C)C2)=O)CC2COCC2C1 C1(NC(C(CC)SC)=O)CCCCN(C(=O)C(c2ccc(F)cc2C)(F)F)C1 C1(C(N2CC(N(CC=C)C)C2)=O)(CC)CCCN(C(=O)CCCCSC)C1 c1(C(=O)NC23CC(CNC(=O)CSc4ccncc4)(C2)C3)onc2ccccc12 c1(C(=O)NC2CCOCC2)cnc(NC2CC(C(=O)O)C2)nc1 N1(CCCN(C(C(C)CC2CCCC2)=O)CCO)CCCCC1C N1(CC(=O)NC2C=CCN(C(COC(CC)C)=O)C2)CCSC(C)(C)C1 c1(C(N2C(C3(NC(CCSCCC)=O)CC3)CCCC2)=O)cnc2ccoc2c1 c1(C(=O)NCCC(C)N(C(c2ccn(CC(C)C)n2)=O)C)ccccc1S(C)=O C1(=CC(=O)NCCC2CCC(NC(=O)C(O)C3CCCC3)C2)CN2CCC1CC2 Cc1ccc(C(C)(C)C(=O)NCC=CCNC(=O)CC2CCCC(O)C2)cc1 C(=O)(C(F)C(C)(F)F)N(CC(C)NC(C1CNC(=O)N1)=O)CC N1(C(C2(CC=C)CCC2)=O)CC2CCC2(CNC(=O)CN2CC(C)(C)C2)C1 N1(C(c2ccc(OC)o2)=O)CCN(C(=O)CC2CCC(C)C(C)C2)CC(C)(F)C1 C1(C(NOCC)=O)C(CC)CCN1C(=O)C(C)Oc1ccc(C)cc1 CC1CCN(C(=O)CN(C23CC2CN(C(c2c[nH]nc2C(C)(C)C)=O)C3)C)CC1 C(=O)(C1=CS(=O)(=O)CCC1)NCC(C1(O)CCN(C(=O)C(C)(C)CCC#N)C1)C CC1(CNC(C23CCC(CC2)CC3)=O)CCCN(C(C2CCCN2C2CC2)=O)C1 c1(C(N(CC(CN(C)C(c2csc(C#N)c2)=O)O)C)=O)ccsc1S(N)(=O)=O O=C(CC(C(F)(F)F)NC(C1CCC2(CCC2)C1)=O)NC1CC(O)C1 c1(-c2nc(CSC)nn2CCCCO)cc(C)c(OCC(C)C)c(C)c1 C1(CC(N2C(C)(CC(=O)N(C3CC4CCC3O4)C)CC2)=O)CC=CCN1C C(=O)(CCCC(C)(C)CC)NCC1CCC(C(=O)NC2C(OCC)C2C)C1 C(=O)(C(C)(C)CCCNC(=O)CC1CCC(C)(C)O1)N(CC(F)(F)CO)C c1(C(=O)NC(CCOC)CNC(=O)COc2cnc(Cl)cn2)ccnc(Cl)c1O C1(CC(=O)NCC2(C)CCN(C(c3ncc(Cl)cc3F)=O)C2)CN2CCN1CC2 C(=O)(C(F)(F)C(O)C1CC1)N1CC(CCNC(C2C(c3n(C)cnn3)C2)=O)C1 c1(C2C(C(=O)NCC3CC(CNC(CCCC#C)=O)OC3)C2)cc(O)ccc1C N1(C(c2ccn(C)c2)C(=O)NC(CC)C)CCn2ncc(S(N)(=O)=O)c2C1 c1(C(=O)NC2CC(O)CN(C(=O)Cc3csnn3)C2)ccc2ccccc2c1 C12(NC(CN(CCC)C)=O)CCCN(C(=O)CSc3ccc(OC)cc3)CC1C2 C(=O)(C(C)CNC(=O)NC(C1CC2(CC2)C1)C(=O)OC(C)(C)C)OC C1(NC(C2CCN(C)CC2)=O)CN(C(C2CN(CC(F)(F)F)C2)=O)CC1N=[N+]=[N-] c1(C(N2CC(NC(CN3CCN(C)CC3)=O)C(O)C2)=O)sccc1S(C)(=O)=O C1(O)(CN(C)C(C2CCC(=O)NC2)=O)CCN(C(=O)C(C)(Cl)Cl)C1 CC1=C(C(=O)N2CCN(C3CN(C(c4n[nH]c(C)c4Cl)=O)C3)CC2)CCC1 C1(NC(c2c(CCC)nco2)=O)(CNC(=O)C(C#N)CC)CCC(F)(F)CC1 N1(c2nc(N3CCC(c4ncc[nH]4)CC3)cc(C)n2)Cc2nn(C)c(N)c2C1 C1(CC(=O)NCc2nc(C(=O)NOCCCC3CC3)co2)CCOC1=O CC1CC(C(=O)NC2C3CCN(C(c4ccnn4C)=O)C23)=NO1 c1(C(N2CC(COC)(CNC(=O)CC3(C)CCOC3)C2)=O)ccc(C)n(C)c1=O C(CCC(C)CC(=O)N1CC(NC(=O)C(C)(C)C(C)C)C(C2CC2)C1)=C(C)C C(=O)(N1CCCc2nccn21)C12N(C(Cc3n(C)cnc3)=O)CCC1CCC2 c1(C(N2CCC(N(C(c3nnc(C)s3)=O)C)C2)=O)cc2cnccc2[nH]1 C(CC1C(=O)N1)OC(=O)OC(C)(C)C.C(C(=O)OC)SCC(C)NOC(C)(C)C N1(C(c2nc(C)oc2)=O)C2CCC1CN(C(=O)CN1CCCCC(O)C1=O)CC2 c1(CN2CC(F)CC(C(=O)NC3CSC3)C2)ccc(I)c(F)c1F Cc1nccc(C(=O)NC(C(=O)NCCCc2c[nH]nc2C)C2(C)CC2)n1 Cc1nc2sccn2c1C(N1CC2CCC1C(CNC(C1CCC(C)C1)=O)C2)=O Cn1cc(NC(c2ccn(C(F)F)n2)=O)nc1C(=O)NCC1CCNC(=O)C1 C1(C(N(C2CCN(Cc3cn(C)nc3C)C2)CC)=O)CC(C)CC(C)(C)C1 C(=O)(N=c1nc(O)c2ccccc2s1)Nc1c(C#N)ncc(C)c1 c1(C(=O)NCC2N(C(c3cc(C)nnc3)=O)CCCC2C)cc(F)c(F)cc1F CCC(CC)(C(C)C)NC(c1ccc(CNC(=O)C(=O)C(C)(C)C)s1)=O c1(NC(C2CC(OC)CN2C(c2[nH]cnc2C)=O)=O)cnc(O)c(Br)c1 N1(C(Cc2c(C)ccs2)=O)CC2CCC2(CNC(C2CCS2(=O)=O)=O)C1 C(=O)(CC(=O)NCC1CC1NC(C1(C(C)C)CCC1)=O)NCC N1(C(C(CN(C)C)(F)F)=O)C2CCC1CC(NC(=O)CCCc1ccsc1)C2 C1(NC(CCc2[nH]c(=N)sc2)=O)CCN(C(=O)C(C2CCCCC2)O)CC1CO N1(C(=O)C#CC2CC2)CCCC(F)(CNC(=O)C(c2ccccc2Cl)O)C1 N1(C(CCC=C)=O)CC(NC(c2cnc(C)cn2)=O)C(C#N)C1 Cc1cc(CNC(c2cc(Cl)ccn2)c2nnnn2CCCF)c(C)o1 Cc1ccc(OCC(C)NC(C2CC(C)N(C(C34CCC(C3)C4)=O)C2)=O)cc1C N1(C(CCCCOC)=O)CCC(NC(=O)CCc2ccon2)C12CCC2 c1(C(=O)NC2CCN(C(=O)NC(c3ccccc3)C)C2)cc(Cl)c(F)c(Cl)c1 C1(C2(O)CCN(C)CC2)(C(=O)NC2CCN(C(C(CC)(C)CC)=O)CC2F)CC1 CCC(C(=O)NC1CCC(NC(c2cn(-c3cnn(C)c3)cn2)=O)C1)N(C)C CCCC(CNC(=O)C1=CCCC1)C(=O)NCc1[nH]ccc(=O)c1O N1(C(C=C(CCC)C)=O)CCN(C(C2(N(C)C)CCCC2)=O)C(CF)C1 S(=O)(=O)(c1ccc(N2CCC(Cc3ccccn3)CC2)c(Br)c1)N(C(C=C)C)C CCCC(C)(O)C(=O)NC(C)CCC(N1CC2CCC(C1)O2)=O CCC(CC(F)(F)F)C(=O)N1CC(NC(=O)CC2(CCOC)CCCC2)C(C)C1 C1(NC(C2CSC2)=O)CCN(C(=O)CC2CCS(=O)(=O)CC2)CC1F C1(C(N(C)Cc2ncn(C)n2)=O)CC(N=[N+]=[N-])CN1C(=O)C1=CCCCC1 c1(OC)ccc(OCC(=O)N(C2CCCN(C(C3C=CCC3)=O)C2)C)cc1 O=C(C(O)CC(F)(F)F)NC1CCN(C(c2ccnnc2SC2CCCC2)=O)C1 c1(OC)ncc(CONC(C(=O)NCCc2ccccc2)=O)cn1 C1(C(N2CCC(OCC(=O)NC3CN(C(C)C)C(=O)C3)C2)=O)CC12CCOCC2 N1(Cc2ccc(C)c(C)c2)Cc2ccccc2C1C(=O)Nc1cc(Br)cnc1Cl N1(CC2C(OCC)CCCC2)CCC(=O)N(CC(=O)N(C)OC)C1=O C=CC(C)N=C(NC1CC(CS(N)(=O)=O)C1)N1CCc2cc(Cl)cc(Cl)c2C1 c1(NCC2(O)CCN(C(C3(CC(C)C)CCC3)=O)CC2)ccc(Br)cc1[N+](=O)[O-] CC1CCC=C1C(=O)N1CCC(O)(CNC(=O)COc2ccccc2Cl)C1 c1(C(N2CCC(C(C)NC(c3cn4c(n3)SCC4)=O)C2)=O)ccc2nccn2c1 C1(NC(C(C)C2CC2)=O)CCCOC12CCN(C(C1CC(C)(F)C1)=O)CC2 C(CN=c1ccc(C)c[nH]1)NC(=O)NCC=CCCOC N1(C(c2cnsc2Br)=O)CCC(c2cn(CC3CC3C(F)(F)F)nn2)C12CC2 c1(C(=O)NC(CCOC)CNC(=O)C(O)CC(C)C)cc(Cl)c(N)c([N+](=O)[O-])c1 c1(C(=O)OCC(C2CCCNC2)=O)cc(=O)n2nccc2[nH]1 c1(C(CNC(N2CCCC(=C)C2)=O)C(F)(F)F)c[nH]c2ccccc12 c1(C(=O)NC2C3OCC(NC(c4c(CC)nco4)=O)(C3)C2)cc2c(s1)CCCCC2 Cc1ccc(C(=O)NCCC2CCC(NC(=O)COCC3CCC3)C2)c(O)c1C CC1CN(C(=O)C=CC(F)(F)F)CCC1CNC(c1cccc(Cl)c1O)=O N12CCCC3(C1)CN(C3)C(=O)Cc1cc(cc(Br)c1)C2=O.C#CC1CC1OC c1(-n2cc(SCC3(C)CCCCO3)nn2)cc(F)cnc1Br c1(OC)ccc(NC(=O)C(c2c(C)cnn2C)N(C2CSC2)C)cc1 CN1CCN(C(c2cncc(Cl)c2)=O)C(CNC(=O)C2=CCCO2)C1 c1(CC)cc(C(N2CC(F)(CNC(c3noc(C)c3Br)=O)C2)=O)c(C)o1 C(=O)(C(C)(C)c1ncco1)NCC1(CNC(C=CC(C)(C)SC)=O)CCC1 c1(CC(=O)NCC(CNC(C(C)OCCN(C)C)=O)C)cc(F)ccc1Cl C1(Cc2cn(CC(C)NC(=O)CCCc3cccs3)nn2)CCCCN1C C(CC(Cc1ccccc1)NC(=O)C(C)C#N)NC(C=C(CC)C)=O c1(CC)nc(C(=O)NC2(C(=O)NC(C)Cn3cncn3)CCSC2)co1 c1(C(N2CC(C)C(NC(CNC(C)=O)=O)C(C)C2)=O)ccc2cccnc2c1 CC(CC(=O)N1CC(NC(C2(C#N)CC3CCC2C3)=O)C(C)C1)CC(C)(C)C C(C)(C)(CCC(=O)NCCOCC(=O)NC1C2CCCC12)N(C)C CN=c1cc(CNC(c2ccccc2CCC(C)C)=O)cc[nH]1 c1(C(=O)NC2CC(CNC(=O)Cc3ccsn3)C2)cnn2c1OCC(F)C2 c1(C(=O)NC(C)CCCCNC(C2CC3CCC2CC3)=O)ccnc2[nH]cnc12 C1(N(C)C)CCN(CCNC(N2CCC(CC(C)(C)C)C2)=O)CC1 c1(C(=O)NCC2(CNC(c3cc(CCOC)on3)=O)CCC2)cn(C)ccc1=O C1(NC(c2cccc(-c3cnco3)c2)=O)CCCCN(C(C2(Cl)CC2(F)F)=O)C1 CC1(C(=O)NCC(CO)NC(c2cscc2Br)=O)COCCO1 C=CC(C)(CCOC)C(=O)NCC(C1CC1)NC(=O)COc1ccc(C)c(C)c1 N1(C(CSC)=O)CCC(OCCCON(C2CCSC2)C(C2CCCO2)=O)CC1 c1(CCC)cc(C(=O)Nc2ccnc(CF)n2)n(-c2ccccn2)n1.C1(=O)CO1 c1(C(N2CC(=O)NCC2)=O)ccccc1OC.C(=O)(CCC1CC1(F)F)OCC.CC C12(CNC(C(C)N(C(CCCOC)=O)CCO)=O)CCC(C1)C(=O)N2 CC(C)CC(C(=O)NCC1(CNC(=O)CN2CCCCCC2=O)CCC1)C(N)=O C1(NC(Cn2ncc(C)c2)=O)CN(C(=O)C(C)(F)F)CCC1C N1(C(C(C)SC)=O)CCN(C(c2ccnc(OC3CC3)c2)=O)CC1C(C)C Cc1ccnnc1C(=O)NC(C)CCCCNC(C1CC(=O)N(C(C)(C)C)C1)=O N1(C(C(C)C(F)F)=O)CC2CCN(C(=O)CCCc3ccc(F)c(F)c3)C2C1 CC(CC(F)F)C(=O)NC1CC(NC(c2ncc(Br)cc2O)=O)C1 C(=O)(CC(C(C)OC)NC(=O)CCC(N)=O)N(CCC(=O)OC)CC=C c1(OC)cc(F)c(C(=O)NC(C)CN(C)C(C2Cc3nncn3C2)=O)c(F)c1 CC(C)CC(C)CC(=O)N1CCOCCC1C(=O)N(C)Cc1cn(C)nn1 N1(C(CNC(c2ccccc2)=O)=O)CCC2(C(=O)NCC3CCC3)CC2C1 C(=O)(C(CC(C)SC)N1CCC(C(=O)NCCC(=O)OC)(OC)CC1)NCC=C c1(NC2CCC3CN(C(CC(C)n4ccnc4)=O)CC32)ncnc2c1CCCC2 C=CCC(C)C(=O)NC(c1ccccc1)CNC(c1sccc1C1CC1)=O N1(C(C2C(CC)C2)=O)CCN(C(=O)CC2(O)CCCC2)CC1 CC1CC2(CC(C(N3CCN(C(=O)CCCC4CCOCC4)C(CO)C3)=O)C2)C1 c1(Nc2cc(C)c(-c3cccc(C(=O)OC(C)(C)C)c3)s2)c[nH]cc(Br)c1=O c1(C(CC)CC)cc(C(=O)NCCC2(NC(c3sccc3SC)=O)CC2)on1 c1(OC)csc(C(=O)N(C)CC2(NC(C3CCSCC3)=O)CC2)c1OC C(C(C)(O)C(=O)NCC1CCC1C(=O)NCC1(CO)CC12CCC2)OC c1(N2CC(O)(CCNC(C3C(C)CC(=O)NC3)=O)C2)cccc(F)c1[N+](=O)[O-] N1(C(C=C(CC)C)=O)CCN(C(=O)C2=COCC2)CC1CCO N1(C(c2c(C)ocn2)=O)CCCN(C(C2CCC3C2C3(F)F)=O)CCC1 C1(NC(=O)CCF)CN(C(c2ccc3n[nH]cc3c2Cl)=O)Cc2nccn2C1 CCC(F)(F)C(=O)NC(CO)C(C)NC(=O)CCN1CCCC(C(N)=O)C1 c1(C(CNC(CN(C2CCC2)C(C2C(=C)C2C(=O)OC)=O)=O)O)ccncc1 C1(CNC(C2(CC(C)C)CC2)=O)CC(C)N(C(=O)CCSc2ccccc2)C1 N1(C(CS(CC)(=O)=O)=O)CC2CCC1CC2NC(C1CCC(C)C1)=O C(=O)(C1CCCc2nnn(C)c21)NC(C1CCCC1)CNC(CCCC#C)=O c1(NCC2ON=C(CC)C2)cc(N2CC=C(Br)CC2)nc(C(C)C)n1 C(C(CN=c1cc(C)nc(CC)[nH]1)C(F)(F)F)NC(C(CCC)OCC)=O C1(CNC(C(COC)NC(=O)Cn2ccc(C)c2)=O)CNC(=O)CO1 C=CC(C)CC(=O)N(C1CCC(NC(=O)Cn2cnnc2O)CC1)C C1(NC(C(C)(C)NC(C=COC)=O)=O)CC2CC(NC(c3ccc[nH]3)=O)C1C2 c1(C(=O)NCC#CCNC(C(c2cccc(OC)c2)C)=O)ccc2c(c1)CCN2 N1(C(CSCC)=O)CC(C(=O)NCc2ncc(C)[nH]2)CC(F)(F)C1 C(=O)(C1=CCc2ccccc21)NCC1CCCC(NC(C(C(C)(F)F)(C)C)=O)C1 Cc1ncc(Br)c(C(=O)NC(C)CCNC(=O)CCOCC2CCCO2)n1 N1(C(C)=O)CCCCC1COCc1ccc(CSC)cc1 C1(C(=O)NCCc2cnc(C)s2)C2CCC(C2)N1C(=O)C(O)CC(N)=O CC1(C)CCCN(C(=O)CC2CCCC(=O)N2)C1C(=O)NCCOC1CCCC1 c1(CC(=O)NC(C)CCNC(C2CCCN2C)=O)ccnnc1O CCCCCC(O)CC(=O)NOCC(N1CCC2(CCSCC2)CC1)=O N1(C(C2ON=C(CC)C2)=O)CC(NC(c2cc(O)ccc2O)=O)CC(C)(C)C1 C=CCN=c1[nH]cc(C(=O)N(C(C)CNC(C2CN(C)C2)=O)C)s1 C1(CNC(CC=C)=O)CN(C(c2cnn[nH]2)=O)CCC1C(F)(F)F C1(C(=O)NC2CCN(c3ncn(C)c(=O)c3)CC2F)CC2(CCCC2)CO1 CC(CNC(c1cocn1)=O)C(F)C(=O)N(C1CCC1)C C(=O)(C(C(CC)CC)OC)N1CCCC(CC)(NC(=O)CCCn2ccnn2)C1 C=CC(CC)CC(=O)NC1(C(N2CCC3C(OC)CC23)=O)CCCC1 c1(C(N(CCNC(C(C=C)CC)=O)Cc2ccccc2)=O)cc(C)cc(C)n1 c1(C(=O)NC(C)(C)CNC(c2ccccc2CC#N)=O)cncc2sccc12 N1(C(c2cc(OC)no2)=O)CCCC(C(=O)NCC(n2cccn2)C)C1 c1(C(=O)NCC(C2CC2)NC(Cn2cc(C(C)=O)nn2)=O)c(C)nsc1C c1(C(N2CCCC(CC=C)(NC(=O)CCF)C2)=O)cnc2nc(O)nc(O)c2c1 C(=O)(C(C)(C)CCC(=O)N1CCC(NC(C2C3COCC23)=O)CC(C)(C)C1)OC CCC(CC(=O)NC1COCC1NC(=O)C(c1ccncc1)C1CCCC1)C(F)F c1(C(N(C2CCN(C(CC3CC(C)C3)=O)C2)C)=O)cc(=O)c2ccncc2o1 CC(CC(N)=O)C(=O)N1CCCN(C(C2(C(F)F)CCCO2)=O)CC1 c1(C(=O)NCC(C)NC(C2(Cc3ccccc3)CCCO2)=O)cc(O)cc(O)n1 c1(CCC)onc(C)c1C(=O)NCCC(C)NC(C1CCOC1=O)=O N1(C(C2(CC=C)CCCN2C(=O)CC=C(Cl)Cl)=O)CC23CCC2(COC3)C1 Cc1ccc(CC(=O)NCC2(NC(=O)NC3CCCC3(F)F)CCCCC2)nc1 c1(C(N(CC(C)NC(CCC(C)N(C)C)=O)C)=O)cc2cc(Cl)ccc2[nH]1 Cc1cc(C(N2CCC(C)(CNC(=O)C(C)C3CCOC3)CC2)=O)ccc1Cl CCC(CNC(C1CC1C(C)(C)C)=O)(CC)NC(=O)CN1CCC(=O)CC1 C(=O)(CS(=O)(=O)CC(F)(F)F)N(C1CCCN(C(C(CCC)OCC)=O)C1)C Cc1cc(-n2cc(C(=O)NC(CCO)C(C)C)nn2)cc(C)c1 N1(C(CSC)=O)CCC(C2CCN(C(C3(n4ccnn4)CC3)=O)CC2)C1 c1(OC)ccc2[nH]c(CN3CC4CC4(C(=O)Nc4ccc(F)cc4Cl)C3)cc2n1 N1(CC(N2CC(C(Cn3cc(CCC(C)O)nn3)F)C2)=O)CCCCCC1=O C1(CN(C(c2c(COC)cc[nH]2)=O)C)CN(C(=O)CCC(CC)OC)CC12CC2 C1(CC(NOC(CC)CC)=O)CCCCN1C(=O)COC1CC1 C1(CC=C)(NC(=O)CCCn2cncn2)CCN(C(=O)C(C)(C)CSC)C1 c1(C(N(C)CC2(NC(C(C(C)O)C)=O)CC2)=O)c(F)cncc1Br N#CC1(F)CCN(C(=NCc2ccc(Cl)cc2F)NCC(F)F)CC1 C(=O)(CCC(C)(C)C(=O)N1CC(NC(=O)CC(C)(C(F)F)N(C)C)C1)OC Cc1cn2c(n1)CN(C(c1csc(CNC(c3cc(O)n(C)n3)=O)c1)=O)CC2 C1(C(N(CC(CNC(c2nccc(C)c2N)=O)(C)C)C)=O)CCn2nnnc2C1 C1(CC(N2CC3(N(C(COCC)=O)CC3)C2)=O)SC(=Nc2ccccc2)NC1=O C(C(O)(CNC(=O)C(CO)NC(C1CC(=O)CS1)=O)CO)OC Cc1nn(-c2ccccc2)cc1-c1nc(CC2CC2)nn1CC1CCCO1 C12(C(=O)NC(C)Cc3ccccn3)CCCC1CCN2C(C1CCC(=O)O1)=O O=C(C1CCc2c[nH]nc21)NCC1(O)CCCN(C(=O)C2=CCCC2)CC1 C1(C)(NC(CC(n2ccc(C)n2)C)=O)CCN(C(c2cccc(C(N)=O)c2)=O)C1 CCC(=O)CCC(=O)NOCC(N1CC(NC(=O)C2CC2)C1)=O N1(C(C2(CC)CCC2)=O)CC(NC(=O)CC2CCCCCO2)C(C2CC2)C1 c1(C(=O)OCC)nc(C(=O)NCCNC(=O)CCNC(N)=O)c(C)s1 CC1(C(=O)NCC2(F)CC(NC(C3COC3)=O)C2)CCNC1=O CCC(C(=O)N1CCN(C(c2ccccc2I)=O)CC1)C(C)O C12(CNC(c3cc[nH]c4nccc3-4)=O)CCCCC1N(C(C1CC=CC1)=O)CC2 N1(C(C=C(CCC)C)=O)CC(NC(=O)CC2COC(=O)N2)CC(C)(C)C1 c1(CC(=O)NCC(C)CN(C)C(C2(C)CCCNC2=O)=O)cccc(Cl)c1Cl C(C(C)(C)C(C)(F)F)(c1n(CC(=C)C)nnn1)Nc1ccc(Cl)c(C(=O)OC)c1 c1(C(N2CCN(C(C(C3CCC3)OCC)=O)C(CF)C2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 Cc1nc(NC(c2ccc(F)cc2Cl)C)cc(N2CCCC(OCC3CC3)C2)n1 C(=O)(C1=NNC(=O)CC1)N(C(C)CNC(=O)Cc1csc(-c2nc[nH]n2)n1)C c1(C(=O)NCC(C2(O)CCN(C(C3CC(O)C3)=O)C2)C)cccnc1N1CCCC1 c1(C(c2nnnn2CC)NC(CCCC)CC)ccc2cnccc2c1 Cc1cccc(C(N2CC(NC(c3nccc(Cl)c3C)=O)C3(CC3)C2)=O)c1C#N C1(C(=O)NCc2cc(Br)no2)CC2(CC2)CN1C(c1ccc(F)c(Br)c1)=O C12(CC)CC1CN(C(c1cc(CNC(=O)C=CCN3CCCC3)on1)=O)C2 C(CC(C)C(=O)NCCN(CC(C)O)C(=O)Cc1cnsc1)=CC c1(C(=O)O)ccc(OCCNC(C2CCC2c2ccc(F)cc2)=O)cc1 C1(O)(CN(C(C(=O)NCCOC)=O)C2CC2)CCN(C(=O)C=CC2CCC2)C1 N1(C(c2ccc(SC)s2)=O)CCC2CN(C(=O)CCCC3CCCC(=O)N3)CC12 C1(C(=O)NCCCC(C)NC(CCC=C)=O)CC2CC(=O)C1C2 C=C1CC(C(=O)NCc2ccc(Cl)s2)N(C(c2ccnc(F)c2)=O)C1 CC(C)(C#N)CC(C)(c1nnnn1C1CCCC1)NC1C2COCC12 C1(C(=O)Nc2ccc(C3CC3)cc2)C2CC1N(C(c1cc(CC3CC3)no1)=O)C2 Cc1nc2cccc(C(=O)NC3CN(C(=O)C=Cc4ccsc4)C3)c2s1 c1(OCC)ccc(Cl)cc1NC(c1csc(Cl)c1)c1nnnn1C1CCC1 C(=O)(C1=Cc2ccccc2C1O)NC1C2C(C)N(C(c3cc(C)c(C)o3)=O)C1C2 N1(Cc2cn(CC(F)(F)F)nc2C2CC2)CCC=C(c2ccco2)C1 N1CCN(C(=O)C#CC(C)(C)C)CC1c1cn[nH]c1.CN1CCCC1CC1CCC1 CCC(C)(C)CC(=O)N1CCCC1(C)CNC(=O)C=C1CN2CCC1CC2 CCC1=NOC(CC(N2CCC(NC(=O)CCN3CCCCCC3)C2C)=O)C1 C(CCC)(C(C)(C)C)NC(CSCCN(C(C(C=C)C)=O)C(C)C)=O C1(C)(CC)C=C(C(=O)N2CCC(C)C(NC(=O)CCc3cncc(F)c3)C2)C1 CN1CC(C)(C(=O)NC2CCC(NC(c3ccc(Cl)cc3)=O)CC2)CC1=O Cc1c(C(N2CCCC(NC(c3cnc(C#N)s3)=O)C2)=O)cncc1Br C1(NC(CSCC)=O)CC2CC(NC(c3scc4c3CCCC4)=O)CC2C1 C(=O)(CCC(=O)c1ccc(Cl)cc1)NCC(CNC(CC(C)C1CC1)=O)(C)O CCCCCCC(C)NC(=O)C(CCC)c1nn[nH]n1 c1(CC(C)NC(C(C)C)=O)ccc(CNC(c2scnc2C(C)C)=O)cc1 C1(CNC(C(COC)(C)O)=O)CN(C(=O)C(F)=C(C)C2CC2)CC12CCC2 N1(C(c2n(CC)cnn2)=O)CC2(C1)CN(C(C1CC13CCCC3)=O)C2 CC1(NC(=O)C(N)=O)CCCCC1C(N1CCC(F)(CF)C1)=O CCC(C)(C)CCN=c1[nH]c(NC2CCn3cnnc3C2)nc2c(F)cccc12 C=CCCC(C(=O)NCC(C)(C)C1CCC1)NC(C1CC2(CCC2O)C1)=O N1(C(=O)CC2CC=CC2)CCC(C2CCN(C(=O)C3=C(Cl)CCOC3)C2)C1 CC(C)(C)C(O)CNC(C1(CNC(c2nocc2Cl)=O)CCCC1)=O CCC(C)(CO)C(=O)N1CCC(CCNC(c2cnc(-c3ccccc3)[nH]2)=O)C1 C(=O)(C1Cc2ccccc21)NCC1C(NC(Cn2cc(C(C)(C)C)nn2)=O)CC1 C(=O)(C1CCCc2cccnc21)NCC(C(C)C)NC(c1ccc(C)c(F)c1)=O C(C)(C(=O)NCCCCN(C(=O)COC1CCOC1)C)OCC=C c1(NC(C2N(C(CN3C(C)CCC3)=O)CCCC2)=O)cn(C)nc1C#N C1(NC(CN(C(C(C)C)=O)C)=O)CC(F)CN(C(c2ccc(Cl)cc2)=O)C1 C(=O)(C(F)CC1CCCCC1)N(CC(C)NC(=O)CCNC(=O)C1CC1)CC C1(CNC(C(C(C)C)OC)=O)CN(C(=O)COCC2CCCCC2)CC(C)(C)C1 C1(CCO)CCCCCN1Cc1nc(Cl)cs1 C1(CCNC(C2C(COC)C2)=O)CC(F)(F)CN1C(c1cc(C2CC2)no1)=O c1(C(=O)NCC2(NC(C3CCC(CC)O3)=O)CC2)c(Cl)cccc1[N+](=O)[O-] N#CCCCC(=O)N1CCC(N2CCN(C(=O)COc3ccsn3)CC2)CC1 C1(O)(CC)CCN(C(=O)C(CCNC(c2c[nH]c(C#N)c2)=O)OC)C1 c1(C(=O)NC2(CC=C)CN(C(C3C=C(C)CS3)=O)C2)ccc(C(C)C)c(C)c1 Cn1nnc(C=CC(=O)NC2CCCC(NC(c3csc(Cl)c3)=O)C2)n1 C1(C(=O)NC2CC2)OCCC1C(=O)N(CCCO)CCOCCCO CCCCCC(O)CC(=O)N1CCN(C)C(CNC(c2occ(C)c2C)=O)C1 C1(C(N(CCCNC(C2CCCC23CCC3)=O)CCO)=O)CC2(CCO1)CC2 N1(C(c2ccc[nH]2)=O)CCC2(CCOCC2C(N2CC(F)C2)=O)CC1 N1(C(c2cnc(C)o2)=O)CCC(C)(C)C1CNC(C1C=CCC1)=O c1(CNC(COCCC#C)=O)ccnc(C(=O)NCc2cnn(CC=C)c2)c1 N1(C(C(C=C)C)=O)CCN(CC(=O)NCCn2cc(C(C)O)nn2)C(=O)C1 C1(CCOC)(NC(c2c(C)csc2Cl)=O)CCN(C(c2nc(Cl)oc2C)=O)C1 c1(C(=O)OCC)cc(C(=O)COCC(=O)N(CCCC2CC2)CC)on1 Cc1nn(C)c(Cl)c1C(=O)NCCC1CCCN(c2ccnc(C3CC3)n2)C1 c1(OCC(C)C)ccc(C(=O)NCC2C=CCN2C(=O)C(O)C(F)F)cc1 CC1OCCC1CC(=O)NC(Cc1ccoc1)C(=O)NC(CC1CCC1)CO c1(C(=O)NCC2N(C(C(CCC)C(C)C)=O)CC2)nccn2nc(C)cc12 c1(CC)onc(C)c1C(=O)NC(C1CN(C(C2CCN2S(C)(=O)=O)=O)C1)C c1(C(=O)NCC2CC(NC(c3cnc(NC4CC4)s3)=O)C2)ccc2c(n1)NCC2 C12(C(=O)NCC(C)N(C)C)CCC(CC1NC(c1cn(C)nn1)=O)C2 N#Cc1cc(F)c(C(N2CCSC(C(=O)NCC3CCC(O)CC3)C2)=O)c(Cl)c1 CCCCC(O)C(=O)N1CCC(CN(C(C2CC=CCC2)=O)CC2CCCO2)CC1 CCC1=NOC(CN(CC(C)NC(c2cnn(C(C)C)c2)=O)CC)C1 n1(CC)nnc(C)c1CN(CCCNC(=O)Cc1cccnc1C(N)=O)C1CC1 n1(Cc2c(OC)c(-c3ncn(C)n3)ccc2)ncc2cc(Br)ccc2c1=O C1(C(=O)NC(CC)C(=O)OC)CC(F)(F)CN1C(C1CCC(C(=O)OC)C1)=O N1(C(CN(CC(F)(F)F)C)=O)CC(NC(c2cocn2)OC)C(C2CC2)C1 c1(N2CCCC(NC(Cc3cc(OC)no3)=O)(CO)C2)ncnc2c1ncn2C c1(OC)ncc(C(N2C(C(=O)NCCn3cc(C)cn3)CC3CC23)=O)cn1 C12(NC(c3occ(C)c3C)=O)CCC1CN(C(=O)CN1CCC(C)(O)C1)C2 c1(NC(N2C(c3onc(-c4c(OC)cccc4)n3)CCC2)=O)c(F)cccc1Cl c1(C(N(CC)CC2CCCN2C(c2cn[nH]c2)=O)=O)cccc(N(C)C)c1 N1(C(CC(=O)ON)=O)CCCC(c2ncon2)C1 O=C1COC(c2ccc(NC3CC4CCC3CC4)cc2)=NN1 C1(NC(C(=O)OC)CC2OCCO2)CCC(P(C)(C)=O)C1 CCC(CC)CCCC(=O)N(C(C)CCNC(=O)C(C)(C)c1cnsc1)C C(=O)(CCCCCCCC1CC1)NC(CCCNC(CC1(CC)CCCC1)=O)C c1(-n2c(Cc3cc(C)no3)nc(-c3ccn(C)n3)n2)ccc(F)cc1C C(CC(C)C)(C(=O)N1CC(CCNC(c2nnc(Cl)cc2N)=O)(OC)C1)OC N1(C(C2CCC(NC(C(C)OC(C)=O)=O)C2)=O)CCc2ncncc2C1 c1(COCC=CC(=O)NC2CN(C(c3sccc3Cl)=O)C2)ccccc1 Cc1cc(=NCCC2CC(C)(C)CO2)[nH]c(=NCC2CCCCC2OC(C)C)[nH]1 c1(OC)cc[n+]([O-])c(C(=O)NCC2(O)CC(NC(C3CCCCC(=O)N3)=O)C2)c1 C(=O)(CCCC(C)(C)C)NCCCN(C(=O)CCc1cncn1C)CC CCC(CC)CCC(=O)NCCSCC(=O)N(CC(C)C(=O)NC)C(C)C N1(C(c2c(C)ncs2)=O)CCCC(C)C1CNC(c1cnc(N(C)C)o1)=O CC1(C)CN(c2nc(Cl)c(C#N)s2)CCC1NC(=O)CC1CC=CCC1 CC(CN(C)C)CC(=O)N1CCC(F)(C(=O)NCc2cc(Cl)no2)C1 c1(CCC(C)C)ccc(C=NOCc2ccccc2)cc1F CC1Oc2ccc(C(=O)N(C3CCCN(C(=O)CN(C)C)CC3)C)cc2C1C C1(NC(Cc2c(OC)ccc(Br)c2)=O)CCCC2CN(C(C3CCCO3)=O)CC12 N1(C(c2ccn(CC)n2)=O)CCCC(C(N2CCOCC(C)C2)=O)CC1 N1(C(c2cccc(CC)c2)=O)CCC(NC(=O)CSCc2cscn2)C(C)C1 C1(C(=O)NCC2CC(OC)CN2C(c2ccn(CF)n2)=O)CC2(CCCC2)CO1 [N-]=[N+]=NC1CCN(C(=O)C(c2cccnc2)NC(=O)Cn2cccn2)CC1O Cc1cnc(C(=O)N(CCCNC(C2CCOC2C(F)(F)F)=O)CCO)c(C)c1 c1(C(=O)NCCCN(C(CC(C)C2CCCO2)=O)C2CC2)cc2ncccc2o1 c1(C(=O)NCC2CC(O)CN2C(C2CCCC2)=O)ccn2ncnc2c1 c1(N2CCC(CNC(c3nc(F)ccc3Cl)=O)C2)nc2cc(F)cc(F)c2o1 C1(NC(CN2C(C)CCC2)=O)CN(C(c2cc(Cl)sc2Cl)=O)CCC1F C1(C(=O)NCCC(C(=O)OC)O)C2CC3C(C2NC(=O)Cc2cn[nH]c2)C13 N1(C(C(C)C)=O)CC2(CCN(C(C3CSc4ccccc4O3)=O)CC2)CC1C C1(CNC(C(C=C)C)=O)C(C2CC2)CCN1C(=O)Cc1ccc(OC)nc1 c1(C(=O)NCCCN(C(=O)CC2CCN(C)C2=O)CC)cnc(N)cn1 c1(C(N(CCC(C)NC(CCCCCC)=O)C)=O)cccc2sncc12 CC(C)CC(F)C(=O)NC1CC(NC(C2(c3cccc(F)c3F)CC2)=O)C1 Cc1cc(-c2nc(CC3(C(F)(F)F)CC3)n(Cc3cnccc3C)n2)ccc1F N1(C(C(CCNC(=O)C=Cc2ccoc2)OC)=O)CCC2(CCC2)CC1 C=CCC(CC=C)C(=O)NCC#CC(=O)N(CC(CC)OC)C CCC(C)C(C(=O)N1CC(NC(C2CC2c2ccccc2Cl)=O)C(C)C1)N(C)C C1(COC)CC(CNC(c2c[nH]c(=N)s2)=O)N(C(=O)C(C)n2cccn2)C1 CC(CCCNC(C12COCC1C2)=O)NC(=O)CSS(C)(=O)=O N1(C(COCC#C)=O)CCC(NC(=O)CCCC2CC2C)C1 C1(C(=O)OCC(C(=O)OCC)O)Cc2ccc(Br)cc2C(=O)O1 c1(CC)c(C(=O)NCC2CC2NC(c2ccoc2C)=O)cnn1-c1ccc(C)cc1 CCC(C)CC(=O)NC1(C)CCN(C(=O)CCCCNC(N)=O)C1 C(=O)(N=c1[nH]cnc(Cl)c1C)c1ccc(OCC#C)cc1 CCC(C)(C)C(O)C(=O)N1CCCC1C(C)NC(=O)CC(C)(C)COC CCCCC(=O)NCC1CCC1C(=O)NC(CCC)C1CC1 C(=O)(C1CCCc2cncn21)NC(CCCNC(c1c(C)cncc1)=O)C C1(N(C(=O)CCC2CCCO2)CC)CCN(C(=O)CC(C)C2CCCCC2)CC1 c1(CC=C)cn(CC2CCC(NC(=O)CCSC)C2)nn1 Cc1ccnnc1C(=O)NC(C)CN(C(=O)CSc1ccccc1)C CN1CCCCC1CCC(=O)NC1CCOCC1NC(c1cnsn1)=O C1(C)(CC)CCC(C(=O)NCC2(F)CC(NC(c3cscc3Cl)=O)C2)O1 C1(NC(Cc2cc(OC)ncc2)=O)CN(C(c2ccc(C)s2)=O)CCC12CCC2 c1(C(C)NC(CCCC2(NC(c3cnc(CC)s3)=O)CCC2)=O)[nH]c(C)nc1C Cc1c(NCCOC2CCCC2)ncnc1NCC1CC(C)OC(C)C1 c1(SCC)nccnc1C(=O)NCC12COC(CNC(=O)CC(F)(F)F)(C1)C2 C1(NC(C=Cc2ccc(SC)s2)=O)CN(C(=O)COC2CCCCC2)CC1(C)C c1(C(=O)NCC2(C)CCN(C(C3CC(C#C)(O)C3)=O)C2)cc(F)c(O)c(F)c1 CCCC(CCC)CC(=O)N1CCOCC1CN(C)C(c1c[nH]cc(F)c1=O)=O Cc1nsc(N)c1C(=O)NC1CCCC(NC(=O)COCCOCCO)C1 c1(C(=O)NCCNC(C(C(C)SC)O)=O)ccc2nc(C(F)F)[nH]c2c1 CCC(CC)(C(=O)N1CCCC(NC(=O)CN2CCP(C)(=O)CC2)C1)OC C(C#N)(c1nc2ccccc2[nH]1)=CC(=O)N(c1nc2c(o1)CCSC2)CCC CC1CN(C(=O)C(c2cn(C)nn2)NC(C2C=CCS2)=O)CC1CO C1(N(C(c2csc(-c3ccco3)n2)=O)Cc2cn(CCF)nn2)CCN(CCl)CC1 c1(CC(=O)N(CC(C)NC(C2ON=C(CC)C2)=O)CC)csc2ccc(C)cc12 C(=O)(CC(C)NC(C1CCN(CCCO)C1)=O)OC c1(C(=O)NC(C)C=CC(=O)NC2CC(C(N)=O)C2)ccc(N)c(F)n1 c1(CC)cc(C(=O)N(CC(C)(C)NC(C2CC(SC)C2)=O)C)cc(O)n1 c1(C(N2CCN(CCC#N)CC2)=O)cn2cc(Cl)cc(Br)c2n1 c1(NC(CC2CC(=O)OC2)=O)nc2c(s1)CC(C(=O)O)CC2 Cc1ccc2cc(C(=O)NCC3CC3CNC(c3[nH]c(O)nc3C)=O)[nH]c2c1 CC(C)CCC(=O)N(CC(C)NC(c1cnn(C(C)C)c1C1CCCC1)=O)C C1(C(=O)NCC2N(C(CC3(C=C)CCCCC3)=O)CCC2)CC2(CCCCC2)C1 C(=O)(CCCCCCNC(=O)CCOC(C)C)NCCC1CC(C)C1 C1(OC)CN(C(=O)C=CC=Cc2ccccc2)CC1NC(=O)C(C)(F)F Cc1c(CNC(=O)Nc2nnn(C)c2C(F)(F)F)cccc1O N1(C(CCSCCCC)=O)CCOC(C(C)NC(c2cc(COC)oc2C)=O)C1 C(=O)(C(C(C)C)NC(c1ccccn1)=O)N1CC(CNC(c2c(C)cco2)=O)C1 N1(C(C(CC#C)C)=O)CCCC(F)(CNC(=O)C(CCSC)NS(=O)(=O)CC)C1 c1(C(=O)NCCCOCCN(C)C(c2cnc(S)nc2)=O)cc(F)cc(N)c1F Cc1ccnc(C(=O)NCC2(F)CCCN(C(C3(C)CCCS3)=O)C2)c1F C(=O)(C#CC1CCCCC1)N1C(CNC(=O)Cc2ccno2)CC(COC)C1 C#Cc1cc(F)c(C(=O)NCCC(C)NC(c2cnnn2C)=O)c(F)c1 N1(c2[nH]c(=NCC3CC=CC3)cc(C)n2)CCc2c(ccc(Cl)c2F)C1 c1(OCCOC)ccc(-c2nc(C(C)C(C)O)n(-c3ccc(CO)cc3)n2)cc1 N1(C(=O)Nc2cccnc2Sc2ccccc2)CCCC12CCCC2 C1(NC(C(CC)c2cccnc2)=O)CN(C(C2CC(C)=NO2)=O)CC2(CCC2)C1 C=CC(C)(C)CCNC(=O)C(C)(CSC)NC(=O)C=C1CCC1 Cc1ccc(C(=O)NCC(CC2CC2)C(=O)NC(CCO)C(C)(C)O)cc1O Cc1noc(C(F)F)c1C(=O)NC1CCCN(C(=O)CC2CCCN2C)C1 c1(C(N2CC3(CN(C(C4CC4C4CCCC4)=O)C3)C2)=O)sc2sccc2c1Cl c1(OCCC#C)cc(F)ccc1NC1CCN(OCc2cccc(Cl)c2)CC1 c1(CNC(C(CCOCC)NC(=O)C(C)CO)=O)cc(C)cnc1O Cc1nn(CC(N2CCCCC2CN(C)C(C23CCC2CC3)=O)=O)cc1Cl C(=O)(C(C)(O)COC)N1CC(CC(=O)NCCc2cnc(C)[nH]2)(OC)C1 C(N=c1ccnc(NC2CCCC2C(C)C)[nH]1)c1ccc(NC(C)C)cc1 C1(c2ccccc2)(NC(C(COC)C)=O)CCN(C(=O)Cc2cnc(C)[nH]2)C1 c1(NC(=O)NC)ccc(C(=O)NC2(c3cncs3)CC2)c(O)c1.c1ccco1 c1(OCC)ncc(C(=O)NC2(CNC(=O)CCc3cc[nH]n3)CCCC2)cn1 C(C)(N=c1[nH]c2cc(F)ccc2o1)C1N(C(CC(=O)NC)=O)CCCC1 C(=O)(C(CCC)S(N)(=O)=O)NCCC(=C)CNC(C1CCC(C)(C)C1)=O N1(C(C(COC)OC)=O)CCCCC1CNC(=O)CCCCN(C)C C(CC(=O)C1=C(c2ccccc2)OCCC1)N(C)Cc1ccc(C#N)cc1O C#Cc1ccc(C(=O)N(CC(C)CNC(=O)C=COCC)C)cc1C c1(C(NS(N(CCCOC)CCC#N)(=O)=O)C)cc(F)c(F)c(F)c1 Cc1nc2cccc(C(N3CCC(C)(C)C(NC(c4cocc4C)=O)C3)=O)c2[nH]1 N1(C(CCC2(C)CC2)=O)CC(NC(c2nnc(O)nc2O)=O)C2CCCC12 N1(C(C=C=C(C)C)=O)CC2(CCC2)CC1CNC(=O)CCCn1ccnc1C Cc1c[nH]nc1C(=O)NC(Cc1cn[nH]c1)C(=O)NC(c1cnn(C)c1)C C#Cc1ccc(C)c(NC(=O)C(CCOC)NC(=O)C(CC=C)OC)c1 c1(C(=O)NCC2N(C(C=CC(=O)OCC)=O)CC2)c(C)c(C)cc(C)c1C C(=O)(C1=NN(C)C(=O)CC1)N1CC(n2ncc(NC(c3noc(C)c3C)=O)c2)C1 N1(C(C23CC(OC)C2C3)=O)C2CCC1CN(C(=O)Cc1cc(Cl)cnc1C)C2 Cc1cnc(C=CC(N2CC(C(C)NC(=O)C=C3CCC(C)C3)C2)=O)[nH]1 Cc1c(C(=O)NCCC(C)(C)CNC(=O)C(C)CC(N)=O)sc2[nH]cnc(=S)c12 C1(NC(C2N(CC)CC2)=O)C2CC3CN(C(c4[nH]ccc4C)=O)C1C3C2 CCC(C)C(C)C(=O)N1CC2CC1(CNC(=O)CCC(C)(C)F)C2 c1(-c2cn(CC(CCNC(C3C(F)(F)C34CCC4)=O)F)nn2)cccc(F)c1F Cc1cc(C(N2CCC(C3CCCO3)C2)C(=O)NCCC2(C)CC2)c(C)o1 CC1(C)CN(C(=O)CCC2CCCCN2C(=O)C#CC2CCC2)CCS1 c1(C(=O)NC2CC(CNC(C3(CC#C)CCOC3)=O)C2)cccc(N(C)C)c1 c1(C(C(=O)NC2C(CNC(C(C)=C(C)C)=O)C2)(F)F)ccc(C)cc1 N1(C(CNS(N)(=O)=O)=O)CCN(C(=O)Cc2ccns2)C2(CCC2)C1 N#CC1(C(=O)NCC2CCCC(CNC(=O)Cc3cc[nH]n3)C2)CC2CC2C1 CC1(CNC(C2(C)CCCO2)=O)CCN(C(C2(C3CCCCO3)CC2)=O)C1 N1(C(CC2CCCN(C)C2)=O)CCC2C1CCN2C(c1cc[n+]([O-])cc1)=O CC1(C)CC(CNC(=O)Cc2c(F)cccc2Cl)N(C(=O)Cc2cnc[nH]2)C1 c1(C(=O)NC2(CC=C)CN(C(c3ccsc3SC)=O)C2)n[nH]c2c1CCSC2 N#CC1CN(Cc2c(F)cccc2F)CC1NC(c1cccc(O)c1O)=O N1(C(c2c(CC)nc[nH]2)=O)CCCN(C(C2CS(=O)(=O)CC(=O)N2)=O)C(CO)C1 C12(C(N3C4CC(NC(Cc5c(C)cccc5)=O)C(C4)C3)=O)CC(C)(C1)OC2(C)C c1(OC)ccc(OC)c2sc(N3CCC(C(C)NC(C4(N(C)C)CC4)=O)C3)nc12 C1(=CCNC(c2scnc2Cl)=O)CCN(c2nc(Cc3ccccc3)ns2)CC1 CC(O)C(C(=O)NC1(C)CN(C(=O)CC(=O)NC2CC2)C1)NC(=O)C(C)(C)C CCCC(C#N)C(=O)N(C1CC2(C1)CN(C(C1(OCC)CCCC1)=O)C2)C C(CCC(O)C(=O)Nc1cccc(CC)c1)NC(CCSCCCC)=O c1(C(CC)=O)cc(NC(=O)C(OC)OC)ccc1Cl.N12CCCC(C1CC)C2=O N1(C(C2CCN(C(c3cn(CCC)nc3)=O)CC2)=O)CC(C)CCC1CC c1(CC)ccc(C(=O)NCC2CCN2C(=O)C(c2cnn(C)c2)C)cc1 c1(CC(=O)N(CCNC(CC2(C)CC2(F)Cl)=O)CC2CC2)ccc2nn[nH]c2c1 N1(C(=O)CCc2c(Cl)cncc2Cl)CC2CCCC(C1)N2C(C1CCCO1)=O N1(C(C(C)N(CC(F)(F)F)C)=O)CCC(NC(=O)C(C)CC2CCCC2)C1C c1(C(N2CCCC(C)(CNC(C(CC)(C)CO)=O)C2)=O)cc2c(cn1)OCCC2 C1(C(=O)NC2CCN(C(=O)C(Cl)=CCl)C2)CC2CCC(C1)C2O N1(CCc2c(OC)cccc2)CCC(=O)N(Cc2nnn(C)n2)C1=O C#Cc1ccccc1CN1CCC(C(=O)Nc2ccnc(C3CC3)c2)CC1 CCCC(CC)C(=O)NC1(C)CCN(C(=O)CNC(c2ccco2)=O)C1 Cc1nc(NC(c2[nH]cnc2C#N)=O)ccc1-c1cncc(O)c1 N1(C(=O)OC(C)(C)C)CC2(CCCC(CC(=O)OCC(=O)C3CCC3)O2)C1 Cc1cc(C(N2CC(N3CC(NC(c4occc4C)=O)CC3=O)C2)=O)ccc1Cl c1(C(N2CC3C(CNC(=O)CC4CCCO4)(C3)C2)=O)cc(Cl)cc(Cl)c1O C(CN=c1ccnc(N2CCC(C3CCC3)C2)[nH]1)OCC(c1ccccc1)C Cc1cc(NC(c2ccncc2Cl)c2nnnn2C(C)(C)C)ccc1F N1(C(c2ccnn2CCF)=O)CC2CCC1CN2C(C1CCn2nncc2C1)=O Cc1c(CNC(C)CC(C)(C)O)c(C(F)(F)F)nc2[nH]nc(O)c12 c1(-c2nn(CCOC(C)C)c(Cc3cccc(Cl)c3Cl)n2)cccc2scnc12 CCC(CCC(=O)NC(c1cscn1)CO)NC(c1ccc([N+](=O)[O-])o1)=O c1(C(=O)NC(CC)CNC(c2ccc(OC(C)(C)C)cc2)=O)ccc(F)cc1C N1(C(C2CCC(CNC(C(CCOC)OC)=O)CC2)=O)CC(OC)CC1(C)C C=CC(C)(O)CC(=O)NCC1CC(NC(=O)CCNS(C)(=O)=O)C1 CC1CC(CNC(C2CCC23CCC3)=O)CCN1C(c1ccco1)=O C1(CCCNC(C=CC(=O)OCC)=O)CN(C(=O)CC2CCOC2=O)CCO1 c1(C(=O)NCCCNC(=O)Cc2cnccc2Cl)cc(Cl)cc([N+](=O)[O-])c1 N1(C(C(CC)c2ccccc2)=O)CC2CCOC2(CNC(=O)CC2CCC2C)C1 CC1CC2(CCN(C(c3ccc(Cl)[nH]3)=O)CC2)CN1C(c1cocn1)=O C1(NC(COCCOCC#C)=O)CCCCC12CCN(C(c1cnc[nH]1)=O)C2 N1(C(CC(CC)(F)F)=O)CC2CCN(C(C3Cc4nc(C)cn4C3)=O)CCC2C1 CCC(O)C(C)C(=O)N1CC2CC(C1)C2NC(=O)CCCCCN(C)C c1(C(N2CC(C(C)NC(c3cnn(C4CC4)c3)=O)C2)=O)ccc(N)cc1O CC(C1COc2ccccc21)NC(=O)C(C)c1nccs1 CCCC(CCC)=CC(=O)NCC1C(C)CCN1C(c1cnoc1)=O N1(C(CC2C(NC(C(CC=C)OC)=O)CC2O)=O)CCN(C)CC1CCO c1(OC)ccc(C(F)(F)C(=O)NCC2CCN(C(c3cc(C)co3)=O)C2)nc1 CCCCCC(O)C(=O)N1CCCC1(C)CNC(c1cccc2ccoc12)=O N1(C(c2nccc(OC)c2)=O)CCOCC(NC(=O)CC23CCCC2C3)C1 c1(C(C)NC(C)C(=O)N(C)C(c2ccc(C#N)cc2)C)ccc2ccccc2c1 c1(C(=O)NC2CC(O)C2)cc2[nH]ccc2cc1-c1cc(CO)ccn1 O=C(CCNCC(F)(F)F)NOCCc1ccccn1 CCN=C(NCC12CC(CC(F)F)(C1)C2)N1CC2CC=CCC2C1 C1(NC(c2cnc3sccn23)=O)CCCN(C(=O)C2=C(Cl)CCCC2)CCC1 CCCCC(CNC(C1CC(C)(C)CO1)=O)NC(=O)Cn1cc(CO)nn1 c1(OC)ccc(S(=O)(=O)N2CCCC2)cc1NC(c1cnc2c(Br)n[nH]c2c1)=O C1(CC(=O)NCCCOCCN(C(CN(C)CC)=O)C)CCCCO1 C(c1ccc(Cl)cc1F)=CC(N1CCC2(NC(C=CC=CC)=O)C(C1)C2)=O C1(N(C(c2scc(CC)c2)=O)CC)CCCN(C(C2C(C)C2C)=O)CC1 C1(C(=O)NC2CC2CNC(=O)Cc2cncc(F)c2)(OC)CCSCC1 c1(C(=O)NC(CNC(CSCC#C)=O)(C)C2CC2)cc([N+](=O)[O-])ccc1NC c1(C(=O)NCCC2N(C(C(CO)NC(N)=O)=O)CCCC2)nccc2n[nH]cc12 c1(C(=O)NCCC(C)NC(C(CC)(C)OC)=O)cc2c(o1)CCCC2 N1(C(C(C(C)C)(C)O)=O)CCC2(CC1)CN(c1ncc3ccsc3n1)CCO2 c1(CC)n[nH]c(CC)c1CC(=O)NC1CCN(C(=O)COC2CCCCC2)C1 C(N=C(NCc1nc(-c2ccco2)n[nH]1)N1CCCCC1)C1C(O)CCCC1 c1(N)nc(=NCCSC(F)F)[nH]c2cc[nH]c12.C1(=CC=C(C)C)CCCC1 N1(SCc2c(Cl)ccc(OC)c2)C(=O)NC2(CC(C[Si](C)(C)C)C2)C1=O O=S(=O)(c1cccc(=NCCCc2ccc(CO)cc2)[nH]1)N1CC2CCC(C1)O2 C1(NC(C2C(CCOC)C2)=O)CCN(C(c2cnn3c2OCCC3)=O)CC(O)C1 C1(NC(c2cccc(C(C)=O)c2)=O)CCN(C(c2ocnc2C)=O)CC1C CC1=C(C(=O)NC2CCC(N(C)C(C3CC3C3CC3)=O)CC2)CCS1(=O)=O C1(C2CC2)(C(=O)NCc2c(C)cccn2)CN(C(c2cc(=N)[nH][nH]2)=O)C1 Cc1cc(C(N2CCCC2CNC(C2CCCC(F)C2)=O)=O)c2c(c1)CCCN2 N1(C(CCOCC)=O)CC(N=c2[nH]ccn3nnnc23)C(C)(C)C1 c1(CC)nc(C)ncc1C(=O)NC1CN(C(=O)CC2CCCO2)CC1(C)C C1(NC(c2cc(C)nc(O)c2)=O)CCCOC12CCN(c1nnco1)CC2 CCCC(C)(C)CC(=O)NC1CC(NC(C2(F)CCCN(C)C2)=O)C(O)C1 c1(C(=O)NCC(CC(C)C)NC(C2CCC(C)(C)OC2)=O)cc(Cl)c(Cl)cc1N c1(OC)ccc2c(c1)OCCC2C(=O)Nc1cc(C)c(F)cc1C CCCC(C)(O)C(=O)NC1CC(CNC(c2ncncc2Br)=O)C1 C#CC1(O)CCN(C(C2CCN(C(=O)Cc3sccc3C)C2C)=O)C1 c1(C2(C(=O)NC3CCN(C(C(COC)O)=O)C3)CC2)nn(-c2ccccc2)cc1C C1(C(N(C(C)C(N)=O)C)=O)(CNC(C2CC2Cl)=O)CC12CCC2 Cc1ccc(C(N2CC(F)(F)CC2CCNC(C2CCN(C)C2=O)=O)=O)c(N)n1 c1(CN(c2nc(C)c(Br)cn2)C2CNCC2F)ccc2cccnc2c1 c1(CC)nnc(CSCC2CC2)o1.c1(C2c3nnnn3CCCN2)csc(Cl)c1 c1(C(N2CCC(N(C(c3cnn(CCC)c3C)=O)C)C2)=O)cnc(O)n(C)c1=O Cc1nn(C)c(C(F)F)c1C(=O)NC(CNC(C1(CO)CCCO1)=O)CC(C)C C1(NC(C2(C)CCOCC2)=O)Cc2ccccc2C1NCc1ncnn1CCF c1(C(N2CCC(NC(COCCCC)=O)C(C)C2)=O)c(F)cc(C)cc1Cl C1(CNC(C2(C=C)CCC2)=O)C(C2CC2)CCN1C(=O)C(O)C(C)(C)CC C1(CN(CC(=O)O)Cc2cc(Br)cs2)CC2(CCOC2)C1 Cc1sc2ncn(CCCC(=O)NC(C)CN(C)C(C3CSC3)=O)c(=O)c2c1C c1(C(=O)NC(CCN(C(C(C)OCCC=C)=O)C)C)cc(C(C)C)nc(O)c1 N1(C(C(CCSC)NC(C)=O)=O)CC(C(=O)Nc2ccc(F)c(C)n2)C2(CC2)C1 Cc1cc(C)c(CC(N2CCC(C)(CNC(=O)C(C)NS(C)(=O)=O)C2)=O)s1 CCCC(C#N)C(=O)NC(C)(C)CCC1CCN(C(=O)C=C(C)C(F)F)CC1 c1(C(N2CC3C(CNC(C4(N(C)C)CC4)=O)(CC3)C2)=O)cc(C#N)ccc1Br C(=O)(C(C)S(C)(=O)=O)N1CC(n2cc(CCCC=C)nn2)C(SC)C1 c1(C(=O)NCCC(CNC(c2cc3ccccn3n2)=O)O)ccc2nc[nH]c2c1 C1(C(=O)NCC2CN(C(C3CC(C)SCC3)=O)CC2C)CCCC12CCOCC2 Cc1cc(N2CCCOCC2)ncc1S(=O)(=O)N(C)CC1CCCC1(C)C O=CN1CCCC1C(=O)NC(Cc1cc[nH]n1)C(=O)NC1CC(CO)C1 C(CCCC(C)(C)C(=O)NNC(=O)C1CC1F)NC(C1=NN(C)C(=O)CC1)=O N1(C(C2C(CC(C)(C)C)C2)=O)CC2CCC(C1)N2C(C1(C)COC1)=O Cn1c(C(=O)NC2CC(NC(c3conc3C3CCCC3)=O)C2)cnc1[N+](=O)[O-] CC(C)C(C(=O)NC1C2CCC1CC2)C(C)NC(c1cnn(C)c1N)=O Cc1cc(=O)c(C(=O)NCC23CC(CO2)N(C(c2cnc(C#N)s2)=O)C3)cn1C c1(OC)nc(Cl)ccc1C(=O)NC1CCCN(C(=O)C(O)C2CC2)CC1 c1(C(=O)OC)nc(C(=O)NCC2CC(NC(=O)CCNC(=O)CO)C2)cs1 N1(C(CC2CN(C(C(CC)C)=O)CC2O)=O)CC2CC1CN2CC C1(F)(CNC(C(c2cnn(C)c2)OC)=O)CCCN(C(c2ccn(C)c2)=O)C1 C#CC1(C(=O)NCCC2(C)CCN(C(c3ccc(CCC)[nH]3)=O)C2)CCCC1 N1(C(C(C)CSC(F)(F)F)=O)CCC(NC(=O)C(=O)Nc2ncc[nH]2)C1C1CC1 c1(C(c2n(CC=C)c(N3CC(OC)CC(O)C3)nn2)(F)F)ccc2c(c1)COC2 C1(C(=O)NC2(C)CC(F)C2)(CC)CCCN(C(=O)CCN=[N+]=[N-])C1 c1(C(=O)NC2CCC(NC(C=NOC)=O)CC2)ccc2ccccc2c1 Cc1ccc(CC(=O)NC2CCN(C(c3cccc(C(N)=O)n3)=O)C2)c(F)c1F N1(C(c2c(NC)cncc2)=O)CCCN(C(c2ccc(F)cc2F)=O)C(CO)C1 C1(CC#N)CCN(C(=NCCC2COCC2O)NC2CC2)CC1 C1(C(=O)OCC)(C(=O)NC2CCCC2NC(c2ccc(OC)s2)=O)CCCCC1 Cc1cn2c(CCC(N3CC4CC3(CNC(C3CCC(F)C3)=O)C4)=O)csc2n1 N1(c2nc(N3CC4CC3CS4=O)cc(C)n2)CC2(CCOCC2)CC1CO N1(C(C(=O)Nc2ncc[nH]2)=O)CC2CC1C2NC(c1ccccn1)=O c1(C(=O)NC(C2N(C(c3occ(C)c3)=O)CCCC2)C)c(C)nn(C)c1F N1(C(C=CCC)=O)CCC(C2CC2NC(=O)CN2CCCCC(OC)C2=O)CC1 N1(C(CC2C(C)(C)C2)=O)CCC(OCCNC(=O)CCc2ccsc2)C1 C1(NC(c2ccc(CC)o2)=O)CN(C(=O)Cn2cc(F)ccc2=O)CCC1F C12(C(=O)NC(CNC(c3c(C)cccc3)=O)CO)OCCCC1C2(F)F c1(OC)cc(N)ccc1C(=O)NC1CCC(CNC(C2CC=CCC2)=O)C1 c1(-c2c(C(N3CCN(C(C)=O)CC3)=O)cccc2)nccc(C(F)(F)F)n1 c1(C(=O)NC(C)C(CO)NC(=O)CCC2CC2)ccc(N2CCOCC2)nc1 c1(C(N2C(C)CNC(=O)C2)=O)cc(O)nc2c1CN(C(C1CC1F)=O)CC2 c1(C(N2CC(CC)(NC(c3ccncc3OC)=O)C2)=O)ccc2nccnc2n1 CC1NC(=O)OC12CN(C(=O)CC(C(F)(F)F)NC(=O)CC(Cl)Cl)C2 c1(C(N(C(CNC(COCCC#C)=O)C2CC2)C)=O)cc(Cl)c(Cl)s1 C1(CNC(C(C)OCCN(C)C)=O)N(C(C2CCC(=O)N2C)=O)CCCC1(C)C Cc1c(N)cc(C(N2CC3CC(NC(c4ncn(C)n4)=O)C3C2)=O)cc1N Cc1nn2c(C(=O)NCCNC(=O)Cc3cccc(Cl)c3Cl)c(C)nc2s1 c1(C(=O)NCC2(NC(C(C3CCC(=O)N3)C)=O)CC2)ccc(Br)c(O)n1 C(C(CCC)C(=O)N1CC=CC1CF)NC(CC1C(CC)C1)=O c1(C(N(C(CNC(Cc2c(C)cnn2C)=O)C)C)=O)cc(F)cnc1O c1(CCC(=O)NC(C2CCCC2)CNC(c2ccoc2Cl)=O)cc(Cl)cs1 N1(C(C2(C)CNC(=O)C2)=O)CCC(O)C(NC(c2cccc(C3CC3)c2)=O)C1 N1(CC(N2CCC(C)(NC(C=Cc3ccc(CC)o3)=O)C2)=O)CC(=O)N(C)C1=O N1(C(C2CN(CC)C(=O)C2)=O)CCN(C(=O)Cc2cncn2C)C(C)C1 C#CC1(C(N2CCCC(CCCO)C2)=O)CCN(C(=O)C=CC2CCCN2C)C1 C1(NC(C2(OCC)CCC2)=O)CN(C(C2CCOCC2(C)C)=O)CC2(CCC2)C1 Cc1ccc(C(=O)NC(C2CCN(C(=O)Cc3nonc3C)C2)C2CC2)nc1 c1(COC)nc(C)cc(=NC2CN(C(=O)CCn3cccnc3=O)CC2C)[nH]1 C1(C(=O)NC2C(C(=O)NCCc3c(C)cncc3)CCCC2)CC2(C1)CC(C)C2 N1(C(C(c2ccccc2)NC(c2ncn(CC)c2)=O)=O)CCOC(C)CC1 N1(C(Cn2c(=N)nn[nH]2)=O)CCN(CC2CC2(F)F)CC1 N1(C(C2(C=C)CCC2)=O)CCCCC2(CCN(C(=O)Cc3cnns3)C2)C1 C(C(CO)(CO)NC(=O)C(C1CC1)OCC)N(C(CCCOCC)=O)C N1(C(CN(C)CC)=O)CC2(C1)C(NC(C13CC(C)(CO1)C3)=O)CCS2(=O)=O C12(C(=O)NC(C3CCN(C(c4cnn(C)c4)=O)C3)C)CCCC1C2(F)F N1(C(CCCC(=O)NC(C)C)=O)CCC(NC(c2cn[nH]c2)=O)C(CO)CC1 c1(C(=O)NCC(C)(C)NC(c2cn(CCOC)nc2C)=O)cc(O)nc(O)n1 N1(C(C2(CCOCC)CCC2)=O)CC(NC(=O)C(F)(F)COC)CC(O)C1 CC1(O)CCN(c2cc(NC3CC4CC3CC4(C)O)ncn2)CC1O C12(C(=O)NCC(CNC(c3cncc4nc[nH]c34)=O)O)C(=O)C3CCC1C2C3 N1(C(C(C)CSC(F)(F)F)=O)CCC(NC(c2ncoc2C2CC2)=O)C12CC2 C(=O)(CCC(C)(F)F)N1CCC(CNC(C(C)C)=O)(CO)C1 c1(CC(N2CCC(O)(CN(C(C(C)NC3CC3)=O)C)C2)=O)cnn2c1CCCC2 n1(SCC)nc(C)cc1C(=O)OC(c1nc(-c2ccccc2C)no1)C N1(C(C(COC)COC)=O)CCN(C(=O)CNc2cccc(C)c2C)C(CF)C1 c1(C(N2CC(CC(C)NC(c3cc(Cl)on3)=O)C2)=O)sccc1CC#N C1(F)(C(N(C2(COC)CC2)C)=O)CCCN(C(C2(C)CCCCO2)=O)C1 c1(NC(C(=O)NC2CCN(C(CC(=O)OCC)=O)C2)(C)C)cc(Cl)ccc1F c1(CC(=O)NCCC2(C)CCN(C(C3CC(C)C3)=O)C2)ccc2c(c1)OCO2 C(=O)(CC1=CCOCC1)N(C)CC1(CNC(c2ccn(C3CC3)n2)=O)CC1 C(=O)(CCCCC(C)(C)C)N1C(C)(C(=O)NC(C)CCC2CCCC2)C=CC1 CC1CCN(C(c2cc(C3CCOCC3)[nH]n2)=O)C(C)C1NC(=O)COCCO N1(C(C=CCCC)=O)CC(NC(=O)Cc2cnn(C)c2)CC12CCCC2 CCCC(CNC(=O)C=Cc1cc[nH]c1)C(=O)NCc1ncc(CC)o1 c1(CC)nc(NC2CCN(C(c3c(OC)ccnc3O)=O)CC2)c2ccsc2n1 c1(NC(C2CC3CC3N2S(=O)(=O)CCCCl)=O)ccc(Cl)cc1I N1(C(=O)Cc2cc(=O)n(-c3ccccn3)[nH]2)CCc2ncc([N+](=O)[O-])cc2C1 c1(CC(N2CCC(NC(C3CCC(C)S3)=O)CC2)=O)ccc(S(N)(=O)=O)s1 Cc1cc(=NC(=O)C2CC(C)CN2C(c2cccc(Br)n2)=O)[nH]c(C)c1C#N N1(C(C(C)N2CCCC2)=O)CC=C(CC(=O)N2CCC(C)C(CO)C2)CC1 C12(CNC(=O)C3=CCCC3)CCC(Nc3ccnc(CO)n3)(CC1)CO2 c1(OC)ccc(CN=C(NCc2nnc(SC)s2)NC2CC2(C)C)cc1 C1(CCNC(CC(C=C)C)=O)CN(C(=O)CC2CCCCCCC2)CCCO1 N1(C(c2cc(C(=O)OC)on2)=O)C2CCC(C2)C1CNC(c1ccc([N+](=O)[O-])o1)=O c1(CNc2c(C(N3CCCC3CO)=O)cc(OC)nc2)cc(Cl)c(O)cc1F c1(C(NC=O)C2CC2)cn(CC2CCCN2C(C2C=CCS2)=O)nn1 Cc1ccc2c(=NCCc3cccnc3Cl)[nH]c(=NC(C)C3CCC3)[nH]c2c1 CC(c1cccc(Cl)c1)=CC(N1CC(NC(c2ccoc2C)=O)CC1C)=O N1(C(C(CC=CC)C)=O)C2CCC1CC(N(C(=O)Cc1cccc(OC)c1)C)C2 c1(OCC)ccc(C(F)(F)F)cc1NC(=O)Nc1ccnn1C1CCOCC1 CN1CCCC1C(=O)NC(C)(CNC(C1CCSC1)=O)C1CC1 c1(C(C)NC(C2(NC(COCCCC(C)C)=O)CSC2)=O)ccc(O)cc1 C1(NC(C(COC)C)=O)CCN(C2CCN(C(=O)Cc3cscc3F)CC2)CC1 CC1=C(C(=O)NC2CCN(C(C3CCCN3C)=O)C2)CCC1 N1(C(C)=O)CCCC1C(=O)NC1(C2CCCN2C(=O)C=CC(C)(C)C)CC1 C(=O)(C1=CCC(C)(C)CC1)NCC1C(NC(CC2CC(=C)C2)=O)COC1 c1(CC)c(NC(C2(NC(=O)C(C)N3CC(C)C3)CCCC2)=O)cnn1C CCCCCC(CC)C(=O)N1CCCCC(NC(=O)Cc2c(C)cccc2C)C1 C=C=CC(C)C(=O)N1CC(OCCNC(=O)CC2CN(C)C2)C1 C(C1=CCN(C(=O)CCC2CC2)CC1)NC(C(c1ccccc1)NC(C)=O)=O N1(C(C(CCCC)F)=O)CCOC2(C1)CN(C(=O)CN(C)CC)C2 Cc1cnc(C=CC(=O)NCC(C2CN(CC3C(C(=O)NC(N)=O)COC3)C2)O)[nH]1 CC(C)CC(C(=O)N1CCOCC1Cc1cn(Cc2cccs2)nn1)N(C)C c1(C(N2CCC(C(N(CCCC(=O)OC)C)=O)CC2C)=O)cccn2nccc12 N1(C(c2n(CC)nnc2)=O)CCCC(C)(NC(=O)CCc2cnco2)C1 C(=O)(C(C)(C)C(F)(F)F)N1CCN(C(c2cncc(OC)n2)=O)C(C2CC2)C1 c1(C(N(C)CC2N(C(CCOCCCOC)=O)CCOC2)=O)cn2c(n1)SCC2 N1(C(C2C(CC)OCC2)=O)CCCC2(CCN(C(c3n[nH]c(C)c3F)=O)C2)C1 C(CC)(CC)(CCNC(=O)Cn1ncn(C)c1=O)NC(C=CCCC)=O C(c1c(F)ccc(Cl)c1F)=CC(=O)NC1C(NC(C(C)c2cccs2)=O)CC1 Cc1nn(C)c2c(NCCN3CCCC3C)nc(N3CC4C(C3)C4(C)C)nc12 c1(C(=O)NCCN(C2CCCCC2)C(=O)C2CC2)cccc2c1NCCC2 N1(C(C(F)OC)=O)CCC(CNC(c2ccccc2C2CC2(F)F)=O)C12CC2 N1(C(C(C)Cc2ccnn2C)=O)CCSCC1CCNC(c1cnsc1)=O C(=O)(C(C)(C)CCC#N)N1CC(C(C)NC(=O)CN2CCSCC2)OCC1 C1(NC(=O)NC(CN(CCCC)C)(C)C)CCCC(O)C1 C(CCO)(CC(C)C)NC(C1(NC(c2c(OC)nn(C)c2)=O)CC(O)C1)=O C1(C2CCCN(C(=O)C=C3CCSCC3)C2)(NC(C(CC)C(C)O)=O)CC1 CCC(O)C(C)(C)C(=O)NCC1CCN(C(c2cc(C)n(C)n2)=O)CC1(F)F C1(CCNC(c2ccn(CCN(C)C)n2)=O)CCCN(C(c2coc(Cl)n2)=O)C1 N1(C(CNC(C2C(C)C2)=O)=O)CC=CC(NC(c2ccc(CC(N)=O)cc2)=O)C1 C1(C(=O)NC(C(=O)OC)CC2CC2)CC2CC2N1C(=O)COCC(=O)NC c1(C(N2C(CNC(C(C(C)C)OCC)=O)CCCC2)=O)cc(=O)n2ccsc2n1 C1(N(C)C)(C(=O)NC2CCC(NC(C3OCC3(C)C)=O)CC2)CCCOC1 c1(-c2cccc(SC)c2)ccc(NC(=O)N(C(C)C)Cc2ccccc2)nc1C C(C)(CCCC(=O)N1OC2CC1C(O)C2O)NC(c1c(C)n[nH]c1)=O N1(C(N(CCC)C(C)C)=O)CCCC(C(=O)NCC(CC)n2cccn2)CC1 C(=O)(CCC(C)CN(C)C)N(CC(C)C)CC(=O)NC1CC2(CC2)CO1 c1(C(N2CCCC(C)(O)C2)=O)cn2c(n1)CN(Cc1cc(F)c(Cl)cc1F)CC2 N1(C(c2n(CCC)ncc2)=O)CCCCC1CN(C(=O)C(C)C1CCCC1)C C1(C(N2CC=CC(C(=O)NCc3ncnn3C)C2)=O)(OC)CCCCC1 c1(CN(C(=O)Cc2csc(Cc3ccc(Cl)cc3)n2)C)cn2cc(Cl)ccc2n1 c1(C(=O)NCC2(F)CC(NC(C(CSC)C)=O)C2)ccc2ncnc(O)c2c1 C(CCC(N)=O)(C(=O)N1CCC(NC(c2cc(F)c(Br)cc2C)=O)C(F)C1)OC c1(C(=O)NCC2(C)CC(NC(C3CCC(CC)CC3)=O)C2)nc(C)c(C)nc1C c1(C(=O)NC(CCCC)CNC(C2(C)COCCO2)=O)cncc([N+](=O)[O-])c1 c1(C(=O)NCCC2CC(NC(CSCCC(C)C)=O)C2)cn2c(n1)CCC(C)C2 c1(C(C(=O)NCC(=C)C)N(c2ccccc2)CCCC)cncc2ccccc12 c1(C(=O)NC2C(OC)CN(C(C3(C#N)CCCO3)=O)C2)cc(F)c(F)cc1Cl N1(C(C(C(=C)C)(C)C)=O)CC2CC(C(=O)NCc3ncnn3CC)CC2C1 n1(CCOC)ccc(=NC(c2csc(Cl)c2Br)c2nnnn2CC2CCOC2)[nH]1 Cn1ccc2ccnc(C(=O)NCC3CCCN(C(C4(C)CC=CC4)=O)C3)c12 N1(C(=O)CC2CC=CC2)CCN(C(c2cn3c(n2)CCC3)=O)C2CCCCC12 N1(C(c2c(C)snn2)=O)CC(CC(=O)N(C(C)CO)C2CC2)C2(CC2)C1 N1(CC)CCOC(C(=O)NCC=CCNC(=O)CCc2ncc[nH]2)C1 C(CNC(C1CCN(c2ccccc2F)C1)=O)(C(F)(F)F)OC C1(F)(CNC(C2CCSC2)=O)CN(C(=O)CCc2nc(-c3ccccc3)no2)C1 c1c(Br)cc(F)cc1Br.Cc1cccc(C(N)=O)c1NC(=O)NCC1CC(N)C1 CC1CCN(CCC(N2CC3C(CNC(C4CC(Cl)(Cl)C4)=O)C3C2)=O)CC1 C1(NC(c2scnc2C(F)(F)F)=O)CCOCC1NC(c1ncccc1F)=O c1(C(=O)NCC(C)(O)CNC(=O)C=CC(=O)N(C)C)ccc(Cl)c([N+](=O)[O-])c1 C1(CC(=O)NC(CC)CN(C)C(C2(N(C)C)CCCC2)=O)CCCC12CC2 Cc1ccc2ncc(C(N3CCCOC(CN=c4ccc(C#N)c[nH]4)C3)=O)n2c1 c1(CC(=O)NCCCOCCCNC(C2COC(=O)N2)=O)ccsc1Br C12(NC(COCCC=C)=O)CCC(CC1)N(C(c1cc(F)cc(C)c1N)=O)C2 c1(CCC)c(C(N2CC(CO)(NC(=O)C(n3nccc3C)C)C2)=O)cnn1C C1(C(N(CCN(C(=O)CC2C=CCCC2)C)C)=O)Cc2ccccc2O1 C1(C(N2CCC(C)OC(C)C2)=O)COc2cccc(F)c2O1 c1(C(N(C(C)CNC(C2CC2(C)C)=O)CC)=O)cnc(C(F)(F)F)s1 c1(CC(C)NCC(C2CCC3(CC2)CC3)=O)nc2ccccc2s1 N(C(=NCCOC(F)F)NCC1(C#N)CC1)C(C1CCOCC1)C C(=O)(C1=C(CC)OCCC1)NCCCN(C(C1(C#N)CCCOC1)=O)CC c1(C(N2CCC(CCOC)C2)=O)[nH]c(Cl)c(Cl)c1Br C1(NC(C(C)(C)CF)=O)COC2(CCN(C(C3CC3c3cccnc3)=O)CC2)C1 Cc1csc2ncc(C(=O)NCCCN(C(=O)C=Cc3ccoc3)C)n12 c1(C(N2CC(C)N(C(=O)C=Cc3cccn3C)CC2)=O)cnc2cc[nH]c2c1 C1(C(c2ccccc2)NC(=O)NC(C)Cn2cccn2)CC12CCOC2 C1(NC(CNC(CNC(C=C(C)C(C)C)=O)=O)=O)CN(C)C2(CCC2)C1 c1(C(N2C(C(=O)Nc3c(C)cc(F)nc3)C3CCC2C3)=O)cc2cccnc2[nH]1 c1(OCCC(=O)NC2(CN(C(=O)C(C)(O)C3CCOC3)C)CC2)ccc(Cl)cc1 n1(C(C)C)cc(C(=O)NCCCN(C2CCCC2)C(c2ccon2)=O)cn1 C1(C(=O)NC(CN(C(CCC=C(C)C)=O)C)Cc2ccccc2)C2CCC1CC2 c1(C(N(CCC(C(C)C)NC(C2CC(O)(CC#C)C2)=O)C)=O)csc2nccn12 C12(CNC(C3(OC)CCC3)=O)CCCN(C(=O)CCOCC(C)C)C1C2 N(C1CCc2cccnc21)C(C1N(C(c2ccc(OCC)cc2I)=O)CC1)=O C1(NC(CC2CC(COC)C2)=O)CN(C(c2cc3n(n2)CCO3)=O)CC12CC2 C=CC1COCCN1C(C12CC1CCN2C(c1cc[nH]c1)=O)=O c1(CNC2C(NC(C3CCN(C(C)=O)CC3)=O)CCCC2)c(F)ccc(F)c1O N1(C(C2CCC(=O)C2)=O)CCCN(C(C2OCC3COCCC23)=O)CCC1 C1(O)(CNC(c2cc(Br)ncc2Br)=O)CCCN(C(c2cnnc(O)c2)=O)C1 Cc1ccc(CNC(c2cc(CNC(=O)CCOC3CCCC3)cs2)=O)cc1C n1(CCCC(=O)N(CC)CC2CCCN2C(=O)CCCSC)nc(C)cc1C CC1CCC(C2CCC2)CN1C(=O)C(N1CC(C)(Cc2ccccc2)C1)=O C1(C(=O)NC(COC)C(=O)N(C)Cc2nncs2)C2CC3C(C2=O)C13 C(=O)(C(=O)N=S(C)(C)=O)NC1(C)CCCN(C(C(COC)N(C)C)=O)C1 c1(CN2CCCC(NC(c3cccc(Cl)c3Cl)=O)C2)cc(F)c(Br)cc1[N+](=O)[O-] CCC(C)(C)C(=O)N1CC(NC(=O)CCc2ncco2)C(c2cncn2C)C1 c1(C(N2CC(CNC(=O)OCc3ccccc3)C2)=O)cc(F)cc(F)c1F CC1Cc2ccccc2C1NC(=O)C(c1ccccc1)Oc1ccc(F)cc1 C(=O)(C(C)CCCC(C)=O)NC(COCC)C(N1CCCC2(C=CCO2)C1)=O c1(NC(c2cc(OC)ncc2-c2ccncc2OC)=O)cc(F)c2cc[nH]c2c1 C(=O)(CC(C(C)C)c1ccon1)NCC(CC)NC(c1cc(Cl)ccc1Cl)=O CC(F)(F)CCC(=O)NCCOCCCNC(c1ncnn1C1CCOCC1)=O N1(CCOCCCCCC)CCC(=O)N(Cc2csc(N(C)C)n2)C1=O c1(C(C)C)ccc(C(=O)NCC2CC(O)CN2C(=O)CC2CCCCC2O)nc1 CCCCCCC(=O)N1CC(CNC(c2n[nH]c(C)c2F)=O)OC(C(F)(F)F)C1 Cc1cc2c(cc1C)OC(C(=O)NC1CC(O)CN(C(=O)CCP(C)(C)=O)C1)C2 N1(C(c2c(O)cccc2Cl)=O)CCCC2C1CCN2Cc1cc(O)cc(F)c1 C1(CC(N2CC(CC(C#C)C)C2)=O)CN(C(=O)CC2(O)CCCCC2)CCO1 c1(NCC2(C)CC2Br)[nH]c(=NCCN2CCNC2=O)nc2sccc12 C1(NC(c2ccc(OC)c(Br)c2)=O)CC2CC1CN(C(=O)CNC=O)C2 N1(C(c2nc(NC(C)=O)sc2)=O)CC(CNC(C2(N(C)C)CCC2)=O)CC1C C(=O)(CS(=O)(=O)c1ccccc1C)NCC1CC2(CN(C(C(F)=C(C)C)=O)C2)C1 O=C(C(Cc1ccccc1)C(F)(F)F)OC1CC2OCCC12 C1(NC(C(=O)N(C)Cc2ccc(OC)cc2)=O)CC2(CCCCO2)C1 C1(NC(C(C)SC(C)C)=O)CN(C(c2ccc(CN(C)C)o2)=O)C2CCCCC12 C1(NC(C2CCC(C)O2)=O)CN(C(=O)Cc2ccoc2)CC12CCCC2 C(=O)(CCCC(F)(F)C(F)(F)F)N1C(CNC(=O)CCC(F)F)COCC1 C1(CNC(C)=O)CN(C(c2ccnc(NC3CCCN3N=O)c2)=O)CCN1C C1(CO)CC(N=c2nc3scnc3c(NCCc3ccc(C)c([N+](=O)[O-])c3)[nH]2)C1 c1(NC2(C3CN(C(C4C=CCCC4)=O)C3)CC2)nc(Cl)nc2ccccc12 Cc1cc(-c2nc(C(=O)NCc3ccc(C(C)C)cc3)ccc2F)cnc1O N1(C(=O)CCC2CCN(C(=O)C(F)C3CCC3)C2)CCc2ncccc21 CS(=O)(=O)c1cccc(C(N2CCC(NC(C3CCSC3)=O)C(O)C2)=O)c1 N1(C(c2c(C(C)C)nns2)=O)CCC2CN(C(c3ccc(N(C)C)nc3)=O)C2C1 C#CCCCC(C)C(=O)NCC(C)N(C(=O)CCCN1C(=O)CN(C)C1=O)C Cc1cc(C(=O)NC(CNC(=O)COCc2nnc(S)n2C)C2CC2)c(C)s1 N1(CCC)C(=O)CCC1C(N1CC(NC(c2cnn(CC)c2CC)=O)C(C)C1)=O CN1CC(C(=O)NCC(C2CCN(C(C3CC=CC(O)C3)=O)CC2)O)CC1=O Cc1ccc(F)c(C(=O)NC(C)CCCNC(C2CC2C(C)C)=O)c1F c1(C(N(CCCCNC(=O)CC2OCCC2(C)C)C)=O)cccn2[nH]c(=N)nc12 C1(C2CCOCC2)(CNC(CC)=O)CCN(C(c2cnc3n2CC(C)CC3)=O)C1 c1(C(N2CC(OC)(CNC(C3CCCC(C)CC3)=O)C2)=O)cc(Cl)c(Cl)cc1N CC1CCCC=C1C(=O)NC1(CN(C(=O)C2=CCCCCC2)C)CC1 C1(CCC=C)CCCCN1C(=O)CCCN(C(=O)COCC(=O)NC)C(C)C N1(C(c2ccc(SC)cc2)=O)CCC2CCN(C(=O)C=CC3CCCN3C)C2C1 C=CCC(C(=O)NC(C(N1CCC(OCCO)C1)=O)c1cccs1)C(C)C C1(CNC(C(CC)CC2CCCCC2)=O)C(C)CCCN1C(=O)C(C)NC(C)=O N1(Cc2cc(C)on2)CCCC1C1CCCCN1C(C1CCCCN1C(N)=O)=O CC1(F)CCC(NC(CC2CCCCC2)CO)CC1 C1(NC(=O)CC2(CNC(C3CC=CC3)=O)CC2)CC(Cl)(Cl)C1 c1(C(N2CCC(N(C)CCc3cccc(Br)c3)C2)=O)cc2ccncc2s1 C=CCCCCCN=c1[nH]c(=NCC2(COC)CCCO2)[nH]c2c1CCCC2 c1(C(=O)NCC2C(C)CN(C(C3CCNC3=O)=O)C2)cc(Br)c(C#N)s1 c1(C(=O)NCC2(F)CC(NC(CS(CC)(=O)=O)=O)C2)cc2ccc(F)cc2o1 c1(C(C)C)oncc1C(N1CCC(N(CCO)C(C2CCCO2)=O)C1)=O N1(C(c2cnc(C)s2)=O)CCOC(CCNC(C2CCCC2(C)C)=O)C1 C12(NC(c3sc4cccnc4c3Cl)=O)CCCCC1CN(C(=O)C=CCO)C2 C1CC(=O)NCCN(CCS(C)(=O)=O)CCO1.C1(C(=O)OC)CC1F C1(c2n(CCCOCC)nnn2)(NC(CC)C(C)(C)C)CCOC(CC(C)C)C1 C12(C(=O)Nc3cc(C)c(NC(C4CC(O)CN4C)=O)cc3)CCC(CC1)C2(C)C C(=O)(C1=NOC2(CCOC2)C1)N1CC(C)(NC(c2c(Cl)cccc2[N+](=O)[O-])=O)C1 C1(NC(c2cscn2)=O)CCN(C(c2ccns2)=O)CC1O N1(C(C=Cc2ccc(C)cn2)=O)CCC(NC(=O)C(C)OCC(C)C)C(C)(C)C1 C1(C(N(CCC(=O)NCC2(C)CC3CC3C2)CC2CC2)=O)CC2(CCC2)CO1 N1(C(C2CN(C(CN(C)C(N)=O)=O)CC2F)=O)CCC12CCC(O)CC2 C1(C(=O)NCCNC(=O)CO)C2CC1N(C(C1CCCSC1)=O)C2 C(CCC(C)C)(C(=O)NC1CCN(C(=O)NC)CC1)NC(CCC(C)OCC)=O C(C(CCNC(=O)CC1(SC2CC2)CC1)NC(COCCOCC)=O)OC c1(CC2(CNC(=O)COc3ccncc3C(F)(F)F)CC2)nccc2ccccc12 n1(CC)cc([N+](=O)[O-])c(C(=O)NCC#CCNC(C2(C3CC3)CCCO2)=O)n1 C(CCCC(=O)N(c1ccccc1)C(C)=O)N(C(C1C(SC)C1)=O)C.C(C(C)(C)C)O N1(C(COc2cc(C)on2)=O)CC2CC(NC(=O)Cc3ccc(Cl)c(F)c3)C2C1 C(=O)(C1CCCc2nncn21)N1CCN(C(CNC(C(C)CC(N)=O)=O)=O)CC1 c1(C(N2CCC(CN(CCC)C)C2)=O)c(C)nn(CC(F)F)c1C Cc1cc(F)ccc1CC(=O)NC1CN(C(=O)C(C)C#N)C(C)(C)C1 C1(NC(C2(CC(C)C)CCCC2)=O)C=CCN(C(C2CCCC(=O)O2)=O)C1 c1(CNC2C(F)(F)CCN(C(C=COCC)=O)C2)cc([N+](=O)[O-])cc(Br)c1O CC1CCN(C(=O)CCN2C(=O)CCC2=O)CC1CNC(C1CC(F)C1)=O C1(CNC(CCS(=O)(=O)N(C)C)=O)CCC2(CN(C(C3CCOCC3)=O)C2)O1 Cc1cnc(Cl)[nH]c1=NCCCCNC(C1CCC(NC(=O)OC(C)(C)C)CC1)=O C1(NC(C(C)CC#N)=O)CN(C(=O)CC2CCC2)C2(CCC2)C1 Cc1cc(C(N2CC3CC3(CNC(c3nnn(C)n3)=O)C2)=O)cc(F)c1 C=CCCC(F)(F)C(=O)NC1CCC(CNC(c2ncc(Cl)cc2Cl)=O)C1 c1(C(=O)NC(CN(C(C2CC2F)=O)CC)C)ccc2c(n1)OCC(=O)N2 c1(C(=O)NCC2C(NC(C(c3ccc(OC)cc3)O)=O)C2)cc2c(ncn2C)[nH]1 C1(CC)(CC)CC(NC(=O)CC(c2ccc(F)cc2)C)CN1C(c1cnco1)=O N1(C(C(NOC)=O)=O)CC(C)CN(C(=O)CSS(C)(=O)=O)CC1C C(C)(CC1=CCCCC1)NC(C(CC)NC(=O)CCc1nccs1)=O C1(C(NOCC=CC)=O)CC(C)CN(C(c2cc(CC=CCOC)[nH]n2)=O)C1 N1(C(CCN=[N+]=[N-])=O)CC2(CCNC(C34CCCCC3C4)=O)CCC1CC2 N1(C(C(CCC)F)=O)CCC(NC(c2ccc(OC)cc2F)=O)C(CO)C1 c1(OC)cc(C)cc(C(N2CC(NC(=O)C=CC3CC3)C3CC23)=O)c1C C1(C(=O)OC)CCN(C(C2(CNC(=O)CN3CCC(C)C3)CC=CC2)=O)C1C N(C1CN(C(=O)COCCSC)Cc2ccccc21)C(CC(C=C)CC)=O C1(=O)C(=O)NCCCC2(CC2)N1.CC1CC1N(C(=O)CC1(N(C(C)C)C)CC1)C c1(CN2CC(C(=O)Nc3nc(SC)nc(O)c3)NCC2)cc(Cl)cc(Br)c1O c1(NC(C2CCC(NC(COCCCC)=O)C2)=O)c(C)ccnc1OCC C1(CNC(C=CCOC)=O)CCC2(CN(C(c3ccc(C(C)=O)cc3)=O)C2)O1 c1(C(N2CCCC(CNC(CCCCOC)=O)C2)=O)nn2c(c1C)CCCC2 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CC)(CC)CCNC(=O)C(C#N)CC N1(C(C(=Cc2ccco2)C)=O)CCN(C(=O)Cc2csnn2)C2CCCC2(C)C1 C1(C(=O)OCC)CCCC(C(=O)N(CCNC(c2csc(C)c2C)=O)C(C)C)C1 C1(CNC(C2CC3CCCC23)=O)CC2CCC1N2C(C1CC1(F)F)=O c1(-c2c(C)nn(C)c2)ccc(=O)n(C(c2ccc(O)cc2)C(F)(F)F)n1 Cc1ccc(C(=O)NCC2CC3CN(C(C4CC4(C)C)=O)CC23)cc1F C1(O)(C(=O)NCC2C(CNC(C(COC(C)=O)C)=O)C2)CN2CCC1CC2 CCC(C)(C)C(O)C(=O)N1CC2CN(C(=O)C(C(C)(C)C)N(C)C)CC2C1 C(=O)(C1=NOC2(CCC2)C1)NC1(C)CCN(C(C2CC(C)SCC2)=O)CC1 C1(CNC(CCCC#C)=O)COCC2(CCN(C(=O)C=CC3CC3)CC2)O1 C12(NC(c3cc(C)[nH]n3)=O)CCCN(C(c3c(C)cc(F)cc3C)=O)CC1C2 N1(C(CNC(C)=O)=O)CC2CCN(C(=O)C(=Cc3ccccn3)C)CC2C1 c1(OC)ncccc1C(=O)C(=O)NCCNC(c1nocc1-c1ccccc1)=O Cc1nc(CO)ncc1C(=O)NCC1(C)CCCN1c1ncc(Cl)cn1 c1(CN2CCCC(C(=O)Nc3nnc(Br)s3)CC2)ccc(F)c(Br)c1F N1(C(c2cn(C)nc2Cl)=O)CCC(NC(c2ccc(F)cc2O)=O)C(CO)C1 Cc1cc(C)c(-c2nc(Cc3ccccc3F)no2)cn1 c1(CC)cc(C(=O)N(CCCNC(c2ncnc(C)c2C)=O)C2CC2)cc(F)c1 O=C1CC(CC(=O)NC23CC(NC(C4CCCCC4(F)F)=O)(C2)C3)=NN1 C=C1CC2CC1CC2(c1nnnn1CCC1CC1)NCCc1ccc(Br)o1 c1(OCc2cn(Cc3cc(SC)nn3C)nn2)ccccc1C#N C(=O)(C1=NOC2(CCC2)C1)N1CCC(COC)(CNC(=O)C2CC2)CC1 C(=O)(C(C)CC(N)=O)NC(C1(O)CN(C(CC2(OC)CC2)=O)C1)C C(C(N=c1[nH]nc(C#N)s1)C1CC1)NC(C1C(c2ccccc2)(C)C1)=O c1(C(N2CCC(C(C(=O)NCC(C)OCC#C)(C)C)C2)=O)ccc(CC)cc1 Cn1cc(C#CCNC(=O)NC2(c3cccc(Br)c3)CCC2)cn1 c1(C(=O)NC(CNC(c2ccc(CCC)[nH]2)=O)C(C)C)ccc(C#N)c(F)c1 c1(C(N(C(C)CNC(c2ccnc(C3CC3)n2)=O)C)=O)ccc(S(C)=O)cc1 C1(NC(C=Cc2ccc(CC)o2)=O)CN(C(c2ccon2)=O)C(C)(COC)C1 N1(C(C2CCC(=O)N2)=O)CCOC(CCNC(c2cccc(C(F)(F)F)n2)=O)C1 c1(C(N2C(CNC(C(CC)OC3CCCCC3)=O)CC2)=O)ccnc(O)c1 Cc1c(C(=O)NC(CNC(=O)CC2CCCS2(=O)=O)C2CCC2)cncc1N C12(C(=O)Oc3nc(C)sc3C)CCC(CC1)N2C(=O)OC(C)(C)C N1(C(CC(C(C)C)C)=O)CCC(CNC(c2cncc(C(F)F)c2)=O)C(F)(F)C1 c1(C(=O)NCCn2ncc(C(=O)NCCC3ON=C(C)C3)c2)ncc(C)cc1C C1(C(N(C)CC2CCCN(C(COCC#C)=O)C2)=O)CN2CCN1CC2 C1(n2ncc(Cl)c2)CN(N2CCC(CN3CCCC3CO)CC2)C1 c1(C(=O)NCCC(C(C)C)NC(COCC)=O)cc(OC)c(OC)c(Cl)c1 S(=O)(=O)(c1cc(C(=O)NCC2CC3(CC3)CN2C(=O)C2=CCSC2)c(C)o1)NC C1(NC(Cn2c(C)ncc2)=O)CCCN(C(c2scnc2C(F)(F)F)=O)CC1F Cc1ccc(N)cc1C(=O)NCC(F)CNC(c1coc(C(F)F)c1)=O C12(NC(=O)Nc3cnc(C(C)OCc4ccccc4)nc3)CC1COC2(C)C N1(C(CCC(C)(C)NC(Cc2cnc(C)s2)=O)=O)Cc2n[nH]cc2C1CO C1(C(=O)NC2(CCNC(=O)CCCC3CCCCC3)CCC2)COC2(CCC2)C1 CC1CC(C(=O)NCC2CCCCC2NC(C2CCOC(C(C)C)C2)=O)=NO1 C1(NC(C(C)S(N)(=O)=O)=O)CCN(C(c2n[nH]cc2Br)=O)CC1(C)C CC(CC(C)NC(c1ccn(CC(F)F)n1)=O)NC(C1CC(F)(CO)C1)=O c1(-n2c(C(c3c(COC)ocn3)NCCCCF)nnn2)c(C)cccc1C N1(C(CC(CC=C)(C)C)=O)CC2CC(C)N(C(C3CCCN3C3CC3)=O)C2C1 CCCC(CCCNC(c1ccc(CC(C)(C)C)cc1)=O)NC(=O)C=CC=CC N1(C(CCOCC)=O)CCN(C(=O)CC2OC(C)(C)OC2=O)CC1C1CCCC1 CC1CN(C(=O)CCCOc2cccnc2)CC1NC(C1CSCCS1)=O c1(N(C)CCc2ccccc2)nnc(-c2cnc(C3CC3)[nH]2)n1CC(=O)N(C)C N1(C(C(C(C)C)n2cnnn2)=O)CCN(C(c2cc(=O)n(C)o2)=O)C(C)C1 C1(C(N2CC(N(C(=O)CSC3CCOCC3)C)C2)=O)CCC2(CCC2)O1 CON1CC(C(=O)NC2CC(NC(=O)C#CC(C)(C)O)CC2O)CC1=O C1(O)(CNCc2c(C(=O)OC)con2)CCCN(C(c2c[nH]nc2Cl)=O)C1 CC(C)C(C)C(C)CC(=O)NCc1ncccc1C(F)(F)F N1(C(CNC(CN(C(CNC(=O)NC)=O)C2CCC2)=O)=O)CCCC1CF CN1CCCN(C(=O)C(C(C)(C)C)NC(c2ccc[nH]2)=O)CC1 C1(CC)(CC)CC(NC(=O)CSC2CCOC2=O)CN1C(c1cc(O)n(C)n1)=O C1(C(=O)NCCCCC(CO)NC(CC=CC=C)=O)CCc2ncccc2C1 C(C(=O)N1CC(O)CCO1)(N(C(C(CC=C)CC)=O)C)C1CC1 CC(C)C(O)CC(=O)N1CCOC(C)(CNC(c2coc(CS(C)(=O)=O)n2)=O)C1 C=CCCC(F)(F)C(=O)N(CCCCCNC(c1cc(Cl)cs1)=O)C N1(c2nnc(CSC)n2CC2CCOC2)CCc2c(ccnc2Cl)C1 Cn1cnc2nc(N3CC(CNC(=O)C(c4ccc(F)cc4)(F)F)C3)ncc12 N1(C(C(CC)Sc2ccccc2)=O)CC2CC(C)N(C(=O)CSC(F)F)C2C1 c1(C(N2CC(NC(=O)C=CC3CCCC3)C(F)C2)=O)cc(Cl)c(Cl)cn1 N1(C(C2=C(C)OCC2)=O)CC2(CCCC2NC(C2CS(=O)C2)=O)C1 C(=O)(C1=CCC(NC(=O)CC2CCCO2)C1)N1C(COC)CC1 C(c1ccc(Cl)cc1F)=CC(=O)OC(C(C)C)C(=O)N1CCCCC1 c1(C(N(C)CCNC(C23CC4CC2C3C4O)=O)=O)csc(=NC2CC2)[nH]1 N1(C(C2C(Br)(C(=O)OCC)C2)=O)CC(C)(c2cn(Cc3csc(C)n3)nn2)C1 C12(C(=O)NC(C)(CNC(=O)Cc3sccc3Cl)CO)CCCC1CC(=O)C2 c1(C(N2C(C)CN(C(=O)CCC3CCCCO3)CC2)=O)ccc2c(n1)CCC2=O c1(SC)ccc([N+](=O)[O-])cc1C(=O)NC1CN(C(=O)CN(C)C2CC2)CC1C Cc1ccc(NC(=O)NC2(C(=O)NC3(c4ccccc4)CC3)CC2)cc1 CC1CCCC(C(=O)NCc2ncccc2C(F)(F)F)O1 CCC(CC(=O)NC1(CCCOC)CCCCC1)NC(=O)C(C)SC c1(C(=O)NC(C)(CNC(c2ccnc(O)c2)=O)CO)cc2n(n1)CCCNC2=O C(=O)(C(C(C)C)NC(=O)NC1(c2ccc(OC)cc2)CC1)OCC N1(S(=O)(=O)C=CC=C(Cl)Cl)c2ccccc2Sc2ccccc21 C12(CNC(=O)Cc3cccc(O)c3)CCCC1CN(C(=O)Cc1csc(S)n1)C2 c1(C(N2CC(CC(=O)NCc3c(C)cccn3)OCC2)=O)cccc2c1OCO2 C1(N(CC(=O)NC2CCCNC2)C)CCN(CC(F)F)CC1 c1(CC(=O)NC2CC(F)CN(C(=O)Cc3ccoc3)C2)coc2cc(F)ccc12 Cc1nc2ccnn2c(C)c1C(=O)NCC1COCCN1C(=O)C(C)NC(N)=O C1(CC)CN(C(c2ccccc2Br)C(=O)NC2CCC2)CC(C)O1 N1(C(CN(C)CC)=O)CC(NC(C23CC(CC)(CO2)C3)=O)C(F)C1 N1(C(c2c(CNC(C3CC4(CC4)CO3)=O)noc2)=O)C2COCC1C2 c1(SCCC(=O)NC2CN(C(c3nc(C(C)C)oc3)=O)C2)nc2ccccc2[nH]1 c1(C(=O)OC)ccc(Br)cc1C(N1CCC(CN=c2ccnc[nH]2)CC1)=O C1(C(C)C)CN(C(C2COCC2C(N)=O)=O)CC1C(N1CC(SC(F)F)C1)=O c1(OC)ccc(Cl)cc1C(F)(F)C(=O)NCC(CO)NC(C1CCSC1)=O C(=O)(N1CCCc2nncn21)C1C(NC(C(C)OC(C)=O)=O)CCO1 N1(C(c2ccn(CC=C)n2)=O)CCN(C(=O)CCC=CCC2CCCCC2)CC1 N#Cc1nccc2cc(NC(C3CN(c4ccccn4)C3)=O)ccc12 C(=O)(CC(F)(F)C(C)C)NC1CCCN(CC(=O)NC(CN(CC)CC)C)C1 C(C(C)(C)CC(=O)NCC1(CCCC(=O)Nc2cccc(C#N)c2)CCC1)OC C1(C(=O)NCC(C2CCCCC2)C)CC2(CCN1C(=O)C(C)CO)CC2 N1(C(C2(F)C(C)C2)=O)Cc2ccccc2CC12CCC2 N1(C(C(CC=C)OC)=O)CC(C)(C)OCC1C(=O)Nc1csnc1OC N1(C(c2cccc(CC)c2)=O)CCCN(C(c2cnc(N)c(Cl)c2)=O)C(C)C1 C=CC(C)(CCOC)C(=O)NCC(CCNC(c1cc(C(C)(C)C)no1)=O)OC C(CCN=C(NCCF)NC1CC(=O)N(C(C)(C)C)C1)=C(C)C c1(C(N2CCC(CNC(CC3(C=C)CCOCC3)=O)C2)=O)ccc2c[nH]nc2c1 Nc1cc(C(=O)NC2CCC2C(=O)NC2CC(CO)(CO)C2)cc(F)c1 Cc1ncncc1NC1(c2nnnn2CC(F)F)CC2CC2C1 N1(C(C(CCC=C)(C)C)=O)CC2COCCC2(NC(c2cc(CCC)[nH]n2)=O)C1 C1(C)(C(=O)NCC(CC)NC(c2c[nH]nc2-c2cccnc2)=O)CC=CCC1 C1(OC)(CO)CN(C(=O)CN(C)C(C2(CO)CCOC2)=O)C1 c1(CC)ccc(C(C)CC(=O)N(C)CCN(C(=O)C=CC2CCCN2C)C)cc1 c1(CC)c(C(=O)NC2CCCCC2NC(=O)CC2CCCCN2CC)nnn1C Cc1nc(C(=O)N(C(C)(C)CC(=O)N2CC(F)(C#N)C2)C)sc1C C1(S(N)(=O)=O)(C(=O)NC2C(CNC(C3N(CC)CC3)=O)COC2)CC1 N1(c2n(CC=C)c(-c3csc(Br)c3)nn2)CC2CN(C)CCC2(CO)C1 c1(CC)cc(C(=O)NCCOC(C)(C)CNC(c2cscc2F)=O)ccc1C c1(C(N2C(C)CC(NC(C(CC)CC3CCCCC3)=O)C2)=O)c[nH]c(=N)cc1C C1(NC(C2(F)CCOC2)=O)CC2(C1)CC(CN=c1nc(C3CCCC3)[nH]s1)C2 c1(C(CN)O)ccccc1Br.CC(C(CO)c1ccccc1)c1ccccc1 Cc1cc(Cl)ccc1C(N1CC(NC(=O)C2=CSCCO2)C(O)C1)=O C1(OCC)CC2(C1)CC2C(N1CC(CC(C)NC(=O)C(C)(F)F)C1)=O Cc1ccc2c(c1)C(NC1CCCCN1Cc1ccccc1)CCCO2 c1(CN2CCC(NC(c3c(C)nc(Br)cc3)=O)C(F)C2)ccc(Br)c2nsnc12 c1(C(N2CC(C(=O)NCCNC(c3cc(C(F)F)on3)=O)C2)=O)ccncc1Cl c1(C(N2CCCCC(C(N3CCC(C(F)(F)F)C3)=O)C2)=O)ccc(Br)c(Cl)c1F N1(C(C(n2cc(Cl)cn2)C)=O)CC2CCN(C(=O)CC3(C)CCCCC3)C2C1C C#CC(CNC(=O)C(CC=CC)NC(=O)C(C)N(C)C(C)=O)CC(C)(C)C C1(C)(CNC(C(C2CC2)SC)=O)CCCN(C(C2CCCC2C)=O)C1 CC(CCCNC(=O)C(C)(F)c1ccccc1)NC(C1(O)CCCC1)=O CCC(C)CCC(O)CC(=O)N(CCN(CC)CC)CCOCC1CC1 N1(CC(=O)NC)C2CCC1CN(C(c1oncc1C)=O)C2 c1(C(=O)NC(C)CNC(=O)CC2CCCC2C)cn2c(n1)CCC2 C(N=c1cc(NCCCn2cnnc2)nc[nH]1)c1c(C)sc(Br)n1 c1(C(=O)NCCN(C(CC=C(C)C)=O)C(C)C)ccnc(OCC2CC2)c1 N1(C(c2ccc(C#N)[nH]2)=O)CCC2CC1CN(C(=O)CC1CCC3(CC1)CC3)C2 C1(CC(C)OC(C)=O)CCN(C(=O)NC2CC(O)C(O)C2)CC1 CC1CC2(CC2)CN1C(c1cc(CNC(c2cncs2)=O)on1)=O c1(C(N2CC(CCNC(C(C)C3CC3)=O)OCC2)=O)cc2n(n1)CCC2 C(C)(CCC(=O)NCC(C)NC(=O)C(C)Cc1ccncc1)OCC C(C)(N=c1[nH]n(C)c(C(F)(F)F)c1[N+](=O)[O-])C1(NC(COC)=O)CCC1 C(=O)(C1=C(Cl)CCC1)NC1C(C)CN(C(C2CC(=O)N(C3CN(C)C3)C2)=O)C1 N1(C(CN2CCC(OC)C2)=O)CCCCC(CNC(=O)CCC2OCCO2)C1 Cc1c(N)cc(C(N2CCC(NC(C3CCS(=O)(=O)N3)=O)C(C)C2)=O)cc1N C1(NC(C2(CSC)CCC2)=O)CC2CC(NC(c3cnccc3Cl)=O)C2C1 c1(C(N(C2CCCC(NC(c3c(C#C)c[nH]n3)=O)C2)C)=O)cccn2nccc12 Cc1sccc1C(=O)NCC(C)(C)OCC(=O)NOCCCC1CC1 c1(C(=O)NCCOCCNC(C(CSC)O)=O)cc(C2OCCO2)ccc1O C1(NC(CCCCC)=O)C2CC3CC(C2)CC1(CNC(=O)C(F)CC)C3 C1(NC(c2c(CC)cco2)=O)CN(C(c2ccc3oncc3c2)=O)C2(CCC2)C1 N1(C(C(COC)O)=O)CCC2(CCCN2C(=O)C(C)c2ccco2)CC1 N1(C(C(C2(O)CCC2)NC(c2cc(CC)n(C)n2)=O)=O)CCC2(CNC(=O)N2)C1 C1(C)(CNC(c2ncc(C)nc2)=O)CCCN(C(C2CCCS2)=O)C1 C1(OCC)CC2(C1)CC2C(=O)NCC(O)CNC(=O)Cc1cn(C)cn1 c1(SCC)ccc(C(=O)N(C)CCN(C(C2CCC(C(C)C)C2)=O)C(C)C)cn1 CC1CN(C(=O)C=CC2CCOC2)CC1NC(=O)Cc1ccc(Br)cc1 C(C(=O)NC1(CNC(=O)C(=O)Nc2cccc(C)c2)CCOC1)(C(C)C)SC C1(CC(=O)NCc2ccc(COC)o2)COCCN1C(=O)CC1CC(OC)C1 N#CC1CCCCC1NC(=O)Nc1ccc(OCC(F)F)cc1 C(CNC(C1CC2CC2N1C(=O)CCC(C)N(C)C)=O)(C(C)(C)C)OC C(=O)(CCC1=NNC(=O)CC1)NC1C(CC)CN(C(C23CC(F)(C2)C3)=O)CC1 C=C=CC(C)C(=O)N1CCC(CC(=O)N(CC(C)CC)C)C1 N1(C(C2(C#C)CCCC2)=O)CC(C2CN(C(C3CCC([N+](=O)[O-])CC3)=O)C2)C1 CC(C)C(C(=O)NCC1CCN(C(=O)CCC(F)F)C1(C)C)C(C)C C(CNC(=O)CCOCC1CCC1)(CCNC(c1nonc1C)=O)OC C1(N(C)C)CN(C(C2CC(NC(=O)CCC(N)=O)C2(C)C)=O)CC1O C1(C(=O)NCC2C(CCC=C)C2)(COC)CCCN1C(c1c(C)cnn1C)=O c1(C(C)NC(C=CC(=O)NCc2cc(C(F)(F)F)[nH]n2)=O)c[nH]nc1F.C1(C)CC1 c1(C(N2CC3N(C(c4cccc(=O)n4O)=O)C(C3)C2)=O)ccc(Cl)cc1[N+](=O)[O-] C(CCCC(=O)N(CCC(=O)NC12CC(CC3CC3)(C1)C2)CC1CC1)N(C)C C(=O)(CC(C)CCC(=O)NCC(C)CNC(C1(C)CC=CC1)=O)OC C=CC1(C(=O)NCCCCCNC(=O)Cc2cccn2C)CCC1 Cc1cc(C(=O)NCC(C)CNC(=O)CC2CCCC2O)ns1 C1(NC(=O)CC2C=CCC2)CC2CC(NC(c3csc4nnsc34)=O)C1C2 c1(CN(C2CN(C(C3CCCOC3)=O)C2)C)c(F)ccc(Cl)c1Br c1(C(=O)NCC(O)CNC(c2ncccn2)=O)cccc(C2CC2(F)F)c1 C(=O)(C(CCC1CCC1)NC(=O)CCn1cnc(=N)[nH]1)N(CCCC)CCOC C(=O)(CCC(CC)NC(CSCC#C)=O)NC1CCC(N(C(C)=O)CC)CC1 N1(CCC#C)CC2CCN(C(c3csc(C(F)(F)F)n3)=O)C2C1 CC1(C)CCCCC1NCCCC1CCCCCC1 c1(C(=O)NC(C(=O)Nc2cc(C)cc(C)c2)CS(C)(=O)=O)ccnc2cc[nH]c12 N1(C(C(C(C)C)SC)=O)CC23CCCC2(C1)CN(C(=O)CC1CNC(=O)O1)C3 CC(C)CC(O)C(=O)N1CCN(C(c2ccc(-c3nc[nH]n3)cc2)=O)C(CO)C1 C(=O)(C(C)(C(F)F)c1ccccc1)N(CC(C)NC(c1n(C(C)C)cnc1)=O)C c1(C(=O)NCc2cccnc2N2CCCCC2)cc2c(cn1)OCCC2 CC1CCN(C(c2cnccn2)=O)CCN1C(C1CC2(C1)CC(C)(C)C2)=O c1(C(=O)NC(C(=O)NCC(=O)NCC=C)CCC)ccn2ccccc12 c1(CC(N2CCC(CCNC(COC(C)(C)C)=O)C2)=O)cccc(S(C)(=O)=O)c1 C1(C(=O)Nc2cc(C(=O)OC)[nH]c2)CN(Cc2cccc(C)c2N)CCC1(F)F CC1(C(=O)NCC2(CNC(c3cc(C#N)no3)=O)CC23CCC3)CCOCC1 CC1CCN(C(C2CCC2C(F)F)=O)CC1NC(=O)C(=O)NC1CC1 N1(C(CC=CC)=O)CCC2CCN(C(c3cn(C(F)F)c(C)n3)=O)CC2C1 N1(C(CSCCC(C)C)=O)CCC2C(C(=O)NCC3CCC(C)(C)CO3)C2C1 C(=O)(C=C1SCC(=O)N1C)NC(C(C)C)CNC(C1CN(S(N)(=O)=O)C1)=O CC1C(NC(c2cc(Cl)ccc2Cl)=O)CC2CCC1N2C(C1(CO)COC1)=O c1(C(N2CC(C)(NC(c3ccc(C)[nH]3)=O)C2)=O)cccc2c1OCC2C CON1CCC(C(=O)NCCN(C)C(c2nocc2CC(C)C)=O)CC1 N1(C(C2N(C)C(=O)CC2)=O)CC(C(N2CC(F)C(F)C2)=O)C(F)(F)C1 c1(C(N2CC3(CN(C(c4ccc(C=C)cc4)=O)C3)C2)=O)cc2c(cc1C)OCO2 C(=O)(CCCC(F)(F)C(F)(F)F)N1C(CNC(C2CC2CF)=O)CCC1 C(=O)(C(O)CC(N)=O)NC1(C2N(C(c3c(OC)cccc3)=O)CCC2)CC1 c1(-c2ccc(C(C)=O)o2)cccc2ccc(C(N3CC(O)CC3(C)C)=O)nc12 S(=O)(=O)(c1cccc(CC(=O)NCCc2nc3c(s2)COCC3)c1)NC C1(CC)CCS(=O)(=O)CC1.C12CN(CCO1)CCNC(=O)CC(=O)N2 C1(C(=O)NCC2(C=C)CCC2)(CC)CCCN1C(c1n[nH]c(O)n1)=O c1(C(=O)NCC2CN(C(C(c3cccc(C)c3)C)=O)C2)ccc2c(c1)C(C)CO2 n1(CCCO)nc(C(C2CC2)C2CC2)nc1-c1ccoc1Cl CC(C)(CO)C(=O)NCCCNC(c1sc(=N)[nH]c1C1CC1)=O N1(C(c2cc(C#N)oc2)=O)CCC(NC(=O)CSCC2CCCO2)C(F)(F)CC1 c1(C(N2CC(C)C(NC(=O)CC3C=NN(C)C3=O)C2)=O)cc2c(s1)CC(C)(C)C2 C12CCCCCC1CN2.Cn1c(C(N2CCCC2CC2(SC)CC2)=O)nnc1S c1(C(N2CCC(N(C(Cc3c(C)con3)=O)C)C(C)C2)=O)ccc2cncn2c1 c1(C(N2CC3C(NC(c4cccc(=O)n4O)=O)C3C2)=O)nccc2occc12 N1(C(C2(C)C(C)(C)C2)=O)CC2=C(C1)CN(C(=O)CCN1CCOCC1=O)C2 c1(OC)cnc(F)c(C(N2CC(C)(C)CC2CNC(=O)CC2CCCC2C)=O)c1 c1(C(=O)NCCN(CCCN(C)C)C(=O)Cc2cccnc2)onc2c1CCCC2 Cc1c(F)ccc(C(N2CCCC(N(C(=O)CC3CSCCS3)C)CC2)=O)c1N c1(C(=O)NCC=CC(=O)NCC2CC(C(C)(C)C)C2)cccnn1 N1(C(C2C3(CN(C(c4ccc(CC(C)C)cc4)=O)C3)C2)=O)CCn2cccc2C1 c1(C(=O)NC(C)CCCCNC(C2CCSCC2)=O)cnc2c(F)cccc2c1 c1(CN(C)C)nccc2c1CCCN2S(=O)(=O)c1ccn(C2CC2(F)F)n1 c1(CC(=O)NC2CC(C)(NC(CCOC)=O)C2)cnc(O)nc1O c1(C(=O)NCCCN(C(=O)C(F)(F)C2CC2)C2CC2)cc(C(F)(F)F)ncn1 C1(C(N(CC)OC)=O)CN(C(C2CC(=O)CS2)=O)CC12CCC2 C1(NC(C2(CCC)CC2)=O)CCC(CNC(C2CC2Cl)=O)CC1 CC1CCCC1(C)NC(C1CCC(NC(=O)C(C)NC=O)CC1)=O C1(C(=O)NCCC2CSCCN2C(c2ccn(C3CC3)n2)=O)Cc2nccn2C1 c1(C(=O)NC2C(C(=O)NCCN(CCC)C(C)C)C2)cc(F)cc(F)c1Br Cc1ccc(C2CC2C(=O)N(CCCNC(C2CCO2)=O)C)cc1C N1(C(Cn2cc(C(N(C3CCCO3)C)=O)nn2)=O)CCCN(C2CCCC2)CC1 c1(C(=O)NC2C(CNC(=O)CCCn3cncn3)CCCC2)cc2cscc2s1 c1(C(=O)NC2CC(CNC(C(CSC)O)=O)CC2O)cncc2c1CCC2 C=CCC(C(=O)N1CC(OC)CC1CNC(c1cc(CC)nc(O)c1)=O)C(C)C c1(N(C)C)ccc(N(C2CC3CC2CN3)C(=O)CCN2CCOCC2)cc1C#N CC#CCCCCNC(=O)C(C)N(C(c1cc(CCO)on1)=O)CC N1(C(C2CCCC(NC(c3c(C#C)cnn3C)=O)C2)=O)CCCC(C)(OC)CC1 C1(NC(C2C(CCC)CN(C(c3c[nH]c(=O)cn3)=O)C2)=O)CCOC12CCCC2 C1(CCC)CN(C(c2c(C(F)(F)F)ncn2O)=O)CCN1C(C1CC12CC2)=O C12(NC(=O)CN3CCCCCC3=O)CCCN(C(=O)CCOC3CC3)CC1C2 c1(CNC(c2cc(C)on2)=O)cc(C(=O)NC2CCCC2C(C)C)ccn1 Cc1ccccc1S(=O)(=O)CC(=O)NC12CCN1C2.C1(=O)CN1.C1(CO)CC1 Cc1cc(C(=O)N(C(C)CN(C)C(C2(N)CCC2)=O)C)cc(C)c1.C(N)=O c1(CC(=O)NCCC2N(C(CC(C)(C)OC)=O)CC(OC)C2)ccc(F)c(F)c1 N1(C(Cc2ccc(C)o2)=O)CC(NC(c2cc(C(N)=O)oc2C)=O)C2CC12 c1(CNC(CC(CCC)CC)=O)nn(C)c2c1CN(C(c1csc(C)n1)=O)CC2 C1(NC(Cc2ccc(OC)c(F)c2)=O)CN(C(C2CC23CC3)=O)C2(CCCC2)C1 c1(C(=O)NCC2N(C(C(CCC)CC)=O)CC=C2)ccc(F)c2c1OCC2 C1(CC)(CC)CC(NC(c2cc(Cl)ccc2N)=O)CN1C(C1CC1(C)C)=O N1(C(CC2(C)CCN2C(c2ncccc2F)=O)=O)CCC(F)(F)C(O)C1 C(=O)(C1=CCc2ccccc21)NCCCCCN(C)C(c1cncnc1)=O c1(C(N(C(C)CN(C)C(C2CCCN2C=O)=O)C)=O)cc(F)ccc1O c1(OC)cccc(C(N2CC(CNS(=O)(=O)CC3CCC3)C2)=O)c1 N1(C(C2CCN(C(CC(C)(F)F)=O)C2(C)C)=O)Cc2cccc(F)c2C1 C1(C(=O)NCC(C)CNC(c2cncc(C(N)=O)c2)=O)COc2ccccc2C1 C(C(C)C(=O)NCC12CC(NC(=O)C(C)NS(C)(=O)=O)(C1)C2)OCC c1(C(=O)NCC(=C)CCNC(C2CC2(C)CC)=O)cn(C)c(=O)c2c1CCCC2 c1(C(=O)NC(C2CCN(C(C3(C)CC3)=O)CC2)CO)cccc2c1CCO2 CC(C)C(C(=O)NCC1CN(C(=O)CCC(=O)OC(C)(C)C)C1)N1CCCC1=O C(=O)(CCCCCn1cnnn1)N1CCC(CN(C(CCC=C=C)=O)CC)CC1 N1(C(COCC(C)C)=O)CC(F)CC1CNC(c1csc(-c2cnc[nH]2)n1)=O N1(C(c2ccc(N)cn2)=O)CCC2CCN(C(c3cc4n(c3)CCOC4)=O)C2C1 C(=O)(C1CCCc2sc(=N)[nH]c21)N1CCNCC1.C(=O)(C(O)CC(N)=O)N(C)C S(=O)(=O)(c1ccc2c(c1)CC(C=O)C2)N1S(=O)(=O)CCOCC1 C1(NC(CCC2N(C)CCC2)=O)CCN(C(=O)CN=S(C)(C)=O)CC1F N1(C(c2cnc3n2CCC3)C(=O)NC(C(=O)OC)C)CCSC2COCCC12 C(C)(C)(CCCC(=O)NC1CCSC1)NC(C(C)C1CCOC1)=O Cc1cc(CN2CCC(F)(CNS(=O)(=O)c3cccs3)CC2)c(O)c(Br)c1 C1(C(=O)OCC)CCCC(C(=O)NCC2(NC(C3CC4(CCC4)C3)=O)CC2)C1 c1(C(=O)NC(C(=O)OCC=C)Cc2ccccc2)ccc(CC(F)(F)F)cc1F N1(C(c2cc(OCC)ns2)=O)CCN(C(=O)C(C)OC)C(c2cn[nH]c2)C1 C1(C(N2CC3(CC(NC(COCC(=O)OC)=O)C3)C2)=O)CC2CC(O)CC(C1)C2 c1(SC)cccnc1NC(c1ccc(Nc2cc(C(F)(F)F)ncn2)nc1)=O C1(CC(N2CC(F)(CO)C2)=O)C2CCCC2N1C(=O)CSc1nc[nH]n1 Cc1cc(C(N2CC=CC2CNC(=O)CC(F)(F)Br)=O)c(F)cc1F N1(CC(=O)NCC(CNC(C2(CO)CCCC2)=O)CO)CC(=O)NC1=O C1(c2ccn(C3C(C)C3)n2)CCS(=O)(=O)CN1.C1C(=O)N1C N1(C(C(CC)(C)C)=O)CCC2(CC1)CC2c1cn(CC2(OC)CC2)nn1 N1(C(C2C(C)(COC)C2)=O)CCC12CN(C(=O)C=Cc1cnc[nH]1)C2 C1(O)(CN(C)C(C2CC(O)CN2C)=O)CCCN(C(=O)CNC=O)C1 N1(C(Cn2c(=N)[nH]nc2)=O)CCCC2(NC(=O)Cn3cnnn3)CC2C1 Cc1cc(CNC(C2CC2C(C)NC(=O)CCOCC(F)F)=O)cc(F)c1 C(C(CC1CC1)CO)NC(CN(C(=O)Cc1ccnn1C)CCC)=O C(N=c1[nH]c(=NCCOC)[nH]c2c1SCC2)C1CCCC(SCC)C1 CCCCC(CC)CC(=O)NC(C1(NC(=O)CC2(C)CC2)CC1)C S(=O)(=O)(c1cccc(NC(=O)CN2CCC(C3CC3)C2)c1)NCC c1(C(N(CCNC(c2cc(C)c[nH]2)=O)CC)=O)cc2ccccc2cc1C C12(NC(CCC=CC)=O)CCOCC1CN(C(C1(C#N)CCN(C)CC1)=O)C2 CC(CCC(=O)NCC1(C)CCC(=O)N1)NC(=O)CCCOC(C)(C)C N1(C(C2CN(CC)C(=O)C2)=O)CCCC2C1CCN2C(c1ccncc1)=O c1(C(N2C(CNC(c3c(O)ncc(CC)c3)=O)CC2)=O)cccc2c1CC(=O)N2 Cc1cccc2c1CC(C(=O)NC1COCC1NC(c1cc(C(C)C)[nH]n1)=O)O2 N1(C(CC(C)(F)F)=O)CC2CC(NC(c3ccnc(-n4cccn4)c3)=O)CC1C2 O=C(CCCCC(F)(F)F)NC(CNC(C1CC(n2ccnn2)C1)=O)C1CC1 C(CC(C(F)(F)F)NC1CC1(F)F)NC(C(=O)Nc1cccc(CS)c1)=O C1(C)(NC(C2CC(=C)C2)=O)CCN(C(c2csc(NC(=O)C3CC3)n2)=O)C1.C1CC1 c1(C(N2C(C(=O)NCCC(=O)OC)CSC2)=O)c(C)ccnc1C N1(C(CCC#C)=O)C2CCC1C(CNC(c1cncc(OC(F)F)c1)=O)C2 C(=O)(C1CC=Cc2ccccc21)NCc1nc(CNC(C(CC=C)(F)F)=O)sc1 CCCC(O)C(CO)NC(=O)CCC1CCCN(C(=O)Cc2ncccc2F)C1 Cc1nc(N2CCCC(CN(C)C(C3CCCCO3)=O)C2)c2c(C)csc2n1 N1(C(C(C2CC(NC(=O)COCC3CCC3)C2)F)=O)CCCC2(CC2)C1 CC1(C)CC(NCc2cncn2-c2ccc(F)cc2)CS1 N1(C(C2CC(CC(=O)OC)C2)=O)CC(C)(NC(=O)C=CC2CCOC2)C1 C(c1cc(Cl)ccc1OC)=CC(=O)NCC(CCNC(C=C(COC)C)=O)(C)C C1(NC(C2(OC)CC2)=O)CC2CC(NC(=O)Cc3ccnc(Cl)c3F)CC12 C1(NC(N2CC(C)(C(F)(F)F)C2)=O)CCOCC12CCC2 c1(CC(=O)N(C(C)C(=O)NCC(c2ccco2)O)CC)cc(C)on1 N1(C(C(CCC)CNC(c2c[nH]c3cccnc23)=O)=O)C2CCC1CC(CO)C2 Cc1cc(S(C)(=O)=O)cc(C(=O)NC(C)CCNC(c2nocc2C)=O)c1C c1(CC(=O)NCC(=C)CCNC(C2CCCN2CC(F)(F)F)=O)cccc(F)c1 N1(C(C2(CC)COC2)=O)CC2ON=C(CNC(=O)CCn3ccc(C)n3)C2C1 C(=O)(C(C)(C)CC(C)(C)C)NCC12C(CN(C(CC(C(C)=O)(C)C)=O)C1)C2 C1(NC(Cc2nc(C)[nH]n2)=O)CCCN(C(c2cnc[nH]c2=N)=O)CC1 c1(C(N2CC(C)(NC(c3onc(CC)n3)=O)C2)=O)cc(C#N)c[nH]1 C1(CNC(CCC2(C)CC2)=O)CN(C(=O)C(C)C(C)(F)F)CCC12CCOCC2 C(CO)(CCCCNC(C1CCC(O)CC1)=O)NC(c1coc(Br)c1)=O c1(CC(=O)NC(CCN(C(C=C(C)C)=O)C)C)cn(C)c2ccccc12 C1(C(N2C(CN(C(=O)CSCCC#N)C)CCC2)=O)CC12CC(C)(C)C2 C1(CCNC(c2cc[nH]n2)=O)CN(C(c2cccnc2C2CC2)=O)CCS1(=O)=O c1(C(N2CC3N(c4nc(CC)cc(CC)n4)C3C2)=O)ccc([N+](=O)[O-])cc1C C1(C(=O)OC)CN(C(=O)NCc2cccc(NC(N)=O)c2)CCS(=O)(=O)C1 N1(C(C(C)N(CC(c2nccs2)C)C)=O)CCOCC1(C)C CC1=C(C)CN(C(C2(CNC(C34CCCC3C4)=O)CCC2)=O)CC1 c1(CC(N2CCC(C)(C(=O)Nc3onc(C)c3Br)C2)=O)ccc(Cl)c(Cl)c1 CC(C)(C)C#CCCNC(C1CC(O)CN1C(=O)Cc1cnns1)=O C1(NC(CCc2cnn(C)n2)=O)CCC(F)(CNC(C2(N(C)C)CCCC2)=O)C1 c1(NC(C=CC(=O)OC)(C)C)cc2c(cnn2C)nc1C Cc1cnc(C(N2CC(C(F)(F)F)C(CNC(=O)CP(C)(C)=O)C2)=O)nc1 c1(C(=O)NC(C(N2CCCN(CCOCCOC)CC2)=O)=O)cnc(C#N)c(Cl)c1 n1(CCC)ncc(C(=O)NCC2CCCC(NC(C3(SC)CC3)=O)C2)c1Cl c1(C(=O)NC2CC(NC(C(CCCC)CC)=O)C2)ccnc2c(C(N)=O)cnn12 c1(CN2CCC(NC(c3cc(C)nn3C(F)F)=O)C2)ccc(F)c(C#N)c1 c1(C(N2CCC(CNC(CCCNC(=O)OC)=O)C2)=O)nnccc1C c1(C(=O)NC(C(C)C)C(=O)NC2CC=CC2)ccc(=O)n(C)c1 c1(CCC(=O)NCC2(F)CC(NC(CC3(OC)CCC3)=O)C2)ccc(SC)cc1 C(=O)(CC(=O)NCC(C)(C)OCC(=O)NCCCC1CCOC1)N(C)C N1(C(c2ccn(CC)n2)=O)CCC2(CNC(=O)CNC(=O)C3CC3)CCCCC12 c1(C2CN(C(Cn3cc(C4(COC)CCCC4)nn3)=O)C2)ccnc(Cl)c1 c1(C(N2CCC3C(C(N4C(C#C)CC4)=O)C3C2)=O)ccc2cc[nH]c2c1 C1(C(=O)NCCC2(NC(C3CC(CC(=O)OC)C3)=O)CC2)CCCOCC1 N1(C(c2c3ccc(C)cc3[nH]c2)=O)CCC(C(=O)N(C)C)c2cc(O)ccc21 N1(C(C(N2CCC(O)CC2)C)=O)CCC12CN(C(=O)CCc1ccc(O)nc1)C2 CCC(C)CC(C(=O)NCC12CCC(CC1O)C2)NC(C1CCN1C(C)(C)C)=O CCCC(C(=O)NC1CCC1C(=O)NCC1C(C)(C)C1(F)F)OCC CCCCC(CNC(C1(C(C)C)CCCO1)=O)NC(=O)C(COC)COC C(CC(C)P(C)(C)=O)NC(=NCC=C)NCC(O)COc1cccc(Cl)c1 C(CCCCCC1CC1)NC(CC1(NC(C2N(CCC)CCC2)=O)CCC1)=O CC(C(C)(O)C(=O)N1CC(C)(NC(c2n[nH]cc2Br)=O)C1)c1ccccc1 c1(C2(CNC(c3cccc(Br)c3F)C)CCC2)cc(Cl)ccc1F N1(C(CC(=O)NCC#C)=O)CC2CCCC(NC(=O)C(C#N)C(C)C)C2C1 N1(C(C2CC3(CC(=O)N3)C2)=O)CCc2nc[nH]c2C12CCN(C(=O)CO)C2 N1(C(C2(NC(c3cnc(C)nc3C)=O)CCSC2)=O)C2CCC1CC(F)C2 C(=O)(C1=CCCSC1)NCC(C1CC1)NC(C1CCCC1O)=O.c1ccccc1C c1(C(N2CCCC(N3CCCCC3)C2)C(=O)NCCC)ccc2c(c1)CCCO2 Cc1ccc(CC(N2CC(CNC(c3cscc3F)=O)C3(CC3)C2)=O)cc1F O=C(Nn1cnc2ccccc12)c1cncc(CNC(C2(CO)COC2)=O)c1 c1(C(=O)NCC(C)CNC(C2CSCCS2)=O)cc(CC2CCC2)c[nH]1 CC(N=c1[nH]c(=NCCC2CCCS2(=O)=O)[nH]c2c1COC2)c1ncn(C)n1 N1(C(Cc2cc(C)cc(F)c2)=O)CCC2CCC(C1)N2C(C1CCO1)=O c1(N(C(CCNC(CCNC(=O)OCC)=O)=O)C)cc(OC)n(C)n1 CC1CN(C(c2cc(Cl)cc(C#N)c2)C(=O)NCCCC2CC2)CCN(C)C1 C(=O)(C(COC)COC)NCCC1(C(N(CC#C)CCF)=O)CCCC1 C1(OC)CCCC(CC(=O)N(C)CCN2CCN(C(=O)CCCC#N)CC2)C1 c1(OC)ccc(C(=O)NC2CCN(C(=O)CN3CCS(=O)CC3)C23CC3)c(Cl)c1 c1(C(=O)NCC(CNC(CC(C=C)C)=O)F)ccc(OC)c2occc12 c1(-c2cn(C(C(=O)NCC(C(=O)OC)C)C)nn2)nnc2n1CCC2 c1(C(N(CCCNC(C2(C)CCOC(C)C2)=O)CC)=O)ccc2cnc(C)n2c1 C1(CNC(C2C(C)CCCC2)=O)(N(C(=O)CCCN=[N+]=[N-])CC)CCC(C)(C)CC1 C(CCCC(C)NC(=O)Cc1ccc(CO)cc1)NC(C1(CSC)CC1)=O C1(CC(=O)NCCn2cc(CNC(C(COC)C)=O)nn2)Cc2ccccc2O1 C1(NC(COCC(=O)NC)=O)CC2(C1)CN(C(c1[nH]c(C3CC3)nc1C)=O)C2 O=C1NC(CC(=O)NCCCOCCNC(c2cnc(C3CC3)[nH]2)=O)CO1 C1(C(C)NC(C(C2CCCC2)OC)=O)CN(C(=O)COC(C)C)CCO1 c1(OC)ccc(C(=O)NCCC(C)N(c2snc(C)c2C#N)C)c(Cl)n1 N1(C(C(c2ccccc2Cl)OC)=O)CC(NC(=O)C=C(C)C(F)F)C2(CCC2)C1 c1(C(N2CC3C(NC(CCC=CCC=C)=O)(C3)C2)=O)cccc2[nH]cc(Cl)c12 S(=O)(=O)(c1cccc(Cl)c1C)N1C(C(=O)Nc2c(Cl)cc(F)cc2Cl)CC(OC)C1 N1(C(C(c2cc(F)cc(F)c2)C)=O)CCC(F)C(NC(C2(NC(N)=O)CC2)=O)C1 N1(C(CN(C(=O)C(F)C2CCC2)C)=O)CCN(C(c2ccc(O)cn2)=O)CC1 c1(OCC(=O)NCC2(C)CCN(C(C(CCC)OC)=O)C2)cc(C)c(Cl)c(C)c1 c1(C(N2CC(F)(CNC(CCCCOC)=O)C2)=O)nn(C)c2ccccc12 c1(CCC)onc(C)c1C(=O)NC(C1CCCC1)CNC(c1sc(=N)[nH]c1C)=O N1(C(c2ccc(C#C)nc2)=O)CCC2(CCC2)C(NC(=O)CCNS(C)(=O)=O)C1 C(=O)(C(C(C)(C)C)C1CCCCC1)N1CCC(n2cc(OC(CC)(C)C)nn2)C1 Cc1nsc(C(=O)NC2CCC(NC(=O)C=Cc3ccc(C(N)=O)o3)C2)c1N c1(C(=O)NC2C(CCC)CN(C(=O)C=C(C)C(C)C)C2)cncc2[nH]ccc12 C(=O)(C(F)(F)C(O)C(C)C)NCCCCCCN(C(CCc1cc(C)[nH]n1)=O)C C1(OC)CC(NC(c2snnc2C)=O)CN(C(c2c(C)[nH]c(C)c2C)=O)C1 Cc1cn2nc(C(N3CC(NC(=O)CCC4(C)CC4)C4(CC4)C3)=O)cc2c(=O)[nH]1 c1(C(=O)NCC(C)(C)NC(C(C)P(C)(C)=O)=O)cccc2c1COCC2 C1(NC(c2cc(COC)sc2)=O)CCCN(C(c2cccn2C(C)C)=O)CCC1 N1(C(c2c(C)cn(C)n2)=O)CC2CC(NC(c3cccc(C)c3C)=O)C2C1 N1(C(c2cc(C)[nH]n2)=O)CCOC2CN(C(C34CCCN3CCC4)=O)CC12 N1(C(c2ncn(CC)n2)=O)CCOCC1CNC(=O)C(C)N1CC(C)C1 N1(C(C(c2cn(CCC)nc2)=O)=O)CC(C)(C)C1CNC1(CC(=O)OCC)CC1 C1(NC(C(C)NC(N)=O)=O)CN(C(c2csc3cccnc23)=O)C2(CCCC2)C1 N1(C(CC(CC)C2CCC2)=O)CCCC(NC(=O)CN2CSCC2=O)C1C C(=O)(C(C)CC(C)(F)F)N(C1CCN(C(c2nccc(C)c2O)=O)CC1)C c1(C(=O)OC)cccc(C(N2CCCC2CNC(C23CCCCC2C3)=O)=O)n1 c1(C(=O)OC)c(C)cc(C)nc1NC1CCN(C(=O)C2=CCC2)CC1C C(=O)(C1=NNC(=O)C1)N(CC(C)NC(C1CCOC1)=O)C n1(COCC)nnc(C(=O)Oc2ccc(SCC(F)(F)F)cc2)c1N N1(C(C(COCC)N=[N+]=[N-])=O)CC2(CCC2)CC1CNC(=O)CC1CCC(=O)O1 N1(C(=O)OCC)CCC(Nc2cnc(C(F)(F)F)cc2C)C(C)C1 c1(CC)noc(C)c1C(=O)NC1CCC(N(C(=O)Cc2ccc(Cl)cc2)C)C1 c1(OCC(=O)NCCCN(C2CCCC2)CC2(O)COC2)ccccc1[N+](=O)[O-] N1(C(c2c(CC)nn[nH]2)=O)C2COCC1CC(NC(c1cc(C)[nH]n1)=O)C2 N1(C(C2(CCCC)CCC2)=O)CCC(NC(=O)CCC2CCCN2C)C(C)C1 N1(C(C(C2CCC2)OC)=O)CC(CNC(c2cc(C)cs2)=O)C(F)(CO)C1 c1(C(=O)NCC(C)(C)NC(CNS(CCCOC)(=O)=O)=O)c(F)cc(F)cc1F C1(C(=O)NCC2(NC(c3ccc(C)cc3F)=O)CC(OC)C2)CC2(C1)CC(C)C2 C(N=c1[nH]c(=N)[nH]c(=NC2CCN(C)CC2)[nH]1)C1(CN(C)C)CC1 CS(=O)(=O)c1ccc(NC(c2nc(-c3cc(F)c(F)cc3F)cs2)=O)cc1 C1(C(=O)NC2CC(C(=O)NCC(C)C(F)F)C2)CC(=O)C12CCC2 c1(C(=O)NCCN(C(C2CC2c2ccccc2F)=O)C2CC2)cc2[nH]ccc2s1 C(=O)(C(O)CC(C)C)N(CCC)CCNC(=O)C(CC1(C)CC1)c1ccccc1 N1(CC(=O)NC)CCN(C(=NCCF)NCC2CCS(=O)(=O)N2)CC1 c1(OC)ccc(F)c(C(N2CCC(NC(c3sc(C)cc3OC)=O)C(F)C2)=O)c1 CC(C)CC(C(=O)N(C)CC1(F)CCC1)NC(=O)CC1(O)CCCOC1 C1(NC(C=CC(CC)C)=O)CCN(C(c2cccc(Cl)c2N)=O)C1(C)C N1(C(CC(=C=C)C)=O)CCN(C)CC1CNC(=O)C(C)OCc1ccc(C)cc1 C1(C(=O)NC2(CCC)CCC2)(C(C)C)CCCN1C(C1CSC1)=O N(C1c2ccccc2CCC1CO)Cc1ccc(C(=O)Nc2c(N)cccc2)o1 N1(C(C#CC(C)(C)O)=O)CCOC2(CCC(NC(c3ccc(O)nc3)=O)CC2)C1 c1(C(=O)NCC2C3CN(C(CC(CC)C4CC4)=O)C2C3)cccc2nc[nH]c12 N1(C(C(COCC)C)=O)CCC(C2CCCN(Cc3csnn3)C2)CC1 Cc1ccc(C(C)C(=O)N(C(C)CCNC(=O)C=C2CCOCC2)C)s1 N1(C(C(N(C)C(C2CNC(=O)O2)=O)C2CC2)=O)CC2CCCC2(CO)C1 C1(COC)(CNC(C2CC3CCC2C3)=O)CCCN1C(=O)C(O)Cn1cncn1 C1(NC(=O)CCc2ccncc2Br)CCN(C(=O)C=Cc2cnc[nH]2)CC1O CCCCC(C(=O)NCC1CCN(CC)C1)NC(=O)CC(CC)C1CCC1 C(=O)(C1Cc2ccc(F)cc21)NCC(C(C)C)NC(=O)CNC=O C(C)(C(F)(F)C(F)(F)F)=CC(=O)NCC1(O)CC(CNC(C(CC)N(C)C)=O)C1 c1(SC)cn(C)nc1CNC(=O)CC(CC1CC1)NC(=O)C(N)=O c1(OC)ccc(CNC2CC(C(=O)NCc3ccc(OC)cc3Cl)C2)cc1Br c1(NC(C(C2CC(NC(CC(C)O)=O)C2)F)=O)cccc2c1OCC2 CC1CCCN(C(=O)Cc2ccccc2)C1CNC(c1ccc(C(N)=O)cn1)=O c1(OCCC(=O)NC(CN(CCCO)CC)C)ccncc1 CCC(CC(=O)NCC1(CCO)CN(C)C1)NC(c1cn(C)nc1C)=O N1(C(C2N(C(c3c(Br)c(C)n(C)n3)=O)CC2)=O)CCc2ccc(C#N)cc2C1 c1(C(=O)Nc2cncc(-c3cccnc3)n2)ncc(F)c2ccccc12 C1(NC(C=C(C)C(C)C)=O)CCC(C)(CNC(c2ccc(F)cc2)=O)C1 CCC(C)(C)CC(=O)NCC=CCNC(c1cc(C(F)(F)F)cs1)=O CC1CN(C(C2(C)CC(C#N)C2)=O)CCC1C(=O)NC1CC2CCCC2C1 N1(C(c2cccc(CC)n2)=O)CC2CCN(C(c3cccc4nccn34)=O)C2C1 C1(CC(N2CC(COC)(CNC(c3cc(C(C)C)no3)=O)C2)=O)CCOC1(C)C C1(C(=O)OC)(OC)CCCN(C(=O)C(c2cccc(Cl)c2F)NC(C)=O)C1 N1(C(C2(C#N)CCCCC2)=O)CCC2(CCC(NC(c3cncs3)=O)CC2)CC1 c1(NC(C2OCCN(C(c3n(CC)ccc3)=O)C2)=O)ccc2c(c1)CCO2 N1(C(C(CC)C(F)(F)F)=O)CCN(C(c2cc3n(n2)CCCO3)=O)C2(CCC2)C1 C=CC(C)(CCOC)C(=O)NCCN(CCC)C(c1cc(C(F)F)cs1)=O C1(N(C(CCC2N(C)CCC2)=O)C)CN(C(=O)CS(C)(=O)=O)CCC1O C1(NC(c2n(CC(C)C)ncc2)=O)CC(C)CN(C(c2cncn2C2CC2)=O)C1 c1(C(=O)NC2CCC(N(C(=O)COC(F)(F)F)C)C2)cc([N+](=O)[O-])n[nH]1 CC1CN(C(=O)COCC2CCCO2)CCC1CNC(c1ccnc(Cl)c1)=O C1(NC(C2CC(OC)C2)=O)(CNC(c2csc(C)c2)=O)CCCCC1C Nc1cnc(Br)c(C(=O)NCCNC(C2CCCS(=O)(=O)N2)=O)c1 CC1C(NC(=O)COc2cccc(F)n2)CCCN1C(=O)CCCC1CC1 c1(CC(=O)NCCC2CC(OC)CN2C(=O)CC=C(C)C)csc2sc(C)cc12 C1(CNC(C=CC(=O)OCC)=O)CC(C)(C)CN1C(=O)CC1CC(C)C1 n1(CC(N2CCC(C(C)(C)NC(C3(F)CC=CC3)=O)C2)=O)ncc2ccccc12 C12(C(=O)NC(C(CCC)C)C)CCC(CC1)N(C(c1cc(C)n(C)c1)=O)C2 C(=O)(CC(C)n1cc(Br)cn1)NCC(C)(C)NC(C(C1CC1)OCC)=O C1(C(=O)NCCC(C)N(C)C(C2COCCN2C)=O)CC2C=CC1C2 c1(-c2occc2)cccc(-c2cnc(N3CCC(CN4CCCC4)C3)nc2)c1 c1(OCC(=O)NCC(CC)NC(=O)C(C)(F)F)cccc([N+](=O)[O-])c1 Cc1ccc(CC(N2CC(O)(Cn3cc(Cn4nc(C)cc4C)nn3)C2)=O)cn1 O=S(=O)(c1cccc(=NC2CCSCC2)[nH]1)NCc1ccc(Br)cc1F c1(C(CC)(C)C)ccc(C(=O)NC2(CO)CN(C(=O)C(C)c3cccs3)C2)cc1 c1(CCCC)nc(C)c(CC(=O)NC2CN(C(C3CC(C)(O)C3)=O)CC2O)s1 C(=O)(CCCC(F)(F)CO)NCCCOC1CCN(C(COC(CC)=O)=O)C1 C(=O)(C(O)C(F)(F)F)NC(C(=O)NCC1(C)CCOCC1)CCC1CCC1 c1(OC)c(NC(=O)C=C2CCN(Cc3c(F)cc(O)cc3F)CC2)cc(Cl)cc1Cl Cc1nc2n(n1)CC(CNC(=O)C(N1CC(CO)OC(C3CC3)C1)=O)CC2 c1(NC(C2CCN(C(C3(F)CC3)=O)CC2)C)c(Br)cncc1[N+](=O)[O-] Cc1nc(O)[nH]c1C(=O)NC1(CNC(C2CCCC2C(C)C)=O)CCOC1 c1(CC)c[nH]nc1C(=O)NC1CC(OCC(=O)NC2CCC(CO)C2)C1 CC1CCC(CNC(=O)CCc2cscn2)N(C(=O)C(C2CC2)C2CC2)C1 C(C(C)(C)C(F)(F)F)N(C(C(c1ccnn1C)NC(C)=O)=O)C(=O)C1CC1 S(=O)(=O)(c1ccc(N(CC(F)Cl)C)c(Cl)c1)NCCC(=O)NC C12(CNC(N3CCC(C(C(N)=O)F)CC3)=O)CC(C#N)(CO1)C2 C1(NC(CSCC)=O)CCCC(C(N2CC(N3CCC3)C2)=O)CC1 c1(C(N(CC(C)CNC(C2(CF)CCOCC2)=O)C)=O)cccc(F)c1F Cn1cc(C(=O)NCCC2CCCN2C(=O)COC2CC=CC2)c(O)n1 C1(NC(CC(c2ccc(C)cc2)(C)C)=O)CCN(C(=O)C(O)C2CCC2)CC1F C1(CCC(=O)NCCC#CCC)CCCCN1C(c1cc(C)nn1C1CC1)=O N1(C(=O)NC2CC(CC)C2)CCC(C)(CSC)CC1 N1(C(C2N(C(c3c(C)[nH]cc3)=O)CCC2C)=O)C2CCC1COC2 C1(CC)(NC(c2nnn3c2CCC3)=O)CCCN(C(=O)CCOC2CC2)C1 N1(c2snc(CCC)n2)CCCC2(NC(C3CCCC4CC34)=O)CC2C1 N1(C(CCN(C)CCO)=O)CCCC(F)(C(=O)NCC2CCC(O)CC2)C1 c1(OCCC)ccccc1C(=O)NC(CC)C(C)NC(c1ccc(CO)cc1)=O C1(C(=O)NCC2C(C)CC2)CNC(=O)CN1C(c1ccncc1N)=O c1(C(=O)NC(c2cccs2)C)c[nH]c2ccc(-c3scc4c3OCCO4)cc12 N1(C(COCC#C)=O)CC(NC(c2ccc(C(F)F)nc2)=O)CC(C)(C)C1 CC(C)C(O)CONC(C1C(C)CN1C(=O)CCN)=O C12(C(=O)NCc3onc(N(C)C)n3)CC1CCN2C(C1CC(O)C(F)C1)=O CS(=O)c1ccccc1C(N1CCC2(NC(c3cc(C#N)c[nH]3)=O)CCCC12)=O c1(CC)ccccc1CC(N1CCC(C(C)NC(c2ccc(CC)nc2)=O)C1)=O C1(C(=O)NC2CC(CC)C2)COCCC1NC(c1cc(Cl)no1)=O C1(NC(c2c(C)ccs2)=O)CN(C(=O)C(N)=O)C2(CCOC2)C1 CCC(C(=O)NCCCCNC(C1CCN(c2nc(=N)[nH][nH]2)C1)=O)NC(C)=O CCC(C)C(O)C(=O)N(C)CC1(NC(=O)CC2COC(C)(C)CO2)CC1 c1(C(=O)NC2CCC(NCc3c(OC)cc(O)cc3)C2)n[nH]c2ccc(Cl)cc12 C1(O)(CNC(=O)CC2(O)CCC2)CCN(C(c2cnnc(Cl)c2)=O)C1 N1(C(c2ccc(Cl)s2)=O)CCC2CN(c3cc4ncnn4cn3)CCC12 C(N=c1[nH]cnc(Cl)c1F)C1CCC(NC(c2c(C)nc(CC)o2)=O)CC1 C=C(Cl)C(C)(C)C(=O)NCC1CN(C)CCN1C(=O)COc1cncc(C)n1 c1(C(=O)NCC(C)N(C(=O)COC2CCCC2)CC)cc(F)cc(F)c1 C1(CC(=O)OCCOc2c(OC)cc(O)cc2)Cc2cc(F)ccc2O1 C#CC1(O)CC(C(=O)N(C2CCN(C(=O)C(C)=C3CCC3)C2)C)C1 c1(C(C(=O)NCCOCCCN(C(C2C(C=C)C2)=O)C)CC)c(C)noc1C C1(CCC)(NC(=O)C(C2CC2)OC)CCCN(C(C2CC(F)(F)C2)=O)C1 C1(CC)CC(CC(=O)NCCC(C)(C)CNC(=O)Cc2ccsc2)CCO1 C1(NC(COCC#C)=O)CCC2CCN(C(C3CCCCN3CC)=O)C12 N1(Cc2c(F)ccc(C)c2Cl)CC(C)Cc2cccc(F)c21 CCCCC(CNC(=O)CC1(C)CCCO1)NC(=O)CC1CN(C)C1 c1(OC)cccc(NCC(=O)N(C)CC2CCCCC2)c1Cl c1(C(=O)NC2CC(C)(NC(c3cc(OC)n(C)n3)=O)C2)cc2c(Cl)cncc2s1 CC1CCC(C(N2CC(F)(CNC(C34CC(F)(C3)C4)=O)C2)=O)C1 c1(C(=O)NCc2c(C(=O)NC(c3nc(C)sc3)C)con2)cnc(O)cc1C C=Cn1ncc(C(=O)NCC(O)CC(=O)N2CCC(CCCO)C2)c1N C1(CCNC(COCCC(C)C)=O)CN(C(C2(C)CC=CCC2)=O)CCS1(=O)=O N1(C(CC2N(C(CC3CC3)=O)CCC2)=O)CCC(COC(C2CCOC2)=O)CC1 c1(CNC(=NCC(C)C)NCC2(CC(N)=O)CC2)ccc2c(c1)C(=O)NCC2 c1(C(=O)NC2CC(C)(NC(C(CC)c3ccccc3)=O)C2)nnn(C(C)C)c1C c1(C(N2CC(CC3C(=O)NC(=O)N3)C2)=O)ccc2c(n1)CCCC2 N1(C(=O)CO)CCCC1CC1CC(Cn2cc(CCCO)nn2)C1 N12CCCC1C1CCCN1C2=O.c1(N)ccc(I)s1 CC1CCN(C(=O)CCc2nncn2C)C(C(=O)NCC2(F)CCOC2)C1 Cc1cc(C(=O)NCC(N2CC3C(C(=O)OC4CCCC4)C3C2)=O)c2cc[nH]c2c1 c1(C(=O)NC(C(=O)NC2C(C)CCC2C)Cc2ccoc2)cn(C)ccc1=O C(C(C(C)(C)C)NC(C1CN(C)C1)=O)NC(C1CC(CC)(CC)C1)=O c1(OC)ccc(-c2cnccc2-c2nccn2CCOc2ccccc2)cc1F C1(C(C)C(N2CC=CC2c2nc[nH]n2)=O)CCCN(C(C2COCC2(C)C)=O)C1 C(=O)(CCCCC#N)N1CCC(C2N(C(Cc3cnc(C)s3)=O)CCCC2)C1 N#Cc1cscc1C(=O)NC1(CNC(=O)CCOc2ccccc2Cl)CC1 C(=O)(C#CC1(C)COC1)NC(CCCOC)C(=O)NCP(C)(C)=O C1(C(=O)NCCC23CC(CO2)C3)CCCCCCN1C(=O)Cc1cn[nH]c1 CC(CN(C)C)C(=O)NC1CC(C)(NC(=O)CC(=O)N(C)C)C1 CCC(CC(=O)N1CCCC1C(=O)NCc1cc(OC)ncn1)C1CCC1 CC1(C(=O)NCC(C2CCOC2)NC(=O)C2=NNC(=O)C2)CCS(=O)(=O)CC1 c1(C(C(=O)NC(C)CCNC(=O)CN2CCCCC2)C)ccc(F)cc1 CCCCC(C)C(=O)N(CC(=O)Nc1cncc(F)c1)C(C)C c1(C(=O)NCCCN(C(CCCc2nc(C)sc2)=O)C)nsc2ccccc12 C1(CNC(C(C(C)C)NC(C)=O)=O)CCC2(CCNCC2)CO1 Cc1cc(CNC(=O)CCN(CCO)C(C2COCC(C)O2)=O)oc1C C1(C(N2CCCC(CCC#C)C2)=O)CCC2CCC1N2C(c1cn2c(n1)CCC2)=O Cc1oc(C)c(C(=O)NCC(C2CC2)NC(C2CCCN2C(N)=O)=O)c1C N1(C(C(C)OCC=C)=O)CC(NC(=O)C(C)(C)c2ccns2)CC2(CC2)C1 c1(CC(=O)NC2(n3ccnn3)CCOCC2)ccc(Oc2ccccc2)c(Cl)c1 C1(C(=O)NCc2ccc(O)cc2C)(CC)CCCN(C(C2CC(C)=NO2)=O)C1 C1(COC)(NC(C2CC(C(=O)NCCc3ccsc3)C2)=O)CCCC1 Cc1cc(N2CC(C)OC(C)C2)ncc1S(=O)(=O)N(C)Cc1ccc(Cl)cc1Cl C1(NC(c2scc(C)c2)=O)CN(C(C2COCCC2(F)F)=O)C2CCCC12 CC(C)(CCNC(=O)CC1CCC(=O)C1)C(=O)NCCCN=[N+]=[N-] c1(C(=O)NC2CC3CC(NC(=O)CC4CC=CCC4)C2C3)cc2sccc2cn1 CC1CCCN(C(c2ncc(F)cn2)=O)C1CNC(=O)Cn1ccccc1=O C1(C(N2CCCC(C)C2)=O)CN(c2ccnc(C(C)(C)C)n2)CC(C)(C)C1 CC1CN(C(=O)Cn2cccn2)CC(C)N(C(=O)CCn2ccnc2C(C)C)C1 CCC(C)CCCCC(=O)NC(C)CN(C(c1ccc(P(C)(C)=O)cn1)=O)CC Cc1nn(CC(=O)NCC2CC(NC(C3CS(=O)(=O)C3)=O)C23CCC3)c(C)c1C N1(C(C(c2cnn(C)c2)OC)=O)CC(NC(c2cnc(O)cc2C)=O)CC(O)C1 Cn1c(CN2CC3CCCC(C2)N3Cc2ccccc2)nc2cc(Cl)ccc12 N1(C(CNC(CNC(C)=O)=O)=O)CCC(F)(F)C(CNC(C2CC23CCC3)=O)C1 C1(CNC(c2ccc(N(C)C)nc2)=O)CN(C(C2CC3CCC2O3)=O)C(C)(C)C1 c1(CNC(=O)CCC2CCCN2C(C2CCCCC2O)=O)cnc2n1CCC2 c1(-c2cn(CC3N(C(C4C=CCC4)=O)CC=C3)nn2)ccc2ccccc2c1 C=C(Br)CCC(=O)N1CC(NC(=O)C(C(C)C)SCC)C(F)C1 c1(CC)nn(C)c(C(=O)NCC(C)NC(c2ccn(C)c(=O)c2)=O)c1Cl N1(C(Cc2nccc(OCC)n2)=O)CCC(NC(=O)C(CCO)N(C)C)C1(C)C Cc1nc(C(=O)NCCC(O)CNC(C2(O)CCSCC2)=O)c(C)o1 c1(CC(N2CCC(Cn3cc(-c4cc(C(=O)OC)sc4)nn3)C2)=O)nn(C)cc1C C1(C(N2CCC(CNC(C3CC(SC)C3)=O)C2)=O)CCCC(C)(C)C1 C(=O)(C1CC(=O)c2ccccc21)NCC(C)N(C(C(C)OCC(C)C)=O)C c1(CC(N2C(CN(C(C=CC)=O)CC)CCCC2)=O)cc(F)c(F)cc1F c1(CCC(=O)NCCC(C)NC(C2(C(C)C)COC2)=O)ccc(N)nc1 N1(C(COCCCCC)=O)CCOCC(NC(=O)C(=O)NCCNC(C)=O)C1 C(=O)(C(C)(CC)CCC)NCC(CCNC(CC=C=C)=O)O c1(C(N2C(C(=O)NC(c3c(OC)cccc3)C)CCC2)=O)ncc(F)cc1C C1(C)(NC(C)=O)CCN(C(C2(CNC(C3C4COCC34)=O)CC2)=O)C1 N1(C(C(CC)NC)=O)CCC2(CC1)CC(C(=O)Nc1ccc(Cl)cc1C)CO2 Cn1cc(Cl)cc1CC(=O)NC1C2CC(NC(C3CC(C)(F)C3)=O)CC12 C1(CCOC)(C(=O)N(CC2=CCCOC2)C)CCCN(CC(C)O)C1 Cc1c(C(N2CC(NC(C34CC(CCO3)C4)=O)C2)=O)sc2ccc(Cl)cc12 c1(C(N(C2CCN(C(c3cc(C(F)F)cs3)=O)C2)CCC)=O)cn(C)cc1C N1(C(c2c(C)scn2)=O)CCC2CN(C(=O)CCC3CCCCN3C)CCC12 C12(CCNC(CC(C)(C)OC)=O)CCC(CC1)N(C(C1CCOC1C(C)C)=O)C2 C1(C(=O)NC(C2CN(C(C(C3CCC3)OC)=O)C2)C)CCC(N=[N+]=[N-])C1 CC1CCc2nc(N3CCC4OCCC4C3)[nH]c(=NC3CCC3)c2C1 c1(C(=O)NCC2OCCN(Cc3scc(C)n3)C2)cc2n[nH]cc2cc1Cl CC(C)C(C(=O)N(CC(C)(C)C#N)C)C(C)NC(=O)CCCn1cccc1 C(=O)CC(C)(CN)C(F)(F)F.C#CCC(C(C)(C)C)c1nc(C)no1 C1(CNC(Cc2nc(C)oc2)=O)CCC(F)(NC(c2nn(C(F)F)cc2Cl)=O)C1 c1(OCCOC)cccc(CC(=O)N(C(C)CNC(=O)C=C(Cl)Cl)C)c1 N1(C=O)CC(S(C)=O)C1.C1(CNC(=O)OC(C)(C)C)(CS)CC1(F)F C(=O)(CCC(C)SC)N1CCC(CCC(N2C(C(=O)NC)C=CC2)=O)C1 CC(C)CC(CNC(=O)CC1CCCOC1)NC(=O)C(C)CO c1(C(=O)NC2C(C(N3CC(OC)(CO)C3)=O)CC2)ccc(Cl)cn1 CC12CCC(CC1)N2C(=O)CNC(c1ccc(F)cc1Cl)=O CC1(C)C(CNC(=O)C(F)F)CCN1C(C1Cc2nncn2C1)=O c1(NC(CC)(CNC(=O)CC2CC3(CCC3)C2)CC)ccc([N+](=O)[O-])cc1C CCC(C)CCC(O)CC(=O)N(CCCCCCNC(=O)C1=CCCS1)C C1(CNC(C2(OC)CCC2)=O)CCCCN(C(C23CCC2C3)=O)C1 c1(C(=O)NCC2(F)CC(NC(C(C)C3CC3)=O)C2)cnc(OCC(F)F)c(Cl)c1 Cc1cc(F)ccc1C(O)C(=O)NCCCC1(NC(c2cnc(S)[nH]2)=O)CC1 c1(C(=O)NCC2CN(C(C)=O)C(C)(C)C2)ccc2c(c1)C=CS2(=O)=O CC1(C(=O)NC2CC(NC(=O)C(O)Cc3ccccn3)CC2O)CCCCO1 C(=O)(CC(C)(C)CNC(=O)C=CC1CCCCC1)N(CC=C)C(C)C C=C(Cl)CCC(=O)N1CCC(N(C(=O)C(C2CCCO2)OCC)C)CC1 C1(C(N2CCC(C3CC3)(NC(=O)CSC(F)F)C2)=O)CCC2(CC1)CC(O)C2 c1(OC)ccc(Cl)cc1S(=O)(=O)NC(=O)C(C1CCC(=O)N1)C CC(C)CC(CN=c1cc(C(N)=O)nc(Cl)[nH]1)NC(C1(O)CCCC(C)CC1)=O CC1C(NC(=O)Cn2ccnn2)CC2CCC1N2C(c1cccc(N)c1)=O C1(NC(c2cccc(OC)n2)=O)CCC(N=c2cc[nH]c(-c3nccs3)n2)CC1 N1(C(C(C=C)CC)=O)CCC2(CC2NC(c2ccc(F)c(C)c2)=O)C1 C#CCCC(=O)NCc1cn(CC(C)NC(=O)C(C)OCOC)nn1 Cc1c2cccc1NC(=O)C(=O)N2.c1(C(CF)OC(C)C)cccc(F)c1 Cc1cc(C)c(CC(=O)NCC2(NC(=O)CCc3ccc(F)nc3)CC2)cn1 N1(C(C=CCOC)=O)CCC(C(C(C)C)NC(=O)Cc2nocc2C(C)C)CC1 C(=O)(CCCCCCC(=O)N1CCCC1C(=O)Nc1ccc(C#N)cc1Br)OC c1(CCN2CC(CNC(C(CN(C)C)O)=O)OCC2)nnc2ccccn12 n1(CC(=O)N(CCCCNC(=O)C=Cc2cccnc2)C)ncc2ccccc12 N12CCC(CC1C)OCCC(O)C2.c1(N(C(CC)(C)C)CC)ccccc1 C(C)(C(=O)NC1CC(NC(=O)CC2(O)CCC2)C1)OC(C)=O c1(C(=O)NC(C(C)C)CCNC(C2CC3CC3C2)=O)ccn2ccnc2n1 CCCCCC(C)(C)C(=O)NC(CC(=O)NC1(C)CCC(=O)NC1=O)C(F)F C1(C(=O)NCCN(C(COC(CC)C)=O)Cc2ccc(F)cc2)CCCC(=O)N1 S(=O)(=O)(c1cc(F)ccc1C#N)NC1CCN(C(CC)CC)C1 c1(C(=O)NC2(CCNC(C(C(C)OC)O)=O)CCC2)cccc2nccn12 C1(NC(COC(c2nnc(C)s2)=O)=O)CCN(C(C2(CO)CCCCC2)=O)CC1(C)C C1(C(=O)NC(CCNC(c2ccc(C(CC)(C)C)cc2)=O)C)CCCCS1(=O)=O c1(C(=O)OCC(C(C)C2CCC2)=O)cccc2oc(C(C)C)nc12 CCC(CC(=O)Nn1ccccc1=O)N(C(=O)CC1CCOC1(C)C)C CN1C(=NC(=O)N(c2cnc3ccccc3c2)CC(F)F)NCC1C(F)(F)F CCCC(CNC(=O)Cc1ccns1)C(=O)NC(C)(C)CC(N)=O C1(CNC(C2(OC(C)C)CCC2)=O)CCCCN(C(c2cccc(CF)c2)=O)C1 N1(C(C=CC=CC)=O)C2CCC1CC(N(C)C(C1C(C)C1C)=O)C2 C1(NC(C(c2ccccc2)OC)=O)CN(C(C2CC(F)C2)=O)C2(CCC2)C1 c1(C(N(CCNC(CC2(COC)CCCC2)=O)C(C)C)=O)cc2cnccc2[nH]1 CCC(C)C(C(=O)NCC(C)(C)OCC(=O)NCc1ccc(OC)nc1)OC Cc1cc(C2CC2)ncc1C(N1CCCN(C(=O)C(C)OCCN(C)C)CC1)=O C1(C)(NC(C(C)CC2CCCC2)=O)CCCC1NC(=O)CN1CSCC1=O C(=O)(CC(C)(O)C1CC1)NCCN(CC)CC1CCC(C)CC1 N(C1CCCc2ccoc21)C(C1(NC(c2ncn(C(C)C)n2)=O)CC(CO)C1)=O c1(NC(=O)COC2CN(C(=O)NCC(c3ccsc3)=O)C2)cc(F)cc(F)c1 c1(C(C)C)ncc(Cl)c(C(=O)NCC2CCN2C(C2(C3CC3)CC=CC2)=O)n1 S(=O)(=O)(CC(=O)NCC1C(C)CCN1c1ncc(O)cn1)NC Cc1nc(Cl)ccc1CC(=O)NC1CCN(C(c2cc(O)no2)=O)CC1C CC(F)(F)C(C)(C)C(=O)NCC1CCC1NC(c1ccc(-c2cc[nH]n2)cc1)=O N1(C(c2c(OC)scc2)=O)CCC(C(F)(F)F)C(CNC(=O)C(F)=C(C)C)C1 C(=O)(CC(CN(C)C)C(F)F)N1CCCC(F)(CNC(C=CCCC)=O)C1 N1(C(C(CC(C)C)O)=O)CCN(C(=O)CCc2cccc(C#N)c2)CCC1C CC(C)(C)C(CO)C(=O)NCC1CC(NC(=O)Cc2ccc(F)c(Cl)c2F)C1 C(CS(=O)(=O)CC(=O)N1CCC1CNC(=O)C(N1CCCCCC1)C)OC N1(CCC#N)C(C)(C)CCCC1(C)C.c1(OC)ccc(Cl)cc1C(O)CN C1(NC(c2cnc(CC(C)C)s2)=O)CCCC(NC(C2(F)CCCCC2)=O)CC1 O=C1CCCCC1Cc1cn(CC(=O)NCC2CC3CCC3C2)nn1 N1(C(c2cc(C)ncn2)=O)CCC(C)C(CC(N2CC=CCC2)=O)C1 C(c1c(F)ccc(Cl)c1F)=CC(=O)NCCNC(c1cn(C(C)C)nn1)=O c1(NC)ccncc1C(=O)NCC1CCCN1Cc1ccc(C(=O)O)s1 CC12CCC(C(=O)C=Cc3cccnc3OC(F)F)(CC1)OC2 c1(OC)ccc(OC(=O)C(C2CC=CCC2)NC(C2CC(=O)CCO2)=O)cc1 C1(CN(C)C)CCCN1C(c1cn(CCNC(=O)C(C)(C)Cl)nn1)=O C(CCCCCN=c1[nH]nc(-c2ccccc2)o1)N(C(C(C(CC)C)OC)=O)C C1(C(=O)NCCN(C)C(C2CCOC2C(F)(F)F)=O)CC2OC(=O)OC2C1 C1(CS(=O)(=O)NC)CCN(CC2CC(=C)C2)CC1C c1(C(=O)NC2CCN(C(Cn3ncc(CC)c3)=O)C(C)C2)cnc2[nH]ncc2c1 C1(C(C)NC(C2(C)CC=CC2)=O)CN(C(c2nn(C)cc2N)=O)CCO1 CC(C(=O)NCC1(O)CC(C(=O)NCC2SCCS2)C1)S(C)(=O)=O C1(NC(=O)CC2COCCO2)CC(NC(c2cscn2)=O)C(O)C1 Cc1cccc(Br)c1CN1CC(NC(=O)N(C(c2nccn2C)=O)C2CC2)C1 c1(NC(=O)C2=CCC2)cccc(NC(C2C3CCCOC23)=O)c1 C1(O)(c2nc(CC(C)OC)nn2-c2ccc(Cl)cc2C)CCN(C)CC1 N1(C(C(C)SCC)=O)CCC2(CCC(CNC(c3ocnc3C)=O)OC2)CC1 C=CC1(C(N2CCC(OC3CC3)C2)=O)CCN(C(C2CC23CCC3)=O)CC1 c1(C(=O)NC2CC3CN(C(C4CCC(C)CC4)=O)C2C3)ncc(P(C)(C)=O)cn1 C=CCC(C(=O)NCCC1(NC(=O)C(O)C(C)C)CC1)C(C)C C(=O)(CC1OCc2ccccc21)N(C)CC1(CNC(CCC=C)=O)CC1 C1(NC(CCN(C(=O)CC2CCOC2)CC)=O)CCC2CC12 N1(C(C2(C)N(C(c3c(C)cc(C)s3)=O)CC(O)C2)=O)CCc2nc[nH]c2C1 Cc1cnn(C(C)C(=O)NCC2CC2NC(C2CC2c2ccc(Cl)s2)=O)c1 c1(C(=O)NC2(C(N3C(CC)CC(C)C3)=O)CCOCC2)cccc(=O)n1C c1(CN2CC3(C(C(=O)NCC4OCC(=O)NC4)C3)C2)cc2n(n1)CCC2 c1(C(=O)NC(C(=O)N2CC(OCCF)C2)c2ccoc2)ncc2ccccn12 CCC(CC(C)C)C(=O)NCCC(C)NC(C1CCC(C)C(C)C1)=O C(CNC(c1csc2cncn12)=O)(CC(F)(F)F)NC(CC(C=C)C)=O C1(NC(C2(C)CCCOC2)=O)CC2CC1N(C(c1c[nH]nc1C1CC1)=O)C2 C1(NC(C(C(CC)O)C)=O)CC2CCCC(C1)N2C(=O)CCSc1ccccn1 C(=O)(C1=CCC2CCC1N2C(c1cncc(Cl)c1)=O)N(CC(CC)O)C C1(C)(CNC(c2c(C)coc2C)=O)CC(F)(F)CN1C(c1ccnn1C)=O C(=O)(NNC(=O)CCCN)NCc1ncc(C(C)(C)C)[nH]1 c1(C(N2CC(O)(CNC(c3nc(CC)oc3)=O)C2)=O)n[nH]c2cc(OC)ccc12 C1(C(N(C)Cc2ccc(CC)o2)=O)CN(C(c2cnn(C)c2N)=O)C(C)(C)C1 C(C)(C(C(=O)NC(C)(C)CC=CC(=O)NCC1COCCN1C)N(C)C)OC n1(CCC(=O)NC(CC)CC(=O)NC2(C3CC3)CCCO2)c(O)nnc1O C1(C(N(C(CNC(c2ncc(CC)nc2)=O)C)CC)=O)CCc2cnnn2C1 C1(NC(C(c2ccccc2F)OC)=O)CCCN(C(C2OC(C)CC2C)=O)CC1 C1(OC)CC(CCNC(c2csc(O)n2)=O)N(C(=O)CCOCC2CCCO2)C1 C=C(C)CC(C(=O)NCC(C)(C)CNC(=O)Cn1ccc(C2CC2)n1)NC(C)=O C1(NC(c2c(CNC(c3nsnc3O)=O)occ2)=O)(CO)CC(F)(F)C1 N1(C(=O)Nc2c(C(C)(F)F)cccc2)CC2(CC2)c2ncccc21 CN1C(=O)CC(NC(N2CCN(C(=O)CCCC#N)CC2)=O)C1c1cnn(C)c1 N1(C(=O)CN2CCN(C(c3cccs3)=O)CC2)CC2CCC(C1)C2O N1(CC(=C)Br)CCc2cc(OC)c(F)cc2C1 N1(C(c2c(C)noc2)=O)CCCC(CCCCNC(=O)CN2CC3C=CC2C3)C1 C1(CNC(=O)CN2CC3CC3C2)CCC(C(N2CCC3CC23)=O)CC1 C(=O)(C(Cc1ccccc1)C1CCCC1)OCC(=O)NC12CSC(C1)C2 N1(C(C(N2CCSCC2)C)=O)CCN(CCNC(C2CCCN2C=O)=O)CC1 C1(CC)(CC)CC(O)CN1C(=O)CCN(C)C(c1ccn(CCF)n1)=O C1(C(=O)NC2CC(CNC(COCC(=C)C)=O)C2)CCCCC(C)(C)C1 c1(C(=O)NCCC(F)Cn2cc(C3CC3C(=O)O)nn2)cnc(O)c2ccsc12 N1(C(C(CCC)(C)O)=O)CCC2(CC1)CC2CNC(c1ccnnc1O)=O C1(C(=O)NCC(C2N(C(COCC(C)C)=O)CCC2)(C)C)C(F)(F)C12CC2 c1(C(=O)NCC2C(CNC(C3(CC)CC3)=O)C2)cc2ccc(F)cc2nc1O Cc1cc(OCC(N2CCOC(C3CC(F)(F)C3)C2)=O)ccc1O C1(C(=O)NC2C(C)CCC2)CC2OCCC2N(C(=O)Cc2ccsc2)C1 c1(C(N2CC(NC(C(C(=C)Cl)(C)C)=O)CC3(C2)CC3)=O)ccc2c(cnn2C)c1 CC1CC(NC(C2C3COCC23)=O)CN(C(=O)C(c2ccc(F)c(F)c2)=O)C1 c1(CC(N2C3C(NC(C4CCC(N=[N+]=[N-])C4)=O)C(C3)C2)=O)cnn2c1OCCC2 CC1CC(NC(C2(O)CCSC2)=O)CN(C(c2cnn(C(C)(C)C)c2)=O)C1 N1(C(c2ccc(Cl)[nH]2)=O)CCC2OCCN(C(=O)CCC3CC3)C2C1 c1(C(=O)NC(CNC(C2CC3(C2)CC(F)C3)=O)CO)cc2cccc(Cl)c2s1 C(c1ccoc1)=NC(=O)NC(C12CC(CO1)C2)C C12(C(N3C(CN(C)C)C=CC3)=O)CCC(CN(C(=O)CCC3CCCC3)C1)C2 c1(C(N2CCC(NC(=O)C#CC3CC3)C(F)C2)=O)cccc2[nH]ncc12 C1(CNC(c2cc(SC)oc2C)=O)CC2(CC2)CN1C(=O)CC1OCCC1(C)C N1(C(C(CSC)(C)C)=O)CC2(CC(CNC(=O)Cc3cc(F)ccc3C)C2)C1 C(CC(C(=O)NCC(C)C1CC1)NC(c1ccc(OC)o1)=O)OCC C(CCN(C(=O)CCSCC)C)(C(C)(C)C)NC(C(c1ccc(CC)cc1)C)=O N1(C(CSCCOC)=O)CCC2(NC(=O)C=Cc3ccsc3)CCCCC12 c1(C(N(C2CCCN(C(=O)Cc3[nH]cnc3C)C2)CC)=O)ccc(C(C)=O)cc1 c1(C(C)=O)cccc(NC(C2CC(F)CN2C(=O)CC#N)=O)c1O Cc1cccc(C2CC2C(=O)NCC(C)(C)NC(C2(O)CC(C)(C)C2)=O)c1 O=S(=O)(c1c[nH]ccc1=NCC1CC2(C1)OCCO2)N1CCCCC1CCCO c1(CCCC)ccc(Oc2ccc(N(S(C)(=O)=O)Cc3nncn3C)cc2)cc1 c1(CC(=O)NC2CN(C(C3COCCO3)=O)CC23CC3)cc(Br)cnc1F C1(CCC)(NC(=O)CNC=O)CCN(C(c2cn(C)nc2C)=O)CC1 C1(CC(=O)NC(C)C(CO)NC(=O)CC2C=CCC2)COCCN1C C1(NC(c2ccc(C(C)=O)o2)=O)CCC(O)CN(C(c2nccc(C)n2)=O)C1 c1(CNC(c2cc(CNC(COC(C)=O)=O)[nH]n2)=O)cccc(Cl)c1 c1(C2N(C(C3C(NC(CC(=O)OCC)=O)CCC3)=O)CCC2)ccccc1F.C(=O)OC Cc1cc(Cl)ccc1C(=O)NCCC1CCCN1C(c1cnc(S)n1C)=O C1(CNC(CC(CC)CC)=O)CCC2C(CC1)C2(F)F n1(CC(C)C)[nH]c(CC(=O)NCC2(NC(=O)Cc3cnc[nH]3)CC2)cc1=O N1(C(c2cc(C)nn2C2CC2)=O)CC2(C1)CN(C(=O)Cc1cnco1)C2 CC(C)(C)CC(C)(C)C(=O)N.N1(C(C(CCCC#CC)C)=O)CCc2c[nH]nc2C1 c1(CCC(=O)N(C2(NC(CN(C(=O)OC)C)=O)CC2)C)ccc(Cl)cc1F CC(C)(O)C(F)C(=O)N1CC2CC1C2NC(=O)CC1=CCCC1 N1(C(c2cc(C)nc(C)n2)=O)CC(NC(C2(C(F)F)CCCC2)=O)CC(C)(C)C1 c1(OC)c(C(N2CC(F)CC2C(=O)Nc2cc(C)c(F)cn2)=O)cccc1Br N1(c2ncnc(C(C)(C)C)n2)CC2CC(NC(=O)C(O)C(C)(C)C)CC2C1 C1(CCC)(NC(=O)C(C)CO)CCN(C(c2cccc(F)c2SC)=O)CC1 C12(NC(CC(=O)OC)=O)CCCC1CN(C(c1nccc3occc13)=O)C2 C1(C(=O)NCC(C)(C2CC2)NC(COCC=C)=O)CCC(C(N)=O)CC1 c1(C(=O)NC2CC(C(C(=O)NCCC=CC)F)C2)cc(OC)n[nH]1 C(=O)(C(F)(CNC(c1cc(O)nc(C)n1)=O)C(C)C)N(C(CC)C)CCO N1(C(c2ncc(C)cc2C)=O)CCC(NC(c2cnn3ccsc23)=O)C12CCC2 N1(C(c2c(C)nn[nH]2)=O)CCCC(C)(C(=O)NC2C3C=CC(C3)C2CO)C1 c1(NC(C23C(CN(Cc4c(O)ccc(OC)c4)C2)C3)=O)cccc(C#N)c1F CN1C(=O)CSC1=CC(=O)NCC1(F)CCC(C(=O)NNC(=O)c2cn[nH]c2)C1 C1(COC)(NC(=O)C(C#N)C2CC2)CCN(C(=O)Cc2ccc(Cl)cc2C)CC1 N1(C(c2cc3c(Cl)cccn3n2)=O)CCC2OCCN(C(C3CC(F)C3)=O)C2C1 C1(C(=O)NCC(c2ccccc2)CNC(CCCOC)=O)(OC)CS(=O)(=O)C1 C1(CC(=O)N(CCC(C)NC(CC2(OC)CC2)=O)C)CCCCN1C c1(C(=O)NC2(COC)CN(C(C3CCCCC3(C)C)=O)C2)ccc(C#N)cc1C CC1(c2cccs2)NC(=O)N(CC=Cc2cccnc2C(F)F)C1=O C(=O)(CC(C)NC(N)=O)NCCC(C)N(C(C=CC(=O)OCC)=O)C CCC(CC(C)C)C(=O)N1CCC2(C1)CN(C(c1ccc(O)c(N)c1)=O)C2 c1(C(N2C(CNC(C(C(C)(C)C)(C)C)=O)CC2)=O)cccc2c1C(=O)NC2 C1(C)(C(=O)NCC(C)NC(c2ccc(NCC(N)=O)cc2)=O)CCCN1C c1(CC(N2CC(CC(C)NC(=O)C(CCO)N(C)C)C2)=O)cncc(C#N)c1 C1(C(N2CCCC(CNC(C(C(=O)OCC)F)=O)C2)=O)CCOCC1(C)C N1(C(c2c(C)nc(C)o2)=O)CC2C=CC1C(C(=O)NC1CN(C(N)=O)C1)C2 C(=O)(CC(C)C(F)(F)F)NCC1(C)C(C)CN(C(c2c(NC)nccc2)=O)C1 CCC(C)C(O)C(C)C(=O)N1CC(CC(NCP(C)(C)=O)=O)(OC)C1 c1(NC(C2CCOCC2)C=C)nccc(N(C)CC2CCN(C)CC2)n1 N1(CC)CCCC(C2CN(c3ncc(C(F)(F)F)cn3)C2)C1.C(=O)(CCCCCO)N CC1(C)CC(NC(=O)Cc2cc[nH]c(=N)c2)CN(C(c2ccc(Cl)s2)=O)C1 c1(C(=O)NC2CN(C(C3(C=C)CCCC3)=O)C2)cc(N(C)C)ccc1F c1(Nc2ccc(SC)cc2)c(NC(=O)C(=O)N(CCCO)C)c(C)nn1C Cc1cc(=NC2CCN(C(c3cccc4cc[nH]c34)=O)CC2C)[nH]cc1C#N c1(OC)nc(Cl)ccc1C(=O)N(CCC(C(C)C)NC(=O)CC(O)C(C)C)C c12cccc(c1)CNC(C)C(=O)N2.c1(C(=O)OC)cnn(CCO)c1 N1(C(C(C)CO)=O)CCC(CNC(=O)CC2CC(F)(F)C2)C(F)(F)CC1 c1(C(=O)NCC(CC(F)(F)F)NC(C(CCOC)C)=O)c(C)cc(C)oc1=O Fc1cc(-c2ccccc2Cl)ccc1CNCCC1COC1 C1(C(=O)NC2(C#C)CC2)CC12CCN(C(=O)CCOCC(F)F)CC2 CC1(C)CN(C(=O)C(CNC(C2(C)C=CCC2)=O)CC2CC2)CCS1 N1(C(C2C(C=C)C2)=O)CCCC12CCC(NC(=O)C=C(C)CCC)CC2 Cc1cccc(F)c1C(N1CCCC(CCCCNC(c2cnn[nH]2)=O)C1)=O C1(CNC(C(COC)OC)=O)CCC2(CN(C(=O)CSc3ccccc3)C2)O1 Cc1ccc(CCC(N2CC3CN(C(c4cncn4C)=O)C3C2)=O)c(C)c1 C1(NC(=O)CSC(F)(F)F)CCCC12CN(C(=O)Cn1cc3ccccc3n1)C2 n1(CCCNC(C(C)(c2cccs2)N(C)C)=O)nccc1C(=O)O N1(C(c2c(C(=O)OC)[nH]cc2)=O)CCC(O)(C(C)CNC(=O)CCN(C)CC)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CC)CNC(C1(COC)CC=CC1)=O C(=O)(C(C)(C)NC(=O)CC(O)C1CCCC1)N(C1CSC1)C n1(CCNCCC2CCOC2)nnnc1C(c1ncoc1C(C)(C)C)OC N1(C(CCOCC#C)=O)CCCCC1CN(C(=O)CCCCF)C c1(CC)cc(N)ccc1C(=O)NCC(O)CN(C(=O)Cc1ccns1)C C(=O)(C1=NOC2(CCC2)C1)N1CCC(CCNC(C(CCC#C)O)=O)CC1 c1(C(=O)NC(c2cccc(O)c2)C)nc2c(s1)CCCC2 c1(C(=O)NC2(C(=O)NC(C)C(F)(F)F)CCCC2)cc(F)ccc1F c1(C(C(N2CCC(NC(C3C4CC4C4CC34)=O)CC2)=O)=O)ccc(Cl)cc1O Cc1cnc(C(=O)NCC2(CCNC(=O)CC34CCC(CC3)C4)CC2)cc1Cl c1(CC(=O)NC2CC(C(=O)O)CC2O)ccccc1-n1cc(-c2nccs2)nn1 c1(CC(=O)NCCCCC2(NC(C(C=C)O)=O)CC2)cccc(OCC(C)C)c1 C1(NC(C2C(=O)NCC2)=O)(CNC(C2(C3CC3)CCCO2)=O)CCCCC1 CC1CN(C(=O)CC2CCCCC2NC(=O)C(C)CC(F)(F)F)c2ccccc21 c1(OCCC)ccc(CNC(C)CNC(C2CN(CC)CCO2)=O)cc1 c1(C(N2C(COC)CN(C(=O)CN(C)C(C)=O)CC2)=O)nc2c(s1)COCC2 c1(C(C)NC(N2CCC(C(N3CC4CC4C3)=O)C2C(C)C)=O)ccc(Cl)cc1 c1(C(=O)NC(CC=C)CNC(c2nn(CCC)cc2Cl)=O)cccc(C)c1CC CCCC(CCC)=CC(=O)NCC1(OC)CCN(C(=O)C(O)C2CCC2)C1 C(=O)(CCCCCCC)NCC1(C(=O)NCCCC)CCCO1 C(=O)(CCC(C)C)N1CCC(n2cc(C(C3ON=C(C)C3)N(C)C)nn2)C1 Cc1cc(C(=O)NCC2CC(NC(=O)CCc3ncc[nH]3)C2)cnc1C(F)F Cc1ccc2c(c1C(=O)NC1CCCC1NC(=O)C(C)c1cc[nH]n1)CCCN2 C(=O)(CCCN(C(=O)CC1C=CCCC1)C)N(C1C(C)CC1)C C1(CNC(C2(NC(C3N(CC)CC3)=O)CC(F)C2)=O)CC[Si](C)(C)C1 Cc1noc2cc(C(=O)NC3CCC34CN(C(=O)CN3CCCC3=O)C4)ccc12 Cc1cc(C(=O)NC2CN(C(c3c(F)cccc3Cl)=O)C2)ncc1C(N)=O c1(C(=O)NC(CCCC)CNC(C2(C(F)(F)F)CC(O)C2)=O)sc(C)c(C)c1C N1(C(C2C(OC)CCCC2)=O)CCC(CNC(c2c(C)nsc2C)=O)C(C)C1 N1(C(CS(CC)=O)=O)CC(C)(C)CCC1CNC(=O)C(C(C)O)N(C)C c1(NC2C(c3ccc(C)cc3)CCC2)ccncc1S(=O)(=O)NCc1cncs1 C1(C(N(C2CCCNC2=O)C)=O)CC2(CCN(C(C3CC34CC4)=O)C2)C1 C1(NC(c2cnc(C)[nH]2)=O)(CO)CCCN(C(C2CCCN(CC(F)F)C2)=O)C1 C(=O)(CS(=O)(=O)CCO)NC(CNC(C(C(C)(C)C)NC(C)=O)=O)(C)C1CC1 C(=O)(CCCC(F)(F)C(F)(F)F)N1C(C)(COC)CC(NC(=O)CC=C(C)C)C1 C(=O)(C1=CC2(CCN(C(c3csc(C#N)c3)=O)C2)C1)N1CC2C(C)(CSC2)C1 n1(C(N(CCN(C(=O)CCOC2CCCC2)CC)CC)=O)nc(C)c(C)c1C N1(C(CC2(CC=C)CCCC2)=O)CC(CNC(=O)C(C)CC)C(C)C1 CC1CCC2(CC2)N(C(C2CCC(C)(C)N(C(=O)CC3COCCO3)C2)=O)C1 C12(CNC(=O)Cc3cnc[nH]3)CCC1CN(C(c1ccc(C3CCC3)nc1)=O)C2 Cc1cc(C(=O)NCC2CC2CNC(C2(C)CCOC2)=O)nn1-c1ccccc1Cl N1(C(c2c(OC)nc(C)cc2)=O)CCN(C(c2ccc(F)cn2)=O)C(C)CC1C N1(C(C2CC(=C)C2)=O)CC(CNC(c2cc(O)nc(OC(C)C)n2)=O)C(F)(F)C1 c1(C(=O)NC2CCN(C(C(C)=CC)=O)CC2CO)ccc2c(c1)NC(=O)C2(C)C N1(C(CNC(N(C)C)=O)=O)CC2CCN(C(=O)C=Cc3ccc(F)cc3)CC2C1 c1(CC(N2CCN(Cc3cc(O)ncc3Br)C3CC23)=O)ccc(Br)cc1I C1(NC(=O)CC2CCOCC2)CC2CCC(C1)N2C(C1CNC(=O)N1)=O c1(C(N2CC(NC(C(c3cn(C)nc3C(F)F)C)=O)C(O)C2)=O)ccc(Cl)nc1N C#Cc1ccc(OC)c(C(=O)NC(C)(CNC(=O)Cc2ccc(F)cc2)CC)c1 Cc1ccc(CC(=O)N(C2CCN(c3nnc(C(C)C)o3)CC2)C(C)C)c(Cl)c1 Cc1cccc(C)c1CC(N1CC(C)(C)CC1CNC(=O)C(c1cccnc1)O)=O C=C(C)CCCC(=O)NCC1CCC(NC(=O)CCCC2CCCO2)C1 C1(CNC(Cc2c(C)con2)=O)CC(C(=O)NCCC2(C)CCCO2)=NO1 C1(O)(C(C)NC(C(C)=C2CC2)=O)CCN(C(C2CCC(=O)N2C)=O)CC1 C=CCCCCCCCC(=O)NCC(O)CCNC(=O)Cc1ccccc1OC CCC(CCC(=O)NC(CNC(C1CCC(=O)N1)=O)C1CC1)OC CC1(C(=O)OC(CCOCCNNC2CC3(CCC3)C2)=O)CC2C=CC1C2 C1(C(=O)O)(CC)CCCN(Cc2ccc(C(N)=O)cc2)C1 C(C(C)N=c1[nH]c2ccccc2nc1NC(=O)CCC(C)C)(C1CC1)OC O=C(CCCC(=O)NC1(CC(N2C3CSCC2C3)=O)CC1)C1CC1 C(=O)(C(C)CC1CCC1)NCCC1(C(=O)NCCC(C)O)CCC1 c1(C(=O)NC2C(NC(Cn3nnc(=N)[nH]3)=O)CCCCC2)cn2ccccc2n1 c1(C(N2C(CNC(CCC3N(C)CCC3)=O)CC2)=O)cnc2cccnc2c1 C(C)(N=c1[nH]c2cc(Cl)ccc2s1)c1ccc(NC(C2C(OCC)C2C)=O)cc1 c1(C(=O)NCC2N(C(c3ccc(C)o3)=O)CC=C2)cc(C)c(F)c(C)c1 C1(C(=O)NC(C)CO)CN(C)CCN1C(=O)CCS(C)(=O)=O c1(NCC2C(OCC)CC2)cc(F)c2nc(C)cn2c1 c1(C(=O)NC(C(N2CC(C#C)C2)=O)C)cncc(F)c1 CC1(C)CC(NC(c2conc2-c2ccccc2)=O)CN1C(=O)CNC(N)=O C1(NC(C2(SCC)CC2)=O)CN(C(=O)C2=COCC2)CC1c1ccccc1 C(=O)(C1=CCCOCC1)NCCC1C(C)CN(C(=O)CC2(C)CCOCC2)C1 N(C(=NCC(C)(C)C(=O)N1CCCC1)NCC1CCSC1)CC(C)(C)C N1(C(C2N(C)CCC2)=O)CCCC(NC(=O)C(F)(F)c2csc(Cl)n2)CC1 c1(OC)cccc2[nH]c(C(=O)NCC(CO)NC(=O)CCCCC(C)C)cc12 Cc1cc(C)cc(C=CC(=O)NC2CCN(C(c3ccoc3)=O)CC2(C)C)c1 c1(CN2CCCC(C(=O)NCCCC3N(CC)CCC3)C2)c(OC)cccc1F N1(C(c2c(C)nccn2)=O)CC(NC(=O)Cc2ccc(Cl)c(F)c2)C(C)(C)C1 C(=O)(CC1=CCCC1)NC1C(NC(CCC=CCC=C)=O)CCC1 N1(C(C2C(COC)(COC)C2)=O)CCC(CC2CN(C(C3COCCO3)=O)C2)C1 c1(NC(N2CC(NC(CN3CC(C)C3)=O)C2)=O)ccccc1OC1CCCCC1C c1(CN2CCC(CNC(C(C)Cc3cnn(C)c3)=O)C2)cc(O)cc(Br)c1 C1(NC(c2n(CCOC)ncc2)=O)CCCN(C(=O)C(n2nc(C)cc2C)C)C1 c1(C(=O)NC(C)CNC(=O)C=CCc2ccccc2)cn(C)c2ccc(F)cc12 C(=O)(CCCCC#N)NC(c1ccc(C)cc1)CNC(C1(Cl)CC12CCC2)=O C=CC(C)(O)C(=O)N(C)CCOCCNC1CCN(C(C)(C)C)C1 C1(C)(C(=O)NCC(CN(C(CCC=C=C)=O)C)C)CCC(=O)NC1 CC(C)CC(C)(O)C(=O)N1CCC(F)(C(=O)NC2CC(CCO)C2)C1 c1(C(N2CCC(NC(c3cnc(CCC)s3)=O)CC2)=O)cnn2c1CN(C)CC2 N1(C(C(CN(C)C)(C)C)=O)CC2(CCC(CNC(=O)CC3CC(=O)NC3=O)O2)C1 Cc1cnncc1C(=O)NCC1CC(C(F)(F)F)CN1C(=O)CCc1cnoc1 CN=c1[nH]cc(C(=O)NCCCCCNC(c2cncc(C(F)F)c2)=O)o1 CCC(CC)C(C(=O)NCCC1(NC(C2CC(OC)C2)=O)CCCC1)OC CC1=C(C(=O)NCC2CCCN(C(C3CCN(CCO)C(=O)C3)=O)C2)CCO1 N1(C(C(C)OCCC#C)=O)CC(CNC(c2csc(CCCCC)n2)=O)C(O)C1 CC(O)C(C(=O)NC1CC(CCC(=O)NCC2COCCC2O)C1)N(C)C C(=O)(C(C)(C)C(C)(C)C)OC.C12CCC3(CCC13)C(=O)NC1CC(C1)CN2 c1(C(N2CCCC(OCCO)C2)C(=O)NCCOC)nc(Br)sc1C C(C)(C)(CCC(=O)NCCOCC1CCC1)NC(CC(C)OC)=O C1(COc2ccc(C(=O)OC)cc2C)CN2CCCN1CC2 N1(C(CC2C(C)(C)C2)=O)CC2CC(C1)CN(C(=O)CN1CCC(CO)CC1)C2 C=CCC(CC=C)C(=O)NCC(c1cccc(C)c1)NC(c1cc(OC)ns1)=O Cc1ccnc(O)c1C(=O)NC1CCCC(N(C(=O)CC2CSC2)C)C1 C1(C)(CN(C)C(c2ccc(CC#N)cc2)=O)CCCC1NC(c1ccoc1Cl)=O C1(NC(=O)C(=Cc2c[nH]cn2)F)CCOCC1NC(=O)CC1CCCC12CC2 c1(C(N(CCNC(C(C)N2CCC2)=O)C)=O)ccc(=O)n2c1CCCC2 C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NCC(C1CC1)NC(C(COC)(C)C)=O Cc1cnc(Cl)c(CN2CC(C)(C(=O)NCc3ccccc3Cl)C2)c1 C1(COC)CC(CNC(c2cc(C3CC3)sn2)=O)N(C(C2CCOCC2)=O)C1 CCC(C)(C#N)C(=O)NCCC1CN(C(c2nccn2C)=O)CCCO1 C1(C(=O)NCC=C(C)C)CN(C(=O)CNC(C2CC2C)=O)CC1C(C)C c1(C(N2CC(F)CC(C(=O)Nc3cc(O)n[nH]3)C2)=O)ccc(F)c(F)c1O C1(NC(c2cc(OC)nc(Cl)c2)=O)CN(C(C2(CO)CC2)=O)CC2(CC2)C1 c1(OC)ccc(C(CNC(=O)C=CC2CC2)NC(C2OCCO2)=O)cc1 N1(C(CC(C)(C)NC(c2cccc(F)c2)=O)=O)CCn2nc(CO)cc2C1 N1(C(C(C(CC)(C)C)=O)=O)CC2CCCC(NC(c3ccno3)=O)C2C1 C1(COC)(CNC(c2ccnn2CC(C)C)=O)CN(C(=O)C(N)=O)C1 C1(C(N2CC3C(N(C(=O)C=C4CCSCC4)C)C3C2)=O)CCN(CCO)C(=O)C1 Cc1cc(C(=O)NCC2CC(CNC(C3CCC(C)(C)CC3)=O)CO2)nc(C)c1 N1(C(CC2CC(=O)NC2=O)=O)CCC2(CC1)CC(NC(c1ccncc1Cl)=O)C2 C(N=c1[nH]nc(C(C)(C)C)o1)C1C(NC(c2cc(CC)no2)=O)CCCC1 C1(NC(c2n(C)nnc2)=O)C2CCN(C(c3cccc(O)n3)=O)CC12 c1(OC)cccc2c(C(N3CCCC(NC(=O)CCC(F)(F)F)C3)=O)c(C)[nH]c12 C1(NC(c2c(CC)oc(C)c2)=O)CN(C(c2cc(COC)no2)=O)C2(CCC2)C1 C1(C(C(=O)NC2(N(C)C)CN(C(=O)CC(C)C)C2)NC)CCc2c(nnn2C)C1 c1(C(=O)OCC)cnn2c1N(C(c1ccnc(N(C)C)c1)=O)C(C)CC2 CC(O)CCCCCC(=O)N(CC(C)NC(c1coc(Br)n1)=O)C C(=O)(C(O)C(CCC)NC(=O)C(C)C(O)C(C)C)N(CC(=C)C)CC#C C1(C(=O)O)Cc2cc(F)ccc2N(C(=O)CC(O)C2CC2)C1.c12ccccc1C2 N1(C(COCC=C)=O)CCC2(CC1)CC(NC(c1cccc(C)c1)=O)CCO2 C(C#CC(=O)NC(C1CCCN(C(c2cccnn2)=O)C1)C)(OCC)OCC C1(CC(=O)C(C)C)CCCN(c2ccc(NCCc3cn(SCC)nn3)cc2)C1 c1(C(N2CC(F)(CNC(c3c(C(C)C)onc3)=O)C2)=O)cccc2c1NCCC2 N1(C(C2N(C(c3c(C)nsc3)=O)CC(=O)NC2)=O)CCCN(C)C(=O)C1 c1(C(N2CCC(C(=O)O)C23CCOCC3)=O)nn(C)c2ccc(F)cc12 N1(C2C(NC(c3cccs3)=O)COC2)CCN(C(=O)C2=CSCS2)CC1 Cc1nc(C(N2CCC(CO)(NC(c3[nH]ccc3C3CC3)=O)C2)=O)cn1C c1(C(N2C(CNC(c3c(C)sc(Cl)n3)=O)CCC2)=O)nc2sccn2c1C c1(OC)cc(F)c(C(=O)NC(C)CNC(c2ccc(C(N)=O)c(Cl)c2)=O)cc1N c1(C(C)C)ncsc1C(=O)NCCC(C)N(C(=O)C(C)Oc1ccccc1)C C1(CC)C(C(=O)NC2(C(=O)NCc3cncc(F)c3)CCOCC2)CCN1C C1(NC(CC(C)(C)O)=O)CN(C(=O)Cc2ccnc(O)c2)CC2(CCC2)C1 N1(C(COCC(=C)C)=O)CC2(C1)CN(C(=O)CCN1CCCC1=O)C2 Cc1cc2c(C(N3CC(CNC(c4ccc(C)s4)=O)CCC3C)=O)cccc2o1 c1(CNC(CCCCC)=O)nnc2n1CCN(C(C1(n3cccn3)CC1)=O)C2 C1(C)(CNC(CC(c2ccc(C)cc2)C)=O)CCCN(C(C2CNC(=O)N2)=O)C1 c1(C(=O)NCC2C(NC(C3(C)CCN(C)CC3)=O)C2)ccn2c1CCCC2 C=CCCC(C(=O)N(C)Cc1cccc(C)c1)NC(=O)Cc1ccccc1O C1(C)(NC(c2cc(CC)[nH]n2)=O)CCN(C(=O)CCc2ccc(Cl)s2)CC1 CC1(CCNC(=O)CCF)CCN(C(=O)C(O)c2ccsc2)CC1 c1(C(C)NCC)ccc(C(=O)OC)cn1.n12cc(nn1)NC(=O)C2 c1(CC(=O)NCCN(C(COCC)=O)CC(C)O)cnn2c1OCCC2 C1(NC(C2CCCC(C)C2)=O)(CO)CCCN(C(=O)COC(F)F)C1 c1(C(C)C)ncc(C(=O)NC(C2CCCCO2)C2CC2)[nH]1 n1(CC(=O)NC2C(C)N(c3ncc(C#N)cc3Br)CCC2)cc2ncccc2n1 c1(C(=O)NC2(CO)CCCN(C(CP(C)(C)=O)=O)C2)ccc(Cl)c(Cl)c1N N1(C(CSCC#C)=O)CC(NC(c2nc(Cl)sc2C)=O)CC2(CC2)C1 Cc1nc(SCC(=O)NCCC(O)CNC(C2C(C)C2C)=O)n[nH]1 C(C1CN(C(C2(CC)COC2)=O)CC1C(N1CC(F)(CF)C1)=O)=CC N1(C(C(CNC(C)=O)(C)C)=O)CCC(NC(=O)Cn2ccc(O)nc2=O)C(O)C1 C(CCC(C)C)(C(=O)N1CCC(C(C)OC)CC1)NC(C(CCCOC)C)=O N1(C(c2c(C)cccc2F)=O)CCOC2(CCN(C(c3cc(C)n(C)c3)=O)C2)C1 c1(OC)cc(CNC2CCCC2C(=O)NC2CCCOC2)cc([N+](=O)[O-])c1 Cc1ccc(C2CCN(C(c3nc(C(C)C)n[nH]3)C(=O)NC3(C)CC3)C2)c(C)c1 C1(C)(NC(C=C(C)C(F)F)=O)CCC(NC(c2cccc(C3CCC3)c2)=O)CC1 CC1CN(C(C2(C)CCCCC2)=O)CCN1C(c1cnn(CC2CC2)c1)=O C1(CC#C)(C(=O)NCC(C)(C2CC2)NC(=O)Cc2c(C)noc2Cl)CCOCC1 CC1CN(C(=O)C(N2CC3CCC2(C(F)(F)F)C3)=O)CC(C)(C)C1 C12(NC(c3n(CCC)nc(C)c3)=O)CC3CCC(C1C2)N3C(C12CC(F)(C1)C2)=O C(=O)(C#CC1CCOCC1)NC(C(=O)NC1CCC(OC)C1)C1(C)CC1 c1(C(=O)NC(CCNC(C2C(CCOC)C2)=O)(C)C)c[nH]c2ccc(Cl)cc12 c1(C(C(=O)NCC2CN(C(c3c(C)nns3)=O)C2)C)ccc(Br)cc1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1C(C)CCN(C(=O)CCc2ncccn2)CC1 C1(CC(N2CCC(N(C(=O)CN(C)S(N)(=O)=O)CCC)C2)=O)CCC(=O)N1C N1(C(c2cn(C)nc2)=O)CCC(C(C)(C)CNC(c2ncoc2C2CC2)=O)CC1 c1(SCC(=O)NCCNC(c2cc3scnc3[nH]2)=O)ccc2c(c1)CCC2 C1(C(=O)NCC2C(NC(CCCN(C(=O)OCC)C)=O)CC2)CC(=O)N(C)C1 c1(C(=O)NCC(CN(C(c2ccc(C)c(Cl)c2)=O)C)C)c(C)sc2ccccc12 C1(CC=C)(NC(=O)C=CC)CC2CCC(C1)N2C(c1c(C)ccnc1O)=O N1(C(C(C)CO)=O)CC(CNC(=O)C=C2CCOCC2)CC1(C)C c1(OC)cccc(F)c1C(=O)NCCCCNC(=O)C=Cc1ncc(C)[nH]1 Cc1cccc(C2(NCc3cc(C)[nH]c3C(=O)O)CCC2)c1 c1(CC)cc(N)cc([N+](=O)[O-])c1.C12CCC(O)(CC1)C(=O)N(CC(=O)C1CC1C)C2 N1(C(c2c(C)n(C)nc2)=O)CCN(C(=O)Cc2nn(C)cc2Cl)C(CC(F)F)C1 C1(C(=O)NCCN(C(=O)C(C)=C2CCC2)CC)CCCN1c1nccs1 S(=O)(=O)(c1ccc(NCCCCCN=[N+]=[N-])c(F)c1)N1CC(C)OC(C)C1 c1(OC)cnc(C(=O)NCCC2(O)CCN(C(C34CCCC3C4)=O)C2)c(F)c1 Cn1ccnc1C(=O)NC1CC(O)(C(=O)NCCOCc2ccccc2)C1 N1(c2nc(C)cc(C)n2)CCN(N2CCc3cc(F)ccc3C2)CC1 c1(CC)oc(C)cc1C(N1CCC(C(=O)Nc2cccc(F)c2)(CF)C1)=O c1(C(=O)NCC(CNC(c2ccc3n[nH]cc3c2)=O)F)nccc2ncncc12 c1(C(=O)NCC2CN(C(C(CCC)(C)O)=O)CC2C)ccc2c[nH]nc2c1 C(=O)(CCS(=O)(=O)c1ccccc1)Nc1ccc(OCC)c(OC)c1 c1(C(N2C3CC(CNC(C4C(C)(C)CO4)=O)C2CC3)=O)cccc2c1NCC2 CC1ON=C(C(=O)N2CC3(CC(NC(C4Cc5nncn5C4)=O)C3)C2)C1C c1(NC(C(C)C)CNC(=O)Cc2cc[nH]n2)cc(-c2cccs2)ncn1 C(=O)(C1COc2ccccc21)N(C1CCN(C(C2(CN(C)C)CC2)=O)C1)CCC N1(C(CCSc2ccc(C)cc2)=O)CCN(C(=O)C(O)C(C)(C)C)CC12CCC2 N1(C(CSCC)=O)CCN(C(=O)CC2CCCCN2C(C)=O)C(C2CCCC2)C1 c1(C(N(C2CCN(C(c3ccnc4ncnn34)=O)C2)C)=O)cc(S(N)(=O)=O)cs1 N1(C(CC2C(=O)OCC2)=O)CCC(N(C(c2cnn[nH]2)=O)CC2CC2)CC1 N1(C(C2=CCC(NC(c3ccoc3)=O)C2)=O)CCCC(C2CC2)CC1 CCN=c1[nH]cnc2cc(C(=O)NCC(C)NC(=O)C=Cc3cccs3)ccc12 C#CCCC(C(=O)NCc1ncnn1CC)NC(c1cc(O)cc(F)c1)=O C(=O)(CC1C(=O)Nc2ccccc21)NCC1CC(OC)CN1C(C1CCOC1)=O c1(OC)nc(Cl)c(C(N2CCC(NC(C34CC(F)C3C4)=O)CC2)=O)s1 N1(C(C(C(C)C)O)=O)CC(CNC(c2cc(C(F)F)ccc2F)=O)C(C)(C)C1 c1(C(=O)NCC2CCCN(C(C3CC(=C)C3)=O)C2)ccc(Cl)c(C)c1 CS(=O)CCC(=O)NCC1CCCCC1NC(=O)C(C1CCOCC1)F c1(CSCC)cc(C(N2CCC(N(C)C(c3cnn(C(F)F)c3)=O)C2)=O)no1 C1(OC)CCCC(CNC(=O)C(CNC(c2sccc2CO)=O)N(C)C)C1 Cc1ccc(CC(=O)NC(C)CCCNC(c2ccc(Cl)nc2O)=O)cc1Cl C1(CNC(C2(C)CC=C(C)CC2)=O)CN(C(=O)C(C)(C)C(C)C)CC2(CCC2)O1 C1(C(N(CC(CNC(C=C(C)C(C)C)=O)C)C)=O)CC2C=CC1CCC2 C12(NC(=O)COC3CC3)CC1CN(C(=O)CCc1cncs1)C2 C1(NC(CC)=O)CCN(C(=O)CCc2scnc2C)CC12CCC2 C1(NC(C=CC)=O)C(C)(C)C(NC(c2ccc(-c3nc(C)cs3)cc2)=O)C1(C)C N1(CCN(C(c2ncc(Br)s2)C(=O)NCCC#N)C)CC(=O)Nc2ccccc21 C1(NC(CCCCOC)=O)CN(C(C2SCCCS2)=O)C2CCCCC12 N1(C(C2(C)CCCN2)=O)CCOCC(C)(C(=O)NCC(c2ccccc2)O)C1 N1(C(Cc2ncc(C)[nH]2)=O)C2CCCC1CN(C(c1ccc(N)cc1Br)=O)C2 Cc1ncc(NC(=O)COCCNC(c2ncccc2O)=O)c(C)c1C CC1CC(C)(C(=O)NC2CC(CNC(c3nc(Cl)c(=O)[nH]c3N)=O)C2)CC(C)O1 C1(C(=O)NCC)CCN(C(c2ccncc2F)C(=O)NCCCF)CC1 c1(CNC2CCCC(COC)C2)c(C)n(C)c2ccccc12 Cc1cccc2c1CCOC2C(=O)NCC(CNC(=O)C1CC1)C(F)(F)F c1(OC)cnc(F)cc1C(=O)NC1CS(=O)(=O)CC1NC(=O)C(=O)N(C)C c1(C(=O)NCC2(C(F)(F)F)CCOCC2)ccccc1C(F)(F)C(F)(F)F C#CC1(O)CCCN(C(=O)C(c2ccc(Cl)cc2)OC)C1 C(=O)(C(C)(C)CC(F)F)NCCC1(C)CCN(C(c2scc(C)c2C)=O)C1 c1(OC)cc(F)ccc1CN1CCC1C(=O)Nc1ccc(CO)cc1 C1(NC(C(N(C(=O)CC2OCCCO2)C)C2CC2)=O)COC2(CCC2)C1 C1(C(N(CC(CNC(C(C)(C)OC(C)C)=O)C)C)=O)CCC(C)C(C)C1 c1(Nc2ccc(Oc3cccc(C(=O)OC)c3)nc2)nccc2ccc(N)cc12 N1(C(C(C)OCCOCC)=O)CC2(C1)CN(C(c1cc(Cl)ncc1O)=O)C2 O(NC(=O)C(C1CN(C(=O)C(F)F)C1)OC)CC#C c1(C(N2CCC(CC(C)NC(C(CC)(C)C)=O)CC2)=O)ccc(F)c(F)c1C N1(C(c2c(C)[nH]cc2)=O)CC(CNC(c2cc(=O)cc[nH]2)=O)CC(C)(C)C1 CC(C)(CC(=O)NCC1(NC(c2cc(C3(C)CC3)n[nH]2)=O)CC(F)(F)C1)C1CC1 N1(C(c2c(CC)c[nH]c2)=O)CC(CNC(C2CS(=O)(=O)C2)=O)C(O)C1 C1(C(=O)NCCCCNC(C(CC)n2cncn2)=O)(CO)CCCCC1 N1(C(c2ccn(CC)c2C)=O)CC2(CNC(C3(CC)CCCC3)=O)CCC1CC2 C(=O)(Nn1cnnc1C)C1N(C)CCN(C(C(C(C)C)OC)=O)C1 N1(C(C2(CCOC)CCC2)=O)CC(C2(NC(=O)CCCc3ccc(C)s3)CC2)C1 C1(CNC(CN(CCC#C)C)=O)CCN(C(=O)C(C)C=C=C)CC1 S(=O)(=O)(c1c[nH]c(=NCC(C)C(C)(F)F)cc1C)NC(C(CC)C)CO C1(NC(C=CC=CC)=O)CC(CNC(=O)Cc2ccc(O)cc2C)C12CCC2 Cc1ccnnc1C(=O)NC1CN(C(c2cc[nH]n2)=O)CC1CC(C)(C)C C12(NC(CCC=C)=O)CC1CN(C(=O)C(C1CCOCC1)OCC)C2 c1(OCC=C)cc(Cl)ccc1C(=O)NCC(C)N(C)C(c1cncs1)=O c1(CCCC(=O)NC2CCC(N(C)C(c3ccnnc3)=O)C2)ccc(CO)cc1 C1(C(N2CCC(C)(CCNC(C(C)(C)n3cccn3)=O)C2)=O)CCS(=O)(=O)CC1 c1(C(=O)NC(C2CCCC2)CNC(c2ccnc(S)c2)=O)ccc2cnoc2c1 N1(C(C2OCC(C)(C)C2)=O)CC(C(N2CCC(CO)C(O)C2)=O)C(C)(C)C1 CC(O)C(C)C(=O)N1CC(CCCCNC(=O)C(=Cc2cccnc2)F)C1 CC(CC1CC1)C(=O)N(C)CC1(NC(=O)CCc2ncno2)CC1.c1ncc[nH]1 CC1=C(C(=O)NC(C(=O)NCC2CCCCN2C(C)C)C2CCC2)CC1 N(S(=O)(=O)N(C)C)CC(N1C(C2CCN(C(CCN(C)CCO)=O)C2)CCC1)=O C(=O)(C(C)(Cc1ccccc1)C(C)C)NCC(CNC(CN(C1CC1)CC)=O)O C(CCCCC(=O)Nc1ccc(F)cc1OC)NC(CC1(NC)CCC1)=O c1(C(=O)NCC(C)OC)ccc2c(n1)CN(C(=O)C1=NOC(C)C1)CC2 c1(C(=O)NC(CNC(CC2C(C)(C)C2)=O)CO)cc(Cl)cc(Cl)c1O C1(N(C(C=CC(C)NC(=O)C(c2cnn(C)c2)O)=O)CCO)CCCCC1 C1(NC(CSCCC)=O)CCC(NC(C2(COC)C=CCC2)=O)C1 N1(C(C2(F)C(C)(C)C2(C)C)=O)CCCC(C2CN(C(=O)COCP(C)(C)=O)C2)C1 N1(C(C2N(C(C)=O)CCC2)=O)CCCC(C)(C(=O)NCc2nn[nH]c2C(=O)O)C1 CC1CCN(C(=O)C#CC(C)(C)C)CC1CNC(c1cnn2c1CCC2)=O C(C(CC(C)C)NC(c1cnnc(O)c1)=O)NC(Cc1cnc(C)[nH]1)=O C(=O)(C(C)(C1CC1)OC)NC(C(=O)N(CCC(=O)OCC)C)C1CCOC1 c1(CC)ccc(C(=O)NCC(C)(F)CNC(c2n[nH]c(C3CC3)n2)=O)o1 S(=O)(=O)(c1ccc(N2CCC(c3cccs3)C2)c(Cl)c1)N(CC(C)C#N)CC c1(OC)cc(C(=O)N(CC(C)O)CCNC(c2cc(C(C)C)nn2C)=O)ncn1 c1(C(N2CCOCC(NC(CCC(=C)C)=O)C2)=O)cc(O)cc([N+](=O)[O-])c1 CS(=O)(=O)CCC(=O)N1CCC(OCCNC(C2OCC3CCCC23)=O)C1 c1(CC(=O)N(CCCCCCNC(=O)Cn2nnc(=N)[nH]2)C)ncn2c1CCC2 c1(C(=O)NC2(CNC(CC3CCN(C)C3=O)=O)CCC2)cccc2c1CCC2=O C12(NC(c3c(CC)nccc3)=O)CCC1CN(C(c1cn3ccnc3s1)=O)C2 N1(C(C(C)CCN(C)C)=O)CCC(c2cn(-n3cnccc3=O)nn2)CC1C N1(C(c2cncc(OCC)c2)=O)CCCCCC(N=c2[nH]nc(O)s2)C1 C1(C(N(C)Cc2cn(CC)nn2)=O)CC(O)CCN1C(C1CCCO1)=O N1(C(c2c[nH]c(=NCC)s2)=O)CC(NC(C2CN(S(C)(=O)=O)C2)=O)CCC(O)C1 C=CC1(C(N2CCCC2C2(C(=O)N(CC(O)CN(C)C)C)CC2)=O)CCOCC1 C1(C2CCC2)(C(N2CC(O)(C(C)NC(C3CCC(F)C3)=O)C2)=O)CC1(F)F N1(C(C(C)OC)=O)Cc2ccccc2C1CNC(=O)CN1C(=O)CCCC1=O C1(OC)CCC(c2cn(C3CCCCC3NC(=O)Cc3nc(=N)[nH][nH]3)nn2)CC1 Cc1ccc(N)c(C)c1C(=O)NC1CN(C(c2cc3c(s2)CCCC3)=O)CC1C c1(C(N(CCCN(C)Cc2c(OC)ncc(Br)c2)C)=O)ccnc2ccccc12 c1(OC)ccc(F)c(C(=O)NCCC2CCCCN2C(=O)CN(C)C)c1OC C(C(C)(C)CCNC(=O)Cc1ccco1)NC(C(C)OCCC#C)=O Cc1c(CNC(=O)CC23CCC2CN(C(c2cc(Cl)no2)=O)C3)cccc1F Cc1ccc(C(CO)NC(=O)NC(C2CCC3(CCC3)O2)C2CC2)c(F)c1 c1(C(=O)NCC(CNC(=O)C(O)C(C)C)OC)cncc(F)c1C(F)(F)F c1(NC2CN(C(c3cccc(C)c3)=O)CC2C#N)ncnc2ccccc12 N1(C(CC(COC)C)=O)CCC(N(C(=O)CCc2cccc(O)n2)C)C2(CC2)C1 c1(C(N2CC(CCNC(C(CC)=CC)=O)OC(C)C2)=O)cc(CC)c(=O)n(C)c1 N1(C(C=C(C)C(C)C)=O)CC(O)(CCNC(C2(Cc3cnn[nH]3)CCC2)=O)C1 C1(C(=O)NCC(C)CNC(c2ccnc(C(F)(F)F)c2)=O)CCc2nncn2C1 CCCCC(O)C(=O)NCC(C)(Cn1cccn1)NC(=O)CCC(=O)N(C)CC CCC(C)(CCO)NC(C1CCC1NC(C1(CN(C)C)CC1)=O)=O n1(CC(=C)C)nc(C(F)F)nc1-c1ccn(Cc2ccc(OC)cc2)c1C c1(CC(C)C)n[nH]c(=NC(CNC(c2ccc(F)nc2)=O)C(C)C)s1 N#CC1CN(Cc2ccc(SC(=O)O)cc2)CCN1C(c1cc([N+](=O)[O-])cs1)=O c1(CCC)c(NCC2CCCC3CC23)nnn1CC c1(C(N2CCC(CC(=O)NC3CCC(C#N)CC3)C2)=O)c(O)cccc1[N+](=O)[O-] C1(NC(C(CC2CCC2)NC(C2CCN(C)C2=O)=O)=O)CCn2cnnc2C1 C12(C(=O)NCCC3(C)CCN3)CCOCC1C2(F)F C1(C(=O)NCCN2CCN(C(C(C(=C)C)(C)C)=O)CC2)C2CCCCCCC12 c1(C(=O)NC2CN(C(Cc3ccn(CC)n3)=O)CC2C)c(C)cc[nH]c1=N C1(CNCCOCCN(C(CCN(C)NCC)=O)C)(OC)CCCCC1 Cc1cncc(C(=O)NC(CNC(=O)Cc2cc(C)on2)C2CCC2)c1 C(=O)(C(C(=O)N1CCC(CN(C(=O)C(F)Cc2ccccc2)C)CC1)OC)OC C1(C(N(CC(=O)NCCCN(C)C)CC)=O)CCC(=O)C1 n1(CC)nc(C(=O)NCC(C)(F)CNC(=O)C(C(C)C)n2cnnn2)c(C)n1 N1(C(C(C(=O)NCCCOC)N)=O)Cc2ccccc2C(C)(C)C1 C1(C(=O)NC2C(NC(c3c(C)nsc3)=O)CCC2)C2CCCCC12 C(C(C(=O)NC1CC(C(C)C)C1)NC(c1coc(C(N)=O)c1)=O)OCC CCC(CN=c1cc(NC(c2ccoc2)C)nc[nH]1)N1CCCC1 Cc1ccc(NC(N2CC(c3c(Cl)cccc3Cl)C2)=O)c(F)c1C N#CC1(NCC(O)CN2CCOCC2)CCOC1 CC1CN(C(C23C(=O)C4CC2C3C4)=O)CCC1CNC(=O)CC1NC(=O)NC1=O C12CC(C)CN1C2=O.C1(CC)CCC(NC(=O)CC2CCSC2)CC1 C(=O)(C(C)C(C)(F)F)NC(C)CN(C(=O)Cc1ccnc(C(F)(F)F)c1)C O=C(C1Cc2ccccc21)NC1CC2(C1)CC(NC(C13CCC(C1)C3)=O)C2 CC1OCCC1C(=O)NCC(C)C(=O)NCCOCC(C)(C)O c12ccc3c(cnn3CNC1=O)c2.c1(C(C)C)cc(C(C)C)n(C)n1 c1(COC)nc(N2CCCC(CNC(=O)CC3CC(F)C3)CC2)cc(C)n1 O=S(=O)(c1c[nH]ccc1=NCc1c(F)cccc1Cl)N1CCC(C23CC(C2)C3)CC1 CN1CC(C(=O)NCC2CCN(C(C3CCNC3=O)=O)C2)C(C(F)(F)F)C1 c1(C(N2CCN(CC(O)C3CC3)CC2)C(=O)NCCC#N)c[nH]c2ncccc12 Cc1cc(C(=O)NC2CCC(NC(=O)CC3CC=CCN3C)C2)c(C)n1C(C)C Cc1cc(C(=O)NC2CCC(C)N(C(c3oc(Br)nc3C)=O)C2)cc(O)c1 c1(C(C)C)ccc(C(=O)N(CCCN(C)C(C2(c3ccccc3)CC2C)=O)C)s1 C(=O)(C(N)CCOC1CCCC1)NCCC(=O)OC(C)(C)C C1(N(C(Cn2c(C)nnn2)=O)C)CN(C(C2CC2Br)=O)CC1(C)C Cc1ccc(C(=O)Nc2ccc(NC(c3cccc(=O)n3C)=O)cc2F)c(C)c1 N1(C(C2CCN(C(C)=O)CC2)=O)CCN(C(c2cscc2Br)=O)C(CC(F)F)C1 C1(C)(NC(C2CCN(C(CCCCCOC)=O)C2)=O)CN2CCC1CC2 C1(NC(c2cnc(C)o2)=O)CC(C(=O)NCCn2ccc(=O)cc2)C1(C)C CC1(C)Cc2cc(NC(c3ccc(OCC4CCCO4)nc3)=O)ccc2O1 c1(C(N2C(C)CCN(C(c3cc(C)c(C)s3)=O)CC2)=O)nn2c(c1C)OCCC2 n1(CC(=O)NC(c2ccc(C)c(F)c2)CNC(C)=O)cc(Br)ccc1=O c1(C(N2CCN(C(C(CCC#C)O)=O)CC2C2CC2)=O)occ2c1CCCC2 C=C(C)CCN=c1cc[nH]cc1S(=O)(=O)N1CC(C)SC(C)C1 c1(C(=O)NCC(CNC(c2cc(Cl)c[nH]2)=O)OC)c(F)cncc1Cl c1(C(=O)NC(c2ccccc2)C(C)C)cccnc1OC(=O)C1CC1 N(C1CCc2ccc(Cl)nc21)C(CS(Cc1scc(C)n1)(=O)=O)=O Cc1nnc(CNC(=O)CN(C2CC(C#N)C2)C(=O)C(F)C2CCCC2)o1 c1(C2C(C(=O)NC3C(CC)CCC3)C2)ccc(F)cc1F CC1=CCC(C(N2CC3CC2(CNC(=O)CCC(C)C)C3)=O)CC1 c1(C(=O)N)cccc2nonc12.N1(C(C2C(=C)C2C(=O)OC)=O)CCN(C)C(=O)C1 CC1CN(C(=O)CC2CC2(C)C)CCCN1C(=O)Cn1cc(S(C)(=O)=O)cn1 c1(C(=O)NCc2nnc(COC)o2)cccc(S(=O)(=O)N2CCCC2C(=O)O)c1 C1(CNC(Cc2cc(C)no2)=O)CCCCN1C(c1ccnnc1)=O CCCC(C)CC(=O)N1CCCCC1CN(C(=O)C(=O)C(C)(C)C)C CCC(C)(O)C(=O)N1CC(N2CCN(C(=O)C(F)(F)C3(OC)CCCC3)CC2)C1 CCS(=O)(=O)c1ccccc1CC(=O)NC1CC2CCC1N2C(c1ccoc1)=O N1(C(CC2C(C)CCC2)=O)CCC2CN(C(c3csnc3Cl)=O)C2C1 C1(C(=O)NCC(C)NC(=O)CCCCN(C)C)CC(O)CN1C(N)=O c1(C(N2CCC3(C(=O)Nc4cc(C)on4)C(C2)C3)=O)cc(C#N)ccc1Cl C(CC(C(=O)NCCc1ncn(C)n1)NC(=O)C=C(C1CC1)C1CC1)OC CCCC(C)CC(=O)NCC(C)CNC(=O)C(F)CC1CCCC1 n1(CC)cc(Cl)c(C(=O)NC(CO)C(C)NC(=O)CCCOC(C)=O)n1 N1(C(c2cnn(CCCl)c2)C(=O)NCCOCC)CC(C)CCC1CCO C1(OC)CN(C(=O)C(=O)Nc2ccccc2CC2CCOC2)CC2CC12 N12CCC(CC1)n1ccc(n1)NC2=O.Cc1nc(SCC2CCCC2)n[nH]1 c1(C(=O)NC(C2(O)CN(C(CCc3c(C)cccn3)=O)C2)C)cc(Cl)cnc1C C(=O)(C(C)CC(F)(F)F)N1CCN(CC2CN(C(C=C(C)C(F)F)=O)C2)CC1 C1(C(=O)NC23COC(CNC(C4CC=CC4)=O)(C2)C3)(OC)CS(=O)(=O)C1 C1(CC(=O)NC2(NC(C3CCC(NC(N)=O)CC3)=O)CC2)SC2=NCCN2C1=O N1(C(CC)=O)CCC2(CC1)CC2NC(c1ccnc(C2CCCC2)n1)=O C12(CCCCO1)C(=O)OC2.C(=O)(C(C)OC(C)(C)C)N(CCNOC)C.C1CC1 c1(CC)ccccc1C(N1CCC(OCC(=O)NOC2CC2)C1)=O C(=O)(C(Cc1cccnn1)NC(=O)NC(C)COC(C)(C)C)OCC N1(C(C=CC)=O)CCN(C(=O)C(C)N(C)C)CC1CS(C)(=O)=O O=C(C1=NOCC1)NCc1cn(-c2ccc(Cl)nc2)nn1 c1(OC)cc(C(N2CCCC(C(C)(C)C(=O)NCC(O)C(C)(C)C)C2)=O)ncn1 N1(C(C(C)OC2CCOC2)=O)CC=C(CC(=O)N2CC3CC(C2)C3(C)C)CC1 c1(C(=O)NCC2(F)CC(CNC(CN(CC(C)(C)C)CC)=O)C2)nnc(S)n1C CN1CCC2CCC(C1)N2C(c1coc(CNC(=O)CNC(=O)CN(C)C)n1)=O c1(C(=O)NC2CCCN(C(C(C)(O)c3ccccc3)=O)C2)c(F)cc(N)cc1F C1(NC(CC(CC)CC)=O)CCN(C(c2cnc(C)c(N)c2)=O)CCC1CO c1(S)ccc(F)cc1.Cc1ncoc1Cn1nnnc1N1CCCC1.N12CCCC1C2 N1(C(CC=C)=O)CC2C(NC(C3(C#N)CCCO3)=O)CS(=O)(=O)C2C1 N1(C(CC2CC(C(C)C)OCC2)=O)CCNC(=O)CCCC1 N1(C(CC)=O)CCCC(N(C2CCCC2)C(=O)Cn2nnnn2)C(F)C1 c1(C(N2CCN(C(=O)C=CCl)CC2)C(=O)NCCOCC)ccnc(Cl)c1F C#CCCCCCCC(=O)N1CCCCC1CNC(C1CCC2CC12)=O C(C)(C)(CCCC(=O)NCC1(O)CC=CC1)NC(C(C)C1CCCO1)=O C1(CNC(C(CC)n2cncn2)=O)CN(C(=O)CC23COCC(C2)C3)CC1N(C)C Cc1cc(C(=O)N(C)CCOCCNC(=O)C(O)C(F)(F)F)c(N)c([N+](=O)[O-])c1 CSC=CC(=O)NCCCN(C(C1COCC1c1ccccc1)=O)C1CC1 Clc1ccc2c(c1)C(NCc1cn(C3CCCC3)nn1)CCCO2 CN1CCC=C(CNC(=O)CC2CC(NC(=O)Cc3ccc(O)nc3)C2(C)C)C1 N1(CC)CCN(C(=O)C(Cn2cncn2)NC(=O)CN2CC(=O)NC2=O)CC1 Cc1ccc2c(C)c(C(=O)NC3Cc4cccnc4C3)[nH]c2c1 CCCCCC(C)(C)C(=O)NCc1cc(C)c(C(=O)NCCn2cnnc2C)o1 C1(C(=O)NCC2CC3CCC3C2)(CNC(=O)Cc2cc[nH]n2)CC12CCC2 C(=O)(CCC(C)(C)C#N)NC(C(C(=O)NC(CC#C)CC#C)(C)C)C N1(C(c2cc(C(N)=O)[nH]c2)=O)CCC2CC12C(=O)NCc1ccncc1Cl Cc1ncncc1C(=O)N(CCCN(C(=O)C(CO)c1ccccc1)C)C c1(C(C2CC=CCC2)(CC)NC2(CC=C)COC2)nnnn1-c1ccccc1 c1(C(=O)NC(CC(C)Nc2nccc(SC)n2)C)ccc2cnsc2c1 CCC(CC(=O)NCCCNC(=O)C(N1CCCCC1=O)C)CC(F)(F)F N1(C(C2(CCF)CN(C(=O)COC)C2)=O)CCN(C2CCC2)CC1 CC(C)CC(C)(C)C(=O)N(CC(=O)NCCC1CCN(C)C1=O)C N1(C(C=CCC)=O)CCCN(C(=O)CC2CC2C2CC2)CC1C Clc1ccc2c(c1)CCC2NCc1cnc2cc(Cl)ccn12 CCCC(C(=O)N1CCC(C)(NC(=O)CC2CC(N(C)C)C2)CC1)C(C)C C12CCC(CC1)C(=O)N2.C(C)(C(=O)NCC(=O)NC1CCC1)NC(C)=O N1(C(c2cc(OCC(F)F)no2)=O)CCC(CNC(C2(F)CC=CC2)=O)C12CC2 C1(CCOC)(NC(c2cn(CC)nc2)=O)CCN(C(=O)Cc2cnns2)C1 CCCCC(CNC(c1ccn(-c2ccncc2)n1)=O)NC(=O)C(C(C)C)SC c1(NC(C2N(C(c3ccn(C)c3)=O)CC=C2)=O)cc(F)c(Cl)nc1Cl c1(C(N(CCCNC(CCc2ncc(C)[nH]2)=O)C)=O)ccccc1OCC(C)C CC1CC(CNC(=O)C#CC2CCC2)CCN1C(c1cc(C(C)(C)C)nn1C)=O CCC(C)C(O)C(C)C(=O)N1CC(C)(C(=O)NCC2(C3CC3)CC2)CC1(C)C CC(C)S(=O)(=O)C(C)C(=O)NCC(C)(C1CC1)NC(=O)CCc1cncs1 c1(C(N2CC(C)CC(NC(CCOCC)=O)C2)=O)cc2c(s1)CCC2=O C1(C(N(CC(=O)O)Cc2cn(CC(C)C)nn2)=O)CCc2cnn(C)c2C1 c1(CC(C(C)C)OC)nc(-c2cccc(C(F)F)c2)nn1CC(N)=O c1(C(=O)OC)cc(N2CCCC2CCCNC(C2CC23CCCC3)=O)ncn1 c1(C(=O)NCC(CC)NC(C2CC2C)=O)nn(C)nc1Br Cc1cc(C(=O)N(C)CC2CCCN2C(=O)Cc2cccc(Br)c2)c(C)cn1 Cc1cc(=NCc2cc(Cl)ccc2F)[nH]cc1S(=O)(=O)N(CC(Cl)Cl)C C(=O)(CCCC#CC)NC(CC=C)C(=O)NC(C12CCC(CC1)C2)CC1CC1 N1(C(Cn2cc(COCC(OCC)OCC)nn2)=O)CCCN2CCCC2C1 CC(C)CC(C)CC(=O)N1CCC(C)(C)C(C(=O)NCc2cc(F)cc(F)c2)C1 c1(C(N2CC(NC(=O)COCC3CCCOC3)C(O)C2)=O)cc2c(s1)CCSC2 N1(C(=O)COC2CCCNCC2)CCC12CCCOC2 c1(C(=O)NC2(COC)CCN(C(=O)C(C)OCCC(C)C)C2)cnc(O)cc1C C1(C(=O)NC(C)C(C)NC(c2cccc(CC3CCCO3)c2)=O)C2CC3C(C2)C13 C1(CNC(c2sc(CCC)c(CC)c2)=O)CCN(C(=O)C(C#N)C2CC2)C12CC2 Cc1cc(C(N2CC(NC(=O)CC(C)CN(C)C)CCC2C)=O)c2nccn2c1 C1(NC(C2ON=C(CC)C2)=O)CC(NC(c2[nH]cnc2C)=O)C12CCC2 C12(C(N3CC(C(=O)NCCC4CCCN(C)C4)(SC)C3)=O)C(=O)C3CC1C2C3 CCC(CC)(CCNC(c1cccc(CO)n1)=O)NC(C1CCC(C)(CC)O1)=O Cc1ccc(Br)c(S(=O)(=O)C(=O)NCCNC(c2c(F)cccc2F)CO)c1 N1(C(C(C2CC2)NC(CCOCCCOC)=O)=O)CC2CCC(C1)C2C#N CC1CC(NC(c2cccc(Cl)c2)=O)CN(C(c2ccc(OCF)cc2)=O)C1 C=CCC(CC(=O)Nc1cc(CC)ccc1C)NC(=O)C(COC)OC C(=O)(CN=c1ccc(Cl)n[nH]1)NC(C)CCCCNC(C12CC(C1)C(C)(C)O2)=O c1(C(=O)NC(CNC(C2C(=C)C2)=O)C2CC2)cc(C(F)(F)F)[nH]c1C c1(CNC(C(C#C)(C)C)=O)ccc2c(c1)CCCC2NC(c1n[nH]cc1F)=O CCC(C)CC(=O)C(=O)N1CCC(CNC(C2CCCS(=O)(=O)C2)=O)C(O)C1 c1(C(=O)NCCOCCN(C)C(c2ccncc2)=O)cc(C(F)(F)F)nn1C c1(C(=O)NCC2CCCC(NC(c3ccc(SC)o3)=O)C2)c(Cl)cncc1Cl CC(O)CCCCCC(=O)NCC1CC2(CO1)CN(C(=O)COC(F)F)C2 C12(C(=O)NCCOC(C)=O)CC(CN(C(=O)CC3CCCCN3C)C1)C2 C1(C(=O)NCCCCC=C)(NC(=O)CSC)CCC(C)(C)C1 c1(C(=O)NCC2CC(NC(C(C(C)O)(F)F)=O)C2)cc2cc([N+](=O)[O-])ccc2o1 C(=O)(C(C)(CC#C)NC(=O)CC1CCCC(C)O1)NCCCCCC#C O=C(CCC(CF)CF)N1CCC(OCC(=O)NCC2CC23CCOC3)C1 C1(CC)CC(C(=O)NCc2cc(C3CCN(CCC(F)(F)F)CC3)no2)CCO1 Fc1ccc(C2(NCC3CC3c3ccc(Cl)cc3)CC2)cc1 CC12CN(C(c3ccc4oc(O)nc4n3)=O)CC1(C)CN(C(C1CC1(C)Br)=O)C2 CS(=O)(=O)c1ccsc1C(=O)OCC1C[Si]2(CCCC2)CN1 C(=O)(CC(C)CC(=O)N1CCC(C(N2CCc3n[nH]cc3C2)=O)O1)OC c1(C(=O)NCC(C)(O)CNC(C2CC(F)C2)=O)ccc2c(c1)NC(=O)CCS2 O=C1COc2ccc(-c3cscc3C(=O)Nc3ccc(Cl)cc3Br)cc2N1 C(=O)(CCCC(=O)NC(C)(CSC)C(=O)NC(c1ncc[nH]1)CO)OC N1(C(CCSCCCC)=O)CCN(C(c2nnn3c2CSCC3)=O)C(C)CC1C c1(CN(CC)CC)ccc(C(=O)NCC(=O)NCc2cc(C(N)=O)no2)s1 c1(C(N)=O)ccc(C(=O)NCC2(CN=c3[nH]nco3)CCC2)cc1 c1(CNC(C2N(CC#C)CCC2)=O)ccccc1CNC(=O)CCCc1ccsc1 C1(C#N)(SCC2(C(=O)NCC(C3CCCCO3)C)CCCCC2)CCOCC1 Cc1cc(Br)ccc1-n1cc(C2CC(NC(=O)CC34CCC(C)(C3)OC4)C2)nn1 Cc1cccc(CCNC(c2ccn(CCNC(=O)Cn3nccc3C)c2)=O)n1 c1(OC)cccc(C(=O)NCC2CC2CNC(=O)CCc2cnco2)c1O C1(O)(CCNC(=O)CC2CCOC2)CCCN(C(C2CCC3(CC2)CC3)=O)C1 CC1CC2(CC(C(=O)NC3(C(=O)NCCS(N)(=O)=O)CCOCC3)C2)C1 CC1CC=C(C(=O)NC2CC=C(C(=O)N(CC(C)C(F)(F)F)C)C2)CC1 c1(OC)cccc(Cl)c1CC(=O)NC1CCC1NC(C1(C)CCC(OC)CC1)=O c1(CCC)ccc(C(=O)NCC2CC(CNC(=O)C=CCO)CO2)[nH]1 C(=O)(C#CC1CCOCC1)N1CC2=C(CN(C(C3C(C)NC(=O)CC3)=O)C2)C1 C1(CNC(c2ncc(NCC)nc2)=O)C(C)CCCN1C(C1(CF)CCC1)=O C(=O)(CC(C)C(=O)OCCNC(=O)C(C)(C)C1CCC1)OC(C)(C)C c1(C(=O)NC2(C)CN(C(c3cc(C(F)(F)F)ns3)=O)C2)cnc2ccccn12 C1(NC(C(CC)C)=O)CCN(C(c2nc(-c3ccccc3C)oc2C)=O)C1C N1(C(C2(C)CC2Br)=O)CCC2(NC(c3cncc(-n4cccn4)n3)=O)CCCC12 C12(NC(C=Cc3c(C)ccs3)=O)CCN(C(=O)C(c3ccccc3)F)CC1C2 c1(CC)ncc(C(=O)NC2(COC)CN(C(=O)CCOC3CCOC3)C2)c(C)n1 Nc1ccc(F)c(F)c1C(N1CCN(C(C2CCCS2)=O)C(C2CC2)C1)=O N1(C(c2c(C)n(C)cn2)=O)CCC2(CC2)CC1C(=O)N(CCC(C)(C)C)C N1(C(C2(C)COC2)=O)CCC2(CCC(C(N3CCOCC34CCC4)=O)CC2)CC1 N1(C(C2CCCCO2)=O)CCN(C(=O)CCn2cccn2)C(CC2CC2)C1 CN1CCC(NC(c2csc(S)n2)=O)C12CCCN(C(C1CS(=O)(=O)N1)=O)C2 C(CC(C(C)C)NC(C1CSCCS1)=O)NC(C(CC)N(CC)CC)=O CON(CCC(=O)N1CCSC2CCC12)C(=O)c1ccnn1C N1(C(CC2CCC(=O)O2)=O)CC2CCC1C(CNC(c1snnc1C1CC1)=O)C2 C12(NC(CC#N)=O)COCCC1CN(C(c1cc(C(F)(F)F)ncn1)=O)C2 C1(C(=O)OC)CN(c2nnc(-c3ccccc3F)n2Cc2cccs2)CC1(F)F C1(NC(C2(C(C)NC(c3cc4ccccn4n3)=O)CC2)=O)CN(C)CCN(C)C1 C(CC(C(=O)NCCCc1c[nH]nc1C)NC(=O)C=Cc1ccsc1)OC N1(C(C2(C(F)F)CC(=C)C2)=O)CC(NC(c2cc(F)ccc2O)=O)CC(O)C1 c1(C(N2CCC(O)(CNC(CN(C)C)=O)C2)=O)n[nH]c2c1COC2 C1(N(C(CCC2(NC(CCC=C=C)=O)CCC2)=O)C)CCC2(CC1)CC2 Cc1ncnc(C(=O)NCC(C2CCN(C(C3C(C)(C)C3(F)F)=O)CC2)O)c1C CC(C)(CC(=O)N1CCCC(C)(NC(=O)COCCO)C1)CC(F)F N1(C(CC(CNC(c2ncn(CC)c2)=O)(C)C)=O)CCC2CCN(C)CC12 CCC(C)CC(C(=O)NC1COCC1OC)NC(=O)C1=C(Cl)CCC1 N1(C(c2ccc(C(F)(F)F)cc2)=O)CCC12CN(Cc1c(Cl)cccc1I)C2 CCC(CC(=O)N1CC(NC(c2csc(C(C)=O)c2)=O)C2(CC2)C1)C(C)(C)C C1(NC(CSCC=C)=O)CCS(=O)(=O)C12CN(C(C1COC(=O)N1)=O)C2 Cc1ncc2ccccc2c1C(=O)NCC1CC(C)N(C(=O)CCC(C)(C)C)C1 c1(C(=O)NC2C(NC(CC(C)F)=O)CCC2)nc2ccccc2[nH]1 N1(C(CCN(C(CC)CC)C)=O)CC(NC(=O)CCNC(C)=O)C(N=[N+]=[N-])C1 c1(CNC(Cc2scc(CC)n2)=O)nc(C(=O)NCc2cncc(Cl)c2)c(C)o1 C(CC(C)C)(C(=O)NCC(F)CNC(c1cccc(F)c1Cl)=O)NC(C)=O C(C)(C)(C(C)NC(c1cn(C2CCCC2)nn1)=O)NC(C(C)O)=O c1(N)ccc(O)cc1.C1(C(C)C)CC(C(=O)NC2CC(NC(C3CC3C)=O)C2)C1 c1(C(C)=O)ccc(C(=O)NC(C)CNC(=O)C(C2CCC(=O)N2)C)o1 C1(NC2(c3n(CC(=C)C)nnn3)COC2)CC(C(=O)OC)C12CCC2 C1(Cc2cn(CCC=C)nn2)CN(C(=O)C(C)CC2CCC2)CCO1 c1(OC)ccc(OC)c(C(N2CCC(CCNC(=O)CN3CC=CC3)C2)=O)c1N c1(C(=O)NC2CCCC(CC(=O)NCc3ccnc(O)c3)C2)c(O)cccc1F C(CN=c1[nH]cnc2c(Br)cccc12)N1CCN(C(c2c(OC)scc2)=O)CC1 c1(N2C(C)C(NC(c3cc(Cl)c[nH]3)=O)CCC2)nc2c(cc1C#N)C(=O)CCC2 Cc1cc(C(N2CCC2C(N2CCC(Oc3ccccc3)CC2)=O)=O)cc(Br)c1 N1(C(c2cc(OCC)no2)=O)CCC2(CCN(Cc3cn4ccccc4n3)C2)C1 N(C1CCCn2ccnc21)C(c1c(CNC(C(CO)OC)=O)nccc1)=O CC1CC(C(=O)O)CN(Cc2ccc(OC(CO)C3(C)CC3)cc2)C1 c1(C(N2CC(NC(C3CC(O)C3)=O)C(CC3CC3)C2)=O)c(F)cc(F)cc1Cl c1(CNC(c2c(OC)csc2)=O)ccnc(Br)c1 C1(CNC(c2ccc[nH]2)=O)C2CN(C(c3ccc(Br)o3)=O)CC12 C(=O)(CC(C)(C)CC(=O)OC)N(C(CNC(c1ccc(C#C)cc1F)=O)C)C CC(F)(F)CCC(=O)NC1CS(=O)(=O)CC1NC(=O)COC1CCCOC1 c1(OCC)ncc(C(=O)NCC2CC(NC(C3CC3[N+](=O)[O-])=O)C2)cn1 Cc1cc(C(=O)NCC(C)NC(C2CC2c2ccccc2)=O)nnc1C C(CC(C)(C)CC(=O)N1CCC(C)(NC(=O)C(C)(C)C(F)(F)F)C1)OC CC1(C(=O)NC2CCCC(CNC(C3CCC4CC4CC3)=O)C2)CC2(CCC2)C1 CC(C)C(C(=O)NCC(C)(O)CNC(c1cncc(Cl)c1)=O)NC(=O)C(F)(F)F CCCCC(O)C(=O)NC1CCC(F)(CNC(C2(C)SCCCS2)=O)C1 C1(NC(=O)CCC2CC(F)(F)C2)CC2CC(C1)N(C(C13CCCC(C1)OC3)=O)C2 CN1CCN(c2cccc(C(=O)OCC3(CNC4CC4)CC3)n2)CC1 Cc1c(C(N2CCCC(C)(CNC(=O)C(C)OC3CCCC3)C2)=O)nn(C)c1N N1(C(c2ccc(C)n2C)=O)CCCC1C1CCCN1C(=O)CNC(N)=O c1(C(=O)NCC(C)N(C)C(c2cnc(C(F)F)s2)=O)coc(Cl)c1 Cc1noc(Cl)c1CCC(=O)NC(C)CC1CN(C(c2cnn(C(C)C)c2)=O)C1 C(C1=CCCN(C(=O)CC2CCCC3CC23)C1)NC(C1CC(OC)C1)=O.C1(C)CC1 c1(NCC(C)C)ccc(-c2nc(C(=O)NC(c3ccccc3)C(=O)O)cs2)cc1 Cn1cc(Cl)cc1C(=O)NCCn1ccc(C(N2CCN(CCF)CC2)=O)c1 c1(-c2cccc(C#C)c2)ccc2[nH]cc(C(=O)Nc3ccc(OC)c(F)c3)c2c1 Cc1cc(C(=O)N(C)CCN(C(=O)CCN2CCC(F)C2)C)cn(C)c1=O c1(C(=O)NCCC(C(=O)N(CCCCC)CCO)O)ccc2cc[nH]c2c1 CC1CN2CCN1CC2C(=O)NCC(C)(O)CNC(c1cnn(C)n1)=O C1(NC(CCc2ccc(C)o2)=O)CCCC(N(C)C(c2cnn(CCF)c2)=O)C1 c1(C(=O)NC2CC(F)CN(C(c3cncn3C3CC3)=O)C2)cc2cccnn2c1 CCC1=C(C(=O)NC(CC(=O)NCC(c2ccsc2)O)C(F)(F)F)CCCO1 N1(C(C(C)C(C)(C)C)=O)CC(C)(C)OCC1CNC(=O)CCC1CCCCCC1 C1(C(=O)NC2CN(C(=O)C(C)(C)COC(C)C)CC2C)(OC)CCC(F)(F)CC1 Cc1cnn(C)c1NCC1CCCC(C(=O)O)C1.c12nc(no1)C(=O)N(CC(C)C)C2 C1(CCNC(C(C2CCOC2)OCC)=O)CCN(C(=O)Cc2ncc(C)s2)CC1 N1(C(c2cc(CC)no2)=O)CC(CNC(=O)C=NOC)C(F)(F)C1 CC1CC(CNC(=O)CC2CSCCO2)CN1C(c1nn(C)cc1Cl)=O c1(C(=O)NC2(CCNC(C3(C)CC3F)=O)CC2)nc2ccccn2c1F Cc1nc(O)[nH]c1C(=O)NCCCCNC(c1ccc(C2CC2)cn1)=O c1(C(N2CC3C(NC)C3C2)=O)cccnc1OC(C)C(F)(F)F C1(C(=O)NCCOCCCNC(C2CC(C)(C(C)(C)C)C2)=O)CC2CC(=O)C1O2 CC1CCN(C(=O)Cc2cccnc2Cl)CCN1C(=O)C(O)Cn1cncn1 c1(C(C)C(=O)N(C2CC2)Cc2nc(C(F)(F)F)n[nH]2)cccc(C#N)c1 CC1CN(Cc2cc(-c3ccc(C=O)s3)ccc2O)CCN1C(c1cccs1)=O C=CC1OCCC1C(N1CCC1CC(=O)NC(CC)CCOC)=O C(C(C)(C)CC(=O)NC1CCC(C)(CNC(=O)CC2CCCCCC2)C1)OC C12(NC(Cc3c(C(C)C)cccc3)=O)CCN(C(c3cccc(O)n3)=O)CC1C2 c1(C(=O)NC2CCCN(C(C3CC(=O)NC3)=O)C2)ccnc(O)c1F c1(C(N2C(CNC(C(C)OCCN(C)C)=O)CCC2)=O)cc(N)cc(O)n1 c1(SC)cc(C(=O)C)ccc1O.C1(N)CCC(C)N(C(=O)CN(C)C2CC2)C1 CCC(CC(=O)NC(CNC(C1NC(=O)CC1C)=O)CC)C(C)C C1(C2CCN(C(c3cn(C(F)(F)CO)nn3)=O)CC2)(NC(CC(CC)O)=O)CC1 C1(C#N)(C(=O)NCC(CNC(c2n(CC(C)C)ncc2)=O)O)CC2(CC2)C1 C1(NC(C(C)NC(CC)(C)C)=O)CCN(C(c2cncc(Cl)c2)=O)C1C(C)C c1(COCC(N2C3CC(NC(CCCCC)=O)C(C3)C2)=O)ccc2c(c1)OCO2 CC(C)C(O)CC(=O)NCC(CNC(=O)CSCC(N)=O)CO c1(C(F)F)ccc(F)cc1-c1nc(CCn2ccnc2)nn1CC(F)(F)F C(=O)(C1=C(C)S(=O)(=O)CC1)NCC1(C)CCC(NC(C(C=C=C)C)=O)CC1 N1(C(c2c(C)ccc(OC)n2)=O)CC2CCN(C(c3nc(C)nn3C)=O)CC2C1 c1(C(N2CCN(C(=O)COCC3CC3)CC2CC2CC2)=O)ccc2occc2c1 C1(CC=C)(NC(C2CCCCN2CC)=O)CCN(C(=O)C(Br)=C(C)C)C1 C1(C)(CC)CC(NC(c2ccc(C3CCCCC3)cc2)=O)CN1C(=O)C1CC1 c1(CNCC(C(C)C)O)ccncc1OCc1ccccc1 Cc1cc(Br)cc(C(N2CC(N(C)C(c3ncoc3C3CC3)=O)C2)=O)c1C c1(C(N2CCC(CC(N3CCCC(C(=O)OC)C3)=O)CC2)=O)c(I)ccnc1Cl CC1(C)CC(CO)CN1C(=O)C(C1(O)CCN(C(=O)OC(C)(C)C)CC1)F C(CCC(F)(F)F)NC(C1(NC(C2CCCS2)=O)CC(CO)C1)=O Cc1ccc(CC(=O)NC(C2CCN(C(=O)C(c3ccccc3)=O)C2)C)c(Cl)c1 Cc1ccc(F)c(O)c1C(=O)NCc1cn(-c2nc3ccccc3s2)nn1 CC(C)C(C(=O)NC1CC2CC(NC(=O)COCCF)CC2C1)C(C)C C1(C(N)=O)CC12CCN(C(=O)C(NC1=NCCC1)=O)CC2.c12cccc(c1)CN2 CC1CN(C(C)C(=O)NCC(O)CNC(=O)CCc2cscn2)C1 C1(C(=O)Nc2c(-c3ncn(C)n3)cccc2)CCOCC12CCC2 n1(CCC)ccc(=NC(=O)CCC2CCC(=O)NC2)[nH]1 C1(C(=O)NCCCC(C)NC(=O)CCOc2ccccc2)CCC(N(C)C)CC1 CCC(CC(=O)NCCc1ccsc1)N(C(=O)CC1CCCC2CC12)C N1(C(CNC(C)=O)=O)CC(C)OC2(CCN(CC(=O)Nc3ccccc3)C2)C1 C=C(F)C1(CC(=O)NCc2ccc(C(=O)NC(CO)C(=O)OCC)s2)CCC1 C1(NC(C2N(C(CCCCOCC)=O)CC=C2)=O)CCCC(F)(F)C1 N1(C(CC(C)(C)SC)=O)CCOCC(NC(=O)C(O)c2cnc[nH]2)C1 c1(C(=O)NC2CCN(C(CC(CC)OC)=O)C2C)cc2c(Cl)cncc2o1 C1(CC(=O)NCC2(N3CCCC3)CC2)C(NC(=O)CCC2CCCOC2)CC1O c1(NC(Cc2ccc(C)cc2C)C)ncnc2c1CCCC2 CS(=O)(=O)c1sccc1C(=O)NCC1(NC(=O)CC2CCOC2=O)CCC1 Nc1c(Cl)cnc(NCC(F)(F)C23CC(C2)C3)c1Cl N1(Cc2ccc(OCC=C)cc2)CCC(O)C(C(=O)Nc2cnncc2Br)C1 c1(C(N2CCC(NC(c3c(C)nc(CO)s3)=O)C(F)C2)=O)cnc2cc[nH]c2c1 N1(C(CCN(C(=O)CCc2ccccn2)CC)=O)CCCC2NC(=O)CC12 CCCCCCCCCCCC(=O)NCC1CN(c2nnco2)CCN1C c1(C(N2CCC(NC(COC(CC)(C)C)=O)C(CO)C2)=O)c2c(nn1C)CCC2 Cc1ccc(C=CC(=O)NCC(C)(Cn2cccn2)NC(=O)C(C)O)c(C)c1 CC(C)(CS(N)(=O)=O)C(=O)NC1CCCN(C(c2ccc(C(N)=O)s2)=O)CC1 CCCC(CNCc1ccnc(C)c1)C(=O)NC1CCCOC12CC2 c1(CC(N2C(CC(=O)NCC3(C(=O)NC)CCOC3)CC2)=O)ccc(NC)cc1 CC1CN(C(=O)Cn2nnc(C3CC3)n2)CC1Nc1ncccn1 C(=O)(C1=CCCCO1)NCc1occ(C(=O)NC2CC(CC(N)=O)C2)n1 Cc1ncnc(O)c1C(N1CCCN(Cc2ccccc2)CC1)C1COC(C)C1 C(=O)(CCC(N)=O)NCC1(O)CC(NC(C2CCN(C)C2)=O)C1 C1(NC(C(C2CCCO2)NC(=O)Cc2ccc(O)nc2)=O)CC2CC3C(C2)C13 CCCC(C#N)C(=O)NC(C)(CO)C(=O)N(C(C(N)=O)C1CC1)C N1(C(C2(C)N(C(c3ncc(C)c(Br)c3)=O)CC2)=O)Cc2cccc([N+](=O)[O-])c2C1 C1(CNC(=O)CCSCc2ccccc2)COCCN1C(=O)Cc1cscn1 C12(C(N3CC(CC)OCCC3)=O)CCC(CC1)N(C(=O)C(C)(O)C1CCC1)C2 C(CN=c1[nH]c(=NCCCN2CCCOCC2)[nH]c2c1CCC2)(C(C)C)OC Cc1c(CCNC(C2CCN(C(c3ccoc3)=O)C2C)=O)cnn1C N1(C(C2C(C)C2)=O)CCOCC1CNCc1ccc(F)nc1 C#CCC(C)(C)C(=O)N1CC(OCCC(=O)N(C(C)C(=O)OC)CC2CC2)C1 N12CCC3CCCC13NC(=O)C2=O.c1(CC=C)nnc(C(=O)OC)s1 C1(NC(COCCOCC#C)=O)CCCC(NC(c2cccc(F)c2)=O)C1 c1(CC(=O)NC(C2CN(Cc3ccc(OC)cc3)C2)C)ccc(F)cc1F c1(OC(C)C)cncc(C(=O)NC2CCCCC2N(C(=O)C(C)CO)C)c1 c1(OCCC)nn(C)cc1OC.c1(OCCCNC(=O)N)ccc(C(=O)OC)nc1 C=CCCC(F)(F)C(=O)NCC(CC=C)C(=O)NCCc1cocn1 C1(CNC(C(C)NC(=O)NC)=O)CN(C)CCN1C(C1CC1C(C)O)=O N1(C(c2cnc(OC)c(C)n2)=O)CC(NC(c2nccnc2N)=O)C(N=[N+]=[N-])C1 C1(NC(c2nn(C)c(=O)cc2)=O)CN(c2ncc(Br)cn2)CCC12CCC2 C1(NC(c2ccc(C)s2)=O)CCC(C)N(Cc2snnc2C)C1 N1(C(CCOCCCOC)=O)CCC(C)N(C(C2CC(C)(F)C2)=O)CC1 N1(C(c2n[nH]c(C)c2C)=O)CCC2(NC(C3CC3C3CCCC3)=O)CCCC12 C1(NC(c2n(C)nc(C3CC3)c2)=O)CCCN(C(=O)C=CC2CC2)CC1F N1(C(c2ccc(OC)c(F)c2)=O)CC2(CC1CNC(=O)CCC(N)=O)CC2(F)F c1(C(=O)NC2(C)CCN(c3n(C)nnn3)CC2)cccc2ccsc12 c1(C(=O)NC2C(C)CCN(C(=O)CCc3cnc[nH]3)C2)cc2ccnn2cn1 c1(NC(=O)CC2CCCN2C(c2sccc2I)=O)cc(Br)cc(Cl)c1O C#Cc1cnn(C)c1C(=O)NCc1c[nH]nc1C(=O)NCCC1CCOC1 C1(NC(Cc2c(C(C)C)con2)=O)CC(C)N(C(=O)CN2CSCCSC2)C1 CCC(C)C(C)C(=O)NCCN(C)C(C1(c2cccc(Cl)c2F)CC1)=O C1(NC(c2cn(CCC)nc2)=O)CC2CC(NC(=O)Cn3ccnc3C)C2C1 N1(C(=O)CO)CCC(n2cc(COc3cncc(Br)c3)nn2)CC1 CON1CCC(C(=O)NC2CCCCC2N(C(=O)CC2CC(SC)C2)C)CC1 N(C1c2cccc(F)c2OC1C)C(c1cc(-c2ccc(OC)cc2)ncn1)=O N1(C(c2n[nH]c(C)n2)C(=O)Nc2ccc(OC)cc2)CCCN(C(C)CO)CC1 N1(C(c2c(C)occ2)=O)CC(C(=O)NCC(C)(O)C(C)C)CCC1(C)C CS(=O)(=O)C1CCCC1C(=O)NCC1CN(C(=O)CCc2ccc(F)cc2)C1 c1(C(=O)NCC(CC)NC(c2c(C(F)(F)F)n[nH]c2C)=O)cncc(SC)c1 c1(C(N2CCC(n3cc(-c4ccc(Cl)s4)nn3)C2)=O)nccc2cc[nH]c12 C(C1CCCCC1)=CC(=O)NC1(CC=CC(=O)NCC(O)C(F)F)CCC1 Cc1cc(NC(=O)CN2CC(C)C2)ccc1NC(=O)COCCOCCO C1(C(=O)NC2(CC(=O)NC(C(C)C)c3cccs3)CCC2)CCCC2CCCCC12 CCCC(C#N)C(=O)NC1(CNC(c2ccc(-c3sccc3C)s2)=O)CC1 C12(C(N3CCCC(F)(CNC(C(C)(C)C)=O)C3)=O)CCC(C(=O)O)(CC1)CC2 c1(C(=O)NC(C2CN(C(CC)=O)C2)C)cnn(-c2cccc(C(C)C)c2)c1C C(C)(CC(=O)NC1(CCCC(=O)NCCC2CCC3CC23)CCC1)OC c1(SCC(=O)N=c2nc[nH]n2CCO)cccc(S(=O)(=O)C(F)(F)F)c1 c1(C(=O)NCC2C(C)CCN(C(=O)C(C)(C)F)C2)cnn2c(N)ccnc12 c1(CN(C(c2cnn(C)c2C)C(=O)NCC=C)C)ccc(Cl)c(Cl)c1Cl c1(C(=O)NCC2CCN(C(c3ccc(CCC)s3)=O)C2)cccc(O)c1[N+](=O)[O-] C=CCC(C(=O)Nc1ncc(C(=O)OC2CN(CC)C(=O)O2)s1)OC CC(C)C(C(=O)NC1CC(=O)N(C(C)C)C1)NC(c1ccncc1Cl)=O c1(NC(C=CC(C)NC(C2(SC)CC2)=O)=O)cc(C#N)ccc1O c1(C(N2CCC3CN(C(C(C(CC)C)OC)=O)C3C2)=O)cc2ccccc2cn1 c1(C(=O)NCC(CN(C(c2cc(C)no2)=O)C)(C)C)cc(C)n(C2CC2)n1 C1(NCc2scc(C(=O)NC(COC)C)n2)CCCC(C)C1 c1(C(N(C)CC2(O)CCCC(C)(C)C2)=O)n[nH]c2c1CCCCC2 Fc1cccnc1C1CCN(c2cnnc(Br)n2)CC1 N1(C(C(CCC(N)=O)NC(C)=O)=O)CCC2C1CCCN2C(=O)CCC(C)C c1(C(=O)NCCNC(=O)Cc2cnc[nH]2)cc(C(F)(F)F)c[nH]1 N1(CC(=O)NCC2CN(C(C3CCC=CCC3)=O)CCCO2)CCCCCC1=O c1(CCC(=O)NC(C2OCCN(C(CC)=O)C2)C2CC2)ccc(N)c(F)c1 c1(-c2scc(C(=O)OC)c2)ccnc(-c2ccnn2C2COC2)c1 Cc1ccc(C)c(CN2CCC(NC(=O)Cc3ccn(C)n3)C(O)C2)c1O C1(NC(c2c(C)csn2)=O)CCCC(C(=O)NCc2c(C)cnn2C)CC1 N1(C(c2c(C)nsc2N)=O)CCC(C2CC2)(NC(=O)CN2CCCC2C)C1 C(=O)(CCN=C(NC1C(C)C1(F)F)N1CCCC(C)C1)NC(C)=O CC1(C)CN(C(=O)CC23COCC(C2)C3)CC1NC(c1ccc(Cl)c(O)c1)=O N1(C(C2(CC)CCN(C(=O)C(CO)OC)CC2)=O)CC2(CCC2)CC1OC c1(CC(=O)NCC2CN(C(c3ccnc(OC)n3)=O)CC2O)ccnc(Cl)c1F O(S(=O)(=O)c1ccc(Br)cc1Cl)c1cccc(CC)c1 C1(C(N2CCC(CC(C)NC(c3cscc3Cl)=O)CC2)=O)CC(=O)C12CCCC2 Cc1nnc(CCCC(=O)NC2CCN(C(C3CN(C(C)C)CCO3)=O)C2)n1C c1(NC2CC(C)SCC2)cc(Br)ccc1S(=O)(=O)N1CC2CSCC(C2)C1 c1(NCC2N(C(C3CC3C3CCCC3)=O)CCCC2)ncnc2c1CCC2 C=CC(C)(C)CC(=O)N(C1CCN(C(c2cn(C)nc2Cl)=O)CC1)CC c1(C(N2CCC(SC)C2)C(=O)NC2CCOC2)ccc(C)c(OC)c1 c1(C(=O)NC(CCOC)CNC(=O)C(C)n2ccnc2)ccc(C#N)c(F)c1 C1(NC(C(=O)N(C)C)=O)(CO)CCCN(C(=O)COCc2ccccc2Cl)C1 CC(C)C#CC(=O)NCC1CC(F)(CNC(C23CC(C(F)F)(CO2)C3)=O)C1 CC1CC(C)N(C(=O)CNC(=O)CC(F)(F)F)CCN1C(=O)C=Cc1cncs1 C1(C(N(C)CC2OCCN(C(C(COC)(C)C)=O)C2)=O)C(C)OC(C)C1C CC1CCCCC1NC(=NCc1cccc(C2CC2)c1)NCC12CC(C1)C(C)O2 S(=O)(=O)(c1ccccc1)NC(C(=O)NC(C1CCCC1)CC)C c1(N2CCC(NC(c3c(CCC)n[nH]c3)=O)C(F)C2)ncnc2ccc(Cl)cc12 c1(C(N2CC(CC(C)NC(c3nn(C)cc3Br)=O)C2)=O)cc([N+](=O)[O-])c[nH]1 c1(C(N2CC3CN(C(CCS(C)=O)=O)CC3C2)=O)cn2ccc(CO)cc2n1 CC1(C(=O)Nc2cc(CO)ccn2)CCN(C(c2c[nH]ccc2=N)=O)C1 c1(OC)ccc(C=CC(N2CC3CC2CN3C(=O)C=C(C)C(C)C)=O)c(OC)c1 CC(C)(C)CC(O)CC(=O)NCCC(O)C(=O)Nc1ccc(F)c(CO)c1 C1(n2cc(-c3n(C)c(S)nn3)nn2)CC2(CCCCC2)CO1 CC(C)C(C)CNC(C1CCCN1C(=O)C=CC1CCC1)=O C1(C(=O)NCC(CNC(CN(c2ccccc2)C)=O)(C)C)CCC2(CCC2)O1 Cn1nc(C(F)(F)F)cc1NC(c1ccc(-c2cncc(O)c2)cn1)=O C(=O)(C1=COCCO1)NC1(CC=C)CCN(C(c2cc(C(F)F)no2)=O)C1 N1(C(c2ccc(N(C)C)cc2)=O)CC(CNC(=O)Cn2ncnn2)C2(CC2)C1 CC1CCc2ccccc2N1CCC(=O)NC(CNC(=O)Cc1cnc[nH]1)CO C1(c2nnnn2C2CC(F)(F)C2)(CCNCC(F)(F)F)CCC(C)(C#N)C1.CCCC C(CCC)(C(=O)N1CC(CNC(=O)CC2CCN(C(C)C)CC2)(OC)C1)=CCC C#CCC(CC#C)C(=O)NC(CN(C(=O)C=C1CCOCC1)CC)CC Cn1ccc(C(=O)NCCOCCNC(c2csc(CO)n2)=O)c1 C12(CNC(=O)Cc3ccon3)CCCCC1N(c1ccc([N+](=O)[O-])cn1)CC2 CCC(CNC(C1CC1C(F)F)=O)NC(=O)CC1(C)CC1 CC1CCCC(C(N2CC(CO)(NC(=O)CC(C)c3ccccc3)C2)=O)CC1 c1(N(C)CC2CC2)[nH]c(=NCC2CC23CCC3(F)F)ccc1[N+](=O)[O-] C1(NC(c2c(C)sc(C(F)(F)F)n2)=O)C2CCC1N(C(=O)C(CO)N(C)C)C2 c1(OC)cnc(C(=O)NC2CCCCC2N2CCCC2)c(F)c1 CCCC(CC1CCCCC1)C(=O)NC1(CNC(c2cncc(OC)c2)=O)CC1 S(=O)(=O)(c1ccc(C(=O)NCC2CC2NC(=O)CCn2ccc(C)n2)o1)NC CC(CCC(=O)NC12CCN(CC1)C2)NC(C1CC(=C2CC2)C1)=O c1(N(C)Cc2nc(C)c(C)[nH]2)nc(N(CC(C)C(C)(C)C)C)c2ncn(C)c2n1 C(C)(CCN=c1[nH]cc(C#N)cc1C)NC(c1ccc(C)c(F)c1)=O N1(C(c2c(CC)cns2)=O)CCCC(C)(C)C1CNC(c1ccc(O)cn1)=O Cc1cc(C(=O)NCC(O)CN(C)C(C23CSCC2C3)=O)cc(O)n1 N1(C(CC(C)OC)=O)CCC(c2ccccc2)(NC(c2cc(C)cnn2)=O)C1 C1(NC(C(C)NC(COC)=O)=O)CCN(C(c2[nH]c(C)cc2C)=O)CC12CCC2 c1(OC)cnnc(C(N2CCC(NC(=O)CN(C)C3CC3)C2C2CC2)=O)c1 c1(C(N2C(C)CC(NC(c3sccc3CN(C)C)=O)C2)=O)ccn2ccccc12 N1(C(C2CCC(N(C)C)C2)=O)CCCC(C2OCCO2)C1 c1(OC)cc(C)c2cc(C(N3CCCC3c3ccccc3OC)=O)[nH]c2c1 C(=O)(CC(C(F)(F)F)n1cccn1)N1C(CNC(c2cnn(C)n2)=O)CCC1 C1(NC(c2scc(C)c2Cl)=O)CCC2CC1CN2C(c1ccc(C#N)[nH]1)=O c1(C(=O)NCCN(C(=O)CCS(=O)(=O)N(C)C)CC)cn(CC)c2ccccc12 CCC(C)N(OC)C(=O)C(F)C1(O)CN(C(=O)Cc2ccccc2OC)C1 c1(C(N(C)CCN(C)C(C2CCOC2(C)C)=O)=O)ccc2cnn(C)c2c1 C=CCC(CC)C(=O)N1CCCC1C(C)(C)CNC(c1ccccc1)=O C1(c2n(C(C)(C)C)cnc2)CCCN(CCc2ccns2)C1 c1(N(C)Cc2cc3cc(OC)ccc3n2C)c(SC)oc2ccccc2c1=O.CN CCCCC(F)C(=O)NCCC1CSCCN1C(=O)Cn1cnc(=N)[nH]1 c1(-c2[nH]cc(C)n2)ccc(NC(=O)C(N2CC(c3ccc(Cl)cc3)(O)C2)=O)cc1 c1(C(N2C(C)CC(NC(c3c(CC)n[nH]c3)=O)C2)=O)cc(C)cc(Br)c1F c1(C(=O)NC2CC(NC(C3(C(N(C)C)=O)CC3)=O)C2)cc(O)nc2ncn(C)c12 N1(C(C2C(C)CCOC2)=O)CCC(C(=O)NCCC2CCCC3CC23)C(C)(C)C1 C1(C(N(CCO)CC)=O)(OC)CCN(CC(=O)NCc2n[nH]c(=N)s2)CC1 C1(NC(C(CCC2CC2)NC(C=CC(CC)C)=O)=O)CCn2nccc2C1 c1(OC)ccc(O)cc1C(N1CCC(O)(C(=O)NCC2CCS(=O)(=O)C2)C1)=O C1(CN(C(CCSC)=O)C)CCCN1C(=O)C(CO)NC(c1ccccc1)=O N1(C(C(CC)C#N)=O)CC(OC)CC(NC(C2(c3ccn(C)n3)CC2)=O)C1 C1(CNC(c2cc(Cl)cs2)=O)CN(C(=O)CN2CCS(=O)(=O)CC2)CC12CC2 N1(C(C2C(=C)C2C(=O)OC)=O)CCCC(CN(C(=O)Cc2cn(C)nn2)CC)C1 c1(OC2CN(C(c3ncc(CN(C)C)o3)=O)C2)cccc(F)c1 c1(C(C)N(c2cccc(F)c2C(c2ccc(Cl)cc2)=O)C)cc2ccccc2s1 Cc1ccc(C(N2CC=CCC2C(N2CCCC(CC3CC3)C2)=O)=O)cc1F C(=O)(C(O)CC(F)(F)F)NC(CC=C)CNC(=O)C=Cc1ccccc1OCC c1(SCC(N2CC3C(NC(C=NOC)=O)C3C2)=O)nnc2ccccn12 c1(OC)ccc(C(=O)NCCCN(C)C(c2cocc2C)=O)nn1 c1(OC)c(F)ccc(F)c1C(=O)NC1CCN(C(C2CSC2)=O)C(C2CC2)C1 C1(C(=O)NCC(CC(F)(F)F)NC(c2cn(C)nc2)=O)CCC(N=[N+]=[N-])CC1 N1(C(=O)OCC)CSCC1C(=O)NC1CCN(C(c2cc(C3CC3)[nH]n2)=O)C1 C1(CC(=O)N(CCNC(CCCC2C(C)C2)=O)CCOCCO)CCC(=O)NC1=O c1(C(N2CC(NC(CCOC(C)C)=O)C(O)C2)=O)ccc(F)c(O)c1F C1(NC(c2c(C)[nH]nc2Cl)=O)CC2CC1N(C(c1cc(Cl)ccn1)=O)C2 N1(C(COCCC)=O)CC(CNC(=O)C=Cc2ccc(C)cc2)CC1(C)C N1(C(C2C(NC(C3CCCO3)=O)C2)=O)CCOC(C2CC2)C1 Cn1ccc2nc(N3CC(CO)(NC(c4ccncn4)=O)C3)ncc12 CC1COCCC1N(C)C(c1cn(CCNC(=O)CCOCC(F)F)nn1)=O CC(C)CC(C)CC(=O)NCC=CC(N1CCN(C)CC1)=O N1(C(CC(C=C)(C)O)=O)CCC(C(=O)NC(c2[nH]c(C)nc2C)C)C(C)(C)C1 C(=O)(C(Cc1ccncn1)NC(=O)OC(C)(C)C)NC(C)CF c1(OCCC(=O)NCC2CN(C(CCN3C(=O)CCC3)=O)C2)c(F)cccc1Cl c1(CNC2(C(=O)OC)CCN(c3ccnc(Cl)n3)CC2)noc2c1COCC2 CCC(CC(=O)N(C)CCN(C(=O)C(C)COC)C)C(C)C c1(C(=O)NCC2CCC(NC(c3c(C)n(C)cc3)=O)C2)cc2n(c1)CCCC2 CCC(C)(CNC(c1cnnn1C)=O)C(=O)N1CC2C=CC1CC2 c1(C(N2CCC3C(NC(C(C)OCC=C)=O)C32)=O)ccnc2c1cnn2C c1(CNC(c2cnn(C)c2C(=O)NC2C3CN(CCF)CC23)=O)cccc(F)c1F c1(CC)ccc(C(=O)N(CC(C)NC(c2nocc2Cl)=O)C)cc1[N+](=O)[O-] n1(CC(=O)NC(CC)CN(C)C(C2CCSC2)=O)nnc(C)n1 C(CC(=O)N(C)Cc1cccnn1)(C(F)F)NC(c1ccc(C)o1)=O c1(C(=O)NCCC(C)NC(CCC2CCC(C)O2)=O)cnc2ccccn2c1=O Cc1nnc(N2CCN(C(=O)Nc3cnc(Cl)s3)CC2)n1C C1(CNC(C=C(C)C(C)C)=O)CCN(C(c2ccc(-c3cccs3)o2)=O)CC1C CCC(CC(=O)NC(C)CNC(c1cccnc1I)=O)SC c1(NC(CC)(C)Cc2ccccc2F)cc(CN(C)C)cc(C(F)(F)F)c1 CC1CC2C(CC(C)(C(=O)O)N2Cc2ccc(C#N)[nH]2)O1 N1(C(c2c(CC)c[nH]c2)=O)CCCC1(C)C(=O)NCC(C)(C)OC Cc1cc(C(N2CCSCC2CCNC(C2CC2C(F)F)=O)=O)sc1C C1(C)(CO)CN=C2NC(=NC3=C2COCC3)N2CCN3C(=O)N(C1=O)CC23.CO C(=O)(CCC1=NNC(=O)CC1)NC1C(C)CN(C(C2CC(N(C)C)C2)=O)CC1 N1(C(Cc2c(CC)n[nH]c2CC)=O)CC2(CC(NC(c3csc(C)n3)=O)CO2)C1 N1(C(C2(OCC)CCCC2)=O)CCOC(C(C)NC(c2cncc(F)c2)=O)C1 C1(C(=O)NCc2ncco2)CCCCN1C(C1CCCN1C1CC1)=O C1(C(=O)OC)CC2C(CCC(C)N2S(=O)(=O)CCOC2CCCCCC2)O1 CC1=NN(C)C(=O)C1CC(N1CCN(C(c2[nH]cnc2C)=O)C(C2CCC2)C1)=O N1(C(CC2(OC)CCCC2)=O)CCCC(NC(c2cncc(C)n2)=O)CCC1 c1(CCC)ccc(S(=O)(=O)NC2CC(C(=O)Nc3cc(O)nc(Cl)n3)C2)cc1 C1(C(=O)NCC=CCC(=O)NCC(C)OC)CCCC(=O)C1 c1(C(N(CC(CO)(CO)NC(=O)C=Cc2cnc[nH]2)C)=O)csc([N+](=O)[O-])c1 CC1(CNC(c2ncnn2C2CCC2)=O)CC(F)(F)CN1C(C12CC(C1)C2)=O N1(C(CCC=C(C)C)=O)CCN(C)C(CNC(c2ccncc2)=O)C1 c1(CNC(C(C2CCC2)NC(c2ccc(O)cn2)=O)=O)cccc(F)n1 C1(C2CCCN(C(C3(c4ncco4)CC3)=O)C2)(NC(=O)C(F)C(F)(F)F)CC1 C1(C)(CNC(CCN(C(CCOC)=O)C2CC2)=O)C=CCCC1 C1(NC(C(C(C)C)OC)=O)CC2(CCCCN2C(=O)C(CSC)OC)C1 c1(C(=O)NC2CC(F)(CNC(C3(C)CCCCO3)=O)C2)cnc2n1CCCCC2 C1(C(N2C(CO)CC(NC(C(CCCC)NC(N)=O)=O)C2)=O)Cc2nnc(C)n2C1 Cc1ccc(F)cc1NC(=O)CONC(c1coc(C(F)F)c1)=O Cc1cc(C(=O)N(C2CCCN(C(c3cc(C(F)(F)F)nn3C)=O)C2)C)cnn1 C(=O)(CC(C(=O)N1CCC(NC(=O)CC(C)OC)C1C)N(C)C)OC c1(OC)cccc(Br)c1C(=O)NC1CCN(C(=O)CNC(=O)OC(C)(C)C)CC1F C1(NC(COc2ccc(C(CC)C)cc2)=O)CCCCN(C(=O)CC(F)F)C1 CCC(C)(C#N)C(=O)N1CCCC1CN(C)C(c1nc(C)oc1OC)=O c1(C(=O)NC(CNC(C(Cc2c(C)noc2C)C)=O)C)ccc(F)c2occc12 CN=c1[nH]c(=NCc2cncnc2)[nH]c(=NCCCN2CCCN(C)CC2)[nH]1 c12cc(on1)CCNC2=O.C1(=O)C(C2CCC2)N1.C=CC(C1CC1)C1CC1 N1(C(CCNC(CC(C)C)=O)=O)CCCN(C(c2ncccc2Cl)=O)CC1C c1(C(=O)NC(CCCC)CNC(=O)C(C)SC)c(C)nc2ccccn12 CC(C)CCCC(=O)N1CCC(NC(c2cn(C(C)C)nn2)=O)C1 CCC1=NOC(CC(=O)NCC(CC2CC2)C(=O)NCCCCCO)C1 Cc1nn(CCO)c(C)c1C(=O)NCC(C)CN(C)C(C1COC(=O)C1)=O Cc1cc(C(=O)NC2CC(F)(CNC(c3cc(C(C)C)on3)=O)C2)c(N)cc1F N1(C(C=C(COC)C)=O)CC(C2CN(C(=O)Cc3ccc(Cl)c(OC)c3)C2)C1 C1(C(N2CCC(NC(c3sccc3Cl)=O)C2)=O)CCCCC12CCC2 C1(C(=O)NC23CC(CNC(c4cnccc4Cl)=O)(C2)C3)CCCC1C1CC1 c1(NC(N(CC(c2ccccc2)CC)CC)=O)nc2ccc(I)cc2s1 C=CCN=C(NCC(=O)N(CC)CC)NCC1(C)CCCCC1 c1(CC(CNC(=O)Cc2cc(C3CC3)ns2)CO)ccccc1F C(=O)(CC1=CCCC1)N1CCC(CC)C1C(N1CC2CC(C)C2C1)=O N1(C(c2c(OC)n[nH]c2)=O)CC(C)C(C)(CNC(c2c(Br)noc2C)=O)C1 c1(NCCOc2c(C)cccc2)ccc(S(=O)(=O)N(C)C(C)C2CC2)c(Cl)c1 c1(NC(=O)NC(C)CC#N)cc(NC2CCCC2C(C)(C)C)ccn1 N1(C(c2n(C=C)ncc2)=O)CCC2(NC(=O)C=C3CCSCC3)CCCC12 c1(CCC(=O)NCC(C)N(C(c2n[nH]c(C)n2)=O)CC)cncc(F)c1 c1(C(=O)NC2C3N(C(C=CC=CC)=O)C(CC3)C2)cc(Br)cc([N+](=O)[O-])c1 N1(C(c2n(CCOC)ncc2)C(=O)NCC2CCCO2)CCc2ncc(C)n2CC1 c1(C(N2CCC(OCCNC(=O)Cc3cncs3)C2)=O)cncc(C(F)F)c1 c1(C(=O)NC2C(C)(CN(C(=O)CC3CC3)C)CCC2)cc(O)c2cnn(C)c2c1 N1(C(c2cc(C)n(C)n2)C(=O)Nc2ccccc2)CCCc2[nH]ccc2C1 Cc1ccc(O)c(NC(=O)CC2CN(C(=O)C(O)CNC(N)=O)CC2C)c1 c1(OCC)cncc(NC(C2CCCN2C(=O)CCc2ncccc2Cl)=O)c1 C(=O)(C(CN(C)C)C(C)C)NC(CC=C)C(=O)N1CCC1C(C)O C1(C(N(CCCNC(CC)=O)C(c2cc(C)c(Cl)s2)=O)=O)CCCCN1CC(F)F C1(C)(NC(N2CCCC(CC)C2)=O)CC2(CCC2)C1.C1(=O)C(OC(C)(C)C)CO1 Cc1nc(CCNC(C2(NC(=O)CCc3ccsc3)CCOCC2)=O)c(C)o1 C(=O)(C1=C(c2ccccc2)SCCO1)N1C2CC(NC(=O)CC(F)(F)F)C(C2)C1 CC(C)(CC#N)C(=O)NCC1(F)CCC(CNC(=O)CSc2ccccc2Cl)C1 N1(C(COC(C)=O)=O)CCN(C(C2(C(N3CCOCC3)=O)CC2)=O)CC(O)C1 C12(C(=O)OCC)COC(CNCCCc3nnc(C)o3)(C1)C2 CCCCCCC(C)(CC)C(=O)NC(CNC(C1(C(N)=O)CCC1)=O)CC CC1Cc2cccc(C(=O)Oc3cccc4c3CCOC4)c2O1 N1(C(C2(C)COC(=O)C2)=O)CCCC(C)(C)C1CNC(=O)Cc1csc(S)n1 c1(C(N2CCC(C(=O)NC3CC(O)CC3O)(CF)C2)=O)cccnc1S C(=O)(C1CCCc2n[nH]cc21)N1CCC(NC(C=COCC)=O)(CO)C1 c1(C(N)=O)ccc(NC(=O)C2CC2)cc1.C1(C2CCOCC(=O)N2)CCOCC1 N1(C(CC(C=C)C)=O)CCC(C)(C)C1CC(=O)NC(C(C)(C)O)C1CC1 C(=O)(C#CC1CCCOC1)NC(C)(C)CNC(=O)C(C)(C)C(C)(C)C C1(CCCNC(C(CC)N(CC)CC)=O)CCCN(C(c2ccccc2Cl)=O)C1 N1(C(C=CC)=O)CCC(CN(C(C2CC(=O)N(C)C2)=O)CC)CC1 Nc1ccnc(C(N2CCC(F)(CNC(c3cncn3C3CC3)=O)C2)=O)c1 c1(CC(C)NCc2cn(CCCCCO)nn2)ccc(O)cc1 C1(C(N2CCC(C)(NC(c3sc(C)c(O)n3)=O)C2)=O)CC1C1CCCCC1 c1(CC)nc(=N)[nH]cc1C(=O)NC(CNC(=O)C1=CCCC1)CC(F)(F)F c1(C(=O)NC2CC(CNC(=O)CC3CCC4CC34)C2)cc2c(=O)[nH]ccn2n1 N1(C(C2CC(NC(CCCC3C(C)C3)=O)C23CCC3)=O)CCCC2(CC(O)C2)C1 N1(C(C(C)NC(CC)=O)=O)CC2CC1C2NC(c1oc(C)nc1C)=O CC1(C)CN(C(C2CC(NC(=O)C=Cc3cc[nH]n3)C2)=O)CCO1 CCCC(CC)CC(=O)NC(C)CCNC(=O)CCSc1ccccc1F c1(CC(=O)NCc2cc3ncccc3[nH]2)cccc2ccccc12 C1(C(N(c2cccc(F)c2)C(C2CN(CC(F)F)C2)=O)=O)C2CC3C(C2)C13 C1(C(=O)NCC(CNC(CSC(C)(C)C)=O)(C)F)CCC(C2CC2)C1 CCC(CC)CC(F)C(=O)NC1CCCC(N(C(=O)Cc2ccnn2C)C)C1 Cc1c(NC(=O)C(CCC2(C#N)CC2)N(C2CC(F)(F)C2)C2CC2)cccc1Cl C(=O)(C(O)CC(C)(C)C)NC1CCC(C(=O)NCc2nn(CC)nc2C)C1 C(=O)(C1=NN2CCCN=C2N1)N1C(CCNC(C=CC2C(C)C2(Cl)Cl)=O)CCC1 c1(C(=O)NCCC(C)NC(=O)C(C)(C)c2ccnn2C)cc(Cl)c(Br)[nH]1 C1(NC(CN2CCN(CC)CC2)=O)CC(F)CN(C(c2cncs2)=O)C1 N1(C(CN(C(=O)CCN2CCCC2)C)=O)CC2(CC(N(C)C)C2)C1 C1(NC(=O)CCC2CCN(C(C3CC4(CCC4)C3)=O)C2)CCCCCCC1O c1(C(N(CC(C)NC(C2CCCN2C2CC2)=O)C)=O)cc2cc(O)ccc2[nH]1 c1(CC)cc(C(=O)NC2CN(C(C3(C)CC3(C)C)=O)CC23CC3)cc(F)c1 C(=O)(C(CC)C(=O)OC)N(C)Cc1ccc(CNC(C2CC(CC)C2)=O)cc1 c1(OC)ccnc(C(=O)NC2CCCN(C(c3csc(COC)n3)=O)CC2)c1F CCC(C)(C)C(C)CC(=O)N1CC(NC(c2c(Cl)ccc(F)c2F)=O)CC(C)C1 C(c1ccc(SC)s1)=CC(=O)NCC(CC=C)NC(=O)C(C)CC1CCCCC1 c1(CNC(c2cnc(CC)o2)=O)ccc(C(=O)N(C2CCCC2C)C)nc1 c1(C(=O)NC(C2CN(C(=O)CC3CCC(C)(C)C3)C2)C)cc(S(N)(=O)=O)c[nH]1 c1(C(N2C3(CN(C(c4c(CC)ncnc4)=O)C3)CC2)=O)cc(C#N)c(N)cc1O CC(C)CC(O)C(=O)NC1(C)CCN(C(=O)C(C)C(F)F)CC1 N1(C(c2ccc(CO)s2)=O)CCC(NC(C2CCC2)=O)C(Nc2ncccn2)C1 c1(NC)cc(N2CCCC(C)(C(=O)NCCC(N)COC)C2)nc(=N)[nH]1 CC1(CNC(=O)C2CC2)CN(C(=O)Cc2ccc(F)cn2)CCO1 c1(C(N2CC(O)(C(C)NC(C3C4CCC34)=O)C2)=O)ccccc1Br c1(OCC)cccc(NC(=O)C(=O)N(C2CCSC2)Cc2ccco2)c1 C(=O)(CCCC(=O)NCC)N1CCC(C(C)NC(C(CCC)F)=O)C1 N12CCOCC1CC2=O.c1(OCC)nc(C(=O)NCCc2ncoc2C)co1 Cc1cc(C(=O)NCC2CCCN2C(c2cc(Br)sc2Cl)=O)ncc1F C1(CNC(C(c2cccc(Cl)c2)C)=O)CCC(NC(=O)C(F)(F)CO)CC1 N1(C(C(CC)SC(CC)CC)=O)CCCCC12CN(C(=O)CN(c1c(C)noc1C)C)C2 N1(C(C(CC(C)C)ONC(CC2ON=C(C)C2)=O)=O)CCCC(C)(C#N)C1 C(C(C)(C)CNC(C1CCC1(C)C)=O)N(C(=O)COCc1ncnn1C)CC Cc1sc(C(=O)NC2CC3CC2N(C(=O)C(C)(C)c2cscn2)C3)cc1[N+](=O)[O-] CCC(C)(C(=O)N1CCN(CC2CCCN(C(C3CC=CC3)=O)C2)CC1)C(F)F N1(C(c2c(F)ccc(C#C)c2)=O)CC2CN(C(=O)C=Cc3ccco3)CC2(C)C1 C1(C(=O)NCC2(NC(c3nccnc3Cl)=O)CCCC2)CC2CCC(C1)S2 c1(C(=O)NC2CCN(c3c(C#N)cncn3)CC2F)cccc2c(Cl)ccnc12 c1(C(=O)NC23CN(C(CCC(C)C)=O)C(CC2)CC3)c[nH]c2cc(F)ccc12 Cc1cn(C)cc1C(N1CC(NC(=O)CC2CSC2)CC1C)=O C(CCC(C)C(=O)N1CCN(C(=O)CSc2nc(C)cc(C)n2)C(C)C1)OC CN1CCC(C)(C(N2CC(NC(=O)C(Cl)=CCl)C(CO)C2)=O)C1 N1(S(C)(=O)=O)CCC(C(=O)N(c2ccccc2)C(c2csc(O)n2)=O)CC1 c1(OC)ncc(Br)cc1NC(C1CC1C(=O)Nc1cccc(C2CC2)n1)=O N1(C(C(C(=O)OCC)OC)=O)CCOCC(NC(=O)CCC2CC(F)(F)C2)C1 c1(C(=O)NC(C)(CNC(C2CCC(O)C2)=O)CO)nnc(Cl)cc1N CCCCCCCC(=O)NC(C)(CNC(c1ccnc(O)c1F)=O)CC C=C(C)CCCC(=O)NC1(C)CCN(C(c2ccc(OC)cc2C(F)F)=O)C1 N1(C(COC2CN(C(C)=O)C2)=O)CCCC2CN(Cc3ncnn3C)CC12 c1(SCC(=O)NC2(C(F)(F)F)CC(O)(CS(C)=O)C2)nc2ccccc2s1 c1(C(=O)NC(C)CNC(C2C=CCCC2)=O)cc(C(F)(F)F)cnc1O N1(C(C2=CC(C)(CC)C2)=O)CC2(CCN(C(c3occ(C)c3C)=O)C2)C1 C(C)(C)(CC(=O)Nc1ccc(C(C)=O)cn1)N(C(CSC)=O)C c1(CCC)c(C(=O)NC(C)CC(C)NC(c2[nH]c(C)cc2C)=O)nnn1CC c1(C(N2CCC(NC(C3C(C=C)C3)=O)C2)=O)cc2ccccc2cn1 CN1CC(O)CC1C(N1CC(CCCCNC(=O)C(c2cccnc2)O)C1)=O CC(C)CCCCC(=O)NC1(CNC(C2CCC3(CCCC3)C2)=O)CCC1 C1(CCN(C)C(C2(O)CCCCC2)=O)CCN(C(=O)CCS(C)=O)CC1 N1(C(C)=O)CCOCC(C)(CNC(C2CCC2Cc2ccc(Cl)c(Cl)c2)=O)C1 N1(C(C2(COCC)CCC2)=O)CC2OCCN(C(=O)C(C)CSC)C2C1 NS(=O)(=O)c1ccsc1C(=O)NC1CC(NC(C2CCCO2)=O)C1 c1(C(=O)OC)ccc(C(=O)N(CC(O)CN(C(=O)CN2CCC2C)C)C)c(F)c1 c1(CC(=O)NC2(CC=C)CCN(C(=O)CC34CCCC3C4)C2)cccc(F)c1Cl C1(OC(C2C=CCC(c3nc(-c4ccncc4)no3)C2)=O)CC2C(C1)C2(F)F Cc1ccc(C(C)C)cc1OCC(=O)NCC(C1CC1)NC(c1ccc[nH]1)=O N1(C(C(CC)C(=O)OC)=O)CCC2(CCC2)C(NC(c2nc(C)ncc2Cl)=O)C1 N1(C(c2cnccn2)=O)CCC2(CC1)CN(C(=O)Cc1nncs1)CC2CO N1(C(c2cncc(OC)c2Cl)=O)CC2CN(Cc3cc(F)c(Cl)c(Cl)c3)CC2C1 C=CC(CC)CC(=O)N1CCC2C(C(=O)NCC3COCC3(C)C)C2C1 C(=O)(C1=CSCCO1)N(CCCCCNC(C1CN(S(CC)(=O)=O)C1)=O)C c1(C(=O)NC(CNC(c2n(CC)ccc2)=O)C2CCC2)cccc(N)c1O Cc1ncc(C(N2CC(NC(c3cnc(S)nc3)=O)CCC2C)=O)cc1Cl c1(C(C(=O)NCC2CCN2C(=O)CNC(=O)C(F)(F)F)C2CC2)cccc(Cl)c1 S(=O)(=O)(c1c[nH]c(=NCC2CCOC2)cc1C)NC(Cc1c(SC)cccc1)C n1(CC(=O)Nc2c(C#N)ccnc2)cc(-c2ccc(F)cn2)cc(C2CC2)c1=O N1(C(c2cc(OCC)no2)=O)CCN(C(=O)C(C)N2CCCC2)C2(CCC2)C1 c1(CC)cc(C(=O)NCC(C(C)(C)C)NC(=O)CCNC(=O)C(C)(C)C)sc1C C(=O)(CCCCN1CCCC1)N(C(C1CCN(C(C2(C#C)CCC2)=O)C1)=O)CCN c1(OC)c(Cl)ccc(C(N2CCC(F)C(NC(=O)CSC(C)=O)C2)=O)c1F N1(C(=O)Nc2cc(-c3ccc(OC)cc3)nn2C)CC(N(C)C)CC1(C)C c1(CC)ncnc(NC2CCCC(NC(c3ccc(CCOC)cc3)=O)C2)c1F c1(OC)cccc2c(C(N3CCC(N(C(=O)C(C)=C4CC4)CCO)C3)=O)coc12 C1(C(=O)NCCC2CC(C)C2)CCN(C(=O)C2=COCC2)CC1(C)C c1(C(=O)NC2C(C)CN(C(=O)Cc3csnn3)CC2)cccc2c1ccn2C C1(C(C)C(=O)NC2(CF)CN(C(=O)CCC3CCC3)C2)CCC(=O)N1C CC1(C)C2CCC1(CC(=O)NC1CCCC(NC(c3cc(F)n[nH]3)=O)C1)CC2 N1(C(c2cc(OC)ncc2)=O)CCN(C(C2CC(C#N)(OC)C2)=O)CC1C C12(CCOCC1)CS(=O)(=O)N2.N1(OC)CC(C(=O)O)C(C)C1 C(CN=c1nc2sccc2c[nH]1)=CCNC(C(COCC)(C)OC)=O N1(C(c2ncc(OCC)nc2)=O)CCN(C(=O)C=CSC)CC1CC C1(OC)(CNC(C2C(C)C2C)=O)CCN(C(c2sccc2C(C)C)=O)CC1 N1(C(c2sc(CC)c(C)c2)=O)CCC(NC(c2cncc(C(C)C)c2)=O)C(C)C1 O=C(C(F)C(F)(F)F)N1CC2(C(N3CC4(CC4)CC3CO)=O)CCC1C2 c1(NC(C2(F)CCN(C(=O)Cn3ccnc3)C2)=O)cc(Br)cnc1[N+](=O)[O-] C1(CC=C)(NC(c2coc(Cl)n2)=O)CCN(C(=O)C(N2CCNC2=O)C)C1 C1(NC(COC2(C)CCCC2)=O)CCC2CN(C(=O)C#CC3CC3)CC2C1 C1(NC(c2cc3ccccn3c2)=O)CCCCC12CCN(C(=O)CCCF)C2 N1(C(CC2C(C)=NNC2=O)=O)CC2(CCN(C(C3CS(=O)(=O)C3)=O)C2)C1 c1(CC(N2CCC(N(C(=O)COCC(F)F)CCO)C2)=O)cc2ccccc2o1 Cc1cc(C(=O)NC2CCCC(N(C(=O)CC3CCOCC3)C)C2)ncc1F c1(C(=O)NCc2occ(C(=O)NCC(CC)C3CCC3)n2)cc(OC)cnn1 C(=O)(C1=C(F)CN(C(=O)CC(C)(C)CC(F)F)CC1)NCCCCCC(C)C C1(CNC(C2(C)CC2Br)=O)(NC(=O)CC2CC3(CCC3)C2)CCOCC1 C1(CCNC(c2c(OCC)scc2)=O)CC(OC)CN1C(c1ccc[nH]1)=O c1(C(C(N2C(C(=O)NC)CCC2)=O)NCc2cn(CC)cn2)c(C)cccc1Br CC(C)(C(=O)NCCC1CCC(NC(=O)CCC2CC2)C1)C1CCC1 c1(OC)cccc(C=CC(=O)NC(C)(C)CCCNC(C2CSC2)=O)c1OC c1(CC)nn(C)c(CC)c1CC(N1CC(N(C(=O)CCCSC)C)C(F)C1)=O c1(C(=O)NC(C)(C)CNC(c2coc(Cl)c2)=O)ccc2c(c1)CC(C)(C)C2 C1(CNC(=O)CCN2CCCC2)C2CCC(C2)N1C(=O)CCc1cnc[nH]1 C1(OC)CN(C(c2nn(C)nc2Br)=O)CC1NC(c1ccc(C)cn1)=O C1(OCC)CCN2C1C2=O.C1(C(=O)NC(C)CCN(CC)CC)CCC(F)(F)C1 C1(CN(C(=O)C(F)(F)CO)C)C2CN(C(=O)C(c3cccn3C)=O)CC12 c1(NCC)cc(Cl)ccc1C(=O)NC1CCC1CNC(C1CN2CCC1CC2)=O n1(CC(N2CCC(N(C(=O)CC3CC(C)C3)CC)C2)=O)sc2ccccc2c1=O c1(N2CCCC(N(C)C(C34CCCC3CCC4)=O)CC2)nc2ncc(Cl)cc2s1 C1(C)(C(N(CC(O)CNC(=O)COC2CCC2)C)=O)CC(C2CC2)=NO1 CC12CCCCC1CN2c1ncc(C(F)(F)F)cc1Br c1(C(N2C(CNC(CS(CC)(=O)=O)=O)CC2)=O)ccc(F)c(Cl)c1F C(=O)(C#CC(C)(C)C)NC(CNC(C(n1cc(C)nc1)(C)C)=O)(C)CO C1(c2n(C)ccn2)CN(C(c2ccc[nH]2)=O)CC1NC(C1CC1[N+](=O)[O-])=O CC(C)CCC(O)C(=O)N1CCN(C(c2cccc(F)c2)=O)C(c2ncc[nH]2)C1 C(=O)(C(C(=O)N1CC(C)C(C)(CNC(=O)C2CC2)C1)C(C)(C)C)OC(C)(C)C Cc1cccc(C(=O)C(=O)NCCO)c1Cl.N1(C(=O)OC(C)(C)C)CC(O)C(C)C1 c1(C(N(CC(C)CNC(=O)CCC(C)N(C)C)C)=O)cc(C#N)ccc1Cl N1(C(c2c(Cl)ccc(C)c2)=O)CCN(C(C2CC(C)(O)C2)=O)C2CS(=O)(=O)CC12 C1(CN(C(=O)CCCc2ccccn2)CC)CCCN(CCCCCF)C1 C1(C(N(C(COC)COC)C)=O)CCC(CNC(C2CCCCC2F)=O)CC1 c1(C(=O)NCCN(CC(C)O)C(C2C(c3c(C)occ3)C2)=O)c[nH]ccc1=N C1(C(N(C(C)CO)C)=O)CN(C(=O)CCC2CCCC2)CC1F Cc1ccnc(C(N2CCC(Cc3cccnc3)C2)C(=O)NC2CCOC2)c1Br c1(CCC(=O)NCC2(CCNC(CSC)=O)CC2)cncnc1 Cc1[nH]cc(C(=O)NC2CN(C(c3cc(C#N)no3)=O)CC2C)c(=O)c1Br C1(C(N2CCC(C(C)NC(c3ccccc3Cl)=O)CC2)=O)CC(=O)CC12CCC2 N1(C(C2CC23CCCC3)=O)CC2CCN(C(=O)Cc3ccc(C(F)F)cc3)C2C1 C1(C(=O)NC(C(C)NC(c2n(CC)cnn2)=O)(C)C)CN(C(C)=O)CCO1 CC(C)(CCNC(c1ccc(C(N)=O)cc1)=O)C(=O)NCCCN1CCCC1=O c1(CN(C)C(C2CCCSS2)=O)ccccc1CNC(=O)C(CO)N(C)C n1(CCCOC)nnnc1C(c1ccn(CC(F)(F)F)n1)NCC1CC1(C)C c1(C(=O)NC(c2cccc(Br)c2)C)cccc(OC(C)(C)C)c1 CCC(O)C(C)C(=O)N1CCCC1CCCNC(=O)CCc1ccccc1 CC(C)CC(C(=O)NC1CCCC(NC(=O)CCc2nncs2)C1)N(C)C c1(C(=O)NCC(CC=C)NC(=O)CC(C)c2ccco2)c([N+](=O)[O-])cnn1CC c1(C(=O)NC2CN(C(c3nc(C)oc3)=O)CC2C)c(Cl)cncc1Cl CCCC(C(=O)N(C)CCOCCNC(=O)C=C(Cl)Cl)C(C)C N1(C(C(CC)Sc2ccccc2)=O)CCC(C)(NC(c2nn(C)cc2N)=O)C1 c1(OC)ccc(C(N2CC(NC(=O)CCC=CC(C)C)C(C)(C)C2)=O)cc1O c1(OC)cc(C(C(=O)NCc2ccco2)N(C2CCS(=O)(=O)C2)C)ccc1Cl C(=O)(C1=CNS(=O)(=O)N=C1C)N1CC(CCOC)N(C(=O)CC2(O)CC2)CC1 N1(Cc2cc(C)on2)CC(NC(c2coc(Br)c2)=O)C(C)(C)C1 C12(CC(=O)N(C(CCNC(C3CN(C(C)=O)C3)=O)C)C)COC(CF)(C1)C2 C(=O)(C(CC(F)F)N(C)C(c1nc(Cl)cs1)=O)NC(c1scc(C)n1)C C1(N(C)Cc2ccc(NC(C3CCC(=O)NC3)=O)s2)CCCCC1(C)C c1(-c2nnc(COC3CCN(CCC(=C)C)C3)o2)cccc(Cl)c1 C12(NC(CCOC)=O)CCCN(C(c3n[nH]c(C)n3)=O)CC1C2 C(=O)(C#CC1CCCCC1)N(C1C(C(N2CCC(C)(CO)C2)=O)CCC1)CCO c1(CNC2CCC(C(=O)Nc3c(OC)nc(Br)cc3)CC2)cc(Cl)cc(Br)c1O C1(CNC(c2cccc(C(C)C)c2)=O)CCN(C(=O)Cc2cncn2C)C1(C)C C1(NC(c2c(C(C)=O)cccc2)=O)CC2CN(C(C3CSC(C)=N3)=O)CC2C1 Cc1ccnc(C)c1C(=O)NCC1(F)CCC(NC(=O)C(C)CC2CCCC2)C1 C1(N(C(CCC#C)=O)C)CCCCN(C(c2ccc(N3CCC(O)C3)cc2)=O)C1 N1(Cc2cc(CC)c(O)cc2)CC2CCN(C(=O)Cc3ccc(Br)cc3)C2C1 C(=O)(CCCC(C)(C)C)NC(C1(C(N2CCC(F)(CO)CC2)=O)CC1)C C1(C(=O)NCCN(C(c2ccc(NC(=O)NCC)cn2)=O)CC)CCOC1(C)C N1(C(=O)OC)CCCC(C(=O)NCC(C)NC(c2onc(OC)c2Br)=O)C1 c1(CNCc2ccc(-c3ccc(COC)c(OC)c3)o2)c[nH]c2ncc(Cl)cc12 Cc1nc2c(s1)CN(C(C1(O)CCN(c3ncnc4c(Br)c[nH]c34)C1)=O)CC2 C1(C(=O)Oc2ccc(C3(C(=O)OC)CC3)cc2)CN(C(=O)C2CC2)CC1(C)C [SH](=O)(=O)CC(C)c1ccccc1.O(COCCO)C(C)=O c1(OCC(N2CC(CCNC(C(C)(C)n3ccnn3)=O)C2)=O)nc(O)nc(O)n1 C=C1CCN(C(c2ccc(C3CCCC3)cc2)C(=O)NCCOCC)CC1 N1(C(c2c(C)coc2)=O)CC2CCC(C1)N(C(c1csnc1Cl)=O)C2 CCCC(O)CC(=O)N1CC2CC2(CNC(c2ccc(C)cc2Cl)=O)C1 CC1CC=C(C(=O)NC2C=CCN(C(c3cccc(F)c3C3CC3)=O)C2)CC1 c1(C(=O)NC2(C)CCN(C(C3C(C)C3(F)F)=O)C2)ncc(C(F)(F)F)cc1N C1(NC(C(C)=CC2CC2)=O)CC2(C1)CC2NC(c1cc(CS(C)(=O)=O)on1)=O C(c1ccccc1Cl)=CC(=O)NC(C)CC(C)NC(=O)C(C)n1cnnn1 c1(C(N(CC)CC)=O)ccc2c(c1)CN(C(=O)CCc1ccc(C)nc1)CC2 C1(C(N(CCC)C)=O)N(C(=O)CN2CSCC2=O)CCC1(C)C c1(C(=O)NCC=CCNC(c2cn(C3CC3)cn2)=O)cc(F)cc(Br)c1O Cc1ccnn1CC(=O)N(CCC(=O)NCCCn1cncn1)C1CC1 CCC1=NOC(C(=O)NCC2CN(C(=O)CC(C)CN(C)C)C2)C1 CON1CC(C(=O)NCC2(CNC(C3CCC4CC3CO4)=O)CC2)CC1=O c1(C(c2nnnn2C2CC(F)(F)C2)NCC(C)C)cccc(C2CCOCC2)c1 N1(C(C(C)n2ccnn2)=O)CC2(CCC2)CC1CNC(c1nnn(C)n1)=O c1(CC)cnccc1CNC(=O)NCC(C)COc1ccccc1C c1(CCC(=O)NCCCN(C(C(CC)O)=O)C)ccc(O)c(OC(F)(F)F)c1 c1(C(=O)NCC(CC=C)C(=O)NCc2cnn(C)c2)cc2cccn2cn1 C1(NC(C2C(C)CCO2)=O)CN(C(=O)CCCCN2CCOCC2)CC1F c1(C(N(CC(C)NC(c2cnn(C)c2)=O)CC)=O)cc(C(C)(C)C)n(C)c1C N1(C(=O)Cc2csc(Cl)n2)CC2C(CNC(C3(F)CC3c3ccccc3)=O)C2C1 C(=O)(CCCCCN)O.C1CCC(=O)N(C)CCO1.C(CC(C)C)OCC(=O)CC=C C1(C(C)(C)C)(C(N2CC(NC(=O)CCc3ccsn3)C2)=O)CCCCC1 c1(C(c2nnnn2C(C)(C)C)NC(c2cc(C)on2)C)c(Br)cnn1C1CC1 Cc1ccncc1NC(c1ccc(CNC(=O)C(O)CC2CCCC2)s1)=O c1(OC)cc(C(N2CCC(NC(=O)C(C)C#N)C2)=O)cc(Cl)n1 C1(NC(C(C)C2CC2)=O)CCC2(CC1)CN(C(c1ccnnc1S)=O)CCO2 c1(C(C)C)nc(CC2CCC(C)O2)n(-c2nc[nH]n2)n1 Cc1cccc(C=CC(=O)N(C2CCN(C(=O)Cn3cc(Br)cn3)C2)C)c1 c1(OC)ccc2c(c1)CC(C(=O)NCC(CO)NC(=O)CC(F)(F)Cl)O2 c1(OC)ccc(NC(C23CC2CN(C(C)=O)C3)=O)c(OC)c1 CCC(COC)C(=O)N1CCCC1(C)C(=O)NCc1ncn(C2CC2)n1 Cc1[nH]c(C)c(C(=O)NC(C)CCNC(=O)CC2NC(=O)NC2=O)c1C O=C1CCC(C(=O)N2CC(CNC(=O)COCc3ccncc3)C3CC23)=NN1 N1(C(C(C(C)(C)C)O)=O)CC=C(CC(=O)NC2CC3(COCCO3)C2)CC1 C(=O)(N=c1nc[nH]n2cc(Br)cc12)c1c(C)nc(-c2ccnn2C)cc1 N1(C(CCc2c(C)ncnc2O)=O)CC2CC1CN(C(=O)C(O)C(F)F)C2 C1(CNC(=O)CCCc2cccs2)CC2COCC2N1C(C1CCC(=O)N1)=O N1(CC(=O)N(C(CCNC(Cc2ccc(C(C)=O)s2)=O)C)C)CSCCSC1 Cc1csc(C)c1C(=O)NCc1cc[nH]c1C(=O)NCc1ccccc1O C1(O)(CN(C)C(c2cn(C3CCC3)nn2)=O)CN(C(c2cccs2)=O)C1 Cc1c(C(=O)N=c2nn[nH]n2C)cc(-c2ccc(CBr)cc2)cc1[N+](=O)[O-] O=C(CC1CCc2ccc(O)cc21)OC1(Cc2ccccc2)CCCC1 CC1(O)CC(C(=O)N(C2CCN(C(=O)CC3CCOC3=O)C2)CCO)C1 Cc1cc(C(=O)NCCC2(O)CCN(C(C34CC(O)C3C4)=O)C2)cc(Cl)c1 C(=O)(C(O)P(C)(C)=O)N1CCCC(N(C(=O)COCCF)C)C1 N1(C(C2CC2(Cl)Cl)=O)CCCC(n2cc(C(c3cccnc3)O)nn2)C1 N1(C(CC=C)=O)CC(NC(c2ccc(=O)n(CCOC)n2)=O)CC12CCOC2 C1(C(N(C)Cc2nnnn2C)=O)CCN(C(C2CC2[N+](=O)[O-])=O)C(C)(C)C1 CC1CCCN(C(=O)C(=O)NC(C)CCN(C(=O)COc2ccsc2)C)C1 c1(CC)ocnc1C(=O)NC1CCC1CNC(=O)CC1CC2(CC2)C1 C(=O)(C(F)C(C)C(F)(F)F)NC(C)CCNC(=O)CC(C(F)F)n1ccnc1 CC1(C)CC(CNC(=O)N(C(C)C2CC2)Cc2cc(Cl)ccc2Cl)CC(C)(C)O1 CC1=C(CNC(=O)NCc2cccc3c2CCCC3)C(C)(C)CCC1 N1(C(c2cc(COC)sc2)=O)CC(C)(C)CC1CNC(c1cccc(OC)n1)=O N1(C(c2cc(C)c(Br)c(Cl)n2)C(=O)NC2(C)CC2)CCn2nnc(Br)c2C1 Cn1ccc2nc(N3CCC3(C)C(=O)Nc3ccc([N+](=O)[O-])c(Cl)c3)ncc12 CC1(C)CC(NC(c2ccc(C#N)cc2)=O)CN1C(=O)C=CI C(=O)(C(C)CC(=O)c1ccc(F)cc1)NCCC(C)NC(c1ccn(C(F)F)n1)=O c1(NC(C2CCC(C)N2Cc2cnc(Cl)s2)=O)cccc2c1C(=O)CC2 C12(NC(c3c(CC)nc[nH]3)=O)CCOCC1CN(C(C1CC(OC)C1)=O)C2 c1(CC)cccnc1C(=O)NCCCC1(NC(C2CCC(C#N)C2)=O)CC1 Cc1sc(S(=O)(=O)NC(c2ccc(OC(C)C)nc2)=O)cc1[N+](=O)[O-] C=CCC(CNC(=O)C=CCOC(C)(C)C)NC(=O)CCC1CCC(C)O1 c1(C(=O)NC(CNC(CS(CC)=O)=O)C(C)(C)C)cnn2c(N)cc(C)nc12 c1(C(=O)NCCOCCC(=O)N(C)CC2(C)CCC2)cccc(=O)o1 CC(C)CC(C(=O)N1CCCC(C)(NC(=O)Cc2coc(C(F)F)n2)C1)N(C)C C=CCCC(C(=O)NC(C1CC1C(=O)OC)C)NC(C1CCCC(CF)C1)=O c1(C(N2CCOC(CCCN(C)C)C2)C(=O)NC)cc(Cl)ccc1Cl c1(C(C)C(N2CC(NC(C3CCCC(=O)N3)=O)C(O)C2)=O)noc2ccccc12 C1(C)(C(=O)NCCCCN(C(C2(CCC)CCC2)=O)C)CC(C2CC2)=NO1 N1(C(c2c(C)nc(COC)s2)=O)CCN(C(c2cnn(CC(F)F)n2)=O)C(C)C1 C1(CC(=O)N(CC(CC)NC(=O)Cc2cc(C)sc2C)C)CCCC2(CC2)C1 N1(C(C2C(C)(C)OCC2)=O)CCOCC(NC(=O)Cc2cc(F)cc(Cl)c2)C1 C(=O)(C1CNc2ccccc21)NC1CCc2n(C)nnc2C1 c1(OCCCC(=O)OCC(C2(O)CN(CC(F)(F)F)C2)=O)ccc(Cl)cc1.C=O C1(C(=O)NC(C)CC2CN(C(=O)CN(C)C(N)=O)C2)C=CC=CC=C1 N1(c2snc(NC(C)C3CC3)n2)Cc2ccc([N+](=O)[O-])cc2C1.C(C)(C)(C)NC(=O)N O(NC(=O)C(C1(C)CC1)NC(C1CCO1)=O)C(CC)CC C#Cc1cccc(CN(C2CN(C(=O)OC(C)(C)C)CCC2F)C=O)c1 N1(C(c2c(OC)c[nH]n2)=O)CC2CCN(C(=O)C=CCO)CC12 C(=O)(CC(C)(C)CNC(=O)CC1CCN(C)C1)N1CCN(CC(C)C)CC1 Cc1nn(C)cc1-c1cn(CC(=O)NOC2CCC(=O)NC2)nn1 C1(C(N(C(CC)C(=O)OC)C)=O)C=CCN(C(=O)CCc2nc(C)no2)C1 Cc1nc(C(=O)NC2CC(NC(=O)C=CC3(C)COC3)C2)c(C)o1 Cc1cnc2n1CCC(C(=O)NCC13CC(NC(=O)CSCCC)(CCO1)C3)C2 C=CC1(C(=O)N(CCC(=O)OCC)C)CCN(C(C2C=CCS2)=O)C1 S(=O)(=O)(c1ccc(NC2CC=CC2)cc1Cl)NC1C(CC)CN(C)C1 Cc1cccc(NC(C2CC23CCN(C(c2ccccc2Br)=O)C3)=O)c1[N+](=O)[O-] Cc1cc(C(=O)N(C)CC2(NC(C3CNC(=O)CC3C)=O)CC2)c2c(c1)CCO2 c1(CC(N2CC(N(C(=O)CC34CCCC3C4)C)C2)=O)ccc(Cl)c(C(F)(F)F)c1 CC1CCN(C(=O)C(O)Cc2cnc[nH]2)CC1NC(c1n[nH]cc1Cl)=O CC(C)(F)C(C)(F)C(=O)NCC1CN(C(C23CC(CC(F)F)(C2)C3)=O)C1 c1(NC(C(CC(C)C)NC(C(C(=O)OC)(C)F)=O)=O)cc(Cl)c(F)cc1F c1(CC(CNC(=O)C(C2CC2)N(C)C)NC(=O)CNC(=O)C2CC2)ccccc1 c1(CC(=O)N(CCCNC(=O)CC2CC23CC3)CCO)ccccc1O c1(C(=O)NCc2c(C(=O)NC3C(COC)C3)scc2)cc(Cl)ccn1 c1(COCCOCCC#C)noc(-c2ccn(CC(=O)O)n2)n1 N1(C(CCCOCCC)=O)CCC12CN(C(=O)CC1COCC(C)(C)O1)C2 CC(CC(Cl)Cl)NC(c1sccc1-c1nn[nH]n1)=O C(=O)(C(F)CC(C)(C)C)N1C(C)(CNC(CCCN(C)C)=O)CCC1 n1(NCCC(c2nc[nH]n2)NC(=O)Nc2cc(C)oc2C)cnc2ccccc12 C#CCCCCCC(=O)NCC(C1CCCC1)NC(=O)CC1COCC(C)(C)O1 CC(C(C)(C)C)NC(=O)CN(C(=O)CC1CCC1)C1CCC1 c1(C(C)C(=O)NC2CCCC(NC(C34CC(CO3)C4)=O)C2)c(F)cccc1F Nc1ccc(C(N2CCC3CC3(NC(=O)C=CC3CC3)CC2)=O)c(Br)c1F Cc1ccc2c(C(=O)N(C3CCCN(C(c4cnsn4)=O)C3)C)coc2c1 N1(C(CCN(C2CCCCC2)C)=O)CCC(NC(C2(F)CCOCC2)=O)C(F)C1 CC1=CCC(C)(C(=O)NC(C2CN(C(=O)C(C)N3CCC3)C2)C)CC1 CC1COCC(CC(N2CC(=O)CC2C(=O)NOCCOCCO)=O)O1 C(c1cnn(C)c1C)=CC(=O)NC1CC(N(C(c2c(C)csc2)=O)C)C1 CC1(CNC(=O)C=CCO)CCC(NC(C23CCC(CC2)C3)=O)C1 C(C1=NOC2CN(C(=O)C3=CCCOCC3)CC12)NC(c1cc(C)nc(O)c1)=O n1(CC(=O)NC(C(=O)NCC(F)(F)Cl)C2CC2)cccn1 N1(C(c2ccc(Cl)c(F)c2)C(=O)NCC=C)CCCC(C2CCCC2)C1 C(=O)(CC(C)C1CC1)NCC(C)N(C)C(c1nc(Cl)cs1)=O N1(C(C(CC)C(C)O)=O)CCCN(C(=O)C(=Cc2ccco2)C)CCC1 N1(c2nc(OCC)c(C)cn2)C2CCC1CC(NC(=O)CCCC(N)=O)C2 C#CCC(O)C(=O)NC1CCC(CC=CC(=O)NCCC2(OC)CCC2)C1 C(=O)(C(C)(O)C(C)(C)C)NC1CCN(C(c2cnc(CCCC)s2)=O)CC1 CCCCC(O)C(C)C(=O)NCc1ccc(C(=O)N(C)Cc2cnccn2)cn1 c1(C(=O)NC2CC(C(C(=O)Nc3cnc(C)nc3)F)C2)c[nH]c(=N)c(C)c1 C=C(Cl)CCC(=O)NCc1ncccc1CNC(c1cccnn1)=O c1(C(c2n(C3(C)CC3)nnn2)NCCc2ccsc2)cnn2c1CCC2 c1(C(N2CC3C(NC(c4ccnc(C)n4)=O)C3C2)=O)cn(C)c(=O)n(C)c1=O c1(C(N(CCOCCNC(CS(C(C)C)(=O)=O)=O)C)=O)ccc2oc(=O)oc2c1 C1(NC(C2N(C)CCC2)=O)CN(C(=O)CCn2cnc([N+](=O)[O-])c2)CC12CC2 C1(CCC)CCCN(C(C2C(C)CN2C(=O)CC(C2CC2)C2CC2)=O)C1 CC(C)(CNC(c1ccc(Br)cc1)=O)CCNC(=O)Cc1cocn1 Cc1nn(C)c2nc(O)cc(C(=O)NC(C)CNC(c3snc(O)c3Cl)=O)c12 N(C(=NCCF)NCc1cc(C)nc(C)c1)CC(CC)(c1ccccc1)N(C)C C(=O)(C(=O)C(C)(C)C)N(C)CC1CCN(C(c2c(CC)ncs2)=O)C1 c1(OC)ccccc1C(C)(C)CNC(=O)NC(C)CC(C)(C)ON C1(C(=O)Nc2cn(SCC)nc2)CCCN(C(=O)C2CC2)C1 c1(CCC(=O)NC2CCC(NC(C(C)OCC#C)=O)C2)ccc2ccccc2n1 c1(C(N(CCN(C)CCO)C(C2CC3CC3C2)=O)=O)ccc(-c2cnn(C)c2)cc1 CC(C(=O)NCc1cc(C(N2CC(C)OCC2C)=O)co1)C(C)(C)C c1(OC)c(C(N2CC(CNC(c3ccnnc3O)=O)C2)=O)cccc1C#N N1(C(C(CC)(C)C)=O)CC2CCC1CN2C(=O)C(=O)NC1CCCC1 N1(C(c2c(C)snc2)=O)CCCCC1C(C)NC(c1csc(-c2nc[nH]n2)n1)=O C12(NC(CS(CC)=O)=O)CCC(CNC(=O)CC3OCCO3)(CC1)OC2 CCCN=C(NCc1nnc(CO)s1)NCC(c1ccncc1)O C(CC(=O)NNc1ncccc1[N+](=O)[O-])(c1ccc(F)c(Cl)c1)N(CC)CC c1(C(=O)Nc2cccc(NC(C(C)n3cncn3)=O)c2)n[nH]c2c1COCC2 N1(CC(=O)NC(C)C(=O)NC2(CN(C)C)CCCC2)CCC(O)CC1 CC1CN(C(c2ccc(Cl)nc2N)=O)CCN1C(c1ccc(C(F)F)c(F)c1)=O C=CCCCCCC(=O)NCCCN(C(c1ncc(C(=O)OC)s1)=O)CC Cn1nnc2cc(C(N3CC(O)CC3C(=O)NCC3CCC3)=O)ccc12 N1(C(C(=O)Nc2n(CC)ncc2)=O)CCC(C(=O)OC)c2cc(Br)ccc21 C(CCC(=O)NC(COC)C1(C)CC1)(C(C)C)NC(c1cn(CC)nc1)=O Cc1ccc(C(N2CC(NC(C3CNC(=O)C3)=O)C3(CCC3)C2)=O)c(N)c1Cl C1(C(=O)NC(C)C(C)(C)NC(c2ccc(O)c(C(N)=O)c2)=O)CC2(CCC2O)C1 c1(C(=O)NCC(CC)NC(c2cccc(CO)n2)=O)cc(NS(C)=O)ccc1F C(=O)(C1CCCc2scnc21)NC1C(CC)CN(C(=O)Cn2nccc2C)CC1 N1(C(c2cccc(F)n2)C(=O)Nc2ccc(OC)cc2C)CCS(=O)CC(C)C1 N1(C(C23N(C(c4n(CCC)ncc4)=O)CC(C2)C3)=O)CCn2nc(C)cc2C1 C(C(C(=O)Nc1cccn2ncnc12)C(C)(C)C)NC(CCC#C)=O N1(C(C(Cc2ccc(C)cc2)C)=O)CCC2CCC(NC(=O)CC3CC3)C12 C=CCC(CC(C)C)C(=O)NC1CN(C(c2cc[n+]([O-])cc2)=O)C2(CCCC2)C1 Cc1cc2cccc(C(N3CCCC(O)(CN=c4[nH]nc(O)s4)C3)=O)c2s1 C(=O)(CCCSC)N(C1CCN(C(=O)CC(O)C2CC2)C1)CC#C N1(C(C(C)(C)C#N)=O)CC2CCC1C(NC(=O)CC1CC(=O)NC1=O)C2 C(=O)(C1CC(=O)Nc2ccccc21)NC1CC(CNC(c2c(C)cnn2C)=O)C1 c1(C(=O)NCC(C2CCC2)NC(C(C)=C(C)C)=O)cc2ccccn2c1C1CC1 CCC(C(=O)NC(C1CCCC1O)CNC(C1(OC2CCCOC2)CC1)=O)N(C)C C(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1CCN(C(C2CC(C)OC2C)=O)C1 N1(C(C2C(C#N)C2)=O)CC(N=[N+]=[N-])CC1C(N1CCC2OCCC2C1)=O N1(C(C(C)OCC#C)=O)CCCC2(C1)CN(C(=O)Cc1cccc3c1CCC3)C2 c1(C(=O)NCC(CC)NC(c2csc(-c3cnc[nH]3)n2)=O)cccc([N+](=O)[O-])c1 c1(OC)nccnc1NC(=O)CC1CCCN1C(=O)COCCSC C1(NC(c2nc(COC)oc2)=O)CN(C(=O)C=C(Cl)Cl)CCC12CCOCC2 CCC(CCCC(=O)NCC=CC(C)(C)C)NC(=O)C(F)C(C)(F)F N1(C(C(C)Oc2ccncc2)=O)CC(CNC(=O)C(C)(O)Cc2ccccc2)C(C)C1 c1(NC(CCOC)C)ccc(C(F)(F)F)cc1S(=O)(=O)NC(C)CCC1CC1 C(=O)(CCCOC)N(C1(C(=O)NC(C(=O)N(CC)CC)C)CC1)C c1(-c2onc(CN3C(C)CCC(CCCOC)C3)n2)cccc2c(Cl)cccc12 c1(C(N(C(C)CNC(=O)C(c2cnccn2)C)CC)=O)c[nH]c2c(F)cccc12 CC#CCCCC(=O)N1CCCC1CC1CCN(C(=O)C(C)(C(C)C)OC)CC1 CCCC(O)CC(=O)N1CCC(CN(C)C(C2(C#N)CC3CC3C2)=O)CC1 C1(CNC(C(CN(C)C)NC(Cc2c(CC)con2)=O)=O)COCC1(C)C N1(C(CC2(OCC)CC2)=O)CC2C(NC(C3(O)CCC3)=O)C2C1 C(=O)(C(O)CC(C)(C)C)N1CC2C(NC(C3N(C)CCCC3)=O)C2C1 c1(C(=O)NCC2(NC(c3csc(Cl)c3)=O)CCC2)cnc(C2CCOCC2)nc1 c1(C(=O)NC(CC2CN(C(c3c(C)nns3)=O)C2)C)nnn(C2CC2)c1C(F)F N1(C(CC(C)F)=O)CC(C2CN(C(c3ccncc3N3CCCC3)=O)C2)C1 c1(N(CC(C2CCOC2)O)C)cc(Br)ccc1S(=O)(=O)NC12CCC(CC1)CC2 C1(C(=O)NC2(CO)CN(C(C3CC=CC3)=O)C2)CCCCCS1(=O)=O c1(C(=O)NC(c2ccc(Br)cc2)C#C)ccnc2ccc(Cl)cc12 C(=O)(C(CCC1CC1)NC(C1CC12CC2)=O)NCC1CC(C(N)=O)C1 c1(SC)cn(-c2ncc(CN3CCCC3)s2)nn1.N12CCC1C2=O N1(C(C2CCN(C(=O)OC)CC2)=O)CCC(C2CC2)(NC(=O)Nc2ccsc2)C1 C12(C(=O)NCc3ccccc3Br)CC1CN(Cc1cnc(-c3ccccc3)[nH]1)C2 N1(C(C2(CCC=C)CC2)=O)CC(NC(=O)CCc2nc(C)c(C)[nH]2)C2(CCC2)C1 c1(C(=O)NCC(CNC(C(COC)(C)OC)=O)(C)F)cccc2cn(C)nc12 N1(C(=O)CC2CCCN2C(c2ccnc(O)c2)=O)CCC2(C1)CC2(F)F C1(C(=O)NC(C(CC)C)CN(C)C)CCN(C(=O)Cn2ncnn2)C(C)(C)C1 Cc1ncc(C(=O)NCC(C2CCC2)NC(=O)Cc2cccc(O)c2)n1C(F)F c1(C(N(C(CNC(C(C)OCCC=C)=O)C)CC)=O)cn(-c2ccccc2)cn1 C(=O)(C1CCCc2nncn21)NCCCCCNC(=O)C(F)C(F)(F)F c1(C(=O)NC(C)C(C)NC(C2CCC(=C(F)F)CC2)=O)n[nH]c2cccnc12 C(=O)(CCC(C)(C)F)N1CC(OC2CCN(C(C3C(C=C)C3)=O)CC2)C1 C(C(=O)NCc1cnco1)(C(C)(C)O)NC(CNC(CC)=O)=O C(=O)(C(C)(C)CNC(C1C(C)C1C)=O)NC(c1snnc1C)C c1(C(=O)NCC(C)NC(C(CC)N(C)C)=O)cnn(-c2ccccc2)c1Cl N1(C(C2CCC(CC)O2)=O)CCC(CCNC(=O)C(N)=O)C(F)(F)C1 N1(C(COC)=O)CCCC1(C)CNC(c1ncoc1-c1ccc(F)cc1)=O C1(NC(CCN(CC)CC)=O)CC(O)CN(C(c2nc(OC)cc(OC)n2)=O)C1 C1(C(N(C2CCN(C(=O)Cn3cnc(C(N)=O)n3)CC2)C)=O)CC(C2CC2)=NO1 c1(C(N(CC)CC2CC2)C)cc(OC)c(Br)cn1 n1(CC(N2CCC(O)(c3scnc3Br)CC2)=O)ncc2cccnc12 CCC(CC(=O)NCCOCCCN(C(=O)CCNc1ccccn1)C)C1CC1 CN1CCN(C(C2CC(O)CN2)=O)C(CNCc2ccc(Cl)nn2)C1 n1(CC)nc(SCC(=O)OCCNC(C)C)c(Br)n1 C1(NC(c2nc(C)oc2)=O)CC(F)CN(C(c2cnn(C3CCC3)c2C)=O)C1 N1(C(C2C(C(C)NC(=O)CC(C)C(F)F)C2)=O)CCN(C)CC(C)C1 N1(C(C2CCCN(CC)C2)=O)CCC(C2(NC(c3ncc[nH]c3=O)=O)CC2)CC1 C1(C(=O)NCCNS(CC)(=O)=O)CCCCCC1NC(C12CCCC1C2(F)F)=O N1(C(C2CC(OCC)C2)=O)CCCN(C(c2ccc([N+](=O)[O-])cc2)=O)CC1C c1(C(N2CC(CN(C(CCOC)=O)C)C2)=O)n[nH]c2ccccc12 c1(C(=O)NCC(N(C(CC=C)=O)C)C2CC2)c[nH]c2nc(Cl)ccc12 N1(C(C(C=C=C)C)=O)CCN(C(c2ccnc(C)c2N)=O)CC(C)C1 CC1(CNC(=O)C(C2(O)CN(C(C3(Cl)CC3)=O)C2)F)CCCC(=O)N1 Cc1cc(C)c(C(=O)NCC2CC3CC3N2C(c2ccccc2O)=O)c(=O)o1 N1(C(C2=C(C)CCC2)=O)CC2OCC(NC(=O)C(CCO)N(C)C)C2C1 CC1c2cccnc2CCN1C(=O)NC1CCN(c2ccnc(Cl)n2)CC1 C1(OC)(OC)CCC1C(=O)NCC(C1CCCC1)NC(C1CCN(C)C1)=O C1(CC)COCCN(C(=O)C(O)C2CN(C(C3CC4CCC(C3)O4)=O)C2)C1 c1(C(N2C(C)CC(CNC(c3cncc(N)n3)=O)C2)=O)coc2ccc(Cl)cc12 C1(CNC(C(C)OCC(C)C)=O)CN(C)CCN1C(c1cn2c(n1)CCC2)=O C(=O)(CCC(N)=O)NCCOCCCNC(C1(CC#C)CCCC1)=O c1(C(=O)NC(C)CNC(C2CCN2C2CCCC2)=O)cnc(O)n(C2CC2)c1=O C1(C(CO)NC(c2ccccn2)=O)CCN(C(=O)C(F)n2ccnc2)CC1 O=C(CCCCCF)NC1CCCC(C(N2CCC3(CSC3)C2)=O)CC1 N1(C(C=NOC)=O)CC2CCN(C(c3cccc(F)c3Cl)=O)C2C1 C#CCCCC(C)C(=O)N1CC=CCC1C(N1CCC(CN(C)C)C1)=O CC1(C)C(O)C2CCCN(C(C3CCCCC3)C(=O)NC3CC3)C12 C1(NC(c2c(OCC)c(F)ccc2)=O)CN(C(c2cnccn2)=O)CC12CCC2 C(CCC(C)(C)C(=O)NCC1(C)CC2(CC2)C1)NC(CC1C(C)CCO1)=O C=CC(C(=O)N1CC(O)(C(F)C(=O)NC(CC)C2CC2)C1)OC CC(C)CCCCCC(=O)N1CC(C)CN(C(=O)CC2CCCSC2)C(C)C1 C1(NC(C(n2ccc(C)n2)C)=O)CCCC(C(N2CCCC2)=O)C1 C1(C#N)(CNC(C2C(NC(C(C3CCC3)OCC)=O)CCCC2)=O)CC(C)(C)C1 c1(C(=O)NCC2CCCN(C(CSCC)=O)C2)ccc(S(=O)(=O)CC(N)=O)cc1 c1(C(N(CCNC(c2c(F)ccc(C#C)c2)=O)CC)=O)cn(C)c(=O)n(C)c1=O c1(OC)ccc2cc(C(N3CC(F)(CNC(C4CC4OC)=O)C3)=O)[nH]c2n1 N1(C(C2C(COC)C2)=O)CCC(C)(NC(c2sc(C3CCCO3)nc2C)=O)CC1 Cn1ccc(C(C)(C)C(=O)NCC(C)(C)CNC(c2ccc(Cl)o2)=O)n1 C=C(C)C(CC(=O)N(C(C)CC(=O)NCC1CCCCC1(C)C)C)OCC c1(OC)cc(CN2CCC(NC(c3ccc(OC)c(I)c3)=O)CC2)ccc1O C1(CNC(c2cc(CNC(CNC(C3C(C)C3)=O)=O)sc2)=O)CCC2(CC1)CC2 Cc1ccc(C(=O)NC2CCC(C)N(C(c3ccc(F)s3)=O)C2)nc1C C1(CNC(c2ccc([N+](=O)[O-])[nH]2)=O)CCN(C(=O)CCCCCF)CC1O c1(C(=O)NCC(CNC(c2cccc(OC(C)C)n2)=O)C)nc2c(s1)CCCC2 C(=O)(CCP(C)(C)=O)N1CC(C)C(CCNC(c2sccc2CO)=O)C1 N1(C(Cn2cc(C(C)=O)nn2)=O)CC(CNC(=O)COC(C)C)CC1C N1(C(C2C(CC)N(C(C3CCCC4CC34)=O)CC2)=O)CC(N(C)C)C2(CC2)C1 CC1=C(C(=O)N2CCCCC2CCNC(=O)Cc2cn[nH]c2)CCC1 c1(C(=O)NCC2N(C)CCN(C(C(COC)OC)=O)C2)cc2cncc(C)c2s1 c1(C(=O)NCCCOC2CCN(C(CC(C)F)=O)CC2)cnc2sccn12 C(C(CC(C)C)NC(C1(C)CCN(C)C1)=O)NC(COCC)=O C1(=O)CC(C)N(C)N1CCCC(C)CC(C)(C)C(N)=O.CCO CCCC(C#N)C(=O)NC12CC(C(=O)N(C3CS(=O)(=O)C3(C)C)C)(C1)C2 C1(C(N2CC(OC)CC2CF)=O)(CC)CCN(C(c2c[nH]c(C)cc2=O)=O)CC1 c1(CC)cc([N+](=O)[O-])ccc1N(CCNC(=O)CC1CCC(C)(O)CC1)CC CC(C)S(=O)(=O)C(C)C(=O)NC1COC2C(NC(=O)C(O)C(F)(F)F)COC12 C(C(CNC(=O)C=Cc1cn[nH]c1)C(F)(F)F)NC(c1c(C#N)csc1)=O N1(C(CC2CN(C(C)=O)C2)=O)CCCC(F)(C(=O)NC(C)(C)CCCF)C1 C#Cc1ccnc(C(=O)NCC2(NC(=O)C=CC3CCC3)CCCCC2C)c1 C#CCCCC(C)C(=O)N1CCC(C=C)(C(=O)N(CC(O)CCC)C)C1 c1(C(N(CC(CN(C(C=C=C(C)C)=O)C)O)C)=O)cc(F)cc(C)c1N N1(C(C2(CC)CCN(C(=O)CCc3ccncc3)C2)=O)CC2CSCC2(C)C1 N1(C(CS(=O)(=O)N(CC)CC)=O)CCC(C)(C)C(NC(c2ccnn2C)=O)C1 N1(CCCC)CCOCC1C(=O)NCCCC(C)NC(c1ccsc1C(F)F)=O c1(CN(C(C)=O)CC2CCOC2)cn(CC(N2CCCC2C(C)(C)O)=O)nn1 C1(CCNC(C2CCCO2)=O)CCCN(C(c2ccc(C(F)(F)F)o2)=O)CC1 c1(OC2CCN(C(N(C(C)C)Cc3c(C)cccc3)=O)C2)ccc(F)c(F)c1 Cc1nccc(CNC(C2(CNC(=O)CCCF)CC(C)(C)C2)=O)n1 N1(C(C2N(C(c3c(O)ccc(C)c3)=O)C3C(C2)C3)=O)CC2CCCC(C1)N2C C1(C(=O)NC2CCCN(C(c3cc(C)c(Cl)s3)=O)C2)CCC(C)(F)CC1 C(=O)(C(C)CC(C)C(C)=O)NCc1c(C(=O)NCC(CCCC)O)n(C)nn1 C1(NC(CN(C(C(C)C)=O)C)=O)CCCC(CNC(=O)C(=Cc2cccs2)C)C1 c1(CC)oc(C(=O)OC)cc1S(=O)(=O)NC1(C(=O)OC)CS(=O)(=O)C1 N#Cc1c(F)c(NCC2CCCN2CC(F)F)nc(F)c1F CC(O)CCCC(=O)N1CC(N(C(=O)Cc2cccc(O)c2F)C)C1 C1(COC)(CNC(C2CC3(CC3)CO2)=O)CCCN1C(=O)C=Cc1cc(C)no1 CCC(C)(C)CC(=O)N(C(C)CNC(C12COC(C1)C2)=O)C N1(C(C(CC=C)OC)=O)CCCN(C(c2cccn3ccnc23)=O)C(C)C1 N1(C(C(CC(C)C)OC)=O)CCC2CCCC(C1)N2C(c1cncnc1C)=O N1(C(C2=C(C)OCC2)=O)CCC2(CC1)CN(C(C1CCCC(C)CC1)=O)C2 c1(OC)cc(C)nc(NNC(=O)NCC(c2ccc3nnc(C)n3c2)=O)n1 c1(NC(C2C(c3n(C)c(S)nn3)CC2)=O)nncc2c1CCCC2 N#Cc1cc(NC2CC(F)CN(C(c3cc(C4CC4)on3)=O)C2)ncn1 C12(C(=O)NCc3cn(C)nc3)CCCC1N(C(C1CCC(F)CC1)=O)CC2 C=C(C)C(C)(C)C(=O)NCC1CC(C(F)(F)F)CN1C(C1COCCO1)=O Cc1cc(Br)ccc1CN1CCN(CC(=O)Nc2ccnc(Cl)c2C)CC1 N1(C(CCS(C)=O)=O)CCC(NC(=O)Cn2ncc3ncccc23)C12CCC2 C(=O)(CCCCN(C)C)NCC(CO)NC(C(c1ccccc1Cl)OC)=O C(CC(C)(C)C)(C(=O)N(CCCCCC(=O)N(C1CCC1)C)C)OC C(=O)(CC(C)(C)CNC(C1CCCN1C(C)C)=O)NCCC(C(=O)OC)C C(=O)(C(F)CC(C)(C)NC(C1CCC(=O)CC1)=O)Nc1c(OC)ccc(C)c1 CCCCCC(O)C(=O)NC(CNC(=O)C(c1cnn(C)c1)C)(CC)CC N1(C(CCC(C)C#N)=O)CCC2C(C1)CN2C(=O)CCc1ccc(Cl)c(Cl)c1 Cc1cc2occ(C(=O)NC3CCCC3NC(C3CCNC(=O)C3)=O)c2cc1C N1(C(CCc2nnc(C)s2)=O)CC2CN(C(=O)Cc3cc(Cl)ccc3O)CCC12 N1(CC(C)(O)C2(NCCC=CC)CC2)CCCC(C(N)=O)C1 C1(N(C(C(=O)NCCOC)C2CC2)CCC)CCCC1 C1(C(=O)Nc2ccc(OC)nc2OC)(CC)CCN(C(C2CC23CCC3)=O)CC1 c1(NC2(C(=O)Nc3cc4c(cc3)C(=O)NC4)COC2)ncnc2cccc(F)c12 Cc1c(C(N2CCC(NC(=O)CC3CCC3)C(CO)CC2)=O)nn2ccccc12 C1(C(=O)NC2(CCC)CCN(C(C3CCCO3)=O)CC2)CC2(CCOCC2)CO1 C(C(C)(CC(C)C)NC(=O)C(O)Cc1cccc(Cl)c1)NC(CCC=CC)=O C1(C)(C(=O)NC(C)CCCNC(c2c[nH]ccc2=N)=O)Cc2ccccc2C1 N1(C(CC=CCCCCC)=O)CC2CCC(CNC(c3cscc3C)=O)C2C1 C1(C(C)C)CN(C(C2(n3cc(C(C)(C)C)nn3)CC2)=O)CCCN1C(=O)CO CC(C)CC(C(=O)NCC1CSC1)NC(=O)C1=CCCC1 c1(C(=O)NC(C(C)(C)C)c2cccs2)ccc(-n2cccn2)c(F)c1 CC1CC1C1CC1NC(=O)CC(C)(C)NC(=O)C(F)n1ccnc1 c1(C(=O)NCC(CO)NC(C(C)OCCC#C)=O)coc2cc(F)cc(F)c12 CN1CC(C)(C(=O)NCCCCNC(C2C(CN=[N+]=[N-])C2(C)C)=O)CCC1=O C(=O)(CC(C(C)C)NC(=O)Cc1ccoc1)NC(CCC)CCC C1(C(=O)NCCN(CCCC)C)COCC1NC(=O)CNC(C)=O C1(C2CCN(C(C3CNc4ccnn4C3)=O)C2)(NC(C2CCCC(O)C2)=O)CC1 c1(C(N(CCCNC(=O)C(F)CC2CCC2)CC)=O)[nH]c2c(C)cccc2c1C c1(CC)[nH]ccc1C(N1CC(CNC(=O)C(C)c2ccco2)(OC)C1)=O C1(NC(c2ccc(CO)cc2F)=O)CCN(C(=O)C(F)=CC2CC2)CCC1(F)F c1(C(=O)NC2C(NC(C(COC)C)=O)CCOC2)cc(C)cc([N+](=O)[O-])c1N c1(N(CONC(C=C(C)C)=O)CC2(c3ncccc3F)CC2)ccc(C#N)cn1 c1(CNC(CCN(CC#C)C(C2CCCS2)=O)=O)nn(C)cc1CO c1(C(=O)NCC2C(CNC(CCC=CC)=O)C2)cn(C)nc1COC n1(CC(=O)NCCC2CCN(C(C3(F)CCC3)=O)C2)nc2c(n1)CCCC2 CC#CCC(C(=O)NC(C)C(=O)N(C)CC)NC(c1cn(C)nc1C)=O Cc1cc(C)c(C(N2C3CC2CN(C(=O)CC2CCC(C#N)C2)C3)=O)cc1C N1(C(CCc2onc(CC)n2)=O)CCCN(C(c2coc3c2COC3)=O)CC1C C1(NC(c2ccc(CO)cc2F)=O)CC2CCC1N2C(=O)CC1CCCCCC1 c1(-c2n(C)ncc2CNC(=O)NC2(C)COCCC2C(=O)O)cc(O)nc(O)n1 C1(NC(C2C(C(C)C)CCC2)=O)CN(C(=O)C=CCOC(C)(C)C)CC(C)(C)C1 N1(C(C(C(C)CNC(=O)Cn2nnc(C3CC3)n2)F)=O)CC=C(C(C)(C)C)CC1 CC(C)C(C(=O)NCCOCCNC(=O)C(C)c1cccs1)c1cccc(Cl)c1 C1(CNC(=O)C=Cc2cccnc2)CCCCCN1C(C1(F)CCOC1)=O N1(C(CCC(C)O)=O)CCCC12CCN(C(c1cc3ncccc3s1)=O)C2 CCC(C)CCCC(=O)NCC1(CC(=O)NCC(O)C(C)C)CC1 C12(NC(Cc3c(C)cco3)=O)CCN(C(c3cnn(CCO)c3N)=O)CC1C2 N1(C(C=C=C(C)C)=O)C2CCC(C2)C1CNC(C1CC(C)(O)C1)=O C1(NC(Cc2cc(C)sc2)=O)CCC(C)N(C(=O)CN2CCOCC2=O)C1 c1(C(=O)NCC(C)N(C)C(c2cc(C3CC3)nc(Cl)c2)=O)c[nH]nc1S(N)(=O)=O c1(OC)ccc2cc(C(=O)N(C)CCNC(C3CCN(C)C3C)=O)ccc2n1 CC1(C2CN(C(=O)CC3COCCN3C(c3ccsc3C#N)=O)CCO2)N=N1 c1(C(=O)NCCC2(O)CCN(C(c3ccc(OC)nc3)=O)C2)c[nH]cc(C)c1=O c1(C(N2CC(C)(NC(c3ccc(=NC)[nH]c3)=O)C2)=O)cnc(O)c([N+](=O)[O-])c1 Cc1cccn2nc(C(N3CCCC(C)(NC(c4ncncc4Cl)=O)C3)=O)cc12 c1(CNCC2N(C(=O)CSc3cccs3)CCOC2)cnc2ccccc2n1 c1(CC)cc(F)ccc1C(N1CCC(O)C(NC(c2cscc2OC)=O)C1)=O CC1Cn2nc(C(N3CCCC(N(C)C(C4CC=CC4)=O)CC3)=O)cc2C(=O)N1 CN1CCN(C(=O)CCCN=[N+]=[N-])CC1CNC(=O)C(C1(O)CCCCC1)(F)F c1(C(N2C(CN(C(c3c(C)con3)=O)C)CC(F)C2)=O)ccc2c(n1)CCC2=O c1(NC(=O)CC2CN(C(C3CC3C(=O)O)=O)C2)nnc(Br)s1 c1(C(N2CC(C)C(NC(=O)CN3CCCNC3=O)C2)=O)cncn(C)c1=O C(=O)(C1CCCc2scnc21)NCCCNC(C1N(C)S(=O)(=O)CC1)=O CCC(CC(=O)NCCCOCCC(=O)NCC(=O)NC(C)C)SC c1(C(C)=O)c(NC(c2sc(NC(=O)CCC3CC3)nc2C)=O)sc2c1CCC2 N1(C(CC2C(C)C(=O)CC2)=O)CC=C(CNC(C2CCC3CC3C2)=O)CC1 N1(C(c2n(C)cc(Cl)c2)=O)CCC(NC(c2ccn(C(F)F)n2)=O)C(C(N)=O)C1 C(=O)(C1=CCCCO1)NS(N)(=O)=O.O=C1CC2C(C(N3CCOC(C(=O)N)C3)=O)C2C1 c1(-n2c(CNC(c3cncs3)C)nnn2)ccccc1OC(F)F CC(c1ccccc1)=CC(=O)NC1CCC1CNC(=O)C(C)(C)C Oc1nc(-c2ccc(OCC3CCCCO3)c(F)c2)cc2nccn12 N1(C(C2(c3cccc(C)c3)CC2)=O)CC(CNC(C23CC2C3)=O)C2(CC2)C1 C1(NC(C(C=C)(C)CC)=O)CN(C(=O)CC2CCCCC23CC3)C2CCCCC12 N1(C(C(CN(C(c2nn(CC)c(C)c2)=O)C)(C)C)=O)CCS(=O)CC1C C1(C(N(CC(C)O)CCNC(C2(F)CCOC2)=O)=O)CCCCCCC1 n1(C(C)C)ncc(C(=O)NCC2(NC(=O)C(c3ccc(Cl)s3)C)CCOC2)c1N N(C(=NCCC(C(F)(F)F)N1CCOCC1)NCc1cccs1)CCC(CC)C c1(C(N2CCC(C)(NC(CN3C(=O)CC(C)(C)O3)=O)C2)=O)cn2ncccc2n1 C1(C(=O)NC2CCC(NC(C3CC=CCO3)=O)C2)(OC)CCCCCC1 N1(C(c2cc(COC)on2)=O)CC2(CC2)CC1CNC(c1c(F)cccc1F)=O C1(N(C(C(=O)NCC)=O)CC)CCCN(C(=O)CCCOc2cccc(Cl)c2)C1 C(=O)(C1=C(C)CCCC1)NC12CC(NC(c3ccc(OC)c(N)c3)=O)(C1)C2 C(=O)(C(C)S(=O)(=O)C(C)C)NCC(C1CCC1)NC(c1cc(C)n(C2CC2)n1)=O N1(C(CC(C)(C)OC)=O)CC(C)C(NC(=O)CC2OCCCC2(C)C)C(C)C1 C1(CNC(COC(C)=O)=O)CCCC1C(=O)NCc1noc(C)n1 c1(OC)ccc(F)cc1S(=O)(=O)N1CC2C(NC(c3cnsn3)=O)C2C1 c1(C(=O)NC2(CO)CCCN(C(C(CC=C)C)=O)C2)cc(F)c(C(C)C)cc1F C=C(C)CCCC=O.CCC(C)(C)N Cc1csc(=O)n1CC(=O)NCC1CN(C(C2CCC(C)CC2)=O)CC1C CN1CC(C(=O)NC(Cc2ccccc2)CCNC(=O)C(C)(C)F)CCC1=O C1(OCCCC)CCC(C)N(N2CCn3ncc(S(C)(=O)=O)c3C2)C1 N1(C(CCC(=C)C)=O)CC(OC)CC(NC(=O)C(c2ccccc2)SC)C1 C1(OC)CC2CC(NC(C3(C(C)C)CCN(C(=O)C(O)CCSC)C3)=O)CC12 C1(O)(CNC(C)=O)CCCN(Cc2cnn(-c3ccc(Br)cc3)c2)C1 c1(C(=O)NC2CCCN(C(C(C)P(C)(C)=O)=O)C2C)nc2ccccn2c1F C(C1CC(C)(C)Oc2ccccc21)NC(=NCC)NCCS(=O)(=O)CC1CCC1 CN1CC(NC(C2(C)C=CCN2C(c2ns[nH]c2=O)=O)=O)C2(CC2)C1 C1(N(CCCCOCC=C)C)CCN(C(=O)CNC(=O)CCCC)CC1 CC(C)C(C(=O)N1CC(CNC(c2ccoc2)=O)C(O)C1)c1ccccc1 c1(C(=O)NC2CC(CNC(=O)C3=CCOC3)C2)cn2c(n1)COCC2 N1(C(C2COCC(C)O2)=O)CC2CC1CN2C(=O)Cn1cccc(O)c1=O N1(C(C(C)=CC=C)=O)CC=CC(C(=O)NC(C2CCC2)C2CC2)C1 c1(SCCNC(c2nnnn2C2CC2)C2(C(F)F)CCC2)cccnc1 N1(C(C(C2CCCO2)NC(C(CC=C)NC(C)=O)=O)=O)CC(CO)C2(CC2)C1 CC(C)C(CO)C(=O)NC1CC(CNC(C2(O)CCOCC2)=O)C1 Cc1cccc(C)c1C(=O)NCC1CCCCN1C(c1cc(O)nn1C)=O C(C(=O)N1CCC(C)(NC(c2cnn(CCO)c2)=O)CC1)(C(C)(C)C)N(C)C C1(NC(C=Cc2occ(C)n2)=O)(CO)CCCN(C(c2ccc(O)c(Cl)n2)=O)C1 C#CCCCCCCC(=O)N1CCN(C(=O)C#CC2CCCOC2)C(C(C)C)C1 Cc1c(C(N2CC=CC2C(=O)N(C)CC2CCC2)=O)ccn1C c1(C(=O)NCCCN(C(=O)CC2CC=CCC2)C)ccsc1Br c1(C(=O)NCC2CN(C(C3CC3(F)F)=O)CCCO2)cc2n(n1)CCCO2 c1(C(N2CC(CC(C(=O)NCCC3(C)CCCO3)F)C2)=O)ccc2c(c1)CCC2 N1(C(C(CN(C)C)(C)C)=O)CC2OCC(NC(=O)CC3COCCN3C)C2C1 c1(C(=O)NCC2N(C(CC)=O)CC=C2)cccc(-c2cnccn2)c1 C1(CC)CCN(C(=O)CC#N)C1CNC(=O)Cc1cc(C)[nH]n1 N#Cc1cccc(NC(C2CN(C(c3c(I)ccnc3Cl)=O)CCN2)=O)c1Cl c1(C(=O)OC(C)(C)C)sccc1NC1CCC1C(=O)NS(C)(=O)=O c1(NC(C2CCN(Cc3cccc(C)c3)C2)=O)cccc2nccn12 O=C(C1=NOC(c2ccccc2)C1)NC1CCN(C(c2ncccn2)=O)CC1O CC(c1ccco1)=CC(=O)Oc1ccc(-c2nnc(Br)o2)cc1 C(=O)(C(C)CC(C)C(C)=O)NC(C(N1CCC(OCCC)CC1)=O)C1CCC1 C1(C(C(=O)NCC)N(C)CC2CCSCC2)C(C)(C)C1(C)C CCCC(C)C(=O)NCCCN(C(=O)CC1CCCCC1C)C(C)C C=CC(C)C(=O)N(C)CCN(C(=O)CC1CC(F)C1)C c1(C(=O)NC(C2CN(C(=O)C(C)(C)CC3CC3)C2)C)ncn2ccccc12 S(=O)(=O)(c1ccc(F)cc1)N1C(C(=O)Nc2cc(CC)nc(Cl)c2)CC(F)C1 N1(C(C(N2CC(C)C2)C)=O)CCC(C(=O)NCC(C)(O)C2(C)CC2)C(C)(C)C1 n1(CC)cc(C(=O)NCCCCN(C)C(c2coc(C)c2)=O)c(C)n1 c1(CC)cc(C(=O)NCC(=O)NCC(=O)NCc2cscn2)no1 N1(C(c2ccc(SC)o2)=O)CC2(CCCCN2C(c2nccn2C)=O)C1 C1(O)(C(C)NC(C(C=CCCC)O)=O)CCN(C(=O)CCc2cn[nH]c2)C1 c1(CC)ccnc(C(=O)NCC2CCCC(CNC(c3nnsc3C)=O)C2)c1 CCCCC(O)CC(=O)NC(C)C(C)(C)C(=O)NCC1(C)CC1(C)C C1(C(=O)Nc2cscc2C(N)=O)(NC(=O)OC(C)(C)C)CC1(C)C c1(C(=O)NCC2N(C(CC=CC)=O)CCC2C2CC2)ncn2cc(Cl)ccc12 c1(CC)c(Cl)nc(C)[nH]c1=NCCCN(C(=O)C(C)(C)c1cncnc1)C1CC1 C=CCCCC(C(=O)NCCC(C)(O)CC)NC(c1cc(C)c(C)s1)=O C12(C(N(CCNC(C(C(C)C)O)=O)C)=O)CCC(=O)N1CCS2 C1(NC(C2(CC)CCOCC2)=O)CCN(c2nc(C3CC3)ns2)C(C)C1 N1(C(COCC(=O)NC)=O)CC(CNC(c2cccc(O)n2)=O)OC(C)(C)C1 C1(CNC(CCOCCCOC)=O)CN(C(c2cc(C)nn2C)=O)CCO1 c1(C(=O)NCC(C2CC=CCC2)(C)O)sc(Br)cc1F C1(CNC(CCc2ncc(C)[nH]2)=O)CN(C(=O)C(C)NC=O)CC(C)(C)C1 C12(NC(c3cnn(CC)n3)=O)CCCC1N(C(=O)C=Cc1ccccn1)CC2 C1(O)(CCNC(C2CCS2(=O)=O)=O)CN(C(c2ccnn2-c2ccccc2)=O)C1 C=C(C)CCCC(=O)N(C)Cc1cn(CC2(F)CCOC2)nn1 CC(CC(=O)NC1(CNC(c2cn(C(F)F)cn2)=O)CCCC1)c1cnn(C)c1 c1(-c2cc(C(=O)NC3C(NC(=O)CC45CCCC4C5)C3)no2)ccc(Cl)cc1 C1(CNC(C2CC(C(=O)OC)C2)=O)CN(C)CCN1C(=O)CC1CCC(=O)NC1 C(=O)(CC(C)CC(=O)NC1CC(N(C(=O)CC(F)(F)Cl)C)C1)OC c1(C(=O)NC(C)CCCNC(=O)C=CC2CCC2)cnc(C(F)F)nc1 Cc1c(Cl)ccnc1C(=O)NCC(C(C)(C)C)NC(C1(C)CC(C)(C)C1)=O N1(C(c2cn(C)nc2)=O)CCN(C(C2CCn3cncc3C2)=O)C2CCCC12 c1(C(=O)NCC(C(C)(C)C)NC(C2CCC3CC2CO3)=O)ncn2c1CCC2 N1(C(CCCC2(C)NC(=O)NC2=O)=O)CC2(CCC(NC(C3CC3F)=O)CC2)C1 c1(C(N2CCC(NC(=O)CCCCC3CC3)C2)=O)ccc2c(=O)cc[nH]c2c1 N1(C(C=CCCC(C)C)=O)CCN(C(c2ccc(=N)[nH]c2)=O)C(C2CCC2)C1 Cc1cc(C(=O)NC2CCCN(C(C3CCC3(C)C)=O)C2)cc(=O)n1C c1(NCC2CCN(C)CC2)ccc(S(=O)(=O)NCCCCC(F)F)cc1C#N N1(C(COC(C)=O)=O)CCCC(C(C)NC(=O)Cc2sc(C)cc2Br)C1 c1(N2CCCN(S(C)(=O)=O)CC2)ncnc2c1ncn2CC(C1CCCO1)O Cc1cc2ncn(CC(=O)NCC3CCN3C(=O)CC3CCCO3)c2cc1C C#CCCCC(C)C(=O)N1CCC1(C)CC(=O)NCC1CC(N(C)C)C1 C(=O)(C(CO)NC(=O)CCOCCCNC(C1CN(C(C)=O)C1)=O)NCC C(=O)(NNC(=O)c1ccc(C(F)F)cc1)C1(C(F)F)CC(=O)C1 C1(C(C)C)CCC(C)CC1CNCc1cn(C)nc1C C1(CC(=O)NCCc2onc(CC)n2)CC(F)CN1C(=O)CC(C)n1cccc1 C1(CC=C)(NC(C2CC(SC)C2)=O)CCN(C(c2cnc(C)s2)=O)C1 N1(C(Cc2nc(C(C)OC)sc2)=O)CC(C)C(C)(CO)C1 N1(CC(=O)NCC(CN(C(c2cnc(C)[nH]2)=O)C)C)C(=O)NC(C)(C2CC2)C1=O C(=O)(CCCCC(=O)NCCN(CCCN(C)C)C(=O)CC1(OC)CCC1)NC C1(CCC)C(=O)NCCN1C(=O)C=CCC(C)(C)NC(c1coc(CO)c1)=O c1(NC(C2CC=CCC2)C)ccc(S(=O)(=O)NCCn2cnnn2)cc1Br C1(NC(N)=O)CCN(C(=O)NC2CCN(C(=O)NC3CCC3)CC2)CC1 C#CCCCC(C)C(=O)NC(C)CC1CCN(C(c2[nH]cc(C)c2C)=O)CC1 c1(C(N2C(CNC(C(N3CC(C)C3)C)=O)CCC2)=O)ccc(SC(F)(F)F)cc1 C(CCNC(=O)CC(C)(F)F)(C(=O)NCCC1COC(C)(C)C1)OC Cc1cc(C(c2nnnn2C2COC2)NCCc2ccnn2C)ccc1Cl N1(C(C(C=C)(F)F)=O)CC(O)(C2(CNC(=O)CN3CCC(OC)C3)CC2)C1 C1(C(=O)NC2(CO)CN(C(C(C)(C)C3CCC3)=O)C2)CCCC2(CCCCC2)C1 Cc1scnc1C(=O)N(C)CCOCCNC(c1cnn(-c2ccccc2)c1)=O N1(C(CCCSC)=O)CC(CNC(=O)CN2CC3C=CC2C3)C(C)C1 CC(C)C(C#N)C(=O)N1CCOCC(NC(=O)CCCOc2cccnc2)C1 c1(OC)ncc(C(N2CC3CC3(N(C(=O)CN3CCOCC3)CCO)C2)=O)cn1 c1(C(=O)NCC(CCCC)NC(=O)COC2CCC2)cc2c(cnn2C)nc1C N1(C(CN2CC(CC)C2)=O)CCN(C(=O)CC2(COC)CC2)CC(C)(F)C1 C1(CNC(c2c(C)cc(F)s2)=O)CC(C)(C)CN1C(C1CCC(F)(F)CC1)=O c1(C(=O)NC2(CC)CCN(C(c3cscc3C)=O)CC2)cnc2scc(C)n12 C1(CNC(CP(C)(C)=O)=O)(NC(=O)CCOCC(F)(F)F)CC2CCC1C2 C1(CNC(C2C(CNC(c3c(C)ocn3)=O)CCC2)=O)CCC(CO)CC1 N1(C(C#CC(C)C)=O)CC(CO)C2(C1)CN(C(=O)CCCc1cccnc1)C2 CC(C)C(O)C(F)(F)C(=O)NCC1(F)CCCN(C(=O)COC(C)(C)C)C1 c1(C(=O)NC(C2CN(C(C3CC(C)(F)C3)=O)C2)C)cscc1-c1ccccc1 c1(CNC(C(=O)N(C2CCOCC2)CCCC)=O)cnc(-c2ccccc2)s1 c1(C(c2noc(C(C)(C)C)n2)C)nnc(CCCc2cccn2C)o1 C12(CCNC(C=CCN(C)CC)=O)CCC1CN(C(=O)C(C)(C)n1cncn1)C2 c1(CSC)cc(C(=O)NC2CC(NC(C3(C#N)CCOC3)=O)C2)ccc1F c1(C(=O)NCC(C2CCC2)NC(c2cc(Cl)ccc2F)=O)ccccc1[N+](=O)[O-] N1(C(C2CCN2C(C2CCOC2C2CC2)=O)=O)CCc2sccc2C1 N1(C(CC(CNC(C=C(C)c2ccccc2)=O)C)=O)CC2(C1)CC(C)(O)C2 N1(C(C)=O)CCCC(C2CN(C(c3cc(C)c(Br)cc3Cl)=O)C2)C1 C1(C(=O)NCC(=O)NCC#C)(OC)CCN(C(C2CN(C)CCO2)=O)C1 S(=O)(=O)(c1cccc(S(C)(=O)=O)c1)NC1CN(Cc2cc(C)[nH]c2C)CC1C#N N1(C(CN(C)CC)=O)CCCC1C1CCN(C(=O)C(F)=CCOC(C)(C)C)C1 N1(C(CCCOCCOC)=O)CCC(F)CC1C(N1CCCN(C(C)C)CC1)=O c1(CCC(=O)NCCN(C(COC)=O)CCOC)cc(Br)ccc1C C(=O)(C(CC)C(=O)NCCC(C)N(C)C(c1ccc(CCF)cc1)=O)OCC C(C(C(=O)C1CC1)NC(c1cc(CSn2c(CSCC)ccc2)n[nH]1)=O)SCC C(=O)(CN=C(NCC(C)(C)C(F)(F)F)NC1COCC1F)NC(C)C C1(CCNC(c2nnn(CC)c2C)=O)CCN(C(c2ccccc2F)=O)C(C)C1 N1(C(c2cnc(SC)s2)=O)CCC(C(=O)NCc2ccc[n+]([O-])c2)C(O)C1 Cc1ccn2cc(CCNC(=O)C(C(C)C)NS(N)(=O)=O)nc2n1 C(=O)(CCCS(C)(=O)=O)NC(C(C)NC(=O)C=Cc1ccccn1)(C)C C1(NC(=O)CCCn2cccn2)CC2CCC1CN2C(C1C=CCCC1)=O N1(CC2(OC(C)C)CCC2)CC(=O)N(Cc2ccc(Cl)cc2Br)C1=O Cc1cc(F)ncc1-c1cn(C2CC(C(N3CC(c4nncs4)C3)=O)C2)nn1 C1(C(=O)NCCc2c(C)nc[nH]2)CCN(C(C2(CO)CCC2)=O)CC1C C12(C(=O)NCC(C)(C)NC(c3c(CC)c(C)ccc3)=O)CCCCCC1OCC2 c1(C(N(C2CN(C(CC3(C=C)CCC3)=O)C2)C)=O)cc2c(F)cc(Cl)cc2[nH]1 c1(C(=O)NCC2CCC(NC(=O)CCC(F)(F)F)C2)ccc2ccsc2c1 C(=O)(N=c1ccn(-c2ccc(F)cc2C#N)[nH]1)NCC(C1CCCO1)OC N1(C(Cc2cc(C)sc2)=O)CC2CC(NC(=O)Cc3ccnc(F)c3F)C(C2)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(CC)N(C(c2ccn(C3CCC3)n2)=O)CC1 C1(N(C(CCC(C)C)c2ccc(Cl)cc2)C2CC2)COC2(CCC2)C1 CS(=O)CCC(O)C(=O)NCC1(F)CC(CNC(=O)C=CBr)C1 C1(NC(C2CC23CCC3)=O)CCC2(CC1)CN(C(=O)CN1CC3CC3C1)CCO2 C(=O)(C(C)C(F)F)N(CCC(=O)NCCC)C(C)CO c1(N(C(C2CCC(CC)C2)=O)C)ccc(OCC(O)CNC)c(OC)c1 N1(C(C2CCCC(C#N)C2)=O)CC(C(=O)NC2C3CCCC23)C2(CCC2)C1 N(C1CCc2ccccc21)C(C1C(NC(c2c(C)ocn2)=O)CCC1)=O c1(C(=O)NC(Cc2cncs2)CO)cc(C2CCCCC2)cc(Cl)c1O N1(C(COCCOCC#C)=O)CCC(F)(CNC(c2sccc2CC#C)=O)CC1 Cc1cc(Cl)cc(C(N2CCN(C(=O)CC34COC(C)(C3)C4)CC2C)=O)c1O C(c1c(Cl)cccc1Cl)=CC(=O)NCC(CNC(C=CCOC)=O)CO C12(Nc3cccc(C(C)Sc4n(CC)cnn4)c3)CCC(C(=O)OC)(CC1)CC2 N1(C(C(C)NS(C)(=O)=O)=O)CCC(CNC(=O)CCOCC(F)F)C1(C)C c1(CNC(CCN(CC#C)C(C2CCC(C)(CC)O2)=O)=O)ccc(Cl)cc1 CC12CC(C(=O)NCC3CN(C(=O)Cn4cc(CC5CC5)nn4)C3)(C1)C(C)(C)O2 C1(CNC(CCC(=O)OCC)=O)CC2CCC1N(C(=O)C(C)CSC)C2 c1(C(=O)NCC2(O)CCN(C(C3(C)CCCS3)=O)C2)ccc(Br)c(F)c1 c1(CCC(=O)NCc2cn(CCNC(=O)CO)nn2)nc2ccccc2s1 c1(OC)cc(C)cc(C(=O)NCC2COCCN2C(c2sccc2C#N)=O)c1C N1(C(C2(OC)CCCC2)=O)CC(NC(=O)Cn2nnc(=O)[nH]2)C(O)C1 c1(CC)cc(CC(=O)NCC2CC(O)CN2C(=O)C(C(C)C)N(C)C)n(C)n1 C1(C(N2Cc3ccccc3C2)=O)C2CC(CC2F)N1C(c1cnnc(O)c1)=O C(=O)(C(O)CC(C)(C)C)N1CCC(C)(NC(C2CC(=O)CC(C)C2)=O)CC1 N(C1c2cc(C)ccc2CC1C)C(=O)NCc1nnc(COC)s1 C(=O)(CC(C)CCC=C(C)C)N(CCCCCC)CCNC(=O)CCC1(C)CC1 N1(C(CNS(C)(=O)=O)=O)CCC2(CCCCN(C(=O)CNC(N)=O)C2)C1 C=CC(C)C(C)C(=O)NCCN(C1CCCC1)C(=O)C=Cc1sccc1C c1(C(=O)NC2CCC(C)(NC(c3ccc(C)s3)=O)CC2)c[nH]c2cccc(C)c12 N1(C(c2nc(C)oc2C)=O)CC2CCC1C1CN(C(c3ccc(O)nn3)=O)CC21 c1(C(N(CC(CC)NC(c2nnsc2N)=O)C)=O)cc(OC)n[nH]1 C1(C)(C(=O)NCCc2c(C(=O)NCc3c(CC)n[nH]c3)c[nH]n2)CCCOC1 CC(C)C(C)C(=O)NCCCC(C)(C)NC(=O)CN1CCCCC1=O N#CC12CC(C(=O)NCC(c3ccccc3)NC(c3cnn(CCO)c3)=O)(C1)C2 c1(OC)ccnc(N(C2CNCC2C#N)Cc2ccc(OC(C)C(=O)O)cc2)n1 CC1CCC(CC(=O)N(CC2N(C(=O)Cn3cccnc3=O)CCC2)CC)CC1 c1(CNc2c(C)c(NC3CCC(C)CC3C)ncn2)n[nH]c2c1CCCC2 N1(C(COCC(C)C)=O)CCC2C1CCCN2C(=O)CN(C)C(C)C n1(CC(=O)NC2CCC(CNC(C3OCC(C)(C)C3)=O)C2)cnc([N+](=O)[O-])c1 c1(C(=O)NCCCCC(C)NC(C(F)=CC)=O)c(F)cc(Cl)cc1F N1(C(CCCC(CC)CC)=O)CC(=O)NC2CN(C(C3CCS3(=O)=O)=O)CCC12 N1(C(Cc2cc(C)nn2C)=O)CCC(NC(=O)C=CC2CCOCC2)C12CC2 CC(C)(C)CC(O)CC(=O)NC(CC1CC1)NC(=O)CCCc1ccc(Cl)cc1 C1(CC2(C(N(C)C(=O)NC)=O)CC2(F)F)CCCN1C(=O)COC1CCC1 C(C(C)(C(C)C)NC(=O)CC(C)N(C)C)NC(c1cnc(CC(C)C)s1)=O S(=O)(=O)(c1cccc(Br)c1F)N1CCC2CN(C(C=C(C)C)=O)CC2C1 c1(C(N2CCC(CN(C(C(C)CF)=O)C)C2)=O)nc(C2CC2)n2ccccc12 c1(C(N(C2CCN(C(CN(CCC)C)=O)CC2)CC)=O)cc2ccccn2c1 C1(CC(=O)NC(C#C)(C)C2CC2)CC2(C1)CN(C(c1ccnc(OC)n1)=O)C2 N1(C(c2c(CC)nns2)=O)CCC(CNC(=O)C(C)(C)C)(OC)C1 c1(COC(C2CCCCO2)=O)ccc(N2CCCCC2=O)cc1 C1(C(N2CCC(NC(c3cccnc3S)=O)C(F)C2)=O)Cc2cccnc2C1 N1(C(c2ccc(C)o2)=O)CCCC2(C1)CN(C(c1ccc(CO)cc1)=O)CCO2 c1(C(N2CCN(C(CCOC(C)C)=O)CC23CC3)=O)c[nH]c2ccc(O)cc12 C1(=O)CCCN1.C(=O)(C(C)N(CCCNCCCN(C)C)C)N(CC)CC C1(C(C)C)C(=O)N2CC(O)CC2C(=O)N1.C1(CSC)CN(C(=O)OC(C)(C)C)C1 CC(O)CC(=O)NCC(O)CCNC(=O)CC1CCSC1 c1(CC(=O)OC)ccc(NC(C2CSCCN2C(=O)C=Cc2ccsc2)=O)cc1 C=Cc1cncc(C(N2CCOCC2CCNC(c2n[nH]cc2Cl)=O)=O)c1 c1(OC)c(C(=O)NCC2CC(NC(C3CC3C#N)=O)C2)sc(S(N)(=O)=O)c1OC c1(C(=O)NCC(C)CN(C(=O)C(C)(C)C)C)nccc2ccccc12 CCC(C)(CNC(c1cccc(F)c1Br)C)C(C)O CN1CCCCN(C(=O)C(c2ccco2)NC(C2CC23CCC3)=O)CC1 c1(OC)ccc(C(=O)NC2CCCC2NC(c2cc[nH]c(=N)c2)=O)cc1C C(c1ccccc1)=C(OC)C(=O)N(C(C)CNC(=O)CCCN(C)C(C)C)C C1(C(=O)NC2(C)CN(C(C3CC4(CSC4)C3)=O)C2)CC(c2ccccc2)=NO1 c1(C(=O)NCC2CC(F)(CNC(C(CC)SC)=O)C2)cn2cc(C)nc2s1 CC(C)CC(CNC(C1C2CCC1(c1ccccn1)C2)=O)N(C)C N1(C(CCCSC)=O)CCN(C(C2C3COCC23)=O)CC1C C1(C(=O)NC(C#C)C(C)C)(NC(=O)Cc2cncc(C)c2)CCOCC1 C1(CC=C)(NC(=O)CCC(F)F)CCN(C(c2cc(COC)no2)=O)C1 C(=O)(C1CCCc2ccnn21)NCC(CNC(C=CCOC)=O)(C)OC C#CCC(C(=O)NC1(C(=O)NCCC(C)N2CCCC2)CCSC1)C1CC1 C(=O)(CC(F)(F)F)NCCCCNC(C1C(C)C1C)=O N1(CCC(N2CC(OCCNC(C(C3CCC(=O)N3)C)=O)C2)=O)C(=O)CCC1=O N1(C(CCC2CC(NC(CC(CC=C)(C)C)=O)C2)=O)CCC2(CC=CCO2)C1 C1(CNC(=O)OC2CCSCC2)C2CCOC2C12CCCC2 C(CCCCC(=O)NC1CCN(C(c2cc(C)ccc2Cl)=O)CC1CO)=CC CC(C(=O)NC1(C)CCN(C(C2(F)CCC(F)(F)CC2)=O)C1)C1=CCCC1 CCCC(O)(CCC)CC(=O)N1CCCC1Cc1ccc(F)cc1 c1(NC(C2(C)N(Cc3cc(C)nn3C)CC2)=O)cc(F)cc(Br)c1 S(=O)(=O)(c1ccc(NCCCC2CCC2)c(F)c1)NCC(CCCCC)O CC1=C(C(=O)N2CCC(O)(c3cn(Cc4ncon4)nn3)CC2)CCCO1 N1(C(C(C)OCC#C)=O)CCC(C)CC1CNC(=O)CCCOCC C1(C(N2CC(NC(C(C(=O)NC)(C)C)=O)C(C)CC2)=O)CC2(C1)CC1(CCC1)C2 C1(CNC(C(C)Sc2ccc(Cl)cc2)=O)(CF)CC12CCOCC2 C1(CNC(C(CCC)=CCC)=O)CCN(C(c2nnc(O)cc2C)=O)CC1(F)F c1(-c2c(NC(C3=C(C)OCC3)=O)sc3c2CCC3)ccc2nc(O)[nH]c2c1 c1(CNC(C(C2CC2)OC)=O)cccc(NC(=O)C=C(C)Cl)c1 C(CC(=O)N1CCC(N2CCC2)C1)(C(F)F)NC(C=NOC)=O C(=O)(C(O)CCC(C)C)NC1CCN(C(C(CC)=CC)=O)C1C(C)(C)C C1(NC(=O)CCC2CC2)CC2CN(C(c3cccc(CO)n3)=O)CC2C1 C(=O)(CCCCC#Cc1ccccc1)NC(CNC(C(C=C)(C)CC)=O)C1CC1 C12(NC(COC)=O)COCCC1CN(C(c1cc3c(s1)CCSC3)=O)C2 c1(NC(C2N(Cc3cc(C)c(F)cc3)CC2)=O)cc([N+](=O)[O-])cnc1C N12CCCC(O)(CC1)C2.c1(C(C)N(C)C)noc(-c2cccs2)n1 C1(N(C(=O)Cc2cnc[nH]2)C)CCC(NC(C2(c3ccccc3)CC2)=O)C1 N1(C(c2c(CC)c[nH]c2)=O)CC(N(C(=O)CS(=O)(=O)NC(C)(C)C)C)C(C)(C)C1 C(CNC(=O)CNc1ccccc1F)(CC(C)C)NC(C(CSC)C)=O CC1C(NC(c2cccc(OC(F)F)c2)=O)CCCN1C(c1c[nH]nc1F)=O C(C(COC)CC(=O)NCC1CC1C(=O)NCc1ncccc1OC)OC C1(C(N2CC(c3n(C)ncc3)C(NC(=O)C=C(Cl)Cl)C2)=O)COC2COCC12 C#CCC(CC(=O)N(C(CC)CC)C)NC(=O)CCc1ncccn1 c1(C(=O)NCCC2CCCN(c3cc(Cl)ncn3)C2)cccc2ncccc12 c1(CN2CCC3(C(C(=O)NCc4ccccc4O)C3)C2)cc2ccccc2[nH]1 C1(C(N(C(C(=O)NCC(n2cccn2)C)C)C)=O)CN2CCC1C2 Cc1ccc(CO)c(NC(C2CCCC2NC(=O)C=Cc2ccccc2)=O)c1 N1(CCc2cn(C3CC(C(=O)NCC4(C)CC4(Cl)Cl)C3)nn2)CCC(O)CC1 c1(C(N2C(C(=O)Nc3cccc(CF)c3)CC(C)C2)=O)ccc(Br)cc1I C(=O)(C1CCCn2ccnc21)N1CCOCC(NC(C(NOC)=O)=O)C1 N1(C(C2CN(C(C)C)C2)=O)CCC(C)(CNC(c2ccc(CSC(F)F)o2)=O)C1 c1(C(N(C2CCCN(C(C3CCS(=O)CC3)=O)C2)C)=O)c[nH]c2nc(Cl)ccc12 c1(C(=O)OCC)ncc(F)cc1NC(=O)Nc1cccc(NS(=O)(=O)C(C)C)c1 c1(C(=O)NCC2(CO)CCN(C(c3c(CC)ncs3)=O)C2)c(F)cc(O)cc1F N1(C(c2cc(C)n(C)c2)=O)CC2CCN(C(c3cc[nH]c(=N)c3Cl)=O)C2C1 Cc1cc(C(=O)NC(CNC(C2CCCC2(F)F)=O)C(C)C)c(N)c(F)c1 C#CC1CCCC(CNC(=O)C(CC2CCCC2)NC(c2cc(Cl)ns2)=O)C1 c1(N2CCC(c3cccc(OC(F)(F)F)c3)C2)c(Cl)cnc2[nH]nnc12 N1(C(c2c(N)non2)=O)CC2(C1)CN(C(C1CC1(Br)Br)=O)C2 N1(C(COCCC=C)=O)CCN(C(c2cocn2)=O)C(C)C1C CC1(C(=O)Nc2ccc3nc[nH]c3c2)CC12CCN(CCC(=O)NC1CC1)CC2 CCCC(O)C(=O)NCC(C1CC1)NC(c1[nH]ccc1-c1ccccc1)=O C=CCC(C(=O)NC(c1cnn(C)c1)C(=O)N1CC(CC)C1)OC Cc1cc(C)c(C(N2CCCC(C3CCCN3C(=O)C(C)(C)CF)C2)=O)[nH]1 c1(C(F)CC2CCCCC2)nc(-c2ccsc2)nn1C12CC(C1)C2 c1(CN(C(c2cccc(CO)c2)C(=O)NCCCCCC)C)cc(Br)ccc1F C(=O)(CC1=Cc2ccccc2C1)NCCCC(CCC)NC(=O)C#CC(C)(C)O C(=O)(C(C)CC(N)=O)NCC1C(C)CCN1C(c1cc(CN(C)C)on1)=O C1(CC(=O)N(CC(=O)NC(CC=C)CO)CCOC)CCCC(=O)C1 Cc1cc(C(N2CCCC2C2CCN(C(=O)CSc3nc[nH]n3)C2)=O)cc(O)n1 C(=O)(C(C)(C)C(=O)N(C)CCN1CCN(C(C2CC2Cl)=O)CC1)OCC C(c1ccc(F)c(Cl)c1)=CC(N1C(C)(NC(=O)OC(C)(C)C)CC1)=O.CN1CC1 C(=O)(CC(CN(C)C)C(F)(F)F)NCC(C)(C)OCCNC(C(CCCC)C)=O C1(c2cn(C3CN(C(C4COC(C)C4)=O)C3)nn2)(OC)CCOC1 C1(C(N(C)CCOCCN(C)C(C2(C)CCC(=O)N2)=O)=O)CCC(C)(F)CC1 Cc1cc(C)c(C(=O)N(CCNC(c2cc(Br)c(C)cn2)=O)C2CC2)c(C)c1 c1(C(=O)NCC2(NC(C(C3CCOC3)OC)=O)CCC2)cnc[nH]c1=N Cc1cc(CC(N2CC(OCC(=O)NCC3(O)CCN(C)C3)C2)=O)nn1C c1(C(=O)NCC(C)CNC(c2c[nH]nc2C(C)(F)F)=O)cc(Cl)ccn1 N1(C(COCCC=C)=O)CCN(C)CC1CNC(=O)CNC(=O)CCC c1(C(N2CC(COC)(NC(=O)CC=C(C)C)C2)=O)cccn2c(C)nnc12 N1(C(CSc2c(C)n[nH]c2C)=O)CCC(C)CC1CNC(=O)C(F)CC1CCC1 C1(CNC(COCCOCC#C)=O)COCCN1C(=O)C(C)SC CCC(C)C(O)CC(=O)NCC1(C(=O)NCC(C)C2CC2)CCCCC1 c1(C(=O)NC2CC(C)(c3ccccc3)C2)cc(CNC(C2CC2F)=O)cc(F)c1 C(C)(CC(F)(F)F)NC(c1n(CC=C)nnn1)c1ccncc1 C1(C(=O)OC)OC(C(=O)OCCCc2nocc2C)CC1C C(=O)(CCC1=NNC(=O)CC1)NC1C(NC(CNC(=O)OCC=C)=O)COCC1 C(CCC(C)CC(=O)N1CCC(=CC(=O)NCC(C)C)CC1)=C(C)C c1(C(=O)NC2CCC(NC(C3(F)CC=CCC3)=O)C2)cc2c(cn1)OCCO2 c1(NC(C(Cc2cccc(OCC)c2)N)=O)cc(C)c(I)cc1C#N Cc1cc(Cl)ncc1NC(C1COC(CNC(c2cc[nH]c2)=O)C1)=O C1(C(=O)NC2(CC=C)CN(C(=O)CCC(=O)N(C)C(C)C)C2)CCCS1(=O)=O C1(CNC(Cc2c(C)ccnc2)=O)CN(C(=O)C(F)C(C)(C)O)CC12CC2 Cc1nn(C)cc1CNC(=O)C(c1ccccc1)n1cccc1 C(=O)(CS(=O)(=O)CC(=O)N(C1CN(C(C2COCC(C)(C)O2)=O)C1)C)OC N1(C(C(CC=C)OC)=O)CC(NC(C2CC(=O)N(C)C2)=O)C2(CCCC2)C1 C1(C(C)(C)C)(CNC(CCC2C(C)(C)C2)=O)CCN(C(=O)CCn2cccn2)C1 Cc1ncnc(C)c1C(=O)NCC12CC(NC(c3snc(Cl)c3Cl)=O)(CO1)C2 C#CCC(C(=O)NCC(F)CO)NC(=O)Cc1cnnn1C C1(CNC(CC=CCC)=O)C(O)C(O)CN1C(c1sc(C)cc1Br)=O C(C(=O)Nn1cccn1)C1CC(C)N(C(c2ccc(CO)cn2)=O)C1 C(CCC(=O)NC(C)Cn1cc(CC(C)O)nn1)OCC=C c1(CNC(=O)CC23CCCC2C3)ccc(C(F)(F)F)cc1F.C12CC(C1)NC2=O c1(OC)cc([N+](=O)[O-])ccc1C(=O)NCC(C)CNC(C1CC(C(F)F)C1)=O C(=O)(C(O)(CC)c1ccccc1)NCC(CC)NC(C1CC1C)=O c1(C(C(=O)NCC(CC)NC(C2CCC3CC3CC2)=O)C)ccc(F)cc1F c1(NC2CC(OC)C2)ccc(S(=O)(=O)N(c2ccc(OC)nc2)C)c(Cl)c1 c1(C(=O)NCC(CC)N(C)C(C2CCOC2C)=O)ncc[nH]c1=O C(=O)(C1(C)CCc2ccccc21)Nc1c(C)cc(NC(c2nocc2Cl)=O)cc1 Cc1cc(C(=O)NC(C)CCCNC(c2nsnc2O)=O)ccc1O N1(C(=O)C(C2CC2)C2CC2)CC2(C1)CN(C(C1CC1(F)F)=O)C2 Cc1ncccc1NC(=O)CCN(C(=O)CCCNC(N)=O)CC1CC1 C1(C(=O)NCC2(CNC(C3(O)CCSC3)=O)CCC2)CCn2cnnc2C1 N1(C(CC(CC)NC(=O)CCOC2COC2)=O)CCCC(C)(O)C1 c1(CC)nc(C)c(C(=O)NCCNC(c2cc(Cl)sc2Cl)=O)o1 N1(C(=O)OC(C)(C)C)C=COCC1C(=O)OCCCCC1CCCO1 CC(C)(C)CCCC(=O)NC1CC(NC(C2CCOC(=O)N2)=O)C1 C1(NC(c2ccc(NC)cn2)=O)CN(C(=O)C=Cc2cccs2)C(C)(COC)C1 CCCC(C)(CCC)C(=O)N(C)CC1(O)CCN(C(C2CC2c2cccs2)=O)C1 C(=O)(C(C)(C)CCC(=O)OC)N1CCCC(CNC(CCSCCCC)=O)C1 N1(C(C(C#N)=CC2CC2)=O)CCC(C2CCCN(C(C3Cc4cscc4C3)=O)C2)C1 c1(C(N2C(C)CC(NC(c3cc([N+](=O)[O-])n[nH]3)=O)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(CNC(C(=O)Nc2ccc(CCC)cc2)=O)cccc(F)c1F CCCC(C(=O)N1CCOCC(NC(c2cnc(OC)c(C)c2)=O)C1)C(C)C CCCCCCCC(=O)NCC(CC(=O)N(c1cc(C)cc(C)c1)C)C1CCC1 C1(F)(C(=O)NCC(COCC)O)CCN(C(c2occc2CC)=O)C1 CCC(CNC(c1ncn(C)c1C)=O)(CC)NC(=O)CC1C=NN(C)C1=O C1(O)(CCNC(C2CN(C)C2)=O)CCN(C(C2CCCC(C)CC2)=O)CC1 C1(C(=O)NC(CCCNC(C=NOC)=O)C)CC(O)c2ccccc2O1 CCCCC(CC)C(=O)N1CCCN(C(c2cnc(OC)s2)=O)CC1 CC(CCNC(=O)CCC1CCCCN1C(=O)Cc1ccn(C)c1)C(F)F C(C(F)(C(=O)N1CCN(CCO)C(C)C1)C(C)C)NC(CNC(C)=O)=O C(=O)(C1=CCC2CCC1N2C(c1coc(C(N)=O)c1)=O)NCC1N(CC)CCC1 n1(CC(=O)NC2CC(C)(CNC(C3CCN(CC)CC3)=O)C2)cccc(O)c1=O c1(C(N)=O)cccc2c1CCN(c1ccnc(-c3nccs3)n1)C2 c1(C(=O)NCC2OCCC(NC(c3ccncc3F)=O)C2)ccc2c(n1)CCC2 c1(NC(=O)NCC(=C)F)ccc(OCCC)c(OC)c1 c1(C(N2CCC(n3cc(CCCC=C)nn3)C(O)C2)=O)cccc2occc12 c1(COC)csc(CNC(c2ncoc2-c2ccccc2)=O)c1 N1(C(c2scnc2C)C(=O)NCCOC)CCCC(C)(C(=O)OC)C1.C(C)(=O)O C1(C(=O)NCC(CC#C)(C)C)CCCCCN1C(=O)CCc1cnc(C)o1 Cc1sc(O)nc1C(=O)NC(C)CN(C)C(c1cncc(-n2cccn2)n1)=O c1(C(N2CCC(Cl)=C(Cl)C2)C(=O)NCCCCCC)nnc2n1CCCCC2 c1(CC)cc(OC)ccc1C(N1CCCC1C(C)NC(=O)C1=CCC1)=O CC1CN(C(=O)CNC(C2CC2C)=O)CCC1C(=O)O CC1(C)CCCCC1C(=O)NC1CC(C(=O)NOCC2CCC2)C1 c1(CC)ccccc1-n1cc(-c2cc(C)c(C)s2)nn1 N1(C(CC(CC)(C)C)=O)CC2(CC(NC(=O)C(c3ccccc3)F)CO2)C1 N1(C(=O)C2=COCCO2)CCCC12CCN(C(C1(Br)CC1(F)F)=O)C2 c1(C(=O)NCCC2C(C)CCCN2C(=O)CCCC2CC2)ccc(C#N)cc1F C1(C(=O)NCCS(=O)(=O)NC)CCCN(C(=O)CCCC2CC2)CC1 CC(=O)CCN=C(NCc1cnccc1Cl)NC1Cc2ccccc21 c1(C(=O)O)cccc(C2(F)CC2C(=O)NC(c2cccc(F)c2)C(F)F)c1 N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CCCC(NC(=O)CCOCCC)C(F)C1 c1(OC)c(COC(C2CCN(C(=O)CC3(CN)CCCC3)C2)=O)cccc1F N1(C(C2C(C#N)C2)=O)Cc2ccnn2CC(NC(c2cc(C(F)(F)F)c[nH]2)=O)C1 N1(C(c2cc(C)cc(F)c2)=O)CCC(NC(c2cnsn2)=O)CC(C)(C)C1 C(=O)(C1CCCc2cccnc21)NC(CC)(CNC(=O)C1=COCCO1)CC c1(C2C(C(=O)NCCS(=O)Nc3ccc(F)c(F)c3F)C2)ccc(F)c(F)c1F C(=O)(CS(=O)(=O)CC(C)C)NC1CN(C(CC2N(CC)CCC2)=O)C1 C(Cn1ccnc1)(C(F)(F)F)N(CCCC)CC.c1(CO)ccccc1OC C#Cc1ccc(C(=O)NC2CC(CNC(c3coc(C)c3)=O)C2(C)C)cn1 N1(C(C2CCCC(NC(CCSCC)=O)C2)=O)CCC2OCCC2C1 c1(C(=O)NC(CC)CNC(C2(C)CCOC(C)C2)=O)cc(C)c(OC)c(C)c1 C1(NC(CNC(C)=O)=O)CN(C(c2cc3c(F)cccc3s2)=O)C2(CCCC2)C1 C1(C)(CNC(COCCCOC)=O)CCN(C(=O)CCc2cncs2)C1 C1(CNC(=O)NCC2(C(C)(F)F)CCC2)C2CC3C(C2)C13 CS(=O)(=O)C(CNC(C1C2CC3C(C2)C13)=O)CNC(C1(C(F)F)CCCCC1)=O c1(CCC(=O)NC(C(=O)NCC(C=C)O)c2cccs2)cc(C)[nH]n1 N1(C(C2(CC#C)CCCC2)=O)CCN(C(C2OCC2(C)C)=O)C(C2CC2)C1 N1(C(C(=O)Nc2cccc(COCC(F)(F)F)c2)=O)CCC2=C(COC2=O)C1 C1(OC)CC(CNC(=O)CSc2cccs2)N(C(=O)CCOCCN(C)C)C1 C(C(C)C(=O)N1CCC(CCNC(c2cc(C(F)(F)C(F)(F)F)on2)=O)C1)SC CON1CC(C(N2CCC(C)(CNC(=O)CCSc3ccccc3)C2)=O)CC1=O CCCCC(C)C(=O)NCC(C)(C)CN(C(c1cn(C)c(C)n1)=O)CC C1(CN(C(CC(C)OC)=O)C)CN(C(c2cc(N(C)C)ccn2)=O)CCO1 c1(COC)ccc(C(=O)NC(C)C(C)NC(C2(CC(=O)OC)CC2)=O)s1 N1(C(C(=O)NC2CCCN(S(C)(=O)=O)C2)=O)CCCC2NCCC12.C1(=O)CN1C N1(C(c2nn(CC)nc2C)=O)CC(C)OC2(CCN(C(=O)CCS(C)(=O)=O)C2)C1 N1(C(CC)=O)CC2(CC(C(=O)Nc3csc(C)c3)CO2)C1 C1(NC(C2CCC(CNC(c3cc(CC)[nH]n3)=O)O2)=O)CCCC(CO)C1 c1(OC)c(Cl)cc(C(=O)N(CC(C)N(C)C(c2cnc(C)cn2)=O)C)cc1Cl CCC(CCCC(=O)N1CCSC(C)CC1)NC(=O)Cc1n[nH]c(C)n1 N1(C(C=C(CC)CC)=O)CCCN(C(c2cc(C(N)=O)cn2C)=O)C(C)C1 c1(C(N2CCC(CNC(C(c3cccs3)SC)=O)CC2)=O)cc(F)ccc1N N1(C(C2CCC(C)CC2)C(=O)NC2CC2)CC=CCC2(CCOCC2)C1 N1(C(c2cc(C)no2)C)CCC(C)C(NC(C2(C(F)F)CCC2)=O)C1 C=CCCCCCC(=O)N1CCCC(C)(C)C1CNC(=O)C(CC)C(C)(F)F N1(C(CN(CCC)C)=O)CCCCCC1C(N1CC(O)C(O)C1)=O N1(C(C(C2CN(C(CCCNC(=O)OC)=O)C2)O)=O)CCC(O)C(F)C1 C(=O)(N1CCC(C(=O)N(C)CCO)O1)C1ON=C(C)C1 C1(CN2CC(C(=O)Nc3ccc4occc4c3)C2)COc2ccccc2O1 c1(C(=O)NC2CC(CCNC(C3(C)CC=CCO3)=O)C2)cncc(S(C)(=O)=O)c1 c1(NC(C)=O)cnc(C)c(C(N2CC(C)C(C)(NCC(=O)C3CC3)C2)=O)c1 Cc1cc(F)ncc1CNC(=O)CC1CC2(CC2)CN1C(=O)CSCCC#N C1(C(=O)NC(c2ccccn2)COC)(NC(C2CCO2)=O)CCSC1 C(=O)(CCC(=O)N1CCC(=CCNC(C2(C)CC2(F)Cl)=O)CC1)OC C1(OC)(NC(=O)C(C)COC)CCN(C(=O)COCCC2CCCC2)C1 N1(C(CC(n2c(C)cc(C)n2)C)=O)CCOCC(NC(=O)COC2CCC2)C1 CCC(CCC(=O)N1CC(CN=[N+]=[N-])C1)NC(C1CCCCN1C)=O C1(CC=C)(NC(C23CCC(C2)OC3)=O)CCN(C(=O)C(C)NS(C)(=O)=O)CC1 c1(C(=O)Nc2ccc(SC)cc2)cc2cc(C(=O)N=c3cc(C)[nH][nH]3)ccc2[nH]1 CC(C)C(C(C)C)C(C(=O)NCc1ccc(F)cc1)N(C1CC1C)C CC1CCC(=CC(=O)NCC2C3CN(C(c4ncoc4Br)=O)CC23)CC1 c1(CC)occ(C)c1C(=O)NC1CN(C(c2ccc(OCF)cc2)=O)CC1C N1(C(C(CCC)N(C)C)=O)CCN(C)CC1CNC(=O)C(F)CC1CCCCC1 C1(CC)C(=O)N(C)CCN1C(=O)C(CC(F)F)N(C(=O)COCC(F)F)C C#Cc1cnc(C(=O)NCC2CC(F)CN2C(=O)CC2CNC(=O)O2)c(C)c1 c1(CC)nnc(CN(CCCNC(=O)CCOCC(F)F)CC)o1 CC1C(C(=O)O)CC2CCC1N2.c12ccc(cc1)CNC2=O.c12noc(n1)C2 NC1(C(=O)NCC2(Cl)CC23CCC3)CC2(CCOCC2)C1 N1(C(C=CC)=O)CC(NC(=O)C=CC2CCOCC2)CC(O)C1 CC(C)C(C(=O)N1CCCC(C(C)NC(C2SCCS2)=O)C1)c1cccnc1 Cc1oc(C(=O)NC(C)(CNC(=O)C(C)CO)CO)cc1Br CC1CN(C(C2CC23CC(O)C3)=O)CC1(C)CNC(c1ccc(F)cc1)=O N1(C(C(C(C)C)C#N)=O)CCCC(C)(C)C1C(N1CCCC1CN(C)C)=O N1(C(C(C)OCOC)=O)CC(NC(c2nc(OC)c(C)s2)=O)C(C)C1 n1(C2C(C)C2)c(N2CCCC(C(=O)NC3CC3)C2)nnc1-c1ccc(Cl)nc1 c1(-c2n(C)nc(-c3ccc(C(C)(C)C)cc3)n2)cnn2ccc(O)nc12 C1(NC(c2ccc(C)o2)=O)CC2CC1CN(C(=O)C(C)(C)C1CCCCO1)C2 Cc1nc(NCCCc2nc3ccccc3[nH]2)cc(=NCC(C)CC(F)(F)F)[nH]1 N1(C(C2CC(NC(C3CN(C(=O)NC)C3)=O)C2(C)C)=O)CC(COC)C2(CC2)C1 c1(NC(C)=O)cc(C(N2C(C(=O)NCC3(O)CCC3)CC3CC23)=O)ccc1F Cc1cc(O)ccc1CNC(=O)C(C)N(C)C(c1cc[nH]c1)=O c1(C(=O)NCc2nccc(C(=O)NC(CCC)CCO)c2)cc(N)cc(F)c1 c1(C(=O)NCCC(C)NC(Cc2cnc(C)[nH]2)=O)cc(N)c(OC(F)F)cc1F C1(C(=O)NCC=CCNC(C=CC2(C)COC2)=O)NC(=O)CC1C(F)(F)F N1(C(C(C)=C2CC2)=O)CC(NC(C23COC(CF)(C2)C3)=O)CC1C CC(C)C(O)C(=O)NCCOC1CCN(C(=O)CC2CC(N(C)C)C2)CC1 C1(C)(NC(CN(C2CCC2)C(c2cnc(CC)nc2)=O)=O)CC(C)(C)OC1=O Cc1nn(C)c(Cl)c1COC(C1CCC(O)CN1C(=O)Nc1ccccc1)=O C1(CC(=O)NCCN(C(=O)C=CC2CCCO2)C(C)C)CC2(CCC2)CO1 CC(C)CC(C(=O)NCCc1nncs1)NC(C1C2CCCC12)=O CC1CCCN(C(=O)C2=NOC(C)C2)C1CNC(c1ccc(N)c(Cl)c1)=O C1(NC(CCC2COC(C)(C)O2)=O)COCCN(C(C2CC(CC3CC3)C2)=O)C1 Cc1cn2c(n1)C(C(=O)Nc1nccc3ncccc13)CCC2 c1(N2CC=CC(NC(c3c(C)nc(O)nc3C)=O)C2)nc(Cl)nc2cnn(C)c12 N1(C(c2nnn(CC)c2C)=O)CC(F)(F)CC1CNC(=O)CS(=O)(=O)CC C1(C(=O)NCc2cnn(CC)c2C)CC2CC1CN(C(=O)CC(F)(F)F)C2 C(=O)(C(C)(CC)CCC(C)C)NC1CC2(CC(CNC(C(C=C)O)=O)C2)C1 c1(C(N2CCN(C(C(C(CC)C)OC)=O)CC(O)C2)=O)nc2nccc(C)n2n1 C1(NC(C2ON=C(C)C2)=O)CCN(C(=O)COc2ccccc2)CC1C c1(OC)ccccc1C=CC(=O)NC(C)CCCCNC(C1CCCOCC1)=O c1(C(N2CCC(C)(CCNC(C3CC3C#N)=O)C2)=O)ccc2c(c1)COC2 c1(C(N2CC(CNC(CSC(C)C)=O)C3C2C3)=O)cc(Cl)cc(Cl)c1N C1(NC(c2nnc(C(C)(C)C)s2)=O)CCC2CCN(C(C3CSCCS3)=O)C1C2 C(=O)(C(=O)N=S(C)(C)=O)NCC1(NC(C(NOC)=O)=O)CCCCC1C c1(C(=O)NC(C2CCCCN2C(=O)C(=O)NC2CC2)C)cnc(=NCCF)[nH]c1 C(=O)(CC(CC)C(C)C)NC(CCCCNC(C=CCOC)=O)(C)C C1(C(=O)NCC=CC(=O)NCC2(C(C)C)CC2)CC(=O)CC12CCC2 CCC(C)C(C(=O)N1CCC(C)C(NC(C2CCNC2=O)=O)C1)NC(C)=O Cc1nc(C(=O)NCC(C)(CO)NC(c2ccc([N+](=O)[O-])[nH]2)=O)ccc1[N+](=O)[O-] c1(CCC(=O)NCC(C)CNC(c2cccc(C3CCC3)c2)=O)cncc(F)c1 C1(C(=O)NC2(CO)CN(C(CCNC(C3C(C)C3)=O)=O)C2)CCCCC12CC2(F)F c1(C(N2C(CNC(Cc3ccc(C)nc3)=O)CC2)=O)c[nH]c2nccc-2c1 Cc1nn(C)c(C(=O)NC(CNC(=O)Cc2cnn(C)n2)CC(C)C)c1Cl C(=O)(C1CCCc2ncnn21)NC(C)CCNC(c1cnc(C(F)(F)F)nc1)=O N(C(=NCC(C)C)NCc1ncccc1Cl)CC(NOCC)=O c1(C(=O)NC2C(CC)CN(C(=O)C(Cl)=CCl)CC2)cc2cc(OC)ccc2[nH]1 Cc1cccc2c(C(=O)NC(C)C(C)(C)NC(=O)CC3CC(=O)C3)coc12 c1(C(=O)NCC(CN(C(C2(C(C)C)CCC2)=O)C)C)nnc(O)cc1O C1(F)(CNC(=O)Cc2ccc(F)cc2)CCN(C(C2CC3(CCC3)C2)=O)CC1 c1(C(=O)[N+](CCNC(C(C)OCCC#C)=O)([O-])CC)cc(S(C)(=O)=O)c(OC)cc1C CC1CN2CCCC2CN1C(c1ccc2c(c1)CCC2)C(=O)NC1CCCCC1 C1(C(C)C(=O)NCCCC2CCCC2O)CCN(C(c2cc(O)ncn2)=O)CC1 c1(C(=O)NC(C)(C)CNC(c2ncc(F)cn2)=O)cccc2c1NCCNC2=O N1(C(c2ncc(NC)nc2)=O)CC(C2(NC(C3CC(CN(C)C)C3)=O)CC2)C1 n1(COCCSc2n(C)ccn2)nc(-c2cccc(F)c2)nc1C1CCC(=O)O1 c1(C(COCC2CCOC2)NC(c2n(CC=C)nnn2)CC)cccc(C)n1 Cc1cc(C)c(C(=O)NC2(C)CCN(C(=O)CCC3CCCCO3)C2)s1 C(=O)(CS(N)(=O)=O)N(C1CN(C(=O)CN2CCOCC2)CC1F)C c1(C(N(C(C)C)CCN(C)C(C2CC2F)=O)=O)cnc2c(F)cccc2c1 C1(C(=O)NC(c2ccccc2F)CNC(c2cnns2)=O)CCCNC1=O c1(C(C)=O)ccc(CC(N2CC3(CCC3NC(c3coc(C)n3)=O)C2)=O)c(C)c1 c1(C(N(CC(CC)NC(c2ccccc2Cl)=O)C)=O)cc2n(n1)CCO2 c1(C(N2CC(CNC(C=C(C)C)=O)C(C)C2)=O)ccn2nccc2n1 N1(CCC(=O)OC2COCC2Oc2ccccc2)C(=O)C2CCCCC2C1=O c1(OCCC)cccc(C(N2CCOC(CNC(=O)C(O)C3CC3)C2)=O)c1 c1(C(=O)NCC(CN(C(c2[nH]cc(CC)c2)=O)C)C)cc(C)c2occc2c1 C(=O)(C1CN(C(=O)C(C)=O)Cc2nnn(CC)c21)OCC.C1C(C)(C)O1 c1(C(=O)NCC(C)NC(C(C(C)C)NC(=O)OCC)=O)noc2c(F)cccc12 C1(NC(=O)CCc2cnn[nH]2)CC2CN(C(C3(F)CC=CC3)=O)CC2C1 C12(C(N3CCC(N4CCC(NC(C(F)=CC)=O)CC4)C3)=O)CCC(CC1)OC2 c1(N(C)CCC2CCCCC2)nc2cccnc2c(=NC2CC2C(C)(C)C)[nH]1 C=CCC(C(=O)N(C1CCCN(C(c2csnc2OC)=O)C1)C)OC N1(C(c2cncc(C(C)(C)C)c2)C(=O)NCC)CC(CO)C2(CC2)C1 CCC(CC(=O)NC1CC(CC(N2CC(OC)CC(C)C2)=O)C1)CC(C)C c1(C(N2CC(C)C(NC(c3ccn(C)c3)=O)C2)=O)csc2nnsc12 Cc1cc(C(N2CC3(CCN3C(=O)C(C)n3ccnc3)C2)=O)nnc1C N1(C(CCC(C)(F)F)=O)CCC2(CC1)C(NC(=O)C=Cc1ccsc1)CS2(=O)=O C1(Cn2cc(C3CN(C(C(C)CCO)=O)C3)nn2)CCCCCCC1 N1(C(C2(COC)CCCO2)=O)CC(NC(=O)C(Cl)=CCl)C(n2cccn2)C1 C12(NC(N3CCC(c4cc(OC)ncc4)C(C)C3)=O)CCCC(C)(C1)OC2 c1(C(=O)NC2CC(NC(CSCC=C)=O)C2)sc(CC)nc1C c1(CCC(N2CCCC(N(CCO)Cc3cc[nH]n3)CC2)=O)cc(F)cc(F)c1 C1(CC(=O)Nc2nc(C(C)C)on2)CCCN(C(=O)NCCCN(C)C)C1 C1(CCOCC)(NC(=O)CSC(C)C)CCN(C(c2ccc(C(N)=O)o2)=O)CC1 c1(C(=O)NCC2C(C)(C)N(C(=O)CCC3(O)CCC3)CC2)ccc2ocnc2c1 Cc1c([N+](=O)[O-])c(C(=O)NC2CC3CC2CN(C(=O)CCCN(C)C)C3)nn1C N1(C(CN(C)C(=O)C2CC2)=O)CCN(C(=O)C(F)C2CCC2)CC1 N1(c2n(C)nc(CC(=O)OCC)c2Br)CCCCC2(CNC2)C1 C(=O)(C#CC1CCOCC1)NCC1CCCC(CNC(c2cc(C)ncc2)=O)C1 C(=O)(C(C)(O)CNC(c1cccc(OC(C)(C)C)c1)=O)OC c1(C(N(CC(C)CNC(=O)CCC2CC2(F)F)C)=O)cc(N)c2ccccc2n1 C1(CC(N2CC(O)(CN(C(CN3CC(CC)C3)=O)CC)C2)=O)CC(=O)NC1=O CCCC(C(=O)NCC1(C)CCCN1C(C1CC(N2CC(O)C2)C1)=O)OC C=CCCN=C(NCc1cc(O)ccc1Cl)NCC1CCCC(C(=O)OC)O1 c1(C(=O)NCC(CCNC(C2C(C)CCC2)=O)(C)C)cc2c(s1)C(C)(C)CCC2 C1(NC(C(CCC)N(C)C)=O)CCOC12CCN(c1ncc(C)c(O)n1)CC2 c1(C(=O)NCC2(NC(C3(C(F)F)CC(=C)C3)=O)CC2)ccc(OC(C)C)cc1 N1(C(c2cnc(C)o2)=O)CCOC(CCCNC(=O)CCc2cncnc2O)C1 Cc1ccc2[nH]nc(C(=O)NCCC3CN(C(=O)CC(C)P(C)(C)=O)C3)c2c1 Cc1c(CCC(=O)N2CCC2CNC(C2CCCCCC2)=O)cccc1Br CCCCCCCCC(=O)N(C1CCN(C(=O)CC23COC(C)(C2)C3)CC1C)C C(=O)(CC(C)(C)N(C)C)NCC1C(C(NOCCCC=C)=O)C1 O=C1CC(C(N2CCOCC(C(=O)NOC3CCOC3)C2)=O)NC(=O)N1 c1(C(N2CC(CNC(c3cc(CCOC)on3)=O)C2)=O)cccc(Cl)c1[N+](=O)[O-] N1(C(C2C(CNC(CC(C)(C)C3CC3)=O)CCO2)=O)CCC(C2=NOCC2)C1 N(C(=NCC(F)(F)F)NCCC1COCCO1)C1CC(NC(C)=O)C1 c1(N2CCC(Cc3n(C)ncc3)C2)cc(C#N)ccc1Br C(=O)(C(O)CC(N)=O)NC(CSC)(C)C(=O)NCc1csc(C)n1 C1(NC(C=C(CC)C)=O)CC2CCC1CN(C(c1ncn(C)c1C)=O)C2 C(C(O)CC(=O)N1CC(C)(C#N)C1)NC(Cn1ccc(C)n1)=O c1(OC)cc(C)c(C(N2CCCN(C(=O)C=C(C)C(C)C)C(C)C2)=O)cc1Cl C1(NC(=O)NCC2OCC(C)C2)NC(=O)OC1(C)C c1(OC)ccc(C(=O)NC2CC(F)CN(C(=O)C=CC3CCCC3)C2)nc1N C(c1scnc1C)=CC(=O)NCC(CNC(C=CCOCCOC)=O)CO C(=O)(C(C)(C)S(C)(=O)=O)NCCN(CCCN(C)C)C(c1cccc2c1NCC2)=O C1(NC(=O)CN2CCCC2=O)CC2CC1N(C(=O)CC(O)C1CCCC1)C2 C1(NC(CCCC(=C)C)=O)CCCCN(C(c2cc(O)ccc2Cl)=O)CC1 C1(C(=O)NCC(CNC(c2cc3nccnc3[nH]2)=O)OC)CCC2CC1C2(C)C c1(CC(=O)N(C2C3CN(C(=O)CC4(C)CC4)CC23)C)ccc(F)c(Cl)c1 CC1CN(C(=O)C=C2CCN(C)CC2)CCN(C(C2CC(=O)C23CCCC3)=O)C1 C(N=c1[nH]c2c(c(=NC3CSC3)[nH]1)CSC2)c1ccc(C(C(F)(F)F)(F)F)s1 Cc1nc(C(N2CCC(NC(=O)Cn3ncccc3=O)C(C)C2)=O)ccc1C#N C(=O)(CCCCCCN=[N+]=[N-])N(C)CC1CCN(c2cc(C)ncn2)C1 C1(F)(CNC(C(C)(C)C)=O)CCN(C(C2(Cl)CC2(C)C)=O)CC1 C(=O)(C(F)CC(C)(C)NC(=O)CCOC1CCCC1)NC(c1n(CC)ccn1)C C#CC1CN(C(C2CCN(C(=O)C(C)OCC3CC3)CC2)=O)CCN1C CC1(C)CC=C(C(=O)N2CC(CNC(=O)CNc3ccccc3Br)C2)CC1 C#CCC(CC(=O)N1CCC(C(N)=O)C1)NC(c1oc(C)nc1C)=O N1(C(C(=O)NC(C)C)=O)CC2(C=C(C(=O)NC3CCCC(O)C3)CO2)C1 N1(C(C2(C(C)(C)O)CC2)=O)CC=C(C(=O)NCc2ccccc2O)CC1 c1(C(=O)OCC)sc2ccsc2c1CNC(c1cccc(OC)c1Br)=O Cc1ccc(N(C)C(c2cc(CNC(C3CC34CC4)=O)cs2)=O)c(C)c1 C(=O)(C(C)(O)CNC(=O)NC1CCC(SC2CCS(=O)(=O)C2)CC1)OC CCC(C)CC(C)C(=O)NC1(C)CC(NC(c2cc(Br)n[nH]2)=O)C1 C1(C(=O)NC2(CN(C(=O)CC3(c4ccccc4)CC3)C)CC2)CC2CC1CC2O CC1(C)CCCC(CNC(=NCCC2CCN2C2CCOCC2)NC2CCC2)O1 C(=O)(CC(F)(F)C(C)C)NC1CCN(C(C=C(C)c2ccco2)=O)C12CC2 CCCC(C#N)C(=O)NCC1(CNC(=O)CCc2nnc(C(C)C)o2)CC1 c1(C(N2CC(CC)N(C(c3csc(=NC)[nH]3)=O)CC2)=O)cc(C)c(=O)n(C)c1 c1(C(N(C2CCN(C(c3n(CC)ncc3)=O)CC2)C)=O)c[nH]c2cccc(F)c12 N1(C(CC(=C=C)C)=O)CCC2C(CCN2C(c2ccc(NC)c(F)c2)=O)C1 C(C)(C(=O)NC1CC(CCNC(=O)CCC2(C)CC2)C1)OCCCC CCC(CC)(CCNC(C1(CCOC)CC1)=O)NC(c1ccnc(OC)c1)=O C(=O)(C(C)CO)N(C(C)CNC(=O)CCN(c1ccncc1)C)CC C1(C(C)C)(NC(C2CCCN(C3CCCC3)C2)=O)CN(CCC#N)CCC1O N1(C(c2cnc(CNC(Cc3n(C)ncc3)=O)nc2)=O)CC(C2CCCC2)C1 N1(C(CC(C(C)C)OCC)=O)CCN(C(=O)C(C)CC(C)(F)F)CC12CCC2 C12(C(N(C)CC3CCN(C(C4CN5CCN4CC5)=O)C3)=O)CCC(N=[N+]=[N-])C1C2 Cc1nnc2n1CC(C(N)=O)N(CCC(=O)N(C)Cc1ccncc1)C2 C1(C(N2CC(SC)C(NC(C3CCOC3)=O)C2)=O)CCN(CP(C)(C)=O)CC1 N1(C(C2(CCC)CC2)=O)CCC(C)C(CNC(c2cccc(OCCF)c2)=O)C1 C(=O)(C1=C(c2ccccc2)CCCC1)NCCCCN(C)C(C1CC1Cl)=O c1(C(C)C)cccnc1C(=O)NC1CCCCC1CNC(=O)C(O)C1CCCC1 C1(CNC(C(C)C2CCC2)=O)CN(C)CCN1C(=O)CC1CCC(C)(C)CC1 C1(C(C(=O)O)CNC(=O)C2CC2)C2CCC(C2)N1CCCl.C12CCCCCC1N2 c1(C(N2C3CCC(NC(CC=C)=O)(C3)C2)=O)cc(S(N)(=O)=O)cs1 C1(NC(C(CSC)O)=O)CCC12CN(C(=O)C(c1ccc(F)c(C)c1)=O)C2 N1(C(C(CC)NC(C)=O)=O)CC2(CC(NC(=O)CC3CC3)C2)C1 C=CCC(CC)C(=O)NC1CCN(C(c2snc(Cl)c2Cl)=O)C1CC N1(C(COCC(=C)C)=O)CCC(C2CCN(C(c3cc(CO)[nH]n3)=O)CC2)CC1 c1(C(N(C)CC2(CNC(C(C(C)C)C#N)=O)CC2)=O)cc(=O)c2ccccc2o1 C#Cc1c[nH]nc1C(=O)NC(C)Cc1ccc(CNC(=O)C(CCC)OC)cc1 Cc1cc(CNC(c2ccccc2N2CC(N)C2)=O)cc(Cl)n1 C1(CC#C)CCN(C(C2(CNC(=O)CNc3ccccn3)CCC2)=O)C1 N1(C(C(CC)F)=O)CCCC(CCCCNC(=O)C(=O)NCCOC)C1 c1(-c2scc(C)n2)nc(CN2CC(C)C2)n(CCC(F)(F)F)n1 CN1CCCC(C(=O)NCC2(NC(=O)CCOC3CC3)CCCC2)C1 S(=O)(=O)(c1ccc(F)c(Cl)c1)N(CCNC(C1C2CC2C2CC12)=O)C(=O)C1CC1 S(=O)(=O)(c1c[nH]c(=NCCc2cccc(N)c2)cc1C)NC(C(C)(C)OC)C C1(N(Cc2c(C)[nH]c(-c3ccccc3)c2)C2CC2)CCC2(CCCCC2)CC1 c1(C(=O)NCC2CC(NC(=O)CNS(=O)(=O)C3CC3)C2)ccccc1O C(=O)(N=c1[nH][nH]c2ncc(Br)cc12)C1(O)CCN(C(c2cccc(Cl)c2Cl)=O)C1 c1(C(=O)OCC)c(C)c(S(=O)(=O)NC2CCCCCC2C)c(C)n1C Cc1nn(C)c(C)c1C(=O)NCC1(F)CN(C(=O)COC2CCOC2)C1 N1(C(C=C(CC)CC)=O)CCC(NC(=O)C(CSC)OC)C(CO)C1 C1(C(=O)Nc2c(C)nsc2)C2CN(C(=O)CC3CCN(C)CC3)CC12 N1(C(CCSc2n(C)nnn2)=O)CC2(COC(CNC(=O)CS(N)(=O)=O)C2)C1 c1(C(N2CCCC(NC(c3c(C)cns3)=O)C2C)=O)ccnc2c(F)cccc12 C1(CNC(C2CCN(C(c3n(CC)nc(C)c3)=O)C2C)=O)CN(C)CCN1C CC(O)C(F)(F)C(=O)NCC1CN(C(=O)C(N)=O)CCCO1 N1(C(c2cn(CC(=O)OCC)nn2)=O)CC2(CCCC2NC(C2CC2(F)F)=O)C1 c1(C(=O)OC)cc(C(=O)NCC2CCN(C(c3cnccc3Cl)=O)CC2)c(C)o1 c1(NCCN2C(=O)CC(OC)C2)nc2c(c(=NCCC(C)N3CCC3)[nH]1)CCC2 S(=O)(=O)(c1cccc([N+](=O)[O-])c1)N1C(C)(C(=O)NCc2c(C)ccc(Br)c2)CCC1 Cc1cnc2cc(-c3nc(Cc4ccccc4F)nn3CC3CC3C)ccn12 CC1CC(C(=O)NCC2CN(C(=O)C(F)(F)c3cnnn3C)C2)CC(C)O1 c1(CNC(c2nc(COC)sc2)c2nnnn2CC2CC2)cc(C)nn1C Cn1nccc1CNC(=O)CCC1CC(NC(=O)C=CC(=O)N(C)C)C1 c1(NC(c2ccc(C)s2)C)nccc(=NCC(F)C2CCC2)[nH]1 c1(CC(=O)NCC2N(C(Cc3cc(CC)no3)=O)CC2)cccc(OC)c1Cl C=CCC(C)(C)C(=O)N(C)CCN(C)C(C1(N2CCOC2=O)CC1)=O Cn1ncc(C(N2CC(NC(=O)COCc3nc[nH]n3)C2)=O)n1 C1(C(N2CCC(NC(CCc3cc(C)on3)=O)CC2C)=O)CCCC2C1C2(F)F c1(C(=O)NCC(C)N(C(CC2(CCC#C)OCCO2)=O)C)cccnc1C1CC1 C1(C(=O)NC2CC(CCC(=O)Nc3c(C)noc3C(C)C)C2)NC(=O)OC1(C)C C1(C(=O)NC(CNC(c2c(O)nc(C)c(C)n2)=O)CO)CCc2cnn(C)c2C1 c1(NC2(CNC(C(C=C)O)=O)CCOCC2)ncnc2c(OC)cccc12 C1(C2(NC(c3nc(CC)oc3)=O)CC2)CCCCN1CC1(CN=[N+]=[N-])CC=CC1 Cc1nc(CCC(=O)NCCC2(O)CN(C(=O)OC(C)(C)C)C2)oc1C c1(C(c2n(CC)nnn2)NC2COC2)cccc(C)c1COC FC1COc2ccccc2C1NCC1CC2(CC2)C1 c1(CN(C(CN2CCC(C)(OC)C2)=O)C)ccc(C(F)(F)F)cc1C C1(CCNC(CCOC)=O)(C(=O)NCC2(N(C)C)CCCC2)CCCC1 C1(CCNC(C(C)C)=O)CC(F)(F)CN1C(=O)C=Cc1ccnn1C C(=O)(CCC(C)(F)F)NC1C(OC)CN(C(c2cc(C3CCOCC3)no2)=O)C1 C1(C(N2C(C(OC)OC)CCC2)=O)CC(=O)N(C)C1c1cccc(F)c1 C(=O)(C(C)(C)C(C)(F)F)N1C(CNC(CNC(CCC)=O)=O)CCC1 c1(C(N2C(CCCNC(C3CCC4CC34)=O)CCC2)=O)cnc2[nH]ccc2n1 c1(NC(N2C(C)COCC2)=O)ccc(Br)c2cccnc12 S(=O)(=O)(CCC(=O)NCC1=CCCN(C(c2[nH]nnc2C2CC2)=O)C1)NC C(=O)(C(C)(C)CC(=O)OC)NC1C(NC(C2C(C=C)C2)=O)CCC1 c1(C(N2CC(NC(C(c3ccccc3)C)=O)C(C)C2)=O)cc(Cl)nc(Cl)c1 c1(OC)ccc2nccc(C(=O)NC3(CO)CCN(C(c4cocn4)=O)C3)c2n1 C1(NC(CCP(C)(C)=O)=O)CCSC12CN(C(=O)CCc1ccc(N)cn1)C2 c1(CC(=O)NC2CC(C)(NC(=O)CC(=O)N3CCOCC3)C2)cc(F)ccc1Cl Cc1cc(C(=O)NCC2(C)CN(C(=O)C(N)=O)C(C)(C)C2)c2c(O)nn(C)c2n1 c1(OC)ccc(O)cc1-c1ccc(C(=O)NCCOc2ccc(Br)cc2)nn1 c1(C(N(C2CCN(C(CC=CC=C)=O)CC2C)C)=O)ccn2cc(C)nc2c1 c1(C(N(C)CC2CCCN(C(c3ccccc3)=O)C2)=O)sc2ncccc2c1Cl Cc1cnccc1CC(=O)NCC1(O)CCN(C(C2CC2C(=O)NCCO)=O)C1 C1(C(=O)NCC2C(NC(c3c(CCC)n[nH]c3)=O)C2)CCOC2(CCC2)C1 CC(C)CC(O)CC(=O)NC1CCCCC1C(=O)NC1CCCC1(C)C C=CC1CN(C(=O)C(C)OC(C)(C)C)CC1NC(c1cccc(C)c1Cl)=O N1(C(CC(C)OC)=O)CCN(C2CCN(C(C3CCCOC3)=O)CC2)CC1 C1(C(=O)O)(NC(c2c(NC)ccc(F)c2)=O)CCc2c(F)cccc21 C1(C(N2CC(C)(NC(C3CCN(C(CC)=O)C3)=O)C2)=O)CCCC(N(C)CC)C1 C1(NC(C2(NC(C(CC3CCC3)NC(C)=O)=O)CCSC2)=O)C2CCC(C2)C1CO N1(C(Cc2c(C)scc2)=O)CCC(C2(NC(c3noc4ncccc34)=O)CC2)C1 C1(NC(c2c(CCC)nco2)=O)CC(CC(=O)NCC2CC(F)C(=O)N2)C1(C)C N(C1CCSc2ccc(Cl)cc21)C(C(c1cccc(OC)c1)F)=O c1(C(=O)NC2CCN(C(COCCCOC)=O)CC2OC)ccc2sccc2c1 C=Cn1ncc(C(=O)N(CC(C)C(=O)NC(CCC)C2CCCC2)C)c1N c1(OC)ccc(C(=O)NCCCCNC(=O)CCCSc2ccccc2)s1 CC1CCCC=C1C(=O)N1CCCC1(C)CNC(C1CCCN1C)=O CC1CC(NC(=O)Cc2cncs2)CCN1C(=O)C(C)N(C)C C1(CC(C)C)COCC1(c1nnnn1CCCF)N(c1ccccn1)CC CC(CC(=O)NC1(CCNC(=O)C(Cl)=CCl)CCC1)C(C)(C)C Cc1cc(C(=O)NCCC2CCN(C(c3cn(C)nc3Cl)=O)C2)cnn1 Nc1c(C(N2CC3CC3(CNC(C3CC4C=CC3O4)=O)C2)=O)cc(Cl)cc1Cl C1(NC(Cc2c(OCC)c(Cl)ccc2)=O)CCN(S(=O)(=O)N2CCCCC2)CC1 C1(C(=O)NCCCOCCCNC(c2c(C)c[nH]c2)=O)CCN(C)S1(=O)=O C1(C(=O)NC(C(=O)N(C2(C#C)CC2)C)CCF)CN2CCC1CC2 N(C1CCCc2nc(O)ccc21)C(C(=O)NCCCCCC)C c1(CN2CC(C)C(C)(CNC3CC(F)(F)C3)C2)ccc2c(c1)COC2(C)C c1(C(=O)NC2C(C)CN(C(=O)CS(N)(=O)=O)C2)cccc(N)c1Br c1(OC)cccc2c1OCC(C(N1CCCN(C(=O)CCF)C(CO)C1)=O)C2 C(=O)(C1=NOC2(CCC2)C1)N1C(CNC(C=CS(CC)(=O)=O)=O)CCC(C)C1 Cc1cc(C)c(NC(=O)CC(C)CNC(C2(CN(C)C)CC2)=O)c(C)c1 Cc1nsc(N)c1C(N1CCC(O)(C(C)NC(C2CCSCC2)=O)C1)=O N1(C(C=COCC)=O)CCC(CCNC(c2csc(C)c2CC)=O)C(F)(F)C1 C1(C)(CNC(CSCC)=O)CCN(C(c2cc(-c3ccccc3)sn2)=O)C1 C1(c2nnnn2CCCF)(NCc2c(C)ccnc2)CCCC(C2CC2)C1 C(=O)(C(C)(C)C(F)(F)F)N1CCC(C(C)NC(C(C(C)C)CN(C)C)=O)CC1 C1(OCC)CCN(C(=NCCSC)NCc2noc3c2COCC3)CC1C c1(C(c2nnnn2C2CC2)NC2(C)CC(=C)C2)cc2n(n1)CC(C)(C)CO2 C1(C(=O)NC2CC(CC(=O)N(C)CC3CC3(F)F)C2)(OC)CCCCC1 C1(NC(C(C)=C(CC)C)=O)CC2CCC1CN(C(c1scnc1C)=O)C2 CC1CN(C(c2ncn(-c3ccccc3)n2)=O)C(C)CN1C(=O)COC(C)(C)C C1(CNC(C(c2ccc(Cl)cc2)C)=O)C(C)CCCN1C(C1CCCC1O)=O c1(C(C2CCCO2)NC(=O)NCCOc2cccnc2)ccc(F)cc1 C(=O)(C(C)C(C)NC(C1(C)CCN(C(=O)Cn2cnc(=N)[nH]2)C1)=O)OC Cc1cc(C#N)cc(C)c1COCC(=O)NCC(C)(CO)CC(=O)O C(=O)(C1=CCC(NC(=O)CC(O)C2CCCC2)C1)NC(CC#C)CC C1(N=c2ccn(CCCO)[nH]2)(c2n(CCC(=O)OCC)nnn2)CSC1C Cc1ccc(C(=O)NCC2COC(CNC(=O)C#CC3(C)COC3)C2)c(=O)n1C C#CCCCC(C)C(=O)N1CC2CC2(C(=O)NCCN2CC=CCC2)C1 c1(C(N2C(C)C(NC(=O)C=C3CCN(C)C3)CCC2)=O)cccc2c1CNC2=O C1(CNC(C2CC(C#N)C2)=O)CC(O)CN1C(=O)CCN1CCC1 C1(CNC(Cn2ncc(CC)c2)=O)CC(C)(C)CN1C(=O)C(C)SC C1(C(=O)NC(c2nc(C)on2)C)CCCCN(C(=O)Cn2ncn(C)c2=O)C1 c1(C(=O)OC)ccc(O)c(C(=O)NCC(O)CNC(=O)C(O)P(C)(C)=O)c1 N1(C(CC(=O)OC)=O)CCC(C=CC(=O)NC2CCC3(CC2)N=N3)CC1 N1(C(c2csc(Br)n2)=O)CCOCC(CNC(C2(F)CCCC2)=O)C1 C1(CNC(c2c(C)con2)=O)CCN(C(=O)C(F)(F)Sc2cnn(C)c2)CC1C c1(OC)cc(C)c(C(=O)NCC2CC(O)CN2C(=O)C2=CCCCC2C)c(C)c1 Cc1ccc(OC(C)C(=O)NCC2(F)CCC(NC(=O)CN(C)C(N)=O)C2)cc1 C12(NC(CCC=CC)=O)CCC(CNC(=O)CC3CCCCC3(F)F)(CC1)OC2 CCC(CC)(C(=O)N(C)CCN(C)C(C1CC1C)=O)c1ccc(Cl)cc1 C1(C(N2CC(C(C)NC(c3ccc(C(F)F)o3)=O)C2)=O)CC(=O)CC12CCC2 c1(CONC(C2(C(N(C(=O)CCSC(C)(C)C)C)=O)CCC2)=O)cncn1C C1(CC(=O)NC2CC(CCNC(CCc3ncn(C)c3)=O)C2)CCCS(=O)(=O)C1 Cc1cccc(Br)c1C(C(=O)NC1CC1(C)CO)NC(c1cc(C(N)=O)[nH]n1)=O CCC(C)(C#N)C(=O)N1CC(CN(C(=O)C=Cc2nc(C)c(C)[nH]2)C)C1 N1(C(c2nnc(C)s2)=O)CCCC(C)C1CCNC(c1cc(C2CC2)no1)=O CC(C)(C)C(=O)CCC(=O)N(CCC(N1CCC(C)(C2CC2)C1)=O)CCO c1(C(=O)NC2CCN(C(C(=O)NCC)=O)CC2C)cccc2c1N(C)C(=O)CO2 CCC(C)CCCC(=O)N(CCC(=O)NC(C)CN(C)C)CC C1(NC(CCCC=C)=O)CN(C(c2ccc(-c3ncon3)cc2)=O)CC2(CC2)C1 c1(NC(C(C(C)(C)C)NC(C(C)S(C)(=O)=O)=O)=O)cnc2[nH]cnc2c1 c1(C(C(=O)N(CCN(C(C(F)=CC)=O)C)C)NC(=O)COC)ccccc1 C1(NC(C2(CC)CCCN2C(c2cnn(C)c2C#N)=O)=O)CCOC12CCCC2 c1(CCCC)cc(N)c(C(=O)NCCCCCNC(=O)C(C)CS(C)=O)c(F)c1 Cc1cccn2ncc(C(=O)NCCCNC(C34CCC3CC4)=O)c12 c1(C(N(C2CCCN(C(C3C(C=C)C3)=O)CC2)C)=O)cnc2sc(C)cn2c1=O N1(C(C2(NC(c3cn(CC)nn3)=O)CC(F)(F)C2)=O)CC(C)=CC(C)C1 C=CC1CN(C(=O)CCc2ncc[nH]2)CC1NC(=O)CCCNC(N)=O c1(C(N2CC(N(C(C(CC)N(CC)CC)=O)C)C2)=O)ccc(OC)c2ccsc12 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1C(C(N(C)Cc2ccccn2)=O)CC(O)CC1 C1(CCN(C)C(C2COC(C)(C)C2)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC1 C1(C(=O)NCCC2(CNC(c3c(C)cn(C)c3)=O)CC2)CC2CCC1CC2 c1(C(C)CC)ccc(OCC2(NC(C)=O)CC2)cc1.N12CCC(CC1)CCOC(=O)C2 C=CC(C)(C)CCNC(c1ccc(SC)o1)c1nnnn1CC C(=O)(C1=C(C(C)F)N(CC)C(=O)NC1c1ccc(N2CCC(C)C2)cc1)OCC c1(C(=O)NC(CN(C(=O)C(C)S(C)(=O)=O)CC)C)coc2c1COC2 c1(CCC(=O)NCC2C(NC(c3cnc(C)[nH]3)=O)C2)ccc(Cl)cc1 CC(C)CC(=O)C(=O)NC1CCC(CC(N2CC(F)(CF)C2)=O)C1 N(C1CN(C(C2CCCC(=O)N2)=O)CCc2ccccc21)C(c1nnn(C)n1)=O c1(C(N2C(CN(C(COC(CC)C)=O)C)CCC2)=O)cc2ncccc2o1 c1(CC)c(Cl)nc(C2CCC2)[nH]c1=NCCN(C)C(C1CN(C)CCO1)=O c1(SC)cnn(C)c1C(=O)NC1(C)CN(C(=O)C(c2ncccc2F)(F)F)C1 C1(NC(c2c(C)csc2)=O)CCCCC1C(=O)N(C1CC1)Cc1ccccc1 N1(C(Cc2cc(C)[nH]n2)=O)CC2COCC2(C(N2CCOCC2C(C)O)=O)C1 c1(NC(C(C2CCC(C)(C)CC2)C)=O)ccc2c(c1)S(=O)(=O)CC(=O)N2 C12(NC(CSC)=O)CCC1CN(C(=O)CC1(N(C)C)CCCC1)C2 c1(C(=O)NC2C(NC(C(C)CC(F)(F)F)=O)CCCC2)cc2c(s1)CC(C)(C)C2 Cc1ccnc(C(C)NC(=O)CCN(C(C2CN(C3CCC3)C2)=O)C(C)C)n1 CCC(C)C(O)C(C)C(=O)N1CC(C)(C)CC1CC(=O)NOC N1(C(c2c(C)nn(Cc3ccccc3)c2)=O)CC2(CC(CNC(=O)C(F)F)C2)C1 C1(C(F)(F)F)(C(N(CC(C)NC(c2coc(C3CC3)n2)=O)C)=O)CCN(C)C1 c1(CC(=O)NC2(COC)CN(C(CCCOCCC)=O)C2)cccc(Cl)c1Cl N1(C(C(CC)OC(C)C)=O)CC2CC1(CNC(=O)CCCOc1ccccc1)C2 N1(C(C(F)=CCC)=O)CC2CCC1C2NC(=O)CC1CCCCC1(C)C c1(SCC(=O)NC2C3CN(C(N4CCC(O)CC4)=O)CC23)cc(F)c(Cl)cc1F N1(C(c2ccc(OC)cc2)=O)CC2CC(NC(=O)COCC(C)C)C2C1 N1(C(CCC2CCN(C(c3ocnc3C3CC3)=O)CC2)=O)CCCC12CCC2 N1(C(C2CC(=C3CC3)C2)=O)CC2(C(=O)Nc3ccccc3)CC1CO2 c1(OC)ncccc1C(=O)N(CCSC(c1ccc(F)cc1)c1cc[nH]n1)C c1(C(=O)Nc2nccn2Cc2ccc(C(F)(F)F)cc2)ccc(F)c(F)c1 CC(C)CCCCC(=O)N(C1CC(NC(=O)COCC2CCCO2)C1)C c1(C(=O)NCC(CNC(c2c(SC)csc2)=O)F)cnc(C)c(C)c1 c1(CC)nnc2c(C(=O)NCCN(C(C3CC4C=CC3C4)=O)CC)cccn12 Cc1cc2ncn(CC(=O)NCCN(C)C(c3c(O)cccc3Cl)=O)c2cc1C CCCC(CCC)CC(=O)NCC=CCNC(C1Cc2cccc(F)c2O1)=O CN=c1[nH]c(=NCc2cnc(C)[nH]2)[nH]c(=NC(C)Cc2nc3ccccc3s2)[nH]1 C(=O)(C(F)(F)Cc1ccccc1)NCC1(C)CC(NC(C2CCOC2(C)C)=O)C1 c1(C(N2C(CNC(c3ncc(C)cn3)=O)COCC2)=O)cnc([N+](=O)[O-])cc1C c1(C(=O)NC2COCCN(C(C3(O)CCCC3)=O)C2)c(Cl)ccc(Cl)c1Cl c1(C(=O)NC2C(CNC(C3(CC#C)CC3)=O)CCC2)ccc(N)c(C(C)=O)c1 C1(CNC(c2ncc(C)nc2)=O)C(C)CCCN1C(c1n[nH]cc1C)=O c1(NC(C2N(c3nc(C)nc4c3c[nH]n4)CCC2)=O)cccn2nc(C)nc12 n1(CCC(=O)NC2CCCC2NC(c2cc(O)cs2)=O)cnc2ccccc12 c1(C(=O)NC2CC3C2CCN3C(C2SC3C=CC2CC3)=O)noc2c1CCCC2 C1(C(=O)NC(c2nccn2C)CC)(CNC(c2cncn2C)=O)CC12CCC2 C(=O)(CC1=CCCCC1)Nc1cc(C)c(NC(=O)CC(O)CN(C)C)cc1 c1(CCC(=O)NCC(C2CCCC2)NC(C(CCC)C)=O)ccc(F)cc1F C(=O)(CC(C)(C)C#N)N1C(C(N2CCC2CC(C)(C)C)=O)(COC)C=CC1 C1(NC(c2ccnc(C)n2)=O)CCN(C(C23CC(CN2C2CC2)C3)=O)C(C)C1 N1(C(CN(CC#C)C(c2cc(C)co2)=O)=O)C2C=CCC1CC2 S(=O)(=O)(c1ccc(Br)cc1NC1CCN2CCCC12)NCC(CSC)OC C(CC(C(=O)NC1CCCSC1)NC(=O)CC1CCOC1(C)C)OC C(=O)(CC#N)NC(C1(CNC(CSCC=C)=O)CC1)C c1(OC)nsc(OC)c1C(=O)NCCOC(C)(C)CNC(=O)Cc1csnn1 c1(C(N2CCC(CC(=O)Nc3c[nH]nc3Br)C2)=O)c(F)cncc1Br C(=O)(C(=O)N=S(C)(C)=O)NCC1(COC)CN(C(=O)CCc2csc(C)n2)C1 c1(N2CCC(=O)NCC2)nc(NCCCn2ccc(C3CC3)n2)c2ncsc2n1 c1(C(=O)NCC2C(NC(C(C=C)(C)O)=O)CC2)cc2cc(Cl)ccc2[nH]1 N1(C(c2ccc(Cl)o2)=O)CC(NC(C2(C(c3ccccc3)=O)CC2)=O)C2CC12 c1(OCCC(=O)NC2C(OC)CN(C(=O)CC3(C)CCC3)C2)ccc(F)c(Cl)c1 C1(CC(=O)NCCc2cccnc2F)COCCN1C(C1CCCC(O)C1)=O C1(NC(C2CCN(C(C=C(CC)CC)=O)C2C)=O)CN(C)C(=O)C12CC2 C1(NC(C=CSC)=O)CC2(CCN(C(=O)CC3CC4(CCCC4)CO3)CC2)C1 N1(C(c2c(C)cn(C(C)C)c2)=O)CC2CCCC2(CNC(c2c[nH]c(=N)s2)=O)C1 c1(C(=O)NC2C(NC(C(Cn3ccc(C)n3)C)=O)C2)ccc(F)c(F)c1F N1(C(c2snc(C)c2N)=O)CC2(CC(C(N3CCC(CC(F)F)C3)=O)CO2)C1 c1(CC(N2CC(CNC(=O)C(O)C3CC3)OCC2)=O)ccc(F)cc1C(F)(F)F C(C(CC)CC(CC)CC)NC(c1n(CC=C)nnn1)c1ncc[nH]1 Cc1cc(N)cnc1C(N1CCC(C(=O)NCC2(C)CCCC(=O)N2)C12CC2)=O N1(CC)CC(C(=O)NC2CCCCC2N(C(=O)CCc2ccco2)C)CC1=O c1(C(=O)NC(CC(C)NC(c2[nH]cc(C(=O)OC)c2)=O)C)c(F)cc(C)cc1Cl C1(C(=O)NCCN(C(C2CC2C2CCC2)=O)CC)CCCCC1(C)C c1(C(C)(C)C)cc(C(N2CCC(N3CCOC3=O)C2)C(=O)NCCCF)on1 n1(CC(N2CCN(C(c3nccc(C)c3)=O)CC2)=O)cnc2c1CCCC2 C1(C(N2C(CNC(CCN(CCC)C)=O)(COC)CCC2)=O)CCCCN1N=O c1(C(=O)NCC(C(C)C(C)C)NC(C2(CCC)CC2)=O)cnc2n(c1=O)CCS2 S(=O)(=O)(c1c(C)o[nH]c1=N)NC(=O)C(n1cc(C)cn1)(C)C.CC N1(C(N2C(CC=C)(CC=C)CCCC2)=O)CC23CCCC2(C1)CN(C)C3 c1(CNC(C23N(C(c4c(OC)nccc4)=O)CCC2C3)=O)nc(C)ccc1O OC1CCCC(N=c2[nH]c(=NCc3ccc(Cl)o3)[nH]c3c2CCC3)C1 Cc1cccc(CCNC(C23CC2CN(C(C2(CO)CCOC2)=O)C3)=O)n1 c1(OC)cc(CNCC2(C(N3CCC(C#N)C3)=O)CC2)ccn1 c1(C(=O)NC(C2CN(C(C3(c4ccccc4)CC3)=O)CCO2)C)cc(O)ncn1 c1(-n2cc(C3N(C(c4cc(C)ncn4)=O)CCCC3)nn2)ccc(Cl)cc1Cl C#CC1CCCN(C(=NCCCC)NCCSc2cccc(OC)c2)C1 C=CCCCCCC(=O)NC1CC2CCC1N2C(=O)CCc1nc(O)n[nH]1 c1(C(COC(N2CC(OCCC(=O)NC3(CCCC)CC3)C2)=O)=O)ccccc1 C(=O)(C1=CC2CCCC12)NCCOC1CN(C(c2nccc(C)c2)=O)C1 c1(C(C)C)ccccc1C(=O)N(C1CN(C(C2CC2c2ccco2)=O)C1)C C(=O)(CCCCCN=[N+]=[N-])NC1(C)CN(C(C2(OC)CCSC2)=O)C1 C(=O)(C(CCN(C)C)NC(=O)CCN(C)C)NCC(C)NC(=O)CO c1(C(N2CCC(NC(Cc3cn(CC)nc3C)=O)(CF)C2)=O)cc(C)nc(O)c1 C1(C(=O)Nc2c(CC)nsc2)CN(C)CCN1C(c1cc(C2CC2)on1)=O c1(N2CCC(S(=O)(=O)NCC)C2)nc(=NCc2ncoc2C)[nH]c2ncn(C)c12 N1(C(C2C(OCC)C2)=O)CCN(C(=O)CC2(OC)CCC2)CC(C)C1 C1(C(N(CC(CN(C(CSc2ncc(C)o2)=O)C)O)C)=O)CC1C1CCCCC1 Cc1nc(CCCNC(=O)CC2CCN(C(=O)Cc3sccc3C)C2)n[nH]1 Cc1cc(C(C)(C)C)ccc1C(=O)NCCCCCNC(=O)Cc1ccno1 N1(CC(CC)(O)C(F)(F)F)CCCC2CCCN(C)C12 C(=O)(C(C)(C)C(=O)N(C)C)NC1CC(NC(C=CCOC)=O)C1 N1(C(C2CN(C)C2)=O)CCCC(C(=O)N(C)Cc2nccn2C)C1 c1(C(=O)NCC(C)NC(=O)C(C)C(C)O)cccc2c1CCOC2 C(c1ccc(F)c(Cl)c1)=CC(=O)NC(C1CCCC1)CNC(C(C)OCC#C)=O c1(-n2c(CNC(CCN(C)C)c3ccco3)nnn2)ccccc1Br c1(SC)cccc(N)c1.C(CC(C(C)C)N)NC(N1CCCC(C)C1)=O C1(N(C(C(=O)NCCOC)C(C)C2CC2)C)CC2CC3CC(C2)CC1C3 c1(C(CSCC)C)cn(C2CN(C(=O)CC3CCSC3)C2)nn1 N1(C(CC2N(C(C(C(C)C)SC)=O)CC2)=O)CCC(O)(CCO)CC1 Cn1nc(C(F)(F)F)cc1CC(=O)NCC(CO)NC(c1cc(CO)on1)=O c1(C(N2C3C(NC(=O)COCCCF)C(C3)C2)=O)ccc2ncccc2n1 N1(C(c2scc(OC)c2)=O)CCC(C#N)(NC(C2CC=CCC2)=O)C1 c1(C(C)C)ocnc1C(=O)NCC1(O)CC(NC(=O)CCc2ccon2)C1 c1(C(C)CC(=O)NCC2CC2NC(=O)CCOCCN(C)C)cccc(F)c1 N#Cc1ccc(F)c(-c2ccc(-n3cc(Br)cn3)cc2)c1 C1(NC(COCCCC#C)=O)CN(C(c2ccc(N)c(SC)c2)=O)CCC1CO N1(C(C(C)NC(=O)OC)=O)CCC(CCNC(C2CC2c2ccncc2)=O)CC1 C1(NC(c2ncccc2F)=O)CN(C(C2CC3CCC(C2)C3)=O)CC12CCCC2 c1(-c2ccc(C)cc2)nnc2n1CCN(N1CCCC(C)CC1)C2C C12CCCCC1N1C(C(CC#N)Nc3cccc(n3)C2)C(CC)CCCC1 c1(C(=O)NC(C2CCN(C(c3ncc(OC)nc3)=O)C2)C)cccc(C#N)c1 C1(NC(C(=O)Nc2c(C)c(N3CCCC3)ccc2)=O)COC2(CCOCC2)C1 C1(C(F)(F)F)(OC)CC(N)(C(=O)NCC2(c3ccccc3C)CCC2)C1 Cc1nncn1NC(=O)C(C)C1CCN(C(=O)C(N)=O)C1 C1(C(=O)NC(CC=CC)C(=O)N2CCC(CC(C)C)CC2)CC2(CCC2O)C1 c1(CC(=O)NCC2N(C(COCCCC)=O)CCC2C)c(Cl)cccc1Cl CC1CC2CC(C(=O)N(C)Cc3cc(C(F)(F)F)ccc3Cl)(C2)O1 C#Cc1ccc(C(=O)NCC(F)CNC(c2cc(C)ccc2Br)=O)cc1C c1(CC)oc(C(=O)NCC2CCN(C(=O)C(C)Oc3ccccc3)C2)cc1C c1(CNC(C(C)Sc2ccccn2)=O)cc(F)c(O)c(F)c1.C12(C)CN(C1)C2=O CC1(C)CC(CNC(C2CCCCNC2=O)=O)N(C(C2(C)CCOC2)=O)C1 c1(OC(C)C(=O)N(C(C)CNC(=O)Cn2nnc(C#N)n2)C)ccc(Cl)cc1Cl Nc1c(C(=O)NC2CCC(NC(c3ccnc4[nH]ncc34)=O)C2)cc(F)cc1F c1(C(N2CC(N(C(CCNC(=O)NC)=O)CCO)C2)=O)ccc(C(C)=O)cc1F C(CC1=CCN(C(c2cc(Br)cc(F)c2F)=O)CC1)NC(C(C(C)O)C)=O C1(C(=O)NCC2C(NC(=O)CCCC(F)(F)F)CC2)CCc2nnc(O)cc2C1 C1(CC)CC(C)CN(C(CCC2(C#N)CCC2)C(=O)NC2CC(F)(F)C2)C1 Cc1nc2cc(C(=O)NC3CC4CC3CN4C(C3CCC(=O)O3)=O)ccc2o1 C1(C(C(=O)NCC(C)NC(C2(N(C)C)CC2)=O)O)CCC(C(C)(C)C)CC1 c1(C(N2CC(O)(CNC(c3c(CC)non3)=O)C2)=O)c(N)cc(C)cc1F C1(C(=O)NCc2c(F)ccc(C)n2)N(C(=O)CC(C)C(C)C)CCCC1(C)C C1(C2CC2)(CNC(C2C(CC)OCC2)=O)CCN(C(=O)Cc2ccncc2Cl)C1 c1(NC(CNC(C(CCC)CCC)=O)C2CC2)ncnc2cc(C)[nH]c12 CN1C(=O)CCC1CC(=O)NCC(C)(C)NC(=O)CCN1CCCCC1=O C12(CNC(C(c3cn(C)nn3)N(C)C(C3CC4(CSC4)C3)=O)=O)CCC(C1)C(=O)N2 c1(N(CC)CC)ccc(C(=O)NC2CCC2NC(c2ncccc2O)=O)cc1 c1(CNC(C(CCF)NC(C2C(C)=CCS2)=O)=O)cccc(F)c1C C1(NC(C(C)N2CCC2)=O)CN(C(c2ccnc(C(F)(F)F)c2)=O)C(C)(C)C1 c1(NC(c2n(C(CC)C)nnn2)c2ccno2)ccc(OC)c([N+](=O)[O-])c1 O=S(=O)(c1ccc(O)cc1)N1CC2(CN(Cc3ncc(-c4ccccc4)[nH]3)C2)C1 c1(C(C)CC(=O)NCC(O)COC(F)(F)F)cccc2ccccc12 c1(CCC)nnc(S)n1CC(=O)N(CC(C)NC(=O)C(C)Cn1ccc(C)n1)C C1(NC(NC(CC)CC)=NCCSC)COc2c(C)cccc2C1 C12(CNC(C(C)(C3CCC3)NC(=O)COCCCF)=O)CCC(CC1O)C2 c1(OC)cc(N2CCC(C(C)NC(c3ccc(C(N)=O)cc3)=O)C2)ncn1 Cc1ccc(C(=O)NC(C)C(N2CC(NC(c3sccc3F)=O)C(C)C2)=O)cc1 CCCCCCN=c1ccn2nccc2[nH]1.C(=O)CC1CC1 C1(O)(CNC(=O)CC2CCN(CCF)C2)CCCN(C(=O)CCC2CCC2)C1 C1(CC(=O)NCC(C2CC2)NC(c2cccc(C(F)(F)F)c2)=O)CCC2CC2C1 C1(C(N(CCSC)CC)=O)(NC(c2cc(C3CCOCC3)on2)=O)CCNC1=O c1(C(N2CC(C)(C(F)F)OCC2)=O)nccn2c(Br)ccc12 C(=O)(C1=NOC(C)C1)NC1CCCC(CNC(c2ccc(COC)o2)=O)C1 CN1CCC(CC(=O)NCC2CC(NC(c3ccco3)=O)C2)C1=O Cc1ccnc(NC(=O)NC(C(C)C)C(O)c2ccccc2)c1Br Cc1cc(Br)cc(F)c1C(N1CC2CN(C(c3cncc(O)c3)=O)C2C1)=O c1(C(=O)OC(C(=O)NCC(C)C)C)cn2c(n1)CC(C)CC2 N1(C(=O)CC2CNCCO2)CCC(CCF)(C(=O)O)CC1 c1(NC(c2cc(-c3ccc(C#C)cc3)[nH]n2)=O)c(C)cc(F)cc1[N+](=O)[O-] c1(NCC(C(CC)CC)O)ccc(S(=O)(=O)N2CCCC(CC(=O)OC)C2)cn1 C1(NC(c2ccc(C(CC)C)cc2)=O)CC2CN(C(=O)CC3CC3C)CC2C1 c1(C(N(C)CC2N(C(C(CSC)C)=O)CCCC2)=O)cc(C)cc(N)c1 C12(CNC(COCCCC#C)=O)CCCC1N(C(c1cc[nH]c1)=O)CCC2 N1(C(c2c(C)onc2)=O)CCC2CN(C(=O)C=Cc3cccc(F)c3F)CC2C1 N(C1CCc2cc(OC)ccc21)C(=O)NCC=Cc1ccc2c(c1)CCO2 N1(C(C(C)Oc2ccccc2)=O)C2CCCC1CN(C(c1ccsc1C#N)=O)C2 N1(C(C2C(c3n(C)cnc3)C2)=O)CCN(C(c2occc2Cl)=O)C(CO)C1 C#CCC(CC(F)F)NC(=O)CC1CCC(NC(c2ccc(CC)[nH]2)=O)C1 C1(CC)CCN(C(=O)C(C)N2CC(C)C2)C1C(=O)NC(CO)C(F)(F)F CC1(C)CN(C(c2n[nH]cc2Cl)=O)CCC1NC(=O)CC1CCC(C)CO1 c1(C(=O)NC(C(C)NC(=O)C(=O)NC2CC2)C)ccc(S(=O)(=O)C2CCC2)cc1 N1(C(C#CC(C)C)=O)CCN(c2cc(O)ncn2)CC(C)(F)C1 CCC(CC)CC(F)C(=O)NC1CC(=O)N(C2CN(C(=O)CCC3CC3(F)F)C2)C1 N1(C(c2n(C)c(-c3ccccc3)c(C#N)c2)=O)CCOc2c(F)cccc2C1 n1(CC)c(C)cc(C(=O)NC(C(C)NC(=O)CCS(N)(=O)=O)C(C)C)c1C C(=O)(C1=CCCOCC1)NC(C(C)CNCC(F)(F)F)=O.N12CCN(CC1)C2=O C(=O)(C1=COCCC1)N1C(C)CC(CNC(c2ccc(OCC(F)F)cc2)=O)C1 N1(C(COC)=O)CC2CCC2(CCNC(=O)CCP(C)(C)=O)C1 C(=O)(C(C(C)(C)C)N(C)C)N1CC(OCCC(=O)N(CC#C)CCN(C)C)C1 C12(NC(c3onc(CC)n3)=O)CCCC1N(C(=O)C=Cc1ccn(C)c1)CCC2 C(C)(C(C(=O)NCc1ccsc1C)C(C)C)NC(C(C1CC1)SC)=O c1(CNC(=O)NC2CCCC(SC)C2)csc2cc(Br)ccc12 N1(C(C(C)(C)OC(C)C)=O)CCCN(C(c2scnc2C2CC2)=O)C(C)C1 C1(NC(C(C)c2ccsc2)=O)CCCC12CCN(C(=O)C=C(Cl)Cl)CC2 C1(CNC(C(C2CCOC2)OC)=O)CN(C(=O)CC(C)C(C)C)CC(C)(C)O1 C1(C(=O)NCCCNC(=O)C=CCN2CCOCC2)CCC(F)(F)C1 N1(C(Cc2cc(C)sc2)=O)CCC(C(F)(F)F)C(NC(c2ccc(N)cn2)=O)C1 C(=O)(C(C)(CNC(c1cc(F)ccc1O)=O)CC)NC(CC)CN(C)C N1(C(C(ONC(c2cc(CC=C(C)C)[nH]n2)=O)C)=O)CCc2nccnc2C1 CCC(C)CC(=O)NCC(C1CC1)N(C(=O)CCC(=O)N(C)C(C)C)C N1(C(C=C(CCC)CCC)=O)CCOCC(NC(=O)CC2(C#N)CCCCC2)C1 C1(OCC)CCCCC1NC(c1cnn(CCNC(C2CC2OCCO)=O)c1)=O c1(C(=O)NC23C(n4cc(CC(C)(C)O)nn4)CC(CC2)C3)cnc2ncccn12 C(C(=O)N1CCC(C(=O)NCc2cccnc2Cl)O1)n1c(=N)nc[nH]1 c1(N(CCC2CCN(C(c3c(C)cns3)=O)CC2)C)cc(=O)n2ccccc2n1 C1(C(=O)NCCCCNC(c2n(C)nc(C(C)(C)C)c2)=O)CC2CCC(C1)O2 c1(C(=O)NCC2(F)CC(NC(CCC)=O)C2)ccc2c(c1)OCCCO2 C1(OC)CCC12CC(C(=O)NC1(CNC(=O)C=C(C)C(F)F)CCC1)C2 CC(C)(CC(=O)NC(CNC(C1C(C#N)C1(C)C)=O)C1CC1)C(F)(F)F Cc1cc(C(=O)OCc2ccn(C3CCCC3)n2)nn1C(C)(C)C C1(c2nnnn2C2(C)CC2)(NCCc2c(C)cccn2)CCN(C)C1C N1(C(C2(CC#C)CCOC2)=O)CC2(NC(=O)CCc3cc(OC)no3)CC1C2 c1(C(C(=O)NCCOC2CN(C(C(CC=CC)C)=O)C2)O)cc(Cl)cc(Cl)c1 N1(C(C(Cn2cncn2)NC(c2c(C)nc(C)o2)=O)=O)CCC2(CNC(=O)O2)C1 c1(C2(C)CCN(c3nnc(C(=O)NCC=C)s3)CC2)nc2ccccc2s1 Nc1c(C(=O)NC2(CNC(C3SC4C=CC3C4)=O)CCC2)cccc1[N+](=O)[O-] c1(C(C)C)cnc(Cl)nc1N1CCC(NC(=O)C(C)OCC2CC2)C(F)C1 N1(C(C(CCC)NC(=O)C(C)C2(O)CCC2)=O)CC(C)C(C)(CO)C1 CC(C)C(C)C(CNC(=O)COCc1nc[nH]n1)NC(=O)C(C)(C)C C(=O)(CCCN=[N+]=[N-])NC1CC(F)(CNC(CC2N(C)CCC2)=O)C1 c1(C(=O)NCC2CCN(C(CCN(CC)CC)=O)CC2)cccn2cncc12 C1(NC(C(C2CCC2)OCC)=O)CC2C(NC(c3cc[nH]n3)=O)C2C1 C1(CNC(C(COC)(C)O)=O)CC2CCC(C1)N2C(c1cc(C(C)=O)oc1C)=O c1(C(N2CCC(C(=O)Nc3nnc(C)o3)C2)=O)cccc(C(F)(F)F)n1 C1(C(N2CCCCC(NC(Cc3nc(C)[nH]n3)=O)C2)=O)CCc2ncncc2C1 c1(NCCCOC(C)C)nc[nH]c(=NCC2(OCCN(C)C)CCCOC2)c1C N1(C(c2c(C)nc(C3CCC3)o2)=O)CCC(F)(CNC(C2(F)CCCC2)=O)CC1 c1(OC)ccc(C)nc1C(N1CCC(O)(C(C)CNC(C2CCCC2)=O)C1)=O N1(C(C2CCC(NC(c3c(C)cc(F)s3)=O)CC2)=O)CCC2(C1)CN(C)C2 c1(C2CCN(C(COc3c(C)cccc3)=O)CC2)cccc2c1OCCO2 N1(C(CCC(CC)NC(c2cnn(C)c2Cl)=O)=O)CC(C)(C)OC(C)(C)C1 c1(COC(C(C)(C)c2ccns2)=O)cc(Br)c(Cl)c(Br)c1 CCC(CNC(c1ccccc1)=O)(CC)C(=O)Nc1ccc2nonc2c1 c1(CN(C(CC(C)N(C)C)=O)Cc2ccsc2)ccc(Br)cc1 N1(C(c2nccc(CC)c2)=O)CCN(c2ncc(Br)c(C)n2)C(CC)C1 c1(NCCN(C(=O)CCN2CCOCC2)C)nccc(-c2ccccc2F)n1 c1(-c2nc(C)nn2-c2cccc(F)c2)ccc2c(c1)CCC2 c1(C(=O)NC(C)CNC(c2ncnc3sccc23)=O)cnc(O)c2ncccc12 C(=O)(CCCC(C)O)NC(C1(O)CCN(C(c2cccc(SC)c2)=O)C1)C Cc1ccc(C(=O)NCC2(O)CCN(C(=O)CC3OCCC3(C)C)CC2)c(C)c1 N1(C(C(OC)OC)=O)C2CCC1C(F)C(NC(C1(CC(N)=O)CCCCC1)=O)C2 c1(OC)ccc2nc(C)c(C(=O)NC(C)CCF)n2n1 C(N=c1[nH]cnc2c1CCC2)C1(NC(C(C)N2CCCC2)=O)CCC1 C1(C(=O)NCCOC(C)=O)CCN(C(=O)CC2(C)CCOC2)C1C(C)C CN1CCC(CC(N2CCOC(CNC(=O)Cc3cn(C)nc3Cl)C2)=O)C1=O c1(C(=O)NCC(CO)NC(C(C(C)C)C)=O)ccc2c(c1)CCCCN2 c1(C(=O)NC2CC(CC)OCC2)c(OC)c(Cl)cc([N+](=O)[O-])c1Cl N1(C(COC2CC(NC(CCC(C(C)C)=O)=O)C2)=O)CCCC2CN(C)CC12 Cc1cc(O)nc(C)c1C(=O)NC1CN(C(=O)CC(C)(C)CN(C)C)C(C)(C)C1 C1(NC(C(C)CN(C)C)=O)CN(C(=O)CSc2ccc(F)cc2)C2(CCCC2)C1 C(CNC(c1csc(C(F)F)c1)=O)(CCOC)NC(CCN(C(CCC)C)C)=O c1(C(=O)NCC=CCNC(C(C)(C)COCC(F)F)=O)cc2n(n1)CCCC2O C1(CCNC(c2ccc(C3CC3)s2)=O)CC(F)(F)CN1C(C1C2CCCOC12)=O N1(C(CCn2ccc(C)n2)=O)CCN(C(=O)CCF)C(C)C1 c1(OCC(=O)NC(C(C)C)(C)CNC(C2(C)CNC(=O)C2)=O)cccc(F)c1F O(NC(=O)CCOCCCN(C1CC1)CC1CC1)CCOCCOC c1(OC)ncc(C(N2CCCC(CCNC(C)=O)C2)C(=O)NC(C)CC)cn1 c1(OC)cc(C(=O)NC2(C)CCN(C(=O)C(C3CCCO3)C3CC3)C2)ncn1 c1(C(N2CC3C(NC(=O)CC4CCCC45CC5)C3C2)=O)cc2sc(F)cc2[nH]1 c1(C(C)NCCC2CCCO2)ccc(I)cc1 c1(C(N(CC(c2ccccc2)C)C2CC2c2ccsc2)=O)ncc(F)cn1 c1(CNC(Cc2ccc(C)s2)=O)ccccc1CNC(C1C=CCC1)=O C(=O)(C(C)C(F)(F)F)N(CC1CCN(C(c2cc(CC)no2)=O)CC1)CC C=C(C)C(CC(=O)NC(COC)C(=O)Nc1cccc(C(N)=O)c1)OCC C1(CC)CN(C(=O)CC(O)C(C)C)CCN1C(c1cnc(C)[nH]c1=N)=O c1(C(=O)NCCCN2CCN(C(C3(C)CC3(F)Cl)=O)CC2)cccc(N)c1O c1(CC(C)C)cn(CCN(C(=O)C(C)c2ccsn2)C(C)C)nn1 c1(COC)nc(NCCCCOC(C)C)cc(=NC2CCCN(C)C2)[nH]1 C1(NC(C(=O)NCC)=O)CN(C(=O)Cn2nnnc2C)CC12CCOCC2 N1(CC#N)CCc2cc(CN3CC(NC(c4cc(CO)on4)=O)C(O)C3)ccc21 n1(CC)nc(C)cc1C(N1CCCC1C(=O)NCc1nn[nH]n1)=O CCC(C)(C)C(C)CC(=O)N1CCCC1CNC(C12CCC(CC1)O2)=O Cc1cc(NC(=O)NCC(=O)Nc2cc(N3CCNC3=O)ccc2C)nc(C)c1 c1(CC)ccc(C(=O)NC(CNC(=O)CCCc2ncco2)C(C)C)c(O)c1 CCC(CC(F)F)C(=O)NCC1CN(C(=O)CSS(C)(=O)=O)CCC1C c1(C(N2CC(C)(NC(C3CC(CCC)OCC3)=O)C2)=O)nccc2occc12 CC1(C)C(C(=O)NCC2CC3CCC2CC3)CCN1C(=O)COC1CCOC1 c1(C(N)=O)ccc(C(=O)NCCNc2ccc(C=O)cn2)cc1.c1(S)ccccc1 C1(=O)CC(CC)N1.C1(CNC(=O)NCCC(=O)OCC)COC(CC)C1 CN1CCN(C(=O)Cc2cscn2)C(CNC(=O)COC2CCCOC2)C1 c1(NC(C)C)ncccc1C(N1CCOC(CNC(=O)Cc2cnnn2C)C1)=O C1(NC(C2(OCC)CCC2)=O)CN(C(c2cc(C)n(C)c2)=O)CC1N=[N+]=[N-] C(C)(C)(C(=O)NCCCNC(=O)CC=C(C)C)OCC CC(C)C(C(=O)OC(C)(C)C)C(=O)NCC(C)NC(c1cc2n(c1)CCSC2)=O C1(C(C(=O)NC(C#C)(C)C)NC(=O)C(=O)N(C)C)CCCCC1 C(C(C)(C)CC(=O)NCC(=O)N(C)C)NC(CCCNC(=O)OC)=O CC(C(F)C(=O)NC1CCN(c2ncnc(Cl)c2Br)CCC1CO)C(F)(F)F c1(OC)ncc(C(N2CCOC(CC(=O)NCCCC(=O)OC)C2)=O)cc1F c1(C(=O)NC(CC=C)CNC(=O)CCCn2ccnc2)cnn(CCC)c1Cl c1(C(=O)NC2CC3CN(C(CCC#C)=O)CC2C3)ccc2c(n1)CCC(C)C2 C(CCCCC(=O)NCC1CC12CCOCC2)N(C(C1C(C(C)C)OCC1)=O)C N1(Cc2c(C)cc(F)cc2)CCC2CC(C(=O)NCC(O)C(C)(C)O)C2C1 c1(C(=O)NCC2(OC)CCN(C(C(C)N(C)CC)=O)C2)nc2ccccc2s1 c1(C(=O)NC23CC(C(C)(C)C)(C2)C3)cc2ncc(-c3nn[nH]n3)cc2[nH]1 c1(C(N2C(C(N)=O)CCCC2)=O)n[nH]c2cccc(-c3ccc4[nH]ccc4c3)c12 N1(CCc2cn(CC)nc2)CCC(NC(=O)Cn2cc(Cl)cn2)CC1C N1(C(CN2CC(CC)C2)=O)CC2CCCCC2(CNC(c2cncc(C)c2)=O)C1 Cc1cccc(C(=O)NCCC2CC(NC(=O)C(C)C(C)C)C2)c1Br C(=O)(C(C)(F)C(C)(C)F)NC(C(C)C)C(=O)NC1(C)CCCCCC1 N1(C(CC(CC)OC)=O)CCN2CCOCC2(CNC(C2CC(O)C2)=O)C1 N1(C(CC(=O)NCC#C)=O)C2CCCC1CC(CNC(=O)C1=NOC(C)(C)C1)C2 c1(C(=O)NC2(CNC(C(C)(C3CC3)OC)=O)CC2)ccc2c(c1)CC2 C1(c2ccc(CC)o2)CCCCCN1C(=O)Cc1cscc1Br CCC(C)C(CNC(C1(SC)CN(C(=O)CCCC(=O)OC)C1)=O)CO C(=O)(C(C)C(C)c1ccc(F)cc1)N1CC(CC=C)(NC(=O)CCOCC)C1 CC1C=C(C(=O)N(C)CCN(C)C(c2csc(C3CCCO3)n2)=O)CC1 C1(CC)CN(C(=O)Cc2ccn(C)n2)CCC1NC(c1cnc(COC)s1)=O CC(CN(C)C)C(=O)NCCSCc1cn(C2CCCC2)nn1 CC(C)C(C)(C(N)=O)NC(=O)NNC(C1OCCN(C)C1c1cnn(C)c1)=O C1(NC(CC2CC(C)OC2C)=O)CCC2CN(C(c3cnsn3)=O)CC2C1 N1(C(c2cnc(-c3cc(=N)[nH]cc3)s2)=O)CCN(C(=O)C=C(Cl)Cl)C2(CCC2)C1 N1(C(C(C)CC2CCCCC2)=O)CCN(C(=O)Cc2cncnc2)CC12CC2 c1(NCC(=O)COC2CCCCC2)ncc(O)cn1.C12CN(CCO1)C2 c1(N2CC(C)C(NC(C3CC34CCOCC4)=O)C2)nc2ncc(Cl)cc2s1 N1(C(CC(C)(C)OC)=O)CC2(CCOCC2)C1c1cn(-c2ccccn2)nn1 C1(CCNC(C2(CC)CCC2)=O)COCCN1C(c1ccnc(C(C)C)n1)=O C(CN=[N+]=[N-])(C(=O)NCC(C)(C)C1CC1)NC(Cc1c(C)n[nH]c1)=O c1(C(N2CC(N(C)C(c3cccc(F)c3N)=O)C(O)C2)=O)cc2cccnc2s1 CC1CC(NC(C2CCCO2)=O)CCN1C(c1ccc(C(F)(F)F)c(O)c1)=O C(C)(C(=O)N1CCCCO1)OCCNC(COC(CC)CC)=O N1(C(c2cc(CNC(=O)CC3CC(F)C3)[nH]n2)=O)CCC2(CNC(=O)C2)C1 C1(C(=O)NC2(CN(C(=O)CCOc3cccc(F)c3)C)CC2)CCCC(F)C1 CCCCC(C(=O)NCCC1(NC(c2c[nH]nc2OC)=O)CC1)N(C)C N1(C(C2(SC)CCC2)=O)CCCN(CCNC(=O)Cc2cccc(C)c2)CC1 c1(C(N(C2CCN(C(C3(C)CC3(F)Cl)=O)CC2)CCO)=O)n[nH]c2c1CCC2 c1(C(=O)NC2(CNC(c3nc(C)sc3)=O)COC2)ccc2occc2c1O C12(CCOCC1)N(C)CC2=O.C1(NC(C=CC)=O)CCC1N(C)C c1(CN(C(C)CNC(c2cc(C#N)c[nH]2)=O)C)nnc(S(C)(=O)=O)s1 c1(C(=O)NCC(CC=C)NC(=O)C(F)CC2CC2)cccc2cnccc12 C(=O)(C(C)(C)c1nncn1C)NCCC(C)NC(=O)CCCNS(C)(=O)=O Cc1nsc(C(N2CCC(C(=O)NC3CCC4CCC34)C2)=O)c1N N1(C(C2OCCN(CC)C2)=O)CC(NC(c2ccnnc2S)=O)CC(F)C1 C(C)(CCC(=O)N1CCCC1CNC(c1cnc(C2CC2)o1)=O)OC Clc1cccc2c1OCC2Nc1nccc(=NCCc2ccoc2)[nH]1 C1(CNC(CCn2c(C)ncc2)=O)CCCCC1NC(C1(CCF)CC1)=O c1(C(N(CCn2cc(C(N3CCOC3=O)C)nn2)CC)=O)cnc2[nH]cncc1-2 c1(NC(C)=O)c[nH]c(C)c1C(N1CCOC(C(C)NC(=O)C=C2CCCC2)C1)=O C1(C2CCC2)(C(N(C(CNC(c2cc(O)cs2)=O)C2CC2)C)=O)CC1(F)F N1(C(C(C)OCCC=C)=O)CCN(C(=O)C2CCc3c[nH]nc32)CC(C)(C)C1 CC1(NC(=O)Cc2ccsc2)CCN(C(C2(C#N)CC2C(F)(F)F)=O)C1 N1(C(COCCC(C)C)=O)CCC2CN(C(c3ccc4c(c3)CCN4)=O)C2C1 C1(NC(C(COC)C)=O)CCN(C(C2CC2c2ccc(C)cc2)=O)CC1 N1(C(CC(C(C)C)C)=O)CC2(CCC(CNC(C34CC(CO)(C3)C4)=O)O2)C1 c1(NC(C2CCCCN2C(=O)NC2CN(C(=O)C3CC3)C2)=O)cccc(Cl)c1 C1(NC(Cc2c(C)n[nH]c2)=O)CCN(C(=O)C(F)C2CCCC2)CC(O)C1 c1(C(=O)NCC2(NC(C3CC3(F)F)=O)CC3CCC2C3)ccn2nccc2n1 N1(C(CCCCOCC)=O)CCCCC12CN(C(=O)Cc1cc(C)on1)C2 Cn1cc(Cl)cc1C(=O)NCC(C)(C)OCC(=O)NCC1CC(C)(O)C1 N1(Cc2nc(C(F)F)sc2)CCCC(c2ccc(Cl)cc2)C1 N1(C(C(N(C(c2cc(C)c(C)s2)=O)C)C2CC2)=O)CC(C)(C)C2COCC12 C1(N=[N+]=[N-])(C(=O)Nc2c(C)cc(O)nc2)CCN(C(c2cccs2)=O)C1 c1(C(=O)NCC(CNC(c2c(C)cc[nH]c2=N)=O)F)ccnc2ccc(F)cc12 S(=O)(=O)(c1cnccc1N1CC23CCC2(COC3)C1)NC(C1CC(F)(F)C1)C N1(C(C2C(C(C)C)C2)=O)CC(CNC(=O)Cn2cc(Br)cn2)C2(CC2)C1 c1(OC)ncc(Br)c(C)c1C(N1CC2(CC(NC(=O)C3=COCC3)C2)C1)=O c1(CCC(=O)NCC(C)CNC(=O)CC2COC(=O)N2)ccncc1 c1(OC)cc(-c2nc(-c3cccnc3)nn2C2CC3CCC2C3)ccc1C(=O)O N1(C(CCNC(CCOCCOCC)=O)=O)CCC(CO)CC1C C1(C)(CNC(c2cnc(OC)nc2)=O)CCC(NC(=O)CC2CC23CC3)CC1 c1(OC(C)C(N2CC=CC(NC(=O)C(C(C)O)N(C)C)C2)=O)cc(F)cc(F)c1 Cc1cc(=N)[nH]cc1C(N1CC(C(F)(F)F)OCC1CNC(=O)C=C1CCC1)=O CC(C)CS(=O)(=O)CC(=O)NC1CC1NC(c1ccc(=O)n(C)c1)=O N1(C(C(=O)NCC)=O)CCC2(NC(=O)C(F)CC(C)(C)C)CCCCCC12 N1(C(c2nc(COC)oc2)=O)CCCCC1C1CCN(C(=O)C(C)=CCO)C1 N1(C(C2(CSC)CC2)=O)CC(C(N2CC(O)(CN(C)C)C2)=O)C(F)(F)C1 C(=O)(C(F)CCCCC)NC(CCC=C)C(=O)NCC1CC(C)C1 C1(NC(c2ccc(OC)s2)=O)CC(O)CN(C(c2nocc2C)=O)C1 c1(C(N2CCCC(NC(CC(C)CF)=O)C2)=O)cccc(O)c1[N+](=O)[O-] C=CCC(C)(C)C(=O)NCc1ncc(C(=O)O)s1 Cc1cc(C)c(C(=O)NCC2CC(NC(c3ccc(C#N)c(O)c3)=O)C2)c(=O)o1 C1(CCNC(C(C)SC)=O)CC(F)(F)CN1C(c1cccc(C2CC2)n1)=O N1(CC(=O)NC(CC)CN(C)C)c2ccccc2CS1(=O)=O CC1=CCC=CC1C(=O)NC1CCC(C(=O)Nc2scc(C)c2C)C1 Cc1nc(N2C3CCC2CN(C(c2ccn4cncc4c2)=O)C3)c2c[nH]nc2n1 C1(CNC(CC(=O)NCC)=O)CN(C(c2c(Br)noc2C)=O)CCO1 Cc1nc(C(N2CCCCC2CN(C(=O)CC2COC(=O)N2)C)=O)c(C)s1 C1(CC(=O)N(C2CCN(C(c3ccon3)=O)CC2)CC)CC2(CCC2)CCO1 c1(CC(=O)NCC2(F)CN(C(C3CC(F)C3)=O)C2)cncnc1O c1(C(=O)NCCCN(C(CC2CC(CC)OCC2)=O)C)c(C)nn(C2CC2)c1Cl c1(OCC)nn(C)cc1NC(=O)C(C)(C1CCC1)NC(C1CCOC1)=O CC1CC2CCC(C1)N2C(C1COCC1NC(c1occ2c1CCC2)=O)=O N1(C(c2ncn(CCNC(Cc3ncn(C)c3)=O)c2)=O)CCCC(CCO)CC1 c1(CC)nccnc1C(=O)NCCC(O)CNC(=O)C=C1CCSCC1 Cc1cc(CNC(=O)C=CC(C)NC(c2ccc(C)c(O)n2)=O)nc(C)c1 c1(C(=O)NC2CN(C(=O)CCNC(N)=O)CC2F)ccc2cncc(Br)c2c1 C1(C(=O)NC2C=CCN(C(CC3(OCC)CCOCC3)=O)C2)CCCC2(CC2)C1 CC(C)CC(C(=O)N1CC(C)(O)C1)N(C(=O)CC1CCCC1O)C N1(C(c2c(OC)cccc2)=O)CC(NC(=O)C(C)C(C)(F)F)C2(CC2)C1 C1(C(N2C(C(C)NC(C(C)NC(COC)=O)=O)CCC2)=O)C(C)(C)C1(C)C C#Cc1cnc(C(N2CCC(C3CC3)C2C(=O)NOC2CC2)=O)c(C)c1 CC(CC(C)(C)C)C(=O)N1CC(OCCC(=O)NC(C2(O)CCCCC2)C)C1 N1(C(C2C(C)(C)C2)=O)CCN(C(N2CCN(C3CCC3)CC2)=O)C2(CCC2)C1 N1(C(CNC(=O)CN(C(c2cn[nH]c2)=O)C2CC2)=O)CCC(C2CCC2)C1 C1(C(=O)NC(CO)C2(C)CC2)(CNC(CCSC)=O)CC=CC1 C(=O)(C1=NOC(C)(C)C1)NC(C1(O)CN(C(c2c(OC)ccc(O)c2)=O)C1)C N1(c2nc(N3CC(=O)NCC3)c3c(n2)scc3)CCCCC2(CCCC2)C1 c1(OC)ccc(C=CC(=O)Nc2cc(C)cc(Br)c2F)cc1C(C)C c1(CN(CCC)C(C2CCCN2C(=O)C=CC2CCCC2)=O)ccccc1 Cc1csc(=NCC(=O)N(CC(O)CN(C)C(c2sc(CO)nc2C)=O)C)[nH]1 Cc1ccc(C(N2CCCC(NC(C3(C4CC4)CCC3)=O)C2)=O)cc1C CC1CCN(C(c2nccc(N)c2Cl)=O)CC1CNC(C1(C(C)(F)F)CCC1)=O c1(C(N(c2ccccc2)CC)=O)cc(OC)ncc1-c1cc(O)ccc1OC N1(C(C2(C=C)CC2)=O)CCN(C2CCC(NC(=O)COc3ccccc3)C2)CC1 CC(C)(C)CC(F)C(=O)N1CCC(C(C)(C)NC(C2CC23CCCCCC3)=O)C1 N1(C(c2cc(OC)ns2)=O)C2CCC1CN(C(=O)C(C)(O)C1CC1)C2 O=C1CCC(C(=O)NC23CC2CN(C(=O)C(F)=C2CCCC2)C3)n2cccc21 Cc1cc(C(=O)NC(C)(CNC(=O)C(F)OC(F)(F)F)C(C)C)c(C)o1 C1(C(=O)NC(C)C(C)(C)C)CCCC(NC(=O)C=CC2CCCN2C)CC1 N1(C(C2C(COC)C2)=O)CCN(C(=O)C=Cc2cncc(O)c2)C(CC(F)F)C1 Cc1sc(=O)n(CC(N2CCC(NC(C3CCN(C)C3=O)=O)C(O)C2)=O)c1C C1(C)(C(=O)NCC2N(C(C(C(C)C)n3cncn3)=O)CCCC2)COC(=O)OC1 c1(C(N2CCC(NC(C3=CC(=O)CC3)=O)CC2)=O)cncc2ccccc12 N1(c2onc(CCC)n2)CC(C(=O)OC(C)(C)C)C2CCCCC12 C(CC(N)=O)(C(=O)N(C(C1CCC(F)(F)CC1)CO)CC)NC(=O)OC(C)(C)C C#CC1(O)CC(C(N2CCC(CO)(CNC(=O)C(C(C)C)NS(C)(=O)=O)C2)=O)C1 CC1=C(C(=O)NC2CN(C(=O)C3COc4ccccc43)C2)Cn2ncnc2N1C C(=O)(CCCCN=[N+]=[N-])NC1(C)CCN(C(=O)C#CC2CC2)C1 C12(CNC(CN(CCOC)C)=O)CCCN(C(c3ccnnc3)=O)C1C2 n1(CC=C)nc(-c2ccc(N)cn2)nc1C(O)Cc1nccn1C c1(NC(C)=O)ccc(C(C)C(=O)OCc2nc(-c3ccccc3)no2)cc1F Cc1ccc(NC(C2CC3CCN(C2)C3)=O)c(-n2cc(C3(O)CCC3)nn2)c1 CS(=O)(=O)c1ccc(Cl)c(C(=O)NCC2CN(C(C3(F)CC3)=O)CCO2)c1 C(=O)(C(CC(C)C)C(N)=O)N1CC(NC(C2CC3(CC(=C)C3)C2)=O)(CO)C1 C(=O)(C#CC1CCCCC1)NC(CN(C)C)C(N1CCC2(CCOC2=O)C1)=O C1(NC(=O)COC2CCC2)CN(C(=O)CCCc2cncs2)CC2(CCC2)C1 C(=O)(C1=CC2CCCCCC12)N1CC(CNC(C2CC3(CCC3)CO2)=O)C1 c1(C(=O)NC(CC)(C)CNC(C2CCCN2c2nccs2)=O)nccc(OC)n1 N1(C(CN2CCCC(CC)C2)=O)CC2(NC(=O)CCCOCC)CC1C2 N1(CC)CC(C(=O)NC2CC(NC(=O)C=CC(=O)N(C)C)C2)NC1=O c1(NC2c3c[nH]nc3CC2)nc2cc[nH]c2c(=NC2CC3CSCC3C2)[nH]1 CC(C)C(C(=O)NCC1CCCC1NC(C1(C(F)(F)F)CC1)=O)N1CCCC1 C(=O)(C#CC1(C)CCCO1)N1CCCC(N(C)C(c2ccc(C(N)=O)nc2)=O)C1 C1(NC(C2C(C=C)C2)=O)CN(C(C2(CF)CC(F)(F)C2)=O)CC1C=C CCC(C(=O)OC)C(=O)NCc1csc(C(=O)NC2CC2c2cnn(C)c2)c1 N1(C(c2cc(CC)nnc2C)=O)CC2CCC1CN2C(=O)C1=CCC(C)CC1 Cc1cnncc1C(=O)NC(CNC(=O)CCCNC(=O)C1CC1)CC(C)C CCCCCCCN(C(=O)CCN(CCCO)C(c1conc1C)=O)C N1(C(CCCCN(C)C)=O)CCN(C(c2ccc(F)cn2)=O)C2CCCCC2C1 CCC(C(C)(C)C(=O)OC)NC(=O)CCCCCn1cc(C(O)C(C)C)nn1 O=C(CCCCC(F)(F)F)NCCC1CCN(C(=O)C(F)OC(F)(F)F)C1 CSC=CC(=O)N1CCC(OCCNC(C2(F)CCC2)=O)C1 CCC(O)C(C)C(=O)N(C(C)CCNC(=O)C(c1ccc(Cl)cc1)C)C CC1(NC(C2CCCCN(C(=O)CCCC3CCCC3)C2)=O)CCCC1(F)F n1(CC(=O)N(CCN(C(C=C(CC)C)=O)C(C)C)C)ccc2c(C)cccc12 Cc1cc2ncnc(N3CCC(NC(C4CC(O)C4)=O)C(C)C3)c2[nH]1 C1(NC(c2cc(OC)n(C)n2)c2n(CC(=C)C)nnn2)CCC2CCCC1O2 c1(C(C2CCCN(C(=O)C(=O)Nc3cc(C#N)ccn3)C2)C)ncc(Cl)cc1F N1(CC(N2CCC(C)C(CNC(C3(C)CCC3)=O)C2)=O)CCc2sccc2C1 c1(C(=O)NCC2CC(NC(CS(=O)(=O)NC)=O)C2)cc(=O)c2ccc(Cl)cc2o1 CCC1=NOC(CC(=O)NC2(CCC(N3CCC(CCOC)C3)=O)CCC2)C1 C(C(C)(C)OCCC(C)C1CCC1)NC(COCCCC)=O.C1C(=O)N1 Cc1ccc2ncc(C(=O)NC3CC4CCC3(NC(=O)C(F)C3CCC3)C4)n2c1 Cc1cc(=NCC2CN(C(=O)CCc3ncc(F)cn3)CC23COC3)[nH]c(Cl)n1 C(CN=c1[nH]cnc2ccc(O)cc12)NC(C1CCn2ccnc2C1)=O c1(SC)cc(N2CCCC2CNC(=O)CSc2cnn(C)c2)nc(SC)n1 C1(C(=O)NC(C)CCCNC(=O)Cc2n[nH]c(=N)s2)CN2CCC1(C)CC2 C(CC(=O)N1CCN(C(c2cc(N)cc(O)c2)=O)CC1CO)(C(N)=O)NC(C)=O c1(C(=O)OC)ccc2c(c1)CC(C)N2C(c1ccc2n[nH]cc2n1)=O Cc1cnc2c(cnn2CC(=O)NC2CN(C(C3(C4CC4)CCC3)=O)CC2C)c1 Cc1c(C(=O)NCCOCCNC(=O)CN2CC3CC3C2)cc(C(C)C)n1C c1(OC)cnc(C)cc1C(=O)NCc1sc(C)nc1COC.c1(C)ccccc1 CCC(O)(CC(=O)Nc1cccc(NC(c2nsnc2O)=O)c1)c1ccccc1 c1(CC)c(C(=O)NCC2(C(F)F)CCN(C(c3cnsn3)=O)C2)cccc1F C=CC(C)(O)CC(=O)NCC1CC(NC(c2scc(C)c2Cl)=O)CCO1 C=CCC(CC(=O)N1CC(c2ccccc2)C1)NC(=O)C(C)CC(=O)OCC Cn1ccnc1C(=O)NCC(C)(O)CNC(C1CC1CC(C)(C)C)=O c1(C(=O)NCC2N(C(C(CCC)(C)C)=O)CCCC2)c2c(nn1C)CCSC2 N#CC1CCC(C(=O)NCC2(NC(=O)Cc3csc(C4CC4)n3)CCOCC2)C1 Cc1nc2cc(C(=O)Nc3ccc4c(c3)CCCC4O)c(F)cc2[nH]1 c1(OC)cc2cnccc2cc1NC(=O)NCC1CCC2(CCCCC2)O1 C1(NC(Cc2ccc(OC)cc2)=O)CN(C(c2c[nH]nc2C2CC2)=O)CCC1C c1(OCC(=O)N(CCNC(=O)CC2(CO)CC2)CC)nc(Cl)c(Cl)cc1Cl c1(C(=O)NC2CCN(C(c3cc(C)cc(O)n3)=O)CC2O)ccnc2[nH]nnc12 Cc1ccnc(C2CCN(C(=O)C(N3CCCC(N(S(C)(=O)=O)C)C3)=O)C2)c1 c1(C(N2CC(C)(C(=O)NC(C)CCO)C2)=O)ccc(F)cc1Br N1(C(C2OCCN(C)C2)=O)CCCC2(C1)CN(C(c1nn(C)cc1N)=O)CCO2 C(=O)(CCS(C)(=O)=O)NC(CCOCC)C(=O)NCC(O)C(F)(F)F N1(C(c2oc(C)c(Br)c2)=O)CCN(C(=O)C(F)CC(C)C)CC2(CC2)C1 c1(C(=O)OC)cncc(C(N2CC(CC(=O)Nc3c(Br)cnn3C)C2)=O)c1 c1(OC)nccc(C(=O)NC2CCCC2NC(c2cnc(-c3ccco3)s2)=O)n1 C#CC(C)(C)C(=O)NCC(CCC)NC(=O)C(C1CCCCC1)O c1(OCC)c(C(C)NC2CCN(c3ccc(Cl)cc3)C2)c(C)nn1C c1(C(C(=O)NC2CCC(NC(C3CC=CC3)=O)CC2)O)ccc(Cl)c(F)c1 c1(-c2cccc(C(=O)NC3CC(CNC(COC)=O)C3)c2)ccc(C(C)C)cc1 Cn1cnc2cccc(CNC3(c4nnnn4C4CCCC4)CC4CCOC34)c12 C=C(Cl)C(C)(C)C(=O)N1CC(CC(C)NC(=O)CSCc2ccccc2F)C1 CCC(C)(C)C(C(=O)OC)N(c1cccc(C(C(=O)OC)C)c1)C c1(CNC(CCCC#C)c2nnnn2C2CCOC2)c(F)cccc1Br C1(CN(C(=O)C(C2CCCCC2)O)C)CCCN1C(C1CCC(F)C1)=O c1(C(N(CC(=O)NCC(=O)NCC2CC2)CCC)=O)sc(C)cc1C Cc1cc(F)sc1C(=O)NC(c1ccccc1)CNC(=O)C(C)NC(C)(C)C c1(C(=O)NCCCN(C)C(c2ccnc(CO)c2)=O)ccc([N+](=O)[O-])nc1 n1(CC(=O)NC(C(C)NC(c2ccn(C(C)(C)C)n2)=O)(C)C)cccnc1=O CCCC(CCCS(C)(=O)=O)C(=O)NC1CC(CO)N(C(c2ccccc2)=O)C1 N1(C(c2c(CC)cccc2)=O)CC2OCC(NC(C3(CC(=O)OC)CC3)=O)C2C1 CN1CCCC(C(C)(C)C(=O)NC2(c3ccccc3)CC(F)(F)C2)C1 N1(C(C(CC)(C)O)=O)C2CCC1CC(NC(c1cc(=O)c(C)c[nH]1)=O)C2 c1(C(=O)NC(C2CN(C(c3c(C)n(CCO)nc3)=O)C2)C)cccc(F)c1C C12(C(=O)Nc3c(OC)cc(C(N4CCOCC4)=O)cc3)CCC(F)(CC1)CC2 C1(CCC)CN(C(=O)C(C)NC(=O)NC)CCN1C(c1cnn(C)c1N)=O Cc1ccc(C(N2CC=CC2CNC(=O)COC(C)C)=O)c(Br)c1 C1(C(N(CC(C)NC(CCc2cc(C)[nH]n2)=O)C)=O)CCC(=O)N1C N1(C(C(C)(C)N2CCCC2)=O)CC(F)CC1CC(=O)NCC1(C)CCC(=O)C1 Fc1cccc(-c2ncc(CN(c3ccc(Br)cn3)C3CC3)s2)c1 Cc1nc(CNC(=O)CC2CCC2)oc1C(=O)NOCCOC(C)C C(CC(C)(C)CC(=O)N1CCCC(CC(N2CCOC(C)(C(C)C)C2)=O)C1)OC C(CC(C)CCNC(=O)C(O)c1ccsc1)NC(Cc1nc(C)[nH]n1)=O N1(CC(=O)N(C)C)CCC2(CC1)CC2C(N1CC2CCC1(C)C2)=O C=CC(CC)CC(=O)N1CC(CNC(c2cc(Cl)n[nH]2)=O)C(F)(F)C1 C1(CCC)CCCN(C(c2cc(CNC(C3(OC)CC3)=O)ccn2)=O)CC1 c1(C(=O)NCCC2(C)CCN(C(CC(=C=C)C)=O)C2)c(C)cccc1N C(=O)(C(=O)N=c1ccn(CC(F)F)[nH]1)N(CCC)C(c1ccccc1OCC)=O S(=O)(=O)(c1ccc(Cl)c(C(=O)N(C)C)c1)NC(c1cn(C)nc1)C1CCC1 C#CC1(C(=O)Nc2cncc(Cl)c2)CCN(C(=O)C(CN(C)C)CC)C1 C1(C(=O)NCCC(C=C)C)C2CN(C(C3(O)CCSCC3)=O)CC12 CCC(CCC(=O)NCCN1C(=O)CNC1=O)NC(c1ccc(Cl)cc1)=O c1(C(=O)NCC(C)N(C(=O)C(O)C(C)C)CC)cc(C2CC2)ncc1Br C1(C(N(CCCN(C(=O)CN2CC=CC2)CC)CC)=O)CCCN1C1CCCC1 c1(NC(c2ccc(-c3c(C)cccc3)cn2)=O)ncc(F)c(Cl)n1 C#CCCCCC(=O)NCc1ccc(CCNC(=O)CC2CCC(C#N)C2)cc1 N1(C(COC(C)(C)C)=O)CCCC(CC(=O)NC2CC(N(C)CCO)C2)CC1 C#CCC(C)(C(=O)N(C)CCc1nccs1)NC(=O)CC1CC(CC)=NO1 c1(OC)ccc(C)c(C(=O)NCC2C(C)CCN2C(=O)Cc2cccc(Cl)c2)c1 c1(C(=O)NC(C)C)cc(C2=CCC(C(C)(C)C)CC2)[nH]n1 C=CC(F)(F)C(=O)NC(C1CCCN(C(c2cc(F)n(C)n2)=O)C1)C N1(C(c2cn(CC)nn2)=O)CCC2CN(C(=O)C(=CC3CCCC3)C)CCC2C1 c1(C(N2C(CNC(C3CCCN(c4ncccn4)C3)=O)CC2)=O)ccc(F)cn1 N1(C(CC=CC)=O)CCC2(CC1)CC2(CO)CNC(=O)C(C(C)C)n1cncn1 c1(C(N2CCC(CC)C2C(=O)NCC2(CF)CCC2)=O)cc(O)cc(F)c1 C(=O)(C1CCCn2ncnc21)NC1CC(C)N(C(c2scnc2Cl)=O)CC1 CC1=NOC(=O)C1CCC(=O)NC(C)CNC(=O)Cc1nccc(C(F)(F)F)n1 C1(C2CN(C(C3(c4cc[nH]n4)CC3)=O)C2)(NC(C(c2cccnc2)C)=O)CC1 N1(C(c2cc(C(F)F)no2)=O)CCN(CCN2CCCC2=O)CC1 c1(C(=O)NC2C(NC(C3C(SCC)CCC3)=O)CCC2)ccnc2c1ncn2C c1(CNC(C2CNC(=O)N2)=O)ccc(C(N2CCC(N3CC(O)C3)C2)=O)cn1 C1(CNC(c2ccc(CC)cn2)=O)COC(C)(C)CN1C(=O)CC1COCCO1 N1(C(C)C)CC(C(N2CCN(C3CCN(C(=O)C=CBr)C3)CC2)=O)CC1=O C12(C(=O)NCCOCCC(C)C)C(NC(=O)CCS(N)(=O)=O)C3CC1C2C3 N1(C(CC(C)C(C)(C)C)=O)CCC2(CC1)CC(NC(=O)CCC1CC1(C)C)C2 n1(CCC)cc(C(=O)NCC(C)(C2CC2)NC(=O)CC2CC(CC)C2)nn1 C12(C(=O)NC(CCCC)CNC(c3sccc3C(C)C)=O)CC(C)(C1)OC2(C)C c1(C(=O)NCCOCCN(C(=O)CC2CCC(=O)O2)C)cnn2c1OCCC2 CCCCC(C)(F)C(=O)N1CCC(N(C)C(C2CCCCC2)=O)CC1 N1(C(c2nc(C)c(C)s2)=O)CCC(C(=O)OCc2c(Br)cnn2C)CCC1=O N1(c2nccc(C(=O)OCC)n2)CCN(C(c2cccc(F)c2I)=O)CC1CC C(=O)(C1CCCc2ccccc21)NCCC1CC(NC(c2cc(C#N)oc2)=O)C1 CCC(CC(=O)NCC1(NC(=O)Cc2ccn(C(F)F)n2)CC1)CC(F)(F)F N#CC1CCCC(C(=O)NCc2ccsc2C(N2CCC(O)(CO)C2)=O)C1 n1(CCC(=O)N(CC(OC)OC)CC(C)C)cnc2sccc2c1=O CC1CN(C(C2CSCC(=O)N2)=O)CCC1NC(=O)C(c1ccccc1F)(F)F C1(CNC(C(c2ccccc2)N(C)C)=O)CCN(C(c2cnc[nH]c2=N)=O)CC1 C(=O)(CCCN(C)C)NCC(CC)NC(c1ncsc1C)=O C1(O)(CNC(c2n(C=C)nnc2)=O)CCCN(C(C2(N(C)C)CCCCC2)=O)C1 Cc1ccccc1CN(CC(O)CN(C)C(c1ocnc1C)=O)C C1(NC(=O)C(N2CCN(CC3CC3)CC2)=O)CN2CCCN1CC2 N1(C(CCNC(C#CC(C)(C)C)=O)=O)CCC2CCC(C1)N2C C12(NC(C3CCCC(N(C)C)C3)=O)CCCC1N(C(=O)CC1CC(F)(F)C1)CC2 CC1CCN(C(=O)C=Cc2ccnn2C)CCN1C(C1CCCNS1(=O)=O)=O N1(C(C2CC=C(C(=O)OC)C2)=O)CC(OC)C2(COC2)C1 N1(C(c2cc(CC)no2)=O)CCOC2(CCCN(C(C3(C)CCSCC3)=O)C2)C1 c1(C(=O)NCCN(C(=O)Cc2cccc(Br)c2)CC)c(C)cc[nH]c1=N Cc1cc(C(N2CCC(C)(NC(=O)COC3CC3(F)F)C2)=O)cnn1 N1(C(C=CC)=O)CCC2C(NC(c3cc(C(C)(C)C)oc3C)=O)C2CC1 N1(C(c2cc(CC)[nH]n2)=O)CCC2(CCCC2C(=O)Nc2ncccn2)C1 C1(NC(CCc2onc(CC)n2)=O)CCCCC1CNC(c1c(Cl)n[nH]c1C)=O c1(CC)ccc(C(=O)NCCC(O)CNC(C2(C(C)(C)C)CCCC2)=O)c(C)n1 CCC(O)C(F)(F)C(=O)NC1CC2(C1)CC(C(=O)NCCCc1ccccc1)C2 N1(C(C(c2ccc(OC)cc2)O)=O)CC2CN(C(=O)C(C)NC=O)CC12 N1(C(c2cccnn2)C(=O)NCc2cccc(OC)c2)CCC2(C=CCO2)C1 C1(NC(c2cc(CCC)oc2C)=O)CN(C(=O)C(C)Cc2ccco2)CCC1F C1(CC#C)(C(=O)NC(CNC(=O)CCn2cnnn2)C2CCC2)CCCCO1 C(CCSC)(C(=O)N1CC(F)CC1CO)NC(c1c(CC)cno1)=O C1(CCC)CN(C(C2CC(=C(F)F)C2)=O)CCN1C(C1CCN(C)C(C)C1)=O N1(C(CC)CC)CC(C(=O)NCC=CCNC(C2OCCOC2C)=O)CC1=O C1(CCN(C(C2C(C)(COC)C2)=O)C)CCN(C(c2scnc2C2CC2)=O)CC1 c12ncccc1CN2.c1(C(=O)NC2CC(CNC(COC)=O)C2)cc(OC)n[nH]1 c1(C(=O)NCC2(C(C)(C)C)CCN(C(=O)C#CC3CC3)C2)cc(O)cc(O)n1 C#CCC(C)(C)C(=O)N1CCN(C(=O)CCN2CCCCCC2)C(CF)C1 C12CC3(CCC3)CN1C2=O.c1(CC)nc(CNC(=O)OC(C)(C)C)ns1 C#Cc1ccc(OC)c(C(=O)NCC2CCN(C(=O)C(=O)NC3CC3)CC2C)c1 n1(CC)nncc1C(=O)NC1CCC(CC(=O)NCC2CC2c2ccncc2)C1 C(=O)(C1=COCCC1)N(C(C)C)CCc1cc(Br)cc(Cl)n1 C12(NC(CCCN(CCC)CCC)=O)CC1CN(C(=O)CSc1cnn(C)c1)C2 c1(C(N2C(CNC(C3(F)C(C(=O)O)C3)=O)CC2)=O)cnn(C2CCOCC2)c1 Cc1ncc(Br)c(C(=O)NCC(C(C)(C)C)NC(=O)CC2CC=CC2)n1 c1(C(N2CC(CC(=O)NCC3CC(C(C)(C)C)C3)(OC)C2)=O)cc(C)c(C)o1 Cc1ccc(C)c(OCC(N2CCC(O)(NC(=O)COC(C)(C)C)C2)=O)c1 N1(C(C(c2cnccn2)C)=O)CCCC1CN(C(=O)CC1CCC(C)C1)C C1(C(=O)NCC(COC)(F)F)C(C)CCN1C(c1ccc(C#N)[nH]1)=O N(C1COc2ccc(Cl)cc21)C(C(c1ccc(C)cc1)(F)F)=O c1(CN(C)C(=O)NCC2CCCN2C(c2ccoc2)=O)cccnc1O S(=O)(=O)(C(C)CN=c1[nH]c(=NCc2cocn2)[nH]c2cc[nH]c12)NC C1(C(=O)NCCC(Cn2cc(C(C)(C)C3CC3)nn2)F)CCCCN1N=O C1(O)(C(C)NC(C2CC(C(F)F)C2)=O)CCN(C(c2csc(Cl)c2)=O)C1 c1(C(=O)NC(CCC)CCCNC(C2CC=CCC2C)=O)n[nH]c2c1CCSC2 c1(OC)ccc(CC(C)C(=O)N(CCCNC(=O)C=Cc2ccoc2)C)cc1F c1(C(=O)NC(C)C(c2ccccc2)NC(=O)CC2(C)CC2)ccn(C)c(=O)c1O CCCCCS(=O)(=O)CC(=O)NC1CN(C(c2cnc(CC3CC3)s2)=O)CC1O c1(C(N(C2CC(C(N)=O)C2)C)=O)coc2c1CN(C(=O)C(C)(C)F)C2 C1(C(=O)NC2(C(N3CCC(CCOC)CC3)=O)CC2(C)C)CCCC12CCC2 N1(C(c2ccc[n+]([O-])c2)=O)CC2(CNC(C34CCC(CC3)CC4)=O)CCC1CC2 C1(C(=O)NCC2(CSC)CCC2)(NC(=O)C(=O)N(C)C)CC(O)C1 C1(CNC(c2ccc(Cl)nc2)=O)CCCCN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 c1(CNCC2(CCC=C)CCCC2)cccc(F)c1OCC(C)C C1(CNC(c2ccnc(-c3nccs3)n2)=O)C2CN(C(C3CS(=O)(=O)C3)=O)CC12 Cc1ccc2cc(C(=O)NC3CC(c4ncc[nH]4)C3)ccc2c1 N1(C(C2(C=C)CCN(C(=O)C(n3cc(C)cn3)C)C2)=O)CCc2nnnn2CC1 CCCC(C(=O)OC)C(=O)NCC1CN(C(=O)CCc2cc(OC)no2)CC1O N1(C(c2c(OC)ccc(O)c2)=O)CCN(C(=O)C(C)=C2CCCC2)CC(C)(F)C1 c1(C(N2C(CNC(c3c(N(C)C)cccn3)=O)CCC2)=O)cc(O)c(F)cc1N C1(O)(NC(C(C)N(CCCCCNC(c2c[nH]nc2C(F)F)=O)C)=O)CCOCC1 N1(C(CNC(CNC(C)=O)=O)=O)CC2CN(C(c3cnsc3C)=O)CC2(C)C1 CC1CN(C(C2CCSCC2)=O)CCC1CNC(c1cc(CO)[nH]n1)=O C(=O)(CCC(C)CN(C)C)NCCC1(O)CN(C(C(C(=O)OC)C)=O)C1 C(CC(=O)N1CC2=C(C1)CN(C(c1c(C)nsc1N)=O)C2)(C(F)(F)F)OC N1(CC(=O)NCCN(C(=O)C=C(C)CCC)CCC)CC=CC1 CN1CCc2ccc(C(=O)NCCC3CN(C(C4CC4(C)C)=O)CCO3)cc21 N1(C(C(CC)CC)=O)C2CCC1CC(NC(=O)C(O)Cn1cncn1)C2 CC(N=c1ccnc(N2CCC(c3ccnn3C)C2)[nH]1)c1cn[nH]c1 C(=O)(C1CCCc2nc[nH]c21)NC1CN(C(C(CC)(F)F)=O)CC1C C1(C(=O)NC2C(CNC(Cc3n(C)ccc3)=O)CC2)CC2(C1)CC(F)(F)C2 c1(CC)nc(CNC(=O)C(=O)NC2(c3ncon3)CCC2)c(Br)s1 N1(CC(CC(C)(C)O)O)CC2(CCCCC2)CC1CO C1(C(N(CCCN(C(COc2ccc(OC)cc2)=O)C)C)=O)CCC2C1C2(F)F C12(CCOCCC(=O)NCc3ncc(Cl)cn3)CCC(CC1)C2 C1(CNC(C(C2CCC2)OCC)=O)(NC(=O)CC2OCCO2)CCCCC1 O=C(C1=CC2CCCCC12)NCC#CCNC(=O)C1Cc2ccccc21 Cc1ccnc(O)c1C(N1CC2CC(NC(=O)CC3CCS(=O)(=O)CC3)C2C1)=O C1(NC(c2nc(OCC)oc2)=O)CCCCN(CC(c2ccccc2)(C)O)C1 c1(C(N2CCC(C)(CNC(C(C)(C)CCF)=O)C2)=O)nc2ncccn2n1 Cc1cc(C(F)F)oc1C(=O)NC(C)CN(C)C(c1ncc(C(F)(F)F)n1C)=O C1(C(N(CC(C)(C)C(=O)NC2CC3CCCC3C2)C)=O)Cc2ccccc2C1 c1(N(CCOCC)C)nnc(-c2ccccc2F)n1CC1CCSC1(C)C c1(C(=O)NCC2(NC(C(C)=C(CC)C)=O)CC2)c[nH]c2cc(F)c(F)cc2c1=O Cc1nc(C)n(O)c1C(N1CCN(C(=O)C(C)C(F)(F)F)C(C2CCCC2)C1)=O CON(C)S(=O)(=O)c1ccc(C(N2CCN(C(c3cc(F)c[nH]3)=O)CC2)=O)cc1 c1(CNC(=O)NNC(c2cc(F)c(F)cc2O)=O)ccc2cnccc2c1 N1(C(C(C)n2cccn2)=O)CCCC(NC(=O)CSCc2ccc(F)cc2)CC1 c1(NCCSC2CCN(CCO)CC2)nccc(=NCc2cc(F)cnc2Cl)[nH]1 N1(C(C(C)(N(C(Cc2ccc(C)nc2)=O)C)C2CC2)=O)CCCC(C)C1CO N1(c2snc(C)n2)CCSCC1CCNc1ccc(-c2ccccc2)cn1 C1(C(=O)NCCN(C(C2CCC2c2nc[nH]n2)=O)CC)CCNC(=O)C1 C(CCC(C(=O)N(C)CCN(C)CCO)NC(=O)C=C(C)C(C)(C)C)OC C1(C(=O)NCC(C(=O)OC)C)CCN(C(=O)C=CC(C)C)CC1C(N)=O N1(C(COC)=O)CCOCC(NC(=O)NCC2(c3cc(C)cc(C)c3)CCC2)C1 C1(C(N(CC(NOC)=O)CC)=O)CCC(C)CN1C(=O)CN1CCC(F)CC1 C1(C(C)C)CC(CC(=O)NC2CCN(C(=O)C3=CCCS3)C2C)CCO1 N1(C(CC2N(CC)CCOC2)=O)CC2CCC(C1)N2C(=O)C(O)CN(C)C C#Cc1cccc(C(=O)NCC23CC(NC(C4CC4(F)F)=O)(C2)C3)c1Cl C(=O)(C1=CCN(C(c2ccc(C)c(C)c2)=O)CC1)NC(C1CCOC1)C#C Cc1cc(C(=O)NC2CC(C(=O)NC(C)C(C)(C)C)C2(C)C)n(C)n1 C(CS(=O)c1ccccc1)Oc1c(OC(c2nc(C3CC3)no2)C)cccc1 Cc1nc(C(C)(C)C)ncc1C(=O)NC1CC1NC(C1CC(=O)N(C)C1)=O C1(C(=O)NCCC2(C)CCN(C(CC3CC(OC)C3)=O)C2)Cc2ccccc2O1 c1(CC)ccccc1S(=O)(=O)N1CCCC(CCN)C1 N1(CC(=O)N(CC=CC(=O)NC2CCC(OC)C2)C)CCC(C)CC1 C(=O)(C(C(C)C)N(C)C)N1C(CNC(CC2(CSC)CC2)=O)CCC1 C12(C(N3CC(N(C(C4(CC)CCCCC4)=O)C)C3)=O)CCC(F)(CC1)CC2 c1(CC(C)OC)nc(C2=NOC3(CCOC3)C2)n(-c2c(F)cccc2F)n1 CC1(C)CC2(CC(C(=O)NCC(N3CCN(C(C45COCC4C5)=O)CC3)=O)C2)C1 C12(C(=O)NCC(C)NC(CC(F)(F)F)=O)CCOC1CCOC2 CC(C(=O)NCC(C(C)(C)C)NC(=O)COC1CCCCCC1)S(N)(=O)=O c1(C(N2C(C)C(NC(c3snnc3C3CC3)=O)CC2)=O)ccc(Cl)c(F)c1 C1(NC(C=CC)=O)CC12CCN(C(=O)C(F)CCC(=O)C=CC(=O)OCC)CC2 C(CCC(C)(C)C(=O)NC(CC)C(C)O)NC(CCC=C=C)=O c1(OC)ccc(Cl)cc1C(F)(F)C(=O)NCC1CN(C(=O)C(C)N(C)C)CC1O Cc1c(O)ccc(C(N2CCC(CNC(=O)CCC3CC3(C)C)C2(C)C)=O)c1C N1(CCNC(=O)Nc2cnc(CO)cn2)c2ccccc2Sc2ccccc21 c1(OC)cc2c(c(S(=O)(=O)NC3c4ccccc4C4CC3C4)c1)OCC2 c1(-c2cn(C(C)C(=O)NCc3ccc(Cl)s3)nn2)cnccc1OC(C)(C)C c1(C(=O)NCC2N(C(Cc3c(C)n[nH]c3)=O)CCCC2)ccc(Br)cc1C#N CC(C)(C)CC(C(=O)N(CCC#N)CCN1CCOCC1)N1CCC1c1cccs1 c1(CC)c(C(=O)NCC2CCCC(NC(c3cc(C)on3)=O)C2)nnn1CC N1(CC)N=C(C(=O)N2CC(OC)C(NC(=O)C(C)CO)C2)CCC1=O CN1CCN(CC(C)(C)C(=O)Nc2ccc(C)s2)CC1.C12CCC3CC13N2 C1(NC(C(CC2CC2)NC(c2c(C)cccn2)=O)=O)CCC(O)C(O)C1 c1(C(N2CC3C(C(=O)NC(C4CCOC4)C)(C3)C2)=O)cc(Cl)cc(Cl)c1 Cc1cc(CC(=O)NC2(C)CC(C(N3CC(O)(CO)C3)=O)C2)nn1C CC1(C)CC(C(=O)NCC2(C)CCCN2C(C2CC23CCOC3)=O)CCO1 Cn1cc(CC(=O)NC2CN(C(=O)C=CCN3CCC3)CC2F)c2ccccc12 c1(OCC#C)ccc(C(=O)NCc2cc(C3CC3)on2)cn1.C1(=O)C(=O)NC1 C1(CNC(CC2CCN(C)C2=O)=O)Cc2ccccc2CN1C(c1cnsn1)=O CCC(CCCC(=O)N1CCS(=O)C(C)C1)NC(C1CCN(C)C1)=O Cc1cccc(OCC(=O)NCC2(NC(=O)CC(C)C3CC3)CCOCC2)c1 N1(C(C(CCOC)C)=O)CC(NC(c2ccnc(C)c2N)=O)CC(C)C1 N1(C(C2N(C(C(C)N(C(C)=O)C)=O)CCCCCC2)=O)CCC2(C=CCO2)CC1 c1(C(N2C(C)CC(NC(C3(COCC)CC3)=O)C2)=O)cncc(Br)c1C N1(C(C(CCCC)C)=O)CCCC2(CCN(C(=O)C(c3c(C)noc3C)C)C2)C1 N1(C(C(C)NC(CC)=O)=O)CCCC(C2CCCN(C(c3cccs3)=O)C2)C1 c1(C(=O)OC2CC(CCC(=O)OC)C2)ccc(Cl)c(NC(=O)OC(C)(C)C)c1N C1(C(=O)NCCn2c(C)nnc2)CC2CC1CC2NC(=O)COC(C)C N#Cc1cc(F)ccc1C(=O)NCCC1CCC(NC(C2(C3CC3)CCC2)=O)C1 Cc1n[nH]c2cnc(C(=O)NC3CN(C(=O)CNC=O)C4CCCCC34)cc12 C1(N(C(=O)CCn2cnnn2)CC)CCN(C(=O)CN2CCOCC2)C1 C(C(=O)Nc1cn(C)nc1C)(C(C)C)NC(CCc1onc(C)n1)=O C(=O)(CCC(C(=O)N(C1CN(C(c2cc(C)ccc2Cl)=O)C1)C)N(C)C)OC c1(C(=O)NC(c2cn(C)nn2)C(=O)NCC(C)N(C)C2CC2)nc(=N)cc[nH]1 C1(C(C)C)CN(C(=O)Cc2nccn2C)CCC1NC(=O)CN(C)S(N)(=O)=O C1(NC(c2ccc(C)c(N)c2)=O)CCC12CCN(C(C1CC1(Cl)Cl)=O)CC2 C1(C(NOCCC(=C)C)=O)C2CN(C(C3CCC(C)(C)C3)=O)CC12 N1(C(C2OCCC(C)C2)=O)CC2CCCC(C1)N2C(=O)C=CSc1ccccc1 CCC(F)(F)C(=O)N1CCCC1CNC(C1CCCCC1n1cccn1)=O C(=O)(C(C)(C)C(=O)NCC1C(C(=O)NC2(CC(F)(F)F)CC2)CCC1)OCC c1(C2(C(=O)NCC(CNC(C(F)=CCC)=O)F)CCCC2)c(F)cccc1F C1(C)(CCC)CCN(S(=O)(=O)Cc2ncoc2CCC)C1 O=C1OC(C(=O)OCCOC2CCCC2)Cc2ccc(F)cc21 c1(CC)cc(C(N2CCC(CN(C)C(c3nccnc3Cl)=O)CC2)=O)c(C)nn1 C(CCC(C(=O)NCCc1cccc(O)c1)NC(=O)Cn1nc(C)oc1=O)OC C(CC(C)C(=O)NCCCN(C)C(c1ccc(C(C)F)cc1)=O)=CCC c1(C(=O)NCC2OCCN(C(C=C(CCC)C)=O)C2)ccc(Cl)c(C(=O)OC)c1 N1(c2nnc(C)o2)CCC(C2CCCN(C(C3CCN3Cc3ccccc3)=O)C2)C1 N#Cc1ccc(=NC2CCCCN(C(c3cnc(Cl)c(Cl)c3)=O)C2)[nH]n1 CC1(C)C(C(=O)NCC2CC(NC(=O)Cn3cccn3)C(O)C2)CCS1(=O)=O C(=O)(C1=NOC2COCC12)NC1C2CC(NC(c3cc4n(n3)CCO4)=O)CC21 c1(C(=O)NC2C(C)CN(C(c3cn(C)cn3)=O)C2)cc2[nH]ccc2s1 N1(CC(=O)NC(C)C(CO)NC(=O)CC2CC2(C)C)C(=O)CNC1=O c1(CCCC(=O)NC2CC23CC(NC(c2occc2F)=O)C3)ccc(O)c(F)c1 c1(C(C)(C)F)cc(C(=O)NCC2C=CCN2C(c2cncc(F)c2)=O)ccc1F O=S(=O)(c1ccc(NCC(Cl)(Cl)Cl)c2cnccc12)NC1CC(Cl)(Cl)C1 C(=O)(C(C)C(C)S(C)(=O)=O)N1C(C(C)C)CN(C(=O)CCC(F)(F)F)CC1 CC(F)(F)C(C)(C)C(=O)NCC1(C2(O)CN(C(=O)Cc3cccc(F)c3)C2)CC1 C(CCN=C(NCC1CCCC1O)N1CCC(C2CC2)C1)OC c1(C(=O)OCC)cc(C(C)NC(C2(c3ccn(C)n3)CC2)=O)c[nH]1 C(=O)(C1=NOC2(CCC2)C1)NC(C(C)(C)C)CNC(=O)COCc1cccnc1 C(CC1=CCN(C(C2(CCN(C)C)CC2)=O)CC1)NC(C(C)OCC)=O c1(CC)sc(C(=O)NC(C)(C)C(C)NC(c2ccc(OC)o2)=O)cc1Br c1(C(=O)NC(CC)CNC(=O)CCOc2ccccc2)cc([N+](=O)[O-])ccc1O CC12CCCCC1CN2C(C1CN(C(C2CC2Cl)=O)CC12CC2)=O CCC(C)CC(=O)C(=O)NCCCN(C(=O)Cc1cnsc1)CC C(CCCN=[N+]=[N-])NC(C(C)N(C(=O)CSc1cn[nH]c1)C)=O c1(-c2n(C)ccc2)ccc(C(N2CC3CC2C3CNC(c2ccc[nH]2)=O)=O)cc1 CCC(C(=O)N(C1CC1)CC)N(C(=O)CN1CCOCC1)C c1(C(N2C(N(CC(N3CC(C)(O)C3)=O)C)CCC2)=O)cc(O)nc(O)n1 N1(C(C(Cn2cncn2)NC(c2cnsn2)=O)=O)CC2CC2(CO)C1 C1(C)(CCNC(C2CC(C)OCC2)=O)CCN(C(=O)CCSCC(N)=O)CC1 N1(C(CC2(CSC)CC2)=O)CCCCC(C(=O)NCC(O)CCO)C1 N1(C(C2ON=C(C)C2C)=O)CCC2CN(C(c3ccc4sncc4c3)=O)CC2C1 C(=O)(CC(C)CN(C)C)N1CCC(C2N(C(C3C(CC)OCC3)=O)CCC2)C1 c1(C(=O)NC(C(=O)N(CC(C(=O)OC)C)C)C2CCOC2)ccnnc1C C(=O)(C(C)(C)C1=CCSCC1)N1CC(O)(C(C)NC(C2CC3CC2CC3O)=O)C1 c1(CC(=O)NC2CCN(C(c3coc(Br)c3)=O)C2)ccsc1Br C(=O)(C(CNC(=O)C(F)=C(C)C)CC1CC1)N(CCN(CC)CC)C Cc1cccc2sc(C(=O)NCC(CO)NC(c3cc(CO)on3)=O)c(Cl)c12 C1(F)(CNC(CCSCCCC)=O)COCCN(C(=O)CC(O)CC)C1 C(=O)(CC1=CCN(C)CC1)N(C1C2CN(C(c3cccc(C)n3)=O)CC21)C N1(C(C2(C(C)NC(=O)CCN3CCCC3=O)CC2)=O)CCC2(CCO2)C1 N1(CC(F)(F)F)CCCC(NC(=NCc2n(C)ncn2)NC2CCS(=O)(=O)C2)C1 N1(C(c2onc(CC)n2)=O)CC2CC(NC(C3CCCS3)=O)C2C1 Cc1c[nH]c(C(=O)NCCC(C)NC(c2cn[nH]c2)=O)c1C CCC(C)C(O)CC(=O)NC1(C)CC(C(N2CC(CO)C(O)C2)=O)C1 N(C1c2cc(Br)ccc2SCC1C)C(CCCOCC=C)=O c1(C(C)C)ccc(C(=O)NCCCN(C(=O)CC2CCCOC2)C2CC2)cn1 Cc1nn(C)c(C)c1OCC(=O)NC(C1CCN(C(=O)CCn2ccnn2)C1)C C(N=c1[nH]c(N2CC3CC2CN3C(C)(C)C)nc2c1SCC2)c1n(C)ncc1 C(=O)(C(C)(C)C(=O)NCC(CNC(=O)C(CC1CC1)CC1CC1)CO)NC CS(=O)(=O)C1(C(N2CCCC(F)(CNC(C3CC3Cl)=O)C2)=O)CCC1 c1(C(c2cccs2)NC(COCC)C(C)C)cc(C)c(OC)cc1C C(=O)(CC(C)(C)CNC(c1cncn(C)c1=O)=O)NCC(=C)Cl C(=O)(CCCCCCCC1CC1)N1CC2(C(NC(=O)CC3=CCOCC3)CC2)C1 CCCCC(O)C(C)C(=O)NCC1N(C(c2cc(OC)nn2C)=O)CCC1(C)C C1(C(N2CCC(NC(CC3CC(OCC)C3)=O)(CF)C2)=O)CCn2ncnc2C1 c1(C(=O)NCC(C)=CC(=O)NCC(C)(CO)CO)cnc(O)cc1C C1(C(=O)OC)CC2(CC(NC(=O)N(CC(C)OC)C)CCO2)C1 N1(C(c2cccc(C(N)=O)n2)=O)CC2CCC2(NC(C2Cc3nccn3C2)=O)C1 c1(C(N2C(C(=O)NCCc3ccccc3)CC(O)C2)=O)ccc2nc(Br)sc2c1 c1(C(N2CCC(F)(C(=O)NC3(CCC)CC3)C2)=O)c(O)cccc1F N1(C(c2cnc(CC)[nH]2)=O)CC(CO)C2(CCN(c3nncs3)CC2)C1 c1(N2C(C(=O)Nc3ccc(N(CC)CC)cc3)C(C)CC2)ncnc2[nH]c(C)nc12 C1(C(N2CCC(N(C(COC(C)C)=O)CCO)CC2)=O)CCC2C(CC1)C2(F)F c1(C(C)(C)C)cc(NCc2ccc(Br)cc2C(=O)O)nc(Cl)c1 Nc1nccnc1C(=O)NCC=C1CCN(C(=O)CCC2CCCC(=O)N2)CC1 CCC(C(=O)NCCn1cc(CNC(C2CN(C3COC3)C2)=O)nn1)C(C)O c1(C(N2C(CCC(N3C(CC)CCC3)=O)CCC2)=O)cc2cnccc2nc1C C(=O)(CC(C)(C)CNC(C1(F)CCCCCC1)=O)NC1CCCC(C(C)C)C1 C(C(C)(C)CCNC(c1cscc1C(=O)Nc1cnc(C2CC2)o1)=O)OC C1(NC(c2cc(C3CC3)cc(F)c2)=O)CN(C(C2(CO)CCC2)=O)CCC1CO CN1C(C(=O)NC(C2CCCC2)CNC(=O)CC2(C3CC3)CC2)CCS1(=O)=O C(C1CN(C(C2CCCC(=O)N2)=O)CC1C(=O)NCCN(CCCF)C)=CC C(CCCC(=O)NCC1CC1NC(=O)Cc1cncn1C1CC1)SC C#CCC(CC#C)C(=O)NC1CN(C(C2CCS2(=O)=O)=O)CC1C c1(CNC(C2(COC)CCN(C(=O)C=CCCC(C)C)C2)=O)nc(C)ccc1C N1(C(C2CCN(OC)CC2)=O)CCN(C(c2cnn(C3CC3)c2C)=O)CCC1C N1(C(C2CCN(C)C2=O)=O)CC(CNC(C2(C)CC2(F)Cl)=O)OC(C)(C)C1 C(c1ccc(O)cc1)=CC(N1CCC(C(C)(C)C)(CNC(C(N)=O)=O)C1)=O c1(CC)cccc(C(=O)NCCCC(CO)NC(C2CCC(N(C)C)C2)=O)n1 c1(OCCC(=O)NC2CN(C(C3C(F)(F)C34CC4)=O)C2)cccc(Cl)c1.OC Cc1c(C(=O)NC2CN(C(=O)CC3(CO)CC3)C3(CCC3)C2)c[nH]c2nccc1-2 C1(C(=O)OC)CCCC(C(=O)N(CC(C)CNC(=O)C(C)Cc2ccco2)C)C1 N1(C(C=CC)=O)CCC2(CCCN2C(C2CCSC(C)C2)=O)C1 C(CC(C)(C)C(=O)N1CC(NC(C2CC=CCC2)=O)C(C(F)F)C1)SC c1(C(=O)NC(C(C)NC(CCSC)=O)(C)C)cc(Cl)c(Cl)cc1C C=CC1(C(=O)N(CC(C)(C)C#N)C)CCN(C(c2cc[nH]c2C)=O)C1 Cc1[nH]nc2c(C(=O)NC(C)CCCCNC(=O)CC(C)C(F)(F)F)cccc12 Cc1cc(C(C(=O)NCCN2CC3CC3C2)C(C)(C)C)ccc1F CN=c1[nH]cc(C(N2C(C(=O)N(C)CC3(N(C)C)CCC3)CC2C)=O)o1 Cc1cc(F)c(C(N2CCC(F)(c3cn(CC(C)C)nn3)C2)=O)cc1F CS(=O)(=O)c1ccc(-c2cccc(N3CCN(S(=O)(=O)c4ccc(Cl)s4)CC3)c2)nc1 N1(C(CSCC)=O)CC(NC(=O)CCCc2sccc2C)CC(O)C1 C=CCC(C(=O)N1CCC(CC=C)(C(=O)NCCN2CC(OC)C2)C1)N(C)C N1(C(C2(C#C)CCC2)=O)CC2CCC(CNC(C3CC3(C)C(F)F)=O)C2C1 C1(C(N2CCCC(CNC(CCCC(=O)OC)=O)C2)=O)CCc2ncccc2C1 C1(C(N2CCCC(CNC(C(C=CC)O)=O)C2)=O)CNc2ccnn2C1 C1(CC(=O)NCC(C)N(C(=O)C(C)(C)C#N)C)CCC(F)(F)CC1 Cc1cc[nH]c1C(=O)N(CC(O)CN(C(=O)C(F)CC1CCOC1)C)C Cn1cnc2[nH]c(C(=O)NC3CC(CNC(c4cccc(F)c4O)=O)C3)cc12 c1(C(=O)NC(CC(C)NC(=O)Cc2c(F)cncc2Cl)C)csc([N+](=O)[O-])c1 CCC(CNC(=O)C(C)OCC1CC1)(CC)NC(=O)CNC(C1CCCC1)=O CCCCC(C)CCC(=O)NCCC(C)(C)C(=O)N(C(C)C(=O)OC)C c1(C(N2CC(N(C(=O)CNC(N)=O)C)C(C)(C)C2)=O)c[nH]c2cc(F)ccc12 C1(NC(C2CC(=C)C2)=O)(COC)CCN(C(c2cnn(CCOC)c2)=O)C1 c1(CC(=O)NC2(C)CCCN(C(C3CC(SC)C3)=O)C2)ccc2c(c1)CCC2 C(CN=c1cc(NCc2nc(C(F)(F)F)cs2)nc(C)[nH]1)NS(CC)(=O)=O N1(C(C(C)SC)=O)CCC1(C)CC(=O)N(CC(C)COC)C N1(c2c(C)ccc(C)n2)CCC(NC(c2snnc2C)=O)CC(C)(C)C1 CC(CC(F)(F)F)C(=O)NC1CCCCN(C(C2(C)CC2C(F)(F)F)=O)C1 C1(C(N2CCCC(C)(CNC(c3sccc3Cl)=O)C2)=O)CC2(C1)CC21CCC1 C1(CNc2nc(C)sc2)C2CN(OC(F)F)CC12.c12cccc(c1)OC2=O c1(OC)ccccc1N1CCC(NC(=O)CNCC2(F)CC2(F)F)C1 N1(C(CCOCC(C)(C)C)=O)CCCCC1c1ccc(C2(O)CCCCC2)o1 N1(C(Cc2cn(C)nc2)=O)CC(NC(C2(CC(F)F)CCC2)=O)CC(O)C1 c1(C(=O)NC2CC(COC)C2)cnn(CCNC(C2(C)CCOC2)=O)c1 N1(C(CC(COC)C)=O)CCN(C(=O)Cc2ccsc2C)CCC1C N1(C(Cc2cc(C)sc2)=O)CCC(CNC(=O)CCc2c(C)noc2C)CC1C c1(NC(=O)OCC)ccc(C(=O)OCSC2CC2C)cc1 c1(C(=O)NCCN(C(C2C3C4CCC(C4)C23)=O)CC)cc2cnccc2[nH]1 CC1CC(C(=O)NCC(C)(C)CO)CN(C(C2(C(F)F)CC3(CC3)C2)=O)C1 C12(C(N3CC(OCC)C(NC(=O)CCSCC(C)C)C3)=O)CCCC(C)(C1)OC2 C1(NC(CCC(C)NC(CCNC(=O)OCC)=O)=O)C2CCCCCC12 C1(C(N(C2CC(NC(=O)C3=CCOC3)C2)C)=O)CC2CCC(C1)C2 C1(CNC(C(C)OCOC)=O)CCCCN(C(C2C3CCCCCC23)=O)C1 c1(NCc2cn(CC)nc2)cccc2cc(O)ccc12.C(=O)(CCCCCBr)NC CC1(C(=O)NCCC2CCC(F)(F)CC2)CCCN(Cc2ccc(F)nc2)C1 C(=O)(C(C)(F)C(C)(C)F)N1CCOCC(NC(C(c2ccccc2F)OC)=O)C1 CC1CCCc2ncc(C(=O)NC3CCCCC3NC(C3(C#N)CC=CC3)=O)n21 c1(C(N2CC[Si](C)(C)CC2)C(=O)NCC2(C(=O)OC)CC2)sc2ccccc2c1Br C(=O)(C(CCS(C)=O)N(C)C)N1CCC(CN(C(C=Cc2ncc(C)[nH]2)=O)C)C1 c1(OCC(=O)NC(C)CCCNC(=O)CCNC(=O)CO)nn(C)cc1[N+](=O)[O-] C1(CNC(C(C)OCCOC)=O)CN(C(c2oc(SC)cc2C)=O)CC(C)(C)C1 c1(C(N2CC(NC(=O)C(c3cccc(Br)c3)O)C(O)C2)=O)c(F)cc(Cl)cc1Cl c1(C(=O)OC)ccc(NC(C2CC23CN(C(=O)Cc2ccsc2)C3)=O)cn1 CS(=O)(=O)c1ccc(C(=O)NCC(C2CCC2)NC(=O)Cc2cncnc2)s1 c1(OC)ccc(Cl)cc1C(=O)NC(C)CNC(c1nnc(O)nc1O)=O C1(CNC(C(COCC)C)=O)CCC(NC(=O)C(C)(C)C)CC1 CCCCC(O)C(C)C(=O)N1CCC1C(=O)Nc1ccc(C2CC2)nc1 N1(C(C2CCN(C(c3cnn[nH]3)=O)C2)=O)CCCCCC1CCO N1(c2cc(SC)ncn2)CCCC(CNC(c2ccc(C)cc2)=O)CC1 C(=O)(CCC(=O)NC(C)CN(C)C(C1CCCN1Cc1nnn(C)n1)=O)OCC C=CC(C)C(=O)N1CC(O)(C(F)C(=O)N(CC(C)C(C)C)CCOC)C1 c1(C(N2CCCC(CCNC(C(CC#C)O)=O)C2)=O)ccnc2cc(C)ccc12 N1(c2ncc(C)cn2)CCN(C(c2ccc(OC(C)C)cc2)=O)CCC1C Cc1cc(N(C(=O)CC(C(F)F)NC(c2cc([N+](=O)[O-])n[nH]2)=O)C)cc(C)c1 CC(C)(C(=O)OCC1(Cl)CCC1)Sc1ccccc1 C(=O)(CCCCC#N)NCC(C)CNC(C1CCCCCC1)=O N1(C(COCCOCC)=O)CCCC(CCNC(C2(C)CCCCC2)=O)C1 c1(C(N(CCN(C(=O)CN2CCC(C)(O)C2)C)C)=O)ccc2sc(O)nc2c1 N1(C(c2cncc(C)n2)=O)CCCC(C)C1CCNC(=O)C(F)(F)CC1CC1 c1(CC)nn(C)c(Cl)c1C(=O)NCC(O)CCNC(c1coc(OC)n1)=O CC(C)C(O)C(=O)N1CCCCC1CCN(C(=O)CC(C)O)C N1(C(c2cccc(SC)c2)=O)CC2CCN(C(=O)C(C(C)O)N(C)C)C2C1 C1(C)(CC)CC(NC(=O)C2CC2)CN1C(C1(c2cccnc2Cl)CC1)=O C#CCCC(C(=O)NCC(=O)OC)NC(=O)C(CC)CC=C c1(C(N(C)CC2(NC(C(CCC)C#N)=O)CC2)=O)ccc2c(c1)C(=O)N(C)C2=O c1(-c2nnc(C(C)OC(c3cc(Br)cc(F)c3O)=O)o2)ccc([N+](=O)[O-])cc1 c1(C(N2CC(CN(C(C(CCC)C)=O)C)C2)=O)c(C)nn(C)c1C C12(CNC(c3n(C)ncc3Cl)=O)CC(CO1)N(C(=O)CC(C)(C)C1CC1)C2 C1(CC(=O)N(CCCN(C)C)CCNC(C(C)n2ccnc2)=O)CCCC1(F)F c1(C(N2C(C)CC(NC(C3(CF)CC3(F)F)=O)CC2)=O)cc2ccc(F)cc2s1 C1(C(=O)NC(C2(O)CCC2)C)CCC(C2CC2)N1C(c1cnns1)=O C1(C)(C(N(CCCNC(c2ccc(C)s2)=O)C)=O)CCc2ccccc2C1 CC(CC(=O)NC(C)(CNC(C1(c2ccncc2)CC1)=O)C1CCC1)NC(N)=O O=C1OC2CN(C(C34CSCC3C4(F)F)=O)CC2O1 c1(C(C(=O)NCCCSC)NCCCN(C(C)C)C2CC2)ccc(F)c(I)c1 N1(C(C(C(C)C)SCC)=O)CC(NC(C2CCC(C)(C)CC2)=O)C2CC2C1 Cc1cc(NC(=O)NCC(c2cc(F)ccc2C2CC2)(F)F)c(Br)nc1C C(=O)(C1=CCS(=O)(=O)C1)NCCC1OCCN(C(c2cc(C#N)sc2)=O)C1 CC(C(=O)NCCCN(C(=O)C(C)(C)Nc1ccccc1)C)C1=CCCC1 c1(OC)ccc(C(N2CCN(CCN3C(C)CCC3C)CC2)=O)cc1C(F)F N1(C(COC(C)=O)=O)CC2(C(=O)NCCCS(C)=O)CC1CO2 C1(C(C)NC(c2cc(CCCO)on2)=O)CCCN(C(=O)COC2(C)CCC2)C1 N1(C(C2(C)CCC(O)CC2)=O)CCC2(CCCCN(C(=O)Cc3cscn3)C2)C1 N1(C(CCC2CCCN(C(c3ccn(C4CC4)n3)=O)C2)=O)CC2CCCC(C2)C1 C1(NC(=O)C=CCc2ccccc2)CCN(C(=O)COCC2CC2)C(C2CC2)C1 CC1CN(C(c2ccsn2)=O)CCN1C(C1CC2C=CC1C2)=O c1(NC(c2ccccc2OC)CCC)ncnc(NCC2CCC(C)(C)O2)c1C C1(NC(C2(CS(N)(=O)=O)COC2)=O)CCCCN(C(C2CC23CCOC3)=O)C1 C(=O)(CCCCCC#N)N1CC(CC(C)NC(c2c(CC)nc(C)o2)=O)C1 C(=O)(C(O)CC(C)(C)C)NCCC(C)NC(c1csnc1Br)=O N(C(=S)N1CCC(N2CC(NC(=O)OC(C)(C)C)CC2=O)CC1)C(CC)C c1(C(N2CC3CC(NC(c4cc(C)on4)=O)C3C2)=O)n[nH]c2c1CCSC2 c1(CC)cccc(C(N2CCC(C)(CC(=O)NCCC3CC(=O)N(C)C3)C2)=O)n1 C(=O)(C1=CCCC1C)N(CC)CC1CCCN1C(=O)CN(c1ccc(Cl)cn1)C C(=O)(CC(CC)C(C)(C)C)N(CCCCCC)CCNC(c1csc(=N)[nH]1)=O N1(C(c2c(C)cno2)=O)CC(CNC(c2n[nH]c3c2COCC3)=O)N2CCC1C2 N1(C(c2ncc(OC)nc2)=O)CC(O)CCC1C(=O)NCCc1ccco1 Cc1c(C(=O)NCC(C)(C)CN(C)C(C2CCS(=O)(=O)N2)=O)ccn1C(C)C C1(CC(=O)Nc2cccc(C(C)C)c2)CC2(C1)CN(Cc1ccncc1O)C2 C(=O)(C(C)(C)CC1CC1)N1CCC(C(C)NC(CCOCCOC)=O)C1 CCC(CC)CC(F)C(=O)NC12CCC(C(=O)NCCCc3ncco3)(CC1)C2 CCC(CC(=O)NOCCN(C)C)NC(=O)Cc1cnnn1C c1(C(=O)NC(CNC(c2c(CCC)occ2)=O)C2CCC2)ccc(CSC)cn1 CC1C(C)N(C(CC2CCC(F)(F)CC2)C(=O)NCCCF)CCS1=O CCC(C)CCCC(=O)NCCCNC(=O)CC1CC2CCC(C1)N2C C1(NC(C(C)C2CCC2)=O)CCN(C(=O)Cc2ccc(Cl)cn2)CC1F c1(C(N2CCC(C)(NC(C(C=C=C)C)=O)C2)=O)cc(S(=O)(=O)C(C)C)ccc1Cl c1(C(N(CC(CC)NC(C2CCCCN2CC(F)F)=O)C)=O)c(C)n[nH]c1C N1(C(CS(CC)=O)=O)CCC(C2CC(NC(=O)CSC3CCCC3)C2)CC1 c1(-c2cncc(NCc3cc(OCC)cc(C)c3)c2)cc(F)c(F)c(F)c1 c1(C(N2CC(NC(c3n(CC)ccc3)=O)C3C2C3)=O)ccc2nc[nH]c2n1 c1(C(N2CC(OCCNC(=O)CCCC3CC3)C2)=O)cccc2c1CCOC2 c1(CCCC(=O)N(C(C)CNC2CC(=C3CCC3)C2)C)ccccc1Cl CC1(C)CC(CNC(=O)C=Cc2cccs2)CN1C(=O)CN1CCSCC1 N1(C(C(=O)NC(c2nccs2)C)=O)CCCC2OCCC12 N1(C(C2=CCC(C)CC2)=O)CC2CC(NC(=O)CCC3CCOCC3)CC(C2)C1 C(=O)(CCCC(CC)CC)NCCN(C(C(CC#C)C)=O)CC1CC1 C1(C(N(CCCN(C(=O)CCCc2ccsc2)C)C)=O)CCc2nnnn2C1 N1(C(c2ccc(C)c(O)n2)=O)CCC2CN(C(=O)CCCCC3CC3)CC12 C(=O)(C1OCCn2ccnc21)NCC1N(C(COc2cc(C)on2)=O)CC1 c1(C(=O)NC(C(=O)N(C)Cc2cncnc2)C2CCCO2)ccc2nccn2c1 C1(CC=C)(C(=O)Nc2ccc(CCF)cc2)CCN(C(=O)CC2COCCO2)C1 c1(CC(C)C)cnc(N(C)CCN(C)C(c2cccc(Cl)c2)=O)nc1 C(=O)(CCCn1cc(CCC(=O)OC)nn1)NC(COC(CC)=O)(C)C c1(C(C)=O)ccc(C(=O)NCC2(O)CN(C(c3coc(C(N)=O)c3)=O)C2)cc1F CC1(C)CC(CNC(C2(C)CC=CCC2)=O)CN1C(=O)CC1CC(=O)NC(=O)C1 C#Cc1ccc(F)c(C(=O)N(C(C)CNC(c2cncc(C)c2C)=O)C)c1 Cc1c(C(=O)N(C)Cc2cccc(C(=O)NO)c2)nnn1C1CCCCC1 Cc1sc(C(=O)NCCCN(CCCNC(C2CCN(C)CC2)=O)C)c(C)c1C c1(C(=O)NCC(C)(C)NC(C2C(OCC)C2)=O)ccc(=N)[nH]c1Cl n1(CC)cc(Br)c(C(=O)NCCN(C(=O)CN2CCC(C)CC2)C2CC2)n1 C(=O)(C1c2ccccc2CC1NC(=O)CC(C)(C)C(C)(F)F)OC c1(OC)cc(C)c(C(=O)NCC#CCNC(c2nc(C)sc2Br)=O)cn1 C1(C(=O)NCCC(=O)NC)COC2(CCN(Cc3ccsc3Br)CC2)C1 N1(C(CCc2nnc(C)o2)=O)CCN(C(=O)C(C)C(O)CC)CC(C)(F)C1 C1(C(=O)NCCCNC(C(c2cccc(Cl)c2)OC)=O)Cc2cc(F)ccc2O1 c1(C(=O)NC2CC(CC)(CC)N(C(=O)NC)C2)[nH]c2ccc(C(C)=O)cc2c1C N1(C(C(CCC)CNC(C2(C#N)CCCO2)=O)=O)CCc2nc(C)[nH]c2C1 N1(C(C2C(C(=O)OCC)CC2)=O)CC(NC(=O)C(CC)(CC)OC)C2(CC2)C1 N1(C(c2cn(C)c(=O)cn2)=O)CCCC2CCN(C(=O)C(C)(C)CC(F)F)CC12 Cc1ccc(SCC(=O)NCCC2(C)CCN(C(C3CC(N(C)C)C3)=O)C2)cc1 N1(C(c2ncc(C)s2)C(=O)NCC=C)CCc2sc(Cl)cc2C1 Cc1cc(Cl)c(C(=O)NC2CC3C2CCN3C(=O)C(C)c2ccco2)c(Cl)c1 N1(C(C(C)(C)c2cscn2)=O)CC2CC(NC(C3(C)CCC(F)(F)C3)=O)C1C2 c1(C(=O)NC(CN(C(C2CCCOCC2)=O)CC)C)cc(C)cc(OC)c1C CCCCCC(=O)NC(c1ccccc1F)CNC(c1nc(C(C)C)oc1C)=O N1(C(CC(CC)SC)=O)CCCN(C(c2cc(O)n(CC)n2)=O)C(C(C)C)C1 Cc1cc(C(N2CCN(C(c3sccc3CO)=O)CC(C)C2)=O)c(F)cc1F N1(C(COCC(=O)OC)=O)CCC(C(C)NC(C2(C)CNC(=O)C2)=O)CC1 Cc1nn(C)c(Cl)c1CC(=O)NC1CN(C(C2CC2F)=O)CCC1C(F)(F)F N1(C(CC)=O)CCCCC1c1nc(-c2ccc(SC)cc2)nn1C(C)CC CCC(C(=O)OC)C(=O)N1CCCC(N(C(=O)COCCNC(C)=O)C)C1 c1(CC)cc(Br)cc(CC)c1NC(=O)CC(C)(C)CCSC N1(C(C=CCOC)=O)CC2(CC(NC(=O)C=Cc3cc[nH]c3)C2)C1 C#CCCCCCC(=O)N1CCCC1C=CC(N1CC(n2ccnn2)C1)=O C(C(=O)NCc1ocnc1C(=O)NC1(C(F)F)CCCC1)(C(C)C)SC CC(C)(O)C(C)(C)C(=O)NCC1CCCC(CNC(c2n[nH]c3c2COC3)=O)C1 C(=O)(C1=CCCC1(C)C)N1CCN(C(CCCC(=C)C)=O)C(CCOC)C1 Cc1cc([N+](=O)[O-])cc(C(=O)NCCCC2(NC(=O)C(=O)N=S(C)(C)=O)CC2)n1 C1(C(N2CC(CC(C)NC(=O)CCCc3cnn[nH]3)C2)=O)CCC2CC2C1 n1(C(CC)CC)nccc1C(=O)NCC(C1CC1)N(C(=O)CNS(N)(=O)=O)C CCC(CC(=O)NC1CC2CC(C1)CN(C(c1cc(F)n[nH]1)=O)C2)C(C)(C)C C(=O)(CC(C)C(F)F)NCC1CCC(C(=O)NC(c2cn(C)nn2)C)CC1 C=C(C)CCC(=O)NC1C2CCN(C(C3CC3c3ccccc3)=O)C12 C1(NC(C2C(CCC)CN(C(C3(O)CCSCC3)=O)C2)=O)CCCC1C1CC1 N1(C(c2ccc(CCCCCC)s2)=O)CC(NC(C2CCC(=O)N2C)=O)C(SC)C1 C1(CN(C(C(C)OCCC=C)=O)CC)CCN(C(c2cccc(C)c2)=O)CC1 C1(C(N2CCC(O)(CN(C(C3(CCC=C)CC3)=O)C)C2)=O)CCS(=O)(=O)C1(C)C c1(C(F)F)cc(N(C2CCC2)C2COC2)n2ncnc2n1 CN1C(=O)NCC1C(N1CC2C(CNC(c3cc(C4CC4)[nH]n3)=O)C2C1)=O c1(CN2C(C(=O)Nc3c(C(=O)OC)n(C)nc3)COCC2)ccc(F)c(F)c1F c1(C(=O)OC(C)C(=O)Nc2nccs2)n[nH]c2c1COC2 N1(C(C(C)NC(C)=O)=O)CC2(CCN2C(c2cnc(O)c(F)c2)=O)C1 Cc1ccc2c(N3CCC(CO)C3)nc(=NC3CCN(C)C3)[nH]c2c1 N1(C(C23CCC(OC)(CC2)C3)=O)CCC2(CCN(C(=O)C(F)C3CCC3)CC2)C1 C(C)(c1cnccn1)=CC(=O)N(c1cccnc1Br)C(C(=O)OCC)C c1(C(N2CCCC3CC(F)(F)CCC23)C(=O)NCC)ccc2c(c1)C=CC(C)(C)O2 c1(C(N2C(C(=O)Nc3cccc(Br)c3Cl)CC(C)C2)=O)cc2ccccn2n1 c1(NC)ccccc1C(N1CC(CNC(=O)CC2CCCSC2)C1)=O Cc1cncc(CC(=O)NCC(O)CNC(c2ccc(C(N)=O)[nH]2)=O)c1 N1(C(C2CC(C#C)(O)C2)=O)CCCC2CN(c3nc(CC)nc(Cl)c3F)CCC12 N1(c2n(CC(COC)(C)C)c(-c3ccc[nH]3)nn2)CCN2C(=O)C(=O)NCC2C1 N1(C(C(CC=C)C)=O)CC2CCC1C(NC(=O)CNC(c1cscn1)=O)C2 c1(OC)cc(C(=O)NC2CN(C(=O)CCCCCO)CC2F)cc(Br)c1Cl C(=O)(C1CCCn2ccnc21)N(CCC(c1cccs1)NC(=O)C=CCO)C N1(C(CC2N(C(C)=O)CCC2)=O)CCN(C(c2cc(C(C)(C)C)no2)=O)CC1C c1(OC(C(=O)N(CCC(C)NC(=O)C=C(Cl)Cl)C)C)ccc(C(F)(F)F)cc1 C1(NC(C(C)NC(N)=O)=O)(CO)CCCN(C(c2ccc(CO)o2)=O)C1 N1(C(c2cc(CC)[nH]n2)=O)CCC2CN(C(c3cc(F)c(Cl)cc3F)=O)CC2C1 CCC(C)C(O)CC(=O)N1CC(CC(N2CC3CC(OC)C(C3)C2)=O)C2(CC2)C1 N1(CCC(C)C(F)F)C(=O)CCN(Cc2ccc(OCC#N)cc2)C1=O C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)NCC1CCC(NC(=O)CCCCC2CC2)C1 C(C(C)C)(C(O)C(=O)NCCSCC(=O)Nc1cc(O)ccc1C)OC C(CNC(=O)C(C)CC)(CC(F)(F)F)NC(c1c(CC)c[nH]c1)=O N1(C(CCCCNC(Cc2ccn(C)c2)=O)=O)CCC(O)C(F)C1 CC(C)C(C)C(C)Cc1nc(-c2ccc(Cl)nc2)nn1C1CSC1 Cc1c(Br)ccc(CN=c2ccc(C(=O)Nc3ncc(C(C)=O)s3)c[nH]2)c1F N1(C(Cc2n(C)ccn2)=O)CCCCC(CNC(C23CC(C(F)F)(CO2)C3)=O)C1 c1(C(N(CC(C)N(C(C(CC#C)C2CC2)=O)C)C)=O)cc2n(n1)CCCC2=O N1(C(c2ccc(C(OC)OC)o2)=O)CCCCCC(NC(=O)CCS(C)=O)C1 C1(CC(=O)NC2(NC(=O)C(O)c3ccsc3)CC2)CCC2CC12.C1CC1 CC1C(C)N(C(c2nncn2C)C(=O)NC(C)(C)C)CCS1(=O)=O C1(CNC(C(CC)n2ccnc2)=O)C2CN(C(=O)Cc3n[nH]cc3Br)CC12 C12(CNC(c3cnc(O)c(F)c3)=O)CCC1CN(C(c1csc(Cl)c1)=O)C2 N1(S(CCCC)(=O)=O)CCN(Cc2c(C)cccc2Br)CC1C#N c1(CC)onc(C(=O)NC(c2ccccc2)C(=O)NCC#CC#CCO)c1C CC1(C)CCCC(CN=C(NCC(F)F)NCC2CC(C(F)F)C2)O1 Cc1cccc(N2CCCC(NC(N3C(C)CC3(C)C)=O)C2)c1 C(CCCC(=O)NC(CCN(C)C(c1sc(F)cc1C)=O)C(C)C)OC N(C(=NCc1cccc(C(F)(F)F)c1)NCc1cnns1)C(CC)C c1(OC)ccc(C(=O)NC(CNC(c2cscc2F)=O)C2CCC2)cc1 C1(O)(CNC(C(C)NC(CC)=O)=O)CCN(C(c2cnc(Cl)[nH]2)=O)CC1 c1(-n2ccc(C)n2)cccc(C(=O)NCC2CC2CO)c1 C=CCC(C)(C)C(=O)NC1CCC(CNC(c2c(C)nn(C)c2C)=O)CC1 Cc1oc([N+](=O)[O-])cc1C(=O)NC12CC1CN(C(C1CCC(=O)N1)=O)C2 c1(NCc2cn(CCn3cc(C(=O)OC)nc3C)nn2)ccc(C#N)nc1C c1(CC(=O)NC2CCN(C(C3CSC3)=O)CC2F)ccc2ncsc2c1 C1(NC(COCCC(C)C)=O)CC(CNC(c2cc(F)ccc2Cl)=O)C12CCC2 c1(C(N2CCC(CCOC)(NC(CCOCC)=O)C2)=O)nncc2c1CCCC2 N1(C(C2C(CCC)C2)=O)CCCCC2(C1)CN(C(c1cc(F)ccc1CC)=O)C2 C1(C)(NC(C(C)NC(=O)Cn2cnnn2)=O)CCCN(C(c2occc2Cl)=O)C1 N1(C(C(CCC)N(C)C)=O)CCC2C(CCN2C(c2cc[nH]n2)=O)C1 n1(CCOC)cc(C(=O)NCC(C(C)C)NC(C2(N3CCCC3)CCC2)=O)cn1 C1(CNC(C(C)(O)C2CCC2)=O)CC2(CCN(C(C3CC(C#N)C3)=O)CC2)CO1 N1(C(C2(C)C(C)C2)=O)CCC(F)(F)C(CNC(=O)C(C2CC2)C2CC2)C1 C(=O)(C(O)Cc1ccccc1)N(CCNC(C(C)N(CC)CC)=O)CCOC C(=O)(C(F)CC(C)(C)NC(=O)CN1CCCCC1)NCC(C)(C)CO c1(C(N2CCC3(C(C(=O)NCc4ncn(CC)c4)C3)C2)=O)cccn2cncc12 N1(C(c2cc(CC)nn2C)=O)CC(C)CCC1CNC(c1csc(COC)c1)=O C1(C(C)C)(C(=O)NCCc2cn(C)cn2)CCCN1C(C1COC(=O)N1)=O CCCC(C(=O)NCCC1CCCN1C(=O)C=Cc1ccc(CC)o1)NC(C)=O CC1CCC(=CC(=O)NC(C)(C)CC=CC(=O)NC2C(C)C2C)CC1 c1(CN(CC(C2COCCO2)=O)C)ncc(Cl)cc1Cl C1(NCc2[nH]nc(-c3ccc(OC)cc3)n2)CCC(C)NC1=O C(=O)(CC(C)(C)C(=O)NCC1CN(C(=O)COC2CCOC2)CC1O)OC CCCC(C)(O)C(=O)N(C)CC1CCN(C(=O)CCCCN2CCOCC2)CC1 C1(CCNC(C=CC)=O)CN(C(C2CCCC(C(=O)OCC)C2)=O)CCN1C C12(CNC(C3C(C)OC(=O)N3)=O)CC(CO1)N(C(C1CC3(CC3)CO1)=O)C2 N1(C(C2N(C(CSCC#C)=O)CC=C2)=O)CCOC(C(=C)C)C1 C1(C(N2CCC(CN(C(C34CCCC3C4)=O)CC)CC2)=O)CC(=O)NC(=O)N1 c1(NC(C2N(Cc3cccc(C)c3)CCNC2)=O)cc(Cl)cc(Cl)c1Br C1(NC(C(C)OC(C)(C)C)=O)CC(F)(F)CN1C(N)=O.C12CN(C1)C2=O CN1CCN(C(=O)C=CC2CC2)C(CNC(c2csc(-c3cnccn3)n2)=O)C1 C1(NC(C2(CCOCC)CCCC2)=O)COC2(C1)CN(C(=O)C(C)(C)COC)C2 C1(NC(CCCCC)=O)CC(C2CCN(C(c3c(C)cc(F)cc3C)=O)C2)C1 c1(C(N2CCC(O)(CN(C(c3c(C)n(C)nc3)=O)C)C2)=O)ccc(F)cc1Cl c1(NC(C(=O)NC2CCN(C)C2=O)=O)cc(Br)cc2[nH]ccc12 c1(C(=O)NC(C(=O)NCC(C)(C)SC)CC2CC2)c[nH]c(=O)cn1 N1(C(C2(C)CCC2)=O)CC2CCCC(NC(c3ncc(Cl)s3)=O)C2C1 C1(C(N2CC(CNC(Cc3c(C)noc3)=O)C2)=O)CCCC(=O)N1C c1(C(N(CC(C)NC(c2cc[nH]c(=N)c2)=O)C)=O)nnc2ccccc2c1O N1(C(c2c(COC)scc2)=O)CCCC(C)(NC(=O)CC2CC2C)C1 N1(C(C(Cn2cccn2)NC(C(C=C)OC)=O)=O)CCOC(CF)C1 C1(C(=O)NCC2C(C(=O)NCc3cnc(C)[nH]3)CCO2)CN2CCN1CC2 c1(C(=O)OC)nc(=NCCN(C(c2cc3sccc3cn2)=O)C(C)C)c(C)c(C)[nH]1 N1(C(c2c(CC)[nH]cc2)=O)CC2CCC(C1)N(C(C13CC(C(C)C)(C1)C3)=O)C2 c1(C2C(C(=O)NCCN(C(C)C)C(C3CCC4CC34)=O)C2)cccc([N+](=O)[O-])c1 c1(CC(=O)NC2CCCN(Cc3sccc3Cl)C2)c(Cl)cccc1Cl c1(C(=O)NCC2CC(NC(C(COC)C)=O)C2)ccc2c(c1)S(=O)(=O)NC2 N1(C(CC)=O)CCN(C(C2CCCN2S(=O)(=O)CC)=O)CC1Cc1ccccc1 N(C1CCOc2c(C)cccc21)C(c1n(C(CC)(C)C)nnn1)CCC1(C)CC1 Cc1cc(C(=O)NCC(C)(C)CNC(c2cc(O)n(C)n2)=O)cnn1 c1(OCC)ccccc1C1(C(=O)NC2CCCOC2)CC1.N12CC3C(C3C1)C2 c1(NC(=O)NC(C2CCCC2)CC)c(-c2ccc(F)cc2)nc2ccc(C)cn12 C=CCCCC(C(=O)OC(C)(C)C)NC1CC(C(=O)OC)C(O)C1 C1(NC(C2C(C)(Br)C2)=O)CCN(C(=O)C(=Cc2ccccc2)C#N)CC12CCC2 O=C1NCc2c(C(N3CC4CC(NC(C56CC5C6)=O)CC3C4)=O)cccc21 c1(NCC2CCN(CC)C2)[nH]c(=NCc2ccc(C)o2)nc2sccc12 CC1CCN(C(=O)C(C)(C)Cc2cnn[nH]2)CCN1c1ccc(C#N)cn1 c1(C(C(=O)OC)N(C2CCC(C)(C)C2)C)cc(Cl)cc(Cl)c1 CC1CCC(NC(=O)Cc2cnoc2)CN1C(=O)CCOC1CC1 CC1CC(NC(=O)CC(C)(O)c2ccccc2)CN1C(C1(c2cc[nH]n2)CC1)=O C=CC1(CNC(=O)CC=CCNC(C2(Cl)CC2C(C)=O)=O)CCOCC1 C1(=CC(=O)N(CC(C)(C)NC(C(C2CC(C)(C)C2)OC)=O)C)CCN(C)C1 CC(C)CC(C(=O)NC1C=CC(C(=O)N(C2CCCCC2)CCO)C1)C(N)=O c1(CC)ncnc(NC(C2C(C(N3CCCC3c3ccc(Cl)cc3)=O)C2)=O)c1F c1(C(=O)NCC(C)(CC)NC(C(C)OCC)=O)cc(-c2ccccc2)ccc1O CC(CN=c1[nH]c(=N)[nH]c(=NCc2cccc(Cl)c2F)[nH]1)C(C)(F)F O=S(=O)(Oc1ccc(OC(F)F)c(F)c1)c1csc(N2CCOCC2)n1 n1(CCC(=O)NCCC(C)NC(c2n(CC)ncc2)=O)ccc2cc(Cl)ccc12 O=S(=O)(C=Cc1ccc(F)cc1)NCc1cncnc1 c1(OC)cc(Cl)ccc1NC(C1(C)CCN(Cc2c(O)cccc2F)CC1)=O c1(OCCC(=O)N(CCCNC(C2C3CCCC23)=O)C2CC2)ccccc1Cl O=C(C1=Cc2ccccc2C1)N1CC2CC1CCC2NC(C1CC(O)C1)=O c1(C(N2CC(C(=O)OC)C(C)(C)C2)C(=O)NCC(F)F)cc(Cl)c(F)c(Cl)c1 C1(CC)CN(C(=O)CC2CN(C(c3ccnc(OC)c3)=O)CCO2)CCN1C c1(C(=O)NC2CC(CCNC(C3OCCN(CC)C3)=O)C2)csc2c1CCCC2 c1(C(N2CCC(CNC(=O)Cn3ccnn3)C2)=O)ccc(C(O)CF)cc1 c1(N2CCCC(CNC(CCOCCN(C)C)=O)CC2)ccc([N+](=O)[O-])cn1 CC1(C2CCCN(C(C34CCCC3CCN4C(C3CCNC3=O)=O)=O)C2)CC1 S(=O)(=O)(c1ccc(NCCCCCCF)cc1Br)N1CC(CC)OCC1 C(=O)(C#CC1CCCC1)NCC1N(C(CCc2ccc(N)cn2)=O)CCC1 N1(CC(=O)NCC2C=CCN2C(c2cnn(C3CCCCC3)c2)=O)CCOCC1 Cc1sc(Cl)nc1C(=O)NC(CNC(=O)CCCC1CCC1)CO CC(C(=O)NCC1CCC(NC(=O)Cn2ccnn2)CC1)C(=O)N1CCOCC1 c1(OC)cc(CCC(=O)NCC2CCOC2)cc(OC)c1O CCC(C)(C)C(C)CC(=O)N1CCCC1CNC(=O)C(C)=CC1CC1 c1(C(N2CCCCC(NC(C(CC)=CC)=O)C2)=O)cnc(O)c2cncn12 C1(C(N2CCC(NC(COCCOC)=O)C(F)C2)=O)COc2cc(Cl)ccc2O1 c1(C(N(CC(C)N(C(C(CCSC)OC)=O)C)C)=O)cc2c(F)c(F)ccc2[nH]1 C1(NC(CC(C)C)=O)(CF)CCN(C(c2ccc(C(N)=O)cn2)=O)C1 CC(CCO)C(=O)NC(CNC(=O)Cc1nncn1C)CO C1(N(C(CN(C(C)=O)C)=O)C)CN(C(=O)C(F)C2CCOC2)C1 N1(C(C(C)Cc2ccco2)=O)CCC2(CC1)CC2NC(c1ccc(CO)cc1)=O C(=O)(C1=CCCCC1C)N1CCCC(C(=O)NCCn2cccn2)(CC)C1 C12(NC(CC)=O)CCN(C(=O)Cn3nc(C(F)F)cc3C3CC3)CC1C2 c1(C(N2CCC(N(C(=O)CNC(N)=O)CC)C2)=O)cc(Br)cc2cccnc12 c1(CC)ncccc1C(=O)NC(C)(C)CNC(=O)C(c1ccc(Cl)nc1)(F)F C(CCC(=O)NCCN(C(=O)C=CCOCC)C1CC1)=CCC=C c1(NC(C2CCC(NC(C3(CCCF)CC3)=O)CC2)=O)cc(Cl)ccc1O N1(C(C(n2ncc(C)c2)C)=O)CCCN(C(=O)CC(C)C)CCC1 c1(C(=O)NCC2(CNC(C3CCCC3O)=O)CC2)cnc2nc(O)nc(O)c2c1 C(=O)(C(C#N)CC1(C(=O)OC)CCC1)N(C(C)CCn1cccn1)CCN(C)CC.CC C(=O)(C(F)C(F)(F)F)NCC(CNC(C1C(CN(C)C)C1)=O)(C)C c1(-n2cc(-c3cncc(C(N(C)C)=O)c3)nn2)ccc(S(=O)(=O)CCO)cc1 C1(C(N2CC(OCC)(CNC(=O)Cc3c[nH]nc3O)C2)=O)CCCCN1C CC1(C)COCCC1C(N1CCOC(c2cn(CCCCO)nn2)C1)=O N1(C(C2CC(=C)C2)=O)CCN(C(c2nc(C)oc2-c2ccccc2)=O)CCC1C CC1(C)CN(C(C23CCCC2C3(F)F)=O)CCC1C(N1CC(S(C)(=N)=O)C1)=O c1(CN(C(C2N(C(=O)C3=CC4C=CC3C4)CCCC2(C)C)=O)C)ccc2cc[nH]c2n1 C(=O)(C1CCCc2nnn(C)c21)N(C1C2CN(C(c3ccc(F)cn3)=O)CC12)C Cc1cc(C(=O)NCC(C2CC2)NC(C2CCCCS2)=O)[nH]c1C c1(C(N2CC3C(C(=O)NCCC=C)(CC3)C2)=O)cc2cc(F)ccc2s1 C(=O)(C(C)(C)CNC(c1cc(C(C)C)no1)=O)NC1(CCCC)CC1 C1(NC(c2cn(CC)nc2)=O)CC(O)CN(C(=O)C(c2cncn2C)O)C1 C(=O)(CC(C)C(F)F)N1CC(Cn2cc(-c3cccc(OC)n3)nn2)C(C)C1 C(=O)(C1=CC2CCCCC12)N1CC(CCNC(=O)C=Cc2ccco2)C1 C12(CNC(CN(C)C(=O)OC(C)(C)C)=O)CCC(CN(C(c3ncn(C)n3)=O)C1)C2 CC1C(NC(=O)C(CO)c2ccccc2)CCN1C(=O)CCC1CCCCO1 C(C(C)(CO)CC=C)NC(C(CNC(C1(CC#C)CCC1)=O)CC1CCCC1)=O C1(CC(N2CC(CC=C)(NC(=O)Cc3nc(=N)[nH][nH]3)C2)=O)CCCC(=O)N1 C1(C(N2CC(CN(C(=O)Cc3ccn(C)c3)C)C2)=O)CCOC1c1nccn1C Cc1ccc2cc(C(N3CCC(N(C(=O)C(C)(C)C(C)C)C)CC3)=O)oc2c1 C1(C(N(C(C)CNC(=O)C(C)CCOC)CC)=O)CCC(N(C)C)CC1 c1(CN(C)C)cccc(C(=O)NC2CCCC2CN(C)C(c2cccnn2)=O)c1 Cc1cc(C#N)sc1C(=O)NC(c1ccccn1)C(C)C C(=O)(C#CC1CCOCC1)N1C(C)CCC(NC(c2c(O)nnc(C)c2C)=O)C1 c1(C(=O)NCCCC2N(C(CS(CC)=O)=O)CCC2)ccc2cnnc(O)c2c1 N#Cc1cc(C(=O)NCC2(CO)CCCCCC2)ccc1Br N1(C(CCN(C(C(CCC)OCC)=O)C2CC2)=O)CCCOC(C)(C)C1 c1(OCCCNC(c2sc(Br)nc2C)c2n(CCC)nnn2)ccccc1Cl Cc1cc(NC(c2cc(Br)cn2C)c2nnnn2-c2ccccc2)cnc1Cl C1(C(=O)NCCNC(C2CC=CCO2)=O)Cc2cc(F)cc(F)c2O1 CN1CC(C(=O)NCCC2(O)CN(C(c3cnc(S)nc3)=O)C2)NC1=O C#CCCCCC(c1nnnn1CC(F)F)NCc1occc1C CCC(CCC(=O)NC1(CCNC(c2ccc(OC)c(Cl)c2)=O)CCCC1)OC c1(CN2C(c3cccs3)CCC(C)C2)n[nH]c2ccccc12 c1(CC)ccc(C(=O)NC(C)C(C)NC(=O)CN(C2CCC2)C)cc1F C1(C(=O)NC(C)CCNC(=O)CCCC2CCOCC2)CCC(C(C)(C)C)CC1 Cc1nc(C(=O)NC2CC(NC(=O)COC3CCCC(C)C3)C2)c(=O)[nH]c1C N1(C(c2cnc(-c3ccccc3F)s2)=O)CCC12CCSCC2 c1(C(=O)OC)nc(N(C)CC2CCN(C(C3CCCC34CC4)=O)C2)sc1C c1(OC)cc(CN=C(NCC(C)(C)C)NC2CCS(=O)(=O)C2)cc(OC)c1C C1(NC(=O)COCC(F)F)(CF)CCN(C(=O)CCc2cccnc2)C1 c1(OC)ccc(C=CC#N)c(C)c1.C12CC(C1(C)C)N(CCCC)C(=O)C2 CCC(C)C(=O)C(=O)N1CCC(C(N2CC(C)(CO)C2)=O)O1 N1(C(C(C(C)C)SC)=O)CCC2CCC(NC(c3cc(C)nc(Cl)c3)=O)C1C2 C1(CNC(C2N(C)C(=O)CC2)=O)CCN(C(=O)Cc2cn(C)nn2)C12CCC2 c1(C(N(C2CCC(NC(CC3C(C)CCO3)=O)CC2)C)=O)cc(F)cc(Cl)c1 CCCCCCC(CC)(CC)C(=O)NCC(CC)NC(=O)CC1CCC12CCC2 N(C1CN(C(=O)CCCC2CC2)Cc2ccccc21)C(C(C)C(F)F)=O C1(NC(C(CC)CC)=O)COC2C(NC(c3nc(C)n(C)c3C)=O)COC12 C1(OC)CN(C(=O)C(C(C)C)NC(=O)CN2CSCC2=O)CC1(C)C C1(CNC(C(CC#C)O)=O)(NC(=O)CC2CCC3(CC3)CO2)CCCCCC1 Cc1nnsc1C(=O)N(C(C)(C(=O)NC(CO)C1CC1)C1CC1)C C1(NC(C2(C)CCC(C)C2)=O)COC2(C1)CN(C(c1c(Cl)csc1Cl)=O)C2 c1(C(=O)NC2(C)CCCN(C(C(CC)(C)CC)=O)C2)cc(OC)c(S(N)(=O)=O)s1 C(=O)(CC(C)(C)C1CC1)N1CC(CC(C)NC(CC(C)F)=O)C1 C1(C(N(C(C2CCC2)C)C)=O)CCC(CNC(c2ccc(C)o2)=O)C1 C12(CNC(C3ON=C(C)C3)=O)CC(CNC(=O)C(C)(C)n3cnnn3)(CO1)C2 N1(C(C2C(NC(C(C)(C)n3ccnn3)=O)CCO2)=O)CCOC2C(O)CC12 CC(C)CC(C)(CO)NC(C1CCCCN1C(C1OCC2CCCC12)=O)=O C1(CN(C)C(N)=O)CCCCN1C(=O)C(Cc1ccc(F)cc1)NC(=O)C1CC1 c1(CC)nccnc1C(=O)NCC1CC1C(=O)NC(COC)CCO c1(C(=O)NC2CCN(C(=O)COc3ccsc3Cl)C2)cc(Cl)cc2ccncc12 C(CCCCCNC(C1CCS(=O)(=O)C1)=O)NC(=O)CCc1ncccn1 N1(C(C2C(C)N(C(C3CCOCC3)=O)CC2)=O)CC2CCCCC2C1C c1(C(=O)NC2CCN(C(=O)C=CCN3CCCCC3)C2)ccc(Cl)c(F)c1 c1(NC(=O)OC(C)(C)C)cnc(C(N2CCC2CC2CCS(=O)(=O)C2)=O)cn1 CC#CCC(C)NC(=O)C(C1CC1)N(C(=O)C(c1ccn(C)c1)C)C C1(NC(CCC(=C)Cl)=O)CCCN(C(c2cccc(C(F)(F)F)c2O)=O)C1C c1(OC)nccc(C(N2CCC2C(=O)N(C)Cc2cnccc2C)=O)n1 CC(C)(C)C(O)C(=O)NCC12CC1CN(C(=O)Cc1nc[nH]n1)C2 C(CCCC(C)C)(C(=O)NCCOC)N1CCN(CC(CC)O)CC1 Cc1nc(CCC(N2CC(CNC(=O)CCc3cc(Cl)no3)C(O)C2)=O)oc1C c1(C(N2CCC(OCC(=O)NC3COCCOC3)C2)=O)cc2ccccn2n1 c1(C(=O)NC2(CNC(c3nc(Br)c[nH]3)=O)CC2)c(Cl)ccc2ncccc12 c1(C(=O)NC2C(C(=O)NC3C(=O)NCC3)CCCC2)ccc2nccnc2c1 Cc1cc(C(N2CCOC(C3CC3)C2)=O)nc(N(C)C)n1 N1(C(c2c(C)nccn2)=O)CCCC(C)(C)C1CNC(=O)CC(C)F c1(C(=O)NCC2C(C)CCN(C(=O)C(N)=O)C2)ccc2sccc2c1 C1(F)(C(=O)NC2CCC(NC(C3(C)CCC3)=O)C2)CS(=O)(=O)CC12CCC2 c1(N2C(C)CCC2C(=O)Nc2ncc(F)cc2Br)ncnc2c1CCCC2 N1(C(CC(C(CC)(C)C)C)=O)CC(NC(=O)C2CC2)C2(CCS(=O)(=O)CC2)C1 c1(C(=O)NC(CCNC(c2nc(C)oc2)=O)C)c[nH]c2nccc(Cl)c12 C1(NC(c2n(CCCOC)nnn2)c2sccc2OC)CCCCCC1 C1(C(N(CCC(O)C(=O)NC2CC(C)(C)C2)C)=O)CCCC2(CC2)C1 N1(C(C(CC)NC(N)=O)=O)CCC(C)C(NC(=O)CC(C(F)F)n2ccnc2)C1 N1(C(CC2C(NC(C3(OC)CCSC3)=O)CCCC2)=O)CC(C)CCCC1C C(c1ccccn1)=C(C)C(=O)NC(C)CNC(c1ccnc(N(C)C)c1)=O n1(CC)ncc(Cl)c1C(N1CCCC(C(C)(O)CNC(=O)Cn2nccn2)C1)=O c12ccccc1CNC(=O)NC(C)C2.N1(C(=O)NCC(=O)OC)CCCC1 C1(NC(c2ccc(OC)cc2OC)=O)CN(C(=O)C(O)C(C)(C)C)C2(CCC2)C1 c1(CNC)cccc(N(C)C)c1.C12CCCN1C(=O)NCC(C)C2 N1(C(CC2(N(C)C)CC2)=O)CCC2(C=C(C(=O)NCCC3CCN(C)C3)C2)C1 c1(C(=O)NC(c2ccccn2)CC)nc(CNC(C2C(C)(C)C2(F)F)=O)oc1C N1(C(CCCN(C(C)C)C)=O)CC(O)CC1(C)C(=O)NC1(c2cccnc2)CC1 C1(C(N2CC(CCCCNC(C(CC)OC)=O)C2)=O)CN(CP(C)(C)=O)C1 c1(C(N2C(C)CN(C(=O)Cn3cc(C(F)F)cn3)CC2)=O)cncc([N+](=O)[O-])c1 c1(C(=O)NCC2CC(CNC(CCCOC)=O)OC2)cc(Cl)cc(Cl)c1 c1(OC)cc(C(=O)NC(C2CCCN2C(C2OCC2(C)C)=O)C)ccc1C(N)=O N1(C(c2cc(Br)nn2C)C(=O)NCCCOC)CCC(S(C)(=O)=O)C1 CC1(C)CN(C(=O)CC2C=CCC2)C1C1CCN(C(C2CC(F)(CO)C2)=O)CC1 N1(C(CCCCC#C)=O)CCN2C(=O)C(NC(c3cn(C4CC4)cn3)=O)CC2C1 n1(CC)nc(C)c(C(=O)N(C)CC2CCCN(C(=O)C=CC3CC3)C2)c1Cl c1(CC(N2C(C(C)C)CN(C(C34CC(C3)C4)=O)CC2)=O)cc(F)c(F)cc1F C1(C(N2CC3CC2C3)C(=O)NCCSC)CCC(C(C)(C)C)CC1 C1(NC(c2sccc2C2CC2)=O)(CNC(=O)CC2CCC2)CCCC1 CC1OCCC1(C)C(=O)NC1CC(NC(c2cccc(C(N)=O)n2)=O)C1 CC(C)C(C(=O)N1CC2CCN(C(C3CC4CC3C4)=O)C2C1)C(C)C CCC(CC)C(C(=O)NC(C)CC1CN(C(c2c[nH]nc2C(F)F)=O)C1)OC c1(CNC(CCN(C)C)=O)csc(C(=O)NC2CCN(CCCO)C2)c1 C1(C(=O)NC2CC(CNC(C(CCSC)O)=O)C2)SC2C=CC1CC2 N1(C(C(c2cccs2)OCC)=O)CC(n2cc(CCNC(N)=O)nn2)C(O)C1 c1(N(CC(CC)(C)OC)C)nncc2c1cnn2C Cn1cc(C(=O)NC2CC2NC(C23CCCCC2NC(=O)C3)=O)c(=O)n(C)c1=O C1(C)(C(=O)NCC(CC)NC(=O)C(O)Cc2cnc[nH]2)CCCCNC1=O C1(CNC(Cc2c(C)nn(C)c2)=O)CN(C(C2CCCC23CC3)=O)C(C)(C)C1 c1(C(=O)NC2C=CCN(C(CC=C(C)C)=O)C2)c[nH]c2c(F)cccc2c1=O C1(C)(C(N2C(C(C)NC(c3n[nH]c(O)n3)=O)CCC2)=O)CCCCCC1 C(C)(C)(CCC(=O)N(C(CC(F)F)C(=O)NCC(C)CC(C)C)C)OC n1(CCC)cncc1CNC(=O)OCC12CC(NC(=O)NC(C)(C)C)C1C2 c1(C(=O)NCC2N(C(C3C(F)(C(=O)OC)C3)=O)CC2)cc(-c2ccncc2)[nH]n1 N1(C(=O)C=C2CCC2)CCC2CN(C(C3(F)CC=CCC3)=O)CC2C1 Cc1cc(NC(=O)Cc2ccccc2O)ccc1NC(C1CCS1(=O)=O)=O c1(C(=O)NCC2CC(NC(C3CCCCC3)=O)C2)cnc2ccc(Cl)cn2c1=O C1(CC)CN(C(=O)C(=O)NCc2cncs2)CC2(CCCOC2)O1 Cc1cc(C(=O)N(C(C(=O)NC2CC3(CCC3)C2O)C2CC2)C)c(O)nn1 C=CCC(C)(CC)C(=O)N1CCC(C(=O)NC(c2ccc(C)o2)CC)O1 Cc1cccc(C(N2CC(NC(=O)CC=CCSc3ccccc3)C(C)C2)=O)c1 c1(CC)c(C(N2CCOC(CC(=O)NCc3nnn(C)n3)C2)=O)nnn1C C1(CC(N2CCN(CCOc3c(C)occc3=O)CC2)=O)CC(C)CC(C)(C)C1 C1(C(=O)NC(C(=O)NCCCS(C)=O)Cc2cc[nH]n2)CC2(CC2)CO1 Nc1cnc(C(=O)NCCCCC(=O)NCCC2(O)CCC2)cn1 CC1(NC(c2ccc(O)nc2)=O)CCN(C(C2CCN2C2CCCC2)=O)CC1 C1(CCNC(CCN(CCC)C)=O)CCN(C(c2snnc2CC)=O)C(C)C1 C(=O)(C(C)C(C)(C)C)N1C(C(=O)NCc2c(C)ccs2)C=CCC1 N1(C(CCC(C)NC(=O)C(C)NC(=O)C(C)(C)C)=O)CCc2ccccc21 N1(C(COC2CC(NC(c3c(CC)cncc3)=O)C2)=O)CCOC(C)(C)C1 Cc1cc(NC(=O)C(c2ccc(Cl)cc2Cl)O)ccc1NC(=O)C1=CCC1 C(=O)(N=c1[nH]n(-c2ncccn2)cc1C)Nc1cccc(C)c1O c1(C(N2CCC(C(C)CC(=O)Nc3nn(C)cc3Cl)C2)=O)ncncc1F N1(C(C=CCCC)=O)CC2CCC2(CNC(c2c[nH]nc2C2CCCO2)=O)C1 N1(C(CCCC#C)=O)CCC2CCC12CNC(=O)COCCC c1(C(N2C(C)C(C(N3CC(C(C)O)C3)=O)CC2)=O)cc2cccnn2c1 C#CCCCC(=O)NC(C)CCN(C(=O)CNC(=O)C(CC)CC)C C1(C(N2CCC(F)(F)C2)=O)CN(C(=O)CCc2nncs2)C2(CCC2)C1 Cc1cc(C(=O)NC2CC(CNC(=O)C=CC(C)C)C(O)C2)c(N)c([N+](=O)[O-])c1 Cc1nc2c([nH]1)CC(C(N1CCC(CO)(CNC(c3cnsn3)=O)CC1)=O)CC2 c1(C(=O)NCC(CNC(c2cc(Cl)ns2)=O)O)cn2c(n1)CCCC2 CN=c1nc(N2CCN(CCC(C)(C)C)CC2)[nH]c(N2CCC(NC3CC3)C2)n1 c1(OC)c(Cl)nc[nH]c1=NCC(C(C)(C)C)NC(c1ccc(F)cn1)=O N1(C(C2C(C)C2)=O)CCN(C)CC1CNC(=O)C(c1ccccc1)C Cc1cc(=NCC2CCC(NC(c3cccnc3-n3cccn3)=O)C2)[nH]c(Cl)n1 Cc1cc(C(N2CCC(O)(C(C)NC(c3ccc(Cl)o3)=O)C2)=O)ccc1C(C)C c1(CC(=O)NCC(C2CC2)NC(C2(OC)CC2)=O)c(Cl)cccc1Br C(CC(C(=O)N1CC2CCC1C2)NC(c1cnccn1)=O)N(C)C C(=O)(C1=CNC2=NCCC2=C1)N1CCC(CNC(=O)C(F)C(F)(F)F)(CO)C1 c1(CC)ncc(C(=O)NCC(C)(CO)NC(=O)CC2(NC(C)=O)CC2)[nH]1 c1(C(N2CC3(CCN(c4c(C)cncn4)CC3)C2)=O)n[nH]c2ccc(C#N)cc12 C(C(=O)NC1(C)CC1)(C1=NOC2CCCCC12)N1CC(C)(C)C(F)(F)C1 C(=O)(C(C(C)CC)NC(C)=O)N(CCC)CCNC(C12CC(O)C1C2)=O N1(C(CN(C(C(C)C(C)(C)C)=O)C2CCC2)=O)CCC(F)(F)C(O)C1 c1(C(N2CCCC(NC(C3CC4C(C)(C)C4C3)=O)CC2)=O)ccc(Cl)c(Cl)c1N CC1CN(C(c2cccc(O)n2)=O)CCC1C(=O)NCC(C)(C)C(C)(C)O C1(C(=O)NCC2N(C(C(C)=CC)=O)C3C(C2)C3)CCn2c(Br)cnc2C1 C1(NC(C2(CCOCC)CCCC2)=O)C2CC1N(C(c1cnn(C)c1C)=O)C2 c1(SC)ncc(C(=O)NCC(C2(O)CN(C(=O)C(C)(O)C3CC3)C2)(C)C)s1 C1(C(N(C2CC(NC(c3nc(OCC)oc3)=O)C2)C)=O)CCC(C)CC1 CC1(c2ccc(Br)cc2)NC(=O)N(CC(=O)NCC2CC2CN=[N+]=[N-])C1=O Cc1cc(C(=O)NC(C2CC=CCC2)C(=O)Nc2csnc2C)cnn1 C1(OC(=O)CC2CCC23CCC3)CCOC2(CCC2)C1 C12(CC)CC(CC(=O)NCC(C)CNC(C3CCN(CC4CC4)CC3)=O)(CO1)C2 C1(CNC(CCC2CCC(NC(=O)CCCC3CCCO3)C2)=O)CC2C=CC1C2 C(CCC(=O)NCc1occc1C(N1CCC1CO)=O)=CCC=C N1(C(C(CC(=O)OC)(C)C)=O)CC2COCCC2(NC(c2ccc(Cl)s2)=O)C1 CCC(CN(C)C)CC(=O)NCCC1(CNC(c2ncoc2C)=O)CC1 N1(C(C(C2CCN(C(C3(C)CCC3)=O)CC2)C)=O)CC2CCCCCCC12 N1(C(C2(CSC)CC2)=O)CC2CCC2(CNC(c2ccc(C3CC3)cc2)=O)C1 CC1CCN(C(c2cnc(C(C)(C)C)nc2)=O)CCN1C(=O)Cn1nccn1 c1(C(=O)NC(CNC(c2c(=N)[nH][nH]c2)=O)C2CC2)cccc2cc[nH]c12 C12(C(N(C)CC3CN(C(=O)COC4CCCOC4)C3)=O)CCCCC1C2(F)F C1(C(=O)OC)CN(C(c2nccc3c[nH]nc23)=O)C2CCCCC12 c1(N2CC(OC)C(F)C2)nc(=NCP(C)(C)=O)nc(N2CCOCC2)[nH]1 C(C(=O)NC1CN(C(=O)C(=O)NCC2CC2)CC1C)(C(C)C)OCCCOC N1(C(CC2(N(C(C)=O)C(C3CN(C)C3)=O)CC2)=O)CCC(F)(CC2CC2)CC1 N1(CC(N)=O)CCN(C(c2scc(Cl)c2Cl)C(=O)NCCC2CC2)CC1 C12(CNC(C=C(CCC)C)=O)CCCCC1CN(C(=O)CNS(N)(=O)=O)C2 c1(C(N2CC3C(C(=O)NC4CCC(COC)CC4)C3C2)=O)c(F)ccc(F)c1F N1(C(c2c(OC)cncc2)=O)CC=C(CNC(C23COCC(C2)C3)=O)CC1 N1(C(CC(COC)(C)C)=O)CC2CC1CN(C(C1CCN(CC3CC3)CC1)=O)C2 c1(C(N2CCC(N(C)C(c3ccccc3O)=O)C2)=O)[nH]nc2ncc(Br)cc12 c1(NC(c2c(Br)cnn2CC2CC2)=O)ccc(OC(F)F)cc1 N1(C(C(C)(C)C)=O)CC2(CCOCC2)CC1CNC(=O)C(F)(F)C(O)C1CC1 c1(NCC2C(=C)C2)nc(C)cc(=NCCn2cc(C3CCOC3)cn2)[nH]1 N1(C(C)=O)CCN(C(c2ccnc(NC3CCC3)c2)=O)C(CO)C1 c1(CNC(COCCC)=O)cc[nH]c1C(N1CCC(C(=O)OC)C1)=O c1(C(N(CCNC(C2(C)CC(=C)C2)=O)C)=O)c(C)ccc(F)c1Br C=CC(CC)CC(=O)N1CCC(CNC(C2(C(F)F)CCCCC2)=O)C1 C1(CNC(c2cc(CC)c(C)s2)=O)CC(NC(=O)CC(F)F)C12CCC2 c1(C(=O)NC(CNC(C2(OCC)CCCCC2)=O)CC)cc(C)nc(C)c1 c1(C(N(C2CC2)CC2CC2)=O)cnn(CCNCCC(=O)OCC#C)c1 N1(C(C2CN(C(C)=O)C2)=O)CCCC(F)(C(=O)NCC(C(C)C)C(C)C)C1 C1(O)(CNC(c2n(CC)ncc2)=O)CCCN(C(=O)C(C)Oc2ccccn2)C1 C12(NC(c3c(C(F)(F)F)ncn3O)=O)CCN(C(C34CC(CO3)C4)=O)CC1C2 C1(C(N2CCC(O)(COC)C2)=O)(NC(C(C)SCCCC)=O)CCN(C)C1 C12CCCCN1C(=O)COC(C)(C)CNC2=O.c1(CC)cnc(C2CC2)[nH]1 C1(CNC(C(CC)C)=O)CCN(C(C2(SC)CCC2)=O)CCC1(F)F Cc1nc2c(C(=O)NC3CCCCC3CNC(c3n[nH]cc3Br)=O)cccc2o1 c1(C(N2C(C(C)C)CN(C(C3(C)CNC(=O)C3)=O)CC2)=O)onc2ccccc12 CC(C)CC(C(=O)N(CC(C)(C)CNC(=O)CN1CCC(=O)NC1=O)C)C(N)=O C(=O)(C(C)(F)C(C)(C)F)NC(C(C)NC(c1ccc(C(=O)C2CC2)cc1)=O)=O N1(C2C(CCC=C)C2)CCCN(C(c2ccccc2)CC)CC1 CC#CCCC(=O)NCCCC1CN(C(C2(CN(C)C)CCCC2)=O)CCO1 c1(OC)c(C(=O)NC23CC(Nc4ncc(Br)cn4)(C2)C3)ccc(Cl)c1Cl c1(C(CC)C(=O)NC(C)C(C)NC(c2cc[nH]c2C(C)C)=O)ccc(F)cc1 CC1(C)CC(NC(C2CCCC2F)=O)CN1C(=O)CCSC(F)(F)F C(CO)(CCC)C(=O)NC(C#C)(C)C1CN(C(=O)C(C)OCCCC)C1 N1(C(CC2(C)CC2)=O)C(CNC(C23CC(C)(C2)OC3(C)C)=O)CC2CCCCC12 Cc1cc(C(N2CCNC(C(N3CCC(C(F)F)CC3)=O)C2)=O)nc(C)c1 C(=O)(CCC(=O)NN(C)C)NCc1c(C(=O)NCC(CC(=O)OC)C)scc1 c1(C(=O)NC2CCC(NC(=O)OC(C)(C)C)C2)ccc2cc(F)c(F)cc2n1 CCCCC(O)C(=O)NCCCCCNC(=O)C(CN(C)C)C(C)C Cc1cc(CC(=O)NC2(CCNC(c3ccsc3C)=O)CC2)cc(C)c1 CC1=C(c2ccc(NC(c3ccc4cc[nH]c4n3)=O)nc2)CCCC1 Cc1cccc(C(C)NC(=O)C(CCC2CC2)NC(c2conc2C)=O)n1 c1(NC(=O)NC2(c3ccccc3)COC2)ccc(=NCc2ccc(Br)cc2)[nH]c1 C1(c2onc(-c3cnc(C)[nH]3)n2)C2CCCOC12 Cc1ccc(C(F)(F)C(=O)NC(C)CC2CCCOC2)nc1 CC(CCCC(=O)NCCNC(C1(C#N)CC1(C)C)=O)c1ccccc1 [N-]=[N+]=NCCCCCCC(=O)NC1CC2(CCN(C(C34CC(F)(C3)C4)=O)C2)C1 c1(C(N2CCN(S(=O)(=O)CCCCl)C3CC23)=O)c[nH]c2c(Br)cccc12 C1(=O)CCC(CC2CCCC2)O1.C1(O)(C(=O)NCC)CCN(C(=O)OCC)CC1 N1(C(C(CC)C(=O)OC)=O)CC2CC(C1)CN(C(C1C3CN(C)CC13)=O)C2 C12(C(N3CC(N(C(C4CN(C)C(=O)CC4)=O)C)C(O)C3)=O)CCC(C)(CC1)OC2 N1(C(c2ccccc2F)=O)CCN(C(c2cscc2Cl)=O)C(C2CCC2)C1 C(=O)(C(C)P(C)(C)=O)NC1CC(NC(CCNC(COC)=O)=O)CC1O C1(NC(COCCCC#C)=O)CCN(C(=O)CSc2ccc(C)c(C)c2)CC1O C1(C)(C(N2CC(CNC(C(CCSC)(C)C)=O)C(O)C2)=O)CC(C(C)(C)C)=NO1 C1(CC)CCC(C)CN1C(c1ccc(C2CC2)cc1)C(=O)NC1CC1C1CC1 Cn1c(Cl)cnc1CC(=O)NCC1(NC(c2nccs2)=O)CCCC1 C1(C)(C(=O)NC(C)CCN(C)C(c2cccc(=O)o2)=O)CC(C(C)(C)C)=NO1 C1(OC)CC(CNC(c2c(C)ccn2C)=O)N(C(c2cc(C(C)=O)cn2C)=O)C1 N1(C(CCN(C(C2(C)C(C)C2)=O)CC2CC2)=O)CC(CO)CC(C)(C)C1 c1(CC(=O)NC2C(NC(CC(CC)C)=O)CCC2)c(C)nc2cc(O)nn2c1C c1(SCC)c(C2CC(F)(CNC=O)C2)nnn1CC.C(=O)(CN(CC)CC)CC c1(-c2nn(C)c(-c3cccc(Cn4cncn4)c3)n2)cc(F)cc(F)c1 C(=O)(C(=O)C(C)(C)C)NC(C)CCC(=O)N1CCC12CCC2 C(=O)(C1c2ccccc2NC1C)N1C(C=C)(c2ccccc2)COCC1 CCC(C)(C)C(O)C(=O)NCC1=CCN(C(C2(Cc3cccnc3)CC2)=O)CC1 C#CCC(C)(C(=O)NCC1(C)CSC(C)=N1)NC(C1CC1(C)C(F)F)=O N1(C(C(CC=C)NC(C)=O)=O)CCN(C(=O)C=C2CCC(C)C2)CC1CCO C1(NC(C(C(C)(C)C)O)=O)COC2C(NC(=O)CCc3n[nH]c(=N)s3)COC12 N1(C(C2CCC(C(=O)OC)O2)=O)C(CNC(c2cnn(C)c2N)=O)CC2CC12 C(=O)(C1OC(=O)c2ccccc21)Nc1cccc(NC(CC=CC(C)(C)C)=O)c1 c1(CCC)ccc(C(=O)NCCCCCN(C)C(c2cc(OC)no2)=O)cc1Cl N1(C(C(CCCC)NC(N)=O)=O)CCC(NC(C2CCCSC2)=O)C(CO)CC1 Cc1cc2n[nH]cc2cc1C(=O)NC1CCC1NC(C1CC(O)C1)=O C12(NC(CCCOC)=O)CCCCCC1N(C(c1cc(C)cnc1N)=O)CC2 C1(C(=O)NCCN(C(=O)C(c2cccnc2)C)C(C)C)CCC2(CC2)C1 C1(CNC(C(C)(Cl)Cl)=O)CN(C(=O)CCNC(c2ccco2)=O)CC12CCC2 C(CC(=O)N1CCC1CC(=O)NCCOC1(C)CCC1)SCCC C(=O)(C1=COCCO1)N1C(C2(NC(=O)Cc3ccc(Cl)s3)CC2)CCCC1 c1(C(N2C(C)COCC2)=O)cc2sccc2n1C C1(C(N(C2CN(C(=O)Cc3coc(-c4ccccc4)n3)C2)C)=O)CN(C)C(=O)N1 c1(C(=O)NCC2CCCC(NC(C3(C)C=CCC3)=O)C2)nccn2nccc12 N1(C(CC2ON=C(C)C2)=O)CCC(CCN(C)C(c2occc2F)=O)CC1 C(=O)(CCC(=O)N(C)C(C)C)N(C1CCN(C(c2cc(O)nn2C)=O)C1)CC Cc1cc(-c2cccs2)c(S(=O)(=O)N(C2CC2)CC2(O)CCC2)cc1C C1(C(=O)NCCCCCNC(C(c2cncc(F)c2)C)=O)CCC(CO)CC1 C1(NC(C2C(C)(C(C)C)C2)=O)CCC2(CCc3ccccc32)CC1 N1(C(C(C)(O)Cc2ccccc2)=O)CC2(CCCN(C(=O)C#CC3CC3)C2)C1 Cc1c(C(=O)NCCOCCN(C)C(C2CCCC2O)=O)cccc1Br c1(CNC(C(C2CCC2)NC(C(C=CC)O)=O)=O)cccnc1F C1(C(N(C)CCc2ccncc2)=O)CC12CCN(c1nnc3ccccn13)CC2 C1(NC(C(C)OCCOC)=O)CC2C(NC(c3cc(SC)c(C)o3)=O)C2C1 N1(C(=O)C=CCF)CC2C3CCC(C2C1)N(C(c1cc(O)cs1)=O)C3 CN1CCc2[nH]nc(C(=O)NCC34CCC(CC3)N4C(=O)C=CBr)c2C1 N1(C(C(COC)O)=O)CCC(CO)(CNC(=O)C=Cc2ccc(C(N)=O)o2)C1 CC(C)CC(C(=O)N1CCC(C(F)C(=O)NC2CCCC(C(N)=O)C2)C1)C(N)=O S1(=O)(=O)c2cccnc2N1.C(=O)(C(F)(Cc1ccccc1)C(C)C)OCC CCCCCCCC(=O)NC(CC(N)=O)C(=O)NC(CC)C(C)C c1(C(N2CCCC(NC(c3ccc(CC)o3)=O)CC2)=O)ccc2c(c1)OCCC2 Cc1n[nH]c(C)c1SCC(=O)N(CCN(C(=O)CC(C)F)C)C(C)C N1(C(C2N(Cc3c(Br)cn(C)n3)CC3(CC3)C2)=O)CCC2(CC1)CC(C)(O)C2 CC1(C(=O)NCC(CO)NC(c2ccccc2OC(F)(F)F)=O)CCC(=O)N1 S(=O)(=O)(c1cnn2ccc(=NCc3cc(Cl)n(C)n3)[nH]c12)N1CCC(C(C)O)C1 C1(CNC(C(C)(C)F)=O)CCCCN1C(c1cccc(NS(=O)(=O)C2CC2)c1)=O C1(NC(c2csc(CO)n2)=O)CCCCCC1C(N1CCC2CCC12)=O c1(C(=O)NC2CC(N(C)C(c3cncc(N)c3)=O)C2)ccc(Br)c(F)c1F c1(C(N2CCC(C)C2c2cn(CC3(O)CCC3)nn2)=O)c(F)ccc(F)c1Cl c1(N(C)C)ccc(C(N2CC(n3cc(C(O)C(C)(C)C)nn3)C(O)C2)=O)cc1F N1(C(C2CC(N(C)C)C2)=O)CCC2CCN(C(c3cccc(CO)c3)=O)CC12 N1(C(CC(C)(F)F)=O)CCCC(C2CCCN(C(=O)CCC3CCC3)C2)C1 c1(C(=O)NC23CN(C(c4cccc(OC)c4)=O)C(C2)C3)c[nH]c2nccc-2c1 C1(C(N2CC(C(C(=O)NCc3c(C)con3)O)C2)=O)CN(C)CCO1 Cc1cc2cc(C(=O)NC3CCN(C(=O)CCc4cccn4C)C3)ccc2cn1 c1(CC)ccc(C(C)C(=O)NC2CCC(Nc3nccc(OCC)n3)C2)cc1 C(CCCCCCN1CCCC1)NC(C(C1(C)CC1)NC(c1cnc(C)s1)=O)=O N12CCN(CC1)CCNC(=O)C2.C1(N(CC(=O)N2CCC2)C(C)=O)CCCCS1 C1(NC(C2CCN(CC)C2)=O)CC2CC(NC(C3(CC(C)C)CC3)=O)C2C1 N1(C(c2c(C)cc(F)c(Cl)c2)=O)CCC2(CC1)CCN(C(C13CC(C)C1C3)=O)C2 N#Cc1c(NC(C2(CNC(=O)CCC(F)(F)F)CC2)=O)cc(Br)cc1F C1(OC)CCn2cc(C(N3CCCC(NC(=O)C(N)=O)C3)=O)nc2C1 N1(C(C(C(C)(C)C)=O)=O)CC2CC(C(=O)NC3(C4CC4)CC3)C(C2)C1 C=CC1(O)CN(C(=O)CCN(C(=O)C=CC2(C)COC2)C(C)C)C1 c1(CC(=O)NCC2(O)CC(CNC(c3coc(Br)c3)=O)C2)ccc(F)cc1 CC1OCCCC1C(=O)NCC1(NC(c2cnc(C3CCOCC3)s2)=O)CC1 c1(CNC(C(N2CCC(NC(=O)OC(C)(C)C)CC2)C)=O)nn(C)c(Cl)c1Br c1(C(N2C(CN(C(C(C)=CC3CC3)=O)C)CC(F)C2)=O)ccc2n[nH]c(C)c2c1 CCC(C(=O)NCC1CCCC1NC(=O)CCNC(C)=O)OCc1ccccc1 C(=O)(C1=CC2(CCN(C(c3sccc3OC)=O)C2)C1)N(CCF)CC c1(NC(CCC)=O)ccc(C(=O)NC(c2cn(CC3CCOC3)nn2)CC)cc1 c1(C(=O)OC)cncc(C#CCNC(C2CCC(c3ccccc3)C2)=O)c1 CCC(C(=O)NC1(CNC(=O)C(O)Cc2ccccc2)CC1)C(C)O CCC(CC)CCC(=O)N(C(C)CCNC(c1cc(C(C)(C)O)ccn1)=O)C c1(CC(=O)NCCCCN(C)C(C2(C)CC(F)C2)=O)cc(F)ccc1F C1(NC(CC(CC)N(C)C(c2c[nH]ccc2=O)=O)=O)CCc2nncn2C1 CCC(C)CCCCC(=O)NCC1(C)CC(F)(F)CN1C(c1cccn1CC)=O C(=O)(C(CC)C(C)(F)F)NCC(=C)CCNC(c1cc(C)n(C(C)C2CC2)n1)=O c1(CC(=O)NCC2CC2NC(C2CCO2)=O)ccsc1Cl CCC(C)C(O)CC(=O)N(C)Cc1ccccc1CNC(=O)Cc1ccc(C)s1 N1(C(C2(COC)CC=CCC2)=O)CCC2(CC(NC(=O)Cn3nnc(=O)[nH]3)C2)C1 c1(CCC(=O)NCC2CC3CCC2N3C(C2CCSC2)=O)ccc2nc[nH]c2c1 c1(N(CC(=O)NC)C)nc(=NCC2CCC(c3ccccc3)O2)[nH]c2c1CCC2 c1(C(=O)NCC(CCOCC)O)ccc(OC)cc1N C1(C(=O)NC2CC(NC(c3sccc3Cl)=O)C2)(OC)CCSC1 c1(CC(=O)N(C2CN(C(C34CCC3C4)=O)C2)C)ccc(F)cn1 C1(CC(=O)NCC(CC)NC(=O)CC2(O)CCCCC2)CCN(C)C1=O N(C(=NCCCC(F)(F)C(F)(F)F)NC1CCCC1(F)F)CC(C)(C)C N1(C(C)C(N2CCCCC2CN)=O)CCCC(CNC(=O)C2CC2)C1 c1(C(=O)NC2CN(C(C(CC)CC3CCCC3)=O)CC2O)cn2cccnc2n1 N1(C(CC(C=C)(C)O)=O)CCC2(CC1)CN(C(C1(CN(C)C)CC1)=O)CC(C)O2 N1(C(C(C2CCCC2)OC)=O)CCC2C(C1)CN2C(=O)CC(C)(C)O C1(C(C(=O)NC2CCCC2)N(C2CCOCC2)CCN(C)C)CCCOCC1 C1(C)(CNC(C2(COC)CCOCC2)=O)CN(C(C2CCCO2)=O)C(C)(C)C1 C1(C(=O)NC(C2CN(C(C3(C)CCCC3)=O)C2)C)(COC)CCCO1 C1(NC(c2n(CC)nc(C3CC3)c2)=O)CC2CN(C(=O)C#CC(C)C)CC12 N1(C(C(CC)N(C)C)=O)CCC(C(F)CNC(=O)Cc2ccsc2Cl)CC1 O=C(CCCNC(=O)NC1(CCO)CC1)NCc1cc[nH]c1 C#CCC(C(=O)Nc1ccc(C(C)C)nc1)NC(c1csc(C)n1)=O C=CC1(CC(=O)NCCC(C2CC2)C2CC2)CN(C(=O)C(C2CC2)SC)C1 N1(C(C(N2CCCCC2=O)C)=O)CC(NC(=O)CC2CS(=O)(=O)C2)C2CC2C1 N1(C(C(CC)C#N)=O)CC2(CCN2C(c2ccc(C(C)(C)C)cc2)=O)C1 C1(C(=O)NCC2C(C)C2C)(NC(c2cc(CCO)on2)=O)CCC(C)(C)C1 c1(CN(C(=O)NCC(COC)C(C)C)C)c(C)cccc1F N1(n2c(-c3ccc(C)c(Br)c3)nc(-c3c(C)cco3)n2)CCCCCCC1=O C1(C(=O)NC(c2ccc(Cl)cc2)c2n(C)ccn2)C2CCC1(C)C2(C)C CCCC(C(=O)N(CC(=O)NC(C)C(=O)N1CCCC1)CC1CC1)C(C)C C(CCCOC)(C(=O)NCc1nnc(C)s1)NC(CC(CC)C1CC1)=O C12(C(N(C)CCNC(=O)CC3(O)CCCCC3)=O)CCC(C)(CC1)CO2 CCC(C)CC(C)C(=O)NCc1cccc(CNC(=O)C(c2ccccc2)O)c1 N1(C(C2(c3ccn(C)n3)CC2)=O)CC2=C(C1)CN(C(c1ccsc1Cl)=O)C2 N1(C(C2(COC)CC=CC2)=O)CC(C)C(NC(=O)Cc2c(C)noc2Cl)C(C)C1 N1(CCCNC(CC2(C)CN(C(CCc3ccc(C)o3)=O)C2)=O)CCCCC1C N1(C(c2cc(C)c(Cl)s2)C(=O)NC)CCCC(N2CCOCC2)CC1 c1(C(N(CC(C)O)CCNC(=O)Cc2ccc(Cl)s2)=O)ccc(C(F)F)cn1 Cc1ncc(C(=O)N(CCCCN(C(=O)CC2(CSC)CC2)C)C)cc1N N1(C(c2cccc(NC(CC3CCCC(C)O3)=O)c2)=O)CC2CCCC(C2)C1 c1(N2CC(CC=C)(NC(=O)CC3COCC(C)(C)O3)C2)cc(C(N)=O)nc(Cl)n1 N1(C(c2c(S(CC)=O)cccc2)=O)CCC2C(CCCN2C(c2ccc[nH]2)=O)C1 C(C)(CCC(=O)NCC1C(CNC(C2COC(=O)N2C)=O)C1(F)F)SC n1(CC)nc(C(C)C)cc1C(=O)NC1CN(C(C2C3CCC(=O)C23)=O)C1 C(=O)(C(C)(C)CS(C)(=O)=O)N(CCN(C)C(c1ccc(Cl)c(C#N)c1)=O)C N1(C(C(C)NC(CC)=O)=O)CCCN(C(C2(OC(C)=O)CCOC2)=O)CC1 C1(NC(c2ccoc2)=O)CN(C(c2cc(C3CC3)ncn2)=O)C2(CCOCC2)C1 c1(C(=O)NC2CCC(C)N(C(C3CC3(Cl)Cl)=O)C2)cccc(N=[N+]=[N-])c1 C(=O)(CC1=NN(C)C(=O)C1)NCC(C)CC(=O)NC1CC(C)N(C)CC1C C(C)(CCC#N)(c1nnnn1C1(C)CC1)NCCNC(COC)=O C1(C(=O)Nc2c(C(=O)OC)n[nH]c2)CC(F)CN(Cc2occc2Br)C1 C12(COC1)CC2.C(C(C)(C1CC1)NC(c1cscn1)=O)NC(=O)OC(C)(C)C c1(C(=O)NCCC(CNC(C(COC)C)=O)O)cc(C)c(C)cn1 Cc1ccc(CNCc2cc(C(F)(F)F)c(C)n2C)cc1-n1nnnc1C(C)C C12(CN)CCC(C(N3CC(c4ccc(F)cc4)C(N)C3)=O)(CC1)C2 Cc1ccc(C(N2CC=CC2C(N2CCOC(C(F)(F)F)C2)=O)=O)cc1[N+](=O)[O-] c1(N2CCCC(CSC)C2)ncc(S(=O)(=O)NC2CCSCC2)cc1Cl CCCC(C)C(CC)(c1nnnn1CCCC1CC1)NCCc1nnc(Br)n1C Cc1c(NCc2ccc(CO)cc2)ncnc1NC1CCOCC1C1CCCC1 C1(C(=O)NC(CNC(CNS(CCOC(C)C)(=O)=O)=O)CC)OC2CCC1CC2 N1(C(c2c(C)oc(CNC(=O)C(C)CC3CC3)n2)=O)CC[Si](C)(C)CC1 N1(C(CN2CC(CC)C2)=O)CCC2(CCN(C(=O)C=C(C)C3CC3)CC2)C(C)C1 c1(CNC(N2CC3(C)C(C)(CC3)C2)=O)ccc2oc(O)nc2c1 C(=O)(C(C)CC(C)(C)C)N(C)CC1OCCN(C(CCc2c(C)noc2Cl)=O)C1 O=C1NC2CCCC1CN(Cc1ccc(-c3ccc(OC(F)F)nc3)s1)C2 CC1(C)CCCN(C(c2cc3ccccn3c2)=O)C1C(N1CC(F)(CO)C1)=O N#Cc1cc(C(=O)NC2(CNC(c3ccc(CO)nc3)=O)CCOCC2)on1 C=CCCC(F)(F)C(=O)NC1CCCCCN(C(c2cc(F)cnc2O)=O)C1 N1(C(c2nc(Br)c[nH]2)=O)CCN(C2CCN(C(C3CCOC3)=O)C2)CC1 C(=O)(CCC(C)C)NC1(CC=C)CN(C(c2cncc(C)c2)=O)C1 c1(CCC(=O)NC2(C)CC(NC(COCc3n(C)ncc3)=O)C2)cccc(F)c1 N1(C(COCCOC)=O)CCC(C(N2CC(C3CCCO3)C2)=O)(C(C)C)C1 C1(NC(C2CC3CCC(C2)C3F)=O)CC2CCC(C1)N2C(c1ccns1)=O Cc1cc(NC(=O)CCOC2COC2)ccc1NC(c1cncnc1C(C)C)=O C(=O)(CCCC(C)(F)F)NCCC1CCCN(C(CCC(=C)Br)=O)C1 C1(CNC(C(CC=C)C)=O)CCC2(CN(C(=O)Cc3cccc(C(C)C)c3)C2)O1 Cc1ccnc(C)c1C(N1CCC(CNC(c2ccc(C3CC3)cn2)=O)CC1)=O N1(C(CCC)=O)CCC2CN(C(C3(C(C)C)CC3C(=O)OC)=O)CCC12 c1(C(N(CC(C)NC(C2(c3ccccc3F)CCC2)=O)CC)=O)cnc(C)cn1 c1(C(N2CCC(N(C(=O)C(C)C3CC3)CCC)CC2)=O)c(F)cc(F)c(O)c1F C(CCN(C)C(c1cc(CSC)on1)=O)(C(C)C)NC(CC1N(CC)CCC1)=O C(C)(c1ccc(F)cc1F)=CC(=O)NCC1(F)CC(CNC(C(C#C)(C)C)=O)C1 c1(Nc2c(C)c(N3CCN(C4CCSC4)CC3)ncn2)cnn2c1OCCC2 C(C(O)CC(=O)N(c1cccc(C)c1)CCO)NC(C1CC(OC)(OC)C1)=O c1(OC)cccc(C)c1C(N1CC(CNC(c2cc(C)sn2)=O)C(C)C1)=O CC(C)CC(C)(CNC(c1ccnc(C2CC2)c1)=O)NC(C1CC12CCC2)=O N1(C(COCc2nnc(C)s2)=O)CCOC2(CCN(C(=O)CCC3CC3)C2)C1 CC1OCCNC1C(N1CCC(O)(c2ccccc2)C1)=O C1(OC)CCN(C(=O)C(CNC(c2ccc(C(C)=O)[nH]2)=O)C(C)(C)C)CC1(C)C C12(CNC(=O)C3=CCCCC3)CCC(CNC(=O)C(F)=C3CCCC3)(CC1)OC2 c1(C(N2CC3C(NC(CC(C)N(C)C)=O)C3C2)=O)cc(Cl)cc(Cl)c1O N1(C(C(C(C)C)CN(C)C)=O)CCC(CNC(=O)CS(=O)(=O)CCO)C(F)(F)C1 NS(=O)(=O)c1cc(C(N2CC(N3CCCCS3(=O)=O)C2)=O)cc(Br)c1 Cc1ccccc1-n1nccc1NC(=O)NCCNS(N)(=O)=O Cc1ccn(CC(=O)NC2C3CC2N(C(=O)C(C)c2ccco2)C3C)c(=O)c1 N1(C(C(CN(C)C)O)=O)CCCC(n2cc(CSc3nccs3)nn2)C1 CCC(C)CCCCC(=O)NCC1CC1NC(=O)CSc1cccc(OC)c1 C1(C(=O)OC)CC(C)N1C(=O)C(C1CC1)NC(c1cn(C(C)C)cn1)=O c1(C(N2CC3C(Cn4cc(-c5ccn(C)n5)nn4)(CC3)C2)=O)n[nH]c2c1CCOC2 c1(N2C(C)C(NC(C3CC34CCSCC4)=O)CCC2)ccc([N+](=O)[O-])cc1 Cn1oc(C(N2CCC(C(F)F)(CNC(C3(c4ccno4)CC3)=O)C2)=O)cc1=O c1(C(=O)NCC(CC)Nc2nc(C)ncc2F)cnc(OC)c(Cl)c1 C1(C(=O)NCC(C(C)C)NC(c2ccncc2O)=O)C2CCN(CC2)S1(=O)=O Cn1cc(C(=O)NC2CCCCC2)c(I)n1 CCC(C)(COC)C(=O)NCCC1(O)CCCN(C(=O)CCc2ccon2)C1 c1(C(N2CCC(C(F)C(N)=O)CC2)C(=O)NCCOC)ccc2nc(C)[nH]c2c1 N1(C(c2ccn(CCCC)n2)=O)CC2CCC(CNC(=O)CCN(C)CC)C2C1 CC(C)C(C(=O)N1CC(CN(C)C(C2CCS2(=O)=O)=O)C1)n1cccc1 N1(C(C(C=C)C)=O)CCOC(CCNC(=O)Cc2c(C)cnn2C)C1 C12(CNC(C(N3CCN(C)CC3)C)=O)CCC(CN(C(=O)COC3CC3)C1)C2 C1(NC(C(c2nccc(C)c2)(C)C)=O)CC12CCN(C(C1(SC)CCC1)=O)CC2 c1(C(=O)NCC(C)(C)NC(c2cnc(NC(C)=O)o2)=O)ccc2cnccc2n1 C1(CCNC(CC(=C)C)=O)CN(C(c2ccc(C)c(Br)c2)=O)CC(C)O1 CC(C)CC(F)(F)C(=O)NCC(C1CCC1)NC(=O)CC12CCC(CC1)C2(C)C C(=O)(C(C)(C)C(N)=O)NC(CCN(C(c1c(C(C)C)ncs1)=O)C)C C(CCN=c1[nH]c2ncc(Cl)cc2s1)NC(C1(C2CCCO2)CC1)=O N1(C(CCC=C)=O)CCCC(CC)(NC(c2cnccc2N2CCOCC2)=O)C1 C1(NC(c2c(C)nc[nH]2)=O)CC2CC(C1)N(C(=O)CN1CCC(C)C1)C2 C1(C(=O)NC(CC(C)NC(C2(C)C(C)(C)C2(C)C)=O)C)CCc2nncn2CC1 c1(C(N2C(C)CCC(NC(=O)C=C(Cl)Cl)C2)=O)ccc(S(N)(=O)=O)c(Cl)c1 C1(NC(C2CC(C)OC2=O)=O)(CNC(c2coc(Cl)c2)=O)CCC(F)(F)CC1 N1(C(C2N(C)C(=O)CC2)=O)CCCC2CN(c3c[n+]([O-])ccc3[N+](=O)[O-])CCC12 CC1=NOC2(C1)CC(C(N1CCCCC(CNC(=O)C(=O)C(C)C)C1)=O)C2 c1(C(N)=O)cc2cc(NC(C34CCCC3CC(=O)CC4)=O)ccc2[nH]1 C1(CNC(=O)C=CC=C(Cl)Cl)CC2CCC1N(C(=O)CCC1CC1)C2 c1(OCCC(=O)NCC2C(NC(c3cc(C)sn3)=O)CC2)ccccc1C(C)C c1(CC(=O)NC(CCNC(c2c(C)c(N)n(C)n2)=O)C)cn2c(C)cncc2n1 N1(C(Cc2c(CC)noc2CC)=O)CCCN(C(=O)C(F)C(F)(F)F)C(C)C1.CSC C=CCCCCCCC(=O)NC1CN(C(c2ccc(C(F)(F)F)o2)=O)CC1OC C1(C(N(C(C)CN(C)C)C(=O)CC2CC(C(=O)OC)C2)=O)CC2(C1)CC2(F)F C(=O)(C(C(C)(C)C)NC(=O)CC1CC2CC2C1)N1CC(NC(=O)OCC)C1 C=CC1(C(=O)N=c2ccn(CC(C)C)[nH]2)CCN(C(=O)Cc2ccc(C)s2)CC1 c1(C(N2CCC(CC=C)(NC(=O)CC(O)C3CC3)C2)=O)cc(=O)n(C)cn1 CC1CC2(CCN(C(C3C4COCC34)=O)CC2)CN1C(=O)COCC1CCC1 c1(C(=O)NC(CCOC)CNC(c2csc(S)n2)=O)cc(COC)oc1C CC1C(NC(c2cnn(C)c2C#N)=O)CCCN1C(=O)CCOC1CC1 c1(C(=O)NCCc2ccc(Cl)c(Cl)c2)nc(Br)n2c1CCCC2 C1(NC(C(C)O)=O)CCCN(C(c2ncsc2Cc2ccccc2)=O)C1 c1(C(=O)NC2(CNC(c3nnc(O)nc3O)=O)CCOC2)cc(F)c(F)cc1Cl N1(C(c2c(CC)onc2C)=O)CC2CCCCC2(CNC(=O)CS(=O)(=O)NC)C1 C(C(COC)C(=O)NCCCCCCN(C(=O)CC1SC(=N)NC1=O)C)OC c1(CC(N2CCC(C3CCCN3C(=O)Cc3ccsc3)C2)=O)ccc(O)c(F)c1 CC1CCCN(C(=O)C(=O)NCc2nc(CNC(c3cn[nH]c3)=O)cs2)C1 CC1CCN(C(=O)CCCC(=O)C2CC2)CC1NC(C1CN2CCC1CC2)=O CON1CCC(C(=O)NC(C)CCN(C)C(c2ccc(C#N)cn2)=O)CC1 c1(OC)cccc(CC(=O)NCC(C)CN(C(=O)C(n2nccc2C)C)C)c1F C1(C#N)(C(=O)NCCC(=O)NCCn2c(CC)nnc2)CCCOC1 C1(C(C)NC(C2(CO)CCCC2)=O)CCCN1C(C1CC(N(C)C)C1)=O C1(OCC)CCC(C(=O)NCCCNC(=O)C(c2ccnn2C)C)CC1 CC(CNC(=O)C(F)n1ccnc1)CC(=O)N1CCCC1CC1CC1 C(=O)(C1=C(C)OCCS1)N1CCN(C(CCSCCCC)=O)CC1CCC C#CCC(C(=O)NCC1CCCNC1=O)NC(c1ccn(C2CC2)n1)=O N1(C(c2c(C(C)C)onc2)=O)CCC(C(=O)N(C)Cc2cnn(C)c2)C(O)C1 N1(C(C2(OCC)CC2)=O)CC2CC(O)C1C2NC(=O)C(C)NC(=O)CC(C)(C)C C1(CNC(CC2C(CNC(CCCOC(C)=O)=O)C2)=O)CCOC1(C)C CC1COc2ccc(C(=O)NCC(C)(C)NC(=O)C(C)C(C)O)cc21 C1(NC(C2N(C(c3ncn(CC)c3)=O)CC=CC2)=O)CC=C(C(C)C)CC1 N12CCC3CC1CN(C3)CC2=O.c1(CCOC)ccc(C(=O)OC)cc1 C=CC(C)(O)CC(=O)NCC1CCCC1NC(C1CC(C(F)(F)F)C1)=O CN1CC(F)CC1C(N1CCC1CNC(=O)CCc1cn[nH]c1)=O c1(C(=O)NCCC(C)N(C(CCc2scc(C)n2)=O)C)cnc2sccn12 CCC(CSC)N=c1[nH]c(N(CC(=O)NC2CC2)C)nc2ncn(CC)c12 O=C(CC1=CCCCC1)NC1CC(CCNC(C2CCCCC2C2CC2)=O)C1 CCCCC(COC)NC(=O)C(CCOC)NC(=O)CCCOC(C)C C(=O)(C1=COc2ccccc2O1)NC1CC(NC(CCNC(=O)NC)=O)C1 c1(C(N(CCC(C(C)C)NC(CC2(C=C)CCC2)=O)C)=O)ccc(C)nc1C Cc1ccc(C#N)cc1C(=O)NCC1(NC(C2C3CC4C(C3)C24)=O)CC1 c1(C(=O)NC2C(CNC(CSCCC=C)=O)C2)cc(CSC)no1 C=CCC(C)(C)CC(=O)N1CCC(NC(c2cc(C(N)=O)cn2C)=O)C12CCC2 CC1(C#CC(=O)NCC2CC3CCC2N3C(=O)Cc2ccnc(O)c2)CCCO1 C1(Cl)(C(N2CC(C(N)=O)(CNC(C3CCCC3)=O)C2)=O)CC12CCC2 c1(C(=O)NC2C(C(=O)NCC(CC)(C)OC)C2(C)C)cnc(Cl)n1C c1(C(=O)NC2CC3CN(C(Cn4c(C)cnn4)=O)CC32)ccnc2c1CC(=O)N2 c1(CNC(C2CCC(C#C)CC2)=O)nc2c(s1)CN(C(=O)CC1CCOC1)CC2 CC1CC(NC(C2C=CCN2C(=O)CCC(C)(C)C)=O)CC(C)(C)C1 C1(NC(c2cnn(CC)n2)=O)(CNC(C2CCCS2)=O)CCCCC1C CC(=O)CC(C)(C)CC(=O)NC(CNC(c1ccc(Cl)cc1C)=O)C1CC1 C1(NC(C(c2ccccc2)OC)=O)CCN(C(=O)Cc2nnc(S)n2C)CC1O c1(OC(C)=O)ccc(C=CC(N2CC(C(=O)Nc3c(F)cccc3Br)C2)=O)cc1 C1(CCNC(c2[nH]cc(C(N)=O)c2)=O)CCCCN1C(=O)Cc1cccc(Cl)n1 N1(C(CC(n2ccc(C)n2)C)=O)CC2CCC(NC(=O)CCCCF)CC2C1 N1(C(CC=CC=C)=O)CCC(NC(C2CCCN2C2CC2)=O)CC1C c1(OC)c(Br)cc(CC(=O)NCC2CCN(c3nccc(C)n3)CC2)cc1Br CC1CCC(NC(C2(CN(C)C)CC2)=O)CN1C(=O)CC1(C2CC2)CC1 N1(C(c2c(C)oc(Cl)n2)=O)CCC(C(=O)NCC2OCC3CCC2C3)C12CCC2 C1(C(N(C(CN(C(c2cncc(OC)n2)=O)C)C)C)=O)CC2C(C1)C2(F)F CC#CC1CCN(C(C2(C3CCCN3C(=O)Cc3cnccn3)CC2)=O)C1 Cc1nc2c(o1)CCN(C(=O)COC(C)(C)CNC(C1COCC1C(N)=O)=O)C2 C1(OCCCNC(CC(=C)C)=O)CCN(C(C2CCC(=O)N2CC)=O)CC1 C1(CNC(c2c(C)nc(CCC)o2)=O)CN(C(=O)CC2CCC(O)C2)CCN1C N1(C(C=C(C)C2CC2)=O)C2CCC(C2)C1C(=O)O.C1(C(=O)NC(C)(C)C)(C(=O)O)CC1 c1(C(N2C(C(=O)NCCOCC(C)C)C(C)CC2)=O)cc2cccnn2c1 c1(NC(N(c2c(C)noc2C)C)=O)cccc2ccoc12.C1(=O)C(C(C)C)CN1 C(=O)(C1=NOC2(CCN(Cc3cc(Br)ncc3Cl)C2)C1)N1CCC(OC(C)=O)C1 N1(C(=O)Nc2ccc(C(=O)OC)o2)CCC2CN(Cc3cc[nH]n3)CCC12 N1(C(C2(OC)CS(=O)(=O)C2)=O)CCCN(C(=O)C(c2ccc(F)c(C)c2)=O)CC1 C1(N(c2cc(C)nc(C(C)(C)C)n2)C)Cc2ccccc2C1C c12ccc(nc1)c(=O)[nH]2.C1(CNC(=O)NC2CC2CC2CCC2)CC1(Cl)Cl C1(NC(CC(=O)NCC)=O)C2CC3C1C3C2C(=O)NC(c1nc(C)c(C)[nH]1)C c1(OCCC(=O)N(CC(CC)NC(c2ncccn2)=O)C)ccccc1O N1(C(CCCOC)=O)CC(O)CC1CNC(C1C2CCC1CC2)=O C(=O)(C(C)(C)C1=CCSCC1)NCC(C)N(C)C(C1CCN(C)S1(=O)=O)=O c1(C(=O)NCc2ccc3occc3c2)n[nH]c2ccc(-c3ccnc(F)c3)cc12 CC1(C)CCC(CCNC(=O)CC=CCNC(=O)C(O)C2CC2)O1 CN1CCCCC(C(=O)NCC2CC3CCC2N3C(C2CCCCN2C)=O)C1=O N1(CCN(CCC)C(c2cc(C(F)(F)F)cs2)=O)CCCC1C(C)C c1(C(=O)NCCC(C)N(C(Cc2cnc(C)o2)=O)C)n[nH]c2c1CCC2 CC(C)(C#Cc1cn(CCCOC(=N)O)nn1)NC(=O)C(C1(O)CCCCC1)O N1(C(C(C)(C)SC)=O)CCC(C2CN(C(=O)C(CO)C(F)(F)F)C2)CC1 CCCCCCC(=O)NC(CCCOC)C(=O)N(C1CCC1)C1CCC1 C(=O)(C(C)(C)C(=O)OC(C)(C)C)N(CCC)CCNC(=O)Cc1sc(C)nc1C N1(C(=O)CC2CCC2)CC(O)(c2cc[nH]n2)C1.C1(NC(CF)=O)C(O)CC1O C1(C(N(CCOC)CCNC(=O)CC(C)(C)C2CCCCC2)=O)C(C)OC(C)C1C N1(C(C(OC)OC)=O)CC2CC(C1)CN(C(c1coc(CC3CC3)n1)=O)C2 n1(CC(=O)NC23CCN(C(C4(O)CCCC4)=O)CC2C3)cnc2ccccc12 N1(C(C(C)(C)OCC(F)(F)F)=O)CC(NC(C2CCC(=O)NC2)=O)C(F)C1 c1(C(=O)Nc2c(C)cccc2)ccn2c1CS(=O)(=O)CC2 N1(C(c2ncc(CC)s2)=O)CCC(NC(=O)C(C(C)C)NC(=O)COC)C1C N1(c2cc(F)nc(-c3ccccn3)n2)CC2C3CCC(CC3)C2C1 c1(OC)cc(NCC2(NC(c3ccc(C4CC4)nn3)=O)CCCC2)nc(C)n1 N1(C(C(CC2CCCC2)OC)=O)CCOCC1CCNC(=O)Cn1cnnc1O c1(-c2nc(CCOC)on2)ccc(C(c2ccccc2)n2cc(Br)cn2)cc1 C1(Cl)(C(COC(CSCC)=O)=O)CC1C(=O)NC1CC1 C1(C(C)(C)NC(=O)Cc2ccsc2)CCN(C(C2CCCN2S(C)(=O)=O)=O)CC1 c1(C(=O)NC2C(CNC(CCCCC#C)=O)COC2)cc(C)c(OC)c(C)c1 CC(=O)CCCC(C)C(=O)NC(Cn1cccn1)C(=O)NCC1(C)CC2(CC2)C1 C1(NC(c2cc(C)c(Cl)s2)=O)CN(C(c2ccc(C#N)c(C)n2)=O)CC1N=[N+]=[N-] C(=O)(CCC(F)F)NC1CC(CNC(CC=CCC)=O)C1 Cc1ccc(N2CC(C(=O)NCC(O)CCNC(=O)C=CCO)CC2=O)cc1 CC1(CNC(c2cccc(CN=[N+]=[N-])c2)=O)CCN(C(C2CCCC3CC23)=O)C1 Cc1scnc1C(=O)NCCCNC(C1(Br)CC1)=O N1(C(N(c2ccccc2)CC)=O)CCC(C)CC1CNC1CCC1 C=CCCCCCC(=O)N1CCC(N(C(=O)CCCSc2ccccc2)C)CC1 C#Cc1cc(C(=O)NC2C3CN(C(c4cnc(CCCC)s4)=O)CC23)cc(F)c1 N1(C(c2c(C#N)scc2)=O)CCC2CC2(NC(=O)C2=COCCO2)CC1 CN1C(=CC(N2CCc3sc(C(=O)O)cc3C2)=O)C(C)(C)c2ccccc21 CC1CN(CC(=O)Nc2cc(Cl)cc(Cl)c2)c2cccc(Cl)c2O1 C(=O)(C(C)S(C)(=O)=O)NC(CC(C)C)CNC(=O)COc1ccccc1 c1(C(N(C(CNC(C(C(C)C)NC(N)=O)=O)C2CC2)C)=O)cccc2c1COC2 N1(Cc2c(CC)noc2)CCOC(C)(CNC(c2ccc(OC)cc2)=O)C1 C1(NC(Cc2cc(OC)no2)=O)CCCN(C(=O)C(=O)NCC(F)F)C1 C1(C(N2CCCCC(CO)C2)=O)CCN(C(c2coc(C(F)F)c2)=O)C12CC2 CC1(C)CCC(O)(C(=O)NC2CC(F)(CNC(=O)CCNC(=O)CO)C2)CC1 N1(C(CC(C)(C)OC)=O)C(CNC(=O)C(C)(C)C(C)(F)F)CC2COCC12 CC1CN(C(c2cnnc(O)c2)=O)CCC1NC(c1cnc[nH]1)=O CN1C(=O)CCC1C(=O)NC1C2CC1N(C(=O)C=Cc1ccccc1)C2 C1(NC(c2ccc(-c3ccccc3)nc2O)=O)CCCCN(C(=O)C2CC2)CC1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CCCC(N(C(=O)CC2C=CCC2)C)CC1 c1(CCNC(=O)NC2CN(C(=O)OC(C)(C)C)CC2O)c[nH]c2cnc(Cl)cc12 N1(C(c2c(F)cccc2Br)=O)CCC2CN(Cc3cc(B(O)O)co3)CC12 C#Cc1ccc(C(=O)N(C2CN(C(c3csc(CC)n3)=O)CCC2C)C)cc1C C1(C)(CC(=O)NCCCOC=C)CCN1C(=O)CCOCCOC CN1CCC(C(N2CC(NC(c3cscn3)=O)C(C)(C)C2)=O)S1(=O)=O C(=O)(C(CCc1cnn(C)c1)N1CCCC1COC(C)(C)C)NC(CC)C C1(CCOC)(NC(c2cnc(C)o2)=O)CCN(C(c2cccc(CO)n2)=O)CC1 c1(C(=O)OC)cc(C(=O)NC2CC23CC(NC(=O)C(C)(Cl)Cl)C3)cc(F)c1 C1(C(N2CCC(N(C(CCOC)=O)C)C2)=O)CCC(C(C)(C)O)CC1 N1(C(C2CCC(OC)CC2)=O)CC(C2CCCN(C(=O)C(F)n3cccn3)C2)C1 CC1CC(CNC(C2(F)CCCCCC2)=O)CN(C(C2(CN(C)C)CC2)=O)C1 c1(OC)csc(C(N2CC=CC2CNC(C2(NC(N)=O)CC2)=O)=O)c1OC c1(C(=O)NC2C(C=C)CN(C(=O)CC3CC3C(F)(F)F)C2)c(C)cc(C)oc1=O CC(CNC(c1ccn(C(F)(F)F)n1)=O)(CO)NC(=O)C=C1CCSCC1 CCCCC(O)CC(=O)NCCC1CCN(C(C2CN(C)CCN2C)=O)C1 CCCCC(O)C(=O)NCc1cc(O)nc(CNC(c2cc(O)n(C)n2)=O)n1 c1(C(N2CCC(C(C)O)CC2)=O)nnn2c1CN(C(C1CC(O)C1)=O)CC2 N#CC1(C(N2CCCC(NC(c3ccncc3)=O)CC2)=O)CCCOC1 c1(C(=O)NCC2(CNC(C3N(C)CCC3)=O)CC23CCC3)cc2ccsc2n1C N1(C(CSSC)=O)CCC2(CCCN2C(=O)Cc2cnccn2)C1 c1(C(N(C2CCN(C(C(CC)(CC)CO)=O)C2)C)=O)sc2ccccc2c1C C1(CC(=O)N(CCC(c2cccs2)NC(C(C)C2CC2)=O)C)CCC=CCC1 C(=O)(C1=CC2CCC(C1)C2)N1CCC(C(=O)NC2CCC(OCC)CC2)C1(C)C c1(OC)cccc(C(O)C(=O)NCC(C)NC(=O)Cc2cnc(C)[nH]2)c1 N1(C(Cc2nc(CC)sc2)=O)CC2CCC(CNC(=O)C(C)(C)C#N)(C2)C1 CCCCCC(O)CC(=O)N1CC(C(=O)NC2CN(C(=O)OC)C2)OC(C)C1 N1(Cc2c(CC)cccc2)CC2(CN(C(c3ccc(C)nc3)=O)CC2C(=O)O)C1 N1(C(C23CC(C(C)(C)C)(C2)C3)=O)CC2CN(C(C3CC3C#N)=O)CC2C1 c1(C(N2C(C(=O)OC(C)C)CCCC2)=O)cc2c(s1)CCC(C(C)(C)C)C2 C(C(=O)NCC1(O)CN(C(=O)CC2CC(=O)NC2=O)C1)(C(C)C)NC(COC)=O N1(C(CC(C)(C)C2CC2)=O)CCC2CCCC12C(=O)NC1CCC(N=[N+]=[N-])CC1 CCC(C(=O)NC1(CO)CN(C(C2(O)CCC2)=O)C1)C1CCOCC1 CC(CC(=O)N1CC2CC2(NC(c2cnc(C3CC3)o2)=O)C1)P(C)(C)=O CP(C)(=O)C(CC(=O)N1CCC(F)(CNC(c2ccc[nH]2)=O)C1)C(F)(F)F C1(CNC(c2cc(C)n(C)n2)=O)CCN(C(c2sc(N(C)C)nc2Cl)=O)C(C)C1 CS(=O)(=O)C1CN(C(C)(C)C)CC1C(=O)NS(=O)(=O)CC1CCC(F)(F)CC1 c1(CC)c(C(=O)NCC(O)CN(C(=O)C(F)=C2CCC2)C)ccn1C C=CCCCCCCCC(=O)N1CCC2(NC(c3cncs3)=O)CCCCCC12 C12CN(N3CCC(CC3)O1)C2.O=C1CCCCN1Cc1ccccc1 Cc1ccc(S(=O)(=O)NC(c2ccc(F)cc2-c2ccc(F)cc2)=O)cc1C C1(C(=O)OC)C2CC(O)C1N(C(c1cc(O)ccc1C)=O)C2 c1(C(N2CC(C(N)=O)SCC2)=O)cccc2c(I)n[nH]c12 C1(C(=O)NC2CCN(C(C3CC(C)(CC)C3)=O)C2C2CC2)CCc2c[nH]nc2C1 N1(C(c2c(C)nn(-c3ccccc3)c2)=O)CC2(N)CCCC2(F)C1 C1(C2CC2)(C(N2CC(N(C(C(C)OC(C)(C)C)=O)C)C2)=O)CC=CC1 N1(C(C2(CC=C)CCCCC2)=O)CC2CC(C1)CN(C(c1n[nH]cc1Cl)=O)C2 C(=O)(C(F)(F)CC)N(CC(C)N(C(C1C(CC)C1)=O)C)C CC(C)CC(O)C(=O)NC1CN(C(=O)Cc2cc(C3CC3)no2)CCC1F C1(C(=O)NCC2(CC)CC2)CCC(C2CC2)N1C(=O)C1=C(Cl)CC1 c1(C(=O)NC2CCN(C(c3c(C)snc3)=O)C(C)C2)c(F)ccc(N)c1F Cc1cccc(N2CCC(NC(=O)Nc3ccc(CCF)cc3)CC2)n1 c1(C(N2CC(N(C(CCC=C)=O)C)C3(C2)CC3)=O)ccc(O)c(C)c1C N1(C(c2n[nH]c(CC)c2C)=O)CC(NC(=O)CN2CCC(C)CC2)CC1(C)CC N1(C(c2ccc(CC)[nH]2)=O)CCC2CCN(C(c3coc(C(F)(F)F)c3)=O)C2C1 C1(CCOC)CCN(C(=O)CCN(C(C2(CO)CCOC2)=O)C(C)C)CC1 c1(OCC)cccc2c1OCC(C(=O)NC(C)C(C)NC(=O)CN(C)C(N)=O)C2 C12(C(=O)NC(CN(C(C=NOC)=O)C)C)CC=CCN1CCC2 C1(C(C)NC2(c3n(CCCC)nnn3)CCOC2)CC2(CCC2)C1 Cc1ncnc(C(N2CCN(C(=O)CC3=CCCC3)C(c3ncc[nH]3)C2)=O)c1C N=c1[nH][nH]cc1C(=O)NC1CC(CNC(c2[nH]nnc2C2CC2)=O)C1 CC(C)CCCCCC(=O)NC(C)CCCNC(c1ccccc1C(F)(F)F)=O c1(C(=O)NC2(COC)CCN(C(=O)C(C)=C(C)C)CC2)n[nH]c2c1CC(C)CC2 C1(CNC(COC(CC2(CC(=O)OC)CC2)=O)(C)C)CC2CC1CO2 c1(C(=O)NCCNC(C2(NC(=O)NC)CCCC2)=O)ccnc(Br)c1N c1(OCC)cc(OC)cc(C(N2C3CN(Cc4cc(Cl)cc(I)c4)CC23)=O)c1 CCC(C)C(C(=O)NC1CCC(CO)CC1)N(C)C(c1cc(C)n(C)n1)=O C12(C(=O)NCCOCCN(C(C(C)CSC(F)(F)F)=O)C)CCC(CO)(CC1)C2 N1(C(C(CCCC)O)=O)CC2CCCC(C1)N2C(=O)CCN1CCN(CC)CC1 C1(NC(C2(CCC)CC2)=O)CCOCC1C(=O)NC1CC(F)C1 C(=O)(CC1=CCOCC1)N1CCCC(CNC(=O)Cc2ccsc2Cl)C1 C(=O)(C(CC)C(=O)OCC)N1CC(NC(C2CC(=C)C2)=O)(CO)C1 c1(C(C)C(N2CCCC2Cc2cn(CCOC(N)=O)nn2)=O)ccccc1F CCCCCCCC(=O)NC(CC)CC(=O)Nc1cnc(C)c(CC)c1 C1(NC(CC=C(C)C)=O)CCN(C(C2C(OC(C)C)CC2)=O)CC1 N1(c2nc(-c3n(C)ncc3)nn2-c2ccccc2)CCc2cc(F)ccc2C1 C1(NC(C(CSC)O)=O)CC2(C1)CC(NC(C1CCCC1O)=O)C2 C=CC(F)(F)C(=O)N1CC(O)(CCNC(=O)COCc2ocnc2COC)C1 O=C1CCCCC(C(=O)NCC2CCCC2NC(=O)CC2(C(F)(F)F)CC2)C1 c1(C(=O)NC2C(NC(c3cnc(C)nc3)=O)CCC2)cc(C)c(F)cc1Cl Cc1sc(=O)n(CC(=O)N(C)CC2CCCN(C(c3cc(Cl)c(Cl)[nH]3)=O)C2)c1C N1(C(C23CCC(COC)(OC2)C3)=O)CC2CN(C(=O)C(C)C)CC2C1 c1(CNC(c2n(CC=C)nnn2)c2sccc2C(=O)O)ccc2c(c1)CCOC2 Cc1ccc(CN(C(C2CC2)C(C)C)CCCOC(C)(C)C)cc1Br CCCCC(C(=O)NCC(C)(C)CNC(=O)C(CCC)N(C)C)NC(N)=O C1(CNC(=O)Cc2ccsc2)CC2(CCN(C(C3C4C5CCC(C5)C34)=O)C2)CO1 CC1Cc2cc(NC(=O)NCCCCCN(C)C)ccc2O1 Nc1ncccc1C(=O)NCCn1cc(CNC(c2coc(C3CC3)n2)=O)nn1 C(=O)(CCCC(=O)N1CCOC(C(C)NC(C2CCCC2F)=O)C1)NC(C)C Cc1cc(NC(c2csc(N(C)C)n2)=O)n(C(=O)Nc2ccccc2Cl)n1 C(C(=O)NC(C)C)(C(C)(C)C)NC(C1(C)CN(C(C(C)OCOC)=O)C1)=O S(=O)(=O)(c1ccc(N(C)Cc2cnccc2Cl)nc1)NCC(CCCCC)(C)C c1(C(N2C3(C(=O)NCCC#C)CC3CC2)=O)cc(C#N)cn1C N1(C(CC(C)(C)O)=O)CCN(C(=O)C(C)(O)c2ccccc2)CC1c1cn[nH]c1 c1(C(N(CC(O)CNC(=O)CC2(CO)CC2)C)=O)cc(Br)c2nccnc2c1 C1(CC)CN(C(c2ccsc2C)C(=O)NC)CCO1 c1(-n2c(C(N(C(C)C(=O)OC(C)(C)C)C)=O)cnn2)cccc(Br)c1 N1(C(C(CC#C)(C)C)=O)CCCC(NC(c2cc(CC(C)C)nn2C)=O)C(F)C1 c1(NC(C(COCC)NC(=O)Cn2cc(C#N)cn2)=O)c(C)nn(C)c1C C(C(O)C(F)(F)F)N(c1ccccc1)CC.N12CCC1C2=O CCN=c1cc(NC2CCCC2CNC(=O)OC(C)(C)C)cc[nH]1 N1(C(CC(COC)C)=O)CC2CCN(C(c3ccc(F)cc3OC)=O)C2C1 C(=O)(C1=NN(C)C(=O)CC1)NC1C(OC)CN(C(=O)C(O)CC(C)C)C1 N1(C(C2CC(C)(C(C)(C)C)C2)=O)CCC2(CCN(C(=O)C(=O)C(C)(C)C)C2)C1 c1(C(N2CCC(N(C(=O)CCc3nncn3C)C)C2)=O)ccc2oc(=O)oc2c1 c1(C(=O)NCC2N(C(C(C)C)=O)C3C(C2)C3)nc2c(Br)cccn2n1 N1(C(C(C)(N(C)C(C2CCCCCC2)=O)C2CC2)=O)CCOC(C2(C)N=N2)C1 CCC(C)(C)CCCC(=O)N1CCCC(C)(C(N2CC(=O)NC(=O)C2C)=O)C1 CC(C(C)(C)C(=O)NCC1CCC(=O)O1)NC(C1CCOCC1(C)C)=O C1(NC(CC=C(C)C)=O)CC(CNC(c2cncc(C(F)(F)F)n2)=O)C12CCC2 c1(C(=O)NC(C(=O)OC)CSC)ccc(S(=O)(=O)NCCC#N)cc1 CC(C)C(C(=O)NCC1(O)CN(C(=O)C(c2ccc(Cl)cc2)C)C1)C(C)C c1(C(=O)NC2CCN(C(C(CC)n3nccc3C)=O)C2)cc(C)c(N)cc1Cl C1(CNC(c2csnn2)=O)CC2(CCN(C(c3cn4ccnc4s3)=O)C2)CO1 c1(CNC(=O)NCC2(C(F)(F)F)CC(=C)C2)cccc2nc[nH]c12 N1(C(C(CSC)O)=O)CCC2CCN(C(c3sc(CO)nc3C)=O)C2C1 c1(CNC(C(CCOCCO)NC(C(C)CO)=O)=O)ccc(=O)n(C)c1 c1(C(=O)NC)ccc(C(=O)NC2(CO)CN(C(=O)Cc3cncs3)C2)cn1 Cc1cc(=NCC2CC2C2CCCC2)[nH]c(=NCC2(CO)CC2)[nH]1 C1(N(C(=O)C(C2(O)CCC2)NC(=O)CC#N)C)CCCCC1O N1(C(C2CCSCC2)=O)CCC2C(CCN2C(c2cnc3[nH]ccc3n2)=O)C1 C(=O)(C(CC(F)F)N(C(=O)COC(F)F)C)N1CCC(N(C)C)(CC)C1 N1(C(CC(C)SC)=O)CCCC2(CCN(C(=O)Cc3nc(C)sc3C)C2)C1 C(=O)(CCCCCSC)NCC(CCC)NC(C1CCN1C(C)(C)C)=O CCS(=O)(=O)CC(=O)N1CC(F)(CNC(=O)CNC(=O)C(C)(C)C)C1 c1(C(N2CCC(C(C)(C)NC(C3N(CCC)CCC3)=O)C2)=O)cn(C)nc1OC C(=O)(C(=O)C(F)(F)F)NC(C1CN(C(C2(C)COC2)=O)C1)C C(CC(C(=O)NCC(C)CNC(c1ccc[nH]1)=O)N(C)C)SC Cn1ncc2cc(C(N3CC4CCC(C3)C4NS(=O)(=O)CC(F)(F)F)=O)ccc12 O=C(C1=CCCSC1)NCC1(NC(c2ccc(O)nc2)=O)CCOCC1 C(=O)(C(C)CCC(C)(C)C)NCCCc1cn(C(c2ncon2)C)nn1 C1(CNC(C=CCOCCOC)=O)CC(NC(C2CCCCC2)=O)C1(C)C c1(C(CC)CC)nc(-c2cc(Br)c[nH]2)n(CCOc2ccccc2F)n1 C12(NC(c3cnc(CC)s3)=O)CCCC1N(C(=O)CCCn1cccn1)CC2 C=CC(C)(CC)C(=O)OCCOCC1(C#N)COC1 c1(OC)ccc(F)cc1C(=O)NC1(CNC(c2cc(C)cc(N)c2)=O)CCOC1 CN1CC2C(C(N3CCOCC3CC(=O)NC3CC(Cl)(Cl)C3)=O)C2C1 C1(C(N(C2CCN(C(C(CC)OCC)=O)CC2)C)=O)CCCC(C)CC1 C1(C)(CC)CC(NC(c2cn[nH]c2)=O)CN1C(=O)CCSc1ccc(F)cc1 C#CC1CCN(C(=O)COC2CCN(C(c3ccc(C)cc3)=O)C2)C1 C1(C(N(CC(C)NC(C2CS(=O)(=O)C2)=O)CC)=O)CCC(COC)CC1 CN1CCN(C2(CNC(C3(O)CCSCC3)=O)CCC2)CC1 N1(C(CC2CCC(C)C2)=O)CC2CN(C(C34CCCC3C4(F)F)=O)CC2C1 c1(C(N2CC(C3CN(C(CC(C)O)=O)C3)C2)=O)cc2n(n1)CCCC2O C(CNC(=O)C(Cc1cnc[nH]1)NC(=O)C(C1CC1)SC)(C(F)(F)F)OC C(=O)(C1=CCCOCC1)N1CCC(NC(c2c(C)ncnc2)=O)C1(C)C S(=O)(=O)(c1ccc(Cl)cc1)N1CC(C(=O)NCCCN2CCOCC2)SCC1 C1(CCC)(NC(=O)CCS(N)(=O)=O)CCN(C(=O)CN(C)S(N)(=O)=O)CC1 CCC(C(=O)NC1(CCOC)CCN(C(c2c(F)cccc2F)=O)C1)C(F)(F)F C1(NC(C(C)OC)=O)CCCN(C(C2CC2c2cn[nH]c2)=O)CC1 c1(C(N2CCN(C(CC(C)(F)F)=O)C(C3CC3)C2)=O)cncc2c(O)nccc12 c1(C(N2C(CN(C)C(C3CCCCC3)=O)CCC2)=O)ccc(F)c(O)c1 c1(SC)ccc(CC(=O)N(C2C3CN(C(C4CCC(=O)N4C)=O)CC23)C)cc1 C1(NC(c2scnc2C(F)(F)F)=O)CCCN(C(C2CC3(C2)CC3F)=O)C1 C(C(Cc1ccc(Cl)cc1)C(=O)NC1CCN(C(=O)CSCC(=O)OC)C1)OC C1(NC(c2cc(C(C)C)no2)=O)CCCCCN(C(=O)CSCc2ncc[nH]2)C1 C1(NC(=O)C2=CCCC2)CN(C(c2ccc(Cl)c(F)c2)=O)CC2(CCOCC2)C1 CCCC(C)CCNC(C1(CO)CCN(C(c2csc(Cl)n2)=O)C1)=O c1(C(=O)NCC2CC3(CCC3)CN2C(c2ccsn2)=O)cc(Cl)c2n[nH]cc2c1 CN=c1nc(N2CCC(CSC3CCOC3)C2)[nH]c(=NCC(C)(C)SC)[nH]1 C1(NC(CCn2c(C)ncc2)=O)CCCC12CN(C(=O)C(C(C)C)N(C)C)C2 N1(c2c(C)c(NC3C=CCCCC3)ncn2)CCC(C)C(F)(F)CC1 C1(CNC(c2c(CC)scn2)=O)C(C)CCCN1C(c1cc2c(s1)CCC2)=O N1(C(Cc2ccc(NS(CC)(=O)=O)cc2)=O)CCNC(=O)c2cc(Br)ccc21 C(=O)(C1=NNC(=O)CC1)N1C(C)(C)C(CNC(=O)C=CC(F)(F)F)CC1 C(=O)(C1OCCc2c(O)cccc21)NC(C)(CO)C(F)F c1(N(C)C)cncc(C(=O)NC2CC(C)(NC(=O)CC3CCCC4CC34)C2)c1 c1(C(C)C)ccc(O)c(C(=O)NC(C)C(C)NC(=O)C2=CCCSC2)c1 c1(CC(N2CC3N(C(c4nn(CC)c(C)c4)=O)C3C2)=O)ccc2c(c1)OCO2 c1(N(CC(=C)Br)C)nc(N2CC(C(N)=O)C3(CC3)C2)c2c(n1)CCCCC2 C(=O)(CCC(O)C(C)(C)C)Nc1cccc(CNC(C2CCC(C)(C)OC2)=O)c1 C1(CC(=O)NC2(C(N(C)CC3CCCO3)=O)CC(CO)C2)CC2(CC2)CO1 N1(C(c2nn(CC)c(C)c2)=O)CCC2CC(NC(=O)C#CC3CC3)CCC2C1 C(CCCCCNC(=O)CN1CCCS1(=O)=O)N(C(=O)C1=CCCS1)C C1(C(N2CC(C)C(NC(=O)C(F)(F)CO)C2)=O)CC2(COC(=O)N2)C1 C=CC(C)C(C)C(=O)N(CCCNC(c1cc(OC)cc(OC)c1)=O)C(C)C c1(OC)csc(C(N2CC(O)(CCNC(C3CC(SC)C3)=O)C2)=O)c1OC Cc1ncc2c(n1)CCC(C(N1CCCC1(C)CNC(=O)Cc1cncs1)=O)C2 C(=O)(C(O)CC(C)(C)C)N(C1CN(C(COc2cccc(CC)c2)=O)C1)C C(=O)(C(C)(C)CN(C(=O)CN1CCCCC1=O)C)N(CC(COC)O)C c1(C(N(CC(CNC(C(C)C2CC2)=O)O)C)=O)ccc2c(c1)CN(C)C2 c1(C(=O)Nc2nc(C)c(C(=O)NCC3(F)CCC3)s2)cc(Br)ccc1Cl C(=O)(CCS(C)(=O)=O)NC1CN(C(c2c(OCC=C)cccn2)=O)CC1C c1(NC(C(C)Oc2c(C)n(C)nc2)=O)ccnc2cc(Cl)ccc12 C(=O)(C(CCOCCO)NC(c1nonc1N)=O)NC1CC(C)(CC)C1 N1(C(c2ccc(CC)cc2)=O)CC2(CC2)CC1CC(=O)NCc1cc(C)ns1 c1(CNC(=O)CNC(=O)Nc2ccccc2)ccc2c(c1)COC2=O.c1nc[nH]n1 N1(C(c2c(SCC)cncc2)=O)CCC(O)(CCNC(=O)CCC(F)F)CC1 C(N=c1[nH]c2c(c(=NCC3CC(n4ccnc4)C3)[nH]1)CCC2)c1snc(C)n1 CC1(C(N2CCC(n3cc(C(C)(C)O)nn3)C2)=O)CCCCCC1 C(=O)(C(CNC(C1CCC(O)CC1)=O)C(C)(C)C)N1CCN(CCOC)CC1 CC1CCN(C(c2ncccc2N)=O)C1CNC(=O)C(C)(C)c1cnsc1 CCC(C(C)O)NC(=O)C(C)(C1CC1)N(C)C(C1CC(=C2CC2)C1)=O C#CCCCCCC(=O)N1CCC2(NC(=O)CC(C)(O)C3CC3)CCCC12 Cn1ccc2sc(C(=O)NC3(C)CCCN(C(c4ccnn4C4CC4)=O)C3)cc12 c1(N(CC(N)=O)C)nc(=NC(CCO)C2CCC(F)(F)CC2)[nH]c2ccsc12 CCCC(C(C)CC)(c1nnnn1CC1CCC1)NCc1cccc(OC)c1 c1(C(=O)NC23CC(NC(=O)C4=CCCS4)(C2)C3)ccc2c(c1)Cc1ccccc1-2 C1(O)(CNC(C(C)CN(C(=O)COc2cccnc2)C)=O)CCOCC1 CCCC(CNC(c1cnc(C)cn1)=O)C(=O)N1CCC1CN1CCCC1 CC1CC(NC(C2(C)CC2)=O)CN1CCSc1cccc(N2CCCS2(=O)=O)c1 N1(C(CCOCCCOC)=O)CCC(CNC(C2CCOC2C2CC2)=O)C(O)C1 CC1CCN(CCC)CCN1CCC.c1(S)css1 C1(CC=C)(NC(=O)C(N2CCC(C)C2)=O)CCN(C(=O)C(F)n2cccn2)CC1 c1(-c2onc(C)n2)ccc(CNC2(c3nnnn3C3CCC3)CCC(C)C2)cc1 Cc1ccn2cc(C(=O)NC3CC4CCC3N4C(C3C(C)(C)C3(F)F)=O)nc2c1 c1(OC)cc(=NC(=O)C(C2(O)CCC2)NC(=O)CC2(O)CCCCC2)[nH]n1C C1(CCC)CCc2ccccc2N1Cc1nnnn1Cc1ccccc1 C1(NC(C(COC)(C)C)=O)CCC2(CC1)CC(NC(=O)CSC)C2 C1(C(=O)NCc2ccc(C)cc2)CN2CCN1CC2C.c1(OC)cccc(Cl)c1N CCC(C)(C)C(C(=O)N1CCC(NC(=O)C(C)(C)c2ccn(C)n2)CC1)OC c1(C(N2C(C#C)CCC2)C(=O)NCC2CCC3(CC3)C2)cc2cc(F)ccc2o1 C1(CNC(c2cc(Cl)ccc2Cl)=O)C2CCC1CN(C(C1CCC1)=O)C2 N1(CC(C)C)CCOC(CNc2cc(NCCC34CCCC3C4)ncn2)C1 N1(C(C(C)(C)OCC)=O)CC2C(C(=O)NCc3ccncc3)C2C1 c1(OC)cccc2[nH]c(C(=O)NCCC(C)NC(c3cnc(Cl)c(Cl)c3)=O)cc12 C(=O)(C1=CCCN(C(C2CCCCCC2)=O)C1)N1CCCC(C(C)O)C1 c1(OC)cccc2c1CN(Cc1cn(COc3ccco3)nn1)C2 c1(C(N2CC(O)CC(NC(CCC(CC)CC)=O)C2)=O)cnc2n1CCCCC2 C(C)(CCC#N)(c1n(C(C)C)nnn1)NC(C)Cc1ccco1 C1(CC(=O)NC(C2CCCCC2)CNC(C2CC2CF)=O)CC2CCC1CC2 C(=O)(CC(C)(C)CC(=O)N1CCCC(O)(CNC(C2(C(F)F)CC2)=O)C1)OCC Cc1[nH]nc2c1CCC(C(=O)NC1CCC(NC(=O)C(C)CS(C)(=O)=O)CC1)C2 C(=O)(C1=CC2(CN(C(=O)Cc3nc(=N)[nH][nH]3)C2)OC1)NCc1ccc(OC)cn1 c1(OCC)ccc(C(C)NC(C2CNCCN2Cc2ncc(Cl)s2)=O)cc1 c1(C(C(=O)O)NC(C(c2cnn(C)c2)NC)=O)ccc(C)s1 C1(CCNC(C=COCC)=O)CCCN(C(=O)C(O)C(C)(C)C)CC1 c1(N(C2CCC(N)C2)C(c2ccc(Br)nc2)=O)cc(N2CCCC2)ncn1 O=C(CC(O)C(Cl)(Cl)Cl)NC1CCOCC1NC(C12CC(F)(C1)C2)=O C(C(=O)N1CCCc2nccn21)(c1cccs1)NC(Cc1c(C)cccn1)=O C1(CC)CN(C(C2CC(O)C2)=O)CC1NC(C1CC=CCC1)=O C1(CNC(CSCCC)=O)CN(C(=O)CCn2ccc(C)n2)C2(CCC2)C1 c1(CC)onc(C)c1C(=O)NC1CCCC(NC(=O)CCCN2CCCCC2)C1 CCCCCC(C)(CC)C(=O)N=S1(=O)CCC2(CC1)CN(C(=O)C(C)C)CCO2 CC(C)C(C)CC(=O)N(CCCn1cc(C2CC3(CCC3)C2)nn1)C1CC1 C(=O)(C(C)N=c1cc[nH]cc1)N1C(C(C)C)(C(N2CCC(F)(F)CC2)=O)CCC1 CC(C)CC(F)C(=O)N1CCCC(O)(CN(C(=O)CN2CCCNC2=O)C)C1 c1(C(=O)NC2CN(C(C(CCC)(C)C)=O)CC(O)C2)cccn2nncc12 c1(CN2CCC(NC(c3cc(Br)ccc3F)=O)C(F)C2)c[nH]c2c(Br)cccc12 C1(CC(=O)N(C)CC2N(C(CN(C(C)=O)C)=O)CCC2)C(=O)ON=C1C c1(CNCCC[Si](C#C)(C)C)cc2c(s1)CCC(C)(C)C2 N1(C(c2c(CCC)[nH]cc2)=O)CC2CCOCC2(NC(=O)C(=O)NCC)C1 c1(CN(C(=O)CN2CCC2C)CCOCC)cc(OC)c(OC)cc1Br C1(C(=O)NCC(C)(C2CC2)NC(=O)CC2CCCC(C3CC3)O2)CCCCC1O C1(CC)(NC(C2C=CCCC2)=O)CCN(C(=O)C(O)COC)CC1 c1(C(=O)NCC(C)N(C(c2cc(OC)cc(F)c2)=O)C)cc2n(c(=O)c1)CCS2 O=C(C1=Cc2ccccc2C1O)NC1CC(CNC(C2(CO)CC2)=O)C1 C1(C(=O)NCC2N(C(CCNC(N)=O)=O)C3CCC2C3)CCCC2(CCC2)C1 N1(C(c2n[nH]c(C)c2O)=O)CCCN(C(=O)Cn2cccn2)CC1C(C)C c1(N(S(CC)(=O)=O)CCN(C(CNCC2CC2)=O)C)ccc(SC)nc1 C=C(C)CN=C(NCC(F)F)N1CCN2C(=O)NCC2C1 N1(C(c2c(C)cc(C#N)s2)=O)CC(C)CN(C(C2CC23CCC3)=O)C(C)C1 N1(C(CN(CCn2cc(Cl)c(C(F)(F)F)n2)C)(C)C)CC(C)OC(C)C1 CC1CC=CCC1C(=O)NCCC1CCCN(C(=O)C=C2CCOCC2)C1 C=C=CC(C)C(=O)N1CCCC(CNC(=O)C(C)OCOC)C1 N1(C(c2c[nH]nc2Br)=O)CC2OCCN(C(c3cnn4c3OCC4)=O)C2C1 N1(C(C)=O)CCc2cc(C(=O)N(C)C)ccc21.C12CCCCN(C1)CCCN2 C1(NC(C2N(C(C)C)C(=O)CC2)=O)CCN(C(c2cc(Cl)nnc2Cl)=O)C(C)C1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CCCC(C(C)(O)CNC(=O)Cn2cnnn2)C1 c1(C(N2CC(NC(Cc3c(C)cco3)=O)C(C)C2)=O)cc2ccccc2cc1N Cc1cc(C(=O)NCC(N2CCC(C)C(CN)C2)=O)ccc1Cl C(CN=C(NCc1cc(C)ccc1O)N1CCN2C(=O)OCC2C1)SC CC1(C)CCN(C(c2c[nH]nc2-c2ccccc2)=O)CC1NC(=O)C=CCO C1(CNC(C(C)N(CC)CC)=O)CCN(C(=O)CCNC(C)=O)CC1(F)F N1(C(C2C(C(=O)NCCc3ncc(C)cn3)C2)=O)CC(C)N(C)C(C)C1 C(=O)(C(O)CCNC(C1CC(O)C(F)C1)=O)NC1C(OC)C(O)C1 CC1OCCOC1C(=O)NC1CCC(F)(CNC(C2(C3CC3)CC2)=O)C1 CCC(C)C(=O)C(=O)NCc1nc(C)c(C(N2CCOCCC2C2CC2)=O)o1 C1(NC(C2N(CC)CC2)=O)CCN(C(=O)C(COC)OC(C)=O)CC1O CCCCC(O)C(=O)NCC(C)(C)CN(C(=O)Cc1ncccc1C)CC c1(C(=O)NC2CN(C(CC3(C=C)CCC3)=O)C(CO)C2)ncnc2c1CCC2 N1(C(CCCCOC)=O)C2COCC1CC(NC(=O)CC1CCCCN1C)C2 c1(OCC(C)C)ccccc1CN1CCC1CNC(=O)C(C)(F)F.C1(=O)CN1 C1(C)(CNC(c2n(CC#C)cnn2)=O)CCN(C(=O)CCC2CCC(C)O2)C1 CCC(CC(=O)NCc1ncccc1C(=O)N(C1CCCC(C)C1C)C)C1CC1 C1(CC(C)C)C(=O)C(CCCC)C(C(=O)NC)N1CCC(=O)OCC.OCC C1(NC(C(=O)NC(COC)C)=O)CCCN(c2ccccc2Cl)C1 C=CCCC(C(=O)N1CC(CO)C(O)C1)NC(=O)CC(=O)N(C)C C(c1ccc(F)c2ccccc12)=CC(=O)Nc1c[nH]nc1Cl CC(C(=O)N(C1CC1)CC1CCCN1C(=O)CC12COC(CF)(C1)C2)C(C)(F)F CC1CCC(NC(=O)CS(=O)(=O)NC(C)(C)C)CN1C(=O)C1=CCCS1 c1(C(=O)NCC(CNC(=O)CC2C=CCC2)O)conc1-c1ccccc1 C(=O)(CC(F)(F)C(F)(F)Br)NCC(C)N(C)C(c1cocn1)=O N1(c2c(C)cnc(C)n2)CC(CNC(C2(O)CCCC2)=O)OC(C)(C)C1 c1(C(=O)NCC2CC(NC(c3cc(OC)ns3)=O)C2)c(CO)noc1C c1(C(=O)NCCN2CCC(C(=O)NCc3c(C)scc3)CC2)c(F)cccc1F c1(C(N(C)Cc2cn(Cc3c(C(C)=O)cccc3)nn2)=O)ccc(Cl)c(Br)c1 c1(C(=O)NC(C)(C)CNC(=O)CCC(N)=O)nc2cccnn2c1Br N1(C(C(CC)COC)=O)CCC(NC(=O)CCc2cccs2)C(F)(F)CC1 C(c1ccncn1)=CC(=O)NCC1CC(NC(C2(c3cccs3)CCCC2)=O)C1 c1(OC)ccc(F)cc1CC(=O)NCCCC1(NC(=O)CNC2CCCC2)CC1 N1(C(C=C(C)C)=O)CCCC2CN(C(C3Cc4ccc(C)cc4S3)=O)CC12 c1(SC)cc(F)ccc1C(=O)NC1CN(C(c2cnccc2Cl)=O)CC1O C(=O)(C(C)CC(C)(C)C)N1CCC(NC(c2c(C)nc(C3CCC3)o2)=O)C1C c1(CC(=O)OC2C(OC(C=CC=CCC)=O)C2)cccc(C(F)F)c1 c1(CC)c[nH]nc1C(N1CC=CC1C(=O)NCCNC(C1CCC1)=O)=O C1(CNC(=O)CCc2cc(Cl)cs2)CCCCCN1C(c1n[nH]c2c1CCC2)=O CC(C)(C(=O)O)C(C1CC1)NS(=O)(=O)CCCOC C1(CNC(CCOCC)=O)CC2CCC1N(C(c1ccc(=O)n(C)n1)=O)C2 N1(Cc2c(CC)noc2C)CC2CCN(C(c3cccc(C(F)F)c3)=O)C2C1 c1(CC)ccc(C(=O)NCC2CCCN(C(C3(C)COC3)=O)C2)cc1N c1(CNC(=O)NC(c2cnn(C)c2)C(=O)OCC)nsc2ccccc12 C1(NC(C(C)C(C)(F)F)=O)CC1C1CCN(C(=O)CC(F)(F)Cl)CC1 c1(C(=O)NCCN(C(=O)CCOc2cccnc2)CCOC)cc(Cl)nnc1O N1(C(C(CN(CC)CC)F)=O)CCCC2(CCCN2C(=O)C#CC2CC2)C1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CCC2CN(C(C3CC=CCC3)=O)CC2C1 C1(C(C)OC)CCCN(C(=O)C(=O)Nc2c(C)cnn2-c2ccc(C)cc2)C1 N1(C(C(N2CCSCC2)C)=O)CCC2C(NC(C3(Cl)CC3(F)F)=O)C2C1 c1(SC)ncc(C(=O)NCC(F)CNC(c2cc(C3CCC3)[nH]n2)=O)c(O)n1 c1(NCCC(=O)NC(C)C)[nH]c(=NCC2CC3(C2)CC32CCC2)nc2scnc12 c1(NC(C2CCN(C(CC)CC)C2)=O)cc(Cl)c(C)c(Br)c1 N1(C(C2C(C)OCC2)=O)CC(C)(C)OC2(C1)CN(C(C1CCSCC1)=O)C2 C1(NC(CN(C2CC2)CC)=O)C2CC3C(C2)C13C(=O)N(C)Cc1cnc[nH]1 C1(C(=O)NC2C3CC2N(C(=O)COCC2CCOC2)C3)CC1C1CCOCC1 CC1COC(C)(C)CN1C(=O)C(Cc1ccco1)NC(=O)Cn1[nH]cnc1=N C(C(Cc1ccccc1)C(F)(F)F)NC(N1CCCC(NCCO)C1)=O N1(C(c2cnc(SCC)c(C)c2)=O)CCC2(CCC(NC34CC(CC)(C3)C4)C2)C1 Cc1ccc2c(c1)CC(C(=O)NCCCNC(c1cccc(P(C)(C)=O)n1)=O)O2 C1(CN(C(=O)CC(C)(C2CCC2)N(C)C)CC)CCCN(C(C2OCCO2)=O)C1 C1(CC(=O)NC)CN(C(=O)Cn2cccn2)CCN1C(c1cocn1)=O N1(C(C2CCCCC2)=O)CCC2(CCN(C(C3CCCC(F)(F)CC3)=O)C2)C1 C(=O)(C(O)CC(F)(F)F)NC1CC(NC(=O)CCOc2ccc(F)c(Cl)c2)C1 N1(C(C2NC(=O)C(F)C2)=O)CC2CCCC(C1)N2C(=O)COc1cccc(Cl)c1 Cc1c(C(N2CCC(CNC(C34CCCC3C4)=O)C2)=O)cnn1-c1ccncc1 Cc1cc(O)nnc1C(=O)NC1CN(C(c2cc(Cl)ncc2N)=O)CCC1CO c1(C(C)=O)ccc(Nc2ccc(CNC3CSCSC3)nc2)cc1C C1(C(N2CC3CC(NC(c4cn(CC)nc4C)=O)C3C2)=O)CCn2cncc2C1 N1(C(C(C)Cc2ccccc2)=O)CCC(NC(c2scnc2C2CC2)=O)CC1C C#CC1(C(=O)NCC2CCC(C(=O)NCCn3cncn3)O2)CCCCC1 N1(C(C2(Br)CC2)=O)CC2(CCNC(C3(c4ccno4)CC3)=O)CCC1CC2 C1(CC)CN(C(c2coc(CNC(c3cnc(OC)s3)=O)n2)=O)CC(=O)N1 N1(C(C2C(C)C2)=O)CC(CNC(C2(n3cccn3)CCC2)=O)OC2CCCC12 c1(OC)c(C(N2CCC(NC(c3ccoc3)=O)C2C)=O)ccc(Cl)c1C C1(NC(C2(c3ccccc3Cl)CC(C)C2)=O)CCC(F)(CNC(=O)CC#N)C1 CON1CCC(CC(=O)NCC2CC2CNC(=O)C=Cc2ccccc2C)CC1 N1(C(c2c(N(C)C)cccn2)=O)CC2CC(NC(c3sccc3F)=O)C1C2 CCCCCC(O)C(C)C(=O)NC1CCC1NC(C1Cc2ccccc2O1)=O C1(C(=O)NC2(c3ccccc3)CN(C(C3(CC)CC3)=O)C2)COC2(CO)CC1C2 CCC(C)(CNC(C1CCCC1)=O)NC(C1C=CCCC1)=O c1(C(=O)OCCN(CCCCNC)C)ccc(-c2ccc(Br)s2)s1 C1(CNC(c2cc(C(=O)OC)sc2)=O)CC(OC)CN1C(c1c(C)cnn1C)=O CC12CCC(C(N3CCCC(NC(=O)CC(F)(F)C(F)F)CC3)=O)(CC1)OC2 c1(CNC(C(Cn2cccn2)NC(c2n(C)nnc2)=O)=O)ccnc(CO)c1 CC(O)(C(=O)N1CCN(C(C2C(F)(F)C23CCC3)=O)C(CO)C1)C(F)(F)F c1(NCCCN(C)C2CC2)ccccc1NC(c1ccccc1)=O C=C=CCC(=O)NCC(COC)NC(=O)CCCn1cccn1 O=C1CCCC(CC(N2CC=CC(NC(=O)CCCc3cc[nH]n3)C2)=O)C1 C1(C(=O)NCC2(SC)CC2)CCC(O)CN1C(C1CC=CC1)=O C(=O)(CCCCC(F)F)N1CC(CNC(C2CC(C)(C)C2)=O)C(C)(C)C1 C#CCC(C)(C(=O)NCCCC1C=NNC1=O)NC(=O)C(COC)COC CC(C)CCCCCC(=O)N(CCCCN(C)C(C1C=CCCC1)=O)C C(=O)(C#CC1CCCO1)N(C(C)CN(C)C(c1cnc(C2CC2)s1)=O)C CC(C(=O)N1CCC1CNC(c1cnn2c1OCC2)=O)C(C)(C)C C1(C)(C(=O)NCCCN(C)C2CC2)CCN(C(C2CC2C2CCCC2)=O)CC1 C(=O)(C(F)C(F)(F)F)NC(CCCCNC(C1(C(=O)OC)CC1C)=O)C CC1CCC(CO)CN1C(=O)COC1CC(NC(=O)C=Cc2ccco2)C1 C1(C(=O)NCc2nc(C)c(C)o2)(C(=O)OC(C)(C)C)CCC2CCCC12 N1(C(CCCOCC)=O)CCCC(CCCCNC(c2cccc(OC)n2)=O)C1 CCC(CNC(=O)C(C)C#N)(CC)NC(c1cc(C2(C)CC2)n[nH]1)=O N1(C(C(C)=C2CCCC2)=O)CCC(O)(C(C)NC(=O)CCC2CCC(O)CC2)C1 c1(C(N2CC3C(NC(c4ccc(CC)o4)=O)(C3)C2)=O)ccc2ccncc2c1 C1(C(=O)NCC2CCC(CNC(CNS(C)(=O)=O)=O)CC2)CCCCNC1=O c1(NC(C2C(CC)CCN2C(=O)Cn2nccn2)=O)ccc(O)c(C)c1 C1(OCC)CCN(C(=O)CC2(COC(c3cncc(NC)c3)=O)CCC2)CC1 C=CCCCC(=O)NC1CN(C(=O)CNc2ccc(C(F)(F)F)cn2)C2CC12 C1(C(C)C(N2CC(F)CC2C)=O)CC2(C1)CN(C(C1CC(F)C1)=O)C2 C#CCCCCC(=O)N1CC(NC(=O)CSc2nnnn2C)C2CC12 C(=O)(C1=NNC(C(F)(F)F)C1)N1C(CNC(=O)CSCCF)CCC1 c1(CN(CC(=O)N(CC(F)(F)F)C(C)=O)CC)ccccc1 C1(CNC(C2(CC#C)CC2)=O)C2CCCC1N(C(c1ccc3c(c1)CCC3)=O)C2 C12(CC(=O)NCCN(C(=O)CCC3CC3(F)F)C)CCC(CC1)CC2 N1(C(C2C(=C)C2)=O)CCC2(CCCN(C(c3nc(C)ccc3OC)=O)C2)C1 n1(CC)nnc(C(N2CCC(C3CCCN3)C2)=O)c1C Cc1oc(CNC(c2cc(C3CC3)on2)=O)nc1C(=O)NC1CS(=O)(=O)C1 C#CC1CN(C(C2CCN(C(=O)Cn3cnnc3)CC2O)=O)CCN1C c1(C(N(C(CCNC(CCOCCCCC)=O)C)C)=O)ncoc1CC N1(C(C2(CC)CN(C(C(CC=C)CC)=O)C2)=O)CC2C=CCC(C2)C1 Cc1cc(C(=O)NC2CN(C(=O)Cn3cccn3)CCC2C)nc(O)n1 c1(CCCCCC)cccc(N=c2[nH]c3cccc(OC)c3n2C)c1 c1(C(=O)NC(C(C)C)(C)CNC(C2(CCO)CC2)=O)ncc(F)cc1F C(=O)(CC(C)CC(C)(C)C)N1C(C)C(C(=O)NC2CCC3(CCCC3)C2)CCC1 c1(C(N(CCC)CCNC(=O)CCn2cccn2)=O)csc(C(C)(C)C)c1 C1(N(C(c2c(C)n(CCO)nc2)=O)C)CN(C(c2cc(Cl)ccn2)=O)CC1(C)C C1(C(=O)NCC2(CF)CC2)CC2CCC(C1)N2C(=O)CC1CCCOC1 c1(C(=O)NC2CC(NC(c3cc([N+](=O)[O-])c[nH]3)=O)C2)ncc2ccccc2c1O C1(C(=O)NC2CC(C)(NC(=O)C(C3(O)CCCC3)F)C2)CN(S(N)(=O)=O)C1 Cc1ccc(C)c(-c2nc(COC(c3csc(C4CCCO4)n3)=O)no2)c1 Cn1nc2c(c1C(N1CCN3CCCC3C1)=O)CN(Cc1cscn1)CC2 C(=O)(C(CO)C(C)(C)C)NCc1ncc(C(=O)NCC(=O)NCC=C)cn1 C1(C(=O)NCC(C)OC)CCN(C(c2ccc(CC#N)cc2)=O)CC1O C1(C(N2CCCCC2CCCNC(C2(CO)CC(F)(F)C2)=O)=O)C2(CC2)C12CC2 c1(C(N(CC(C)NC(=O)C(C)(Cl)Cl)CC)=O)oc2c(OC)cccc2c1C N1(C(C(C)OC(C)(C)C)=O)CC(C(C)(C)O)(CNC(C2CCCCS2)=O)C1 c1(NC(CC2OCCN(S(CCCC)(=O)=O)C2)=O)cc([N+](=O)[O-])c(F)cc1C C=CCC(C(=O)NCCCCC(C)NC(=O)Cc1ccccc1OC)C(C)C c1(C(N2C(CC(=O)NCC3CCC(CO)C3)COCC2)=O)cccc2c1CCN2 CC(F)(F)C(C)(C)C(=O)NCCC1CC(NC(=O)C2=C(Cl)CCCC2)C1 c1(C(=O)NCCCC2N(C(C(CC)N(C)C)=O)CCC2)noc2c1CCCC2 c1(N2CC(NC(c3cccc(O)c3)=O)C(F)(F)C2)ncnc2cc(Br)sc12 N1(C(C2(SC)CC2)=O)CC(CN(C)C(C2(C)CCNC2=O)=O)C2(CC2)C1 N1(C(C(C=C)(C)C)=O)CCC2(CC1)CC2CNC(=O)C=C(C)c1ccccc1C N1(C(CC2C(C)=NNC2=O)=O)CCC2(CC2C(=O)NOCCN(C)C)C1 C(C(=O)N=c1ccc(C)c(Cl)[nH]1)Nc1c(CC)nn(C)c1-n1nc(C)nc1C N1(C(CCCn2ncc(C)c2)=O)CC(F)CC1CN(C(=O)C(O)CC1CCCC1)C C(=O)(C(O)CC(C)C)NC1CNCC1F.C1(SC)CCCC1n1cc(C2CC2)nn1 c1(C(=O)NCC(CC=C)NC(=O)CN(CC)CC)cc(Cl)cc(Cl)c1Cl c1(C(=O)NCCC2CCCN2C(c2sc(F)cc2Cl)=O)ccc2cccnc2n1 c1(C(N)=O)ccc2c(c1)CCC2NC(=O)N(CCC1CC2CC1C2)C1CC1 C12(NC(c3nnc(C)o3)=O)CCC(CC1)N(C(=O)CCOC1COC1)C2 c1(N(C2CC(C#N)C2)CC)cccc(C(CF)NC(c2ccccc2)CCO)c1 c1(C(N2C(CNC(C3C(OC)(OC)CC3)=O)CC2)=O)ccccc1C1CC1 N1(C(c2cc(C)c(C(F)F)cn2)=O)CC2(CCCCN(C(C3CCCC3)=O)C2)C1 Cc1cccc(Cl)c1CC(=O)NC1C=CCN(C(=O)C=CCN(C)C)C1 c1(CNC(C2CCC(C)C(C)C2)=O)nc2c(s1)CN(C(=O)CC1(CO)CC1)CC2 N(C)(S(=O)(=O)N1CCNC(C2CCC2)C1)CCN(C)C C1(Cc2onc(CCCS(C)(=O)=O)n2)CC2C=CC1CC2 C1(OC)CC(CNC(C2CCC(F)CC2)=O)N(C(c2n[nH]c(C)c2Cl)=O)C1 c1(C(=O)NCCCN(CCC)C(C2CCCSC2C)=O)cc[nH]c(=N)c1 N1(C(C(C2(O)CN(C(c3c(CC)ncs3)=O)C2)F)=O)Cc2c[nH]nc2C(C)C1 N1(C(C2CCC(C)(CC)O2)=O)CCC2(CCCN2C(=O)C(=O)N=S(C)(C)=O)CC1 c1(C(=O)NCC2C(CNC(CCOCCCOC)=O)C2(F)F)c(C)n[nH]c1C c1(C(=O)NCCCC2(NC(c3cccnn3)=O)CC2)ccc(O)nn1 Cc1c(C(=O)NCC2CCN(C(C3CC3C3CCC3)=O)CC2)cncc1Br C#Cc1ccc(C(=O)NC2C3CC4C2C4C3C(=O)NC(c2nccs2)C)cc1 c1(CC(C)NC(C2CC3CC3N2C(=O)CS(C)(=O)=O)=O)ccc(O)c(O)c1 N1(C(C2CC(=O)NC2)=O)CCC2C1CCCN2C(c1cnc2cccnc2c1)=O C1(OC)CC(NC(=O)CCC(C)SC)CN(C(c2ccc(CO)cn2)=O)C1 N=c1ccn(CC(=O)Nc2nc(N3CCNC3=O)no2)[nH]1 N1(C(C2(c3ccc(Cl)nc3)CC2)=O)CCC2CN(C(C3CCC4CC34)=O)CCC12 C(=O)(C(F)C(C)CC(C)(C)C)N1CCC(N(C(CCCOCCOC)=O)C)C1 c1(CSC)ccccc1NC(C)(CCn1cccn1)c1nnnn1C(C)C CC1(C)CC2(CC(NC(=O)C(CC3CCOCC3)NC(c3ccsc3Cl)=O)C2)C1 N1(C(CC(=O)OC)=O)CC2COCC2(C(=O)NC2CN(C(C)=O)CC2(C)C)C1 Nc1c(C(N2CCC(C(F)C(=O)NC3CC=CC3)C2)=O)cccc1F C1(C(N(C(C)C)CCN(c2nc(Cl)c(C#N)s2)C)=O)CS(=O)(=O)CC(=O)N1 c1(C(=O)NC(C2CCN(C(C3CCC(SCC)CC3)=O)C2)C)cc(O)ccc1F Cc1nc(O)c(C(=O)NCC(C)NC(=O)C2=CCCC2C)nc1C c1(CC)c(C(=O)NC2CCN(C(=O)C(O)CCSC)CC2)csc1C N1(C(CCC#C)=O)C(C(=O)Nc2cccc(CCC)c2)CCC12CC2 Cc1nc(C(=O)NCC(C)(C)NC(=O)CC(C)C(F)F)ccc1C#N C1(C(=O)NC)(OCCNC(=O)NC2(CC=C)CC2)CCOCC1.c1cn(C)nn1 C1(C(C)NC(C2(C(F)(F)F)CC2)=O)CCN(C(=O)CNC(=O)C2CC2)CC1 c1(OCCN(CC)CC)cccc(SCCc2ccccc2F)c1.C(C#N)O Cc1oc(S(N)(=O)=O)cc1C(=O)NC1CN(C(c2cc[nH]n2)=O)CCC1C C(C)(CCC(=O)NC1(C(=O)NC2CC(O)(CN(C)C)C2)CCC1)SC c1(CNC(c2cnc(OC)s2)=O)cc2n(n1)CCN(C(=O)CC1CCC(C)C1)C2 CCC(C)CCC(O)CC(=O)NCC(C)(C)OCCNC(=O)CNC=O CC(C)C(C(=O)N(Cc1ccccc1)CC1CCCC1)S.c1(N)cccnc1 C1(OC)CN(Cc2cscc2Br)C2(CCC2)C1 c1(C(=O)NCC(C)N(C(C(C)C2CC2)=O)C)oc(Br)nc1C(F)(F)F c1(C(=O)NC(C(=O)NCCC(CCC)O)CCOC)cc(C#N)ccc1N c1(OC)nccnc1-c1nc(CCc2scnc2C)n(C2CCCOC2)n1 Cc1ccc(C=CC(=O)NCCC2COCCN2C(c2csnc2C)=O)cc1Cl c1(C(=O)NC2CCC(N(C(=O)CC3(C#N)CCC3)C)C2)ccc(F)c(F)c1 C(=O)(C(O)CCOC)N1C(C(=O)NCC2(OCC)CN(C)C2)CC2CC21 Cc1cc(C(N2CC(NC(C3C4COCC34)=O)C(F)(F)C2)=O)cnc1F c1(CCN=C(N(C)Cc2c(C)occ2)NC2CC2C)c[nH]c2cc(F)c(F)cc12 N(C(=NCCC1CCCC(C)C1)NC1CCOCC1)Cc1c(C)cccc1 C(=O)(CC(C)C(=O)NCC1CN(C(C2(OC)CCSC2)=O)CC12CC2)OCC C1(C(N(C2CN(C(c3ncccc3Cl)=O)CC2(C)C)C)=O)CCCCCS1(=O)=O C=CC(C)(C)CC(=O)NCc1csc(CNC(=O)CCCOCCC)n1 N1(C(c2cc(COC)[nH]n2)=O)CC2(CCCC(CNC(=O)C(C)(C)CSC)O2)C1 N1(C(c2sccc2OC(F)F)=O)CCC2(C1)CN(C(C1(F)CC=CCC1)=O)C2 N1(C(CCc2cc(OC)c(O)cc2F)=O)CC2CCCCCCC2C1 N(C1CCCn2ccnc21)C(C1N(C(Cc2c(C)scc2)=O)CCC1C1CC1)=O c1(CNC(CC(CNC(CC(COC)C)=O)(C)C)=O)ccc2c(c1)CCC2 C1(C)(CC)C=C(C(=O)NCC2(O)CCN(C(c3csc(C(C)(C)C)c3)=O)CC2)C1 C12(C(=O)NC(c3nc(C(N4CCC5CC45C)=O)co3)C)CC(C#N)(C1)C2 N1(CCC(C)CC(=O)O)CCc2c(ccnc2Cl)C1 c1(OC)ncc(N(C)Cc2ccc(F)c(Cl)c2)cc1Br N1(CC)CN(Cc2ccccc2)CC1COC.c1ccccc1 C1(CC(C)(C)C)CN(C(c2cnns2)=O)CCN1C(c1ccc(C#N)s1)=O c1(CC(N2CCN(C(c3c(SC)nccn3)=O)CC2)=O)ccc(C)c(Cl)c1 C1(CNC(CCCn2ncc(C)c2)=O)CN(C(=O)C(O)C(C)C)CC1(F)F N1(C(C(CC)C)=O)CCC2(CC1)CC(NC(=O)Cn1cnc(C#N)n1)CCO2 c1(NCCn2c(C(C)C)nnc2)ccc(S(=O)(=O)NCCCN2CCCC2)cn1 C(=O)(C(C)(C)C(C)(C)C)NC(CC1CN(C(C2(C)ON=C(C)C2)=O)C1)C C#Cc1ccc(C(=O)NC2CC3(NC(=O)CN4CCC(C)(C)C4)COC2C3)cc1 c1(C(=O)NCC2C(NC(CC=C(C)C)=O)CC2)cc(Cl)c(Br)cn1 c1(CC)ccc(C(N2CC(OCCNC(=O)C(CC)OC)C2)=O)c(Cl)c1 C(=O)(CCC1=NNC(=O)CC1)N1C(C)CCN(C(=O)C(F)CC2CCC2)CC1 C(CC(=O)NC(C)(C)CC(C)(C)C)(C(F)(F)F)NC(C1C(=C)C1)=O CC(CC(C)(C)C)C(=O)N1CCN(C(c2coc(C(F)(F)F)c2)=O)CC1 c1(N(CCCC)C)nc(=NCc2cc(C)cc(Cl)n2)[nH]c2c(F)cc(F)cc12 CCC(C)CCC(=O)N1CC(C(=O)NCc2cnn(CCF)c2)CCC1C CN1CC=C(C(=O)NCC(C)(O)CNC(=O)C(C(C)(C)C)C2CCC2)C1.C(C)(=O)N NC(=NCC(C)c1ncc(C)s1)NC(C)C.c1(CC(=O)OC)ccccc1 N1(C(c2cn(C3CCCC3)nn2)C(=O)NCCCF)CCCCC12CC2 c1(SC)nc2ncnc(NC3CS(=O)(=O)CC3NC(c3cccc[n+]3[O-])=O)c2s1 C(=O)(C1CCCc2nc[nH]c21)N1CC2C(N(C(C=CCN(CC)CC)=O)C)C2C1 c1(C(=O)NCC2OCC(CNC(=O)CCCCC3CC3)C2)cnn2ncccc12 N1(C(C(C)=C(CC)C)=O)CC2CCCN(C(c3ncnc4c3CCC4)=O)C2C1 N1(C(Cc2c(C)non2)=O)CCCC(CCNC(C2CC3C(C2)C3(F)F)=O)CC1 C(=O)(CS(=O)(=O)CCOC)NC(COCCOC)C(=O)NC1CN2CCC1CC2 C1(CC(=O)N(C)CC2COCCO2)CC2(C1)CN(C(C1CCCCC1(C)C)=O)C2 c1(CC)nc(=NC(=O)NCC2COCC2n2cc(COC(C)(C)C)nn2)n(C)[nH]1 N1(C(C2(CCCC)CC2)=O)CCC(C)(C)C(NC(=O)CCCCC(=O)NC)C1 Cc1cc2[nH]c(C(=O)NC3CC3CNC(=O)CC=Cc3cccc(F)c3)cc2o1 Cn1ccc(C(=O)NC2CCCC2(C)NC(C2CC2c2ccco2)=O)cc1=O C1(C(N2CCCC(c3onc(-n4c(C)ncc4)n3)C2)=O)COC2COCC2O1 c1(C(N(CCNC(C(C)OC)=O)C(C)C)=O)ccc2c(c1)CC(C)O2 c1(C(=O)NCC2CCC(C(NOCC#C)=O)O2)csc(C)c1C c1(OC)ccc(Cl)c(C(c2nnnn2C2CC2)NC(C)CC2CCOCC2)c1Cl c1(SC)cc(C(=O)N(C2CC(NC(=O)C(C)S(N)(=O)=O)C2)C)ccc1N C1(CNc2c(C)c(N3CCC=C(Br)C3)ncn2)CCCC2(CNC2)O1 N1(C(C(c2ccn(C)c2)C)=O)CCCC(O)(CN(C(=O)CSC(F)F)C)C1 C1(C(=O)NCC(CC=C)NC(=O)C=CC)CC2CC(=O)C1O2 C12(C(N(CC(COC)O)C)=O)CCCC1N(C(=O)CC1CC(C)C1)CC2 C1(CC(N)=O)(NC(C2COC(=O)C2)=O)CCN(C(=O)CCF)CC1 N1(C(CCC(=O)NCC)=O)CCC2CCCC12CNC(c1nccnc1CC)=O C1(CC(=O)NCC2CCCCO2)CC(O)CN1C(=O)C=CC(F)F C(C(CC(=O)N(C1(CCC)CC1)C)OC)NC(C1(CC)CCC1)=O c1(C(N2C(CNC(Cc3c(C)cccc3)=O)CCC2)=O)cc(C#N)ccn1 c1(C(=O)NC(C)CNC(c2csc(Br)c2)=O)cc(C(F)(F)F)ncn1 C1(NC(c2cccc(CSC)c2)=O)CCCCN(C(=O)C(O)C(C)(C)C)C1 C1(C(=O)NCC(CC=C)NC(c2cc(C)c(CO)cn2)=O)COCC2(CCC2)O1 c1(C(=O)NC(CC=CC)C(=O)N(C)Cc2cnccn2)nccc(C)c1N N1(C(c2c(CC)[nH]cc2)=O)CC2OCC(NC(c3ccc(OC)cc3F)=O)C2C1 c1(C(=O)NCC(CC=C)NC(=O)C(C)CC=C)ccc(Br)cc1 n1(CC)cc(C(=O)NC(C2(CNC(=O)CCC3CCCN3C)CC2)C)c(C)n1 c1(CS(C)(=O)=O)nc(Cl)cc(=NCCCC2CCCC2)[nH]1 C(=O)(CCCC(=O)NC(C)CC(=O)N1CCC(CF)C1)OCC C(CC(C(=O)NCc1cnn(C)c1C)NC(C1CCCCS1)=O)OC c1(CN2CCC(CC(=O)NC(C(C)O)CO)C2)c(F)cc(Cl)cc1Br C(=O)(C1=C2CCCN=C2NN1)NC1C(NC(=O)C=CC(F)(F)F)CCOC1 c1(N2CC(NC(C3C(C(F)(F)F)C3[N+](=O)[O-])=O)C2)nc(C2CC2)nc2c1CCC2 C1(F)(CNC(=O)COc2ccccn2)CCCN(C(c2cc(O)ccc2O)=O)C1 c1(C(=O)NC(C2CCN(C(C(F)=CCC)=O)C2)C)coc2cc(F)cc(F)c12 N1(C(CC=CCC)=O)CC(NC(c2coc(-c3cccnc3)n2)=O)C2(CC2)C1 c1(CC)ccc(F)c(C(N2CCCCC(NC(=O)C(C)(Cl)Cl)CC2)=O)c1F c1(NC(C2CC(NCc3ncn(C)n3)C2)=O)cc(F)c(Cl)cc1Cl C1(CCNC(C(C(C)O)NC(N)=O)=O)CCCN(C(C2(O)CCC2)=O)CC1 c1(C(=O)NC2(C)CN(C(C(C)NC(=O)NC)=O)C2)cc(F)cc2nn(C)cc12 O=S(=O)(c1ccc(Br)cc1NCc1nc(Cl)cs1)NCc1cc(F)ccc1F C1(NC(c2nc[nH]c2C(F)(F)F)=O)CCOCC1NC(C1CCOCC1)=O C(=O)(C1=CCCOCC1)N1CCCN(C(c2c(C#N)ccs2)=O)CC1 C1(CCNC(C(C)n2cncn2)=O)CCCCN1C(c1n[nH]cc1C(F)(F)F)=O c1(C(=O)OCC)nnc(SC)nc1N1CC2CC2(C(=O)NCCSC)C1 O=C1CC(C(=O)NCC23CCC2CN(C(=O)CN2CCCC2)C3)=NN1 N1(CC(=O)NCC(C2CCCC2)C)CCN(C(=O)CCc2nncs2)CC1 c1(C(N2C(C(=O)Nc3ccc(Br)nc3I)C(O)CC2)=O)ccc2occc2c1 C(CC#CC(C)(C)C)NC(CCC(C)NC(=O)CC1CC(=O)NC1=O)=O C1(C(N2CC(C)(CC)C2)=O)N(C(=O)C(C)N2CCCC2)CC12CCCC2 C1(NC(C(=Cc2ccco2)C)=O)C2CC(O)C1N(C(c1cnnc(O)c1)=O)C2 CC1CCCn2c(CC(=O)NCC3C4CN(C(=O)CCC(C)(C)C)CC34)cnc21 C1(C(N2CC(C)(OC)C2)=O)CC2CC1CN(C(=O)CC1CCC(C)(C)O1)C2 CC(C)(C)CCC(=O)N1CCC(CC(=O)NC2(c3ccncc3)CC2)C1 N1(CC)CCC(NC(=O)C=CC(C)(C)SC)CC1.c12sccc1CNC2=O c1(C(=O)NCCC2(CNC(C3CC4CC3CO4)=O)CC2)ccc([N+](=O)[O-])cn1 C1(C)(C(=O)NCCCC2N(C(c3cc(OC)n(C)n3)=O)CCC2)CCCC1(F)F n1(C(C)C)cc(C(=O)NC2CN(C(=O)C(CO)N(C)C)CC23CC3)c(O)nc1=O C#CCC(C)(C(=O)Nc1cnc(C)c(C)c1)NC(=O)CC(C)C(F)F CC1(C)C2CCC1(C(=O)NCC1CC1CNC(=O)CCSc1ccccn1)CC2 C1(CNC(c2nc(OCC)oc2)=O)CC(C)N(C(c2cnn(CC)n2)=O)C1 c1(C(=O)NCC2CC2NC(C23C=CC(CC2)C3)=O)cccc2nncn12 N#Cc1nccc(N2CCC(O)C2c2ccccc2OC(F)(F)F)n1.C1(=O)CO1 c1(C(=O)NCC2(CN(C(C(C=C)O)=O)C)CC2)cc2c(=O)[nH]ccn2n1 Cn1cc(C(N2CCC(CO)(NC(=O)CC3(C#N)CCC3)C2)=O)c2ccccc12 N1(C(CC2C(C)=NNC2=O)=O)CC2CCN(C(c3cc4sc(F)cc4[nH]3)=O)C2C1 [N-]=[N+]=NCC(F)CCNC(C1(NC(=O)CC2CCCC2O)CC1)=O C(=O)(CCCCC(F)(F)F)NCC12OCC(NC(c3nccc(C)c3)=O)C(C1)C2 C1(NC(C(C(C)C)C#N)=O)CN(C(C2CC3(C2)CC(O)C3)=O)C2(CCC2)C1 CC(C)CC(C(=O)NCC(O)C(C)O)ONC(C1CCC2(CCC2)O1)=O c1(C(C)OC)nn(CC(=O)OC(C)(C)C)c(=O)o1.C1C(=O)N1 C1(C(N2CCC(NC(C=CCC)=O)(CF)C2)=O)Cn2c(C)nnc2CN1C c1(SC)cc(F)ccc1C(=O)NC(CO)C(C)NC(=O)Cn1ccc(C(F)F)n1 C1(C(N(C2CC(=C)C2)C)=O)CN(C(C2(C(=O)OC)CC2)=O)CC(C)(C)C1 C1(CNC(C2(CC)CC2)=O)CC(F)(CNC(c2ccc(C(C)C)o2)=O)C1 N1(C(CCN(C)C)=O)Cc2[nH]nc(C(=O)NCCN3CC(C)(O)C3)c2C1 N1(C(CC=CC)=O)CCC(C)(CNC(C2C=CCS2)=O)C1 N1(C(c2c(COC)cccc2)=O)CC(C)C(N=c2ccc(C#N)c[nH]2)C(C)C1 N1(C(c2c(C)nsc2)=O)CCCC(CNC(C2CC3CCC2C3)=O)C1 c1(C(N2CC(CC)C(NC(=O)C(=O)NCC(F)F)CC2)=O)c([N+](=O)[O-])cnn1C CP(C)(=O)c1cnc(C(=O)NCC2(O)CN(C(C3COCCC3(F)F)=O)C2)nc1 N1(C(CC(=O)NCC)=O)CCCC(N(C)C(c2ccc(C(N)=O)[nH]2)=O)C1 Nc1ccc(O)c(C(N2CCC(OCCNC(C3CCOC3)=O)C2)=O)c1 N1(C(=O)OC(C)(C)C)CC2CC(F)C1C2C(=O)NCc1ccco1 C1(C(N(C)CC2N(C(C=CC(CC)=CC)=O)CC(F)C2)=O)CC2CCC(C1)C2O C(C(O)CC(=O)NCC1=NOC(C)C1)NC(c1cn(CC=C)nn1)=O c1(C(C)=O)cc(C(=O)NC(C)CN(C)C(C2CC2(C)C(C)C)=O)c(C)o1 N1(C(C(CCSC)OC)=O)CCC2(CCCN(C(c3ccc(CO)s3)=O)C2)CC1 Cc1cc(CNC(=O)C(CCF)NC(c2nnsc2C)=O)c(C)s1 n1(CC)nc(C(=O)NCc2cnn(C)c2C(=O)NOCC(N)=O)c(C)n1 N1(c2ncc(C)s2)CCC2(CC1)CCN(C(=O)COc1ccc(Cl)cc1)CC2 S(=O)(=O)(c1ccc2c(c1)COC2)NCC(=O)NC1C(NC(COC(C)C)=O)CC1 S(=O)(=O)(c1ccc(F)cc1Br)NC(C(c1cc[nH]c(=N)c1)(C)C)=O c1(C(N2CCC(NC(CCC(=C)C)=O)(CF)C2)=O)cccc([N+](=O)[O-])c1Cl C(=O)(C(COC)CC(C)C)NCC(CC=C)C(=O)NC(C)Cc1ccco1 N#Cc1cccc(OC2(C(=O)NC3(c4ccccc4)CCC3)CCCC2)c1 C(C(F)(C(=O)N(c1ccsc1)C)C(C)C)NC(C(C1CC1)OC)=O C1(C(C)N(C)CC)CCCN(C(=O)CC2CCN(C(C3(CCCF)CC3)=O)C2)C1 C1(NC(CCN(CC)CC)=O)CC2CCC(C1C)N2C(=O)C(CC)CC(C)C N1(C(c2n(CC#C)ccc2)=O)CC2CC2(C(=O)NC(C)CCC2CC2)C1 CCCC(O)(CNCC(=O)NCc1ccn(-c2ccccc2)n1)CCC C1(NC(=O)CC2COCCO2)CN(Cc2ccc(F)nc2F)CCC1(F)F c1(C(N2C(CNC(C(c3ccc(Cl)cc3)CC)=O)CCC2)=O)cccc(F)c1N C(N=c1[nH]c(Cl)ncc1Cl)C1C(NC(CC2CCC(C)CO2)=O)CCCC1 c1(C(N2C(CCNC(c3c(C)nsc3C)=O)CCCC2)=O)ccc(N)c(F)c1 N(C1CCCc2n[nH]cc21)C(=O)NC1C(N=[N+]=[N-])COC1 CC1CC(NC(=O)Cn2cccn2)CCN1C(=O)CCc1cc(F)ccc1F c1(C(=O)NCC(C)(CNC(C2(C)CCCC2O)=O)OC)ccc(N(C)C)nc1 n1(CC(=O)NCCNC(C(C)(F)c2ccccc2)=O)nc(O)ccc1=O Cc1cc(C(=O)N(CC(C)(C)CNC(=O)CCN2CCCC2)C)cc(C)c1O c1(C(N2CC(NC(C34C(CN(C(C)=O)C3)C4)=O)C2)=O)cnc2c(c1)N(C)CCO2 N1(C(C2OCCN(C)C2)=O)CCC(NC(c2cn[nH]c2)=O)C12CC2 C1(C(C)NC(c2cncn2C)=O)CN(C(c2cc(Cl)cs2)=O)CCO1 N1(CC(=O)NC(CN(C(=O)CC(=O)N(C)C)CC)C)C(=O)NC2(CCCC2)C1=O C(CS(=O)(=O)C(C)(C)C)c1cc(N2CCC(c3nncs3)C2)nc(COC)n1 C1(CNC(=O)C2=CCC2)C2CCCC1N(C(c1cnc3ccoc3c1)=O)C2 C1(n2cc(CCCOC)nn2)CN(C(=O)CNC(=O)CC2CCOCC2)CC1C C=C=CCCC(=O)N1CC(C2CN(C(c3cnc[nH]3)=O)CCO2)C1 C1(F)(C(=O)NCCOC)CCN(Cc2ccc(C(=O)O)o2)C1 N1(c2ccnc(SC)n2)CC2CC(NC(c3c[nH]nc3C(C)C)=O)CC2C1 c1(C(=O)NCC(C(C)C)NC(c2cc(OC)ns2)=O)ccc(CCF)cc1 c1(CC(=O)N(CC(O)CNC(=O)C(C)(C)S(C)(=O)=O)C)ccc2c(c1)CCCO2 C1(C(N2CC(C)(NC(c3cc(-c4cccnc4)[nH]n3)=O)C2)=O)CCCS1(=O)=O C(=O)(C(F)(F)C(C)(C)O)NC1CCN(C(Cc2ccc(C)cc2Cl)=O)CC1F CCC(CC(=O)NC1(C)CC(NC(=O)CCN2CCCCC2)C1)OC CC1(C)CCCC(CC(=O)NCC(C)(C2CC2)NC(=O)CCCCNC(N)=O)C1 c1(C(N(C(C)C)CCN(C(=O)CNc2nccs2)C)=O)cccc[n+]1[O-] CC(C)CS(=O)(=O)CC(=O)NCC(=C1CN(C(=O)CCN2CCC(F)C2)C1)F C(C)(C(C(=O)NCC(C)(C)CNC(=O)C(=Cc1ccccc1)OC)N(C)C)OC c1(NCc2c(CC)nn(C)c2)nc(N2CC3CC3(CO)C2)nc2sccc12 c1(N(C)C)nc(C(=O)NC2CC(CNC(=O)CCc3ccccc3)C2)[nH]c(=N)n1 CC1CN(C(=O)CCC2CCOC2)CCCN1C(c1ccc2nn[nH]c2c1)=O c1(C(=O)OCC)cc(CNC2CCC3(CC3)C2)c(C)o1 N1(C(C(CCCC)C)=O)CCC2OCCN(C(=O)CN(C)C3CC3)C2C1 Cc1cc(C(=O)NC(CNC(=O)C(CO)N(C)C)C(C)(C)C)nc(C)c1 c1(C(N(CC(=O)NC(C(O)CO)C2CC2)C(C)C)=O)c[nH]c(C#N)c1 c1(NC)c(C(=O)NCC2CCN(C(c3scnc3COC)=O)C2)cccc1F c1(OC)ncnc(C(N2CC3CC(CNC(c4cc(CO)on4)=O)C3C2)=O)c1F C1(CNC(C2(CCCC)CCCC2)=O)COCCN(C(c2cc(C#N)no2)=O)C1 c1(C(=O)NC(C2OCCN(C(c3ccc(C)nn3)=O)C2)C)cnc(C)cc1C c1(C(=O)NCCC(C)NC(C2C(C)C2C)=O)nn(C)c2c(=O)[nH]cnc12 c1(CN2CC(C(=O)NCCc3ccccc3)(CF)C2)c(F)ccc([N+](=O)[O-])c1F C(Cn1ccnn1)(C(=O)N(C(C(N)=O)C1CC1)C)NC(C(C1CCOCC1)C)=O C(=O)(C(C)(CNC(=O)C=CCF)CC)NCCC(CC)C C(=O)(CC1OCCc2sccc21)NC1C(C)N(C(=O)C=CC(C)(C)C)CCC1 C=C1CCN(C(C2CCC(C)(C)CC2)=O)C(C(=O)NC(C)CC2CCCCC2)C1 c1(CCNC(CSCC#C)=O)ocnc1CNC(=O)C(c1cnn(C)c1)O C1(CNC(CC2C=NN(C)C2=O)=O)CN(C(=O)CCCn2cccn2)CC1(C)C C1(CNC(n2cnccc2=O)=O)CCCC12CCN(C(=O)COCC1CC1)CC2 CC1CC(C(=O)NCC2(C(=O)NC3CC3C3CC3C)CC3(CC3)C2)CN1C C(=O)(C(C)CN(C(=O)CCN(C(=O)CNc1ncccn1)CCO)C)NC c1(CCC)cc(C(=O)NCCN(C(=O)CC(C)COC)CC2CCCC2)ccn1 CC1CN(C(c2cc(O)ncn2)=O)CC(C)N1C(=O)C(C)(C)Cc1cnn[nH]1 C(C(CNC(C1CCCC(C)(C)O1)=O)S(C)(=O)=O)NC(C1(CC)CC1)=O C1(NC(CC2(C)CCOCC2)=O)CC2CCC1CN2C(c1ccnc(S)c1)=O c1(CC(C)C)ccc(CCNC2CCCC(NS(C)(=O)=O)C2)cn1 C(=O)(CC(C)C(F)F)NCC(CO)NC(CN(C(=O)OCC)C)=O N1(C(c2nc(C)oc2C)=O)CC2CC(NC(=O)Cc3ccco3)CC2C1 c1(C(=O)NCC2CC(NC(C=CC(C)C)=O)C2)ccc(OCF)cc1.C1CO1 c1(C(N2CC(OC)C(NC(c3cncc(SC)c3)=O)C2)=O)ccc(F)c(Cl)c1 C(CCCC(C)(C)C(=O)NNC(=O)c1c[nH]nc1Br)NC(C(C)=C(C)C)=O N1(C(CCCCOCC)=O)CCC2CCN(C(=O)C3=NNC(=O)C3)CC2C1 N1(C(C(C)N(C(=O)C(=O)N(C)C)C)=O)CCC(C(C)(C)C#N)C1 c1(C2(C(=O)NCC(CO)NC(C3(C)CC(C)C3)=O)CCC2)ncccc1F c1(C(=O)NCC(CC=C)NC(c2ccsc2C(F)(F)F)=O)cc2n(c1)CCC2 Cc1c(C(=O)OC2CCOC(C)(C)C2)[nH]c2cc(Cl)ccc12 N1(C(c2ccc(C)o2)=O)CC(C)CN(C(=O)CCc2nc(C)no2)CC1C N1(C(=O)C#CC2CCOC2)CC2CCN(C(c3ccc(Cl)[nH]3)=O)CCC2C1 C1(NC(c2cc(CN(C)C)on2)=O)CCN(C(C2CCCN2N=O)=O)C12CC2 c1(COC)nc(=NC2CS(=O)(=O)CC2NC(c2ccc3c(c2)NC(=O)C3)=O)s[nH]1 c1(C(=O)NC2CC3CC(C2)N(c2nncs2)C3)ccc2ncc(=O)[nH]c2c1 c1(C(N(CCC(C)NC(C2(O)CCC2)=O)C)=O)ccc2nc(O)cn2c1 C(=O)(C(C(C)C)NC(=O)OC(C)(C)C)NCCN(C(C=C(C)Cl)=O)C1CC1 C1(N(C(C=CCN(C)CC)=O)CC)CCCN(C(=O)Nc2coc(C(N)=O)n2)C1 C(c1cccnc1)=C(C)C(=O)NC1CC1NC(c1ccn(C(C)(C)C)n1)=O C1(C(=O)NC2C(C(C)C)C2)(CNC(=O)CC(C)F)CCOCC1 c1(C(N2CC3C(CNC(Cc4cc(C)on4)=O)(C3)C2)=O)ccc(Cl)c(F)c1 C1(NC(CNC(CCCCC)=O)=O)CCCCN(C(c2cccc(CO)c2)=O)C1 N1(CCCC(=O)NC(CCC)CCCc2ccccc2)C(=O)NC(C)(C)C1=O C(C(=O)N(CCC(=O)NC(C)C(C)SC)CCO)(C(C)C)OCC.C(C)=O c1(C(=O)NCc2cncc(C(=O)NCC(C(C)C)CO)c2)cnn(C)c1C#N C1(C(C)NC(C2CC(CN(C)C)C2)=O)CCN(C(=O)C(O)Cc2ccccc2)C1 N1(C(c2c(C)nsc2C)=O)CCC2(CC1)CC2CNC(=O)CC(=O)NCC1CC1 C1(CNC(C(C)O)=O)CN(C(c2ncc(OCC3CC3)cc2F)=O)CC(C)(C)O1 N1(CC)C(C)CN(C(C2CCN(C(C3CC(=O)CCO3)=O)CC2)=O)CC1C N1(C(Cc2ccc(C)cc2C)=O)CCC2(CC1)CN(C(=O)C(C)CF)CC2CO Cc1cccc(NC(=O)CC2CN(Cc3cccc(CC(=O)O)c3)CCO2)c1I C(CC(C(=O)NC(C)C(=O)NCCOC)NC(c1ccoc1C)=O)OC c1(C(=O)NCC(C)NC(CCc2cc(C)no2)=O)cc(C#N)ccc1N C(C(=O)NCC(C)(C(C)C)NC(=O)CCn1ccnc1C(C)C)(C(C)C)OCC N1(CC(N2CC(NC(C(C)N(CC)CC)=O)C2)=O)CC2CC2C1 c1(C(=O)NCC2CCCN(C(C3(C)CCCCO3)=O)C2)cc2ccccc2s1 C(=O)(C1SCCc2ccccc21)N(CCCNC(C1CC2(CC2)CO1)=O)C1CC1 C(=O)(N1CC(n2cc(-c3ccccc3I)nn2)CO1)C1CCC(=O)N1 Cc1cncc(C(=O)NCC2(O)CCN(C(=O)C(N)=O)C2)c1C C(=O)(CCCC(C)(C)CC)N(C1CCCN(C(C(c2ccccc2)OC)=O)C1)C C12(C(=O)NCC3CCN(C(c4ccn(C5CC5)n4)=O)CC3)CCCC1OCC2 CC(C)C#CC(=O)NCC(C1CC1)NC(=O)CCCOc1ccccc1Br C#Cc1ccc(C(=O)NC2(CC=C)CCN(C(c3coc(C(F)F)c3)=O)C2)nc1 N1(C(c2ccc(NC)cn2)=O)CCC(C)(C)C(NC(c2oc(C)cc2C)=O)C1 c1(C(=O)NC(C2CCOC2)CNC(CC2CC(=C)C2)=O)cc(C(=O)OC)n(C)c1 N1(C(C(COC)C(F)(F)F)=O)CCC2C(=O)OCC12CO c1(OCC)cccc(C(=O)NC(C2CCCN(C(=O)C(C)(C)CF)C2)C)c1 C1(C(N2CC(CCC)C(NC(C3CCCCC3C)=O)C2)=O)CC2(CCO1)CC2 N(C1CCCc2nc(C)[nH]c21)C(C(=O)Nc1ccc(OC)cc1)C CN1CC(O)CC1C(=O)NCCCCCCN(C)C(C1CC2CCC2C1)=O C1(C)(C(NOC(C=C)C)=O)CCN(C(C2CCC(CC)C2)=O)CC1 C1(NC(=O)CSCC(=O)NC(c2ccccc2)=O)CC(=O)N(O)C1 CC1=C(C(=O)N2CC3CC2CCC3NC(=O)Cc2coc(C)n2)CCCO1 C1(NC(C=C(CC)C)=O)CC2CC1CN(C(c1n[nH]c(CC)c1Br)=O)C2 c1(CNC(=O)NCC2(C)CCOCC2)ccc2c(c1)CC(=O)N2 C(C)(CN=c1ccc([N+](=O)[O-])c[nH]1)N(C(c1ccc(OCC=C)cc1)=O)C Cc1ccccc1C=CC(N1CCN(C(c2cccn2C)=O)C(C)C1)=O C#CCC(CC(=O)NCCN(CC(F)F)C)NC(=O)CCCCC c1(CC(N2C(C3CCN(CC)CC3)CCOCC2)=O)cc(C(F)(F)F)cc(F)c1 C1(C)(CC)CCN(C(C2(CNC(c3cnc(C)cn3)=O)CC=CC2)=O)CC1 c1(-c2cn(CC(=O)NC(C(=O)NC)Cc3ccccc3)nn2)cc(F)ncc1F c1(C(N(C)CC2CN(C(C3(SC)CCC3)=O)C2)=O)cc2nn[nH]c2cc1F C1(OCc2cnc(C3CCC3)s2)CCN(C(=O)NCC(n2cncn2)C)CC1 c1(NCCCCCC)ccc(-c2csc(C(=O)CN3CCC(CO)CC3)c2)cc1 C#CC1(C(=O)N2CC=CCO2)CCN(C(=O)CSC(F)F)CC1 CC(C)(C(=O)NNC(=O)c1ccc(O)c(I)c1)C1CCO1 n1(CC(N)=O)cc(C(N2CC(CO)(NC(c3coc(Br)c3)=O)C2)=O)nn1 C1(CNC(C(CC)O)=O)(CO)CCN(C(=O)CCC(C)C)CC1 C(C1Cc2ccccc21)OC(c1ncc(C#C)cn1)=O c1(NC(C2=CCN(C(CC3CC(=O)OC3)=O)C2)=O)cccc2c1CCC2 c1(C(N2C3CN(Cc4ccc(CO)cc4)CC23)=O)cc(F)c(Br)c(F)c1 C1(CC)CN(C(c2cn(C)cn2)=O)CCN1C(c1[nH]cnc1-c1cccnc1)=O n1(CCC(=O)N(CCCCCC)CCNC(C2C(C)C2C)=O)ccccc1=O C1(C)(C(=O)NCCN(C2CCCC2)C(c2ccc(SC)o2)=O)CC2CC2C1 Cc1ccc(F)cc1C(=O)NC1CC(NC(C2CCC3CC23)=O)CC1O c1(C(=O)NC2(CF)CCN(C(CCCCC)=O)C2)cnn2c(Cl)cccc12 C1(C)(C(=O)NC(c2nc(C(=O)NC3CN4CCC3CC4)co2)C)CCCN(C)C1 c1(CC)ccc(C(=O)NCCCOCCNC(c2ocnc2C)=O)c(OC)c1 N1(C(C(C)=C(C)C)=O)CCC2(C1)CN(C(C1CC3CCC1O3)=O)C2 C1(OC)CC2CC(C(N3CCN(CCNC(C4(C)CCCC4)=O)CC3)=O)CC12 c1(C(=O)NCC2(C)CCN(C(=O)C(F)=C3CCC3)C2)cnn2c1S(=O)(=O)NCC2 O=S(=O)(c1c[nH]ccc1=NCC1CCC12CCOCC2)NCCc1nncs1 N1(CC(=O)NC2C(CNC(CCS(C)=O)=O)COC2)C(=O)CC(C)(C)C1=O N1(C(c2cc(COC)cn2C)=O)CC2CC1CN2C(c1c(C)nn(C)c1C)=O C1(NC(c2cc(CF)on2)=O)CC2(CCCCN2C(=O)CCC[N+](=O)[O-])C1 Cc1ccc(F)c(NC(C2(C)CCN(C(C3CC3C3CC3)=O)C2)=O)c1 O=C(CCCC(F)(F)F)NCCC1CCN(C(=O)CCC2CCOC2)C1 c1(C(=O)NCCOCCN(C)C(C2CC2(C)C(F)(F)F)=O)c(F)ccc(N)c1F C(C)(C)(CC(F)C(=O)NCc1cnc(C)n1CC)NC(C(C(CC)O)C)=O c1(C(N2C(CNC(C(CCC)C(C)C)=O)C=CC2)=O)ccc2ccccc2c1F C(=O)(CS(N)(=O)=O)N(C(C)C)CCNC(=O)CCN(C)CCc1ccccc1 c1(OC)cccc(C2(NC(C3CN(C(=O)Nc4ccc(=N)[nH]n4)C3)C)CC2)c1F C(C1C(C(=O)N(C(C)C)CC23CC(NS(=O)(=O)CCCCl)(C2)C3)C1(C)C)=C(C)C Cc1ncc(C(N2CCCC2C(=O)NCCC2CCC(C)O2)=O)cn1 c1(C(C(=O)NC(C)CCNC(=O)COCC(C)(C)C)(F)F)nc2ccccc2s1 CC1(C)C(CNC(c2ccncc2)=O)CCN1C(C1COCCO1)=O Cc1ccc(C(=O)NCCC2(NC(=O)CSCCC#N)CCCC2)c(=O)n1C CC1CCn2cc(C(N3CCCC(c4nnc5ccccn45)C3)=O)nc2C1 C(=O)(CCCCC(=O)c1ccccc1)NCC1N(C(C(COC)O)=O)CC(O)C1 CC(CS(C)(=O)=O)C(=O)N1CC2CCN(C(c3cccc(CN(C)C)c3)=O)C2C1 N1(C(C)=O)CC2CCCC2(C(=O)NC2CC(=C3CCC3)C2)C1 c1(C(=O)NCC(=O)NC(C)CC(C)NC(c2cnnn2C)=O)ccc([N+](=O)[O-])cc1 CC1CN(C(=O)C(c2ccc(F)cc2)=O)CC1NC(=O)CC1CCC(=O)N1 C1(CNC(C(CC)(C)CC)=O)CN(C(=O)CCCc2nc(C)no2)C2CCN1C2 CCC(C(=O)NCCC1CC(NC(=O)C(=O)Nc2ncc[nH]2)C1)C1CCOCC1 CC1(C)CCN(C(C2CCCC2NC(c2ccc(OC(F)(F)F)cn2)=O)=O)CC1 C1(F)(CNC(CC(C)OC)=O)CCC(CNC(=O)Cn2nccn2)C1 C1(NC(CCCC#CC)=O)COC2CN(C(C3C=CCCC3)=O)CC12 CCC(O)C(F)(F)C(=O)NCC1CN(C(c2ncccc2Cl)=O)CC1(F)F C1(CC=C)(C(=O)NC(c2csnn2)C)CN(C(=O)CCC2CC2(C)C)C1 C1(CC(C)C)COCCN1C(c1sccc1CNC(c1cc(Cl)n[nH]1)=O)=O N1(C(C(C)CC2CCC2)=O)CCC(C(C)(O)CNC(C2(O)CCC2)=O)CC1 CC(C)CC(C)C(=O)NCC(C)(C)CNC(C1CSCN1C(=O)C(C)(C)C)=O C1(C)(C(c2cn(C(C)C(=O)O)nn2)N(C)C)CCN(C(=O)C=C2CCOCC2)CC1 C1(CC(=O)NC(CCC)(C)CC)C2CCC(C2)N1C(=O)C=C=C(C)C CN=c1cc(C(=O)NC(C(=O)NCCCn2ccnn2)C2(C)CC2)cc[nH]1 c1(C(N(C)CC2N(C(CCC(=C)C)=O)CCOC2)=O)cc(C)c2nc(C)cn2c1 c1(CC(N2CCC(NC(C3CC4(CSC4)C3)=O)C2)=O)ccc2ccccc2c1 C1(CNC(C=Cc2nc(C)sc2)=O)CN(C(=O)C(C)C2CCCC2)C2(CCC2)C1 CC1CCC=C1C(=O)NCC1(CNC(=O)COC2CC(F)(F)C2)CCC1 CC(C)(CNC(=O)CC1C(NC(c2cc[nH]n2)=O)CC1O)CC(F)F C1(C(=O)NCCCCNC(c2occ(C)c2)=O)CSC(c2ccccc2)=N1 C1(CNC(=O)NC2(C(N)=O)CCOC2)CCCOC1C1CC1 c1(C(=O)NC(C(=O)N(CCOC)CCO)CSC)cc(CSC)n(C)n1 C1(CNC(C2(CC)CCC2)=O)CN(C(=O)Cc2cc(C)no2)CC12CC2 c1(C(C(=O)NCC(F)F)N(CC(=O)OCC)C)cc2ccccc2o1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NCC1OCCN(C(c2ccoc2)=O)C1 c1(C(c2nnnn2C2CC2)NC(=O)CCCCN2CCCC2)ncc(F)cc1F N1(C(COC(CNC(COCCOC)=O)(C)C)=O)CCSC(C)CC1 C1(NC(CN(C)C(C2CCC(C)(C)C2)=O)=O)CCN(CCO)CC1 C1(c2c(OC)cccc2)CN(C(c2c[nH]ccc2=O)=O)CCN1C(=O)CC(C)O CCCCC(CC(=O)NCC(C)(C)C(N)=O)NC(=O)C(C)(O)CCN(C)C Cc1coc(C=CC(=O)N(CCNC(=O)CCC2CC2)CC2CC2)n1 N1(C(C(C)N(C)C)=O)CCC2(CC2C(=O)N(CCCC(O)CO)C)C1 CC1CN(C(c2ccc(N)c(O)c2)=O)CCC1CNC(=O)CCNC(N)=O C1(O)(CNC(C(C)n2cnnn2)=O)CCN(C(=O)CC(C)NC(N)=O)CC1 C1(NC(=O)CN2CCCC2=O)CCC2CC1CN2C(C12CCC(C1)OC2)=O c1(C(N(CC(C)NC(c2ccc[nH]2)=O)CC)=O)cccc(OCCOC)c1 N1(C(CCCCCC)=O)CCCCC1C1CCCN1c1cc(O)ncn1 N1(C(c2ccc(F)s2)=O)CCOC2CN(C(C3(F)CC3)=O)CC12 C12(C(=O)NC3CC(CCNC(C(C4CCCC4)SC)=O)C3)CCC(O)(CC1)CC2 C1(C(N2C(CSC)CCC2)=O)CN(C(c2cnccn2)=O)CC(C)(C)C1 c1(OC)ccc(-c2cnc(-c3ccccc3)s2)cc1CN1CCC2(CCC2)C1 C(=O)(CCC(=O)NCC1CC(NC(c2cc(Cl)ns2)=O)C(O)C1)NCCC c1(C(N(C2(C)CN(C(C(N3CCOCC3)C)=O)C2)CCO)=O)cn(C)cc1CN N1(C(C(C)N(C(=O)CC2(C(=O)OC)CC2)C)=O)CCCC(N(C)C)CC1.N(C)C Cc1ccc(Cl)c(C(C(=O)NC2COC2)N(C)CC2CC2)c1 N1(C(C(CC)Br)=O)CCC(N2CCC(N(c3ccccc3)C)C2)C(C)CC1 CC1OCCC12CN(C(C(=O)NC1CC1)C1CC1c1ccnn1C)CCO2 C1(NC(c2cc(C(=O)OCC)n[nH]2)=O)CCCC(NC(C2CNC(=O)N2C)=O)C1 c1(C(=O)NCC2(CC(=O)N(C3CCCCC3)CC#C)CC2)nnc(O)nc1O C12(C(N3CC(CNC(C4CCSCC4)=O)OCC3)=O)CCC(F)(CC1)C2 c1(C(=O)NC(C2CCCN2C(=O)C(C)CC(C)(C)C)C)ccc2cncn2c1 N1(C(C(C)C2CC2)=O)CCC(C2(O)CN(C(=O)CC(C(F)F)C(C)(C)C)C2)CC1 CC1(OCC(=O)NCC(C2CCC2)NC(C2CC2C(F)(F)F)=O)CCOCC1 CC(N=c1cc[nH]cc1S(=O)(=O)NCC1CC(=O)N(C)C1)c1n[nH]c(=N)s1 C1(C(=O)NCCCCC(C)NC(CCC(=C)C)=O)CN2CCCC2CO1 C1(CNC(CC(CN(C)C)O)=O)CC(C(=O)NCCC(N)=O)=NO1 C1(CNC(COCCOC)=O)CC(F)(F)CN1C(c1cc(C(C)C)ccc1C)=O CCC(CC)(CCNC(C1(C)CCC(OC)C1)=O)NC(c1cnsc1)=O C1(NC(=O)NC2CCOCC2C(=O)O)Cc2ccccc2C1 N1(C(C2CC(OC)C2)=O)CCCC(C2CCN(C(=O)Cc3cccnc3Cl)C2)C1 Cc1c(C(=O)N(C(C)CNC(C2OCCC2(C)C)=O)C)csc1Br CCN=c1[nH]c(C(=O)NC2CN(C(=O)CC=C(Cl)Cl)C(C)(C)C2)cs1 c1(C(C)NC(CCOC(C)=O)=O)nocc1C(=O)NCC12CCCC1C2 c1(CC)nc(C)c(CC(=O)NC2CC(=O)N(C3CN(C(=O)C(C)C)C3)C2)c(C)n1 c1(NCCCN2CC(C)(C(=O)NC(CC3CN(C)C3)=O)C2)ccc(F)cc1F c1(CC)nocc1C(N1CC(C(C)NC(c2cc(CO)[nH]n2)=O)C1)=O C1(C(=O)NCC(C)NC(=O)CC(C)c2ccncc2)(CO)CCCO1 N1(C(C(C(C)C)SCC)=O)CC(CNC(=O)Cc2nonc2C)C2(CC2)C1 c1(OC)cc(C(=O)NC2CC(C)(NC(=O)C(C)NS(C)(=O)=O)C2)cnc1O CC1CCc2c(C(=O)NC3(C)CCC(NC(=O)CC4CC=CC4)CC3)csc2C1 c1(C(=O)NC2C(C(N3CC(C(=O)OC)C(F)C3)=O)CCCC2)ccc(Br)c(Cl)c1F c1(C(N(c2nccc(C)n2)C2CCNCC2)=O)ccc2c(c1)c(C)c(C)n2C N1(C(C(F)=CCC)=O)CCC2(CCN(c3nc(CC)nc4sccc34)C2)C1 C1(NC(c2c(CC(C)(C)C)cccc2)=O)CC2CC1N(C(c1cnn[nH]1)=O)C2 C=C(Cl)CC(C(=O)NCc1nnc(O)n1C)NC(=O)C(C)COCC c1(C(=O)NC2CC(NC(CC(C)(C)OCC)=O)C(O)C2O)nc(O)ccc1C c1(C(=O)NCC(CC)NC(=O)CCSCC(=O)OC)cnn2c1NCCC2 C1(C(N2C(C)CCCC2C(N2CCNCC2)=O)=O)Cc2cccnc2C1 c1(C(C(=O)NCC2CC2C=C)N(CC=C)C2CC2)ccc(CCCC#N)cc1 N1(C(CN(C(C)=O)C)=O)CCCC12CCN(C(=O)C(C)(N(C)C)C1CC1)CC2 N1(c2cc(C(N)=O)nc(Cl)n2)CC2(CCC(NC(=O)C(F)C(F)(F)F)CC2)C1 N1(C(c2c(C)cc(-c3ccccn3)nn2)=O)CCCCNC(=O)C(F)(F)C1 C1(C)(CNC(c2cc(COC)sc2)=O)CCCN1C(c1c[nH]nc1C)=O c1(CN(C(c2csnc2C)C(=O)NCC)C)cccnc1OC Cc1nn(CC(=O)NC2COCC2NC(C2CCC(C)(C)O2)=O)c(=O)n1C C1(C(N(C(CC)CC)C)=O)CC=CCN1C(C1CC(O)C1)=O c1(OC)ccc(F)c(C(N2CCN(C(=O)Cn3cnnc3O)C(CO)C2)=O)c1N c1(C(=O)NC2C=CCN(C(C3CCN(C)C3=O)=O)C2)c[nH]c2nccc-2c1 C#CCCC(C(=O)NCC1(O)CCCC1(C)C)NC(=O)CCCCC CCCCC(CC)C(=O)NC1(CO)CCN(C(c2nc(Cl)c(Cl)s2)=O)C1 c1(C(N(CC)Cc2ccco2)=O)cc(Cn2cccn2)on1 N1(C(C(CC)OC)=O)CCN(C(=O)COc2cccc(C#N)c2)CC1C1CCC1 c1(C(N2CC3C(NC(c4cnc(Cl)s4)=O)(C3)C2)=O)cc2c(Cl)nccc2o1 N1(C(C=Cc2n(C)cnc2)=O)CC2(CCCCN(C(c3cccnn3)=O)C2)C1 c1(-n2ncc(C(=O)NC(C)CNC(C3(CO)CC3)=O)c2)ccc(Br)cc1 Cc1c(C(=O)NCCCCNC(C2(C)CCC(C)(C)CC2)=O)nn2ccccc12 Cc1ccc(F)c(-c2cn(C(C)CNC(=O)C(C)(C)CC3CCOC3)nn2)n1 C(=O)(C1=CS(=O)CCC1)NCCCNC(C(N1CCC(C)CC1)C(C)C)=O c1(NC(c2cnc(SC)nc2)c2n(C(C(=O)OC)C)nnn2)ccnc(OC)c1 Cc1cnc(C(=O)NCC(C2CC2)NC(C2CC2c2ccccc2C)=O)c(F)c1 N1(C(C2ON=C(CC)C2)=O)CC(NC(C2CC(n3cnnc3)C2)=O)CC1(C)C CC1CC2CN(C(=O)CC(C)(C)F)CC2N1C(c1cccc2ccncc12)=O C1(CNC(C2(SC)CC2)=O)CN(C(C2CC3(CCC3)C2)=O)C2CCCCC12 Cc1cc[nH]c1C(N1CCC(N(C)C(c2csc(CC(C)C)n2)=O)C1)=O C=CC1COCCN1C(C1CC(F)CN1C(c1ncccc1N)=O)=O N1(C(C(C)OC)=O)CCC(NC(=O)CCn2nc(C)nc2C)C(OC)C1 C1(C(N2CCC(NC(C3CC3(F)F)=O)C(O)C2)=O)C2CCCCCCC12 CCCCCCCCN(C(=O)C(C)(C)NC(=O)COC(CC)CC)C Cc1c(C(=O)NC2CCCC2(C)CNC(=O)CC2CCCSC2)noc1C1CC1 c1(C(N(CCCCC=C)C)=O)cc2ccc(-c3cc(C)cnc3OCC)cc2o1 C1(NC(c2cnc(C)s2)=O)CC12CCN(C(c1c(F)cncc1F)=O)C2 C(=O)(C(Cc1ccsc1)NC=O)NCC(CC)NC(=O)C(F)F C(=O)(N=c1ccn(C)[nH]1)C1(O)CCN(C(c2c(C)nc[nH]2)=O)CC1 C1(CC(=O)NCC(C)(C2CC2)NC(c2cnc(C3CC3)o2)=O)CCCOC1 c1(CC)ncncc1C(=O)NC1CC2(C1)CC2C(=O)NCc1cc(C(N)=O)co1 N#Cc1cccc(C2(C(=O)NC3CCC(NC(=O)Cn4ccc(F)n4)C3)CC2)c1 N1(C(CCC(C)NC(c2cc(=O)n(C)cn2)=O)=O)CC2CC1C(F)(F)C2 C1(C(=O)NCCn2c(C)ncc2)CC(O)CN1C(C1COC(=O)N1)=O C(=O)(C(F)(F)C(C)O)N(c1ccc(CC(=O)NC)cc1)CC.C1(C)(CO)CCCC1 c1(C(N(C(CCNC(CCC(C)CN(C)C)=O)C)C)=O)cc2n(n1)CCCO2 c1(C(=O)NCC(O)CNC(C2OCCCO2)=O)n[nH]c2c1COc1ccccc1-2 C1(CC(=O)NCc2ccncc2N2CCOCC2)CCc2ccccc2N1 C(C(=O)N1CCC(C)(CCNC(=O)CC(C)(C)C2CC2)C1)(C(C)C)NC(=O)OC c1(C(=O)NC2(C)CC(NC(C=CC)=O)C2)ccc(C(C)(F)F)nc1 c1(C(=O)NC(CNC(c2ccc([N+](=O)[O-])o2)=O)CO)ccc(O)nc1Cl C#CCC(C)(C)C(=O)N1CCCC1CNC(=O)C(c1cccc(C(F)(F)F)c1)(C)O C(C(C)(C)CC(=O)NC1C(C(=O)NCCCN(C)C(C)C)C1(C)C)OC(C)=O c1(C(=O)NCCC2OCCN(C(C(C)OCC3CC3)=O)C2)cc(N)nc(Cl)c1 c1(CN2C3C(C(=O)Nc4c(C#N)scc4)C(C3)C2)nc(Br)ccc1F C1(O)(C(=O)NC2C(C)CN(C(c3ccc(CO)cn3)=O)C2)Cc2ccccc2C1 CC(C)C(C(=O)N1CC(NC(c2ccc(CSC(F)F)o2)=O)C1)c1cnn(C)c1 C1(C(=O)NCC2CC(C)N(C(=O)CCOC3CC3)CC2)CCC2(CCC2)CC1 c1(C(CC)NC(C(CC(=O)NC)=O)=O)ccc2nccnc2n1.OC C(CCCCC(=O)NC1(CN(C)C(C2(C)CCCC2C)=O)CC1)=CC c1(NC(C(C)C)CNC(c2cc(C(C)(C)C)no2)=O)cc(=O)n2ccccc2n1 c1(SC)ccc(CC(=O)NC2CC(C)(NC(c3ccc(C(C)=O)o3)=O)C2)cc1 C(=O)(CCC(C(C)C)NC(C1C2CCC(F)C12)=O)N1CC(C#C)C(O)C1 C(=O)(C(F)C(C)CNC(=O)C(C)(C)c1ccno1)NCc1nc(C(C)C)on1 C(=O)(C1=CCCSC1)N1CCC(CCNC(C(C(C)C)SC)=O)C1 c1(C(N2CCC(O)(CCNC(C(CCC)(C)C)=O)C2)=O)cccc2occc12 c1(C(=O)OCC)cc(Br)ccc1N(C)Cc1sc(C)cc1C c1(N2CCC(C)C2CNC(=O)C(C)(C)CO)cc(Cl)nc(-c2ccc(F)cc2)n1 C1(NC(CC)=O)(CNC(c2cc(C)[nH]n2)=O)CC2CCC1C2 C(C(C)C(C)(C)C)N(C(C(CSCC)NC(c1cnsn1)=O)=O)C C1(C(=O)NC(CNC(CC(=O)NCC)=O)(C)C2CCC2)CCC2CC1C2(C)C N(C(=NCCCF)NCc1ccnc(NC2CC2)n1)C(c1ccccc1)C c1(OCC(=O)NCc2cc(C(C)=O)oc2)cccc(C(C)(C)C)c1 CC(CC(=O)NC1C2CC1N(C(c1ccc3c(c1)CC3)=O)C2)CC(C)(C)C c1(C(C(=O)NCCN(C(c2c(CC)csc2)=O)CCOC)C)cccc(Cl)c1 CC(C)(CC(F)(F)F)C(=O)NC1COCCC1NC(=O)CN1CCCOC1=O C(C)(CN=c1[nH]nco1)(CC(C)C)NC(c1cc(OC)n(C)n1)=O N1(C(C2(CCC)CC2)=O)CCCC(CNC(=O)C(C(C)(C)C)C2CCCC2)CC1 c1(C(N2CC(C=C)OCC2)C(=O)NC(C)C)cccn2ccnc12 N1(C(CSCC#C)=O)CCC(=C)CC1C(=O)NC1CC(C)OC1=O C1(C(=O)NCCC2CC(NC(c3ncn(CC)c3)=O)C2)(CC)CC=CCC1 c1(OC(=O)NCC2(COC)CCC2)ccc(C(=O)OC(C)C)cc1O C1(OC)CC(C(N2CC=CC(NC(C3CCN3C)=O)C2)=O)CC1OC N1(C(c2ccc(OCC)cc2)=O)CC2CC(C1)N2C(c1ccc(C)cc1O)=O C(=O)(C(C)(C)CN(C)C)NCC1(CNC(n2ccc(C)n2)=O)CCCC1 C1(NC(C(C=C)O)=O)CN(C(=O)CCCOc2ccc(C(C)(C)C)cc2)CC1C C1(C(=O)NC2CC(CO)N(C(C3CCCN3c3nccs3)=O)C2)C2CCCCC12 c1(C(N2CC(OC)C(NC(=O)CC3CN4CCC3CC4)C2)=O)cc(C)cc(O)c1 c1(CC(n2cc(C3COCCN3C(C3(C)CC3)=O)nn2)C)ccccc1F c1(C(N2C(C)CC(CNC(=O)C#CC3CC3)C2)=O)ncc2ccccc2c1O N1(C(C(C)C(=O)N2CCOCC2)=O)C2CCC1CN(C(C1(CF)CC1)=O)C2 N1(C(C(CNC(=O)C(C)(C)OC(C)=O)OC)=O)CCC2(CCOC2)C1 C(c1ccc(F)cc1)=CCC(=O)NCC1CCCC(NC(=O)C2=CCCOC2)C1 c1(CC2C(=O)N2)ccc(Cl)cc1Cl.N1(C(COCCSC)=O)CCOCC1CO c1(CN=[N+]=[N-])ccc2c(c1)CN(S(=O)(=O)C1CCOC(C(F)(F)F)C1)CC2 Cc1nc(C(=O)N(C)CC=CC(=O)N(CCC(C)(C)C)C)cc(O)n1 N1(C(c2cc(OC)ncc2)=O)CCN(C(=O)C=C2CCCCC2)CC1CC1CC1 c1(OC)cc(C(=O)NC(CNC(=O)C(=O)NC(C)C)C2CCC2)cnc1O c1(CCNC(CCN(C(=O)CC(=O)NC2CC2)CC#C)=O)ccccc1 Cc1cc(C(=O)NC2CCN(C(=O)CNC(c3nnc(C)s3)=O)CC2)cc(C)c1 c1(C(=O)NC(CNC(C(C(C)(C)C)SC)=O)CCOC)cc(C)ccc1[N+](=O)[O-] C1(C(C)(C)C)CCC(C(O)C(=O)NC2CN(C(=O)CSCC(=O)NC(N)=O)C2)CC1 c1(C(=O)NC2CCCN(C(C3(C)CC(C)OCC3)=O)CC2)ccc2c(c1)CCC2 N1(CC(=O)N(CCn2cc(Cn3ccnc3)nn2)CC)CCOCC1=O C1(NC(C2C(CC)C2)=O)CCCN(C(=O)C(c2ccc(Cl)cc2O)=O)CC1 CCCCC(C(=O)NCCn1cnc(C(N2CCCC(OCC)C2)=O)c1)C(C)C C1(CC(=O)N(CCC)C)CCCCN1C(c1cccc(F)c1)=O C(=O)(CCCCC#N)N1CCC(C(=O)NOC(C)(C)CO)(CC=C)C1 c1(C(N(C)CC2N(c3snc(C)n3)CCC2)=O)cc2cccc(Cl)c2o1 C(C)(CC(=O)NCCCCN(C)C(c1cn(C(F)(F)F)cn1)=O)SC C1(NC(COc2cccc(C)c2)=O)CN(C(=O)Cc2ncn(C)c2C)C(C)(C)C1 CC(C)C(F)C(=O)NC1CCC(CNC(c2ccccc2Br)=O)CC1 c1(SCC(=O)N(CCN(C(C(C)O)=O)C)C(C)C)cc(F)ccc1F c1(NCC2CCC(NC(C(c3ccc(C)cc3)=O)=O)C2)ccc(C)cc1[N+](=O)[O-] C1(NCC(CNC(c2nnccc2C)=O)OC)CC2(C1)CC2C(=O)NOCCO C1(NC(=O)Cn2nnc(=O)[nH]2)CN(C(c2cocn2)=O)CC12CCOCC2 c1(C(=O)NC2CCCC(NC(c3onc(C)c3C)=O)C2)c2c(c[nH]c1=N)CCC2 C(=O)(C(C(C)(C)C)c1cnno1)NCC1(F)CN(C(C2(C)CCCS2)=O)C1 N1(C(C=C(CC)CC)=O)CCC(N(C)C(C2CC(C(=O)O)C2)=O)CC1 CN1CCCCC1CC(N1CCC(O)(CCNC(=O)C(C)(C)c2cnc[nH]2)C1)=O C(=O)(CC1COc2ccccc21)O.c1(OC)ccc(SC)c(NCC2(C)CC2)c1 c1(C(=O)NC2C(F)CCN(C(CC#C)=O)C2)ccc2occc2c1O CC1COCC(CC(=O)N(CC(CO)(CO)NC(=O)COCc2nc[nH]n2)C)O1 N1(C(C(C)c2cccs2)=O)CSCC1C(=O)NC1CCNC1=O C#CCC(C(=O)N(C)CC1(F)CCC1)NC(=O)Cn1ccccc1=O C12(NC(CCCOCC)=O)CC1CN(C(C1COCCN1C)=O)C2 C(=O)(C(C(C)(C)C)N(C)C)N1C(CC)C(C(=O)NCC=C(C)C)CC1 N1(C(C2C(CC)C2)=O)CC2CC1CCC2NC(=O)CC1COCC(C)(C)O1 n1(CC(=O)NCC2(C(N)=O)CN(C(CNC(CCC)=O)=O)C2)ccccc1=O N1(C(C(C)CC(C)(C)C)=O)C2CCCC1CN(C(=O)C(N1CCCCCC1)C)C2 N1(C(C(OC)OC)=O)CCN(C(=O)C(c2cncn2C)O)CC1c1ccncc1 CCCC(C(=O)NC1CCN(C(=O)C(C(C)O)N(C)C)CC1)NC(N)=O C(=O)(C1=CCCCC1)N1CCCC(C(C)NC(c2nc(Cl)c(Cl)s2)=O)C1 Cc1ccc(N)c(C(=O)N(CCCNC(=O)C(C)C)Cc2cccnc2)c1F C(=O)(CCC(=O)NC1CCCCC1CNC(C1CN(C(C)C)CCO1)=O)NC C1(NCc2c(CC)cccc2)CN(C(C2CC=C(C)CC2)=O)CCC1F C(=O)(C(=O)NNc1ncc(Br)cn1)Nc1c(C(=O)OCC)ccs1 c1(CN2C3C(C(=O)NCCc4nn[nH]n4)C(C3)C2)ccc(F)c(O)c1 C(=O)(C1=CCS(=O)(=O)C1)N(C(C)CNC(=O)C(c1ccccc1C(F)(F)F)O)C C1(C(=O)NCC2C(NC(c3ccc(CC)cn3)=O)CCC2)CCC(C#N)CC1 C1(CNC(C(C)(C)OC)=O)CC2(CCOCC2)CN1C(c1cnc(C)n1C)=O C1(C(=O)OC)N(C(C(=O)Nc2ccc(F)cc2C)C2CC=CC2)CCSC1(C)C CC1CC(CC(=O)NC(C)CC(C)(C)C)CN1C(=O)CSc1cccnc1 c1(C(N2CCN(C(C3CC3F)=O)C(CC(F)F)C2)=O)cn2ncccc2n1 C(CC(=O)N1CC(CNC(=O)C(C2CC2)SC)C1)NC(=O)OC N1(C(c2c(C)[nH]c(C(C)(C)C)c2)=O)CC2CCC1CN2C(C1CC1(C)Br)=O c1(-c2onc(C)n2)ccc(N2CCOCC2)cc1.C1C(C(F)F)NC(=O)N1 c1(C(=O)NCCN(C)C(C23CC(C(C)(C)C)(C2)C3)=O)ncn(C(F)F)n1 CCC(C(O)C(C)C)NC(C1C2CC3C(C2NC(=O)CCc2ccnn2C)C13)=O c1(C(C)(CO)NC(=O)CC2CC3CCC2O3)ccccc1Cl C1(NC(C=CCCC)=O)CN(C(c2cccc(OC(F)F)n2)=O)CCC1O C(=O)(C1=CCN(C(=O)CCOC2CCC2)CC1)NC1CCCN(C)C1 c1(NCC2C(C)CCNC2=O)ccc(S(=O)(=O)N2CCc3ccccc3C2)cc1Br C1(CNC(CNC(c2c(C)occ2)=O)=O)CCCCCN1C(C1CC(C#N)C1)=O N1(C(=O)Cc2c(Cl)cccc2Cl)CC2CCCC(C1)N2C(=O)C(F)Br N1(C(Cc2cc(C)c(Cl)cc2)=O)CC(CNC(=O)C2=NNC(=O)C2)C2(CCC2)C1 c1(C(=O)NC(CCCNC(c2c(OC)cccn2)=O)C)noc2c1CCCC2 C1(C(N2CCC(SC(F)(F)F)CC2)=O)(OC)CCN(Cc2ccccc2C)CC1 N1(C(c2c(CC)noc2C)=O)CCC(C2(O)CCN(C(=O)C(O)C3CC3)C2)CC1 C1(CNC(c2ccc(CC)cc2)=O)CC(NC(c2cnc(C)[nH]2)=O)C12CCC2 C(c1cc(F)c(O)c(F)c1)=CC(=O)NCC1CCN(C(CNS(NC)(=O)=O)=O)C1 N1(C(c2c(Cl)sc(C)c2C)=O)CC2CCC1CN2C(=O)CCNC(C1CC1C)=O N1(C(C(=O)NCC2CCN(C(c3c(C(C)C)n[nH]c3)=O)C2)C)CCP(C)(=O)CC1 N1(C(c2cc(C(C)C)nn2C)=O)CC(NC(C2CC2(C)Br)=O)C2(CCOCC2)C1 N1(C(CC=C(C)C)=O)CCCOC(CCNC(=O)CN2C(=O)CNC2=O)C1 CC(C1CC1)=C(F)C(=O)N(CC(O)CN(C(=O)CCOCC1CC1)C)C N1(C(C(=O)C2CC2)=O)CC2(CCCN2C(=O)CCN2C(=O)C=CC2=O)C1 c1(C(N2CCC(CNC(=O)C=CC(=O)NC3CC3)C2)=O)ccncc1F c1(C(N2C(CCNC(C3(SC)CCC3)=O)CSCC2)=O)ccc2cnccc2c1 c1(C(N=c2[nH]ncc(C)c2)=O)ccc(-c2ccc3c(c2)C(=O)NC3)c2c1OCO2 C(C(C)NC(=O)CC1(N(C)C)CC1)N(C(=O)CC1CCC1)CC n1(CCC)nc(C)cc1C(N1CCOCC1CCNC(C1CCCO1)=O)=O CC12OCC(CNC(=O)CNc3ccc(F)c(Cl)c3)(CO1)CO2 c1(C(=O)NCC(C(C)(C)C)NC(C(C)(C)OCC)=O)ccc(Br)c(N)n1 N1(C(CN(C(c2ccccc2)C)CC)=O)C2CCC1CN(C(C1CCC1)=O)C2 C1(NC(=O)CC2CC(F)(F)C2)CCC2(CCN(C(=O)C(O)C3CC3)C2)C1 c1(C(=O)NCC2C3CN(C(c4cnn(C5CC5)c4)=O)CC23)cccc2[nH]ccc12 C1(F)(CNC(CN(C)CC)=O)CCC(NC(=O)CSc2cccc(C)c2)C1 Cc1cccc(CC(=O)NC(C)(CNC(C2C(C)C2C)=O)C(C)C)c1Cl C(c1ccc(C)cc1)=CC(=O)NCCN(C(C=COCC)=O)CC C12CN(CCO1)CCNC2=O.c1(CNC(c2cnon2)=O)cccnn1 N1(C(CC(CC)C)=O)CCC(CC(N)=O)(NC(C2CCCS(=O)(=O)N2)=O)CC1 N1(C(c2cc(COC)[nH]n2)=O)CC2CC3CC2C1C3NC(C1CCC1(C)C)=O c1(C(=O)OC)ccc(C=CC(=O)NCC2CCC(NC(C3CCC3)=O)C2)o1 Cc1ccc2cc(S(=O)(=O)N3CC(S)CC3(C)C)ccc2c1 c1(C(N2C(CCCC)CN(C(C3(F)CC3)=O)CC2)=O)cc(F)cc([N+](=O)[O-])c1 C1(C(=O)NC(C(=O)NCC2CCC(C)(C)C2)Cc2ccoc2)CCCCC(=O)N1 N1(C(c2cc(C)[nH]c2)=O)CCCC(C2(NC(=O)CC3CCC(=O)N3C)CC2)C1 CC(C)(CC(=O)NCC1(CNC(c2ccccc2Cl)=O)CCC1)C1CC1 C1(C(C)(C)NC(C2C(C)C2)=O)CCN(C(C2(c3ccccc3)CC2(F)F)=O)CC1 c1(C(=O)NC2C(NC(C=Cc3c(C)n[nH]c3)=O)COCC2)cnc2cccnn12 c1(CN(C(=O)NC2CN(C)C3(CCCC3)C2)CC)ccc2c(n1)NCCC2 c1(C(C(=O)N(CCOC)Cc2c(C)noc2C)(C)C)ccccc1C(F)(F)F Cc1ccc(C=CC(N2CC(NC(=O)C3=CCOCC3)C3CCCC23)=O)c(C)c1 C1(CCNC(c2nc(CSC(C)C(N)=O)sc2)=O)COCC1(C)C N1(C(c2c(C)c[nH]n2)=O)CCC(C)(C)CC1C(=O)NC1CCOC2(CCC2)C1 C1(NC(Cc2ccc(C)nc2)=O)CCCC12CCN(C(=O)CSCC(N)=O)CC2 c1(CC)ccc(C(=O)NCCOCCCNC(C2CC3CCC2O3)=O)cc1 C1(C(N(C(CC)CNC(c2cc(C)nn2CCO)=O)C)=O)CC12CCOCC2 C1(C(=O)NCC(C)NC(CC=CC=C)=O)CCN(c2ccc(F)cc2)C1=O Cc1ccn2ncc(C(=O)NC(C)CCNC(C3(NC(N)=O)CCCC3)=O)c2c1 C1(CC(=O)NCC2N(C(c3c[nH]c(=N)s3)=O)CCC2)(OCN)CCCCC1 C1(NC(C2(NC(c3c(C)csn3)=O)CCSC2)=O)CCCCCC1CO c1(-c2n(-c3ccc(C)c(Cl)c3)nc(-c3cnn(C)c3)n2)cc(F)cc2ccoc12 c1(C(=O)NC2CC(F)(CNC(CN(CCOC)C)=O)C2)ccc(C(C)(F)F)nc1 n1(CC)c(C(N2CCC(CCNC(c3cnn(CCOC)c3)=O)C2)=O)cnc1O Cc1ncnc(C)c1C(=O)NC1CC(F)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C1 N1(CC2C(CCC)C2)C(=O)CN(Cc2cc(Br)cnc2-n2cccn2)C1=O c1(OC)nccc(I)c1CN1C(C(=O)Nc2ccccc2SC)CC2CC12 C1(CNC(C2(CCNC(C(COC)C)=O)CCC2)=O)C2CCCCCC12 c1(C(N2C(C(=O)Nc3c(C#C)nccn3)CC(OC)C2)=O)cc2cccnc2[nH]1 Cc1c(C(N2CC3CC2CN3C(C2(CCF)CC2)=O)=O)oc2ccc(Cl)cc12 Cn1ncc2cc(C(N3CC4CC4(CNC(=O)C(C)(C)C(F)F)C3)=O)ccc12 C1(C(=O)NCC2CC(NC(C3(CC#C)CC=CCC3)=O)C2)COC(C)(C)CO1 C#Cc1ccc(C(=O)N(C2CCN(C(=O)C(C)=C3CCCC3)C2)C)c(F)c1 C1(CNC(c2cccc(OC)c2O)=O)CC2CCCC2N1C(=O)C(C)S(C)(=O)=O C=C(C)CCC(=O)N1CC(O)(C2CCCN2C(=O)CC(C)(C)SC)C1 N1(C(C2CCN(C(=O)C3CC3)CC2)=O)CCN(C(c2cnns2)=O)C(CF)C1 C1(C(=O)NCC(CNC(c2cc3ccccc3o2)=O)F)CCc2ncccc2C1 C1(NC(C(c2ccc(Cl)cc2)CC)=O)CCCC(CNC(c2cnsc2)=O)C1 C(=O)(C(C)(C)C1=CCN(C(=O)C(=O)Nc2ccc(S(C)(=O)=O)c(C)c2)CC1)OC n1(CC(=O)N(CCCNC(C(N)=O)=O)C2CC2)cc(Br)c(O)nc1=O C(CNC(C1CC2C=CC1O2)=O)(CC(F)(F)F)NC(CC(C)(F)F)=O C=CCCCCCC(=O)N1CCN(C(=O)CC(O)CN(C)C)CC1CCO C1(C(=O)NCC2(CC(F)F)CC2)CCCN(C(=O)Cc2ccco2)C1 N1(CCC(=O)NC2C(NC(C3(C)CCOC3)=O)CCC2)CCOCC1=O C1(CC(=O)NCC2C(CNC(C(C)(C)F)=O)C2)CCCCCC1 c1(C(=O)NC2C3CN(C(CCS(C)=O)=O)C2C3)cncc2ccccc12 CCC(C)C(O)C(=O)NC1CC(C)(CNC(=O)C(F)(F)C=Cc2ccccc2)C1 CC1CCCCN(C(=O)C=CC(C)(C)NC(=O)CC2(O)CCC2)C1 N1(C(COCc2c(C)cccc2)=O)CC(C)N(C(=O)Cc2csc(S)n2)CC1C CCC(CC(=O)OC)NC(=O)C(C1(O)CCC1)NC(=O)CC1CSC1 Cc1cc(F)ccc1C(=O)NCC#CCNC(C1COCC1c1ccccc1)=O CCCC(CC)CC(=O)N1CC(OC)CC1CNC(c1ncoc1C)=O c1(OC)ccc(CC(N)CC(=O)N2CC(C)(CC(N3CCCC3)=O)C2)cc1 N1(C(C(C(C)C)F)=O)CCN(C(c2cc(C3CCC3)on2)=O)CC1C1CCCC1 Cc1ccn(C)c1C(=O)NCC(C1CC1)NC(=O)C(C)CF c1(OC)nsc(OC)c1C(c1nnnn1C1CCC1)NC(c1cc(C)no1)C C12(C(N3CC(NC(c4cnn(CCF)c4)=O)C3)=O)CCN(CC1)C2 N1(C(c2nc(C3CC3)cs2)=O)CCc2c(F)ccc(Br)c2C1 C(=O)(C(C)C(=O)N1CCOCC1)N1CC(C)(NC(C2C(C)C2)=O)C1 N1(C(C(C)NS(C)(=O)=O)=O)CCCC2(NC(=O)C=Cc3cccn3C)CC2C1 C12(C(=O)NC(c3ccccc3)C(C)NC(=O)C(N)=O)CC(C1)C(C(F)(F)F)O2 N1(C(C=C(CC)C)=O)CCCC2(NC(c3cn(C)cn3)=O)CC2C1 C1(C(N2C(C(C)NC(CCSCCCC)=O)CCC2)=O)COCCN1C=O CC1CCCCC1(CNC(=O)C=Cc1ccncc1)NC(=O)CCc1cc[nH]n1 CCC(F)(F)C(C)(C)C(=O)NCCC1CC(NC(c2oc(CO)cc2C)=O)C1 N1(C(C(=Cc2cccs2)C)=O)CC2CC(NC(=O)CCc3ccncc3)CC(C2)C1 C1(C(N2CCC(F)(CNC(C(F)=C(C)C)=O)CC2)=O)Cc2ccccc2C(=O)O1 CN1C(=O)C(=O)N(CC(=O)NC2CC(CCNC(C3(C)CC3(F)F)=O)C2)C1=O c1(C(=O)NCC2(CNC(C=C(C)C3CC3)=O)CC23CCC3)cc2n(n1)CCO2 c1(C(C(=O)NCCC(C)NC(=O)C(C)(C)CF)O)ccc(F)c(Cl)c1 c1(C(=O)NCC2(O)CN(C(C3C4CCCC34)=O)C2)cncc(O)c1 c1(C(=O)NC2CN(C(CCOCC#C)=O)C2)cncc(SC)c1 C(C1=NC2(CCN(CC(F)(F)F)C2)ON1)c1cccc(COC)c1 c1(C2CN(C(=O)Nc3nc(OCC)c(C)s3)C2)ccnc2ccccc12 Cc1cc(CCC(=O)NCCNC(=O)CN2CCC2c2ccccc2)cc(C)n1 C1(NC(CCc2ncc(C)[nH]2)=O)(CO)CCN(C(=O)CS(N)(=O)=O)C1 Cc1nsc(C(N2CC=CC(NC(c3ccc(C(F)F)o3)=O)C2)=O)c1N N1(C(C2C3N(C(C(c4ccn(C)n4)C)=O)C(CC3)C2)=O)CCCCC(C)(F)C1 c1(C2C(C(N3C(Cn4cc(C(CC)O)nn4)CCC3)=O)C2)ccc(Cl)c(Cl)c1 c1(C(=O)NC2CC3CN(C(C(CC)(CC)CO)=O)C2C3)cc(=O)n2ccsc2n1 c1(C(N(CCCNC(CC=C=C)=O)Cc2cccnc2)=O)cccc(CC)c1 c1(C(=O)NC2C3CC(NC(COCCCN(C)C)=O)CC32)ccc([N+](=O)[O-])cn1 c1(C(N2CC(CCNC(C(CC(=O)OC)C)=O)OCC2)=O)ccc2ccoc2c1 Fc1cc(CNCC2CC23CCOCC3)cc(Br)c1 c1(C(N2C(CN(C(=O)CC3CC4(CC4)C3)C)CCC2)=O)ccc2cnnn2c1 C(CCC(C)(C)C)(c1nnnn1CC1CCOC1)NCc1cnn(CCC)c1C c1(OC)ccc2c(C(=O)N(C3CCN(C(=O)C(O)P(C)(C)=O)C3)C)c[nH]c2c1 Cc1nccn1CC(=O)NC1(C(=O)NCCC(C)O)CC1C c1(OC)ccc(CNC(C2(F)CCN(C(=O)C(C)C3(O)CCC3)CC2)=O)cc1Cl C(=O)(CC(C)(O)C1CC1)N(C1CCN(C(c2ncoc2C2CCCO2)=O)C1)CC C1(CC=C)(C(=O)NCCN2CCC(C)C2)CCN(C(=O)COCC(=C)C)C1 C(=O)(C#CC1(CC)COC1)NC(CC#CC)C(=O)NC1CCC(=O)NC1 n1(CC(=O)N(CC(C)NC(c2cc(=O)n(C)o2)=O)C)cnc2sccc2c1=O N1(C(C(C)C#N)=O)CCN(C(CNC(c2cscc2F)=O)C(F)(F)F)CC1 C(C(C)(C)C(=O)NC(c1nnc(C)o1)C)NC(C=C(C)C(C)C)=O CCC(C)C(C(=O)NC1CC1CNC(=O)C(C1CCCCC1)F)NS(C)(=O)=O C(=O)(C(O)CC(N)=O)NCC(C)(CO)NC(c1n(CC)nc(C(F)(F)F)c1)=O CCCC(CNC(c1cc(CCC)[nH]n1)=O)C(=O)NCC(=O)OC(C)C N1(C(Cn2nnc(C)n2)=O)CC(O)CC1CNC(c1cc(Br)n(C)c1)=O CN1CCN(C(=O)CC2(NC(c3cncc(O)c3)=O)CCC2)C(CO)C1 c1(C(=O)NCC(CN(C(c2ccc(C#C)cn2)=O)C)O)ccc2nccnc2c1 C1(C(N(CCOC)CCSC(C)=O)=O)COCC1C(N)=O.C1CC(=O)N1 c1(NC(=O)NCCC(=O)N(CC)CC)nc(Cl)c2ccnc-2[nH]1 C1(C(N(CCO)CC)=O)CC12CN(C(C1CCN(C3CCCC3)CC1)=O)C2 N1(C(C2C(CC)N(C(=O)CC(C)(C)C(F)F)CCC2)=O)CCCC(C2CC2)CC1 Cc1cc2[nH]c(CN3CCn4c(C5CCNCC5)nnc4C3)cc(=O)n2n1 C1(CC)CC(CC(=O)NC2CN(C(C3(C)CCCC3)=O)CC2C)CCO1 N1(C(C(CC#C)C2CC2)=O)CC(C(=O)NC2CC(O)C(F)C2)C(F)(F)C1 N1(C(C(CC)NC(N)=O)=O)CC(C2(NC(c3nccc(OC)c3F)=O)CC2)C1 c1(C(=O)NCC2N(C(CCSCCCC)=O)CC(C)CC2)[nH]nc2ncccc12 Cc1c(C(=O)N(CC(O)CNC(C2CC2c2cccc(O)c2)=O)C)c(Cl)nn1C Cc1cc2c(NC3CCN(C(c4cnccc4C(=O)NN)=O)CC3)ncnc2[nH]1 C1(CN(C(=O)CSCc2cccc(Cl)c2)C)CCCN(C(C2CC2[N+](=O)[O-])=O)C1 C1(NC(CCC)=O)COC2(CCCN(C(c3cc4cc(Cl)ccc4n3C)=O)C2)C1 O=C(N=c1nc(Cl)[nH]n2ccnc12)C(C1CCCCC1)c1ccccc1 Cc1ccc(N)c(C(=O)NCC2(CNC(C3(C)CC3F)=O)CC2)c1F C1(C(=O)NCC2N(C(Cc3nn(C)c(Cl)c3)=O)CC2)CCc2ccnn2C1 Cc1cn2cc(C(=O)NC(CNC(C3COC4(CCC4)C3)=O)C3CCC3)nc2s1 C12(CNC(C(C)(C)n3cnnn3)=O)CC1CN(C(=O)CCc1ccncc1)C2 C(CC1CCc2ccc3c(c21)CCO3)NC(C1CCC2(CN(C(CC)=O)C2)O1)=O c1(CC)ccccc1C1CC1C(N1CC(OCC)C(NC(=O)C(CC)OC)C1)=O c1(OC)ncc(Br)c(=NC(=O)C2CC3CC3N2Cc2occc2C)[nH]1 C1(CNC(Cn2ncc(CC)c2)=O)C(C)CCCN1C(C1CC(F)(CO)C1)=O N1(C(CC2(COC)CCOCC2)=O)CCC(COC)(NC(C2(C)CC2Br)=O)CC1 C1(CNC(Cc2n(C)ccc2)=O)C2CN(C(=O)CCNC(C3CCCO3)=O)CC12 C(CCCCC(=O)NCC12CCC(F)(CC1)C2)N(C(=O)C(O)C1CC1)C Cc1cn2c(C(=O)NCC3CCCCN(C(C4C5CCCC45)=O)CC3)cnc2s1 c1(NC(C(C)S)=O)cncc(C2=CCC(C(F)(F)F)CC2)c1 C=C=CCCC(=O)N1CCC(N(C(=O)CSC(F)(F)F)C)C1 N1(C(c2c(CC)nccc2)=O)CC(NC(c2cnoc2C(C)C)=O)CCC(O)C1 Cc1nc(O)c(C(=O)NCC2CCCCN(C(C3(CF)CC3(F)F)=O)C2)nc1C N1(C(c2c(CC)c[nH]c2)=O)CC2CC(C(=O)NC(C)CC3=CCCCC3)C(C2)C1 N1(C(c2n(C)ccc2)=O)C(CNC(=O)C=Cc2cncc(F)c2)CC2COCC12 N1(C(C2C(COC)CC2)=O)CCC2CCN(C(=O)COCC(C)(C)C)CC12 O=C(CC1CCc2ccccc21)NCC1(CNC(C2CC3CC(=O)C2C3)=O)CC1 c1(C(=O)NCC2CN(C(CC(C)C)=O)C(C)C2)cnc2c(c1)N(C)CCO2 c1(C(=O)NC2C(C(=O)NCC(CC)(C)COC)OCC2)cc(C)ccc1F C1(C(=O)NCCC2CCCCN2C(=O)C(Cl)=CCl)(OC)CCC12CCC2 Cc1cccc(OC(C)C(=O)NC(C)CN(C)C(c2cc(CO)[nH]n2)=O)c1 CC1(NC(c2csc(C(F)F)n2)=O)CCCN(C(C2CC3CC3C2)=O)C1 C(C(CC(C)C)C(=O)NCC1CC2CCC1N(C(=O)Cc1cncnc1)C2)OC Cn1ncc2c(N(C3CCCNC3)Cc3cc4ccccc4s3)ncnc12 C1(N(C(=O)CC2(CNC(c3ncnn3C)=O)CC2)C)CC2CCC1O2 CCCCC(O)C(=O)OC1CCCC1COC(=O)C(c1ccc(Cl)cc1)=O C1(C(N(c2ccccc2)C)=O)CCC(NC(c2ccn(C(F)F)n2)=O)C1 C(C(C)(C)CC(=O)NC1(CN(C)C)CCC1)NC(C1CCN(C)CC1)=O C(=O)(CS(=O)(=O)C1CC1)NC(C)CC1CN(C(=O)CCS(C)(=O)=O)C1 N1(C(Cn2c(C)ncc2)=O)C(C(N2CCC2C(N)=O)=O)CCC1C CC1CCC(CC(=O)NC2C3CC2N(C(=O)COCC(C)(C)C)C3)CC1C C1(=CC(N2CC3(N(C(c4cnc(CC)[nH]4)=O)CC3)C2)=O)CCOc2ccccc21 N1(C(c2c(NC(C3(C)CCCC3)=O)cncc2)=O)CCCC(F)(F)CC1 CCCCC(CC)CC(=O)NCc1ccccc1CNC(C1(O)CCCC1)=O C1(CNC(C(C2CC2)OCC)=O)CC2(CC2)CN1c1ccnc(C)n1 c1(CC(=O)NC(CC(=O)NCC(C)=O)Cc2cccs2)cc([N+](=O)[O-])ccc1C C1(C(=O)NCCc2ncc(C(F)(F)F)[nH]2)CC2(C1)C(C(=O)O)C21CCC1 C(=O)(C1=NOCC1)NC(C1(CNC(=O)CCCn2cccc2)CC1)C C1(NC(c2c(SCC)nccn2)=O)CCCN(C(=O)C(C#N)=CC2CC2)C1C c1(C(=O)NC2CC(NC(C34CC(CO3)C4)=O)C2)c2ccccc2cc2ccccc12 C(=O)(C(CCc1cnccn1)NCC(=O)OC1CCCN(C(=O)OC)C1)OC c1(C(C(=O)NCCN(C(=O)C(CO)N(C)C)CC)(F)F)cc(Cl)ccc1Cl c1(-c2c(CNC(C=C(C)CNC(=O)C(C)=C(C)C)=O)nco2)ccc(C)cc1 c1(C(=O)OC)c(C)noc1NC(C1CC(O)CN1C(c1cc[nH]n1)=O)=O C(=O)(CCCCN1CCOCC1)NCCCN(C(C=CC=CCC)=O)CCO C1(C(N2C3C(CNC(CC(C)n4ccnc4)=O)C(C3)C2)=O)CCOCC12CCC2 c1(CCNC(=O)NCCC2CCCSC2)cccc2[nH]ccc12 c1(CC(=O)NC2CCCN(C(CC3CCC(=O)NC3)=O)C2)cc(F)ccc1Cl N1(C(c2c(C)nc(N(C)C)s2)=O)CC(C2(NC(=O)COC(C)(C)C)CC2)C1 c1(C(=O)NC2C3CCC(C3)C2C(=O)O)cnc2c(F)cccc2c1 c1(COc2ccccc2)nc(C(C)OCC(CC)C)n(-c2ccn(C)n2)n1 C(=O)(C(C)(C)C(F)(F)CC)N1CCC(C(C)NC(CCC(CC)OC)=O)CC1 C1(NC(c2n(C)nc(C(C)(C)C)c2)=O)CCC(C)(NC(C2(C)COC2)=O)CC1 C1(c2nnnn2-c2ccc(SC)cc2)(NC(CC)(C)C(C)C)COCCOC1 C=CCC(F)(F)C(=O)NCC1CC(C)N(C(c2ccoc2C2CC2)=O)C1 Cn1c(=O)c2cc(C(=O)NC3CC3c3ccc(Br)c(F)c3)n(C)c2n(C)c1=O CCCC(C(=O)N1CCCC(Cn2cc(CN(C)CCO)nn2)C1)C(=O)O N1(C(=O)NC2CC(C)C2)CCCSCC1C(=O)O C12(OC(C3CCOC3)=O)C3C4C1C1C2C3C41C.CCC1CCC(=O)OCC(=O)O1 C(C)(CCCNC(C1(COC)CCOC1)=O)NC(C1C(=C)C1)=O c1(C(=O)NCCCCCN(C)C(c2c[nH]cc(Cl)c2=O)=O)ccn2nnnc2c1 C1(CNC(Cn2c(C)ccn2)=O)CC(C(C)C)CCN1C(=O)C(C)NC(N)=O c1(C(C(=O)NC2CCN(C(C3(C4CCC4)CC3)=O)CC2)O)ccc(F)c(Cl)c1 N1(C(C2C(C(N)=O)COC2)=O)CCOCCC1C(=O)NC12CCC(CC1)C2 C1(N(C(=O)CNC(c2ccccn2)=O)C)CCCN(C(C2CCCNC2=O)=O)C1 C1(CN(C2(CC(=O)O)CCCCC2)C)CCCN(C(=O)CC2CC2C2CC2)CC1 C1(NC(=O)C(c2cccc(F)c2)O)CC2C1CCN2C(=O)CCCn1cccc1 C1(OC)(CNC(c2ccnnc2C)=O)CCN(C(C2CC2C(F)(F)F)=O)C1 Cc1cc(C(=O)NC2(C(=O)NCC3CC4C=CC3C4)CC2)ncn1 N1(C(c2c(C)n(C)c(C3CCCC3)c2)=O)CC(NC(C2CC2C)=O)C2CCCC12 C1(C(N2CCC(C)C(NC(C3(CC4CC4)CC3)=O)C2)=O)CC2(COC(=O)N2)C1 c1(CNC(=NCC)NCC2(OC)CCCOC2)ccc(C)cc1SC c1(CCN(c2nnc(-c3ccc[nH]3)n2CC2CCCCO2)C)ccc(F)c(F)c1 c1(C(C(N2CCC(CCCC3CCCNC3)CC2)=O)=O)ccc(F)cn1 C(C(C(CC)CC)OC)NC(C1(CC)CCCOC1)=O C1(C(=O)NCCC(C)N(C(c2c(C)n(C)nc2)=O)C)CC2(CCCO2)C1 Cc1ccc(C)c(C(N2CCCC(NC(=O)C=Cc3ccccc3F)CC2)=O)n1 c1(C(N2CC3CCC(C2)N3C(c2cc3cscc3s2)=O)=O)ccc2nn[nH]c2c1 N12Cc3cc(OC)c(cc3C1)O2.N1(c2cc(CC)on2)C(=O)OC2CNCC12 N1(CC(=O)NC(C2CCOC2)CNC(c2nn[nH]c2Cl)=O)C(=O)CCC1=O C1(C(N2CCCC2CCCO)=O)NC2CC1CC2O N1(C(c2cc(C)n(C)n2)=O)CC2OCCN(S(=O)(=O)c3cn[nH]c3)C2C1 C=C(C)C(C)(C)C(=O)N1CCCC(CCC)(NC(c2ccc(C(F)(F)F)[nH]2)=O)C1 Cc1cc([N+](=O)[O-])cc(C(=O)NCCC2(O)CCCN(C(=O)C(O)CF)C2)c1C C(c1cc(F)cc(F)c1)=CC(=O)N(CCCN(C(C1CC(C)OCC1)=O)C)C c1(C(=O)NCCC(C)N(C(C(CC)F)=O)C)cc(C(F)F)ccc1F c1(C(=O)NC2C(CC=C)N(C(=O)CCCCCSCC)CC2)ccc(F)cc1F C#Cc1cc(F)c(C(N2CC3=C(C2)CN(C(=O)C(C)=C2CC2)C3)=O)cc1F c1(C(=O)NC2C(CC)CN(C(c3ns[nH]c3=O)=O)CC2)cnc2c(Cl)cccn12 C1(CC(=O)NC2CCN(C(c3cc(Br)no3)=O)C23CC3)CCC2(CCC2)O1 C1(C(=O)NCc2ccc(F)c(N)c2)(CC)Cc2ccccc2C1 c1(C(N2CCC(CNC(C(c3cn(C)nc3)O)=O)C2)=O)cnc2ccc(F)cn12 c1(OC)ccn2c(C(=O)NCC3CCN3C(=O)Cc3ccc(N)cc3)cnc2c1 C=CC(C)(C)C(=O)N(CCC(C)NC(C1CCCN1C(C1CCCC1)=O)=O)C C1(C(=O)N(CC2CSCCO2)CC2CC2)CC(NC(=O)OC(C)(C)C)C12CCC2 C1(C(N(CCNC(c2cnoc2-c2cccs2)=O)CC)=O)CCC(=O)N(CC)C1 CC1(C(=O)NC2CCC(CSc3ccccc3)C2)CC2(CC2)C1 C1(NC(CCCN(CCCC(C)C)C)=O)(CNC(=O)C(O)C(C)C)CCOCC1 CC1CN(C(C2(NC(=O)COCCCF)CC2C)=O)CCN1CCO c1(NC(=O)NC(CC)(COC)c2ccccc2)cc(OC)cc2ncccc12 N1(C(c2c(C)ccnc2)=O)CCC(O)C(NC(=O)Nc2cccc(Br)c2)C1 C1(CNC(C2CCOC2CNC(=O)C(=O)NCC(F)F)=O)CCC(CO)CC1 Cc1cc(F)c(C(=O)NC(c2ccc(Cl)cc2Cl)c2ccccc2)c(F)c1 C(C)(C(=O)NCCC(C)CO)(N(C(C(C)OCC)=O)C)C1CC1 CCC(C)(C)C(=O)N1CC2CC1C2NC(c1c(-c2ccccc2F)noc1C)=O CC1OC(C)C(C)C1C(=O)NC(C1(O)CN(C(C2CC23CCSCC3)=O)C1)C c1(OCC)ncccc1C(N1CC(NC(c2ncoc2C)=O)C(C(F)F)C1)=O C(CN=c1[nH]c(N2CCCC3(CC3)C2)nc2cc(C)ccc12)(CC(C)(C)C)OC C(=O)(CCCN(C)N=O)NC(CCC)CCCNC(c1ccc(C(C)O)cc1)=O C(C(F)(F)F)(C(F)(F)F)NC(c1cc(CC(C)C)on1)=O CC1(C)CC(CNCC2CCCN2C2CC2)CN(Cc2ccc(F)cc2F)C1 N1(C(c2cc(C)ns2)=O)CCN(C(C2CCCN(C)C2)=O)C(c2cn[nH]c2)C1 N1(C(CC2(NC(C(C)NC=O)=O)CCC2)=O)CC2COC(=O)C2C1 N(C1CCc2cc(CNC(C3CCC3)=O)ccc21)C(C(C)Cc1cnn(C)c1)=O N1(C(C(CCOC)NC(C2(C#C)CCCC2)=O)=O)CC(C)(C)CCC1C CCC(CCc1ccccc1)C(=O)NC(C)CC(C)NC(=O)CN(C)C Cc1cnc(C(N2CC(C(F)(F)F)CCC2C)C(=O)NC(C)C)cc1Br C1(CCNC(CNS(NC)(=O)=O)=O)CCCCN1C(c1cn(C2CC2)nc1C)=O c1(OC)cc(CC(=O)NCCCN(C(=O)CCc2nc(C(C)C)no2)C)on1 N1(c2ncnc3ccc(C#C)cc32)CCc2cc(Br)cc(C)c2C1 n1(CC(N2CCN(C(Cc3cc(C)cc(C)c3)=O)CC2)=O)cc([N+](=O)[O-])nc1C C1(CNC(C2CN(C(C)C)C2)=O)CCCC(NC(C2CC2c2cccnc2)=O)C1 CC(C)(C)CC(C)(C)C(=O)NCC12COC(CN=c3nc(O)c(Cl)c[nH]3)(C1)C2 c1(C(CC2CC2)NC(c2ccc(Cl)s2)CC)nnnn1C1(C)CC1 C(=O)(C1=C(C)S(=O)(=O)CC1)N(C)CC1CN(C(c2cc(OCC)c(C)cc2)=O)C1 c1(C(=O)NCC2N(C(CC3(CC(=O)OC)CC3)=O)CC2)csc(-c2nc[nH]n2)n1 N1(C(CC2CC(C)N(C(=O)CC3CC(F)C3)C2)=O)CCC2C(C(N)=O)C2C1 N1(C(C=CCC)=O)CCC(NC(C2CCC(C)C2)=O)C(F)C1 CCC(C)CC(C(=O)N(C1CN(C(C)C)C1)C)NC(c1sccc1C#N)=O C(=O)(C1=CCCN(C(c2ccc(O)nc2C)=O)C1)N(CCCC)CCOC Cc1c(C(N2CCC(CN(C)C(C3CCCSC3)=O)C2)=O)oc2c(F)cccc12 C(C1=NOC2CCCC12)NC(C1C(C)N(C(c2ns[nH]c2=O)=O)CC1)=O Cc1nccc(C(=O)N(CC(C)(C)C(=O)NC2COCC2N(C)C)C)n1 C1(C)(C(N2CC(C)(NC(COCCOCC#C)=O)C2)=O)COCCO1 N1(C(C2C(OC)C2)=O)CC(NC(c2csc(-c3ncccn3)n2)=O)CC12CCC2 C1(C(=O)Nc2nc(COC)c(C)cn2)CCOCC12CCC2.C(C)(C)O c1(C(=O)NC2CN(C(C(CC)NC(C)=O)=O)CC2C)cnn2c1CCC2 c1(CC)c(C(=O)NCC(CNC(c2cc(C3CC3)sn2)=O)OC)cnn1C c1(SCCNC(CC(c2cccs2)NC(N)=O)=O)ccc(Br)cc1 C1(C)(NC(C(CSC)OC)=O)CCN(C(=O)CNC(c2ccncc2)=O)C1 CC1CCC(CNC(=O)C=Cc2cnn(C)c2)N(C(=O)Cn2ncnn2)C1 CC12CC(C(N3CC4C(CNC(C5CC(F)C(=O)N5)=O)C4C3)=O)(C1)C(C)(C)O2 N1(C(CSC)=O)CCCC(N(C(=O)CN(C2CCCCCC2)C)CCO)C1 c1(-c2c(C)ccs2)nc(C2CSC2)nn1CCC(F)(F)F N1(C(Cn2c(C)nnn2)=O)CCC(C)(CC(=O)NC(C)CC2(O)CCC2)C1 N1(C(CCCCCNC(c2cn(CC)nc2C)=O)=O)CC2CC(OC)C(C2)C1 c1(C(N2CC(C)(C)C(NC(=O)COC3CCCC3)C2)=O)cnc2[nH]ccnc1-2 N1(C(CC=CC)=O)CCCCC1C1CCCN(C(c2cccc(=O)o2)=O)C1 N1(C(c2ccc(C)s2)=O)CCN(C(C)CNC(C2CCC(N(C)C)CC2)=O)CC1 N(C(=NCCC(=O)Nc1ccccn1)N1CCC(NCC2C(CC)C2)C1)C(C)C C1(F)(C(=O)Nc2ccc(OCC)cc2)CCN(C(=O)C(C)(C)CCF)CC1 c1(C(=O)NC2C(C)(C)C(CNC(c3cn[nH]c3)=O)C2)sc(C#N)cc1Cl N1(C(C(CCC)NC(C)=O)=O)CC2CCCC(C1)N2C(c1nn[nH]c1C(=O)O)=O C(=O)(C(C)(C)CS(N)(=O)=O)N(CCC(C)NC(=O)CC1Cc2ccccc2O1)C C1(C(N(CCN(C(C2CCN(C)C2=O)=O)CC)CC)=O)CCOC2(CCCC2)C1 C#Cc1ccc(C(=O)NCC(c2ccccc2)CNC(C2CC2CC)=O)c(C)c1 N1(C(C(CC)C)=O)CCC(O)(CCNC(=O)CCc2cn(C)nc2C)C1 C1(C(N2CCC(=CCC)C2)=O)CCCCCN1C(=O)CNC(=O)C1CC1 CC(C(=O)N(C)Cc1ccc(Br)cc1)C(F)(F)F N1(C(c2c(C)c(Cl)ccc2)=O)CC23CCCC2(C1)CN(C(C1CCC(=O)C1)=O)C3 N1(COC)CC(C(=O)NCC(C(C)(C)C)NC(=O)C=C(C)c2ccsc2)CC1=O c1(C(N2CC(C(N)=O)(OC)C2)=O)c[nH]c(=NC2CCOCC2)cn1 N1(C(C2CCCN(C)C2)=O)CCC(C(=O)NCC(O)C(C)(C)O)CC1(C)C C1(O)(c2cn(CC(CNC(C(C)CC3CC(F)(F)C3)=O)(F)F)nn2)CCOCC1 C(=O)(C#CC1CCOC1)NC1CC(Cn2cc(-c3cccc(N)n3)nn2)C1 Cc1[nH]c(=NCc2ncc(Cl)s2)sc1C(=O)CCOc1ccc(Cl)cc1 c1(C(=O)NCC(C2CC2)NC(C(CC=CC)CC)=O)cc2c(C)n[nH]c2cn1 C12(NC(C3ON=C(C(C)(C)C)C3)=O)CCOCC1CN(C(c1cscn1)=O)C2 Cc1ccc2c(C(N3CC4CC(C3)C4NC(=O)COCCN(C)C)=O)n[nH]c2c1 N1(C(CCC2(NC(C3C(C)OCC3)=O)CCC2)=O)CC2CSCC2C1 c1(C(N2CCC(NC(=O)CSC(F)F)(CF)C2)=O)c(Cl)ccc2ccncc12 c1(C(CC(=O)NCCC(C)NC(c2cnn(C)c2C2CC2)=O)C)ccc(F)cc1 c1(CC(=O)NCC(C)(CO)NC(C=C(C)C(C)C)=O)cc(C)sc1C N#Cc1cc(C(N2CC3CC(C2)C3(F)F)=O)c(O)nc1S c1(N(CCOCC=C)C)cc(C)c(S(=O)(=O)NCC2CC(C)(C)CO2)cn1 C1(C(=O)NC2CC(CNC(Cc3n(C)ccn3)=O)OCC2)CCc2c[nH]nc2C1 N1(C(C(=O)NCC2N(C)CCOC2)=O)CCC2(CCCOC2)CC1 CC1Cc2cc(CC(=O)NCC3CC(NC(=O)C(F)(F)CO)C3)ccc2O1 N1(C(c2cc(C)ncc2)=O)CC(C(=O)NCCC2(C)CCOCC2)C2(CC2)C1 Cc1ccc2c(C(=O)NC3CN(C(C4COC(=O)O4)=O)CC(C)(C)C3)c[nH]c2c1 c1(CCC)ccc(CC(=O)NCCOCCCNC(=O)CC(C)SC2CC2)cc1 N1(C(CCC#C)=O)CC(CNC(=O)CSCCc2ccccc2)OC2CCCC12 N1(C(c2cc(OCC)no2)=O)CCC(O)(C(C)NC(=O)C(CC)SC)CC1 c1(CCNC2CCC(O)C2)ccc(Br)cc1 c1(C(=O)NC2CC(N(C(c3c(C)nc(CCC)o3)=O)C)C2)cncc2[nH]ccc12 C(=O)(C(CC=CCl)c1ccccc1)NCCN(C(c1nc(Cl)cs1)=O)CC C(=O)(CCCC(C)NC(C1CCC2CC12)=O)NCC(C(C)C)(C)C N1(C(c2n(C=C)nnc2)=O)CCCCC2(CCN(C(c3nccnc3C)=O)C2)C1 Cc1cncc(CNC(C2CC(C)(NC(=O)C(C)C3(O)CCC3)C2)=O)c1 C(=O)(C(C)(C)C(N)=O)N1CC(OC)C(C(N2CCC(C)(C(=O)OC)C2)=O)C1 c1(C(N(CC(C)N(C)C(c2cnn[nH]2)=O)C)=O)c(F)ccc(F)c1Cl c1(C(=O)NC2CCCC(N(C)C(c3cc(F)n(C)n3)=O)C2)cncc2n[nH]cc12 N1(CC(=O)NC(c2ccccc2)C(C)NC(C=C(CCC)C)=O)CC2CC2C1 C1(CC)C(NC(=O)C(O)C(C)C)CCN1C(c1ccnc(OC2CCC2)c1)=O C1(CNC(CC2CC(=C)C2)=O)CC(F)(CNC(=O)C(=O)NCC(F)(F)F)C1 c1(C(N2CCCN(C(C(C)CN(C)C)=O)CC2C)=O)ccc(S(N)(=O)=O)cn1 C1(CC(=O)NCC(CC=C)NC(C2(C)CCCCO2)=O)CCC2(CCCC2)CC1 C(=O)(C(C)(C)CCSC)NCCn1cc(CNC(C=Cc2ncc(C)[nH]2)=O)nn1 C(C)(CCCCNC(=O)Cn1nnc(C2CC2)n1)NC(c1n(C(C)C)ccn1)=O c1(CN2CC3C(N)(CC3C(F)(F)F)C2)c(F)cc(O)cc1Cl C1(CC)(NC(=O)C(C)c2cccs2)CCN(C(C2C=CCC2)=O)CC1 C1(NC(CC(C)OC)=O)CC2(C1)CN(C(=O)CCNC(C1CCCO1)=O)C2 CC1CCN(C(c2ccccc2C2(CON)CCC2)=O)CC1c1ccc(O)cc1 Cc1c(S(=O)(=O)N2CCC(S(=O)(=O)C(C)C)CC2)sc2cccc(Cl)c12 Cc1ncnc(C)c1CC(=O)NCC#CCNC(c1ccc(N)c(Br)n1)=O c1(NC)cc(C)c(C(=O)NC(CNC(c2c(SCC)nccn2)=O)C)cn1 C1(N(C)C)CN(C(=O)Cc2cccc(Cl)c2)CC1CNC(C1CCC(O)CC1)=O C1(C(N(C(C)C(=O)NCC(F)(CC)CC)CCC)=O)CC2CC1CC2O N1(C(C(C)NS(CCCC)(=O)=O)=O)CCN(C(=O)CC2(C)CCC2)CC(C)(F)C1 N1(C(C2C(C)(C)COCC2)=O)CC(CNC(=O)C#CC2CCC2)OC2(CCC2)C1 N1(C(C2(CC=C)CCC2)=O)CCC(CO)C(NC(c2snc(C)c2N)=O)C1 C(C1(O)CCc2ccccc21)NC(CC(C)C)c1nnnn1CC1CCOCC1 c1(C(=O)Nc2cccc(-c3c(C)nn(C)c3)n2)cc2cc(F)ccc2[nH]1 c1(C(=O)NCC(CC)NC(c2coc(Cl)c2)=O)sc(N(C)C)nc1C c1(C(N2CC(OCCNC(c3cc(OC)no3)=O)C2)=O)cc(Cl)cc(Cl)c1F C1(CN(C(C2N(CC)CC2)=O)C)COCCN1C(c1nc(C)sc1C)=O C1(NC(C(=O)N(C)C)=O)C(CNC(c2ncc3[nH]ncc3n2)=O)CCC12CCC2 N1(c2nnc(CC)s2)CCN(C(c2cn(CC3CCOC3)nn2)=O)CC(O)C1 c1(OCC)nc(C)cc(=NC2CN(C(C3CCCNS3(=O)=O)=O)CC23CCC3)[nH]1 N(C(=NCCCF)N1CCC(C2CCC2)C1)Cc1scc(C)n1 c1(C(=O)NCCN(CCC)Cc2ccccn2)ccc(C(C)(C)OCC)cc1 CC1CCN(C(=O)CC(C)(C)O)CC1CC(=O)NCc1nncs1 c1(C(N2CCN(C(c3ccc(CC)s3)=O)CC2CC)=O)cc2ccccc2cn1 C1(C)(C(=O)NC(CC(C)C)CNC(c2cnn(C)c2)=O)CCS(=O)(=O)CC1 Cc1cc2ccc(C(=O)NC3CN(C(c4cc(Cl)c5n[nH]cc5c4)=O)C3)cc2o1 N1(C(=O)OC(C)(C)C)CCC2(CCN(Cc3csc(-c4ccco4)n3)C2)C1 C=CCCC(C)(C)C(=O)NCCC1CCCCN1C(=O)C(C)OC C(c1c(Cl)nc2ccc(Br)cn12)=Cc1c(C)ccc(C)c1 Cc1cccn2cc(CC(=O)OCC3(C)CC3Br)nc12 O=C(C#CC1CCCCO1)OCc1noc(-c2ccc(F)cc2F)n1 C(=O)(C(CNC(C1CCCCNC1=O)=O)CCC)NCCC(=O)NCC#C N1(CCCNC(CN2CC(C)(C)C2)=O)CCN(C(c2sccc2F)=O)CC1 CC1CCCC1(C(=O)NCCOC(=N)O)NC(c1cc[nH]c1C1CC1)=O n1(CCC)ncc(C(=O)NCCC2(O)CN(C(c3cccc[n+]3[O-])=O)C2)c1Cl Cc1nccnc1-n1cc(CC2CCCN(C(=O)C(C)Cc3ccoc3)C2)nn1 c1(C(N2CCC(C3N(C(C(CC)F)=O)CCC3)C2)=O)ccnc(C2CC2)n1 CCC(C)C(O)CC(=O)NC(C)(CNC(=O)CSC(C)(C)C)Cn1cccn1 N1(C(C2(C#N)C(C)C2)=O)CC(C2(NC(=O)C=CCF)CC2)C1 C=C1CC2(C1)CC(C(=O)NC1CN(C(c3ccc(Cl)nc3OC)=O)CCC1C)C2 c1(-c2cn(CC(=O)NCc3c(C)nc(C)o3)nn2)c[nH]c2nccc-2c1 C1(O)(CNC(c2cnc(O)o2)=O)CCCN(C(=O)C2=CCCS2)CC1 c1(CC)nc2c(C(N3CCCC3(C)CNC(=O)CS(C)(=O)=O)=O)ccnc2[nH]1 C(C(=O)NCc1nc(C(=O)NCC2(C)CSC(C)=N2)c(C)o1)(C(C)C)SCC CCC(O)C(F)(F)C(=O)NCCCN(CCO)C(c1cc(C(=O)OC)ccn1)=O c1(CCC(=O)NC(CNC(c2c(C)ncs2)=O)C2CCC2)c(C)n[nH]c1C N1(C(CCCOC)=O)CCCC(C2CN(C(=O)CC3CSC3)C2)C1 N#Cc1cccc(CCC(=O)Nc2nc(CC(=O)NCCC#N)cs2)n1 C1(N(C(CCN(C(c2cscn2)=O)CC)=O)C)CCCCCCC1 CC1(CNC(=O)CC(CC#N)c2ccccc2)CC(F)(F)CN1C(=O)C=CCO CC1(C)OCC(n2cc(C(N3CCC(OC4(O)CCOC4)C3)=O)nn2)C1O c1(C(=O)NCC2CCN(C(CCCCSC)=O)CC2)cccc(C(C)C)c1O C1(C(N2CCC(CC)OCC2)=O)COC2(C1)CN(C(c1coc(C)n1)=O)C2 C1(C(=O)OC)CCOC1C(=O)NC1(CNC(C2(N(C)C)CC2)=O)CCOC1 C1(CNC(C2(CC(C)C)CC2)=O)C2CC1N(C(c1cncn1C(F)(F)F)=O)C2 c1(OC)ccc(CN2CC3C(C2)N3C(C2CCC(=O)NC2)=O)cc1C(C)C C1(=O)CC(C)(C)CC(=O)NC(C)(CC(C)C)CN1.C(=O)(C(C)SC)OC.C(=O)NCC N1(C(c2c(C)[nH]cc2)=O)CCC(C)C(NC(=O)C=Cc2ccc(Br)o2)C1 c1(C(=O)NC2C(NC(=O)Cc3ccnc(Br)c3)CC2)n[nH]c2c1CCCC2 c1(OCCC)ccccc1.C1(=O)C(C)N(C)C(=O)NC2(CC2)C(=O)NCC(C)N1 C#Cc1cc(NC(C2(C)CCCN(C(=O)Cn3ccnn3)C2)=O)cc(F)c1 CC(C(=O)NCC(O)CNC(C1OCCCC1(C)C)=O)S(=O)(=O)C1CCOCC1 c1(C(N2C(COC)CN(C(=O)C(C)(F)C(=O)OC)CC2)=O)ncn2c1CCCC2 C(=O)(C1=CS(=O)(=O)CCC1)NCCCCC(C)NC(=O)C(S(C)(=O)=O)C1CC1 C(=O)(CC(C)(C)COC)NCC1C(NC(C(C=C)c2ccccc2)=O)CC1 c1(CC)ccc(C(N2CC(C)C2C(=O)NC(C)Cc2cn[nH]c2)=O)cn1 Cn1nnc2ccc(C(=O)NC3CC(C)(NC(=O)C=Cc4cccs4)C3)nc12 CC(C)CCC(O)C(=O)N(C)CCOCCCNC(c1ccc[n+]([O-])c1)=O c1(C(=O)NCC2N(C(C(C)OCOC)=O)CC(F)C2)cc2cccnc2cc1F C1(C(=O)NC(CC(=O)NC)C)(CF)CCN(C(C2CCCN2C)=O)C1 Cc1cc(F)c(C(=O)NC(C)CC(C)NC(=O)CCC(C)(C)F)c(F)c1 C(=O)(C(C)CN(C(=O)CCCN(C)C(C1CCCN1C)=O)C)OC CCCCC(COC)NC(=O)CCN(C(c1ccn(C)c1)=O)C1CC1 c1(C(=O)NCC23OC(C)C(NC(=O)C4CC4)(C2)C3)cc(Br)c(F)cc1N c1(OC)cc(F)cc(C(=O)NCC2CCN(C(c3ccns3)=O)CC2C)c1N C12CC1C1CCCN(C1)C(=O)C1C(NCC)C1CC(C)C(=O)N2.C=CCCOC Cc1ccn(CC(=O)NC2CN(C(c3cccnc3)=O)C2)c(=O)c1 N1(C(CCN(C(=O)C(C(C)C)SC)CC)=O)CCOC2COCC12 C1(NC(C(C)c2ccco2)=O)CCCCN(C(=O)CN2CCC(F)CC2)C1 CCCCCC=CCC(=O)N(CC(=O)NC(C1CCOCC1)C)CC c1(C(=O)OC)cc(F)cc(S(=O)(=O)NC2CCc3cc(F)ccc32)c1 CCCC(C(O)C(=O)N(CCCO)C1CC1)NC(c1cc(C)nnc1C)=O Cc1nocc1C(=O)NCC(F)CNC(C1C=CCCC1)=O N1(C(c2ccc(Cl)nc2)=O)CC2CCN(Cc3ccn(CCF)n3)C2C1 CC1(C)CN(C(c2cc(NC(C3CC4CC4C3)=O)ccc2N)=O)CC1NC(N)=O c1(C(=O)NC(CNC(=O)C2=CCCS2)C2CC2)nccc2cccnc12 C1(NC(c2c(CCCC)ocn2)=O)COC2(C1)CN(C(=O)C(C)OC(C)(C)C)C2 N1(C(C2(CCC)CC2)=O)CC2(C)CN(C(=O)CCCC(C)O)CC2(C)C1 c1(C(N2CCCC(C(C)(O)CNC(=O)Cn3ccnn3)C2)=O)ccc(O)c(Cl)n1 c1(C(=O)Nc2cncc(F)c2)nc2n(c1Cl)CCN(C(c1ccno1)=O)C2 n1(C(CC)C)ccc(=NC(=O)C2C(C3CC3)CCN2C(c2cccnc2O)=O)[nH]1 c1(C(=O)NCCC2(O)CN(C(c3cnccn3)=O)C2)cc(Cl)c(F)cc1Cl C1(C(=O)NC2C(C)CN(C(c3ccc(F)c(Cl)n3)=O)C2)CCC2C(C1)C2(F)F CCC(CC(=O)NCC1CC1NC(c1cn(-c2ccccc2)nc1C)=O)C(F)F C(=O)(C(CC(F)F)SC)N1CC(N(C(CNC(c2ccc(OC)cc2)=O)=O)C)C1 C1(CC)CN(C(c2cnc(F)c(C)c2)=O)CCN1C(=O)CCc1ccccc1F c1(OCCC(=O)NC2CCC2NC(c2cc(C(F)F)no2)=O)ccc(F)cc1 N1(C(CN(S(CC)(=O)=O)C)=O)CCC(C2CC2)(CNC(=O)C(C)(C)CF)C1 C(CSC)(C(=O)NCCC1(NC(c2ccnn2C2CC2(F)F)=O)CC1)OC C(=O)(C(CO)C(F)(F)F)NC(C)CNC(c1ccn(C(C)(C)C)c1)=O c1(C(N2CCN(C(CNC=O)=O)CC23CC3)=O)c(F)ccc2cnn(C)c12 c1(C(N2CC(O)(CCNC(c3cc(Cl)n[nH]3)=O)C2)=O)c[nH]c2nccc(Cl)c12 C(c1c(C)nn(C)c1Cl)=CC(=O)N(CC(CC)NC(c1cc2sccc2s1)=O)C c1(OCC)ccc2c(c1)CC(C(=O)Nc1ccc(C=CC(F)(F)F)cc1)CO2 N1(C(=O)NCC=C)CCCC(N=c2[nH]nc(CCC)s2)C1 C(=O)(C1CCCc2nc[nH]c21)NCC(CN(C(C1C=CCCC1)=O)CC)(C)C c1(NC)ccc(C(=O)NCCN(CC(C)O)C(=O)COCc2nccn2C)nc1 C=C1CCN(C(=O)CC(CC)CC)C(C(=O)NCc2ccnn2CC)C1 C(=O)(CC(C)C(F)(F)F)NCC(CC=C)NC(=O)C(c1ccc(Cl)cn1)(F)F C1(CC#C)(C(=O)OC)CCN(C(c2csc(Cl)c2)C(=O)NCCCF)CC1 C1(C(C(=O)NCC(CCC)NC(=O)CCOCCOC)O)CCCCCC1 C12(C(N(C)CCOCCNC(c3cc(C4(C)CC4)n[nH]3)=O)=O)CCC(CC1)OC2 S(=O)(=O)(c1ccc(C#N)cc1)NCC(=O)NC(C(C(C)C)Nc1ccccc1)C N1(C(C2C3CCC2CC3)=O)CCCC(C2CCCN(C(c3cnc(O)o3)=O)C2)C1 C(C(C)(C)C(=O)NC1CN(C(=O)C(c2ccc(C)cc2)F)CC1SC)OCC c1(C(C(F)(F)F)NCC2C(C(OC)OC)C2)ccc(C#N)cc1 Cc1cc(C(=O)NCC2CCC2NC(c2ccc(C3CC3)nc2O)=O)cnc1O c1(OCC)cc(Br)nc(NC(c2ccc(NC(C3CCCCO3)=O)cc2)=O)n1 c1(C(=O)NC2(CNC(C(C)NC(N)=O)=O)CC2)cc2n(n1)CCO2 c1(OC)ccccc1C1CC(O)CN1Cc1cn(C)nc1C1CC1 C1(NC(=O)C(O)CC2CCCCC2)CC2CN(C(=O)Cc3ccccc3)CC2C1 N1(C(c2[nH]cc(C)c2)=O)CC(NC(C2CN(C(C)C)C2)=O)CC(C)(C)C1 c1(C(N(C)CC2(NC(=O)Cn3cnnc3O)CC2)=O)ccc(-n2ccnc2)cc1 C(=O)(C(C)(C)C(C)(C)CO)NCc1c(C(=O)NCCOCC(=O)OC)nco1 c1(C(N2C(CNC(=O)C(F)(F)C3CC3)CC3CCCC23)=O)cccc2oncc12 C1(NC(C2CC=CC2)=O)COCCC1C(N1CCC(CC(F)F)C1)=O C1(C#N)(C(N(CCCNC(=O)CC2(C)CC2)CC)=O)CCCO1 CCC(O)CC(=O)N1CCOCC1CN(C(=O)C(c1cnccn1)C)C N1(C(CCCCC#C)=O)CCCC2(C1)C(NC(=O)CC1CC=CCC1)CCN2C C=CC1(C(N2CC(CC(F)C(=O)NCCOC(=N)O)C2)=O)CCCCC1 C12(C(=O)NCC3N(C(=O)CC4CCCC4)CC(O)C3)CC(CO)(C1)OC21COC1 C1(CNC(C(C(C)C)NC(N)=O)=O)CN(C(=O)CCc2nc[nH]n2)CCN1C N1(C(COC(=O)CO)=O)CC(O)CC1CNC(C1(F)CCCCC1)=O c1(C(C2CC2NC(=O)N)N(C)C)ccc(OCC(=O)OC(C)(C)C)cn1.C(N)(=O)N N1(C(C2C(C)CCO2)=O)CCN(C(c2ccc(O)c(Cl)n2)=O)C2(CC2)C1 C1(CC)CN(C)C(=O)CN1C(=O)COC1CC(NC(=O)CCc2nccn2C)C1 Cc1nc(N2CCC(NC(c3cnn(CC(F)(F)F)c3)=O)C2(C)C)c(F)c(C)n1 c1(C(=O)NCC2(O)CN(C(C3C(F)(F)C34CCC4)=O)C2)ccc2c(c1)NCCC2 CC1OC(C)(C)N(C(=O)OC(C)(C)C)C1CNC(C1CS(=O)(=O)C1)=O c1(C(=O)NCC2(CNC(c3cc(C(=O)OC)no3)=O)CC2)cc2c(ncn2C)[nH]1 C(=O)(CCS(N)(=O)=O)N1C(CC)C(C(=O)N(C(C)C)Cc2ccco2)CC1 c1(NC(C2CC(=O)NC2=O)C)ccccc1C1CCOC1 N1(C(CNc2c(C)cccc2C)=O)CC2(CCCC2NC(=O)Cn2ccnn2)C1 N1(C(C2CCN(C)C2=O)=O)CCOCC(F)(CNC(=O)CSC(F)(F)F)C1 C1(C#N)(C(=O)NCCC2CCN(C(COCC(C)(C)C)=O)CC2)CC12CCC2 N1(C(C(=O)NCCCC(C)NC(=O)C=Cc2cccnc2)C)C(C)CCC1C c1(NC(C)(CNC(=O)COCC2CCC2)c2nn[nH]n2)cncc(C2CC2)c1 c1(NC(C2(CNC(CC)=O)CCCC2)=O)cnn(C(C)C)c1C c1(NC(C2(COC)CCCOC2)=O)ccccc1S(=O)(=O)C(F)(F)F C(C1=C(C)CCC1)NC(c1nn(C)cc1C)c1n(CCCC)nnn1 C1(F)(C(=O)NCC(CNC(C2(CC#N)COC2)=O)O)CCOC1 c1(N2CC(NC(C(C)(F)F)=O)C(O)C2)ncnc2c1CCCC2 C(C(C)(C)C(=O)N(CCC(=O)NCCSCCCO)OC)OCC CCCCN(C(=O)CC1CCN1C(C1(CSC)CC1)=O)C C1(CNC(c2ccn(CC)n2)=O)(COC)CCN(C(=O)C2=CCCS2)C1 N1(C(C(C=C)(F)F)=O)CCC(C2(NC(=O)CCc3cncc(F)c3)CCC2)CC1 CC1(OCC(=O)NCC2CC(NC(=O)CCc3nc[nH]n3)C2)CCCC1 Cc1cc(Cl)cc(C(N2CC(C)(NC(=O)CCNC(C3CCCO3)=O)C2)=O)c1O CC(CCC(=O)NCC1(O)CN(C(c2ccccc2C(F)F)=O)C1)S(C)(=O)=O c1(CC)ncncc1C(=O)NC1(C)CCN(C(=O)C(F)n2cccn2)C1 c1(OC)cc(F)c(Br)cc1NC(=O)CC1CCN(c2ccncn2)C1 c1(CC(=O)NCC(C(=O)NCC2CCN(C)C(C)C2)OC)ccc2c(c1)CC2 c1(-c2cn(C(C(=O)NC(c3ncc(C)s3)C)C)nn2)cnn(C)c1C c1(CC)cc(C(=O)NC2CC(C)(OCC)C2)c2c(c1)CCO2 N1(C(COCC(C)C)=O)CC(CNC(=O)C(c2ccc(F)cc2)=O)C2(CC2)C1 Cc1ccc(O)nc1CNC(C1CNC(=O)CN1C(=O)CN1CCC(C)CC1)=O C1(C(N2CC3C(C(=O)OC)(C3)C2)=O)CCC2(CC2)N1C(=O)C(C)(C)n1cnnn1 c1(OCC)ccc(C(c2nnnn2C)NCc2sccc2OC)nc1 c1(CC)ccc(C(=O)NC(C(=O)NCC2(CO)CCC2)C2(C)CC2)o1 c1(NC(COC)(C)CO)cccc(CC(=O)OC(C)(C)C)c1 c1(C(N(C(C)CNC(C2CCc3cncn3C2)=O)CC)=O)c(Cl)ccc(C)c1N c1(CC(=O)N(C2CCCC2)CCOC)ncn2c1COCC2.C1C(=O)NCC1 C1(CNC(C2(C=C)CCC2)=O)CN(C(=O)C(C)Cc2ccco2)CC1C Cc1cc(Cl)ccc1OCC(=O)N(C(C)CCNC(c1ccc(N)c(Cl)c1)=O)C c1(C(C(=O)NCC(C)C)N(C(c2ccccc2)CF)C)ccc(OCC#N)cc1 N(C(=NCC1CCCCO1)NCC(C)(C)C(=O)NC)C1CCN(CC)C1 c1(NC(C)=O)cccc(NC(C2CC(C)N2C(=O)C#CC2CC2)=O)c1C C(C1CN(C(c2c[nH]c(=N)o2)=O)CC1C(N1CCC(C)(C(C)C)CC1)=O)=CC N1(C(C2CN(C(N)=O)C2)=O)CCN(C(C2(O)CCOCC2)=O)CC1CC(F)(F)F CCCCC(CNC(C1CCN1C(=O)CC1=CCOCC1)=O)CCC C(=O)(CC(C)P(C)(C)=O)NCCN(CCOC)C(C1CC(C)OC(C)C1)=O C1(NC(C(C2CC2)OC)=O)(CNC(C2(CCF)CCC2)=O)CCCCC1 c1(C(=O)NCC(CC=C)NC(=O)C(C)OCCC(C)C)cc(CC)cc(F)c1 c1(C(=O)NCC2C(NC(C(CCC#C)O)=O)COC2)cnc2cc(C)ccn12 C1(NCC(=O)NCC(S(C)(=O)=O)c2ccccc2)CCc2nnnn2C1 N1(C(c2cc(CC)[nH]n2)=O)CCCC(C)C1CNC(=O)C=Cc1ccc(C)nc1 C(=O)(CCCCNC(=O)C(F)n1ccnc1)N(CC(C)O)CCO C1(NC(c2cc(SC)oc2)=O)CC2CCC(C1)N2c1ncnc2[nH]ccc12 CC1CN(C(=O)CSc2cccc[n+]2[O-])CC1CCNC(=O)CCn1cncn1 c1(CC(=O)NCCn2cc(CN(C(C)C)C(C)C)nn2)c(F)cccc1Cl c1(C(=O)NC(CCC)CCCNC(c2ccoc2C)=O)ccc([N+](=O)[O-])cc1F CC(C#N)CCC(=O)NCC(O)CN(C)C(c1ccnc(-n2cccn2)c1)=O C1(C(=O)NCC#C)COCCN1C(=O)C(C(C)C)OCC C12(C(=O)NCc3cc(CC)on3)CCCC1CCN2C(c1cnn(CCO)c1)=O C1(NC(=O)CC2(N3CCCC3)CC2)CN(C(=O)CC2C=CCCC2)CC12CCC2 C1(C(=O)NCc2c(C)nn(C)c2)CS(=O)(=O)CC12CC2 C(=O)(CC(C(C)CC)NC(C1(OC)CCSC1)=O)NC(C=C)C1CCC1 C#CC(CC(C)(C)C)NC(C1(F)CCN(C(c2cc(C)n(C)n2)=O)C1)=O c1(C(N(CC(O)CNC(c2cnc(N(C)C)c(Cl)c2)=O)C)=O)cccc([N+](=O)[O-])c1 C1(C(=O)O)C2CC2CN1C(=O)C(F)(F)C1(O)CCC1 c1(CC)oc(C)cc1C(=O)NC(C)(C)CCNC(=O)Cc1sccc1C N1(C(Cc2c(OC)nccc2)=O)CCC2CN(C(C3CC(SC)C3)=O)CC12 C1(C(N2CCC(OCC)C2)=O)C2CCN(C(C3OCCC3(C)C)=O)CC12 C12(NC(c3c(CNC(C(CCC)OCC)=O)ocn3)=O)CCCN(CCC1)C2 c1(C(C)C)cccc(F)c1C(=O)NCC1CC(NC(c2cnc(C3CC3)s2)=O)C1 CC1CCCC(C(=O)NC2CCC(N(C)C(c3nccnc3N)=O)CC2)CC1 Cc1oc(Br)cc1C(N1CC=CC1CN(C(=O)COC1CCOCC1)C1CC1)=O N1(C(c2cccc(OC)c2)C(=O)NCC=C)CCC2C(C1)C2(F)F C(CCCCCC(=O)N1CC(O)C(O)C1)NC(C(C)(C)c1ccno1)=O c1(OC)ncc(C(N2CCC(C)(N3CCOCC3)C2)C(=O)NC2CCOC2)cn1 N1(C(C2C(CC)C2)=O)CCCC1C1CCN(C(=O)CCc2cnn[nH]2)C1 c1(C(c2n(CC=C)nnn2)NCC2CC=CC2)cnn2cc(Br)cnc12 N1(C(c2c(C)nc(CCC)o2)=O)CC(NC(c2sc(SC)cc2C)=O)CCC1C C#CCC(C(=O)N1CC=CC(NC(C2(c3cccs3)CCCC2)=O)C1)C1CC1 c1(C(=O)NC2(C)CN(C(c3cnc(C(C)OCC)s3)=O)C2)cn2c(n1)CCCC2 N1(C(COCC#C)=O)CCCC(C2CN(C(c3ccc(O)cc3F)=O)C2)C1 c1(CNC2C3CN(C(C4=C(C)OCC4)=O)CC2CC3)n[nH]c2cc(Br)cc(F)c12 CN1N=C(CC(=O)NC2(C(=O)NCCC3CCC(C)(C)O3)CCN(C)C2)CC1=O C1(CNC(C2CCCC(C)(C)C2)=O)N(C(c2csnc2Cl)=O)CCCC1(C)C C(=O)(C(O)C1=CCCCC1)N1C(N(C(C)=O)CC)CC1C.N12CCCC1C2 CC1CN(C(=O)COc2ccon2)CC(C)N(C(c2cccc(=S)n2O)=O)C1 c1(C(=O)NC2CN(C(C(CC#C)O)=O)CC23CCC3)ccc(=O)n2c1COCC2 CC(C)C(C(=O)N(C1CCN(C(c2cn(C)cn2)=O)C1)CCO)c1cnn(C)c1 Cc1ccccc1-c1cccc(N(CCCCCCC2OCCO2)C(C)C)c1 C(=O)(C(C)C(C)COC)NCCN(CCC)C(c1cncc(N)n1)=O C1(C(=O)NCc2cncc(C(=O)NC(C)CCC3CC3)c2)CCCCC1(C)C C1(CNC(C(COC)C)=O)CCC2(CCC2)CN1C(=O)C=C1CN2CCC1CC2 C=CCC(C(=O)N1CCC(CCNC(c2c(N)cc(Cl)nc2Cl)=O)C1)C(C)C C1(CNC(CC2(NC(c3c(C)snc3)=O)CC2)=O)CCC(=O)NC1C C1(C(=O)OC)CCC(Cc2cccc(-c3ccccc3)n2)CN1CC.C(C)(C)(C)OC=O CC(C)CC(C(=O)OC1CCCCC1)N(C)CCC1NC(=O)NC1=O N1(C(Cn2c(C)nc(C)n2)=O)CC2CC(NC(C3(S(C)(=O)=O)CC3)=O)CC2C1 N1(C(CSCC)=O)CC(CCNC(c2cnc(SC)nc2)=O)C(C)C1 C1(C(=O)NC2(C)CC(F)(F)C2)CCOCCN1C(C1CCC(F)(F)C1)=O C(C)(C(=O)NCC1CCCC1N(C)C)(N(C(C(C)=CC(C)(C)C)=O)C)C1CC1 C1(C(N(C)CC2(O)CCCN(C(=O)CNC=O)C2)=O)CCC2(CCCC2)C1 N1(C(C2CC(C)(C)C2)=O)Cc2nccn2CC(NC(=O)CN2CCC(C)(O)C2)C1 N1(C(C2CC(C#C)(O)C2)=O)CC2CCC1CN2C(=O)Cc1cc(C)cs1 Cc1oc(S(=O)(=O)Nc2cc(Cl)nc(Cl)c2)cc1S(C)(=O)=O N1(C(c2ccc(NC)cn2)=O)CCN(C(c2cc(C)cc(C)c2)=O)C(C2CC2)C1 c1(C(=O)NC2C(CNC(CCP(C)(C)=O)=O)CC2)cc(F)c(F)cc1Br c1(C(N(CCN(C(c2cccc(F)c2)=O)CC)CC)=O)cc2sc(C)nc2[nH]1 c1(C(=O)NC2C(C)CN(C(=O)CCc3nncn3C)CC2)cnn2ccncc12 c1(CC)ccc(C(F)F)c(F)c1.c12ccc(s1)CN(C)C2C(=O)NC1CCOC1 N1(C(C(c2cncn2C)N(C)C)=O)CCC(C)(C)C(NC(=O)Cn2ccnn2)C1 c1(C(=O)NCC(=O)NCC2CCCN(C(c3cscn3)=O)C2)[nH]cc2c1CCC2 N1(C(c2cc(CNC(=O)CCc3csnn3)sc2)=O)CCOC2(CC2)C1 C1(NC(CCCCSC)=O)CC1C1CCCN(C(c2nnn(C)c2N)=O)C1 N1(CC=C)CCCN(C(=O)C(CNC(c2ccncc2)=O)CC2CCCC2)CC1 C#Cc1cc(C(=O)NCC2CCN(C(C3CC3F)=O)CC2(F)F)cc(Br)c1 CC(C)(C)C(C(=O)NC12CCC1CN(C(=O)CC1COC3CC1C3)C2)NC(N)=O c1(C(N2CCCC(N(C(=O)CCc3cnn(C)n3)C)C2)=O)cc2cccnc2o1 C1(C(=O)NC(C2CCCC2)C#C)CCCCC1(C)NC(=O)C(C)NC=O C1(CCNC(C(C=C)O)=O)CN(C(=O)CCc2c[nH]c(C)c2C(C)=O)CCO1 c1(N(C(C(C)NC2C3COCC23)=O)S(C)(=O)=O)cc(-c2ccccc2)nn1C c1(OC)cc(NC(=O)C(C2CCN(C(=O)CCC(C)SC)CC2)C)cc(OC)n1 N1(C(C2C(C)C(=O)C2)=O)CCOCC1CNC(c1ccn(C(F)F)n1)=O CC1(C)CCN(C(=O)CC2CCCC23CC3)CC1CNC(C1(F)CC1)=O CC(C(N)C(=O)NCC1(C#N)CCNC1)C1CC1 C1(C(C)C)CN(C(=O)CSCC(F)F)CCC1NC(=O)C=Cc1cccnc1 N1(CC(=O)NCCC(C)(C)NC(=O)C=CC(=O)N(C)C)CCCCC1=O N1(CCc2cccc(OCC)c2)CCC(=O)N(Cc2cc(Cl)ccc2C)C1=O N#Cc1ccc(C(=O)NNC(=O)C2(C#N)CCCC2)nc1Cl Cc1nsc(C(N2CCCC(CNC(c3cc(Br)nn3C)=O)C2)=O)c1N c1(C(N2CC(CC)SCC2)=O)ccc(F)c(-c2cn(-c3ccccn3)nn2)c1 Cc1c(C(N2CC3CC(O)C2C3NC(=O)C2=CCOC2)=O)oc2ccc(F)cc12 C1(CNC(COC)=O)CC2(CCN(C(c3c[nH]nc3OC)=O)CC2)CO1 N1(C(CC2(CC=C)CCCC2)=O)CCCC(CCNC(C2CNC(=O)N2)=O)CC1 c1(CC(=O)NCC(CNC(CC2(C(=C)F)CCC2)=O)F)ccc2c(c1)COC2 n1(Cc2cc(OCC)on2)c(N2CCC(CC(=O)OC)C2)nnc1C1CCCO1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CCC2(CCC2NC(C2CC(C)N(C)C2)=O)CC1 CN1CCC(C)(CNC(=O)CC2CCCN(C(C3CC(O)C3)=O)C2)C1 CCCC(C=O)C(=O)NCC1CCCC(CNC(C2CC2COCC)=O)C1 C1(NC(C2(CCC)CCC2)=O)CCN(CCNC(C2(C)CCCCO2)=O)CC1 C(=O)(CCCCCCCBr)NC(C1CCN(Cc2cc(F)c(F)cc2Cl)CC1)C C(c1cnc(O)nc1O)=CC(=O)NCCCCCCNC(C(C)CS(C)=O)=O CC(C)C(O)C(C)C(=O)N1CCC(CF)(NC(=O)CSCCN(C)C)C1 CCCN(OC)C(=O)C1(C)CC(O)CN1C(c1cc(F)n(C)n1)=O N1(C(CCCc2onc(C)n2)=O)CC(C)(C)CC1CNC(c1ncccc1O)=O N1(CC(C)NC(c2nc(C(C)C)oc2)=O)CCN(C(=O)COC(C)(C)C)CC1 CCCCCC(C(=O)Nc1cccc(Cl)c1C)N1CCN(C(C)CC(=O)OC)CC1 c1(C(=O)NC(CNC(c2cc(CCCO)on2)=O)CO)ccc(Cl)nc1O C1(N2C(=O)CC23CC3)CCCN(C(=O)C(C)OC(C)=O)CC1.C1(OC)CCCC1 N1(C(CN(CC(C)(C)C)C)=O)CCCN(C)CC1.N1(C(=O)C2CC2)CC(C)(CC)C1 c1(CC)nc(=N)[nH]cc1C(=O)NC1CCN(C(C2(c3cc[nH]n3)CCC2)=O)CC1 N1(C(C#CC2(CC)CC2)=O)CCN(C(=O)CCc2nc(C)no2)C(C)CC1C N1(C(c2[nH]cc(CC)c2)=O)CC2CCC(CNC(c3cc(COC)on3)=O)(C2)C1 C12(CN)CCN(CC1)C2=O.c1(OCCOC)ccc(C2CCC2)cc1 c1(C(=O)NC(C(=O)NC(C)CC(F)(F)F)(C)C2CCC2)cc2cccnc2[nH]1 c1(NC(C2N(C(Cc3cnc(C)s3)=O)CC2)=O)cc(Br)ccc1[N+](=O)[O-] c1(C(N2CCC(C(CNC(CC(=C)C)=O)O)CC2)=O)ccc(NC(C)=O)c(F)c1 N1(C(C(=O)NCc2onc(C(C)OC)n2)=O)CCC(SCc2nc(Br)sc2C)CC1 c1(N2CC(C)C(NC(c3cccnc3F)=O)C2)nc2ncc(Cl)cc2o1 c1(C(N2CC(OC)CC2(C)CNC(c2sccc2C)=O)=O)cc2n(n1)CCOC2 N1(C(CCC(=C)Br)=O)CCCC(N(C(=O)CC2CCOC2)CC)CC1 c1(C(N2CC(C)C(NC(c3coc(C(F)F)n3)=O)CC2)=O)ccc2[nH]ccc2c1 C1(NC(CC=C=C)=O)CCC2(CC1)CN(C(=O)Cc1n[nH]c3ccccc13)C2 CCCC(CCC)CC(=O)N1CCCCC1CCCNC(C12CC(OC)C1C2)=O N1(C(C2N(C(C)C)C(=O)CC2)=O)CCCC(N=c2nc(C(F)(F)F)[nH]s2)(CO)C1 CC1CCCN(Cc2ccccc2NC(=O)COCc2ccccc2)C1 C(C(=O)N(CCC(=O)NCC(C)(C)OCC1CC1)C)(OC)OC C1(C(N(C(C)C(C)(C)C)C)=O)(CF)CCN(C(=O)Cc2ccc[nH]2)C1 c1(CCNC(C(C)n2cnnn2)=O)ocnc1CNC(=O)Cc1ccco1 c1(NC(C2CCN(C(c3c(C)cc(Br)cn3)=O)C2)=O)ncc(S(=O)(=O)O)cc1Br C1(CNC2(c3nnnn3CC3CCCCC3)C(C)CSC2)CCCCC1(F)F Cc1sc(=O)n(CC(=O)NCCCCN(C(=O)C(C)c2cc[nH]n2)C)c1C C1(CNC(Cc2n(C)nnc2)=O)CN(C(C2(C)CCOC2)=O)CC12CCC2 N1(C(CCc2cn(C)nc2)=O)CCCc2c1cnn2OCCN1CCCC1 N1(C(c2ccc(C)s2)=O)CC2(NC(c3cc(C)n(C)c3)=O)CC1C2 O=C(CS(=O)(=O)c1ccc(Cl)cc1)NCCOCCNC(c1ccncc1O)=O C1(C(CC)CC)CCC(NC(=O)N(C)CC2CCOC2)CC1 C(CNC(C1(COC)CCOCC1)=O)(C(C)C(C)C)NC(c1cc(CC)[nH]n1)=O c1(C(=O)NC(C(C)NC(C(C)OCCOC)=O)CO)nc(-c2cccs2)oc1C C(=O)(C(C(C)(C)C)N(C)C)OC(c1ccc(C)o1)C1CCCCC1 CCC(C(C)C)C(C(=O)Nc1ccc2c(c1)CCC2)N1CC(F)(F)C1 C#Cc1ccc(C(=O)NC(C)CCCNC(C23CCC(CO)(CC2)C3)=O)cc1C Cc1cnc(NCC2C3CN(C(C4COCCC4(F)F)=O)CC23)c([N+](=O)[O-])c1 C(C(C(=O)N(C)CC1CCOC1C)C(C)(C)C)NC(CC(C)C)=O c1(C(=O)NC(C2(O)CN(C(C3CN(C)CC3C)=O)C2)C)cc(O)ncn1 N1(C(c2c(C(N)=O)coc2)=O)CCCC(C(=O)NCC(CO)NC(N)=O)C1 c1(CNC(C(C(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)=O)cc(Br)ccc1[N+](=O)[O-] C#CCCCCC(=O)NCC1CN(C(=O)C=C(C)C)CCC1C N1(C(C2(C)N(C)CCC2)=O)CC(C2CN(C(=O)CN3CC4CC4C3)C2)C1 CC(C)CCC(=O)N1CCCC(NC(c2cc(C(F)F)cs2)=O)C1 C1(C(N2C(C(=O)NC3(CC#C)CCC3)CC2)=O)(COC)CCCO1 c1(OC)ccc(C(N2CC3(CCC3)C2C2CCOCC2)=O)nc1N c1(CC)ncsc1C(=O)NCC1CCC1NC(C1CCCN1c1ccncn1)=O C1(NC(c2cn(CCN(C)C)nc2)=O)CC(O)CN(C(C2(C(N)=O)CCC2)=O)C1 N1(C(c2ccc(F)cn2)C(=O)NCC)Cc2ccccc2C(c2ccccc2)C1 CC1(C)CCCC1(C)NC(C1CN(C(c2ccnc(O)c2)=O)CCO1)=O c1(CNc2c(SCC)nccc2)cc(F)c(Cl)c([N+](=O)[O-])c1 c1(Cn2cc(C3(O)CN(C(=O)CCCCC4CC4)C3)nn2)cc(Cl)ccc1Cl N1(C(C(c2ccc(C)cn2)(F)F)=O)CCCC(O)(CNC(=O)C(F)C2CCC2)C1 c1(C)ccncc1.C(=O)(CCN(C)COC(=O)CCCNCC1CCC1)C1(N)CC1.C=O C1(NC(=O)CC2CCOC2)CCCC2CN(C(c3ccc(O)c(Cl)c3)=O)CC12 c1(NC(CSC)C)ccc(S(=O)(=O)NCC2CCOC3(CCC3)C2)c(Cl)c1 c1(OC(C2C(c3ccc(C)cc3)C2)=O)cc(F)ccc1C C(c1cc2ccccc2o1)=CC(=O)NC1CC(NC(c2n(C)ccc2)=O)C1 C1(C)(C(N2CC(C(N(C)C)=O)C2)=O)CCN(C(=O)COCCCN=[N+]=[N-])C1 N1(C(c2c(OC)csc2)=O)CC(NC(C2CC23CCOCC3)=O)CC(F)(F)C1 c1(N2CCCC(CN(C(c3c(CC)noc3C)=O)C)C2)nc(OC)c(F)c(C)n1 N1(C(C2(CC#C)CCCC2)=O)CCC(C)(CC(=O)NCCCC(=O)NO)C1 c1(CC(=O)OCCOc2c(C)cc(Cl)cc2)ccccc1N=[N+]=[N-] C=CCC(C(=O)N1CCC(F)(F)C(CNC(=O)Cc2cnoc2)C1)C(C)(C)C C(=O)(CC(CCCC)NC(=O)Cc1cncnc1O)N1CCCC(C#C)C1 CCCCCC(O)CC(=O)N1CCN(C(C2CC2C(N)=O)=O)CC1C1CCC1 C#Cc1ccc(C(c2nnnn2C2CCOC2)NCC2(CO)CC2)cn1 c1(NC(C(=O)NC(c2noc(C(F)(F)F)n2)(CC)C)=O)cc(OC)nn1C c1(OCC#C)ccc(C(=O)NCC(C)(CO)NC(=O)CCC=CC(C)C)cc1 C=CCC(C(=O)OC)NC(=O)CCOCCN(C)C(C1C2CCCC12)=O N1(C(c2ccc(COC)o2)=O)CCC(NC(C2CCN(C)C(=O)C2)=O)C(C)(C)C1 Cc1cc(C(=O)NC2CC2CNC(=O)C(C(C)C)N2CCCCC2)c(O)nc1C CC1CN(CC(c2ccccc2Br)O)CCN1c1ccncc1 C1(NC(c2nn(C)c(O)c2)=O)CCN(C(=O)C(c2cccnc2)O)CC1(C)C C(=O)(CC(C)C(C)(C)NC(c1ccn2ccccc12)=O)NC(c1nc(=O)o[nH]1)C c12ccc(nc1)SCC(O)CNC2=O.c1(C(N)=O)ccncc1.C1CC(=O)N1 N1(C(C=CC=CC)=O)CCN(C(=O)C(c2cccc(Cl)c2)O)CCC1C c1(C(=O)NC(C)C(C)NC(C2(C#N)CC2)=O)ccc2nn(C(F)F)cc2c1 c1(C(=O)NC(C)C(CO)NC(c2ncncc2C#N)=O)ccccc1[N+](=O)[O-] N1(C(c2cc(Cl)ccc2F)C(=O)NC)CCCc2cc(C(C)(C)C)ccc21 C#CCC(CC(=O)OC)NC(=O)C(CC(C)C)NC(C1CC1C(F)(F)F)=O C1(CNC(=O)CN2CC3CC3C2)CN(C(=O)CN2C(=O)CNC2=O)CC1O N1(C(C2CCN(C)CC2)=O)CCC2(CCN(C(C3(C)CC=CCO3)=O)C2)C1 Cc1cc(NC(C2CSCCN2C(c2ccc3n[nH]cc3c2)=O)=O)c(F)cc1F c1(OC)cccc(NC(C2(C)CCCN2C(c2cc(C#N)cs2)=O)=O)c1O N1(C(C=CC(=O)OCC)=O)CCC(C(=O)NCCSCCC(F)(F)F)C1 c1(OC)ccc(CC(N2CC(NC(=O)CCn3ccccc3=O)C(C)C2)=O)cc1 c1(CC2CC2)cccc([N+](=O)[O-])c1.c12cccc(c1)Cn1c(ncc1)NC2=O c1(C(N2CC(NC(C3(CF)CCC3)=O)CC(O)C2)=O)cc2c(o1)CCCC2 N1(C(CCCCOCC)=O)CCC2(CCCN2C(=O)CC2NC(=O)NC2=O)CC1 c1(C(=O)NCCC2CC(NC(C3(OC)CCC3)=O)C2)cnc(C)nc1 C1(O)(CNC(c2cc(CNC(C3(CC4CC4)CC3)=O)on2)=O)CCSC1 c1(CNC2(c3ccccc3)CN(C(c3c(C)onc3O)=O)C2)cnc(O)c(F)c1 c1(C(c2noc(-c3cc(C4CCCN4)[nH]n3)n2)C)ccc(CC(F)F)cc1 N1(C(C2(C)CCCCCC2)=O)CCCC(C2CN(C(C34CC5CC3C4C5)=O)C2)C1 OCC(Cc1ccoc1)CN=c1nc(N2C3CCCC2COC3)c2c([nH]1)CCC2 Cc1cn2nc(C(N3CC(CN=c4cc(C)nc[nH]4)C(C)C3)=O)cc2c(=O)[nH]1 c1(C(C(=O)NCCOCC(=O)NCC(CO)C2CCC2)O)cccnc1 C1(C2(O)CCOCC2)(C(N2CC3CCN(C(=O)C4=C(Cl)CCCC4)C3C2)=O)CC1 C1(C(C)NC(=O)CCCN2CCCCC2)CN(C(c2ccnc(F)c2)=O)CCO1 c1(C(=O)NC2C(CNC(C=CC(C)C)=O)CC2)cc(C(C)(C)C)n(C)n1 C1(C(N2CC(C(C(=O)NCC(O)CSC)OC)C2)=O)CCOC1(C)C n1(CC(C(=O)NC2(CF)CCN(C(C(C#C)(C)C)=O)C2)C)ccc2ccccc12 C1(CNC(C2(CCC)CC2)=O)CCCCN(C(C2(F)CCCN(C)C2)=O)C1 N1(C(Cc2ccc(C)o2)=O)CCCC(NC(c2ncc(Br)cn2)=O)C1 C(=O)(C(CC#N)c1ccccc1)NCC(CN(C(=O)COCCOC)C)O N1(C(C(CC)N(C(=O)C=Cc2cnn(C)c2)C)=O)CCC2CCN(C)CC12 O(NC(=O)C1CC(=O)O1)C(=O)OC(C)(C)C.c1(CC)cc(-c2ccn(C)c2)[nH]n1 CC1(C)CC2(CC(C(=O)NCC3(O)CCN(C(C4CC(F)(CF)C4)=O)C3)C2)C1 Cc1cc(Cl)n[nH]c1=NC(=O)C1CC1C(=O)NCc1cccc(Cl)c1Cl CC(F)(F)C(F)C(=O)NCCOC1(CC=CC(=O)NCC2CCC2)CCC1 C1(c2n(CCC)nnn2)(NCc2cn(C3CC3)nn2)CCC(CC)C1 N1(C(C(n2cc(-c3cccc(C)c3Cl)nn2)C)=O)CCC(O)C(C)(C)C1 N1(C(CC2CN(C(c3ccc(CC)nc3)=O)C(C)C2)=O)CCC(F)(C#N)C1 c1(C(N2CCC(CCC(=O)NCc3onc(CC)n3)C2)=O)c(C)ccnc1O C#Cc1ccc(OCC(=O)NC2CC3CC(NC(C4(CO)CCC4)=O)CC23)cc1 N1(C(C=CC(C)(C)SC)=O)CC2CC1C2C(=O)NC1CCCC1N(C)C N1(C(C23CC(C)C2C3)=O)CC(N)CC2(CC2)C1 C1(C(=O)NCc2c(C(=O)NCC(CC)C)n[nH]c2)CN(C)CC(C)O1 C1(c2n(CCCCCC)nnn2)(Nc2cnc(C)c(C)c2)CN(C)CC1C c1(C(=O)NC2CCN(C(c3cc(C)nc(O)c3)=O)CC2O)ccc2oncc2c1 CC1CC2CN(C(C3COC(=O)C3)=O)CC2N1C(c1ccncc1)=O N1(C(C2CC(OC)C2)=O)CCN(C(c2oc(CO)cc2C)=O)CC1CS(C)(=O)=O Cc1nn(CC(=O)NCC(C)(C)CNC(=O)C(F)(F)c2cnccn2)c(=O)o1 c1(C(N2C3CN(C(C(C)Br)=O)CC2C3)=O)ccc(I)c([N+](=O)[O-])c1 N(C1CCC(NC(=O)CC(C)(C)O)c2ccccc21)C(CC=C=C)=O c1(CN(C2CCCC2)CC(C)C)c(F)ccc(C#N)c1F C1(NC(c2cc(CC)no2)=O)COC2C(NC(=O)C(O)CN3CCCC3)COC12 N1(C(C(COC)(F)F)=O)C(CC(=O)Nc2cnccc2CO)C2CCCC12 N1(C(CCOCC)=O)CCCCC(NC(C2CC(F)(CO)C2)=O)C1 CS(=O)CCC(=O)NC12CC(CNC(c3ncoc3-c3cccc(F)c3)=O)(C1)C2 C1(CNC(CS(=O)(=O)NC)=O)CN(CCC2CCS(=O)(=O)C2)CCC1(F)F Cc1ccc(C(N2CCN(C)C(C(=O)N(C3CCN(C4CC4)C3)C)C2)=O)cc1O C1(C(=O)NC2CCC(C(NOC(C)(C)CO)=O)C2)CCCC2(CC2)C1 CCCC(C)C(=O)N(C(C)(C(N1CCC(C)(CO)C1)=O)C1CC1)C N1(C(c2scc(C(C)=O)c2)=O)CCCC(N(C)C(c2cc(C)c(C)o2)=O)CC1 N1(C(CCC(=O)NCCC)=O)CCOCC(NC(c2cc(Br)ccc2C)=O)C1 Cc1ccnnc1C(=O)N(CCCCCNC(=O)CCC1COC(C)(C)O1)C N1(C(CCCc2onc(C)n2)=O)CC2CCCC(NC(C34CC(C3)C4)=O)C2C1 CC1(NC(=O)CC2CC(F)C2)CC(NC(=O)CC2(C3CC3)CC2)C1 C1(NC(=O)CNC(=O)C2CC2)CCN(C(c2ccc(C3CC3)nc2O)=O)CC1F C(C)(C(C)(C)C(=O)NCCOC(=O)C1CC1)NC(CCC(C)OCC)=O Cc1ccccc1C(N1CC(CNC(=O)Cc2ccnnc2O)C1)=O C1(OC(C)C)CC(NCCCc2ccccc2)C1(C)C c1(CC(N2C(C)CC(NC(CCOCC)=O)C2)=O)c(Cl)cccc1Br C1(C(=O)NCC2(C(=O)NC(C)C)CC2)CCCN(C)C1.C1(C)CCCN1C=O c1(C(=O)NC2CCCC2NC(=O)C(O)CC2CC2)cc2cc(F)cc(F)c2[nH]1 C1(CNC(c2c(C)cc(C)s2)=O)CC2CCC1N2C(c1cc(CO)on1)=O c1(NC(C2CN(Cc3ccc(Cl)o3)CCS2)=O)ccnc(-c2ccccc2)n1 N1(C(C2CC(C)SCC2)=O)CCN(C(c2cnco2)=O)CC1C(C)(C)C Cc1cc(C(N2CC(CO)(NC(C3CCCC3O)=O)C2)=O)c2c(C)n[nH]c2n1 C1(CCNC(C23CC(F)C2C3)=O)(OC)CN(C(=O)CCc2ccn(C)c2)C1 C12CCCN(C1)CCCOC2=O.CCCCNC(=O)N(C)C c1(OC)nccc(C(N2CCC(C)C(NC(=O)CCc3cn[nH]c3)C2)=O)c1Br c1(C(=O)NCCCC2N(C(CN(C)C(N)=O)=O)CCC2)cnncc1O Cc1nc(N2C(C(N3CCC(O)C(F)(F)C3)=O)CC3CC23)nc2ccc(Br)cc12 C1(CC(=O)NCC2C(C(=O)NC)CCC2)(CC)CCOCC1.C12(CC1)C(=O)N2 C#CCC(CC(F)F)C(=O)N1CC(CNC(=O)C2=C(C)OCCS2)C1 c1(C(=O)NCC(CC)NC(=O)CCCS(N)(=O)=O)cccc2oc(=N)[nH]c12 CN1CCc2c(C(N3CC4CCC3CN4Cc3csc(Br)n3)=O)cccc21 C1(NC(C(C)N(C(=O)C(F)OC(F)(F)F)CCC)=O)CCCCC12CCC2 C12(CC)CN(C(C3CC=C(C)CC3)=O)C(CNC(=O)Cc3cnccc3Cl)(C1)C2 O(NC(=O)C1CCc2c[nH]nc21)C(CC(C)C)C(=O)NCCCCCCF C(=O)(C1SCCc2sccc21)NC(C(C)C)(C)CNC(c1cnnn1C)=O C1(OCC)CC2(C1)CC2NC(C1(C(=O)Nc2cccc(OCC)c2)CC1)=O C12(CNC(C(C)C)=O)CC(CO1)N(C(=O)CCc1nc(C3CC3)no1)C2 c1(CC(=O)NC23C(CN(C(CS(CC)=O)=O)C2)C3)ccc2nc[nH]c2c1 O=C(C1=COc2ccccc2O1)NC12CCC(CF)(C1)OC2 C(C1(C)COC1)=CC(=O)NC1(CN(C(=O)Cn2ccc(Br)n2)C)CC1 c1(C(=O)NC(CN(C)C(C2CC3(CC3)CO2)=O)(C)C)ccccc1SCCO c1(C(=O)NCC2(C)N(C(c3nc(C)c(C)s3)=O)CCC2)cccc(F)c1Cl CCCC(C#N)C(=O)N(C)CC1CCN(C(C2(C(C)(F)F)CCC2)=O)C1 c1(C(=O)NC(C(C(C)C)NC(CCNC(=O)OC)=O)C)cc2c(s1)CCCCC2 c1(C(=O)NCCC(C)CCNC(C2CCC(C#N)CC2)=O)ccc2cncn2c1 C1(C(=O)NCC2(O)CCCN(C(CC#N)=O)C2)CCCc2ccccc2C1 C1(CC=C)(NC(c2cn(C(F)(F)CO)nn2)=O)CN(C(C2CC(=O)N2)=O)C1 Cc1nc(C(N2CCC(O)(CCNC(c3ccns3)=O)C2)=O)c2n1CCCC2 CCC(CC)CCC(=O)N1CC2(C1)CN(C(c1cncnc1)=O)C2 C1(CNC(c2c(C)nco2)=O)CC2CCC1N2C(c1scc(Br)c1C)=O N1(C(C(CC(C)C)OC)=O)CCCN(C(c2cncc(N)c2)=O)C(C(=O)O)C1 N1(C(C(CC#C)O)=O)CCCC(NC(c2ccc(-c3nnc(C)o3)cc2)=O)C1C C(CC(C)C)(C(=O)N1CCC=C(F)C1)C(=O)NOCC1(COC)CCC1 C1(CN(C(c2ccc(COC)[nH]2)=O)C)CN(CC(C)C)CCO1 c1(N(C(=O)COC(c2c[nH]nc2-c2cnccn2)=O)C)nc(Cl)c(Cl)s1 C(C)(CO)(CC(C)C)NC(c1cc(CNC(c2ccc(OC)s2)=O)ncc1)=O Cc1ccc(C(N2CCN(C(c3ncncc3Cl)=O)C3CC23)=O)cc1OC(F)F CC(C)S(=O)(=O)C(C)C(=O)NC1CN(C(c2ccccn2)=O)CC1F c1(C(C)=O)cc(C(=O)N(C2CCCCC2)CCCNC(=O)C(C)N(C)C)co1 C12CC(C)CN(C1)C(=O)C(=O)N2c1cccc(C#N)c1.c1(CC)cc[nH]c1C(=O)O O=C1CC(NC(c2coc(CNC(=O)CC3CCCCO3)n2)=O)CC(=O)N1 CCC(CO)CCNC(C1CCN(C(c2ccnn2C)=O)C1)=O c1(N(C)Cc2ccc(I)cc2Br)ncnc2ncn(C3CC3)c12 c1(C(CC(=O)NC(CNC(CN(CCOC)C)=O)C(C)C)C)ccc(F)cc1F C#CCC(C)(CC)C(=O)NCC(C)(CNC(=O)Cn1cccc1)OC C1(C(N2C(C(C)NC(c3c(COC)ccs3)=O)CCC2)=O)C2CCCCC12 c1(C(=O)NC2C(NC(CC3C(C)(C)CCC3)=O)CC2)cc(Cl)c2n[nH]cc2c1 N1(C(c2ccc(C(C)C)s2)=O)CCC2(NC(c3nc(Cl)sc3Cl)=O)CC2C1 C1(CN(C)C(c2ccn(C)c2)=O)CCCN(C(=O)COCC2CCCC2)C1 C1(C)(NC(c2nc(C)n(-c3ccccc3)n2)=O)CCCN(C(C2CCCS2)=O)C1 N1(CC)CC2CCCC2(Oc2cccc(C)c2)C1.C(C(O)C(F)(F)F)N1C(=O)C1 O=C(CCCCCn1cc(C2CCCCC2)nn1)NC1(CC2CCOCC2)CC1 C1(C)(CC)CCCN(C(=O)C(CCC2CC2)NC(c2ccc(CO)cc2)=O)CC1 N1(C(C2CC(OCC)C2)=O)CC(C(N2CCC(C(C)(C)C)C2)=O)C2(CC2)C1 C(CC1=CCCCC1)N(C(CCCC=C)c1nnnn1C)CCCC CC1=CCC(C(=O)NC(C)(C)CCNC(=O)CNc2ccc(C(N)=O)cn2)CC1 C(c1ccc(F)cc1)=C(C)C(=O)N1CCC1CNC(=O)C1=CCC1 S(=O)(=O)(c1cccnc1NCc1ccc(F)cc1F)NCc1c(F)ccc(C)c1 c1(C(N2CCCN(C(C(CCC)(C)CC)=O)CC2)=O)cnc2c(c1)CCCC2 c1(C(N2CCCC(OC)CC2)C(=O)NCC(=C)C)cc2n(n1)CCCCO2 C12(CNC(=O)CCC3CCCC3)CC(C1)C(NC(=O)Cc1cnns1)CO2 C(=O)(CC(C)(C(F)F)N(C)C)NC1CCC(N(C(CC(CC)C)=O)C)CC1 C=C(Cl)C(C)(C)C(=O)N1CCCN(C(=O)C=C2CCC2)CC1 CC1CC(NC(=O)C=CI)CN1C(C1CCC(C(=O)N(C)C)CC1)=O S(=O)(=O)(c1cccc(F)c1)NCC(=O)NC1CC(CNC(CCOC)=O)C1 c1(CCC(N2C(CN(C(c3cnsc3)=O)C3CC3)CCC2)=O)ccc(O)cc1 c1(OC)c(NCC2CCCC(NC(=O)C(C)C(C)C)C2)ncnc1Cl C#CCC(C(=O)N(C)Cc1cccc(O)n1)NC(c1cnn(C)c1C)=O c1(C(=O)NCCNC(C(C)(C)N2CCCCC2)=O)cc(Cl)c(F)c([N+](=O)[O-])c1N Cc1ccc(Cl)c(C(=O)NCC2(C(F)F)CCN(C(=O)COC(F)F)C2)c1 C(C1CCCCC1)=CC(=O)NCC1(O)CC(C(=O)NCCC(C)N(CCC)C)C1 C1(CNC(CC(C)n2ccnc2)=O)CCCN(C(c2cnn(C(C)(C)C)c2)=O)C1 C1(C(N(CC=CC(=O)N(C(C)C(=O)NC)CC)C)=O)CCC2(CC1)CC2 C1(NC(c2c(Br)n[nH]c2C)c2n(CC(=C)C)nnn2)CCn2ncnc2C1 C=CC(C)(CC)C(=O)NC1C2CCN(C(c3ccnn3CC)=O)CC12 c1(CCC(=O)NC2CN(C(C=Cc3cccc(C)c3)=O)C2)nc2ccccc2[nH]1 c1(-c2scc(CC(N3CC(c4ccccc4)C(O)C3)=O)n2)ccc(O)cc1 n1(CC)nc(C(N2CC(C(C)NC(C3CCC(=O)N3C(C)C)=O)C2)=O)ccc1=O N1(C(c2ccn(CCC)c2)C(=O)NC(C)CC)C2CCC1CC(CO)C2 c1(C(=O)NCC2(CC(=O)NCC(C)(C)OC)CC2)cn(C2CC2)nc1C CCC(CC)CCCC(=O)NOC(CC(C)C)C(=O)N1CC(C)(OC)C1 C#CCCCCCCCC(=O)NCC1CCC2CN(C(C3CNC(=O)N3)=O)CC12 C(=O)(C(F)C(=O)Nc1cn(C)nc1CNC(C12CC(C(C)C)(C1)C2)=O)OCC c1(C(=O)NC2(C)CCN(C(c3c(C)csc3Cl)=O)C2)cc2ccncc2[nH]1 c1(OC)ccc([N+](=O)[O-])cc1S(=O)(=O)N(C)Cc1cc(Cl)cc(Br)c1 C(C(CC1CCCC1)C(=O)NCC(C)(O)C(C)C)NC(COCC(=O)OC)=O N(C1CCc2cc(CNC(c3cnnn3C3CC3)=O)ccc21)C(CCOCC)=O C(CC(=O)NCCCOCCC(=O)NC1CC1)(C1CC1)NC(COC)=O CC1C(NC(C2CC2C(F)F)=O)CCCN1C(c1cc(C(F)(F)F)cnc1O)=O c1(CC)cc(N)ccc1C(=O)NCCC(O)CNC(=O)CC1(CC)CCC1 N1(C(C2(SC)CC2)=O)CCC(C(F)CNC(=O)C(O)CCN(C)C)CC1 C=CCCN=C(NCCC1C=CCC1)N1CCc2cc(Br)cc(F)c2C1 N1(C(C(C2CN(C(=O)C=Cc3ccncc3)C2)OC)=O)CCS(=N)(=O)CC1 c1(NC(C2CCC(N(C(=O)CCCNC(N)=O)C)CC2)=O)cc(F)c(F)cc1O C(=O)(C1=CS(=O)(=O)CCC1)NC1C(CC)CN(C(=O)C=Cc2cnc(C)s2)CC1 CC1(C)CC(CNC(c2ccccn2)=O)N(C(=O)COc2cc(F)cc(Cl)c2)C1 C#CCC(CC(F)(F)F)C(=O)N1CCC(Oc2cccc(C)c2)CC1 C12(C(=O)NC(CC=C)(C)C)CC(CN1C(=O)Cc1csc(C)n1)C2 C1(C(C)NC(CSCCOC)=O)CCN(C(=O)Cc2cnn(C)c2)CC1 C(c1ccccc1)(C(F)(F)F)=CC(=O)NCC(C(C)(C)C)NC(C1CCSC1)=O C1(NC(C(C)OCC)=O)CC2CC(C1)N(C(=O)Cc1noc3ccccc13)C2 Cn1cnc2c1CN(c1nc(N3CCC(C4CC4)C3)c3[nH]ccc3n1)CC2 c1(-c2nnc(N3CC(OC)C3)n2C)cc(C)c2ncccc2c1C c1(C(N2CCC(NC(C3C(=C)C3)=O)CC2)=O)ccc(C)c(S(=O)(=O)NCC2CC2)c1 N1(C(C=CC)=O)CCCC(C2CCN(c3nnc(C(C)C)c4ccccc34)C2)C1 c1(CC)cccc(C(N2CCCC(C(C)C(=O)NCC(C(C)CC)OC)C2)=O)c1 Cc1n[nH]c(C)c1CC(=O)NC1CCC(CCNC(c2cn(C)nc2Cl)=O)C1 c1(N(CCCN2CCCC(N(C)Cc3ccco3)C2)C)cc(C=O)ccn1 C(=O)(C(C)CCC(C)(C)C)N(CC(N1CCSC(C)CC1)=O)CCC Cc1ccc(C(=O)NC23CCN(C(c4oc(C)nc4C)=O)CC2C3)c(C)c1 N1(C(C2C(CCC)CCC2)=O)CC2(C1)CN(C(=O)C(C1CCOCC1)C)C2 C1(C(=O)NCC(C)NC(C(C2CC(F)(F)C2)OCC)=O)CCC(=C2CCC2)CC1 c1(C(N2C3CN(Cc4c(Cl)cccc4I)CC23)=O)cc(F)c([N+](=O)[O-])cc1F c1(OC(C)C(=O)NCC(CO)NC(C2(n3cccn3)CC2)=O)ccc(Cl)cc1 N1(C(C(c2c(C)cccc2Br)NC(C2CC2C2CC2)=O)=O)CC(C)(C)C12CCC2 O=C(CCCCOCCO)NCC1CC2(C1)CC2F c1(CNC(=O)NCC23CCCN(CCC2)C3)cccc2nn[nH]c12 C1(CNC(c2ccc3cc[nH]c3n2)=O)C(C2CC2)CCN1C(=O)C=C1CCC1 N1(C(c2n(C)nc(Cl)c2)C(=O)NC2CCOC2)CCC(N(C)C)(CO)CC1 c1(C(N2CCCC(C)(F)C2)=O)noc2c1CN(C(C1CC1C1CC1)=O)CC2 CCCC(C)(C)C(=O)NC(C)C(C(C)C)NC(c1cn(C)c(C)n1)=O C(CCCCC(=O)N1CC2C(CNC(c3cc(C)cc(C)c3)=O)C2C1)OC C12(NC(COC(CC)(C)C)=O)COC(C1)C(NC(C1(n3cc(Cl)cn3)CC1)=O)C2 C1(C)(NC(C(C)Cn2ccnc2)=O)CCCN(C(c2ccc(O)cc2)=O)C1 N1(C(C(C)(C(C)C)OC)=O)CC2CCCC2(NC(=O)CCNC(=O)C=CCl)C1 C1(NC(=O)CCCc2cccs2)(CF)CCN(C(C23CC(C2)C3)=O)C1 CC#CCCC(=O)N1CCC(CN(C(=O)C(C(C)C)N2CCCC2=O)C)CC1 N1(C(c2cnn(CC)c2C)C(=O)NCCOCCOC)C2CCC1CN(C)CC2 c1(CC)cccnc1C(=O)NC(C)(CNC(=O)C(C)NC(=O)CC(F)(F)F)CO c1(C(=O)NCC2(F)CC(NC(c3c(C)coc3C)=O)C2)ncn2c1CCCCC2 c1(C(=O)NCC(N(C(c2c(C)ccs2)=O)C)C2CC2)cccc(C2CCOC2)c1 C(=O)(C#CC1(C)CCCO1)N1CC(C)(C(=O)NCC(CCC=C)(C)C)C(C)C1 c1(SC2(C(=O)NCC(C(C)C)NC(c3noc(CN)n3)=O)CC2)ccccc1F N1(C(C(C)N(C)C)=O)CCN(C(c2nn[nH]c2C(F)(F)F)=O)CC1CO c1(CC)n[nH]cc1C(=O)NCC1(CCNC(c2cc(C(F)F)cs2)=O)CC1 N(C=CC(=O)C(F)(F)F)C(C1CC2(C1)CN(C(c1cc3ccoc3s1)=O)C2)=O C(CN=c1ccc(Br)c(S(=O)(=O)NC(C)CC(C)O)[nH]1)c1scc(C)n1 CCCCC(CCC)N=c1[nH]c(N2CCCOC(CC)C2)nc2ccsc12 C(C)(CO)(C(=O)NCC(C(C)(C)C)NC(=O)CCc1cc[nH]n1)OC C1(N(C(C(c2ccnn2C)C)=O)C)CN(C(=O)C=C2CCSCC2)CCC1O C1(N(C(c2ccc(C)cc2)=O)C)CN(C(c2onc(C)c2C)=O)CC12CC2 c1(C(=O)NCCNC(=O)CCCn2ccnn2)c(-n2cccc2)sc2c1CCC2 C1(C(=O)NC2(C)CN(C(C(Cc3c(C)nc[nH]3)O)=O)C2)CCc2n[nH]c(C)c2C1 N1(C(=O)CC(F)(F)Cl)CC2(C1)CN(C(C1CCOC3(CCC3)C1)=O)CC2CO N1(S(CC=C)(=O)=O)CC2OCCN(C(=O)Cc3ccc(OC)cc3Br)C2C1 CCC(C)C(C(=O)NCC(C)C)N(C)C(c1cc(C)on1)=O c1(CC)cc(OC)ccc1C(=O)NC(C)C(C)NC(=O)CCCCN(C)C(C)C N1(C(c2cnc(OC)c(C)c2)=O)CCOCC(F)(CNC(c2[nH]nnc2C)=O)C1 c1(COC)nc2ccccn2c1C(=O)NC1CCCN(C(=O)CCCCSC)C1 C#CCC(C)C(=O)NC1COCC1NC(=O)COc1ccc(CC(=O)NC)cc1 c1(NC)ncccc1C(N1CCCC(CCC(=O)NCC(C)F)C1)=O C(C(CNC(C1(C#N)CCC1)=O)CO)NC(C1CC(C)C1)=O c1(CC(=O)N(C2CC(NC(CCCc3onc(C)n3)=O)C2)C)cccc(F)c1F C1(NC(c2cc(C)sc2)=O)CC12CCN(C(c1c(O)cc(O)cc1O)=O)CC2 c1(C(N(CCCNC(CC(C=C)C)=O)CC)=O)ccc(C(C)C)cc1O C1(C(N2C(C=CC(=O)NC(C=C)C(F)(F)F)CCC2)=O)CCCCNC1=O CN1C(=O)CSC1=CC(=O)NC1CCCN(C(c2cccc(Cl)n2)=O)C1C C1(C(=O)NCC2C(CNC(c3c[nH]cc3C3CC3)=O)C2)CC1C1CCCC1 N1(C(CC(c2ccc(F)cc2)=O)=O)CCOCC(NC(C23CC(O)C2C3)=O)C1 N1(CCCC)CCCC2(CCN(C(=O)CCc3c(C)noc3C)C2)C1 N=C1NC(=O)C(CC(N2CCC(C(C)(C)C)(CNC(C3CCS3(=O)=O)=O)C2)=O)S1 C1(C(N2CC(C)(NC(=O)C=Cc3ncc[nH]3)C2)=O)(COC)C=CCC1 c1(CN(C)C(C2C(CNC(=O)C(O)Cn3cncn3)C2(C)C)=O)cccc(O)n1 Cc1nn(CCO)cc1C(=O)N(CC(O)CNC(=O)CCc1cnoc1)C Cc1ccc(OCC(=O)NC(C)CC2CCN(C(=O)C3=CCCS3)CC2)cc1 C12(NC(c3scc(C(N)=O)c3)=O)CCN(C(c3cnnn3C3CC3)=O)CC1C2 C1(C(=O)NCCC#C)CCC(C)(C)N(C(=O)C(CC)C(=O)OCC)C1 CCCC(C(=O)NC1CCCCC1CC(=O)N(C)Cc1nncn1C)OC CCCC(C)(C)CC(=O)N1CCN(C(C2CCCC(CF)C2)=O)C(CC)C1 C(=O)(CCCCN=[N+]=[N-])NCCC(C(=O)NCC1CCC(C)CC1)OC c1(NC(C2CSCCN2C(c2cnccc2Cl)=O)=O)ccc(Br)nc1F N1(C(C(C=C)O)=O)CC2(CCN(C(c3cnc(C)nc3C3CC3)=O)CC2)C1 N1(C(c2c(C)oc(C(C)C)n2)=O)CC(NC(C2CCCSC2)=O)C2CCCCC12 N1(C(CCN(C(c2c(C)cnnc2)=O)C2CC2)=O)CCOC(C)(C(C)C)C1 C1(NS(c2c(C)cc(SC)nc2)(=O)=O)CCOC2(CCS(=O)(=O)C2)C1 C1(CC#C)(C(=O)Nc2csc(Cl)c2)CCN(C(C2CCC3(CC3)C2)=O)C1 C(CC(F)(F)Cl)NC(C(C1CCCC1)NC(C)=O)=O c1(C(N2CC(N3CCN(C(C(CC)CC)=O)CC3)C2)=O)cc(=O)n(C)c(=O)n1C C1(CNC(C2CC(C)C2)=O)CN(C)CCN1C(c1ccc(-c2cnco2)cc1)=O c1(C(=O)NCC2(O)CC2)cc2n(n1)CCCN(C(C1(F)CCC1)=O)C2 C=C(C)CC(C)C(=O)Nc1ncc(-c2ccccc2Cl)s1 Cc1cc(C(=O)NCC2(CNC(=O)C(C)(C)N(S(C)(=O)=O)C)CC2)ncc1Cl N1(C(c2c(OC)c(C)sc2)=O)CCC2C1CCCN2C(c1csnc1C)=O N1(C(CCC=C)=O)CCCOC(CNC(c2occc2C(=O)OC)=O)C1 C1(C)(CC)C=C(C(=O)N2CCCC2CNC(C2CC3CCC3C2)=O)C1 C1(CC=C)(NC(=O)C(CCC)OCC)CCN(C(=O)Cc2cccc(Cl)c2)C1 CC1CN(C(=O)CC2CCOC2=O)CC(C(=O)N(CC(CO)N(C)C)C2CC2)O1 c1(C(N(C)CC2CN(C(C3CN(C4CCC4)C3)=O)C2)=O)ccn2cncc2c1 Cc1ccc(C(=O)NC2CC(NCc3cnc4ncccn34)C2)cc1[N+](=O)[O-] N1(NCC2N(CCC)CCC2)CCCC(O)(CC)CC1 N(C1CCCc2c[nH]nc21)C(C(C)CN(C(=O)CCc1nccs1)C)=O C12(CNC(C(CC)N(CC)CC)=O)CCC(CC1)N2C(c1cc(F)ccc1C)=O C1(CNC(C(C)N(C(=O)CNC(=O)OC)CC)=O)CCC(=O)N1 Cc1cccc(N)c1C(=O)NC1CC(F)CN(C(C2CC2CF)=O)C1 C(CN=c1[nH]c(Cl)nc2c1CS(=O)(=O)C2)c1ccc(OC)c(F)c1 c1(NC(c2c(OC(C)(C)C)ncc(-c3csc(=N)[nH]3)c2)=O)ccc2[nH]ncc2c1 C(C)(C)(CCC(=O)NCCCCCCNC(=O)C(c1cnn(C)c1)O)OC C(=O)(C(F)CC(C)(C)C)N1CCC(CC=C)(C(=O)NCC2(CO)CC(C)C2)C1 C1(CN=c2[nH]nc(CO)s2)(NC(c2cc(CCC)oc2C)=O)CCCCC1C c1(=O)n2c(C(F)(F)F)cc(=O)n1nc2C(=O)NC(C)CF.CCO C1(C(N(CC=C)Cc2ccccc2)=O)CN(C(=O)C(F)C(CC)CC)CC(C)(C)C1 C(=O)(C1=CS(=O)(=O)CCC1)NC(CNC(C1(CC)CCOCC1)=O)CO CC1CCC(NC(=O)CC2(n3cnnn3)CCSCC2)CN1C(=O)OC(C)(C)C c1(C(=O)NC(C)CC(C)NC(C23CC(CO2)C3)=O)csc(=NC2CC2)[nH]1 CCC(CC)C(F)C(=O)NCC(C)(C)CC(=O)NC(COC)C(C)C c1(CC(=O)NCC(C)(C)NC(CSCC)=O)ccc2c(cnn2C)c1 c1(CC(N2CCC(OCCOC)CC2)=O)csc(=NCc2c(Cl)ccnc2Cl)[nH]1 C1(N(C(Cc2c(C)n(C)nc2)=O)C)CCN(C(c2ccc(C#N)[nH]2)=O)CC12CC2 C1(NC(c2nccc(CC)c2)=O)CCCN(C(C2CC(C(C)=O)C2(C)C)=O)CC1 c1(COC)cccc(NC(=O)C(=O)NCC2CN(C(=O)OC(C)(C)C)C2)c1 c1(C(N)=O)ncccc1C(N1C(C(N)=O)CC2CC12)=O N1(C(C(C)CO)=O)CCN(C(N2CC3(CC3C(=O)O)C2)=O)CC1 c1(C(=O)NC2C(C)(C)N(C(c3cc(Cl)ccc3F)=O)CC2)occ2c1CCOC2 C1(CCCC(=O)N(C(CC)CC)CNC(=O)CS(=O)(=O)NC)CCC(C)C1(C)C c1(CC)cc(C)ccc1C(=O)NCC1C2CN(C(c3cc(O)ccc3Cl)=O)CC12 C1(CC)CCN(C(=O)Cc2cc[nH]n2)C1C(N1CCC(OCC(N)=O)C1)=O C(=O)(C(O)(CN(C)C)C(F)(F)F)NCC(C)NC(C1(C(F)F)CCCCC1)=O C1(NC(c2ncc(C)c(Cl)c2)=O)CC2CCC(C1F)N2C(c1cccc[n+]1[O-])=O c1(C(N2CCN(Cc3cnc(SC)nc3)CC2C)=O)cc(F)cc(F)c1Br O=C(C#CC1CCCC1)NCc1cccc(NC(c2ccsn2)=O)c1 CCC(O)C(C)(C)C(=O)N1CCN(C2CCN(C(=O)CCCN=[N+]=[N-])CC2)CC1 c1(C(N2CC(NC(c3cnc(C)n3C)=O)C(C)C2)=O)nc(Cl)ccc1OC(C)C C1(NC(CS(CC)=O)=O)CC2CN(C(=O)C(O)C(C)(C)CC)CC2C1 N1(C(c2c(C)oc(C)c2C)=O)CCN(C(c2cncs2)=O)C2(CC2)C1 C1(CN(C(=O)Cc2cccs2)C)C2CN(C(=O)C(C3CC3)C3CC3)CC12 CC1CN(C(=O)CC(C2CC2)C2CC2)CCC1NC(c1cc(Cl)ccc1F)=O C1(CNC(C(CC)NC(C)=O)=O)CN(C(c2sccc2CC#N)=O)CCC1(F)F C(=O)(C(C)CC(=O)N(C1(CC(=O)NCC2(F)CCCCC2)CC1)C)OC N1(C(CONC(C2C(C)CCO2)=O)=O)CCSCC1CO C(=O)(CCC(O)C(C)(C)C)NCC12N(C(C3(C)CCN(C)C3=O)=O)CC(C1)C2 c1(C(N2C(C)C(C(=O)NC3(C(F)(F)F)CC3)CC2)=O)ccc2cc[nH]c2n1 C1(C(=O)NCc2ccc(CC)o2)CC12CC(NC(=O)Cc1ccsc1C)C2 C12(CNC(=O)C3=CCCOCC3)COCCN1CCN(C(c1cc(Cl)cs1)=O)C2 C1(CN(C(=O)NC2CC(C(=O)O)C2)Cc2ccccc2)CN(CC(F)(F)F)CCO1 c1(C(=O)NCC(C)CN(C)C(C2CC2c2ccccc2)=O)cc[nH]c2nccc1-2 Cn1cc(C#N)cc1C(=O)NC(C(=O)NCCn1ncccc1=O)C(C)(C)C Cc1ccc(Br)c(NC(C2CC23CN(C(=O)Cn2cc(C)nc2C)C3)=O)n1 c1(OC(N(CCOC(CCC)C(=O)OC)CCOC)=O)cc(C)cc(C)c1 c1(CNC(=O)NC2(n3cnnn3)CCOCC2)ccnc(-c2ccccn2)n1 O(NC(=O)C(C)(C)CC(F)F)C(CC(C)C)C(N1CCC2(CNC(=O)O2)C1)=O C(=O)(C1=CC2CC(C1)CC2O)NC12CC(CNC(c3c(CC)noc3)=O)(OC1)C2 N1(C(CC=CCC)=O)CC(C2CCCN(C(c3c(Br)cc(Br)c(O)c3Br)=O)C2)C1 c1(C(=O)NC(C(=O)NC2CCC(SC)C2)C(C)O)ccc2ccsc2c1 c1(CC(=O)NC2C(CNC(C3(C(C)(C)C)CCC3)=O)C2)cncnc1O C1(CNC(c2cc(C3CC3)[nH]n2)=O)C2CN(C(c3sccc3F)=O)CC12 Cc1nc2c(F)cccc2cc1C(=O)NCCN(C(c1ccon1)=O)CC1CC1 c1(N(C)C(c2ccnn2C)=O)ccc(S(C)(=O)=O)c([N+](=O)[O-])c1 c1(C(=O)NCC(C2CCOC2)NC(CCC=C)=O)c(C)coc1C CCCN=C(NCc1ccsc1S(C)(=O)=O)N1CCC(C(=O)OC)(CC)C1 c1(C(=O)NCC(CNC(CCCOC)=O)CO)cnc(C)nc1 C1(C(=O)NCC(C2CCCC2)NC(COCCCC)=O)CCC(N(C)C)CC1 c1(C2(C(N3C(CNC(CCC4CCN(C)C4)=O)CC3)=O)CCC2)ccccc1Cl C1(C(=O)Nc2ccc(-c3ccc(C)cc3)cn2)(CN)CCC(F)(F)CC1 c1(SC(CC)COC)ccc(OC)cc1Oc1ccc(Br)cc1 CC(C)CC(CNC(=O)OC(C)(C)C)C(=O)NC(C)CNC(C1CC1OC)=O C1(CC(=O)NC(CNC(C2(CC)CCC2)=O)(C)CO)CC2(CC2)CO1 N1(C(C(C)N2CCC2)=O)CCC(NC(c2occc2CN2CCOCC2)=O)C1C C(=O)(CCC(=O)c1cc(C)sc1C)N1CC(O)(CCNC(CCNC(C)=O)=O)C1 N1(C(c2c(CC)ccs2)=O)CCN(C(C2CCCS2(=O)=O)=O)C(CC)C1 c1(C(N2C(CCNC(c3c(CC)n(C)nc3)=O)CCCC2)=O)ccc(O)c(Cl)n1 c1(CCN=C(NC(C=C)C)NC2CC23CCCC3)cccc2cc[nH]c12 CC(C)CC(C(=O)NC1CC(F)C1)NC(c1cccc(Br)c1)=O c1(C(=O)NC2CCN(C(C(CC)SC)=O)C2(C)C)cc(CC)c2n[nH]cc2c1 Cc1cn(C(C)C)cc1C(=O)NC1C2CN(C(C3(C(=O)N(C)C)CC3)=O)CC12 C(=O)(C#CC(C)(C)CNC(C1CC12CCC2)=O)NCc1c(OC)cccn1 c1(CNC2CN(C(CC(C)O)=O)CC23CC3)n[nH]c2ccc(Br)cc12 Cc1nc(N(C2CCCNC2)C(C2CCC(O)CC2)=O)c2cc(Br)ccc2n1 C(=O)(C(=O)CC(C)C)N1CCC(C(=O)NCc2cscc2C)(OC)C1 C=CC(CC)CC(=O)N(C1CCCN(C(=O)C=Cc2ccncc2C)CC1)C N1(C(CCNC(=O)OC)=O)CCC2C(C1)CN2C(=O)CCc1cccc(Cl)c1 Cc1c(C(N2CCCC(C)C2CNC(=O)Cc2cn[nH]c2)=O)sc2ccccc12 N1(C(C2CCC(=O)N2)=O)CCCCC(NC(c2cc(F)ccc2Cl)=O)C1 c1(OCCC(=O)NCC(C)CNC(C2CCC3(CC3)C2)=O)ccc(Cl)cc1Cl N1(CC)CC(NC(=O)C(C2CCN(C(=O)CCC3OCCO3)C2)C)C(C)C1 C1(NC(C2C(C(C)(C)C)C2)=O)CC2CCC1CC2NC(C1CCCCO1)=O n1(CC=C)nnnc1C(c1cc[nH]n1)NC(C1CCOCC1)C N1(C(CC(=O)NCC(F)(F)F)=O)CCOC2CCN(C(C3(F)CCCC3)=O)CC12 N1(C(C=C(C)C(F)F)=O)CCC2CN(C(C3CC=CC3)=O)CCC2C1 C(=O)(C1=CC2(CCN(C(c3nc[nH]n3)=O)C2)C1)NCCC(CCC)C1CC1 C1(C(=O)NC2(CNC(C(C)(C)n3cccn3)=O)CC2)CCS(=O)(=O)C1 CC1=C(C(=O)NC(CNC(C2CCS2(=O)=O)=O)C2CC2)CC1 C=CCC(C)(C)CC(=O)NC1CS(=O)(=O)CC1NC(=O)COCCN=[N+]=[N-] C1(NC(c2cnc(O)s2)=O)(CNC(c2ncc[nH]c2=O)=O)CCOCC1 N1(C(C(C=C)(C)C)=O)CC2CC(C1)CN(C(C1CNC(=O)CC1C)=O)C2 CCCCC(O)C(C)C(=O)N1CC(O)CC1CNC(=O)CCOCCOCC C1(NC(CC=CC)=O)CC(O)CN(C(c2ncncc2Cl)=O)C1 c1(CCC(=O)NC(CC)CNC(C2(CCOC)CC2)=O)ccc2ncsc2c1 c1(CNC2C(C(=O)NC(C)C(N)=O)C2)c(F)ccc(F)c1O C=CCCC(C(=O)NCC(C)C#N)NC(c1ccc(OC)nc1)=O n1(CC)nc(C(N2CC(F)CC2CNC(c2cnsc2C)=O)=O)c(Br)n1 c1(OC)cc(N)c(Cl)cc1C(=O)NCC1CC(NC(C2(F)CCOC2)=O)C1 C(c1cncc(O)c1)=CC(N1CC(NC(C2C(C)(C)CC2)=O)C(O)C1)=O N(C(=NCCC(C)=O)NCc1c[nH]nc1-c1cccs1)C1CC(OC)C12CCC2 C1(C(=O)NC(C(C)C)CCNC(C2(Cl)CC2)=O)CCc2ncncc2C1 c1(C(=O)NC(CC)CNC(C2CCN(C3COC3)C2)=O)ccc(C)c(C)n1 CC(CCC(=O)NCC12CCCC1C2)NC(=O)C=Cc1cccnc1 Cc1ccc(CN(C(=O)C(CC(C)C)ONC(=O)CCc2cn[nH]c2)C)c(C)c1 C1(C(=O)OC(COC)CO)CCN(C(=O)OC(C)(C)C)C2(CC2)C1 C12(NC(C3CC3(F)F)=O)CCC(C(N3CC4C(C3)C4(F)F)=O)(CC1)C2 CC1COCCC1C(=O)NCC1CC1CNC(c1cnn(C2CCCCC2)c1)=O C1(C(N(CC(=O)NCC=CC2CC2)C(C)C)=O)CCC(CO)CC1 Cc1cc(C#N)cnc1C(=O)NC1CS(=O)(=O)CC1NC(c1ccc(Cl)o1)=O Cc1nc(=N)[nH]c(C)c1C(N1CC(NC(=O)C=Cc2cccc(Cl)c2)C(C)C1)=O C(=O)(C(C)(C)COC)OC(C)(COC(=O)NC)C1(C(=O)OCC)CC1 c1(OC)ccnc(O)c1C(=O)NCCCCC(C)NC(C1(Br)CC1)=O C=CC1CN(C(=O)CCOCCNC(c2cccn2CC)=O)CC1O CCC(C)C(C)C(=O)N(C1CCN(C(=O)C=CSC)CC1)CCO CC(CC(N)=O)C(=O)N(C)CC1CCCC1NC(c1ccc(=O)n(C)n1)=O CC1CCN(C(c2cscc2C#N)=O)CC1CNC(c1cncnc1)=O Cn1nc2c(c1C(=O)NC1CC(C)(NC(c3cnn(C(C)(C)C)c3)=O)C1)CCC2 CC1(C)CCC(C(=O)NC2(C(=O)NCCOC3CCC3)CSC2)C1 C=CCC(F)(F)C(=O)NCC1CC2CN(C(=O)CCCOC)CC12 N1(C(C(C)NC(=O)NC)=O)CCC(CNC(c2n[nH]cc2[N+](=O)[O-])=O)(OC)CC1 c1(-c2cccc(C)c2F)cn(CC(F)(F)F)c(=O)nc1O c1(OC)ccc(C)c(C2CCCN2C(=O)C(=O)OCCN2CCC(F)CC2)c1 N1(C(CSCCC(C)C)=O)CC(NC(=O)C#CC2CC2)C2(CCC2)C1 C1(=O)C(C(C)(C)C)OC2CCN1C2.C=CCC(C)(C)NC(=O)COC CN1N=C(CC(=O)NCC23CC2CN(C(C2(C(F)F)CCC2)=O)C3)CC1=O c1(C(=O)NCC2CC3CCC2N3CC2(C(=O)OCC)CC2)cc2occc2n1C C1(C)(CNC(c2ccc(COC)cc2)=O)CN(C(=O)CC(C2CC2)C2CC2)CCO1 C12(NC(=O)Cc3ncc(-c4ccccc4)o3)CCCC1N(C(=O)CCF)CCC2 Cc1cnc(N2CC3C(C(=O)Nc4c(C(F)(F)F)cccc4Cl)C3C2)nc1C C(=O)(CCC(=O)N1CC(OC)CC1CNC(C1CCCO1)=O)NCC N1(C(c2c(OC)n[nH]c2)C(=O)NCC(C)C)CCN(C(=O)CC(C)SC)CC1 C(=O)(C1=CC2CCCCCCC12)N1CCN(C(C(=O)OC)(C)C)CC1 CC(C(=O)NCC1CN(C(=O)CCc2ccco2)CCO1)C(F)F C12(C(=O)NCC(C)N(C(C(C)=CC)=O)C)CCC(O1)c1ccccc12 n1(CC)ccc(CC(N2CC(C)C2C(=O)NCCOC2CCCCC2)=O)n1 C(=O)(CC1OCc2ccccc21)N(C(CCNC(c1cn(C(C)C)nc1)=O)C)C C1(C(=O)NCCN(C(C)C(=O)NC2CCCCC2)CC)CCCCN1C N1(C(CCc2ccc(C)o2)=O)CCCC(NC(c2ccsn2)=O)C1 C12(CNC(C(C)NC(C)=O)=O)CN(C(C3CC(N(C)C)C3)=O)CC1CCO2 C1(NC(c2cc(C)nn2C)=O)CCC2CCN(C(=O)CCCc3cc(C)no3)C12 C1(C(N2CC(C)C(NC(=O)Cc3cn[nH]c3)C2)=O)CC(C)(C)OC1(C)C O=C1COc2cc(NCC3CCCC3O)cnc2N1 C=CC(C)CC(=O)N1CC2CC1C2NC(=O)Cc1ccccc1C C1(CN(C(Cc2nnc(C)o2)=O)C)CN(C(=O)CSC(F)F)CCO1 N1(C(C2C(CN)CC2)=O)CC(O)C(C#N)C1 c1(C(=O)NC23CCC(NC(=O)C(O)C(F)(F)F)(CC2)C3)coc(=O)c2ccccc12 C#CCCC(C(=O)N=c1cc(C)n(CCO)[nH]1)NC(c1cccc2[nH]ncc12)=O C#Cc1cnc(C(N2CCC(C(=O)OC(C)(C)C)CC2C)=O)c(C)c1 C1(N(C)C(=O)C2CC2)CN(CC2CN3CCN2CC3)CC1(C)C.c1ccc(F)cc1 C1(C(F)(F)F)(C(=O)NC2CCC(C)(CC(C)C)C2)CCCCCC1 c1(NCC(C2CC2)NC(c2ncn(CC)c2)=O)ncnc2c1SCCC2 c1(C(=O)NC(CCOC)C(=O)NC2CC(=C3CCC3)C2)cnc(C)c(C#N)c1 c1(C(N2CCN(C(CCC3(C)CC3)=O)C(C(C)(C)C)C2)=O)cnc2ccnn2c1 C#CC1CN(C(=O)CC2CN(C(=O)C=C(C)C(C)(C)C)C(C)(C)C2)CCN1C c1(C(C)C)nccc(C(=O)NC2CCC(NC(=O)C(c3cccc(F)c3)O)CC2)n1 CCC(CC(=O)N1CCCC(CCNC(c2cc(Cl)ns2)=O)C1)C(C)C S(=O)(=O)(c1cccnc1)N1CC(CC(N2CCCC(N3CCCC3=O)C2)=O)C1 c1(C(N2CC(O)C(F)C2)=O)cc2n(n1)CCCN(C(C1(O)CC1)=O)C2 C1(OC)CN(C(c2cccc(C(F)(F)F)c2)=O)CC1NC(c1ns[nH]c1=O)=O c1(C(=O)NC2(CNC(C(C)N(CC)CC)=O)CCC2)cccc2ccnn12 CC1CCN(C(C2CC(F)(CO)C2)=O)CC1NC(=O)Cn1cccc(C)c1=O C#CCC(CO)NC(=O)CCNC(=O)CCc1cncs1 C1(C(=O)NC2CCC2)CC(O)CCN1C(=O)CCCSCCC(C)C N1(C(C(C)NC(=O)COCC2CCCO2)=O)CC2CCC(C1)C(=O)O2 c1(C(N2CCCC(CCCO)C2)=O)cc(O)nc(O)n1.c1(N)cc(Cl)cc(Cl)c1 c1(C(=O)NC2C(NC(C(C)NC(=O)NC)=O)CCCC2)c(OC)ccnc1O C1(CNC(C=CCNC(CNC(C2C(C)C2)=O)=O)=O)CC(=O)N(C)C1 N1(C(C2CCN(C(C)=O)C2)=O)CCN2CCN(C(C3COC(=O)N3)=O)CC2C1 C1(C)(C(N(CC(=O)NC2CC(CC(C)(C)C)C2)CCOC)=O)CSC1 c1(N2CCC(NC(C)=O)C2)nc2c(c(=NCc3csc(Br)n3)[nH]1)CSC2 CC(CC(=O)NC1(C(=O)NCc2cccnn2)CCN(C)C1)C(F)F C1(NC(C2CCC(C)O2)=O)C2CC3C(C2)C13C(=O)NC1CC(O)C(F)C1 c1(N(CCNC(c2cc(OCC)no2)=O)CC)ccnc(COC)n1 c1(C(=O)NC(CN(C(C=C(C)C(C)(C)C)=O)C)(CO)CO)nccc2cc[nH]c12 c1(C(N2CC(CNC(COC(C)=O)=O)C2)=O)ccn(C)n1 C12(C(=O)NC(CC)(C)CO)CC1CN(C(=O)CC=CC(C)(C)C)C2 Cc1cc(=O)n(C)cc1C(=O)NCCN(C)C(C1(C)CCNC1=O)=O N1(C(c2c(-c3ccc(C(=O)NC(C)(C)C)nc3)ncs2)=O)CC2COCC2C1 c1(C(N(C2CCN(C(=O)Cn3ccnn3)C2)C)=O)c(C2(CO)CC2)cccc1F S(=O)(=O)(c1ccc(=NCC(C)N2CCCC2)[nH]c1)NC(c1ccc(S(C)=O)cc1)C C(=O)(C(C)(C)C1=CCSCC1)N1CC(CC(C)NC(=O)C(F)C(C)(C)O)C1 N1(C(c2c(C)onc2)=O)CCC(C)C(NC(=O)C=Cc2ccc(C3CC3)s2)C1 CCC(C)CCC(=O)NCC(C)(CO)NC(=O)CCc1cc(Cl)no1 C=CCCC(C)C(C(=O)NCCCC)N(C)Cc1ccsc1 N1(C(COCCC=C)=O)CCC(F)(F)C(CN(CCOC)CC)C1 N1(C(C(C)C2CC2)=O)CCCC(N(C(=O)CCc2nc(-c3ccco3)no2)C)C1 c1(CN2C(CC)CN(C(c3cnc(C)nc3C)=O)CC2)cc2ncccc2[nH]1 CC1OCCC1CC(=O)NC(CC1CCC1)C(=O)NCCc1nccs1 c1(C(N(CC(CC)NC(=O)C(=O)C(C)(C)C)CC)=O)cccc(C#N)c1F C#CC1(C(=O)NC2CCC(=O)N(CC)C2)CCN(C(=O)CCCn2ccnn2)C1 c1(C(N2CCN(C(C(COC)OC)=O)CC2CCO)=O)cnc2cccc(C)n12 Cc1ccc([N+](=O)[O-])cc1C(N1CC2CC1CC2NC(c1ccco1)=O)=O Cn1cnc2[nH]c(=NCC3COCC3C(N)=O)nc(N3CC4CC4(CO)C3)c12 C(C(C)N=c1cc(C)[nH]c(=NCC2(OC)CCCC(C)(C)C2)[nH]1)N(CC)CC C1(CNC(c2cc(C)n(C(C)C)n2)=O)CCN(C(C2CC(F)(CO)C2)=O)C1(C)C C(=O)(C1CC(=O)Nc2ncccc21)NC1(CNC(C(COC)(C)C)=O)CCOC1 C(=O)(C(C)C(O)C(C)C)NC(CC#C)(C)C(=O)NC1CC2C=CC1C2 c1(C(=O)OC)cc(=NC(=O)C2CCN(Cc3cc(Br)c(F)cc3O)CC2O)[nH][nH]1 c1(C(N2CCCC(N(C(=O)COC3CC3)CC)C2)=O)cc(F)c(N)cc1OC C(=O)(C1=CC2CCCCC12)NCC1(F)CCCN(C(CSCC=C)=O)C1 Cc1nc(C2CC2)nc(C)c1C(=O)NCCCNC(C1CN2CCCC2CO1)=O C1(C)(NC(CCc2c(C)ncs2)=O)CCCN(C(=O)CNC(c2cccs2)=O)C1 N1(C(c2ccc(CNC(c3ccc(CC)o3)=O)o2)=O)CCCC(F)(F)CC1 C#CCCN=C(NCC(C)OCC=C)N1CC(O)C(C)(C)C1 CC1CCN(CCc2cccs2)CC1NC(c1nc(Cl)sc1Cl)=O C1(CN(C)C(C2CCNC2=O)=O)COCCN1C(=O)C=Cc1cn(C)cn1 C(c1cccc(F)c1F)=CC(=O)NC1CCC(NC(c2c(C)scn2)=O)CC1 c1(NC(C)=O)ccc(C(N2CC3C(CN(C)C(c4occc4F)=O)C3C2)=O)cc1 CC1=C(C(=O)NCC2=CCN(C(c3ncc(C(F)(F)F)cc3O)=O)CC2)CCO1 C(=O)(C1=CCCOC1)NN(CCCCC1CCCN(C(CSC)=O)C1)C1CC1 CC1CC(NC(=O)CCC2CCN(C(=O)CCc3nc(O)n[nH]3)C2)CC(C)(C)C1 C(=O)(CCCN=c1[nH]c2c(c(=NCC(COC)CO)[nH]1)CCCC2)NC N1(C(C(CC)(C)CNC(=O)CC(COC)COC)=O)CCCOC(C)(C)C1 C1(NC(C2(C=C)CC2)=O)CCCOC1C1CCN(C(=O)C=CSC)CC1 CC(C)CCCCC(=O)N1CCCC(O)(CCNC(C2CC3(C2)CC(C)C3)=O)C1 c1(OC)cc(CC(N2CCOC(CNC(=O)C(C)(C)CO)C2)=O)ccc1O C(=O)(C(C)(C)CN(C(=O)CC(=O)N(C)C)C)NCc1n(C(C)C)ccn1 N1(C(NS(=NCC=C)(C)=O)=O)CC(OC(C)(C)C)C2CCCC12 Cc1nc(C(=O)NCC2CCCN2C(c2ncccc2O)=O)n(C)n1 C(=O)(C(C)(CO)NC(c1scnc1Cl)=O)N(C)CC1(C#N)CC1 N1(C(c2c(OCC=C)cccn2)=O)CCCC2CN(C(=O)C(C)(C)CC)CCC12 c1(OC)ccc(F)c(C(N2CC3CN(C(c4c(OC)cccc4I)=O)CC23)=O)c1 C(C)(C(C(=O)NC1C(c2csc(C)n2)C1(C)C)NC(=O)CC(C)(C)N(C)C)OC C=CCCC(C)(C)C(=O)NCCCC1CCCCN1C(c1[nH]c(C)nc1C)=O N1(C(C2C(C(=O)OC)C=C2)=O)CC2CC1C2NC(c1n[nH]c(C)c1Br)=O C1(CC(=O)N(C2(CC(=O)NCc3cccnc3)CC2)C)CCC(=O)N1C CC(CCCNC(=O)C(C)OCc1ccccc1)NC(c1csc(C2CC2)n1)=O C1(C(=O)NC(C=C)(C)C)CN(C(C2CC(OC3CC3)C2)=O)CC1F c1(CN(S(N(CCC)CC)(=O)=O)C)c[nH]c2c(Cl)cc(F)cc12 S(=O)(=O)(c1cnn2ccc(=NCCC(F)F)[nH]c12)NC1CC(C=C)C1 c1(NC(=O)Cc2ncccn2)ccc2c(c1)CN(C(=O)C1=CCCCO1)CC2 N1(C(C2N(CC)CC2)=O)CCC(C)(CC(=O)NCC(C2CC2)OC)C1 c1(C(c2c(NC(C3CCN3C3CC3)=O)ccc(F)c2)=O)c[nH]c2ncc(F)cc12 Cc1ccc(C(N2CCN(C(=O)CSC(C)(C)C)C3CC23)=O)c2c1CCCN2 c1(C(=O)NC2CCN(C(C=C(CC)C)=O)CC2CC)cc([N+](=O)[O-])ccc1O N1(C(C(C(C)(C)C)OC)=O)CC2CCN(C(C3(CO)COC3)=O)CC2C1 C1(N2CCN(C(=O)OC)CC2)CCN(C(c2ccc(CO)o2)=O)CCC1C C#Cc1ccccc1CC1CCC(C=Nc2ccccc2OCC)C1 CC(C)(CNC(c1ccc(C(F)F)o1)=O)CCNC(=O)C=CC1CC1 c1(C(N2CC3C(NC(C4CNC(=O)O4)=O)C3C2)=O)cc2cccc(Br)c2[nH]1 C(C(F)F)(C(C)(C)C)NC(CC1N(C(c2c(CC)nccc2)=O)CC(O)C1)=O C1(CNC(c2cc3ccccn3c2)=O)CCCC2CN(C(c3cncs3)=O)CC12 C1(F)(CNC(=O)CN2CCC(O)CC2)CCN(C(=O)C(=O)NCC(F)F)CC1 N1(C(C(C)(C)SC)=O)CCN(CC2CN(C(c3nsnc3O)=O)C2)CC1 N1(C(Cc2ccc(C)o2)=O)CCC2(CC1)CCN(C(C1CN(C)C(=O)N1)=O)CC2 N1(C(CCCCCCC)=O)CCOC2(C1)CN(C(=O)C(C)C(=O)OC)C2 C(C(C(=O)NCCN1C(=O)CNC1=O)C(C)(C)C)NC(c1n(C=C)ncc1)=O c1(C(=O)OCC)cc(C)nnc1N(C(C)CNC(=O)CN1CC(=O)NC1=O)C c1(OC)c(C)cc(C(=O)NCCC2CC(NC(C3CC(C)CO3)=O)C2)cc1C O=C(CCCn1ccnc1)NCC1(CNC(c2csc(C(=O)C3CC3)n2)=O)CC1 CC(Cc1ccccc1Cl)N=c1nc(N2CCC(F)CC2)c2c([nH]1)CCC(C)C2 CC(C)CC(C(=O)NC1CCCC(O)C1O)NC(c1nc[nH]n1)=O Cc1ccc(CC(N2CCC(N(C)C(c3n[nH]cc3Cl)=O)C2)=O)cc1C CS(=O)(=NC(=O)c1cc(Br)cc2c1OCCC2)C1CC(O)C1 Cc1cc(C(N2CC3CCC2CN3C(C2(C)CCC(C)C2)=O)=O)c(C)nc1C N1(C(c2c(O)ncc(C(C)C)c2)=O)C2CCC1CN(C(c1ncn(C)n1)=O)C2 Cc1cc(C(=O)NC2(CNC(c3[nH]c(O)nc3C)=O)CCC2)ccc1Cl Cc1ccc(NC(=O)NCCC2CC3C=CC2C3)c(-n2cc(Cl)cn2)n1 C=CCC(CC(=O)NC(C)CCF)NC(C1(C=C)CCCCC1)=O c1(C(CC(=O)NC(c2nccc(=N)[nH]2)C)N)cccc(F)c1 c1(N(CCOCC)C)nnc(C2COCCN2C)n1CC1CCCO1.C1CCOC1 CC(C)CC(C)C(=O)NC(C)(CNC(c1c[nH]cc(Br)c1=O)=O)C1CC1 C1(NC(CNC(CC(C)(C)C)=O)=O)CCCC12CCN(C(c1sccc1F)=O)C2 C=CC(CC)C(=O)N1CCC(C(=O)N(CC(O)C2CC2)C)(CO)C1 c1(NC(C(C)NC(CCC2CC(OC)C2)=O)=O)ccc2ccoc2c1 c1(CC(=O)NCCNC(c2c(CC)scn2)=O)ccc2c(c1)NC(=O)C2 N1(C(C2(C#C)CN(C(c3csnc3Cl)=O)C2)=O)CCOC(C)C1CO N1(C(c2cc(C)oc2)=O)CCC2CN(C(=O)Cc3c(O)ncnc3O)CCC2C1 C(=O)(C1=COCCO1)N1C(CN(C)C(C2(c3ccc(F)cn3)CC2)=O)CCC1 c1(C(N2C3(CNC(c4n(C)ncc4)=O)CCC2CC3)=O)c[nH]c2cccnc12 CC(C)C(CCNC(C1(C)CCOCC1)=O)NC(=O)C(C)NC(C)(C)C c1(C(C)NC(C(C)NC=O)=O)nocc1C(=O)NC1CC2CC2C1 c1(C(N2CC(CNC(COc3c(OC)cccc3)=O)C2)=O)cc(S(C)(=O)=O)co1 n1(C(C)C)nc(C2CC2)cc1NC(=O)CCCN(C)C c1(NCc2ccc(C)nc2Cl)ncccc1S(=O)(=O)NC1CC(C)CC(C)(C)C1 N1(C(CN(CCC)C)=O)CC2CCC1C(CNC(=O)Cc1ccccc1F)C2 C1(N(C(c2cnc(CC)s2)=O)C)CCCC(NC(=O)C(C)(C)NC(C)=O)C1 N1(C(C2(C#C)CCN(C(=O)C(C)C(C)(C)C)C2)=O)CC2CCCCC2C1C C1(CNC(C=CC=CCC)=O)COC(COC)C1.C1(=O)CCC2CC(C2)N1 c1(CC(=O)NCC(c2ccc(F)cc2)NC(c2c(C)nc[nH]2)=O)ccc(F)cc1 CC1=CC(C)=NS(=O)(=O)N1CC(=O)NC(C)CNC(c1cc2n(n1)CCC2)=O C1(NC(CC2N(CC)C(=O)CC2)=O)CN(C(c2ccc[nH]2)=O)C2(CCCCC2)C1 C1(CCC)CN(C(=O)C(N2CCNC2=O)C)CC1NC(c1cc(OC)n(C)n1)=O N1(C(C(C)OCC=C)=O)CC(n2cc(-c3ccc(F)cn3)nn2)CCC1(C)C C1(c2n[nH]c(=N)o2)C2CN(C3(C(=O)O)CCOC3)CC12 C=CC(O)C(=O)NC1CCCC1CNC(=O)CC1(O)CCCC1 c1(SC(N2CCC(Oc3cccc(C#N)c3)C2=O)COC)cccc2cc(C)oc12 CCCC(C)CC(=O)NCCCCN(CCCNC(=O)Cc1cccn1C)C O=C(N=c1ccn(C2CN(C(=O)CC3CCC3)C2)[nH]1)c1cc(F)c(Br)cc1F C1(C(N2C(CCCNC(C(C)S(C)(=O)=O)=O)CCCC2)=O)CC2(C1)CC(F)(F)C2 Cc1nn(CC(=O)NC2CN(C(C3CCC(C(N)=O)C3)=O)CC2(C)C)c(C)c1Cl C1(CNC(C(C)N(C)C)=O)CN(C(c2n[nH]cc2Cl)=O)C2COCC2O1 N1(C(C2(OC)CCCOC2)=O)Cc2[nH]nc(C(=O)N(C)CCF)c2C1 N1(C(Cc2cc(OCC)ncc2)=O)CCC2CCN(C(c3ccsc3C)=O)C2C1 C1(NC(C2CN(C(c3c(CC)nn(C)c3)=O)CC2C)=O)C(O)C2CCOC12 C(CCN=c1cc(C)nc(OC)[nH]1)N(C(C(C)OC)=O)C c1(C(N2CCC=CC2C(=O)OC)C(=O)NCC=C)ncccc1Cl N1(C(C=CCN(CC)CC)=O)Cc2[nH]nc(C(N3CCC(C)C3C)=O)c2C1 N1(C(CCC(C)OC)=O)CCN(C(c2cccnc2)=O)CC1CN(C)C C1(NC(C(C)(C)c2ccns2)=O)CN(C(C2CCC(C)CC2)=O)CCC1CO C1(N(CC(F)F)C(=O)OCC(C)O)C=CCN(C(=O)OC(C)(C)C)C1 C1(C(=O)NC(CC=C)(C)C)CCCN(C(C2(CO)CCCO2)=O)C1 C1(C(N(C)CCN(C)C)=O)(NC(=O)CC(=O)NCC#N)CC1(C)C C12(COC)CC(CNC(=O)CC(C)F)(CN1C(c1ccc(C)s1)=O)C2 c1(C(=O)NC2COCCN(C(CC(CC)(F)F)=O)C2)ccc([N+](=O)[O-])n1C C1(CC(N2CC(CC(=O)NC(c3ccccc3)C)C2)=O)NC(=O)NC1=O CC1CCN(C(=O)CC2CCN(NC(c3cc4occc4[nH]3)=O)C2)C(C(N)=O)C1 C(CC(C)C(=O)N1CCC(C(=O)N(CCC(N)=O)C)C1C)OC c1(C(N(C)CC2N(C(C(=O)NC(C)C)=O)CCCC2)=O)nc[nH]c2ncnc1-2 Cc1ccc(C(=O)NC2CC(C(=O)NC3CCCC(F)C3)C2)nc1 C(=O)(C(CCC(N)=O)N(C)C)NCC1N(C(Cn2c(C)csc2=O)=O)CCN(C)C1 c1(C(N2CCC(c3cn(-c4ccc(C#N)s4)nn3)CC2)=O)c(Br)ccnc1Cl N1(C(c2cncc(C=C)c2)=O)CCC(C(=O)NCc2ccccn2)C(C)(C)C1 C1(OC)(OC)CC(C)(C(N2CCCC(NC(C3CC(=O)N(C4CC4)C3)=O)C2)=O)C1 C(=O)(C(c1cccs1)=Cc1cccc(Cl)c1)NC1CCN(C(C(C)N(C)C)=O)C1 C1(NC(c2c(CC)ocn2)=O)CCN(C(=O)C(C2CCOC2)OC)CC1C N1(C(c2cncc(OC)n2)=O)CCOCC(C(=O)NCC2(CCO)CCCC2)C1 C1(CNC(CC2(CSC)CC2)=O)CCC(CNC(C2SCCS2)=O)CC1 N1(C(CCN(C(=O)Cc2cccs2)CC#C)=O)CC=CCC(C)(C)C1 C1(CNC(CCCOC)=O)CN(C(=O)Cc2cn(C(C)C)nn2)CC(C)(C)C1 C(=O)(CC1OCCc2sccc21)NC1C2(CC(NC(CCC(=C)C)=O)C2)C1 c1(OCC)c(CC(N2CCCC(CNC(C3CC(SC)C3)=O)C2)=O)cccc1Cl C(=O)(CCCC(=O)N1CC(NC(=O)CCn2ccnc2C)CC1C)OCC c1(SC)cscc1CNC(c1nnnn1CC(F)F)(C1CCOCC1)CF C1(CNC(c2cc(Cl)sc2Cl)=O)C2CCCC1N(C(=O)CC1CC=CC1)C2 c1(C(=O)NC(C)CNC(=O)CC2CCC(=O)C2)ccnc(C(F)F)c1 c1(C(N2C3C(NC(c4c(C)sc(O)n4)=O)CC(C3)C2)=O)ccc2c(c1)C(=O)NC2 Cc1sc(Cl)c(C(=O)NC2(CNC(=O)CC3CC(C)C3)CCOC2)c1C Cc1cc(O)c(F)cc1NC(C1CN(C(c2nnsc2C)=O)C2(CCC2)C1)=O c1(C(N2C(CNC(c3ccns3)=O)CC(F)C2)=O)cnc2c(c1)CNC2=O c1(N(CCNC(=O)C(c2ccccc2)F)CC)nccc(C(C)(C)C)n1 C1(NC(c2c(C)onc2C(F)(F)F)=O)CCC(C)N(C(C2C3CCCCC23)=O)C1 CCC(C)(C)C(C)CC(=O)NCC1C=CCN1C(=O)CSc1ccc(OC)cc1 c1(C(=O)NCCCCN(C(C(c2cnccn2)C)=O)C)ccc(F)c2ccsc12 CC1CC(C(=O)N(C)CC2CCCC2(C)C)CN(C(=O)CCc2ncccn2)C1 C1(CNC(C(C=CCCC)O)=O)CC12CCN(C(=O)C=C(C1CC1)C1CC1)CC2 Cc1ccc(C=CC(N2CC(CC(C)NC(=O)C(c3ccccc3)C)C2)=O)cc1 N1(c2n(C3C(C)COC3=O)nnn2)CCS(=O)(=O)N2CCOCC12 CC1=C(C(=O)NCC2(C)CCN(C(=O)C(c3ccccc3)F)C2)C(=O)OC1(C)C CCC(C)(O)C(=O)NC(C1CN(C(C2(c3cccc(Cl)c3)CCCCC2)=O)C1)C c1(NCC(=O)N(CCNC(c2c(CCC)nns2)=O)C2CC2)ccc(C)cc1 c1(C(N2CCC(C)(C(N3CCC(CO)C(F)C3)=O)C2)=O)nc2ccc(F)cn2n1 C#Cc1ccc(C(N2CC(CNC(=O)CC3CCC(=O)NC3=O)C(C)C2)=O)cc1 c1(CN(CCNC(C(CC)OCC)=O)CC)ccc(C(F)(F)F)cc1 CC#CCC(CO)NC(=O)CN(C(=O)C(C)CC1CC1)C1CCC1 Cc1c(N)ccc(C(N2CCCCC2CN(C)C(c2scnc2Cl)=O)=O)c1Cl c1(C(N2CC=C(CCNC(CCCCSC)=O)CC2)=O)cnn2ccc(C)cc12 C(N=C(NC1CCCCC1)N1CC(C)CC(C)C1)C1Cc2c(ccc(CC)c2)O1 CC1(C)CC(n2ccnc2-c2cccc(C(F)(F)F)n2)C(=O)N1 C1(NC(CCCc2onc(CC)n2)=O)CCN(CC2CCC(C)O2)C(C)C1 c1(CC(=O)NC(C2CC2NC(=O)CNC(=O)CC(C)(C)C)C)ccc(O)nc1 c1(CC)ccc(O)c(C(N2CC(C)(NC(=O)C(C)Oc3cccc(C)c3)C2)=O)c1 Cc1cc(N)ccc1C(N1CCC(CN(C(=O)CN2CCN(C)C(=O)C2)C)C1)=O c1(OC)nc(C(=O)NCC(C)CNC(C2COCC2C(F)F)=O)ncc1F c1(OC)nccc(=NC(=O)C2(C)CCN(Cc3ccc(Br)nc3Br)C2)[nH]1 C1(NC(C(CC)CCOC)=O)CC2CCC(C1)N2C(=O)C(c1ccccc1)=O c1(OC)cc(Cl)ccc1C(=O)NCCCN(C(=O)C(F)(F)CC1CC1)C1CC1 CC1CCN(C(=O)CCc2cccnc2)C1CNc1cc(O)ncn1 c1(OC)cc(C(=O)NCC2CC2CNC(c2ccc(Cl)nc2C)=O)ccc1C O=C1NC(=O)C(CC(=O)NC(Cc2ccoc2)C(=O)N2CC(c3ccncc3)C2)N1 C1(C)(CNC(C(CCC)NC(=O)C(C)OCCC(C)C)=O)CCCC(C)(C)C1 CCS(=O)(=O)C=CC(=O)N1CCC(OCCNC(=O)CC2=CCCCC2)C1 CCC(CC)CN=c1[nH]c(=NCC2(C)CC3(C2)CC(F)(F)C3)c2cccc(F)c2[nH]1 CCC(CCC(=O)NCC1CC(C)=NO1)NC(=O)CCCOC(C)(C)C C1(CC=C)(NC(=O)CN(C2CCSC2)C)CCCN(c2ncc(OC)c(C)n2)C1 c1(C(C(N2CC3(CC(NC(C(C=C=C)C)=O)C3)C2)=O)C)cccc2ccccc12 C1(COC)(NC(c2cc(O)n(C)n2)=O)CCCN(C(=O)CCCC(C)C)C1 C1(CC)CN(C(C23CCC(C2)C3(C)C)=O)CCC1NC(=O)CCCC1CC1 C(=O)(CC(C)CF)N(CCC)CCNC(=O)C(F)(F)c1csc(C)c1 C1(C(=O)NC2C(OC)CN(C(=O)C(C(C)C)N(C)C)C2)CC2CCC1C21CC1 Cc1ccc2c(c1)CC(C(=O)NCCCCCCN(C(=O)C(C)(C)C)C)S2 c1(C(N2CC(NC(Cc3c(C)noc3C)=O)C2)=O)ccc(F)c(F)c1O Cc1ncc(C(=O)NCC2CC3CCC2N3C(=O)Cc2ccccc2C)c(C)n1 c1(C(=O)NCCC(C(C)C)NC(=O)CC(O)C2CC2)nccc2occc12 c1(C(N(C2CCCN(C(=O)CCC(C)SC)CC2)CC)=O)cn2cc(C)sc2n1 C(=O)(C1=CCCCC1C)NC1CC2CC(NC(c3c[nH]cc(C)c3=O)=O)CC21 C1(C(=O)NCCS(CC)=O)CCCCN1C(=O)Cc1cncnc1 c1(C(=O)NC2CC(NC(C3CCOCC3)=O)C23CCC3)ccc2[nH]ccc2c1 C1(C(N(CC(=O)NCC)C)=O)CCCC(NC(=O)CCC=CC(C)C)CC1 c1(CC)ccc(C(=O)N(CCCCCCNC(C2(C#N)CCCO2)=O)C)cc1Cl C(=O)(CC(C)(C)C(F)F)N(C1CCCN(C(C2COC(=O)O2)=O)CC1)CC c1(C(C(=O)NC(C)CCNC(c2ccc(C(F)F)cc2)=O)O)ccc(F)c(Cl)c1 CCCCC(C)(CO)NC(c1ccc(C)c(C(=O)O)c1)=O C#CCC(C)(CC)C(=O)N1CCC(CNC(c2cccc(F)c2C)=O)C(F)(F)C1 c1(C(=O)NCC(CC)NC(=O)C(C)(C)C(N)=O)oc2c(Cl)cccc2c1C C(C)(C)(CCC(=O)NCCN(CC)CC)NN(CCC)CCN(C)C C1(NC(c2c(C)nc(O)cc2)=O)CC2CC(NC(C3C=CC=CC=C3)=O)CC2C1 Cc1ccc(C)c(C(=O)NCC2CC2NC(c2cnc(O)c(F)c2)=O)c1O C(CO)(C(C)(C)C)NC(c1nnnn1C(C)(C)C)CCOCC C1(NC(c2c(C)nc(O)[nH]2)=O)CN(C(C2CC2C)=O)C2(CCCC2)C1 Cc1cc(-c2nc(Cc3ccc(Cl)cc3)nn2CC2CCCOC2)nnc1O N1(C(C(=O)NCCN(CCOC)C)=O)CCCCNCC(F)(F)C1 C1(CC(N2CCCCC2C2(NC(=O)COC(F)(F)F)CC2)=O)(CC)CCOCC1 N1(C(C(CCSC)OC)=O)CC2CCN(C(c3sc(F)cc3Cl)=O)CC2C1 O=S(=O)(c1ccc(NC2CC2O)nc1)NC(c1cccc(F)c1)CC1CC(O)C1 S(=O)(=O)(c1cccs1)NC(CCSC)C(=O)Nc1cc(CS(C)(=O)=O)nn1C C(CC(C(=O)N1CCN(c2ccncc2C(F)(F)F)CC1)OC)OC N1(C(CCOC)=O)CC2(C1)C(NC(=O)Cn1cccc(C)c1=O)CCS2(=O)=O N1(CC)CCN(CC(=O)Nc2cccc(C(=O)O)c2)C(C)C1=O C1(NC(c2cnc(Cl)s2)=O)COCCN(C(=O)C(C2CCS(=O)(=O)CC2)O)C1 CC1OC2(CO)CC1(C(=O)NCCN(C)C(C1CCCN(CC(F)(F)F)C1)=O)C2 N1(C(C(C)O)=O)CCOCC1CN(C(=O)CSc1ccccn1)C c1(C(=O)NCCN(C(C2C(=C)C2)=O)CC)nnn(CCC)c1C(F)(F)F c1(C(=O)NC(CC)(CC)C(N)=O)n[nH]c2c1CN(C(=O)C(C(C)C)SC)C2 Cc1c(Cl)cnn1CC(=O)NC(C)CN(C(=O)Cc1sccc1Cl)C C1(C2CCN(C(c3cnn(CC)c3C)=O)CC2)(NC(CC(C=C)(C)C)=O)CCC1 C1(C(N(CCC#C)CCO)=O)CC(CCNC(=O)CCOC2CCCC2)C1 C(=O)(CS(=O)C(F)(F)F)N1CC(NC(CC(C)CCOC)=O)C1.C1CC1 C(=O)(CCCN=[N+]=[N-])NCCCC(=O)NC(C)CC1(O)CCC1 N1(C(C(C(C)(C)C)CO)=O)CCC2(CC1)CCN(C(c1csc3nnsc13)=O)C2 c1(CC)cnsc1C(=O)NC1COCC1n1cc(-c2ncc(CC)o2)nn1 C(=O)(C1=C(Cl)CCOC1)NCC1CCC(C)N(C(=O)CCc2ncc[nH]2)C1 CN1CCN(C)CC(C(N2CCCC2CCNC(C2(C)CC2(F)Cl)=O)=O)C1 C1(C(C)NC(c2coc(Br)n2)=O)CN(C(=O)C(C)OCc2ccccc2)CCO1 CCC(C(=O)NC1CC1NC(C1CC(O)C1)=O)Oc1ccccc1 c1(C(=O)NCC2(CN(C(C)C(=O)O)CC)CC2)c[nH]nc1-c1ccoc1 Cc1ccn2c(=O)c(C(=O)NCC3(NC(=O)C(N)=O)CCCCC3C)cnc2c1 CCS(=O)CC(=O)N(CC(O)CN(C)C(c1cc(Cl)ns1)=O)C N1(C(C(c2cc(C)sc2)(F)F)=O)C2CCC1CN(C(c1cc(O)cc(O)n1)=O)C2 N1(C(CCC(=O)OC)=O)CCC(NC(=O)Cc2ccc(Br)cc2I)C(F)C1 CCCCC(c1nnnn1CCSc1cccs1)NCCn1cc(Br)cn1 C1(C(N2CC3CC(NC(C4CC(O)(C#C)C4)=O)C3C2)=O)(CC)CCC(F)(F)CC1 C1(N(C(CCCC#C)=O)C)CC2CCC(C1)N2C(C1CCC(C)C1)=O CC1CCCCN1CCNC(=O)C(C)(C)NC(=O)CC(C)N(C)C c1(OC)cccc(C2CC(C)CN2C(c2ccsc2Br)=O)c1 N1(C(CCCCC=C)=O)CC(CNC(c2cnc(C)[nH]2)=O)CC12CCOCC2 N1(CCC(=O)N(CC(C)(C)NC(C(C2CCOC2)OC)=O)C)CCOCC1=O C1(C(=O)NC(CC#CC)C(=O)NC)CN(C(=O)C(CCC)N(C)C)CCC1(C)C c1(C(=O)NC2C(NC(COCC=C)=O)CCC2)cc(F)cc2nc[nH]c12 C(=O)(C1CCc2cccnc21)NCC1CC(NC(C=Cc2c(C)cccn2)=O)C1 CC(C)(F)CN=c1[nH]c2c(c(=NC3CN(c4ccncn4)C3)[nH]1)CCCCC2 CCC(C)(CCNC(=O)C(=Cc1cccnc1)F)NC(=O)C(O)CSC c1(OC)ccc2c(=NCCC3CCC3)[nH]c(=NCC(C)(C(C)C)C(C)C)[nH]c2c1 CC1(C)CC(CC(N2CCCC(C)(NC(c3cocn3)=O)C2)=O)C(=O)O1 C(=O)(C1=NN(CC)C(=O)CC1)NCC1(C)N(C(CCC=CC)=O)CCC1 n1(CC(=O)NC2CC(NC(=O)CCC3CCCC(O)C3)C2)ncc2ccccc12 C(=O)(CCC(=O)NN(C)C)N1CCCC(N(C(c2cc(OC)ns2)=O)CC)CC1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC(C(C)NC(c1ocnc1C1CC1)=O)C C1(CCNC(CN(S(CC)(=O)=O)C)=O)COCCN1C(=O)C(N1CCC(C)C1)=O c1(C(C)C)cc(C(=O)NCC(C)NC(c2ccncc2Cl)=O)cc(F)c1 C1(NC(C(C)(C)CF)=O)CC(F)CN(C(c2c[nH]nc2C2CCOC2)=O)C1 CS(=O)(=O)c1ccc(NC(=O)C(=O)Nc2ccc(C(N)=O)c(Cl)n2)cc1 C12(C(=O)NCCCN(C(=O)CC3CCCCC(=O)N3)C)CCC(CO)(CC1)CC2 C1(N(C)C)CN(C(C2CCC(NC(=O)Cc3ccsc3)CC2)=O)CCC1O C=CCCCC(C(=O)NCC(CC)N(C)C)NC(=O)C#CC(C)(C)C Cc1cc2ncc1S(=O)(=O)N2.C1(NCCN(C)CCO)CC=CCC1C(F)(F)F c1(C(N2CCCC2C(=O)NC(C)(C)C)C(=O)NC)cc(Cl)cc(Br)c1F c1(C(=O)OC)cc(COC)cc(S(=O)(=O)N2CCC(=Cc3cccnc3)CC2)c1 N1(CC(=O)NCCCCNC(c2nc(CC)oc2)=O)C(C)CCC1C C1(NC(c2c(-c3cn(CC)nc3)n[nH]c2)=O)CCC(CNC(=O)C(C)CF)CC1 CCC(C)(C(=O)NCC1CCN1C(c1cc(C2CC2)[nH]n1)=O)OC N1(C(N2C(c3onc(C)n3)CCC2)=O)CC(=O)Nc2cc(C(F)(F)F)ccc21 N1(C(c2c(C)noc2)=O)CCC(N(C(=O)Cc2cc(Cl)n(C)n2)C)C(C)C1 c1(C(N2CC(NC(C3CC(C)(F)C3)=O)C3(C2)CCC3)=O)cc(O)ccc1[N+](=O)[O-] c1(CC)ccoc1C(=O)N(C)CCOCCC(=O)NC(c1cnsc1)C C1(NC(Cc2cc(C)on2)=O)COCCC1NC(=O)C(C)c1ccco1 C1(C(=O)NCCc2scc(C)n2)CC2CCC(C1)N2C(C1C2CC3C(C2=O)C13)=O CCCS(=O)(=O)C(C)C(=O)NC1CCC12CN(C(=O)C=C(C)C1CCCCC1)C2 N1(C(C(C)(C)SC)=O)CCC(NC(c2oc(C(F)F)cc2C)=O)C(C)C1 c1(OC)ccc2oc(C(N3CCC(NC(C4(O)CCSC4)=O)C3)=O)c(C)c2c1 C(C(=O)NCC1(O)CN(C(C2(C)CCN(C(C)=O)C2)=O)C1)(C(C)C)SCC c1(NCC2(O)CCN(C(CC(=C)C)=O)CC2)ncnc2sc(C)c(C)c12 c1(CC)c(C(=O)N(CCNC(C2CC2c2cccnc2)=O)C(C)C)cnn1CC Cc1cc(C(F)(F)F)ccc1CC(N1CCC(NC(c2n[nH]c(C)c2C)=O)C1)=O c1(OCC)ccc(NC(=O)CCC2CCN(C(=O)C=CCO)C2)cn1 c1(C(=O)NC(C)CNC(=O)CCCCO)cncc(N=[N+]=[N-])c1 C1(CS(C)(=O)=O)CN(C(=O)CCCc2ccccn2)CCN1C(C1CC1(F)F)=O c1(-c2ccc(C(=O)NC)cc2)ccn2nc(C(=O)NC(CO)CO)cc2c1 n1(CC(=O)NC(C)(C)CC2CCCC2)cc(CNS(=O)(=O)C2CC2)nn1 CCCCC(F)C(=O)N1CCCC1CCC(=O)NCc1cccc(F)c1O N1(C(CC(CC)C)=O)CC(NC(c2ccoc2C(F)(F)F)=O)C(N=[N+]=[N-])C1 C#CCCCCCCCCCC(=O)NCCOC1CCN(C(=O)CC=C(Cl)Cl)C1 C1(C(=O)NC)CCN(C(C2CN(C(=O)CN3CSCC3=O)CCO2)=O)C1C N1(C(C(C)c2cccs2)=O)CCN(C(C2(F)CCCCC2)=O)CC2(C)CCCC12 C(C)(C(C(=O)NCc1ccc(C#N)cc1)C(C)C)NC(C(C1CCCC1)OC)=O C1(NC(CCC(C)=O)=O)CC(NC(=O)C=Cc2cnc[nH]2)C12CCC2 c1(C(CN2CCC(CC(c3cn(CC)nc3)=O)C2)OC)ccc(F)cc1 C1(C(C(=O)N(C2CCN(C(c3cnc[nH]c3=N)=O)C2)C)O)CCS(=O)(=O)CC1 N1(C(CN2CCCC(c3nnc(C)o3)C2)=O)CC(C)OC(C)C1 c1(CCC)nc(C)c(C(=O)NC(CNC(C23CC(C2)C(C(F)(F)F)O3)=O)CC)o1 c1(N2CC(c3ccc(C)o3)OCC2)nc(=NCCC2CC2)[nH]c2cccc(F)c12 N1(C(c2cncc(C)c2C)=O)CCC(NC(C2(F)CC=CC2)=O)C(CO)CC1 O=C(C#CC1CCCC1)NC1CCCCN(C(=O)CCc2nccs2)C1 c1(C(=O)NCCCN(C(c2c(C)n(CCO)nc2)=O)C(C)C)cnn2c1CCC2 Cc1cccc(CNC(C2CC3CC3N2Cc2nccn2C)=O)c1O N1(C(CC2(OC)CCC2)=O)CCC(F)(F)C(NC(=O)CCCc2ccccc2)C1 C1(C(=O)NC2CC(NC(CC)=O)C(O)C2)CCc2nc(C)nc(C(F)(F)F)c2C1 CCC(CC(=O)N(C)CCOCC(C)(C)C)NC(=O)C(C)C1CCCC1 Cc1nc(N(CCCCN(C(=O)CC(C)(O)C(F)(F)F)C)C)c2scc(C)c2n1 c1(C(C(=O)N(CCC)CCNC(=O)C(C)COC)N(C)C)c(F)cccc1Cl O=C1CC(NC(C2C3CC2N(C(C2CCCC4(CC4)C2)=O)C3)=O)CC(=O)N1 C1(C(=O)NC(C(=O)NCC(CC)(C)Cl)CO)C2CC3C(C2)C13 c1(C(=O)NC23CCCC(NC(C(C)OCCOC)=O)(C2)C3)cc2ccccn2n1 C(CC(=O)N1CC(C)CC1CC)(C(F)(F)F)NC(C(CC)C)=O Cc1nc(N)c(CC(=O)NCC(CNC(=O)CC2CC2(C)C)CO)c(O)n1 c1(CC)cnc(CNC(=O)CC=CCNC(=O)CSCCC#N)o1 N1(C(c2nccc(C)n2)=O)CCC(NC(=O)C(CCS(C)=O)N(C)C)C(C)(C)C1 C1(CNC(C2(CC)CC2)=O)CN(C(=O)C(F)C(F)(F)F)C2COCC2O1 N1(C(CCNC(=O)OC(C)(C)C)=O)CCN(C(=O)COC(F)F)C2CCC12 C1(NC2(c3n(C4(C)CC4)nnn3)CCSC2)CCCC(C(C)(C)C)C1 c1(CC(C(=O)N2CCC(OCCF)C2)NC(=O)CN2CCCC2)ccccc1Br C1(C2(O)CN(C(=O)C(CC(C)C)C3CC3)C2)(CNC(CNC(C(C)C)=O)=O)CC1 C(C(C)C(F)C(=O)NCc1ccn(C)n1)NC(c1cnc(C(C)C)o1)=O C(=O)(C(C)(C)CC(C)C)NCC1(OC)CCN(C(c2nocc2Cl)=O)C1 Cc1ccc2scc(CC(=O)N(C(C)CN(C(=O)CC3CC=CCC3)C)C)c2c1 c1(CC(=O)N(CCC(C(C)C)NC(c2cnn(C)c2)=O)C)c(F)cccc1F C1(C(=O)NC(CCNC(C2(CC)CCC2)=O)(C)C)CC(Cc2ccccc2)=NO1 C1(CC(=O)N(CC(C)NC(=O)Cc2ccc(Cl)nc2)C)CCC(C)CC1 Cc1c(F)ccc(Br)c1C(=O)NCC(F)CNC(c1nc(=N)cc[nH]1)=O C(=O)(C(C)(C)CCCc1ccccc1)N1CCC(NC(CN(C)CC)=O)(CO)C1 C(=O)(CCCCCC(=O)NCC1(C)CCN(C(=O)C=NOC)C1)OCC C(=O)(CCCCC(C)(C)C)N1CCC(CNC(CCC(C)C)=O)C(F)(F)C1 C1(NC(CCC(=O)NC)=O)CN(C(c2cc(C)cc(O)n2)=O)C2CCCC12 c1(N2CCCC(CC=C)(NC(=O)C(C)OCC3CC3)C2)ncnc2[nH]ccc12 c1(C(N2C(CNC(C(CCCC)N(C)C)=O)CC(OCC)C2)=O)nccc2occc12 N1(C(C2CC(C)C2)=O)CC2CCCC1C2CNC(c1c(Cl)n[nH]c1C1CC1)=O C1(CNC(c2csnn2)=O)CCCN1Cc1cc[nH]c1 N1(CCCCCCSC)C(=O)CN(CC23CCCC2C3(F)F)C1=O c1(CC(N2CCOCC(NC(CCC(N)=O)=O)C2)=O)c(F)cc(F)cc1F N(C1CN(C(c2ccc3c(c2)CC3)=O)Cc2ccccc21)C(CCOCC#C)=O C1(NC(=O)CSc2ccc(F)cc2)CCCCN(C(=O)C=CC(F)(F)F)CC1 Cc1cccc(C(N2CCOC(CN(C(=O)C(C)OCC3CC3)C)C2)=O)c1C C1(C(=O)NCCCOCCNC(=O)CCc2cn[nH]c2)C2CC3C(C2=O)C13 Cn1cc(C(=O)NC2CC(NC(=O)CCC3CCCC(=O)N3)CC2O)ncc1=O N1(C(c2ccc(Cl)c(Cl)c2)=O)CCN(C(C2CCc3nnnn3C2)=O)CC(O)C1 N1(C(c2ccn(CC)c2C)=O)CCN(C(c2ncncc2C)=O)C(COC)C1 N1(c2scc(C)n2)CCN(C(=O)CC(C)C2CC2)CC1 N1(Cc2cnc(C)s2)CC(NC(=O)C(C)Sc2ccccn2)C(C#N)C1 c1(C(=O)NCC(C)(CO)NC(=O)CC2C=CCCC2)ccc(F)cc1Br Cc1nc(C)c(C(N2CC(NC(=O)C3=CCCCO3)CC(F)C2)=O)c(C)n1 C(=O)(C(C(C)(C)C)NC(N)=O)NC(C1CCN(C(Cn2ccc(C)n2)=O)C1)C N1(C(CCCC(=O)OC)=O)CCC2C(CCCN2C(=O)CCC=C(C)C)C1 c1(OCC)ccc(OCC(=O)NC2CCC(NC(=O)CC(CC)OC)CC2)cc1 c1(C(=O)NCCC2(OC)CN(C(=O)Cc3cnnn3C)C2)nccc2ccsc12 CC(C)CC(CNC(=O)C(C)(O)C1CCC1)NC(=O)CSc1ccc(F)cc1 c1(-c2nc(-c3ccc(C)cc3)nn2C23CC(C2)C3)c(C)cccc1F c1(NCc2c(C)scc2)ccc(C(N2CCC(Br)C2)=O)cn1 CC1CCCC=C1C(=O)N(C)CC1CCCN(C(=O)C(F)(F)c2cscn2)C1 C1(CNC(C=CS(C)=O)=O)(NC(c2cnn(C3CC3(F)F)c2)=O)CCCCCC1 c1(C(=O)NCCC(=C)CNC(=O)Cc2ccc(Cl)c(F)c2)cc(O)nc(OC)n1 N1(C(c2snnc2C2CC2)=O)CCOC2(CCN(C(=O)CCC3CCC3)C2)C1 C1(C(N(CC(=O)NCC(O)CO)C)=O)CCCC(F)C1 C1(NC(C(C)OCC2CC2)=O)CN(C(=O)C(C2CCCO2)C2CC2)CC1C N1(C(Cn2ccc(C)n2)=O)CCCC(C)(NC(=O)CSCc2ccccc2C)C1 N1(C(C2C(CCC)C2)=O)CCC(NC(=O)C(=O)N(C)C)C(F)(F)CC1 c1(CC(=O)NC2CC(NC(c3cscc3F)=O)C2)cn2c(n1)CCCC2 C1(C(=O)NCC2CC2NC(C2C=CCS2)=O)CCC(F)(F)CC1 N1(CCOC(C)C2CC2)CCC(Cc2ncoc2C(F)(F)F)C1 CC1(C)C(NC(c2n[nH]cc2F)=O)CC1CNC(=O)CCNS(C)(=O)=O c1(C(C)C)cnn(C)c1C(=O)NC1CC(C)(NC(=O)C2CC2)C1 c1(Cc2nc(C(C)(C)NC(C)=O)sc2)cccc(S(=O)(=O)C(N)=O)c1 C#CCC(C(=O)NCC=C=C)NC(=O)C(F)OC(F)(F)F C(=O)(C1=NOC2(CCC2)C1)NC1CC(C)CN(C(c2cccn3nncc23)=O)C1 N1(C(CC2CC(OC)C2)=O)CC(C(=O)OC)CC2CCCCC12 C(=O)(CC(O)CC(C)(C)C)N1C(CCNC(C2(NC(C)=O)CCC2)=O)CCCC1 CC(CS(C)(=O)=O)C(=O)N1CCC(C)(NC(=O)C2=CC3CCCC23)CC1 CC1CC2(CCN(C(c3cncc(CO)c3)=O)CC2)CN1C(=O)C1=CCC1 C(CN=c1cc(Cl)nc(CC)[nH]1)(C1CC1)NC(Cc1c(CC)cccc1)=O N1(C(c2onc(C)n2)=O)CCC2(CC2C(=O)NCC2CN(C)C2)C1 N(C1CCCn2cnnc21)C(CC1(C)N(C(C2(CCN(C)C)CC2)=O)CC1)=O c1(C(=O)NCCC2CCN(C(=O)CCC(F)F)C2)ncc(Cl)cc1Cl c1(C(=O)NCC(CC)NC(c2sc(COC)nc2C)=O)noc2cc(F)ccc12 C12(NC(=O)C=CC3CC3)CCCN(C(C3(c4ccccc4)CC(O)C3)=O)CC1C2 C1(c2n(CC)nnn2)(NCc2n[nH]cc2Br)CCOC(CC(=O)OC)C1 Cc1ccc2nonc2c1C(=O)NC(C)CCNC(=O)CCCc1n[nH]c(=N)s1 CC(C(=O)N1CCC(C(=O)NC2C(=O)OCC2(C)C)O1)=C1CCC1 c1(C(N(CCNC(CCC)=O)CCOC)=O)cc(Cl)cnn1.CC1CCC1 c1(C(N(C2CCN(C(=O)C(F)F)C2)CC)=O)ccc(-c2ccc(Br)cc2)n1C CC1CN(C(=O)CS(=O)(=O)NC(C)(C)C)CC(C)C1NC(=O)Cn1nccn1 C1(C)(CC)NC(=O)N(CC(N2CC(NC(c3cccn4nncc34)=O)C2)=O)C1=O CC(C)(CCC#N)C(=O)N1CCCC2(NC(C3CCOC3)=O)CC2C1 C(=O)(C1CCCn2nccc21)NCC(C)N(C(C(C)Sc1ccccc1)=O)C C1(C(N2CCC(C3N(c4nnn(C)n4)CCC3)C2)=O)CCC(=C(F)F)CC1 c1(N2CC(C#C)OC(C)C2)ncnc2c1ncn2C(CCO)c1ccco1 C#Cc1ccc(C(=O)N(CC(C)O)CCNC(C2(C)CCCS2(=O)=O)=O)cc1Cl C1(N(C)C(=O)NC2CCN(S(C)(=O)=O)C2)CCCC(N)C1 c1(C(=O)NC2(CNC(C3C(OCC)C3)=O)CC2)cnc2ccccc2c1OC c1(C(N(C2CCN(C(C3(CO)CCCO3)=O)C2)CC)=O)ccc(OC2CC2)cc1 C1(F)(CNC(C2C(CC)C2)=O)CCCN(C(c2cnc3n2CCS3)=O)CC1 C1(C)(CC)CC(NC(=O)CCNC(C)=O)CN1C(c1ncnc(C)c1C)=O CC1CC(N(C(=O)CCCN(C)C(c2csc(Cl)c2)=O)C)CC(C)C1 N1(C(c2nc(N(C)C)oc2)=O)CC(F)(F)CC1CNC(C12CCC(F)(CC1)C2)=O CC(C)(CNC(c1conc1CNC(C1CCCC(=O)CC1)=O)=O)CCCO Cc1cccc(O)c1C(=O)NC(CCCNC(=O)C(C)(C)F)c1ccccc1 Cc1c(F)ccc(C(=O)NCCC2CCN(C(=O)Cc3cc[nH]n3)C2)c1N N1(C(c2c(C)nncc2)=O)CCC(C2CCN(C(C3(F)CC3C)=O)C2)CC1 c1(C(=O)NC(CNC(C(C)O)=O)CO)cnn(-c2ccccc2)c1F c1(C(N(C2CCN(C(c3nncn3CC)=O)C2)CCC)=O)ncc(Br)cn1 C1(C)(C(=O)NC2C3CC(NC(c4n(C)cnc4)=O)CC32)COC(C)(C)CO1 C(=O)(CCC(CC)CCCC)NC(CNC(CCC(=C)Cl)=O)C(C)C N1(C(C2CN(C(CCC(C)OC)=O)CC(C)O2)=O)CC2NC(=O)OC2C1 c1(CNC(C2CC2C(=O)NCc2ccnn2-c2ccccc2)=O)cccc(O)c1 N1(C(C(C)CF)=O)CCC(NC(=O)C(O)C2CCCC2)CC1 C(CC(CO)C(C)C)NC(C(C(C)C)NC(=O)C=CC1CCCN1C)=O N1(C(C)=O)CCOCC1C(N1CC(CNC(=O)CC2CCC2)C1)=O N(CP(C)(C)=O)(CC(=O)NC1CCCN(CC(=O)OS(C)(=O)=O)C1)CC C1(NC(C=C(C)C)=O)CC2CCC1(CNC(c1nc(C)n(-c3ccsc3)n1)=O)C2 C(=O)(NN1CCCC1C(=O)NCC1(C)CCC(=O)N1C)c1c(C)n(C)nn1 c1(C(=O)NC(CC)(CNC(=O)C(F)n2cccn2)CC)c[nH]c2cc(F)ccc12 C1(N(C(C=C(C)C)=O)C)CC2CCC(C1)N2C(=O)CCc1ccc(O)c(O)c1 C1(c2cn(CC3(O)CCN(C(c4sncc4C)=O)C3)nn2)(OC)CCCCC1 N1(C(c2cc(C(=O)OC)n(C)n2)C(=O)NC2CCCCC2)CCC2CCN(C)CC12 C(=O)(C1=CCCCO1)NC1CN(C(CCOc2ccc(C(N)=O)cc2)=O)C2C1C2 c1(C(=O)NCC(CC=C)NC(C2(C(C)C)CNC(=O)C2)=O)ccc([N+](=O)[O-])cn1 c1(CC)noc(CC)c1CC(=O)NCCC(C)(C)NC(=O)CSCc1cscn1 C(=O)(C#CC(C)(C)C)NC(C1CCCN1C(c1ccc(N2CCCC2)nc1)=O)C C1(C(c2nn[nH]n2)NC2(CCC(=O)OC)CCOC2)CCc2c[nH]nc2C1 c1(C(N2CCN(CC(N3CCC(C#C)CC3)=O)CC2)=O)cccc2c1CCC2 N1(C(n2ncc(C)c2N(C)C(=O)C2CC2)=O)CC2CCC(CSC)C2C1 C1(CC(=O)N(CC)Cc2cncn2C)CN(C(c2c[nH]nc2C)=O)C(C)(C)C1 N1(c2cc(OCC)ncn2)CCCOC(CNC(=O)CN2CC(=O)N(C)C2=O)C1 C(=O)(C1CCCn2c(Br)cnc21)N1CCCN(C(C(C(C)C)(C)O)=O)CC1 c1(OC)ccc2c(c1)C(Nc1ccc(S(C)(=O)=O)nc1)CCCS2 c1(C(=O)NC2(CC=C)CCN(C(=O)C(=Cc3c[nH]cn3)F)C2)ccn(O)c(=O)c1 C(=O)(C1=CCCC1(C)C)NC(CCCC)CNC(=O)CCc1nc(CSC)no1 N1(C(C(C)C)=O)CCN(C(C2(C)CC2)=O)CC1.c1(C2C(C=O)C2)ccc(F)cc1 CCC(CC(=O)NCC1CN(C(=O)C(C)C#N)C2(CCC2)C1)CC(C)C CCCC(CNC(=O)COCC(F)F)C(=O)NCc1cn(CCC)nn1 CC1(C)C2CCC1(C)C2C(N1CCN(C(=O)CCC2CCOC2)C(CF)C1)=O C1(NC(C(C)c2cccs2)=O)CCN(C(c2cc(CF)on2)=O)C1C1CC1 C1(O)(CCNC(C(C)CC2CCCO2)=O)CCN(C(c2ccoc2Cl)=O)CC1 Cn1ncc(C(=O)NC(C(=O)NC2CCN(C(N)=O)C2)C2CCCO2)n1 C#CC1CN(C(C2CCS(=O)(=O)C2)=O)CCN1C(=O)C(COC)N(C)C c1(C(N2CCC(CCCNC(CN(CCC)C)=O)CC2)=O)nc(O)nc(O)c1N c1(C(N2C(CN(C)C(c3ncccn3)=O)CCC2)=O)nccc(Cl)c1F c1(C(C2CCCN2C(c2ccc(Oc3ccccc3)s2)=O)=O)ccnc(Cl)c1F c1(CC(N2C(CN(C(C3(COCC)CC3)=O)C)CCC2)=O)cnn(C)c1C C1(C(=O)NCc2n(C)ccc2)CCC(NCC2CCC(O)CC2)CC1 c1(NC(c2n(CCOC)nnn2)C2CCCSC2)ccc(N(S(C)(=O)=O)C)cc1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCN(C(Cc2c(C)nn(C)c2Cl)=O)CC1 CC(C)(C(=O)N1CCC(C2CCCN2C(C2CCCC2)=O)C1)C(F)(F)F N1(c2n(Cc3c(Cl)cc(Cl)cc3)nnn2)CCc2nc[nH]c2C1c1ccc(Br)cc1 N1(C(C(C(C)C)(C)C)=O)C(CNC(=O)CN2CCNC(=O)C2)CC2COCC12 N1(C(c2c(CC)nc(C)[nH]2)=O)CCN(C(=O)CCCC(C)=O)C(C)C1 N1(C(c2c(C)n(C(C)C)nn2)=O)C2CCC1CN(C(c1c[nH]ccc1=N)=O)C2 C1(O)(CNC(C(Cc2ccccc2)NC(C)=O)=O)CCCN(C(=O)C(F)F)C1 C1(C(=O)NCC(C)CCCO)CCCN1NC(=O)C1(C#N)CCCC1 C1(C(=O)NCC(C)CC2CC2)COCCN(C(=O)C2=CCCC2C)C1 N1(CC(=O)N(C(=O)C(C)NC(c2ccc(Cl)cc2)=O)CC)CCN(C(C)(C)C)CC1 c1(CC)nn(C)cc1C(=O)NC1CCCC1NC(=O)CCC(=O)C1CC1 C1(NC(c2onc(CC)n2)=O)CN(C(=O)CCc2cncc(C)c2)CCC1C Cc1cc(C(=O)NC(C)(CO)C(=O)N2CC(F)(C#N)C2)oc1C N1(C(C(c2n(C)ccn2)(F)F)=O)CCOC(CNC(=O)CCN2CCCC2)C1 C(=O)(CCC(C)(F)F)N1CCC(C(N2CC(CSC)C2)=O)(CF)C1 c1(OC)cncc(C(=O)NC2CCC(CNC(C3CC4CCC3O4)=O)C2)c1 C1(C(=O)NCC2(C(=O)OC)CCC2)CC2CCC1N2C(=O)CC(C)C1CCCO1 C1(CCNC(C2(CO)CCCO2)=O)CCN(C(C23CC(CC(F)F)(C2)C3)=O)C1 c1(CCC(=O)NC2CN(C(=O)C3=CCCSC3)CCC2F)c[nH]c2ccccc12 N1(C(C(CC)CCOC)=O)CCCC2(C1)CN(C(=O)CCc1cccc(O)c1)C2 N1(C(C(CNC(c2n(CCC)ncc2)=O)C(C)C)=O)CCOc2ccccc21 c1(C(=O)NC2(CC)CCCN(C(=O)C(O)C(C)(C)C)C2)cc(Cl)ccc1[N+](=O)[O-] C=CC1CN(C(c2cc(C)ccc2OCC)=O)CC1NC(=O)C(C)(C)CO C1(NC(C(C)NS(CCC)(=O)=O)=O)(CNC(=O)C(C)O)CCOCC1 N1(C(CCc2ccc(C)o2)=O)CCC(C)C(NC(=O)CSc2n[nH]c(O)n2)C1 C1(CC(N2CCC(C)(NC(c3cnccn3)=O)CC2)=O)CCn2cncc2C1 N1(C(CC2(C(=O)OC)CCC2)=O)CCN(C(=O)C(C(C)(C)C)SC)C(CC2CC2)C1 C(CN=C(NCc1cc(C)on1)NCC(F)F)C1CC(CC)C1 C(=O)(C1=CC2(CCN(C(=O)C(=O)C(C)C)C2)C1)NC(CCCC)CC CC(C)CCC(O)C(=O)N1CCCCC(CNC(=O)CCc2ccc(Cl)nc2)C1 C1(O)(CC(=O)NCC(=O)N(C2CCCO2)C)CN(C(=O)COC(C)(C)CC)C1 N1(c2cccc(OC)c2)CCCC(NC(C2(C(C)C)CCCO2)=O)C1=O Cc1cc(C)c(C(=O)NCC2CC3CCC2N3C(=O)C2=CCC2)cc1Br c1(C(=O)NC2CC(CNC(C(C3CC3)SC)=O)C2)c(C)nc2sccn12 C1(NC(Cc2ncc(CC)[nH]2)=O)CCN(C(c2cc(C)[nH]n2)=O)CC1CO N1(C(CCC2C(C)(C)C2)=O)CCOC(CNC(c2ccoc2Br)=O)C1 C(=O)(C1CCCn2nccc21)N(CCNC(c1cc(OC)c(O)c(Br)c1)=O)C N12CCN(CC1)c1ccnc(n1)COC2=O.c1(CCNC(C)(C)C)cnc[nH]1 N1(C(c2oc(C)c(CO)c2)=O)CC(CNC(=O)C(F)C2CCOC2)CCC1C N1(C(CNC(CC)=O)=O)CCOCC(CNC(C2(C)CCOC(C)C2)=O)C1 N1(C(C(CC)SC)=O)CCCC(C2CCN(C(c3nc(C)ncc3Cl)=O)CC2)C1 CC1CCN(C(=O)C(c2cnccn2)C)CCN1C(c1ccc(=O)oc1)=O c1(C(N2CC(NC(COC)=O)C(O)C2)=O)c(Cl)ccc(F)c1C c1(OCC=C)ccc(CNc2cccc(N3CCOCC3=O)c2)cc1Cl C1(NC(CN2CCN(C)CC2)=O)COC2C(NC(c3ccc(Cl)o3)=O)COC12 C1(C(=O)CC2(C(N(CC)Cc3ccc(F)cc3)=O)CC2(F)F)CC(C(C)C)=NO1 c1(OC)nc(Cl)c(C(N2CC(NC(C3CC(F)C3)=O)C(C)C2)=O)s1 C12(CNC(CNC(CC(C)C)=O)=O)CCCC1N(C(=O)Cc1ccsc1)CCC2 Cc1ccc2sc(CN(C3CCN(C(=O)CCOc4ccccc4)C3)C)nc2c1 CCC(F)C(=O)NCC(O)CN(C)C(c1cnn(C(F)(F)F)c1)=O C1(C(N(C)CC2N(C(C(CC)n3cccn3)=O)CCCC2)=O)CCCC(C)(C)C1 c1(COC)sccc1C(N1CC(C(C)NC(C2CN(CC(F)(F)F)C2)=O)C1)=O C1(C(N2CC(O)(CNC(CNS(CC)(=O)=O)=O)C2)=O)CC2CCC1C2 O=S(=O)(c1ccc2c(Cl)ccc(Cl)c2c1)NC1C2Cc3c(F)cccc3C12 C=C1CC2(C1)CC(C(N1CCOCC(NC(=O)C(c3ccc(C)s3)C)C1)=O)C2 CC1(C)CCCN(C(c2cc(C(N)=O)[nH]n2)=O)C1C(=O)Nc1cnc(Cl)nc1 C1(C(=O)NCc2oc(C(=O)NCc3c(C)ccs3)c(C)n2)CC(C2CC2)=NO1 C1(CNC(C(C)=C(CC)C)=O)CN(C(=O)C=CCN(C)C)C2(CCOCC2)C1 c1(C(N2CC3(CN(C(C(C(COC)C)C)=O)C3)C2)=O)ccc2ccncc2n1 c1(C(N(C(CN(C(C(CC)=CC)=O)C)C)C)=O)ccnc(N2CCN(C)CC2)n1 c1(C(=O)NC(CC)(C)C(N)=O)nc(C)c(C)cc1N C1(CNC(CSCCCC)=O)CC12CCN(C(c1ccsc1CC)=O)CC2 Nc1c(CNC(C2CCN(c3ccc(F)cc3F)CC2)=O)cccc1O c1(NC(c2c(C(C)NC(c3c(C(C)C)onc3)=O)noc2)=O)cccn(C)c1=O N1(C(CN(CCCCCC)C)=O)CCC2CCN(C(=O)Cc3nc(C)cs3)CC12 CC(CC(C)C(F)F)NC(=O)C(C1CC1)NC(=O)CCC(=O)C1CC1 C(c1ncccc1C)=CC(=O)NC1CC(CNC(c2c(CC)cco2)=O)C1 c1(NC(C2CN(C(CNC(CCC(C)C)=O)=O)CC2C)=O)ccc(F)cc1Cl c1(C(N(CC(CNC(Cc2cc(C)on2)=O)(C)C)C)=O)cccc([N+](=O)[O-])c1Cl N1(C(C(c2ccc(F)cc2)CC)=O)CCC(NC(=O)Nc2cnncc2C)CC1 N1(C(CCC(C)OC)=O)CCCCC(C(=O)NC(CO)CCC2CC2)C1 N1(C(CCC)=O)CCC2(CCCCC2NC(=O)CN(C)CCO)C1 O=C(CCC(F)(F)F)NCCCCC1(NC(=O)COC2CCCO2)CC1 c1(C(=O)NC(CC)C(=O)NCC#CC(F)(F)F)cc(C)sc1N c1(CC(=O)NC2C(NC(C3C(CN(C)C)C3)=O)C2)cccc(OC(F)(F)F)c1 c1(C(=O)NCCC2CN(C(C(C)(C)C3CCCO3)=O)C2)ccc(N)cc1Cl c1(-c2ccn(CCCC3(F)CCN(C(=O)OC(C)(C)C)C3)n2)cc(F)ccc1F CCC(C#N)C(=O)N1CC(O)(CCNC(=O)C2CC2)C1 c1(OCCC)cccc(C(=O)NCC2(O)CCN(C(=O)Cn3ccc(C)n3)C2)c1 c1(C(N(CCCCNC(C=C(C)C)=O)C)=O)sc2cccnc2c1Cl C(=O)(CCC(N)C(=O)O)N1CCCC(CNC(Cc2c(CC)noc2CC)=O)C1 C1(C)(C(=O)NC(c2ccccc2)C(C)NC(c2ccc(C(C)=O)o2)=O)CCOCC1 C#CCCCCCCC(=O)N1CCC(C(N2CCC(OC)C2C2CC2)=O)C1CC c1(OC)cc(C(N2CC(NC(=O)CCN3C(=O)CCC3=O)C(O)C2)=O)nc(C)c1 c1(C(=O)NC(CC)CN(C)C(C23CCCC2(C(N)=O)C3)=O)ccc(O)c(C)c1C c1(C(=O)NCC2(F)CC(NC(C(C)n3cccc3)=O)C2)ccc2c(c1)nnn2C c1(CC)cc(NC(c2nnnn2C2CCC2)(C)CC2CCOC2)ccc1C c1(OC)cc(C(N2CC(NC(c3nc(=N)cc[nH]3)=O)CCC2C)=O)cc(C)n1 C1(CNc2ccnn2CC(F)F)CNCC1(F)CO.O=C(C(=O)C1CC1)NCC1CC1 c1(N(C)C(c2ccc(CCF)cc2)=O)cc2cc(Br)ccc2s1 C1(NC(C(Cn2ccc(C)n2)C)=O)CCN(C(c2cc(Br)no2)=O)CC1O C(=O)(CC(C)(C)CC(F)(F)F)NCC12CC(NC(C=CC(C)(C)SC)=O)(C1)C2 C1(C(=O)NC(C#C)CC)CCN(C(=O)Cc2cccc(O)c2)C(C)(C)C1 N1(C(C(CNC(C2(CCOC)CC2)=O)O)=O)CC(C)(C)C1C(N)=O Cc1ccc(NC(C2(NC(=O)C(c3ccnn3C)C)CCN(C)C2)=O)cn1 C1(NC(C2C(C)C2)=O)CC2(C1)CC2NC(=O)CCSc1cccc(Cl)c1 c1(C(N2CC(C)CC(NC(c3c(CC)nc(C)[nH]3)=O)C2)=O)ccn2c1CCCC2 N1(C(Cn2ccc(C)n2)=O)CCC2(CC1)CCN(C(C1CCCC1C)=O)C2 n1(CC)ncc2c(-c3ccc(CN(CC(=O)OC)C)cc3)ncnc12 c1(C(=O)O)sc2ccccc2c1S(=O)(=O)NC(C1CCC2(CC2)C1)=O c1(C(C)OCC)nc(CC(=O)NCC(O)CNC(=O)Cn2cn[nH]c2=N)cs1 N1(C(c2n(C)ncc2C#N)=O)CC2CCCC(NC(=O)CC3(O)CCOC3)C2C1 C12(C(=O)NC(C3CCCCC3)C#C)CC(CO1)N(C(c1ccc(CO)s1)=O)C2 Cc1ccc(CC(=O)N(C)CCN(C(=O)C=Cc2nc(C)co2)C)cc1 N1(C(c2c(C)cccc2)=O)CC(NC(=O)C=CC(C)C)C(C2CC2)C1 C1(CC(=O)NCCCCCNC(=O)CN2CCCNC2=O)CC2CCC1CC2 N1(C(c2[nH]c(=NC)sc2)=O)CC2CCC(C1)N2C(=O)C=CC1CCCC1 C1(CCN(C)C)CN(CC2(n3cc(Br)nn3)CC2)CCCO1 N#CC1(CNC(=O)C(O)CCCNC(C2CC2C#N)=O)CCCCC1 Cc1cc(C)n(CC(N2CCCN(C(=O)CCC(N)=O)C(C)C2)=O)c(=O)n1 C=CC(C)(O)C(=O)N1CC2CC2(NC(=O)C=CC(CC)=CC)C1 Cc1ccc(NC(C2CCCN(C(=O)Cn3cccnc3=O)C2C)=O)cc1C CS(=O)CCC(=O)NC(C1CCCC1)CNC(=O)C=Cc1cc(C(N)=O)co1 CCCCCCCNC(=O)COC1CC(NC(=O)C(O)CC2CCCC2)C1 c1(C(=O)NC)ccc(Cl)c(NCc2cn(C)nc2C(F)(F)F)c1 CCC(C)C(CNC(=O)COCCNC(=O)CNC(C)=O)OC C1(N(C(CN(CCC)C)=O)C)CN(C(=O)CNC(=O)NCC2CC2)C1 c1(C(=O)NCCC(C)N(C)C(c2cc(Cl)on2)=O)ccncc1F c1(C(N2CC(O)(CNC(CCc3c(C)n[nH]c3C)=O)C2)=O)ncnc2c1CCC2 C1(NC(c2ccc(C)c(C)n2)=O)CN(C(=O)C(C)Cc2ccco2)CC(F)(F)C1 N1(C(CN(C)CC)=O)CCOC2(CCC(NC(c3cc(O)ccc3C)=O)CC2)C1 N1(C2C(NC(C3C(c4c(C)ccs4)C3)=O)CCC2)CCN(C(=O)C=CBr)CC1 C1(F)(C(=O)NC(C)C(=O)NC(C)(C)C)CCN(C(C2CCC(=O)N2C)=O)C1 N1(C(CC(=O)NCC)=O)CCN(C(C23CC(CC(C)O2)C3)=O)CC1CCO C1(NC(C2C(C)CCO2)=O)CN(C(=O)CC2(C(F)(F)F)CCC2)CC1O CC(C(=O)NCC(C(=O)N1CCC(CC(C)(C)C)C1)N(C)C)C(C)(C)C c1(CNC(C(CC)N(C)C)=O)cccc(C2CCC2)c1 N1(c2cc(NCC3(Br)CC3(F)F)nc(C)n2)CCCNC(=O)C(F)(F)C1 c1(NC(C(C(C)(C)C)NC(C2=C(C)CC2)=O)=O)ccc2c(c1)OCC2 c1(C(=O)NCCC(C)N(C(C(CC)n2cccn2)=O)C)cc(C)nn1C c1(CCC)cc(C(=O)NCC(C)(C)CNC(=O)CC(C)n2cccn2)[nH]n1 c1(C(=O)NCCN(C(c2nc(C)n(C)c2)=O)C2CC2)cc2c(C)nn(C)c2s1 N1(C(CC(C(C)C)C)=O)CC2CC3CC2C1C3NC(C1CC=CCC1)=O c1(C(=O)NC(CC(C)C)CNC(C2(F)CCCN(C)C2)=O)cncc2c[nH]nc12 N1(C(c2c(C)nc(CC)o2)=O)CC(N(C)C(C2CC2c2ccsc2)=O)C(C)(C)C1 C1(C2CCOCC2)(C(N(CC(CC)NC(=O)CCCNC(C)=O)C)=O)CC1(F)F n1(CC(N2CC(N3CCN(C(C=C=C(C)C)=O)CC3)C2)=O)cc(F)ccc1=O C(C(C)(C)C#CC(=O)NC1CCCN(CC)C1)NC(c1c(CC)non1)=O c1(CC(=O)NC2C3CN(C(C(C)=C4CC4)=O)C(C3)CC2)cccc2c1OCCO2 C1(NC(C2(C)CCC2)=O)COC2(CCCN(C(C3CC(F)(F)C3)=O)C2)C1 C1(NC(Cc2n(C)ncc2)=O)CCCCC1NC(=O)Cc1cnc[nH]1 C=CCC(C(=O)NCC1CC2CCC2C1)NC(c1ccc(OC)s1)=O C1(CC(NOCC2CC(=C)C2)=O)CCCCN1C(=O)C(n1ccnc1C)C N1(C(C2C(CC)OCC2)=O)CCC(CCNC(=O)C(F)(F)c2cnn(C)c2)CC1 C1(C(N(C2CCCN(C(=O)CC3(CO)CCC3)CC2)C)=O)CC12CCOCC2 C1(NC(CS(=O)(=O)N(CC)CC)=O)CCN(C(=O)Cn2ncnn2)C12CCCC2 C1(CNC(=O)Cc2cccnc2)COCCN(C(c2cn3c(n2)SCC3)=O)C1 c1(CC)cnc(N(C2CCNCC2F)C(=O)Cc2ccccc2Br)nc1 O=C1CCC2(C(=O)NCCNC(c3ccc4occc4n3)=O)CCCCC2N1 C(c1ccc(Cl)cc1)=CC(N1CCC(F)(Cc2ccc(Cl)cc2)CC1)=O C1(OC)CS(=O)(=O)CC1N=c1[nH]c(=NCCC(C)(C)CC)[nH]c2c1CCCC2 C(=O)(C(C(C)(C)C)N(C)C)N1CC2C(CNC(c3c(C)ccs3)=O)(C2)C1 Nc1c(C(=O)NCC(O)CNC(c2cnn3cnnc3c2)=O)ccc(Br)c1F CC(C(C)(C)C(=O)NC1(C2CC2)CC1)NC(c1cnc2n1CCC2)=O C(=O)(CC(C)(C)CNC(c1ccc[n+]([O-])c1)=O)NCC(C)N(C)C1CC1 N12CC3(CO)CC1(C3)C2=O.c1(CN(CC=C)CC=C)cn(CC(=O)O)nn1.C(C)(=O)OC n1(CN(c2ccccc2)C)cncc1CC1CN(C(=O)CCNC(=O)CO)C1 c1(-c2cn(C(C(=O)NCC(C)OCC=C)C)nn2)cc(OC)ccc1Br Cn1nc(CN(C2CCCC2)Cc2conc2C2CC2)c2c1CCSC2 C(C1CC1)(C1CC1)=CC(=O)NC(C1CCOC1)CNC(=O)CCc1cccs1 C12C3CCC(C3)N1C(=O)C(C)(C)CNC2=O.C1(OC)(CO)CC1 Cn1c(=O)n2c3c1CCN(C3)C(=O)N1CCN(C2)CC1.c1ncc[nH]1.C(C)(C)C N1(CC(=O)NCCOCCNC(c2c(CCC)n(C)nn2)=O)CCN(C)C(=O)C1 N1(C(Cc2c(C)n(C)cn2)=O)CC2COCC2(C(=O)NOCCCC2CC2)C1 N1(C(C2CCC(C)N2C(=O)OC(C)(C)C)=O)CC(CCCCl)C2(COC2)C1 N1(C(Cc2cc(C)no2)=O)CCC(F)(CC(=O)Nc2cnc(Cl)c(C)c2)CC1 N1(C(C(=O)N(C2CCN(C(c3cc(OC)n[nH]3)=O)C2)CCC)C)CCC(O)CC1 CCCC(CC)C(=O)N1CCC(CNC(C2(C(F)F)CCCC2)=O)C(O)C1 CC1(C(=O)NCCC2COCCN2C(c2nnc(C(F)(F)F)s2)=O)CCOCC1 C1(CC(=O)NC(C(C)C)CNC(=O)CSCCN(C)C)CCC(=O)NC1 N1(C(=O)NC(c2ccc(OCC(=O)NC)cc2)CC)CC(C(=O)NC)C(F)(F)C1 C12(CC(=O)NCCC(C)N(C(=O)CC3C=CCC3)C)CCC(CC1)C2 c1(C(=O)NCCNC(C2CC=CCO2)=O)nc(-c2ccccc2)oc1C1CC1 C1(C(=O)NCC2CCC(NC(CC(=C)C)=O)CC2)CCn2c(C)nnc2C1 N1(C(CC(=O)OC)=O)CCC2CCN(C(C3CC(=O)N(OC)C3)=O)C2C1 C1(CNC(=O)C(F)=CCCF)CCCC12CCN(C(C1(O)CCCCC1)=O)CC2 c1(C(=O)NC(CC)(CNC(C2CC2(Cl)Cl)=O)CC)noc2c1COCC2 N1(C(c2ccc(=N)[nH]n2)=O)CC(C(=O)NCC2CCCC(CO)C2)C(F)(F)C1 CC1(NC(=O)C(CCC2CC2)NC(=O)CCc2nncs2)CC2CCC1C2 C(N=c1nc2scnc2c(NC2CCCC2)[nH]1)C1CN(CCC2=COCCO2)C1 N1(C(CCSCCC)=O)CC2CCOC2(CNC(c2cn(C)nc2O)=O)C1 C1(CC(=O)NCCCCN(C)C(c2cn(CC3CCOC3)nn2)=O)COC2(CCC2)C1 C1(NC(c2cc(Cl)sc2Cl)=O)CN(C(=O)CCN2CCC(F)C2)CCC1F C(=O)(C(F)C(C)CNC(C1(CC)CCOCC1)=O)N(CC#CC)C c1(-n2cc(C3C(N(C)C)CN(C(C4(CC)CC4)=O)C3)nn2)nnc2ccccn12 C1(NC(C(C)C2(O)CCC2)=O)CC(C(=O)NCc2ncc(CO)[nH]2)CC1O c1(C(N(CCC(C)NC(=O)CC2COCCO2)C)=O)cnn(C(C)C)c1F c1(C(N2C(CNC(=O)CCn3cc(Cl)cn3)CC2)=O)cc(Br)sc1Cl c1(NC(C2CC3(CC(OC)C3)C2)=O)ncnc2c1CCC2 c1(C(=O)NCC(CO)NC(=O)C(c2ccccc2)=O)ccccc1C(F)F CCCCCC(C)(C)C(=O)NC1CS(=O)(=O)CC1NC(=O)Cc1ccc(C)cc1 C#CCCN=C(NCC1(C2CC2)CC1)NCC(C)(O)CC C(=O)(CCC1=NNC(=O)CC1)NC1CC(NC(c2c(C)ncnc2)=O)C(O)C1 C1(CC)CN(C)CCCN1C(=O)CCCCCNC(=O)C=CCCC(C)C c1(-c2c(OC)cncc2)ccn2cc(C(=O)Nc3cnc[nH]3)nc2c1 CC(=NO)C1CC(NC(=O)NC2(C)CCN(C(=O)OC(C)(C)C)CC2)C1(C)C Cc1cc(=NCC(C)CNC(=O)Cc2[nH]cnc2C)[nH]c(C(C)(C)C)n1 C1(NC(=O)CCn2cccn2)CCOCC1NC(c1nccc(C(F)(F)F)n1)=O CC1=CCSC1C(N1CCC(OCC(=O)NC2CC(F)(F)C2)C1)=O c1(CC)cccc(NC(=O)CONC(=O)Cc2ccon2)n1 CC(C)CC(C)CC(C)C(=O)NCC1CC(C)N(C(=O)C(C2CC(F)(F)C2)O)C1 c1(CC)ccc(C(=O)NC2CCN(C(=O)CNc3cnn(C)c3)C2(C)C)c(F)c1 CCC(CC)(CC)C(=O)N1CCCC(C)(NC(=O)C(n2ccnc2C)C)C1 CCC(C)C(CC(=O)NCCCCC1CC1C)NC(c1cocn1)=O C1(C(=O)NC(CC)(C)CC)Cc2cccc(OC)c2O1 C1(C)(NC(C(CC)C)=O)CCN(C(=O)CCCN(C)C(C)=O)C1 N1(C(CN(C)CCO)=O)CCOC2(CCN(C(C3CCC(F)(F)C3)=O)C2)C1 C1(O)(C(=O)NC2C(CNC(c3coc(C(F)F)n3)=O)CCC2)CCSCC1 N1(Cc2ccc(C(=O)OC)o2)CCC(NC(=O)CSc2ccncc2)C12CC2 N1(C(C(C)Oc2cccc(F)c2)=O)CCCCC(NC(c2nnc(S)n2C)=O)C1 c1(C(N2CCN(C(C(CC)O)=O)CC2CCOC)=O)n[nH]c2c1COCC2 N1(C(CC=CC(=O)NCCC)=O)CC2CC2(C(=O)O)C1 C1(N(C)C)Cc2ccccc2C1NC(=O)CCCOc1cc(F)cc(F)c1 c1(C(c2nnnn2C)NC2CCCC2)ccccc1C(=O)NC.CCS CC(C)C(CCC(=O)NCC1CC2(C1)CC(O)C2)NC(C1COCCN1C)=O c1(SC)ccc(CN2CCCCC2C(=O)Nc2ccc(C(=O)OC)cc2)cc1 C1(NC(C(C(CC)C)N(C)C(c2sccc2C)=O)=O)CCCCC12CCC2 c1(CCN(C)CC)cn(C2CCC(C(=O)NCc3ncoc3C(C)(C)C)C2)nn1 N1(C(Cc2c(C)n[nH]c2C)=O)CCCCCC1CNC(C1COCCN1C=O)=O N1(C(C2CCN(C(=O)CC3CCOCC3)CC2F)=O)CC(F)(F)C(F)(F)C1 c1(C(=O)NCC(CC(=O)NC(C2CCCC2)C)OC)ncc(F)cc1F c1(CC(=O)NC(C(CO)NC(C(CC)n2ccnc2)=O)C)ccc2c(c1)CCO2 C1(NC(=O)C=Cc2ccc[nH]2)CCC(NC(c2ccncc2C2CC2)=O)CC1 c1(OCC)ccc(NC(=O)C(N2CC(O)C(O)C2)=O)cc1S(N)(=O)=O c1(C(N2CCC3CN(C(c4[nH]c(=N)sc4)=O)C3C2)=O)cccc2nc(O)ccc12 C(=O)(CC1=NNC(=O)C1)N(C1(C(=O)NC2(C)CCN(C(C)=O)C2)CC1)C1CC1 C1(CNC(C(CCC)NC(=O)CCc2ccncn2)=O)CCOCC1(C)C c1(CCC)nc(C)c(C(=O)NCCN(CCC)C(C2CC2c2cccs2)=O)s1 c1(CC(N)C(=O)NC23CCCCC(F)(C2)C3)ccc([N+](=O)[O-])cc1Cl c1(C(=O)Nc2ccc(CNc3c(C(N)=O)cncc3)cc2)scc2c1OCCO2 Cc1cc(N(C)C)ccc1C(N1CCOCC1c1cn(CCO)nn1)=O c1(COCC)nc(N(C)CCNC(C2CC(Oc3ccccc3)C2)=O)cc(Cl)n1 c1(C(=O)NC(C2N(C(C3C(C=C)CC3)=O)CCC2)C)cc(C)c(Br)cn1 N1(C(CC2(C(=O)NCC(O)CCC3CC3)CC2)=O)C2CCC1CCC2.CN(C)C Cc1cc(C(=O)NCCC2(O)CCCN(C(=O)COC(F)F)C2)c2occc2c1 C12(C(=O)NCC3(NC(C4(O)CCCC4)=O)CCCC3)CCC(O1)c1ccccc12 C(CCCC(=O)NC(C)CCN(C)C(c1cccc(NC(=O)OC)c1)=O)OC c1(C(=O)O)ccc(Br)c(CNC2C=CS(=O)(=O)C2)c1F C(=O)(C(C(C)(C)C)NC(c1cnns1)=O)NC(C)CC1CCCC1 C(=O)(CC(CC)C(C)C)N1CCN(C(CCCC)=O)CC1CF N1(C(CCC#C)=O)CCC(C)(C)C1C(=O)NCCN1CCCCC1 C1(CCC(N2CCCC2Cc2cn(C3CC4CC4C3)nn2)=O)C2CCCCC12 Cc1cc(C(N2CC3CC3(C(=O)Nc3cc(Br)nc(Br)c3)C2)=O)cc(C#N)c1 N1(C(CSCCC)=O)CCCC2C(NC(=O)C(N3CCSCC3)C)C(C)(C)C12 C(=O)(CS(=O)(=O)C(C)(C)C)NC1C(CNC(C(c2ccc(OC)cc2)(F)F)=O)C1 N1(C(c2ccc(SC)o2)=O)CCC(O)C1C(=O)NC1(C)CCCC1C C=Cn1nncc1C(=O)N(C1CCN(C(c2ccc(C(C)=O)cn2)=O)CC1)C c1(CN(C(C(C)C)CO)Cc2ccccc2)cc(Br)n(C)n1 N1(C(c2cnc(C(C)C)o2)=O)CC2CN(C(=O)CSc3ccccn3)CC2(C)C1 C(CC(O)CNC(C1CNC(=O)N1)=O)NC(=O)Cc1cc[nH]n1 c1(-c2onc(C3(OC)CCCC3)n2)coc2c(F)cc(F)cc12 C(C(CC(C)C)C(=O)NC)c1nc(-c2cccnc2-n2c(C)nc(Br)n2)nn1C C1(O)(CNC(C2(CC#C)CCOC2)=O)CCCN(C(c2nc(Cl)sc2Cl)=O)C1 C(=O)(C1=CCCS1)NC1C(NC(C=CC(C)NC(=O)OC(C)(C)C)=O)CCC1 N1(C(C(CC[S+](C)C)O)=O)CC2(CCCN(C(=O)CC3CC4(CC4)C3)C2)C1 Cc1cc(C(=O)NCC2CCN(C(c3ncoc3C)=O)C2)ncc1F c1(OC)ccc(Cl)c(C(=O)NC2CCCN(C(=O)Cc3ccc(Br)cc3)CC2)c1 Cc1cc(Br)c(NC(C2CC3(C2)CN(C(=O)C(C)c2cccs2)C3)=O)cc1C C(=O)(C(C1=NOC2CC12)N(C1CC2(CCC2)C1)C)NCCC N1(C(C2(CNC(Cc3nc(C)oc3)=O)CC2)=O)CCn2cnnc2C1 c1(NCc2c(C)nc(Cl)s2)cccc2cccc(Cl)c12 N1(C(c2ccc(C)nc2C)=O)CC(NC(=O)CC2CCCCC2O)CC(C)(C)C1 C1(NC(C(CCOC)C)=O)CN(C(=O)CCCc2nc(C(C)C)no2)CCC1C c1(CCCC)cc(C(=O)NCC2CCCN2C(=O)CN(C)C2CC2)c(C)o1 N1(C(C2C(C)(Br)C2)=O)CC=CC1Cn1cc(CC2(O)CCC2)nn1 c1(C(=O)OCC(c2ccccc2)(C)OC)c(OC(C)C)nn(C)c1C n1(CC(=O)NCC#CCNC(c2cnc(C#N)s2)=O)nc(C(F)F)c2c1CCC2 C1(CNC(C2(CC=C)CCCN2C(=O)CC2CSCCO2)=O)CC2(CCO1)CC2 c1(N(C)OC(Cc2nc(C)oc2)=O)ccc2c(ccn2C(C)C)c1 c1(C(N2CCC(NC(c3c(C)cn(C)c3)=O)C(CO)C2)=O)cccn2nncc12 c1(C(N2CC(NC(C3N(C)CCC3)=O)C(F)C2)=O)cc(C(F)(F)F)nc(Cl)c1 C1(C(=O)NC(CCC)C2CCCC2)N(C(c2csc(C)c2C)=O)CCCC1(C)C c1(CC(=O)NCC(C(C)C)NC(c2ccc(C(F)F)cn2)=O)cc(F)ccc1F C1(C(N2CCC(C)(CNC(c3cc(Cl)c[nH]3)=O)C2)=O)CCOC2(CCCC2)C1 C1(Cl)(NCc2cn(CCCOCC(N)=O)nn2)CCCCC1 c1(C(C)Nc2sc(Br)cc2N)cc(F)ccc1F c1(C(N(CC(CC)NC(c2ccnc(O)c2)=O)C)=O)cnc(C)c(C#N)c1 C(=O)(CCCS(C)(=O)=O)NCC1C(NC(CCn2ncc(C)c2)=O)CC1 N1(C(c2cnc(C(C)OC)s2)=O)CC2CCCC(C1)N2C(=O)CSS(C)(=O)=O c1(C(N2C(C3CCN(C(=O)C4CC4)C3)CCC2)=O)[nH]nc2ncnc(O)c12 C1(NC(C(CC=C)C)=O)CC2CC1N(C(c1c[nH]nc1-c1ccsc1)=O)C2 N1(C(c2c(Br)ccc(C)n2)C(=O)NC2CCOC2)CCC2(CC(C(F)F)=NO2)C1 c1(CC)ncsc1C(=O)NCC1CCCC1NC(=O)CC1C(CC)C1(F)F CC(CCCNC(=O)C(C)OC1CCCC1)NC(C1CC1c1ccccc1)=O c1(C(N2CCC(OCCNC(C(C=C)O)=O)C2)=O)nn(CC(F)F)cc1[N+](=O)[O-] C1(N(C)Cc2cncc(C)c2)CCCN(C(=O)C(n2ccnc2C)C)CC1 Cc1cc(=O)c(C(=O)NC2(CNC(C3COC3)=O)CC2)nn1-c1ccccc1 C1(C(N2CCC(CNC(c3c(C)c(N)cnc3)=O)C2)=O)CC2(C1)CS(=O)(=O)C2 C(CC(C(=O)Nc1ccc(OC(C)C)nc1)NC(=O)CC1CN(C(C)=O)C1)OC Cc1cc(N)c(C(=O)NCC(F)CNC(C2CCC3CC2CO3)=O)c(F)c1 C1(CC(=O)NC2(CC(C)C)CC2)CCN(C(=O)C=CCF)C1 c1(N2CC(NC(c3ccn(C(C)(C)C)n3)=O)C(F)(F)C2)ncnn2cc(Br)cc12 CN1CC(O)CCC1C(N1CC(CC(=O)NCc2nccs2)C2(CC2)C1)=O c1(CC(=O)NC(C)CCNC(C2(CO)CCC2)=O)cc[nH]c(=N)c1 C1(C(=O)NCCOC2CCN(C(c3ccncc3F)=O)C2)CCC2(CC1)CC2 C(=O)(CCCCCCS(N)(=O)=O)N1CCC(C2(NC(C=COCC)=O)CC2)C1 C1(C(=O)OCC(=O)NC(c2c(C)cccc2)C)CCC2(COC2)OC1 C1(CC(C)NC(=O)C2CC2)CC2CCC(C1)N2C(=O)C=Cc1ccccc1 c1(CC)c(C(=O)NC2CCC(NC(=O)C(C)P(C)(C)=O)C2)[nH]c2ccccc12 C1(NC(=O)Cn2nc(Cl)ccc2=O)COC2(CCCN(C(=O)CC3CSC3)C2)C1 c1(OC)ccc(C(N2CCC(N(C)C)C(C)C2)=O)c(N)c1 N1(C(c2c(CCCC)ocn2)=O)CCCC(CNC(=O)C(=O)NC2CC2)C1 C1(C(=O)OCc2ccccc2)CS(=O)(=O)CN(C(C2CCCC2C2CC2)=O)C1 C(=O)(C1COc2ccc(F)cc21)NCC(CNC(c1[nH]cc(OC)c(=O)c1)=O)O c1(OCC)cc(C(N2CCCC2CNC(=O)CC2CCC(F)(F)C2)=O)oc(=O)c1 C#Cc1ccc(OCC2CC23CCOC3)cc1.N12CC(CNC)(C1)CC2=O Nc1cccn(CC(=O)NCC2CC(CNC(C3(C(F)(F)F)CC3)=O)CO2)c1=O c1(C(=O)NC2CN(C(Cc3cc(C(C)C)no3)=O)CC2F)ccc(S(C)(=O)=O)s1 C1(CC(N2CC(NC(=O)CN3CCCNC3=O)(CF)C2)=O)CCC2(CCC2)O1 c1(CC)nc(-n2cccc2)sc1C(=O)NC1CCC1NC(c1scnc1CC)=O CC(CS(=O)(=O)c1ccc(Cl)c(Cl)c1)NS(=O)(=O)c1ccc(Cl)s1 C(=O)(C1=CCC(C)CC1)N1CCC(COC)(NC(=O)C=CC2CCOC2)CC1 Cc1nc(C(N2CCC3(CCCN3C(C3CCC(=O)N3)=O)C2)=O)c2n1CCCC2 c1(OC)ccc2[nH]c(C(=O)NC3CC(CNC(c4ccc(CO)o4)=O)C3)cc2n1 C1(CC(=O)NC2(CC(=O)N(C3CCSC3)C)CCC2)CCC(=O)C1 CCCC(C)(C)C(=O)NC1CCCC(CNC(C2CC3CCC2C3)=O)C1 c1(NCC(CC)(CC)NC(=O)C(CC(C)C)OC)ccnc2nc(C)nn12 NC(=O)CCC(=O)NCC(CNC(c1cccc(OCC(F)(F)F)n1)=O)CO N1(C(C2CCC(CNC(C(C)(C)SC)=O)CC2)=O)CCOC2COCC2C1 C#CC1(O)CCN(C(=NCCc2c[nH]nc2C)NCC(=O)NC(C)COC)C1 N1(C(c2c(C)cno2)=O)CC2CCCC(CNC(=O)C3=C(Cl)CCOC3)(C2)C1 CC1=C(C(=O)NC(C2CCCC2)CNC(=O)CCC(=O)c2ccc(C)s2)CCC1 c1(C(=O)NC2CC(N(C(C(C)SCC)=O)C)C2)c(F)ccc(Cl)c1N C1(C(=O)NCC2CC(OC)CN2C(=O)C=C(C)C(F)F)CCc2c(cnn2C)C1 CCC(C)(C)C(=O)NCCCN(C(=O)CN1C(C)CCC1C)C c1(CC)c[nH]c(C(=O)NCC2(O)CC(NC(=O)C(C)OCC(F)(F)F)C2)c1 C1(CNC(c2ccc(OC)o2)=O)CC2CCC1N2C(c1cnnc(Cl)c1)=O C1(O)(C(CNC(C2C(CCC)C2)=O)(C)C)CN(C(=O)Cc2csc(C(C)C)n2)C1 N1(CC=C)C(=O)NC(c2cnc(OC)cn2)C(C(=O)OCC)=C1C(C)OC C(=O)(C(C)CC(C)(C)C)NC(C(CO)NC(CC(C)NC(=O)OC(C)(C)C)=O)C C#CCCCC(C)C(=O)NC1CC2CC1N(C(=O)Cc1ccc(C)nc1)C2 O=C(CC1=CCOCC1)NCCC1CCC(NC(C2CS(=O)C2)=O)C1 N1(C(C(C=C)(C)O)=O)CCCN(C(c2cncc(OC(C)C)c2)=O)CC1 CCCC(CCC)C(=O)N1CCOC(C(C)NC(c2ccc(N)c(Cl)c2)=O)C1 O(NC(=O)C(C)(C)C1CCCN1C(C1CCCC2(CC2)C1)=O)CCC(C)O N1(C(C2C(c3cn(CC)nc3)OCC2)C(=O)NCCCSC)CCC2C(O)CC12 C=C(CNC(c1nnnn1C1CCOC1)c1ncc[nH]1)c1ccc([N+](=O)[O-])cc1 C1(CN(C)C(c2ncc[nH]c2=O)=O)CC(F)CN1C(C1C2COCC12)=O CC(C)C(C(=O)N(C)Cc1cncs1)NC(=O)C(C)Cn1ccnc1 N1(C(CSCC=C)=O)CC(C=C)(CC(=O)NC(CC)C(=O)NC)C1 C(=O)(CC(O)C(Cl)(Cl)Cl)NCC(C)Cc1cn[nH]c1 C1(C(=O)NCC=CC)CC(C)(C)CCN1C(=O)C(N1CCOCC1)C C(N=c1cc(C)nc(Cl)[nH]1)C1CCC(NC(c2c(OC)cccc2F)=O)CC1 C(CCC(C(=O)NCC12CCC(CC1)O2)NC(c1ccncc1Cl)=O)OC Cc1ccc2sc(C(=O)NC3CC4CC3N(C(C3(C)COC(=O)C3)=O)C4)cc2c1 c1(C(C)(C)C)noc(CCC(=O)NCC2CCN(C(=O)C(F)C3CCOC3)C2)n1 C1(C(=O)NC(CC#C)C(N)=O)CCCCCCN1C(C1CC(=O)OC1(C)C)=O c1(CC(=O)NCCSCC(=O)N(CC(CCC)C)C)ccc(F)nc1 C(=O)(C1=CCCOC1)NCCCCCCNC(C(c1ccn(C)n1)(C)C)=O C(C(=O)N1CC(CNC(=O)CC(O)C2CC2)C1)(C(C)C)NC(COC)=O C(CCC(C(=O)N1CC(CO)C(CO)C1)NC(C1CC1C1CCC1)=O)OC c1(C(=O)NCC2N(C(C(=O)NC3CC3)=O)CCOC2)ccc(CO)cc1F C(=O)(C1=CCC(C)CC1)NC1CCCCN(C(C(=O)NCCOC)=O)C1 Cc1ccccc1-n1cc(-c2csc(C(=O)NCC3(C#N)CC3)n2)cn1 CCC(CCC(=O)NCC(O)CCO)NC(=O)Cc1ccc(O)cn1 N1(C(C(c2nc(C)sc2)=O)=O)CCC(CO)C(NC(c2cocn2)=O)C1 CC(C)C#CC(=O)NC(C1CN(C(=O)C(CN(C)C)c2ccccc2)CCO1)C c1(CCC)ncoc1C(=O)N(CCCCCNC(=O)C(O)CN1CCCC1)C N(C(=NCC1CC1)NCC(=O)Nc1ccccn1)CC(c1cccc(F)c1)CO C(=O)(CC(CC)CCCC)NCC12C(CN(C(C(CCCCC)F)=O)C1)CCO2 C1(C(N2CCC(C)(NC(=O)C#CC3CC3)CC2)=O)C2CCC(CC2)C1C(F)(F)F Cc1cc(C(=O)NNC(=O)C2CSCCN2)c(C)n1-c1ccccc1 c1(C(=O)NC2CCC(NC(c3cncc(O)c3)=O)C2)c(F)c(F)cc(F)c1F N1(C(c2c(COCC)ncs2)=O)CCCC1(C)CNC(C1CCCC12CC2)=O Cc1cc2c(C(=O)NC3CCC(NC(=O)CC(C)C(F)F)CC3)ccc(C)c2[nH]1 c1(NC(C2COCCN2Cc2ccc(CO)o2)=O)ncc(I)cc1C(F)(F)F Cc1cccn2ncc(C(N3CCN(C(=O)C(C)(C)C(C)C)CC3C3CC3)=O)c12 C1(CNC(C(c2cnn(C)c2)OC)=O)CC2CCC(C1)N2C(C1C2CCCC12)=O CC1(C(=O)NCCCN(C(c2cscc2C2CC2)=O)C2CC2)CCCC1O CC1(C)CCCN(C(=O)CC2COCC2O)C1C(=O)NCC1=NOC2COCC12 C1(NC(C(CC#C)C2CC2)=O)CCC2(CCN(C(=O)CC(=O)OCC)C2)C1 Nc1cc(C(=O)NCC(CO)NC(=O)C(F)C(F)(F)F)cc(F)c1Br C1(C(=O)NCC(C(N2CC(C)(OCC)C2)=O)C)CC(=O)NC(=O)N1 C1(C(=O)OC)N(CCOc2cccc(F)c2)CC12CCC(F)(F)CC2 N(C1CCc2cccnc21)C(c1[nH]c2c(Br)cccc2c1-c1ccccc1)=O c1(C(N2CCC(C(=O)Nc3c(C)cnc(F)c3)C2)=O)ccc(Br)c(O)c1Br C1(C(=O)NCCc2cc(C)cc(C)c2)CCN(Cc2sccc2Cl)CC(C)(C)C1 C1(OCC)CC2(C1)CC2C(N1CCCCC1CN(C(=O)CC(C)(F)F)C)=O C1(NC(C(=Cc2ccco2)C)=O)CN(C(C2CC(C)(C)CN2C)=O)CCC1CO N1(C(c2n(C(C)C)ccc2)=O)CCC2CN(C(=O)C=Cc3ccco3)C2C1 C1(N(C(CCSCCC)=O)C)CCC2CN(C(=O)Cn3cnc(C(N)=O)n3)CC12 N1(C(C(C)SC)=O)CC(NC(=O)CCc2cnn(C)n2)Cc2ccccc21 C1(NC(CC2(C)CC2(Cl)Cl)=O)CCN(C(c2cccnn2)=O)CCC1CO c1(OC)cc(C(=O)NC2CC(c3ccccc3)(CNC(C3(C)CC3F)=O)C2)sn1 C(=O)(NNc1ccc(Cl)c(C)n1)c1cnc(OC)[nH]c1=N c1(C(N2CCC(OCCNC(C(C(C)O)N(C)C)=O)C2)=O)ccc(S(C)(=O)=O)o1 c1(C(=O)OC)c(CSC2CCCCN2C(=O)C=CCOC(C)(C)C)occc1=O C(=O)(CC1=NNC(=O)C1)NC(CN(C(C(c1c(C)n[nH]c1C)C)=O)C)C n1(C(C(=O)N(CC(C)NC(=O)CC2(C)CC2)CC)CC)ncc2ccccc12 N1(C(C(COC)COC)=O)CCC(C)(NC(=O)CSC2CCOC2=O)CC1 Cc1ccc2[nH]c(C(=O)NC3CCC4CC3CN4C(C3CC3C)=O)cc2c1C CCCC(CNC(=O)Cc1cn(C(C)C)nn1)NC(=O)C=C(CC)CC c1(CC)ccc(C(C)C(=O)NCC(CO)NC(=O)C=CCF)cc1 c1(C(CO)NC(CN(CC)CC)=O)ncc[nH]1 O=[N+]([O-])c1cc(Cl)c(Cl)c(S(=O)(=O)NCC(O)COc2ccccc2C(F)(F)F)c1 N1(C(CCC=C)=O)CCOCC1CN(C(=O)C(C)(C)COC)C C1(C(=O)NCCCOCC)CCCCN1C(=O)CC1CCC(C)CO1 C(=O)(C1CCc2ccccc21)NC1C(C(N(C(C)(C)C)CCN)=O)C1 c1(CC)cccnc1NC(=O)NC1CCN(C2CCC2)C1=O N1(C(C(CN(CC)CC)F)=O)CCCC(C)(CNC(c2cnncc2C)=O)C1 C1(NC(C(C(CC)O)C)=O)CCCC12CN(c1ncnc(C(C)(C)C)n1)C2 N(C(=NCCNS(C)(=O)=O)NCC1CC2CCC1O2)CC(C=C)(C)C C1(N(C(c2n(CC)ccc2)=O)C)CCCN(C(=O)CCC2COC(C)(C)O2)C1 N1(C(C2(CF)CCN(C(c3cc(C)cc(C)c3)=O)C2)=O)CC2CCCCC2C1C C1(NC(C(=O)NC(C)C)=O)CCN(C(=O)COCc2ccccn2)C(C2CC2)C1 N#Cc1ccc(CN2CC(Nc3ncc(C4CC4)cn3)CC(CO)C2)c(Br)c1 c1(NC(C(c2n(C)cnc2)N)=O)ccc(C(F)(F)F)cn1 c1(C(=O)Nc2ccc(-c3ccc(C(=O)OCC)nn3)s2)cc(OCC)ccc1I c1(C(=O)NC2CCC(F)(CNC(Cc3n[nH]c(=N)s3)=O)C2)c(F)ccc(F)c1F n1(C2(C(=O)NC3CC(NC(CCN(C)CC)=O)C3)CC2)cc(Cl)cn1 C1(NC(c2c(CC)nco2)=O)CC2CCC1CC2NC(=O)CCc1ncnn1C C1(CC=C)(NC(=O)C(c2ccccc2C)C)CCN(C(=O)CC=CCC)C1 O=C(C#CC1CCOCC1)NCC12CCC1CCN2C(c1ccc([N+](=O)[O-])o1)=O c1(C(=O)NC23CC(CNC(C(C)c4ccsc4)=O)(OC2)C3)cccn2nccc12 c1(COC)ccc(C(=O)NC2CCC(NC(C3CCNC(=O)C3)=O)C2)cc1F c1(C(=O)OCC)ccc(Cc2ccccc2)cn1.C12(COC1)C(=O)N2 c1(C(=O)NCC2OCC(CNC(C(CC)(C)C)=O)C2)c(N)sc2c1CCSC2 C1(NC(C(CC)n2ccnc2)=O)CCC(C)N(C(c2ccc(Br)cc2)=O)C1 C1(CN(C)C)CCCCN1C(C1C=CCN1C(=O)CCC1CCCC1)=O N1(C(CC(CC2CC2)NC(Cc2cc(C)on2)=O)=O)C2CCCC1CN(C)C2 C1(c2ccon2)(CC(=O)N(C)CC2(CNC(C3CCS3(=O)=O)=O)CC2)CS(=O)(=O)C1 N1(C(C=CCOCCOC)=O)CCC2CCN(C(=O)CCCn3ccnc3)C2C1 C1(C(N(C2(c3nn[nH]n3)CC2)CC)=O)CC(C)N1C(C1CN(C2COC2)C1)=O N1(C(C2(C)CCOC2)=O)CC2(NC(=O)COCC3CCCOC3)CCC1CC2 C(=O)(CC1(O)CCOc2ccccc21)NCC(C)NC(CCCC#C)=O C1(C(N(CCCNC(=O)CCC2CC2(F)F)C)=O)CCCCN1S(N)(=O)=O C=CCC(CC=C)C(=O)NC1CCN(CCCNC(=O)C(O)P(C)(C)=O)C1 C1(NC(c2csc(Cl)n2)=O)CC2(CCCN(C(=O)CC3CCCO3)C2)C1 C1(N(C(C(=O)Nc2c(C)nn(CC(F)F)c2)=O)C(C)CN)CC(C)(C)CC(C)(C)C1 Nc1ccc(C(N2CCCC(c3cc(O)n[nH]3)C2)=O)c(F)c1 C(=O)(C(O)CCCC)NCC1CN(C(CC=C)=O)CC1c1ccc(OC)cc1 c1(CNCc2ccc(CC)cn2)cn2c(C)cc(C)nc2n1 C=CCC(C)C(=O)NCc1ccc(CNC(c2cc(C(F)(F)F)ncn2)=O)cc1 C1(C(=O)NC2CN(C(=O)C3=CCSC3)CC23CC3)CC(c2ccc(F)cc2)=NO1 C(C)(CCN=c1ncc(C(F)F)c[nH]1)NC(C1CCC(=C)CC1)=O S(=O)(=O)(c1c[nH]ccc1=NCCn1ncnn1)Nc1c(C(C)C)cn(C)n1 C=C(C)C1CN(c2cc(N(C)Cc3cccs3)nc(C)n2)CCO1 C1(CNC(CCCC#C)=O)CN2CCCCC2CN1C(c1cncc(SC)c1)=O c1(C(=O)NC(C(C)C)(C)CNC(C2(C)CCCNC2=O)=O)cnc2occc2c1 N1(C(CC(CCC)O)=O)CC2CC1CCC2NC(=O)CC1OCCCC1(C)C c1(CN2C(CC(=O)NCC3(CO)CCC3)COCC2)ccc(Cl)cc1O CCCCC(C)C(=O)N1CCCC(F)(CNC(=O)C(O)C2CCCC2)C1 C(=O)(C1SCCc2ccccc21)NC1CN(Cc2nc(CC)[nH]n2)C(C)CC1 C(=O)(C1=CC2(CN(C(c3cccc[n+]3[O-])=O)C2)OC1)N1CC2C(C)(C)C2C1 c1(C(=O)NC(C)CCN(C)C(c2ccc(N)cc2)=O)cc2c(=O)[nH]ccn2n1 C(=O)(C(F)(CNC(C1CCCOCC1)=O)C(C)C)NCCC1CC(C)C1 C1(C(=O)NCC(CN(C)C(C23CCC2C3)=O)O)CCOCC1 c1(NC(c2nc(C(=O)OC)oc2)=O)ccc([N+](=O)[O-])cc1Cl C=C=CC(C)C(=O)NC(c1nocc1C(=O)NC1CC(C)(C)C1)C C1(C(=O)NCC(CC)(C)Cl)CC(O)CN1C(c1nccnc1C)=O O=S(=O)(c1nc[nH]n1)NCCCCCc1cccs1 N1(C(c2n(CC=C)ccc2)=O)CCC2(NC(=O)CCOC3CC(F)(F)C3)CC2C1 c1(C(=O)NCc2c(C)ncs2)cn(C)nc1C1CCC1 N1(C(C(c2ccccc2)NC(C)=O)=O)CCCN(C(c2cc(C)n(C)c2)=O)CC1 C(=O)(CCCC(C)C)N1CC(CC(C)NC(C(CCSC)OC)=O)C1 C(CCC(N)=O)(C(=O)N1CCC(C)(C(C)=O)C1)NC(=O)OCc1ccccc1 Cc1cccc(O)c1C(=O)NCCc1ccc(CNC(C2(CO)CCC2)=O)cc1 c1(C(=O)NCC=CCNC(C2CCCO2)=O)ccc(N2CCOCC2)cc1F C1(C(=O)NC2CC(O)(CNC(c3ccc(Br)o3)=O)C2)CCc2nnc(O)cc2C1 C12(C(=O)NCC(C(=O)OCC)C)CC1CCN2C(=O)Cn1cncn1 c1(C(N(CC(CN(C(C(C)NC(C2CCC2)=O)=O)C)O)C)=O)cc(O)cs1 c1(C(=O)NC(C2CCN(C(=O)CCOc3ccc(F)cc3)C2)C)c(Cl)cnn1C C(C(=O)NC1(C)CCC(CC(N2CCC(CO)(CO)C2)=O)C1)(C(C)C)SC C1(C(N(CCN(C(=O)Cc2cccc(C(F)(F)F)c2)C)C)=O)CC2(CCC2)C1 c1(C(=O)NC2C(NC(Cc3cnc(C)[nH]3)=O)COC2)csc2c1CCCCCC2 c1(C(N2C(C)CC(NC(=O)C(=O)N=S(C)(C)=O)CC2)=O)nccc2c1NCCC2 C1(C(=O)O)(NC(=O)NC2CC2C2CCCO2)CCS(=O)(=O)CC1 c1(CNC(C(CC)NC(=O)C=CC2CCC2)=O)cncc(C)c1 c1(C(=O)NC2CN(C(c3cc(C)c(C)[nH]3)=O)C(C)CC2)n[nH]c2c1NCCC2 c1(NC(CCC2N(C(c3c(C)cco3)=O)CCC2)=O)cc(C(N)=O)ccn1 N1(C(CC(CNC(C(C=C)(C)C)=O)C2CCC2)=O)CC2(CNC(=O)OC2)C1 c1(C(=O)NCC(C)N(C(C(CCC)OCC)=O)C)c(OCC2CC2)cccc1Cl C1(C(C)C)C(=O)O1.c1(CCC=CC)ccc(F)cc1 C1(CNC(Cc2cc(C)[nH]n2)=O)C(C2CC2)CCN1C(c1cnccc1C#N)=O CC1CN(CC(=O)COCC(F)(F)F)CCN1C(c1coc(C2CCOCC2)n1)=O CS(=O)(=O)c1ccccc1CN1CCCC(C(=O)NCc2c(Cl)cccc2Cl)C1 c1(OC)cc(F)c(F)cc1C(N1CC2CC1CN2C(c1cc(O)cc(=O)o1)=O)=O Cc1cccc2c(C(N3CC(NC(c4cc(=N)[nH]c(Cl)n4)=O)C(C)C3)=O)n[nH]c12 N1(C(C=CC(C)C)=O)CCN(C)CC1CNC(c1[nH]c(=N)ccc1C)=O N1(C(C(CC)(C)O)=O)CCC(C)(CCc2ccccc2)CC1 Cc1cc(CC(=O)NCC2(C)CCN(C(C3CN(S(C)(=O)=O)C3)=O)C2)ccc1F Cc1cc(C)nc(N2CCCC(NC(=O)CCn3cccnc3=O)C2)n1 c1(C(N(CCN(C(C(C(=O)OC)(C)F)=O)C)C)=O)ccc(O)c(C)c1C Cc1csc(C(=O)NCc2ccc(C(N3CCCC3C3CCCC3)=O)cc2)c1C c1(OC)ccc(CC(C)CNC(=O)N(C(C)C)Cc2ccoc2C)cc1F N1(C(C(CCC)CC2CCCC2)=O)CC2(CCN(C(C3(CF)CC3)=O)CC2)C1 CC(C)C(C(=O)NCC1C2CC1N(C(=O)CC(C)c1ccco1)C2)n1cnnc1 C1(c2nc(C)[nH]n2)CN(C2CC(C(=O)OC(C)(C)C)C2)CCO1 Nc1cc(Cl)cc(Cl)c1C(=O)NC1CC(O)CN(C(=O)CSC(F)(F)F)C1 C1(C(C)(C)NC(C=C(COC)C)=O)CCN(C(c2ccncn2)=O)C1 c1(CC)nc(C)[nH]c1C(=O)NCC(C)N(C(=O)CCC1CC1(Cl)Cl)C n1(CCC)nnnc1C(c1ccoc1C)NC(C)C(=O)OC(C)(C)C C1(NC(c2c(C)snc2)=O)CC2C(NC(=O)CC3CCCN(C)C3)C2C1 Cc1cnc2c(cnn2CC(=O)NC2(CN(C)C(C3CCN(C)C3)=O)CC2)c1 N1(C(C2(n3cc(-c4n(C)ccn4)nn3)CC2)=O)CCN(CC2C3CCCC23)CC1 c1(C(N2CC3C(CNCc4n(C)cnc4)(C3)C2)=O)c(Br)ccc2c1OCO2 c1(CC)oc(C)cc1C(=O)NC(CN(C(C1(C(F)(F)CC)CC1)=O)CC)CC c1(CCN(C)C)ccc(C(=O)NNC(=O)c2ccc(N(C)C)cc2)cc1[N+](=O)[O-] Cc1nc(C(N2CCC(O)(C(C)CNC(=O)CCCc3ncco3)C2)=O)c(C)s1 C1(CC)CCCC1(C)C(N1CCC(CF)(NC(c2ccc(C(F)(F)F)[nH]2)=O)C1)=O CC1CC(C)N(C(=O)CNC(N)=O)CCN1C(c1ccc2nc(O)[nH]c2n1)=O CCC(C)(C)C(O)C(=O)N1CCC(C(=O)NC2CCN(C(C)=O)C2)C1 C#CCCCCC(=O)N1CCC(C(C)NC(=O)CC2CC3(CCC3)CO2)C1 CC1(O)CCN(C(C23CC2CN(Cc2cnc(C(F)(F)F)nc2)C3)=O)CC1 N1(C(=O)COCC2CCOC2)CCOC2(C1)CN(C(=O)C=C1CCCCC1)C2 C(=O)(C(C(=O)OC(C)(C)C)C(C)C)NC(C(C)NC(c1c(CC)cno1)=O)(C)C Cc1cc(=NCC2C3CCCC23)[nH]c(N(C)Cc2ccc(OC(C)(C)C)cc2)n1 c1(C(N2CCC(C3CCC3)C2)C(=O)NCCC(=O)OCC)cnc2cnccn12 C1(C(=O)NC2C(NC(CCN(C)CC)=O)CC2)CCc2nnc(O)cc2C1 C12(C(=O)NCC(C3CC3)NC(c3c(C(C)=O)cccc3)=O)CC3CC1C2C3O c1(C(=O)NC(C2CN(C(c3sccc3F)=O)CCO2)C)cncc(F)n1 S(=O)(=O)(c1cccc(F)c1)NCC(=O)NC1CCC(CNC(C2OCCO2)=O)C1 N1(C(c2c(C)cc[nH]2)=O)CC2OCC(NC(c3cccn4nccc34)=O)C2C1 C1(C)(CC)C=C(C(=O)NCC2CC(OC)CN2C(c2cc(SC)ccc2Cl)=O)C1 CC1=C(C)CC(C)(C(N2CC(CNC(=O)CP(C)(C)=O)C(C)(C)C2)=O)CC1 N1(C(C(Cc2cn[nH]c2)NC(CC2CC(OC)C2)=O)=O)CC2(CCN2C)C1 C=C(Cl)CC(C(=O)NCc1nc(C)cc(O)n1)NC(c1cc(C)nnc1C)=O CC(C)C(C(=O)N(CCC(C)NC(C1CC(C2CCC2)C1)=O)C)C(C)C c1(-c2cn(CCCC(=O)N(C(COC)C)C)nn2)cc(Cl)ccc1C(=O)O c1(C(N(CC)CC2CCCN2C(=O)CC(C)n2cccn2)=O)ccc(C)c(C)n1 C1(CNC(C(=Cc2ccco2)C)=O)COCCN(C(=O)C=CSc2nc[nH]n2)C1 Cc1ccc(CNC(=O)C(C)NC(c2cnccn2)=O)c(F)c1 C=C1Cn2c(C(=O)NC34COC(C3)C(NC(C3(C#N)CC=CC3)=O)C4)nnc2S1 c1(N2CC=CC(NC(=O)CC3CC4(CC4)C3)C2)ccc2nnnn2n1 c1(C(=O)NCC2(NC(C3C(C=C)C3)=O)CCCC2)sc(C)nc1C(F)(F)F N1(C(CCC=C)=O)CCCC2(NC(c3cnc(OCC)cn3)=O)CCCC12 Cc1cccc2cc(C(=O)NC3CCN(C(=O)CC4CCOC4)C(C)C3)[nH]c12 N1(C(C(CCC)C)=O)C2CCC1CN(C(c1cc(C(N)=O)cc(C)c1)=O)C2 C1(C(N2CC(C)(CSC)C2)=O)CCCCC1CNC(=O)C(C)c1cc[nH]n1 C1(C(N2CCC(F)(CF)C2)=O)CCCN(C(C2CCCCS2)=O)C1 C#CC1CC2(CC2)CN1C(c1ccnc(CNC(=O)C(C)(C)CC(F)F)c1)=O CC1CC(C(=O)NCCC2CCCN2C(c2cnc(-c3cnccn3)s2)=O)=NO1 N1(C(C2(OC)CCOC2)=O)C2CC1CN(C(c1sc(C)nc1C(=O)O)=O)C2 N1(C(CCCC(=C)C)=O)CCCCCCC1C(=O)NC1CC(=O)N(C(C)C)C1 c1(CN2C(CSC)CCC2)ccnc2cc[nH]c12 C1(CC(=O)NCCCCC#CC)C2CCC(C2)N1C(c1cc(C)nn1C)=O C1(OC)C(N=c2[nH]c(=NC3CC(NCC(F)(F)F)C3)[nH]c3c2COC3)CC1(C)C C1(C(N2CCC(O)(Cn3cc(CC(C)(C)O)nn3)C2)=O)Cc2cc(Cl)ccc2O1 C1(N(C(C(=O)NCCNC(C)=O)=O)C)CN(C(C2CCNC2=O)=O)CC1(C)C C1(CCCC)CN(C(=O)C(C)CSC)CCN1C(c1nn(C)cc1C)=O CC1=C(C(=O)N2CCC(NC(C3CC(F)(F)C3)=O)CC(C)(C)C2)C(C)(C)CCC1 C#Cc1cc(F)c(C(=O)NC2CC3(C2)CC3NC(c2coc(Cl)n2)=O)c(F)c1 N1(C(C(CSC)O)=O)CCCC2CN(C(=O)CNC(=O)Cn3cncn3)CC12 c1(C(N2CCC(C(C)NC(c3cccc(CC)n3)=O)CC2)=O)ccc(N)c(F)c1 c1(CC)ccc(C)cc1C(N1CC(C(=O)O)(CNC(=O)OC(C)(C)C)C1)=O C1(c2nocn2)C2CCCC2CN1N(CCO)CCO.C1(C)(CC)CCC(NC)O1 C1(NC(CCC=C(C)C)=O)CN(C(c2ccc(C)nc2O)=O)CCC1CO Cc1ccc(C(=O)NC2(CNC(=O)C(C)C(C)O)CCCC2)cc1Cl c1(C(C)(F)F)cc(C(=O)NC2CC(NC(C34CC5CC3C4C5O)=O)C2)ccc1F Cc1cc(Br)cnc1C(=O)NCCCCN(C(=O)C(C1CC1)C1CC1)C C1(OC)CCCN(C(=O)CC(C(C)C)NC(=O)CC=C(C)C)CC1 C1(NC(c2cc(CC)nn2C)=O)CC2CN(C(=O)CC(=O)OC)CC12 C(=O)(N=c1ccn(C(F)F)[nH]1)C1(C)N(C(COCC(=O)NC)=O)CCC1 CN1CCN(C2CN(C(C3(C(=O)NC4(C(=O)N(C)C)CCOC4)CC3)=O)C2)CC1 O=C1N(CC(c2nc(Cl)cs2)=O)CC2CCCCN12 C(C(CC(F)(F)F)NC(c1ccnn1C1CC1)=O)NC(c1c(C(C)C)[nH]cc1)=O C1(CC(C)C)(C(=O)NCC2CC(NC(c3nc(CCC)oc3)=O)C2)CCNC1=O c1(NCC(CCCCC)O)ncc(C)cc1S(=O)(=O)NC(c1ccccc1Cl)C Cc1cc(C(=O)NC(CCNC(c2csc(Cl)c2)=O)C(C)C)nn1C1CC1 c1(C(N2C(CO)CC(NC(CNS(CC)(=O)=O)=O)C2)=O)cc2ccsc2n1C N1(C(c2c(OC)ccs2)=O)C2CCC(C2)C1C(=O)NCc1cccnc1SC CCC(CCCC(=O)NCCC(=O)NC(=O)C=C1CN2CCC1CC2)NC(N)=O c1(C(N2CCC(CNC(C(C)n3cnnn3)=O)C23CC3)=O)cn2ccncc2n1 C(C(C)CC(=O)NC1(CCOC)CCN(C(=O)C(C)=C2CC2)C1)OC c1(CC)ccccc1OCCOCC(=O)NCC=CCNC(=O)C(C)CO N1(CC)N=C(C(=O)N2CCC(=CCNC(=O)CCCCC(C)C)CC2)CCC1=O c1(NC(C(c2cc(Cl)cs2)N(CCN(CC)CC)C(C)C)=O)cccc(Cl)c1C c1(C(N2CCCC(CC=C)(NC(CCC)=O)C2)=O)cc2c(cn1)OCCO2 C12(C(N3CCC(OC(C)=O)C3)=O)CC(C)(C1)OC2C c1(C(N(CC(C)NC(C(CC=C)C)=O)C)=O)noc2cc(Br)ccc12 Cc1cccc(C2(C(=O)N(CC(C)N(C)C(c3cccnn3)=O)C)CCC2)c1 c1(-c2ccc(NC(C3C4CCC(F)(F)C34)=O)cc2)nnc2n1CCC2 CONC(=O)CNC(C1C=CCN1C(=O)COCC(F)F)=O c1(OC)ccc(N(C(=O)NNC(=O)c2cc(Br)c[nH]2)C(C)=O)cc1 N1(C(C=CCC)=O)CCCC12CCN(C(c1cc(C)sc1C)=O)C2 c1(C(=O)OCC)ccc2c(c1)CC(NC(=O)NC(CC(C)C)C(C)(C)C)C2 CC1CN(C(C2CC3C=CC2C3)=O)CCC1CNC(C1COC(C)(C)C1)=O c1(CNC2CN(C(Cc3c(C)ccc(Br)c3)=O)CC(F)C2)cc(F)cc(C#N)c1 Cn1c(=O)sc2cc(CN3CCCC(c4ncns4)C3)ccc12 C1(CN(C(C(C)C)=O)C)CCCC(NC(=O)C=C2CCC(C(C)(C)C)CC2)C1 CC(CCc1ccccc1F)C(=O)NCCCOCCNC(=O)CC1CCCC1 c1(C(=O)NC2(CC)CCCN(C(=O)CCC(C)(F)F)C2)ccc2nc[nH]c2n1 CC1CCCC1(C)C(N1CCN(Cc2cn(Cc3cnn(C)c3)nn2)CC1)=O c1(CN2CC(C(N(CCCC)CCCC)=O)SCC2)cc(C)cc(C)n1 N1(C(C(N2CCOCC2)C)=O)CC(CNC(c2nn(C)cc2N)=O)CC12CCC2 N1(C(C(CSC)O)=O)CC(NC(c2ccc[nH]2)=O)C(CC(C)(C)C)C1 C=CC1(NC(C2(CC)CCN(C(c3cc(Cl)cs3)=O)C2)=O)CCCCC1 N1(C(C(CC)CC(C)C)=O)CCC(NC(=O)CC(F)(F)C(C)C)C2(CCC2)C1 C(=O)(C1=NOC(CNC(c2cn(C)cc2C)=O)C1)N1CC(OCC(=O)NC)C1 C1(NC(c2nc(CC)[nH]n2)=O)CCC2(CC1)CN(C(c1nc(O)c(C)s1)=O)C2 c1(C(C(=O)NCCC#N)N(CCCC)CC)cc(S(N)(=O)=O)cs1 C(=O)(C(O)C(C)C)N1CC(OCCNC(c2n(COC)ncc2)=O)C1 c1(C(N2C(CNC(C(C(C)C)F)=O)C(C)(C)CC2)=O)ccc2c(c1)CCN(C)C2 c1(SC(C)C(=O)NCC(C)(C2CC2)NC(=O)CSC(=N)N)ccccn1 C=CCC(C)(C)CC(=O)NC1CCCC1CNC(=O)COC(C)(C)C N1(C(c2csnn2)C)CCC(O)CC1.C123CC(C1C2)n1cc(nn1)CNC3=O N1(C(CCC=C=C)=O)CC(CNC(=O)CC2CCC(=O)NC2)C2(CCOCC2)C1 N1(C(c2cc(C)[nH]c2C)=O)CCC2CN(C(c3ccc(F)c(F)c3Br)=O)CC2C1 N1(C(C2C(C)(C)C2(C)C)=O)CC(C(=O)NOCc2cncc(C#N)c2)C2(CCC2)C1 N1(C(c2cn(C)nc2I)C(=O)NC(C(=O)OC)CC(C)C)CCC(C)C(F)(F)C1 CC1CC(NC(C2(C)CC(C)(C)C2)=O)CCN1CCCN1C(=O)CNC1=O S(=O)(=O)(c1cc(C(=O)NC2(C3CCCN3C(c3ccsc3)=O)CC2)co1)N(C)C N1(C(CCc2cnc(C)o2)=O)CC(O)CC1CNC(=O)CCN1CCCCC1 N1(C(C(CNC(=O)CC2CCOC2)N(C)C)=O)CCn2ncnc2C1 C(=O)(N=c1ccn(CC2CC2)[nH]1)C1N(C(C2NC(=O)C(F)C2)=O)CCOC1 Cc1ccc(S(=O)(=O)N2CCCC2)cc1N(C)Cc1c(Br)c(C)nn1C C(=O)(CC1=NNC(=O)C1)NC1CC2C(NC(CC3(COC)CCOCC3)=O)C2C1 S(=O)(=O)(c1ccccc1)N1CCC(C(N(CCC)CCNC(=O)C2=CCC2)=O)C1 N1(C(C(CCCOC)C)=O)CCCN(C(=O)C(F)(F)CN2CCCC2)CC1C N1(C(C(CC=C)(C)C)=O)CCC(C2(NC(C3(C(C)(F)F)CCC3)=O)CC2)CC1 C(=O)(CCCCCC(C)C)N1CCCC(NC(c2n(CC)nc(C)c2)=O)CC1 Cc1nc2cccc(C(N3CCC4(CC3)CC4NC(=O)C(C)C3CCC3)=O)n2n1 CN1N=C(C(=O)NC2C=CC(CC(=O)N3CC(O)CCO3)C2)CCC1=O c1(OC)cccc(C(CNC(C2C=CC(NC(c3c[nH]nc3C)=O)C2)=O)OC)c1 c1(C(=O)NC2CN(C(C3C(C)(CC)C3)=O)C2)ccc(CCc2ccccc2)[nH]1 n1(CCCC)nc(C)c(C(N2CC(O)(CNC(=O)CC3CCOC3=O)C2)=O)c1Cl C(=O)(CCCC1CC1)NCC(C1CCOC1)NC(C1(CC)CCC1)=O CCCCCCC(C)C(=O)N1CC2(C1)CN(C(c1cc(C)n(C)c1)=O)CCO2 C1(CCNC(=O)Cc2cnccn2)COCCN1C(=O)Cc1cncs1 C1(CC)CCCN(C(c2ccnn2C)C(=O)NCc2ccco2)CC1 n1(CC)nc(C2CC2)cc1C(=O)NCCC1CC(NC(=O)COC2CC=CC2)C1 C1(C(=O)NC2CN(C(C3CCC(C)CC3)=O)C2)CCCC2(CC2)C1 c1(CC(=O)N(C)CC2CCN(C(C3CC(O)C3)=O)C2)csc2nccn12 C1(C(F)(F)F)(C(=O)NC2CN(C(c3cc(C(=O)CF)c[nH]3)=O)C2)CC=CCO1 CON(CCO)C(=O)COC1CN(C(=O)C=C(C2CC2)C2CC2)C1 C(CCCC(CO)NC(C12CCC1C2)=O)NC(C1CCN(C)CC1)=O c1(C(N2CC(O)(CNC(C3CCn4cncc4C3)=O)C2)=O)ccc(F)c(F)c1F N1(C(c2c(C)scc2)=O)CCN(C(=O)C(C(C)C)n2cncn2)C2CCC12 c1(C(C)=O)ccc(SC(C)C(=O)NCc2ccc(Cl)cn2)cc1 C#Cc1cn(C)nc1C(=O)NCC1CCN1C(c1cn(CC2CCOC2)nn1)=O C(=O)(C1(C)CCCc2ccccc21)NCCN(C(=O)C#CC(C)(C)O)CCC C1(NC(C2CC3CCC3C2)=O)CCN(C(=O)C(O)C2CCC2)CC1 c1(C(c2nnnn2C2CCC2)NCCCCCC=C)cccn(CCSC)c1=O CC(CC(=O)NCCCCO)C(C)(C)NC(c1cn2c(n1)CCC2)=O Cc1ccn(C(C)(C)C(=O)NCC2(F)CC(NC(=O)C(N3CCNC3=O)C)C2)n1 CCC(CC)C(C)C(=O)NCCCCNC(c1cnc2sccn12)=O c1(C(=O)NCc2c(CCNC(C(CC)OC)=O)ocn2)nnc(O)cc1O C1(NC(C(c2cncnc2)C)=O)CCCC(C(=O)NC2(CCF)CC2)C1 c1(N(CCOCC)CC)nnc(CC(C)C)n1CCCC1CCCCO1 N1(C(C=C(C)C2CC2)=O)CCC(C2CCCN(C(C3CCOC3)=O)CC2)CC1 c1(CN(CCN2CCOCC2)CC)ccc(-c2ccnnc2)c(CO)c1 CC1(C)CCC(NCCCc2ccc(C(C)(C)C)cc2)c2ccccc21 N1(C(CC2CC(=O)C2)=O)CCC(CNC(c2nc(Cl)c(Cl)s2)=O)C12CCC2 N1(C(c2c(OCC)ccs2)=O)CCC(O)C(C(N2CC(C(=O)OC)C2)=O)C1 c1(C(N2C(CNC(c3c(C)[nH]c(C#N)c3)=O)CCC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 c1(NC)ccc(C(N2CC(CO)(NC(c3cccnc3C)=O)C2)=O)cc1 c1(NC(C2(C)CCN(C(c3cc(F)cc(F)c3)=O)C2)=O)ncc(Cl)nc1Br C1(COC)(NC(=O)CCSCC(=O)OC)CCCN(C(=O)C(C)(F)F)C1 CCCCCC(O)CC(=O)N(C)CCNC(c1cc(F)cc(Cl)c1)=O c1(C(N2CC(NC(C3CCCSS3)=O)CC3(C2)CC3)=O)cc(F)c(F)c(O)c1F C1(CNC(=O)C=Cc2ccco2)CC2CCC(C1)N2C(=O)CCC(F)F c1(C(N(C(CNC(C2(CC=C)CCOC2)=O)C2CC2)C)=O)cc2nnn(C)c2s1 C1(C)(C(=O)NCCCOCCNC(c2nc(COCC)sc2)=O)CCCCC1C C1(C2CC2)(NC(C(F)=C(C)C)=O)CCN(C(c2ccc(Cl)cc2)=O)C1 c1(C(=O)Nc2ccnc(C(N3CCC(O)CC3)=O)c2)ncn2c1CCCC2 Cc1nocc1NC(=O)CC1CCN(C(C2(C)OCCO2)=O)C1 c1(CCC(=O)NCCC2(O)CCN(C(C3CCSC3)=O)C2)nc2cccnc2[nH]1 c1(C(=O)NC2CN(C3CN(C(CSC(=N)N)=O)C3)C(=O)C2)csc2cncn12 Cn1nc2c(c1C(=O)NCC1CCC(F)C1)CN(C(=O)C1=COCCC1)CC2 C(=O)(C1=CCCOC1)NC1CCCN(C(C(CC)F)=O)C1 C1(CCC)CN(C(c2ccc(Cl)o2)=O)CCN1C(=O)CCC1CCC(=O)N1 N1(c2ncc(OC)cn2)CCC2CN(C(c3c(F)ccc(C)c3F)=O)CCC12 N1(C(CCOCC)=O)CCC2(COC(CNC(=O)CN3CC4CCC3C4)C2)C1 C1(NC(C(c2ccccc2)NC(=O)OC)=O)CCOCC1NC(C1(Cl)CC1)=O c1(C(=O)NC(CNC(C2CC(CC)OCC2)=O)(C)C)cn(C(C)C)c(=O)nc1O c1(C(=O)NC(CNC(C(CC)(C)C)=O)(C)CC)coc2c1CS(=O)(=O)C2 Cc1sc(C(N2CCCC2CCNC(=O)C(C)CC2CCC2)=O)nc1O c1(CC(N2CCN(C(C(C(C)C)F)=O)C(C3CCC3)C2)=O)cccc2nonc12 N1(CCC(N2CCCC(N(C)Cc3cc(C)on3)C2)=O)C(=O)NC(C)(C)C1=O c1(C(=O)NC(C(=O)NC(c2n(CC)ncc2)C)CC2CC2)cccc2[nH]ccc12 C1(C(N2C(CN(c3c(C)cncn3)C)CCCC2)=O)CC(=O)NC1(C)C C1(C(=O)NCC2(CC(C)C)CC2)CCC(C)(C)N(C(C2CCCN2C=O)=O)C1 CCC(C)C(C(=O)NC1CC(CC(C)(C)C)C1)N(C(=O)Cn1ncccc1=O)C c1(C(=O)NC(C2CN(C(=O)C(F)C3CCC3)C2)C)ccc(OC(F)(F)F)nc1 N1(C(CCNC(C)=O)=O)CCCC12CCCN(C(c1cc(Cl)c[nH]1)=O)C2 CN1CC(=O)Nc2ccc(C(=O)NCC3CC(NC(C45CC(O)C4C5)=O)C3)cc21 CCC(C(=O)NCCCN(C(=O)Cc1cnn(C2CC2)c1)CC)N(C)C C1(CCC(=O)NCC(=O)OC(C)C)CCCN(C(c2cscn2)=O)C1 C1(CC=C)(C(=O)NCCCc2cnn(C)c2)CCN(C(c2cc(Cl)no2)=O)C1 C(CCCC(=O)N1CCC(NC(c2cc(C)c(C)s2)=O)CC1)OCCC=C CC1=C(C)CC(C(=O)NC(C2CCCN2C(c2nn(C)c(C)c2Cl)=O)C)CC1 C1(NCc2cc(SC)c(Br)cn2)CCCC12CCOCC2 n1(Cc2c(C)cccc2)nc(C)c(NC(=O)C(C)C(C)O)c1C c1(NC(c2nc(C(N3CC(O)C3)=O)cs2)=O)cc(O)ccc1Cl c1(CC)ccccc1C(=O)NCCC1CC(NC(c2ccccc2OC)=O)C1 CCC(CC(=O)N(C)CC1(O)CCN(C(=O)CC2(C#N)CCCCC2)C1)C(C)C C1(S(C)(=O)=O)(C(N2C3CC(CNC(C(C)C#N)=O)C2CC3)=O)CCOCC1 C1(C(N(CCNC(c2cc(CCOC)on2)=O)CCOCCO)=O)C2COCC12 N1(C(c2c(C)cnn2C)=O)CCCN(C(C2CC2C)=O)C(c2ccccc2)C1 c1(C(N(C2CCN(C(=O)C(C)CO)CC2)CC)=O)noc2ccc(Cl)cc12 N1(C(C#CC(C)C)=O)CC=C(C(C)(C)C(=O)NC(C)C(=O)N2CCCC2)C1 c1(C(=O)NCCC2CCN(C(CNC(=O)NC3CC3)=O)C2)cc(Cl)c(F)c(Cl)c1 c1(NC(CC)CSC)cc(Br)ccc1S(=O)(=O)NCc1cc(C)cc(C)n1 CN=c1[nH]cc(C(N2CCN(CCNC(=O)COC3CCCC(C)C3)CC2)=O)s1 C12(NC(c3ccn(C)c3)=O)CCC(C(=O)Nc3nccc(Br)c3Cl)(CC1)CC2 c1(N2CC(C)C(NC(C3CCCC3(F)F)=O)CC2)ncnc2sc3c(c12)CCC3 C(CC(C)(C)CNC(=O)C(C)Oc1ccccc1F)NC(C(CC)O)=O CCC(C)C(C(=O)N1CCC1Cn1cc(-c2ccc(OC)c(N)c2)nn1)N(C)C C1(CN(C2CCCCN(C(=O)OC(C)(C)C)C2)C)CCCCCCCCCCCC1 C1(C(=O)NCC2CCC(CC)O2)CCCCN1C(=O)C(CC)OC CCCCCC(C)(c1nnnn1C1CCOC1)NCc1cc(Cl)cs1 Cc1nc(F)ccc1-c1noc(C(C=O)CCC#N)n1.C(N)=O n1(CCC(N2CC(NC(CC(C)C3CC3)=O)(CO)C2)=O)cccnc1=O N1(C(c2cc(C)ns2)=O)CC(C(=O)NCc2nonc2C)C2(CCC2)C1 c1(C(=O)NC2C(NC(C3CN(C(=O)OCC)C3)=O)C2)nnc(O)nc1O CC1CN(C(=O)CCN(C)CCO)CC(C)C1NC(c1ccc(S(C)(=O)=O)o1)=O C(CC(C(=O)N(C(C)(C)CC(=O)N(C1CN(C)CC1O)C)C)OC)OC c1(OC)ccccc1OC(C)C(=O)N(CC(C)NC(=O)CCc1cn[nH]c1)C CC1=C(C)CC(C(=O)N(C(C)CN(C)C(c2cn(C)[nH]c2=N)=O)C)CC1 C12(C(=O)NCC(C)(CO)NC(c3ccc(O)nc3Cl)=O)CC3CC(CC(C3)O1)C2 C12(NC(CS(CC)(=O)=O)=O)CCN(C(c3cnc(C(F)(F)F)nc3)=O)CCC1C2 C(C)(C)(CCC(=O)NC1CC(CNC(C2CCO2)=O)C1)OC C1(NC(c2nc(C)sc2)=O)CCCN(C(C23C=CC(CC2)C3)=O)CC1 C1(CCC2C=CCCC2)CCN(c2nnnn2CCC2CCCS2)CC1 CN1CC(O)CC1(C)C(=O)NCC1CCCCN1C(=O)CN1CC2CC2C1 c1(C(N2C(CNC(C(CCC)c3ccccc3)=O)CC2)=O)nc(O)[nH]c(=O)n1 N1(C(C(C)=C2CCCC2)=O)CCCC(NC(c2cnc(C)c(Cl)c2)=O)C1C CC1(C)CC(C(=O)Nc2cnoc2C2CC2)CN(C(=O)COCP(C)(C)=O)C1 C1(NC(c2cc[nH]n2)=O)CN(C(C2(c3ccccc3)CC(O)C2)=O)CC1C1CC1 Cc1ccc2c(=O)c(C(=O)NC(C)(C)CNC(=O)CC3CC=CC3)c[nH]c2c1 c1(C(=O)NCC(CNC(Cc2c(C)cc(C)s2)=O)F)cnn2ccc(O)nc12 CCC(C)(C(=O)NCC1(O)CCN(C(=O)CN2CCS(=O)CC2)C1)C(N)=O C1(C(=O)NC(c2ccc(OC)cc2)CC)CC2COCC(C1)C2N c1(CSC)ccc(C)cc1-c1cscc1C(N(C)CC1CCCN1C)=O c1(CC(CNC(=O)C=Cc2nccs2)NC(C2C(CC)C2)=O)ccccc1 C(=O)(C(C)(C)C(=O)NC(CNC(c1ncsc1Br)=O)C1CC1)NC c1(C(N2C(CCNC(c3ocnc3C)=O)CC(OC)C2)=O)ccn2ccccc12 c1(C(N2CC(c3cn(-c4c(C)nn[nH]4)nn3)(C)C2)=O)nc(S(C)(=O)=O)ccc1Cl N1(C(CC2N(C(C(C(C)C)O)=O)CC2)=O)CCOC2(CCC2)C1 c1(CNC2CN(C(C3CC(=O)OC3)=O)C2)ccc(C(F)(F)F)cc1 C(=O)(CC=C(Cl)Cl)N1CC(CC(CN(C)C(=O)OC(C)(C)C)=O)C1 Cn1cc(C=CC(=O)NCCC(O)CNC(=O)Cc2cccc(Br)c2)nn1 Cc1sc(Cl)c(C(=O)N(C)CCOCCNC(=O)C(N2CCCC(O)C2)C)c1C N1(C(C(CC(C)C)CNC(=O)CCCCN(C)C)=O)CCc2ccc(F)cc21 C1(C(N)=O)(NC(C=CC(C)NC(C2CC(=O)C2)=O)=O)CCN(C)C1 c1(OC)ccc2c(c1)OCC(C(=O)NCC(C)CNC(=O)C(C)C)C2 C1(N(C(C2N(C(CCNC(C)=O)=O)CC(C)C2)=O)C)CC(C)CC(C)C1 C(C)(CO)(C(=O)N1CC(C(O)C(N2CCOC(C(C)(C)C)C2)=O)C1)OC c1(C(=O)NCC(n2cc(-c3c(C(=O)OC)n[nH]c3)nn2)C)ccc2sccc2c1 c1(C(N2CC=CC(NC(c3cnn(C)c3F)=O)C2)=O)cc2nccnc2cc1F N1(C(C(C)(C)C)=O)CC2CCC(NC(=O)CCc3cccc(C(=O)OC)c3)(C2)C1 N1(C(c2c(CC)nn[nH]2)=O)CCOC(C(C)NC(C2(CO)CCCC2)=O)C1 C1(CNC(=O)CC2(N3CCCC3)COC2)CN(C(=O)C2CC2)C2CCN1C2 CC1=CCCN(C(C2CC(C)N2C(c2nccn2C)=O)=O)C1 CC(C)CC(CNC(=O)C(C)C(C)C)C(=O)NC(C(C)(C)CO)C1CC1 c1(C(N2CCCC(C)(NC(c3ccoc3)=O)C2)=O)ccc(F)c(N)c1F C(=O)(CC(CC)CCCC)NC(CC=CC)C(=O)NCc1ccnn1C c1(C(N(C)Cc2c(CNC(C(C=CC)O)=O)cccc2)=O)cnc2cccnn12 N1(C(C2OCCN(C(C=CC(C)C)=O)C2)=O)CCCC12CCOC2 C1(C(=O)NC(CC=C)CNC(C23CC(COC)(C2)C3)=O)CC(OC)CN1C(C)=O C(=O)(C1=CC2C=CC1C2)N(C(C(=O)N(C(CC(CC)C)C)C)C)C N1(C(c2cccc(CC)c2)=O)C2CCC1CC(N=c1ccn3ncc(I)c3[nH]1)C2 CCC(C(=O)NC(C)CCNC(C1(CC)CCC1)=O)OC1CCCC1 N1(C(CCCC(C)C)=O)CC2(CCC(C(=O)NCc3cnccn3)O2)C1 CCC(C)C(C(=O)N1CCC1C(=O)NCc1ccc(C)nc1O)NC(=O)OC CCN(C)NC(=O)Cn1cc(CCN(C2CCCCC2)C(=O)CNC(C)=O)nn1 C1(CC(=O)NC(C2CN(C(c3cccs3)=O)CCO2)C)CC2CCC1CC2 Cc1ccc(C(N2CC(C)(C)CC2CNC(=O)C(C)n2ccnn2)=O)c(F)c1 c1(CCC(=O)NC2CCCN(C(c3c(C)nccc3)=O)C2)ccc(Cl)cc1O N1(C(c2n(CC)ncc2C)=O)CCC2(C=C(C(=O)Nc3ccc(F)nc3C)C2)C1 c1(OC)ccc(C(N2CCC(NC(=O)C(C)CC(C)(F)F)CC2)=O)c2sccc12 c1(CCC(=O)N(C(C(=O)OC)C2CCCO2)C2CC2)ccc(O)c(OC)c1 C1(NC(C2C(N(C)C)CCC2)=O)CC(NC(c2cc(C3CC3)no2)=O)C(O)C1 C#Cc1ccc(NC(=O)Nc2ccccc2C(=O)NC2(C#C)CCCCC2)cn1 C(CC(C)C)(C(=O)NCCC(C)(C)C)NC(C(CCCC)O)=O N1(C(C2(C(=O)OC)CCCC2)=O)CC2CC2(C(N2CCNC(=O)C2)=O)C1 C1(NC(CC(C)(C)F)=O)CCCN(C(=O)CCc2ccc(Cl)cc2Cl)CC1 N1(C(Cn2c(C)nc(C)n2)=O)CCC(C)(C)C1C(=O)NOCC1CCCCC1 C1(NC(C(C)OCCCC)=O)CN(C(c2scnc2Cl)=O)CCC12CCOCC2 CCC(C(C)(C)O)NC(C1CCC(NC(=O)CC2CCC(=O)C2C)CC1)=O CC1(C)Cc2cc(C(=O)NC3CCN(c4cc(F)ncn4)CCC3CO)sc2C1 C1(NC(COC(C)C)=O)CCCC(C(=O)N(C)CC2(C#N)CCC2)CC1 CC(C)CC(CNC(c1ncccc1Br)=O)NC(C1CCCS1(=O)=O)=O C(=O)(C1=CCCCC1C)N1C(C)(C(=O)Nc2c(C)cc(F)cc2)C=CC1 c1(OC)ccc(C#N)c(NC(c2cc(-c3cnn(CCN(C)C)c3)[nH]n2)=O)c1 Cc1ccc(C(=O)NC(C)CCNC(C2(CC(F)F)CCC2)=O)cc1Cl N1(C(C(C)OCCOC)=O)CC2CCC(N(C(=O)Cc3cncs3)C)C2C1 C1(C(C)C)C(=O)NCCN1Cc1cn(C)nc1C(F)F O=NN1CCCC1C(=O)NCCC1CC(NC(C23CC(F)(C2)C3)=O)C1 Cc1noc(C)c1C(C)CC(=O)N(C1CCN(C(=O)CCC2CC2)C1)C C1(C(=O)NCCC2(NC(COc3cc(C)on3)=O)CCCC2)CC(=O)N(O)C1 N1(Cc2cn(CCC)nc2)CCSC(C(=O)Nc2ccnc(OC)n2)C1 N1(C(c2ncn(CC)c2)=O)C2CCC1(CNC(=O)CC1CCCC(F)(F)C1)CC2 N1(C(c2c(C)ocn2)=O)CC(O)CC1C(=O)Nc1ccccc1CC#N c1(N2CC(C(=O)Nc3c(OC)nccc3C)SCC2)ncnn2ccc(Br)c12 n1(C(C)C)ncc2cc(C(=O)N(C3CN(C(c4cnsn4)=O)CC3F)C)cnc12 c1(C(=O)NC2CC(NC(Cc3c(C)cccc3)=O)C(O)C2)c(Cl)ccc(F)c1N C(=O)(C1=CCCSC1)NCC1CC(N(C(=O)CCCNS(C)(=O)=O)C)C1 C(=O)(C1=CCCOCC1)N(C1CCCC1)CCNC(C1CCCS1(=O)=O)=O CCC(CC)CC(=O)N1CC2CC(NC(C3CCN(C(=O)NCC)C3)=O)C2C1 CC1=CCN(CCNC(=O)CCCCNC(C2CC2C2CC2)=O)CC1 N1(C(CN(C)C(=O)C2CC2)=O)CC2CCC1C2NC(=O)COC1(C)CCC1 Cc1ccc(Br)c(CC(=O)NC2CC2C(=O)NC2(c3cc(C)on3)CC2)c1 c1(C(N(C2CCN(C(C(CC#C)C)=O)C2)C)=O)ncc(C(=O)OC)cc1Cl C(=O)(CC(C)C(C)C)N1CC(CNC(c2nc(C)n(C)c2)=O)C(C(F)(F)F)C1 C1(OC)CCCCC1C(=O)NCC(C1CCCC1)NC(=O)C=CC1CCCC1 c1(C(=O)NCCCOCC(C)(C)NC(C2CC(C)OC2)=O)cnc([N+](=O)[O-])n1C CC1CC(c2ccccc2)CCN1C(c1occc1C(=O)OCC1CCCC1)=O N1(C(c2c(N)cncn2)=O)CCCCC(CNC(C2C3CCCOC23)=O)C1 C=CCC(CNC(C1(CF)CCOCC1)=O)C(=O)N(CC)Cc1ccc(Br)cc1 C1(c2cn(CC(=O)N(CC)CC)nn2)CN(C(=O)CN2CCCCCC2)CCO1 Cc1cc(I)ccc1C(=O)NC1CC(NCc2c(Cl)ccnc2Cl)C1 c1(NC(CCC)C)ncccc1S(=O)(=O)NCC1CCC1.N1S(=O)(=O)N1 C1(CC)CC(C(N2CCC(CCO)CC2)=O)CCN1C(c1cccc(O)c1F)=O Cc1ccc(CC(=O)NC2CC23CCN(C(C2CCC(C)C2)=O)C3)cc1F N1(C(=O)C(c2ccccc2)O)CCCN(C(C2(F)CC=CC2)=O)CCC1 C1(C)(C(=O)NC(C)C)CCCN1CC1CCC(C(F)(F)F)CC1 C(C(=O)NCC1(C(N2CCC2CC(C)C)=O)CC2(CC2)C1)(C(C)C)OCC C1(CNC(c2nc(C(C)OCC)sc2)=O)CC2(C1)CN(C(=O)Cc1csnn1)C2 N1(C(c2c(C)snn2)=O)CCCCCC1CNC(C12CCC(C(F)F)(CC1)C2)=O Cc1cnc(NCC(C)NC(c2nn(C)c(Cl)c2Cl)=O)nc1S(C)(=O)=O C1(CNC(CN(S(C)(=O)=O)C)=O)CC2(CCN(C(c3ccncn3)=O)C2)CO1 Cc1ccc(SCCCCc2cn(CC(=O)NCC3CCCC4CC34)nn2)cc1 CC(F)CC(=O)NC(C)(C)COCCCNC(C1CCCN1C1CC1)=O C1(F)(CNC(C=CCOCCOC)=O)CN(C(=O)C(C)(C)c2ccsc2)C1 Cc1cccc2sc(C(=O)NC3CCC4CC3CN4C(=O)CCCC#N)c(Cl)c12 c1(NC)snc(C)c1C(=O)N(C1CCCC(NC(=O)Cc2n[nH]c(C)n2)C1)C C1(CCNC(c2n(CC)ncn2)=O)COCCN1C(=O)CCOCCCOC Cn1ccc(=NC(=O)C23CC(CN(C(C4CC4(C)C)=O)C2)C3)[nH]1 n1(CC(N2C(C)CCC(NC(=O)CCC(F)F)C2)=O)cc2ccccc2n1 N1(C(c2nncc(NC)c2)=O)CC2CCC1C(C(=O)NCC1CC(C(=O)OC)C1)C2 C=CCC(C(=O)N1CC2(CC(CC(=O)NCC3CCOC3=O)C2)C1)C(C)C N(C)(CP(C)(C)=O)C(C1C(NC(c2cnc(C)o2)=O)C1(C)C)=O Cc1ccccc1C(C)CC(=O)NC1CCC1CNC(c1c(C)cnn1C)=O C(=O)(C1CCCc2nn[nH]c21)NC(CCOC)CNC(=O)CCC1CCCC1 c1(C(=O)NC(CCCNC(C(CCSC)OC)=O)C)nc(C)c(C)nc1O CC1CN(C(C)C)CCCN1CC(=O)CC1CC(C)(C)N1c1cnc2[nH]cncc1-2 N1(C(CN2CC(C)(OC)C2)=O)CC2CCC1C(NC(=O)Cc1c(Cl)cnn1C)C2 C1(CNC(C2C(CC)C2)=O)CCN(C(c2ncccc2F)=O)CCC1(F)F C12(CNC(C(CC)(C)C)=O)CCCC1CCN2C(=O)CNC(=O)C(CC)CC c1(SC)cc(C(=O)NC2CCC(N(C(=O)CC3(CO)CC3)C)C2)ccc1F c1(C(=O)NCC(CC=C)NC(=O)C(CO)N(C)C)cnc(C(N)=O)cn1 C12(C(N(CC)CC3CCC3)=O)CCC(NC(=O)Cc3ccccc3F)(CC1)C2 O(N1CCC(N=c2cc(C)[nH]c(-c3cccs3)n2)CC1)CC N1(Cc2ccn(CC=C)c2)CCC(O)C(C(=O)NCCCc2ccccc2F)C1 c1(OCC)c(Cl)cc(C)nc1C(=O)NCC1CCN1C(=O)Cn1ncnn1 C1(C(=O)NCCCCC(=O)N2CC(C(CC)C)C2)CC12CCOCC2 Cc1nc(C=CC(N2CCCC2CNC(C2CC(C)(O)C2)=O)=O)[nH]c1C C(CC(C)(C)CC(=O)N1CCCCC1CC(N1CC2CC(F)CC2C1)=O)OC C(C(CC1CCCCC1)CO)NC(=O)C(N1CCC(OCc2cccnc2)C1)=O Cc1ccc2oc(C(=O)NCC(C3CC3)NC(=O)C(C)C(C)(F)F)c(C)c2c1 CC1=C(C(=O)NC(CC(=O)N2CCSC(C)CC2)C(F)F)COCC1 N1(C(C(N2CC(C)C2)C)=O)CC2CC(O)C1C2NC(=O)CCN1CCCCC1 CCCC(C#N)C(=O)N1CCN(C(CNC(c2cc(C)c(C)o2)=O)C(F)F)CC1 c1(CCOC)nc(=NC(C)C2CCN(C(C3COCCN3C)=O)C2)s[nH]1 c1(C(=O)NC(CN(C(=O)C(C)CC2CC2)CC)C)ccc(OC)cc1Br N1(C(c2c(C)ocn2)=O)CC2CC2(NC(c2ccc(SC(F)(F)F)o2)=O)C1 c1(OC)cc(C(=O)NC23CC2CN(C(=O)COCc2ccccc2)C3)ccc1C N1(C(c2nc(COC)oc2)=O)CCCC(CCNC(C2CC3(CC3)C2)=O)CC1 N1(C(C2(C#C)CCC2)=O)CCC(C)C(N(C)C(C2CC2c2cnccc2C)=O)C1 S(=O)(=O)(c1cccnc1N1CCC(C#N)C1)NCC1OCCN(C(C)(C)C)C1 N1(C(c2c(OC(C)C)n[nH]c2)=O)CCCCC1CNC(C1CC2CC2C1)=O Cc1nc2cc(Br)cc(NC(c3ccc(Cn4cccn4)o3)=O)c2o1 c1(C(N2C(C(=O)Nc3c(C#N)scc3)CCCC2)=O)c(Cl)cccc1Cl N1(C(c2cc(COC)[nH]n2)=O)CC2CCC2(CNC(=O)CCC(C)N(C)C)C1 c1(C(=O)NC2C(OC)CN(C(=O)C(F)C3CCC3)C2)cc2cccc(F)c2s1 C(=O)(C(c1cccs1)=Cc1cccs1)NC1CN(C(C2CCN(CC)C2)=O)C1 N1(C2CCN(C(C(F)=CC)=O)C2)CCN(C(C2OCCC2C(C)C)=O)CC1 CC1OC2(CNCC(c3cccc(Cl)c3)O)CC1(CO)C2 c1(C(=O)NC(c2ccccc2F)CNC(c2ccc(C)s2)=O)cncc(N)c1 CC(C)(CC(=O)NC1CN(C(C2CCN(C(N)=O)CC2)=O)C2CC12)c1cccs1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1CC2CCN(C(c3cn(C)nn3)=O)CC2C1 c1(OC)cc(NC(C2C3CC2N(Cc2scnc2C)C3)=O)cc(F)c1 C(=O)(CCCCC(C)C)NCCC(=C)CNC(c1c(Cl)sc(C)c1C)=O C1=CC(=O)NC1(C)C.C1(=O)C(C2CCOC2)N1.C1(=O)CC2(CC2)N1.CO.OC N1(C(C2CCN(C(CC3(OC)CCC3)=O)C2C)=O)CC2(CNC(=O)OC2)C1 CC(C)(C)C(C)(C)C(=O)N1CCC(=CCNC(C2Cc3nccn3C2)=O)CC1 Cc1cc(C)c(S(=O)(=O)NCc2ccc(F)c(S(N)(=O)=O)c2)cc1[N+](=O)[O-] c1(OC)ncccc1CC(=O)NCC(C)NC(C1(C)CC2CC2C1)=O N1(C(C2CN(C(c3c(C)ccnc3)=O)CC2(F)F)=O)CCSC2(CCC2)C1 C12(N(C(C(Cc3ccc(C)cc3C)C#N)=O)C)C3C4C1C1C2C3C41C.C1CN1 CC(C)CC(C)C(=O)NCC1(O)CC(CNC(c2csc(Br)c2)=O)C1 C1(CNC(=O)Cc2ccsn2)C2CN(C(C3CC3c3cccc(Cl)c3)=O)CC12 Cc1cnc(C(N2CCC(CCNC(C3(c4ccsc4)CC3)=O)CC2)=O)c(F)c1 c1(OCC(N2C(C(=O)NCC3(C)CCC3)CCC2)=O)ccc(C#N)cc1 N1(C(CNC(C(CC)C)=O)=O)CCN(C(c2coc(C3CC3)n2)=O)CC1C C1(CC(=O)NCCC(C)N2CCCC2)CN(C(C2CCCC(=O)N2)=O)C(C)(C)C1 c1(C(=O)NC2CCC(CNC(C3CC(CC)C3)=O)C2)nccc2ncccc12 C(CNC(=O)C(c1ccccc1)O)(CC(F)(F)F)NC(C1N(C(C)=O)CCC1)=O N1(C(COC)=O)CC(NC(=O)CC(C)(C2CCC2)N(C)C)C2(CC2)C1 N1(C(C(C)=C2CCC2)=O)CC2CC(NC(=O)C(C)(C)c3cncnc3)C2C1 CCCS(=O)(=O)CC(=O)NCC12CN(C(=O)C(C)(C)n3cccn3)CC1CCO2 N1(C(C2C(C)=C2)=O)CCOC(C(C)NC(C2CC3C=CC2C3)=O)C1 C12(CNC(C3(C#C)CC3)=O)CCC1CCN2C(=O)Cc1ccc(C#N)cc1 c1(CC)cc(N2CCC(C(C)NC(c3oc(C(F)(F)F)nc3C)=O)C2)ncn1 CC1CCSCCN1C(C1(NC(C2CCCC2O)=O)CCC(C)(C)C1)=O c1(CC)oc(C)cc1C(N1CCCC(CNC(c2ccc(C3CC3)cc2)=O)C1)=O C1(CC=C)(C(=O)NC(C)CN(C(C2CC(OCC)C2)=O)CC)CCC1 N1(C(C(C)NC(N(C)CC)=O)=O)CCCC(C(=O)NCCCc2ccccn2)CC1 c1(N2CCOCC(NC(c3c(C(C)C)cccc3)=O)C2)c(Br)cccc1[N+](=O)[O-] C#Cc1cccc(C(=O)NC2CCCC2NC(=O)CCCN=[N+]=[N-])c1 C1(CC)(CC)CC(NC(c2nnc(S)n2C)=O)CN1C(=O)CC1CC1(C)C n1(CC(=O)NCCN(C(=O)C(O)C(C)CC)CCCCCC)c(C)c(C)sc1=O C(=O)(CC(=O)N(CCCNC(C1(C(=O)OC)CC1)=O)C)C1(C(C)C)C(C(=O)OC)C1 n1(C(C)C)cc(C(=O)NCC2CCN(C(c3coc(C(F)F)n3)=O)C2)ccc1=O CC1CCN(C(c2ccccn2)=O)CC1NC(C1CCN(CC2CC2)CC1)=O C1(CNC(=O)NC(c2ccccc2Br)CC)(OC)CCC(C)C1 N1(C(=O)OC(C)(C)C)CCOCC(NC(=O)NCC(c2ccc(Br)cc2)O)C1 O=C1CCC(CCC(N2CCCC(CNC(c3ccsn3)=O)C2)=O)CN1 c1(CC)ccc(C)c(NC(=O)C(F)C(C)CNC(=O)C(=O)NC2CC2)c1 N1(C(C2C(c3cn(C)nc3)C2)=O)CCCCC12CC(NC(=O)CC(F)(F)F)C2 CN1CCC(C(=O)NCCC2CCC3CC23)(NC(C2(C(=O)NC3CC3)CC2)=O)C1 N1(C(C(CC)(C)O)=O)CCCC2(CCN(C(=O)CC3CCCC34CC4)CC2)C1 c1(COCC(=O)NC(C2CCCC2)CNC(C2(CC)CC2)=O)cccc(Cl)c1 c1(N(CC(C)CO)C)nc(N2CCCNC(=O)CC2)nc2ncn(C)c12 CC12CN(C(c3cc(Cl)c(F)cc3O)=O)CC1C1C=CC2C1 N1(C(c2ccc(CC)o2)=O)CCCCC1CC(N1CCC(C)(F)C1)=O c1(OCC=C)ccc(C(=O)NCC(CO)NC(=O)C(C(C)C)NC(C)(C)C)cc1 C1(C(=O)NC2C3OCC(NC(=O)CC(F)F)C3OC2)CC(C2CCOCC2)=NO1 C(=O)(CC1=NNC(=O)C1)NCC(OC)OC(C1CC(OC(F)F)C1)=O CCCC#CC(C)(C)NC(=O)C(C)NC(=O)C(C)n1cccn1 C(=O)(CS(=O)(=O)CCOC)N1CCC(NC(C(COC)OC)=O)C1C1CC1 c1(C(C)NC(C(CC)SC)=O)ccc(CNC(c2c[nH]nc2F)=O)cc1 C1(C(N2C(C)CN(C(c3cccn3C)=O)CC2)=O)CC(c2ccncc2)=NO1 c1(CC)ccccc1C(=O)N(C1CN(C(=O)CCN(C(CC)CC)C)CC1F)C C1(C(=O)NC(c2ccccc2)C(C)NC(C2CC(C#N)C2)=O)CC12CCOCC2 C1(C(=O)NCC(CN(C(c2cc(Cl)c[nH]2)=O)CC)(C)C)C(F)(F)C12CCC2 N1(C(Cc2ccc(OC)cn2)=O)CCC(C)(C)C(CNC(=O)C(O)C(F)F)C1 O(NC(=O)CN=c1ccnc(N(CC(N2CCCC2)C)C)[nH]1)CC.N(CC)CC n1(CC)ncc(Cl)c1C(=O)NC1CC(F)(CNC(=O)C(c2ccc(Cl)s2)=O)C1 c1(CCN2CC(C(CC)CC)C(C(F)(F)F)C2)ccc([N+](=O)[O-])cc1F CC1CC=CCC1C(=O)N(CC(O)CN(C)C(c1ccc(OCCF)cn1)=O)C c1(C(N2CCN(C(COC(CC)C)=O)CC2C)=O)ccc2c(c1)nnn2CC c1(C(=O)NC2(CC(N3CCC(C)(O)C3)=O)CCC2)ccc2[nH]ccc2c1 c1(OC)cncnc1C(=O)NC(C(N1CCC(C)(NC(C)=O)C1)=O)C1CCC1 c1(CC)ccc(Cl)cc1C(=O)N(CC(CC)NC(=O)COC(C)C)C c1(C(=O)NCC(C)CNC(=O)C(C)(C)c2ccno2)ccc2nccn2c1 C1(NC(COC(C)C)=O)CC2CCC1N2C(=O)C(O)Cc1cccc(Cl)c1 c1(C(=O)NCCCN(C2CCCC2)C(C2CCC(=O)N2)=O)ccccc1F c1(-c2cnc(OCC)nc2)cccc2[nH]nc(C(=O)NCCc3nn[nH]n3)c12 c1(CC(N2CC(N(C)C(c3cc(Br)no3)=O)C2)=O)ncc(F)cc1F N1(C(CSCCCC)=O)CCC(C(=O)NC(C)C)C12CC2 Cn1cnc2ccc(C(N3CCCCC(CNC(=O)C(O)CC(N)=O)C3)=O)nc12 CCCCCC(F)C(=O)NCCNC(c1cc(O)ccc1F)=O C(=O)(CN=S(C)(C)=O)NCc1c(CN(C)C(C2(CO)CC(F)(F)C2)=O)cccc1 C12(NC(C3C(C)CN(C)C3)=O)CCC(CC1)N(C(c1cc(Cl)no1)=O)C2 C1(CC)CN(C(=O)C=C2CCCCC2)CC1NC(=O)C(F)CN(CCOC)CC c1(C(=O)NCC2(NC(c3ccncc3Br)=O)CCC2)cc2cccnc2cn1 N1(C(C2CC2[N+](=O)[O-])=O)CC2CC(C1)N(C(c1ccc(-c3cccnc3)s1)=O)C2 c1(C(=O)NC(CNC(COCCOCC)=O)CC)c2n(c(=O)n1C)CCCC2 Cc1cnc(C(=O)NC(C)(CNC(c2onc(C)c2C(F)(F)F)=O)CO)cc1C CC(C)CC(c1nnnn1C1CCCC1)NCc1csc(Cl)c1 N1(C(Cc2cccc(C#C)c2)=O)CCC(F)(F)C(CNC(c2sccc2C)=O)C1 N1(C(c2c(CC)nccn2)=O)CCC2C(CCCN2C(=O)C(C)CSC)C1 C1(NC(CCCOC)=O)CC2CCC(C1)N2C(c1ncsc1C(F)(F)F)=O c1(C(=O)NC2C(CNC(C(C)CF)=O)CC2)ccc(C(F)(F)F)nc1 CC(C)CC(=O)C(=O)N1CC2C(NC(=O)COc3ccsn3)C2C1 CCC(C)C(O)C(C)C(=O)NC(COC)CC(=O)N(C)CCN1CCCC1=O C(=O)(C(F)(F)C(F)(F)F)NC(C1(O)CCN(C(C2CCC(C)(C)CC2)=O)C1)C c1(CC(=O)NC2CC(C)N(C(=O)CCN3CCC3)C2)cc2cc(Cl)ccc2[nH]1 C(=O)(CC(C)C(=O)N1CCCC(NC(=O)C(=O)NCC(F)F)C1C)OC CC(CC(=O)N1CCCC(C)(CNC(=O)CC2CC3CCC2O3)C1)P(C)(C)=O Cc1cc(F)ccc1C(N1CC(=O)CC1C(N1CCC(F)CC1)=O)=O C#Cc1ccc(C(=O)NC2CCCCC2CNC(=O)C2=CCC2)nc1 C#Cc1ccc(F)c(C(C)NCC2CCN(c3ccc(F)cc3F)C2)c1 c1(C(=O)NCC2CCN(Cc3cccc(C)n3)C2)ccc(Br)nc1Br CC(C)(C)CCC(=O)NCC12CC(NC(C3CCCN3C3CC3)=O)(C1)C2 c1(CC(=O)NC2CC(C)N(C(=O)CP(C)(C)=O)CC2)cn(C)c2ccccc12 c1(COCC(=O)N(CCNC(=O)C(F)OC(F)(F)F)CC)ccc(F)cc1 N1(C(C(C)Cn2ccnc2)=O)CCC(CO)(CNC(=O)Cc2cn(C)cn2)C1 Cc1ccc(SCC(N2CC3CCC3(NC(=O)C(O)C3CC3)C2)=O)c(C)c1 C12(C(=O)NCC(C)OCC#C)COC(C1)C(NC(=O)C(C)NC(C)(C)CC)C2 Cc1cc(=NCCCC(C)(C)NC(=O)C=Cc2ccco2)[nH]c(C2CCC2)n1 CCC(CC)C(=O)NCC(=O)NC(C)CCNC(=O)C(C)(CC)OC CC(C)C(CNC(C1CC2COCC2C1)=O)C(=O)N1CCCC1CN(C)C c1(C(N2CC3C(NC(CN(CCC)C)=O)(C3)C2)=O)cc(Cl)cc2c1CCC2 n1(C(C)C)nc(-c2ccc(N)cn2)nc1C(C)Sc1nncn1C CC(N=c1nc(N2CC(=O)NC(C)(C)C2)c2ncccc2[nH]1)c1ccoc1 C1(C(=O)NCC2(O)CC(NC(C34COCC3C4)=O)C2)CCC2(CCCCC2)CC1 C1(NC2(CC(=O)OC)CCCOC2)CC2(CCCCCC2)C1 c1(OC)ccc(CNC2CC2C(=O)NCC2CCC(O)CC2)c(OC)n1 CCC(C(=O)NCCOCCNC(=O)Cc1c(C)nn(C)c1Cl)C(C)(C)CC C(=O)(C(C)(C)N=[N+]=[N-])NCc1c(C(=O)NCCc2nc(C)[nH]n2)occ1 C1(NC(CCC2CC(OCC)C2)=O)CCC(CC(=O)Nc2cnn(C(F)F)c2)C1 C(=O)(CC1=CCCC1)N(C1CCCN(C(C(C)OCC(C)C)=O)C1)C N1(C(C2C3(CC(OCC)C3)C2)=O)CC(NC(C2CC3CC3C2)=O)CC2(CC2)C1 C1(CNC(C(C)CC(F)(F)F)=O)CCCC2(CN(C(=O)CC3CC(C)(C)C3)C2)O1 CCCCC(O)C(C)C(=O)NCC(C)=CC(=O)NCc1cnc(C)s1 Cc1ccc(F)c(C(=O)NCC2CCCC(NC(=O)CN(C)C(=O)C3CC3)C2)n1 c12ccc(cc1)[nH]c2=O.c1(C(N2CCC(CO)C2)C(=O)OCC)cccc(F)c1 CC(=O)CCCC(=O)NC(C)(CNC(=O)CCCc1nncn1C)CO CCCC(F)C(=O)N1CCC2CC12C(=O)N(C)Cc1ccncc1 c1(CCC(=O)NCC(CNC(=O)Cc2noc(C(C)C)n2)OC)cncnc1O CC(C)C(O)C(F)(F)C(=O)N(C)CC1CCCC1NC(=O)C(C)Cc1cnco1 C1(CN(C(COC(CC)CC)=O)C)CCCN(C(=O)CCCC2(NC)CCC2)C1 c1(C2(NC(C3CC(O)(c4cccnc4)C3)=O)COC2)cccc(Cl)c1 C(=O)(CCP(C)(C)=O)NCCC1(O)CCN(C(Cn2cc(CN(C)C)nn2)=O)C1 C(CCCCCCCO)=CC(N1CC(CNC(C(C(C)C)OC)=O)N(C)CC1)=O C(N=c1cc[nH]c(-c2nccs2)n1)C1CN(C(=O)NC2C(C)(C)CCC2)C1 c1(C(C)OC)nc(C)c(S(=O)(=O)N2CCCCC2C(=O)OC)s1 Cc1ccc(C(=O)NC2CCC(C(=O)N(CC(C)C(C)(C)C)C)CC2)nn1 C(N=c1ccn2nccc2[nH]1)C1CCCN(Cc2c(OC)cccc2F)C1 c1(OC)ccc([N+](=O)[O-])c(C(N2CCN(c3ccc(S(N)(=O)=O)cc3)CC2)=O)c1 c1(C(N2CC(C)(C)C(C(=O)NCC3(C)CC4CC4C3)C2)=O)c[nH]c2cnccc12 N1(C(C(CC)OC)=O)CCCCC(C(=O)NC2CC2(C)C)C1 C1(NC(C(CCCC)O)=O)COC2(CCN(C(c3cncs3)=O)CC2)C1 Cc1ccc(C(C)NC(=O)C(CNC(=O)C(O)C2CCCC2)N(C)C)nc1 Cc1nc(C(N2CCN(C(C3(Cl)CC3(F)F)=O)CC(C)(F)C2)=O)c2ccnc-2[nH]1 c1(CCC)cccc(OC(c2ccnn2Cc2ccccc2)=O)c1 C(=O)(C1CCc2c[nH]nc21)N1CCC2(C(NC(c3n(C)c(S)nc3)=O)C2)C1 C(=O)(C(C)CCO)NCC(C1CCCC1)NC(CN1C(C)CC1)=O C1(CNC(=O)Cc2csnn2)CCN(C(C2CCC(=O)N2C2CC2)=O)C12CCC2 c1(C(=O)NCC(CNC(CSCCC)=O)F)cnn(CCF)c1 C1(C2(NC(CC(=C)Br)=O)CC2)CCCCN1C(c1ccccc1SC)=O c1(C(=O)NCCOC(CNC(CC2N(CC)CCC2)=O)(C)C)ccc(C)n1C c1(OC)cc(C)c(CCC(=O)OC(CC(F)(F)F)c2ccc(F)cc2)c(C)c1 N(C1CCCc2cc(N)ccc21)C(Cn1cc(OC)c(=O)cc1C)=O C1(CC)CCN(C(=O)CN2CCOC2=O)C1CNC(C1CC(N(C)C)C1)=O c1(OCC)cc(C(N2CCS(=O)(=O)CC2)=O)c(-c2cc(O)cc(F)c2)cn1 Cc1cc(CNC2CC(NC(C3CCCO3)=O)C2)cc(C)c1Cl N1(CC)CCOCC1CC(=O)NCC1(NC(C2CCCC(C(=O)OC)C2)=O)CC1 N1(c2ncc(C)cn2)CCOCC(CNC(=O)CC2CCCCCC2)C1 c1(C(CNC(C2C(C)C2C)=O)NC(=O)C=CCN2CCOCC2)ccccc1F N1(C(C(C)C(C)O)=O)CCCC(C)(NC(=O)C=Cc2cccc(Cl)c2)C1 c1(C(=O)OCc2c(C)ccc(OC)c2)ccc(=NCCN(C)C(C)C)[nH]c1 C1(C(N2CC(C(N)=O)(CNC(c3cc(CC)[nH]n3)=O)C2)=O)CCCC(NC)C1 C1(NC(c2cc(OC)nn2C)=O)CS(=O)(=O)CC1NC(=O)C(C)(C)c1ccns1 c1(NC(c2n(C(C(=O)OC)C)nnn2)C2(SC)CCC2)ccc(C)c(C#N)c1 CCC(CC(=O)NCC1CC(C(=O)NC(C)Cn2ccnn2)C1)OC C12(CC(=O)NCCNS(CC)(=O)=O)CCC1CN(C(=O)C(C(C)C)N(C)C)C2 S(=O)(=O)(CC(=O)N1CCC(O)(CN(C(=O)COCc2cccc(C)c2)C)C1)NC Cc1nc(N2CC(O)(CCNC(c3ccco3)=O)C2)cc(-c2ccco2)n1 Cc1cncc(C)c1C(=O)NCc1cn(C2CN(C(=O)C(O)P(C)(C)=O)C2)nn1 C1(C)(COC)CC(NC(=O)C2=CCCC2)CN1C(=O)Cc1ccc(Cl)s1 C1(CNC(c2cnc[nH]2)=O)CC2CCC(C1)N2C(=O)C=Cc1ccccc1 CCCCCCCCNC(=O)C(=O)NCC(c1ccc(OC)c(OC)c1)C C(=O)(C(F)C(C)C(F)(F)F)NCC(CNC(c1cc(C)c(C)s1)=O)O CCCCCC(O)C(C)C(=O)N1CC2CC(NC(C3COCCN3C=O)=O)C1C2 c1(C(N2CCC3CN(C(CCC(C)C#N)=O)CC32)=O)ccc2cccc(F)c2n1 C(=O)(C(O)C(F)(F)F)N1CCC(CNC(c2ccc(CC(C)C)s2)=O)C1 C1(N(C)C)CCCC(C(=O)NC2CCCN(C(C34CC(CF)(CO3)C4)=O)C2)C1 c1(C(n2cc(C3(N(C)C)CN(C(=O)CC(=O)O)C3)nn2)C)nc2ccccc2o1 c1(C(=O)NC(CNC(C(C)NC(=O)NC)=O)C(C)C)cc2ccccc2oc1=O C=CC1(C(=O)NC(C)CC2CCCCC2)CCN(C(=O)C=C2CCCCC2)CC1 CC1(C)CN(C(=O)C=CC2CCOCC2)CC(CNC(=O)C(C)(C)CF)O1 c1(OC)cc(CC(=O)NC(C)CCNC(C2(CSC)CCC2)=O)cc(Cl)c1 C(=O)(C(CC(C)C)C(N)=O)N1C(C(N2CC(F)=C(C)CC2)=O)CCCCC1 C1(O)(CN(C(C2C(CCC)C2)=O)C)CCN(C(=O)CNS(=O)(=O)C2CC2)C1 N#Cc1cnccc1COC(=O)C=Cc1cccc(-c2ccc(Cl)cc2)c1 O=C1C2CCCCCCCC2=NN1c1cc(Cl)cc(Cl)c1 C(S(=O)(=O)CCNC(N1CCC(C(=O)O)C1)=O)c1cn(CCCC)nn1 c1(OCC)ccccc1CC(=O)NCC#CCNC(C1(C(=O)OCC)COC1)=O C1(CNC(C(CO)N(C)C)=O)CCC(CNC(C2(C)CC=CCC2)=O)CC1 C#CC1(C(N2CCC(CCO)C2)=O)CCN(C(=O)CC(C2CC2)C2CC2)C1 N1(CCOC)CCC2(CCN(C(=O)OCc3ccc([N+](=O)[O-])cc3)C2)C1 C1(C)(NC(c2cccc(OC)c2)=O)CCC(NC(=O)Cc2ccccc2Cl)CC1 c1(-c2c(C3(C(=O)OC)CC3)cccc2)cc(OC(C)C)c(F)c(F)c1 c1(CCC)cc(C(=O)NCCOCCNC(C2CC(C#N)C2)=O)c(C)o1 c1(C(N(C)CCN(C(=O)C(C)(C)c2ccccn2)C)=O)cnn(C)c1N c1(C(N2CC(NC(CC(C(C)C)C)=O)C3C2CCC3)=O)cccc(C#CCO)c1 c1(C(=O)NCC(C)CN(C(=O)CCC2(C#N)CCC2)C)sccc1Cl N1(C(c2cn(C)nn2)=O)CCC(C2CCCN(C(c3ccc(F)nc3)=O)C2)C1 Cc1ccc(C#N)cc1C(N1CCC(C)C(CC(=O)NC(CF)C(F)(F)F)C1)=O c1(OCC)cc(CCC(=O)N(CCCCCN)C)on1.c1(C2CCC2)ccc(C)s1 N1(C(C(=O)NC)C)CCCC(NC(=O)CC(C)OC)CC1 N1(C(CCC=CCC=C)=O)CCC(CNC(c2scc(C)c2C)=O)(OC)CC1 CC1(C)CCOC(C(=O)N2CCC(C(=O)NCc3cc(C(N)=O)no3)O2)C1 C1(C(=O)NC2C(C)COCC2)CC2C=CC1N(C(C1Cc3nccn3C1)=O)C2 N1(C(C(C(C)C)SC)=O)CCC2(CCC(NC(C3(F)CC=CC3)=O)C2)CC1 C1(C2(O)CCOC2)(C(=O)NCC(C2(O)CCN(C(=O)CC(C)(C)O)C2)C)CC1 c1(C(=O)NCC(CCNC(C(C)OCC)=O)O)ccnc2ccncc12 C(=O)(CCCC(=O)N(C1CCCN(C(c2coc3c2COC3)=O)C1)CC)NCC S(=O)(=O)(c1ccc(C(=O)N(CCC(C)NC(=O)C(O)CCSC)C)cc1)NC N1(C(C(CCC)c2ccccc2)=O)CCCC(F)(CNC(=O)C=CC(F)(F)F)C1 c1(C(=O)NCC(CNC(=O)CC2COC(=O)C2)OC)ccc(F)c(F)c1 N1(C(C2N(CC(C)C)CCC2)=O)CCC(O)(CNC(=O)CCc2cnoc2)CC1 c1(C(N2CC(N(C(CCCC)=O)C)C(C)(C)C2)=O)cnn2c1OCCCC2 N1(C(C2(C(C)C)CCCO2)=O)CC2CC1CN2C(=O)CNS(C)(=O)=O C1(C(=O)N(CC(C)C(C)C)C)(CC)CCCN(C(c2ccc(C(C)C)o2)=O)C1 c1(C(N2CCC(NC(CCc3cn(C)nn3)=O)C2)=O)c(C(F)(F)F)cccc1O c1(CC)nn(C)cc1C(=O)NC1CN(C(c2sccc2C(C)(C)C)=O)CC1C N1(C2CCC(NC(CCOC)=O)C2)CCN(C(=O)CCN2CCC(O)CC2)CC1 N1(c2c(C)c(NCc3ncsc3Cl)ncn2)CCC2(CCCN2C)C1 N1(C(c2cnn(C)c2Br)C(=O)NCC2CCCO2)CCC(C(F)(F)F)C(F)(F)C1 CC1(C(=O)NCC2C3CN(C(=O)Cc4cnco4)CC23)CNC(=O)C1 Cc1ccc([N+](=O)[O-])c(C(=O)NC2CN(C(C3CC4CCC4C3)=O)CC2O)c1C N1(C(=O)Cc2ccc(Cl)cn2)CC2CCC(C1)N2C(C1CC1F)=O C1(N2CCC(COC)C2)CCC2(CC1)CN(C(c1c(F)cccc1Br)=O)C2 C12(CNC(=O)Cc3ccon3)CC(C1)C(NC(=O)COC1CC=CC1)CO2 C1(C(N2CC(C3CN(C(c4csc(O)n4)=O)CCO3)C2)=O)CCN(CCF)CC1 N1(C(CN(C2CCC(C)CC2)CC)=O)CCC(C2CCCN(C(C)C(N)=O)C2)CC1 Cc1cccc2nc(C(=O)NC(C)(C)CCN(C(=O)C3=COCCC3)C)cn12 C1(C)(C(=O)NC2C(C)(C(C)C)C2)CCCN(C(C2CCN(S(C)(=O)=O)C2)=O)C1 C(=O)(C(O)CCCNC(C1CC(C)N(C)C1)=O)N(CC(=C)C)C C1(C(=O)NCC2C(NC(=O)Cc3ccno3)CCC2)Cc2cccnc2C1 CC1(C)C(CNC(C2CCCO2)=O)CCN1c1ncc(O)cn1 N1(C(CCNC(COC)=O)=O)CC(N(C)C(C2CC23CCCC3)=O)C(C)(C)C1 N1(C(Cc2ccc(C)cc2)=O)CC2CCC2(CCNC(c2ccc(C)nn2)=O)C1 N=c1[nH]c2ccc(C(N3CCC(NC(=O)C#CC4CC4)CC3)=O)cc2[nH]1 N1(C(C#CC(C)(C)C)=O)CC23CCCCC2(C1)CN(C(C1CC(C#N)C1)=O)C3 N1(C(c2cncc(CC)c2)=O)CCC2CCC(C1)N2C(=O)CC(=O)OC CC1c2c[nH]nc2CCC1C(N1CCCCC(CNC(=O)Cc2ccns2)C1)=O N1(C(c2ccc(C=O)s2)=O)CCC2(CCC(C(C3CCCCC3)=O)O2)CC1 C1(NC(c2cc(CNC(C3(CC)CCC3)=O)ncc2)=O)CN(C)CC1(F)F c1(N2C(C=O)CC2)c(CNCC)noc1C.c1(C(=O)NCC)nsc(OCC)n1 Cc1nc(N(C)C)sc1C(=O)NC1CC(CCNC(=O)C=CCO)C1 c1(C(N2CCCCC2CF)C(=O)NCCC2(C)CC2)cccc(Br)n1 N1(C(CCS(C)(=O)=O)=O)Cc2ccc(-c3cc4cc(F)ccc4[nH]3)cc2C1 c1(C(N2CC(O)(C(C)NC(CC=CCC)=O)C2)=O)cccc(C)c1Br C1(NC(Cn2cc(SCc3c(C(=O)OC)csc3)nn2)=O)CCS(=O)(=O)C1 c1(OCC(C)C)ccc(SCC(N2CC(NC(=O)CNC=O)C3CC23)=O)cc1 N1(C(C(CC)COC)=O)C2CCC1C(C(N1CCC=CC1C(=O)OC)=O)C2 c1(C(CC(C)NC(=O)C#CC(=O)N(C)C)=O)ccc(O)cc1 C12(C(=O)NCCC(C)N(C)C(c3csc(-c4cnc[nH]4)n3)=O)CCC(CC1)CO2 CN1N=CC(CC(=O)NCC(C(=O)NCCN2CCNC2=O)N(C)C)C1=O C(=O)(C(C(C)NC(C1CCCC1O)=O)C(C)C)NCc1nccc(C)n1 c1(C(=O)NC(C)Cn2cc(CN3CC4CC4C3)nn2)c(Cl)nc2ccccn12 C1(C(=O)OC)CC2(CCC(CNC(c3ccc(-n4ccccc4=O)cc3)=O)O2)C1 CC1CN(C(=O)CC2CC3(CC3)CO2)CC1NC(c1cnc(O)s1)=O c1(C(=O)NCCOCCCN(C(c2cc(OCC)no2)=O)C)ccccc1C c1(CC)nnc(O)c(C(N2CCC(CNC(=O)C(O)CCC(C)C)C2)=O)c1CC CCCCCC(C)(C)C(=O)NCC(C)(C)CNC(C1CCCN(C(C)=O)C1)=O c1(OC(=O)NCC2(COC)CC2)cc(F)ccc1N1CCCCC1 CC(C)C(F)(CNC(c1ccccc1C#N)=O)C(=O)NCCN1CCOCC1C N1(C(c2c(C)ccs2)=O)CCC2(CC1)CN(C(=O)C(C)(C)N1CCCC1)C2 C1(CNC(CSCCC)=O)CCCC1C(=O)NOCCCCCC1CC1 C12(C(N(CCCNC(c3coc(C4CC4)n3)=O)CC)=O)CCCN1CC(OC)C2 N1(C(c2c(C)nncc2)=O)CCC(C)C(CC(N2CC3CC(C)C3C2)=O)C1 Cc1cccc(C(=O)NC2(CCCCNC3CC4CC4C3)CC2)c1 N1(C(CC2CC(C)N(C(C34CCC(C3)C4(C)C)=O)C2)=O)CC=CCC(C)(C)C1 c1(COC(=O)NC(CC(C)C(C(=O)OC(C)(C)C)OC)C)cccn2c(C)cnc12 c1(C(N2CC(C)(OCC(=O)NCC(C#C)CCC3CC3)C2)=O)nnccc1C C1(OCC(=O)N(C(C)C)CCN(C(=O)CCn2cccc2)C)CCCCC1 c1(C(N2CCC(CNC(C(C)N(C(C)=O)C)=O)C2)=O)cc2c(nn1)CCCO2 c1(C(N2CC(NC(C(C=CCCC)O)=O)C(C(F)F)C2)=O)c(F)ccc(F)c1Cl N1(C(CC2C(C)CCN(C(c3cc(C)nn3CO)=O)C2)=O)CCC12CCOCC2 C(=O)(CCCCNC(=O)C(C1CCCO1)NC(=O)C(c1ccccc1)C)OCC N1(C(CC(=O)OC)=O)CCC(O)(C(N2CC3C(C(=O)OC)C3C2)=O)C1 N1(Cc2nnc(C)o2)CC2(CN(C(c3ccc(F)c(O)c3)=O)CCO2)C1 c1(C(N2CCC(C)(NC(=O)C3=C(C#N)CCC3)C2)=O)cnn2c(Br)cccc12 CCS(=O)CC(=O)NCC1(F)CC(NC(c2cccn2-c2ccc(F)cc2)=O)C1 Cc1c(C2(CN(C(C34CC(CO3)N(C(=O)C(C)C)C4)=O)C3CC3)CC2)cccc1F C1(NC(c2csc(C)c2C)=O)CCCCCCC1NC(=O)CC1CCCN(C)C1 CCCC(C(=O)N1CC(CCNC(c2ccccc2SC(C)C)=O)C1)OC C(=O)(C(C(C)(C)C)c1cc[nH]n1)NCC(C)N(C(=O)CO)C C#Cc1ccc(Br)c(C(=O)NCCC2(O)CN(C(c3c[nH]nc3F)=O)C2)c1 N1(C(c2cn(CCC)nn2)=O)CC2OCC(NC(c3ncc(Cl)cc3Cl)=O)C2C1 c1(C(=O)NC2CC(O)(CNC(C3CCC3(F)F)=O)C2)ccc(F)cc1Br c1(CNC(N2CCC(C(=O)Nc3ncc(OC)nc3)CC2)=O)ccc(F)c(Cl)c1 c1(C(=O)NCCC2(O)CN(C(C3OCCN(C)C3)=O)C2)ncnc(O)c1F O=C(CCC(=O)c1ccc(F)cc1)NCC(CO)NC(C1CC2CC2C1)=O Cc1noc(C)c1CC(=O)NCC1C2CN(C(C3CC(=O)N3)=O)CC12 c1(CC)cncc(CC(=O)NCC2CN(C(=O)C=Cc3ccc(C(F)F)o3)C2)c1 C1(CN(C)C(=O)C2CC2)CC(NC(C=CC=CC)=O)CN1.n1(C(C)O)cnnn1 C(=O)(C#CC1CCCOC1)NCC(C(C)C)NC(C1(CC=C)CCC1)=O N1(C(c2ccc(C(=O)OC)c(Cl)c2)=O)CCOC2CCN(C(=O)C=C(Cl)Cl)CC12 N1(C(CCC=C(C)C)=O)CC(NC(=O)CCOCC(F)F)CC12CCCCC2 CC(C)CC(CNC(=O)C(C1CCOCC1)F)C(=O)N(CCC(N)=O)C c1(N(C)Cc2cccc(F)c2)nc2ccsc2c(=NCCN(S(C)(=O)=O)C)[nH]1 C1(C(N(CC(C)CNC(=O)CC(C)NC(N)=O)C)=O)COCCN1C=O Nc1c(C(=O)NC2COCC2CNC(C2OCCC2C(F)F)=O)cc(Cl)cc1Cl C(c1cscn1)=CC(=O)NCC1(CN(C(C(C)=CC2CC2)=O)C)CC1 N1(C(C2(CCNC(c3n(CC#C)cnn3)=O)CCC2)=O)CCC(O)CC1C C1(NC(C(CC)COC)=O)CC2CCC1CC2NC(=O)COC1CC(F)(F)C1 C1(NC(c2nc(CC(C)C)sc2)=O)CC12CC(NC(c1cscc1Cl)=O)C2 N1(c2n(CCC=C)c(CCCS(N)(=O)=O)nn2)Cc2c[nH]nc2C(C)(C)C1 C(C(=O)N1CC(NC(c2cnco2)=O)C(C)C1)(C(F)(F)F)OC(C)=O c1(OC)cc2nc(C)sc2cc1NC(=O)C(c1ccccc1N)OC c1(CNc2c(C)scc2)c(OC(F)F)cccc1Cl c1(CNC(C(CC)N(C)C)=O)ccc(CNC(c2cncn(C)c2=O)=O)c(F)c1 C12(NC(=O)Cc3ccccc3)CCOCC1CN(C(=O)CCC1OCCO1)C2 CC1CCCC1(C)C(=O)NCC1CC(NC(c2ccc(C3(C)CC3)cc2)=O)C1 C=CCC(C(=O)NC(C)CNC(=O)CCC(=O)Nc1c(F)cccc1F)C(C)C c1(C(=O)NC)ccc(O)c(NC(C2CCCCC(=O)C2)=O)c1 C(=O)(C#CC(C)(C)C)N(CCC1CC(NC(Cc2cc(C(=O)OC)sc2)=O)C1)CC CC(=O)C(C)(C)CC(=O)N1CC2COCC2(C(N2CCOC(CC(N)=O)C2)=O)C1 C1(C(=O)Nc2sccc2CO)CC2(C(N3CCC(CCCO)CC3)=O)COC1C2 Cc1ccc(CC(=O)NCC(O)CNC(C2(C)COCCO2)=O)c(Cl)c1 Cc1cc(CNC(c2occc2CNC(C2(O)CCOC2)=O)=O)nnc1C C1(NC(=O)C#CC2CC2)C2CC3C(C2)C13C(=O)NCC1CC2(CC2)C(=O)O1 c1(C(CC)CC)cc(C(=O)NC2CC2CNC(=O)CCCn2cccn2)on1 C1(NC(CS(N)(=O)=O)=O)C2CCCC1CC(NC(c1cc(=O)cc(Cl)[nH]1)=O)C2 C1(C2N(C(=O)C(F)C3CCCC3)CCC2)CCN(C(C23CC(C2)C3)=O)CC1 CC1CCC(C(=O)NC(C2CCN(C(=O)C(CO)N(C)C)CC2)C)CC1 N1(C(C(=O)C(=O)NC2(C(F)(F)F)CCC2)=O)CC2CN(C(=O)CO)C2C1 CON1CCC(C(=O)NC2(CC(=O)NCC3CCSC3)CC2)CC1 Cc1nc(C=CC(N2CC(NC(C3(C#N)CC3(C)C)=O)C(C)C2)=O)[nH]c1C N1(C(C(CC=C)OC)=O)CC2CC(C(=O)NC3CCCC3(C)N(C)C)(C2)C1 N1(C(c2cc(CC(=O)OC)no2)=O)CCC2CN(C(=O)CCC(C)C)CCC12 C=C(Cl)CCC(=O)N1CCCCC1CC(=O)NCc1ccn(C(C)C)n1 C1(CNC(c2nnn(C)c2C(F)(F)F)=O)CCN(C(c2cc(Cl)cs2)=O)C1(C)C N1(C(C=C(CCN(C)C)Cl)=O)CCN(C(=O)C=CC2CCCN2C)CC1CF c1(CC)ccc(C(=O)NCC(CC)N(C(=O)C(c2ccnn2C)C)C)s1 N1(C(C#C)=O)CCC2(CCCC2C(=O)Nc2ccc(F)cc2C)C1 c1(C(c2nnnn2C2CCCC2)NC(c2c(C)nn(C)c2)C)ccc(Br)cc1I C(=O)(C1=NOC(c2ccc(F)cc2)C1)NCC(CNC(CCSCCCC)=O)C c1(CC)nc(C)oc1C(=O)NCCOCCC(=O)N(C)Cc1occc1C CC(CC(C)(C)C)C(=O)NC1CN(C(c2csc(O)n2)=O)CC1c1nccn1C C(C1CCc2nccn21)NC(CC(CNC(CSCC#C)=O)O)=O C1(NC(C(=O)N(C)C)=O)CCCC(NC(=O)CSc2ccccc2Cl)CC1 c1(C(=O)NC(C2CCCN2C(c2cc(N)ccc2Cl)=O)C)nccc(Cl)c1F c1(CC)cccnc1C(=O)NCC1CCCCN1C(=O)C=Cc1cn(C)nn1 c1(C(=O)NC2C3(CCC(NC(C(N)=O)=O)CC3)C2)c[nH]c2nc(F)ccc12 C#Cc1ccc(C(=O)N(C)CC2CC(F)CN2C(C2CN(CC)CCO2)=O)cc1 C1(CC(=O)NCCCCCN(C(C)=O)Cc2csc(Cl)n2)C(=O)NN=C1C Cn1ccc2c(COC(C3CCCCS3(=O)=O)=O)ncnc12 C1(CC(=O)NC23C(CN(C(CCCOCCC)=O)C2)C3)CCC(F)(F)CC1 c1(C(=O)NC2CN(C(c3cc[nH]n3)=O)C2)ccc2nnc(O)n2c1 N1(C(C(C)CF)=O)CCC(CO)(CNC(=O)C(C)COc2ccccc2)CC1 c1(CCCC)ncc(C(N2CC(O)C2)=O)s1.C1(C(=O)NC)(C(=O)C2CC2)CC1 CN1C(=O)CCCC1C(=O)N(c1ccns1)C CC1CC2(CC(C(N3CC4CC(NC(=O)Cc5cocn5)C3C4)=O)C2)C1 N1(C(C(COC)C(F)(F)F)=O)CCc2sccc2C1CNC(=O)CCC(N)=O CCCCCCC(C(=O)NC1CC(NC(=O)CC2CC=CC2)C(O)C1)NC(C)=O C#CCCCCCC(=O)NC1(C)CCN(C(=O)CSc2cc(C)ccc2C)C1 c1(CC)cc(Cl)ccc1C(N1CCC(NC(C2CCN2CC)=O)C1(C)C)=O n1(C(C)C)ccc(C(=O)NC(C)(C)CNC(=O)CCCC2CCOCC2)n1 CN1C(=O)CCC1C(=O)NC1CN(C(c2cnc(N)cn2)=O)CC1O c1(-n2cc(-c3cn(C)nc3)nn2)cncc(C(N2CCC(CCO)C2)=O)c1 Cn1cnc2cccc(C(=O)NC3CCC3NC(c3cnc(S)n3C)=O)c12 C1(CC=C)(NC(C2CC(C)CO2)=O)CCCN(C(=O)CN2CCC2)C1 CC(C)CC(CNC(=O)C(C)c1ccco1)C(=O)NC(c1cncc(F)c1)C N1(C(C2C(C)CC2)=O)CCCC12CCN(C(c1cc3cccc(Br)c3o1)=O)C2 CCC(C)CCC(=O)N(C1CC2CC1N(C(=O)Cc1cc(Cl)n(C)n1)C2)C C#Cc1ccc(NC(=O)NCC2(NS(=O)(=O)C3CC3)CC2)nc1C C1(NC(C(CCC)NC(N)=O)=O)CC2CC(NC(=O)CCCSC)C2C1 C1(C(N2CC(N(C(c3nnc(C)o3)C)C)C2)=O)(OCC)CCCSC1 C12(OC)CCC1CN(C(=O)C(CC(N)=O)NC(=O)CC13CCC(CC1)C3)C2 c1(C(=O)NC(CCCC)CNC(c2ccnn2COC)=O)cccc2c1COC2 c1(C(=O)NCCN(CCC)C(C2CC2(F)Cl)=O)cnoc1-c1ccccc1 C1(NC(CCSCCC)=O)CN(C(c2c[nH]cc2CC)=O)CCC12CCC2 C1(OCCNC(CCC=CCC=C)=O)CCN(C(=O)CC(C2CC2)C2CC2)CC1 C(=O)(CC(C)CC(F)(F)F)NC1CC(CCNC(c2c(C)ncnc2C)=O)C1 C1(C(N(CCCCS(C)(=O)=O)C)=O)CC2(CNCC2C#N)C1 Cc1nn(-c2ccccc2)c(NC(N2CCCC2C(O)C(F)F)=O)c1Br C(C(C)(C(C)C)NCC)NC(CC1CC(OC(=O)CP(C)(C)=O)C1)=O N1(C(C2C(C(N)=O)CC2)=O)CC=CC1C(=O)NC(C1CC1)C1CC1 c1(C(N2CCC(C)N(C(C3CCCS3)=O)CC2)=O)c2c(nn1C)CCCC2 C1(C)(C(=O)NC(C)CNC(=O)CCCc2n[nH]c(=N)s2)CCCCC1(F)F C1(C(=O)NC(CCNC(C(C=C=C)C)=O)(C)C)Cc2cc(Br)ccc2O1 N1(C(C)CNC(C2CNC(=O)C2)=O)CCN(C(c2ncncc2N)=O)CC1 N1(C(C2CN(S(C(C)C)(=O)=O)C2)=O)Cc2cccc(Cl)c2C1 c1(C(=O)NCCCOCCN(C(CC=CC)=O)C)cnn(CC)c1C c1(C(C)C)nc(NCCSc2nccn2C)cc(N2CCC(C(C)O)C2)n1 c1(C(=O)NC2CC(NC(C3(C(F)F)CC(=C)C3)=O)C2)ccc(Cl)c(S(N)(=O)=O)c1 C1(C(=O)NCc2nc(-c3ccco3)n[nH]2)CC2CCC(C1)C2(F)F N1(C(c2c(OC)cccc2)=O)CCCN(C(C2CC(=O)N(OC)C2)=O)CCC1 c1(NC(C2N(C(C(C)CF)=O)CCC2)=O)ccccc1C1CC1 N1(C(N(c2ccc(F)cc2)C2(C)CC2(Cl)Cl)=O)CCCNCC1 c1(C(C)CNC(=O)C(=O)NCCC2CCCCC2)ccc(Cl)cc1 Cc1cc(C)n2nc(C(=O)NCCC3CCN(C(C4CCC(=O)N4)=O)C3)nc2n1 c1(C(=O)NCC2(O)CN(C(c3ccc(F)cc3)C(N)=O)C2)ccnc2ncnn12 c1(C(N(CCNC(c2n[nH]c(C)n2)=O)CC)=O)ccncc1Cl c1(C(=O)OC)cncc(S(=O)(=O)NCCc2ccc(Br)cc2F)c1 CCC(C)C(C)C(=O)OC(C1CC(F)(F)C1)OC(C1(CS(C)(=O)=O)COC1)=O C1(=O)CCN(OC)C(=O)C(CO)N1.CCC(C1CC1)(C1CC1)C1CC1 C=C(C)C(C)(C)C(=O)NC1CCCCCC1C(=O)N(C)CCc1ncon1 N1(C(Cc2ccn(C)n2)=O)CCCC(C)(C)C1C(=O)NCCCn1ccnn1 c1(C(=O)NC2CC(C)N(C(=O)C(N)=O)C2)cc([N+](=O)[O-])c(F)cc1N C1(NC(C(C)OCC=C)=O)CN(C(c2ccc(-n3cncn3)cc2)=O)CC1F C1(NC(C2OC3CCC2C3)=O)CCC(NC(C2C(Cl)(Cl)C23CC3)=O)CC1 c1(OC)ccc(C(C)C(=O)NCCNC(=O)C(c2cnn(C)c2C(C)C)C)cc1 N1(C(c2c(C)ccs2)=O)CCN(C(c2ccn(-c3ccccc3)n2)=O)CC1CO Cc1nnc2n1C(C(=O)NCC(C1CC1)NC(c1ccn3cncc3c1)=O)CC2 n1(CC)nc(C(=O)NCC2C3CC3CN2C(C2CC2F)=O)ccc1=O C1(NC(c2c(C)sc(O)n2)=O)CCN(C(=O)C(C)CC(C)C)CC(C)(C)C1 N1(C(CN(S(C)(=O)=O)C)=O)CCCN(C(=O)C=CC=Cc2ccccc2)CCC1 C=CC1(CNC(=O)C(CC2CCC2)NC(=O)CC(C)n2cccn2)CCC1 Cc1cc(NC(C23CC2CN(C(=O)C#CC2CC2)C3)=O)cnc1C C1(CC)(CC)CN(C(=O)CC(C2CC2)NC(=O)CC2CCC(O)C2)CCO1 c1(C(N2C(C(=O)NCCOc3cccnc3)CC(OC)C2)=O)ccc(O)cc1Cl C(=O)(C(C)(C)CC(C)(C)C)NCC(C)N(C(CCOC(C)C)=O)C CN=c1nc(N(C)C(=O)N)cc(C)[nH]1.N1(CCC2ON=C(C)C2)CCC(C)(C)C1 C=Cc1cnn(C)c1C(=O)NCC=CCNC(=O)Cc1cnn(C)c1 N1(C(C2(COC)CCCC2)=O)CCC(O)(C(C)NC(=O)COC2CC=CC2)CC1 C1(NC(CCc2onc(C(C)OC)n2)=O)CN(C(c2[nH]c(C)nc2C)=O)CC1C c1(OC)ccnc(C(N2CCC(NC(C3CN(C(C)=O)C3)=O)CC2C)=O)c1OC C12(C(N3CCCN(C(CC4COCC(C)O4)=O)CC3)=O)CCC(N=[N+]=[N-])C1C2 Cc1ncc(Cl)cc1NC(C1OCCC1NC(=O)CC1CCC(C)(C)C1)=O Oc1cccc2cc(CN=c3ccc(Br)c(F)[nH]3)ccc12 C#CC1CCC(NC(C2(CNC(c3nn(C)cc3Cl)=O)CC=CC2)=O)C1 c1(CNC(=O)OC(C)(C)C)cc(C(=O)NC2CC(OCC(F)F)C2)co1 C1(C(N2CC(C(C)(C)O)(CNC(C=C3CCN(C)C3)=O)C2)=O)CC(=O)OC1(C)C c1(OC)cc2nn[nH]c2cc1C(=O)NCC1CCN(CC2CC3CCC2O3)C1 Cc1nc2c(C(N3CCC(N(CCO)Cc4cccnc4C)C3)=O)cccc2o1 Cc1c[nH]c(C(=O)NC(C)CCC(=O)NCCC(O)C(C)C)c1C c1(OC)c(C)cc(C(N2CCN(C(c3ccc(O)cc3)=O)CC2CO)=O)cc1C N1(C(c2n(CC)ccc2)=O)CC2(CCC2NC(c2ccc(OC(F)F)cc2)=O)C1 CC1(F)CN(C(c2ncn(C(C)(C)C)n2)=O)CCN(C(C2(C)CC2Br)=O)C1 c1(C(N2C(C(=O)NCC3CN(C)CCO3)CC(C)C2)=O)ccc2ncnn2c1 N=c1ncc(C(N2CCOC(Cn3cc(CNC4CCOCC4)nn3)C2)=O)c[nH]1 C1(O)(C(=O)NC23CN(C(C(C)(C4CC4)NC(C)=O)=O)C(C2)C3)Cc2ccccc2C1 N1(C(N(C)CCN2CCOC(C)(C)C2)=O)Cc2ccccc2-c2ccccc21 n1(CC(N2CCN(Cc3c(O)cccc3O)C3CC23)=O)ccc2c(F)cccc12 c1(-c2nnc(-c3ccc(-c4n(CC(C)O)ccn4)s3)s2)cc(=O)cc[nH]1 Cc1ccnc(C(=O)NCC2(CO)CCN(C(C3(C)CC3C)=O)C2)c1N C1(NC(c2c(C)nc[nH]2)=O)CN(C(c2cc(Cl)c(O)c(Cl)c2)=O)CC(C)(C)C1 CC1C(NC(c2snnc2C2CC2)=O)CCCN1C(c1cc(C2CC2)on1)=O C(CN=C(NCc1ccsc1Br)N(C)Cc1ncnn1CC(F)F)SC Cc1sc(CNC(=O)C(Cc2cccc(Cl)c2)NC(=O)OC(C)(C)C)c(C)c1C CCCN=c1[nH]c(=NC2CCCCN(Cc3ccccc3)C2)c2sccc2[nH]1 C1(C(=O)NC2C(NC(c3n[nH]c(CC)c3C)=O)COCC2)CC2OC1C1CC21 N1(C(C(=O)N(C)C)=O)CC2CCCC(N(C)C(c3cnc4sccn34)=O)C2C1 c1(C(=O)NC2(C)CC(NC(C3COCC(C)O3)=O)C2)ccc2nccnc2n1 Cc1nc(CNC(=O)C(CNC(=O)CC23CCCC2C3)N(C)C)sc1C CC(C)(CC#N)C(=O)N1CCC(NC(c2sccc2OC(F)F)=O)C(O)C1 c1(C(=O)NCC(C2CC2)NC(C(C)(C)OCC)=O)cc2c(F)ccc(F)c2s1 n1(CCN(CC)Cc2ccc(-c3ccccc3CO)nc2)ccc2ccccc12 CC1CC(C(=O)NCC2CN(C(=O)CCCc3ccccc3N)CCN2C)=NO1 N1(C(c2c(C)nns2)=O)CCCC2(CCN2C(C2CCCSC2)=O)C1 C(=O)(C(F)C(F)(F)F)NCCCOCCNC(Cc1c(CC)cccc1)=O CCCCCC(O)C(=O)NCc1ncccc1C(=O)N(CCC(N)=O)C N1(CCC)CCCC1C(=O)NC(C)CCNC(c1cnoc1C1CC1)=O C(C(C)CC(=O)NCCCC(C)NC(=O)CSCCCc1ccccc1)OC C1(C(=O)NCC2N(C(C=CCC)=O)CC(F)(F)C2)CCOC2(CCCC2)C1 CC(C)CS(=O)(=O)CCC(=O)NCCCN(C)C(C1(C)SCCCS1)=O N1(C(COC(C)=O)=O)CC2C(NC(c3ccc(CO)cc3)=O)C2C1 c1(OCC(=O)N(CC(CC)NC(=O)C(C)(C)N(C)C)C)ccccc1C Cn1ncc2c(=O)n(C(=O)N3CC(n4cc(-c5cccnc5Cl)nn4)C3)[nH]c(=O)c12 N1(CCC(C)(C)CBr)CC2CCC(O)CC2C1 c1(CC)cc(C)ccc1NC(=O)CC1CCCCC1NC(c1c[nH]ccc1=O)=O c1(C(=O)NCc2ccsc2)n[nH]c2c1CN(C(=O)CN1CC=CC1)C2 O=S(=O)(c1ccc(NC(c2ccccc2)CO)c(Cl)c1)N1CCC=C(F)C1 CC(C(=O)NCc1cscn1)NC(=O)C(C)C1CCCC1 C1(C(=O)NCCC2OCCN(C(c3c[nH]c(=NC)o3)=O)C2)CC(C)(C)OC1(C)C C12(C(=O)NC(c3nc(C(F)(F)F)cs3)CC)CCCCC1C2Br C1(NC(CSSC)=O)CCCC2CN(C(c3cnc4cccnn34)=O)CC12 CCCCC(C)C(=O)N1CC(CNC(=O)CCC2(NC(=O)OC(C)(C)C)CC2)C1 N1(C(C(N(C)O)=O)=O)CCC(O)(CNC(=O)NC)CC1 C1(C(C)NC(C2CCCO2)=O)CCCN(CC(=O)Nc2ccccc2)C1 c1(CC)cc(C(=O)NCC2(O)CC(NC(=O)CC3CC=CC3)C2)c(C)nn1 c1(C(N(C2CC(NC(=O)CCn3cc(Cl)cn3)C2)C)=O)csc2nccn12 CC(C)(C#N)CC(=O)N1CC(NC(C2CCC(=O)N2)=O)C(O)C1 c1(CNC(C(=O)NCC(CNC(C=C(C)C(C)C)=O)C)=O)ccc(F)cc1 N1(C(c2n(CC(=O)OC)cnc2C)=O)CCCC(F)(CNC(c2cnn[nH]2)=O)C1 c1(CN(C(CCCOC)=O)C)cnn2c1CN(C(=O)C(C)S(N)(=O)=O)CC2 c1(CCCCC(=O)N(CCNC(=O)C2CC2)CCOCF)nc2ccccc2s1 C1(NC(C(N2C(CC(=O)NC3CC3)CCCC2)=O)=O)CC2OC(=O)CC12 Cc1cn2c(C=CC(=O)OCc3cnc(C#N)cn3)c(C)nc2s1 C=C(C)CC(C(=O)N1CCN(C)C(CNC(=O)C(O)CCSC)C1)OC CCC(CC(=O)NCC(c1ccc(F)cc1)NC(C12CC(F)(C1)C2)=O)C(C)(C)C C1(CC(N2CC(CSC)C2)=O)CC(F)CN1C(C1CC12CC2)=O c1(C(=O)NCCC2CC(NC(c3cc(CCC)on3)=O)C2)n[nH]c2c1CSCC2 C(=O)(C1=CCC(C)(C)CC1)NCC(C(C)(C)C)NC(c1cnc(O)n(C)c1=O)=O c1(C(N2CCC(OCC(=O)OC)C2)=O)cc(C#N)[nH]c1C C#Cc1cc(NC(=O)C(C2(O)CCC2)NC(C2CCCS2)=O)ccc1C C(=O)(C(CN=[N+]=[N-])NC(C1CC2C=CC1CC2)=O)N(C1CCN(C)CC1)C N1(Cc2ccn(C(C)C(=O)O)n2)CCC(c2nn[nH]n2)CC12CC2 c1(C(N(CC(CN(C(c2c(OC)nsc2)=O)C)O)C)=O)cc(C)c(Cl)c(C)c1 C(CN=c1[nH]ccc(=NC2CC2c2ccc(C)c(C)c2)[nH]1)n1c(C)cc(C)n1 N1(C(C2(NC(C3C(C)C3)=O)CC(O)C2)=O)CCCCCC1 c1(C(=O)NCC(CC)(C)NC(=O)C(F)=C(C)C2CC2)ccc(C)c(F)c1 N1(C(C(C)OCC)=O)CCCC2(CNC(=O)CC3CC(C)=NO3)CCCC12 Nc1cccc(C(=O)CCC(=O)NC2CC2NC(C23CCCC2C3)=O)c1 c1(C(N2C(CC)C(NC(c3cnncc3C(F)F)=O)CC2)=O)ccc(Cl)cc1O C=CCC(CNC(=O)COCC(C)C)NC(=O)C#CCN(C)C N1(C(CN(C(=O)OCC)C)=O)CCCC(CCC(=O)NCC(O)CC)C1 C(=O)(C1=NN(C)C(=O)CC1)N1CCN(C(C2CC(CC)OCC2)=O)C2(C1)CC2 C1(C(=O)NC2C3(CN(C(c4cc(=NC)[nH]cc4)=O)C3)CC2)CC2(C1)CC(C)(C)C2 N1(C(C(CC)(C)O)=O)CC(CNC(c2ccoc2C2CC2)=O)CC(C)(C)C1 C1(C(=O)OC)(NC(C2CC(N(C)C)C2)=O)CCN(C(=O)C(C)Cc2ccco2)C1 c1(OC)ccc(C(N2CCC(CNC(=O)CCF)C(F)(F)C2)=O)c(Br)c1F N1(C(C(c2ccccc2)C)=O)CC2CC(C1)CN(C(c1ocnc1C1CC1)=O)C2 c1(C(COC)(C2CC2)NCCOC)nnnn1C1CCCC1.C1CCN1.C1(C)CCC1 C1(C(=O)NC(C2CCCC2)C#C)CCCCC1(C)NC(=O)CC1(O)CCOCC1 CN1CCC(C)(C(=O)NCC23CC2CN(C(=O)CC2CSCCO2)C3)CC1 c1(OC)cc(OC)nc(-n2cc(C3CCCN3C(=O)CC3COC(=O)C3)nn2)n1 C=CC(CC)C(=O)NC(CO)C(C)NC(c1cnn(CC)c1CC)=O N1(C(C2C(COC)C2)=O)C(C)CC2CN(C(=O)CCC3CCC3)CC12 c1(N(C)CC2CC2)ccn2ncc(S(=O)(=O)NC3(C)CCOC3C3CC3)c2n1 c1(C(N2CCCC(N(C(=O)CCC3(C)CC3)CC)C2)=O)c(F)ccc(C#N)c1F c1(C(N2CC(C)(NC(c3cc(COC)oc3C)=O)C2)=O)cccn2nnnc12 C1(F)(CNC(C(c2ccc(F)cc2)OC)=O)CCN(C(=O)CC2CCC(=O)N2)C1 C(CNC(c1cccc(COC)c1)=O)(C(C)(C)C)NC(c1c(CCC)nns1)=O c1(C(=O)O)ccn(CC(=O)NC2CN(C(C3CC(N4CCCC4)C3)=O)C2)n1 c1(OCC)ccc(C)nc1C(N1CCOCC(NC(C)=O)C1)=O Cc1cc(F)c(CC(N2CCC3(C2)CN(C(=O)CC2(O)CCCOC2)C3)=O)cc1F O=C(CCCCCCNC(c1ocnc1C1CC1)=O)NCCC#CCO C1(NC(c2ccnn2CCF)=O)CCCCC1CNC(C1CCCO1)=O CC1(C)C(NC(=O)Cc2ccc(F)cc2F)CCN1C(C1COC(=O)O1)=O C1(CNC(CC=C=C)=O)CCN(C(=O)CNC(C2CCCCC2)=O)CC1C Cc1nc(F)ccc1-c1cn(CC2CCN(C(C3C=CCC3)=O)C2)nn1 Cc1nn(C)c(N)c1C(=O)Nc1c(C)nn(CC(C)C)c1C N1(C(Cc2ccc(CC)cc2)=O)CCCN(C(c2ccc(F)c(Cl)c2)=O)C(C)C1 c1(OC)cc(C(=O)NCCC2COCCN2C(c2ccsc2)=O)cc(C2CC2)c1 C1(NC(CC(CC)C)=O)CC2CC(NC(c3cc(C(C)C)[nH]c3C(C)C)=O)C1C2 CN1CCC2(C(=O)N=c3cc[nH]cc3Cl)CCCCC12 C1(CCNC(C2CS(=O)(=O)C2)=O)CCN(C(=O)CC23CCC(CC2)C3)CC1 C1(NC(CSCCCC)=O)C(C)CN(C(c2occc2CC)=O)CC1C C1(C2CCCN(C(=O)C=CCF)C2)(NC(CC2C(C)=NN(C)C2=O)=O)CC1 Cc1nn(C)c2cc(NC(=O)CC3CCC(C)C3)ccc12 C(c1nc2ccccc2[nH]1)=CC(=O)NCC1C(NC(c2c(N)cccc2Cl)=O)C1 N1(C(C=Cc2n(C)ccc2)=O)CCN(C(C2CC3COCC3C2)=O)CC1CO N1(C(CSC)=O)CCOC2CN(C(=O)C(C(C)C)n3cc(C)cn3)CC12 C=CCC(C(=O)N1CCC(C(C)(C)C)C1)NC(c1ccc(OCC)nc1)=O c1(OCC(N2CCC(N(C)C(C3CCC(F)C3)=O)C2)=O)ccc(F)c(Cl)c1 c1(OC(C)(C)C)ccc(C(N2CC(NC(=O)C=C3CCCCC3)C3CC23)=O)cc1 C12(NC(CCOCC)=O)CC(C)(C1)OC21CCN(C(C2CCC(F)(F)C2)=O)CC1 c1(OC)ccc2c(c1)CCCC2C(=O)NC12CC(NC(=O)CO)(C1)C2 c1(C(N2CCN(C(C(C=C=C)C)=O)C(CC)C2)=O)nnn2ccccc12 c1(NC(C2CCCC(NC(C3(Br)CCC3)=O)C2)=O)cccc(F)c1Br c1(CNC(c2nc(CNC(C=C(C)C(C)C)=O)oc2C)=O)cncc(C#N)c1 N#Cc1ccc(Cl)c(C(N2CCC3(CNC(c4cscn4)=O)CCCC23)=O)c1 CC(C)C(C)(CNC(=O)CCCN1C(=O)CNC1=O)NC(C1C=CCCC1)=O C(=O)(C(C)(C)CC(F)F)N(C)CC1CCCC(NC(c2cn(C)c(=O)cn2)=O)C1 N1(C(C(C2CN(C(C3(OC)CCOCC3)=O)C2)O)=O)CCCC(N=[N+]=[N-])CC1 C1(C(=O)OC2CC(c3ccccc3)C2)CCC2(C1)CC2(F)F c1(C(N2CC3CN(Cc4c(Br)cn(C)n4)C3C2)=O)ccc2c(c1)CCO2 C(=O)(C(F)(F)F)NCC(=O)N(C1CCN(C(=O)C(O)c2ccco2)C1)C Cc1ncnc(C(=O)NCC2(F)CN(C(=O)C(c3ccccc3)F)C2)c1C Cc1cccc2[nH]cc(CC(=O)NC3CCCN(C(c4coc(C#N)c4)=O)C3)c12 C=CCCCC(C(=O)NCC1CCCO1)N1CC(F)(F)CC1CC(=O)OC Cc1cc(C(=O)NC(C)CCN(C(=O)CNC(=O)CCC(C)C)C)c(O)nc1C c1(NC(c2cccc(O)n2)=O)ccc(NC(c2ccc(O)cc2O)=O)c(F)c1 c1(OCC)ccc(Cl)cc1CC(=O)NCC(O)CN(C(=O)CCCNC(C)=O)C C(=O)(C(CC)(CC)CC(=O)OC)NCCC(CNC(C(CCC)CC)=O)O C1(C(=O)NCc2ccc(C)o2)CC2C=CC1N(C(=O)CC1CCC(=O)C1C)C2 c12cccc(n1)C(=O)NCCN(C)C2.c1(C(=O)NC(C)(C)C)ccc(F)s1 N1(C(CC(C)N(C)C)=O)CC2(CCN2C(c2ncccc2Cl)=O)C1 C(=O)(CCCN=[N+]=[N-])NC(C(C)NC(C1N(C(C)=O)CCC1)=O)CO N1(C(C2C(C)(C)C2)=O)CCN(C(=O)Cc2cnc[nH]2)CC1c1ccc(F)cc1 N1(C(Cc2nc(CC)sc2)=O)CCCC(C2CC2NC(c2cnsc2)=O)C1 C1(CC(=O)NC(CNC(=O)CC23CCC(CC2)OC3)C2CC2)CC2(CCC2)CO1 c1(CC)cc(C)nc(N2CCCC2C(C)(C)CNC(C2CC(=O)NC(=O)N2)=O)n1 N1(C(C2C=C(C)CS2)=O)CCCC(CO)(NC(c2ccnc(O)c2)=O)C1 c1(C(=O)NC(CCNC(C=C(C)C(C)C)=O)(C)C)ccc2cnoc2c1 c1(C(N(C)CC2(NC(Cc3cncc(C)c3)=O)CC2)=O)ccc2[nH]ccc2c1 C(=O)(C(C)(C)C(C)(F)F)N1CCN(C)CC1CNC(C1(CCO)CC1)=O c1(C(=O)OC)cccc(NC(C2CC2C(=O)Nc2ccc(C)cc2F)=O)c1C C1(C(F)(F)F)(N(C(C2CC2c2ccco2)C)C(C2CC2)C2CC2)CC=CCO1 N1(C(c2[nH]cc(C)c2)=O)CC(NC(=O)C=Cc2cn(C)cn2)CC12CCCC2 C1(C(C)NC(=O)C(C)(C)c2ccsc2)CCN(C(c2ccc[n+]([O-])c2)=O)CC1 c1(OC)ccccc1OC1CN(C(C2(N)CCSCC2)=O)C1 N1(C(C(C)NC(C)=O)=O)CCC(CNC(=O)COc2ccc(C)cc2C)C12CC2 Cc1ccc(CNC(=NC(C)C)NC2CC(=O)N(C(C)C)C2)c(=O)n1C C1(C(C)C)CCC(C)CC1(O)CNC(=O)Cc1c(F)ccc(Br)c1F C(=O)(C1=CC2CCCCCCC12)NCC1N(c2nnc(C(N)=O)s2)CC(F)C1 C(=O)(CC(C)C(F)(F)F)NC1C(CNC(c2c(-c3ccc(C)o3)onc2)=O)CC1 c1(C(C)C)cnc(CNC(=O)NC23CSC(C2)C3)o1 CS(=O)(=O)c1ccc(CN2CCN(Cc3c(Cl)ccc([N+](=O)[O-])c3Cl)CC2)cc1 C1(NC(c2ccc(C(=O)OC)o2)=O)CCC(NC(=O)C(C)c2ccon2)CC1 N1(CC=O)CCC(O)C1.C(=O)(CC(=O)NCC1CC1)NCCN(CCOC)C CN1CC(C)(C(=O)NC2CCN(C(=O)CC3CNC(=O)O3)CC2)CC1=O c1(C(=O)OC)cc(C)cnc1NC1CN(C(=O)C(C)(C)C(C)C)CC1C C1(NC(C=C(CC)CC)=O)CN(C(C2CC2(COC)COC)=O)CC1C c1(C(=O)NCC(CNC(Cc2cc(C)cc(Br)c2)=O)C)cccn2ccnc12 N1(C(c2cc(CC)no2)=O)CCC2(CCCCC2NC(=O)CCCN(C)N=O)C1 N1(C(CNC(CCCC)=O)=O)CCN(C(=O)OC(C)(C)C)C(Cc2ncco2)C1 c1(CCNCc2ccc(-n3c(C)cc(C)n3)nc2)cccc(F)c1F c1(C(N(CCNC(c2cnccc2Cl)=O)CC)=O)cn2ncnc2nc1C C1(CNC(c2ncn(C(C)C)n2)=O)COCCN1C(=O)Cc1cscn1 C(=O)(C1=CC2CCC(C1)C2)N1C(C(=O)NCC(CC(C)O)(C)C)C2(C1)CCCC2 N1(C(CNC(=O)OCC)=O)CCC(F)C(NC(=O)C(C)(C)N2CCCC2)C1 C1(NC(C2CCCC(CF)C2)=O)CCCC2CN(C(=O)C=C3CCCC3)CC12 c1(C(N2CCCC(CNC(C3ON=C(C)C3)=O)CC2)=O)cc(C)cc(C)c1C CC1CN(C(=O)CC2CCCN(C)C2)CC1NC(c1cc(CCCO)on1)=O C12(C(N(CC(=O)NC3C=CC(C(=O)NC)C3)CC3CC3)=O)CCN(CC1)CC2 C=CCC(CC(F)F)C(=O)N(C)CC1(O)CCCN(C(=O)CCC(C)CC)C1 N1(C(C2(C#N)CC3CC3C2)=O)CC(NC(c2cnc(Cl)s2)=O)CC(F)(F)C1 Nc1ccc(S(=O)(=O)NCCC(=O)NCC2CCN2C2CC2)cc1 N1(C(C(CC)(C)F)=O)CC(NC(=O)CCn2cccn2)CC(F)C1 C1(C(=O)NCC2C(C)CN(C(=O)CN3CCCCC3)C2)CCC(C2CCCO2)O1 c1(C(N2CCOC(C(F)(F)F)C2)C(=O)NCCCC)ccc(COCC)cc1Br Cn1c(CO)nc2cc(C(=O)NCC(C3CC3)NC(C3CSCCS3)=O)ccc12 CC1Cc2cccc(O)c2N(CCC2(C#N)CCOCC2)C1 CC1CC=C(C(=O)NC2CC3CC2N(C(=O)CCc2cnn(C)n2)C3)CC1 C1(CNC(CCS(C)=O)=O)CCN(C(=O)CSCc2ccc(F)cc2)C12CC2 C1(CNC(c2ncc(C)cn2)=O)CCN(C(=O)CSC2CCOC2=O)C12CCC2 n1(CC)ncc(Cl)c1C(=O)NC(C)CC1CN(C(=O)C=C2CCOCC2)C1 C1(C(N2CC[Si](C)(C)C2)=O)CN(C(=O)C2=CCCOC2)C2(CCC2)C1 Cc1noc(Cl)c1CC(=O)NC1CCCC(CN(C(=O)CCn2cnnn2)C)C1 CCCC(CCNC(C1OCCC1CNC(c1occc1C(C)C)=O)=O)CCC N1(C(C(=O)NC(CCCCC)C)=O)CCSC2(CCCCC2)C1 CC1CCOC(C(N2CCC(NC(c3ccc(C(F)(F)CF)cc3)=O)C2)=O)C1 C1(Nc2cc(NC(CC=C)CC)nc(C)n2)CCc2nn[nH]c2C1 c1(C(C(=O)NC2CCC2)N(CCCC)CC)nscc1Br CC(C)(C(=O)N(CC(S(C)(=O)=O)C1CC1)C(C)(C)C)C(=O)N1CCCC1 Cc1c(Cl)ccc2[nH]c(C(N3CCCN(C(C4CCOC4)=O)C(C)C3)=O)cc12 O=C1OCCCN1CNC(=NCc1ccccc1)NCC(C1CCOCC1)(F)F N1(C(CC=CC=C)=O)C2CCC1CC(CNC(c1cc(O)nc(Cl)c1)=O)C2 c1(C(N2CCC(CN(C)C(c3cncc(C(F)(F)F)c3)=O)C2)=O)cccc(O)n1 c1(N2C3CS(=O)C(C3)C2)nc2ccccc2c(=NCc2cccc3nc[nH]c23)[nH]1 C(=O)(C1CCC(=O)c2cccn21)NCCN(C(C1CCC(C)(C)CC1)=O)C1CC1 CC(CC(=O)N(CCCCC(=O)N1CC(O)(C(N)=O)C1)C)C(F)F c1(C(=O)NCC2C(NC(c3ccns3)=O)COC2)cncc2c1CCC2 CCC(F)(F)C(=O)NCC1(O)CC(NC(c2ccnc(NC(C)=O)c2)=O)C1 Cc1cc(N(C(C)CNC(=O)C(C)C(C)S(C)(=O)=O)C)n2ncnc2n1 CCCCC(C(=O)N1CCC(F)(CNC(c2c(C)cccc2O)=O)CC1)C(C)C S(=O)(=O)(c1ccc2c(c1)C(=O)NC2=O)Nc1c(C)n(C)nn1 c1(CC(=O)NCC2(F)CCCN(c3ccnc(OC)n3)C2)cnc2ccccn12 C1(C(=O)NCCc2nc(C)sc2)COCCN1C(=O)CC1C=CCC1 N1(C(C=CCCC)=O)C2CCC1C(NC(c1sc(Cl)c(Cl)c1C)=O)C2 C=CC(C)(CCOC)C(=O)NC1CCCN(C(c2cc3cscc3s2)=O)C1C CCCCC(C)C(=O)NCC1(CN(C(=O)CC2CCCC2O)C)CC1 c1(NC(CN(C)CC2CCN(C(C3CCCN3C)=O)C2)=O)ccc(Cl)cc1 c1(C(N(c2ccc(C)s2)CC(C)OC)=O)ccc2c(c1)OCCN2C(=O)OC Cc1ccc(C(=O)NC2COCCN(C(c3cn(C)nc3C)=O)C2)c(I)c1 O=C(C1CCCCCc2ccccc21)NC12CC(NC(=O)C3=CCSC3)(C1)C2 Nc1cccnc1C(=O)NCC(c1ccccc1)CNC(=O)CNC=O c1(NC2CCN(C(=O)OCC)CC2OC)ccc2ncc(Br)n2c1 CC1CCN(C(C2COC(C)C2)=O)CC1NC(=O)CNC(c1ccc(N)cc1)=O CCC(CNc1ccccc1Cc1ccccn1)CC(C)O N1(C(N(c2cn[nH]c2)C)=O)CC2(C1)CN(C(=O)OC(C)(C)C)C2 N1(c2ccnc(CC)n2)CCn2ncc(CN(C(=O)CCC(C)OC)C)c2C1 Cc1cnn(CC(c2ccccc2)C)c1.n12cc(nn1)CCNC(=O)C2C c1(C(N2CCOCC(NC(C(C)O)=O)C2)=O)c2c(nn1C)CCSC2 N1(C(C(C#C)(C)C)=O)CCC2(NC(=O)CC(COC)Cc3ccccc3)CC2C1 C(=O)(C(CC1CC1)NC(=O)CC(C)F)N(c1cnn(C)c1)CC c1(C(N(CCNC(c2nc(CCC)sc2)=O)CC)=O)cnc2c(cnn2CC)c1 c1(C(=O)NCc2ccc(O)c(O)c2)ccc(C#N)nc1.CC12CC(C1)C2 C1(O)(CNC(C(Cc2cn(C3CCCC3)nn2)NC(=O)OC)=O)CCCN(C)C1 c1(C(=O)NCC2CC(NC(C(=O)NC3CC3)=O)C2)cccc(-c2ccccc2)n1 C1(C(=O)NC(CCC)c2ccco2)(NC(=O)Cc2cncn2C)CC1(C)C N1(C(C2CCCN(C)C2)=O)CCC(F)(C(N2CCCC(CC3CC3)C2)=O)CC1 N1(C(C2(CCCC)CC2)=O)CCN(C(=O)CC2=CCCC2)C(CO)C1 C1(C(=O)NCC(=O)NCC(C)C)C2CCC(C2)C1NC(c1cc(Cl)cn1C)=O C1(C(N(CC)CC2CC2)=O)CCCCCCN1C(=O)CC1(COC)CC1 C1(NC(C=Cc2nc(C)sc2)=O)C2CC1CN(C(c1nc(O)sc1C)=O)C2 c1(C(N2CCC(C)(NC(CCN(S(C)(=O)=O)C)=O)C2)=O)nc(Cl)ccc1N Cc1[nH]c(C(=O)NCC(O)CO)c(C)c1C(N1CCC(O)(CF)CC1)=O N1(C(c2c(CC)n(C)nc2)=O)C2CCC1CC(NC(C1CCN(CC)C1)=O)C2 C1(CNC(c2cccc(C(C)C)c2)=O)(NC(c2cscn2)=O)CCCCC1C c1(C(=O)NCC(C)N(C(C(CC)O)=O)CC)cccc(-n2ccnc2O)c1 Cc1[nH]nc2c1CCC(C(N1CC(C)(NC(c3ccccc3Br)=O)C1)=O)C2 c1(C(=O)NC2(C(=O)NCCCN=[N+]=[N-])C(C)(C)C2)ccc(O)cc1F C1(C(=O)NC(CCC=C)C2CC2)CC12CCN(C(c1ncsc1NC)=O)CC2 Cc1nsc(C(=O)N(C2CCN(C(=O)Cn3nccc3C)C2)C)c1Br N1(C(c2c(C)cco2)=O)CCN(C(c2cnn(C(C)C)c2N)=O)CC(C)(F)C1 c1(-c2n(CC)c(O)nn2)cnc(OC)c(CN(CC(F)(F)F)C)c1 Cc1nc(C(=O)NC(C)C(=O)N(C2CC(C)C2)C)ccc1C#N c1(OC)cccc(S(=O)(=O)N2CCC23CN(c2cc(C#N)ncn2)C3)c1 c1(NC(=O)CSCCOC2CN(C(C3(CO)CCCO3)=O)C2)ccncn1 N1(C(c2c(C)scc2)=O)CC(NC(=O)CC2CCSCC2)C(O)C1 N1(C(C)=O)CCCCC1C(=O)NC1CCC(CNC(c2cc(CCO)on2)=O)C1 c1(OC)cncc(C(=O)N(CC(=O)NCCC2CC(C)(C)C2)CC(C)C)c1 Cc1ccc2occ(C(=O)NC3CCCN(C(=O)C#CC4CCCO4)CC3)c2c1 C1(NC(c2c(C)[nH]cc2)=O)CC(O)CN(C(=O)CCCc2ccc(F)cc2)C1 c1(C(N2CCC(NC(c3nnn(C)c3C(F)F)=O)C2)=O)cccc2c1CCOC2 CCCC(CCCNC(=O)C(C)Cc1ccco1)NC(=O)CS(=O)(=O)NC c1(CC(=O)NC2CC(NC(c3ccc(C)cn3)=O)CC2O)cnn2ccccc12 N1(C(CC(=O)OCC)=O)CC(C(=O)NC(CC)C(C)O)C(C2CC2)C1 N1(C(c2cc(C(C)=O)on2)=O)CC(F)CC1CNC(=O)CC(C)(C)N(C)C C1(CCOC)CN(C(C2(C)COC(=O)C2)=O)CCN1C(=O)C1=COCCO1 Cc1cc(=NCc2nc(C3CCCCC3)no2)nc(-c2cccs2)[nH]1 C(=O)(CCC(=O)NN(C)C)NCC(CC)NC(=O)Cc1[nH]cnc1C C(CC(C(C)(C)C)NC(=O)C(C)OCC=C)N(C(CCCC#C)=O)C CC1CCC(CNC(c2ccc(CO)cc2)=O)CN1C(c1n[nH]cc1Cl)=O C1(NC(c2n[nH]c3c2CCCC3)=O)CCCCN(C(c2ccoc2)=O)CC1 C1(C(N2CCN(C)CC2)=O)C2CCC(C2)C1NC(C1CC=CC(O)C1)=O N1(C(C(C)(C2CC2)OC)=O)CCN(C(c2csnn2)=O)C2(CCC2)C1 C#CCCCC(=O)N(C)Cc1ccc(CNC(C2C3CNC(=O)C23)=O)cc1 Cc1cc(=NC(=O)C(F)C2CCN(C(=O)C3CC3)C2)[nH]n1C CC1=NN(C)C(=O)C1CC(=O)N(C)CCN(C)C(c1ccnnc1S)=O C#CC1(C(N2CCOCC(O)C2)=O)CCN(C(=O)OC(C)(C)C)C1 CC1C(NC(C2CC3(CC3)CO2)=O)CCN1C(=O)C(O)C1CC1 c1(N(C)CC2CCN(C(=O)C3=COCCC3)C2)nccc(S(C)(=O)=O)n1 C(=O)(CC(C)(C)CNC(c1cnn(C)c1)=O)NC(C)CSC(F)F c1(CC)cccc(C(=O)NC(CNC(=O)CC2CCC2OC)C(C)C)c1F C(=O)(C1=CCCCCC1)NCC1(C(C)NC(c2coc(Br)n2)=O)CC1 C1(CNC(=O)OC(C)(C)C)CCC2(CC(C(=O)Nc3cncc(Br)c3)C2)O1 c1(NCC(=O)NC2CN(C(c3ncn(C(C)C)n3)=O)C(C)C2)cccc(C#N)c1 C1(NC(c2n(CC)ncc2)=O)CC(CNC(=O)COCCF)C1(C)C C1(NC(CC2(COC)CCCC2)=O)CC2CCC1N(c1ncc(C)c(O)n1)C2 c1(C(=O)NC2C(NC(C(C)CO)=O)CCC2)cncc(C(F)(F)F)c1 C1(C(=O)NCC2CCCCN(c3nnc(CO)s3)C2)CCCCC12CCC2 c1(C(=O)NCCCCCN(C)C(C2CC23CCOC3)=O)cncc(N)n1 c1(C(N(C2CCN(C(C3CCC(N(C)C)CC3)=O)C2)CC)=O)cncc(Cl)c1C S(=O)(=O)(C1CCCCC1)NC(C1CC(c2ccc(Br)cc2)(C)C1)=O C=CCC(C(=O)N1CCC(=CCNC(=O)C(O)CC(=O)OC(C)(C)C)CC1)C(C)C c1(NC(C2C(C(N3CCN(CC(=O)NC)CC3)=O)C2)=O)c(C)cc(Br)cc1Cl C1(CNC(C)=O)CC2(CCN(C(=O)CC3CCC(O)C3)C2)CO1 O=C1NC(=O)C(CNC(C2CCCN(C(c3ccnc(C(F)F)n3)=O)C2)=O)N1 CCCC(C(=O)NCC12CCC(CN(C(c3cnnc(C)c3)=O)C1)C2)C(C)C C1(NC(=O)CCNC(C2COC(=O)N2)=O)CN(C(c2cnns2)=O)CC12CC2 Cc1nc(C(F)(F)F)sc1C(=O)NC1CCCN(C(C2CC3CC2CO3)=O)C1 N1(C(C(c2ccccc2)SC)=O)CC(NC(c2ccc(Cl)c(O)c2)=O)C2(CC2)C1 c1(C(=O)NCCC(C)NC(c2cc(N(C)C)ccn2)=O)cc(F)n(C)n1 CCC(C(=O)NCC1CN(C(=O)CCOC(C)C)CCN1C)C(C)(F)F C1(N(C(Cc2c(CC)con2)=O)C)CCCN(C(C2CC(Cl)(Cl)C2)=O)CC1 c1(C(C)=O)ccc(C(=O)N(C(C)C(=O)N(C)Cc2nc(C)cs2)C)o1 c1(CC)ccc(C(=O)NCC2COCC2NC(=O)C(C)n2cccc2)cc1F C1(NC(CC(=C)C)=O)CC2(C1)CC2NC(C1CCC(CCO)CC1)=O C1(CN(C(c2cnc(C)s2)=O)C)CN(C(=O)CCc2cc(C)n(C)n2)CCO1 C1(NC(CCCC(C)=O)=O)CCC2(CCCN2C(=O)C2Cc3ccccc32)CC1 c1(CNC(C2CCCCO2)C)cc(Br)cc(Cl)c1O C1(C(=O)NC(c2cn[nH]c2)C)CC2CC2N1Cc1cccc(OCCO)c1 C1(C(=O)NCc2occ(C(N(CC(C)(C)C)CCC#C)=O)n2)CN(C)CCO1 c1(C(=O)NCC2(OC)CCN(C(c3ccoc3)=O)CC2)ccn2c(C)cnc2c1 N1(C(=O)Nc2cc(C)cc(Br)c2)CC2(CCCC2)OCC1C C(c1ccc[nH]1)=CC(=O)NC12CC(CNC(C3CC3c3cccs3)=O)(C1)C2 C=C(C)CCC(C)NC(=O)CC1(N(C(=O)C(C)COCC)C)CC1 N1(C(=O)C(O)C2CC2)CCN(C(C2CCCCN2C(=O)Cc2cnc[nH]2)=O)CC1 N(C(=NCCN1CCn2nccc2C1)NC(C)CCC1CC1)C(CC)C C1(NC(CCC=C)=O)(CO)CCN(C(c2cn(CC3CCCO3)nn2)=O)CC1 CC(Cc1ccco1)C(=O)N1CC(C(C)NC(=O)Cn2cnc(C(F)(F)F)c2)C1 N1(C(C(=O)NCC)c2ccns2)CCCCC1CNC(c1ccccc1)=O c1(C(=O)NC(CN(C(C(CCCC)=O)=O)C)(CO)CO)cc(S(=O)(=O)NC)c[nH]1 C1(NC(C(=Cc2ccccn2)C)=O)CCC2(CC1)CC2NC(=O)COCC1CC1 C(=O)(C1CCc2ccccc21)NC1CC(NC(c2n[nH]c3c2CN(C)CC3)=O)C1 N1(C(c2cccc(SCC#C)c2)=O)CCN(C(C2CCC3(CC3)C2)=O)CC1CO C12(NC(CC3CC(SC)C3)=O)CC1CN(C(=O)Cc1sc(O)nc1O)C2 c1(CC(=O)N(C2CCN(C(C(C)C)=O)C2)C)ccc(Br)cc1[N+](=O)[O-] c1(CC)nc(C(=O)NC2CC2CNC(c2cc(F)cnc2O)=O)c2ccccn12 C1(C(N2CCC(Br)C2)=O)CCc2nc(-c3ccc4n[nH]cc4c3)sc2C1 N1(C(=O)CCC2CCC(O)CC2)CC2CCC(C1)N2C(=O)CC1CC1 c1(C(=O)NCC2CCN(C(C3CC3F)=O)CC2(F)F)ccc2ccnc(O)c2n1 c1(C(=O)NCC2CCCN2C(c2occc2Cl)=O)cc2ncccc2cc1Cl C1(NC(C(CCCC)C)=O)CN(C(=O)COCC(C)C)CC2CCCC12 c1(N2C(C(=O)NC3CCN(C)CC3)CC(O)C2)ncnc2sc(Br)cc12 c1(NCC(=C)Br)ccc(S(=O)(=O)NCC2(S(N)(=O)=O)CCC2)cc1F CC1=C(C(=O)N2C3CCCC2CC(CNC(=O)C(O)C(C)C)C3)CCC(C)(C)C1 c1(C(N2CC(C(C)NC(=O)CCC(=O)N(C)C)C2)=O)cc2cnccc2[nH]1 Cc1cnc(F)c(C(N2CCC(CNC(=O)CC3(C(F)(F)F)CC3)C2)=O)c1 c1(OCC)ccnc(N2CC(C(C)NC(C3(Cl)CC3)=O)C2)n1 C1(N(C)C(C2CC2C2CC2)=O)CN(C(C2CCCCC2)=O)CC1O CC1=C(C(=O)N2CCOCC2CNC(C2CC2c2ncccc2F)=O)CCC1 C(=O)(C1=CSCCO1)N(CC(C)NC(c1c(C)nc(C(C)C)o1)=O)C C1(NC(CN(C2CCC2)C)=O)COCCC1C(=O)N(C)OCC(F)(F)F N1(C(C2CCCCC2)C(=O)NC)CCC(C)CCC1CCC.C(C)(C)(C)OC=O N1(C(C(C)(C)c2cnco2)=O)CC2C3CCC(C2C1)N(C(C1CC=CCC1)=O)C3 N1(C(C2CCC(OC)CC2)=O)CC2CCCC(NC(=O)Cc3cc(C)no3)C2C1 N1(C(c2ncc(C)nc2)=O)CCC(C)(C)C(CNC(c2coc(N(C)C)n2)=O)C1 CC1=CC(C)CN(C(=O)COC2CC(CNC(=O)CN3CCOCC3)C2)C1 c1(CC(=O)NCCN(C(=O)C(C)C2(O)CCC2)CC)cccc2nonc12 c1(C(=O)NCC(C)NC(=O)CC(=O)NC2CC2)ccnc2c1nnn2C C1(NC(CCCOCC)=O)CCN(C(C2CCN(CC(C)C)C2)=O)CC1C N1(C(c2c(CC)cno2)=O)CCOCC(NC(=O)C=Cc2scnc2C)C1 C(N=c1ccnc(-c2ccc(C)cc2)[nH]1)C1(NC(=O)C(C)n2cccn2)COC1 c1(C(N2CCCC(NC(c3n(CC)nc(C)c3)=O)C2)=O)cc2ccccc2o1 C1(CNC(COC)=O)CCN(C(c2cccc(C)c2O)=O)CC1C C(=O)(CC(C)CC(C)C)N(CCNC(c1cncc(C(N)=O)c1)=O)CC C1(C(C)NC(C=C(C)C(C)(C)C)=O)CCCCN1C(=O)C(=Cc1c[nH]cn1)F N1(C(c2cnc(OC)s2)=O)CCC2(CCN(C(c3cc(Cl)c[nH]3)=O)C2)C1 c1(C(=O)NCC23C(CN(C(C(F)=C(C)C)=O)C2)C3)cc(Br)cc(N)c1C N1(C(c2nc(C)oc2)=O)CC(CNC(=O)COCc2ccnn2C)C2(CC2)C1 C(=O)(CCCC(=O)OC)N1CC(NC(CCSCCC)=O)C2C1C2 N1(CC(C)(C)NC(Cc2c(C)ncs2)=O)CCN(C(C2(C(N)=O)CC2)=O)CC1 N1(C(C2(C)CC3CCC2O3)=O)CC2(C1)C(NC(c1ccns1)=O)CCS2(=O)=O n1(CC(=O)NCCCN(CCC)C(C2CC2(C)C(F)F)=O)ccc(=O)cc1C C1(C(N2CC(C(N3CCC(C(=O)NCc4ccco4)C3)=O)C2)=O)(CC)CCCO1 C(C(=O)N(C1CN(C(=O)CC2CC=CCC2)C1)C)(C(C)C)c1cnc(C)s1 C1(C(N2C3CC(NC(Cc4nc(C)[nH]n4)=O)(C3)C2)=O)CCS(=O)(=O)C(C)C1 O=[N+]([O-])c1cc(OC)c(OCc2ccc(I)c(Cl)c2)cc1F C(C(=O)Nc1ccc(Cl)cc1F)(C1=CCCSC1)N(CCC)CC1CCOC1 N1(C(CSc2n(C)nnn2)=O)CC(C2CN(C(c3cccc(N)n3)=O)C2)C1 C(=O)(CCS(=O)(=O)NC)NC1CCCN(C(C(=Cc2ccccc2)CC)=O)C1 c1(C(=O)NC(CCNC(C(C)Cn2cccn2)=O)C)cc(Br)cnc1O O=C1Nc2c(C(N3CC4CN(C(C5CCCS5)=O)CC(C3)O4)=O)cccc2C1=O c1(OCC)ccnc(N2CCN(C(=O)CCN3CCOCC3)CC2)n1 C(=O)(C(O)CC(F)(F)F)NCC1C(C(=O)NCC(CC=C)(F)F)CCCC1 C#Cc1ccc(C(=O)NCC(C)N(C)C(c2ccc(F)c(CO)c2)=O)cc1Cl c1(NCC(CC)O)ccc(S(=O)(=O)NCC2CCOC3(CCCCC3)C2)cc1Br N1(C(c2ccc(N)cn2)=O)CCC(CNC(=O)CC(F)(F)C(F)F)C(F)(F)CC1 c1(-c2c(C(N(c3ccc(CC)cc3)CC)=O)ccs2)ccc(C)nc1F c1(OC)nc(NC(=O)CN2CCN(S(C)(=O)=O)CC2)ccc1-c1nn[nH]n1 Cc1cnc(NC(c2ccnc(-c3cccc(O)c3)c2)=O)c(Br)n1 C1(Nc2ncc(C(=O)OC)cn2)CCC2CN(C(=O)Cn3cccn3)CC12 C1(C)(CC)C=C(C(=O)N2CC(NC(=O)CC(C)(C)OC)CC2C)C1 Cc1ccc(C(N2CC3CC2C3NC(=O)CC(C)C)=O)nn1 Cc1noc(C)c1CC(N1CCC(C(C)(C)NC(C2COCCO2)=O)C1)=O c1(NCC(N(C)C(C2CC2C2CCCCC2)=O)C2CC2)cc(S(C)(=O)=O)ncn1 Cc1ncn(C)c1C(=O)NC(C)CCNC(=O)CCCCC1CCCCC1 C(=O)(C(C)CC(F)(F)F)N1CCC(CNC(C(CCC)(C)O)=O)CC1 C1(C(=O)OC)Cc2n[nH]cc2N(C(=O)C(c2ccc(Cl)cc2)O)C1 C1(CC(N2CC3C(NC(C4C5CC6C(C5)C46)=O)C3C2)=O)CCC2(CCC2)O1 c1(C(=O)NC2(CCC(N)=O)CC2)ccc(OCC(=O)N(C)Cc2ncco2)cc1 CCCC(C)(CC)C(=O)N1CCC(O)(C(C)NC(=O)COC)C1 C(CC(C)(C)C)(C(=O)NC(C)C(=O)N(C1CN(C)C1)C)OC Cc1cc(N2CCC(CC(N3CCNCC3C3CCC3)=O)C2)nc(C)c1 C(=O)(C1c2ccccc2C2CC1C2)N1C(CC)CN(C(=O)CC(C)SC)CC1 N1(CCC(=O)N(CC)Cc2ccccc2)CCc2nc(O)ccc2C1 CN(C)NC(=O)CCC(=O)NCC(C1CCCN(C(C2SCCS2)=O)C1)(C)O C=CCCC(C(=O)OC)NC(=O)CCN(CCO)C(c1cnc(O)n1CC)=O C1(NCC(CN(c2ccccc2F)C=O)O)CCCC(c2cccs2)C1 N1(C(C(C)(N(C(C(C)N(C(C)=O)C)=O)C)C2CC2)=O)CCC(NC(N)=O)CC1 C(C)(CC(=O)N1CCC1CC(=O)N(CC(C)CO)C)=C(C)C c1(C(=O)NCCCCCNC(c2cc(CC)sn2)=O)cc(C)nn1C(C)(C)C c1(CC(=O)Nc2cnc(OC)nc2)c[nH]c2cccc(-c3cnc(F)c(F)c3)c12 C(CS(=O)(=O)N(CCC(C)C)CCC#N)(C1CCOC1)OC O=C(C1CCCn2cnnc21)NC1CC(NC(C2CCCCNC2=O)=O)C(O)C1 C12(NC(C(CC)O)=O)CC(CNC(c3cnc(S)[nH]3)=O)(C1)OC21CCC1 c1(C(=O)NC2C(CNC(C3(C(=O)NC)CC3)=O)C2)ccc2cc(OC)ccc2c1 C1(C2CC2)(OC)CN(C(=O)CC(C)CNC(=O)OC(C)(C)C)C1 C1(C)(C(N(CCCC)C)=O)CCCN(Cc2cccc(CC(=O)O)c2)C1 CC1CCN(S(=O)(=O)CC(=O)N(CCCNC(C2CC3(C2)CC3F)=O)C)CC1 c1(OC)cccc2c1N(C(C1NCC13CCOCC3)=O)CC2 c1(NC(C)=O)ccc(F)c(C(N2CC=CC2CNC(=O)C(O)C(C)(C)C)=O)c1 Cc1cccc2oc(C(=O)NCC3CCN(C(C4(C5CC5)CC4)=O)CC3O)cc12 c1(C(N(C(C)C(=O)N2CC(C3CCCO3)C2)CC)=O)cnc(C2CC2)o1 c1(OC(C)C(=O)N(c2cccc(CN3CCC(O)CC3)c2)C)cc(Cl)ccn1 N(C)(C1CN(C(=O)CCCCSC)CCc2ccccc21)C(C1(CC#C)CC1)=O c1(NC(=O)NC2C(CC=C)C(O)C2)cccc(P2(=O)CCCC2)c1 c1(CCCC)cc(C(N2CCCC2CN(C)C(C2(C#N)CCCO2)=O)=O)c(C)o1 c1(C(=O)NCC2CCN(C(=O)C(F)C3CC3)C2)cnc2[nH]nnc2c1 c1(C(N2CC(CCC)C(NC(=O)Cc3cccnc3)C2)=O)cc(C)ccc1CC C1(N(CCOC)C(c2cscc2Cl)=O)CCN(C(C2(Cl)CC2(F)F)=O)CC1 C(C1CCCc2scnc21)N1CC(=O)CC12CCC2 c1(C(N(CCC)CCNC(c2ccnn2C2CCC2)=O)=O)cccc2c1OCC2 C(C(CO)(CO)NC(c1ocnc1C)=O)N(C(CSCCOC)=O)C c1(C(c2ccccc2)N(CC(C)C)CCCO)ccc(Br)c(C(F)(F)F)c1 N1(C(CC2CCC(=O)NC2)=O)CC2(C1)CN(C(=O)C=C1CCC1)CC2CO N1(C(c2cncc(OC)n2)=O)Cc2n[nH]cc2C1C(=O)N(C)C(C)C1CC1 C1(c2ccccc2)(NC(C(CC)n2ccnc2)=O)CCN(C(=O)CSC2CC2)C1 CC(CC(C)NC(c1ccnn1-c1ccccc1)=O)NC(=O)CCC1CCOC1 C1(C(=O)NC2CCCC(CNC(Cn3c(C)ncc3)=O)C2)CC2CC(=O)C1O2 C1(CC)CC(N=c2cc(C)nc(NCc3nnc4cccnn34)[nH]2)C1 N1(C(C=CC(N)=O)=O)CC2CC(C1)C(CO)C2NC(c1cc(C(F)(F)F)no1)=O c1(SC)c(C(=O)N(C2CC(NC(c3snc(Cl)c3Cl)=O)C2)C)cnn1C c1(C2(C(=O)NCC(CNC(C3(OC)CC3)=O)(C)O)CC2)ccc2c(c1)OCCO2 C1(C)(NC(CC2(OC)CCCC2)=O)CCN(C(c2nnc(C)s2)=O)CC1 Cc1cc(N(CCCNC(c2ccc(F)cc2C)=O)C)nc(C(C)C)n1 C(=O)(C(CCN(C)C)N(C)C)NC(C1CCN(C(=O)CC=C(Cl)Cl)CC1)C c1(CNC(c2c(COC)onc2C)=O)nnc2n1CCN(C(=O)C=CC(=O)OC)C2 c1(C(=O)NC2(C)CCN(C(C3CCCOC3)=O)C2)ccc2c(c1)CCC2=O CC1CC(C(=O)N(C)CCOCCNC(C2(C3CCCO3)CCCC2)=O)CN1C c1(CC(=O)NC2CCC(NC(C3(C)C(C)C3)=O)CC2)cccc2ncccc12 C#Cc1ccc(C(=O)NC2CCN(C(=O)CC3CC4CC4C3)C2(C)C)cc1 N1(C(CSCC#C)=O)CC2CC(C1)CN(C(=O)CCCCCC(C)C)C2 N1(C(c2cnc(CCCC)s2)=O)CC2(C1)CN(C(c1n[nH]cc1CC)=O)CC2CO n1(CC)cc([N+](=O)[O-])c(C(=O)NCC2CN(C(=O)C(C)(C)C(C)(F)F)CCO2)n1 CC(C)C(C(=O)N1CCOC(CC(=O)N(CC(O)CO)C)C1)C(C)C c1(C(=O)NCC2CCC(CNC(COCC)=O)CC2)cc(=O)c(OCCO)co1 Cc1cc(C(=O)NCCCCNC(C2(C)CNC(=O)C2)=O)cc2ccoc12 C(=O)(CCCC(C(=O)OC)N(C)CCNC(C1CCOCC1)=O)OC C1(C(C)NC(=O)C2=CCC2)CCCN(C(C2CC(=O)N(c3nccs3)C2)=O)C1 C#Cc1ccc(CNC(=O)CCC2CC(NC(C3CC(F)C(=O)N3)=O)C2)cc1 CCC(CC)C(C)C(=O)NCC1CC2(CC2)CN1C(=O)Cc1cnco1 C1(CC(=O)N(C2CCCN(C(C3(C(N)=O)CC3)=O)C2)CC)CCCC(=O)N1 Cc1cnc2c(C(N3CC(NC(=O)CC4CCCC4)CC(O)C3)=O)cnn2c1 c1(OC)ccnc(CN2CCN(CCCNC(c3cncc(O)c3)=O)CC2)c1 C(=O)(C(CCOCCO)NC(=O)CN1CC2CC2C1)NCC1(N(C)C)CCCC1 C12(C(N3CCC(CNC(CN(C)CC)=O)C(C)C3)=O)CCC(CC1)C(C)O2 N1(C(c2c(N)c(Cl)ccc2)=O)CC2(CCC(CNC(=O)CCc3cnn[nH]3)O2)C1 CCC(C)CC(C)C(=O)NCCNC(C12CCC(F)(CC1)C2)=O C=C(C)C1OCCC1C(=O)NC1CC(NC(=O)C(C)(C)C2CCCCC2)C1 N1(C(c2c(C)ccnn2)=O)C2CC1CN(C(=O)C(N1CCOCC1)C)C2 Cc1c[nH]cc(C(=O)NC(C2CCN(C(=O)CCCOC(C)(C)C)C2)C)c1=O N1(C(CCCc2cc(C)no2)=O)CCC2OCCN(C(c3csnc3C)=O)C2C1 Cc1cccc(C)c1CC(=O)NCCCNC(=O)CC1CN2CCN1CC2 N1(c2sc(C(=O)OC)c(Cl)n2)CC(C)(C)CC1CNC(=O)C1=NOC(C)C1 N1(C(c2nnn(C)n2)=O)CCC(C2CCN(C(c3snc(O)c3Cl)=O)CC2)C1 C1(CC)CC(C(F)(F)F)CCN1C(C12COCC(COC1)O2)=O c1(C(N2CC(NC(c3c(C)cccc3)=O)C(F)C2)=O)ncnc(O)c1Cl N1(C(C2CCC(CC)O2)=O)CC2(CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)C1 c1(C(=O)NC2(C)CC(NC(C3C(C)(C)C3(C)C)=O)C2)cc(Cl)ccc1C(F)(F)F c1(C(N2CCC(N(C(=O)C(F)OC)CC)C2)=O)ccnc(C)c1C C(CC1=CCN(C(c2cnnc(Cl)c2)=O)CC1)NC(=O)CCc1ccc(Cl)cc1 N1(C(c2cc(CC)on2)=O)CCOC2(C1)CN(C(C1(S(C)(=O)=O)CCCC1)=O)C2 C(CCCC(CO)NC(c1ccc(F)s1)=O)NC(COCCCCCC)=O CC(C(=O)N(C)CCNC(=O)COCCF)NC(c1cccs1)=O C(C(C)C(=O)Nn1ccccc1=O)N(C(C(CCC)CCC)=O)C C1(C(=O)NCC(C)(C2CCC2)NC(C(C=C=C)C)=O)CCOC2(CCOCC2)C1 N1(C(c2cnc(Cl)s2)=O)CCN(C(c2cc(O)ccc2F)=O)C(CC(F)(F)F)C1 Cc1cc2ncc(C(N3CCC(C(=O)Nc4ccc(CCO)cc4)C3)=O)cn2n1 C1(C(F)(F)F)(C(=O)NCC(=C2CN(C(CCCOC(C)C)=O)C2)F)CCOCC1 C(c1ccc(OCCN(C)C)cc1)=CC(=O)NC1CN(C(Cc2c(C)ccs2)=O)C1 C(=O)(C1=CCCN(Cc2cnc(Br)c(F)c2)C1)NC(CC=C)CO N1(C(c2cc(CCC)on2)=O)CCN(C(C2CCN2CC)=O)CC1CS(C)(=O)=O Cc1nc(C(C)C)nc(O)c1C(N1CCC(CF)(NC(=O)C(C)O)C1)=O C1(CNC(C=CCC)=O)CC(NC(c2ccc(C(C)CC)cc2)=O)CCO1 C1(N(C(c2ccccc2OC)=O)CC)CN(C(=O)C(C(C)O)N(C)C)C(C)(C)C1 C1(C(=O)NC2C(CN(C)C)C2)CC(C)(C)CCN1C(C1CCCCC1(C)C)=O C(=O)(C(O)CCN(C)C)NCCC(C)NC(=O)CC(c1ccccc1)N(C)C CC1=C(C)C(NC(=O)C(=O)NC(c2ccccc2)CC2CCOCC2)CCC1 C1(CNC(c2cc3ccsc3s2)=O)CC2CN(C(=O)C=Cc3ccncc3)CC12 c1(CC)conc1C(=O)NCC1CCCC1NC(c1ccc(-c2ccco2)o1)=O N1(C(Cc2nc(C)sc2)=O)C2CCCC1CN(C(C1CCCC(F)(F)CC1)=O)C2 C1(C(N2CCCC(N(C(c3ncn(C)n3)=O)CC)C2)=O)CCCCC(=O)N1 Cn1cc(C(=O)NC2CN(C(=O)C(=Cc3cccnc3)F)CC23CC3)ncc1=O c1(C(C(N2CC(NC(C3CC3CF)=O)(CO)C2)=O)O)cccc(F)c1 S(=O)(=O)(c1c[nH]ccc1=NCCCCCS(C)(=O)=O)NC(C)CCC1CCCO1 c1(CNC(C2(COC)COC2)=O)cncc(C(=O)NCC(O)(CO)CO)c1 C(=O)(C1=COCCO1)NC1C(CNC(c2cnc(C(C)(C)C)nc2)=O)CCCC1 N1(CC(=O)NC2C(CNC(=O)COC3CCCOC3)CCC2)CCC(CO)CC1 C1(C)(CC(=O)N(CCCNC(=O)CCCn2cccn2)C)CCS(=O)(=O)N1 N1(C(C2N(CC)CC2)=O)CCC(O)(CN(C(=O)CC2CCCC(OC)C2)CC)CC1 c1(C(N(CC(CNC(Cc2ccc(CC)cc2)=O)O)C)=O)ccc2nn[nH]c2c1 c1(OC)cccc(OC)c1C(=O)NCC1CCC(NC(=O)C=C(Cl)Cl)CC1 O=C(CC1COc2ccccc21)NC1CN(C(c2nc3c(Br)cccn3n2)=O)C1 c1(C(N2CCC(CN(C(C(c3ccccc3Cl)C)=O)C)C2)=O)ccc(F)c(N)c1 C1(C(N2CC(O)(CCNC(Cc3cc(C)n(C)n3)=O)C2)=O)CCn2cnnc2C1 C1(C(N(CC(C)CNC(C2CC3(C2)CC(CO)C3)=O)C)=O)CCC2C(C1)C2(F)F N1(C(CC(CC)CC)=O)CCC2(NC(c3ccc(SC)o3)=O)CCCC12 N1(C(C(CC)SC)=O)CC(CC(=O)NC2C(C)(C)C2(C)C)C2(CC2)C1 C1(C(=O)NC2COCCC2O)CC2(CC2)CN1Cc1ccncc1Br C1(NC(c2ccc(O)cc2)=O)CC(C(=O)NC2CC3CCC2O3)C12CCC2 N1(C(c2c(C(=O)O)nc(-c3ccccc3)s2)=O)CC2CCC1C2N C(=O)(CCC(C)(F)F)N1CC(C(C(=O)N(C)Cc2cncnc2)O)C1 C=CCC(C)(C)C(=O)N(CC)CC1CN(C(=O)CCOC(C)CC(C)C)CCO1 c1(C(=O)NCC(c2cn(CC)nc2)=O)cnc2c(Br)c(C)nn2c1 C(C)(N=c1[nH]nc(C(C)(C)C)o1)C1OCCN(C(c2ccc(C(C)C)s2)=O)C1 C1(F)(COC)CCN(C(c2ccc(-n3cnnc3)c(I)c2)=O)CC1 C1(S(N)(=O)=O)(C(N(C2CCCCC2)CCNC(CN(CC)CC)=O)=O)CCC1 c1(CC)nn(C)c(Cl)c1C(N1CCOCC(C(C)(C)C)C1)C(=O)NCCC#N N1(C(c2cc(C3CC3)[nH]n2)C(=O)NCc2ccccc2)CCc2cccnc2C1 CCC(C)C(O)C(C)C(=O)NCC(C)(O)CNC(c1cccc(O)c1F)=O Cc1nc(Cl)nc(N2CCC(N3CCN(C(C4CCCN4C)=O)CC3)CC2)c1Cl CC(Cc1ccco1)C(=O)NCCOCCNC(=O)Cc1coc(C(F)F)n1 c1(N(C(C)C)C)ccccc1C(=O)NCC1CCN1C(C1CNC(=O)N1C)=O c1(C(=O)NC2C(CNC(CCC3CCC(C(N)=O)O3)=O)C2)ccc2n[nH]cc2c1F c1(N(C(=O)NCCCC2CCOC2)CC)nc(C)nc(=N)[nH]1 c1(OC)csc(C(N2CCN(C(C3(C(N)=O)CCC3)=O)CC2)=O)c1OC C1(CNC(C(CC)F)=O)CN(C(C2(COC)CCOCC2)=O)CC(C)(C)O1 n1(CC)nc(C(=O)NC2(CNC(=O)CC3CCC(=O)NC3)CCCCC2)cc1O C1(NC(C(C)(C)NC(C)=O)=O)CC2(C1)CC(C(=O)NC1COCCC1O)C2 N1(C(c2cccc(SCC)c2)=O)CC(N(C)C(C23CC(OC)C2C3)=O)C2(CC2)C1 c1(C(=O)NCC2(O)CCCN(C(C(C=C)O)=O)CC2)cccc2c1nc(O)n2C N1(C(c2c(C)ccs2)=O)CCN(C(c2cn(C)nn2)=O)CC1C1CCCC1 N1(C(Cc2c(C)cccc2)=O)CCN(C(=O)C(CO)c2ccccc2)C(C#N)C1 Cc1cncc(C)c1C(=O)NC1CC(N(C(=O)CC(F)(F)F)C)C1 C1(CN(C(C(=O)NCC(=C)C)C)C)CCN(C(c2coc(C3CCC3)n2)=O)C1 C=CC1(C(=O)NC2CN(C(=O)C(C)CC3CCCC3)CC2C)CCOCC1 CCCC(C(O)C(=O)Nc1cc(C)ccc1C)NC(=O)C(C)(C)COC C=C1CC(C)(C(=O)NC)C1.C(C(C)(C)CN)C1CN(C(=O)CNc2ccccn2)C1 c1(CC)csc(C(C(=O)NC(C)(C)C)N(CC)Cc2nc(C)cs2)c1 C1(NC(C(C)(C)CC2CC2)=O)CCOC12CCN(C(C1(C)CC3CC3C1)=O)CC2 C(=O)(CCN=c1[nH]ccs1)N1CC(F)(CNC(c2cnc(CC(C)C)[nH]2)=O)C1 c1(-c2cccc(CNC(C3(O)CC3)C)c2)c(O)cccc1O N1(C(CCCC#C)=O)CC(CNC(c2nc(Br)c(C)s2)=O)C(F)(F)C1 C1(C)(C(=O)OC)CCCN(C(c2ccc(-c3ccc(C)c(OC)c3)nc2)=O)C1 CC1CN(C(c2cscc2C(F)(F)F)=O)CC1NC(=O)C(C)(C)c1cnn(C)c1 CC(CCC(F)(F)F)NC(=O)CCNC(C1CCCCC(=O)C1)=O Cc1c(C(=O)NCC=CCNC(=O)C(C(C)C)NC(N)=O)[nH]c2c(C)cccc12 N1(C(C(C)S(N)(=O)=O)=O)CC(C)CN(C(C2CCCC(C)(C)C2)=O)CC1C N1(C(C)C)CCCC(CC(=O)NC2CCCC(NC(=O)Cc3ncc(Cl)s3)C2)C1 O=C(CC(F)(F)C(F)(F)F)NC1CN(C(=O)COC2CCCCC2)C2CC12 C1(CCOCCO)C(=O)N1.C(CNC(C)=O)(C(=O)N1CCC(CSC)C1)OC c1(C(N(CCN(C(C2C(C)=C2)=O)C(C)C)C)=O)ccc(F)c(C)c1Cl Cc1n[nH]c(C)c1SCC(N1CC(CNC(=O)CSCC(C)C)C(C)C1)=O C(=O)(C(CN(C)C)C(C)C)NC1(C)CN(C=O)C1.C1(CC#C)CCOC1 c1(C(=O)NC(C2CCCN2C(=O)CC(C)(C)C#N)C)c(OC(F)F)cccc1Cl C(=O)(CC(C)C(F)F)NC1(CNC(CSCCOCCOC)=O)CCCC1 CCCC(C)(CC)C(=O)NCc1cc(C)c(C(=O)NCCCN(C)C)o1 C(=O)(CC(C)C(=O)OC)NC1(C(=O)NCC(=O)OCC)CC1C C1(NC(c2ccccc2Cl)=O)CN(C(=O)C(O)c2ccsc2)CC1O C1(C(=O)NCC(C(=O)OC)O)N(C(=O)CN2CCNC(=O)C2)CCC1(C)C c1(OC)ccccc1C1(C(=O)N(CCCCCCNC(=O)C(C)O)C)CCC1 n1(CC(=O)N(C(CNC(c2ncn(CC)c2)=O)C)C)c(C)cc(C)nc1=O Cc1ccc(Cl)c(C(=O)N(C)CC2(NC(=O)C(c3ccc(Cl)cc3)CO)CC2)c1 N1(C(c2cc(OC)cc(OC)c2)=O)CCCCC12CC(NC(C1CC1CF)=O)C2 C1(CC)C(NC(=O)CC2CCCOCC2)CCCN1C(=O)C=Cc1cnccn1 CCC(O)(CC)CCNc1ncnc(NC2COCC2OCC)c1C CC(C)(C(=O)NC1CC(O)(CNC(c2ccc[nH]2)=O)C1)Oc1ccccc1 c1(C(N2CCN(C(C(CCC)CCC)=O)CC2C)=O)ccc2c(C#N)c[nH]c2c1 C1(C)(CNC(Cn2c(C)cnc2)=O)CCN(C(=O)CC2CCC(F)(F)C2)C1 CC1CCC(O)(C(=O)NCC2CCN2C(C2CCC(C)(C)C2)=O)CC1 C(N=c1cc(C)[nH]c(=NCc2n[nH]cc2C2CCC2)[nH]1)c1c(OC)cc(F)cc1 c1(C(=O)NCC2(O)CN(C(C(C)NC(C)=O)=O)C2)[nH]nc2ncc(Br)cc12 N1(C(CCCSC)=O)CCC(C(F)(F)F)C(NC(c2cc(C(N)=O)no2)=O)C1 C1(C(=O)NC2CN(C(C(=O)NCC)=O)C2)CC(c2cc(F)ccc2F)=NO1 N1(C(C(CC)C)=O)CCN(C(c2cc(C)sc2C)=O)CC(C)(F)C1 c1(CCOCC)nc(C(=O)NCCN(C(c2cncs2)=O)CC2CC2)co1 c1(SCC(N2CC(O)(CNC(CC3C(C)OCC3)=O)C2)=O)cccc(C(F)F)c1 C(CC(=O)N=c1[nH][nH]c(-c2ccccn2)c1C)(c1cccnc1)N(C1CCOC1)C N1(CCCNC(CC(C)NC(N)=O)=O)Cc2ccccc2C1 C(=O)(C1=CCN(C(=O)C2=NOC(C)C2C)CC1)NC(C1CCOC1)C#C N1(C(CNC(CNC(C)=O)=O)=O)CCC(CO)(NC(c2n[nH]c(C)c2C)=O)C1 c1(C(=O)OC)cc(F)c(F)cc1-c1cn(CC(C)CC2(C)OCCO2)nn1 c1(C(C2CCOCC2)CNC(c2cc(C)no2)=O)cnc(C(F)(F)F)nc1 N1(C(C)=O)CCCCC(CNC(=O)Cn2c(-c3ccccc3)c(C)sc2=O)C1 C1(N(C(C2CC2CF)=O)OCC)CCN(C(=O)CCCN(C)C(C)C)CC1 c1(C(N(CCCNC(C2CC2(Cl)Cl)=O)C)=O)cnn(-c2ccccc2)c(=O)c1 C1(O)(CNC(CCSCC)=O)CCCN(C(c2cncn(C)c2=O)=O)C1 CC(C)(CO)CCN=c1[nH]c(=NCc2cccc(N)n2)[nH]c2c1CCCC2 C1(C(=O)NC(C(C)(C)NC(CCc2cnc(C)o2)=O)C)CC2OC1C1CC21 C1(C(=O)NC2(CN(C(C(C)OCCCC)=O)C)CC2)CC(c2ccccc2)=NO1 C(=O)(C(CCSC)OC)NC1CC(CCNC(CN(CCC#C)C)=O)C1 O(NC(=O)C1=CC2(CCN(C(=O)C(C)NC=O)C2)C1)CC(C(C)C)O C(=O)(CC(CC(N)=O)CC(C)C)N1CC2(CCN(C(COCCOC)=O)CC2)C1 C1(CC=C)(NC(=O)CC2CC(C)(C)CO2)CCN(C(=O)CS(C)(=O)=O)CC1 Cc1cc(C(=O)NC2CCN(C(=O)COCC(C)(C)C)C2C)nc(C)c1 N1(C(C(C)=C2CCCC2)=O)CC2CCC1CN(C(=O)CN1CCCNS1(=O)=O)C2 c1(C(C)NC(=O)NC2(C3CC3)CCCCC2)cc2cc(Br)ccc2[nH]1 c1(OC)cncc(OCC(C)OC(C2CCCC2c2ccccc2)=O)c1 N1(c2ncc(OC)c(C)n2)CCC2(CCCN2C(c2ccc(Cl)c(O)c2)=O)CC1 C1(C(=O)NC(C2N(C(CNC(=O)NC)=O)CCC2)C)CCn2ncnc2C1 CC(C)C(F)(CNC(=O)CN1CCN(C)CC1)C(=O)N1CCC1C1CCCC1 C1(O)(CNC(c2sc(C)c(O)n2)=O)CC2CCC(C1)N2C(C1(C)CCCOC1)=O CCCCCN(CCC(=O)NC1CN(C(C2(CS(N)(=O)=O)COC2)=O)C1)C c1(C(=O)NC2CC(C)(NC(CC(CC)OC)=O)C2)cc(Cl)c2c(c1)OCCO2 c12ccc(F)cc1CN2C.C(O)(C(F)(F)F)C1CCC1.C12CC(C1)CNC(=O)N2 c1(C(=O)OC)cccc(NC(C(C)CC2CCOCC2)c2nnnn2CCF)c1 N1(C(C(C)=CC2CC2)=O)CC(C)(C)OCC1CNC(C1(C2CCC2)CC1)=O C1(C)(C(=O)NCCN(C(=O)COCC2CCCCO2)CC)CCN(C)C1 C12(NC(C(C)NC(=O)NC)=O)CCCC1N(C(=O)CCc1ncc(F)cn1)CC2 C1(CNC(CC2C(C)(C)C2)=O)CC2CC2N1C(C1(F)CCCCC1)=O c1(C(C)C)nc(NC(c2csc(C3CC3)n2)C)cc(N2CCC(Cl)=C(Cl)C2)n1 C(=O)(C(CC(C)C)C(C)C)NC1(CC)CCCN(C(c2cn(C)nn2)=O)C1 c1(OC)ccnc(C(=O)NCCC2CC(NC(C3(C)CC3(Cl)Cl)=O)C2)c1N N1(C(COC)=O)CC2CCN(C(c3cnn(C4CCCCO4)c3)=O)C(C2)C1 N1(CCNC(C(C)NC(CC)=O)=O)CCN(C(=O)CC2CN(C(C)=O)C2)CC1 N1(C(C2CC(OC)C2)=O)CCC2(CCN(C(=O)CC3(n4cncn4)CC3)C2)C1.C CCCC(C(O)C(=O)NCC(C1CCC1)OC)NC(C1CC(=O)CC12CCC2)=O N1(CC)CCN(C(=O)CC2CCC(NC(c3cc(C)ncc3Cl)=O)CC2)C(C)C1 c1(C(=O)NCC2CN(C(C3(C(F)F)CC(=C)C3)=O)CC2C)cc(C)c(C)nn1 c1(C(N(C2CCOC2)CC)=O)ccn(CCNC(=O)CCC2CCCC2)c1 C(C)(C(=O)NCC1(C(=O)NCC2(CNC(C)=O)CCC2)CCC1)OCCCC c1(N2CCCN(C)CC(C)C2)cccc(S(=O)(=O)N2CC3CCOC3C2)n1 CC12CN(C(C3CC4CCC3O4)=O)CC1(C)CN(CCC1=CCCCC1)C2 Cc1nc2cc(C(=O)NC3CCC3NC(c3c[nH]nc3C(C)C)=O)c(F)cc2[nH]1 Cn1ccc2c(C(=O)NC3CN(C(=O)CCc4cnco4)C4CC34)ccnc12 CC1(C)CC(C(=O)NC2CC(=C3CC3)C2)CN(C(C2(F)CCOC2)=O)C1 N1(C(c2cc(C)c(Br)o2)=O)CCCC(CNC(C2(C)CCCO2)=O)CC1 C(C(C(=O)NC(C)C(C)C)NC(=O)C(C)=C(C)C)OCC c1(N2CC3CN(C(c4sc(Br)cc4Br)=O)CC32)ncc2sccc2n1 c1(C(N2CC(COC)N(C(C3CC3C3CCC3)=O)CC2)=O)c[nH]c(C)c(Cl)c1=O N1(C(c2cnn(C)c2F)=O)CCC(NC(=O)Cc2ccc(F)cc2F)CC(O)C1 N1(C(C(C)NC(COC)=O)=O)CC2(CC2)CC1CNC(=O)CC1CC2(CCC2)C1 N1(C(CCC=C)=O)CCC(c2ccccc2)(NC(=O)Nc2ccc(NC)cc2)C1 C(C(CCC)CC(C)C)NC(C(CCCOC)NC(CCCC#C)=O)=O C(CC(O)C(=O)N1C(C(=O)NCCC2CCN(C)CC2)CCC1C)N(C)C c1(OC)c(-c2sc(CN3CCC(CN(C)C)CC3)cc2C)cccc1F N1(C(C2C(=C)CC2)=O)CC(C(N)=O)(CNC(c2ccn(-c3ccccc3)n2)=O)C1 c1(CN2C(C(=O)Nc3cc(OC)ncn3)CC2)ccc(F)c(F)c1Br N1(C(C(CCCCC)O)=O)CC2(C=C(C(=O)Nc3ccc(C)nc3C)CO2)C1 CN1C(=O)CCC(NC(C2COCCN(C(c3cc4n(n3)CCO4)=O)C2)=O)C1=O C1(NC(C(c2c(C)noc2C)C)=O)CN(C(=O)C2=CSCCO2)CCC1CO Cc1nc(C(=O)NCc2ccsc2C(=O)NCC2CCSC2)cc(O)n1 c1(NC2CC(OC)C2)cc(C)c(S(=O)(=O)N2CCCN3CCCCC3C2)cn1 N1(C(C2CCS(=O)(=O)N2)=O)CCC(F)(F)C(CNC(C2(C3CC3)CCC2)=O)C1 C1(NC(c2ccccc2Cl)=O)COCCN(C(c2cc(Cl)ncc2F)=O)C1 N1(C(=O)CCn2cccn2)CCC2CCC(C1)N2C(=O)C=CCOC1CCOCC1 C(=O)(C(CC(F)F)N(C)C(C1CCCC1F)=O)NC(CC)C(C)(C)O N1(C(c2c(CC)ccs2)=O)CCCCC1CCC(=O)NCC(Cl)Cl C1(NC(CCC(C)OC)=O)COC2C(NC(=O)Cc3cc(C)cc(F)c3)COC12 Cc1ccc(C(=O)NC2CC(NC(C3CCCC3(F)F)=O)C2)c(C)c1 C=CCC(F)(F)C(=O)NCCC(CC)(CC)NC(C1CC(CF)C1)=O c1(CNC(=O)CN2CCCC(c3ncc[nH]3)C2)cc2c(s1)CCC2 C12(NC(CCCOCC)=O)CCN(C(c3conc3CC)=O)CC1C2 n1(CC(=O)NC(CCN(C(CC(C)OC)=O)C)C)c(O)nc2ccccc12 C=C(C)C(C)(C)C(=O)NCC1(NC(=O)C(c2ccnn2C)C)CCOC1 N1(C(c2cnc(C)[nH]2)=O)CC2(CC2)CC1C(=O)N(C(C)C)Cc1cccnc1 C1(NC(C(C)C(F)F)=O)CC(C2CCN(C(c3c[nH]nc3C3CCC3)=O)CC2)C1 N1(C(c2c(CC)nc(C)[nH]2)=O)CCN(C(=O)C(C)Cn2ccc(C)n2)C(C)C1 c1(C(=O)Nc2cc(Cl)ccn2)cc(F)ncc1NS(=O)(=O)CC1CC1 CC1CC(C)CN(Cc2ccc(CN3CC(C(F)(F)F)CCC3=O)cc2)C1 c1(C(=O)NCc2c(C(=O)OCC)cc[nH]2)ccc(-n2ccc(CC)n2)cc1 C1(NC(CSCC(C)C)=O)CCOCC1NC(=O)CC(c1ccc(F)cc1)O N1(C(Cc2c(C)ccnc2)=O)CC(NC(=O)C(C)N(C)C)C2(CCOCC2)C1 CCC(CC(F)(F)F)C(=O)N(C)CC1(CNC(c2cccc3nc[nH]c23)=O)CC1 C(CCCC(=O)NCC12COC(CNC(=O)CC(C)N(C)C)(C1)C2)N(C(C)=O)C N1(C(c2c(C)ccnc2F)=O)CC2(CCC(C(=O)NCc3ccnc(F)c3)O2)C1 N1(C(C(C(CC)C)OC)=O)CCN(C(c2nc(Cl)cs2)=O)CCC1C CCC(CC(=O)N(c1ccccc1F)CC)NC(=O)C(C)(C)OCC N1(C(c2n(C(C)C)ncc2)=O)CCCC2(CCN(C(=O)CC(C)(C)F)C2)C1 C1(NC(C=CCCC)=O)CCC(C)(CNC(c2cc(C)oc2C)=O)CC1 c1(C(=O)NCC2(F)CN(C(C(C)=CC3CC3)=O)C2)ccc2sc(C)nc2c1 C1(CC=C)(C(=O)N(C2CCC3CC23)C)CCN(C(c2c[nH]nc2OC)=O)C1 n1(CC(=O)NC2N(C(CNS(CCOCC)(=O)=O)=O)CCOC2)cc(F)ccc1=O S(=O)(=O)(c1ccc(N(C)Cc2cccnc2)c(Cl)c1)N1CC2N(C)C(CCC2)C1 Cc1cn2cc(C(N3CCN(C(=O)CCCC4CCC4)C(C4CC4)C3)=O)sc2n1 C12(C(=O)NC(C(C)NC(C3CC=CCO3)=O)C)CC3CC(F)(C1)CC(F)(C3)C2 C(CCCCC(=O)N(C1CC1C)C)n1cc(-c2ccc(C)n2C)nn1 Cn1nc(C(=O)N(CCNC(C2CC23CC3(F)F)=O)C2CC2)c(Cl)c1Cl C(CO)(C(F)(F)F)NC(C1CCC(C(=O)Nc2cc(-c3ccco3)on2)C1)=O C=CCCCC(=O)N(CCCNC(=O)CCCOOC(C)(C)C)C.N1C(=O)OCC1 N1(c2ccnc(C(C)C)n2)CCC2(CC(NC(=O)CC(C)c3ccncc3)C2)C1 N1(C(C(CC)n2ccnc2)=O)CCOCC1CNC(c1cnn(C(F)F)c1)=O C(=O)(CC1OCc2cc(Cl)ccc21)N1CCC(N(C(c2c(C)ccnn2)=O)C)C1 N1(C(C(CC(=O)OC)(C)C)=O)CC2(C1)CN(C(C1C=CCCC1)=O)CCO2 C1(C(=O)NCCCCNC(C2COC3(CCC3)C2)=O)SC2=CCC1CCCC2 c1(CNC(c2coc(C(C)NC(CCCSC)=O)n2)=O)cncc(C2CC2)c1 N1(C(c2cnn(CC)c2C)=O)CC(NC(C2CC3(CCC3OC)C2)=O)C2(CC2)C1 c1(C(N2CCC(C)(NC(C)=O)CC2)C(=O)NC)ccc(C#N)cn1 CCC(C(=O)N1CCC(CC)(NC(c2cc(C(N)=O)cn2C)=O)CC1)C(F)(F)F C(CCCCCNC(c1coc(-c2cccc(Cl)c2)n1)=O)NC(C(CSC)C)=O C1(CNC(c2c(CCC)n[nH]c2)=O)CN(C(C23CC2CNC3=O)=O)CC1OCC c1(C(=O)NCC=CCNC(c2cnc(CCC)s2)=O)ccc(NC(C)C)c(F)c1 c1(C(C(=O)OC(c2onc(CCC)n2)C)C)cccc(Br)c1 N1(C(c2[nH]c(=N)sc2)=O)CC2(C1)CN(C(=O)CCOCC1CCCO1)C2 C1(NC(CCc2onc(C(c3ccccc3)OCC)n2)=O)C(=O)OCC1(C)C Cn1nnc2cc(C(=O)NC3CCN(C(C4C5CCC45)=O)CC3)cnc12 CCC(CC)C(C)C(=O)NC1CCC(NC(=O)C(c2ccc(C#N)cc2)(C)C)C1 N1(C(C(CC)SC)=O)CC(NC(c2cc(Cl)c(Br)[nH]2)=O)C(C)C1 c1(C(N(C2CCN(C(C3CCCC3O)=O)C2)CC)=O)sc2cncn2c1C c1(CNC(CCCOCCC)=O)nc2c(s1)CCN(C(c1cncnc1)=O)C2 C1(C(N2CC(C(=O)N(CCCOC)C)(SC)C2)=O)CC1C1(C)COC1 c1(N(C2CC2)CC2N(C(=O)OC(C)(C)C)CCC2)cc2sccc2s1 c1(N2CCC(OC)CC2)nc2c(c(=NCC(C(C)C)N3CCCCC3)[nH]1)COC2 c1(C(=O)NC(CN(C(=O)CC2COCCO2)C)(C)C)n[nH]c(C2CC2)n1 N1(C(C=CCOCCOC)=O)CCCCC1CC(=O)NCCCCC1CCCC1 N1(C(N2CC(N3C(=O)COCC3=O)C2)=O)CCS(=O)(=O)CC1C1CC1 CC(CNC(=O)C=CCN(C(=O)C(C)n1cncn1)C)CO c1(C(=O)NC(C)(CNC(=O)C(F)C2CC2)CO)cc(F)ccc1F C1(C(N(CCC)CCC)=O)CCN(C(C2C=CCCC2)=O)C(C)(C)C1 CCCCCC(F)C(=O)NC1CC(CNC(=O)C(n2ccc(C)n2)C)CC1O N1(C(C(CSC)C)=O)CCCC(CCNC(=O)C(F)CC2CCOC2)CC1 c1(N2CCCN(C(c3ccccc3)C)CC2)ccc2cnc(C#N)cc2c1 C=CCC(C)(C(=O)N1CCCC(CCNC(c2nn(C)c(Cl)c2Cl)=O)C1)N(C)C C12(NC(CCC(=O)NCC)=O)CC(CNC(C3CCC3C)=O)(C1)OC2(C)C c1(CN(C(Cc2ccc(C)s2)=O)C)ccc(CNC(=O)C=C2CC2)cc1 c1(CC)ccc(C(C)C(=O)NC2C=CC(CNC(c3ccccc3)=O)C2)cc1 c1(OCC)ccnc2sc(C(=O)NC3CN(C(C4CCCC45CC5)=O)C3)cc12 c1(SC)nc2ncnc(N3CCCC(CN(C)C(c4nccnc4Cl)=O)C3)c2s1 Cc1cc(N)cnc1C(=O)NCC1CCN(C(C2CCOC2C)=O)CC1O c1(C(=O)NCC2CN(C(C=C=C(C)C)=O)C(C)C2)ccc(C)cc1F CC1CCC2(CC1)CCN(CC(=O)Nc1cccc(S(N)(=O)=O)c1)C2 N1(C(CCCCSC)=O)CCCC(NC(=O)Cc2ccc(F)cn2)C(F)C1 CCC1=NOC(C(=O)NC2CCC2NC(=O)CN2CC(=O)NC2=O)C1 CC1CC(CNC(c2ccc(C3CC3)s2)=O)CN1C(c1cc(O)nn1C)=O CC1(C)CC(CC(=O)NC2(CO)CCN(C(c3c[nH]ccc3=N)=O)CC2)CCO1 Cc1ncc([N+](=O)[O-])cc1C(N1CC(C)(NC(=O)C=C2CCOCC2)C1)=O c1(C(N(CCCCNC(CCCOC(C)C)=O)C)=O)ccc2c(c1)COC2 c1(NC(CCC2N(C(CCN(C)C)=O)CCC2)=O)c(Cl)cccc1Br c1(C(=O)NC(CC)CNC(c2csc(O)n2)=O)cc[n+]([O-])cc1 CC(C)CC(C)CC(=O)NC(C(=O)NCC(F)CO)c1cccs1 C1(NC(CCNC(N)=O)=O)CCCN(C(c2cc(Cl)ccc2N)=O)CC1 C#CCC(C)C(=O)N1CC(NC(=O)C(c2ccccc2OC)(C)C)C(O)C1 c1(C(N2CCC(CCCNC(C(COC)(C)OC)=O)CC2)=O)cn2ccsc2n1 N1(C(CCNS(CC)(=O)=O)=O)CC(C)(CNC(=O)Cc2nc[nH]n2)CC1(C)C c1(C(N(CCCC(N2CCC(CC)(CC)CC2)=O)C)=O)cncc2[nH]ccc12 C1(Nc2ncc(C(=O)OC)cc2Br)CCC2(CN(C(=O)CC(=O)OC)C2)O1 N1(C(Cc2nc(C)sc2)=O)CCC2(NC(c3ncccc3Cl)=O)CCCCC12 C1(NC(C2N(CCC)CCC2)=O)CN(C(=O)C2=CCCCO2)CCC1CO c1(C(C)=O)cccc(C(N2CCC(O)(CCNC(=O)CC(C)N(C)C)C2)=O)c1 c1(C(=O)NC2CC3CN(C(CCOCCN(C)C)=O)CC32)ccnc2[nH]nnc12 N1(C(C(F)=C(C)C)=O)CCOC2CN(C(=O)C(C3CCCCC3)N(C)C)CC12 CN1CCCC(C(C)(C)C(N2CCC(NC(C3CC(O)C3)=O)CC2)=O)C1 C(C(C)(O)CC(=O)N1CCN(CC(=O)NC2CCC(CO)CC2)CC1)OC C1(C(N2C(C)(CNC(C3C(C)C3)=O)CCC2)=O)Cc2cc(Cl)ccc2O1 N1(C(c2cc(OCC)c(OC)cc2)C(=O)NC(C)C)CCOC2(CCCSC2)C1 C(=O)(C1=NOC2(CCNCC2)C1)NC(C)CCO c1(C(N(CC(C)(C)CNC(=O)CC2=CCCC2)C)=O)cncc(P(C)(C)=O)c1 c1(OC)cc(C)c(Cl)cc1C(=O)NCC(C)(C1CC1)NC(=O)C(C)OC N1(C(CNC(C(CC)C)=O)=O)CC2CCCC(NC(c3ccc(OC)s3)=O)(C2)C1 N1(C(c2ccsc2Cl)=O)CC(CNC(=O)C(F)(F)C2(O)CCC2)C(O)C1 n1(CCOCCN(C(c2ccoc2Br)=O)CC(C)C)cc(C2CCCC2O)nn1 C#CC1(C(=O)NCC2CN(C(=O)C=C(Cl)Cl)CCC2C)CCOCC1 N1(C(C(CC)SC)=O)CCC(C2CCCN2C(c2ocnc2C)=O)CC1 c1(C(N2C(C)CC(CNC(C(C(CC)C)OC)=O)C2)=O)cc(F)cc2nn[nH]c12 CC1OCCC1CN(C)C(C1CC(CCNC(=O)Cc2ccn(C)n2)C1)=O c1(C(=O)NC(C(=O)N(CC(C)(C)C)CCC)Cn2cncn2)cnc(C)cn1 C(=O)(C(CC(C)C)C(C)C)NC1C(C(N2C3CC(=C)C(C3)C2)=O)COC1 CC(CC(=O)NC(C)(C)CC=CC(=O)N(C1CCCC(C)(C)C1)C)CC(C)(C)C c1(NC(C(CC2CCC2)NC(C(CCCC)F)=O)=O)cc(C)cn(C)c1=O N1(C(c2c(OC)cc(O)nc2)=O)CC2CC3CC2C1C3NC(=O)CS(C)(=O)=O Cc1cc(C(=O)NCC2CCC(NC(c3ocnc3C)=O)CC2)cc([N+](=O)[O-])c1 c1(C(N(C2C3CN(C(CC(C=C)C)=O)CC32)C)=O)cccc(=S)n1O C1(C(N2CCC(N(C(c3ccn(CCC)n3)=O)CCO)C2)=O)CC2(C1)CC(F)C2 C1(C(N(CCCCCC)CCNC(=O)CNC=O)=O)CCc2n[nH]cc2C1C Cc1cc(C(N2CC3=C(C2)CN(C(C2(CO)CCCO2)=O)C3)=O)cc(N)c1O N1(CCC)CCCCC1C(=O)NCC(C)NC(=O)C(=Cc1c[nH]cn1)F N1(C(C(CC)O)=O)CCN(c2ccc(C(=O)N(C)Cc3cccs3)cn2)CC1 N1(C(C2(OCC)CCC2)=O)CC(NC(=O)C=CC(C)C)C2(CCC2)C1 C1(C(=O)NC(CC=C)CC=C)COCCN(C(=O)C(F)C2CCCC2)C1 NS(=O)(=O)c1cc(C(=O)NC2CN(C(C3CCCO3)=O)CCC2CO)cs1 c1(CCC(N2CC(C)(NC(c3cncs3)=O)C2)=O)cccc(C#N)c1 N1(C(CCCC#C)=O)CCC(F)(F)C(NC(c2cc(F)cc(F)c2Cl)=O)C1 c1(C(N2CCC(N3CCCC3)CC2)C(=O)NCC2CC2)cc(F)cc(I)c1 Cc1ccccc1OCCCC(=O)NC(C)CNC(=O)CCC=CBr C1(C)(C(=O)NC(CNC(C2(C(C)=O)CC2)=O)C2CC2)CCCC1 Cc1snc2sc(C(N3CC4C(C3)N4C(C3CCCCC3)=O)=O)cc12 C1(NC(CCCCCOCC)=O)CCN(C(=O)Cc2csnn2)C12CCC2 C(CC(C)(C)C(=O)N1CCC(O)(CNC(=O)CCSC(F)(F)F)CC1)OC N1(C(C2(CC)CC2)=O)C2CCC1CC(C(=O)NCC(C)Sc1ccc(F)cc1)C2 c1(CNC(C2(OC)CCC2)=O)nc2c(s1)CN(C(=O)CC1CCC(=O)N1C)CC2 c1(NCCC(=O)NCC(CCCC)NC(C2CCCCC2)=O)c(C)cccc1Cl c1(C(C(=O)NCCSC2(C)CC2)N(C(C)COC)CC)ccc(C(Cl)Cl)cc1 C(=O)(C(F)C(C)(F)F)NCC(N1CCN(C(=O)CCc2ncc[nH]2)CC1)C C(CC(N)=O)(C(=O)NC(C)CCC1CC1)NC(C1C(C(C)C)CCO1)=O C1(NC(CC2CCN(C)CC2)=O)CCCCCC1C(N1CCC1CO)=O C1(NC(C(F)OC)=O)CCN(C(=O)CNC(=O)CC2CCCC2)C12CCC2 N1(C(c2cn(CCC)nc2)=O)CCC(CNC(C2CCC2C(F)(F)F)=O)C12CC2 c1(CC(CC)NC(=O)NCCCCOCC(=O)NC2CC2)cc(C)ccc1C C1(NC(C(C)(C)Cc2cnn[nH]2)=O)CCN(C(C2CCOC2)=O)CCC1CO C(=O)(C#CC1(C)CCCO1)N1CCC(NC(C2CCN(C(=O)NC)C2)=O)C(C)C1 C=CCC(C)(C)C(=O)N(CC(C)(C)CNC(=O)CC(=O)NCC(F)(F)F)C CC1CN(C(c2cccnc2)=O)CC1(C)CNC(=O)CSCc1ccccc1Cl C1(N=c2[nH]nc(C3CCCC3)s2)(CCNC(CCCCC#C)=O)CCC1 C#CC1(C(=O)NC(C)CC2CCOC2)CCN(C(c2ccc(C)cc2)=O)CC1 C1(OC)C2CC3CN(C(C4CCC5(CCCC5)O4)=O)C1C3C2 c1(C(=O)NCC(CN(C(C(C)SCC)=O)C)O)ncc(Br)cc1C N1(C(COCCC#C)=O)CCC(C2CCN(C(c3cnc(C)n3C)=O)C2)C1 c1(C(N2CC3C(NC(C4CC(C)(O)C4)=O)C3C2)=O)ncc(C(N)=O)cc1Cl N1CCC1C#CC(=O)OC(F)F.C(=O)(N=c1ccn(C2CCCC2)[nH]1)C(C)(C)C C1(CC(N2CCC(F)(CNC(=O)CCOCC(F)F)C2)=O)CN2CCN1CC2 C1(CNC(CC(=O)N(C)C)=O)CCC(CN(C(=O)CC2CCC(=O)NC2)C)CC1 c1(C(C)NC(C2CC(CNC(=O)CCN3CCCC3)C2)=O)ccc(F)cc1F N1(CC2CN(C(C(C)OCC(C)C)=O)C2)CCN(C(=O)Cc2cn[nH]c2)CC1 c1(C(N2CCOCC(NC(c3nn(CC)nc3C)=O)C2)=O)cccc2c1OCC2 c1(CC)n[nH]c(=NCc2ccc(CNC(=O)CCC(C)OC3CC3)c(F)c2)o1 C1(NC(CC2CCN(C)CC2)=O)CN(C(=O)CP(C)(C)=O)C2(CCCCCC2)C1 Cc1cc(-c2ccnc(Cc3ccccc3)c2)c[nH]c1=NCc1ccc(Cl)cc1C c1(Oc2ccc(C#CC)cc2)nnc(C2CCCc3ccccc32)s1 Cc1cc(CC(N2CC(CN(C(=O)C(c3cccc(F)c3)(C)C)C)C2)=O)n(C)n1 C1(C(N(CCCCN(C(C2ON=C(CC)C2)=O)C)C)=O)CC2(CCOCC2)CO1 C1(C(C(=O)OC)NC2(c3nnnn3C)CC3CC3C2)CC(F)(F)C1(C)C c1(C(=O)NC2CN(C(C(CSC)C)=O)CC2O)ccc(S(=O)(=O)N2CCCC2)o1 C(=O)(C(C#N)=CCl)NC1C(NC(CC(=O)OC)=O)CCC1 C(=O)(C(O)C(C)(O)CC)NCC(C(C)(C)C)n1cc(COCCCOC)nn1 c1(C(=O)NC2(CCNC(c3cc[nH]n3)=O)CC2)ccc2c(n1)NCC2 C1(CNC(C(CC)C)=O)CC12CCN(C(c1sc(Cl)cc1Cl)=O)CC2 C(=O)(N=c1nc2n([nH]1)CC(C(=O)OC)CC2)NC(CCCN(CCO)CC)C C1(C(=O)NCC2(F)CC(NC(=O)CCF)C2)CC12CCOc1ccc(Cl)cc12 N1(C(c2c(CC)nc(C)[nH]2)=O)CC(C)CN(C(=O)COC2CCCC2)C(C)C1 N1(C(CCC(C)OC)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)CCC1C C1(N(C(=O)C(=Cc2ccco2)C)CC)CCCN(C(c2n[nH]cc2Cl)=O)CC1 c1(C(C(=O)NCC2(CS(C)(=O)=O)CC2)(F)F)cccc(C(=O)ON)c1 Cc1cc(CNC(C2CSCCN2C(c2cc3ncsc3[nH]2)=O)=O)ccc1Br C(CC(C(=O)N1CCCC(CCNC(=O)C2=CCOC2)C1)OC)OC C(=O)(C1=NOC2(CCC2)C1)N1CC(N(C)C(c2ccn(C3CCC3)n2)=O)C(O)C1 CCCCC(CC)CCC(=O)NCC1(NC(=O)CC(C)F)CCCCC1 C1(NC(=O)CCF)CCN(C(C2(N3CCCCC3)CCCCC2)=O)CC1F N1(C(COCCOCC#C)=O)CCCC(NC(C2CCN(C)C2=O)=O)C1C CC(C)C1=NOC(C)(C(=O)NCCCCNC(=O)CCc2ccn(C)c2)C1 c1(-c2cn(CC(=O)NCCOCC(=O)O)nn2)cc(F)ccc1F C1(NC(=O)Cn2cncn2)CN(C(C23CCCC(CO2)C3)=O)CC12CC2 c1(C(N2C(CNC(c3cnn(CC)n3)=O)CC2)=O)cc(OC)ccn1 C#CCC(C(=O)NCCC(C)NC(C1CC(N(C)C)C1)=O)C1CC1 C1(C(N(CCCN(C(C(c2ccc(C)o2)C)=O)C)C)=O)NC(=O)OC1C S(=O)(=O)(CC(=O)NCC(C(C)(C)C)NC(=O)CC1CCCCN1C)NC C(C(=O)N1CCC(C(=O)NCC2(CC)CCCO2)O1)C1(CCC)CC1 N1(C(CC2CCC(OC)CC2)=O)CCC2(CNC(=O)C(C)(C)CO)CCCCC12 C12(C(N3CC4C(C)(C)C4C3)=O)COCC1CN(C(=O)Cc1ccn[nH]1)C2 n1(CC(N2CCC(C(CNC(C3C(C)C3)=O)F)CC2)=O)c(=O)oc2ccccc12 Cc1ccc(C(=O)NC2CCN(C(c3cnoc3)=O)C(C)C2)c(O)n1 c1(C(C)C)nnc2n1CCN(C(=O)C=Cc1nc3ccccc3o1)C2C CC(C(C)C(=O)N(C)CC1CCC(C)CC1)NC(=O)C=Cc1cncn1C c1(OC)ccccc1C(=O)N(C(=O)NC1CCCSC1)C1CC1.C1CO1 C(c1ccc(CC#N)cc1)=CC(=O)NCC1CC(NC(CC(=O)NCC#C)=O)C1 c1(C(N2CC3CCC(O)C3C2)C(=O)NCCCSC)cc(F)c(F)cc1F CC(CO)C(C)NC(=O)CCN(C(=O)CN(C)CCO)C c1(CNC(=O)CCOC(F)F)ncccc1C(=O)NC1CSC1 C1(NC(c2ccc(C)cc2)=O)CCN(C(c2nc(O)[nH]c(=O)n2)=O)CC1C N1(C(C(C)(C)CF)=O)CCCC2CN(C(c3cccn3C3CCCC3)=O)CCC12 c1(NC(c2nc(-c3c(OC4CC4)ccc(C)c3)sc2)=O)cccc(F)c1[N+](=O)[O-] C1(C(=O)NCC(C(=O)N(CCN2CC=CC2)CC)C)CCCC(=O)C1 Cc1ccn(CC(=O)NCCOCCC(=O)NC(c2nc[nH]n2)C2CC2)n1 N1(C(c2cnc(C)nc2)=O)CCC(C)(C)C(CNC(=O)CNC(=O)C(C)(C)C)C1 NS(=O)(=O)CCCC(=O)N1CCCCC(CNC(=O)Cc2ccc(Cl)nc2)C1 c1(C(=O)NCCC2CC(NC(c3c(C)cn(C)c3)=O)C2)cc2c(s1)COCC2 C1(c2nc(C(c3cccc([N+](=O)[O-])c3)OC)on2)CCC2CCCCC2C1 c1(C(N2CCCC(NC(=O)C(F)CC3CCCC3)CC2)=O)ccc2snnc2c1 CCC(C)(CCC(C)C)C(=O)NC1C2CC3CN(C(=O)CC(C)(C)SC)C1C3C2 CCCCC(C(=O)NCCCN1CCCC1C)NC(c1ccc(=N)[nH]n1)=O C(=O)(CCCC(F)(F)F)N1CC2C(NC(C3CCC34CCOCC4)=O)(C2)C1 c1(CNC(=O)Nc2c(C)n(CCC(C)C)nc2)cccc2c1OCCO2 CC1(C2CC2C(=O)NCC2CCOC2C(N2CC3CC3C3CC23)=O)COC1 Cc1cc(Cl)cc(C)c1C(N1CCOC(CNC(=O)Cn2c(C)csc2=O)C1)=O N1(C(C)C(=O)NCC2CCCO2)CCSC2(CCOCC2)C1 O=C(CCCN1CCOCC1)NC1CC1CNC(C1(C(F)F)CC(O)C1)=O C1(C(C)C)CCC(C(=O)N(C)CC2CCOCC2)N1C(C1CCN1C(C)(C)C)=O c1(CCC)c(C(=O)NC2CC2NC(=O)C(C)c2ccco2)cnn1CCO C1(NC(C(C)(C)CF)=O)CS(=O)(=O)CC1N=c1[nH]nc(C2CC2)o1 N1(C(C(CC)N2CCCC2=O)=O)CC2CCC2(CNC(=O)C(=O)C(C)(C)C)C1 c1(C(N2C(CCNC(C3(C)CN(C)C3)=O)CCC2)=O)cncc(C#N)c1 C1(C)(CNC(C2(SC)CC2)=O)CCC(NC(=O)CCc2cccs2)C1 N1(CC(N2C(C(C)(C)CNC(=O)CC3CCC(O)C3)CCC2)=O)CC2CCC1C2 N1(C(C(=O)OC)C)CCN(CCCNC(c2csc(Cl)c2Br)=O)CC1 Cc1ccc(C(=O)NC2CCC3CCN(C(=O)C(C)(C)F)C2C3)c2ccccc12 c1(N2CCC(C)(C(=O)NC)C2)nc2c(c(=NCC(C)(C)NC(C)=O)[nH]1)COCC2 C1(NC(c2n[nH]c(CC)c2Cl)=O)CCCCN(C(c2cc(N)ccc2F)=O)C1 S(=O)(=O)(c1ccc2[nH]c(=NCc3csnc3C)sc2c1)N1CC(CC)N(C)CC1 c1(CNC(C2CC(OC)C2)=O)c[nH]nc1C1CCN(C(c2c[nH]c(=N)s2)=O)C1 c1(NC(C2CCCCC23CC3)=O)cc(Br)ccc1OCC(F)(F)F C(=O)(C1CCCc2nncn21)N1CCCC(NC(c2cc(C)c(C)[nH]2)=O)C1 C1(N(C(CC(CCC)C)=O)C)CCC2CN(C(=O)CN(C)C(N)=O)CC12 N1(C(C(c2ccc(F)cc2)C)=O)CCC(CF)(NC(c2cc(Cl)ns2)=O)C1 N1(C(COCC=C)=O)CC2(C1)CN(C(c1sc3ccsc3c1C)=O)CCO2 C(C(=O)N(OC)C1CCS(=O)(=O)CC1)c1n(C(C)C)nc(C2CC2)c1Br N1(C(c2cnc(CC)[nH]2)=O)CC2CCCC(CNC(=O)CC3CC3)C2C1 c1(CNC(C2(CNC(COCC)=O)CC2)=O)ccc(O)c(OC)c1 C(=O)(C(O)CCCNC(C12CCC(CC1F)C2)=O)NCC(C1CCCC1)OC C(=O)(CCC(C)(C)N(C)C)NC(CNC(CCCC#C)=O)(C)C1CCC1 N1(C(C2CC(C)C2(C)C)=O)CC2CCC1CN2C(C1C=CCCC1)=O C#CCC(CC(=O)N1CCC(O)(CO)C1)NC(=O)Cc1sccc1C C(=O)(C(C)C(C)(C)C)N1CC(OC)C(NC(=O)CCn2cnccc2=O)C1 N1(C(C(=O)Nc2ccc(C)cc2Cl)C)CCS(=O)(=O)C(CNC(=O)CC2CC2)C1 c1(NC(C(C)OC(c2cccc(C3CCC3)c2)=O)=O)cc(C(F)(F)F)ccc1F C1(C)(C(N(CC)Cc2cccnc2)=O)CCCN(c2cc(OC)nc(C)n2)C1 c1(C(N2C(CNC(c3cnn4ncccc34)=O)CC2)=O)cc2c(nn1)OCCS2 c1(CC(=O)NCCN(C(=O)CC2CS(=O)(=O)C2)CCOC)cnc(Cl)cc1C Cc1cc(C(N2CCC(NC(=O)CCc3ccn(C)n3)CC2C)=O)cc(C)c1Cl C1(C)(NC(C(CCC)OC)=O)CCCN(C(c2cccc(C3CC3(F)F)c2)=O)C1 CCC(CC)CC(=O)NC(c1ccccc1F)CNC(=O)C(COC)CC CC(C)(C#N)C(=O)NCc1ccccc1CNC(c1ncccc1N(C)C)=O c1(NC(CCc2ccc(NC(=O)OC(C)(C)C)[nH]2)=O)cccc(C(F)F)c1 C1(CNC(C=C(C)C(F)F)=O)CC12CCN(C(=O)CN(C)CCO)CC2 c1(C(N2CCC(CNC(C(n3ncc(C)c3)C)=O)C2)=O)nccc(Cl)c1C N1(C(CC(C=C)CC)=O)CCCCC12CC(NC(=O)COC1CCC1)C2 C1(C(N(C)Cc2c(C)nsc2)=O)CC(NC(c2cncs2)=O)CCO1 C(CC(=O)NCC1CCCSC1)(C(C)(C)C)NC(c1c(C)nc(C)o1)=O Cc1ccc(C=CC(=O)NC2CCC(CCNC(c3ccc(C)nc3)=O)C2)nc1 N1(C(CN(C2CC2)CC)=O)CCCC(C(=O)NC2CCN(C(=O)NC(C)C)C2)C1 C1(O)(CN)CN(C(C2CC(C(F)F)C2)=O)C1 c1(CC)nccnc1C(=O)NCC1CC(O)CN1C(C1CC1c1cccs1)=O C1(C(N(C2CCN(C(=O)CC3CCCOC3)C2)CCO)=O)COC2CC1C2 Brc1csc(CN2CC(n3cncn3)C2)c1 CCCC(C(=O)N(CCCNC(C1CC2(C1)CC1(CC1)C2)=O)CC)C(C)C C(=O)(CCC(C)NC(=O)C=Cc1ccnn1C)N(C(CCCC)C)C C1(NC(C=Cc2n(C)cnc2)=O)CCCC12CN(C(C1NC(=O)OC1C)=O)C2 c1(OC)cc(C(=O)NCCC(C)NC(=O)C=C(C)c2cnn(C)c2)cc(Cl)c1 C#Cc1ccc(CC(=O)NCC(C)NC(=O)C(c2ccc(F)cc2)(F)F)c(F)c1 c1(C(=O)NCCC2(C(=O)NC(C3CCOC3)C#C)CC2)cc(CCO)on1 C1(C(N2CC(NC(C3(C4CCOCC4)CC3)=O)C3C2C3)=O)CN2CCCN1CC2 C1(C(=O)NC(C)(C)CCNC(c2ccccc2CC#N)=O)CCc2ccnn2C1 C1(C(C)C)CN(C(c2ccc(O)nn2)=O)CCN1C(=O)Cc1nc[nH]n1 O=C1CS(=O)(=O)CC(C(=O)NC2(CO)CCN(C(=O)CC3CC3)C2)N1 CS(=O)(=O)CCc1cn(CC2CCN2C(=O)Cc2nccn2C(F)F)nn1 c1(SC(C)(C)C)ccccc1C(=O)NC1CCC(Cn2cc(C(C)OC)nn2)C1 Cc1nscc1C(=O)NC(CC1CC1)C(=O)NCc1nc(CO)n[nH]1 Cc1cc(O)c(F)cc1NC(C1(CNC(=O)C(C)CO)CCOCC1)=O c1(C(=O)NC(C(C)NC(C(C)Cc2cnc[nH]2)=O)(C)C)cc(Cl)c(F)cc1O c1(NCC2(CO)CC(C)C2)cc(Br)ccc1S(=O)(=O)N1CCC2CC12 C(C(C)C(C)C(=O)NC1(CNC(=O)CSC)CCOCC1)OC C12(C(=O)NCCN(C(=O)COCc3nccn3C)CCC)CSCC1C2(F)F c1(CC(CNC(=O)C(C2CCCC2)SC)NC(C(F)OC)=O)ccccc1 c1(C(N2CCC(c3cn(Cc4cnn[nH]4)nn3)CC2)=O)ncccc1Br C1(CC)CCC(C)CN1C(=O)C(CC(F)F)N(C)C(c1cc(C#N)[nH]c1C)=O N1(C(=O)Nc2c(SCC)nccc2)CC2(NC(=O)C(F)(F)F)CCC1CC2 c1(NC(C2N(C(C(C)C)=O)CCCC2)C)nccc(S(C)(=O)=O)n1 N1(C(C(=O)N(CC(C)OC(C)(C)C)C)=O)CC2CCCC12 Cc1nc(Cl)sc1C(=O)N(Cc1ccc(Cl)cc1)Cc1ccsc1 c1(CC(=O)NC2(CN(C)C(C3CCCCC3(C)C)=O)CC2)cc(O)nc(O)n1 N1(C(c2cc(C)c(O)nc2)=O)CCCC2(NC(c3cc(Br)co3)=O)CC2C1 N1(C(C(C(C)C)OC)=O)CC(C(=O)NC2CSC2)C(C)(C)C1 Cc1ccc(F)c(CNC(c2cncc(CNC3(C)CC3)c2)=O)c1 N1(C(C=CC(=O)OCC)=O)CCC(C2CC2)C1CNC(C1CC2C=CC1CC2)=O c1(C(C)C)ncc(C(N2CCC(NC(c3ccn(C4CCC4)n3)=O)CC2)=O)cn1 N1(C(c2cc(C)n(CC#C)c2C)=O)C2CCC1CC(N(C(=O)CC(=O)NC)C)C2 C(=O)(C(C)CC(C)(C)C)N1C(C(=O)NCC(CC(=O)NC)C)(COC)C=CC1 C12(C(N(CCCC=C)CC)=O)COCC1CN(C(c1ccc(C(N)=O)cc1)=O)C2 C1(OC)C(CN=c2[nH]nc(-c3ccccn3)o2)CCCN1C(C)=O CC1CCC(C(N2CCCCCCC2)=O)CN1C(C1CCN1C(C)(C)C)=O N1(C(CCC#C)=O)CCCC12CN(S(=O)(=O)CCC(=O)OCC)C2 C=CCC(C(=O)NCCN1CCN(C(C2CCCCC2O)=O)CC1)OC C1(CN(C(c2cnc(CC)s2)=O)C)C2CN(C(c3ccn(CCO)c3C)=O)CC12 CC(C)C(C)C(=O)N1CC(C)C1C(=O)NCCc1cocn1 N1(C(C(C)n2ccnn2)=O)CCC2(CC1)CC2CNC(c1cocc1C(N)=O)=O CCCC(CC)CCC(=O)NC1CC(NC(=O)CC(C)C2CC2)C1 C1(CC(=O)NCC2(Nc3nc(C)nc(O)c3)CC2)COc2ccccc2O1 Cc1cc(CN2CC(O)CC2C(N2CC3CCC2C3)=O)c(C)cc1Br C12(CNC(C3C(C)(C)C3)=O)CC(CCO1)N(C(C1CC3C=CC1O3)=O)C2 C1(O)(CN(C(C(CC#C)O)=O)C)CCN(C(=O)C(CC)N(CC)CC)CC1 C12(C(N3CC(C)(NC(c4n(C(CC)C)ncc4)=O)C3)=O)CCC(CC1=O)C2 C1(CN(C)C(=O)OC(C)(C)C)CC(C(=O)OCc2nnc(O)o2)=NO1 C1(CNC(c2c(C(C)C)cco2)=O)CCCCN(C(=O)CC2CCCC2(C)C)C1 c1(C(=O)NC2C=CCC(C(=O)NC(CCCC=C)C)C2)c(C#N)ncn1C C(=O)(C(C(C)(C)C)N1CCCC1=O)N1CCC(n2cc(CCN(C)C)nn2)C1 c1(Cn2cc(CN3CC(N(C)C)CC34CCC4)nn2)c(F)cc(Br)cc1F C1(CS(=O)(=O)N(C(C)C)Cc2cccc(C)c2)CC12CCCc1ccccc12 C1(O)(CNC(C2CC(=C3CC3)C2)=O)CCCN(C(c2cnsn2)=O)C1 C1(C(=O)NCCCOCCN(C(c2c(C)c[nH]n2)=O)C)OC2CCC1CC2 c1(C(C(=O)NC(CC)C)N(C2CC2C)C)cnc(C(C)C)s1 c1(OC)ncc(C(=O)N(C2CC3CC2N(C(C2(C)CS(=O)(=O)C2)=O)C3)C)c(C)n1 c1(NC(C2(C(=O)OC)CCNC2)=O)ncnc2cc(C(C)(C)C)sc12 c1(NC(C2(NC(C3CN(C(C)C)C3)=O)CC2(C)C)=O)ccccc1N=[N+]=[N-] Cn1nc(C(=O)NCC2CC3(CC3)CN2C(=O)CC2(C)CC2(Cl)Cl)c2c1CCC2 C(=O)(C(C)(C)CNC(C1CCC(NC(C2CCC(O)CC2)=O)C1)=O)NC C1(C(=O)NCC(C2CCC2)OC)CCCC(NC(c2nnsc2N)=O)C1 c1(COC)ccc(C(=O)NCC2(F)CN(C(c3ncoc3C3CC3)=O)C2)s1 C1(NC(C2(CC)CCNC2=O)=O)CCC2CC1CN2C(=O)Cn1cncn1 C1(NCC)CCCC(CNC(=O)CCC2CN(C(=O)OC(C)(C)C)C2)O1 c1(C(=O)NCC2CCN(Cc3cc(Br)cs3)C2)cnn2cccc(F)c12 C12(NC(c3c(C)n[nH]c3)=O)CCCN(C(c3c(Cl)csc3Cl)=O)CC1C2 c1(SC)cc(C(N2CCCC2CCC(=O)NCC(C)(C)C2CCCO2)=O)co1 N1(C(c2c(C)nc(CCC)s2)=O)CCC(C)C(NC(=O)CC2(O)CCOC2)C1C C(=O)(C1=CS(=O)CCC1)NC(C(C)C)CNC(=O)CCCc1cccnc1 C1(N(C(=O)CC(C2CC2)C2CC2)C)CN(C(=O)CC2CC(F)(F)C2)CC1F N=c1[nH]c(-c2c[nH]c(C(=O)NCC#CCNC(=O)CCn3cccn3)c2)cs1 C(C(C)(C)C(=O)N1CC(C(=O)NC2C3CCCC23)C(C)C1)OC(C)C CC(CCCCNC(=O)CC1CC1(Cl)Cl)NC(C1CC(F)(CO)C1)=O c1(C(=O)NC2C(NC(CCc3nnc(CC)o3)=O)CCCC2)n[nH]cc1[N+](=O)[O-] c1(-c2c(CNC(N3CC(CC)OCCC3)=O)ccc(F)c2)ccc(C)cc1NC CCCC(C)(CCC)C(=O)NCc1ccnc(C(N2CCC2(C)CCO)=O)c1 CC1(C)CCC(C(=O)NC2CC(CNC(c3cnn(CC(F)(F)F)c3)=O)C2)C1 CCCC(C(=O)NCCCNC(=O)Cc1cccc(OCC2CC2)c1)N(C)C c1(-c2ccc(C(N3CCC(C(=O)NCC)CC3)=O)nc2)nc2ccccc2s1 C1(NC(C(C)CN(C)C)=O)CCN(CCNC(C2C3CCC2CC3)=O)CC1 c1(CCC(=O)NC2CCC(CCN(C(C(C)(C)C)=O)C3CC3)C2)ccnc(Cl)c1 C1(OC)CC(NC(=O)CCc2ccccc2)CN(C(C2CC23CCC3)=O)C1 Cc1cccn2nc(C(=O)NC3CCN(C(C4CCCC4)=O)C(C4CC4)C3)cc12 N1(C(c2cccc(C=CC(F)(F)F)c2)=O)CCC2CCC(F)(F)CC2C1 N1(C(=O)Nc2c(OCC#C)cccc2)CCc2[nH]c3ccc(F)cc3c2C1 c1(C(=O)Nc2cncc(C)n2)cnc2ccc(-c3ccc(F)c(C#N)c3F)cn12 c1(-c2nc(C(C)C3CC3)nn2C2CCC2)ccc(S(=O)(=O)C(F)(F)F)cc1 N1(C(C2(c3c(C)c[nH]n3)CC2)=O)CCC(NC(=O)C(C)NC(=O)C2CC2)C1(C)C C1(OC)CN2CCCC2(C(=O)NCCC2(COC)CC2)C1.c12ncnc(Cl)c1N2 N1(C(C2CCC(NC(CC)=O)C2)=O)CC2(CCCCN(C(=O)C3=CCCC3)C2)C1 N1(C(CCSCCC)=O)C(CNC(=O)CCc2csnn2)CC2CC12 CC(CCC(C)(C)C)C(=O)NC(C)C(c1nc2ccccc2s1)C CC(C)C(O)CC(=O)N1CC(C)(C)CC1CC(=O)NCc1nn(C)c(=O)n1C c1(N2C(C)CN(C(=O)CC(=O)NCC(F)(F)F)CC2)nc2ccc(F)cc2o1 CCCC(C(O)C(=O)N(CCCO)CC)NC(=O)C(O)CCN(C)C C1(CNC(C#C)=O)C(C)CCCN1C(=O)CC1CC1 C1(C)(NC(C(CC)C)=O)CCN(C(C2(c3cc[nH]n3)CCC2)=O)C1 c1(C(N2C(CNC(CSCC)=O)C(C)(C)CCC2)=O)cnc2n1CCCC2C C1(C(=O)NC(C(=O)NC2(CN(C)C)CC2)C2CC2)CCCC2(CC2)C1 c12cc(N(C)C)cc(c1)NC(=O)N2.Cc1n[nH]cc1CCOC(C)(C)C C1(C)(OC)CC(NC(=O)C(CCOC)NC(c2cc(C)nc(O)c2)=O)C1(C)C C(=O)(C1=CCN(C(C2CC(OC(C)=O)C2)=O)C1)N(CCC(=O)NC)C C1(CC(N2C(CC)CC(O)C2)=O)CCN(C(=O)CCC2CCCOC2)C1(C)C C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCCNC(c1cncc(C=C)c1)=O)C C=C(CNC(c1ccccc1)=O)CCNC(=O)CCNC(=O)CC12COC(C1)C2 c1(NC(C2(OC)CCSC2)=O)cc(NC(c2ccc[n+]([O-])c2)=O)ccc1C C1(CC(=O)NC(C)CN(C)C(C2CCN(C3CCCCC3)C2)=O)C(C)(C)C1(C)C CC1CC(C)CCN(C(C2C=CCN(C(c3ccnnc3O)=O)C2)=O)C1 c1(C(=O)Nc2c(C(=O)OC)c(C)cs2)ccc(-c2ccc(F)cc2)nc1C c1(CC)c[nH]cc1C(=O)NCC1OCCC1C(=O)NCc1ccsc1C C1(CNC(C(C2CC2)OC)=O)N(C(=O)CC(C)NC(N)=O)CCCC1(C)C CC(C(=O)N1CC2CC(NC(C3CCCCCC3)=O)C1C2)C(C)(F)F CCCCC(C(=O)NC)NC(C12CC(CN1C(=O)CC1CC(C)(C)CO1)C2)=O C1(O)(CNC(C(CC)SC)=O)CCCN(C(c2cc(OC)ccn2)=O)CC1 c1(OC(C(=O)NCC(CNC(C(C)CC2CCC2)=O)(C)C)C)ccccc1F n1(CC)ccc(=NC(=O)CCC2CCN(C(=O)Nc3ccc(F)c(F)c3)CC2)[nH]1 Cc1cccc(CCN(C2CCOC(c3ccncc3)C2)C)c1 N1(C(CCOCCNC(C(C)(C)OC)=O)=O)CC(=O)NC(C(C)C)C1 C=CCCC(F)(F)C(=O)N1CC2(CCCC2NC(c2cn(C(F)F)c(C)n2)=O)C1 N1(C(C2CC(C)OCC2)=O)CC2CC(C1)C2NC(c1ncccc1C(F)F)=O S(=O)(=O)(c1ccccc1Cl)NC1C(NC(Cc2ccc(C)nc2)=O)C2CCC1C2 c1(C(=O)NCC2CCC(NC(c3c(SC)snn3)=O)C2)nn(C)cc1[N+](=O)[O-] C(=O)(C1CCCc2c[nH]nc21)N(C1CCN(C(=O)CSCCOC)CC1)CCC CC1=C(C(=O)N2CCCC2C2(NC(c3cc(Cl)cn3C)=O)CC2)S(=O)(=O)CCO1 C=CC12CN(C1)C(=O)C2.C1CCC(=O)N1C.C1(C(N)=O)CC12CCC2 CC1CCC(NC(C23CC(C2)C3)=O)CN1C(C1CCC(C(N)=O)C1)=O c1(C(=O)NCC2CCCCN(C(C3(OC)CC(C)C3)=O)C2)nc(O)nc(O)c1F c1(OC)ccccc1CNC(C1(CC)CCCN1C(=O)C(O)C1CC1)=O O=C1CC(C(=O)NC(C2CC2)C2CC2)N(C(C2CC=CC2)=O)C1 C1(Cn2cc(-c3c(C)ccs3)nn2)CCCN(C(c2ccccc2Cl)=O)C1 N1(C(C(C)OCC=C)=O)C2CC1CN(Cc1ccc(CC)cc1)C2 C1(CNC(C=CC=CC)=O)CC2CCC(C1)N2C(C1CCC1c1nncn1C)=O c1(C(N2CC(C)(CNC(CSCC)=O)OCC2)=O)cc2nccnc2cc1F C#CCCCCCC(=O)NC1CCC(C)(CNC(=O)CCc2cc(OC)no2)C1 C1(CNC(C(CC#C)C)=O)CC2CCC1N2C(c1cc(C)cc(F)c1)=O N1(c2ncc(C)c(C)n2)CCC2(NC(=O)Cc3ccc(F)cc3Cl)CCCC12 C=C=CCCC(=O)NC(C)CN(C(=O)CCC(C)c1ccc(Br)cc1)C c1(OCC2(n3cccn3)CN(C(=O)OCC3CC3)C2)cc(Cl)c(C)cc1[N+](=O)[O-] CC(C)(C)[Si](C)(C)OC1(CC(COC)NC(=O)Cc2c(O)ncnc2O)CCC1 C(=O)(C1=C(C#N)CCC1)NCCn1cc(C(N2C3CN(C)C(C3)C2)=O)nc1 C1(NC(c2ccc(F)s2)=O)CN(C(c2cc3c(o2)CCCC3)=O)CC2CCCC12 Cc1cc(F)ccc1C(N1CC(C)(C)CC1CC(=O)NC(c1ccnn1C)C)=O C(C)(c1cccs1)=CC(=O)N(C(=O)C(CNC(C)=O)N(C(C)(C)C)C)CCCC Cc1cc(O)ncc1C(N1C2CCC(C2)C1C(=O)NCC1(C)CCCO1)=O N1(C(CCCC#CC)=O)CCC2(C1)CN(C(C13CC(C1)C(C)O3)=O)CC(C)O2 Cc1n[nH]c(C)c1CC(N1CCCC(C(C)C(=O)N(C)CCO)C1)=O Cc1cc(=NC(COC(C)(C)C)C(C)C)[nH]c(N2CCC(N(C)C)C2)n1 Cc1cnnc(O)c1C(=O)NCCC1CC(F)(F)CN1C(c1ccnnc1O)=O CCC(CC(=O)N1CCC=C(C(=O)NCc2ncoc2C(C)C)C1)C(F)F N1(C(c2c(OC)cccc2)=O)CCN(C(=O)Cc2cccn2C)C(CC2CC2)C1 c1(C(=O)NCC2CCCN2C(C2CC23CCCC3)=O)n[nH]c2cc(Cl)ccc12 CC(C)CCCC(C)C(=O)N1CCC(O)(CN(C(=O)CC(=O)N(C)C)C)C1 Cc1nc(O)nc(C)c1CC(N1CCCN(C(C2OC3CCC2CC3)=O)CC1)=O c12ccc3cnnc(c3c1)n2C.c1(C(=O)OC)cc2ccccc2n1C Brc1ccc(-c2ccc(CN(CCCSC3CCCO3)C3CC3)s2)cc1 c1(C(N)=O)cncc(C(=O)NCCN(C2CCCC2)CC=CC2CCCC2)c1 CC(C)C1=CCC(C(N2CC(C)N(C(C3CC34CC4)=O)CC2C)=O)CC1 Cc1cc(C(N2CC(C)CCC2C(=O)NCCC(F)=C(F)F)=O)ccc1C#N N1(C(c2c(CC)nc(C)[nH]2)=O)CCCC(C)(NC(c2nn(C)cc2Cl)=O)C1 C=CCC(C(=O)NCCC1CCCN1C(=O)C(=O)Nc1ncc[nH]1)N(C)C C=CCCCCCC(=O)NC1CN(C(=O)Cc2cncnc2O)CC1C c1(C(=O)NCC23CC(CNC(C(CC)O)=O)(OC2)C3)cccc(F)c1F N1(CCNC(CCSCC)=O)CCN(C(C2(C)CCC(=O)N2)=O)CC1 C1(CNC(C(c2cccs2)NC(c2cn(CCOC)nc2)=O)=O)CN(C)CCO1 c1(C(N2CC(C(C)NC(c3c(C)c[nH]n3)=O)C2)=O)cc2c(Br)cccc2[nH]1 CC(C)(CC(=O)NCC1CCCC(NC(c2cc(=O)cc[nH]2)=O)C1)CC(F)F c1(CCNC(C(N2C(C)COCC2)=O)=O)cc(C#N)ccc1I C1(C(=O)NC2(CSC)CC2)CC(O)CCN1C(c1cnnc(C)c1)=O CC1CCN(C(=O)CCS(C)(=O)=O)CCN1C(=O)C(C)CC1CCCCC1 C1(N(C(CN(CCOC)C)=O)C)CCCN(C(c2ccnn2C2CC2(F)F)=O)C1 C1(C(C(=O)NC(C)(C)C)N(C(c2nc(C)[nH]n2)C)C)CC=CCC1C CC(C)C(N=c1[nH]c(Cl)ncc1Cl)C(C)NC(=O)OC(C)(C)C c1(C(C)=O)cc(C(=O)NC(COC)C(=O)NC2(c3n[nH]c(C)n3)CC2)no1 c1(CCC)ccc(Nc2cccc(OCC(=O)OC)c2)cc1S(N)(=O)=O C1(C)(C(N2C(CNC(C(CC)(F)F)=O)CCCC2)=O)CCCNC1=O C1(C(=O)NCCCC2N(C(c3c(CC)nns3)=O)CCC2)CCC(O)CC1 Cc1cc(C2CC2)ncc1C(=O)NC1CCN(C(c2cc(CF)on2)=O)CC1F C123CCC(CC1)(OC2)CNC(=O)CCc1c(ccc(F)c1)C(=O)N3.C1(CO)CC1 N1(C(Cc2cc(C)ncc2)=O)CCOC2(CCN(C(C3CC4C=CC3C4)=O)C2)C1 c1(NCC(CC(C)C)NC(=O)C2=NOC(C)(C)C2)nc(O)n(C)c(=O)c1[N+](=O)[O-] N1(C(NNC(C23C(C(=O)OC)CC(CC2)C3)=O)=O)CCCC(C2CCCCC2)C1 c1(C(N(C(C)CN(C(=O)C(O)C2CCC2)C)C)=O)cccc(-c2ccco2)c1 c1(N(C)C)cnccc1C(N1CC(F)(CNC(=O)C=Cc2cccs2)C1)=O c1(C(N2CCC(N(C(=O)CCCc3cccc(Br)c3)CCO)C2)=O)ccc(O)nc1 Cc1ncnc(C)c1C(=O)NCC1(NC(=O)CCC2CCCOC2)CCCC1 CC(C)(COCCCl)CC(=O)C(N)=O.C(=O)(C(F)(F)F)NCCO.C1CN1CCN C1(NC(C(C)=CC)=O)CC2(C1)CC(CNC(=O)C(c1cccn1C)=O)C2 C1(C(=O)NCC2C(NC(Cc3c(C)cccc3C)=O)C2)CCn2nccc2C1 C(=O)(C(C)CC(C)C)NCC(C)(CNC(=O)C(c1c(C)n[nH]c1C)C)OC c1(NC(C(C)O)COC(C)(C)C)ccnc2c1CCO2 C1(NC(Cc2ccc(CC)cc2)=O)CC2CC1N(C(=O)C(C)(C)CNC(N)=O)C2 C1(CNC(COCC)=O)(N(C(C2C(C(C)=O)C2(C)C)=O)C2CC2)CCCC1 N1(C(CC2(COC)CC2)=O)CC2COCCC2(NC(c2csc([N+](=O)[O-])c2)=O)C1 C1(OC)CC(CNC(=O)CCCOc2ccccc2F)N(C(c2ccc[nH]2)=O)C1 NS(=O)(=O)c1n[nH]cc1C(N1CC2CC1CN2C(C12CC(CF)(CO1)C2)=O)=O N1(C(C2CC(C)(O)C2)=O)CCC(N2CCN(C(C3CCC4CC4C3)=O)CC2)CC1 C1(C(=O)Nc2cccc(C(C)C)c2)CNC(=O)CN1C(=O)CCc1ccsc1 Cc1c(NCCF)nc[nH]c1=NCC(CC)(c1ccc(F)cc1)c1ccccc1 c1(OC)ccnc(N(C)CCN(C)C(C2CCN(Cc3ccccc3)CC2)=O)n1 N1(C(CC(C(F)F)NC(c2c(CC)nn[nH]2)=O)=O)CCC12CCC(C)CC2 N1(C(C(CNC(C=CC=CC)=O)C(C)C)=O)CCc2c(F)cccc21 N1(C(c2c(CC)nns2)=O)CCN(C(c2ccc(OC(C)C)nc2)=O)C(C)C1 Cc1[nH]nc(C(=O)NC2CCCC2CNC(c2sccc2Br)=O)c1C c1(C(N2CCC(CNC(C3CC4CC4C3)=O)C2)=O)c(Cl)cncc1Br c1(C(=O)NCC2(F)CC(NC(C=CC(C)(C)SC)=O)C2)cc(Cl)ncc1NC N1(C(C(C)(C)C#N)=O)CCC(C2CN(C(=O)CC3OCCOC3(C)C)C2)CC1 Cc1nc(C(C)C)nc(O)c1C(N1CCN(C(C2C3CCCC23)=O)CC1)=O c1(C(=O)NCCCC(C)NC(c2cc(OC)c(C)cc2)=O)cc(Cl)cc(Cl)c1O C1(NC(c2c(C)coc2)=O)CCCCC1CC(N1CCC(CC2CC2)C1)=O C=CCCC(C(=O)NC1CCOC(C)(C)C1)NC(=O)CCC(C)(C)C c1(C(N(CCCN(C(C2C(CCOC)C2)=O)C)C)=O)ccn(-c2cccnc2)n1 C1(NC(C(CCNC(C2C(C)CC2)=O)(C)C)=O)CCC(C2CC2)CC1 c1(OCC)cc(F)c(-c2cn(C3(C(N4CC5CC(C4)C5O)=O)CC3)nn2)cc1F CC1OC(C)C(C)C1C(=O)NCC(C)CNC(C1CC(O)(C(F)(F)F)C1)=O c1(C(C)C(=O)NC2(C)CCN(C(=O)Cc3ccoc3)C2)ccc(C#N)cc1 C(=O)(CCC(=O)c1ccc(Br)cc1)NC1CC(NC(C(COC)C)=O)C1 C(CC(C(=O)NCC12CC1CN(C(=O)COCC1CCC1)C2)NC=O)SC C=CCC1C(=O)N1CC.C(C)(C(=O)NOCC1CC1)NC(C)=O C1(NC(c2cccc(C3(OC)COC3)c2)=O)CCN(C(=O)C(C)NC(N)=O)C12CC2 C(=O)(CC(C(F)F)CC(CC)NC(=O)NC(C(F)F)C1CCCC1)OC Cc1ncncc1C(=O)NC(C)C=CC(=O)NCc1ncoc1C C(=O)(CS(=O)(=O)CC)N1CC(C(=O)N(C)Cc2ccccn2)(SC)C1 N1(c2nnc(C(=O)OC)s2)CC2CC(NC(c3cc(CC(C)C)on3)=O)C2C1 C1(F)(CNC(C2(C(=O)NC)CCC2)=O)CC(CNC(=O)C(C)COC)C1 Cc1ccnc2c(C(=O)NC(C)CNC(=O)CCCCCC(C)(C)C)cccc12 Cc1cc(F)cc(C(=O)NC2CCC2NC(c2c[nH]nc2[N+](=O)[O-])=O)c1N Cc1cc(C(=O)N(CCCNC(C2CC2Cl)=O)C(C)C)c(C)n1NC(N)=O CC(CN=C(NCC1CCCO1)NCC1CC2CCC1CC2)OC(F)F c1(C(N2CC(COC)N(C(=O)CCSC)CC2)=O)ccc2ncn(C)c(=O)c2c1 c1(C(N(CCN(C)C(c2cc(Br)cnc2N)=O)C)=O)cc([N+](=O)[O-])nn1C c1(NC(C2C(CC)CN(C(=O)CC(C)NC=O)C2)=O)cc(CO)cc(F)c1 c1(C(CC)NC(C2C=CC(NC(=O)C(C)=O)C2)=O)cc(OC)ccc1O C1(C)(C(=O)NCC(C)(C(C)C)NC(CC=C=C)=O)CCCS1(=O)=O C(C(CCC)C(=O)NCC(C)(C)F)NC(COC1(C#C)COC1)=O C1(NC(C(C)OC(N)=O)=O)CCCC1Cn1cc(C(C)(C)N(C)C)nn1.C1CO1 c1(C(N2CC(NC(CC3(COC)CC3)=O)C3C2C3)=O)cc(Cl)cc2c1OCC2 C1(C(=O)NC(C2CN(C(CCCNC(=O)OC)=O)C2)C)CCCCC1F C(=O)(C1CCCc2nn(C)cc21)N(C)CCNC(=O)Cc1cnn(C)c1 N1(C(c2ccc(C(C)C)cc2)C(=O)NCCSC)CCC(C)C(CO)C1 CCCCC(=O)C(=O)NCC(C(C)(C)C)NC(c1scnc1COC)=O CC1(c2ccccc2)CCN(C(=O)C(N2CCOC(c3ccc(Cl)s3)C2)=O)C1 CCCC(C(=O)N1CCC(C)(CNC(c2ccc(C(F)F)nc2)=O)C1)NC(N)=O C=C(C)CCC(=O)NCC1(C)CCN(C(=O)C(N2CCNC2=O)C)C1 C(CN=c1cccn[nH]1)NC(C1N(S(C)(=O)=O)CCCC1)=O N1(C(c2[nH]cc(C)c2)=O)CCN(C(C2CC(C#N)C2)=O)C2CCCC2(C)C1 c1(NCC(C)CN(C)C)[nH]c(=NC2C3CC(Cl)CC23)nc2sccc12 c1(CN2C(C(=O)NCCNCCO)CCC2)c(C(F)(F)F)cccc1O N1(C(C=CC)=O)CCN(C(c2ccccc2Br)=O)CC1c1cn[nH]c1 N1(C(C(CC)NC(N)=O)=O)CCC2(CC(C(N3CC(N4CCC4)C3)=O)C2)C1 c1(SCC(=O)NC2CC(NC(=O)C=CC3CCOC3)C2)ccc(C(F)(F)F)cn1 C(=O)(CCCC(F)(F)F)N1C(CNC(CC(C)NC(N)=O)=O)CCC1 c1(C(=O)NCCC2CC(NC(c3cc(OC)n[nH]3)=O)C2)nn(C)cc1Cl CC1=NN(C)C(=O)C1CC(N1CC=CC1CNC(C1(CC2CC2)CC1)=O)=O C=CC(C(=O)N1CSCC1C(=O)NCC=C=C)OC C(CCCCCNC(C1CCCC(=O)O1)=O)N(C(CC1N(C(C)C)CCC1)=O)C c1(OC)cc(C(N2CCC(CNC(c3ccccc3F)=O)C(C)C2)=O)ccc1F CC1CN(C(=O)C=CC(F)(F)F)CCN1C(c1cccn(CC(F)(F)F)c1=O)=O C1(NC(C(CN(C)C)NC(CNC(CCC)=O)=O)=O)CCC(C(C)O)CC1 N1(N(CCC)C)CC=C(CCNC(c2cc3oc(C(=O)O)cc3[nH]2)=O)CC1 N1(C(c2c(C(C)=O)ccs2)=O)CCC(CNC(=O)COCC(C)C)C12CC2 c1(N(C2CC3CC2CN3)C(C(CC)NC)=O)ncc(OC(F)(F)F)cc1Br C1(CNC(C2C(OC)CCC2)=O)CN(C(c2ccncc2F)=O)CCN1C Cc1ccc(Cl)cc1C(=O)NCC1C(C)CCN1C(C1(C(N)=O)CCC1)=O Cc1cccc2oc(C(=O)NCC3CCCN3C(=O)C#CC(=O)N(C)C)cc12 Cc1cnc(C)c(C(=O)NC(C)CC2CN(C(=O)C=Cc3cn(C)cn3)C2)c1 C1(NC(C(C=C)(C)C)=O)CC2CCC(C1C)N2C(=O)CCc1nnc(C(C)C)o1 C1(NC(c2c(OC)ccs2)=O)CCN(C(=O)CC2(O)CCC2)CCC1CO C#CC1(NC(=O)C(CC)N(C(=O)C(C)CC(C)(C)C)C)CC2CCCC12 C12(CNC(C3C(C(N)=O)C3)=O)CCC(CN(C(=O)CN3CC4CCC3C4)C1)C2 C12(C(N3CCCN(C(C(CCC)OCC)=O)CC3)=O)COCC1CN(CCC)C2 C1(OCC(N2CC(OCC(N3C(C4(C)CC4)CCC3)=O)C2)=O)CCC(C)(O)CC1 CC1(C)CC(=O)CCC1C(N1CCC(n2cnnc2S)CC1)=O c1(OC(C(=O)N(CC(C)NC(c2cocn2)=O)CC)COC)ccc(Cl)cc1C C1(CNC(C2(NC(c3c(CSC)occ3)=O)CCOC2)=O)NC(=O)NC1=O N1(C(c2ccn(C)c2)=O)CCN(C(=O)CCS(N)(=O)=O)C(c2ccccc2)C1 C1(NC(CCOCCC)=O)CCS(=O)(=O)C12CN(C(=O)CCCC(F)F)C2 c1(CC(C(=O)NC(CNC(c2c(CC)con2)=O)CC)F)ccc([N+](=O)[O-])cc1 C=CCCCCNC(=O)CC1(C)CN(C(=O)COC(C)(C)CC)C1 c1(C(=O)NCC(C(C)C)NC(C(CC)NC(N)=O)=O)cc2c[nH]cnc-2n1 c1(Cc2cn(C3CN(C(C(=O)N(CCC#C)C)=O)C3)nc2)cccc(C)c1 c1(OC)nc(C)c(C(c2nnnn2C(C)C)NCCn2cnnn2)c(C)c1Cl Nc1sc2c(c1C(N1CC3(NC(=O)CC4(CO)CC4)CCC1C3)=O)CCC2 N1(C(CCC=C)=O)CCC2(CC1)CC2C(N1CCOCC(C(=O)O)C1)=O C#CCC(CC(F)F)C(=O)NC1CC(CO)(NC(C2CCN(C(C)(C)C)C2)=O)C1 Cc1cc(F)cc(C)c1C(=O)NCC1CN(C)CCN1C(=O)C(C#N)C1CC1 Cc1ncc(C(N2CCCC2(C)C(=O)NCc2ccc(NC(C)C)cc2)=O)n1C C1(NC(c2ccc(CC)cc2)=O)CN(C(=O)C(C#N)C(C)(C)C)C2CCCC12 C(=O)(CC(C)(C)NC(=O)CC(C)(C)NC(c1cnc[nH]c1=N)=O)NC N1(C(COCC)=O)CC(NC(c2nc(C)n(-c3ccccc3)n2)=O)C(CC2CC2)C1 C(=O)(C(CC)C(F)(F)F)N1CC(OCCNC(c2n(C=C)nnc2)=O)C1 C1(NC(C(C)OCc2ccc(C)cc2)=O)CCN(C(C2CCCCO2)=O)C1(C)C C1(NC(C2(OC)CC2)=O)COC2CN(C(=O)CC3(O)CCCCC3)CC12 C(N=c1cc(C)c(S(=O)(=O)NCC(C)(C)CCC)c[nH]1)C1C(=C)C1 N(C1CS(=O)(=O)c2ccccc21)C(CC1C(C(=O)OCC)C1)=O n1(CC)nc(CNC(C2CC(NC(c3ccnn3C)=O)CCO2)=O)c(C)n1 N1(C(c2cc(CCC)on2)=O)CC2CCC1CN2C(=O)C1=NOC(C)(C)C1 C(C)(CCCC(=O)N1CCC1CN=[N+]=[N-])NC(CCCC=C)=O C(C(=O)N1CCCC(CCNC(c2nc(C3CC3)oc2C)=O)C1)(C(C)C)OC c1(C(C(N)=O)NC(C2(F)CN(C(C3CC3F)=O)C2)=O)ccccc1Br C1(CC(=O)NC)CN(C(=O)CCCN(C)C(C)=O)CCN1C(=O)CC(C)C1CC1 Cc1ccc2c(c1)CN(C(C1(NC(=O)CC(=O)NC3CC3)CC1(C)C)=O)C2 C1(CC(=O)N(CCCCNC(c2c[nH]cc2Br)=O)C)CCOC(C)(C)C1 C=CC1(O)CCN(C(=O)COC2(C)CN(C(=O)C=C(C)C)C2)C1 C1(NC(C2(C)CCOC2)=O)CN(C(=O)Cc2ccc(O)cc2)CC2(CC2)C1 C(N=c1ncc(Cl)c[nH]1)C1CC(NC(c2cccc(C(N)=O)n2)=O)C1 N1(C(C(C=C)(C)O)=O)CCOCC(C)(CNC(c2c(Cl)c(C)nn2C)=O)C1 c1(CCNC(C(c2ccoc2)NC(CC(C)c2ccco2)=O)=O)ccncc1F N1(C(C(=O)N(C2CCN(C(=O)CSc3ccccn3)C2)CC)C)CCOCC1 c1(C(C(=O)NC(C2CCN(C(C3C=CCC3)=O)C2)C)=O)cccn1C c1(OC)cc(C(=O)NC2CN(C(=O)Cc3cocn3)CC2(C)C)c2c(c1)CCO2 O=C(C1CCOc2ccccc21)NCC12CCCN(C(c3cscn3)=O)C1C2 C1(Cn2cc(C(c3cccc(C)c3)O)nn2)CCC2(CC1)NC(=O)N(C)C2=O C(=O)(C1CCc2ccccc21)N(C1CCN(C(=O)C(C)(C2CC2)OC)CC1)CC c1(C(N(CC(=O)NC2(CNC(C3CCCC3(C)C)=O)CCC2)C)=O)ccccc1Cl Nc1c(C(=O)NCC(CNC(c2cncc(C3CC3)c2)=O)CO)cccc1F c1(OC)ccc(Cl)c(CC(N2CCC(O)(C(N3CCCC(F)(F)C3)=O)C2)=O)c1F c1(OCC(=O)NCCCC(C)NC(CSCCC)=O)ccc(Cl)c(C)c1 CC1NC(=O)C(N(C)C)=C1NCC(O)C(C)(F)F C1(NC(c2cccnc2O)=O)CCCN(C(C2(Cl)CC2(F)F)=O)C1 Cc1ccc(F)cc1CC(=O)NC1C2CN(C(C34CSCC3C4)=O)CC12 N1(C(c2c(C)csc2)=O)CCC(C)C(CC(=O)NC(Cn2cncn2)CC)C1 CC1CCN(C(c2cccc(Cl)c2)=O)CC1NC(=O)CC1CC2CCC1C2 N#Cc1cc(S(=O)(=O)NCC2CCN(Cc3cc(Br)c(F)cc3O)C2)ccc1F C1(C(=O)NCc2c(C)occ2)CC(=O)CN1C(C1CC(=O)C1(C)C)=O CC1(C(F)(F)F)c2cc(Br)ccc2CCN1C(=O)N(C1CCOC1)CC.C(C)(C)C c1(C(N2C(C)CC(NC(=O)CCCCC3CC3)C2)=O)ccc(N=S(C)(C)=O)s1 c1(CC)nc(N2CC(OCCNC(c3ccc(C)c(Cl)c3F)=O)C2)c(F)c(Cl)n1 C1(C(=O)NCC(C)(C)OC(C)C)CC12CCN(C(=O)C(C1CCCCC1)F)C2 C(=O)(CCCCCCNC(C1C2(CC2)C12CC2)=O)N(CC#C)CCOC CC(C(=O)NCC1CN(C(c2coc(C(F)F)c2)=O)CCO1)S(C)(=O)=O C(c1ccc(F)cc1)=C(C)C(=O)NCC(C)NC(c1ccc(N)cc1F)=O C12(CNC(c3ccc(C)cn3)=O)CCC1CN(C(=O)C(c1ccccc1F)C)C2 N1(C(CSCCN(CC)CC)=O)CC2(C)CC1CC(C)(C)C2 N1(C(C#CC(C)C)=O)C2CCC1CC(NC(C1CCCCC1C)=O)C2 N1(C(C2(NC(=O)CN3CSCC3=O)CCN(C)C2)=O)CC(O)C(C2CC2)C1 Cc1cn2c(n1)C(C(=O)NC1(C)CCN(C(C3(CF)CC3)=O)CC1)CCC2 C(CSC)(C(=O)NCCC1CC(NC(=O)CCCn2ccnc2)C1)OC c1(CC(=O)NCCCNC(C(C)OCCOCC)=O)cc(F)ccc1Br CCC(C)C(O)C(=O)N1CC2(NC(=O)C(N3CCC(C)CC3)=O)CC1C2 c1(CC(=O)NC(C(C(C)C)NC(=O)CCC2CCCC2)C)nc2c([nH]1)CCCC2 c1(OC)ccnc(C(=O)NC2(C)CC(NC(C3CC3(Cl)Cl)=O)C2)c1OC c1(CC(=O)OCC(c2nnco2)=O)ccco1 N1(C(CCCSCC)=O)CCC2(NC(=O)COc3ccc(F)c(C)c3)CC2C1 CC1(NC(=O)CCc2cc[nH]n2)CCN(C(C2CC2C(F)(F)F)=O)C1 Cc1ccc(O)c(C(N2CCCC2C2(NC(C3CC(C)OC3C)=O)CC2)=O)c1 OC12CC1C2.c1nc(C2(c3ccccc3)CC2)no1.[nH]1cccn1 C=CCCC(C(=O)N1CCCC(C)C1)NC(c1cc(C)cc(F)c1)=O C=CC1(C(N2CC(NC(c3ccoc3C3CC3)=O)C2)=O)CCCCC1 C1(C(N2CCCCC(NC(COCCCC)=O)C2)=O)Cc2n[nH]cc2C(=O)N1 C1(C(N(c2ccc(Cl)cc2)C)=O)CCC(C)(C)N(C(=O)C2=CCCOC2)C1 N1(C(C=CC(CC)=CC)=O)CCc2sc(CNC(C3(F)CCCOC3)=O)nc2C1 c1(C(=O)NC2CCCCCC2NC(C2CCCS2)=O)ccc2nonc2c1 N1(C(CCC#N)=O)CCC(NC(c2c(C(F)(F)F)cccc2F)=O)CC1C1CC1 N1(C(C)C(N2CCCC2CNC(C2(CC3CC3)CCCO2)=O)=O)CCCCCC1 c1(CC(=O)NC(CNC(CC(C)=C(C)C)=O)(C)C2CC2)ccc(F)c(C)c1 C1(NC(C2C(CC)CCO2)=O)CN(C(c2coc(Cl)n2)=O)CCC1C C(N=c1cc(C)nc(C)[nH]1)C1N(C(C(c2cccc(C)c2)(F)F)=O)CCCC1 Cc1ccc(C(=O)NCC=CCNC(C2CC2C(C)C)=O)c(F)c1F C1(O)(C(=O)NCC2CC(NC(c3ccc(C)nn3)=O)C2)CCCC(C)CC1 C1(CNC(C(COCC)C)=O)CN(C(=O)C(F)C(C)(F)F)C2(CCC2)C1 C1(CNC(Cc2ncc(CC)[nH]2)=O)CC2CCC1N2C(C1C(C(=O)OC)C1(F)F)=O N1(C(C(F)OC)=O)CC2CN(C(c3cccc4c3OCC4)=O)CC2(C)C1 c1(C(=O)NCC(C(C)C)NC(C(C2CC2)OC)=O)sc(C)cc1C N1(C(C(C)n2cnnn2)=O)CCC2(CC1)CN(C(=O)CSC(F)F)C1COCC21 C1(F)(C(=O)NC(C)CCCCNC(C2CCC2C)=O)CCCCCC1 N12CCC(CC1)C(C)Nc1cc(on1)CC2=O.C1(C(=O)N)CCN(C)C1C.CO.C1CC1 c1(CN(C(C2CCCN2Cc2ccco2)=O)CCO)cc(F)cc(Br)c1 c1(C(N2CC(C)C(Nc3ncnc(O)c3Br)C(C)C2)=O)ccc2nc(O)oc2c1 c1(C(N2CC3C(NC(CCCC(=C)C)=O)C3C2)=O)cc2c(=O)[nH]ccn2n1 Cc1csc(CC(=O)NC(C)CC(C)NC(=O)C(C)Cc2ccco2)c1 N1(C(c2cccc(CC)c2)=O)CCC2CN(C(C3(CC=C)CCCCC3)=O)C2C1 N1(C(CCCNC(C)=O)=O)C2CCC1CC(C(=O)NC(c1nncn1C)C)C2 Cc1c(C(=O)NC(CNC(C2(Cl)CCCCC2)=O)C(C)C)cccc1F c1(C(=O)NCC(=C)CCNC(=O)COC(F)(F)F)ccc(=O)n(C)n1 c1(N(C)CC)ccc(C(=O)N(C2CCN(C(=O)C(C)CC34CC(C3)C4)C2)C)cc1 C1(CC(=O)NNC(=O)C2OCCO2)C(F)(F)C12CCOCC2 C1(C2CCN(C(c3cc4c[nH]cnc-4n3)=O)C2)(NC(C2CCCSS2)=O)CC1 c1(C(N2CCN(C(C3C4CC5C(C4)C35)=O)CC2CCO)=O)nccn2ccnc12 N1(C(CC(CC=C)(C)C)=O)CCC2CN(C(c3cc([N+](=O)[O-])c[nH]3)=O)CCC12 c1(C(C)C)cc(=NC(C)C2CCCN2C(=O)C#CC(C)(C)C)[nH]c(CC2CC2)n1 N1(C(c2oc(C)c(CO)c2)=O)CC(C(=O)NOCC(C)(C)C)CCC1(C)C C12(C(N3CC(NC(c4cc(CCC)nn4C)=O)C3)=O)CCOC1CCOC2 C(=O)(CC(C)NC(=O)CCC1CCC(NC(=O)CC(C)N(C)C)C1)OC C(=O)(C#CC1(C)CCCO1)NC(CCC=C)C(=O)Nc1ccc2ccccc2c1 O=C1NC(c2ccccc2O)C(=O)N1CN1CCC(c2ccc(O)cc2)C1 c1(C(=O)NCC2C(CNC(C(C)=CC3CC3)=O)C2)cnc(S(C)(=O)=O)s1 c1(C(C(=O)NC)N(C2CC3CC3C2)C)cc(C2CC2)[nH]n1 N1(C(C(CC)CC)=O)CC2CCC2(CNC(=O)C=CS(C)=O)C1 CCCCC(O)CCC(=O)N1CCCOC(CNC(C2(C)CCN(C)C2=O)=O)C1 C1(CC)CCC(C(=O)NC2(C)CN(C(C3(CF)CCOCC3)=O)C2)CC1 C(=O)(C(C)(C)CCCO)NCC1C(NC(c2c(=O)ccn(C)c2)=O)CCC1 N1(C(C2C(C)(C)OCC2)=O)CCC2(CCC2)C(NC(=O)C(=O)NCC(F)(F)F)C1 CC1CCC(NC(=O)CC2(O)CCCOC2)CN1C(c1cc(=O)n(C)cn1)=O Cc1oc(C2CC2)nc1C(=O)NC1CCCC(CNC(=O)COC(F)F)C1 CCCC(C)C(C)(c1nnnn1C)NCc1ccc(-c2nc[nH]n2)cc1 C1(NC(c2nc(C(C)=O)sc2)=O)CCCN(C(C2(C)CCCC2)=O)CC1F C1(C(C)C(=O)N2CC(C(F)(F)F)C2)CCN(C(c2cncnc2C2CC2)=O)CC1 N1(C(C=COCC)=O)CCC(NC(c2cc3n(c2)CCC3)=O)C(F)C1 N1(C(c2c(CC)c[nH]n2)=O)CCCC(C)(NC(C2CN(C(=O)OC)CCO2)=O)C1 N1(C(CN2CC(C)C2)=O)CC(O)(CNC(=O)CC2(C)OCCO2)C1 c1(NC)ccc(C(N2C(C(=O)NCC(C)(O)C3(C)CC3)CC2C)=O)cc1 CCC(C(=O)N(CCC(=O)N(CC(C)(C)N(C)C)C)CC)NC(N)=O Cc1ccccc1CC(=O)NC1CN(C(C2(CCCF)CC2)=O)CC1C(F)(F)F c1(OC)ccc(CC(C)C(N2CCNC(C(=O)N(C)C(C)C)C2)=O)cc1OC C1(Nc2nccc(OCC)n2)CN2CCN1CC2C.C12(F)CC(C1)CNC2=O c1(CC)c(C(=O)N(C)CC2COCCN2C(c2cnnn2CC)=O)nnn1CC c1(NC(C2N(S(c3c(C)n[nH]c3C)(=O)=O)CC2)=O)cccc(C#N)c1[N+](=O)[O-] c1(NCC2OCC(C)C2)[nH]c(=NCC2(C(F)(F)F)CC2)nc2c1ncn2C c1(N(c2sc(=NCc3ccccc3Br)[nH]c2C)CC)c(F)cc(Br)cc1[N+](=O)[O-] c1(C(N(CCOCCCN(C(C2C(C)(CC)C2)=O)C)C)=O)cccc([N+](=O)[O-])c1 c1(CC(=O)NC2(C)CCN(C(C3(C)CC=CCC3)=O)C2)c(F)cccc1F N1(C(CC=CC)=O)CC2=C(C1)CN(C(=O)Cn1nc(C)c(Br)c1C)C2 C1(CNC(Cc2c(C)nsc2)=O)(NC(=O)C(O)CC2CCCCC2)CCOCC1 c1(C(=O)NC2CC(CNC(C3(OC)CCSC3)=O)C2)cnc2c(c1)COCC2 c1(CC)cnc(Cl)[nH]c1=NC1CCN(C(c2sncc2C)=O)CC1C C1(NC(CCC#C)=O)CC2(CCC(CNC(C3CC(C(F)(F)F)C3)=O)CC2)C1 N1(C(C2CC(C(C)C)C2)=O)CCCC(N(C(=O)C(C)C2CCCC2)C)C1 c1(CCNC(C(COC)(C)C)c2nnnn2C2CCOCC2)c(Br)cncc1Br N1(C(C(C)NC(=O)C2CC2)=O)CCCC2(C1)CC2(F)F Cc1ccc(C(=O)NC2CCN(C(c3cc(C(N)=O)cn3C)=O)CC2)cn1 c1(C(=O)OCC)cnc(NCc2nnc(CO)s2)s1 c1(C(N2CC3C(NC(CSCCC)=O)(C3)C2)=O)cc(SC)c(Cl)cc1Cl N1(C(C(CCC)NC(C)=O)=O)CCCC(C2CN(C(=O)C3=NOC(C)C3)C2)C1 CN1CCC2C(CCN2C(=O)CCC2CCCN(C(C3(C4(C)CC4)CC3)=O)C2)C1 C12(NC(CC=CC)=O)CCOCC1CN(C(c1cccc(Br)c1)=O)C2 CCCCC(CNC(c1cnccc1N(C)C)=O)NC(=O)CC(=O)NCC1CC1 C1(C)(CC)CC(NC(c2ccc(C(C)(C)C)s2)=O)CN1C(=O)CC=C(C)C Cc1sc(Br)cc1C(=O)CC(=O)OC(=O)Cc1ccc(C)n1-c1ccccc1 C(=O)(CCCC(=O)N1CCCC(NC(=O)C(C)(C)n2ccnn2)CC1)OC C1(CN(C)C(C2CCC2(F)F)=O)CCCCN1C(c1ccc(=O)oc1)=O C(CC1=CCCCC1)NN1C(CC(=O)N(C(CO)CO)CC)CCC1 C1(CC=C)CCCCN1C(=O)CNC(=O)CC#N c1(C(N(C(CNC(C(F)=CC)=O)C2CC2)C)=O)nn(C(F)F)cc1Cl N1(C(Cc2cc(C)sc2)=O)CCC2(CC1)CC(NC(=O)CCC1CC1(Cl)Cl)CO2 c1(NC(c2cc(OC)ns2)C)cc(C)c(S(=O)(=O)N2CCCC(O)CC2)cn1 c1(CNC(CC(COC)(C)C)=O)ccc2c(c1)COC2(C)C c1(C(=O)NCC(C)NC(c2cc(C(F)(F)F)c[nH]2)=O)cccc2cccc(O)c12 C1(NC(c2cnc(OCC)s2)=O)(CF)CCN(C(=O)CC(C)n2cccc2)C1 C1(OC)CC2(C1)CC(C(=O)NCC(c1ccccc1)CNC(=O)CC(C)C)C2 C1(NC(C(CC)N(CC)CC)=O)CCC2CC1CN2C(=O)CCC(C)(C)OC CC1CN(C(=O)Cn2nnc(=N)[nH]2)CC1CNC(c1cn(C2CCCC2)nn1)=O C1(C(N2CCC(SC)CC2)=O)CN(C(=O)C=CC(F)F)C2(CCC2)C1 Cc1cc(CNC(C2CCN(C(c3cc(C)nc(C)c3)=O)C2(C)C)=O)cc(F)c1 c1(C(=O)NCC2CCC(C)N(C(=O)COc3ccon3)C2)cccc2[nH]ncc12 N1(C(c2ccc(C3C(C)OCC3)nc2)=O)CCOCC1(C)c1ccccc1 C1(C(N(CCCCO)C)=O)C2CCCC2CN1C(C1CCC(=O)N1C)=O O(N(CC)C(=O)C1CC=CC(NC(c2ccnc(OC)c2)=O)C1)CC C1(CCCNC(C(COC)OC)=O)CCCCN1C(=O)C=C(C)c1ccco1 C1(CCNC(CCC(=O)NCCC)=O)CCCN(c2nccc(CC#N)n2)CC1 N(C)(C(=NCCF)NCC1C2CCC(C2)C1(C)C)CCOCCOC Cc1cccc2c1C(=O)NCCN2C(c1cnc(-n2cccn2)cn1)=O CCCC(C)(O)C(=O)NC1CC(OCC(N2CCC(n3cnnn3)C2)=O)C1 O=C1CC2(CCC2)C(C(=O)NCCN2CCN(CCO)CC2)CN1.C(CO)O c1(C(N2CC(CNC(=O)CCOCC3CCCO3)C2)=O)cc2ncccn2n1 C(=O)(C1=CC2C=CC(C1)C2)NCCC(=C)CNC(=O)CCc1cnn(C)c1C Cc1ccnc(C)c1C(=O)NCC(CO)NC(=O)CC1CC(c2ccccc2)C1 C1(F)(CNC(C(n2ncc(C)c2)C)=O)CCN(C(=O)C(F)C(C)C)CC1 c1(C(N2C(C)CCN(C(C3(OC)CC3)=O)CC2)=O)cc(O)nc2cc(F)ccc12 c1(C(=O)NC2CS(=O)(=O)CC2NC(c2ncccc2O)=O)cnc2n1CCOC2 Cc1c(C(N2CCN(C(C3(C)CC3F)=O)CC2)=O)sc2[nH]cnc(=O)c12 C1(OC2CN(C(C(C)C)=O)C2)CN(C(=O)C(C)(O)c2ccccn2)CCO1 N1(C(CCNC(N)=O)=O)CC2C(CO)C2C1.C12(CC1)C(=O)NCCO2 c1(CNC(=O)NCCC2CCOC2)ccc(CO)c(Cl)c1 N1(C(C(C)(C)O)=O)CC(NC(C2CC3CCCCCCC23)=O)CC2(CCC2)C1 C(=O)(CCC(C)CN(C)C)NC(CC1CCN(C(C(C)OCCC=C)=O)CC1)C C1(C(=O)NCCC2CC(NC(C(C=C)O)=O)C2)CCCCN1Cc1ccccc1 n1(C2CC(C(=O)OC)C2)nnnc1C(c1cncnc1)NCCn1cnnc1 c1(CC)cc(C(N2CCC(N(C)C(c3ncccc3F)=O)C(C)C2)=O)cc(Cl)c1 N1(C(CSc2ccc(C)cc2C)=O)CC2CCCC1CN(C(=O)C1CC1)C2 C1(CNC(C(c2ccc(F)cc2F)C)=O)CC2CN(C(C3CCC3)=O)CC12 C1(C(=O)NCC2(F)CN(C(C(CC=C)NC(C)=O)=O)C2)CCC2(CCOCC2)O1 c1(C(=O)NCC2CCC(NC(c3ccc(CC#N)cc3)=O)C2)cc2n(n1)CCC2 N1(C(c2n(CC)nnc2)=O)CC2CC1C2NC(c1cc(C2CCOC2)[nH]n1)=O c1(C(N2CCCC(O)C2)C(=O)NCC)cccc(N(C)C)c1.c1(CC)ccccc1Cl C1(C(=O)NCCc2ccccc2OC(F)(F)F)CNCC1C1CCOC1 N1(C(C(c2ccccc2F)(C)C)=O)CCC(CF)(NC(C2CCCO2)=O)C1 c1(C(=O)NC2(CC=C)CN(C(c3nsnc3O)=O)C2)coc2c1COC2 CC(C)(C)CC(O)C(=O)NCCCCCCC(=O)NCCCC1(O)CC1 C1(OC)CC2C1CCN2N1CC(c2nc(O)c3ccccc3n2)C1 C1(C(=O)Nc2cn(C3(CN)CC3)nc2)CCCC2(C1)CC2(F)F c1(C(N2CCC(NC(C(CCC#C)O)=O)CC2)=O)c[nH]c2ccc(C#N)cc12 c1(C(=O)NC2C(NC(c3c(C)n(C)nc3)=O)COCC2)ccn2c1CCC2 c1(C(N2CCC(C(=O)Nc3c(C#N)scc3)C2)=O)ccc(O)c([N+](=O)[O-])c1 N#CC1(C(=O)NCCCCCNC(c2ccc(C3CCOC3)s2)=O)CC2CC2C1 n1(CCC#C)c(N2CCC(CCCOC)CC2)nnc1-c1ccc(C)o1 O=C(C(F)(F)CCn1cc(C2CCC2)nn1)NCC1CCSCC1 C1(NC(CC(=C)C)=O)CN(C(=O)CC2(OCC)CC2)CC1Cc1ccccc1 C1(CNC(CC2(CNC(=O)Cn3nccn3)CC2)=O)(OC)CC2CCCC12 CCC(CCCC(=O)NCCC1CCCC(C)C1)NC(C1COCC(C)O1)=O c1(CNC(=O)NCC(=O)Nc2cnc(O)nc2O)cnc2[nH]cncc1-2 c1(C(=O)OC)cc2c(s1)CCC2NC(=S)Nc1cccc(F)c1C c1(C(N(C2CCN(C(C(CC=CC)C)=O)C2)CCC)=O)ccc(C2CC2)c(Cl)c1 n1(CCOCC)nnnc1C(c1ncoc1C(F)F)NC1CC(C)C1 c1(OCC)cc(-c2nccn2Cn2cccc2)cc(C2CC2)c1O C(=O)(C(C)CCCC(C)C)N1CC(CC(=O)NC(CC)C(=O)NC)OCC1 CC(C)CC(CNC(c1ccc(C(O)CF)cc1)=O)NC(c1cc(Cl)n(C)n1)=O C1(C(=O)OC)CCC2(CCOCC2)CN1C(=O)C(c1ccccc1F)C N1(C(C=C(C)c2ccccc2F)=O)CC2CC(C1)CN(C(=O)C(C)C(C)O)C2 C(=O)(C1SCCc2sccc21)NCC(C1CCC1)NC(c1cc(C)n(C)c1)=O N1(C(CCC2CCCCN(C(c3cccc[n+]3[O-])=O)C2)=O)CC2CCC(C1)C2O C1(C(C)(C)NC(CNC(CC)=O)=O)CCN(C(=O)C(F)=C2CCCC2)C1 C(CC(O)C(=O)NCC1CCN(C(C2CCCC2c2nc(S)n[nH]2)=O)CC1)SC N1(C(c2ccc(C3CCC(=C)CC3)cc2)=O)CC2CCOCC2C1 Cc1nc(C=CC(N2CC(F)(CNC(C3CCC3C(F)F)=O)C2)=O)cs1 C12(NC(C=CC(=O)NC3CC3)=O)CCN(C(=O)Cc3ncc[nH]3)CCC1C2 N1(C(C2C(C)OCC2)=O)CC(C)(C)C(NC(C2CCN2S(C)(=O)=O)=O)C(C)(C)C1 n1(CCC(=O)NCC(CC)NC(=O)Cc2cn(CC)nn2)ncn(C)c1=O C(C(C)(C)CC(=O)N(C1CCCN(C(=O)C(C)CC(N)=O)C1)C)OC N1(C(c2nc(OCC)sn2)=O)CCC2(CC(NC(C3(C)CCOC3)=O)C2)C1 C1(C(=O)OCC)CCC(CCC(C)C)CC1.n12ccnc1CCCCN(C)C2=O Cn1nccc1C=CC(=O)NC(C1CCOC1)CNC(=O)C(C)(C)n1cc(Cl)cn1 CCC(C)(C)CCCC(=O)N1CC(C(=O)NC(CO)CC(C)(C)C)C(C)C1 C1(C2CCC2)(C(N2C(C3(O)CN(C(C4(COC)CCCC4)=O)C3)CCC2)=O)CC1 N1(C(Cc2c(C)nsc2)=O)CCC2(NC(=O)Cn3ccc(O)nc3=O)CCCC12 CC(C)CC(O)C(C)C(=O)NC1CCCC(CC(N2CC(N(C)C)C2)=O)C1 C1(C(=O)NCC(CN(C(=O)CN2CC(=O)NC2=O)C)(C)C)CC2CCC(C1)S2 C1(C(=O)NC2(CC(=O)NCCCn3cccn3)CC2)CCS(=O)CC1 c1(CC)ncc(C(=O)NC2CCCN(C(c3ccnc(Cl)c3N)=O)C2)c(C)n1 C1(CC)CN(C(=O)COC(F)(F)F)CCN1C(C1CCN(C)C(=O)C1)=O N=c1[nH]c(CC(=O)NCC2(CNC(=O)C=CCF)CC2(F)F)cs1 C1(NC(C(C)C)=O)CCN(C(C2(CF)CC2)=O)CCC1(F)F c1(C(C)NC(=O)OC(C)(C)C)nc(C(=O)NCc2nc(C(C)C)ns2)cs1 c1(C(=O)NC2(CN(C(CN3C(=O)CN(C)C3=O)=O)C)CC2)nccc2cc[nH]c12 C1(CC)(NC(c2cc(F)cs2)=O)CCN(C(C2CCCNC2=O)=O)CC1 c1(C2(CNCC3N(C(c4ccc(Br)o4)=O)CCC3)CC2)ccnc2ccccc12 C1(C(N2C(CN(C(CN(CC(=O)NC(C)C)C)=O)C)CCC2)=O)SC(=N)NC1=O Cc1c(C(N2CC(CNC(=O)Cc3cccnc3O)CC2C)=O)cnn1CCO C1(C(=O)NCC(C2CC2)N(C(CNC(=O)OC)=O)C)(C(=O)OC)CCNCC1 C1(CNC(C(CC=CCC)C)=O)CN(C(c2cnc(CC)nc2O)=O)CC1(C)C CCCCC(CNC(=O)CCc1cn[nH]c1)NC(=O)C(C)SCC c1(-c2ccc(OC)c([N+](=O)[O-])c2)cnc(N=c2[nH]c(C3CC3)cc(C)n2)nc1 c1(C2CN(C(c3n(C4(C)CC4)nnn3)=O)C2)noc2c1CCC2.C1(N)CCOC1 Cc1ccc(OCCC(=O)NCCC(C)NC(=O)CSC(F)F)cc1 N1(Cc2cc(C)on2)CCCC1C1CCCCN1C(c1cc(C2CC2)no1)=O N1(C(C(C)CF)=O)CCCC(C)C1CNC(c1cnn(C2CC2)c1)=O C1(NC(C2C(=C)CC2)=O)C2CC1N(C(C1CCCN1Cc1ccccc1Cl)=O)C2 Cc1cc(C(=O)NC2CCC3CC2CN3C(=O)CCNS(C)(=O)=O)cc(C)c1C N1(C(c2cc(C(C)=O)oc2)=O)CC(NC(=O)CCc2cccnc2Cl)C(C)C1 CC(C(=O)NC1CN(C(c2cn3cc(Br)ccc3n2)=O)C1)C(F)(F)C(F)F N1(C(CCCCCOCC)=O)CCC2CN(C(C3CCS(=O)(=O)N3)=O)CC12 N1(C(C)=O)CCC(CNC(=O)CCC(=O)c2cc(C)sc2C)C(C)C1 C1(OC)CCCN(C(=O)C(C)(C2CCC2)NC(c2ccc(SC)s2)=O)C1 Cc1nc(C(N2CCCC(N(C(=O)CCCc3ccc(Cl)cc3)C)C2)=O)nn1C c1(-c2onc(-c3cccc(SC)c3)n2)cnn2c(C)c(C)ccc12 c1(NCC)ccccc1C(=O)NC(CO)C(=O)NCCC12CC(CCO1)C2 C123CCC(CC1)(CO2)CNC3=O.C(=O)(C(C)c1ccco1)CNCCOC(C)C N1(CCC)CCN(C(=O)C(C)CN(C(=O)CC(CC)SC)C)CC1 C1(C(=O)NCC(C)N(C(=O)COCC2CCCO2)C)CNC(=O)CC12CCC2 N1(c2nnc(C)o2)CCC2(CCC(CNC(C3(Br)CC3)=O)OC2)CC1 C1(CN(C(C(COC)OC)=O)C)CN(C(c2cc(C)c(C)o2)=O)CCO1 c1(C(=O)NC(C)CNC(c2cc(C(F)(F)F)cc(F)c2)=O)coc(S(N)(=O)=O)c1 Cc1cccc(F)c1CC(=O)NCC1(NC(C23CCCC(C2)OC3)=O)CCCC1 C1(CNC(C2(C(C)(F)F)CCC2)=O)CC2(CC2)CN1c1nc(CC2CC2)ns1 CC1(C)CCC(O)(CNC(C2(CCNC(=O)C=CC3CC3)CC2)=O)C1 C(=O)(CC(F)(F)C(F)(F)F)NCC12C(CN(C(c3c(N)c(O)ccc3Cl)=O)C1)C2 CC(C)(C)C(C#N)C(=O)N1CCC(C(N2CCCC3(CC3)C2)=O)(CF)C1 Cc1cnc(NC2CCCCNC2)c(S(=O)(=O)NC2CCCC2F)c1 Cc1ccc(Cl)c(O)c1C(N1CCC(N(C)C(C2CCCN2N=O)=O)CC1)=O c1(NC(CN(C(=O)CC2CNC(C(F)(F)F)CO2)C)=O)ccc2nccn2c1C c1(C(N2C(CNC(CC(=C)C)=O)CCC(C)C2)=O)onc2c1CCCC2 N1(C(C2C(C)OC(=O)N2)=O)CCC(CNC(C2(CF)CCC2)=O)C(C)C1 N#Cc1cc(C(N2CC3(C2)CN(C(c2n[nH]c4c2COC4)=O)C3)=O)ccc1F C1(CC(=O)NC(C2CCN(C(C3CC(O)C3)=O)C2)(C)C)CC2CCC(C1)N2C c1(OCC)c(CN2CCCC2)cccc1Cl.c1(C(=O)NO)cncc(OCC)c1 C(=O)(C#CC1CCCCC1)N(CC1CCN(C(C23CC(C(C)(C)C)(C2)C3)=O)C1)C1CC1 c1(C(N2CCN(C(C(C)OC)=O)C(C3CC3)C2)=O)cccc2ccccc12 C=CCC(C(=O)NCCc1ncoc1C)NC(c1cncc(F)c1)=O C1(CNC(Cc2cc(C)sc2)=O)CN(C(=O)CCCC(C)(F)F)CCC12CCC2 CC(C)C(C(=O)Nc1ccc2ncnn2c1)C(C)NC(=O)C(O)CN1CCCC1 N1(C(CCN(CCC)C)=O)C2CCC(C(=O)NCc3n[nH]c(C)n3)C1CC2 c1(N2CC(NC(c3c(OC)cncc3)=O)C(C)CC2)ncn(C)c(=O)c1Br c1(SCC)cccc(C(N2CC(C(=O)Oc3ccccc3C)CC2=O)=O)c1 c1(OC)ccccc1OCCC(=O)NCC1(O)CCN(C(=O)C(C)NC(N)=O)C1 C1(NC(C(N(C(c2snc(C)c2N)=O)C)C2CC2)=O)CCc2c[nH]nc2C1 N1(C(=O)OC(C)(C)C)CCC(O)(COC(=O)NCCC2CCC(F)(F)CC2)CC1 c1(NC(C2(F)CN(C(c3n(C)cc(F)c3)=O)C2)=O)ccnc2c1ccn2C N1(C(C=CCN(C(c2cc(CC)no2)=O)C)=O)CCN(C)C2CC12 C(=O)(C1=CCCN(C(=O)CN2CC3CC3C2)C1)NCc1ccc(C#N)s1 C1(CC(=O)NCC2(COC)CCCO2)CC(C)N(C(c2cc(=N)[nH][nH]2)=O)C1 CC1(C)CC1(CO)NC(c1cccnn1)=O.c1(CC(=O)O)ccccc1 C1(N(C(CSCC=C)=O)C)CC2CCC(C1)N2C(c1cnc(N(C)C)o1)=O Cn1c(C(N2CCCC(CCCCNC(=O)C(O)C3CCC3)C2)=O)ccc1C#N N1(C(c2c(CCC)n[nH]c2)=O)CC(O)CC1(C)C(=O)NCc1ncn(C)n1 Cc1ccnc2c(S(=O)(=O)NCCc3ccc(=N)[nH]c3)cccc12 C1(C(=O)NC(CCC)C(=O)NCC2(C)CCC(=O)N2)CN(C)CC(C)O1 C=Cc1cc(C(N2CCN(C(=O)CC3(O)CCOC3)CC2CC)=O)cc(F)c1 c1(C(COC)NC(C2(c3ccc(Cl)cc3)CCC2)=O)ccccc1F C1(NC(C2C(OCC)C2)=O)CC2CCC1CC2N(C(=O)CN1CCOCC1)CC c1(C(=O)NCC(CO)NC(C2(CCCC)CCC2)=O)cc2ccsc2n1C Cc1coc(C(N2CC(N(C(=O)CSCC(=O)NC3CCCCC3)C)C2)=O)c1C CCC(C)C(C(=O)NCCCS(C)(=O)=O)N(C(=O)C(F)C(C)(F)F)C C(CO)(C(=O)N1CCC(C(F)(F)F)C1)NC(C(C)=C1CC1)=O N1(C(C2N(C)C(=O)CCC2)=O)CC(F)(F)CC1(C)CNC(=O)CC1CCOCC1 CCC(C)C(C(=O)NCC(C)CNC(c1ncc(C)s1)=O)NC(=O)OC(C)(C)C N1(CC(=O)NC(CNC(COCCOC)=O)C2CC2)CC2CCC1C2 CC1C(C(=O)NNC(=O)c2ncccn2)CCN1CCSC(C)(C)C S(=O)(=O)(c1cccc(Cl)c1Cl)N1CC(NC(c2scc(C)n2)=O)C(F)(F)CC1 c1(OCC)ccc(N)c(C(N2CCCC2C2(NC(c3ccns3)=O)CC2)=O)c1 c1(C(=O)NC2(CNC(C(c3cccc(Br)c3)C)=O)CC2)nc2ncccn2n1 C1(NC(c2c(CC)[nH]cc2)=O)CCC12CN(C(c1cc(C(N)=O)c[nH]1)=O)C2 C(=O)(C1=CS(=O)(=O)CCC1)N1C(CNC(c2cnc(SC)n2C)=O)CCC1 S(=O)(=O)(c1ccc(NC(CO)CC(F)(F)F)c(F)c1)NC1(C)CCCOC1 C1(CSCC(=O)NCCC2(NC(c3ccccn3)=O)CCC2)CC1C1CCCC1 [N-]=[N+]=NC1CCC(C(=O)NC(C2CCCOC2)CO)CC1 CC1CCC(NC(=O)CCN2CCCC2=O)CN1C(=O)CNC(N)=O C1(O)(C(C)NC(Cc2ccc(CCC)cc2)=O)CCN(c2nnnn2C)CC1 c1(C(=O)NC2(CC=C)CN(C(=O)C(O)CC(C)C)C2)c(C)nn(CC)c1Cl C1(NC(c2nc(C)[nH]n2)=O)CC(=O)N(C2CN(C(=O)Cc3ccc(Cl)cc3)C2)C1 N1(C(CCC=C(C)C)=O)CCC(C(=O)N(CC(N2CCCC2)C)C)CC1C C(=O)(C1=CCC2CCC1N2C(c1ccc(N)cn1)=O)NCCCC(C)C C=CC(C)N=c1[nH]c(=N)[nH]c(=NCc2cccc(SC(F)F)c2)[nH]1 c1(C(=O)NCC(C2CCC2)NC(C(C)O)=O)ccc(S(C)(=O)=O)cc1Br Cc1cnn(CC(=O)NC2CCC2NC(=O)Cn2ccc(C)n2)c1 C(=O)(C1NCCc2nn(C)cc21)NCCc1c(C(=O)OC)cccn1 C1(N(C(C(C2CN(C(C3CC3CC(C)C)=O)C2)OC)=O)C)CCOC(C)(C)C1 C(C(CC1CC1)C(=O)N(C)Cc1cn(C)nn1)NC(C1(SC)CC1)=O c1(C(C(=O)NCC2(OC)CCN(C(CCC#C)=O)C2)C)cc(C)cc(F)c1 c1(CC)ccc(C(=O)NCCn2cc(-c3csnn3)nn2)c(F)c1 O=C(C(F)Cc1ccccc1)NC1(CNC(C2CC2(Cl)Cl)=O)CC1 C1(NC(C2(C(N)=O)CC2)=O)CC2(CCC(NC(c3ccnn3C3CC3)=O)CC2)C1 C=CCC(CNC(c1scnc1C)=O)NC(C1CCCCO1)=O C(CC)(C(=O)N1CCC1CNC(c1c[nH]nc1OC)=O)=CCCC c1(C(NOCc2cn(CC(CC)O)nn2)=O)ccc2cc(OC)ccc2c1 C(=O)(C(C(C)(C)O)NC(c1cc(C(C)C)[nH]n1)=O)NCCC(CCC)O C1(CCNC(CC=C=C)=O)CCCN(C(=O)CCc2ccc(CC)cc2)C1 c1(CC(C)C)nccc(C(N2CCC(C)(CCNC(=O)C(F)=CC3CC3)C2)=O)n1 N1(C(CCCC#N)=O)CCCCCC1C(=O)NCCn1cncn1 C1(C(N2CC=C(CNC(Cc3nc(CC)sc3)=O)CC2)=O)CCCCC(=O)C1 CC1N(C(C2CC23CC(NC(=O)COCCN(C)C)C3)=O)CCC1(C)C C1(CNC(c2c(OCC)scc2)=O)CCCCCN1C(=O)CC(C)C1CCCC1 c1(-c2onc(-c3nc(N4CCOCC4)ccc3)n2)ccc2n[nH]cc2n1 c1(C(N(CC(=O)OC)CC#N)=O)cc(C)c(C(=O)O)cc1C Cc1ccc(CNC(C2CCN(C(C3COCC3(C)C)=O)C2C)=O)cc1 Cc1cc(F)c(C(N2CCC(O)(C(C)NC(=O)CCC(F)(F)F)CC2)=O)cc1F N#Cc1ccsc1C(N1CC=CC(C(N2CC(OCCO)C2)=O)C1)=O C1(c2n(CCCC)nnn2)(NCCOCC)CCC2CCCC2C1.CCF C1(NC(C2C(C=C(C)C)C2(C)C)=O)CCCN(C(=O)CC2(OC)CCCC2)CC1 c1(C(N2CCN(C(C3(C=C)CC3)=O)CC2CO)=O)cc2oc(Br)cc2s1 CN1CCOC2CN(C(C3(C)C=CCN3C(C3CC3c3ccccc3)=O)=O)CC12 C(CCCC(c1nnnn1CCSC)NCC1CCSC1)OC c1(C(=O)NCC2N(C(c3noc(CC)c3C)=O)CCCC2)cc(S(N)(=O)=O)cs1 c1(C(N(C2CCN(C(=O)C(C)(C)CF)C2)CCC)=O)ccc(C(C)C)cc1F C1(C(=O)NCC(C)N(C(=O)CNC(=O)NCc2cccnc2)C)C2COCC12 C1(CC(=O)N(C)CC2CCCN2C(=O)CCn2cncn2)COC2(CCC2)CO1 C=CCC(CC)C(=O)NC12CC(CNC(=O)CCc3cccnc3F)(C1)C2 C1(SC)CCC(NC(c2cn(CCNC(C3(c4ccno4)CC3)=O)cn2)=O)C1 c1(OCC(N2CCN(C(C3(C)CC3)=O)CC2CCO)=O)ccc2c(c1)CCCC2 c1(OC)ccc2c(ccn2CC(=O)NCC2CCCCCN2C(C2CCSC2)=O)c1 c1(CNC(C2C(C)=C2)=O)ccc(CNC(=O)CC2CCCC(O)C2)c(F)c1 C1(NC(COCCCC)=O)CCCOC12CCN(C(=O)C(C)(C#N)CC)CC2 c1(CCC(=O)N(C(C)CCNC(=O)CCC[N+](=O)[O-])C)c[nH]c2ccccc12 c1(C(=O)NCC(N(C(Cc2scc(CC)n2)=O)C)C2CC2)ccc(S(C)=O)cc1 CC1CCCC1C(=O)NCC1CC1CNC(=O)C(c1ccn(C)c1)C c1(NC(C2N(C(c3n(C)c(C(F)(F)F)cc3)=O)C3C(C2)C3)=O)cc(Br)cnc1I CCC(CC)C(=O)NCC(=O)N(CC(C)NC(=O)Cc1cc(Cl)ccn1)CCOC c1(OC)nc(C)ncc1C(=O)NC1CN(C(c2cc(C)c(O)nn2)=O)CC12CC2 c1(NC(c2ccccc2-n2cc(CCCO)nn2)=O)cccc(Cl)c1.N12CC(C1)C2 n1(CC)cnc2cc(C(=O)NNC(=O)C(C)SC(F)(F)F)[nH]c2c1=O c1(-c2cn(C(CNC(COCCCC)=O)C)nn2)ccc(-c2cn[nH]c2)cc1 N1(C(c2cnc(C)nc2)=O)CCC(C2CC2)C1CNC(c1cc(CCO)on1)=O N1(C(c2cnc(NCC)c(Cl)c2)=O)CC2(COC(CNC(=O)C(C)C(C)C)C2)C1 c1(NCc2cccc(F)c2I)ccc(C2=CCSCC2)nc1 c1(C(N(C(C)CNC(C2(n3ccnn3)CC2)=O)C)=O)cc2c(F)c(F)ccc2[nH]1 C(CC(CC)C(=O)N1CCC(F)(CNC(=O)CC)C1)=CC.c12cccc(c1)N2 c1(C(=O)NC(CC)CNC(c2c[nH]nc2C(F)F)=O)cccc(C#N)c1C CC1CN(C(=O)CCc2ccc(CCC(=O)O)cc2)CC1NC(=O)OC(C)(C)C N1(CC(N2C(C3(NC(=O)C=CCF)CC3)CCC2)=O)C(=O)CNC1=O c12cc(on1)COC2=O.C(=O)(C(CC1CCCO1)SC1CC(F)C1)OCC C1(NC(c2ncc(F)cn2)=O)CCC2(CC1)CN(c1cncc(Cl)n1)C2 c1(NC(C)=O)cccc(C(N2CCCC(C3CC(N)CCO3)C2)=O)n1 c1(C(=O)OCC(=O)NC(c2ccccc2)C)cnc(-c2ccco2)s1 N12CC3(CCC1C3)CCNC(=O)c1nc(cs1)C2=O.C1(OC(C)=O)CC(O)CN1 N1(CC2N(C(=O)NCCc3ccn(CC)n3)CCC2)CCN(C)CC1.CCO C1(CCNC(c2c(C)coc2)=O)CC(F)(F)CN1C(c1ncc(C(F)F)s1)=O c1(OC)cncnc1C(=O)NCC(C1CCOC1)NC(c1nncs1)=O C1(CC(=O)N(CCCCC)C)CN(C(C2(CC)CC2)=O)CCO1 c1(C(=O)NC(C2CCN(C(=O)C(C)n3cnnn3)C2)C)cccc2c1CC(=O)N2 C1(CC=C)(NC(=O)C(C)NC(=O)CC)CCN(C(c2c[nH]nc2C(C)C)=O)C1 C(=O)(CCS(C)(=O)=O)NC(C(=O)N(C1CCNC1=O)CC)Cn1ccnn1 c1(C(=O)NC(CCCNC(C(CC)CC2CCCC2)=O)C)cc(N)cc(F)c1 c1(C(N2CCN(C3CCN(C(C4C(C)C4)=O)CC3)CC2)=O)ccc(Br)nc1O c1(CC(=O)NC2C(NC(=O)C=Cc3cc[nH]n3)C2)ccc2ccccc2c1 c1(C(=O)NCC2N(C(c3ccc(C)cn3)=O)CCC2C)cc2c(s1)CC(C)(C)C2 CC1(C)OCC2CC12C(=O)NCC1CCN1C(c1nocc1Cl)=O c1(C(=O)NCCC(=C)CNC(=O)CC=C(C)C)cc(C2CC2)ncc1Br CCCC(C(=O)NC(C)CNC(=O)C(C)(C)OCC)OCC c1(C(=O)NC2CC(CC(C)C)OCC2)cc(S(C)(=O)=O)ccc1F CC1(C(=O)NC2CCCC2NC(C2CC(F)(CO)C2)=O)CCc2ccccc21 CC1(C(=O)NC2CCCC2NC(C2(C3CCCO3)CC2)=O)CC1(F)F c1(N2CCN(c3c(C)cccc3C)CC2)cc(C(F)(F)F)nc2ncnn12 c1(C(N2CCN(C(C#CC3(CC)CC3)=O)C(C)CC2)=O)ccc2oc(=O)oc2c1 N1(C(c2c(C)nccc2)=O)CCCN(C(=O)C(F)CC2CCCCC2)CC1C C(=O)(C(=O)N=c1ccn(CC(=O)Nc2cccc(Cl)c2Cl)c(O)n1)N(c1nccs1)C CC1C(NC(c2cc3c(F)cccc3s2)=O)CC2CCC1N2C(c1cnns1)=O c1(C(N2C3C(NC(c4c(COC)cc[nH]4)=O)C(C3)C2)=O)cccc2cnccc12 Cc1ocnc1CC(=O)N(C(C)CCNC(=O)CC1CC1C1CC1)C C=CCC(CC)C(=O)NC(C(=O)N1CCC(C(=O)OC)C1C)C(C)(C)C C1(C(=O)NC2CC(C(=O)OCC)OC2)COCCC1C1CC1 CCC(C(=O)NCCC1CC(NC(=O)CCC2CCCN2C)C1)C(C)(C)CC N1(C(C2CCC(CC)CC2)=O)CCCC2(CCN(C(=O)C(F)C(F)(F)F)CC2)C1 Cc1[nH]nc(Br)c1C(=O)NC1CC1CNC(=O)C(c1ccccc1)C C12(CNC(COCCC)=O)CC(NC(=O)C(OC)OC)(CO1)C2 CC(=O)CCCCCCC(=O)N1CCC(CF)(NC(=O)C2=CS(=O)(=O)CCC2)C1 C(=O)(CCC(=O)NCC1CCCCC1NC(=O)CSCC(=O)OC)NC C1(C)(C(=O)NCC=CCNC(C(N2CCOCC2)C)=O)CCCS1(=O)=O c1(C(N2CCC(OC)C2)C(=O)NC2CCCCC2)ccc(C)c(C)c1F CCC(COC)C(=O)N1CC(C(=O)Nc2csnc2C)(CC)C1 C(=O)(CCC(C)(C)F)NC(C1(O)CCN(C(C2CCC(C)O2)=O)C1)C N1(CC(c2cscn2)N(C)C)C(=O)NC(c2cccc(F)c2)C1=O c1(C(C)C)ccc(CC(=O)OCC(=O)NC2CC=CCC2)cc1F Cc1oc(-c2cccs2)nc1C(=O)NCC1(F)CC(NC(=O)C=C2CCC2)C1 c1(CNC(CC(C)C)=O)cnn(C)c1C(N1CCOCC1OC(=O)C1CC1)=O c1(C(=O)NCCN(C(C=Cc2ncc(C)[nH]2)=O)C2CCC2)ccc(O)c(F)c1F C1(C)(CCC(=O)NCCCCC2C(C)C2)CCCN1C(C1CCCCCC1)=O N1(C(c2cc(C(CC)CC)no2)=O)CC2(CCN(C(C3(F)CCOC3)=O)C2)C1 c1(C(N(C(CNc2ncc(C(=O)OCC)nc2)C)C)=O)cc2cc(C)ccc2s1 N1(C(c2c(CC)n[nH]c2)=O)CCCCC1CNC(=O)Cc1nonc1C C1(C(=O)OC)Cc2c[nH]nc2CN1C(c1ccc(OCc2ccccc2)nn1)=O C1(C(=O)NCCCC2(CNC(C(C)OC3COC3)=O)CCCC2)CCCC12CC2 c1(NC(CCN(CC=C)C(C2OCCC2CC)=O)=O)cn(C)c(=O)nc1O c1(C(=O)NCC(C)(CO)NC(c2cccs2)=O)cccc(-n2ccnc2O)c1 O=C1CC2(CNC2)C(CNCC2CCN(c3ccccc3)C2)O1 C1(C(N(C(CNC(c2c[nH]c(=NC)o2)=O)C)C)=O)CC2C=CCC(C1)C2 COn1cnc(C)c1C(=O)NC1CCCCC1CC(N1CC(O)(CN(C)C)C1)=O Cc1cc(F)ccc1NC(=O)C(N1CCOCC1c1nc[nH]n1)c1ccoc1 c1(NCCC(CCC)C)cc(=NC(C)c2cnc(Cl)c(Cl)c2)[nH]c(COC)n1 CC(Cc1ccncc1)C(=O)NC1CC(CCNC(c2[nH]ncc2Cl)=O)C1 Cn1nc(CNC(C2CCS2(=O)=O)=O)cc1C(=O)NCCn1ccc(=O)cc1 c1(CC(=O)N(C2CCN(C(c3c(C)csc3)=O)C2)C)ccccc1I C1(CNC(C2C(C)CC=CC2)=O)CN(C(=O)CCCC#N)C2CCN1C2 c1(OC)ccc(Cl)c(C(=O)NC2CC(CNC(c3ccnn3C)=O)C2(C)C)c1 N1(C(c2c(C)cns2)=O)CC=CC(C(=O)NCC2CNC(=O)CO2)C1 C1(NC(C2(C(=O)NC)CC2)=O)CCCC2CN(C(c3conc3CC)=O)CCC12 N1(C(c2c[nH]c(=NC)o2)=O)CCC(CNC(=O)C(C)CS(C)(=O)=O)C(F)(F)C1 CC(C(=O)NC1CN(C(C2CC(F)(CO)C2)=O)CC(C)(C)C1)C(C)S(C)(=O)=O Cc1cccc(C)c1C(N1CCC(C(F)C(=O)N(C2CC(O)C2)C)C1)=O N1(C(=O)Nc2cccc(O)n2)CCCN(C(c2cnc(C(F)(F)F)cn2)=O)CC1 c12ccc(c([N+](=O)[O-])c1)c(=O)[nH]2.N1(C(=O)OC)CCN(CCNC2CC2)CC1 c1(CC)cccc(F)c1-c1ccc(Nc2nnc(-c3ccco3)o2)nc1 C1(C(=O)OC)CC(NC(=O)C(C2CCCN(Cc3ccc(C)s3)C2)C)CN1C c1(C(=O)NCC23CC(NC(CC(C)O)=O)(C2)C3)ccc(OC(F)(F)F)cn1 N1(C(COCCCC#C)=O)CCCC(CNC(=O)C(C)N(C)C)CC1 c1(CC2N(C(c3cccc(CC)n3)C(=O)NCC)CCOC2)c(C)cccc1C CCC(CC)(CC)C(=O)NCC1CC(C)CCN1C(=O)CS(C)(=O)=O c1(OC)cccc(C)c1C(N1CCC(c2ccccc2)(NC(=O)COC(C)C)C1)=O N1(C(Cc2c(SC)cccc2)=O)CC(C)CCC1CNC(=O)CNS(N)(=O)=O c1(NC(C2(C)CCN2C(c2ccc(Cl)cc2)=O)=O)ncc([N+](=O)[O-])cc1O Cc1cnn2cc(C(=O)NCCC(C)(C)C(=O)OCC(C)C)cnc12 C1(C(=O)NCc2cc(CC)no2)CC2(CC2)CN1NC(=O)CC1CCCOCC1 C(C)(C)(CCCF)NC(C(CN(C)C)NC(=O)CC1(CN(C)C)CCC1)=O c1(C(N(CCC)CCNC(c2sccc2Cl)=O)=O)ccccc1OCC(C)C c1(C(=O)NC(CC)CN(C(=O)C2=C(Cl)CC2)C)cc(C2CCCCC2)n(C)c1C c1(N(C(CC2(C)CN(C(c3cc(COC)no3)=O)C2)=O)CC#N)ccc(C)cc1C C1(CNC(C=CCCC)=O)CCN(C(=O)C(F)(F)c2cnn(C)c2)CC1 CC1CC2CN(C(=O)CCOC3CCCC3)CC2N1C(c1cnc(C2CC2)s1)=O N1(C(c2c(OC)ccs2)=O)CC2CCC(CNC(=O)CC3CCCC3O)C2C1 Cc1nc(-c2ccc(Br)cc2)sc1C(C)NC(c1cc(C2CC2)ccn1)C C1(NC(c2c(C)coc2)=O)CC2(C1)CC(NC(c1ccn(C)n1)=O)C2 O=C(CS(=O)(=O)C1CC1)NCC1CCC(CNC(=O)CCOC2COC2)C1 c1(C(=O)NC2CCC(NC(c3c(C)nncc3)=O)C2)ccc2c(c1)C(=O)OCC2 C=CCCCCCC(=O)N1CCC(F)(CNC(C2(C(C)(C)C)CCCC2)=O)CC1 C=CCCCCC(=O)NC(C)(CNC(c1ccc(C(C)C)cn1)=O)CO C1(C(=O)NC2C(CNC(c3cccc(N)c3O)=O)C2)Cc2cc(F)cc(F)c2O1 Cc1nn(-c2ccc(F)cc2)c(C)c1CC(=O)NCC1CC(Cl)=NO1 C#CC1CCCCN1C(c1n[nH]cc1CNC(=O)C(CC)N(C)C)=O c1(CCc2n(CCCOC)c(N(c3ccccc3)C)nn2)cc(C)cc(C)c1 CC(=O)C(C)CC(C)C(=O)NC1CCCC(CC(=O)NCCN2CCOC2=O)C1 C=CC1CC1C(=O)NCC1(CC(=O)OCC)CC1 c1(C(N2C(CCNC(C(C)=C(CC)C)=O)COCC2)=O)cnc2n1C(C)CCC2 N1(C(C(F)=CC)=O)CCN(C(=O)Cc2sc(C)cc2C)C2CCCCC12 C1(C(=O)OCc2ccccn2)CCC(=O)N1C(=O)CCN1CCCCCC1 C(C)(C1OCCc2sccc21)N(C(C(C)(C)Nc1ccc(OC)cc1)=O)C C1(C(=O)NC(C)CC(=O)O)C2CN(C(=O)C(N3CC4CC4C3)C)CC12 c1(CC)ccoc1C(=O)NCC(C)CN(C)C(C1CC(OC(F)(F)F)C1)=O c1(C(=O)NCCOC2CN(C(C3CCC(C)C3)=O)C2)ccc(CC(C)(C)C)cc1 c1(-n2cc(C(C)O)nn2)cccc(F)c1C(=O)NNC(C1CC2CCC(C1)N2)=O C(=O)(CCCN=c1nccc[nH]1)NCCOCCNC(C(C(C)C)(C)O)=O n1(C(C)C)ncnc1C(=O)N(CC(C)NC(=O)CCC1CCC(=O)N1)C c1(-c2n(C)cnc2)ccc2nnc(C(=O)Nc3scc(O)c3C#N)n2c1 C(=O)(C1=CCC(C)(C)CC1)NC(C(=O)Nc1c(C)cc(Cl)cc1)Cn1ccnn1 N1(C(C=Cc2nc(C)sc2)=O)CCCCC(C2CN(C(=O)C3=NOCC3)C2)C1 C1(OC)CCCCC1C(=O)N(C)CCN(C(=O)C(F)(F)c1cccnc1)C c1(C(=O)NC(CNC(C2C(C=C(C)C)C2(C)C)=O)(C)C)ccc(S(C)(=O)=O)s1 C1(COC2CN(C(CC(=C)C)=O)C2)CCN(C(=O)CN2CCCC(CC)C2)CC1 O=C1COc2ccc(S(=O)(=O)Oc3cnn(N4CCOCC4)c3)cc2N1 Cc1ccc2c(c1)CCN2C(C1CCC(F)CN1C)=O N1(C(C2C(CC)CCCC2)=O)CC(CNC(=O)C(C)(C)C(C)C)C2(CCC2)C1 Cc1ccc(C(=O)NC(C)C(C(C)C)NC(=O)CC(C)(C)C2CC2)nc1C c1(C(=O)NCC2(NC(CC(CC)OC)=O)CCCC2)cccn2cncc12 C1(C(=O)NC2(CCC)CC2)C=CCN1C(=O)C=CCN1CCOCC1 C(=O)(C1=C(C)CCC1)C(c1cnn(CCNCC2CC(SC)C2)c1)=O C1(CNC(c2cc(C)c(Cl)s2)c2nnnn2C(C)(C)C)CCCC(C)(C)C1 c1(C(=O)NCC(C(C)C)NC(C(NOC)=O)=O)cc(C)cc(F)c1 c1(C(=O)NC(CNC(C2OCCN(C)C2)=O)C2CC2)cc(F)cc(F)c1 c1(C(N(C2CCCN(C(=O)CN3CCCCCC3)C2)C)=O)ncccc1Cl N1(C(C(C)CN(C(=O)CN2CCCC2=O)C)=O)CCC(=O)N(C)CC1 C(=O)(C(C)SC(F)(F)F)N(C)CCN.C(=O)(C=C(C)C)N(CC)CC C12(CNC(CC=CC)=O)CCC(CNC(=O)CCCC3OCCO3)(CC1)CO2 C1(CC)CC(C(=O)NCCCc2ccsc2)CCN1C(=O)CC1CC(C)(C)CO1 C#Cc1cc(C(=O)NCC2CN(C(=O)CC=C=C)CC23CCC3)cc(N)c1 C(=O)(C(O)C(C)CC)NC1C(CNC(COc2c(C(C)=O)cccn2)=O)CCC1 Cc1ncc(C(=O)NCC2(NC(=O)C=CC(F)(F)F)CC2)n1C c1(C(N(CCCNC(C(C(CC)O)C)=O)C2CC2)=O)ncccc1N=[N+]=[N-] C(=O)(C1=C(Cl)CCOC1)N(C)CC1COCCN1C(c1cc(F)n[nH]1)=O C1(CNC(c2[nH]ccc2CO)=O)CC12CCC2.C12(CCC1)C(=O)N2.CCOC C(CC(C)N=c1nc(C2CC2)[nH]c2c(C)csc12)NC(C(C(C)C)NC(C)=O)=O Cc1cc(C)c(C(=O)Nc2ccc(CN3CC(C)C(C)C3C)cc2)cc1O N1(C(CN2CCN(C)CC2)=O)CCC2CC2(NC(=O)CC2CCC=CCC2)CC1 N1(Cc2ncn(C)c2)CCC2(CC1)CN(C(C1CC1F)=O)C2 N1(C(CCc2cc(C)no2)=O)CCN(C(C2CN(C)CCO2)=O)C(C)C1 N1(C(CCCC=C)=O)CCC2CCC12COC(c1c(I)c(OCC)nn1C)=O c1(CC(C(C)C)NC(=O)COC2(CO)CCCNC2)ccc(Cl)cc1 N1(C(=O)Cc2ccccc2NCc2cc(I)cc(I)c2O)Cc2ccccc2C1 CC(c1ccccc1Cl)=CC(=O)NC(C1CCCC1)CNC(=O)C#CC(C)C c1(SC)ccc(Cl)c(C(=O)OC2CCN(C(=O)C(C(C)=O)NC(C)=O)CC2)c1 CCCCC(CNC(=O)Cn1cnnc1O)NC(=O)CN(C)CC C=CCC(CC)C(=O)NC1(CO)CCN(C(=O)C(C)(C)c2cscc2Cl)CC1 N1(C(c2c(CC)[nH]nc2Cl)=O)CC2CCC(NC(=O)CNC(N)=O)(C2)C1 C1(C(=O)NCC2ON=C(CC)C2)CN(C(C2CC2(C)C(F)F)=O)C2(CCC2)C1 c1(C(N(C)CC2CCCN2C(=O)C(c2cncn2C)O)=O)cccc(F)c1 N1(c2n(CCOCC(=C)C)c(CS(N)(=O)=O)nn2)CCc2cc(COC)ccc21 C(CC(CNC(=O)C=C(Cl)Cl)NC(=O)C(C)OC(C)(C)C)OC C1(CNC(CC(=C=C)C)=O)CCC(C)(C)CN1C(=O)CCSc1nnnn1C c1(C(=O)NC(C(C)C)C(C)NC(c2c[nH]cc2C2CC2)=O)cc2sccc2n1C CC1CC(C(=O)NCC2CCC(NC(=O)COc3cccc(F)c3)CC2)C1(C)C Cc1noc(C)c1CNCCCn1nnc(N(CCC(=O)O)CC(F)(F)F)c1C c1(C(N2OCC(n3cc(COC)nn3)C2)=O)cnc2c(c1)c(C)nn2CCO c1(C(=O)NC2CC(NC(c3cnsn3)=O)C2)ccnc(I)c1F Cc1nc(C)c(-c2nnc(SC(c3ccccc3)C(=O)N(C)C)n2C)s1 N1(C(C2C(=O)NCCCC2)=O)CCCC12CCN(C(=O)COC1CC=CC1)C2 c1(C(=O)NCC2CN(C(C(CC)C)=O)CC2O)c(C)nn2cc[nH]c(=O)c12 c1(OC)c(CC(N2CCC(O)C(N(C)C(C3CC3C)=O)C2)=O)cccc1F N1(C(c2ccc(N)cc2O)=O)CCC(C2CC2)(NC(=O)CSCc2ncc[nH]2)C1 N1(C(C=Cc2c(OCCC)cccc2)=O)Cc2[nH]nc(C(=O)O)c2C1 C#CCCCC(C)C(=O)NCC1CN(C(=O)CN2CCCCCC2)C1 c1(CC)cc(C(=O)NCCNC2CC(=O)NC2=O)c(C)o1 C1(OCC)CCCN(C(=O)C(C(C)O)NC(C2(OC)CCSC2)=O)C1 N1(C(c2cccc(COC)c2)=O)CC2CCCC2(NC(=O)CCF)C1 Nc1cnc(C(=O)OCc2cccc(C(F)(F)F)n2)cn1 C1(NC(C2CC(F)C2)=O)CCCCN(C(=O)Cc2cccnc2O)CC1 c1(OC)ccc(SCCC(=O)NCC2CCCN(C(=O)CN(C)C)C2)cc1 C1(C(=O)NC(C(=O)NC(CC(=O)OCC)C2CC2)C)C2CCCCC12 N1(C(C(C)(CO)OC)=O)CCOC(C)(CNC(=O)CSC)C1 C1(CC)SC(C)CC(N2CCC(O)C(C(N3CC4CCC(C3)O4)=O)C2)C1C C1(C(=O)NCCS(CC)=O)CCCCCN1C(c1n[nH]c2c1COC2)=O C1(C(N2C(CNC(c3ccnc(C)c3N)=O)CC2)=O)Cc2ccc(F)cc2O1 Cc1c(Cl)nc[nH]c1=NCC(O)CNC(c1cc2cccnc2s1)=O CC1(C)OC(=O)CC1C(=O)NCCN(C(=O)CC1CCC1(F)F)C1CC1 N1(C(C2OCCC(C)C2)=O)CCC(CNC(c2ccc(O)c(N)n2)=O)CC1C Cc1nn(C)c2c(NCc3cnns3)nc(N3CCC(C4CC4(F)F)CC3)nc12 C1(C(=O)NCC(C)(Cn2cccn2)NC(C=CCCC)=O)CN(C)CC(C)O1 c1(C(N2C(CNC(=O)C=Cc3cnc[nH]3)C=CC2)=O)cnc2c(c1)CCCC2 N1(C(c2c(C)n[nH]c2)=O)CCOC(CN(C(=O)C(F)CC2CCCCC2)C)C1 C12(C(N(CC(=O)NC(C)(C)C)C)=O)CC(CO)(CN1C(C1CC3(CC3)C1)=O)C2 c1(C(N2CCC(NC(C3(OC)CC3)=O)CC2C2CC2)=O)ccc2c(n1)CCC2=O c1(OC)cc(OC)nc(CNC(C2CCC(C)(C)OC2)=O)n1 CN(C1CCc2ccc(Cl)cc21)C(=O)C(=O)NCCc1ccc2c(c1O)OCO2 C1(N(C)C(c2coc(OCC(F)(F)F)n2)=O)CCN(C(c2ccnn2C)=O)CC1F c1(OCCCC(=O)NCC(CCNC(C(C)(C)NC(N)=O)=O)O)ccc(Cl)cc1 N1(C(c2cn(CCNC(CSCC#C)=O)nc2)=O)Cc2ccc(O)cc2C1 c1(SC)ncc(CNC(c2nnnn2CC2CC2)CC2CCCC2)s1 c1(N(CCC)C)cc(NCC(C)(C)COC)nc(C(C)C)n1 c1(C(N(CC(C)(C)NC(C2CC(C)OCC2)=O)C)=O)cnc(O)cc1C(F)(F)F C1(NC(c2nn(C)c(F)c2)=O)CC2CN(C(c3cnn4cc[nH]c34)=O)CC12 c1(C(=O)NCCCC(=O)NCc2nc(C)sc2C)ccc(C)c(C#N)c1 c1(CC)ncc(C(=O)NC(C2CCC2)C)[nH]1 C1(CC(=O)NCC2CN(C(C)C)C2)CCCCN(C(=O)CC(C)O)C1 N1(C(C(CC)F)=O)CCC2(CCC2)C(CNC(c2cccc3cccnc23)=O)C1 c1(C(=O)NCc2c(CNC(CC(=C=C)C)=O)nccc2)nnn2c1C(=O)NCC2 c1(C(=O)NCC(C)NC(C2CCCC23CCC3)=O)cccc(C(N)=O)c1F c1(OC)ccc(C=CC(=O)NC2(CF)CCN(C(C3(C#N)CC3)=O)C2)cc1F c1(OC)cccc2c(N(CCCNC(C3CCCN(C)C3)=O)C)ncnc12 N1(C(C(CC)SC)=O)CC2CC1CN2C(=O)C(c1cncn1C)N(C)C CC1CCN(C(c2cn3c(n2)SCC3)=O)CC1N(C(=O)Cc1cccc(O)c1)C CC1CCC(C)(C(=O)N(CC(C)N(C(=O)Cn2ncnn2)C)C)CC1 C(=O)(CC1=CCN(C(c2cc(C(C)=O)[nH]n2)=O)CC1)NC(C#C)(CC)CC CC(CCS(C)=O)N(C(=O)C(=O)C1CC1)C CCC(C(=O)NC(C)CCCNC(C1(Br)CC1)=O)Sc1ccccc1 c1(C(N(CC(CC)NC(=O)Cn2nnc(C)n2)C)=O)coc(-c2ccccn2)n1 C1(C(=O)NC(C2CCCC2)CNC(C2CN(C3CCOCC3)C2)=O)COC(=O)C1 C1(NC(c2cc(CO)[nH]n2)=O)CN(C(=O)Cn2ncc(Br)n2)C2CC12 c1(CC)ccccc1-n1nnnc1C(C1(CC)CC(O)C1)NCc1ccoc1 S(=O)(=O)(c1cccc(Cl)c1)NCCC(=O)NCC(CNC(C(CC(C)C)C)=O)C C1(CNC(CCC#N)=O)CCCCC1NC(c1nn[nH]c1Cl)=O C=C1CCN(C(=O)C=CC(F)F)C(C(N2CCNC(=O)C2)=O)C1 c1(C(=O)NCCCCNC(C2C(C)(C(=O)OCC)C2)=O)cnc(C2CCC2)s1 O=C(C1=NOC2(CCOC2)C1)NC1CCN(C(c2ccc(F)c(C(F)F)c2)=O)C1 c1(NC(C(CCNC(CC(CC)C)=O)O)=O)cc(C)ccc1OC Cc1nsc(C)c1C(=O)NCC1(C)CCN(C(=O)Cc2cc(Cl)n(C)n2)C1 C(CN=c1[nH]c2cccc(Br)c2o1)C1CCN(C(CSCCCC)=O)CC1 C(=O)(CCCC(C)C)NCC1(CO)CCN(C(c2c(C)nc(C3CC3)o2)=O)C1 c1(CN2CC(C(=O)Nc3ncc(Br)s3)SCC2)c(O)cccc1Cl C1(CNCC(CC)(C)CC)(CO)COCCN1Cc1ccccc1 Cc1nc2cc(C(=O)NCCC3CCCNCC3)c(F)cc2[nH]1 c1(CN2C(C(N(C)CCc3ccccc3)=O)C=CC2)cc(F)c(O)cc1F CCCCC(C)C(=O)NCC1(NC(=O)CCC2OCCO2)CC(OC)C1 N1(C(C(=O)NCC)=O)CCCC(NC(c2oc(C(C)C)nc2C)=O)C(F)C1 Cc1c(C(N2CCC(CN(C)C(C3CCC(N(C)C)CC3)=O)C2)=O)cncc1N c1(C(N2CCC(C(=O)NC(c3cnccn3)C)C2)=O)cc(Cl)nc2n[nH]cc12 CC1CCC(CC(=O)NCCCCCCNC(=O)CCCN2CCCCC2)OC1 CC1CCN(C(=NCCC2(C)CC2(F)F)NCCF)C1 c1(CC)ccc(C(C)(C)C(=O)NCCCOCCN(C)C(C2CC2CC)=O)cc1 C1(N(C(C(C=C=C)C)=O)C)CCCN(C(=O)OC(C)(C)C)CC1 N1(C(=O)CC2(CO)CC2)CCN(C(=O)C2=COCCO2)C(C2CCC2)C1 c1(CCC(C)C)cc(C(=O)OCC(CN2CCN(CC)CC2)O)nn1CCO c1(OC)cccnc1C(=O)NC1CN(C(c2cc(C3CCCC3)no2)=O)C1 C1(CNC(c2ccc(F)cc2O)=O)CC2CCCC2N1C(=O)CCC1CC1(F)F O(NC(=O)C(O)CCCNC(C1(C#N)CCC1)=O)CC(CC)C c1(CC)cccc(C)c1C(=O)NCC1(F)CCCN(C(=O)C(C)n2cnnn2)C1 c1(C(=O)NCCN(C(=O)CC2CCCOC2)C2CC2)cnc2ccccc2n1 c1(C(=O)NCC(CNC(COCCC)=O)C)cc2cc(C(=O)OC)sc2s1 O=C1NCCc2ccc(C3CC34CC(NCCSc3ccc(Cl)cc3)C4)cc21 c1(OC)ncc(C(=O)NC(C)CCCNC(C2CCNC2=O)=O)cn1 N(C(=NCCCF)NC1CCS(=O)(=O)C1)CCc1c(OCCC)nccc1 C1(CNC(C(CC=C)CC)=O)CCC12CCN(C(=O)C(C)(C)CC)CC2 C(=O)(CC(F)(F)C(F)(F)F)N1CCC(Cn2cc(CCOC(C)=O)nn2)C1 N1(C(C2CC(NC(c3cccc(I)c3)=O)C2)=O)CCC12CCCCC2 c1(OC)csc(C(=O)NCC2CN(C(=O)CCOCC(F)F)CC2C)c1OC c1(OC)cc(Br)c(F)cc1C(c1nnnn1C)NCC(=O)Nc1ccc(F)cc1 c1(NC(CC2CC3(CN(C(C(C(C)(C)C)O)=O)C3)C2)=O)cccc2ncsc12 N1(CC)CC(CNC(c2ccc(CNC(C3CCO3)=O)s2)=O)CC1=O c1(NC(C2CC(F)CN2C(C2CCCS2)=O)=O)nc(Br)cnc1Cl c1(C(=O)OCC)cc2c(s1)CCOC21CCN(N2CCCC(OC)C2C)CC1 C(CNC(=O)C(COC)N(C)C)(CC(C)C)NC(C1(CC#C)CCOC1)=O C(=O)(CCCCc1cnn[nH]1)N(C1CN(C(=O)C=C(Cl)Cl)C1)C c1(C(=O)NCC(C)NC(=O)Cc2cnc[nH]2)cccc2nc(O)n(C)c12 c1(CC)[nH]nc(C(=O)NC2CC(CCNC(=O)COCCc3cccs3)C2)c1Cl C(C(F)(F)C(=O)N1CCC(F)(CNC(=O)CN2CCCC(N(C)C)C2)C1)N(C)C C(C(C)(C(C)C)NC(C1CCCCC1O)=O)NC(C(C)OCCOC)=O C(c1cnn(C)c1)=CC(=O)N(C1CCN(C(CCc2onc(CC)n2)=O)C1)C C(=O)(C(CNC(c1ccc(O)nc1)=O)C(C)(C)C)NC(c1cncnc1)C c1(C(N2CCC(NC(c3c(C)ccnc3)=O)CC2C)=O)cc2c(nn1)OCCS2 c1(CC)noc(C)c1CNC(C12CC(n3cc(COCC(N)=O)nn3)C1C2)=O C1(NC(c2ccc(CC)nc2)=O)CC2CCC1C(NC(C1(N(C)C)CCC1)=O)C2 C(=O)(CC(=O)NCC(C)CN(C(=O)C(C)COCCOC)C)NCC#C N1(C(C2CC(O)(CNC(c3sccc3Cl)=O)C2)=O)C2CCC1CC(O)C2 N1(C(c2c(-c3ccc(C)cc3I)nccc2)=O)CCc2nc(C)sc2C1 c1(C(N2C(CCCNC(C(COC)(F)F)=O)CCC2)=O)cccc(C(N)=O)c1F C=C(C)CCCC(=O)N1CCN(C2CCN(C(=O)C(C)C3CCCO3)C2)CC1 N1(C(C(C=CCCC)O)=O)CCC2(CCCN(C(c3cn(CC)nn3)=O)C2)C1 C(=O)(C(CCC1CC1)NC(c1csc(CO)n1)=O)NC(C1CC(F)(F)C1)C O=C(CCCCCc1ccc(F)cc1)NC1CC(NC(=O)Cc2ccccn2)C1 c1(CCC)ccc(Cl)cc1-c1nc(-c2ccn(C)n2)nn1CC1CCCOC1 C1(C(N(CC(=O)N(CC(CC)OC)C)C)=O)CCC1(F)F C1(NC(C2CCCCS2(=O)=O)=O)CC2CN(C(C3CCC4CC4C3)=O)CC12 CCCCCC(C)(C)C(=O)NCCC1=CCN(C(c2cccc(C)c2C)=O)CC1 C1(NC(C(NOC)=O)=O)CC2CCC1C(NC(C1CC3COCC3C1)=O)C2 C=CCCC(CC(C)C)C(=O)N1CCC(NC(=O)CC2OCCC2(C)C)C1C N1(C(C2N(C(CCSCC)=O)CC(=O)C2)=O)CCC(O)CC(C)(C)C1 Cc1ccc(C(N2CCCC(C)(NC(=O)C(C)C#N)C2)=O)cc1Br C1(CNC(C2C(C)=C2)=O)CN(C(c2occ3c2CCC3)=O)CCC1(C)C c1(C(=O)NCCCNC(C(C(CC)CC)OC)=O)c(O)nnc2c1CCC2 C1(C(=O)N(C2CCC(O)CC2)C)(COC)C=CCN1C(c1csc(C)n1)=O c1(SC)nn(C)cc1C(=O)N(C)CC1CCN(C(C2OCCO2)=O)CC1 N1(C(C)=O)CCc2ccc(NC(=O)C(C)Oc3ccc(CO)cc3)cc21 C1(OC(C(c2cc(C)no2)(C)C)=O)CCC(F)(F)C1 Cc1cc(=NC(=O)C(=O)NCC(C2CCCC2)NC(C2CC=CCO2)=O)[nH]o1 C1(C(=O)NC(C)CC(C)NC(=O)Cn2cc(N)cn2)(CC)CCNC1=O C(=O)(C(C)(C)C(=O)N1CC(NC(=O)C=CCN2CCC2)C(CO)C1)OCC N1(C(C)=O)CCN(C(=O)NCc2ccc(N3CCCC(O)C3)cc2)C(C)C1 c1(NC(C2CCCN2C(c2cc(Cl)sc2Cl)=O)=O)c(Cl)ccc2cccnc12 C1(C(=O)NCC2CCC(CNC(c3cc(C)oc3C)=O)CC2)CC2CC2CC1C Cc1ccc(C)c(SCC(=O)NCCCCN(C)C(c2ccc(CSC)o2)=O)c1 c1(C(C)=O)cn(C)nc1C(=O)NC(C)CC(C)NC(C1CCC(=O)N1)=O O(NC(=O)C(C)C(C)NC(c1coc(CC)n1)=O)CC C(C)(C)(C(C)CC(=O)NC1CN(C)CC1(F)F)NC(CCSCC)=O c1(CC(=O)NC2CC(CCNC(c3ccc(OC)s3)=O)C2)csc2nccn12 Cn1cnc(C(=O)NCC23CC(NC(C4CCCN4C=O)=O)(CO2)C3)cc1=O C=CCC(C(=O)N(CCCCN(C)C(C1(CN(C)C)CCCC1)=O)C)OC N1(C(C(n2ncc(C)c2)C)=O)CC2CCOC2(CNC(C2(N(C)C)CC2)=O)C1 N1(C(CSCC)=O)CCN(C(=O)C(N2CCCC2CC)=O)CC1c1ccccc1 Cc1noc2nc(C3CC3)cc(C(N3CCc4ccnc(O)c4C3)=O)c12 C(=O)(C1CCc2ccccc21)NCC(C)N(C(=O)Cn1nnc(=N)[nH]1)C n1(CC)ccc(C(=O)NC23CC2CN(C(C2C(Cl)(Cl)C24CC4)=O)C3)cc1=O C(CCCC(=O)N=S(=O)(C(C)C)C1CCNC1)Oc1cccc(OC)c1 c1(C(=O)NCC23CC(NC(CC4C(C)=NOC4=O)=O)(C2)C3)c(C)nc(C)nc1C C1(CN(C(CC2(COC)CCCC2)=O)C)CCN(C(=O)C(C)N(C)C)CC1 CC(C)C(C)(C)C(=O)NCCN(C)C(C12C3C4C5C3C1C5C24)=O c1(C(N(CC(O)CN(C)C(C2(C(F)(F)F)CCCC2)=O)C)=O)cc(C#N)ccn1 C(=O)(C(C)(C)C(F)F)NCC(CN(C(C(c1ccc(C)cc1)C)=O)C)C c1(C(=O)NCC2C(CNC(COC(C)(C)C)=O)C2)c[nH]nc1-n1cnnn1 C1(C(=O)NC(c2cn(C(C)C(=O)NC3CC3)nn2)CCC)CCCS1(=O)=O C(C(O)CN=c1[nH]nc(C(F)F)o1)NC(c1cn(CCOC)nc1C)=O C1(C(=O)NCC=CC(=O)N(CC(C)O)CC(C)O)CCCC(F)C1 c1(C(=O)NC2CCCN(C(c3n(CC)ccc3)=O)C2C)cccc2c[nH]nc12 N1(C2CCN(C(c3c(SC)ccs3)=O)C2)CCC(NC(=O)C2=CCC2)CC1 CN1N=CC(CC(=O)N(C2CCCC2)Cc2ccccc2)C1=O C1(NC(C2CCC(N(C)C)C2)=O)CC(CO)N(C(=O)CCC2CCC2)C1 C#CCCCCC(=O)N1CC(=O)NCC1C(N1CCC(O)(C#C)C1)=O C1(C)(NC(C(C)OC2CCCC2)=O)CCN(C(=O)COCC2CCCCO2)CC1 C1(NC(c2nc(C3CC3)cs2)=O)CN(C(C2CCCCCC2)=O)C2CCCCC12 c1(CNC(=O)NC2(C3CCCC3)CC2)c(Cl)oc2ccccc12 N1(C(C2(C#C)CN(C(=O)C(C)=C3CCCC3)C2)=O)CC(C)C(C)C1C C12(CC(=O)NC(C3CCN(C(C=CCN(C)CC)=O)C3)C)CCC(CC1)C2(C)C Cc1ccc(C=CC(N2CCC(C(C)NC(c3cc(O)nc(Cl)c3)=O)C2)=O)cn1 c1(N2C(COC)CCC2)nnc(-c2ccccc2C)n1Cc1ccc(CSC)o1 C(=O)(CC(F)(F)F)NCC(=O)N(CCNC(C1C(C)CC1)=O)CC1CC1 N1(C(C(C)(C)c2cccs2)=O)CC2CC(O)C1C2NC(C1CCCS1)=O C(=O)(CN(C(=O)CN(C)CCOCCOC)C)N(CCC)CCC N1(C(C(=O)NC(C)C)=O)CCN(C(c2ccncn2)=O)C(c2cccc(F)c2)C1 Cc1ccc(C(=O)NCCC2CN(C(=O)COC3(C)CCC3)CC(C)O2)c(Cl)c1 c1(C(=O)NCCOCCNC(c2c(C)ccnc2C)=O)sccc1S(N)(=O)=O N1(C(C(C)SCC)=O)CCN(C(=O)C(O)C2CCCC2)C(CCO)C1 CCCC(O)(CCC)CC(=O)N1CC(O)(C2(CNC(=O)CCNC(N)=O)CC2)C1 Cc1ccc2scc(C(=O)NC3CCN(C(=O)CCCC(C)(C)C)CC3F)c2c1 C1(F)(CNC(C2(CC)CC2(F)F)=O)CCCN(C(c2ncccc2O)=O)C1 c1(C(=O)NC(CN(C(C(C)O)=O)C)C)ccc(Sc2ccccc2Cl)cc1 C(=O)(C1CCSc2ccccc21)Nc1c(C#N)cc(Br)cn1 c1(C(c2nnnn2C(C)C)NC2(CC=C)CCC2)ccc(Cl)cc1F Cc1cc(CC(=O)NC2CC(=O)N(c3cnn(C)c3)C2)ccc1O C(C)(C)(CC(=O)N1CC(O)(CNC(=O)Cc2ccccc2C(C)C)C1)OC c1(OCC)cccc(C(=O)NC2CC(C#N)C2)c1F CCCC(C)(O)C(=O)NC1CCC(CNC(c2ccc(Cl)o2)=O)CC1 C12CN(CCN1c1nnc(C3CC4(CCCC4)C3)n1C)C2.c1(CC)ccccc1 c1(C(=O)NCC(CCOC)NC(c2ccc(C)o2)=O)ccc2c(c1)OCCC2 c1(OCC(C)(C)NC(C2CCC(CC)C2)=O)ccc(F)cc1 c1(CC(=O)Nc2cccc(CNC(C3CCC(F)(F)C3)=O)c2)cc(Br)ccc1O N1(C(=O)NC(C2(C)CCCO2)c2cccs2)CCC(Oc2ccccc2)CC1 C(N=c1[nH]c2cc(F)c(F)cc2s1)C1CCCCN(C(c2nc(CC)oc2)=O)C1 c1(C(N2C3CN(C(c4cc(I)ccc4F)=O)CC32)=O)cnc2ccccc2n1 c1(CC)n[nH]c(=NCN2C(=O)CCC(C(=O)NC3CCC3)C2)s1.OC Cc1ccc(CC(=O)NC2CN(C(C3CCC(C(N)=O)CC3)=O)CC2C)c(C)c1 C1(NCC(N)CC(F)(F)F)CCc2c(cnn2Cc2ccccc2)C1 N1(C(C(C(C)(C)C)n2cc(-c3c(C)cccn3)nn2)=O)CCOCC(C)(C)C1 CCC(C)C(C)C(=O)NC1CN(C(=O)CNS(=O)(=O)N(C)C)CCC1C c1(CC)ccc(C)c(C(N2CCC(C)(CCNC(C3CC(OC)C3)=O)C2)=O)c1 N1(C(n2cc(Br)cn2)C(=O)NC)CCCCC1c1cn(-c2ccccc2C)nn1 n12cc(cn1)C(=O)NCC2.n1(CCOC)cc(-c2csc(C)c2)nn1 c1(C(N(CCCN(C)C(c2cc(CO)n(C)n2)=O)C)=O)ccc2ccoc2c1 N1(C(c2ccsc2)=O)CC(C2CN(C(C3CCSC3)=O)C2)C1 c1(CC(=O)NC2CCC(F)(F)C2)cnc2n1CCOC2.n12cc(nn1)CNCC2 c1(CN2CCC(F)(C(N(C)CC3CCC3)=O)C2)cnc2[nH]ccc2c1 N1(C(C)=O)CCCCC1C(=O)N(C1CC1)CC12CCC(CO1)C2 C1(C(=O)NCc2cn(CC(=O)NC3CC(CC(N)=O)C3)nc2)C2CC3C(C2)C13 CC1CCCC(CC(=O)NC(CN2CCC2)C(C)(C)C)O1 N1(C(CCOC)=O)C(CNC(=O)C(C)(C)OC(C)C)CC2CC12 c1(C(=O)NCCC2CCCN(C(CC(COC)C)=O)C2)cn2cccnc2n1 n1(C(C(=O)NCCOCCNC(Cc2cnc(C)[nH]2)=O)C)cnc2ccccc12 c1(C(=O)NC2CCC(NC(C3N(C)CCCC3)=O)CC2)ccc(O)c(CO)c1 N1(C(C(C(C=C)C)C)=O)CC2(CCN(C(=O)CCCc3cccc(Cl)c3)CC2)C1 C1(NC(CC2(C=C)CC2)=O)CCC(O)CN(C(=O)C(F)C(F)(F)F)C1 N1(C(C2C(=C)CC2)=O)CCN(C(c2cccc3cncn23)=O)C2(CC2)C1 N1(C(CC(C)CF)=O)CC(NC(c2cncc(C(F)(F)F)c2)=O)CC(F)C1 c1(N2CC(C(C)NC(c3cncc(Cl)c3)=O)C2)ncnc2ccc([N+](=O)[O-])cc12 N1(C(c2cnccc2Cl)=O)CCC(N=c2[nH]c3cc(F)cc(F)c3o2)C1 N1(C(CCc2ccc(OC)nc2)=O)CC2CCC1CN2C(=O)C(C)NC(N)=O c1(C(N2CC3C(CN(C(C4C(=C)CC4)=O)C)C3C2)=O)csc2c(OC)cccc12 C1(CC(=O)NCC2(F)CC(CNC(c3cc(CC4CC4)on3)=O)C2)CCC2CC12 c1(CC)cc2c(N3CCN(C(C4CCC(F)(F)C4)=O)CC3C)ncnc2s1 c1(-c2onc(C)n2)ccc(C(=O)NC(C)C(C)NC(C2(O)CC2)=O)cc1 C1(CNC(C=CC)=O)CN(C(c2nnn3c2COCC3)=O)CCC12CCOC2 C(=O)(CS(=O)CCC(F)(F)F)NC(CNC(C=CC)=O)(C)CC CC(O)(CC(=O)N1CCCC(F)(CNC(=O)Cc2ncc(Cl)s2)C1)C(F)(F)F C1(CCC(=O)NCC2C(NC(c3cc(C)sn3)=O)C2)CCCN(C)C1 C(=O)(C(F)(F)CCn1cccn1)N1CC2C(CNC(C(C)(C)SC)=O)(C2)C1 c1(CC)nc(C(=O)NC23CC(C(N4CCC(OCCN(C)C)C4)=O)(C2)C3)c(C)o1 c1(NC(C(c2cnn[nH]2)N(CCCCC)C)=O)ccc2c(c1)OCCO2 C(C)(CNC(c1n[nH]cc1Br)=O)(CO)NC(CC1CN(C)C1)=O N1(C(COCCOCC#C)=O)CCC(C(=O)NCC2C=CCCC2)C(C)(C)C1 C12(NC(c3nc(C)c(C)s3)=O)CCN(C(=O)CC(C)(C)O)CC1C2 N1(C(=O)NC(c2ccc(SC(F)(F)F)cc2)C)CCN(C)C(C)C1C N1(C(c2ccnc(C)n2)=O)CC2CCC2(CC(N2CCC(OCC(N)=O)C2)=O)C1 Cc1c(C(=O)NC2CN(C(=O)CN3CC(=O)NC3=O)CC23CC3)sc2nccn12 Cc1oc(CO)cc1C(=O)NCC(C)(F)CNC(C1(C)CCCC1C)=O N1(C(Cc2ncc(CC)[nH]2)=O)CCC2C(CCN2C(=O)C(C)NS(C)(=O)=O)C1 C(CCCCCC(=O)N1CC(CNC(=O)C(=Cc2cccnc2)F)C(C)C1)SC c1(C(C)C)ccc(C(=O)N(CC(C)CN(C(C2CCOC2)=O)C2CC2)C)o1 C1(NC(C(C)C(F)(F)F)=O)CCN(C(=O)CC2CNC(=O)O2)CCC1CO C1(C(=O)NCCOC2CCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)C2)Cc2cscc2C1 c1(CC(=O)NCC(C)NC(C2(F)CCOC2)=O)ccc(C(N)=O)nc1 N12CC3CC(CC3C1)C2.c1(C(=O)NCc2ccccc2C(=O)O)cnccc1F C1(C(=O)OC)CCc2sc(NC(N3CCC(N4CCCC4)C3)=O)nc2C1 c1(CC(=O)NC(C)C(C)NC(=O)OC(C)(C)C)nc(CNC(=O)CCF)no1 CC(CN=c1ccc([N+](=O)[O-])c[nH]1)N(C(=O)Cn1ncn(C)c1=O)C Cc1cc(C(N2CCCN(C3CC3)CC2)C(=O)NC(C)C)c2c(c1)CCC2 C=C(C)C(O)CC(=O)NCC(C1CC1)NC(=O)C(C)SCCCC c1(C(=O)NC2C(NC(C(C)(C)n3cnnn3)=O)CC2)cnc2c[nH]nc2c1 N1(C(C2C(COC)C2)=O)CCCC(C(=O)NCCc2ccc(C)s2)C1 N1(C(C(=O)NCC)=O)CC2CC2(NC(=O)CCC2CC(C)(C)CO2)C1 C#Cc1ccc(C(=O)NCC(C)N(C)C(c2cnn(C3CCC3)c2C)=O)nc1 C1(NC(c2cscc2F)=O)CCN(C(C2CCC(F)CC2)=O)C1C1CC1 c1(C(C)=O)cnc(Cl)[nH]c1=NC1CCCC(NC(c2cnc(C)o2)=O)C1 C1(C(=O)NCC2C(C)CN(C(C34CCC(C)(CO3)C4)=O)C2)CNC(=O)CC1(C)C Cc1cccc(NCCC(N2CC(F)CC2CN(C2CN(C)CCO2)C)=O)c1 C1(NC(C(c2cccs2)NC(CCC=CCC=C)=O)=O)CNC(=O)C12CC2 C1(CSC)CCC(NC(=O)C(C2(O)CCC2)N(C(=O)CCNCCC#N)C)CC1 C(=O)(CCCCC(=O)NC)NCC1(NC(CCc2nnc(C(C)C)o2)=O)CCC1 N1(C(C(c2ccccc2Cl)C)=O)CC(N(C(=O)CCCC2CCC2)C)C(O)C1 C1(CC(=O)NCC(CNC(C(c2cccnc2)OC)=O)C)CCCC(F)(F)C1 CCCCC(C(=O)N1CCC(CCC(=O)NCCCn2ccnc2C)C1)N(C)C CCC(C)CC(=O)NCC1CCCN1C(=O)C(C#N)=CC(C)C N12CCC(CC1)C2.C1(CC(C)O)CCCN1C(=O)C(n1cc(C(C)(C)C)nn1)C CCC(C(C)(F)F)NC(=O)COC1CN(C(=O)CC(F)(F)F)C1 c1(C(=O)NCC(C)C)cccc2c1CCCN2C(=O)Cc1ccccc1 C#CCC(C)(CC)C(=O)NCCC1CC(NC(C2(C#N)CCSCC2)=O)C1 c1(C(=O)NC(C(=O)OC)(C)C)ccc(OC(F)(F)F)c(-c2ccccc2F)c1 Cc1ccc(N2CCC(C(N3CC4C(NC(=O)CC(C)(C)C)C4C3)=O)C2=O)cc1 N1(C(COCCC)=O)CC2CCCC(NC(=O)C(N3CCC(O)CC3)C)(C2)C1 c1(C(C)(C)NC(c2ccc(OC)cc2)=O)ccc(-c2nn[nH]n2)c(O)n1 C(c1cn(C)cn1)=CC(=O)NC1C(NC(c2ccc(C(C)=O)o2)=O)CC1 C(=O)(C(C)(O)C(F)(F)F)NCCCC(C)NC(CCc1nnc(C(C)C)o1)=O Cc1nc(NCCN(C(c2ccc(C(N)=O)o2)=O)C2CC2)c2cnn(C)c2n1 Cc1nccc(C(N2CC(C3CC3)(C(N3CCCC3CC(N)=O)=O)C2)=O)c1N c1(CC)oc(C(N2CCCC(CNC(C3CCCC(CF)C3)=O)C2)=O)cc1C c1(C(=O)OC)nccc(NCc2ccc(CNC(=O)CCc3ccoc3)cc2)n1 C1(NC2CCCN(CC(C)(C)C)C2=O)CC2CCC1N(S(=O)(=O)CC1CCC1)C2 N1(C2CCC(NC(CCCOCC)=O)C2)CCN(C(c2cnc(OC)s2)=O)CC1 c1(C(N(CC(=O)NCC2CCN(C(N)=O)C2)CCOC)=O)sccc1C#N C#CCCCCC(=O)Nc1cccc(CC(=O)NCCCN2CCC(O)C2)c1 c1(C(C(=O)N(C(C)CO)CC)C)cccc(Br)c1 N(C(=NCCC1OCCC1(C)C)NCC1CCOC1)Cc1c(Br)cn(CC)n1 C1(OC)CCC(C(=O)NCC2(OC)CCN(C(=O)CCn3ccnc3C)C2)CC1 Cc1ncc(C(N2CCC(O)(CN(C)C(C3CCC(=O)N3C)=O)C2)=O)cc1N N1(C(CC2CCC(C)C2)=O)CCOCC(CNC(C23CC(CN2C2CC2)C3)=O)C1 C1(OC)(CNC(=O)C(C2CCCCC2)NC(=O)C(CO)N(C)C)CCCCC1 C1(C(N(CCC(C)NC(=O)CCC(F)(F)F)C)=O)CCCC(C)(C)C1 c1(C(N(CCN(C(=O)CCNC(=O)CO)C(C)C)C)=O)c[nH]c(Br)c1 C1(C(=O)OC)COC2(C1)CN(C(=O)C(c1ccccc1)OCC1CCCC1)C2 Cc1ccc([N+](=O)[O-])c(C(N2CCC(NC(c3ccc(Cl)s3)=O)C2)=O)c1 N1(C(CC=C(C)C)=O)CCCC(n2cc(CNC(C3C4CNC(=O)C34)=O)nn2)C1 N1(C(c2cnn(CCC)c2Cl)=O)CCC(NC(=O)CC2CC=CCN2C)CC1C C1(O)(C(=O)NC2CCCC(NC(c3ccsc3Cl)=O)CC2)CC2(CCOCC2)C1 N1(C(C(C(C)OC)NC(C2CNC(=O)O2)=O)=O)CC2CCN(C)C2C1 C1(C(=O)NCC2N(C(C(C)(C)NC(=O)C(F)(F)F)=O)CCC2)CCC(C#N)C1 Cc1ccc(OCC(=O)NCC(C)CN(C)C(c2ccc(O)c(N)c2)=O)c(C)c1 C1(NC(=O)Nc2cccc(C(N)CO)c2)CCn2nnnc2C1 C1(NC(C(CC)=CC)=O)CN(C(c2cnn(CCO)c2N)=O)CC2(CCC2)C1 N1(C(C2(NC(c3cc(C)on3)=O)CCCC2C)=O)CC2CC(C)C2C1 C1(O)(CC(N2C(C(CNC(Cc3c(C)ccs3)=O)(C)C)CCC2)=O)CCCCC1 C(=O)(CCCN=[N+]=[N-])N1CCC(O)(CNC(C2CC(C)(F)C2)=O)C1 C1(c2n(C)ncc2)CN(C(=O)CCS(C)=O)CC1NC(c1cnc(C2CC2)o1)=O Cc1ccc(Cl)c(O)c1C(=O)NCCNC(C1(C)C=CCCC1)=O Cc1cccc(S(=O)(=O)N2CCCC(C)(C(N3CCC4(CCCCC4)C3)=O)C2)c1 C(=O)(C(F)CC)NC1CC(CCC(N2CC(CC)C2)=O)C1 c1(CN=C(NCC2(COC)CCC2)NC2CCOCC2)cccc(C#N)c1F CC(C)(O)CC(=O)NCC1(F)CC(NC(c2ccnnc2NC2CC2(C)C)=O)C1 c1(C(N(CCNC(CC(C)C(C)(C)C)=O)CC2CC2)=O)cc2c(cn1)COCC2 N1(c2cc(NC(CCCN(CCO)CC)C)ncn2)CCC2(CCCCC2)C1 Cc1coc(C(C)C)c1C(=O)NC1CC(C)(NC(c2ncc(Br)cn2)=O)C1 N1(C(C2(C#C)CC2)=O)CCCC(C2(NC(=O)C(C)OCCN(C)C)CC2)C1 C(=O)(CC(C(F)F)c1ccccc1)NC(CC(C)NC(c1cnc[nH]1)=O)C c1(CNC(C(C)(C)CCC#N)c2n(CC)nnn2)ccc2ccccc2c1C C(C(C)C)(C(O)C(=O)NCCN(C(C1(c2ccccc2)CC(C)C1)=O)CC)OC c1(CCNC(C2CN(CCN3CCCC3)CCC2O)=O)ccc2c(c1)OCO2 c1(C(N2CC(CNC(c3cc(OC)n(C)n3)=O)C(O)C2)=O)nc2sccn2c1C C(=O)(C(C)(O)C(C)(C)C)NCC(C)NC(c1nccn2ccnc12)=O C1(NC(Cc2c(C)nco2)=O)CC2(C1)CC(NC(c1onc(C)c1C)=O)C2 CN1CC(NC(=O)CC2CCCN(C(c3ccn(C4CC4)n3)=O)C2)CC12CCC2 C1(C(N(CCC(=O)NCCCc2cc(C)no2)CC#C)=O)CC=C(C)CC1 N1(C(c2cc(OC)no2)=O)CCN(C(=O)CC2(CO)CC2)C(C)CC1C CC(C)C(CC(=O)NC1CC1)NC(=O)C#CC(C)(C)C.C1C(C)C(=O)N1 CC(C)C(O)CC(=O)NC1CN(C(c2scnc2C(C)(C)C)=O)CC1CC1CC1 C1(F)(CNC(C=CCOC)=O)CC(NC(=O)C=Cc2cocn2)C1 N1(C(C2CCCC(C(=O)OC)C2)=O)C(C)CC2CN(C(c3coc(C)n3)=O)CC12 C(CC(C)C(=O)N1CCC(C(C)C(=O)NC(CCOC)C(C)C)C1)=CC c1(CN(CC(F)(F)F)CC2CCCC2)ccc2cccc(Cl)c2n1 CC(N=c1[nH]c(=NCc2nnc(CO)s2)[nH]c2c(F)cc(F)cc12)c1csnn1 c1(NC(C2(NC(CC=C)=O)CC(CO)C2)=O)cnc(Cl)c(C)c1 c1(C(N2CCCC(NC(c3cc[nH]n3)=O)(CO)C2)=O)cc(Br)ccc1[N+](=O)[O-] N1(C(CCC(C)(C)F)=O)CCC2(CC1)CCN(C(=O)CN1CC3C=CC1C3)CC2 c1(-c2c(SC)cccc2)ccc(C#N)c(CC(=O)NC2CC2)c1 Nc1cccc(C(=O)NCCCNC(C2(Cc3cnn[nH]3)CCCC2)=O)c1F C(=O)(C1CCc2c[nH]nc21)N1CCC(C(=O)NC2(C#C)CC2)C(O)C1 C1(CC(=O)NC2COCCN(C(c3csc4cncn34)=O)C2)CC2(CCC2)CO1 C=CCC(C)(CC)C(=O)N1CSCC1C(N1CC2(C1)CC2(F)F)=O c1(CC)nc(N2CCCC(NC(c3c(C(F)(F)F)cnn3C)=O)CC2)[nH]c(=N)n1 c1(CNC(=O)CC2CC2)nnc2n1CCN(C(c1ccc3cccnc3n1)=O)C2 Cc1ccc(C(=O)NC(C)C(C)NC(c2cnn(C)c2C(F)F)=O)c(N)c1Cl N1(C(C2(C)CCN(C(c3c(C)cc(CC)o3)=O)C2)=O)CCC2(CCC(O)C2)C1 N1(C(C(CSC)(C)NC(=O)C#CC2CCC2)=O)CCc2nc[nH]c2C1 c1(NCC2CCC(CCCCC)O2)ccc(=N)[nH]n1 Cc1ccoc1C(=O)NCCC1CN(C(=O)C=CCN2CCCC2)C1 O=C(C#CC1CCOC1)NCC1(C(=O)NCC(F)C2CCC2)CC2(CC2)C1 N1(C(c2ccc(CCC)s2)=O)CCN(C(=O)CC2CC(CC)C2)C(CCOC)C1 C1(CC(=O)NC(CNC(c2cc(CCC)[nH]n2)=O)CC)CC(O)C12CCC2 N1(C(=O)Cc2ccc(Cl)cc2)CCCC2C1CCN2C(=O)Cc1ccncc1 N1(C(C=CC)=O)CC(C2CCCN(C(c3[nH]c(=N)sc3-c3ccccc3)=O)C2)C1 c1(N(C)CC2CCCN(C(=O)CCc3cscn3)C2)nnccc1C#N CC(C)C(O)CC(=O)N1CC(F)(F)CC1CNC(c1cnn(C(C)(C)C)c1)=O c1(SC)c(CNC(c2cnc(OCC(F)F)cn2)=O)cccc1C c1(CC)cccc(CC)c1CC(=O)NCC(C)CN(C)C(C12CC(F)(C1)C2)=O c1(C(c2nnnn2CCCC2CC2)NC(C(=O)NCC(C)C)C)ccnc(F)c1 c1(C(=O)NC2C(CCC)CCCC2)cccc2ccc(OCC)cc12 C1(C(N2CC(C(C)OC)C2)=O)C=CC(NC(=O)Cc2cn(C)cn2)C1 c1(C(N2C(CNC(C3CCO3)=O)CCC2)=O)ccc(Cl)c(C(F)(F)F)c1 C1(C2CCNCC2)(C(=O)NCC(C(C)C)=O)CCOCC1 C#CC(C)(C)C(=O)NCC1CCCCN1C(c1c(C)noc1CCC)=O c1(C(=O)NCC2N(C(C(C)n3ccnc3)=O)CCOC2)noc2ccc(Cl)cc12 c1(C(N(C(C2CCC2)C)C)C)cccc2ccccc12 C(CCCCC(=O)NC1CN(CC)CC1(C)C)NC(C=CC(CC)C)=O N1(C(c2c(CC)n[nH]c2)=O)CC(C)(C)CC1CC(N1C2C=CCC1CC2)=O c1(C(N2C3CCN(C(C(CCC)O)=O)CC3C2)=O)cc(=O)c2ccc(F)cc2o1 C1(C(=O)NCC=CCNC(c2c(C)nn(C(C)C)c2)=O)CN2CCN1C(C)C2 c1(CN(C(C2CC(OCC)C2)C(=O)NCC(F)F)C)cccc(Cl)c1 C(c1ccnn1C)=CC(=O)NC(=O)CC(N(N1CCCC1)C(C)CCC)=O CCC(C)(CC)NC(=O)C(C)CN(C(=O)C(F)F)C c1(OC)cc(CNC(C2CCC2CNC(=O)C=CC(C)(C)SC)=O)n(C)n1 C=CC(C)(O)CC(=O)N1CC(OCC(=O)NC2CCC3CCC23)C1 c1(CC(N2C3(CN(C(c4ccnnc4)=O)C3)CC2)=O)nc2ncccn2n1 C1(C)(C(=O)NC(CCCNC(C2C(C)=CCS2)=O)(C)C)CCCCNC1=O N1(C(c2c[nH]nc2C2CC2)=O)CCC2C(C1)CN2C(=O)C1=CCCCO1 CC(C)(CC(=O)N1CC(NC(C2CCO2)=O)C(C(F)F)C1)CC(F)F c1(C(c2nnnn2C2CCOCC2)NCC(CO)C2CC2)c(F)cc(Cl)cc1Cl c1(CC)cnccc1C(N1CC2C(C(N3CC(C)=C(C)C3)=O)C2C1)=O CC(CN(C)C)CC(=O)N(C1CCCN(C(=O)CC=Cc2ccccc2)C1)C N1(Cc2cc(C)sc2C)Cc2ccc(C(=O)Nc3cc(Br)cc(F)c3F)cc2C1 c1(CC(=O)NC(C2C(C(=O)NCC3(OC)CC3)C2)C)n[nH]c(C)n1 c1(C(C)=O)ccc(N(C)CCN(C)C(C23CCC(CC2)CC3)=O)c([N+](=O)[O-])c1 c1(NC(C=CC(CC)C)=O)nn(C)cc1N N1(C(CC(C=C)(C)O)=O)CC(C2CCCN(C(=O)CCc3cn(C)cn3)C2)C1 C(CC1=CCOCC1)NC(c1c(CNC(C(COC)(C)C)=O)ccs1)=O C1(C(=O)Nc2cccc(NC(CCCCC(N)=O)=O)c2)Cc2c[nH]cc2S1(=O)=O N1(C(C2C(CC)C2)=O)CCCC(C2CCN(C(c3ncn(C(C)C)n3)=O)CC2)C1 C1(NC(CN(CCC)C)=O)CC2(CCN(C(=O)C(C)CC(F)(F)F)CC2)C1 C1(C(C(=O)NCc2cn(CC)nn2)C)CN(C(=O)C(C(C)O)N(C)C)CCO1 Cc1ncc(C(=O)NCc2ccc(C(=O)NCCc3ncc[nH]3)s2)s1 C1(NC(c2n[nH]c(C)c2Cl)=O)CN(C(C23CC(F)(C2)C3)=O)CC1S(C)(=O)=O c1(C(=O)NC2(CO)CCN(C(c3n(C)ccn3)=O)C2)cnccc1N1CCCC1 N1(C(C2C(C)C2)=O)CC2OCCN(C(=O)C(O)Cc3cnc[nH]3)C2C1 C(=O)(C(CC)CC(F)F)NCC1C(NC(CC=C)=O)CCC1 c1(C(C(=O)NCCN(C(C2CCC(CC)C2)=O)CCOC)(F)F)cccc(C)c1 N1(C(C(CC)OC2CCCC2)=O)CCC(C2(NC(=O)C3=CCCOC3)CC2)CC1 C(C(=O)N1CCCC1(C)C(N1CCC(CN=[N+]=[N-])C1)=O)(C(C)(C)C)OC Cc1cc(N2CC(C(N)=O)C3(CC3)C2)nc(=NCCN(C)CCO)[nH]1 c1(CNC(C2C3CCC2(c2nccs2)C3)=O)cncc2cnccc12 C(=O)(C(F)CC(CC)CC)NC1CC2(C(C(N3C4CC(=C)C(C4)C3)=O)C2)C1 C1(NC(C(CNC(=O)OC(C)(C)C)C2CCOCC2)=O)CCC(F)CC1 C(=O)(C#CC1CCCO1)NC1(C)CCN(C(c2nc(OC)c(C)s2)=O)C1 N1(C(C=CC(C)(C)C)=O)CCCC(CCC(=O)N2CC(F)C2)C1 C1(C(=O)NCC(CNC(C(CCSC)NC=O)=O)F)CC(=O)N(C)C(=O)N1 Cc1ccc(NC(C2(C(F)(F)F)CCN(C(=O)CCC3CC3)C2)=O)c(Br)c1 C1(CN(C(CCN(CCC)C)=O)C)COCCN1C(=O)C=Cc1cscn1 C(=O)(C1=NOC(C)(C)C1)NC1C2(CCN(C(CCCNC(=O)OCC)=O)C2)C1 C1(NC(=O)CCCc2nccs2)(CO)CCN(C(=O)CC2CCC=CCC2)C1 C1(C)(NC(CN2CCC(C)CC2)=O)CCN(C(C2CC2C(F)(F)F)=O)CC1 C(=O)(C(CC)CCCCC)N1C(CC=C)(C(=O)NC2CC3(C2)CC3(F)F)CCC1 C(=O)(C(C)(F)C(C)(C)F)NC1C=CC(C(=O)NCc2[nH]nc(C(C)C)n2)C1 C1(C(=O)NC2C(NC(CCC(C)(C)F)=O)COC2)CSC(c2ccccc2)=N1 Cc1cn2cc(C(=O)OC3CCC(C)CC(C)(C)C3)nc2c(C)n1 C#Cc1cnn(C)c1C(=O)NCC1CC(NC(c2c(C(=O)OC)n[nH]c2C)=O)C1 CC1CCCC(C)N1CC=CCSC1CC2(CN(C(=O)OCC(C)(C)C)C2)C1 c1(CN2CC(NC(C(c3ccc(OC)cc3)C)=O)C(C)C2)cc(Cl)c(O)cc1F N=c1[nH]nc(CCC(=O)NC2CC(F)(CNC(=O)C(=C3CCCCC3)F)C2)s1 C1(NC(C2CCC3C(C2)C3(F)F)CCl)CCSC12CN(CC1CCCCCC1)C2 Cc1cc(=NCC2CC=CCC2)[nH]c(N2CCC(N3CCC3)CC2)n1 Cc1ncnc(C)c1CC(=O)NC1CCN(C(C2CC(C)(C)O2)=O)C1 c1(N(C)C)nc(C(N2CCC(CNC(C3CCCC(=O)O3)=O)C2)=O)cc(O)n1 C(=O)(N1OC2CC1C(O)C2O)C1C2(CC(NC(=O)CCc3nc[nH]n3)C2)C1 C(=O)(C(O)Cc1cnc[nH]1)N(CC(CN(C(=O)COC(F)F)C)O)C c1(C(=O)OC)cc(C(C(=O)NCc2nnn(C)n2)N(CC(C)C)C2CC2)c(C)o1 CC1CN(C(c2ccc(CF)cc2)=O)C(C)CN1C(=O)C(O)CC1CCCC1 CCCC(C)CC(=O)NCCC1CN(C(c2cccc(C)c2O)=O)CCO1 Cc1cc(Cl)cnc1S(=O)(=O)N1CCSC(c2ccccc2)C1 O=C(CC1OB(O)c2ccccc21)NC1(C2CCN(C(=O)COC(F)F)C2)CC1 C(=O)(C(F)(F)C(O)C(C)C)NCC1(C)CCCN(C(C2(CC#C)CCC2)=O)C1 c1(C(N2CC(CNC(C(C)C(C)(F)F)=O)CC2(C)C)=O)cccc2nc(O)oc12 c1(C(N2CC(NCCC(=O)NCc3ncc(C(=O)O)[nH]3)C2)=O)cccc2oncc12 C1(C(=O)NCC(C2CC2)NC(c2cc(C(=O)OC)on2)=O)CN(C)C(=O)N1 Cn1cc2cccc(CCN(c3nnnn3CCC3CC4OC3C3CC43)C)c2n1 Cc1ccc(C)c(C(=O)NC(C2CCCCN2C(C2CC3(C2)CC(C)C3)=O)C)c1 C1(C(N(C)CC2CCCN(C(c3c(OC)noc3C)=O)C2)=O)CCCCN1N=O N1(C(C(C)(C)c2cccnc2)=O)CC2(C1)CN(C(C1CC13CCCCC3)=O)C2 c1(-c2ccc(C(=O)Nc3c(C#N)cccc3)cc2)nc2ccccc2o1 CC1(C)C(CNC(c2nn(C(F)F)cc2Cl)=O)CCN1C(=O)CCC(N)=O N1(C(C(F)=CC)=O)CC2CCC(C1)N(C(c1ncc(C)cc1Br)=O)C2 C(=O)(C1CCCc2nc[nH]c21)NCCC(CNC(Cc1c(C)cccn1)=O)O N1(C(CS(=O)(=O)NC)=O)CC(C)N(C(=O)CCc2cscn2)CC1C c1(C(=O)NC2(C3CN(C(C(C)OCC=C)=O)C3)CC2)cncc2nnn(C)c12 C(C1C(C)C1(Cl)Cl)=CC(=O)N(C(CC)C1CCC1)C1CC1 CC1COC2(C1)CN(C(C1(NC(=O)OC(C)(C)C)CCOC1)=O)C2 c1(C(=O)NCC2(O)CCN(C(C3CN(C)C(=O)C3)=O)C2)cc2sc(Cl)cc2[nH]1 C(=O)(C(C)CCCC(C)C)NC1(C(=O)NCCc2cc(CC)no2)CCCC1C CCC(C(=O)N1CCOCC1CNC(c1ccccc1OC1CCC1)=O)C(C)C Cc1nc2cncc(C(N3CCC(CNC(=O)C4=CCSC4)C34CC4)=O)c2[nH]1 N1(C(CC(C)(F)F)=O)Cc2ccnn2CC(NC(=O)COCc2ccccn2)C1 C(CN=c1[nH]nc(-c2ccccc2)o1)C1(NC(N2CCOCC2)=O)CC1 C(=O)(C(C)(O)CCN(C)C)NCC(C(=O)N(CCCCO)CC)N(C)C c1(N2CC(COC(C)C)OCC2)nc2cc[nH]c2c(=NCCc2ccccn2)[nH]1 c1(C(=O)NCC2N(C(C3C(C=C)C3)=O)CC2)cc(C(C)C)nn1C c1(C(=O)NC2CC(C)(NC(CCC(C)C)=O)C2)cc2sccc2[nH]1 CCCCC(CC(=O)Nc1ccc(OC)cc1F)NC(=O)Cc1ccnc(C)c1 CC(CNC(C1CCCS1)=O)(C1CCC1)N.c1(CC(=O)NC2CC2)ccsc1 C(=O)(C(CCC(N)=O)N(C)C)N1CCCCC(NC(CCCOC)=O)C1 c1(C(=O)NCC2(C(C)(C)O)CN(C(CN(C)C)=O)C2)cc2cn[nH]c2cn1 C#CCC(C)(CC)C(=O)NCCC(C)(C)NC(c1nc(C)n(-c2nc[nH]n2)n1)=O Cc1cccc(C(=O)NC2C=CC(CNC(=O)Cc3csc(C)n3)C2)c1 N1(C(c2cc(C(C)C)no2)=O)CCN(C(=O)Cc2ccnc(O)c2)C2(CCC2)C1 c1(C(=O)OC)ccncc1C(=O)NCC1(NC(C2CC2(C)C(F)F)=O)CCC1 c1(C(=O)NCC(CNC(=O)CCc2ccncn2)F)c(O)cc(F)cc1F C1(NC(Cc2cc(C)on2)=O)CCN(C(=O)CCC(F)F)CC1C c1(OC)ccc(C)cc1C(N1CCCC(NC(c2ncc(F)cc2F)=O)CC1)=O C=CC1COCC1NC(=O)COC(C1CC2(CC2)C1)=O c1(-n2cc(CSC(C)C)nn2)ccc(CNC(C2CC2F)=O)cc1 N1(C(C(C)(C)O)=O)CCC2(CC(NC(c3ccnc(C(F)F)c3)=O)CO2)C1 c1(C(=O)NC(C)C(c2c(F)cccc2Cl)O)cc2n(n1)CCCCC2=O N1(C(C(CCC)NC(c2cc(OCC)no2)=O)=O)CCCC(C)(CC)CC1 CS(=O)(=O)c1coc(COC(C2CCN(CC(F)(F)F)CC2)=O)c1 Cn1ncnc1CCC(=O)NCC1CCN(C(=O)COC2CCOC2)C1 c1(C(=O)NCC(CC)(C)NC(=O)CC(F)(F)C(F)F)cccn2cc(C)nc12 Cc1cc2c(Br)ccc(C(=O)NC3(CF)CCN(C(=O)C(C)O)C3)c2o1 N1(C(c2c(CNC(CCC(=O)NC)=O)nnn2C)=O)CCOCC12CC2 N1(C(C2C(C(C)C)CCC2)=O)CCC2(CC1)CC(NC(=O)CC(C)C(F)F)CO2 CC1(CNC(=O)CCC2CCOC2)CCN(C(C2(C(F)(F)F)CCOCC2)=O)C1 C(=O)(C1CCCc2nn(C)cc21)N(CCNC(C=Cc1c(C)cccc1)=O)C N1(C(CSCc2ccc(C)cc2)=O)CC2(CC(NC(=O)CCC[N+](=O)[O-])CO2)C1 C1(NC(=O)CC2CCS(=O)(=O)C2)CN(C(=O)C2=CCCSC2)Cc2ccnn2C1 CC1CCC(NC(=O)CCCn2cncn2)CN1C(=O)C=CC(C)(C)C c1(OC)ccc2c(C(=O)NC34CC3CN(C(C3CCCCCC3)=O)C4)cnn2c1 C(C(O)CC(F)(F)F)NC(C1(F)CC(CNC(=O)C(O)CN2CCCC2)C1)=O C(C1=CCCOC1)N(C(CCN(C(CNC(C1C(C)C1)=O)=O)C)=O)C C1(CNC(C2CC2C2CCC2)=O)(CO)CCN(C(c2cccc(O)n2)=O)CC1 CC1CCN(C(c2cnc3n2CCC3)=O)CC1CNC(=O)Cc1cncc(O)c1 Cc1c(C(N2CCC(NC(=O)CSCC(=O)Nc3ccccc3)C2)=O)ncn1C C1(CNC(CC(C2CC2)NC(CCN(CCC)C)=O)=O)CCC2(CC1)CC2 N1(C(c2cc(C)nn2CC(F)F)=O)CC2CC(NC(c3sccc3C)=O)C2C1 Fc1ccc2c(c1)C1C(c3nc(CC(F)(F)F)nn3CC3CC4CCC3C4)C1C2 c1(N(C(C)=O)Cc2ccn(CC)n2)ccccc1OCc1ccncc1 c1(C(=O)NC(CC=C)CNC(C)=O)ccc(OC)c(S(C)(=O)=O)c1 CC1CCN(c2nnc(C(F)F)n2CC2CCCCO2)CC1F c1(C(=O)NC2(C)CN(C(C(COC)COC)=O)C2)cc2cc(Cl)ccc2nc1C c1(COC(COc2c(C)nn(C)c2C)=O)ccc(S(C)(=O)=O)nc1C c1(CC(N2CCCC(CCNC(C3CCOC3)=O)C2)=O)coc2cc(Cl)ccc12 C(=O)(CCC(C)(F)F)NC(CNC(CC1N(C(C)=O)CCCC1)=O)(C)CO c1(C(=O)NC23CC(NC(=O)CC(O)c4ccccc4)(C2)C3)ccc(F)cc1 C1(C(N2CCC(C(CC)CC)C2)=O)CC2CN(C(=O)C(C)(C)OC)CC2C1 N1(C(C(C(C)C)C#N)=O)CCC2(CCC2NC(c2ccc(CN(C)C)o2)=O)CC1 C(=O)(CCCC(F)(F)CO)N1CCCC(C)(NC(c2cc(C)n(C(C)C)n2)=O)C1 c1(CC(C(=O)N(CCOC)CCNC(=O)Cc2cnsc2)OC)ccc(C)cc1 CC1=C(C(=O)NC2CC3(C(N4CCC(CC(N)=O)C4)=O)COC2C3)CCCO1 c1(CCC)ncc(C(=O)NC2CC2NC(C2CC(O)C2)=O)s1 N1(C(CNC(=O)CC2CCCCC2)=O)CC2CCCC2(NC(=O)C2=CCCOC2)C1 c1(C(=O)NC2CCCN(C(C3(C)CC=C(C)CC3)=O)CC2)cc2c[nH]cnc-2n1 CCC(C)(C)C(=O)N(CC(C)(C)NC(=O)CCc1ccc(SC)cc1)C N1(C(CC2CC(OC)C2)=O)CC(NC(=O)C(C)CC#N)CC(O)C1 C(C)(C(C)CC)N(c1ccccc1)C(CSCC)=O C1(C(C)NC(=O)CCC2CNC(=O)N2)CCN(C(c2cn(C)cn2)=O)CC1 N1(C(C2CC(C)(C)N(C(c3ccc(C#N)cc3)=O)C2)=O)CCCN(C=O)CC1 c1(CC(N2CCC(N(C(C(CC)O)=O)C)C2)=O)coc2ccc3ccccc3c12 S(=O)(=O)(c1ccc(N(C)CCOC2CC2)nc1)N1C(CC(C)O)CCCC1 CCC(C)(CO)C(=O)NC1CCC(CC(N2CCOCC2CCO)=O)CC1 N1(C(C(C(C)NC(=O)Cn2ccnn2)C)=O)CC2(CCCCC2)C1 CC1CCCC1C(=O)NCc1c[nH]nc1C1CCN(C(=O)C(=O)NCC(F)F)C1 CC1CN(C(c2ccc(Br)o2)=O)CCC1NC(=O)C=CC(N)=O C(=O)(CC(C)C(=O)OC)N1C(CCC(N2C(C(=O)OC)CCC2C)=O)CCC1 C1(C(N2C(C#C)CC2)=O)CN(C)CCN1C(c1cscc1OC)=O N1(c2c(C(=O)OC)cc(C)cn2)CC2CN(C(=O)C(C)SC)CC2C1 C(=O)(NNC(=O)CN1CCCC1)C12CC(NC(=O)OC(C)(C)C)(C1)C2 C(CC1=CCCCC1)NC(C1C(CNC(Cn2cnc(=N)[nH]2)=O)CCCC1)=O N1(C(C2CC(C#N)C2)=O)CC=C(CCNC(=O)C=CC2CCC2)CC1 c1(CNC(C2(CC#C)CCCO2)=O)ccc2c(c1)CN(C(=O)C1=CCOC1)C2 Cn1c(Cl)c(C(c2nnnn2Cc2ccco2)NCC23CCC(CC2)OC3)sc1=O C1(C(=O)NCC2C(CNC(CCC=C(C)C)=O)C2(F)F)CC(C)(C)CO1 Cc1cc(C(=O)NCC2CCN(C(c3nocc3C)=O)CC2C)cc(C)n1 C1(OC)CN(C(=O)Cc2cscn2)C(C)(CNC(=O)Cn2cccc2)C1 N1(C(C2(CC)CCC2)=O)CC2C3CCC(C(NC(c4cc(C)no4)=O)C3)C2C1 C1(C(C(=O)NC)N(CC(C)S(C)(=O)=O)C)CCN(CC(C)(C)C)CC1 CCCC(C)(C)CC(=O)N1CCC2(CC2C(=O)NCc2ccc(F)cn2)C1 Clc1ccc(-c2csc(CSc3cccc(Cl)c3)n2)cc1 N1(C(C2CC(CC)C2)=O)CC2CC(C1)C(CO)C2NC(c1cccc(F)c1Cl)=O c1(CN(c2cc(NC(c3cc(O)n[nH]3)C)nc(C)n2)C)ccc(N=S(C)(C)=O)s1 CC1=C(C(=O)NC2(CF)CN(C(c3cc(C)nc(O)c3)=O)C2)CCO1 C1(C(=O)NCCCC(C)NC(C=C(CCC)C)=O)CCC(C(=O)OC)CC1 C1(C(=O)NC2C(C)CCN(C(c3c(CC)scn3)=O)C2)CCc2nc(C)cn2C1 C(C(C(C)C(C)C)NC(=O)CN1CCCC1=O)NC(CCc1c(C)cccn1)=O Cc1ccc(O)c(C(=O)NC(CNC(=O)CN2CCC(=O)NC2=O)C2CC2)n1 N1(C(C(CC)N(C)C)=O)CC2CC(C(=O)NCC3(SC)CCCC3)C(C2)C1 N1(C(CC(CC)(F)F)=O)CC2(C1)CN(C(c1cc3c(=O)[nH]ccn3n1)=O)CCO2 N1(C(C2CN(CC)C(=O)CC2)=O)CC2CCCN(C(c3cc(=O)n(C)o3)=O)C2C1 c1(C2(N(C)C(=O)NCC3(c4cc[nH]n4)CC3)CC2)ccc(F)c(F)c1Cl C1(NC(CCOc2cccc(C)c2)=O)CN(c2nccc(CO)n2)CC(C)(C)C1 C1(C(N2C(CCCC)C=CC2)=O)CCN(c2nc[nH]n2)CC1 C(=O)(C(C)(CC)CC)NCC(CC(=O)N(C(CC#C)C)C)O CC1C(C(=O)N2CC(NC(c3ccc(F)cc3F)=O)CC2(C)C)=NOC1C C1(CNC(CP(C)(C)=O)=O)CCC2(CO1)CC(NC(C1CC(O)C1)=O)C2 c1(C(N(CCCOC)CCNC(=O)CSC2CCCO2)=O)ccccc1C C(C(O)C(=O)NC(C1CCCCC1)C)NC(C(F)=C(C)C)=O C1(C)(C(=O)NCC2CCC(NC(C3C(C)CCCC3)=O)C2)CCC2(CC1)OCCO2 N1(C(c2c(C)cc(N(C)C)cc2)=O)CC2CN(C(C34CCC3C4)=O)CC2(C)C1 N(C(=NCCc1ccccn1)NCc1ccc(CO)cc1F)C(COC)C1CC1 N1(c2cc(NC3CC(O)C3)nc(COC)n2)CCCN2CCCC2C1 N1(C(C2CC(OC)C2)=O)CCC(=O)NC2CN(C(=O)C(C)CO)CCC12 C(=O)(CC(CC)CC(C)C)NC(C(=O)N1CCC(O)(CC#C)CC1)CC(F)(F)F C(c1ccc(S(=O)(=O)NC)cc1)=CC(N1CCCC(CNC(C(CC)O)=O)C1)=O n1(CC)cc(C(=O)NCC2COCC2NC(=O)Cc2cc(C)nn2C)c(C2CC2)n1 C12(C(=O)NCc3cc(C)[nH]n3)CCCC1CCN2C(c1cc2ncccc2[nH]1)=O C(=O)(C(C)CC(C)CC)N1CCC(NC(Cc2c(SCC)cccc2)=O)C1 CCC(CC)(CO)C(=O)NC1CCN(C(c2cccc(C3CCC3)c2)=O)CC1F N1(C(C(CC)COC)=O)CCC(C(N2CC3CC=CC2C3)=O)C(C)(C)C1 c1(CC(C(=O)NC(C#C)CC2CCCC2)NC(=O)C(O)C(C)C)ccccc1Br c1(CCNC(=O)C(c2sc(Br)nc2Cl)N2CCCC23CC3)cccc(F)c1 N(C1CN(C(=O)CCC(F)F)CCc2ccccc21)C(C1(COC)CCC1)=O N1(C(C2(CSC)CC2)=O)CCCC1CCCNC(=O)COc1cc(C)on1 N1(C(c2c(CC)nco2)=O)CC2CC(C1)N2C(C1COCC(C)O1)=O Cc1cc(=O)ccn1CC(=O)NC1CC2CC(NC(=O)Cn3ccnn3)C1C2 c1(C(=O)NC(c2cccc(OC)c2)C(=O)OC(C)C)c(Br)nc2n1CCOC2 N1(C(c2nc(OC)sc2)=O)CCCC(CC2CN(C(c3ccncc3Cl)=O)C2)C1 c1(C(=O)NC2CCC(CC(=O)NCC3(CCOC)CCC3)C2)sc(F)cc1C C(=O)(CCN=[N+]=[N-])NC(C(=O)NCCCC#C)CC1CCC1 Cc1ccc2nc(C(=O)NC3CCCC34CCN(C(=O)CC3CSC3)C4)cn2c1 CC(CCC(C)(C)C)C(=O)N(C)CC1(NC(=O)C2=CSCS2)CC1 Cc1cnn2c(NCC(=O)Nc3ccc(O)cc3)cc(Cl)nc12 c1(C(=O)NC2CN(C(c3c(C)cc(C)nc3)=O)C(C)C2)ccc2c(c1)COC2=O CCC1=C(C(=O)N2CCC(NC(c3cnc(S)[nH]3)=O)C2(C)C)CCCO1 N1(C(CC2CC(=O)C2)=O)CC2CC(NC(c3n[nH]cc3Cl)=O)C1C2 n1(CCC)cncc1CNC(C1(CNC(=O)C=Cc2cncs2)CC1)=O C1(NC(c2cnc(NC(C)=O)o2)=O)CN(C(C2CSC2)=O)CC1F N1(C(CCC)=O)CC2(CCC(NC(=O)C=Cc3ccc(OC)cc3)C2)C1 c1(C(N2CC(N(C)C(C3CCC(=C4CCC4)CC3)=O)C2)=O)ccc(N)c(CO)c1 N1(C(C(C(C)C)NC(C(CC)=CC)=O)=O)CC2(CC(N(C)C)C2)C1 N1(C(C2(CC)CCN(C(=O)C(C)(C)n3cncn3)CC2)=O)CC(C)CCCC1C C(=O)(C(CC(F)F)N(C(=O)CC(C)N(C)C)C)NCC(C#C)OC N1(CCNC(=O)Cc2cnc[nH]2)CCN(C(=O)C=C2CCC2)CC1 CC(CCNC(=O)C(c1ccccc1Br)(F)F)CCNC(=O)C=CCF C1(C(N2CC(CCCCNC(Cc3cn(C)nc3)=O)C2)=O)CCOC(=O)CC1 C1(NC(=O)CC2CC(F)(F)C2)CCN(C(C2CCCC(F)(F)C2)=O)C12CCC2 c1(C(N2CC(O)(CNC(=O)COCc3nc[nH]n3)C2)=O)cc(C(F)F)ccc1F C(=O)(C1CCCn2ncnc21)NC1CN(C(c2c(C)nc(CC)s2)=O)CC1(C)C C(CCS(=O)(=O)Nc1cccnc1OC(F)F)N(C)C1CC1 CCC1=NOC(CNC(C2(CC)CCN(C(C3CC(C(C)C)C3)=O)C2)=O)C1 C1(CC(=O)NCCCNC(=O)CC2C=CCC2)Cc2cc(C(F)(F)F)ccc2O1 C1(CC#C)(C(=O)N(CCCNC(=O)CC2CC2(Cl)Cl)C2CC2)CCOC1 c1(C(=O)OC)cccc(NCC(c2ccccc2)(O)NC(C)=O)c1Cl c1(C(=O)OC)ccc(SC(C)CO)cc1.C1(CC2CCC2)C(=O)N1 C12(CNC(C3N(C(C)C)CCC3)=O)CCC(C1)N(C(C1(C(C)C)CCC1)=O)C2 C(Cc1cnc[nH]1)(C(=O)NCCC(C)NC(=O)CCC1CC1)NC(C)=O CC1CC(NC(c2ncoc2-c2ccon2)=O)CN1C(=O)C=Cc1ccnn1C c1(C(=O)NCCN(C(c2csc(CO)n2)=O)C2CC2)ccc2ccnc(O)c2n1 c1(OC)ccc(O)cc1C(=O)NC1CCCC(CNC(C2CC(O)C2)=O)C1 N1(C(C(CC)NC(N)=O)=O)CC(CNC(C2CN(CC(C)C)C2)=O)C(O)C1 N1(C(C(C(C)C)N(CC)CC)=O)CCC(CNC(=O)CCSC)C(F)(F)CC1 CC(C)C(C)(CNC(C1OCCC1C)=O)NC(c1cn(C(F)(F)CO)nn1)=O c1(C(N2C(CNC(CC(=O)NCC)=O)CC3(CC3)C2)=O)cc(C)c2c(c1)CCC2 c1(C(N2C(C(=O)NCC(C)NC(=O)OC)C=CCC2)=O)ccc(C)nc1C c1(C(N2CC(N(C(CCCCSC)=O)C)C(F)C2)=O)cc(C)nc(O)n1 c1(C(=O)OCC)ccc(C(N2CCCC(N(C)C(C3(CF)CCC3)=O)C2)=O)nc1 C1(OC)CC(N(C)C(c2occc2C)=O)C12CCC2 N1(C(c2n(C)ccn2)=O)CCc2nc(CNC(C3CC3C3CC3)=O)sc2C1 C(=O)(C1=CCCN(C(=O)CC2(CSC)CC2)C1)N(C(C=C)C1CC1)C c1(NC(C(c2cccnc2)NC(c2ccc(COC)s2)=O)=O)cc(C)ccc1C c1(C(=O)NC(C2CCN(C(c3cccc(OCCF)c3)=O)C2)C)cnnc(O)c1 N1(C(C2CC(NCc3c(C)cccc3)C2)=O)CCCC2CCCCC12 N1(C(C2C(CC)OCC2)=O)CCC2(CC1)CC(NC(c1cncnc1)=O)CCO2 c1(C(=O)NC2(CN(C)C(c3ccc(Br)nc3F)=O)CC2)c[nH]c2cccc(C#N)c12 C(=O)(C(COC)CC(C)C)N1CC(C(=O)NCC(F)C2CCC2)(COC)C1 CC1CN(C(c2ccco2)=O)CCC1CNC(=O)CCc1ccc(Cl)cc1 c1(C(N(CC(CC)NC(C2(CC#C)CCCO2)=O)C)=O)ccccc1C(C)=O C1(C(N2CCOC(C(F)(F)F)C2)C(=O)NCC(=C)C)CC2CCC1CC2 CC1CCC(=CC(=O)NCCCC(C)NC(c2ccn(C3CCC3)n2)=O)CC1 C1(C=O)CC(C)=NO1.C1(=O)CCN1CC1CC1.C(C(C)N)SCC c1(NC(C2C=CC(NC(C3CC(O)CN3)=O)C2)=O)cc(Cl)ccc1[N+](=O)[O-] N1(C(C(C)(C)F)=O)CCC(F)(F)C(CNC(C2(CC3CCCC3)CCCC2)=O)C1 C1(C)(CC)C=C(C(=O)NC2(C(=O)NCC(O)CC3CCC3)CCCCC2)C1 C1(C(=O)NCC(CNC(C2(NC(C)=O)CCCC2)=O)CO)CC=C(C)CC1 c1(OC)c(C)cnn1C.c12ccc([nH]1)CC(=O)NCCOCCOCCNC2=O N#CC1CC(C(=O)NC2CC(CNC(c3occc3-c3ccccc3)=O)C2)C1 N1(C(c2ccc(C=CC(=O)OC)o2)=O)CCN(Cc2cccc(F)c2)CC1CF c1(C(C)C)ncc(C(=O)NCC2CCCC2NC(=O)Cc2ccoc2)cn1 c1(OC)ccc(Cl)c2c(=O)c(C(N3CCC(C)C(C(F)(F)F)C3)=O)c[nH]c12 c1(SCC(N2CCCC(NC(C(C(=O)OC)C)=O)C2)=O)ccc(C)c(C)c1 C1(S(N)(=O)=O)(C(=O)NCC(CNC(Cc2c(OC)ccc(F)c2)=O)F)CCCC1 N1(C(=O)Cc2cc[nH]n2)CCC(O)(CNc2cc(C(=O)O)no2)C1 N1(C(CNC(CCC)=O)=O)CCCC1CCNC(=O)C(C)(C)c1cncs1 N1(C(C2CN(CC)C(=O)CC2)=O)CCC2(NC(=O)CC3CC3C)CCCC12 C1(N(C(Cn2ncc(C)c2)=O)C)CC2CC1N(C(C1CCC(=O)N1)=O)C2 CC(C)C(O)C(F)(F)C(=O)N(CCNC(c1cnc(O)o1)=O)C1CC1 c1(OC)cc(I)c(Cl)cc1CNc1cc(Cl)ccc1C(=O)N(C)C C1(NC(CC2ON=C(C)C2)=O)CCC(F)(CNC(=O)Cn2ccc(C)c2)C1 c1(C(=O)Nc2c(CC)ccc(F)c2)cc([N+](=O)[O-])ccc1OC C=CC(C)(C)CC(=O)NCC(C(F)(F)F)N1CCN(C(=O)CC2CSC2)CC1 N1(C(c2n(CCC)ncc2)=O)CC(NC(c2coc(OCC)n2)=O)CC1C C(=O)(CS(=O)(=O)C(C)(C)C)NCC(C)(CO)NC(C1C(C)(C)C2CCC1C2)=O C12(C(=O)NCC3(CCOC)CC3)CC(C)(CN1C(=O)Cc1ccns1)C2 c1(NCc2cnc(C)s2)nccc(=NC(C)CS(C)=O)[nH]1 C12(OCC)CN(C1)C(=O)C1(CC(C)C1)OCC(=O)NC2.S(C)CC C(C1=CCN(C(C2CCC=CO2)=O)CC1)NC(CC1(OC)CCC1)=O c1(CC)ccc(C)cc1C(=O)NCCC(C)NC(C1(C)CCNC1=O)=O c1(C(N2CC(N(C(=O)CC3CCC4CC34)C)C2)=O)cc2c(s1)CCC2 c1(NCC2CN(C(CC(C)N(C)C)=O)C2)ncnc2cnccc12 NC(=O)CC(O)C(=O)N1CCCC(CO)(NC(c2ccc(N)c(Cl)c2)=O)C1 C1(CC(=O)OC)(NC(=O)Cc2cccc(F)c2)CS(=O)(=O)C1 N1(C(C(CCC)CC)=O)CCC(C2CC(NC(=O)Cc3scnc3C)C2)CC1 C12(C(=O)NC3CC(NC(C(CCC)c4ccccc4)=O)C3)CCN(CC1)CC2 CC(CS(C)=O)C(=O)NC12CC(CNC(c3ncccc3C3CC3)=O)(C1)OC2C c1(C(C)C)ccc(C(C)(C)CNC(C)(CCI)c2nnnn2C2CCOC2)cc1 N(C1CCCn2ncnc21)C(c1ccccc1OC)CC C1(CNC(CNC(CCC)=O)=O)CCCN(C(=O)C(C)(CC2CCC2)OC)CC1 N1(C(COCCSC)=O)CC(CNC(=O)CN2CCOCC2)CC1C C1(CC)C(C(=O)NC2CCC2(C)C)CCN1C(=O)CN(C)C(=O)OC c1(C(N2CCC(NC(c3ccc(CC)cn3)=O)C(F)C2)=O)ccn2c1CCCC2 n1(CC)ccc(C(=O)NC2(CC(=O)NCc3cnn(C)c3)CCC2)n1 CCC(CC(=O)NCC(C)(C)CN(C)C(C1(F)CCCCC1)=O)SC C(=O)(C1=CCOCC1)NC1C(CNC(CC2N(C(C)=O)CCC2)=O)C1 C(C)(C)(C(=O)N(CCNC(c1cn(CC2CCCOC2)nn1)=O)C1CC1)N(C)C Cc1ccc(Br)cc1C(=O)NCCCCCCN(C(=O)C(C)C1CCCO1)C N1(C(C(=O)NC)CC2CCCO2)CCC(C)=C(Br)C1 N1(C(CC2N(C(C(C)NC(=O)NC)=O)CC2)=O)CCCC2CNC(=O)C12 c1(C(=O)NCCN(C)C(c2coc(Br)c2)=O)cc(OC(F)F)cc(F)c1 C(=O)(C1=CCCSC1)NC1C(CCC)CN(C(c2c(SC)cnn2C)=O)C1 c1(CC)ccc(C(C(=O)Nc2ccccc2Cl)N(C)CC2CCCCC2)c(Cl)c1 c1(CNC(c2cnn(CC3CC3)c2F)c2n(CC)nnn2)cc(F)c(Br)cc1F C(=O)(N=c1cc2n([nH]1)CCCC2)C1C(C)N(C(=O)CC=C(Cl)Cl)CC1 C1(CNC(C(C(CC)C)=O)=O)CCC2CN(C(=O)C(=Cc3cnn(C)c3)C)CC12 C1(O)(CNC(C2CC(C)N2C(=O)OC(C)(C)C)=O)COC2CC1C2 N1(C(C2(CC#C)CCCO2)=O)C2CCC1CN(C(c1cccc(CCO)c1)=O)C2 C1(COC(C)(C)C)CC(F)CN1C(=O)NCC(=O)NCc1ccnc(C(=O)O)c1 c1(C(C(=O)NS(=O)(=O)CCCC2CCC2)O)ccc2ccccc2c1 C1(C(C(=O)NCc2c(-n3cc(CC(C)(C)C)nn3)ccs2)C(N)=O)CCCCC1 CN1C(=O)CCC1C(=O)N(C1CCCCC1)CCNC(=O)CC1(CO)CC1 c1(-c2n(-c3ccc(OC)cc3)nc(CO)n2)cc(F)ccc1O N1(C(c2cccc(Br)c2)C(=O)NC(C(=O)OC)C)CC(CN(C)C)CC(C)C1 c1(N2CC(C(C)NC(=O)CCc3cnn(C)n3)C2)ccnc(-c2nccs2)n1 n1(CCC)nc(C(=O)N(C2CCNCC2)CC)ccc1=O C1(NC(CC2(COC)CC2)=O)CN(C(=O)C(C)(C)CC2CC2)CC1C(F)(F)F C1(C)(CNC(c2cnn(CC)c2C2CC2)=O)CCN(C(=O)C2=CCOC2)CC1 Cc1cnc(NCC2CCCC2NC(=O)CSc2nc[nH]n2)nc1 Cc1cc(NC(c2nncs2)=O)ccc1NC(=O)C(C)n1cncn1 c1(CCC(=O)NCC(CNC(C(C)OCCC#C)=O)OC)ccccc1C(N)=O C1(NC(C(CC=CC)C)=O)CC12CCN(C(c1c[nH]c(C(F)(F)F)c1)=O)CC2 N1(C(CCc2cccc(C)c2)=O)CCN(C(c2nc(=N)cc[nH]2)=O)CC12CC2 CCC(C)(C)CC(=O)NCCCC(C)NC(=O)C(C)C1CC1 CCCCCCCN(C)C(C1C(C)CCN1C(c1ncn(C)n1)=O)=O c1(N(C)C)ncc2c(n1)CCC(NC(=O)C(=O)NCc1c(F)cc(F)cc1F)C2 C1(C(=O)NC2C(NC(C3CCCN(C(=O)OC)C3)=O)CCC2)CC2C=CC1CC2 c1(CC)oc(C(=O)N(C)CCC2CCN(C(=O)C=CC=C(C)C)CC2)cc1C N1(C(c2cnc(C)[nH]2)=O)CC(NC(c2ccc(I)c(O)c2)=O)CC(F)(F)C1 C1(NC(C2C(COC)C2)=O)CC2CC1N(C(=O)CN1CC(C)(OC)C1)C2 c1(CC)ccc(NC(C23CC(CO2)N(C(=O)CC2CC2(C)C)C3)=O)c(C)c1 c1(OC(F)F)cc(C)ccc1C(N1CCCC(N(C)C(C2(OC)CC2)=O)CC1)=O CC1CN(C(c2ccccc2)=O)CCC1Nc1cc(C(F)(F)F)cnc1O C12(C(N3CCN(C(CCc4cc(C(C)=O)c(C)o4)=O)CC3)=O)CCN(CC1)CC2 C=C(F)C1(CC(=O)NCC(=C2CN(C(c3noc(CC)c3C)=O)C2)F)CCC1 c1(C(N2CC(C)(NC(c3cnc(O)c(Cl)c3)=O)C2)C)ccc(C#N)cc1F CCCC(CC)C(=O)N1CCOCC1CNC(c1cnn[nH]1)=O C1(NC(CCSCC)=O)CC(CC(=O)NCc2ccc(SC)o2)C1(C)C N1(C(C(CC)=CC)=O)CCC(C)N(c2ccncn2)CC1 c1(C(N2CCC(NC(C(c3cnn(C)c3)OC)=O)C2)=O)n[nH]c(C2CC2)c1Br Cc1n[nH]c(C)c1S(=O)(=O)N1CCC2(CC1)CN(C(C1CC1F)=O)C2 c1(CC(=O)NC2CCC(CCNC(C3(CC=C)CC3)=O)C2)ccc(C)nc1Cl Cc1ccc(C(N2CCN(C)C(CNC(C3(CC(C)C)COC3)=O)C2)=O)c(O)n1 CCC(C)C(C)CNC(=O)CC(C)(C)N(C)C(C1(CC)CCCCO1)=O c1(OC(C(N2CCC(c3cccc(OC)c3)(C)C2)=O)C)ccc(F)cc1Br C1(CNC(COCCC#C)=O)CN(C(c2cc(C(F)F)[nH]n2)=O)C2(CCC2)C1 C(=O)(CC(C)C(C)(C)C)N(C(CC(=O)N(CCCC#C)C)(C)C)C c1(CC)cc(C(=O)NC2C=CC(C(=O)Nc3cnncc3Br)C2)cc(C)n1 Cc1coc(C(=O)NC2(CNC(=O)Cc3cccc(CO)c3)CCC2)c1C C(C1c2ccsc2CCN1C(=O)C(C1CCOCC1)F)NC(=O)CCOC1CC1 C(c1ccc2ccccc2n1)=CC(=O)NC12C(CN(C(c3c(OC)ccs3)=O)C1)C2 c1(CC)ccc(Br)cc1C(=O)NCC1(F)CCCN(C(c2nc[nH]n2)=O)C1 N1(C(CN(C)CC)=O)CCCCC1CNC(c1cc(C(=O)NC(C)(C)C)on1)=O C(=O)(C1=CC2(CCOCC2)C1)N1CCC(N(C(=O)Cc2nc([N+](=O)[O-])n[nH]2)C)C1 N(C1c2ccccc2CC1NC(=O)CCS(C)(=O)=O)C(Cn1nc(C)c(Cl)c1)=O c1(NC(C(C)NC(CN(C(C2CCCC2)C)C)=O)=O)ccccc1CCO Cc1cc(=O)n(C)cc1C(=O)NCc1nc(C(=O)NC2(C)CCCC2C)co1 Cc1ccc2[nH]c(C(N3CCC(C)C3CNC(=O)CC3C=CCC3)=O)cc2c1C c1(C(=O)NC2CC(NC(CC(C)C3CCCO3)=O)C2)csc2c1CCCC2 Nc1ccc(C(N2CCC(OCCNC(c3cncc(Cl)c3)=O)C2)=O)cc1Cl N1(C(C2CC(=C)C2)=O)CCCC2(CC(NC(=O)C(C)(C)OC)CO2)C1 C1(NC(Cc2ccc(CCC)cc2)=O)CC2CC(C1)N(C(C1(C)CC1(F)Cl)=O)C2 C1(C#N)(C(N2CCCN(C(C(=O)NC(C)C)=O)C(CO)C2)=O)CC2CCC1CC2 c1(C(N(C(CNC(C2CC(NC(CC)=O)C2)=O)C)CC)=O)[nH]nc2ncccc12 c1(-c2c(C#N)nccc2)nc2c(s1)CC(C(=O)NCCn1cc(CO)nn1)CC2 CC(c1cccs1)=CC(=O)NCC1CN(C(=O)CN2CCCNC2=O)CC1O Cc1cccnc1S(=O)(=O)NCCC(N1CCS(=O)(=O)CC1)=O Cc1nc(C)n(CCC(=O)NC2CCN(C(=O)CSCCC(C)C)C2C2CC2)n1 c1(-c2scc(CCN(CCn3ccnc3C)CC)n2)ccc(F)cc1 c1(C(N(C)CCC2CCN(C(C3CC3Cl)=O)CC2)=O)ccnc2ccccc12 CCC(C)(CNC(=O)C(n1cc(Cl)cn1)C)NC(c1ccn(C)c1)=O c1(C(=O)NC2C(CNC(c3cc(C(C)=O)sc3)=O)C2)cc(C)nc(O)c1[N+](=O)[O-] N#Cc1ccc(C(N2CC3(CNC(=O)CC4CCCCO4)CC2CO3)=O)cc1F C1(C(=O)NCCN(C(=O)C(F)(F)CO)CCC)CC2CCCN2C(=O)N1 N1(C(C2CC(n3ccnc3)C2)=O)CCCC(O)(Cn2cc(CCCO)nn2)CC1 Cc1ncnc(C)c1CC(N1CCC(NC(C2CCOC(C(C)C)C2)=O)CC1)=O N1(C(C(c2cn(CC)nc2)(F)F)=O)CCOC(CNC(=O)C(C)(C)CC2CC2)C1 C1(CC(N2CC(COC)(CNC(=O)C(C)CN(C)C)C2)=O)CCC(F)(F)C1 N1(C(c2cc(C)sn2)=O)CCC2(CCC2NC(C2CNC(=O)CC2(C)C)=O)CC1 N1(C(C(CCSC)O)=O)CCN(C(=O)CC(C)N(C)C)CC2(CC2)C1 N1(C(c2ccc(OC)cn2)=O)CCN(C(=O)C=Cc2cncnc2O)C(CO)C1 CC1CC(NC(=O)CCC(C)(F)F)CN(C(c2cccc(C(F)F)c2F)=O)C1 N#Cc1cccc(CC(N2CCC(CNC(C3CC4CCC(C3)O4)=O)C2)=O)c1 C1(c2cccs2)(CC(N2CC(CCC(F)(F)F)C2)=O)CCCCC1 Cn1ccc(C(=O)NC2CCOCC2NC(C2C3(CC3)C23CC3)=O)c1C1CCC1 C1(C(=O)OCC)CCCC(C(=O)N(c2cncc(C)c2)CC)C1.C(=O)C(Cl)(Cl)Cl c1(CC(=O)N(CCNC(=O)CC2CC=CC2)CC)ccc(O)cc1Cl c1(N2CC3(CN(C(C4(c5ccccn5)CC4)=O)C3)C2)nc(O)c2c[nH]nc2n1 C(CCN=C1NCC2CCCCC2N1)c1c(F)cccc1 Cc1ccc(C(O)C(=O)NCC2(CO)CCN(C(c3sncc3C)=O)C2)nc1 N1(C(c2cc(CCC)[nH]n2)=O)CC2CC1(C(=O)NCc1scnc1C)C2 C1(C(=O)NC(C#C)C(C)(C)C)CCC2(CC2)N1C(=O)CS(=O)CC Cc1cc(C(N2CCC(CNC(=O)CCCNC(N)=O)CC2C)=O)c(N)c(F)c1 c1(N2CCN(CCOC)CC2)nc(=NCC(C)n2cccn2)[nH]c2c1CCCC2 Cc1cnc2n1CCCC2C(=O)NC(C)CNC(c1cnc(Br)s1)=O C1(C(=O)NCC(CN(C)C(C2(C(C)(F)F)CC2)=O)O)CCOC1(C)C c1(C(=O)NC2(C(=O)NC(COCC)C)CC2)cc(C)on1 c1(N2C(CCNC(c3ccc(CC4CCCC4)cc3)=O)CCC2)nccnc1F c1(NC(C2C(C)C2)=O)cc(F)c([N+](=O)[O-])cc1F c1(OC(C(N2C(CNC(c3cc(C)ncn3)=O)CCC2)=O)C)cccc(C)c1C N1(C(c2scc(C)c2)=O)CCN(C(=O)CCOc2ccccc2F)CC1C N1(C(c2cccc(C(C)C)c2)=O)CC(C)(CNC(=O)C2=CCOC2)CC1(C)C C12(C(N(CCN(C)C)CC)=O)CCN(C(c3cccc(CC#N)c3)=O)CCC1C2 N1(C(C2C(CC)CCO2)=O)CC(C)(C)CC1CC(=O)N(C)Cc1cnn(C)c1 C1(F)(CNC(C(C)NC=O)=O)CCCN(C(C2CCC2c2nc[nH]n2)=O)C1 CCC(O)C(C)(C)C(=O)NCC(CC(=O)NC1(CO)CC(OC)C1)C1CCC1 Cc1cc(N2CCC(CS(N)(=O)=O)C2)nc(NCCCCN2CCC2)n1 c1(C(=O)NCC2N(c3cc(OC)nc(C)n3)CCCC2)cc2cccnc2[nH]1 C1(CC(=O)NC2CN(C(C3CCC(CC)CC3)=O)CC2O)CCC(C)(C)CO1 N1(C(CC(C)(C)O)=O)CCC2(CCCCC2NC(c2cc(O)nc(Cl)c2)=O)C1 C=Cc1ccccc1-c1cnc(CNc2cc(C#N)ncn2)nc1 CCC(C)C(C(=O)Nn1nnc2c1CCCC2)N(C(=O)C=Cc1cncn1C)C N1(C(C(c2cnn(C)c2)NC(c2ccnc(OC)n2)=O)=O)CCCC2(CCCO2)C1 CC(C(=O)N1CCC(CNC(c2ccc(C3CCC(=O)N3)cc2)=O)C1)C(F)F C(=O)(C(C)(C)CCOC)NC1C2(CC(NC(C(C=C)(F)F)=O)C2)C1 c1(NC2(c3n(C4(C)CC4)nnn3)CCCSCC2)ccc(F)c(S(N)(=O)=O)c1 Cc1csc(-c2cn(CC3CCN3C(=O)C(O)Cc3ccccn3)nn2)n1 c1(OC)cc(C(=O)NCC(CC(C)O)c2ccccc2)cc(SC)c1OC N1(C(c2cc(OC)cc(Cl)c2)=O)CC2(CCC(N3CCCC3C(N)=O)CC2)C1 O=C(CCCCNC(C1CC1C1CCCO1)=O)NCc1cn(C2CC2)nn1 C1(CN(C(CCc2onc(CCC)n2)=O)C)CN(C(c2ccc(F)o2)=O)CCO1 C(=O)(CCS(=O)(=O)CC(C)C)NCC(CCNC(C1CC=C(C)CC1)=O)O CCC(CC(=O)N1CCC(CNC(c2cnsn2)=O)(COC)C1)CC(F)(F)F CC1(NC(=O)CC(F)(F)Cl)CCC(NC(=O)Cc2ccc(C#N)cc2)CC1 C1(CNC(c2nc(COCC)sc2)=O)C(C)CCN1C(c1cnc(NC)cn1)=O CCC(CN(C)C)CC(=O)N1CCCC(NC(=O)C=Cc2cccnc2)C1C C1(C)(C(=O)NCCC(C)C)CCCN(C(c2cc(CO)n(C)n2)=O)C1 c1(C(=O)NC2CC(C)(NC(CC=C)=O)C2)cc(Cl)cnn1 CCN=C(NCCCS(=O)(=O)C1CC1)N1CCC(F)(C#N)C1 S(=O)(=O)(c1c(Cl)cccc1Cl)C(=O)CNC1CCNCC2CCC12COC N1(C(COCCCC#C)=O)CCCN(C(=O)CSc2ccc(F)c(F)c2)CC1C C1(NC(CCC#CC)=O)COCCN(C(=O)CCCSC(C)(C)C)C1 C1(CS(=O)(=O)NCC(C(C)C)c2ccccc2)CC2OC1C1CC21 N1(C(C(F)=CCC)=O)CCC(O)(C(C)NC(=O)Cc2ccc(C)nc2)C1 C1(C)(CNC(CS(CC)=O)=O)CC(F)(F)CN1C(C1CC2(CC(=O)N2)C1)=O c1(C(=O)NCC(C)CNC(C2CCC(O)CC2)=O)ccc(N(C)C)cc1F N1(C(CC(CC)C)=O)CCC(NC(c2cc(-c3ccc(C)o3)[nH]n2)=O)C12CCC2 N1(Cc2ccc(-c3ccc(C(=O)NC(C)(C)C)cc3)cn2)CCn2cncc2C1 Cc1ccc(Cl)c(N(C(C)=O)CC2CCCN(Cc3nn[nH]n3)C2)c1.C1C(=O)O1.OC c1(N2CC(NC(C(=O)OCC)=O)C(F)(F)C2)ccn2ncc(I)c2n1 C=CCC(C(=O)NC(CO)CCCNC(=O)C=C1CCCCC1)C(C)C N1(C(C2(COC)CCOC2)=O)CCN(C(=O)CCCC(F)F)C(CCO)C1 C=Cn1nncc1C(N1CC(O)(CNC(=O)CC2CC2C)C1)=O Cn1ccc(CCC(=O)NCCOC2CCN(C(=O)CC3OCCO3)C2)n1 N1(C(COCCOCC)=O)CCCN(C(c2ccccc2-n2cncn2)=O)CC1 C(=O)(CN=c1[nH]c2ccccc2s1)N1CC(F)CC(NC(CCCN=[N+]=[N-])=O)C1 N#Cc1ncn(CC(N2CC(F)(C(=O)NCCc3cn[nH]c3)C2)=O)n1 N1(C(=O)NCC(c2ccsc2)C)CCC(NS(C(C)C)(=O)=O)CC1 Cc1cc(C(=O)NCCOC2CCN(C(=O)CCC3(C#N)CCC3)C2)cc(C)n1 C1(N(C(c2c(C3CC3)cnn2C)C(=O)NC2CCCCC2)C)CNC(=O)C12CC2 Cc1nnc2n1CCN(C(C1COCCN(C(c3ccc(N)c(F)n3)=O)C1)=O)C2 c1(C(N2CC(=C(CNC(COCCC=C)=O)F)C2)=O)cc(F)ccc1Br c1(C(=O)NC(c2cn(CC(CC)CC)nn2)(C)C)cc(C)ccc1F CC(C)C(C)CC(=O)NC(C1CC(NC(C2CCC(C(N)=O)C2)=O)C1)C N1(C(c2cc(SC)ncc2)=O)CCCOC(CCNC(C2C(C)C2C)=O)C1 c1(C(=O)NC2C(NC(=O)CCc3ccoc3)CC2)ccc(Br)o1 C1(CC(=O)OCC)CCCCN1C(c1cnn(CC)c1)C(=O)NCC1CCC1 C1(CNC(c2cc(CC)nn2C)=O)C(C)CCCN1C(c1csc(COC)n1)=O Cc1nc(CO)ncc1C(N1CCCN(C(c2cc(C(C)(C)C)no2)=O)CC1)=O c1(CC(=O)NC2C(NC(c3[nH]cc(C(C)=O)c3)=O)C2)coc2c(F)c(F)ccc12 c1(C(=O)NC2CC(NC(CNC(C(CC)C)=O)=O)C2)ccc(C)nc1N C(C)(C)(CCCC(=O)NC1CC(O)C1O)NC(c1nc(C)sc1)=O C(CC(F)F)(C(=O)NC(C)CCN1CCCC1)NC(CCCC)=O N1(C(C(C)(C)OC(C)C)=O)CCCCC(CNC(=O)NCc2ccc(Cl)cc2)C1 C1(C(N(C2CCN(C(=O)C(O)CC)C2)C)=O)N(C(=O)OC(C)(C)C)CC1(C)C C(=O)(C1=C(C#N)CCC1)N1CCN(C(Cn2c(=O)sc(C)c2C)=O)CC1C(C)C CC(=O)CCCCCCC(=O)N1CCC2(CCOC2=O)C1 C1(C(=O)NC(c2nccn2C)CC)CCCCC1CNC(=O)CCC=CC(C)C N1(C(C=CC=CCC)=O)CC(F)CC1C(=O)Nc1cnn(C(F)(F)F)c1 C1(C(N2CC(OCC)C2)=O)CN(C(=O)CN2CCC(C)CC2)CC1C N1(C(C2CN(C(C(CC)NC(N)=O)=O)CC2C)=O)CC2CC1CN2C C1(NC(c2cnc[nH]2)=O)CC2(C1)CN(C(=O)CC1CC=CCC1)C2 C1(C(=O)NCC2(NC(=O)CC34CCCC3C4)CC2)CCCN2CCCC12 N1(C(C(CC(C)(C)C)O)=O)CCCCC(N=c2[nH]nco2)C1 C1(COCC)(NC2CC(C(=O)OCC(C)(C)C)C2)CCOC1 c1(C(N2C3CC(CC(C)O)CC2CC3)=O)cc2ccncc2c(O)n1 C1(COC)(NC(=O)CCCc2nc(C3CC3)no2)CC1(F)F c1(C(=O)NCCCN(CCC)CC2(CC)CC(C(=O)NC)C2)ccc(CC)s1 C1(C(=O)NCCCCN(C)C)CCOCC1NC(c1nccnc1N)=O C1(C(=O)NCc2cc(OC)ncc2)CN(C)CCN1C(c1ccco1)=O N1(C(=O)C(c2ccccc2Cl)O)CC=C(CCNC(C2(n3nccn3)CC2)=O)CC1 CC(CF)CC(=O)NC(C)CC1CN(C(=O)C(F)(F)C2(O)CCC2)C1 C1(C(=O)NC2(CO)CCN(C(c3cccc(CSC)c3)=O)C2)CCC2(CCC2)C1 C(CNC(c1cccc(OC(F)F)n1)=O)(C(C)(C)C)NC(C(CN(C)C)O)=O n1(CCC(=O)NCC2CCC(CC)CC2)cnc2ccccc12 c1(OC)cccc(C)c1.N1(CC(=O)NC)CCC(OC)C1.C12CC(C1)C(=O)N2 C1(C(NOCC)=O)CCN(C(C2CC3CCC(C2)O3)=O)CC1O.C123CCC(C1C2)N3 C(=O)(C#CC1CCC2(CC1)OCCO2)NC(C(CC)C)C(=O)OC Cc1c(C(=O)NC2COCC2NC(c2cn(C)nc2Br)=O)nnn1C C1(C(=O)NCC(C)(CO)NC(c2c(C)cc(CC)o2)=O)CC2(C1)CS(=O)(=O)C2 N(C1CCc2cc(CNC(=O)C3CC3)ccc21)C(c1ccc(C(C)(C)C)cn1)=O Nc1ccc(F)c(C(=O)NCCCN(CCCNC(c2cccnn2)=O)C)c1F C(CC(C)(C)CC(=O)NCCCOCCC(=O)NCCc1ccc(C)s1)OC CCC(CC(C)C)C(=O)N1CCC(C(=O)NCC(n2ccnn2)C)(CC)C1 C1(COC)COCCN1C(=O)CCN(C(=O)CC1CCSC1)C(C)C CCCCCC(O)C(=O)NC1CN(C(c2nn(-c3ccc(C)cc3)cc2O)=O)C1 C1(NC(c2c(CC)ccs2)=O)CC2CN(C(c3ccc(N)cc3C)=O)CC2C1 n1(CC)nc(C(C)C)cc1C(N1CC(NC(C2(C)CC=CCC2)=O)C(O)C1)=O c1(C(N2C(CNC(CC(C)OC)=O)CCC2)=O)cc([N+](=O)[O-])ccc1C(F)(F)F Cc1nc(C(=O)NCC2(C)CCC(NC(c3cccc(C(N)=O)n3)=O)C2)n(C)n1 c1(C(N2CCC(CC)C2C(=O)NCc2nnn(C)n2)=O)cc(O)cc(F)c1 N1(C(=O)Cc2cccs2)CCN(C(=O)C(F)(F)C2CC2)CC1c1cccc(F)c1 c1(C(N2CCCC(C(C(=O)NCCCOCC#C)C)C2)=O)ccc(C)cc1C c1(C(=O)NCCC2CCCCN2C(c2cc(Cl)c(Cl)s2)=O)cc2ccccn2c1 Cn1cnc2c(CNC(c3ccc(N4CCC(CO)CC4)nc3)=O)cccc12 c1(C(N(CC(C)(C)CNC(C2CCCN2C2CC2)=O)C)=O)ccc(CCO)cc1 C1(NC(CNC(C(CC)C)=O)=O)CC(C)CN(C(c2ccc(C3CC3)o2)=O)C1 c1(C(N2C(CNC(Cc3ccc(C)s3)=O)CCCC2)=O)cc(C)c(N)cc1F C(=O)(C1CCCc2ncnn21)N(CCOC)CCNC(=O)CC1CC(C)OC1C CC(C(=O)NCC(C1CC1)N(C)C(C12CC(C)(CCO1)C2)=O)C(F)(F)F C1(CC)CC(O)CN1C(=O)CC1CCC(NC(=O)CC2(OC)CCC2)C1 c1(OC)cnc(Cl)cc1C(=O)N(CCCNC(C1CC12CC2)=O)C(C)C C1(CC)CC(O)CN1C(=O)C(C)(C1CC1)N(C)C(c1cn(C)nn1)=O c1(CCC(=O)NC(CCOC)CNC(c2ocnc2C2CC2)=O)ccccc1Cl N1(C(c2c(C)nc(C)c(C)n2)=O)CCCC2(CCN(C(=O)CCC(C)(C)F)C2)C1 C1(NC(Cc2n(C)ncc2Cl)=O)CC(O)CN(C(c2cnc(O)cc2O)=O)C1 c1(C(=O)NC(COC)CC(=O)NC2(C)CC2(C)C)cc2cccnc2[nH]1 c1(C(N(C)CC2CCN(C(c3c(C)cc(F)cc3)=O)C2)=O)cc(N)cc(O)c1C c1(C(=O)NC(C2CCCN2C(C2CC2C2CC2)=O)C)cccc(C2CC2)c1 c1(C(=O)NCC(C)(Cn2cccn2)NC(C(CC)O)=O)c(CC)oc2ccccc12 C1(C(=O)NC(CNC(C(CSC)O)=O)(C)C)CN2CCN1CC2C C1(CNC(c2ccn(CCCC)n2)=O)CN(C)CCN1C(=O)Cn1ncnn1 N1(C(C2(C)C(C)CN(C(COC(CC)C)=O)C2)=O)CCN(C)C2(CCC2)C1 N1(C(C(c2cc(Cl)cnc2F)CF)=O)CCN(C2CC2)c2c(Cl)cccc21 c1(SCC(=O)NCC(CNC(c2cnn(CCO)c2N)=O)OC)ccccc1F C1(CCC(=O)NCC2(Cl)CCC2)(NC(C(C)n2cnnn2)=O)CCCC1 N1(C(c2cnccn2)C(=O)NC(C(=O)OC)C)CCC2(C1)CN(C)C(=O)CO2 c1(OC)cccnc1C(=O)NCC12CC1CN(C(C13CC(C)(C1)C3)=O)C2 N1(C(CCCOC)=O)CCCCC(NC(=O)C=CC2CCCO2)C1 c1(SC)ccc(C)c(C(=O)NC2CCCCN(C(=O)CC3CCC4CC34)C2)c1 N1(C(c2nnc(CC)s2)=O)CC(NC(c2ncccc2OC)=O)CC2(CC2)C1 c1(C(=O)NCC(CN(C(C2CC(CC)C2)=O)C)O)cccc2[nH]ccc12 c1(C(=O)NC2CCCCCN(C(C(C)O)=O)C2)cn(C)c2ncccc12 C=CCC(C)(C)CC(=O)N1CCC(C(C)C(N2CCC2(C)CC)=O)CC1 N1(C(C(n2cc(-c3c(OC)ccs3)nn2)C)=O)CCOC(c2ccccc2Cl)C1 c1(CC)ccc(C(=O)NCC(C2CCN(C(C3(O)CCOC3)=O)CC2)F)cn1 c1(SC)cc(C(=O)NC2CN(C(=O)CC3CCOC3=O)CC2F)cc(Cl)c1 C(N=c1[nH]nc2cccnn12)C1CN(CC2(CCCC)CC2)C1.N12CC(C1)C2=O c1(NC(c2c(C)cccn2)C)nccc(=NCC2C(F)(F)C23CCC3)[nH]1 C#CCC(CC#C)C(=O)NCC1(O)CN(C(=O)CSCCC#N)C1 C1(CC(=O)N(CCCOCCN(C(=O)CCF)C)C)(C(F)(F)F)CCC1 C(C(C)(C)CNC(C1(OC)CC1)=O)N(C(=O)COCC1CCCOC1)CC N1(C(C(c2cccnc2)NC(CCC(=O)N(C)C)=O)=O)CC2CCCC(C1)N2C C1(C2CC2)(C(=O)NCC2(F)CC(NC(CNC(C)=O)=O)C2)CCOCC1 CC(C)C(C(C)NC(=O)CC(C)(C)C)NC(c1ccnc(C(F)(F)F)c1)=O C1(CNC(CCNC(COC)=O)=O)C2CC1N(C(C13CCCCC1C3)=O)C2 c1(C(=O)NCC2CN(C(C3CC34CC4(F)F)=O)C2)cccc2c3c([nH]c12)CCC3 N1(C(CC(c2cccs2)NC(C)=O)=O)CCN(C(=O)C=C2CC2)C(CO)C1 c1(NC(C2CC(O)CN2C(=O)C2CC2)=O)cnc2cccc([N+](=O)[O-])c2c1 c1(C(N2CCC(O)(C(C)NC(c3nc(CCC)sc3)=O)C2)=O)cnc(O)c(F)c1 C1(C(N(C(C(=O)OC)C)C)=O)(NC(=O)CCc2nccs2)CCC(C)(C)C1 c1(OC)cccc(C=CC(N2CC(NC(C3CC3c3ccsc3)=O)C(C)C2)=O)c1 C1(NC(C2C(C)N(C(=O)Cn3cccc3)CC2)=O)CCC(=O)NC1(C)C C(=O)(C1CCCn2cc(C(C)(C)C)nc21)NC(CCOC)COC C(=O)(CCCCON1CCC(N2CCC(CS(N)(=O)=O)C2)C1)N(C)C CCCCC(C)CCC(=O)NCC(CC(=O)NCC(C)(CO)OC)C1CCC1 C1(CNC(c2ccc(COC)cc2)=O)(NC(=O)CNC(C)=O)CC2CCC1C2 C1(=CC(=O)NCC(CCNC(C2CC=C(C)CC2)=O)O)CCOc2ccccc21 N1(C(COCC=C)=O)CCCC(NC(=O)CCC2CCCC(=O)N2)CCC1 CC(C)C1=NOC(C(=O)NCc2cc(C(=O)NC3(C)CCOCC3)cs2)C1 O=C1CCc2ccc(C(=O)NC3CCC3NC(=O)C(Cl)=CCl)cc2N1 c1(C(=O)NC2(C)CCN(CCCCCC)C2)cccc2occc12 C1(NC(c2ccc[nH]2)=O)CN(C(c2cnn(C3CCC3)c2)=O)CCC1O CC1(C)CC(F)(F)CCC1C(N1CCN(C(=O)CCCNC(N)=O)C2CCC12)=O c1(OC)cc(C)c(C(N2CC3(CCC3NC(=O)CC3CCCC3O)C2)=O)c(C)c1 c1(C(=O)NCC(CC=C)NC(C2C=C(C)CS2)=O)ccc(CO)cc1F c1(CC)cc(C(=O)NC(Cn2cc(C3(O)COC3)nn2)CC(C)C)sc1C NC1CCc2c(C)cccc21.Cc1nn(C)c(Cc2nnnn2C)c1Br C1(OC(C)(C)C)CCCC(CCNC(=O)NCc2cc(=N)[nH]o2)C1 CC(O)C(C(N)=O)NC(c1ccc(CNC(C2CCC=CCC2)=O)cn1)=O N1(C(C2(SC)CC2)=O)CCC2CN(C(=O)C3=NOC(C(C)(C)C)C3)C2C1 CC1CC(c2cn(CC(F)(F)F)nn2)CCN1C(c1cc(Cl)sc1Br)=O CC1CN(C(=O)COCC2CC2)CCC1CNC(c1ccccc1C(N)=O)=O C1(C(=O)NCCCOC(C)C)CCN(C(c2ncnn2C2CCOCC2)=O)CC1 c1(C(=O)NCC2N(C)CCN(C(c3ccsn3)=O)C2)nc2cncnc2nc1O C1(OC)CN(C(=O)CCC2CCCOC2)CC1NC(c1cc(C)cs1)=O N1(CC)C(=O)CCC1C(=O)NCCC(C)CCNC(=O)C(F)(F)C1CC1 C(=O)(CC1COc2ccccc21)N(CC(C)(C)NC(c1ccc([N+](=O)[O-])[nH]1)=O)C Cc1ccc(C)c(OCCC(N2CC3(NC(=O)CC4CC(CF)C4)CC2C3)=O)c1 C1(C)(C(=O)NCC2CC(C(=O)NCC(CC)(O)CC)C2)CC2C=CC1C2 N1(C(C2(OC)CCOCC2)=O)C2CCC1CC(NC(C1(C)CCC(=O)NC1)=O)C2 C12(CCC(=O)OCc3ccn(C)c3)CCC(CC1)C2 c1(NC(=O)NCCC(=O)NCc2ccccc2Br)cccc2c1NCC2 c1(C(N2CCC(NC(CCC=C(C)C)=O)C2C)=O)nc(Br)n2ccccc12 C1(NC(C(CC)C(C)C)=O)CN(C(=O)C(C)(C)C2CCCC2)CC(F)(F)C1 C1(NC(C(C(C)C)N2CCCC2)=O)CCc2nnc(-c3ccccc3)n2C1 N1(C(CSCC=C)=O)CC2CC1CCC2NC(c1ccc(C(C)(C)C)c(Cl)c1)=O N1(C(C2(C#C)CC2)=O)CCC(N(C(=O)Cc2ccn(CC)n2)C)C1 Cn1cc(C(N2CC=CC2CNC(=O)CCN2CCOCC2)=O)cn1 C1(c2n(CCCSC)nnn2)(NC2CCC3(CC2)CSC3)CCCC(C2CC2)C1 c1(CCC(=O)N(CC(C)N(C(=O)Cn2ncnn2)C)C)cccc(Cl)c1 N1(C(c2nc(SC)sc2)=O)CCCCC(NC(c2cncc(N(C)C)c2)=O)C1 CN1C(=O)C(NC(=O)NCC(N2CCCC2C(N)=O)=O)CC1c1ccc(Br)cc1 C(c1cc(F)c(O)c(F)c1)=CC(=O)NC(CNC(c1cnnc(O)c1)=O)C1CC1 c1(CC)ccc(C(=O)NC2CC(C(=O)OC)(CO)C2)nc1.C1C(=O)NCC(=O)O1 N1(C(CCc2ccc(C)o2)=O)CCC(NC(C2CCN2S(C)(=O)=O)=O)C(O)C1 N1(C(CCC=C)C(=O)NCCC#N)Cc2ccc([N+](=O)[O-])cc2C1 N1(C(c2scc(C)c2C)=O)CC2(CCN(C(=O)Cc3ccsn3)CC2)C1C(C)C C12(C(N3CC(NC(C(=O)NC(C)C)=O)C(F)CC3)=O)CC=CCN1CCC2 c1(C(=O)NCC(C)CNC(=O)CCc2ccc(O)c(F)c2)ccc2nn[nH]c2c1 c1(C(N2CCC(CC(C)C)C2)=O)cn2c(n1)CCN(C1CCC(C)(C)C1)CC2 NS(=O)(=O)c1ccc(CC(=O)NCCCCCNC(c2cnnn2C2CC2)=O)s1 N1(c2ccnc(C)n2)CC2CCC(NC(c3coc(C(C)C)n3)=O)CC2C1 c1(CC(=O)NCCOCCNC(=O)Cc2ccns2)ccc([N+](=O)[O-])cc1Cl C(=O)(CC(C(F)F)c1ccc(F)cc1)NC1C(NC(CCC(=C)Cl)=O)C1 C(=O)(C(C)(O)C(C)(C)C)NCC1CC2(CC(NC(c3c(CC)noc3)=O)C2)C1 c1(OC)ccc(C(C)NC(=O)NC2CCC2)cc1SC(C)(C)CC(F)(F)F C1(COC)(CNC(=O)CCC2CC2(Cl)Cl)CCCN1C(=O)Cc1c(C)noc1Cl C1(NC(c2ccc(C#C)cn2)=O)CC2CCCC(C1)N2C(=O)C(F)=C1CCCC1 Cc1ccncc1C=CC(N1CC2C(NC(c3cc(=N)[nH]cc3Br)=O)C2C1)=O C#Cc1ccc(C(=O)NC2(CF)CCN(C(=O)C(C)NS(C)(=O)=O)C2)c(F)c1 CC1CN(C(=O)C(C)N(C)C)CC1CC(=O)NC(C(N)=O)C1CC1 C1(CC(=O)NC2CCN(CCOC)C2)CN(C(C2(N3CCCC3)CC2)=O)CC12CC2 Cc1occ(C(F)(F)F)c1C(N1CC(CNC(c2cn[nH]c2)=O)C(C)C1)=O c1(C(N(CC(C)NC(C=CCC)=O)C)=O)ncnc(C)c1C N1(C(C(CC2CCC2)NC(Cc2c(C)n[nH]c2)=O)=O)CCOC(CN=[N+]=[N-])C1 c1(C(=O)NC(CNC(C2(COCC)CC2)=O)(C)C)nn(C)c(=O)cc1C N1(C(C(COC)(C)OC)=O)CCCCC(NC(C2CC(N3CCCC3)C2)=O)C1 C1(C)(C(N2CC(C)(C(N3CC(C)(N(C)C)C3)=O)C2)=O)CC=CCC1 Cc1c(C(C)NC(C)CC(C)(C)c2ccccc2)cccc1Cl N1(C(C2(C(F)(F)F)CC=CCO2)=O)CCCCC1CC(O)C(F)(F)F c1(C(=O)NC2(C)CN(C(C3(CO)CC(C)(C)C3)=O)C2)cc2ccsc2s1 S(=O)(=O)(CCC(=O)NCC1CCN1C(c1cnc(C(F)(F)F)c(F)c1)=O)NC c1(CNC2CCC(C(=O)NCc3c(OC)cccc3)C2)ccc(Br)cc1O c1(C(=O)NC(CCNC(Cc2c(C)n[nH]c2C)=O)C(C)C)ncc2[nH]ncc2n1 c1(CC)ccc(Cl)c(NC2CN(Cc3cnc(C(F)(F)F)nc3)CC2C)c1 C1(NC(c2cnc(OC)c(C)n2)=O)CCC12CCN(C(=O)C1=C(Cl)CCC1)CC2 Cc1sccc1C(=O)NCC(F)CNC(=O)C(F)(F)C1CCOCC1 C1(CC)CN(C(=O)CC2CCN(C)C2=O)CCN1C(=O)Cc1ccc(OC)nc1 C1(CNC(c2ccc(C)nc2O)=O)CC12CCN(C(C1(CO)CCCO1)=O)CC2 c1(C(=O)NCC2N(C(C3C(OC)CC3)=O)CC2)cc(SC)ccc1C O=C1NC(C(=O)NCCC2(CNC(c3ccc(F)cc3CO)=O)CC2)C2CCC12 C12(CNC(C(c3cccnc3)C)=O)CC(CN1C(=O)CNC(c1cccnc1)=O)C2 C(C(C)(C)C(=O)NC1CC2(C1)CC2NC(=O)CCNS(=O)(=O)C(F)(F)F)OC c1(CCC(=O)NCC2CC(O)CN2C(=O)CN2CC=CC2)cnc2n1CCOC2 C1(NC(c2nc(C(C)OC)sc2)=O)CN(C(c2cc(C3CC3)[nH]n2)=O)C(C)(C)C1 N1(C(C(C)c2ccsc2)=O)CCC2(CCCCN(C(=O)C(C)c3cc[nH]n3)C2)C1 N1(C(CN(C)C(C2(CS(N)(=O)=O)COC2)=O)=O)CCCCC1CO c1(OC)cc(O)ncc1-c1nc(C2(Oc3ccccc3)CC2)nn1CC1CCOC1 C1(C#N)(C(=O)NC2(C)CCN(C(C3CCCS3)=O)C2)CC2CCC1CC2 C(CC(C(=O)NC(C)(C)CN(C(=O)CCc1ccco1)C)OC)OC C=CC1(C(=O)NC2CCC(CNC(=O)Cn3cnc([N+](=O)[O-])n3)C2)CCCCC1 C1(NC(=O)Nc2c(OCC)ccs2)CCCCCC1c1ccccc1 CC1CN(Cc2ncc(Cl)nc2Cl)CCN1C(C1CCC(=O)N1C)=O c1(C(=O)NCCC(Cn2cc(CC(COC)O)nn2)F)ccc(F)c(OC)c1 C1(CN(C(c2ccn(C3CC3)c2C)=O)CC)CCN(C(=O)C2=CCC2)CC1 c1(C(=O)NCCC2CCCN2C(=O)C(F)OC(F)(F)F)cnc2n1CCOC2 C=CCCC(C)(C)CNC(=N)NC(C(CC)CC)c1ccccc1 N1(C(c2ccc(NC(c3cc(I)ccc3F)C)nc2)=O)Cc2ccccc2C1 N1(C(C2C3(CCN(C(CC(C)F)=O)CC3)C2)=O)CCc2ccncc2C1 c1(NC(c2ccncc2F)C)cc(NCC(N2CCCCCC2)(C)C)ncn1 CC(C)CC(C)(CNC(=O)CCOC1CCCC1)NC(C1CCC1C(C)(C)C)=O Cc1nc(C(C(C)C)NC(=O)CC2CC3CC3C2)no1 C(=O)(CC1=NN(C)C(=O)C1)N(C)CC1(O)CCCN(C(C(C)SC(C)C)=O)C1 CC1CN(C(c2ccnc3ccnn23)=O)CCCN1C(C1CC=CCC1)=O N1(Cc2cn(CCC)nc2)CC(NC(c2cc(Cl)c(Cl)nc2Cl)=O)CC(F)(F)C1 C1(NC(C(c2n(C)ccc2)=O)=O)CS(=O)(=O)CC1NC(C1CCC1)=O C(=O)(C(CC(C)C)C(C)C)NCC#CCNC(c1c(C)nc(N)cn1)=O N1(CC(=O)NC(C2CCCN2C(c2conc2C(F)(F)F)=O)C)CCC(C)(O)C1 C(C)(CC(=O)N1CC(F)(CNC(C2(C)CC2(F)F)=O)C1)(C(F)F)N(C)C Brc1ccc(CN2CCOCC2)c(N2CCOC(c3cccs3)C2)c1 N1(C(C(CCC)c2ccccc2)=O)CCCC(NC(=O)C(F)(F)COC)C1C C1(C(N2CCC(O)(CCNC(C(CC)C#N)=O)CC2)=O)CCC2(CCOCC2)O1 c1(C(=O)NCCc2c(OC)c(Cl)ccc2)ccc2nc(F)ccc2c1O c1(C(N2C(C(=O)NCC(C)(O)CCO)CC(C)C2)=O)ccc2n[nH]cc2c1 c1(CNC2C3CN(C(C4CCC(OC)CC4)=O)CC32)cc(C)c(Br)cc1F N1(C(CCCCC)=O)CC2CCN(C(c3c(C)ccc(Cl)c3F)=O)CCC2C1 CCC(CC(=O)NC(C)C(C)(C)CO)N(C(=O)C=CC1(C)COC1)C Cc1ccc2[nH]c(C(N3CCC=C(CNC(C4CCO4)=O)C3)=O)cc2c1 CCCC(O)CC(=O)NC1CN(C(C2(c3cccs3)CC2)=O)CC1C c1(C(=O)NC(C2(O)CN(C(COC)=O)C2)C)cc2c(Br)c(F)ccc2[nH]1 C(=O)(CC(C(F)(F)F)P(C)(C)=O)NC(C(C)NC(CCC(C)C)=O)C Cn1ncc2cc(C(=O)NCC34CC3CN(C(c3cc(N)cnc3Cl)=O)C4)sc12 c1(OC)cc(OC)cc(C(=O)NC2COCC2NC(C2CC2(F)F)=O)c1 C(N=c1[nH]c(=NC(C)c2ccc(Br)c(F)c2)[nH]c2c1SCC2)c1cc(C)on1 C(C1CC1)(C1CC1)=CC(N1CCC(OC(C(=O)N(CC(F)F)C(C)C)=O)C1)=O c1(C(=O)NCCCCC(C)NC(C(CCC)C)=O)ccc(N2CCC(C)=N2)cc1 C1(NC(c2c(C)sc(Br)n2)=O)CN(C(=O)C=C(Cl)Cl)CCC1C N1(C(C2CC2CNC(C2(NC(C)=O)CC2)=O)=O)CCCN(C=O)CC1 N1(C(=O)NCc2c(COC)ocn2)CC=C(c2cccc(C)c2C)CC1 C1(CNC(CCCC#C)=O)CN(C(=O)Cc2cc(F)cc(F)c2)C(C)(C)C1 N1(C(C(CC)C#N)=O)CCOC(C)(CNC(=O)COc2ccn(C)n2)C1 Cc1c(C(=O)NC(C)C(C)NC(c2cncc(F)c2)=O)cccc1C#N C(=O)(CC(C)C(F)F)N1CC(OC)C(C(=O)NCc2cccc(C)c2O)C1 C(CCC(=O)NCCc1ocnc1CNC(C1(C)CC1(F)F)=O)OCC=C C(CCCC(=O)N(C)CC1CCCN(C(=O)CCSc2ccccn2)C1)OC N1(C(C2=NOC(C)C2)=O)CCN(C(=O)Cn2ncccc2=O)CC(O)C1 c1(C(=O)NC2CCN(C(C(C)(C)Cc3ccccc3)=O)C2)nccc2[nH]ccc12 C(C(CNC(=O)C(Cc1ccco1)NC(=O)CSc1ccccn1)C(C)C)OC c1(OC)ccc(C(=O)C(=O)NCC2CCC(C)CN2C(c2cccs2)=O)cc1Cl c1(C(=O)NCC(CNC(c2cc(OC)ns2)=O)C(F)(F)F)ccn2nncc2c1 c1(OC)cncnc1C(=O)NC1COCCC1NC(C1C(C)C1C)=O C1(n2cc(COC)nn2)CCN(C(c2c[nH]nc2-c2cccnc2)=O)CC1O N1(C(c2cnn(C)n2)=O)CCC(O)(CNC(c2nccc(C(F)(F)F)n2)=O)C1 c1(OC)c(O)cc(C(N2CCCC2C(=O)Nc2cnc(C)c(Br)c2C)=O)cc1O C12(C(N3CCC(O)(CN(C(C(CCN(C)C)O)=O)C)C3)=O)CCC(O)(CC1)CC2 C(=O)(C(C)C(O)C(C)C)NC(CC=C)CC(=O)NC(C)(CO)C1CCCC1 C(=O)(C1CCCc2sccc21)NCC(C)N(C(c1c(C)n2c(nc1)ncn2)=O)C N1(C(CC2(C=C)CC2)=O)CCC(O)(CNC(c2cnc(C(C)(C)C)[nH]2)=O)C1 C1(C(=O)NCCn2ncc(C)c2)CN(C(=O)CC23CCCC2C3)C(C)(C)C1 c1(OC)cc(OC)c(Cl)c(C(N2CC3(NC(=O)C(C)N4CCC4)CC2C3)=O)c1 CC1(C#N)CCN(C(C2CC3C=CC2N(C(c2c[nH]nc2C2CC2)=O)C3)=O)CC1 CC1C2CCC(C2)C1C(N1CC2(C)CC1(C(=O)NC1CCCCCC1CO)C2)=O c1(C(=O)NC)cc(S(=O)(=O)NCC2(O)CCOCC2)cn1C C=CC(C)C(=O)N(CC(CC)NC(=O)CCc1cncn1C)C C(=O)(C(CO)C(F)(F)F)NC1CC(C(=O)NC(C2CCCO2)CC)C1 Cc1cc(O)c(C(=O)NCCCC(=O)N(C)C)cc1F Nc1c(C(=O)OCC(=O)NCC(C2CCOC2)O)ccc(Cl)c1Cl C(CC(C)C)(C(=O)NC(CNC(C1(CF)CCC1)=O)C(C)(C)C)NC(C)=O CC1CCN(c2nccnc2F)CC1NC(c1ccccc1C(F)F)=O C(c1cc(OC)cc(OC)c1)=CC(=O)NC(C(C)NC(C(CC)CC)=O)C C1(C)(C(=O)NC(C(=O)OCCC)C)CC(O)CN1C(=O)CCc1cc(C)on1 c1(CC(=O)N(CCN(C(c2c(NC)cnnc2)=O)C)C(C)C)csc2nccn12 C1(C)(NC(c2nnnn2C2CCC(C(=O)NC(C)C)C2)(COC)C)CCCC1 C1(C(=O)NCC2(C(=O)Nc3nnc(O)o3)CC(=C)C2)CSCC(=O)N1 C1(NC(c2c(OC)nsc2)=O)(CO)CCCN(C(c2n[nH]cc2C)=O)C1 N1(C(c2cc(C)[nH]c2)=O)CCC(NC(C2CCC(C3CC3)CC2)=O)CC(C)(C)C1 C(=O)(CCCCCCN=[N+]=[N-])N(CCCCCCNC(=O)CC1CCC1(C)C)C c1(C(=O)NC(C=C)COC)nc(CNC(C2(C#N)CCCO2)=O)oc1C N1(C(c2cc(CC)no2)=O)C2CCCC1CN(C(c1c[nH]c(C)c1)=O)C2 c1(N2CC(C(C)NC(C(c3cccnc3)OC)=O)C2)nn2cc(C)nc2s1 N1(C(c2c(C)oc(CO)c2)=O)CC(N(C)C(C2(F)CCCCC2)=O)C(C)(C)C1 C1(C(=O)NCCN(CCOC)C(c2cc(Cl)ncc2O)=O)CC2COCC(C1)C2 N1(C(c2c(C)cc[nH]2)=O)CC2(CCN(C(C3CC3c3ccccn3)=O)CC2)C1 N1(C(C2CCSCC2)=O)CC2CCC1C(CNC(C13CCCN1CCC3)=O)C2 N1(C(CC(COC)C)=O)CCN(C)C(C(N2CC(CO)C2(C)C)=O)C1 C1(NC(C2(OC)CCOCC2)=O)CC1C1CCCN(C(=O)CCC2CCOC2)C1 Cc1cc(Cl)ccc1Nc1ccc(C(=O)NC2CC2NC(=O)C(C)N(C)C)nc1 C1(NC(c2cnnc(Cl)c2)=O)CCCCC1NC(c1occc1Br)=O C1(C(=O)NCC(C)C)COCCN1C(c1cnc(Br)s1)=O C1(C(=O)NC(CC)CNC(c2nnsc2C)=O)CCCCC1O N1(C(CCC2CC(OC)C2)=O)CCCC(CCNC(=O)CCCN(C)C)C1 c1(Sc2n(C)ccn2)ccccc1NC(=O)NCC1(C)CNC(=O)O1 C1(C(C)NC(C2(CCOC)CCC2)=O)CCCN(c2nnc(C#N)s2)C1 C1(C(N2CC(COC)(CNC(c3ccc(C)s3)=O)C2)=O)CCS(=O)(=O)C1(C)C N1(C(C=CCN(CC)CC)=O)CC=CC1(C)C(=O)NCc1cn(CC2CC2)nn1 c1(CCC(N2CCN(C(C3CC3(F)F)=O)C3CC23)=O)c[nH]c2ccccc12 c1(C(=O)NCc2c(C(=O)NC3C(CN(C)C)CCC3)scc2)ccc(N)c(F)n1 N1(C(CCCCN(C)C)=O)CCCC(C2(NC(=O)C3Cc4ccccc43)CC2)C1 C1(C)(NC(c2ccn(C)n2)=O)CCC(NC(c2c(Cl)cccc2Cl)=O)CC1 c1(C(N(C)CCNC(C2(Cl)CC2(C)C)=O)=O)cc(Br)cc([N+](=O)[O-])c1 Cc1ncnc(O)c1CCC(=O)NCC(C)(CO)NC(C12COCC1C2)=O C1(F)(C(=O)NCC(C)(C)NC(c2cc(OC(F)F)n(C)n2)=O)C2CCCCC12 O(C1CCc2cc(Br)cnc21)C(C(c1cccc(F)c1)C)=O C(=O)(C(C(C)O)N(C)C)N(CCNC(c1cc(CC)n[nH]1)=O)C N1(C(Cc2c(C)noc2)=O)CC(NC(=O)Cc2ccc(Br)c(F)c2)C2(CC2)C1 c1(C(C(=O)N(C2C3CN(C(=O)Nc4ccccc4F)CC23)C)O)cccc(Cl)c1 C1(C(=O)NCC(c2ccncc2)O)(CC)CCCN(C(=O)C=Cc2ccoc2)C1 c1(C(N2CC(CNC(C(CC=C)OC)=O)(OC)C2)=O)ccc(N)cc1Br C1(CCCCC)CCC(C(N2CC(O)CC2C(=O)Nc2ncc(F)cn2)=O)CC1 N1(C(CN2C(=O)CSC2)=O)CCN(C(c2cccc3cc[nH]c23)=O)C2CCC12 c1(CC)[nH]nc(C(N2CCCC2CN(C(C2C=CC=CC=C2)=O)C2CC2)=O)c1Cl N1(C(C2C(C(C)C)C2)=O)CCC(C(F)(F)F)C(CNC(=O)C2=CC(C)(C)C2)C1 c1(C(C)Oc2ncc(NS(=O)(=O)CC3(N(C)C)CC3)s2)ccc(Br)cc1 C1(C(=O)NCCc2cn(C)nc2)CC(O)CN1C(=O)CC1CC2CC2C1 O=C(O)CC(c1ccccn1)NC(=O)C(c1ccccc1)OCCn1cnnn1 Cn1nncc1C(c1cnc(CC(F)(F)F)s1)=O C1(CC)C(NC(=O)C=C(C)C2CC2)CCN1C(=O)CCCOc1ccc(C)cc1 Cc1ccc(NC(C2(C)CC(NC(=O)C(Cl)Cl)C2)=O)c(C)c1 N1(C(C2(n3ccnn3)CC2)=O)CCCC1.O=C1CC2(CC2)CO1 N(C(=NCCSc1nccn1C)NCC1CCCC(=O)N1)C(c1ncccn1)C c1(C(=O)NC2CC(C)C2)cnc2nc(NS(=O)(=O)C3CCCCC3)ccc2c1 C1(C(C)NC(C2(SCC)CC2)=O)CCN(C(=O)Cn2ccc(C)c2)CC1 c1(C(C)C)nocc1C(=O)NCC(C1(O)CN(C(=O)CN2CC3CC3C2)C1)(C)C c1(OC)cccc(C(C)CC(=O)NC2(CO)CN(c3ncc(C)cn3)C2)c1 C=C1COCCN(C(c2cnc(C(F)F)s2)C(=O)NC2(C)CC2)C1 N1(C(c2c(OC)ccnc2)=O)CC2(C(N3CC4(C)CC3CCO4)=O)CCC1CC2 c1(CCC(=O)NCCC(C)NC(=O)C(C)(C)CO)ccc(Cl)cc1Br C#Cc1ccc(C)c(NC(C2CC3CC3N2C(c2cnn(CC)c2)=O)=O)c1 c1(C(N2CCN(C(C(C(C)C)SCC)=O)C(C)C2)=O)ccc2c(C)noc2n1 C(=O)(C#CC1(C)COC1)NCC(C)NC(c1ccc(C(F)(F)F)[nH]1)=O CC1(C)C2CCC1(C(N1CCC(OC3CCOCC3)C1)=O)C2 CC1C(=O)N(CC(=O)OCCC2CCC(C)C2)C(=O)C1C C(=O)(C(C)S(=O)(=O)C(C)C)N(CC(C)NC(c1c(NCC)ccc(Cl)c1)=O)C N1(C(C2CC(C(C)C)C2)=O)CCC(N(C)C(c2coc(CC3CC3)n2)=O)C1 N1(C(C(CC)N(CC)CC)=O)CCC(C2(NC(=O)C(COC)OC)CC2)C1 C1(NC(C=CCC)=O)CC2CCC1(C(=O)NCC1(OCCO)CCCC1)C2 CC1CC(CNC(C2CCC(CNC(=O)COCC3CC3)CC2)=O)CCS1 c1(CC)noc(CC)c1CC(N1CC(O)(C(C)NC(c2ncnn2C)=O)C1)=O N1(CC)C(=O)CCC1CC(=O)N(C)CC1CN(C(c2cc(C3CC3)ccn2)=O)C1 N1(C(CCC=C)=O)CCOCC(CNC(c2nn(C)nc2Br)=O)C1 C(CCO)(C(F)F)N(C(C(C1(O)CCC1)NC(CCC)=O)=O)C C1(C(=O)NC2C=CCCCC2)Cc2c[nH]nc2CN1 Cc1cc(C(=O)NC2C=CC(C(=O)NCCC3CC=CC3)C2)[nH]c1C c1(OC)ccc2c(N(C3CCNCC3F)C(c3ccc(Cl)c(O)c3)=O)ncnc2c1 Cc1c(OC(F)(F)F)cccc1C(=O)N(C1CCCNC1)C N1(C(c2ccc(OC)nc2)=O)CCC(C2CCN(C(=O)C(C)P(C)(C)=O)CC2)C1 c1(OC)ccc(C2CCCN2C(c2ccc(C3CCOC3)cc2)=O)cc1OC N1(C(CCOC(C)C)=O)CCN(C(c2ccccc2C(F)(F)F)=O)CC(O)C1 N(C(=NCC(C)C)N1CCC2(CC(C(F)F)=NO2)C1)CCc1ccc(CC)cc1 c1(C(C)C)ccc(NC(C2CC(NC(=O)Cc3cccc(F)c3)C(O)C2)=O)cc1 c1(SCC)ccccc1C(=O)N(CC(C)CNC(C1CC1c1nccn1C)=O)C c1(CC(=O)NC2CC(NC(CC3C(OC)CC3)=O)C2)cccc(OCC#N)c1 N=c1nnn(CC(=O)NC(c2ccccc2)CNC(c2nn[nH]c2Cl)=O)[nH]1 c1(OC)nn(C)cc1C(N1CCCC1(C(=O)NC1(CF)CC1)C(C)C)=O O=C(C#CC1CCCC1)NC1COCCN(C(=O)CN2CCSCC2)C1 CCCC(C)CC(=O)N1CC2(CNC(C3CN(C)C3)=O)CCC1C2 C(=O)(CCC(O)C(C)(C)C)N1CCC(CNC(Cc2cnc(C)o2)=O)C1 c1(CC)cccc(NC(C2(NC(=O)CC3CCCC3C)CC2)=O)c1 c1(C(N2CC(CC)N(C(=O)C3=CCSC3)CC2)=O)cnc2n1CCOC2 CCC(C)C(C)(O)CNC(=O)CCC(C)(C)NC(c1cnc(C)nc1)=O CP(C)(=O)CC(=O)NCC1(O)CN(C(c2cc(CCCO)on2)=O)C1 c1(OC(C)C)cccnc1C(=O)NC1CCC1NC(=O)C=Cc1cscn1 O=C1NCC(C(=O)NCC#CCNC(=O)CCCn2cccn2)N1 C#Cc1ccc(CC(N2CCC(NC(=O)C=C3CCN(C)CC3)C(O)C2)=O)cc1 c1(NCC2(CNC(c3nnn4ccccc34)=O)CC2)c(Br)cccc1[N+](=O)[O-] C(C(=O)N1CC(O)CCO1)N(C(C)CC(N(C)C[Si](C)(C)C)=O)C C#Cc1cccc(C(N2CCOCC2CNC(C2CC2C=C)=O)=O)c1Cl c1(OC)c(C(=O)NCC2CN(C(=O)C(C3CCCOC3)OC)C2)cccc1Cl C(=O)(CC(C(F)F)n1ccnc1)NCCC(C(C)C)NC(=O)CCCOC(C)C O=C(C1=C(Cl)CCC1)NC1CC(NC(c2cccc(-n3cncn3)c2)=O)CC1O c1(NC(C(C2C3CCCC23)N(C2CCC2(C)C)C)=O)ccc(F)cc1 N1(C=O)CC(N(C)C)CC(C)C1.c1(NC(C)=O)ccc(CN(C)C)cc1 C(C1=NOC2CN(C(c3scc(C)c3OC)=O)CC12)NC(COCC=C)=O c1(C(N(CC(C)NC(C2(N=[N+]=[N-])CC2)=O)CC)=O)cccc([N+](=O)[O-])c1Cl c1(OC)noc(C)c1C(=O)NC(C)CCCCNC(c1cc(C(C)=O)c(C)o1)=O C(CC(C)C(=O)N1CCC(C)C1C(=O)NCCN1CCC(OC)C1)=CC c1(NC)cc(C(N2CCC(NC(C3CCN(CC(C)C)CC3)=O)C2)=O)cc(Cl)n1 C1(OCC)COCCC1CC(N1CCCC1CNC(=O)CC1CCCC1)=O C(C(C)CC(C)O)NC(=O)NC(c1ncn(-c2ccccc2)n1)C C1(C(=O)NC2CN(C(c3cc(CCC)n(C)n3)=O)CC2C)CN2CCN1CC2 C1(C(=O)NC)CC(C)CN(C(c2cnccc2)=O)C1.n12cc(nn1)CNC(=O)C2 CC1=NOC(C(N2CC(O)(CCNC(=O)C(C)Sc3ccccn3)C2)=O)C1 C(=O)(NNC(=O)C(=O)NC(C)CC1CCCCC1)NCC1CC(C)CC(C)C1 C1(NC(c2c(CC)nccc2)=O)CN(C(=O)C2=CCSC2)C2(CCCC2)C1 c1(CCC)sc(C(=O)NC(C)(CNC(=O)C(C)c2ccsc2)CO)cc1CC C12(CC)CC(NC(c3cc(CNC(=O)C(C)n4cncn4)on3)=O)(CO1)C2 C1(C2CC2)(CNC(CN(C)C2CC2)=O)CCN(C(c2cnsc2)=O)C1 C(=O)(CCCC(=O)N(C)C)N(CC(CNC(C1(C)C(C(=O)OCC)CC1)=O)O)C O=C(C#CC1CCCCO1)NC1CCC2(CC1)CC(NC(=O)C1=NNC(=O)C1)C2 C1(CCNC(C2(CC)CC2(F)F)=O)CN(C(c2cncnc2C2CC2)=O)CCO1 C(CC(C)(c1nnnn1C1CCCC1)NCCCCO)(OC)OC c1(C(=O)OCCSCc2cccc(OC)c2)ccc(F)c(C(F)(F)F)c1 O=C(N=c1nc(O)[nH]c(O)n1)c1[nH]nc2cc(-c3ccc(F)c(CO)c3)ccc12 CN(NC(=O)NCc1ccc(C2(C)NC(=O)NC2=O)cc1)c1cnccn1 C12(NC(c3c(Cl)ccc(OC)n3)=O)CCCC1N(c1nnco1)CCC2 c1(C(=O)NCC23C(CN(C(C4(NC(C)C)CC4)=O)C2)C3)nccn2ccnc12 N1(C(CC(CC)OC)=O)CCC2CN(C(c3ncc(C)cc3OC)=O)CCC12 N1(C(c2c(C)onc2Br)=O)CCN(C(C2CC2F)=O)C(CO)C1 C(=O)(C(C)(C)CN1CCOCC1)NCC(C)N(C(CCN(CC)CC)=O)C C#Cc1ccc(C(N2CC3(CC3)CC2C(=O)Nc2cnccc2CC)=O)c(C)c1 C1(NC(c2n(CC)ncc2)=O)CC=CCC1C(=O)NCC(O)C(F)(F)F CC1(CNC(=O)Cn2ncccc2=O)CCC(NC(C2CN(C3CCC3)C2)=O)C1 Cc1nn(C)cc1C1CCC(CO)N1C(=O)CCc1cccc(Cl)c1 N1(C(CCOCC#C)=O)CCSCC1CCNC(c1cc(C)n(C)n1)=O C1(CCC(=O)NCC(C)(C2CCC2)NC(=O)C2=CCOC2)CCCC(O)C1 N1(C(c2ncn(CC)c2)=O)CCCN(C(=O)Cc2ccc(C)cc2F)CC1 c1(C(=O)NCC(C)(O)C)cc(Cl)n[nH]c1=N.C1(CC)CC1CC(=O)NCC=O Cc1cc(C(=O)NCC2(CNC(C3(C#N)CCC3)=O)CC2)ccn1 CC(C)(C)C(O)C(=O)NCC(C)(C1CC1)NC(c1cc(Cl)cc(Cl)c1)=O C1(CNC(CCOC)(C)c2nnnn2C(C)(C)C)(CO)COCC2CCCCN12 c1(OC)cccc2c(C(N3CCCC(NC(=O)COC4CCOC4)C3)=O)coc12 C1(NC(c2n(CC)cc(Cl)c2)=O)CC2CCC1C(NC(=O)CC1COCC1O)C2 C#CCC(C)(C(=O)NC(CCC)CCO)NC(c1cccc(CO)n1)=O C12(NC(CC(CC=C)NC(=O)Cc3cc(C)cs3)=O)CC3CC(CC1C3)C2 c1(OC)ccc(C2(NC(c3cnn(CC(C)C)c3)=O)CCOCC2)cc1Br C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCC2C(NC(CS(CC)(=O)=O)=O)C21 C1(C(=O)NC2C3CC2CN(C(=O)C=Cc2nccs2)C3)CC2C=CC1C21CC1 C(CN=c1[nH]c(C2CC2)nc2c1CCC2)NC(=O)NC1COC(=O)O1 C(=O)(C1=CCC(C)(C)CC1)NCC1(C(=O)Nc2c(Br)cn(C)n2)CC1 C1(CC)C(NC(C2CC(N(C)C)C2)=O)CCN1C(c1csc(C2CCCO2)n1)=O C(C1CCOCC1)=CC(=O)NCC(C(C)C)NC(=O)Cc1ccn(C)n1 c1(C(=O)NC(CNC(C(=O)NCCOC)=O)CCOC)cccc(F)c1Cl C1(CC(=O)NC2(CC=CC)CC2)CCCCN1C(c1nnc(S)n1C)=O C(C(C)CCCC(C)C)NC(CC1(C)N(C(c2c(CC)nns2)=O)CC1)=O C(=O)(C1=CCC2(COC2)OC1)NC1C(NC(c2cc(OC)c(C)cc2)=O)C1 c1(C(N2CCC(C(C)(C)NC(C3CC34CCCC4)=O)CC2)=O)ncc(Cl)cc1Cl C1(C(N2CC(CC)C2)=O)CC(O)CN1C(=O)CCCCNC(=O)C1CC1 c1(OCC)cc(F)c(-c2ccc(NCc3ccc(NC(C)=O)cc3)nc2)cc1F c1(C(=O)NCC2CCN2C(=O)CCOC2CC2)c(C(F)(F)F)nc2n1CCCC2 N1(C(C2CC(SC)C2)=O)CCOCC1.C1(=O)CSCC(=O)NC2(CC2)CC1=O c1(OC)cccc(O)c1C(N1CCCC(CO)(NC(=O)CC2CCCCC2)C1)=O c1(NC(C2(CNC(c3ncoc3C)=O)CC(=C)C2)=O)cn(CC)nc1C#N C12(C(=O)OC)COCCC1(F)CN(C(=O)NCc1ccnc(S(N)(=O)=O)c1)C2 C1(C(N2CCC(=C)C2)=O)CC1C1CN(C(=O)CC2CCCCN2C)C1 CC(CS(C)=O)C(=O)NC1CCCCC1NC(c1cc(O)nc(N(C)C)n1)=O C1(OC)CC(CNC(c2ccsc2Cl)=O)N(C(C2CC(=O)CCO2)=O)C1 c1(C(=O)NC2(CO)CCN(C(=O)CCc3cncs3)C2)cc2ccccc2[nH]1 c1(C(=O)NC(CC)CNC(=O)C=CC(=O)N(C)C)cccc(C(C)(F)F)n1 C1(C2CCN(C(C3(CO)COC3)=O)C2)(NC(C(CC(C)C)OC)=O)CC1 n1(C(CC)(C)C)nnnc1C(c1ccc(C)o1)NC(C)CCc1cn[nH]c1 C1(NCC2OCC(CC(=O)OC)C2)CCCN(CC#C[Si](C)(C)C)C1 C1(NC(CC(CC)O)=O)CCN(C(C2(N3CCCCC3=O)CC2)=O)CC1C C1(OC)CN(C(=O)C(F)=CC2CC2)C(C)(CNC(=O)C=CC2CC2)C1 C(CCCC(=O)O)n1cc(CN(CC(c2ccccc2OCC(F)F)O)C)nn1 C(=O)(C1=NN2CCCN=C2N1)NC(CCN(C)C(c1cc(Cl)ns1)=O)C(C)(C)C C1(NC(Cc2cn(CC)nc2)=O)CC(F)CN(C(=O)CN2CCOCC2=O)C1 C1(C(=O)NCC2(NC(c3[nH]c(=NC)sc3)=O)CCOCC2)COC2(CCC2)CO1 N1(C(C(N2CCSCC2)C)=O)CCCCC2(CCN(C(c3ccc(Br)o3)=O)C2)C1 c1(NC(c2ccc(OC(C)C)cc2)=O)cc(C2=CCC(O)CC2)ccn1 c1(C(=O)OC)nn(C)cc1S(=O)(=O)NC1CC(CCC(N)=O)C1 c1(OC)ncc(Cl)cc1C(=O)NCC1CCN(C(c2ccn(C)c2)=O)C12CC2 C1(OC)CC(CNC(=O)COCc2ncc(C)o2)N(C(=O)CC(C)F)C1 N1(CCN(C2CCCCC2)Cc2cccc(C)c2)Cc2ccccc2CC1CO c1(NC(C)=O)ccc(C(=O)N(C(C)CCNC(=O)C2=CCCS2)C)nc1 C(=O)(CC(F)(F)F)NCCCC(C)NC(C1CCC(c2ccccc2)O1)=O O=C(C1=CCSC1)NCCC1CC(NC(c2ccnc(-c3ncc[nH]3)c2)=O)C1 c1(C(N2CC(=O)NCC2C(N2CCC2CF)=O)=O)cccc2[nH]ncc12 N1(C(c2n(C(C)C)ncc2)=O)CCC(CNC(=O)CC2CCCCC2)CC1C N1(CCC(N2CC(CC(C)NC(=O)CCF)C2)=O)Cc2ccccc2C1=O c1(C(=O)NC(CNC(c2onc(CC)c2C)=O)C)ccc2c(c1)C(=O)OC2 c1(C(=O)NCCCCNC(C(C)(C)N(C)C)=O)ccc(S(C)(=O)=O)o1 C(CCC(=O)NC(C)CCNC(=O)Cc1csc(C(F)(F)F)n1)=CC CC(C)C(C(=O)NCCC(C)NC(c1cnccn1)=O)c1cnn(C)c1 N1(C(C(C)C2CCCO2)=O)CCN(C(C2CC(O)C2)=O)C(C)C1 C#Cc1ccc(C(=O)NC2CC2NC(=O)C(C)CN2CCOCC2)cc1Cl C1(CNC(c2c(CC)nc[nH]2)=O)CCN(C(=O)CSc2cccc(Cl)c2)CC1C c1(NC(C2CCN(Cc3ccc(OC)cc3Br)C2)=O)ccc2c(c1)c(Br)nn2C C(=O)(C(O)CC(C)(C)C)NC1CC(NC(C(C)(C)OCC)=O)C1 c1(C(CNCC2(C(=O)NCCOCC)CC2(F)F)C)ccc([N+](=O)[O-])c(OC)c1 N1(C(c2cnc(Cl)cn2)=O)CC2CCN(C(=O)COCC(F)(F)F)C2C1 c1(CC)c(C(=O)N(CCCCN(C)C(C2CCCN(C)C2)=O)C)ccn1C CC1CCCC1(C)NC(=O)NCC(=O)N(C(F)C(=O)O)C1CCCC1 C(N=c1[nH]cc(Cl)c(C)c1C#N)C1CN(C(C(C(CC)C)C)=O)C1 CN(Cc1ccc(N2CCCC(C(N)=O)C2)cc1)N1CC2(CC=CC2)C1C(=O)O N1(C(c2c(CC)ocn2)=O)CCOC2(CCN(C(C3CCCC34CC4)=O)CC2)C1 c1(C(=O)NC(CNC(C(C)OCC(F)(F)F)=O)C(C)(C)C)c(NC)cccc1F C(CN=c1ncc(C(C)(C)O)c[nH]1)CCN(C(=O)CC1CCn2cncc2C1)C C1(C(=O)NC2CC(NC(C(C3CCCC3)OC)=O)C2)CCC(=O)O1 C(=O)(CS(=O)(=O)CC(F)(F)F)NC(CN(C(c1c(CC)ccc(OC)c1)=O)C)C CC#CCC(C(=O)N(CC)CC1CCOCC1)NC(=O)C(C)C(C)(C)C C12(CNC(C(C)(O)C3CCC3)=O)CCCCC1N(c1nccc(C#N)n1)CC2 N1(C(c2c(CC)ccs2)=O)CCCC(NC(c2c(C)noc2C)=O)C(F)C1 c1(CC(C(=O)NCC(C)CNC(c2cn(C)nn2)=O)O)ccc(F)cc1 c1(C(=O)NCC(CN(C(c2c(C)cns2)=O)C)C)cccc(NC(=O)N(C)C)c1 C(C)(CNC(c1cc(C(N)=O)cn1C)=O)(CC(C)C)NC(c1[nH]cc(C)c1)=O N1(C(c2c(CCC)n(CC)nn2)=O)CCN(C(=O)CO)C(C2CC2)C1 n1(CC(=O)N(C2CCN(C(C(C)(C3CC3)OC)=O)C2)CC)nnc2c1CCCC2 C12(C(=O)NC(CCOC)C(=O)NC(C)Cc3nn[nH]n3)CCCC1OCC2 Cc1[nH]c(CN2C(C(N3CC(O)CC3CO)=O)CCC2C)c(C)c1C(=O)O N1(C(c2cccc(OCc3ccc(F)cc3)n2)=O)CCCC2(CCNC2)CC1 C1(OC)CC(C(N2CC(C(C)NC(=O)CSC)C2)=O)CC1OC N(C(=NCCCCl)NCCN1CCCCCC1)C(c1cc(F)cnc1Cl)C C=CCC(C)C(=O)N(C1CCN(C(=O)CNC(=O)Cc2cccc(F)c2)CC1)C n1(CC)nc(C(=O)NC(CC2CC2)CC(=O)NCc2ccc(C)s2)cc1C N1(C(c2ccc(COC)s2)=O)CC(NC(=O)C=C(C)c2ccsc2)CCC(O)C1 Cc1ncccc1C=CC(=O)NC(C)CN(C(=O)C(c1cccc(O)c1)C)C c1(C(=O)NC(C)CC2CN(C(C3(CO)CCC3)=O)C2)nn(C)c2c1C(O)CCC2 N1(C(c2ccn(C)n2)=O)CC2CC(NC(C3(c4ccnn4C)CC3)=O)CC2C1 c1(C(=O)NCC2CCC3(CN(C(C(=O)NCC)=O)C3)O2)cc(C)ccc1S(N)(=O)=O c1(C(c2n(CC)nnn2)NCCC=C(Cl)Cl)cc(F)cc(Br)c1 C(C(COC)CC(=O)NCC1CN(C(C2(C(C)(F)F)CC2)=O)CCCO1)OC c1(C(=O)NC2CCN(C(C(C)NC(=O)OC)=O)CC2C)ccc2ocnc2c1 c1(OC)ccccc1C1CCN(C(=O)C(N)Cc2nc(C(C)C)no2)CC1 c1(CC)ccc(F)c(C(=O)NCC(C)N(C)C(c2cnsc2C)=O)c1F C(=O)(C(Cc1ccccc1)CC(C)C)N1CCN(C(C(=O)OCC)C)CC1 C(CCC(=O)N(C)CC=CC(=O)NC1CC1Cl)N(C(C)C)C CCC(COC)(C(=O)O)NS(=O)(=O)CCCCOc1ccccc1 CC(CC(C)(C)C)C(=O)N(CC(Cc1ccccc1)NC(=O)CC(C)(C)C)C C(=O)(CC(CC)CC)NCC1C(C(=O)NCCC)CCC1 C1(CNC(COCC(C)C)=O)(CNC(=O)Cc2ccco2)CC1(F)F C(C1CCCc2ccccc21)NC(=O)Nc1nc(C)c(-c2cccs2)cc1 C(=O)(C(CNC(=O)CC(F)(F)F)CC(C)C)N(CCCC)CC CC1CCN(C(=O)C=C2CCCCC2)CCN1C(C1CC=CCO1)=O N1(C(C=CC=CC)=O)CCCC(C(=O)NC(C2CCCCC2)C2CC2)C1 Cc1nc(S)sc1CC(N1CCC(C(C)CNC(c2ccc(Cl)s2)=O)CC1)=O c1(OC)cc(C)[nH]c(=NCc2ccccc2C(N(C)Cc2ccccc2)=O)n1 c1(C(=O)NCC2C(CC)CCN2C(=O)CS(=O)(=O)NC)cc2ccccc2o1 C(=O)(C1CCCc2c[nH]nc21)N1C2C(CNC(c3c(COC)n[nH]c3)=O)C(C2)C1 C(CN=c1[nH]c(=NCc2cc[nH]n2)[nH]c2c1CSC2)n1c(C)ncc1 C1(CNC(=O)COC2COC2)CCCN(C(c2scnc2Cl)=O)C1 C1(NC(C(Cn2cccn2)NC(c2c(C)[nH]cc2)=O)=O)CCN(C)CC1C C1(C#N)(C(=O)NCC2CC(NC(C(COC)O)=O)C2)CCCCC1 C1(C(N2CC(CC)N(C(c3cnc(C)cn3)=O)CC2)=O)CCC2CC1C2(C)C C1(NC(C(=O)Nc2n(C)nc(C3CCCO3)c2)=O)CC(C2CCCC2)C1 Cc1cccc(C(=O)NC2(CNC(=O)CCC3CCCCO3)CC2)c1Cl Cc1sc(C(N2CCC(C(O)C(F)(F)F)CC2)C(=O)NCC(F)F)c(C)c1Br c1(C(=O)NCc2nc(CNC(CNC(=O)NC)=O)sc2)cnc2cc(C)[nH]c2c1 C1(C(N2CCC(O)CC2)=O)(COC)C=CCN1C(=O)C(COC)OC N1(C(C(C(C)C)NC(C2COCCN2CCO)=O)=O)CCCC(C)(CO)C1 C1(C(=O)NC2CN(C(C3(C(=O)NC)CC3)=O)CC2C)CC(=O)CC(=O)N1 c1(C(=O)NCCC2(CNC(=O)C3=CCOC3)CC2)cc(C(F)F)ccc1Cl.C1CC1 C(CC(C(=O)NCCC1CCCN1C(C1CC1F)=O)OC)OC C1(NC(C(CSC)C)=O)CCN(C(c2ccc(-c3nc[nH]n3)cc2)=O)CC1O c1(C(=O)NCCCNC(C2CC3(C2)CC(F)C3)=O)cc(F)c(F)c(O)c1F C1(NC(Cc2c(C)n(C)nc2)=O)CC2(CCC(CNC(c3ccoc3)=O)OC2)C1 Cc1cccc(=O)n1CCCC(=O)N(O)Cc1cn(CC2CCCO2)nn1 C1(CNC(c2cnc(C)n2C)=O)CN(C)CCN1C(=O)CCc1cccs1 N1(C(C(CC2CC2)NC(CC2(CC)CCC2)=O)=O)C2COCC1C2 CN1CCc2ccc(C(N3CCC3CNC(=O)Cn3ccc(Br)n3)=O)cc21 CCCC(C(=O)NCC1CCC1NC(=O)C(c1ccccc1OC)=O)NC(C)=O C=CC(C)(CC)C(=O)NCCCN(C(c1cc(Cl)ns1)=O)C1CC1 C=Cc1cncc(C(=O)NC(C2CCN(C(c3snc(O)c3Cl)=O)CC2)C)c1 c1(OC)cc(CN2CC(O)CC2C(=O)Nc2cnc(C)cn2)cc(C(F)(F)F)c1 c1(CC(=O)NC(CCCCNC(CC(C=C)C)=O)C)c[nH]c2c(Br)cccc12 c1(CC(=O)NC2C(NC(C3(C)CC(F)(F)C3)=O)C2)n[nH]c2ccccc12 c1(C(=O)NCCOC2CCN(C(CCC(C)OCC)=O)C2)cc(F)cc(F)c1N c1(CN(C(c2cc(Cl)cs2)C(=O)NCC2CC2)CCN(C)C)cccc(Cl)c1 n1(CC)ncc2c(NCC(C(C)C)OC)nc(N(CC(C)SC)C)nc12 c1(OCC)nccc(C)c1C(N1CCC1CNC(=O)Cc1ccc(C)c(Cl)c1)=O C(=O)(C1=CCCCO1)N1CCCC(C2N(C(CC=C=C)=O)CCC2)C1 c1(C(=O)NC2CC(C(C(=O)NC)F)C2)cnc(C)nc1 c1(C(N2CCC3(C(C(N(C(C)C)CC4CC4)=O)C3)C2)=O)cc2ncccc2[nH]1 C(=O)(C1=CC2(CCOC2)C1)NC1CCC(NC(CN2C(C)CCCC2)=O)CC1 C1(C)(C(N2CC(COC)(NC(=O)CCn3cc(C)cn3)C2)=O)C=CCCC1 CCC(CC)(CO)C(=O)N1CC(CCNC(c2ccnc3c2CCO3)=O)C1 N1(C(=O)NC(C2CC3CCC2C3)C)CCC(Cc2cc(C(C)(C)C)n[nH]2)CC1 C1(NC(CN(C(C)=O)C)=O)CCCC(C(=O)NCCCOCCO)CC1 c1(C(=O)NCCCCC(C)NC(c2ccnc(CO)c2)=O)cn2cnnc2cn1 C1(C(=O)NCC2CCC(C(N(CC(=O)OC)C3CC3)=O)CC2)CCCC(=O)N1C C12(NC(CCc3ccc(C)s3)=O)CC1CN(C(c1cc(CO)oc1C)=O)C2 Cc1noc(C(C)C)c1NC(C12CC(CN1C(C1CN3CCC1C3)=O)C2)=O c1(N(CC(C)NC(=O)CC2CCCC(C)(C)O2)C)ccc([N+](=O)[O-])cc1Br C12CCC(O1)C(=O)NC2.C(CC(=O)NC1CC1)NC(=O)NC.C(=O)N(C)C(C)C c1(SCC(N2C(CNC(c3cc(CC)on3)=O)CCC2)=O)nc2ccccc2o1 C1(C(=O)NC(CNC(CCNC(COC)=O)=O)C)COCCC1c1ccccc1 C(C(C)(C)CNC(c1nocc1C(C)(C)C)=O)N(C(C(C1CCC1)OC)=O)C C1(NC(C2CC=CCO2)=O)CC2CN(C(c3ccnc(Cl)c3)=O)CC12 C1(NC(c2c(OC)csc2)=O)CC(CNC(c2csc(=N)[nH]2)=O)C1(C)C c1(C(N2CC3CC(C(=O)NCC(C(CC)CC)O)(C2)C3)=O)cccn2ccnc12 CCCCC(C(=O)NCC1CN(C(=O)COC(C)C)CCO1)C(C)C N1(Cc2n(C)c3c(n2)c(Cl)ccc3)CCc2c(Cl)c(Br)cc(F)c2C1 N1(C(C(OC)OC)=O)CCCC1CCNC(c1nonc1C(C)C)=O C(=O)(C1=NOC2COCC12)NC1CCCC(CC(=O)NC(C)(C)CCCF)C1 C1(NC(C=NOC)=O)CCCC(C(N2CC(C(=O)NC3CC3)C2)=O)C1 CCCCC(C(=O)NC(CCN(C)C)C(=O)NCCCCOCC)C(C)C C1(C)(CC)COCCN1CC(=O)Nc1cn(C)nc1-c1cccc(F)c1 c1(C(N2CCC(N3CCCC3)C2)C(=O)NC)cccc(C(N)=O)c1.C1CC1 C1(NC(C2CC(=C)C2)=O)CCCC2CN(C(C34CC(CO)(C3)C4)=O)CC12 Cn1cc(C=CC(=O)NC2(C(=O)NCCC(N)=O)CSC2)cn1 N1(C(C=Cc2nc(C)sc2)=O)CC(NC(=O)C(n2nccc2C)C)C2CCCC12 C1(C(=O)NC2(CNC(CN(C(=O)OCC)C)=O)CC(OC)C2)CC2CCC2C1 Cc1ncc2n1CC(C(=O)N(C)CCNC(=O)C(C1(O)CCOCC1)(F)F)CC2 CCCC(CC)CCC(=O)NC(c1nocc1C(=O)NCCCN1CCC1)C N(C(=NCCN1CCCC1)N1CCCC(CC2CC=CCC2)C1)CC1CCOC1 C=Cn1nccc1C(N1CCCC1CC(=O)NCC#CCN(C)C)=O c1(CNC(=NC)NCc2csc(C)n2)sccc1S(C)(=O)=O N1(C(C2C(C)C2)=O)CCC(c2cccc(F)c2)(NC(=O)C(=C2CCCCC2)F)C1 c1(CCN=C(NCC(CC(=O)OC)C)NC2CC=CC2)cc2ccccc2o1 C(=O)(CC(C)CCC)NC1C(CNC(CNC(CCCCC)=O)=O)CCC1 N1(C(CCCC(C)O)=O)CCC2CCN(C(c3c[nH]nc3C3CC3)=O)CC12 O=C(C1=COCC1)NC1CCCC(NC(c2cc(C3CCOCC3)[nH]n2)=O)C1 C(=O)(C1=CCCSC1)N1C(CNC(C(C)(C)C2(O)CCC2)=O)CC1 CC1CN(C(=O)CN2CCOCC2=O)CC1n1cc(CC(C)(C)NC(N)=O)nn1 c1(C(CC(=O)NC(CS(C)(=O)=O)c2ccccc2)(C)C)c[nH]c2c(Br)cccc12 c1(C(=O)NCC2N(C(CC(CCC)(C)O)=O)CC2)cc2cccc(OC)c2o1 c1(C(N(CC(C)NC(=O)CC2CCCCCCC2)C)=O)ccccc1S(C)(=O)=O c1(CC(N2C(CNC(C(F)=CCC)=O)CC(OC)C2)=O)ccc(C)nc1Cl C=CC1(CC(=O)NCCCN(C(C2C3CCCCC23)=O)C(C)C)CCCCC1 Nc1cc(F)cc(C(=O)NC2(C3CCCCN3C(C3CCC(O)C3)=O)CC2)c1F C1(NC(C(C)(C)NC(Cc2c(C)n(C)cn2)=O)=O)CCCCCC1(C)C c1(N(C)C)ccccc1NC(=O)COC1CC(NC(=O)Cc2ccc(O)nc2)C1 C1(C(=O)NC(c2nnc(C)o2)C)(NC(CSCC)=O)CCC(C)(C)C1 C1(n2cnnn2)(CC(=O)NC2C(NC(CC(=O)N(C)C)=O)C2)CCOCC1 C1(CCNC(CC2N(C)CCC2)=O)COCCN1C(c1ccccc1CC#N)=O c1(C(=O)NCCCN(C(CCC(=O)NCCC)=O)CC)cc(Cl)c(F)cc1Cl N1(C(c2cc(C)sn2)=O)CCC(NC(=O)CC2(C)CCCCCC2)CC1C c1(C(=O)NCC2(O)CCN(C(C3N(C)CCC3)=O)C2)cn(C)c2c(Cl)cccc12 Cc1ccc(C(=O)NC(C2CCN(C(=O)CCOC3CCC3)CC2)C)cc1F CC1CCCCC1n1cc(CC(O)Cc2ccccc2)nn1 C1(NC(c2c(C)snn2)=O)CCN(C(c2nnc(S)n2C)=O)CCC1(F)F N1(CC)CCOC(C(=O)NC2(CC(=O)NC3C(C)CCC3C)CCCCC2)C1 C(C(C)C(=O)NCC1CCN(C(=O)CC2(OCc3ccccc3)CC2)C1)SC C(=O)(C(C(O)C(F)(F)F)C(C)(C)C)NCCN(C(c1cnnc(O)c1)=O)CC C1(C(=O)NCC2(F)CN(C(CCSc3n(C)ccn3)=O)C2)CCCC2CCCN12 C1(N(C(CNS(CCCC)(=O)=O)=O)C)CCC2CN(C(=O)C(=O)C(C)CC)CC12 c1(CC=C)cccc(C(N2CCCC(CN(C)C(C3CC3F)=O)C2)=O)c1 c1(C(N2C(C(=O)NCC(=O)OCC)CCCC2)=O)cc2c(s1)CCC2 CCCC(C(=O)NC(C)(C)CCCNC(=O)COc1cccc(Cl)c1Cl)C(C)C c1(CC)c(C(=O)NC2CCCC(NC(=O)CCn3nc(C)nc3C)C2)nnn1C c1(C(=O)NCCCOCCC(=O)NCc2ccc(F)cc2)c[nH]c(=S)cn1 CCC(CCCC(=O)NC1CC2(CCCC2)C1)NC(C1(C)CC(F)C1)=O C1(C(N2CC(C3(NC(CCC(=C)Br)=O)CC3)C2)=O)CCc2nncn2C1 O=C(C1=COCC1)NC(Cn1cncn1)C(=O)NCCCc1cccs1 c1(NC)ccc(C(N2CC=CC2(C)C(=O)NC(C)Cc2ccncc2)=O)nc1 c1(C(=O)NC(CC)CNC(C2CCC(N(C)C)CC2)=O)ccc2oc(C)nc2c1 N1(C(C(C)C2CCCO2)=O)CCC(C2(O)CN(C(=O)C3=CCCCC3)C2)CC1 c1(C(=O)NCC(CC(C)C)NC(=O)CS(C)(=O)=O)ccc2c(O)n[nH]c2c1 N1(c2ccc(S(=O)(=O)NCC=CC)cc2Cl)CCCCC(C2CCOCC2)C1 C1(NC(C=C(C)C2CC2)=O)CC=C(C(=O)N2CCCC(CCO)CC2)C1 C1(C(=O)NCC(c2ccc(F)cc2)NC(c2c(C)n[nH]c2)=O)CC2CC1CO2 N1(C(C2(OC)CC2)=O)CC2CC1CC2NC(=O)CCc1cccc(C(F)F)c1 Cc1ccn2ncc(C(N3CC4C(NC(C5CCCN5C=O)=O)C4C3)=O)c2c1 N1(C(C=C2CCC(C)C2)=O)CC2(C)CN(C(C3CCC(C)C3)=O)CC2(C)C1 CC(C)CC(CC(=O)NCC1OCCC1(C)C)NC(c1c[nH]c2cnccc12)=O C(=O)(C1CCc2cc(F)ccc21)NC1(C)CCCN(C(c2sccc2Cl)=O)C1 c1(C(=O)NCC2=CCN(C(CS(CC)=O)=O)CC2)c(F)ccc2ccncc12 C(N=c1[nH]cc2ccnc-2[nH]1)C1(C)CCN(C(c2cc(C(C)C)on2)=O)CC1 c1(N2CCC(C)(C(F)(F)F)CC2)nc(N2CC3CCC3(N)C2)nc2ccccc12 c1(C(=O)NC(C2CN(C(C(n3ccc(Br)n3)C)=O)C2)C)c(F)cccc1F C1(NC(c2c(C)nn(CC)c2Cl)=O)CCC2CC1CN2C(=O)C1=NOC(C)C1 C(=O)(C1CCCc2cncn21)N(CCCN(C(C1N(C(C)=O)CCOC1)=O)C)C c1(C(=O)NCC2CC(NC(C3(COC)CC3(F)F)=O)C2)nccn2nc(C)cc12 N1(C(C2CCCN(CC)C2)=O)CCC(C(=O)NCCCSC)(OC)CC1 N1(c2cc(NCC(C)CC(C)O)nc(COC)n2)CCc2sc(Br)cc2C1 c1(CC(C)(C)C)cc(=NC(=O)NC2CCC2OC(F)F)[nH]o1 O=C1CN(c2nc(=N)nc(N3CCC(c4ncccn4)C3)[nH]2)CC(=O)N1 c1(C(N(C2CCCCC2NC(C2CCC(F)(F)CC2)=O)C)=O)cc2scnc2[nH]1 C1(C(=O)N(CC(C)CO)C)(CC)CCCN1C(=O)Cn1cnc(C#N)n1 Cn1cnc2[nH]c(=NCC3(C)CCOC3)nc(N3CCOCC3)c12 N1(C(C2(CCC)CCC2)=O)CCC2(CC1)CN(C(=O)C(C)(C)c1csc(C)n1)C2 CC1(F)CCC(C(N2CCCC(C)(NC(c3cnn[nH]3)=O)C2)=O)CC1 c1(C(c2nnnn2CCCF)NCC2(CC)COC2)ccnc(Cl)c1 C#CCC(C)(CC)C(=O)N(C)CC1CCCN1C(=O)C(C)=CCC C12(CC(N3CC(OCC)C3)=O)CCC1CN(C(=O)C(c1ccc(F)cc1)(F)F)C2 C1(C(=O)NCCCCCC)N(C(c2cccnn2)=O)CCC1(C)C N1(C(C(C)S)=O)C(C(=O)NC2COCCC2O)CC2CCCCC12 c1(CC(N2CC(CCNC(=O)CC3(C)CCOC3)(OC)C2)=O)cn2ccsc2n1 N1(C(CCN(C)CC)=O)CC2CC2(C(=O)NC(c2ccco2)C)C1 c1(C(=O)NC(C(C)NC(=O)CCNC(C2CCC2)=O)(C)C)cc(C(F)(F)F)ncn1 C1(CNC(CCC=C)=O)CCN(C(c2ncoc2-c2cccs2)=O)CC1C1CC1 C1(C(=O)NCCNC(CN(C)C(=O)C2CC2)=O)CC=CCC1C(F)(F)F C(=O)(CC(CC)C(C)C)N1CCC(C(=O)Nc2cnc(CCC)nc2)C1C N1(C(C(c2c(C)n[nH]c2C)C)=O)CCC(CNC(C23CCC(C2)C3)=O)C(C)(C)C1 CC(C)C(C#N)C(=O)N(C)CC1CCCN1C(=O)C(C)C=Cc1ccccc1 C(=O)(C1=CCC2CCC1N2C(=O)Cc1cccn1C)N1CC(C(=O)OC)(CC)C1 c1(C(=O)NC2CC(OCC(=O)N(CC(CCC)C)C)C2)cncnc1C.OCCC c1(COC)ncc(CNC(=O)CNC(C2(C#N)CC2)=O)[nH]1 Cc1c(NCCCSc2ccc(Cl)cc2)nc[nH]c1=NCc1cocn1 C(=O)(CCCCCc1cccs1)NC1CN(C(c2cc(CC)c(C)s2)=O)CC1O c1(CC)cc(F)ccc1C(=O)NCC1CCCC(NC(C2(O)CCSC2)=O)C1 Cc1csc(=NCC(=O)N2CCCC(C)(NC(C3CCCCC34CC4)=O)C2)[nH]1 C1(CC(=O)N(C(CNC(C2(C#N)CC2)=O)C2CC2)C)CC2(CCC2)C1 c1(CNC(C(COC)NC(C2CCN2C)=O)=O)nnc(O)n1C C1(C(=O)NCc2nc(CC)on2)CCN(C(=O)C2CC2)CC1 N1(C(C23OCC(COC)(C2)C3)=O)CCC(CO)(CNC(=O)C(C)O)CC1 CCC(F)C(=O)NCCC(C)(C)NC(c1ccc(CC(C)C)s1)=O CN1CCC(C(N2CCC(NC(c3csc([N+](=O)[O-])c3)=O)CC2)=O)CC1=O c1(C(=O)NC2C3CN(C(C4C(COC)C4)=O)C2C3)c[nH]c2cc(Cl)ccc12 N1(C(c2ccc(OC)nn2)=O)CC(N(C(=O)CC2CC=CC2)C)C2(CC2)C1 C1(CCC#N)CC=CC(NC2(CC3CC=CCC3)CC2)C1 C(CCS(=O)(=O)C(C)C)N(C1CCN(C(c2cc(CC)[nH]n2)=O)C1)C C(=O)(C1OCCc2ccc(C)cc21)N(CCC)CCNC(=O)CCC1CC1C Cc1[nH]c(=N)nc(O)c1CCC(=O)NC1CC2CC1CN(C(=O)C1=CCCS1)C2 N1(C(c2c(C)n[nH]c2)=O)CC(F)CC1C(=O)NCC1CC1[N+](=O)[O-] CC1CN(C)CCC1N(C)C(C1CCC(NC(c2ccnc(O)c2)=O)CC1)=O C(CN=c1ccc2c([nH]1)CCCC2=O)C1N(C(C(COC)O)=O)CCCC1 N1(C(C2(CC)CN(C(=O)CNc3cccnc3)C2)=O)CC2(CC2)CC1C c1(C(=O)NCC(O)CNC(c2cscc2C(F)F)=O)ccc(SCCO)cc1 N1(c2c(C(=O)Nc3cc([N+](=O)[O-])ccn3)cccn2)CCc2cccnc2C1 C12(NC(C3CC(C#C)(O)C3)=O)CCCCC1CN(C(=O)CC(C)CCCCC)C2 C1(NC(=O)CCN(CC(F)F)C(c2ncoc2C2CC2)=O)CC2CC2C1 c1(NC(c2n(C(CC)C)nnn2)c2c[nH]nc2C2CCC2)ccc(O)cc1C C1(NC(C(C)OCC#C)=O)CC2CC1CN(C(=O)C(C)SC(C)C)C2 c1(CC)n[nH]c(=NC2C(C)CN(C(=O)C3=C(C)OCC3)CC2C)s1 N1(C(C(CCC)C#N)=O)CCC2CCN(C(c3ccc([N+](=O)[O-])o3)=O)C2C1 CC(=O)CCCCC(=O)N1CC(OCC(=O)NCc2c(C)cccc2F)C1 c1(SNC(C)CN(C(=O)C(C)(C)C)C)ccccc1NC(=O)COC1CCCOC1 Cc1cccc2c1CC(C(=O)NCC(O)CNC(c1ccc(CO)o1)=O)O2 N1(C(C2N(C(=O)OC(C)(C)C)CCC2)=O)CCC2(CCCN2C(C2CCO2)=O)CC1 C#Cc1cccc(CNC(=O)C(C)CN(C(=O)Cc2csc(C)c2)C)c1 N1(C(C=CCCC)=O)CC(CCNC(=O)C=Cc2ccc(F)cc2)OC(C)C1 C1(NC(CCCC)=O)CN(C(c2cc(C)n(CC3CCCO3)n2)=O)CCC1CO C#CCC(CC(=O)NCC(C)(O)CO)NC(=O)CS(C)(=O)=O C(=O)(C(C(C)(C)C)SC)N1CC(NC(Cc2ccc(OCC)nc2)=O)C(OC)C1 CCC(C)C(C(=O)N(C)Cc1ncco1)NC(C1C(C)(C)C1(C)C)=O CC1(C)COCC1C(=O)NCC(c1ccccc1F)NC(c1cccnc1)=O C1(NC(C(CCN(C)C)NC(=O)CC2CCC(=O)CC2)=O)CN(C)C(C)(C)C1 C(CC(O)C(=O)NCC=C1CCN(C(C2CCOC2=O)=O)CC1)SC N1(C(C2=CCN(C(CC(CC(C)C)O)=O)C2)=O)CCC2(COC(C)C2)C1 C1(COC)CCCN1C(=O)CC(C)NC(c1cccs1)=O N1(C(COCC=C)=O)CCC(C)(NC(=O)CC2CCCCCC2)C1 c1(CC)cc(C)nc(NC2CCC(NC(=O)CC3CCCCC3C)CC2)n1 c1(CC(=O)NC2CC(NC(C3(O)CCC3)=O)C(O)C2)cc2nc[nH]c2cc1Br c1(NC(C)(CNC(=O)C=CS(C)=O)C2CCC2)ccc(C(F)(F)F)cc1[N+](=O)[O-] Cc1cn2cc(C(N3CCCC3CCCNC(C3CCCN(C)C3)=O)=O)nc2s1 C1(CC=C)(NC(=O)C=CC2CCCC2)CCN(C(=O)CC2CCN(C(C)C)C2)C1 CCS(=O)(=O)CC(=O)N1C(C(=O)NC(CCO)C(C)C)CC2CC12 c1(OCC(=O)NCC2CCCC(NC(CC3(OC)CC3)=O)C2)cc(C)ccc1O C(=O)(CCC=O)NCC.C12(OCC)CN(C1)C(=O)c1ncoc1CNC2.NC c1(SCC)ccccc1C(=O)NC1CC1CNC(=O)CC1CCCC(=O)N1 CCCS(=O)(=O)CC(=O)N1CC(CNC(=O)CCc2ccccn2)CC1(C)C c1(C(N(CCCNC(C2(C)CC2(C)C)=O)CC)=O)cnccc1N1CCOCC1 CC(C)CCC(O)C(=O)N(C)CC1CCCN1C(c1cccc(C(C)(C)C)c1)=O N1(C(C(c2ccc(C)o2)C)=O)CCC2C(C1)CN2C(c1cn(C(C)C)nc1C)=O C(=O)(C(CO)C(C)(C)C)N1CCN(C(c2n(CC)ncc2)=O)C(C)C1 N1(C(C(c2n(C)ncc2)NC(c2cnsn2)=O)=O)CCCC2(CC2)C1 c1(-c2cn(C(CCC(=C)C)C(=O)OC(C)(C)C)nn2)cnc2cccnn12 c1(C(=O)NCC2CCN(C(c3cnns3)=O)C2)ccc2c(c1)S(=O)(=O)NC=N2 c1(NCc2cc(COC)on2)nc(N2CCC3C(CCN3C)C2)nc2sccc12 C1(C(=O)NC2CC(C(F)F)(NC(C3CCCO3)=O)C2)CCC2CC1CO2 N1(C(C(C)(C2CCC2)NC(c2c(CC)cccn2)=O)=O)CC(C2CCCCC2)C1 C(=O)(C(C)C(C)(C)C)N1C(CCNC(c2c(C)cn(C)c2)=O)COCC1 C1(CC(=O)N(CCN(C(=O)C(c2cnn(C)c2)C)CC)CC)CCC(=O)N1 c1(N2CCN(C(CS(CC(C)C)(=O)=O)=O)CC2)ccc2c(c1)COC2(C)C O=C1NCc2cc(C(N3CCC(NC(C4CC5CC4C5)=O)C(F)C3)=O)ccc2N1 C(=O)(CCCCC(F)(F)F)N1C(C2(CNC(c3cnc(OC)s3)=O)CC2)CCC1 N1(C(c2n(CCCC)ncc2)=O)CCC(C)C(NC(c2ncc(Cl)s2)=O)C1 C1(C(N2CCC(C)(N(C)C)C2)=O)CCc2ccnn2C1 C1(NC(COCCCCC)=O)CC2CC(C1)N(C(C1CCCC3(CC3)C1)=O)C2 CN=c1nc(C(N2CCOC(CNC(c3cnc(SC)s3)=O)C2)=O)cc(C)[nH]1 C12(C(=O)NCCC3(NC(=O)CSc4nc[nH]n4)CCC3)CCCCC1C2 S(=O)(=O)(CCC(=O)N1CCCC(N(C)C(c2sc(CO)nc2C)=O)C1)NC N#CC1CN(C(c2cc(O)nc(Cl)c2)=O)CCN1C(=O)CCc1ccoc1 C1(CNC(=O)NC(c2cccc(-n3cccn3)c2)C)CCC(C)c2ccccc2C1 S(=O)(=O)(c1cccc(-c2ccccc2OC)c1)N1C(C(=O)OC)C(=O)NCC1 N1(C(C(C(C)C)C2CCC2)=O)CCC2(CCC(NC(=O)CC3CCCC3)C2)C1 N1(C(CCC#CC)=O)CCCN(C(=O)C(C#N)Cc2ccc(C#N)cc2)CC1C CC(C)CC(C)CC(=O)N1CCCC(C)C1CNC(=O)CC1(C)CCCCC1 C1(NC(c2cccn2C2CC2)=O)CC2CC1N(C(C1CCC1)=O)C2 N1(C(C2C(OC(C)(C)C)C2)=O)CCN(C(c2ccncc2F)=O)C(CO)C1 Cc1cn2ccc(C(N3CC4CC(NC(=O)C(C)(O)C5CCC5)C3C4)=O)cc2n1 C1(COC)(NC(=O)CCc2nncs2)CCN(C(c2nccnc2C(N)=O)=O)C1 Cc1cc(C)n(CCCC(=O)NC2CCN(C(=O)Cn3ccnn3)C2)n1 N1(CCCCOCCCN)CCN(C(c2cccc(Cl)c2)=O)CC1 c1(NC2(c3n(CCSC)nnn3)CCC2)cc2n(n1)CC(O)CO2 CCCC(C)CCCC(=O)NC1CCC(NC(c2c(C)nsc2N)=O)C1 c1(N2Cc3n(cc(C)n3)CC2)nc2ccsc2c(=NC2CCCSCC2)[nH]1 Cc1ccc(C(=O)N(CCNC(=O)C(CC(C)C)n2ccnc2)C(C)C)c(O)n1 c1(OC)ccc(OCC(F)F)c(NC(=O)C(=O)NCCCN(C)C(C)=O)c1 C12(CNC(c3nc(CCC)sc3)=O)CC(C1)C(NC(C1(C)CC=CCC1)=O)CO2 c1(C(=O)NC2CC(C(N3CC(C)OCC3C)=O)C2)cnc2ccoc2c1 CC1OCCOC1C(=O)NC(C)CC(=O)NC(C)C(C)F C1(C(=O)CC23CC(CN2C(=O)Cn2ccnc2)C3)CCOc2ccccc2O1 C(=O)(C(C)CC(C)(C)C)N1CCC(C)C1CNC(c1ccnc(C(F)F)c1)=O N1(C(C(C)C2CC2)C(=O)NC(C)(C)C)CCCC(c2nncn2C)C1 Cc1cccn2nc(C(=O)NCCC3CC3C)cc12 C1(CC=C)(C(N2CCC(C(C)NC(c3ncsc3NCC)=O)C2)=O)CCCC1 CCC(C(=O)NCC(C1CC1)NC(c1ccco1)=O)NC(c1ccccc1)=O CC1CN(C(c2cnc(C3CC3)[nH]2)C(=O)NCc2ccc(F)cc2)CC(C)(C)C1 C1(CNC(C2CCO2)=O)(CO)CCN(C(C2(CO)CC2)=O)CC1 C(C(C)C)(C(O)C(=O)N(CCC(C)NC(C1(C)CCN(C)C1=O)=O)C)OC C1(CC=C)(C(=O)N(CCC2CC2)CC)CCN(C(=O)Cc2ncccc2C)C1 C1(CC(=O)NC2CN(C(COC(C)C)=O)CC(C)C2)COc2ccccc2O1 CC(C)CC(C(=O)NCc1cnccn1)ONC(c1n[nH]cc1[N+](=O)[O-])=O c1(C(=O)NC2(C3N(C(CCN(c4ccncc4)C)=O)CCC3)CC2)ccc(F)cn1 c1(C(=O)NCC(CC=C)NC(C2CCS2(=O)=O)=O)cc(C(F)(F)F)cn1C N1(C(C(C)n2ccnc2)=O)CCSCC1C(=O)NCC(O)(CO)CO CN1CC2CN(C(c3c(Br)cc(Br)c(O)c3Br)=O)CCN2C1=O c1(NC2CC(F)(CNC(=O)CC3CCC(O)C3)C2)nc2c(cc1C#N)CCOC2 C1(C(N2CCCCC(NC(=O)COC3CCOC3)C2)=O)CCCC12CCOCC2 C1(C(=O)NCC(CNC(c2c(CCC)n[nH]c2)=O)F)CCCCN1S(N)(=O)=O C1(C(=O)NCC2C(OCC)CN(C(C3CCCC3O)=O)C2)CC(C(C)C)=NO1 CC1(CNC(c2csc(-c3ccsc3)n2)=O)CCCN1C(C1CC1F)=O CC(C)(O)CC(=O)N1CCC(C)(NC(c2cc(-c3ccccc3)ccn2)=O)C1 N1(C(c2cnc(C)nc2)=O)CCN2C(=O)C(NC(c3nn[nH]c3Cl)=O)CC2C1 c1(C(c2n(CCC=C)nc(C3CCCCCC3)n2)C)ccc(F)c(F)c1 C1(C(=O)NC(CNC(c2cccc(F)c2Cl)=O)C2CC2)CCc2ncsc2C1 C1(C)(OC)CC2CC1CC2NC(=NCCOCCF)NCC1CCC1 C1(C(=O)NCCCN(C(COCCOCC)=O)CC)CCC2CNCC2O1 N1(C(C)C(=O)NC2(CN(C)C)CN(C(=O)CC(Cl)Cl)C2)CCC(O)CC1 N1(C(=O)CO)CC2CN(C(c3c(F)ccc(Cl)c3F)=O)CC2(C(F)(F)F)C1 Cc1ccnc(C)c1CNC(=O)C1=CCC(NC(C2CCNC(=O)C2)=O)C1 c1(C(=O)NCC(=O)NCC2(O)CN(C(C3C(C)CCS3)=O)C2)cc(Cl)ccn1 C1(C)(C(=O)NCc2ccc(C)nn2)CC(O)CN1C(=O)C=Cc1ccncn1 c1(OC)ccc2c(C(=O)NC3CCCCC3NC(=O)C(O)CC(C)C)coc2c1 C1(C(=O)NCCC(=C)CNC(=O)CCC)CC2CCC1CC2(F)F C(=O)(C(C)(C)C(F)F)NC1CCN(C(c2cc(CC)[nH]n2)=O)C1c1ccccc1 C(C(C)(C)CNC(c1cnn(CC(F)(F)F)c1)=O)NC(=O)CCSC(F)(F)F C1(NC(CC=CC=C)=O)CC1C1CCCN(C(c2c(C)noc2C2CC2)=O)C1 N1(C(C(COC)C)=O)CCC(C(=O)NCc2ncc(C(C)C)s2)(C(C)C)C1 C1(CC=C)(C(=O)NCCCC(=O)OC)CN(C(=O)CC2COCCO2)C1 Cc1c(NC(=O)C(=O)NC2CN(C(=O)CC3(C)CC3)C3CC23)cccc1F O=C(C1Cc2c(Cl)cccc21)NC1(CNC(C2Cc3nccn3C2)=O)CCC1 N1(C(C(CC#C)(C)C)=O)CC=C(CC(=O)NCC2(n3ccnn3)CC2)CC1 C=C(Cl)C(C)(C)C(=O)N1CC(NC(C2(C(F)F)CCN(C)CC2)=O)C(O)C1 CC(CC1CC1)N=c1ccnc(NC2(c3cc(F)ccc3F)CC2)[nH]1 C1(C(=O)NC(C)CNC(c2ccccc2Cl)=O)CCCCC(=O)C1 C1(CC(=O)N(C(CNC(C(C)Cc2cnc[nH]2)=O)C)C)CCC2CC1C2(C)C N1(C(CC=C)=O)CC2(COC(CNC(c3c(C4CC4)cccc3F)=O)C2)C1 C(=O)(C(C)(O)C(F)(F)F)NC1C(C(=O)NC(C(=O)OC)C)CCC1 C1(C(N(C(C)CO)CCC)=O)CN(C(=O)C(N2CCOCC2)C)CCC1O C1(C(N2CC(CNC(=O)CC3CSCCS3)C2)=O)OCC2CCCCC12 N1(Cc2cccc(OCC=C)c2)CCC(C(=O)Nc2cc(C)n(CC)n2)C(C)C1 CCCCC(C)C(=O)NCC=C1CCN(C(c2cnc(C(N)=O)cn2)=O)CC1 C1(C(=O)NC2CCC(CNC(C(C)C)=O)C2)CC2CCCCCCC12 N1(C(C(C)NC(CN(C(C)(C)C)C(C)=O)=O)=O)CCCC1(C)CCC(N)=O CC1(C)Nc2ccccc2C1NC(C1CCC(C)(CN)CC1)=O N1(CC(=O)N(C)CC2C(OC)(OC)CC2)CCCC(C)(c2ccccc2)C1 C1(C#N)(C(=O)NCC2N(C(CCCSC)=O)CCC2)CC12CCC2 C1(c2cn(CC(C3CN(C(C(CC)n4cncn4)=O)C3)F)nn2)CCC(C)CC1 c1(C(=O)OC(C)(C)C)cc(NC(c2cc(C(C)(C)C)n[nH]2)=O)cs1 C(=O)(C#CC1(C)CC1)N(CC(CC1CN(C(CC(CC)SC)=O)C1)(C)C)C1CC1 Cc1cc(F)ncc1-c1cn(CCN(C2CCN2C)C)nn1 c1(C(=O)NC(C(C)NC(=O)CNc2ccccn2)C)c(Cl)cncc1Cl N1(C(C(CC#C)(C)CC)=O)CCCCC2(CCN(C(C34CCC(CC3)C4)=O)C2)C1 C(C1=CCN(C(=O)CCC2CCCC2)CC1)CCNC(=O)COC(F)(F)F C1(C)(C(N(C)CC2(C#N)CCC2)=O)CC(O)CN1C(C1CC(C)(O)C1)=O c1(C(=O)NC2CCCN(C(C(CC)OC3CCCC3)=O)C2)ccn2ccccc12 c1(C(N2CC(O)(C(C)NC(c3csc(CO)n3)=O)C2)=O)cc2ccccc2nn1 N1(C(c2cn(CCCC)nn2)=O)CCC(O)C(NC(c2csc(Cl)n2)=O)C1 n1(C(C)C)ncc2c(NC(C)C(C)CO)[nH]c(=NC(C)c3ccccc3Cl)nc12 C1(C(=O)NC(c2n(C(C)C)ncn2)C)CCCN(C(C2CCC(=O)N2C)=O)C1 c1(C(N(CC(F)(F)F)CC)=O)ccncc1C1=CCC(C(F)(F)F)CC1 C(=O)(CCC(C(=O)OC)Nc1ccc(NC(c2ccccc2)=O)c(F)c1)OCC Cc1cccc(CCC(N2CCC(NC(=O)CCC=CBr)C2C)=O)c1 n1(C(C)C(=O)NC2(C)CN(C(c3csc(Cl)c3Cl)=O)C2)cnc2ccccc12 C1(C(=O)NC(C=CC(=O)NC(COC)C)(C)C)CCC(C)O1 c1(C(=O)NCC2N(C(C3(CC=C)CCC3)=O)CCCC2)nc(C)n(C)c1C c1(OC)ccc(C(N2CCN(C(C3CC3F)=O)C(CC3CC3)C2)=O)c(F)c1 C#CCC(C)(C(=O)N1CCC(OCC=C)C1)NC(C1CC2CCCC2C1)=O N1(C(c2n(C)cc(C(N)=O)c2)=O)CC(C)(C)CC1CNC(C1CC(CC2CC2)C1)=O c1(C(=O)NCC2(F)CC(NC(c3cn(CC)nc3)=O)C2)c(C)nc2ccccn12 C1(C)(N(C(=O)CCCCS)C(=O)NC)CCCCCC1.c1(-c2ccccc2)ccc(N2CCCC2)nc1 c1(CNC2CCC(CC(=O)Nc3cn(CC)nc3C)CC2)ccc(Cl)nc1Cl c1(OC)ccc2c(c1)CC(C(=O)NC(C)(C)CN(C(=O)Cn1cccn1)C)O2 Cc1oc(-c2cnn(C)c2)nc1C(=O)NC(C)C(C)F c1(C(=O)OC)c(OC)ccc(C)c1NC1CS(=O)(=O)CC1CO N1(C(c2cnc(S)nc2)=O)CCC(F)(C(=O)N(C2CCOC2)CCO)C1 C1(NC(C2(C)CCCS2)=O)C=CCN(C(c2cnn(C(C)(C)C)c2N)=O)C1 c1(C(=O)NCC(CC)(C)NC(=O)Cn2cccn2)cc(C)c2c(c1)CCC2 N1(C(c2c(C(C)C)cco2)=O)CC2CCC2(NC(C2CC2(C)C(F)F)=O)C1 N1(C(c2cn(CCC)nc2)=O)C2CCC1CN(C(c1cn(C(F)F)c(C)n1)=O)C2 c1(C(=O)NC(C)C(C)NC(c2cc(O)ncn2)=O)cccc2c1nnn2C C1(CC)(NC(C2CN(c3nncs3)C2)=O)CCN(C(=O)C(C)OC)CC1 N1(C(CC2ON=C(C)C2)=O)CC(C(N2CCC(C3CC3)C2)=O)CC12CCC2 O=C(C1CCCc2sccc21)NC1CN(C(c2cccnn2)=O)CC1O C1(NC(c2scc(OC)c2)=O)CC(O)CN(C(C23CCC(CO)(CC2)C3)=O)C1 C12(CC(=O)NCC3(O)CCCN(C(=O)CC4CC5CC5C4)C3)CCC(CC1)OC2 c1(C(=O)NC2(C)CCCN(C(CC(C)F)=O)C2)cc2cc(Br)cn2cn1 C1(C(C)(C)C)(CNC(C2(OC)CC2)=O)CCN(C(c2c(C)nsc2N)=O)C1 N1(C(CC(=C)Br)=O)CCOC(CN(C)C(C2CC(=O)N(CC(C)C)C2)=O)C1 N1(C(c2c(CCC)nns2)=O)CCC2(CC1)CC2NC(C1(OC)CCOCC1)=O C1(SC)CN(C(=O)C(=O)Nc2cc(C(c3cccs3)=O)co2)C2(CCC2)C1 C1(CNC(c2cc(C(N)=O)[nH]n2)=O)CN(C(=O)CCn2ccnn2)CCC1(F)F CC1(C)COC(C(=O)NCC2CCN2C(=O)COC2CCCCCC2)CO1 n1(CCOC)nnnc1C(c1cncn1C(C)(C)C)NC(C1CCCCC1)C C1(NC(CCc2c(C)nn(C)c2)=O)CN(C(=O)C(C)OCC2CC2)CC1C1CC1 C(=O)(C(O)CCC(C)C)N1C(CN(C(c2noc(CC)c2C)=O)CC)CCCC1 c1(CNC(C(C)C(C)O)=O)cccc2c1CN(C(C1(F)CC=CC1)=O)C2 c1(C(=O)C=CC(N2CCN(CCO)CC2CC(F)(F)F)=O)ccnc2[nH]ncc12 C1(CNC(C2C(CC)C2)=O)CN(C(=O)Cc2cccc(C)c2)CC1O N1(C(C23N(C(c4cc(C)c(O)nn4)=O)CC(C)(C2)C3)=O)CCCC(C)(O)CC1 c1(C2(CNc3nccc(N(C)CC4CCC4)n3)CCC2)ccc(F)cc1F c1(OCC(=O)NCCC(C)NC(=O)Cc2ccsc2)ccc(F)cc1O c1(C(=O)NCC(CN(C(COCCCC#C)=O)C)O)c(F)cc(OC)cc1F C1(C(C)=O)CC(C(=O)NCC(C)CNC(=O)CC2(CSC)CC2)C1(C)C Cc1cn(C)cc1C(=O)N(C(C(=O)NCc1nccs1)C1CC1)C C(CC(C)C(=O)NC(C)CNC(=O)Cc1ccccc1OC(C)C)OC c1(NC(C2CN(C(=O)OC(C)(C)C)C3C2C3)=O)cccc(C(=O)O)c1Cl N1(C(C=CC=CC)=O)CCCC(C)(NC(c2ccc(Cl)nc2Cl)=O)C1 C1(C(N2CC(N(C(c3c(C)c(Br)sc3)=O)C)C2)=O)SC2C=CC1CC2 C1(CC(=O)NC2CC(CNC(CCc3cn(C)nc3)=O)C2)CCCC(=O)N1 c1(C(N2CCC(O)C(O)CC2)C(=O)NCCCSC)ccc2ccc(Br)cc2n1 c1(CC(=O)N(C2CCCCC2)CCNC(C(C2CCC2)OCC)=O)sccc1Cl C1(C2CC2)(C(=O)NCC2CN(C(Cc3c(C)cccc3)=O)C(C)C2)CCOCC1 c1(C(=O)NC2CN(C(CC3CC(=O)NC(=O)C3)=O)CC2O)cccc2nccn12 c1(C(C(=O)N(C2CCN(C(C3C=CC=CC=C3)=O)C2)CCC)C)ccc(F)cc1 C1(NC(CC2(C=C)CN(C(=O)COC)C2)=O)CCc2n[nH]cc2C1 c1(NCC(C)(C2CC2)NC(c2cc(C3CC3)on2)=O)ccc([N+](=O)[O-])cc1C#N C1(C)(CNC(C(C)NC(CC)=O)=O)CN(C(=O)CCNC(=O)CO)CCO1 C1(CC(N2C(CN(C(C3ON=C(C(C)C)C3)=O)C)CCC2)=O)CCCNC(=O)C1 c1(C(=O)NCC(N(C)C(c2coc(CC3CC3)n2)=O)C2CC2)ccn2ccsc12 N1(C(c2n(C)ncc2C2CC2)=O)CCN(C(c2ccnc(Cl)c2Cl)=O)CC(O)C1 C12CCCN(C1)CC(=O)N(CC1CC1)C2.c1(CC)ccon1 N#Cc1csc(C(=O)NCC(O)CNC(=O)CC2CC(C(F)F)C2)c1 N1(C(C2CC(OC)C2)=O)CC(C)CN(C(=O)C=CC=C(Cl)Cl)C(C)C1 Cc1cc(C(N2CCC(CO)(NC(=O)C=CC(=O)N(C)C)CC2)=O)cc(C)c1O C(=O)(C1OCCc2ccccc21)N1CCC(NC(c2cnc(C(F)F)s2)=O)CC1 C(=O)(C(O)CCCCC)NCC1(F)CC(CNC(C2C(=C)C2)=O)C1 S(=O)(=O)(c1cccc(=NCCCn2ccnc2)[nH]1)NCC(C)(C)F c1(C2C(C(=O)NCC3(N(C)C)CC3)(COC)C2)ccccc1 S(=O)(=O)(c1[nH]c(=NCc2cncs2)ccc1Br)NCC(CC)(CN(C)C)CC C1(CNC(c2c(C)ccs2)=O)CN(C(C2CN(C(C)C)CCO2)=O)CC12CCC2 C(=O)(C(C)(C)C1CCN(C(=O)C(C)NC(=O)C(C)(C)C)C1)NCCOCC c1(C(N2C3(CNC(c4c(C)nc(C5CC5)o4)=O)CC(C2)C3)=O)nc(Cl)ccc1Cl C1(S(C)(=O)=O)(C(=O)NC2CC(C)(NC(CC3C(C)(C)CCCC3)=O)C2)CCCC1 c1(NCCN(CC(CC)C)C)ccc(S(=O)(=O)NC(C(C)O)C2CCC2)cc1C#N C1(NC(C=CCN(C)CC)=O)CCC(C)(NC(=O)CC2NC(=O)NC2=O)CC1 N1(C(=O)NC2(N(C)C)CCCC(C)C2)CCC2(C1)CC2(F)F C(=O)(C1Cc2ccccc21)N(CC(C)NC(C(CC(=O)OC)(C)C)=O)C C1(CC(=O)NCC(C2CCCC2)NC(=O)COCC2CCCC2)CCCC12CC2 CC1C(C(=O)NC2(CCF)CCC2)CCN1C(=O)Cc1ccsn1 N1(C(c2c(C)onc2)=O)CCC(C2CC2)C1CNC(C1NC(=O)CC1C)=O N1(C(=O)CC2CCCCCC2)CC2(CO)CC1(C(=O)NCc1cn(CCO)nn1)C2 C(CCCCC(=O)N1CCC=CC1C(=O)N(C1CC2CC2C1)C)OCC C1(CNC(c2nc(C3CC3)no2)C)CCC(c2ccccc2)CC1 C(=O)(CC(C)(C)CC(=O)NCCC(O)CNC(=O)CCC1CC(C)C1)OC CC(C)(O)C#CC(=O)N1CCCC1CC(=O)NCCCN1CC=CC1 N1(C(CC(C)F)=O)CC2(CO)CC1(C(=O)NCC(C)OCCO)C2 CON1CC(C(=O)NC(CC(=O)NC2(C(O)CO)CC2)C2CC2)CC1=O C1(CN(C(C=CC(=O)OCC)=O)C)CN(C(c2ccon2)=O)CCO1 C(=O)(C(CCC(C)C)OC)NCC(CC)(CC)NC(C1CC1OC(C)(C)C)=O C(=O)(C(F)(CNC(C1CNC(=O)N1)=O)C(C)C)N1CCC(C(CC)C)CC1 CC(C)C(CNC(=O)CN(C1CC(C#N)C1)C(=O)C(C)n1ccnn1)C(C)C C1(C(=O)NCCCN(C(=O)C2=CCC(C)CC2)CCC)OCC2CCCCC12 c1(NC(C)=O)cnc(C)c(C(N2CCC(NC(=O)CC3CCCN3C)CC2)=O)c1 N1(C(C2C(OC)CC2)=O)CCN(CCNC(C2CCCN2C(C)C)=O)CC1 N1(C(C(COC)OC)=O)CCC(COC)(NC(C2Cc3nccn3C2)=O)CC1 c12cc(Cl)ccc1C(=O)N1CCCC1CNC(=O)C2.C1CC1C(=O)OC.CCS c1(C(N(C(C)CNC(=O)CC2CC3(CCC3)CO2)C)=O)ccc(S(C)(=O)=O)o1 CC1(C)C(CNC(c2ccnc(F)c2)=O)CCN1C(c1ncc(Cl)cc1Cl)=O c1(C(=O)NCC(C(C)(C)C)NC(CCC=C=C)=O)nn2cccnc2c1Cl c1(C(=O)NCC=C2CCN(C(c3cc[nH]c3)=O)CC2)cc2c(Cl)cccc2s1 C(C)(CO)(C(=O)NCC1(CNC(=O)CCc2ccccc2C)CCC1)OC N1(C(C2C(C)CCO2)=O)CC2CN(C(c3occc3Br)=O)CC2C1 C1(NC(c2cn(CC)nn2)=O)CC(O)CN(C(=O)CCC=CC(C)C)C1 N1(C(C(F)=CC)=O)CCC(C(C)(O)CNC(=O)CC23CCC(CC2)C3)CC1 C1(C(=O)NCC2(CCCNC(c3c(C)csc3)=O)CCCC2)CC2COCC2C1 N1(C(C2(C#N)CCCC2)=O)CC2CCC(CNC(C3C=CCCC3)=O)(C2)C1 O=C(NNc1cc(F)c(Br)c(F)c1)C1CN(Cc2ccc(F)cc2)CCO1 c1(C(=O)NCC(C)NC(C2(c3cccc(C)c3)CC2(F)F)=O)cnc(Cl)c(N)c1 C1(CC(=O)NC(c2cnc[nH]2)C)COCCN1C(c1cncc(C(F)(F)F)c1)=O N1(C(C(C2CCN(C(C(C)NC(N)=O)=O)C2)C)=O)CCOC(C#N)C1 N1(C(C2(SC)CC2)=O)CCC(C(=O)Nc2sc(C)c(C)c2C(N)=O)(OC)CC1 C1(OC)CC2CC(NC(=O)C=CC3CCN(C(=O)CSC(F)(F)F)CC3)CC12 c1(C(=O)NCCC(=O)N(c2ccnc(C)n2)CC)cncc(OC)n1 C(C(C)CC(=O)Nn1cnc2ccccc12)NC(CCCCCNC(C)=O)=O c1(OC)ccc(CCC(N2CCC(CN(C)C(C3(C(F)F)CC3)=O)CC2)=O)cn1 c1(COC)nc(C)c(C(N2CCCC2C(C)NC(C2(O)CC2(C)C)=O)=O)s1 O=C1NC(=O)C2(CCCC23CN(C(c2cccc(-n4cnnc4)c2)=O)C3)N1 c1(OC)ccc(OC(C2CC(Sc3ccc(Cl)nc3)C2)=O)cc1F C(=O)(C(C)(C)C(=O)NC)N1CCC(c2c(CNC(C(C3CC3)OC)=O)c[nH]n2)C1 c1(C(=O)NC2CCCN(C(CC(CC)O)=O)C2)cc(Br)c(C)cn1 c1(C(=O)NCCCCC(C)NC(C2(CC)CCOC2)=O)ccc2c(n1)CCC2=O N1(C(c2c(CC)c[nH]c2)=O)CCC2CCCC12C(=O)NC1(C)CC(O)C1 C1(NC(C(CC)(O)c2ccccc2)=O)CCN(C(=O)Cc2ccsc2C)C(C)C1 c1(C(=O)NCCC2N(C(C(C)=C(CC)C)=O)CCOC2)cc(O)nc(C2CC2)n1 c1(NC(C(c2c(C)cccn2)N2CCSCC2CCO)=O)ccc(Cl)cc1F CC1CN2CCN1C(C(=O)NCCC1CC(NC(=O)CC(C)(C)O)C1)C2 C1(F)(C(N2CC(C(C)NC(C(CC)C)=O)C2)=O)CC=CCC1 O=C1CCCCC(C(=O)NC(c2cccnc2)C(=O)Nc2cccc(C3CC3)c2)N1 C(=O)(C1(O)CCCc2ccccc21)NCC(Cc1c(C)c(Br)ccc1)CO C1(NC(CN2CCC(n3c(C)n[nH]c3=N)CC2)=O)CC2(CC(=O)N2)C1 c1(OC)cc(Cl)c(Cl)cc1NC(=O)C(=O)NC(C1CCCOC1)CCO c1(N2CCC(CC)C2)nc(N2CCn3nc(C(C)(C)C)cc3C2)nc2c1CSC2 C(c1ccc(Cl)cc1)=CC(=O)NCC1C=CC(NC(C(C)n2cccc2)=O)C1 C(=O)(C#CC1CCCO1)N1CCN(C(=O)Cc2ccc(F)c(C(F)F)c2)CC1CO c1(C(=O)NCC(CCC)C(=O)NCC(F)Br)ccc2n[nH]cc2c1 Cc1cccc(C2CCCC(OC(C3CCN(C(=O)CC(C)C)CC3)=O)C2)c1C C(=O)(C(F)C(C)(C)O)NCC1C(CC(=O)N(CCC(N)=O)CC)C1 C1(CCNC(C2CCCOCC2)=O)CCCN(C(c2cnc(Cl)cn2)=O)CC1 c1(N2C(C(=O)NCC3CCCOC3)CC3(CC3)C2)ncnc2ccc(F)cc12 c1(CN2C(COC)CN(C(C3CCCCN3C)=O)CC2)cc(Br)cc(C)c1O c1(C(N(C(C)C(=O)NCCOC2CCOC2)C)=O)cscc1Cl Cc1ccc2c(N3CCN(C(=O)C(C)(O)CC(C)C)CC3)ncnc2c1 C1(NC(c2cc(C)c(C)[nH]2)=O)CC=C(C(=O)NCC(C)C2CCC2)C1 CS(=O)C=CC(=O)NCC1CCN(C(C2CCCN2C(=O)CC2CC2)=O)CC1 N1(C(C=CC(=O)N(C)C)=O)CCC2CCC(NC(c3cc(Cl)nnc3O)=O)C1C2 N1(C(C(C)NS(CC)(=O)=O)=O)CCOC(C(C)NC(c2cnn(C)c2N)=O)C1 O=C1CS(=O)(=O)CC(C(=O)NC2CC2CNC(=O)CC(F)(F)Cl)N1 N1(C(COCCC#C)=O)CC2CCCCN2CC1CNC(=O)CCNC(=O)CO C(=O)(C(CNC(=O)C(C)=CC(C)(C)C)C(C)(C)C)N1CCCC(C#C)C1 N1(C(c2c(C)csc2Cl)=O)CC2OCCN(C(c3c[nH]c(=O)cn3)=O)C2C1 c1(CNC(C=CCN(C)C(C2CCSC2)=O)=O)ccc(Cl)cc1 N1(C(CCOCCCOC)=O)CCC(C=C)(C(N2CC(c3ncccn3)C2)=O)C1 CC(CC(=O)N1CCCC1C1(NC(=O)C=CC(C)(C)C)CC1)CC(F)(F)F c1(C(N2CCC(CSCc3nnc(CC)o3)C2)=O)ccc2c(Br)cccc2n1 C1(C(=O)NC2(CF)CN(C(C(C)CN(C)C)=O)C2)CCCCN(C)C1=O N1(C(Cc2c(C)scc2)=O)CCOC(CCNC(=O)CC2CC(F)C2)C1 N1(C(c2c(CC)n[nH]c2)=O)CCC(NC(c2scc(C)c2Cl)=O)C(C)C1 N1(C(C(=CC2CCCC2)C)=O)CCCCC(NC(=O)CN2CCNC(=O)C2)CC1 Cc1ccc(C(=O)N(CC(C)NC(=O)C2=CCOC2)C)c(F)c1F C1(C(=O)NCCC(CC)CO)CN(C(=O)CN2CC3CC3C2)CC12CC2 c1(-c2cccc(OC)n2)cc(C(=O)Nc2ccc3cncn3c2)cc2cc[nH]c12 C(C(=O)NCCC1CN(C(c2ccccc2)=O)C1)(C(C)C)N(CC)CC c1(C(=O)NCC(C)(C(C)C)NC(c2ccc(OC)cc2)=O)cnn2c1N(C)CC2 N1(C(COCCCC#C)=O)CC(CC(=O)NCCn2cncn2)CC1C C1C(C)(C)CNC(=O)C(C)CC(C(=O)NC)N1CC1CC1.CCOC C12(C(=O)NCCCC3CCOC3=O)CC(CN1C(=O)CCC1OCCO1)C2 O=C1NC(=O)C2(CCCN(C(=O)C(F)(F)c3cccnc3)C2)N1 C=CCC(F)(F)C(=O)NCC(C1CC1)NC(=O)C(CCCC)N(C)C C1(N(C(=O)CC2CC3(CC3)C2)CCO)CCN(C(=O)Cc2nc[nH]n2)CC1 c1(C(=O)NCC2CC(NC(C3(OC(C)C)CCOC3)=O)C2)cnc[nH]c1=N n1(C(C)(C)C)nnnc1C(C1(c2cccs2)CC1)NCCC1CCCO1 CC1CC=C(C(=O)N2CC3CN(C(c4cc(C#N)ccc4N)=O)CC3C2)CC1 Cc1nc(F)ccc1CN1CCCCC1C(=O)NCCC(C)C N1(C(c2cc(C)c(F)cn2)=O)CC=C(CCNC(=O)CNC(=O)C(F)(F)F)CC1 C(=O)(C1c2c[nH]nc2CN1C(=O)Cc1ccoc1C)NCc1c(C)cccc1 c1(C(N2CC(OCCNC(C3(CCC)CC3)=O)C2)=O)ccnc(COC)c1 c1(OCC)ccc(NC(c2c(OC(C)=O)cccc2)=O)cc1NC(=O)COC O=C1CC(=O)NC(C(=O)NC2(CC(N3CCOCC3CO)=O)CCCCC2)C1 c1(C(N2CC(CC)C(NC(=O)Cn3nccn3)CC2)=O)ccc(S(=O)(=O)NC)o1 C1(O)(CNC(CS(N)(=O)=O)=O)CCN(C(=O)CCC(=O)c2ccc(F)cc2)CC1 C1(CC(=O)NC(CC)CC)CCN(C(=O)C(=O)NCCSC(C)C)C1 N1(C(CC=CC)=O)CCC(N(C)C(C2CC(CC(C)(C)C)C2)=O)CC1 c1(C(N2C(CNC(C3(C)N(C)CC(OC)C3)=O)CCC2)=O)c(O)ccc(Cl)c1F C(=O)(CCCCCC(C)(C)C)NC(C)CCCNC(c1cncc2ccsc12)=O C1(C(C(N2CC(OC)C2)=O)F)CCN(C(c2n[nH]cc2C2CC2)=O)C1 C#Cc1ccc(OCC(=O)NCC2(C)CN(C(c3cnn[nH]3)=O)CCO2)cc1 C1(C(N(C(C)CCNC(c2ncoc2C2CC2)=O)C)=O)OCCC1(C)C C(C1=CCN(C(=O)C2=CCCCO2)CC1)NC(C(C(C)C)C)=O C=CCC(C)(C)C(=O)NC1CCOC(CNC(=O)Cc2cscn2)C1 C1(NC(c2csc(CNC(=O)C(O)C3CC3)c2)=O)CCCC(CO)C1 N1(C(c2c(C)con2)=O)CCN(C(=O)CCc2cccn2C)CC1CF C1(C(=O)Nc2cn(C)nc2)C2CCC(C2)C1NC(=O)Cc1ccco1 C1(CNC(C2N(S(CC)(=O)=O)CCC2)=O)CCSC1(C)C C1(C(N2C(CN(C)C(c3ccc(Cl)o3)=O)CC(F)C2)=O)CC2(C1)CC(F)(F)C2 N1(C(C(CC)COC)=O)CC2(C1)CN(C(c1cc(C3CC3)ns1)=O)CCO2 C12(CCCC1)NC(=O)CSC2.C1CCCCO1.C12CC(C1)C(=O)NCC2.CS C(C(F)(F)CCC(=O)NC12COC(C1)C(O)C2)n1cc(CCC(CC)O)nn1 CC1(C)C(CNC(C2CCCN2S(C)(=O)=O)=O)CCN1C(=O)CC(F)(F)F C(C1=CCCSC1)(c1n(C2(C)CC2)nnn1)NC1CC1F c1(OC(C)C(=O)N(C)CC2(C(C)(C)O)CC2)cccc(F)c1.C1(=O)C=CCN1 c1(C(=O)NCC(N(C(CSCC)=O)C)C2CC2)ccc(-c2ccccn2)s1 CC1CN(C(C2CC(O)C2)=O)CC1NC(=O)C(c1ccc(O)cc1)(C)C CN=C(NC(C)(C)C=Cc1ccccc1)N1CN(C)C(=O)C1C CC1(NC2CC23CCCC3NC(=O)NC2CCCCCCC2)CCCC1(F)F c1(OC)ccn2cc(C(=O)NCC#CCNC(c3ccn(CC#N)n3)=O)nc2c1 C1(C(N2CC(C)(CC)C2)=O)CC(C)(C)CN1C(C1CC(=O)C1)=O C1(C(N2CC(NC(c3cc(CCC)on3)=O)C(C)C2)=O)CC2(CCC2OC)C1 c1(C(N2CCC(F)(CNC(Cc3nc(C)sc3C)=O)C2)=O)ccccc1[N+](=O)[O-] N1(C(c2ccn(C(C)(C)C)n2)=O)CC2(CCCC2NC(=O)Cc2cnsc2)C1 c1(CCCC(=O)NC2CN(C(Cc3cnc(C)[nH]3)=O)C2)ccc(F)cc1Br C1(OC)(CNC(C2(C)CC2F)=O)CCN(C(c2c(Cl)sc(C)c2C)=O)CC1 N1(C(CC(CC)(C)C)=O)CC2OCCN(C(=O)CCOC3CCCCC3)C2C1 O(NC(=O)C(CNC(C1CC(=O)C12CCC2)=O)C(C)(C)C)CCC(C)O CC(C)C(C)CC(=O)NCC12CC(NC(=O)CN3CC4CCC3C4)(C1)C(C)O2 c1(C(=O)NCC2(CNC(Cn3ccc(C)n3)=O)CCC2)cc2cc[nH]c(=O)c2s1 S(=O)(=O)(c1ccccc1F)NCC(=O)N(CCCNC(C1(C#N)CCC1)=O)C C1(NC(C2CCN(C(c3cc(OC)nn3C)=O)C2(C)C)=O)CCOCC12CCC2 c1(C(C)NC(C2C(=C)C2C(=O)NC2CC(N3CCCC3)C2)=O)nn(C)cc1O c1(C(=O)NCC(C)NC(=O)CC2(C(F)(F)F)CC2)nccnc1OC1CCCC1 C1(NC(=O)NCC(C)CN2CCCC2)CC12CCCCC2 N1(C(C2CCC(NCc3cn(C(C)C)nc3)C2)=O)CCC2SC(=O)C=C2C1 c1(C(N(CCNC(CCNC(COC)=O)=O)CCOC)=O)n[nH]c(C)c1F N1(C(c2ncnc(C)c2C)=O)CC2(CNC(c3cnc(C)n3C)=O)CCC1CC2 C=CCN=c1[nH]cc(C(N2CCN(C(c3cc(F)n(C)n3)=O)C(CCC)C2)=O)s1 C(=O)(C1=CC2CC=CCC12)N1CC(O)(CCNC(c2[nH]c(CC)c(Cl)n2)=O)C1 N1(C(CN(CC)CC)=O)CCC2(C=C(C(=O)NCCNC(C)=O)C2)C1 C1(NC(CCSCCC)=O)CC2CCC1(C(=O)NCc1cc(C)co1)C2 C(=O)(C1CCCc2sccc21)N1CC(O)(C(C)NC(C2COCC(C)(C)O2)=O)C1 c1(C(=O)NC2CC(C)N(C(c3ccnc(Cl)c3Cl)=O)C2)cccc2cnnn12 C1(C(=O)NCCCN(C(C2CSCN2C(C)=O)=O)CC)OC2CCC1CC2 N1(CCCC)CCN(C(=O)CN2CCN(C(=O)C(C)(F)F)CC2)CC1 N1(C(CN(CCN(CCC)CC=CC=O)C)=O)CC(F)CC1CO C(CCCC(C)(C)C)NC(C(C(C)O)NC(=O)COCCF)=O C1(C(C)(C)C)(CN)CCN(C(C2(C3CCCCO3)CCOCC2)=O)C1 n1(CC(C(C)CN2CCCC2=O)=O)ccc2c(C(=O)O)cccc12 C(C#CC(C)n1cc(C(c2ccccc2)C)nn1)(OCC)OCC CC1CN(C(c2ccoc2C(F)(F)F)=O)CCC1NC(=O)CCCC(=O)N(C)C CC1(NC(c2cnc(S)[nH]2)=O)CCN(C(c2cnc(CC(F)(F)F)s2)=O)C1 C1(C(N(C2CC(C#N)C2)CC(=O)N(C(CCO)C(F)F)C)=O)C(C)(C)C1(F)F c1(CC(=O)NC2CC2NC(C2CCC(=O)N2)=O)csc(C2CC2)n1 CC(CC(=O)NC(C(=O)NCc1ncco1)c1cccs1)n1cccc1 CC(C)(Cc1ccc(Br)cc1)C(=O)Oc1ccccc1-n1ccnn1 CC(N=c1[nH]c2c(c(=NC3CCCS(=O)(=O)C3)[nH]1)CCCCCC2)c1ccoc1 c1(C(=O)NC2CC(NC(c3ncc(OC)cc3F)=O)C2)cc2cc(F)ccc2[nH]1 C(CC(C(=O)Nc1ccccc1OC)NC(C1CC12CCCC2)=O)OC C1(CCCNC(c2c(C)nco2)=O)CN(C(c2cnccc2N(C)C)=O)CCO1 N12Cc3ccc(cc3C1)CNC(=O)C2.C1(NC(c2cnns2)=O)CC2CCC1C2 c1(C(=O)NC2CN(C(c3cccc(OCCC)c3)=O)C2)cnc(Cl)c(C)c1 N1(C(C(CC#C)C)=O)CCC(CCOC)(NC(=O)CC(C)c2cnn(C)c2)CC1 c1(OC)cccc(C(C(=O)NCC(F)CNC(c2nc(C)sc2C)=O)OC)c1 c1(C(N(CCCN(C(=O)CCc2cccnc2F)C)C)=O)ccccc1O C1(CN(C(=O)CCc2cncnc2O)CC)CCCN(C(c2ccsc2Cl)=O)C1 O=C(C1Cc2ccc(Cl)cc21)NC1CN(C(c2ccc(Cl)o2)=O)CC(F)(F)C1 c1(C(=O)NCCCC(C)NC(C2CC(OC)C2)=O)ccnc(OCCO)c1 N1(C(C(C(=O)OC)C)=O)CCC12CCN(Cc1cc(Br)cc(C)c1O)CC2 CC(CC(C)NC(=O)CCC1CC1)NC(c1ccn(-c2ccncc2)n1)=O N1(C(CC(CCC)O)=O)CCC(C(=O)N2CC(C(N)=O)C(C)C2)=C(F)C1 C1(NC(N2CCC(O)C2)=O)CCN(c2nnnn2-c2ccccc2)CC1 C(c1ccccc1F)=CC(N1CC2CC1CC2NC(C1(C2CC2)CC1)=O)=O N1(C(c2n(CCCC)ncc2)=O)C2CCC1C(NC(=O)COCC)C2 C(=O)(CC(C)COC)NCC1(C(=O)NCC(C)OCC#C)CC=CC1 CN1C(=O)CN(CC(N2CC(C3(Nc4ncnc5sccc45)CC3)C2)=O)C1=O C(=O)(CCCn1cncn1)N(C(C)C(=O)NC(C)CSC)CC C1(C(=O)NC(C2CCN(C(c3csc(-c4cnc[nH]4)n3)=O)C2)C)CC(F)(F)C1 C1(C(N(CCNC(C2(N(C)C)CCCC2)=O)C2CC2)=O)CC12CCC(F)(F)CC2 C(=O)(C#CC1CCOC1)N1CCC(NC(CCS(=O)(=O)NC)=O)(CO)CC1 c1(CNc2cccc(C(CC)O)c2)c(C)ccc2ccccc12 C1(C(C)C)CCCN(C(=O)CN(C(c2ccnnc2)=O)CC2CC2)CC1 CC1(C)CC(C(=O)NCC(O)CCC(N2CC(c3cc(O)no3)C2)=O)=NO1 C(=O)(C1=NOC(CNC(c2c(C)oc(C)c2C)=O)C1)N1CC(CCC)OCC1 c1(C(C)C)cc(C(=O)NCCC(O)CNC(=O)CN(C2CCSC2)C)ccc1O c1(C(=O)NCC2CC(NC(C(C(C)C)OC)=O)C2)cc(Cl)c(F)c([N+](=O)[O-])c1N C(=O)(C(O)CCc1ccccc1)NC12CC(NC(C(C)NC(=O)OC)=O)(C1)C2 N1(C(c2ccc(OC)cc2OC)=O)CCC2CCC(NC(c3cc(C)c[nH]3)=O)C12 CCCS(=O)(=O)C(C)C(=O)NCC(C1CCCN1C(c1ccncc1O)=O)(C)C C1(CNC(c2cncc(C#C)c2)=O)CCN(C(=O)C(F)C(F)(F)F)C12CCC2 Cc1ccc(-c2cc(NC(=O)C(C)OC(c3cnn(C)c3C)=O)n[nH]2)cc1 N1(C(C=CCC)=O)CC(CC(=O)NC2CC2(C)C(F)F)CC1(C)C C(=O)(C1=C(Cl)CCC1)NCC1C(NC(C(CC)Oc2ccccc2C(C)C)=O)C1 N1(C(COCCCN(C)C)=O)CC2(CC2)CC1CC(=O)NCC(F)(F)CO c1(CCCC)cc(N)c(C(=O)N(CCNC(=O)CC(O)CN(C)C)CC)c(F)c1 N1(C(C2CCN(C(C)C(=O)NCCNC(=O)OC(C)(C)C)C2)=O)CC(O)(C2CC2)C1 c1(OC)ccc2cc(C(=O)NCCc3ccc(S(N)(=O)=O)s3)[nH]c2n1 c1(C(N)=O)ccnc(C(=O)NC23CC2CN(C(C2CSCCS2)=O)C3)c1 c1(C(=O)NC2C3(CC(NC(C(COC)(C)OC)=O)C3)C2)cnc2c(C)cccn12 c1(Cc2onc(C(C)(C)NC(c3ccccc3)=O)n2)ccc(N)c(Cl)c1 C=CCC(C(=O)NC(CNC(=O)CCNS(C)(=O)=O)C(C)(C)C)NC(C)=O C1(CCC)CN(C(c2ccncc2Br)=O)CCN1C(C12CC(O)C1C2)=O c1(C(=O)NCC2N(C(CC3N(C(C)=O)CCC3)=O)CCCC2)cc([N+](=O)[O-])c[nH]1 Cc1cc(C)n(CC(N2CC(CNC(C3CC3(C)Br)=O)C2)=O)n1 Cc1cc(C)c(C(=O)NC2CC(NC(c3cc(C4CC4C)on3)=O)C2)cn1 CCCC(C(O)C(=O)N1CC2C(CO)C2C1)NC(=O)CC1CC(CC)=NO1 C1(C(=O)NC(c2cccnc2)CC)CC12CCN(C(=O)CC1CC=CC1)CC2 C#CC1CC2CCC1N(C(=O)C(c1cnn(C)c1)NC(=O)C1=C(C)OCC1)C2 CCC(CNC(C12COCC1C2)=O)(CC)NC(c1cncnc1)=O C(=O)(C(C)C(C)C(C)(C)C)N1CC2(CCN(C(c3cnn(CCC)c3C)=O)C2)C1 CCC(CCC(=O)NCC(O)CC(F)(F)F)NC(c1cccnc1NC)=O N1(C(CCN(C)C(c2nc(C#N)cs2)=O)=O)CCN(C(N)=O)CC1 C1(COC)(CNCc2ccc(C(C)(C)C)s2)CCCO1 C(N=c1ccc(C#N)c(C)[nH]1)C1C2CN(C(C(CC)CC(C)C)=O)CC21 C(CCC(C(=O)NOC1CCC1)NC(C1CCCN1C)=O)OC CC1CCC(NC(c2ccc(C3CC3)cc2)=O)CN1C(=O)Cc1cccnc1 N1(C(c2cc(C)nnc2O)=O)CC2ON=C(CNC(=O)C3=CCCCC3)C2C1 c1(C(C)NC(C(Cc2cn[nH]c2)NC(COCCCOC)=O)=O)ccc(O)nc1 C1(C(N2C3CC(NC(COCC=C)=O)C3CC2)=O)COc2ccccc2C1 c1(C(N2CCC(C)(NC(CN(C3CCCC3)C)=O)C2)=O)cncc(O)c1Cl C1(C2CCN(C(C3CCC4(CC3)CC4)=O)CC2)(NC(CCNC(C)=O)=O)CCC1 Cc1cccc2oc(N3CC(NC(=O)CC(c4cccc(F)c4)C)CC3C)nc12 c1(C(N2C(CSC)CCC2)=O)ccc2nccn2c1.c12cccc(c1)NC(=O)N2 c1(C(=O)NCC=CCNC(C2(C)CC(F)C2)=O)cc(-c2ccccc2)ccn1 C1(C)(CC)CCC(C(=O)N(CCC(=O)N)C(C)C)O1.C12(CC1)C(=O)NC2.C1CC1 c1(CC)ccc(C=CC(=O)NC2CC2CNC(=O)Cn2ncc(Cl)c2C)cc1 CC(C)CC(CN(C(=O)Cc1ccnn1C1CCC1)CC)NC(c1ccc(F)s1)=O C1(CNC(C=CC)=O)CC(C)(C)CCC1NC(c1cncc(NS(C)(=O)=O)c1)=O c1(C(C)C)ccc(C(=O)NCC2CCC(NC(C3(C)CSC3)=O)CC2)cc1 N1(C(C2CC(CC)C2)C(=O)NCCC2CC2)CCC(CNC(=O)C2CC2)C1 Cc1sncc1NC(=O)C(C)NC(=O)COC1CC=CC1 CCCCC(F)C(=O)N(CCCNC(=O)C(C)(C)C(F)F)C1CC1 C1(CCCC)CN(C(C2CC23CC3)=O)CCN1C(=O)Cc1ccnn1C(F)F c1(CNC(C(C)(O)C2CC2)=O)cncc(C(=O)NCCn2cnnn2)c1 C#Cc1cccc(C(=O)NCCOCCNC(=O)CC2(C)CCS(=O)(=O)N2)c1C N1(C(C(C2CCCC2)OC)=O)CCN(CCNC(C2(C)CCOC2C)=O)CC1 N#CC1CCC(C(=O)NCCCCCCNC(=O)C(F)C2CCC2)CC1 c1(CS(=O)(=O)N(C2(C(OC)OC)CC2)CC2CC2)cc(C)ccc1C c1(OC)ccc(CN(C(c2cccc(Cl)n2)C(=O)NCC2CCOC2)C)cc1F CC1(C)C(O)CC1(C(=O)O)NCc1ccc(-n2cncn2)cc1Cl c1(NCCOC)cncc(C(=O)NCCN(C)C(C2CC(C)(F)C2)=O)c1 N1(C(c2ccc(C(=O)NCC)nc2)=O)CCOC(C)(C(=O)OC(C)(C)C)C1 N1(C(CNC(C2CCN(C)C2)=O)=O)CCN(C(=O)CC23CCCC2C3)CC1 C(CNC(=O)Cc1ccc(Cl)cc1)(C(C)C(C)C)NC(Cc1cc(C)n(C)n1)=O C1(CC(N2CC(C#C)(F)C2)=O)CC2(C1)CN(C(C1CCCC(F)C1)=O)C2 C1(C(=O)NCC(C)CN(C(=O)C(c2cccc(F)c2)O)C)CN(C)CCO1 C(=O)(CCC(C(=O)NCC1CN(C(c2cccc(C(F)F)c2)=O)C1)N(C)C)OC N1(C(CCC=CC(C)C)=O)CCC(C)C(CNC(=O)CCC#N)C1 C(=O)(C(C)CC1CCCC1)NCC(C)N(C(=O)COCCc1cccs1)CC C(=O)(CC(CC(C)C)NC(c1cc2ccccn2c1)=O)N1C(CC=C)CCCC1 N1(C(COCCC)=O)CC=C(CNC(c2ncc(F)cn2)=O)CC1 C(CC(=O)Nn1ccnn1)N(C(=O)C(CC)C(=O)CC)C1CC1 N1(C(Cn2nnc(C)n2)=O)CCCCC1Cn1cc(CCN2CCCCC2)nn1 c1(OC)ccc(Br)c(C(N2CC3(C2)CN(C(=O)Cn2ccc(C)n2)C3)=O)c1F c1(CC)ccc(C)cc1C(=O)NC(C1CN(C(=O)CCn2cnccc2=O)C1)C Cn1c(=O)ccn(CC(=O)NCC2CN(C(=O)CC3CC3)CC2(F)F)c1=O CC1(C)CC(C(=O)NCCOCCNC(c2cn3cnnc3cn2)=O)CNC1=O c1(C(N2CC(NC(c3c(OC)cccc3)=O)C(C)C2)=O)cc(Cl)ccc1N Cc1ccc(C(N2CC(NC(=O)CC3CCCSC3)CC23CCC3)=O)cc1C#N CC(CC(F)(F)F)N(C(C(=O)NC1COCC1)C(C)C1CCCOC1)C C1(NC(C2C(C#C)C2)=O)CC2CN(C(=O)C=Cc3cnc[nH]3)CC2C1 CC(CNC(=O)C=CCNC(c1ccc[nH]1)=O)CN1CCCC1 C=CC1(CC)COCCN1C(=O)CS(=O)(=O)CC1COCCO1 C(C(C)(O)CC(=O)NCC1CC(C)(C)CN1C(=O)Cc1ccc(C)cc1C)OC C1(NC(c2cncc(Cl)c2)=O)COC2CN(C(C3CCC34CCOCC4)=O)CC12 c1(C(N2CC(C(=O)NC3CCN(C(C)C)C3)C(F)C2)=O)ccc2cncn2c1 c1(CN2CCC(O)(C(=O)NC3CC3)C2)cc([N+](=O)[O-])ccc1Cl C(=O)(C1Cc2ccccc21)NC1CCN(C(c2c(OC)ccs2)=O)C(C2CC2)C1 Cc1cc(NC(=O)C(C)NC(C2CCCC2)=O)ccc1Cl.C12CCC(C1)C(=O)N2 c1(-c2c(CN3CCN(C(C(C(C)C)O)=O)CC3)cccc2)cc(O)c(F)c(F)c1 CC(=O)CCCCC(=O)N1CC2CC2(C(N2CCC3(CCO3)C2)=O)C1 Cn1nnnc1C(c1cnn(-c2ccccc2)c1)NC1CCSCC1 c1(C(CCN2CC(NC(=O)OCC)OCC2)=O)ccc(Cl)c(F)c1 CC1CCCN(C(=O)CC2CC3CC3C2)C1.c1ccccc1-c1nn[nH]n1 C1(NC(c2cnc(N(C)C)o2)=O)CN(S(=O)(=O)Cc2ccccc2Cl)CC1O N1(C(C(CSC)(C)C)=O)CC2OCC(NC(C3CC4(CCCO4)C3)=O)C2C1 N1(C(C(CC=CC)C)=O)CC(NC(=O)Cn2nc(C)n(C)c2=O)CC12CCC2 CCCC(CNC(c1ncccn1)=O)C(=O)NC(c1ccccc1)C1CCC1 N1(C(CS(=O)(=O)NC)=O)CCC(NC(=O)CC2CCC(C)(C)C2)C(F)(F)CC1 C12(C(N(CCCCNC(CC3CCC(C)O3)=O)C)=O)CC3CC1(CO)CC3C2 C1(C(=O)NC(C2N(C(CCCOCC)=O)CCC2)(C)C)CS(=O)(=O)CC12CC2 c1(OC)cccc2c(N3CC4CC3CN4Cc3ncc[nH]3)ncnc12 c1(CC(=O)NCCC(C)NC(c2nccnc2C(N)=O)=O)ccc2c(c1)COC2 C=CC(CC)CC(=O)NCC(CO)NC(=O)C(C)=C1CC1 N1(C(C(C2(O)CCC2)NC(C(CCOC)C)=O)=O)CCCOCC1C c1(C(N2CCC(C(N(C(C(C)SC)C)C)=O)C2C)=O)cc(=O)n(C)cn1 CC1Cc2cccc(C(=O)NCC3CCCCN3C(c3ncccc3F)=O)c2O1 C1(CNC(=O)NCCc2c(C)ccnc2)CCC2(CCC2)CO1 n1(CC(=O)OCCC2CC(F)C2)ccc(=O)c([N+](=O)[O-])c1 Cc1nc(C(N2CCC(O)(C(C)CNC(=O)COC3CCCC3)C2)=O)c(C)s1 C=CC1OCCC1NC(C1(OC)CCN(C(=O)C=CC2CCOCC2)C1)=O C1(CCC)C(=O)NCCN1C(=O)C(CC)N(C)C(c1ocnc1C)=O C1(C(=O)NCC2(C(=O)NC3CCCC(C)CC3)CC(=C)C2)C2CCCCCC12 C(=O)(C(C)(C)CS(N)(=O)=O)N1CC(N(C(c2cc(C)n(C3CC3)n2)=O)C)C(F)C1 c1(C(N(C)CC2(NC(C3ON=C(C)C3C)=O)CC2)=O)sc2cccnc2c1Cl CC(=O)CCCC(=O)N1CC(CNC(c2cccnn2)=O)C2(CC2)C1 C(=O)(C1SCCc2sccc21)NCc1ccc(CN(C(CC(C)C)=O)C)cc1 c1(C(N(CC(O)CNC(c2ccnc(C3CC3)n2)=O)C)=O)cccc2oc(O)nc12 C=C(C)CCC(=O)NC(CNC(c1ccncc1OCc1cccs1)=O)C(C)C c1(C(=O)NCC2(O)CCN(C(c3cc(F)ccc3F)=O)C2)ccc2cncn2c1 N1(C(=O)CCCC2CCC2)CCCC(F)(CNC(C23CC(F)(C2)C3)=O)C1 C1(CCNC(c2cc(COC)on2)=O)COCCN1C(=O)CCC1CCCOC1 C(C(C)C#N)NC(CN(C(=O)C=C(C)C1CC1)CCOC)=O c1(C(N(CC(CN(C(=O)CC2C(C)(C)C2(C)C)C)O)C)=O)ccc2c[nH]nc2n1 c1(C(=O)NC2CC(C)(NC(CC34CC(C)(OC3)C4)=O)C2)ccc2oc(=N)[nH]c2c1 C(=O)(C#CC1(C)CCCO1)NC1CC(N(C(Cc2ccc(C)nc2Cl)=O)C)C1 c1(C(=O)NC2C3(CC(NC(C4(C)CNC(=O)C4)=O)C3)C2)nc2cccnc2s1 N1(C(C2CC(C)C2)=O)CCC2(CC1)CCN(C(=O)CCC(N)=O)C2 C=C(C)CN=C(NC1CC(CC(=O)NC2COC2)C1)N1CCC(OCC(C)C)CC1 C1(C(=O)NC2CCN(C(CCSC)=O)CC2)CCc2n[nH]cc2C1C C(CCC1CCC1)(C(=O)NOC1CCOC1)NC(COC(c1nc[nH]n1)C)=O c1(C(=O)NC(CN(C(c2cnc(C(C)=O)s2)=O)C)C)coc(S(=O)(=O)N(C)C)c1 C1(CNC(C(C)=C2CCCC2)=O)CN(C(c2cccc(N)n2)=O)CCN1C N1(C(CC(=C=C)C)=O)CC2(CC)CC1(CNC(=O)C(c1ccccc1)O)C2 c1(C(=O)NC2C(C)(C(C)C)C2)cnn(CCNC(C2(CCN(C)C)CC2)=O)c1 N1(C(c2ccsc2)=O)CCC2CN(C(C3CN(CC4(CO)CC4)C3)=O)CC12 N1(C(C(C)OC2COC2)=O)CCC(O)(CNC(c2cc(F)cnc2O)=O)CC1 c1(C(N2CCCC(N(C(C(CC=CC)C)=O)C)C2)=O)cc(CC)ccc1F C=C(Cl)CC(C(=O)NCC1(S(C)=O)CC1)NC(=O)CC1CCCNC1=O N1(C(C2C(C(=O)NCCc3ccccc3)C2)=O)CCCC1c1ccccc1 N1(C(CN(S(C)(=O)=O)C)=O)CCCC1CCNC(C1(CO)CCCO1)=O CC(CNC(=O)OC(C)(C)C)CC(=O)NCCNC(=O)C(C)Cc1ccncc1 c1(C(=O)NCCCCN(C(C2CCOC2)=O)C2CC2)cc(OCC(F)F)ccn1 c1(NC(C)Cc2ccc(C3CCCC3)cc2)cccc2c(C(=O)O)nccc12 c1(C(NOC(CC)C(=O)OC)=O)c(CNC(c2ncoc2C(C)C)=O)nnn1C N1(C(C=CSC)=O)CCCC2CN(C(c3ccc4c(c3)OCO4)=O)CCCC12 N1(C(C2CC(C(C)C)C2)=O)CC2CCN(C(=O)CCc3cccc(O)c3)C(C2)C1 c1(CC)nc(=N)[nH]cc1C(=O)N(C)CC1CC1C C1(C(=O)NCCCOCCCNC(C(CSC)(C)C)=O)CC2(CCOCC2)C1 c1(N2CC(C(C)N(C(=O)CCc3cn(C)cn3)CCO)C2)cc(O)nc(=O)n1C CN1CCOc2c(C(=O)NC3CC4CC(NC(=O)C(C)(C)C)C4C3)cccc21 C1(NC(C2(SCC)CC2)=O)CN(C(C2CCCOCC2)=O)CC1C1CC1 C1(NC(c2ccc(C)cn2)C2CC2)CCNC2(CCC2)C1 C=CC(C)CC(=O)N1CC2CC1C2NC(=O)CNC(c1cc(C)oc1C)=O C(=O)(C1CCCc2nc[nH]c21)NCC1CCN(C(c2c(N)nc(Cl)cc2Cl)=O)C1 N1(C(CNC(C(CC)C)=O)=O)CC2CC(C1)C2NC(C1CCCCO1)=O N1(C(C2CCCSC2)C(=O)NC(C)C)CCCCC2(CCC2)C1 N1(C(C(C(C)C)F)=O)CCCC(O)(CNC(c2ccnc(OC3CC3)c2)=O)CC1 c1(OCC(N2CCC(C)(NC(C(CC=CC)C)=O)C2)=O)c(C)cc(Cl)cc1C Cn1nc(C(=O)NCCC2CCCN2C(=O)C(F)C2CCC2)c2c1CCCC2 C#CC1(C(N2CCC(N(CCC)C(C3CC3c3cccs3)=O)CC2)=O)CCCC1 C1(F)(C(N2CCC(OCC#C)C2)=O)CCN(C(c2n[nH]c(O)n2)=O)CC1 c1(NC(c2cc(F)ncc2Br)=O)cccc(F)c1C(=O)Nc1ccc(Br)c(Br)c1 c1(C(=O)NC(CNC(c2[nH]cc(C)c2)=O)C2CC2)ccccc1N1CCCC1=O Cc1coc(C(=O)N(C(c2ccccc2)CNC(=O)Cc2ccsc2)C)c1 C1(C(=O)NC(CNC(COc2c(C)cc(Cl)cc2)=O)C)CC2CCCCN2C1 C1(N(C)C(c2ccco2)=O)CN(C(c2cc(Cl)ccn2)=O)CC12CC2 c1(CC)cc(F)ccc1-n1nc(CCCO)nc1C1CC12CCOCC2 S(=O)(=O)(c1ccc(C#N)c(N2CCC(C(C)O)CC2)c1)NCCC(CC)C n1(C(C)C)nc(C(=O)NCCCC(C)NC(C2(C)CCCO2)=O)c(Br)n1 c1(C(N(C)CCN(C)C(c2cc(C3CC3)ns2)=O)=O)sc2cccnc2c1Cl C1(CC(=O)N(C)CCn2cccn2)CCCC1NC(c1nsnc1O)=O C1(CCNC(C2C(OC)C2)=O)CSCCN1C(=O)C(=O)Cc1ccc(Cl)cc1 C#Cc1ccc(C(=O)NCCCN(C)C(c2ccn(CC(C)C)n2)=O)cn1 N1(C(COCC(C)(C)C)=O)CCCC(C2CCN(C(=O)C3=COCCC3)C2)C1 CC1(c2nn[nH]n2)CCCN(CCS(C)=O)C1 CCC(C)(C(=O)N1CCC(N(C(=O)Cc2cc(-c3ccccc3)on2)C)C1)OC N1(C(c2cc(NC(C)=O)ncc2)=O)CC2CCC(C1)N2C(=O)CC1(C)CC1(F)F N1(C(c2ccc(-n3ccnc3)c(F)c2)=O)CCC(C)N(C(=O)CSC2CC2)CC1 C1(NC(C(c2ccccc2)=O)=O)CN(C(C2CC2c2cccc(F)c2)=O)CC1O C#CC1(C(=O)NC2(C)CC3(CC3)C2)CCN(C(=O)CCc2nccs2)CC1 c1(C(=O)NCC2CC(CNC(C(CC=C)C)=O)C2)ccc2c(c1)COC2=O C(CN=[N+]=[N-])(C(C)C)NC(c1c(OC)cccc1)C(N1CCNC(=O)C1)=O C(c1cncc(C)c1)=CC(N1CCC(N(C(C2CC2(F)Cl)=O)CC)C1)=O C=CCC(CC=C)C(=O)NC(C)CCC(=O)N1CC(CC23CC(C2)C3)C1 c1(C(=O)NC2C(C)CN(C(=O)CN(C)S(N)(=O)=O)CC2)[nH]nc2c1CCC2(C)C N1(C(C(C)NC(=O)Cc2ccco2)=O)CC2C(Cc3ncccn3)C2C1 C(=O)(C(=O)CCC(C)C)N1C(C(=O)NC(CC=C)(C)CC=C)CSCC1 c1(SC)ccc(O)c(C(=O)NCC2CC2CNC(=O)C(N2CCNC2=O)C)c1 c1(C(=O)NCCn2cc(C3(OCC)CCOC3)nn2)nc2cc(Cl)ccc2o1 c1(C(CC)C)ccc(C(C(C)C)Nc2ncc(C3CCC3)s2)cc1 C1(NC(c2c(OC)nc(Cl)cc2)=O)CN(C(C23C=CC(CC2)C3)=O)CC(F)(F)C1 C(=O)(C(O)CNC(c1coc(C)n1)=O)NC(c1cnn(C)c1)CC Cc1ccc(Br)c(C(=O)NCC2CCCC2NC(=O)CC(C)C)c1 CC1CC(CNC(c2cc(C3CCC3)on2)=O)CN1C(=O)CN1CCSCC1 CS(=O)(=O)CC(=O)N1CCC(C2N(C(c3cnccn3)=O)CC2(C)C)CC1 C(CCC1CCC1)(C(=O)Nc1ccsc1)NC(C(OCC)OCC)=O C1(C(N2CCC(=C)CC2)=O)CCC2(C1)CC2(F)F N1(C(CS(=O)(=O)NC)=O)CCC2CCC(NC(=O)Cc3cnn(C)n3)C1C2 CCC(O)C(C)C(=O)NCC1(NC(C2CN(S(C)(=O)=O)C2)=O)CC(F)(F)C1 C1(C)(CC)CC(C(=O)N(C(C)CCNC(C2(COC)CCC2)=O)C)CCO1 C(=O)(C1(C)OCCc2ccccc21)NC1C(NC(C2(CC)CC2)=O)CC1 C(C(=O)NOCC=C(C)C)(C1CCOC1)NC(c1cc(OC)n[nH]1)=O c1(C(=O)NC(C)CCCNC(C2(C)C(C)(C)C2(C)C)=O)ncc(Cl)c(N)c1Cl c1(C(C)C(=O)NCCN(C(C2CC(N(C)C)C2)=O)C2CC2)ccc(F)c(F)c1 n1(CC(=O)N(CCC)CCNC(c2csnc2C)=O)nc(C)n(C)c1=O C1(C(N2C(CNC(c3c(CC)[nH]cc3)=O)CC(F)C2)=O)Cc2ccccc2C1 C(=O)(CCCC(=O)OCC)N1CC(CNC(C2(CC=C)CCCC2)=O)C(C)C1.O Cn1nc2c(c1CNS(=O)(=O)c1cscc1C(F)(F)F)CCCC2 C1(CC=C)(NC(C2CCCC2CC)=O)CCCN(C(C2COC(C)(C)C2)=O)C1 C(=O)(CC(C(C)(C)C)NC(c1ccc(O)c(C)c1)=O)NCC(C(=O)OCC)C C1(NC(c2ccc(Br)nc2O)=O)CCCN2CCCC12 n1(CC)cc(Cl)c(C(=O)NCC(C2CCCCC2)NC(C2CCC(C)(C)C2)=O)n1 Cc1ccc(-c2ccc(C(N3CC4CC4(C(=O)NC4CC4)C3)=O)cc2)cc1 C12(C(=O)Nc3ccc(C(=O)OC)c(O)c3)CCN(C(C3CCNC3=O)=O)CC1C2 c1(C(N2CC(NC(CN(C(=O)OC)C)=O)C(F)CC2)=O)cn2c(n1)CC(C)CC2 S(=O)(=O)(c1ccccc1Br)NCCC1CCCN(C(c2ccsn2)=O)C1 C1(CCCCCNC(C(C)OC2COC2)=O)CCN(C(c2nonc2N)=O)CC1 C=CC(C)(C)C(=O)NC1CCCN1C(C1COCCN1C(=O)NC(C)C)=O Cc1c(C(=O)NCC(C)(C)NC(=O)Cc2cnco2)cnn1-c1ccccc1F Cc1cc(C(=O)NCC2(NC(=O)CC3C=CCC3)CCOCC2)n(CC(F)F)n1 N1(CC(=O)N(CCNC(c2c(C)con2)=O)CCOCCO)CC(=O)NC1=O C1(NC(CN2CC(CC)C2)=O)CC(NC(c2cc(C)cc(C)c2)=O)C12CCC2 CON(CCC(=O)NCCN1CCCCCC1)C(=O)C(C)OC(C)(C)C C(N=c1[nH]c2c(c(=NCCc3c[nH]nc3O)[nH]1)COCC2)C1(CO)CC1 c1(OC)ccc(Cl)c(CC(=O)NCc2ccc(NC(c3cscn3)=O)cc2)c1F C1(CC)CC(C(=O)NC23CCCC(NC(=O)C=C(C)Cl)(C2)C3)CC(=O)N1 O=C1CCC2CCN(C(=O)Cc3cccc(C4CC4)c3)C1C2 CCC(CC)CC(F)C(=O)NC1CC2(C1)CC2C(=O)NCCC1CC(C)C1 C1(SC)(CNC(c2nnc(NC(=O)NCc3ccc(Cl)cc3)o2)=O)CCOCC1 c1(C(=O)NC23C(CN(C(C(C(C)C)SCC)=O)C2)C3)ccc2ccccc2c1C c1(C(=O)OCC2(C)CCC(C(=O)OCC)C2)onc2c1CCCC2 c1(OC)nc(C)ccc1C(N1CC(N2CC(NC(c3cnns3)=O)CC2=O)C1)=O c1(OC)c(C(N2CCC(CC(=O)Nc3cc(O)nc(OC)n3)C2)=O)cccc1F Cc1cc(C(=O)NCc2ccc(CN(C(=O)C=CS(C)=O)C)cc2)c(C)nc1C c1(NC(C2CC(C)(NC(COCc3onc(CC)n3)=O)C2)=O)cccc(C)c1 c1(NC(CN(C(=O)C(F)CC2CC2)CC)=O)ccc(OC)c(C)c1 c1(C(=O)NCCOCCCN(C(=O)CCn2cnc(=N)[nH]2)C)ns[nH]c1=O c1(C(N(CC(C)NC(C(C(C)C)SCC)=O)C)=O)nn(C)c(Br)c1C c1(C2(C(=O)NCC(CO)NC(C3(C)CCC(=O)N3)=O)CC2)cccc(F)c1F C(=O)(CC(C)(C)SC)N(CCCCN(C(C1C(=C)C1)=O)C)C CC(C)CC(CCO)NC(=O)CC1C2CCCC2N1C(=O)CC1CC2(CCC2)C1 Cc1c(NC(C2CCN(C(C3CN(C)C3)=O)C2)=O)cccc1F N(C(=NCCN1CCOCC1)NC1CCS(=O)(=O)C1)Cc1cn(C(C)(C)C)nc1 c1(C(N2C(C(=O)OC)CN(C)CC2)=O)ccc2c(c1)CCCNC2 Cc1[nH]nc(C(=O)NC2CN(C(C3CCC=CCCC3)=O)CCC2F)c1[N+](=O)[O-] CCCCCCC(C(=O)N1CC(CO)CC(O)C1)NC(=O)CCCCC(=O)OC C(=O)(C1CCCn2ccnc21)NC1(C)CCN(C(CC2CCN(C)CC2)=O)CC1 C12(CNC(CCCC(C)=O)=O)CN(C(c3cc(O)ccc3C)=O)CC(F)(C1)C2 C#Cc1cccc(C(N2CCCC(C)(CNC(c3ncn(CC)n3)=O)C2)=O)c1Cl C1(NC(C2C(C(C)C)C2)=O)CCc2onc(C(=O)NCc3cncc(F)c3)c2C1 Cc1nc(N2CC3C(NC(C4(C)CS(=O)(=O)C4)=O)C3C2)c2cnn(C)c2n1 Cc1cncc(CC(=O)NCc2ccc(C(=O)NC3C(C)CCC3C)nc2)c1 C1(NC(C(CC=C)OC)=O)CN(C(c2cc(C(C)=O)cn2C)=O)C2(CCC2)C1 C1(C(=O)NCC(C(C)(C)O)F)C2CC(O)C(C2)N1C(C1CCCS1)=O c1(C(N2C(C)(CNC(C(COC)(C)C)=O)CCC2)=O)cccc2c1CCCCC2 Cc1cc(-n2cc(CCN(C(=O)CC3OCCOC3(C)C)C)nn2)cc(F)c1 N1(C(c2cc(CCC)[nH]n2)=O)CC(CNC(C2CC(SC)C2)=O)C(C)C1 CCC(CC(=O)NC1CC2CCC1C(NC(=O)CCC(N)=O)C2)C(C)C N1(C(C2CC(C)(O)C2)=O)CC2(CC(NC(=O)C=Cc3cncnc3O)CO2)C1 N1(C(C(C(C)C)OCC)=O)CCC2(CC2NC(c2cc(C#N)c[nH]2)=O)C1 CC1(C(=O)NCCC2CCCN(C(=O)CCOC3CCCC3)C2)CCOCC1 Cc1cc(C(=O)NC2(N3CCN(C(=O)C(C)(C)C(N)=O)CC3)CC2)n2nccc2n1 N1(C(c2ccc(C)s2)=O)CCC2(CCCN(C(=O)CCCCN(C)C)C2)CC1 C=CCC(F)(F)C(=O)NCC1CC(CNC(C2CCC(CC)C2)=O)C1 c1(C(=O)NCCCOCCNC(c2cc3scnc3[nH]2)=O)cnc2[nH]cncc1-2 C1(NC(c2cscn2)=O)C=CCN(C(=O)CCC(F)F)C1 C(N=c1[nH]cnc2ccccc12)C1CN(C(c2c(OC)cccc2)=O)C(C)C1 C1(NC(CCCNC(N)=O)=O)CC2CCC1(C(=O)NCCOCCF)C2 N1(C(CNC(C(CC)C)=O)=O)CCCC12CCN(C(c1nnccc1C)=O)C2 CCCCC(=O)NCC1(C(=O)NC2COCC2CC)CC=CC1 c1(C(=O)NC2CCCC(NC(c3cc(C)no3)=O)C2)cc(O)ccc1Br N(C(=NCC1OCCC1(C)C)NCC1(C)CCC1)C(c1ccccc1)C C(C)(CN=c1nc2[nH][nH]cc-2c(O)n1)NC(CNC(CCNC(C)=O)=O)=O CC1CCOCCN1C(=O)CCc1ccccc1 Cn1nc(C(F)F)c2cc(C(=O)NC3CCOCC3N3CCCC3)sc12 N1(CC(=O)N(C(C)Cc2ccccc2Cl)CC)CCCCC1n1ccc(C)n1 c1(C(=O)NC2C(NC(C(C)OC)=O)C2)cccc(C2(O)COC2)c1 c1(CCC(=O)NCC(C)CN(C(=O)CC2CCCC2)C)nc2ccccc2s1 C(N=c1nc2sccc2c(NC2CCCC2C#N)[nH]1)c1c(OC)c(C)cc(C)c1 c1(SC)ncc(C(=O)NC(C)CC(C)NC(=O)Cc2c(C)cccc2Cl)c(O)n1 C1(NC(c2c(C)n(CC(C)(C)O)nc2)=O)CCN(C(c2n[nH]cc2Br)=O)C1(C)C N1(C(C=Cc2c(C)n(C)nc2)=O)CCCN(C(c2ns[nH]c2=O)=O)CC1C N1(C(C)=O)CCCC(NC(C2C3CC2N(C(C2CC(=O)CS2)=O)C3)=O)C1 CN(C)C(=NCC1(C(N)=O)CC1)NCC1(c2ccc(Br)cc2)CCC1 c1(O)ccc(C2CCCCC2)cc1C.C(C1CONC(=O)N1)OC c1(C(N2C(C)(CNC(C3CC3C(F)F)=O)CCC2)=O)cc(O)c2ccoc2c1 C1(C)(CC)CC(NC(C2(C(=O)OC)CC2)=O)CN1C(=O)Cc1cnc(C)o1 C(=O)(CC(F)(F)C(=O)OC)NC1(COC)CN(C(CCCCOC)=O)C1 n1(CCOC)nc(C)c(C(N2CCC(C(C(F)(F)F)C(=O)OC)C2)C2CC2)c1C C1(C(=O)NCCN(C(C(CC)F)=O)C)CCc2cnn(CC)c2C1 CCC(CC(=O)N(CCNC(=O)C(=CC1CCCCC1)F)C1CC1)C(C)(C)C c1(C(=O)NCC=CCNC(c2cc(=O)cc(Cl)[nH]2)=O)ccn2ccnc2n1 N1(C(C2CCC(=C)CC2)=O)CCC(CC)(NC(c2c(C)cccc2C)=O)CC1 C1(NC(c2cn(C)nc2Br)=O)CCCC(NC(=O)Cc2cnn(C)c2)CC1 c1(C(=O)NC(CCNC(C2C(C)(CC)C2)=O)(C)C)ccc(C=CC(=O)OC)cc1 CCC(CC)(CN=c1[nH]c2c(cc1C#N)COCC2)NC(C1CC2CCCC12)=O C1(CNC(CCOC(C)=O)=O)(COC)CCN(C(C2CCOC2C)=O)CC1 C(CCC(C)C(=O)N1CC(CCNC(c2occ(C)c2C)=O)C(C)C1)OC Cc1nc2ccc(C(=O)NCC3CCCCN3C(c3cnco3)=O)cc2nc1C CCCCCCCCC(=O)N1CC2CCC2(C(=O)NOc2ccccc2F)C1 C1(OC)CN(C(C2(C(C)(F)F)CC2)=O)CC1NC(c1cc(C2CCC2)no1)=O Cc1ccc(C)c(OCC(=O)NC(C)CNC(=O)CC=C(Cl)Cl)c1 C1(NC(CCCN=[N+]=[N-])=O)CC2CCC(C1)C2NC(C1CC(=O)N(C2CC2)C1)=O N1(C(Cc2cc(C)cc(C)c2)=O)CC2CCN(Cc3ccc(C)c(Br)c3)CC2C1 C(=O)(CC(C)(C(F)F)N(C)C)NC12C(CN(C(C3CC(CC)NC(=O)C3)=O)C1)C2 C1(CNC(c2c(C(C)C)cco2)=O)CN(C(=O)C(C)C(F)F)C2(CCOCC2)C1 Cc1cc(C(C)C)ccc1CN(C)C(=NCC1CCOC1)NCC(C)C(C)(C)C N1(C(C2CC(CC)C2)=O)CCOCC1CN(C)C(c1sccc1C(=O)OC)=O C1(NC(c2c(C)cn(C(C)C)c2)=O)CC2CC1CN(C(=O)C(c1ccn(C)n1)C)C2 CC1(C)CN(C(=O)CCn2ccc(=N)[nH]2)CCC1NC(c1ccc(CO)cn1)=O Cc1cccc(C(C)C(=O)NCC(C)NC(c2cnc(S)n2C)=O)c1 c1(C(=O)NC(C)(C(N2CC(F)C(F)C2)=O)C2CCC2)ccc2cc[nH]c2c1 C(c1ccc(F)cc1F)=CC(N1C(C(=O)NCCc2ccc(Br)s2)CCCC1)=O O=C(C1CS(=O)(=O)c2ccccc21)NC1C=CCN(C(C2(C3CC3)CCC2)=O)C1 N1(C(=O)CCCn2cc(CC(O)C3CC3)nn2)CCC(S(=O)(=O)C(F)F)C1 Cc1c(Cl)c(C(=O)N(CCC(C)NC(c2cc(Cl)c[nH]2)=O)C)nn1C Oc1c(CN=C(NCC2CCCCO2)NC2CCCCC2F)cccc1Br c1(OC)cccc2c1OCC(CNC(=O)NC1CCN(c3cc[nH]n3)C1=O)C2 CCC(CC)CCC(=O)NCC1CCCN1C(=O)C(c1cccc(F)c1)F c1(C(N2C(C)CC(NC(CNC(=O)NC)=O)C2)=O)cc(C)c(O)c([N+](=O)[O-])c1 c1(C(=O)NC2CN(c3nc(SC)nc(C)c3)CC2F)ccc(F)c([N+](=O)[O-])c1 CN1CCOCC1CC(=O)NC1CC(CCNC(=O)CCSc2ccccc2)C1 CCC(CCC(=O)NCC1(O)CCCC1(C)C)NC(C1CCC(CC)CC1)=O C1(NC(c2cc(C)ncc2)=O)CN(C(c2sc(Cl)c(Cl)c2C)=O)CCC1C Cc1nc(C2CCC2)oc1C(=O)NC(C1CN(C(c2c(Br)nnn2C)=O)C1)C Cc1ccc(C(N2CC(NC(=O)C(c3cn(C)nc3C)O)C(O)C2)=O)c(C)n1 c1(OC)ccc(C(N2CCC(NC(=O)CSS(C)(=O)=O)C2C(C)(C)C)=O)c(F)n1 N1(CC(NOCCC(C)O)=O)CCN(C(C2CCC(=O)CC2)=O)CC1 CC1CN(C(c2ccccc2SCCO)=O)CCN1C(C1COC2COCC12)=O N1(C(C2(CC(C)C)CC2)=O)CCC(C(O)CNC(=O)CC2CSCCO2)CC1 c1(CNC(=O)NCC(=C)C)cn(C)nc1Br C1(NC(C(CCC)OC)=O)CCC2(CC1)CN(C(=O)C=C1CCC1)CCO2 c1(CN(C(C2N(C(C=CCN(C)CC)=O)CC2)=O)C)ccccc1C c1(C(c2n(C3(C)CC3)nnn2)NC2CC(=C3CC3)C2)ccc2cc(Br)ccc2c1 O=C1CN(C(=O)C(F)CC2CN(C(c3cnn(C(F)F)c3)=O)C2)CC2(CC2)N1 S(=O)(=O)(c1ccccc1S(C)(=O)=O)N1C(C(=O)Nc2ccc(OC)nc2)CCC1 C1(CCCC)CN(C(=O)CCC2CCCN2C)CCN1C(=O)Cc1sccc1Cl C1(NC(C2(C)COC(=O)N2)=O)CN(C(C2CC(C3CC3)C2)=O)C2(CCCCC2)C1 C1(n2cc(-c3nc(CC)sc3)nn2)CCCN(C(C2(C)CC2C)=O)CC1 C1(NC(C(C)CC#N)=O)CC(C(=O)NCC(C)(C)N2CCCC2)=CC1O C1(O)(CCNC(=O)CC2CC(C(=O)OC)CCO2)CCN(C(=O)C2CC2)CC1 c1(C(=O)NC2CCC(NC(=O)C3=CCCS3)CC2)cnn2cc[nH]c(=O)c12 N1(C(=O)C(c2cccc(F)c2)O)CC2(CCN2C(C2CCS(=O)(=O)C2)=O)C1 N#Cc1ccc(NC(c2coc(-c3ccccn3)n2)=O)cc1-c1ccncc1 CC(C)CC(CNC(=O)Cc1cc(C(F)(F)F)n[nH]1)NC(=O)CSc1nc[nH]n1 c1(SC)ncc(C(N2CC(F)CC2CNC(C2(CO)CC2)=O)=O)n1C C(CC(O)CC(=O)NC1CCN(C(=O)CCC(=O)c2cnn(C)c2)CC1O)SC c1(C(=O)NC2CN(C(c3cnc(N)c(Cl)c3)=O)C3C2C3)ccc2c(c1)COC2 N1(C(c2cn(CCC=C)nn2)=O)CC2CN(C(c3ccsc3Cl)=O)CC2(C)C1 c1(OC)ccnc(C(=O)NC(C)C(C)NC(c2cc(C3(O)COC3)on2)=O)c1F C#Cc1ccnc(C(=O)NCC2(C)CCCN2C(c2ccc(C)c(NC)c2)=O)c1 c1(C(N2CCC(n3cc(CC(C(C)C)O)nn3)C(O)C2)=O)cc(I)cc(Br)c1C CC1Cc2ccccc2N(C(c2cc(F)c(N)c(F)c2)=O)C1C C1(CC(=O)NCc2ccc(F)cc2)CCN(C(=O)Cc2cc[nH]n2)CC1 c1(CN2CC3CN(C=O)CC32)sc2ccccc2c1Cl.c1(N)cccc(Cl)c1F N(C1CCCc2occc21)C(C(CCSC)NC(C1CCN(C)CC1)=O)=O N1(C(CC2(N(C)C)CC2)=O)CC(NC(=O)CC2(C(=O)OCC)COC2)CC(O)C1 N1(C(c2cc(C)oc2)=O)CCCC(N(C)C(c2cc(C3(C)CC3)n[nH]2)=O)C1 c1(CC(=O)NC2CCC(NCc3c(C)ncs3)C2)ccc(Br)cc1Cl C(CC(C)C(=O)NCCN(CCOC)C(C1(c2ccc(F)cc2)CCC1)=O)=CC N1(C(C(CC=CC)NC(C2CCC(C)(C)OC2)=O)=O)CC2COCC2(C)C1 O=S(=O)(c1ccc(Br)cc1NC1(C2CCCO2)CCC1)NCC1(N2CCCC2)CC1 C1(CC)CN(C(C2COCCC2(F)F)=O)CCN1C(c1cncc(C(C)C)c1)=O C12(NC(C3C(SC)CCC3)=O)CCC(NC(c3oc(C)nc3C)=O)(CC1)C2 Cc1nc(C)c(-c2nc(C3CC=CCC3)nn2C2CCCOC2)nc1C N1(C(C2(CCNC(C3(F)C(C)(C)C3(C)C)=O)CC2)=O)CC2(CCNC2=O)C1 Cc1oc(C)c(C(=O)NCC2CC(C)CN(C(c3cc(F)c[nH]3)=O)C2)c1C c1(OC)nc(Nc2nc(Cl)ccc2C(=O)Nc2cc(C(N)=O)ccn2)ncc1F c12ccc(c(F)c1)CO2.c1(CNCC(CCC)C)ccccc1OC Cc1cc(-c2cccnn2)cc2c1NC(=O)CC2 C1(NC(C2CCS(=O)(=O)N2)=O)CC2CN(C(c3ccsc3C(F)(F)F)=O)CC2C1 c1(COC)ncc(NC(C23CC(NC(c4ncncc4Cl)=O)(C2)C3)=O)cn1 CC(C(=O)NCC(C1CC1)NC(C1(C(N)=O)CCC1)=O)NC(C)(C)C N1(CCCCC2(C)OCCO2)CC(C2=NOCC2)C1 C1(NC(=O)NCc2cccs2)CN(C(C2(c3ccccc3)CC2)=O)CCO1 C1(O)(CNC(c2c(CCC)[nH]cc2)=O)CCN(C(=O)C(C)SC(F)(F)F)C1 N1(C(COCCOCC#C)=O)CCC2CC12C(=O)NC(CN(C)C)CO c1(C(CC(=O)OC2CC2C(=O)NCC=CCNCC)C)cccc(F)c1 N1(C(CCC)=O)CCCC1(C(=O)NCC1CN(C2CC2)C1)COC C1(CC)CCC(C(=O)NCc2sccc2C(=O)NCCc2ncccc2C)CC1 c1(OC)cc(Cl)c(C(N2CCC(c3cn(CCO)nn3)(N(C)C)C2)=O)cc1Cl c1(Cc2n(C3CN(C(CCCSC)(C)C)C3)nnn2)ccc2cccc(C)c2n1 c1(C(N(CCCCN(C(c2nc(CC)sc2)=O)C)C)=O)cc2n(n1)CCCC2=O C1(C(F)(F)F)(C(=O)NC(CC=C)CC)CC(C)(C)C1 CCCC(CNC(C1CCCCC1OCC(F)(F)F)=O)C(=O)O C1(N(C(=O)Cc2cnoc2)C)CCC2CN(C(C3CC(C)(C)CN3C)=O)CC12 C#CC1(NC(=O)CCC2(C)CCCN2C(C2C(C)(C)C2(F)F)=O)CC2CCCC12 C1(O)(C(C)NC(=O)CCc2cccs2)CCN(C(c2c(N)cccc2Cl)=O)CC1 N1(C(C(c2ccccc2)N(C)C)=O)CC2(C1)CN(c1cc(O)ncn1)C2 c1(C(=O)NC(C2(O)CN(C(C(CC(CC)C)C)=O)C2)C)ccc(F)c2ccsc12 OC1CC2CC1CC2CN(c1cccc(C(F)(F)F)c1)C1CC2(CNC2)C1 C1(NC(COC)=O)(COC)CCN(C(=O)CNC(=O)C(F)(F)F)C1 c1(C(N2CC(NC(C3CC(C)(CC)C3)=O)C2)=O)cncc(-n2cccc2)c1 c1(NC(C2(C)CN(Cc3ncc(C)c(Br)c3)C2)=O)ccc2c(c1)NC(=O)CCC2 c1(CN(C)Cc2cncc(C(N)=O)c2)cc(C#N)cs1 C1(NC(=O)CCCn2cccc2)CCCC(c2ccccc2)C1 N#Cc1cc(CN2CC3CC3C2)ccc1Cl.c12cccc(c1)C(=O)N2 CCCC(C(=O)NCCC1CCOCC1)NC(c1ccc(F)cn1)=O c1(C(N2C(CNC(CC3C(C)C3)=O)CC2)=O)ccc(C(F)(F)F)[nH]1 N1(C(c2ccc(OCOCC)o2)C(=O)NCC2CCCO2)CCC(C2CC2)CC1 N1(C(c2cccc(OC)c2)=O)CCN(C(=O)C(n2nccc2C)C)CC12CC2 c1(C(N(CCN(C(CCC2C(C)C2)=O)C)C)=O)cn(C)nc1C1CCC1 C(C1CN(C(c2sccc2F)=O)Cc2ccccc21)NC(c1[nH]n(C)c(=O)n1)=O c1(C(=O)NCC(C)NC(c2ccc(-c3ccccc3)s2)=O)cc2cccnc2[nH]1 c1(NC(C2C3CC2N(C(C2CC4C=CC2C4)=O)C3)=O)ccc(F)c(F)c1F N1(C(c2ncc(-c3c(OCC)c(C)ccc3)cn2)=O)CC(O)C(O)C(O)C1CO C1(NC(c2c(C)ncn2O)=O)CC12CCN(C(=O)COCc1ccccc1)C2 C(=O)(C(O)CC(C)(C)C)N1C(C(C)C)CCC1C(=O)NCCC1COCC1O C1(C(=O)NC(C(C)C)CNC(C2CCCCS2)=O)CCCC(C)CC1 c1nc(N(c2cnn(-c3ccccn3)c2)C)ncc1F.CC1(C2CC2)CNC1 NS(=O)(=O)c1ccsc1C(=O)NCC12CC1CN(C(c1ccoc1)=O)C2 C1(NC(Cc2ccc(OC)nc2)=O)CC2CC1CN(C(=O)C=C(C)Cl)C2 c1(C(=O)NC2C(NC(=O)C=Cc3cccc(O)c3)CC2)cc2n(n1)CCCC2O CCC(C(N)=O)NC(C1CCN1C(c1cnn[nH]1)=O)=O C1(C(=O)NC2CC(OC)CN(C(C=CCC)=O)C2)CCn2c(C)nnc2C1 c1(C(=O)NC(CC)CNC(c2cn(C)cc2C)=O)coc2ccc(O)cc12 c1(C(C)C)ccc(C(=O)N(C)CCOCCNC(=O)CCc2ccoc2)nc1 c1(-c2scc(NC(c3cn[nH]c3)=O)n2)ccc(O)cc1F C12(C(N3C4C(NC(c5cc(F)ccc5Cl)=O)CC(C4)C3)=O)C3CC(CC13)C2(F)F c1(C(=O)NC2CC(C)N(C(c3ccccc3)=O)C2)ccc2nnn(C)c2n1 c1(C(N(CC(CC)NC(=O)CCC2CC2(C)C)C)=O)cc(Cl)c(F)cc1F C(=O)(C1=CCC2CCC1N2C(=O)CCOCC(C)C)NCC(CC=C)(C)CO C1(C(N(CCN(C(C)=O)C)C)=O)CCCN(C(=O)C=CC2CCC2)C1 C1(C(=O)OC)CCN(C(C2C(CNC(c3cc(CO)on3)=O)C2(C)C)=O)C1C C(=O)(C1CCc2cc(F)ccc21)N1CCCC(CN(C(=O)CCC2(C)CC2)C)C1 c1(C(N2CCCN(C(C3C(COC)C3)=O)C(C)C2)=O)cc2nc(C)cc(C)n2n1 c1(C(=O)NC2CC(NC(C(C)Cc3cccnc3)=O)C2)cccc(F)c1 Cc1ccc(O)cc1C(N1CCC(NC(c2ccc(C3CC3)o2)=O)C(O)C1)=O CCCC(C)CCCC(=O)NCC12CC1CN(C(c1cnc(O)n1CC)=O)C2 C(C)(C(=O)N1CCC(NC(c2cc(CCO)on2)=O)C1)(C(C)C)OC c1(C(=O)NCC(CNC(=O)C=CCO)F)ocnc1-c1ccccc1 CCCCCCC(C)C(=O)NCCC(C)N(C(=O)C=Cc1cncc(OC)c1)C C12(C=O)CC1CCN2C(=O)CC1CC(OCC)C1.C(=O)(C(C1CC1)NC1CC1)NCC C1(C(C)C)(C(N2CC(F)(CO)C2)=O)CCN(C(c2cnn(CCF)c2)=O)C1 c1(C(=O)NCCC(C)N(CCC)C)c[nH]nc1CNC(=O)C(O)C1CCCC1 CON(C(=O)C1CCCCN1C(=O)Cc1cncc(C)c1)C1CCCC1 N1(C(c2cc(C)nnc2C)=O)CC2(C=C(C(=O)N3CCC(C)(O)C3)CO2)C1 N1(C(CCCC#C)=O)CC(NC(c2sccc2F)=O)C2CCCCC12 n1(CC)ccnc1C(=O)NCC1CCCC1NC(c1cnc(Cl)s1)=O N1(C(c2n(C)c(=O)ccc2)=O)CCC=C(C(=O)Nc2cc(C(C)(C)C)no2)C1 C(=O)(C(C)CCCC(C)C)N1C(C(=O)NC(CC(C)C)C)CC2(CC2)C1 n1(CC(N2CCCCC2C2CCCC2)=O)nc2ccccn2c1=O Cc1ccc(C#N)cc1NC(C1CCCC(NC(C2(O)CCC2)=O)CC1)=O N1(C(C2CC(OC)C2)=O)CC2(CNC(=O)C(C(C)(C)C)SC)CC(F)(C1)C2 CC1(C)CCCC(C(N2CC3CC2C3NC(=O)Cc2ccns2)=O)CC1 C1(CC)CCCN(C(=O)CC(C)C(F)F)C1C(N1CC(C)(C(N)=O)C1)=O N1(C(c2cc(C)sc2)=O)CC(C)CN(C(c2n[nH]c(O)n2)=O)CC1C c1(OC)ccc(CC(=O)NCC(O)CNC(c2sccc2C2CC2)=O)cc1 C1(NC(C(C(C)OC)NC(C2CCC(=C)CC2)=O)=O)C2CCC(F)(F)C12 C(N=c1[nH]c2c(c(=NC3CCC3C3CCCC3)[nH]1)CCC2)c1cc(O)nc(O)n1 c1(OC)ncc(F)c(=NC(=O)c2cc(F)ncc2NC(=O)C(O)C(C)(C)C)[nH]1 CCC(C)(CCNC(C1CCOC(C)C1)=O)NC(c1cn(C(C)C)nn1)=O N1(c2n(Cc3c(OC)ccc(OC)c3)nnn2)CC=CCC2(CCCC2)C1 CCCCC(F)C(=O)N1CC(C(C)NC(=O)CC2CNC(=O)O2)C1 c1(C(=O)NC2(C(=O)NC(c3noc(C)n3)CC)CC2(C)C)oc(CSC)nc1C C1(NC(=O)CC2(NC(=O)CC3CCCCO3)CC2)CCCC(F)C1 C(CC(C(=O)NCC1(F)CC(CNC(=O)C=C(C)Cl)C1)NC(N)=O)SC C(CC1CCCC1)(C(=O)NCC1CC=CCC1)NC(CN(C)C(=O)C1CC1)=O C1(O)(CCNC(Cc2nc(CC)sc2)=O)CCN(C(=O)COC(C)(C)C)CC1 N1(C(C(C)NC(c2ccoc2)=O)=O)CC(NC(C2CC2(Cl)Cl)=O)C(C)C1 Cc1cccc(Cl)c1C(N1CCC(NC(=O)CS(=O)(=O)NCC2CCCO2)C1)=O N1(C(c2c(CC)cncc2)=O)CC2(C=C(C(=O)N3CCOC(CC)C3)CO2)C1 C1(NC(c2nccc(C)c2)=O)C2CC1CN(C(C1CCS(=O)(=O)N1)=O)C2 CC1(C)CN(C(=O)CCN2CCC(O)CC2)CC1NC(c1cc2ccsc2[nH]1)=O N1(C(c2snc(C)c2N)=O)CCC(C)(NC(C2CC3C=CC2CC3)=O)CC1 C=CC1(CC(=O)NC(C2CCCO2)CC)CN(C(=O)CCC(N)=O)C1 C(=O)(C(F)C(F)(F)F)C(c1ccnc(N2CCC(C)C2CN)c1)=O.CC(C)N Cc1cc(N2CCC(F)(CF)C2)nc(=NCC2CCC(CO)O2)[nH]1 c1(CC(=O)NCCC(C)NC(=O)CC2CC2)ccc(C#N)nc1 CCC(C)(CCC(C)C)C(=O)NCCNC(=O)C(C1CCCCC1)N(C)C C1(CNC(C(C)CC2CCCC2)=O)C(C)CCCN1C(=O)CCCOC(C)(C)C c1(N2CCC(CC=C)(NC(c3cc(C)n(CC)n3)=O)C2)ncc2ccsc2n1 C(=O)(C(CC(C)C)ONC(c1oc(C)nc1C)=O)NC1C(CCOC)C1 c1(OC)ccc(CCC(=O)N(CC(C)NC(=O)Cc2ccc(Cl)cc2)C)cc1N C1(NC(Cc2ccc(OC)cn2)=O)C2CC(O)C1N(C(=O)C(C)(F)F)C2 c1(C(C)=O)cc(C(N2CCC(O)(C(C)NC(C3CCOC3C)=O)C2)=O)ccc1C c1(C(=O)NCC(CNC(C(C)OCCCCCC)=O)C)ccc(SC2CC2)cc1 C1(C2(O)CN(C(c3cnc(N(C)C)o3)=O)C2)(CNC(C(C(C)C)SC)=O)CC1 C(=O)(CC(C(F)F)n1cccn1)NC(CNC(c1n(C(C)C)ccn1)=O)C C1(COC(c2c(OCC)cnnc2)=O)COCCC1(F)F N1(C(CCN(C)C)=O)CC2(CCC(NC(c3nc4ccccc4[nH]3)=O)C2)C1 c1(NCC(C)(C)CCCO)nc(N2CCC(C3CC3)CC2)nc2scnc12 CC1CN(C(C2CCCCC2CNC(C2CC(C)(C)CO2)=O)=O)CCC1(F)F C(=O)(C(F)CCC(C)(C)C)N1CC2C(C(N(C3CCC4CC34)C)=O)C2C1 C1(CNC(C(F)=CC)=O)CCN(C(c2cc3cccnc3[nH]2)=O)CC1(F)F c1(SC)cc(C(=O)NC2(CCNC(=O)Cc3csc(C)c3)CC2)oc1C c1(C(=O)NC(CN(C)C)C(=O)NCc2ccnc(F)c2F)ccc2cccnn12 CCC(C(=O)N1CC2C(C(N3CC4(C3)CN(C(C)=O)C4)=O)C2C1)C(F)(F)F N1(C2C(NC(C(C)NC(N)=O)=O)C2)CCCCC1 C1(OC)CC(NC(C2(SC)CC2)=O)CN(C(=O)C=Cc2ccc(C)s2)C1 C1(CC(=O)NC(C)(C)COC(F)(F)F)CCCN(C(=O)CCCNS(C)(=O)=O)CC1 CCCC(CCC)C(=O)N1CCN(C(c2nc(C)sc2C)=O)C(C(C)C)C1 C12(C(N(CC(C)NC(c3cc(Cl)cc(F)c3F)=O)C)=O)CC(C)(C1)OC2(C)C N1(C(C2CCN(OC)CC2)=O)CC2CCCC2(CNC(=O)CCF)C1 c1(C(=O)NCCC(C)(C)NC(=O)COc2ccon2)c(F)ccc(Cl)c1F C1(C(=O)NCC(CC)NC(c2ccncc2NC)=O)CC12CC(O)C2 CC1CN(C(c2ccc(Cl)nc2N)=O)CCC1NC(c1c[nH]nc1C(F)F)=O c1(C(=O)NC(CNC(C2(COC)CCC2)=O)C)ccc(N)c(F)c1 C1(OC)C(NC(=O)CN(CC(C)C)C(=O)C=CC2CCCC2)CC12CCC2 S(=O)(=O)(c1ccc(=NCCN(C)C)[nH]c1)N1CCC(C)(C(=O)NC)C1 C1(C(=O)NC2CC(N3CCCC3)C2)(NC(C2(C)C(C)C2)=O)CC(O)C1 C(=O)(C(O)CC(C)(C)C)Nc1snc(-c2ccc(C)cc2)n1.N12CCC(C)(CC1)C2 N1(C(CC(=O)OC)=O)C2CCC1CC(CNC(c1cnc(-c3ccco3)s1)=O)C2 C1(C)(CNC(C(C)c2cccs2)=O)CCN(C(C2(c3cccnc3)CCC2)=O)C1 C1(NC(Cc2n(C)nc(C3CC3)c2)=O)CC2CC1N(C(c1cscc1F)=O)C2 C1(C)(CNC(C(=O)NC(C)C)=O)CCC(NC(c2cc(CC3CC3)on2)=O)C1 C1(C(=O)NC2C(c3onc(C)n3)C2)CC1C1CN(C(=O)Cc2ccccn2)C1 C1(CNC(c2c(C#C)c[nH]n2)=O)C2CCCC1N(C(=O)Cc1c(Cl)cnn1C)C2 c1(C(=O)NCC(=C)CCNC(=O)CC(CC)OC)cccc(OC(C)C)c1F c1(Nc2scc(C(=O)Nc3ncc(Cl)cc3O)n2)ncnc2sccc12 Cn1ncc(S(C)(=O)=O)c1NC(=O)C(=O)NCCC1CCCN1 CCCC(C)C(=O)N(CCC(=O)NCC(C)(O)CC)CC C1(C)(CNC(=NCC2CC(OC)C2)NC2CCCCC2C)CCS(=O)(=O)CC1 c1(CNC(c2cncc(O)c2)=O)ccc(CNC(C2CC3(CC3)C2)=O)cc1 CCCCC(C)CCC(=O)N1CCCC(C)(CNC(c2ncn(C(C)C)n2)=O)C1 C1(NC(C(C)C)=O)COC2(C1)CN(C(C1(C)CCC(F)(F)C1)=O)C2 O=C(CC(C(F)(F)F)n1ccnc1)NCC1(O)CCCN(C(=O)CC2(O)CC2)C1 N1(C(C(C)SCC)=O)CC(OC)C(NC(c2ccc(-c3scnc3C)cc2)=O)C1 C1(C(N2CC3C(CNC(c4cn(C)nc4Br)=O)C3C2)=O)CC2(C1)CC2(F)F N1(C(C(C(C)C)N(C)C)=O)CCOC2(CCC(NC(c3nc(=N)[nH][nH]3)=O)CC2)C1 c1(CC)cscc1NC(=O)C(O)C1CN(C(=O)C=Cc2cscn2)C1 C1(CNC(c2cc3ccoc3s2)=O)CC2COCC2N1C(C1CC2(CC2)C1)=O N1(C(c2c(C)ncs2)=O)CC(NC(c2cnn(C3CCC3)c2)=O)CC1C C(=O)(CCC(F)(F)F)N(CC(=O)NCCOCC=C)C N1(C(CN2C(C)CCCC2)=O)CCC(C(=O)N(C2CCC2)C2CC2)C1(C)C C1(C(=O)NCC#C)CC2CCC1N2C(C1CCC(C)(C)C1)=O c1(C(N2C(CNC(C(COC)OC)=O)CCC2)=O)cccnc1C N1(CC(C)NC(c2c(CCC)nco2)=O)CCN(C(C2C=CC=CC=C2)=O)CC1 c1(C(=O)NC2CC(NC(C(C)N(CC)CC)=O)C2)c[nH]cc1Cc1ccccc1 C(CCCNC(=O)CC#N)(c1ccccc1)NC(COC1(C)CCC1)=O N1(C(CN(C)CC)=O)CCCC(C(=O)NCCC(C)C)C1C C(=O)(C1CCCc2c[nH]nc21)NC1C=CCN(C(c2c(C)cc(=O)oc2C)=O)C1 C(=O)(CCc1cccs1)NC1(CCNC(COCCN(C)C)=O)CC1 C1(NC(=O)CCCNC(C2(F)CC=CC2)=O)CCC(F)(C(=O)Nc2ccco2)C1 Cc1cccc(C(=O)NCC(CNC(C2CCCCC23CC3)=O)CO)c1Cl C1(NC(C2CCC3(CC2)CC3)=O)CCC(=O)N(CC(F)(F)F)C1 C(CC(C(C)(C)C)NC(=O)OC(C)(C)C)N(C)C(C1CCCN(CC(F)(F)F)C1)=O c1(C(=O)NC2(CNC(C=CC3C(C)C3(Cl)Cl)=O)CC2)cccc([N+](=O)[O-])c1 c1(N2CCC(CCNC(C3(C)CCOCC3)=O)C2)ncnn2c(Br)ccc12 C1(C(N(C)CC2CCN(C(c3occc3F)=O)C2)=O)CC(C2CC2)=NO1 c1(CCC(=O)NCC2N(C(C3C(OC)CCC3)=O)CC2)ccc2ccccc2c1 c1(-c2n(Cc3ccc(OC)cc3)nc(C3CC34CC4)n2)cc2cc(C)ccc2[nH]1 N1(C(C(Cc2ccco2)NC(COCCOCC#C)=O)=O)CCC(N(C)C)C1 n1(CC#C)cccc1C(=O)NCCN(C(=O)C(F)C1CCC1)C(C)C CCC(CNC(c1cc(C)c(CO)o1)=O)(CC)C(=O)NCC1CCCC1N(C)C C1(SC)CN(C(c2cnn(CC3CC3)c2)=O)CC1NC(C1CCC(=O)NC1)=O Cc1cc(Cl)ccc1OC(C)C(=O)NC1CCCC1CNC(c1cnoc1C)=O c1(NC2CCCCN(C(c3c(C(C)C)ncnc3)=O)C2)ncc([N+](=O)[O-])cc1F C(=O)(C(C)CC(C)C(C)=O)N(CC(=O)N(C(CCO)C(F)F)C)C(=O)NCC CC1=C(C)CC(C(N2CCN(C(c3cncc(N)c3)=O)C(C3CCC3)C2)=O)CC1 S(=O)(=O)(c1cc(NCC(c2cccs2)O)ccc1C)NC C(C(C)C(F)C(=O)NCCCN1CCCC1)NC(c1cncc(OC)c1)=O c1(NC2(C(=O)OCC)CC2)cc(Cl)nc(C(=O)OCC)n1 Cc1ccc(C(=O)NCC2CC3CC3N2C(=O)CC2CCC(=O)N2C)c(O)n1 N1(C(c2cnc(C(C)C)nc2)=O)CCN(C(=O)C(C)N(C)C)CC1C1CCCC1 C1(CNC(c2cccc(OC)n2)=O)CC2(C1)CN(C(C1CCOC1C)=O)C2 c1(CC(=O)NCC(C(C)(C)C)NC(C(CCC)C#N)=O)cncc2ccccc12 C=C(C)CC(C)C(=O)NC(C)CN(C(=O)COCCCC)CC c1(C(N2C(CNC(C(C(C)C)F)=O)CCCC2)=O)cc2oc(Cl)cc2[nH]1 N1(CC)CCOC(CNC(c2cc(I)ccc2Cl)=O)C1c1cnn(C)c1 O=C(C1=CCCCCC1)NCCCN(C(c1cnc(Cl)s1)=O)CC1CCCC1 CC1CN(C(C2CC2(C)C)=O)CC1NC(C1CSCCS1)=O CC(C)CC(O)C(C)C(=O)NCC(C)C(=O)N(CC(C)C(C)C)C CC(C)CC(C)(O)CNCC(=O)NS(C)(=O)=O n1(CC)nc(C(=O)NC2CN(C(c3cnnn3CC)=O)C2)c(=O)c2ccccc12 C(=O)(CS(=O)(=O)CC)N1CC(CC=C)(C(=O)NC(COC)C(C)C)C1 N1(C(c2c(COC)n(C)nc2)=O)CCCN(C(=O)CCCc2ccsc2)CC1 c1(N(C)CC)ccc(S(=O)(=O)NC2CCC(NCCF)C2)c(Cl)c1 N1(C(C(C)(C)C2CCCO2)=O)CC2OCCN(C(=O)Cc3ccoc3)C2C1 c1(-n2cc(C(N(C(C(CC)NC(=O)CO)=O)C)C)nn2)ccccc1C Cc1ncc(NC(C23C(NC(=O)C(C)Cn4ccnc4)C4CC2C3C4)=O)c(C)n1 CC(C)C(CCc1ccccc1)C(=O)NCCN(C)C(c1ccc(N)c(O)c1)=O N1(C(C2CN(C)C2)=O)CCN(C(=O)C(C)(C)F)CC1Cc1cncs1 CC(CNC(=O)CSS(C)(=O)=O)(Cc1ccccc1)NC(=O)CC1CCCOC1 CC1(C)OC2(CNC(c3cc(F)c(Cl)cc3Cl)=O)CC1(NC(=O)C1=CCOC1)C2 N1(C(CSCCC)=O)CCCC(N(C(=O)Cc2cc(C(F)(F)F)n[nH]2)CCF)C1 C=CC1(CNC(=O)C(c2ccoc2)NC(=O)COCCn2cncn2)CCC1 c1(CC(=O)NC(CN(C(C(C2CC2)OCC)=O)CC)C)cc(C(F)(F)F)n(C)n1 CC1CN(C(=O)CCC2CCC(NC(C34CC(C#N)(C3)C4)=O)C2)CC(C)N1C c1(CC(N2CCCC(C)(CNC(C(C)OC)=O)C2)=O)csc2cc(C)sc12 C1(F)(NC(c2ccc(OC)cc2C)=O)CS(=O)(=O)CC12CCC2 C12(CNC(C(CC)CC)=O)CCCC1N(C(=O)COCCCF)CCC2 c1(CN(C)C)ccc(C(=O)NC2CCC(C)(CNC(=O)C(C)(C)C)C2)cc1 c1(OC)c[nH]c(C(=O)NCC2(NC(C3CNC(=O)N3)=O)CCCC2)cc1=O C1(NC(=O)NC2CCN(C3CCCCC3O)CC2)CCS(=O)(=O)NC1 C1(CC)CC(C(N2CC(=C(F)CNC(=O)CC3COC(C)(C)C3)C2)=O)CCC1=O O(C=C(C#N)C(=O)N1CCCC1CCNC(c1cc(C(C)C)on1)=O)CC CCCCCCN(C)C(C1CCOC1CNC(=O)CNC(C1CC1C)=O)=O N1(C(c2nc(C)sc2)=O)CCC(O)C1C(N1CCC(C(F)(F)F)C1)=O N1(C(c2n(CC)nnc2)=O)CC2CCC(C1)N2C(c1cc(C)c(F)cc1Cl)=O C1(NC(c2ccc(O)cn2)=O)CN(C(c2csc(S)n2)=O)CC2(CCC2)C1 C1(CN(C(C(C)=C(C)C)=O)C)CCCN1C(c1cc(Cl)no1)=O c1(-c2nnc(C)o2)cccc(CNC(C2CC(=O)N(c3ccccc3F)C2)=O)c1 C12(C(N(CCCC#C)C)=O)CCN(C(c3cnc(CC)nc3)=O)CCC1C2 C1(N(C(C2CC3CC3C2)=O)CC)CCCN(C(=O)C=Cc2ncc(C)[nH]2)C1 CN1CCC(C(=O)NCCN(C(c2csc(C(C)(C)C)c2)=O)C2CC2)CC1 C12(C(=O)NCCc3cc(C)no3)C(NC(C3CC3[N+](=O)[O-])=O)C3CC1C2C3 Cc1ccc(O)c(CC(N2CCCC2(C)CNC(=O)COc2cc(C)on2)=O)c1 n1(CC(=O)N(CC(C)CNC(=O)Cn2nccn2)C)nc(-c2cccs2)oc1=O N#Cc1cccc(Br)c1NC(C12CC(C(=O)Nc3cc(F)cc(Cl)c3Cl)(C1)C2)=O C(=O)(CCCCCSC)NCC(C(=O)NCc1ccc(OC)cc1)OC CC(C(C)(C)C)=CC(N1CC(F)(CN(C(=O)CCCOc2ccccc2)C2CC2)C1)=O Cc1c(C(C)(C)C)o[nH]c1=NC(=O)OCCCOC(C)(C)C c1(CC2(C(=O)NCC3(O)CN(C(c4cc(C)sn4)=O)C3)CC2)c(F)cccc1F CCC(CC(C)C)C(=O)NCCC(C(C)C)NC(C1CNC(=O)CC1(C)C)=O n1(C(C)C)cccc1C(=O)NC1CCC1NC(=O)C(C)OC1CCCCC1 C(C)(C)(C(C)NC(c1ccnn1CC1CCC1)=O)NC(COCCC)=O c1(OC)nc(C)c(C(=O)NC2CCC(N(C)C(C3CC(CCO)C3)=O)C2)s1 CC1(n2cc(CCNC(N)=O)nn2)CCOCC1.c12cccc(c1)C(=O)O2 c1(C(C(=O)NCCC#C)NC(=O)C(C)NC(N)=O)cnn(C)c1 C1(NC(C2C(=C)C2)=O)C2CC3C(C2)C13C(N1CC(C)(C(F)(F)F)C1)=O Cn1cc(-n2cncc2C(N2CC(OC(=O)Nc3ccccc3)C2)=O)cn1 c1(NC(c2ccc(-c3cn[nH]c3)cn2)=O)ncc(F)cc1O C1(NC(=O)C=Cc2cscn2)COC2(CCN(C(c3ccccc3CO)=O)C2)C1 C=C(C)CCC(c1nnnn1CCC(=O)NCCC)NCCC1CC2CCC1O2 c1(C(=O)NCC(=O)NCC2CCC2NC(=O)CC2CC=CC2)cc(O)cc(=O)o1 c1(C(=O)NC(CNC(C(C)=C(CC)C)=O)(C)C)cncc2c[nH]nc12 C#CCCC(O)C(=O)N1CCN(C(C2SCCS2)=O)C(C)C1 CC1(C(N2CC3CCC3(NC(c3csc4nnsc34)=O)C2)=O)CCC12CCC2 c1(CC)cnn(CC(=O)NC(C)(CNC(=O)CC2CCCOC2)C2CCC2)c1 N1(C(=O)Nc2c(C(C3CC3c3ccco3)OC)nn[nH]2)CCCCC(C)C1 C1(CNC(c2cnc(C)s2)=O)CC12CCN(C(=O)CCn1cc(Cl)cn1)CC2 c1(CNC(Cc2cc(C)on2)=O)ccc(CNC(C2CCC(C(N)=O)O2)=O)cn1 c1(OCC(=O)NC2CCCCC2NC(=O)CCC2CCC2)cc(F)cc(Cl)c1 C12(CC)CN(C(c3sc(SC)cc3C)=O)C(CNC(C3CNC(=O)C3)=O)(C1)C2 c1(NC(=O)C(=O)NC2COC3(CCCC3)C2)ccc2sccc2c1 C(=O)(CC1=CCCCC1)NC1CCC(N(C(c2c(Cl)cncc2Cl)=O)CC)CC1 C(=O)(CCCC(=O)N(C1CCCCN(C(c2cc(C)oc2C)=O)C1)C)OCC Cc1nc(C(=O)NC2(C)CCN(C(=O)C=CCN3CCCC3)C2)ccc1C#N N1(C(c2cncc(OC)c2C)=O)CCC2CN(C(c3ccncc3O)=O)CC2C1 C(=O)(CC(C)(C)CC(C)=O)NCCCCCCCn1cc(C(CC)O)nn1 N1(C(C(C#C)(C)C)=O)CCN(C)C(C(=O)NCc2ccccc2C)C1 CC1(C(=O)NCC2(C)CCCN2C(=O)CCC[N+](=O)[O-])CCc2ccccc21 CCCC(C)(CC)N(c1nnnn1Cc1cn(C)nc1C1CCC1)CC C1(N(C(=O)CCn2ccnn2)CCC)CCN(C(=O)CN2CCC(C)C2)C1 c1(CN2CC(OC)C(C(=O)O)CC2)ccc(F)c(F)c1Cl N1(C(C(CNC(C)=O)(C)C)=O)CCC2(CCCC2CNC(C2CC23CC3)=O)CC1 C(C(C(=O)NCC(N1CCCCC1)C)C(C)(C)C)NC(C(c1ccc(C)o1)C)=O N1(C(C(=O)NC(=O)NC)C)CC2CN(C(=O)CC3C(C)(C)C3(C)C)CC2C1 CC(C)C(C)(CNC(=O)C=C1CCOCC1)NC(C1CC(Cl)(Cl)C1)=O C1(CNC(CCOCCCOC)=O)CCC(NC(=O)CCCC2CCOCC2)C1 N1(C(c2nncn2C)C(=O)NC(C(=O)OC)C)Cc2nccn2CC(CO)C1 c1(C(=O)NC(C(C)NC(c2cc(CC)nc(O)c2)=O)C)cnc2ccnn2c1C N1(C(c2c(C)ccnc2)=O)CCC2CN(C(=O)C(=O)NCC3CC3)C2C1 N1(C(c2ccc(CCC)cc2)C(=O)NC2CCCC2)CCOC2(CCCSC2)C1 CC1CN2CCN1CC=CC2=O.C1(CCC(=O)N(C)C)CC(C)(C)CO1 N1(C(c2cnns2)=O)CCN(c2ncnc3[nH]ccc23)CC(O)C1 c1(C(C)(O)C(=O)NC2CN(C(=O)C(O)C3CC3)C2)ccc(Cl)cc1 C(=O)(C(C)CC(C)C)NCc1occ(C(=O)Nc2c(OC)nn(C)c2)c1 Cc1cc(C)c(C(=O)NC(CNC(=O)Cn2ccc(C)n2)CC(C)C)cn1 c1(C(=O)NC2(C)CC(NC(C(C(C)C)c3cnc(C)s3)=O)C2)cc(N)cc(F)c1 C1(NC(C(C)SC)=O)C2CC3CN(C(=O)CCc4cnc(C5CC5)o4)C1C3C2 C(c1ccc(SC(F)F)cc1)=CC(=O)NC1CN(C(c2cc(C)sc2)=O)C(C)C1 CC(C)C(C)CC(=O)NCC1(C(=O)NOC2CC3CCC2C3)CC2(CC2)C1 C1(CC)Cc2c(Br)cccc2CN1CCC(=O)NCCOC C1(C(N2CCC(NC(c3ccc(Cl)cc3Cl)=O)(CO)C2)=O)Cc2cccnc2C1 C#CCC(CC(F)F)C(=O)NCC(CC)N(C(=O)Cn1nnnc1C(C)C)C N1(C(COCC=C)=O)CC(C)(C)OCC1CNC(=O)CC(F)(F)C(C)C N1(C(c2c(C)[nH]cc2)=O)CC2COCC(C1)N2C(c1ccc2cn(C)nc2c1)=O c1(C(N2CC(CNC(CC(CC)C)=O)C(F)(F)CC2)=O)cnc2n1CCCCC2 Cc1cccc(-c2nc(-c3nc(CS(C)=O)no3)cs2)c1C N1(C(CC2CC(C)C2)=O)CCN(C(=O)CCCN2CCCC2)CC1CCO N1(C(c2nc(C)nc(O)c2)=O)CC2C3CCC(C2C1)N(C(c1occc1C)=O)C3 C(=O)(C(C)Cc1cnc[nH]1)NCC1(CC(=O)NC(CN(CC)CC)C)CCC1 c1(CN(C(COC(C(C2CCCCC2)OC)=O)=O)C)cnc2ccccn12 c1(NC(C(c2cn(C)nn2)NC(=O)C(=O)C2CCCC2)=O)ccc2c(c1)OCC2 C1(NC(C(C2CCCC2)OCC)=O)CCCC2CN(C(C3COC(C)C3)=O)CC12 CC(C(=O)NC1CCN(C(=O)COC(F)(F)F)CC1O)C(F)(F)F C1(NC(C(CC)C(F)(F)F)=O)CN(C(=O)Cc2cnc[nH]2)CC2CCCC12 CCC(CC)(CO)C(=O)NC1CC(F)(CNC(=O)Cc2cc(F)ccc2F)C1 c1(-c2c(C(=O)NCc3cc(C)on3)ncs2)ccccc1C C1(C(=O)NCC(c2cnc[nH]2)C)CSCN1C(=O)Cn1cccc1 CCC(C(=O)NCc1ccon1)N(C)C(C1CC(C)(F)C1)=O c1(CCC)nc(C(=O)N(CC(=O)NCCCCCC2CC2)C(C)C)co1 C12CCN(C1)C2=O.c1(NCCNC(C(=O)NC)=O)ccn(C)n1 N1(C(CCc2ccc(C)nc2)=O)C2CCCC1CN(C(=O)C(C)C1CC(=O)C1)C2 CCC(C)(C)CCCC(=O)N(C)CC1CCC(NC(c2[nH]c(O)nc2C)=O)CC1 C1(O)(C(C)NC(c2cnn(CC)n2)=O)CCN(C(=O)CC2(O)CCCOC2)C1 C1(NC(CCc2cc(OC)no2)=O)CCCN(C(c2ccncc2)=O)C1C C1(NC(c2ccnn2CCF)=O)CCC2CN(C(C3CCCOC3)=O)CC2C1 N1(C(C=NOC)=O)CCCC2(CNC(c3cc(F)cc(Br)c3)=O)CCCC12 Cc1[nH]nc2c(C(=O)NC3CCCC3CNC(=O)CCCC(C)(C)C)cccc12 c1(C(N2CC(c3ccccc3)(NC(C3C(C)(C)COC3)=O)C2)=O)ccc(O)c(F)c1 C1(CC(=O)NC2CC(OCC(=O)N(C3CC(O)CC3O)C)C2)CCC(=O)NC1 Cc1ccc(Cc2nc(NC(=O)C(=O)NC(C34COC(C)(C3)C4)C)cs2)cc1 N1(C(C(C)(C)OCCC)=O)CC2CC(C(N3CC(C(N)=O)C4(CC4)C3)=O)CC2C1 Cc1cnc(C(N2C3CC2CN(C(c2cnnn2C)=O)C3)=O)cc1Cl Cc1cc(CON)cc(Cl)n1.C12CC(C)N(C1)c1n(nnn1)C1CCC(C1)OC2=O c1(C(=O)Nc2c(C)ccc(CO)c2)cn2c(n1)CN(c1ncncc1C#N)CC2 C(=O)(CCCCC(C)C)N1C2CN(C(CCCCCOCC)=O)CC1C2 c1(OC)cccc(I)c1C(=O)NCCNC(=O)CCC(C)C#N CCC(C)(C(N)=O)NC(C1CCCC(NC(=O)CCc2ncccn2)C1)=O C1(OC)CC(NC(c2ccc(C)cc2)=O)CN(C(=O)C(C(C)C)SC)C1 N1(C(C2(COC)CCCO2)=O)CC2(C1)CN(C(C1(COC)CCOC1)=O)C2 c1(CC)ccc(C=CC(c2ncc(I)cc2Br)=O)cc1 C1(C)(CC)CC(NC(=O)C(F)F)CN1C(=O)CCCCCc1ccccc1 CCCC(C)CC(=O)NC(C1(O)CCN(C(=O)C(c2ccccc2)C2CC2)C1)C c1(C(C)(C)CNC(=O)Nc2ccccc2)ccc([N+](=O)[O-])cc1 C(=O)(CC(C)(C)C(=O)NC1CCCCC1NC(C1CCCCS1)=O)OCC C1(C(=O)Nc2cn(CC(N3CCCC3)=O)nn2)CCc2ccccc2C1 c1(C(N2C(C)CC(CNC(=O)Cn3cncn3)C2)=O)cc(N)cc(F)c1 CCCCCC(F)C(=O)N1CCC(NC(c2c[nH]nc2CC)=O)C1 c1(C(=O)NC2CCCC(NC(C3CC(C)(C)C3)=O)C2)cc2scc(Cl)c2[nH]1 c1(C(C)C)ccc(C(=O)NC2(CC3NC(=O)CC3c3ccc(Cl)cc3)CC2)cc1F c1(CC(N2CCC(CCOC)(NC(C(CC#C)C)=O)C2)=O)cccc(C)c1C Cn1nc(O)cc1C(N1CCC(Cn2cc(Cn3cc(N)cn3)nn2)CC1)=O c1(C(N2CCC(NC(CCSCC(C)C)=O)C(F)C2)=O)ccc2nc[nH]c2c1 C1(NC(C(c2cccs2)SC)=O)CC(F)(F)CC1NC(c1cnccc1Cl)=O C12(C(N3CC(CCNC(CS(=O)(=O)N(C)C)=O)C3)=O)CCCCC1NC(=O)CC2 c1(C(N2CC3CC2CN3CCOc2cccc(Cl)c2)=O)cnn2c1CCCC2 c1(CC(N2CC(N(C(C(C)C3CCC3)=O)C)C2)=O)nn(C)cc1Br n1(CC)ccc(CC(=O)NC(CN(C)C)C(=O)NCC2(C3CC3)CCCO2)n1 C1(C(=O)NC2CC(CCC(=O)NCc3ccc(C)o3)C2)(CC)CCNC1=O N1(C(CCNS(CC)(=O)=O)=O)CCC(NC(c2cnn(CCO)c2)=O)CC1C c1(NCC23CC(C(=O)NC4COC(n5cccc5)C4)(C2)C3)ccc(OC)c(Cl)c1 Cn1nc(C(N2CCCC2(C)CNC(C2C3CCCC23)=O)=O)c2c1CCCC2 CN(C)S(=O)(=O)N(C)CC(=O)NC1CCCC1NC(c1cc(Cl)ccc1O)=O c1(CC(=O)NCC(C(C)C)NC(c2ccnn2C(C)C)=O)cnccc1C(F)(F)F c1(C(=O)NCC(c2ccccc2)CNC(C2CC(=C)C2)=O)sccc1Br C1(CNC(=O)CC(F)F)CC2CC2N1C(C1CC(=O)N(C2CC2)C1)=O C=C(Cl)C(C)(C)C(=O)NCC1(C)CCN(C(C2(CCCC)CCC2)=O)C1 c1(OC)ncccc1CC(=O)NC(C1CCCN1C(c1ccncc1Cl)=O)C N1(C(C(SC)SC)=O)CC2CCCC(N(C)C(C3CCS(=O)(=O)C3)=O)C2C1 C=CC(CCC)CC(=O)NCCOCCCN(C(=O)CC1CC=CC1)C c1(NC(C2(F)CCN(C(C(CCCC)O)=O)C2)=O)cc([N+](=O)[O-])ccc1Br C#CCCN=C(NCC12CCC(CC1)CC2)NC1CCN(S(C)(=O)=O)C1 C12(C(N3CC(CC)SCC3)=O)CC(C)(CN1C(=O)CCCC(C)C)C2 N1(C(c2c(CC=C)cccc2)=O)CCCN(C(c2c[nH]cc2CC)=O)CC1C Cc1conc1C(=O)NC1(CCCCNC(=O)Cn2ccc(Br)n2)CC1 N1(C(=O)NC(c2ccc(OC)c(C)c2)C)CCC(C2CC(F)(F)C2)C1 C(=O)(C(C)(O)CC(F)F)N(CCCNC(=O)COCC1CCC1)C N1(CCC)CC(C(N2CC(NC(c3nocc3C3CC3)=O)C(F)C2)=O)CC1=O N1(C(C2C(c3c(C)ccs3)C2)=O)CCC(NC(=O)C(C)N(C)C)C(O)C1 N1(C(C(CC(=C)C)C)=O)CCN(C(c2noc(CC)c2C)=O)CC(O)C1 C1(C(N(CCCCN(C(c2c(SC)n(C)nc2)=O)C)C)=O)CC(S(C)(=O)=O)C1 c1(C(N(c2c(C(=O)NC)cccc2)C)=O)cc(C2=CCS(=O)(=O)CC2)cs1 c1(C(=O)NCCC2CCC(NC(c3scc(C)c3)=O)C2)cc(C)cc2c[nH]nc12 N1(C(C(C)OCC#C)=O)CCCC(C(=O)NC(C)C)C1 c1(N(C)Cc2cc(C)no2)ncc(N)c2ccccc12 CC1(C)CCN(C(c2ccncc2)=O)CC1C(=O)NCC1(C)CCC(=O)N1 c1(-n2c(=O)c2=O)c(C)cccc1C.c1(SC)cccnc1.CO C1(C(N(CCC(=O)OCC)C)=O)C2CCN(C(=O)C(c3cncn3C)O)CC12 N1(C(Cn2c(C)nnn2)=O)CCC(CNC(c2ncccc2OCF)=O)C(C)C1 c1(NC(CC2CC3(CN(C(C(C)S)=O)C3)C2)=O)cc(Br)cc(Cl)c1O C(C(C)C)(C(F)(F)F)NC(C1(N(C(C(CCC)NC(C)=O)=O)C)CC1)=O c1(C(=O)NC(CN(C(c2nc(C)oc2C)=O)CC)C)c(C)oc(C)c1Br C1(F)(CNC(C2(C)CCCC2(F)F)=O)CCCN(C(C2COCCO2)=O)CC1 N1(C(C2(C)CCCOC2)=O)CCCCC(NC(=O)Cc2n[nH]c(=N)s2)C1 C1(C(=O)NCC2(OC)CCN(C(c3cn[nH]c3)=O)CC2)C2Cc3ccccc3C12 N12CCN(C(C3CC3)C1)CC2=O.c1(OC)ccccc1NCc1cn(C)nc1C C1(NC(c2cc(C)c(C)s2)=O)CN(C(c2cc(Cl)cnc2O)=O)CC2(CCC2)C1 C1(O)(CN(C(Cc2c(CC)con2)=O)C)CCN(C(c2ccc(CO)nc2)=O)C1 C(=O)(C1=CCC(NC(=O)C(C)(C)n2cnnn2)C1)NCCSCCOC C(C(C)(C)C(=O)N1CCCC(OC(F)F)C1)NC(=O)NC(CCC)COC C(N=c1[nH]c2c(c(=NC3CC4(CCCC4)C3)[nH]1)COCC2)C1(C)CCCO1 c1(NC(C2CCN(C(CN(CC)CC)=O)CC2(C)C)=O)ccc2c(c1)OCCC2 c1(OCC)sccc1C(=O)NC(C)CNC(c1ccc(Cc2ccccc2)s1)=O c1(NC(C2(S(N)(=O)=O)CC2)c2n(CCOCC)nnn2)ncccc1F c1(OC)ccc(C(=O)N(CCCN(c2ncncc2Br)C)C)cc1C#N c1(OC)ccc(I)cc1C(N1CC(NC(c2ccncc2O)=O)C(F)C1)=O c1(-n2cc(CCCNC(c3cc(CO)[nH]n3)=O)nn2)cnccc1Cl c1(C(=O)NCC=CCNC(C(CC)CC)=O)c[nH]c2nc(Br)ccc12 C(CC(O)CC(=O)NCC1(F)CC(CNC(c2ccccc2OC(F)F)=O)C1)SC C=C(Cl)CC(C(=O)NCc1[nH]nnc1C)NC(c1ccnc(O)c1F)=O C1(C(N2CC(COC)(CNC(C3CC(C)(O)C3)=O)C2)=O)CCS(=O)(=O)CC1 CC(CCCc1ccccc1)C(=O)NCCCNC(C1CC1OC(C)(C)C)=O CCC(C(=O)NC(C1CN(C(=O)C(C)n2cncn2)C1)C)OC1CCCCC1 c1(C(N(C(C)C)CCNC(C2(Cl)CC2(C)C)=O)=O)ccc(C(F)(F)F)cn1 c1(CC)ccc(Cl)c(C(=O)NC2CC(F)CN(C(=O)Cc3ccoc3)C2)c1 c1(COC)nc(NCCN2CCS(=O)(=O)CC2)cc(=NCC(C)N(C)C)[nH]1 C1(OC)(CNC(=O)C(F)C2CCC2)CN(C(C2CCCN2C2CC2)=O)C1 C1(NC(C2CN(C(N)=O)C2)=O)CCOCC1NC(=O)Cc1cc[nH]c1 c1(C(=O)NCC(CN(C)C(C2C(F)(F)C23CC3)=O)O)cc(F)cc2nc[nH]c12 C1(C(=O)NC(Cc2ccccc2)CCCO)C2Cc3c(Cl)cccc3C12 c1(CNC(CC2OCCN(C(c3cnc(C(C)C)o3)=O)C2)=O)cccc(F)c1F c1(C(=O)NCC2C(NC(c3c(C(C)C)onc3)=O)CCC2)cccc(F)c1 C1(C(=O)NCC(CNC(c2ccc(CC)o2)=O)(C)O)CNC(=O)C(C)(C)C1 N1(C(CCC=C)=O)CCC2CN(C(=O)CCc3nccn3C)CC12 c1(C(N2CCN(C(CC(CCC)C)=O)CC2COC)=O)c(F)ccc(Cl)c1F C(=O)(C(CNC(=O)CCc1cnn[nH]1)Cc1ccoc1)N1C(CC)CCC1 c1(NC(C2CC(C(=O)OCCSC)C2)=O)cc(C(F)(F)F)ccc1OC(F)F C1(C(N2CC(CC(CNC(C3C(C(C)C)C3)=O)(C)C)C2)=O)(N(C)C)CCCSC1 c1(NCC(=O)NCCN(C(=O)CC2(O)CCC2)CC)ccccn1 CN1CCc2cc(C(=O)N(C3CCC(NC(=O)CS(=O)(=O)C4CC4)C3)C)ccc21 N1(C(Cc2ccc(NC(C)=O)cc2)=O)CC(F)(F)CC1C(N1CC(=O)NC(C)C1)=O N#Cc1ccccc1C(=O)NCC1CCCN1C(=O)CCc1ccc(F)cc1 CCC(F)(F)C(=O)N1CC(CNC(c2ccncc2C(F)F)=O)(OC)C1 N1(C(C(C)OCC#C)=O)CCC(C)(C)C1CC(=O)NCC(C)(O)CO N1(C(C23CCCC2C3)=O)CC2(CCN(NC(c3[nH]cc(CC)c3)=O)CC2)C1 C1(C(=O)NCC(C)CNC(=O)C(c2ccccc2F)(F)F)Cc2nnsc2S1 C(=O)(C(C)(C)OC1CN(C(CCC)=O)C1)NC(C1(CNC(=O)NC)CC1)C CC(C)(C)C(CNC(c1c[nH]c(Br)c1)=O)NC(C1(C)CC2CC2C1)=O C1(C(=O)NCC2CC(OCC)C2)CN(C(c2coc(C(N)=O)c2)=O)CC(C)(C)C1 C1(N(C(C(C(C)C)(C)O)=O)C2C(C)C2C)CCC2CN(CCC(C)CC)CCC2C1 C(=O)(C(C(C)CC)N(C)C)NC1(C)CN(C(COCC(=O)OCC)=O)C1 C(N=c1cc(C)nc(-c2ccccn2)[nH]1)C1CCN(C(C(CC)C)=O)C1 C1(CC(=O)NCCCOCCNC(CN(C(=O)OCC)C)=O)C=NN(C)C1=O C1(C(N2CCCC(C(C)C(=O)NCc3ccc(N)cc3)C2)=O)CCCC(C)(C)C1 Cc1cc(C(=O)N2CC(n3cc(COc4ccc(Br)cc4)nn3)CO2)cc(F)c1 Cc1ccc(CNC(C2CCN(C(c3nn(C)c(C)c3Br)=O)CC2O)=O)c(F)c1 N1(C(C=CC(C)C)=O)C(C(=O)Nc2cnc(Br)cn2)CCC1C C12(CNC(CC(=O)N(C)C)=O)CC(NC(c3cc(F)c[nH]3)=O)(C1)C(C)(C)O2 C(=O)(CC(C)CC(C)C)N1C(CC(=O)NCC2(OC)CC2)CCCC1 N1(C(c2c(-c3ccc(OC)nc3C(F)(F)F)ncs2)=O)CCc2n[nH]cc2C1 CC(C)(C)C(C#N)C(=O)NC1(CNC(=O)C=Cc2cccc(Cl)c2)CCCCC1 N1(C(c2nc(OCC)sn2)=O)CCCCC1C(C)NC(c1cc(Cl)c(Cl)[nH]1)=O C1(C2(O)CCN(C(C34CCCCC3CCC4)=O)CC2)(NC(C2CCC2)=O)CC1 c1(OC)cccc(Cl)c1C(=O)Nc1ccsc1C(=O)Nc1ccc(C)nc1 C1(N(C(=O)CCSc2ccccn2)C)CCCCN(C(C2CCC2C#N)=O)C1 c1(C(=O)NC2CC(NC(c3n[nH]c(CC)c3Cl)=O)C2)c(OC)ccn2ccnc12 c1(C(N2CCN(C(C(CCC)NC(N)=O)=O)C(CC)C2)=O)c(F)cc(N)cc1F c1(-c2ccc(-c3n(CC(C(C)C)(C)O)ccn3)s2)cc(F)cc(Cl)c1 C1(NC(C(C)=C2CC2)=O)CN(C(=O)CCC2CCC2)C2(CCCOC2)C1 C1(CNC(C=C(C)C(F)F)=O)CCCCCN1C(=O)CC1COC(C)(C)C1 c1(OC(C)C(=O)NC2CCCC2NC(=O)C(C)CF)cccc(Cl)c1 C1(O)(C(=O)NC(C)C(N)=O)CCN(CCNc2ncccn2)CC1 C(=O)(C(S(C)(=O)=O)C1CC1)NC(CNC(C(C)C1CCC1)=O)C1CC1 CCC(CCC(=O)N1CCCC(F)C1)NC(C1CC2(CC2)CO1)=O C1(C)(C(N2CC(N(C)C(C3CC(F)C3)=O)C2)=O)C=CCC1 N1(C(COCCC=C)=O)CCN(C(=O)Cc2ccsn2)C2CCCC12 N1(C(CC)=O)CC(Nc2nc(OC)cc(OC)n2)C2(CCOCC2)C1 C1(NC(C2CCS(=O)CC2)=O)CCCN(C(C2CC(OC(F)(F)F)C2)=O)CC1 N1(C(C(C)NS(CCC)(=O)=O)=O)CCC(NC(c2cc(=O)cc[nH]2)=O)C12CC2 CC(C)C(C)(O)C(=O)N(C)CC1CCCN(C(=O)C2=CCCOC2)C1 c1(C(=O)NCC(C)(O)CNC(=O)COc2ccsn2)cnc2ccccn12 CC1(C)COCC1CNC(=O)CC1(NC(C2CC=CC(O)C2)=O)CCC1 c1(NC(c2n(CCOC)nnn2)C2CCCSC2)cc(-c2ccccc2)n(C)n1 c1(-c2c(C(N(CCCN(C(CN(C(C)C)C)=O)C)C)=O)c[nH]c2)ccccc1F C1(C(N2CC3(CCN(C(Cc4nc(C)sc4)=O)C3)C2)=O)CC2CS(=O)(=O)CC2C1 C1(CNC(CCC(CC)OC)=O)CC12CCN(C(C1(C(N)=O)CCC1)=O)CC2 c1(OC)cnc(C(=O)NCC2CCCN(C(C3CC4CCC3C4)=O)C2)nc1 c1(C(=O)NCC2C(CNC(C3CCC(C)(F)CC3)=O)C2)noc2ccc(Cl)cc12 C(CCCCC(=O)NC1CCC(CO)C1)N(C(C1ON=C(C)C1)=O)C c1(CC(N2CCC(NC(c3cc(CO)[nH]n3)=O)C(O)C2)=O)nc2c([nH]1)CCCC2 Cc1nsc2ncc(C(=O)NC3CCCC3CNC(c3ccncc3O)=O)cc12 CC1(C)C2CC1CN(C(=O)COC1CN(C(C3CC(C)(O)C3)=O)C1)C2 c1(SC)c(C(=O)N(CCNC(=O)CCCN(C)C)CC2CC2)cccc1F c1(C(=O)NC(C)C(C)NC(=O)C(c2cccc(Cl)c2F)(C)C)cc(O)cc(O)n1 CCCC(C(O)C(=O)N1CC1CC(=O)OC)NC(=O)C=CC(N1CCCCC1)C c1(C(=O)NC2C(C(N3C(C)CN(C)CC3)=O)CCC2)c(Br)ccc(F)c1F Cc1oc2nc(Cl)ccc2c1C(=O)N(CC(O)CNC(C1OCCO1)=O)C C(=O)(C1=CC2CCCCC12)NC1(C)CC(NC(c2ccc([N+](=O)[O-])c(O)c2)=O)C1 c1(C(N2CCC(CNC(CC3(C)CC3)=O)C2)=O)ccc(Cl)c2occc12 c1(CCC(=O)N(C)CCOCCCN(C)C(c2ccns2)=O)cccc(O)c1 CON(CCC(=O)NCC1CC12CCOCC2)C(=O)C1(C)CC(C)(C)C1 O=C(N=c1cc(C(=O)NC2(c3ncccn3)CCC2)[nH][nH]1)c1cc(F)ccc1F c1(C(N2CCC(N(C(c3c(CCC)nns3)=O)C)CC2)=O)c(C)cc(Cl)cc1N C1(CC(C)NC(c2cc(C)sc2)=O)CCN(C(=O)CC(C)O)CC1 N1(C(CCNC(CC2CCC(C)C2)=O)=O)CCNC(=O)CC1 Cc1ccc(C(=O)C(=O)NCC(C)NC(=O)CCC2CCCO2)cc1 C1(C(N2CCN(C(=O)NC)CC2)=O)COCCN(C(=O)CCc2cccn2C)C1 c1(C(=O)NC2CCC(CNC(C=C3CCN(C)C3)=O)C2)cnccc1Cl C1(C)(CC)C=C(C(=O)NCC(=O)NCC(=O)NC(Cc2ccco2)CO)C1 CCCC(CC)CCC(=O)N1CCCCC1CCNC(=O)CCN1CCCC1=O Cc1cc(F)c(C(N2CCC3C(C2)CN3C(=O)Cc2cc[nH]n2)=O)cc1Br c1(CC)occ(C)c1C(=O)NCC1(C(F)F)CCN(C(C2CCOC2CC)=O)C1 C1(C(=O)NCC(C)N(C)C(c2nc(C3CC3)cs2)=O)(OC(C)C)CCOC1 c1(OC)ccc(NC(=O)OC(C)(C)C)cc1SC.n12cc(nn1)CC(=O)N2 c1(C(=O)NCC=CCNC(CCCCSC)=O)nc2c(Br)cccn2n1 c1(C(N2CC(F)(CNC(=O)CC(C3CC3)C3CC3)C2)=O)cc2c(nn1)CCOC2 C(=O)(C1=CCCCCC1)N1CC(CNC(C(C(CC)C)O)=O)N(C)CC1 C12(C(=O)NC(C)C3CC3)COCC1CN(C(=O)Cc1ccccc1Br)C2 c1(OC)cncc(C=CC(=O)NC2C=CCN(C(c3ccoc3Br)=O)C2)c1 c1(OCC(C)C)ccccc1C(=O)NCCC1(O)CCN(C(=O)CC(C)(F)F)C1 C12=CC=C(C=C1)C2.c1(C(C(=O)NC)N(CCF)C2CC2)c[nH]nc1C c1(C(=O)NCC(CC(C)C)NC(c2c(Cl)cnn2C)=O)ncc(C(N)=O)cc1Cl N1(C(CC(CCC)NC(c2c(CO)n[nH]c2C)=O)=O)CCN(C)C(C)(C)C1 c1(C(=O)NCC(CC=C)NC(C23CCN(CC2)CC3)=O)cc(C#N)ccc1O N1(C(CC(CC)C2CCC2)=O)CC2CCC1C2NC(c1ccc(OC)cc1N)=O C1(CC(=O)NCC(CNC(C(CCOC)C)=O)(C)OC)CCC(C)(C)CO1 C(CC(C)P(C)(C)=O)NC(C(=O)Nc1ccc(CCCCC)cc1)=O N1(C(C2(CC=C)CCN(C(c3cc(CC)no3)=O)C2)=O)CCC2(CC(OC)C2)C1 n1(CCC)nccc1C(=O)NCC1(NC(=O)CC2CC2(Cl)Cl)CCOC1 CC1(C(=O)NCc2cn(C3CN(C(C4CC(O)C4)=O)C3)nn2)CC2CCC1O2 CN1C(=O)CCCC1C(N1CCOCC1CNC(C12CC(CO1)C2)=O)=O C=CCC(C)C(=O)N1CC(CC=C)(NC(=O)CCCn2ccccc2=O)C1 c1(C(N2C3CC(CN(C(C(C(C)O)N(C)C)=O)C3)C2)=O)cn(C)c(=O)n(C)c1=O C(=O)(C1CCCc2n[nH]cc21)N1CC(F)CC(NC(c2c(C)ccc(C)n2)=O)C1 n1(CCC)nnnc1C(C1CCCCC1)NCC1(CCC)CCC1 C1(C(=O)NCC2C(C(N(C3CCN(C)C3)CC)=O)CCO2)CCN(C)C(=O)C1 c1(C(=O)NCC2(CNC(c3snc(O)c3Cl)=O)CCC2)cn2cccc(F)c2n1 c1(OC)cccc(OC)c1CC(=O)NCC1C=CCN1C(C1CC1c1cnc[nH]1)=O c1(OC)ccc(S(N)(=O)=O)cc1C(N1CCC(C)C1CNC(=O)CC1(O)CC1)=O C(CO)(C(=O)N1CC2COCC2O1)NC(c1c(OC)cncn1)=O CC1CN(C(C2(O)CCOCC2)=O)CCC1C(=O)N(C)OC1CCCC1 N1(C(C2(C)CCCN(C)C2)=O)CC2CC(NC(C3CCC4CC3CO4)=O)CC1C2 C(=O)(C1=CC2CCCC12)NCC1CC(NC(c2cccc(OCC)c2O)=O)C1 C(N=c1[nH]c(N2CCc3ccnc(N(C)C)c3C2)nc2c1CSC2)c1c(C)scn1 C(=O)(CCCCCNC(N)=O)NCCC1CCN(C(Cc2nc(=N)[nH][nH]2)=O)CC1 c1(OC)ncccc1C(=O)NCCC(Cc1ccccc1)NC(=O)C1=CCCS1 N1(C(c2c(OC)cc(C)s2)=O)CC2(CCCCN2C(c2cc(C)c(C)nn2)=O)C1 C1(NC(C2(OCC)CCOC2)=O)C2CN(C(=O)CCCCC3CC3)CC12 C(=O)(C(C)C(=O)N(C)CC1CCCN1C(c1ncc(F)cn1)=O)OC Cc1cnn(CC(=O)NC2CCC(N(C)C(c3ocnc3C3CC3)=O)C2)c1 c1(OC)ccc(O)c(C(=O)NCC(N2CCN(C(c3ccco3)=O)CC2)C)c1 C(C(CO)N=c1nc[nH]n2c(Br)ccc12)NC(=O)C=C1CCC1 C(=O)(C(F)CC(CC)CC)N1CCC(CNC(CCC=C)=O)(CO)CC1 c1(C2(C(=O)NCC(CNC(c3cc(C4CC4)on3)=O)OC)CCC2)ccc(C)cc1 c1(C(=O)Nc2ccnc(-c3ccccc3)n2)nc(Cl)ccc1Br c1(C(=O)NCC(CNC(C2CCS(=O)(=O)CC2)=O)OC)nn(C)c(N)c1C Cc1c2c(-c3cnc(F)c(C(=O)NCC(N4CCCC4)=O)c3)cccc2nn1C c1(C(=O)NCC2CC(NC(C(CC=C)C)=O)C2)cc(O)nc(CC)n1 CCS(=O)(=O)CC(=O)N1CCC(C2CCCN2C(=O)C=C2CCC2)C1 CN1CCCC1C=CC(=O)NCC(C)(C)NC(C1C=CCCC1)=O N1(C(C2CC2C(F)F)=O)CCN(C(c2snc3ccccc23)=O)C2(CCC2)C1 C1(C(N2CCCCC2)C(C2CCCCC2)=O)CC12CCC2 N1(C(CCCC(=O)NC)=O)CCC(F)(F)C(CNC(C2CCN2C(C)(C)C)=O)C1 c1(C(=O)OC)cc(C(=O)O)cc(S(=O)(=O)NC2(CC(F)F)CC2)c1 c1(OC)ccc(C(=O)NC(C2(O)CN(C(=O)C=CCN3CCC3)C2)(C)C)cc1 Cc1occc1C(=O)NCC1CCN1C(=O)C(C)c1cc[nH]n1 C1(NC(C(CC)NC(C)=O)=O)CC2CCC1(C(=O)NCCCCCCCO)C2 c1(C(N2C(CNC(c3cccnc3O)=O)COCC2)=O)ccc2c(c1)CCCO2 N1(C(=O)NC2COC(C(F)F)C2)CCCc2ncccc21 C1(C)(C(N2CC(NC(c3cc(C)ncn3)=O)C3(C2)CC3)=O)CCCCNC1=O C1(NC(CC=C)=O)CN(C(c2cc(N(C)C)nc(Cl)c2)=O)CCC1O C1(NC(C2C(c3c(C)occ3)C2)=O)CCN(C(c2ccc(C3CC3)cc2)=O)C1C C1(CNC(c2cc(C)[nH]n2)=O)CCCCN1C(=O)CCC1(C)CCC(=O)N1 c1(N2CC(OC)(CNC(c3c(C)ncn3C)=O)C2)c(C)cncc1[N+](=O)[O-] C=CCC(CC(=O)N1CCOCC1CCO)NC(=O)Cc1cccc(O)c1 CCC(C)(CO)C(=O)N1CCCC(CCNC(=O)Cc2cnc[nH]2)CC1 C1(CC)CCN(C(c2cnccc2C)=O)C(C(=O)NC(C)CN=[N+]=[N-])C1 Cc1ccc(NC(=O)CS(=O)Cc2ccc(Cl)cc2C#N)c(Cl)c1O C(CC(=O)NC1CCC(NC(=O)C2=CS(=O)CCC2)C1)(C(F)(F)F)OC C(=O)(C(C)=Cn1ccnn1)NCC12CN(C(C(C(C=C)C)C)=O)C(CC1)CC2 c1(C(=O)NCC2C(NC(c3cc(-c4ccncc4)on3)=O)C2)ncccc1F C(=O)(C(C)C(C)NC(c1sc(F)cc1C)=O)NC(C1CCCCC1)CC C(CN=C(NCC(N1CCOCC1)=O)N1CC2C(CF)C2C1)N1C(=O)NCCC1 CCC(CCOC)C(=O)NC(C)(CNC(=O)Cc1cc(C)nn1C)C(C)C C(CC)(CS(=O)(=O)c1ccccc1)Cc1[nH]c(=NC(C)C(C)C)cc(CC)n1.N C1(C(=O)NCCC(C)NC(=O)C(C)(O)C2CC2)COC(=O)N1C c1(C(N(C2CCN(C(c3ccc(C#C)cc3)=O)C2)C)=O)cccc(F)c1C#N N1(C(C2CC(C)OC2)=O)CCC(C(O)CNC(=O)CCCN(C)C)CC1 N1(C(CN(C(=O)OCC=C)C(c2cn(CC3CC3)nn2)C)=O)CCS(=O)(=O)CC1 c1(NC(=O)CSc2cc(F)c(C(=O)O)c(F)c2)ccc2c(c1)OC(F)(F)O2 c1(CC)cc(OC)cc(C(N2CCC2CNC(c2cc([N+](=O)[O-])c[nH]2)=O)=O)c1 n1(CC(=O)N(CC(=O)N(CCCC=C)C)CCC)cccnc1=O CC1(C)CC(NC(=O)COc2cnn(C(C)(C)C)c2)CN1C(=O)CCF N1(C(Cc2c(C)cccc2C)=O)CCN(C(=O)C2=CC(C)C2)C(C)C1C c1(CNC(c2cc(C)[nH]n2)=O)cc(C(=O)NC2(C)CCSCC2)n(C)n1 c1(C(=O)NC2C(CNC(c3ccccc3)=O)CCCC2)[nH]nc2ncnc(O)c12 c1(CC(=O)NCCCCNC(C2N(CCC)C(=O)CC2)=O)cnn2c1CCCC2 C1(C(=O)NC(C(=O)NCCOC(CC)(C)C)(C)C)CC12CCOC2 c1(CCC)cc(C(=O)NCC2COCCN2C(=O)Cc2ccccc2C)ccn1 c12cnc(nc1)o2.C1(C(=O)NCC)CCCN(C(=O)C(C)=CC)C1 Cc1cc(C(=O)NCC2C(C)CCN2C(=O)COc2ccccc2Cl)c(C)cn1 c1(CC(N2CC3C(NC(c4c(C)nsc4)=O)C(C3)C2)=O)c(C)oc2ccccc12 C(=O)(NN=c1[nH][nH]c(=Nc2ccccc2Cl)s1)c1ccc(C(N)=O)nc1 C#CC1(O)CCCN(C(=O)CC2CCN2C(C2CC(OC(C)=O)C2)=O)C1 CCCC(C(=O)OC)C(=O)N1CC=CC1C(=O)NOCCCCC1CC1 c1(OC)ccc2cc(C(=O)NC(C)CN(C)C(C3CCSC3)=O)[nH]c2c1 c1(OCCN(C)C)c(C(N2CCCC(C3CC(N)CCO3)C2)=O)cccc1N c1(C(=O)NCC(C)(CNC(C2CCCN2C2CC2)=O)OC)ncc(C)cn1 c1(C(N2C(CCNC(C3OCC(C)(C)C3)=O)COCC2)=O)cnc2ccccn12 C1(CCN2CC(O)CC(OC)C2)Sc2ccccc2NC1=O N1(C(c2n(C=C)ncc2)=O)CCN(C(=O)C2=C(Cl)CCOC2)CC2(C)CCCC12 c1(C(CNC(C=C(CSC[SH]=C)C)=O)NC(=O)CC2CSC2)ccc(OC)cc1 C(C(C)CC(=O)NCC1(C)CC1(C)C)NC(c1ccn(CCC)n1)=O c1(-n2c(C)ncc2)ccnc(C(=O)NCC2(CNC(c3cn(C)nn3)=O)CC2)c1 C1(NC(Cc2c(OC)cccc2)=O)CN(C(C2COCCN2C)=O)CCC1O Cc1nc(C(C)(C)C)sc1C(=O)NCC(O)CN(C(=O)CCCN(C)C)C C(N=c1nc(O)c2ccccc2[nH]1)C12CCC(NC(c3cnns3)=O)(CC1)CO2 CS(=O)CCC(=O)N1CC2CC2(NC(=O)Cc2ccsn2)C1 C1(C(N(C)Cc2nncn2C)=O)(NC(=O)C=CC2CCCN2C)CCC(C)(C)C1 c1(C(=O)NCC23C(CN(C(C4N(C)C(=O)CCC4)=O)C2)C3)ccc([N+](=O)[O-])cc1 FC1CCCCCC1N=c1[nH]c(N2CCN(c3nc[nH]n3)CC2)nc2cc[nH]c12 N1(C(C2(C#C)CCC2)=O)CCC(N(C(=O)CSC2CCCC2)C)C(C)C1 C1(CCC(=O)NCC2C(NC(c3n(C)ncc3)=O)CCC2)CCCC(O)C1 C=CCC(C(=O)NCCC1CCN(C(c2c(NC)c[nH]c2C)=O)C1)NC(C)=O N1(C(c2c(C)nn(C3CC3)c2)=O)CCCC(NC(=O)CC2CCOCC2)C(F)C1 CC1COc2c(C(=O)NC3CCCCC3CNC(=O)CS(C)(=O)=O)cccc21 C1(CCC)CCN(C(C2(NC(=O)C(C)COC(C)=O)CC(O)C2)=O)C1 Cc1ccc2c(c1)CC(C(=O)NC1CN(C(c3ccc(=N)[nH]n3)=O)CCC1F)S2 C1(NC(=O)COCc2ccccc2)CCCC(CNC(CCCOCC)=O)C1.O c1(SC)nc(Cl)cc(=NC2CCCC(NC(c3cc(N(C)C)ccc3F)=O)C2)[nH]1 C1(=CCNC(CCn2ccc(C)n2)=O)CCN(C(C2(C#N)CC2C)=O)CC1 N1(CC(=O)N(C)C)CCC2CC(C(N3CC(C(=O)O)OC(C)(C)C3)=O)C2C1 CC(C)CC(C(=O)NCC(C)(C)OCCO)ONC(C1CCCCC1)=O CC1(C)CC(CC(=O)Nc2cccc(CNC(c3ccsc3)=O)c2)CCO1 C1(CNC(c2ccc(C(F)F)cc2)=O)C2CC1N(C(=O)CCN1CCCC1=O)C2 c1(CC(CCC(C2CCCOC2)F)CO)ccc(Cl)cc1.N c1(NC(C2CN(C(c3noc(C)c3C)=O)CC(F)C2)=O)cc(C#N)c(F)cc1Br C1(CC)CN(C(=O)CC2(C)CC2)CC1NC(C1(c2ccc(OC)cc2)CCC1)=O CC1(F)CC2(CN(c3cc(NC(c4cccc(Br)c4)C(N)=O)ncn3)C2)C1 C(CC)(CCCC(=O)NCc1cc(C)cnc1F)NC(C1(CC=C)CC1)=O C1(CNC(C(P(C)(C)=O)O)=O)CC12CCN(C(c1ccn(C(F)(F)F)n1)=O)CC2 c1(OC)c(C(=O)NCC2CCN2C(c2cc(C(C)(C)C)n(C)n2)=O)cccc1Cl CC1=C(C(=O)NCc2cc(C(=O)NCC(c3ccccn3)O)on2)SCCO1 c1(OC)nc(=NC(=O)C2=NOC3(CCN(CC4CC4(F)F)CC3)C2)nc(OC)[nH]1 C12=C(Cl)N=CNC1=NCC1(CC1)CC2.C(=O)(C(N)=O)OC c1(C(=O)NCC2CC(NC(=O)C(O)CCc3ccccc3)C2)cc(O)nc(O)c1 C1(C)(C(N2CC(F)(CNC(Cc3cc(C)sc3)=O)C2)=O)CCC(=O)C1 c1(C(N2C(C(CC)O)CCCC2)=O)sc2ccccc2c1Cl C#CCCC(C(=O)N1CCC(C(N)=O)CC1)NC(=O)CCC1CCC(=O)C1 c1(C(N(C(C)C)CCNC(C2CCC2(F)F)=O)=O)cnc(CC2CC2)nc1O c1(C(N2C3CCC(NC(c4c(C)nsc4)=O)C(C3)C2)=O)cccc(P(C)(C)=O)c1 c1(C(=O)NCC2(CN(C(=O)CC3CSC3)C)CC2)cc[nH]c2nccc1-2 CC(CC(=O)c1ccccc1F)C(=O)NC(Cc1ccccc1)CO CN1CCC(C#N)(C(=O)NC2CCCCC2CNC(=O)C2=C(Cl)CC2)CC1 c1(C(N2CCC(CNC(c3cnn(C4CC4)c3)=O)C2)=O)cccc(F)c1C(F)F N#CC12C3C4C1C1C2C3C41C(=O)NCC(C1CCC1)NC(=O)CCNS(C)(=O)=O N1(C2CCN(C(C(C)C)=O)C2)CCC(NC(C2(c3nccn3C)CC2)=O)CC1 C=CCCC(C)(C)C(=O)N1CC(CCCCNC(=O)C#CC(=O)N(C)C)C1 N1(C(=O)CCNS(=O)(=O)c2cccc(Br)c2)CCc2c(O)ccc(F)c2C1 C1(C(=O)NCC(C)NC(c2cnc(C3CC3)[nH]2)=O)CCCC2C1C2(F)F CCC(CC(=O)NCC(Cc1ccccc1)NC(C)=O)SC C(=O)(C1=C(Cl)CCOC1)N(C(C)CNC(C1(COCC)CCCCO1)=O)CC CC1=C(C(=O)NC2(CO)CN(C(=O)C(C)(O)C(C)C)C2)CCC(C)(C)C1 Cc1c(C(=O)NC2COCCN(C(=O)C(C)n3ccnc3)C2)sc2nnc(S)n12 C(c1cnn(C)c1C)=CC(=O)N(CCOCCNC(C(n1ccc(C)n1)C)=O)C N1(C(CCN2C(=O)COCC2)=O)CC2(CNC(=O)C(=O)NCC(F)F)CC1CO2 C(CCC(C)(F)F)N(C)C(C1CN(C(=O)Cc2cccnc2O)CCO1)=O C(=O)(C(C)(C)CCF)NCC(C)CC(N1CC2CC2C2CC12)=O S(=O)(=O)(c1cccc(NCc2nc(C#N)cs2)n1)N(CCF)CC C1(C)(C(=O)NC(C)CCN(C(=O)C(C)CF)C)Cc2ccccc2C1 N1(C(c2c(CC)n(C)nc2)=O)CCC2(CC2NC(=O)CCc2cncnc2O)C1 C(=O)(C(C)CCC(C)(C)C)NC(CN(C(c1cc(N(C)C)nc(Cl)c1)=O)CC)C C1(NC(c2cc(C)ncn2)=O)COCCN(C(=O)CCc2ccc(F)cc2Cl)C1 c1(CCC(=O)NCCCN(C(=O)C(Cl)=CCl)C)nc2ccccc2s1 n1(CCN(C)C)cc(C(=O)NC2(CNC(C3CC(CCO)C3)=O)CC2)nn1 N1(C(=O)C2=COCCO2)CC23CCCC2(C1)CN(C(c1occ2c1CCC2)=O)C3 CC1(NC(C2CCCC2N2CCOCC2)=O)CCCN(C(c2cccnc2)=O)C1 CCCCC(O)C(=O)NC1(CC)CCCN(C(c2scc(C)c2Br)=O)C1 CCCCC(CC)NC(C1C=CCCN1C(c1ccccc1OC)=O)=O C1(NC(C(C)(C)C2(O)CCOC2)=O)COCCN(C(=O)CCc2cccs2)C1 C1(CNC(c2[nH]cc(C)c2)=O)COCCN(C(=O)C(C(C)O)N(C)C)C1 C(=O)(CCCC(C)(C)C)N1C(C(=O)NCCOCCOC)C=CCC1 C1(NC(C=CCN(C)CC)=O)CC2CC1N(C(C1(COC)CCC1)=O)C2 c1(NC(C2(NC(C(C)=C(CC)C)=O)CCCC2C)=O)cc(F)ccc1OC C#Cc1cncc(C(=O)N(C2(C(=O)NOCC=CCl)CC2)C)c1 S(=O)(=O)(c1cccc(F)c1C)N1CC2CCN(Cc3ccc(OC)cc3O)C2C1 c1(C(N2C(c3c(C)noc3C)CCC2)=O)cc(Br)cc(=N)[nH]1 N#Cc1ccc(C(=O)NCC2CC(NC(C3CC4CCC4C3)=O)C(O)C2)cc1 C(=O)(CC1NC(=O)c2ccccc21)N1C(C)CCN(C(COC)=O)CC1 C1(C(C)C)CCC(CC(=O)NCCNC(c2cc(C3CC3)[nH]n2)=O)CC1 c1(C(=O)NCC2CCC(NC(Cc3c(C)cnn3C)=O)C2)ccn(C)c(=O)c1 C1(CC(=O)NCC(C(=O)NC)O)N(C(=O)C=CC(F)(F)F)CCC1(C)C C1(C(=O)OC)(N(C(=O)C(F)=C(C)C)C)CCC1 c1(CN(C(=O)C(c2cccc(Br)c2)CN)C)ccccc1OC(F)(F)F N1(C(c2c(C)cc(C)n2C)=O)CCC2(CC1)CC2c1cn(CC2C3CCCC23)nn1 c1(C(C(=O)NC(C)CC)N(CCOCC)CC)cc(C)cc2c1CCC2 C1(NC(C(c2cn(C)nc2)=O)=O)CN(C(=O)CSC2CC2)CC1F c1(CC(=O)NC2CC(NC(C(CC)(C)C)=O)C2)c[nH]c2cccc(Cl)c12 Cn1ccc(C(N2CC3CC3(CNC(=O)CCOC3CCCOC3)C2)=O)cc1=O c1(CC(=O)NC2CN(C(C3(CC=C)CC3)=O)CC3C2C3)cccc([N+](=O)[O-])c1C N1(C(Cc2sc(C)c(C(C)C)n2)=O)CCC(C)(NC(=O)CCS(C)=O)CC1 CC(C)(O)CC(=O)NC1CCOC(CNC(c2cn(CC(F)(F)F)cn2)=O)C1 C#CCC(CC(F)F)NC(c1coc(CNC(=O)C2=NOC(C)C2)c1)=O c1(C(=O)NCC2CC(F)(CNC(C3CC3F)=O)C2)ccc2ccoc2c1 Cc1ccc(C(CNC(=O)Cc2cc(C)on2)NC(=O)Cn2ccc(C)n2)cc1 CC(C)C(C(C)NC(=O)Cc1csc(C2CC2)n1)NC(c1cocn1)=O CC(CS(C)(=O)=O)N=c1[nH]c(N2CCOC3(CCC3)CC2)nc2c1CCCC2 C1(CNC(C2(OC)CCOCC2)=O)CC2CCCC2N1C(=O)CC1COCCO1 N1(C(C(C)=CC)=O)CCC2C1CCCN2C(=O)COCCCC(C)C C1(NC(CC2C(C)C2(F)F)=O)CCC2CCN(C(c3ccc(N(C)C)nc3)=O)C12 N1(C(Cc2cnc(C)o2)=O)CC(NC(=O)CSc2nncn2C)CCC1C C1(C(N(C2CCN(C(C=CCOC)=O)CC2)C)=O)CC(COC)C12CCC2 N1(CC)CCN(C(C2CN(C(C3CC3CCOC)=O)CC(C)O2)=O)CC1C Cn1c(C(=O)NC2CN(C(C3CC3(C)C(F)F)=O)C2)ccc1-c1ccccc1F N1(C(Cc2cn(CC)nn2)=O)CCC(C)C1CNC(c1ccc(C)n1C)=O C1(NC(c2n[nH]cc2C2CC2)=O)CN(C(c2cc(F)c[nH]2)=O)CCC1CO C1(C(N2CCC(C(=O)NCC(F)F)CC2)=O)CCC(=O)N2CCOCC12 c1(SC(C)C(N2CCN(C(=O)CCC#N)CC2)=O)ccccc1Br CC1CCN(C(=O)CCC(C)(C)NC(=O)CSC2CC2)CC(C)O1 CC1OCCOC1C(N1CCOC(CN(C)C(c2cccc(C(F)F)n2)=O)C1)=O c1(CC)ccsc1C(=O)NCc1ncoc1CCNC(c1ccc(C(C)C)s1)=O C1(CC#C)(C(=O)NC(c2cccc(C)n2)C)CCN(C(C2CC23CC3)=O)C1 C(N=c1cc(C)nc(N2CC3C(CO)C3C2)[nH]1)c1c(C)ccs1 Cc1cc(CCC(N2CCOCC2CCNC(=O)CCC(C)N(C)C)=O)nn1C c1(C(=O)NC(CCC)CNC(C2C=CCS2)=O)cccn(C)c1=O CCC(C)C(O)C(=O)N1CC(OCC(=O)NCC2CCC(C)(C)CC2)C1 C=C1CC2(C1)CN(C(C1CCCC(NC(c3ncccc3F)=O)CC1)=O)C2 N1(C(=O)NC2C(NC(=O)Nc3ccccn3)CCC2)CCCc2ccccc21 c1(C(N2CC3CC2C3NC(C2(Cl)CC2(F)F)=O)=O)nc2ccccc2s1 N1(C(C(CSCC)(C)C)=O)CCN(C(c2ccc(COC)[nH]2)=O)C(CCO)C1 CC(C)C(C)C(CNC(=O)C(C)(F)F)NC(c1cc(C(F)(F)F)ccc1O)=O C1(N(C(C=CC=CC)=O)C)CS(=O)(=O)C12CCN(C(=O)C(C)CCC)CC2 C(=O)(CCC(C)(C)C#N)N1C(C(C(N2CCC(NC(C)=O)C2)=O)(C)O)CCC1 C(CCN=C(NCC(C)(C)C(C)(C)O)NC1CCCN(c2cc(C)nn2C)C1)OC N1(C(C2(OC)CC(CF)C2)=O)CCC(CNC(C23CC(O)C2C3)=O)CC1 CC1CC(C(N2CCC(C(C)C(=O)NC3CCC(CO)C3)CC2)=O)CN1C N1(c2c(C)c(NCCc3cnc[nH]3)ncn2)CCC(C2CCCOC2)CC1 c1(C(=O)NC(c2ccccc2)CNC(C(C)(C)OC)=O)cc(C)n(C)c1C C1(NC(CCCNC(C(C)(C)NC(CC)=O)=O)=O)CC2CC1CC2CO N1(C(c2nccc(Cl)c2F)=O)CCC2CCN(C(=O)C(F)(F)CO)CC2C1 CCC(CC)(CO)C(=O)NCC1(NC(c2cc(C(C)(C)C)n(C)n2)=O)CC1 C12(C(=O)OC)C3C4C1C1C2C3C41C(N1CC(CO)C(O)C1)=O N1(C(C(N2CCCCC2)=O)=O)CCCC1(c1ccccc1)CO C1(C)(CN(C(C(C)=C(CC)C)=O)C)CCCC1NC(=O)C(N1CCSCC1)C c1(C(=O)NCC2CC(NC(CCOCCCOC)=O)C2(C)C)ncc(F)cc1F c1(CC)nc(C)c(C(=O)N(C2C3CN(C(C4OCCC4C)=O)CC23)C)o1 N1(C(=O)CCc2ccc(F)nc2)CCC2(CCN(C(=O)CCc3cocn3)C2)C1 C1(CNC(c2ccc(CC)s2)=O)CCC(C)N(C(C2CCC(O)C2)=O)C1 c1(CN(C(C2CCC(CCCCC)O2)=O)C2CC2)nc(C)c(C)s1 C(CC(C(=O)N1CC(C(N2CCC(O)(COC)C2)=O)(SC)C1)OC)OC C(c1ccccc1)=C(CC)C(=O)NCC1CCC1NC(=O)CCC1CCCO1 c1(C(N2CC(OC)C(NC(C3OCCCO3)=O)C2)=O)ncc(F)c2ccccc12 Cc1ccccc1C(C)CC(=O)NCC(C)NC(=O)Cn1nnnc1C1CC1 c1(C(=O)NC(C2(O)CN(C(=O)C=Cc3cscn3)C2)C)ccc2nnn(C)c2c1 c1(C(N2C3CC(CN(C(C(C)OCCCC)=O)C3)C2)=O)c[nH]c2nc(F)ccc12 N1(C(C(CCC)(C)C)=O)CCC(C2CCN(C(=O)CCc3ccc(Cl)nc3)C2)C1 c1(C(=O)NCC2(F)CCN(C(c3cncc(OC)c3)=O)C2)cc2c(s1)CCSC2 C(=O)(CCCC(F)(F)CO)N1CC(NC(=O)COc2cccc(F)c2)C(CO)C1 N1(C(CN(C)C(N)=O)=O)CCC(C2(NC(C3CCS3(=O)=O)=O)CC2)CC1 C1(NC(CC2C(C)C2)=O)CN(C(=O)CN2CCC(N(C)C)CC2)CC1(C)C Cn1nc(C(=O)NC2CCC(CNC(=O)CC3CC(C)(C)CO3)CC2)cc1O CN1CCC(N(CCC#N)C(C2CCC(=O)C2)=O)CC1 C1(CNC(C=C(CC)C)=O)CCCCC1NC(=O)COC1CC(F)(F)C1 c1(CNC(C2C(NC(C(CCC)C)=O)C2)=O)cnc2[nH]ccc2c1 C1(CC(=O)NC2(CNC(C=CCN(C)C)=O)CCCC2)OCCC1(C)C Cn1ncc2c1CC(NCC(=O)Nc1ccc(F)c(F)c1F)CC2 C1(N(CC#C)C(C2(C)CC2Br)=O)CCN(C(=O)C(C2CCC(=O)N2)C)CC1 C(CCN(C(=O)CCOCC)C)(C(C)C)NC(C12CC(CCC)(C1)C2)=O c1(C(=O)NCC2CC(C(=O)NCC(F)(F)F)C2)cc2occc2[nH]1 C1(CCC)CCCN(C(C2CCC(n3cc(-c4cccnc4C)nn3)C2)=O)C1 c1(C(N2CCC(C)N(C(=O)CC3C=CCC3)CC2)=O)cc2ccccc2c(O)n1 C1(CCNC(=O)CCOC2CCOC2)CCN(C(c2ccco2)=O)C1 C(C)(C)(CCC(=O)NC(C1(O)CCN(C(c2ccc(CO)cn2)=O)CC1)C)OC c1(C(=O)NCc2c(C)c(F)ccc2)ccc2nc(C3=CCCC3)cn2c1 c1(CC)cc(C(=O)NCC(O)CN(C)C(c2cn(C)nc2SC)=O)cc(N)c1 C1(C(=O)NCC#CCNC(Cc2n(C)ccc2)=O)CN2CCN1CC2 C1(C2(NC(CN(CC)CC)=O)CC2)CCCCN1C(c1ccc(C(C)=O)[nH]1)=O c1(C(N2CC3C(NC(CC(COC)C)=O)(CC3)C2)=O)cccc2c1CCC2 Cc1ccc(CC(C)C(=O)NCCC(O)CNC(=O)CC2CC(F)(F)C2)cc1 N1(CCN=C(NCC(=O)NCC=C)NC2CC(=C)C2)CCn2nccc2C1 C1(NC(C(C)=CC=C)=O)CCC(C(=O)NCCSCC)C1 c1(C(C)=O)cc2ccc(NC(=O)CN(C)S(=O)(=O)N(C)C)cc2o1 N1(C(CCc2scc(C)n2)=O)CCC(F)(CNC(c2cc(Cl)cn2C)=O)C1 C=C(C)CCCC(=O)NC1(c2ccccc2)CCN(c2ncncc2C#N)C1 N1(C(C2CC(OCC)C2)=O)CCCOC(CNC(=O)CC(C)F)C1 C(=O)(CCC(C)(C)N(C)C)NC(C(=O)NC(C(CO)SC)C)COC c1(C(=O)NCCCN(C)C(c2c[nH]nc2C(C)(C)C)=O)cc(C2(O)COC2)on1 c1(C(=O)NCC2C(C)(C)CCN(C(C(C)SCC)=O)C2)coc2c(Cl)cccc12 Cc1ccc(F)c(CNC(=O)C=CC(C)NC(c2occ3c2CCC3)=O)c1 C1(CC)CN(C(c2ccc(OC)cc2)=O)CCC1NC(=O)CCCC(C)C N1(C=O)CCCC(O)C1.Cc1ccccc1C1(NC(=O)CNC(=O)C2CC2)CC1 N1(C(CCC(C)C)=O)CCC(NC(=O)C=Cc2cnccn2)C(F)(F)CC1 CC12CCOC(C(N3CCC(NC(c4ncnc(O)c4Cl)=O)CC3)=O)(C1)C2 c1(NC(c2ccc(-c3nc(C)sc3)cc2)=O)cc2n(n1)CC(O)CO2 N1(C(c2n(C(C)C)cnc2)=O)CC(NC(C2CCCN2CC(F)(F)F)=O)C(C)C1 CCC(C)(CC)C(=O)N1CC(CNC(c2cncs2)=O)OC(C(F)(F)F)C1 C1(C(CNC(C(C)OCC)=O)(C)C)CCN(C(=O)C(C)CC2CC2)CC1 N1(C(C(=CC2CCCC2)C)=O)CC(O)CC1(C)C(=O)NOCCC(C)O C(=O)(C1CCc2ccccc21)NC(CNC(C=CC=CC)=O)CO CC(C)C(C(C)NC(c1ccnn1CC(F)(F)F)=O)NC(=O)CSCC(N)=O C1(C(=O)NCC2(COC)CC2)CC12CCN(C(c1cn3c(n1)CCC3)=O)CC2 C1(C(=O)NCC2C(NC(C3CCC(C)(CC)O3)=O)CCCC2)CN2CCN1CC2 N1(C(C(CC)NC(C)=O)=O)CC(C)CN(C(c2ccc(C(C)=O)[nH]2)=O)C(C)C1 c1(CC(=O)NC23C(CN(C(c4cccc(OC)c4)=O)C2)C3)cc(Br)ccc1C C12(C(=O)N(c3ccccc3)C3COC3)CCCN(CC1)C2 CCCC(C)(O)C(=O)N1CC(NC(c2cn(C)nc2I)=O)C1 Cc1c(C(=O)NC2CCN(C(=O)CC3OCCO3)CC2O)sc2[nH]cnc(=O)c12 C(=O)(C1=NOC(C(=O)NC(C)(C)CCCNC(C2CC2C)=O)C1)NC(C)C N12CCC3(CC1)CC3CC1(COC1)C2=O.CC1CCCN(C(=O)CC(F)(F)F)C1 N1(C(C(C(CC)CC)C)=O)CCC2(CC1)OC1(CO)CC2(NC(=O)C(C)CF)C1 C(=O)(C#CC1CCOCC1)N1CCC(C(N2CC(C)=C(C)C2)=O)C(C)C1 C1(Cc2ccc(C)o2)CCN(C(=O)C(=O)Sc2cccc(C(=O)O)c2)CC1 N1(CC(=O)NCCC(CNC(=O)C(C)C2CCOC2)OC)CCC(C)(C)C1 N1(C(COCCC#C)=O)CCC(CN(C)C(C2C(c3ccccc3)C2(C)C)=O)C1 c1(C(c2ccccc2OCC(=O)NCc2cccc(Cl)n2)C)cccc(Cl)c1F C(CC(C)(C)C(=O)NCC1(C)CCC(NC(C2(C(C)(F)F)CCC2)=O)C1)OC c1(C(=O)NC2C(C(N(CCOC)C)=O)CCOC2)ccc(O)nc1C c1(C(N(C(CC)CNC(=O)C(c2ccn(C)n2)C)C)=O)ccc(C)c(Cl)c1 C1(CCOC)(NC(CCC#C)=O)CCN(C(c2nc(Br)c[nH]2)=O)C1 C1(NC(C2CCN(C)C2)=O)CN(C(=O)CCC(C)(C)N(C)C)CC12CCC2 n1(CCC(=O)NCC2(O)CC(CNC(C3CC3F)=O)C2)nc(O)c2c1CCCC2 C(C(C)C(F)C(=O)NCC1(F)CCN(C)C1)NC(c1cc(C)sc1)=O C(=O)(C(C)(C)C(C)NC(=O)CCC=CC(C)C)NCCn1c(C)nc(C)n1 c1(C(=O)NCC2C3CN(C(c4on(C)c(=O)c4)=O)CC32)ccc(Cl)nc1N C1(CN2CC(C(CC)=O)C2)CCCN(C2CCSC2C)C1 N1(C(C(C2CCC(=O)N2)C)=O)CCC(NC(c2cccc(F)n2)=O)C2(CCC2)C1 c1(C(N(C2CCCC(NC(C(C)=C(C)C)=O)C2)C)=O)cc(F)c(O)c(F)c1 C1(C(=O)NC(C2CCN(C(C3(O)COC3)=O)C2)C)CCc2nnc(O)cc2C1 C=CCCC(F)(F)C(=O)NCC(O)C(=O)NC1COC(C)(C)C1 Cc1cccc2cc(C(=O)NCCCNC(c3c(Br)noc3C3CC3)=O)nn12 C#CCC(C)(C)C(=O)N1CCC(NC(=O)CCCCCc2ccccc2)C(F)C1 c1(NC(C(=O)N(CCC)CC2CCCOC2)=O)ccc(C(F)(F)F)nc1 N1(C(CCC=C(C)C)=O)CCC2(NC(C3CCCC(C)CC3)=O)CCCCCC12 c1(SC)cccc(CC(N2CCC2CNC(=O)CC(c2ccc(F)cc2)C)=O)c1 c1(C(=O)NCCCNC(C(C2CCCO2)OC)=O)c(N)cccc1[N+](=O)[O-] c1(N2CCN(c3ccc(C)cc3)CC2)nc2c(c(=NCC(C)CC(C)O)[nH]1)COC2 C(C(=O)N1CCN(C(=O)CNC(c2cccc(O)c2)=O)CC1C)(C(C)(C)C)OC C(CC(C(=O)NCCC1CC(C)=NO1)NC(c1cscn1)=O)=CC C(CCCCCC(=O)NCC(O)CNC(C1CCC1C(F)F)=O)SC C(=O)(C(C)(F)C(F)(F)F)N(CC(C)N(C)C(c1coc(Cl)n1)=O)C CCC(O)C(=O)NC1(CNC(C2(CO)CCCO2)=O)CCCC1 C1(CC(=O)NC(C2N(C(C3(C(=O)OC)CC3)=O)CC2)(C)C)CC(C)(C)CO1 C1(C(N2C(C=C)CCC2)=O)CCN(C(=O)c2cc(C(N)=O)c[nH]2)O1 CC1CN(C(C2CCC(C(F)(F)F)O2)=O)CCCN1C(c1ncc(Cl)cc1F)=O c1(C(=O)NCC2(O)CCN(C(Cn3c(=N)[nH]nc3)=O)C2)[nH]cc2c1CCS2(=O)=O c1(COC)nccc(=NC2CS(=O)(=O)CC2NC(c2ccc(O)nc2)=O)[nH]1 CCC(C(=O)NC)NC(C1(CNC(C2CCCN2C(N)=O)=O)CC=CC1)=O C#CC1(F)CN(C(=O)COCCCn2cc(C3CCCC(C)C3)nn2)C1 CC1CCCN(C(=O)CCn2ccnn2)C1CNC(=O)CCC(=O)N(C)C C(C(CNC(=O)C(c1cccnc1)OC(F)(F)F)CO)NC(C1(C)CCC1)=O Cc1nc(F)ccc1C(=O)NCC1(C(N)=O)CN(C(=O)CC2COC3CC2C3)C1 c1(C(=O)NCC2(NC(C(c3ccc(CC)s3)=O)=O)CCOC2)cnnc(O)c1 C(CC(C)(C)NC(=O)CCN(CC)CC)NC(C1C(C=C)C1)=O C1(C(=O)NCC(CC)F)(C(C)N)CCOCC1 C1(C(C)NC(C=CSC)=O)CN(C(=O)Cc2csc(C(F)(F)F)n2)CCO1 C1(C2CCCC2)(NC(C2CC(C)CN(C(=O)C=CCF)C2)=O)CCC1 C1(NC(c2cccnc2F)=O)CC2(C1)CC(NCc1ccc(F)nc1F)C2 c1(C(=O)NCC2(NC(C=CCC)=O)CC(C(F)(F)F)(OC)C2)sc(C)c(C)c1C c1(OC)cccc(CC(=O)NC(C)CC(C)NC(C2CCC(C)C2)=O)c1 C(N=c1[nH]c(=NCC(CO)OC)c2sccc2[nH]1)c1ncc(CC)s1 c1(C(=O)NCC(C2CC2)NC(C(P(C)(C)=O)O)=O)cccc2c1CCC(=O)N2 C1(NC(CS(N)(=O)=O)=O)CN(C(C2CCCC3(CC3)C2)=O)CC12CCOCC2 N1(C(C(CCCC)O)=O)CCC2C1CCCN2C(=O)Cn1ncc2cccnc12 CC(C)(C#N)CCC(=O)NC1CCCCC1C(=O)NC1(C2CC2)CCCC1 c1(NC(C2OCCN(C(c3cc(OCC)n[nH]3)=O)CC2)=O)ccc(N=[N+]=[N-])cc1 Cc1ccc2[nH]nc(C(N3CC4(CCNC(=O)C=CC(C)C)CCC3C4)=O)c2c1 N1(C(C(CC)=CC)=O)CCOCC1CCNC(=O)C(O)C(C)C CC1CN(C(=O)CCOc2cc(Br)ccc2F)CC(C)C1N CCS(=O)CC(=O)NCC1(OC)CN(c2ccc(COC)cn2)C1 C(=O)(CC(C)CNC(=O)CC1CC(F)C1)NC1CCN(CCC)C1 c1(C(N2C(CCNC(c3sc(F)cc3Cl)=O)CCC2)=O)ccn2ccnc2c1 c1(C(N(C)CC2(NC(C34CCC3CC4)=O)CC2)=O)nccc2[nH]ccc12 C1(CCNC(CCC=C)=O)C(C)CCCN1C(c1cccc(-c2cnco2)c1)=O S(=O)(=O)(c1cc(C)cnc1N1CCCCC(N2CCCC2)C1)N1CC=C(C)CC1 C1(COC)(CNC(=O)CC=Cc2ccccc2)CCN(CCO)CC1.C1CCC1 CC1(C)CCCC(CC2CC2)O1.N12CC(C1)C2=O c1(CN2C(C(=O)Nc3c(OCC)cc(F)cc3)CC3CC32)cc(F)c(Br)cc1Cl c1(-c2cn(C(C)(C)CCN3CCOCC3)nn2)ccnc(CO)c1 CC(CN(C)C)CCC(=O)N(C)CC1CN(C(=O)Cc2c[nH]ccc2=O)CCO1 c1(C(N2CCC(CC#C)(C(=O)NC(C)CC3CC3)C2)=O)cccc(C#C)c1C C(=O)(C1=CC2CC(C1)CC2O)N(CC(c1ccc(Cl)c(Cl)c1)=O)CC1CC1 C(N=c1[nH]cnc2[nH]ccc12)C1N(C(C2CCCN2C2CCCC2)=O)CCC1 c1(SC)nc(N2CCC(O)C(C(N3CCn4nccc4C3)=O)C2)ncc1F C1(NC(CCCCN(C)C)=O)CC12CCN(C(=O)CC(C)(F)F)C2 c1(OC)cccc2cnc(NC(C3CC3NC(c3cccnc3C)=O)=O)nc12 c1(C2(O)CC(C(N(CC(C)N(C(C(=O)NC(C)C)=O)C)C)=O)C2)cccc(Cl)c1 c1(CCN(C)Cc2ncon2)cc2ccccc2o1 S(=O)(=O)(c1ccc(NC(C)C2CC2)nc1)NC(C=C)(C)CC c1(C(=O)NCC2CCCN(c3cc(OCC)nc(C)n3)C2)cc2n(n1)CC(F)C2 CCC(C)(C)C(C)CC(=O)N1CCCC(C)(C)C1CNC(=O)COCC(=O)NC N1(C(c2cccc(-c3cc[nH]n3)c2)=O)CCC2CC1CN(C(C1(O)CCC1)=O)C2 C(C)(CCCNC(=O)C(O)CNCc1cc(C(=O)COC(C)C)no1)OC1CCC1 N1(C(CCn2c(C)ncc2)=O)CC2CC1CN2C(C12CCC1CC2)=O Cc1ccn(C(C)C(N2CCC(C(=O)NC(c3scnc3C)C)C2)=O)n1 C1(CCC#C)CN(C(=O)CC)CCN1C(=O)CCCc1ccc(C2CC2)cc1 C1(CNC(C(C)CC(F)F)=O)CN(C(=O)CCC(C)(C)F)C2(CCC2)C1 N#Cc1ccc(Cl)c(C(=O)NC(Cc2cn(-c3ccccn3)nn2)C(=O)O)c1 Cc1ccc(C(=O)NC2CC(CNC(=O)CC3CC4C=CC3C4)C(O)C2)c(N)c1 N1(C(CC(C=C)CC)=O)CCC2(CC1)CC2CNC(c1conc1C1CCC1)=O O(NC(=O)CC(C)C(C)(C)NC(C1CCCCO1)=O)CCCOCC C1(NC(C=Cc2scc(C)n2)=O)C2CC1CN(C(C1(F)C3CCCC13)=O)C2 C1(CC(N2C(CNC(C=CC(CC)=CC)=O)CC2)=O)CC2(CCC2)C1 c1(CC)cccc(CC)c1CC(=O)NCC1CC(O)CN1C(=O)CC1(C)CCC1 c1(N2CCC(C(C)(C)NC(=O)COCC3CCCO3)C2)ccc(C#N)nn1 C(C#CC#CCO)NC(C1CCCCN1C(=O)COc1cccnc1)=O C1(CC(=O)NCC(CNC(=O)OC)F)CCC(NC(c2ncsc2C(C)C)=O)C1 C1(F)(CNC(c2ccc(C)o2)=O)COCCN(C(c2ccc(CO)c(F)c2)=O)C1 C1(NC(CC(CC)OC)=O)CC2CC(NC(=O)CCCCN3CCCC3)CC12 C1(C(=O)NCC(C)N(C(=O)C(=O)C2CCCC2)C)CCC2(CCOCC2)O1 C1(C(N2CC(O)(C3CCCN3C(C3CC(=C4CC4)C3)=O)C2)=O)CC12CCOCC2 c1(CN(C(C(C2CN(C(CC)=O)C2)OC)=O)C)c[nH]nc1C c1(CC(=O)NC2C(NC(C(CC#C)C)=O)C2)cc(F)cc(Br)c1 C1(C(=O)NCCC2(O)CN(C(c3cc(Cl)ncc3N)=O)C2)(OC)CCCC(C)C1 CCC(C)C(C)C(=O)N(C(C)CCNC(c1cnnc(Cl)c1)=O)C c1(OCC(N2CCC(C(C)NC(C=C(CC)C)=O)C2)=O)ccc(CC)cc1 C1(CC#C)(C(N2CC(OCCO)C2)=O)CCCC1.C1(C=O)(CNC=O)CC1C C1(CC)CC(C(=O)NC2CC(N(C(=O)CC=CC(C)(C)C)C)C2)C1 CC(CCCC(=O)NC1CC1)NC(=O)C(C1CC1)C(c1cn(C2CC2)nn1)(C)C c1(N(C)C)ncc(C(N2CCC(c3ccccc3[N+](=O)[O-])C2)=O)cc1C#N C1(NC(C(CC)C(F)(F)F)=O)CCC12CCN(C(C1CN(S(C)(=O)=O)C1)=O)CC2 C1(N(C(C(C=CC)O)=O)CCF)CCCN(C(=O)COC(C)=O)C1.CCCCCC C1(F)(C(N(CCC(=O)NCCC(C)CCC)CC=C)=O)CC=CCC1 C(=O)(CCCCCN=[N+]=[N-])NCCC(C(=O)N(CC(=C)C)CC(=C)C)O N1(C(c2n(C=C)nnc2)=O)CCC(NC(C2CC23CC(O)C3)=O)C(F)(F)CC1 N1(C(Cn2c(C)cnc2)=O)CC(O)CC1(C)C(=O)NCCC(F)(F)CO c1(-c2nc(CSC)nn2C2CCCS(=O)(=O)C2)ccc(=O)n(-c2ccccc2)n1 c1(CC(CC)NCC2CCCCC2C(F)(F)F)ccc(C(F)F)cc1 O=C1Cc2cc(C(N3CCC4CCC(C3)N4c3nnc(C#N)s3)=O)ccc2N1 c1(C(N(CCCn2cc(COC(=N)O)nn2)C)=O)ccc(-c2cnco2)cc1 c1(C(N2CCN(C(C(CC)OC)=O)C(CF)C2)=O)ccc2ncsc2c1 C1(NC(=O)CC2CC3(CCC3)C2)CC(CNCc2ccc(Cl)cc2Cl)C12CCC2 C(=O)(CCS(N)(=O)=O)N1CCC(N2CCC(NC(C3C(OC)CC3)=O)CC2)CC1 C1(NC(c2cc(C3CC3)ccn2)=O)CC2(CCN(C(=O)C=Cc3cscn3)C2)C1 C(C)(C)(CCC(=O)NCCc1ccncc1)NC(C1CC(C(=O)OC)C1)=O c1(OC)ccc(C)nc1C(N1CC2CC1CC2NC(=O)CCOCC(F)(F)F)=O c1(C(N2CCN(C3CCC3)CC2)C(=O)NC(C(=O)OC)C)ccc(Cl)c(C)c1 C1(C(=O)NC2CC3(C(NC(c4c(CC)n(CC)nc4)=O)C3)C2)CN2CCN1CC2 N#CC1CCN(C(=O)CCOCCNC(=O)C(c2ccccc2)F)CC1 C1(C(N2CC(CC(C(=O)N(C3CCCC3)CC=C)F)C2)=O)CC2COCC2C1 C(=O)(C1CSc2ccccc21)NCCC1=CCN(C(C23OC(C)C(C2)C3)=O)CC1 C1(N(C(C2(C(N)=O)CC2)=O)CC)CCN(C(=O)C=Cc2c[nH]nc2C)CC1 N1(C(c2c(C)oc(Cl)n2)=O)CC2CN(C(c3cnn[nH]3)=O)CC2C(F)(F)C1 N1(C(C(CCC)CC)=O)CCC2(CCCN2C(c2cnc(C(F)F)cc2C)=O)C1 N1(C(c2cc(C)[nH]c2)=O)CCSCC1CCNC(c1ncccc1C(C)(C)C)=O C(=O)(C1CS(=O)(=O)c2ccccc21)N1CC(NC(CC2C(C)(C)C2)=O)C1 C(c1nc2ccccc2o1)=CC(=O)N(CCNC(c1c(C)cnnc1O)=O)CC C1(CNC(CC(C(CC)C)O)=O)(NC(=O)Cn2ncnn2)Cc2ccccc2C1 C(=O)(C1CCc2nccn21)N1CC(NC(c2c(CC)nco2)=O)CC12CCC2 C1(NC(c2cncc(OC)c2)=O)CC2CN(C(=O)CC(=O)NC3CC3)CC2C1 C1(NC(c2c[nH]cc(C)c2=O)=O)CC2CC(C1)N(C(C13CCCN1CCC3)=O)C2 C1(NC(c2cn(C)c(=O)n2C)=O)CC12CCN(C(=O)C#CC1CCOC1)CC2 c1(C(=O)NC2COCCN(C(C(C)(F)F)=O)C2)occ2c1CCCC2 N1(C(CC)=O)CC(N(C(=O)Cn2ccc3ccccc23)CC)CC(C)(C)C1 c1(-c2ncc(CNC(c3ccsc3)C)s2)ccccc1F N1(C(C2(CCNC(C(n3c(C)ncc3)C)=O)CC2)=O)CCC(C)(C)C1C CCC(CC(=O)NCC1(C)CCN(C(=O)C(COC)C(F)(F)F)C1)C(F)F C1(NC(C(CC)C)=O)(CNC(=O)Cc2ccc(F)cc2F)Cc2ccccc2C1 n1(C(C)C)ccnc1CNC(=O)C=CCNC(c1ccccn1)=O CC(C)C(C)CN=c1[nH]c(=NCCOC(=N)O)[nH]c2ccc(Cl)cc12 c1(C(=O)NCCCCNC(CCOCC(C)C)=O)cc2c(s1)CCS(=O)(=O)C2 N1(C(C2(C)CC=CCO2)=O)CC2CCCC2(CNC(=O)Cn2cc(CO)nn2)C1 CCC(CC(=O)NCCCCCSC)NC(=O)CC1CC=CCN1C N1(C(C2N(C(C=CCCC)=O)CC(F)C2)=O)CCS(=O)C(C)C1 C1(CC)CCN(C(=O)COC2CC(NC(=O)CC3CC=CCC3)C2)CCO1 CN1CCOC(C(=O)NCC2(C)CN(C(c3ccns3)=O)CCO2)C1=O c1(CSC)cccc(C(=O)N(CCNC(=O)C(C)CO)CC2CC2)c1 CC(CC(=O)NC1(C2CCCN2C(=O)CO)CC1)C1CCCO1 Cc1nc(CC(=O)NC2CC(NC(c3ocnc3-c3ccccc3)=O)C2)c(C)s1 C=C(C)CC(C(=O)NC(C)Cc1cn[nH]c1)NC(=O)C(C(C)C)SC n1(CC(=O)N(C2CCC(CNC(C(CCSC)O)=O)CC2)C)cccc(C)c1=O C(C(C)(C(=O)NCCOC1CN(C(C2CCN(C)C2=O)=O)C1)OC)OC Cc1nc2c(o1)CCN(C(C1CCCCCN1C(C1CCC=CCCC1)=O)=O)C2 N1(C(C2C(C)(C)C2)=O)CCC(O)(CCNC(=O)C2=CCCCC2)CC1 C12(NC(c3c(C#C)cn(C)n3)=O)CC(C)(C1)OC21CN(C(C2CC2(Cl)Cl)=O)C1 C(=O)(C1=CCC(C)(C)CC1)N(CC(C)NC(c1cc(OC)ccc1O)=O)CC c1(OC)ccc(N)c(C(=O)NC(C)CNC(=O)COC2CCCOC2)c1 CCC(N=c1[nH]c(N2CC3CC3(CC)C2)nc2cc[nH]c12)c1cccc(OC)c1 c1(CC(=O)NC2C(NC(=O)CCOCC(F)F)CCC2)cn2c(n1)CCCC2 Cc1ccc(C(=O)NC(C)(CNC(=O)C(O)CF)CC(C)C)c2cccnc12 C1(NC(C2(CNC(c3cn(CC)nn3)=O)CC2)=O)CCCC(C(N)=O)C1 c1(C(C)=O)cccc(N(C(=O)NC(C)CN2CCOCC2)Cc2ccco2)c1 C1(C)(C(=O)NC2CC(C)N(C(c3cnn(C)c3)=O)C2)Cc2ccccc2N1 c1(C(N2CC(NC(CC=C)=O)C(C)CC2)=O)ccc2nc(O)n(C)c2c1 C1(C)(C(=O)OCC=CCCC)C2CC3CC(C2)CC1C3 CCCCC(CC)n1cc(NC(c2cnn(C3CC3)c2)=O)nn1 c1(CC)cccc(C)c1C(=O)NCC1(F)CN(C(c2nc(C(C)C)oc2C)=O)C1 C1(NC(c2c(CCC)n(C)nc2)=O)CCCCN(C(=O)Cc2ccnnc2O)C1 C12CN(C)CCN1C2.Cc1cc(C(=O)O)nn1CCn1cc(CC2CC2)nn1 c1(CN(C(C2N(C(C)C)C(C)(C)OC2)=O)C)cc(Br)cc2c1OCC2 C(=O)(C1=CCC(C)CC1)NCC(C)CNC(c1ccc(-c2ncn(C)n2)cc1)=O C1(C(C)(C)C)(CNC(CCC=CC)=O)CCN(C(C2(c3cc[nH]n3)CCC2)=O)C1 c1(C(=O)NCC2N(C(C(C=C)(C)C)=O)CCC2)c(Br)ccc(Cl)c1F N1(C(COCCCCC)=O)CC2CC2(CNC(c2cc(C(C)(C)C)c[nH]2)=O)C1 C1(CN(C(=O)COCC2CC2)C)CCCN(C(c2ncc(Br)cn2)=O)C1 Nc1ccc([N+](=O)[O-])cc1C(N1CCOCC1CNC(C1(F)CCCOC1)=O)=O c1(C(C(=O)NC(C)(C)C)N(CCCC(F)(F)F)CC)noc2c1CCC2 CC1CCC(O)CN1C(c1ccc(Cl)cc1O)=O O=S(=O)(c1cnc(N2CCOCC2)c(Cl)c1)NCCCOc1ccc(F)c(F)c1 c1(C(=O)NCCCCNC(c2ccn(C)c(=O)c2)=O)c(F)cc(F)c(F)c1F N1(C(=O)Cc2nc(F)c(F)cc2F)CCCC2C1CCCN2C(=O)CC1CC1 N1(Cc2ncc(OCC)cn2)CCC(NC(=O)Cc2ccc(Cl)c(F)c2)C(C)C1 c1(CNC(C)(CCCO)c2nnnn2CCCF)c(Cl)cccc1[N+](=O)[O-] C1(NC(C(c2ccccc2)C)=O)CC2(C1)CC(NC(c1sccc1Br)=O)C2 C1(CN(C(C=C(C)C)=O)C)CCCCN1C(=O)CC(C)c1ccncc1 N1(C(c2nccc(C)c2)=O)Cc2ccc(C(=O)Nc3cc(Cl)cnc3C)cc2C1 C(=O)(CCCN(C(=O)C(C1CCC1)NC(=O)CCCF)C)NC CC1CC=C(C(=O)N(C(C)(C)CC(N2CC(=O)NCC2C(N)=O)=O)C)CC1 N1(C(C(CSC)(C)C)=O)CCOC2(CCN(C(=O)Cc3sc(C)cc3C)C2)C1 C1(C)(C(=O)NCC(C)(C)NC(C2(F)CCOC2)=O)CC(c2ccccc2)=NO1 CC(CCCC(=O)N(C1CCCC1C#N)C)NC(=O)C=C1CCC1 c1(C(=O)NC(CNC(C2(c3cc[nH]n3)CC2)=O)CO)cc2ncccc2[nH]1 Cn1cc(Cl)c(C(=O)NC2CC3C(NC(C4CCS(=O)CC4)=O)C3C2)n1 c1(C(=O)NCC2C(NC(CCC(CC)CC)=O)C2)cc2cccc(OC)c2o1 c1(C(=O)NC2CCCCN(C(c3n(CC)nc(C)c3)=O)C2)ccc(F)cc1C#N N1(C(COCCN(C)C)=O)CC(NC(=O)C(=C2CCCCC2)F)CC(F)C1 c1(C(N(C)CCOCCNC(=O)Cc2cnccn2)=O)cncc(Cl)c1Cl N1(C(c2ncc(C)cc2C)=O)CC(NC(C2CC3CCC3C2)=O)C2CCCC2C1 C(=O)(CC(C)C(F)(F)F)NCCCC(C)NC(c1snc(Cl)c1Cl)=O C1(NC(CC(C)NC(=O)Cc2ccccn2)=O)CC2CCC(C1)C2O c1(C(N2C(CNC(C3(OC)CC3)=O)CC(C(C)C)CC2)=O)cn2cc(Cl)cnc2n1 N1(C(C2N(C(C)C)CCCC2)=O)C2CCC1CN(C(=O)C(O)C1CCC1)C2 N1(C(COC(C)C)=O)CCn2c(CNC(C3CCC4CCC(=O)N34)=O)nnc2C1 C(CCCCCN=[N+]=[N-])NC(C(C)(CO)NC(c1cc(F)cnc1O)=O)=O N1(CC(=O)NC2CCC(NC(C(C)(C)C)=O)C2)CCCS1(=O)=O N1(C(c2n(C)nc3c2CCC3)=O)CCC2C1CCCN2c1ncncc1F c1(NC(CC2N(C(C3CCC(=O)C3)=O)CCOC2)=O)cccc2[nH]ccc12 C1(C(N(CCOCC=C)C)=O)CN(C)CCN1C(=O)CC(C)(O)C=C C12(CNC(CCOC)=O)CC(NC(=O)CC(C)C(C)C)(C1)C(C)O2 N1(C(C(C(=O)OC)OC)=O)CC2(CCCC2)C1C(=O)N(C)Cc1ccns1 c1(OC)cccc2[nH]cc(CC(N3CC(NC(C4CSC4)=O)CC3C)=O)c12 C(c1cccc(O)c1)=CC(N1CCC(NC(c2c(CC)nc(C)o2)=O)C1)=O c1(C(=O)NCC(C2CCCC2)NC(=O)CCC2CCOC2)cncc2[nH]ccc12 C1(NC(=O)NCC2C(c3ccc(Br)cc3)(C)C2)CCCC2OCCC12 C1(C(N)=O)CN(C(=O)C(=O)NCCC2(C)CCCO2)c2ccccc2O1 O=C1CC(C(=O)NCC(C2CC2)SCC2(c3cn(CC(=O)O)nn3)CC2)=NN1 c1(OC)cccc(C(=O)NC2(CCNC(=O)C(F)(F)C3(OC)CCC3)CC2)c1F c1(C(=O)NCC(=O)NCc2ccco2)cccc(-n2cncn2)n1 c1(C(=O)NCCN(C(C2CCSC(C)C2)=O)CC)coc(C#N)c1 c1(OC)cccc2[nH]cc(C(=O)NC3CCC(NC(c4ccccc4I)=O)C3)c12 N1(C(c2n(CC=C)ccn2)=O)CCCC(C2CCCN(C(=O)C(F)OC)C2)C1 Cc1ccc(-c2cnc(NC(C3CC4CCC3O4)=O)c(O)c2)c(C)n1 C(=O)(C(O)CC(C)(C)C)N1CC(N(C(=O)Cn2nc(C(F)(F)F)cc2Cl)C)C1 c1(CCC(=O)NCC2C(NC(CC3(OC)CC3)=O)C2)nc(C)c(C)[nH]1 c1(C(=O)NC2(C)CC(NC(C3(CCC)CCNC3=O)=O)C2)ccc(C#N)cc1C C(=O)(C(C)(C)C(F)(F)F)N1C2CC(C(=O)NC(C(C)C)C3CC3)C1CC2 C1(NC(CSCC)=O)CN(C(c2cc(OC)cc(Cl)c2F)=O)CC12CCC2 c1(C(=O)NC(CC)CNC(c2cccnc2S)=O)c(C)nn2c(C)cc(C)nc12 C1(C(=O)NC2CC(C)(NC(CC3CCC(C)CC3)=O)C2)C2C3CCC(C3)C12 C(=O)(C1=CC2CCC(C1)C2)NCC(C(=O)N(CC(C)C)CC(N)=O)CC1CC1 C(=O)(CC1CS(=O)(=O)c2ccccc21)NCC1CCN(C(C#C)=O)CC1 C1(NC(c2c(CO)cccc2F)=O)CN(C(=O)C2=COCCC2)C2(CCOC2)C1 C1(NC(=O)OC(C)(C)C)CC12CCC(C(=O)NCc1n[nH]cc1C1CC1)CC2 N=c1cc(C(=O)NC2CCC(NC(=O)Cn3cccn3)C2)c(Br)c[nH]1 C1(NC(CN(CCOC)C)=O)CC12CCN(C(c1csc(C(C)C)n1)=O)CC2 c1(C(=O)NCC(=O)N(CCNC(C(CC)N2CCCC2=O)=O)C)ccccc1C N(C1CCCc2cc(CNC(=O)CC(C)c3ccco3)ccc21)C(CC(=C)C)=O c1(OC)cc(C(=O)NC(CNC(=O)C(C)SC)CC(F)(F)F)ccc1Cl C1(C(=O)NC2CC(F)(F)C2)CN(C(c2cccc(F)c2O)=O)CCC1O c1(CC)ncoc1C(=O)NC(C)(C)CC=CC(N1CC(c2nncs2)C1)=O C1(NC(COC)=O)CCCC(CNC(=O)C(CCSC)OC)C1 C1(NC(c2cnc(C3CC3)nc2)=O)CN(C(C2CC2F)=O)CC2(CCC2)C1 C(=O)(C(C)CN(C)N1CCOC2c3ccccc3OCC12)c1c(C)cccc1[N+](=O)[O-] C1(O)(CNC(c2ccsc2)=O)CCCN(C(C2CCCOC2c2cc[nH]n2)=O)C1 C1(CNC(CCCOCC)=O)CC2(CCOCC2)CN1C(=O)C(F)(F)CO N1(C(C(CCC)C)=O)CCN(C(c2ccc(Cl)cc2OCC=C)=O)CC1C Cc1cccc(O)c1C(=O)NC1CC1CNC(c1cc(C)n(C2CC2)n1)=O N1(C(c2scc(COC)c2)=O)CC(CNC(=O)Cc2cnn(C(F)F)c2)C(O)C1 c1(C(=O)NCC(CC)NC(C2CCCN2C2CC2)=O)cc(OC)cc(OC)c1 c1(C(=O)OC)cc(C(=O)NCCNC(=O)COCC2CCOC2)c[nH]1 C1(CNC(C(C(C)C)N(C)C)=O)CC12CCN(C(c1cc(Cl)c(Cl)n1C)=O)CC2 N1(C(C2CN(C(C(CCC)C#N)=O)C(C)(C)C2)=O)CCC2OCCC2C1 c1(C(=O)NCC2C(CNC(c3nc(C)nc(O)c3)=O)C2)nc2nccc(C)n2n1 CC1(C)CCC(CC(=O)NCC(C(C)(C)C)NC(=O)C2=CCC2)C1 c1(CC)cc(C(=O)NC2CCC(NC(C34CCOC(C)(C3)C4)=O)C2)ccc1OC C12(C(=O)NCCN(CC(C)O)C(c3c(C=C)cnn3C)=O)CCCC1CC(=O)C2 C1(O)(CCNC(=O)CCC2CC2)CCN(C(=O)Cc2c(Cl)cccc2Cl)CC1 C(=O)(C(COC)CC(C)C)NCC(=C)CCNC(=O)C(C)COC(C)=O C1(N(C(C(COC)C)=O)C)CCC2CN(C(c3cc([N+](=O)[O-])ccn3)=O)CC12 N1(C(C2(CCN(C)C)CC2)=O)CC2CCC1C1CN(c3nnco3)CC21 CCC1=NOC(C(=O)NCc2cccc(NC(c3scnc3C3CC3)=O)c2)C1 C=CC1(CC(N2CCCC(N(C(=O)CNC(=O)NC3CC3)C)C2)=O)CCCCC1 c1(C(=O)NCCC(C)N(C(=O)C(C)C2CCC2)C)csc(-c2ncc[nH]2)n1 N1(C(C2(CC)CCN(C(=O)CC3CC4CC4C3)CC2)=O)CCCC2CC1C2(C)C C(C1=NOC2CN(C(c3c[nH]nc3C(=O)NC)=O)CC12)NC(CCC(=C)Cl)=O C12=NC3=C(C(=NC4CCN(C4)N1C)N2)SCC3.c1(C=O)cn(C)cn1.C1(NC)CCC1 N1(c2nccc(C(=O)OC)n2)CC(C(N2CC3CC2CN3C)=O)CC(F)C1 Brc1ccc2c(c1)OCCN2Cc1cnc2n1CCC2 C(=O)(CC(C)(C)CC(=O)NC1CN(C(=O)C2=C(C)CCC2)CC1C(F)F)OCC C1(C(N2CC(C)N(c3ccncc3)CC2)c2ccccc2)CCOCC12CCC2 C1(C(N(CCOCCC(=O)NC(C(=O)OC)C)C)=O)COC(C)C1 C1(CNc2cccc(CN(C)C(C3CC(N(C)C)C3)=O)c2)CC2C=CC1C2 O=C(C(O)C(F)F)NCCOC1CCN(C(=O)C(F)(F)Cc2ccc(F)cc2)C1 C(C(C)(C)C#CC(=O)NC1(CO)CC2CCCC12)NC(c1nc(C)oc1)=O C(CCC(C)(C)C(=O)N1CCCC(CCF)C1)NC(C(CC)CC)=O C1(C(=O)NC(CCC)C(=O)NC)CCCCCN1C(C1CCOCC1)=O C1(CC(C)C)CCN(C(=O)C(C2(O)CCCCC2)NC(=O)CSC(C)C)CC1 N1(C(c2ccc(CC)[nH]2)=O)CCCCC2(CCN(C(=O)CCC3CCOC3)C2)C1 c1(C(N(CC(CC)NC(C2(O)CCCCCC2)=O)C)=O)cc(C)cc(Br)c1 Cc1ncn(C)c(=O)c1C(=O)NCC#CCNC(C1CC2CCC1O2)=O c1(C(=O)NC2CN(C(C(C3CCC3)OC)=O)CC2O)ccc(F)c2ccccc12 c1(CC)cc(C(=O)NCC2C3CN(C(=O)C(C)(CC)CC)CC23)ccc1O C1(NC(c2n(CCCC)nnn2)c2nc(CO)cs2)CCC(C)(C)CC1 c1(C(=O)NC(C2CCCN(C(C3CC(C#N)C3)=O)C2)C)cnc2c(c1)CCC2 N1(C(C(CCNC(C2(CC=C)CC=CC2)=O)OC)=O)CCc2ccccc2C1 N#Cc1ccc(N)c(C(N2CCCN(C(=O)CCS(N)(=O)=O)CC2)=O)c1 C=CC1(C(N2CCC(CC(C)C)CC2)=O)CCN(C(c2ccnc(C)c2)=O)C1 C(=O)(C1CCc2snnc21)NC(CCCNC(CCNS(C)(=O)=O)=O)(C)C C(=O)(CCCCC(=O)N1CCCC1CCNC(C1(C)CC1(Cl)Cl)=O)OC C1(NC(c2n(CCOC)nnn2)c2n[nH]cc2Br)CCN(C(=O)OC(C)C)CC1 N1(C(c2c(NC(C)=O)cccn2)=O)CCCC12CCN(C(C1CC(F)C1)=O)C2 CC(CNC(=O)CN1CCSCC1)C(=O)N1CC=CCC1 C1(CC#C)(C(=O)NC2C=CC(CNC(=O)Cc3ccc(C)s3)C2)CCCO1 c1(C(N(CCN(C(C)C)C(c2ccnnc2S)=O)C)=O)ccc(S(C)(=O)=O)cc1 C1(NC(c2ccn(CC)n2)=O)CC2CC1N(C(c1cnn(CCN(C)C)c1)=O)C2 N1(C(=O)OC(C)(C)C)CCC1CCCNC(CCCC1CCCO1)=O C=CCC(C)(C)C(=O)N1CCC(C(=O)NCc2cc(O)ccc2O)C1 c1(C(=O)NCCC2(CNC(C3NC(=O)OCC3)=O)CC2)nnc2ccccc2n1 CC(C)C(O)C(=O)NC12CC(C1)N(C(C1(c3ccc(F)cc3)CCC1)=O)C2 c1(C(=O)NCC23CC(CN2C(c2cc(O)ccc2O)=O)C3)[nH]nc([N+](=O)[O-])c1Cl c1(C(=O)NCC2(CNC(C(N3CCC(O)CC3)C)=O)CC2)cc(N)c(Cl)c(O)c1 C1(F)(NC(CN(CCOC)C(=O)OCCCNC(=O)NC(C)(C)C)=O)COC1 N1(C(C(CC=CC)CC)=O)CC(O)(C2(CNC(=O)CC3C=CCCC3)CC2)C1 c1(COC(C(C)C(C)c2ccccc2Cl)=O)cn2ccccc2n1 c1(C(C)C)ncc(C(=O)N(C(C)CNC(=O)C(C)C2CC2)C)s1 n1(CC(=O)NC2CC(CCNC(C3CN(C(C)C)C3)=O)C2)ncc(O)nc1=O N1(C(C=C(C)C2CCCCC2)=O)CC(NC(=O)CCC2CCCC2)CC(C)(C)C1 Nc1c(C(=O)NC2(CCNC(c3n[nH]c4c3CCC4)=O)CC2)sc2nccnc12 C1(C(=O)NCC2CCC2)CCC2(CN(C(c3ccn(-c4ccccc4)n3)=O)C2)O1 CCC(C)C(C)N=c1[nH]c(CC(N2CCOC(C3CCCCC3)C2)=O)cs1 C1(CNC(C=CC(CC)=CC)=O)CN(C(=O)CN(C)C(c2ccoc2)=O)CC1C C1(C2CCN(C(=O)C(C)(C)C(C)(C)O)CC2)(NC(C(C=CC)O)=O)CC1 N1(C(C(C)OCC)=O)CCN(C(C2CC(F)(F)C2)=O)C(CC)C1 c1(C(=O)NC2C3CN(C(CCSCCCC)=O)C(C3)C2)cc(F)c(F)c(F)c1 c1(C(N2C3C(CNC(CC4(OC)CCC4)=O)C(C3)C2)=O)cnc2[nH]cnc2c1 CC1COC(CO)CN1C(=O)Nc1ccc(-c2ccsc2)nc1 c1(C(=O)NCC2COCCN(C(c3cc(C)c(C)s3)=O)C2)ccnn2ccnc12 CC(C)C(CNC(C12COCC1C2)=O)NC(=O)C(=O)NC1CC1 S(=O)(=O)(c1cccnc1NCC1(OC)CCS(=O)(=O)C1)NC1CC2(CC(OC)C2)C1 N1(C(c2nc(CC)oc2)=O)CCC(C(C)C(N2CCOCC2)=O)CC1 C=CC(CC)CC(=O)NCC1(NC(c2ccnc(N(C)C)c2)=O)CCCC1 c1(OC)cc(C(=O)NCC(C)(C)CN(C(=O)Cc2ccc(F)cn2)C)ccn1 CC1(C)COCC(C(N2CC(CNC(c3nn[nH]c3Cl)=O)C(F)(F)C2)=O)O1 c1(CCC)nc2cc(C(N3CC(C)(NC(=O)CCCCOC)C3)=O)cc(C)c2[nH]1 C1(C2CC2)(NC(=O)CCc2ccsc2)CCN(C(C2CCNC2=O)=O)C1 c1(OC)cccc(OCc2cc(C)on2)c1N(C)C(=O)NCC.C(CC(C)C)O C1(CC(=O)OC)CCCC(NC(C2CC(C(F)F)(NC(=O)OC(C)(C)C)C2)=O)C1 Cc1cn(C)cc1C(=O)NC(C)CN1CCN(C(C2(CN(C)C)CC2)=O)CC1 C(C(=O)NCCC(C)N(C)C(C1CC(C(N)=O)C1)=O)(C(C)C)c1cnc(C)s1 N1(C(c2cc(CC)ncc2)=O)CCCCCC1CNC(=O)CCN(C)CCO O=C(CN1CCCC(O)(c2cnn[nH]2)C1)C1Cc2ccccc21 Cc1ccc([N+](=O)[O-])cc1Cn1cc(CN2CC(c3ccc(Br)c(F)c3)C2)nn1 CS(=O)(=O)c1ccc(NC(=O)Cc2csc(-c3ccsc3)n2)cc1 CC1(C)OCc2cc(C(N3CCOCC3CNC(=O)Cc3ccon3)=O)ccc21 C(C(F)(F)CCC(=O)NCCCNC)n1cc(C2(C(=O)OC)CC2)nn1 c1(CNC(CC(C)NC(N)=O)=O)cccc(NC(=O)Cc2ccccc2Cl)c1 N1(C(c2ccsc2Cl)C(=O)NCC2CCCO2)CCC12CCCS(=O)(=O)C2 C(CC(CC)C(=O)N1CCCCC1CCN(C(=O)COCCOCC)C)=CC Cc1ccc(CCC(=O)N(C2CC2)CC2CN(C(=O)CC(C)c3ccccc3)C2)o1 C(CC(O)C(=O)NCC(=C1CN(C(C2CN(C)C(=O)N2)=O)C1)F)N(C)C C1(OC)CC2CC(NC(=O)CC(C)(C)OC)C2C1 CC1N(C(C2C3CCC(C3)N2C(C2CCC2C#N)=O)=O)CCC1(C)C CC1CN(C(C2(c3cccc(F)c3)CC2)=O)CC1CNC(c1ncn(C)n1)=O c1(NC(C2CCCN2C(C2CCCN2C(c2cccs2)=O)=O)=O)cccc(I)n1 C(=O)(C1=NOC2COCC12)NCCCCC1CN(C(C2(S(N)(=O)=O)CC2)=O)C1 N1(C(C(CCCOC)C)=O)CC2(CCCCN2C(c2snnc2C)=O)C1 C(C)(CCC(=O)NCC(c1ccccc1)NC(c1cc(C)nn1CCO)=O)OC C1(N(C(CCCN(C)C)=O)C)CN(C(C2C(Cl)(Cl)C23CC3)=O)CC12CC2 c1(C(=O)NOCC(C)NC2CCC2)cc(O)sc1C.C(CCOC(C)(C)C)OC NS(=O)(=O)c1ccc(CC(=O)NC2CCN(C(=O)Cc3ccno3)CC2F)cc1 C1(NC(C2CC2F)=O)CCC12CN(C(=O)CCc1ccccc1F)C2 CC(C)C(O)CC(=O)NCC1(CNC(C2CC3CC3C2)=O)CCCCC1 c1(C(=O)NCC=C(CCC)CCNC(=O)OC(C)(C)C)ccc2c(n1)CCC2 N1(C(C)=O)CC2CCN(C(C3CCC4CCCC4C3)=O)CC12 Cc1nnc(O)c(C(=O)NC2CC(CNC(=O)COCC3(F)CC3)C2)c1C c1(C(N2CC(C)(NC(c3ccc(-n4cccc4)nc3)=O)C2)=O)cc(=O)cc(Cl)[nH]1 C1(NC(COC(CC)C)=O)CCN(C(c2ccc(NC(C)=O)cn2)=O)CC1F CCC1C(=O)Nc2ccc(C(N3CC(CNC(c4csc(SC)n4)=O)C3)=O)cc21 N1(C(c2cccc(C#N)c2)C(=O)NC(C)C)CCN2CC(F)(F)CC2C1 CC1(C)CC(CC(=O)NCCC(F)(F)F)CN1C(=O)C=CC(F)F C1(NC(C2(OCC)CC2)=O)CC1C1CCN(C(C2CCCCN2CC)=O)CC1 C(CC(C(=O)N1CCC(COC)CC1)NC(=O)CC1CCC(=O)CC1)OCC O=C1CCN(CC(=O)NC(Cc2ccco2)C(=O)N2CC(OC(F)F)C2)CC1 C=C(Cl)CCCN=c1cccc(S(=O)(=O)NC2(C)CCC(C)(C)C2)[nH]1 N1(C(C(CC)SC)=O)CC2CC(NC(=O)COC3CCN(CC)CC3)C1C2 C1(O)(CN(C(=O)C(F)n2ccnc2)C)CN(C(=O)CCc2cncs2)C1 N1(C(CCCSC)C(=O)NC2CCC(F)(F)CC2)CCC2CCC(O)C1C2 c1(CNC(=O)NCc2c(OC)cc(Br)cn2)cc(Br)cc2c1OCC2 c1(C(N2CCN(Cc3c(OC)c(Br)ccc3)C3C2C3)=O)ccc(F)c(F)c1O C(c1ccccc1F)=CC(=O)N(C)CC1(O)CCN(C(=O)Cc2ccc(Cl)s2)C1 N1(C(COC)=O)CCC(O)(C(C)NC(c2cn(C3CC3)cn2)=O)C1 C1(NC(=O)CCn2ccnn2)CN(C(=O)Cn2ncnn2)CC12CCC2 c1(OCC(=O)NCc2cc(C(N(CC)Cc3nc[nH]n3)=O)no2)ccn(C)n1 c1(C2C(C(=O)NCc3cn(CC)nc3C(F)(F)Cl)C2)ccc(C)cc1C c1(OC)nc(C(=O)NCC2CN(C(=O)C=CC(C)C)C3CC23)cc(O)n1 c1(C(=O)NCCC2(O)CN(C(C3(CC)CC3(F)F)=O)C2)cc2[nH]nc(C)c2cn1 C1(F)(CNC(=O)C=CCn2cncn2)CCN(C(=O)CSCC2CCOC2=O)C1 Cc1nc(C)c(CCC(=O)NCC(C)(C)CC2CC2)c(O)n1.C(=O)(CCCC(F)F)N N1(C(C2CC(C)=C(C)CC2)=O)CCC(NC(C2CN(C)C2)=O)C(C)(C)C1 O=C(C(O)C1=CCCCC1)N1CC(C(N2CCCC23CCCCC3)=O)C(F)(F)C1 c12ccc(C)cc1CC(=O)N2.N1(C(CCN(CCC)C)=O)CCCC(C(=O)OC)C1 N1(C(=O)Cc2cnc(C3CC3)[nH]2)CCCC2CN(C(C3CCCO3)=O)CCC12 c1(C(N2CC(CNC(C(COC)COC)=O)C(O)C2)=O)sc2cccnc2c1Cl c1(C(=O)NC2CCOC(C(N3CCC(F)(F)CC3)=O)C2)nnc(O)nc1O C1(C(=O)NC2CC(NC(C3CC(C(=O)OC)C3)=O)C2)Cc2nn[nH]c2C(C)C1 C1(COC(Cc2cccc(OC)c2)=O)CC(C)(C)CC(C)(C)C1 Nc1cc(Cl)cc(Cl)c1C(N1CC2CCC1CN2C(C1CCCC12CC2)=O)=O N1(C(c2ccc(CO)o2)=O)CC2CCC2(C(=O)NC2CCC(F)(F)CC2)C1 CC(C)(C(c1nnnn1C1CCCCC1)NCC1CCC(=O)O1)c1ccncc1 c1(OC)cnccc1C(=O)NCCCCNC(C1CCC2(CC2)C1)=O c1ccc2oc3c(c2c1)CCCC3.O=CN=c1ccc(Cl)c(Cl)[nH]1 C1(C)(C(=O)NC2CC(CNC(Cc3c(C)cccn3)=O)C2)COC(C)(C)CO1 C1(CC(N2CC(c3cn(CCOC)nn3)(O)C2)=O)CCN(C)CC1 N#Cc1ccc(C(N2CCCCC2C(O)C(F)F)=O)cc1[N+](=O)[O-] c1(C(=O)NC2CN(C(C(C)CF)=O)CC(C)(C)C2)c2c(nn1C)CCSC2 C1(NC(COCC)=O)CN(C(=O)CC2CSCCO2)CC1C(F)(F)F C1(OC)CN(C(c2cnncc2C)=O)CC1C(N1CC(O)C1(C)C)=O c1(C(=O)NC(C)Cn2cc(-c3ncoc3C(=O)O)nn2)cnn(C)c1S(N)(=O)=O CS(=O)C=CC(=O)NCCOCCn1cc(CN)nn1.C1(C)CCCNC1=O n1(CC)nnc2c(N3CCN(C)C(CNC(C4(O)CCSC4)=O)C3)ncnc12 C=CCC(C(=O)N1CC(NC(=O)CCc2ccc(Cl)c(F)c2)C(C)C1)C(C)(C)C c1(C(=O)NC2CCC(NC(C34CC(CO3)C4)=O)C2)c[nH]c(=O)c2ccnn12 C1(NC(c2c(OC)c[nH]n2)=O)CC2(CCCN(C(c3ccc(O)nc3Cl)=O)C2)C1 CC1(CC(=O)NCC2(CNC(c3c[nH]cc3-c3ccc(Cl)s3)=O)CC2)CCCO1 C1(NC(CCC(=O)Nc2ccccn2)=O)CC2CC(C1)N(C(=O)OC(C)(C)C)C2 N1(C(c2cc(CC)oc2C)=O)CCCN(C(=O)CN2CCCC2C)CCC1 c1(OC)ccc(C(=O)NC2CC(C)N(C(C3CCCC(N(C)C)C3)=O)C2)nc1Cl N1(C(c2ccc(SC)o2)=O)CCN(C(=O)CC(F)F)C2CCCCC2C1 c1(OC)cc(C)c(C(=O)NC2CN(C(c3ccc(=N)[nH]n3)=O)C2)cc1Cl C1(C)(C(=O)NCC2(O)CN(C(c3c(COC)nn(C)c3)=O)C2)CCCCNC1=O C1(C)(C(=O)NC(CNC(C2(CC=C)CCCC2)=O)CO)CCN(C(=O)NC)C1 CC1(C)CC(CNC(C2CC(F)(CF)C2)=O)N(C(C2CCOC2(C)C)=O)C1 C(=O)(CC(C(F)(F)F)NC(=O)CCCNC(N)=O)N1CCN(CC)CC1C c1(C(N2C(C)(CC)CC(NC(c3cc(C)c[nH]3)=O)C2)=O)cc(S(N)(=O)=O)cs1 N1(C(CCC(=C)C)=O)CCC(NC(=O)C(C)OCCc2ccccc2)CC(O)C1 O=C1OCC2CN(CC(c3ccc(Cc4ccccc4)cc3)=O)CCC12 CC1(C)CCCOC1C(=O)NCCCC(=O)NCC1C2CCCCC12 C(=O)(CCC(=O)N(C)C)NC(C)C(CO)NC(C1CC(=O)N(O)C1)=O C1(NC(C2CCC2CF)=O)CN(C(c2ccc(CO)o2)=O)Cc2nccn2C1 C(=O)(CCCS(C)(=O)=O)NC(C)C(CO)NC(C1CC(n2cnnc2)C1)=O c1(NC(C(N2CCC(C)(CC#N)C2)=O)=O)cc(Br)c(F)cc1Cl CC1CCCCCCN1C(c1coc2c1CN(C(c1cn(C3CC3)nn1)=O)C2)=O C(=O)(C(C)(C)C(C)O)N1CCC(C)(CC(=O)NC(c2ccncc2F)C)C1 N(C(=NCC(F)(F)Cl)NCc1ccccc1)CC(C)(C)F c1(C(N2CCC(NC(COCCCC#C)=O)C(CC)C2)=O)ncnc2ccsc12 C1(NC(Cc2cccc(C)c2)=O)CN(C(c2ccc(Cl)c(O)c2)=O)CC1(F)F N(C1CN(C(=O)Cc2cccc(Cl)c2Cl)Cc2ccccc21)C(CSC)=O C(=O)(C#CC1CCCCC1)NCC(CNC(c1c(CC)con1)=O)CO C1(C(=O)N(C(CNC(c2snnc2C)=O)C2CC2)C)(COC)CCCCC1 CCC(C)C(=O)N(C)CCOCCN(C)C(c1cc(Br)no1)=O CC1CCC(CNC(=O)C=C2CCN(C)C2)N(C(=O)Cc2ccc(F)c(F)c2)C1 N1(C(c2c(CNC(c3ccc(CC)[nH]3)=O)nnn2C)=O)CC23CCC2(COC3)C1 C1(F)(CNC(c2n(CC)ccc2)=O)CCC(NC(=O)CCC2CCCO2)C1 C1(C)(CNC(C=Cc2n(C)cnc2)=O)COCCN(C(C2CCNC(=O)C2)=O)C1 c12nc(n(-c3ccc(OC)cc3)n1)C(C)O2.O(C(F)(F)F)CC N1(C(COC(CC)C)=O)CCC(C)(NC(c2ccsc2C(F)(F)F)=O)C1 c1(N(C(C(=O)NC(c2ncc(CC)o2)C)=O)CC)ccc(N2CCOC2=O)cc1 c1(C(=O)NC2CCN(C(C3CC4C=CC3C4)=O)CC2)ccn2ncnc2c1 C=CC(C)C(=O)NC(CSCC)C(=O)N1CCC(CF)C1 Cc1ncc2n1CCC(C(=O)NCC1CN(C(=O)C(=O)NC(C)C)CCC1N)C2 O=C1CN(Cc2ccccc2)C(=O)N1Cc1ccccc1.C1CCCN1CCO Cc1nc(CSCC(=O)N(C)CCNC(c2cn(-c3ccccc3)nn2)=O)cs1 CC1CC(NC(c2c(C3CCC3)cnn2C)=O)CN1C(=O)C(C1CCC(=O)N1)C N1(C(C(C2CCC2)OCC)=O)CCC(CN(C)C(C2(CSC)CC2)=O)CC1 c1(C(N2C(CC)CN(C(C3C(F)(F)C34CC4)=O)CC2)=O)cn2ccc(C)cc2n1 C1(O)(COC)CCN(C(=O)C(C2CCCO2)NC(=O)C=C(C)C)C1 Nc1cc(C(N2CC3CC3(NC(C34COCC3C4)=O)C2)=O)cc(O)c1Cl c1(C(N2CC(CN(C)C(C3CCCC3O)=O)C2)=O)cc(C(C)(C)C)no1 Cc1ccc2c(c1)C=C(C(=O)NC1CC1CNC(=O)CCCCC(N)=O)CO2 N1(C(CCc2cc(C)no2)=O)CCC(F)C(NC(c2ccc(F)c(Cl)c2)=O)C1 C1(CNC(C2(C(C)C)CC2)=O)CN2CCCCC2CN1C(=O)CC1(C)CC1 N1(C(C(C=C)(C)C)=O)CCC(NC(C2(C)CC(OC)CN2C)=O)C(C)C1 n1(CC(=O)NC(C2CCCN(C(c3cc(CO)on3)=O)C2)C)ncccc1=O C=CCC(CNC(=O)CC(Cl)Cl)C(=O)NC(CO)CCC(C)C C1(CNC(=O)C(F)n2ccnc2)C=CCOC1.C12(CCC1)C(=O)NCC2 C1(C(N(C(C)CNC(c2cccc(C(C)(C)C)c2)=O)C)=O)CCC2(C1)CC2(F)F N1(C(C2(CC(C)C)CC2)=O)CC=CC(NC(=O)C(C(C)C)N2CCCCC2)C1 c1(CC(=O)NC(C)CF)cccc(C(F)(F)F)c1.C12CC(C1)CNC2=O n1(CC)cnc2[nH]c(=NCC(C)CCCO)nc(N3CCc4nc[nH]c(=N)c4C3)c12 c1(C(N2C(C(C)(C)NC(C(CCCC)O)=O)CCC2)=O)cc2sccc2cn1 c1(C(=O)NCC(C)N(C)C(c2c[nH]nc2C(F)(F)F)=O)cccc(C2CCC2)c1 N1(C(CC(C)c2ccncc2)=O)CCN(C(c2ccn(C(F)F)n2)=O)CCC1C C=CCC(C(=O)NCc1cncc(OC)n1)NC(=O)Cn1[nH]cnc1=N Cc1c(C(=O)NCC(C)(O)CNC(=O)C(F)F)sc(Cl)c1Cl C1(C(=O)NCCCN(C(c2c(C)coc2)=O)C2CC2)CCCN(S(C)(=O)=O)C1 N1(C(C2CCN(C)C(=O)C2)=O)CCC2(CCCN2C(=O)C(Cl)=CCl)CC1 C1(C(=O)NC(CCC)(C)CC)CCC2(CC2)N1C(c1c[nH]nc1CC)=O Cc1cc(F)cc(CN2CCC(F)(C(=O)Nc3cc(C(N)=O)ccc3F)CC2)c1O N1(C(C2N(CC)CC2)=O)CCC2CCC(NC(c3cccc4[nH]ncc34)=O)C1C2 c1(NC(C2CCOCC2)CC)ccc(S(=O)(=O)NC(C)C(C)(C)OC)cc1Br C1(CNCc2nnc(CC)s2)COCC(C)O1 Cc1ccc(CC(=O)NC2CCN(CCC3CCCCC3(F)F)CC2)cc1C C(=O)(C1=CCCOCC1)N1CCC2C(C(N3C(C)CC(O)CC3)=O)C2C1 c1(C(=O)NC2(CC=C)CCN(C(=O)C=CC)C2)cc(OC)cc2c1OCC2 CCC(C)(C)C(O)C(=O)NC1(C(N2CCN(CC(C)O)CC2)=O)CCCC1 N1(C(CSSC)=O)CCC2(NC(c3cccc(Cl)c3)=O)CCCCCC12 C(=O)(C(O)CC(N)=O)NCC(=O)NC(CN(C(=O)Cc1ccc(F)nc1)CC)C C1(OC)CC(CF)N(C(=O)COC2(C)CN(C(=O)C=C3CCC(C)CC3)C2)C1 CCC(C(O)C(C)C)NC(C1CCN(c2ccccc2Cl)C1)=O Cc1cn2cccc(C(=O)NC3(C)CN(c4nc5ccc(N)cc5s4)C3)c2n1 c1(OC)c(Cl)ccc(C(=O)N(CCCNC(c2ccc([N+](=O)[O-])cc2)=O)C)c1F c1(NC(=O)Nc2c(C)cc(N3CCN(C)CC3)cc2)noc2cc(Cl)ccc12 CCC(CO)C(=O)N1CC(=C(F)CNC(C2CCCS2)=O)C1 C=C(C)C(C)(C)C(=O)NC(CNC(c1cnc(-c2ccccc2)o1)=O)CCCC c1(C(N2CCCC(N(C(=O)CN3CC4CC4C3)CC)C2)=O)cc2c(ccn2C)[nH]1 N1(C(CN(C(COC)=O)C)=O)CCN(C(c2snnc2C)=O)CC(C)(F)C1 C(=O)(C#CC1CCOCC1)N1CC(O)(C(C)NC(C2(C)CCCC2(F)F)=O)C1 c1(C(=O)NC(C(C)NC(c2c(C)nc(CC)s2)=O)C(C)C)c(N)cccc1F c1(C(N2CCC(N(C(C3N(C)CCOC3)=O)C)C2)=O)ncc(Cl)cc1O CCC(CC(=O)NC1(CCCC(=O)N(CCCOC)C)CCC1)SC Cc1nc(C(=O)N(C)CCC2CCCCN2C(C2CC=CCC2)=O)sc1C Cc1cccc(Br)c1C(C(=O)NCC1CC2CC1CC2=O)NC(=O)C(F)OCF C1(C(=O)Nc2scc(CC(=O)N(c3cn[nH]c3)CC)n2)CCOCC1(C)C c1(C(=O)NCC2CC(NC(C(C(C)(C)C)N(C)C)=O)C2)cc(F)c(C#N)c(F)c1 c1(OC)cc(NC(=O)C(C)(C)C)c(CNC(C2(C)C3CCCC23)=O)cc1OC C1(C)(NC(C(C)OC)=O)CCCN(C(c2ncn(C(C)(C)C)n2)=O)C1 S(=O)(=O)(c1cccnc1NCCCCC1CCCC1)NC(c1ncc(C)o1)C C(CC(=O)N(C(C)C(=O)OC)C(C)C)(CC(C)C)NC(C(COCC)C)=O C1(C2CC2)(C(=O)NC(CCCC)CC)CN(C(=O)C(CC2CC2)OC)C1 n1(CC(OCC)OCC)ccc2c(C(=O)N(CC(N)=O)C)cccc12 n1(CC(=O)OC)nc(C)c(=NCCc2cccc(C(=O)OC)c2)[nH]1 N1(C(c2c(C)[nH]nc2Cl)=O)CC2(C1)CN(C(C1CCCC1C(F)(F)F)=O)CCO2 c1(N(C)CCOC(F)F)nc(N2CCC(Cc3ccccc3)C2)c2sccc2n1 CC(O)CCCCCC(=O)N(CC(O)CN(C)C(c1ccc2c(n1)CCC2)=O)C c1(C(=O)NC2CN(C(=O)C=CBr)CC23CC3)cccc2[nH]cc(Cl)c12 c1(C(=O)NCC2N(C(c3c(C)nc(C)o3)=O)CCCC2)cncc(C)c1Cl C=CCC(CC(=O)N(C1CCOC(C)(C)C1)C)NC(=O)C(C)CC1CCC1 C1(C(=O)NCCN(C)C)CC12CCN(C(=O)C(c1ccccc1)O)CC2 C1(C(=O)NC2CC(OCC(=O)N(C(CC)CO)C)C2)COC(=O)N1 c1(C(=O)NC2CCCC(NC(c3ncc(N(C)C)cn3)=O)C2)ncnc(O)c1F N1(C(CC2(COC)CCCC2)=O)CC2CCC1C1CN(C(=O)C(F)OC)CC21 N1(CCNC(C(C2CN(C(=O)C(C)C(F)F)C2)OC)=O)CCCCC1C c1(NC(CNC2(CC(=O)OC)CCCS(=O)(=O)C2)=O)ncnc2c1COC2 C(C(=O)NC1CCC(F)(F)CC1)(C(C)CC(C)(C)C)N(CCC=C)CC S(=O)(=O)(c1ccc(=NCCNS(=O)(=O)CC)[nH]c1)N1CC(C=C)OCC1 c1(C(C(=O)NC2CCOC2)N(CCF)CC)cccc(C(F)(F)F)c1F c1(C(=O)NCC(CNC(C2C(C(C)C)C2)=O)(C)C)ccccc1CCC(F)(F)F C1(NC(=O)C=Cc2ccc(F)cc2)CCN(C(c2ccc(Cl)o2)=O)CC12CCC2 C(=O)(CCCCC(F)F)N1CCC(CNC(C(C2CCCCC2)OC)=O)C1(C)C N1(C(CCC(=O)NCCC)=O)CCC(C(=O)NCCCc2cncnc2)C1(C)C c1(C(N2C(C)(C(=O)NCCC(CCC)O)CCC2)=O)cc(C)cc(O)n1 C(CC(=O)NCc1cnn(C)c1C)(C(F)(F)F)NC(c1cc(CC)sn1)=O CS(=O)(=O)c1nccc(N2CCC(O)(C(=O)Nc3c(Cl)ccnc3Br)C2)n1 Cc1cn2cc(C(=O)NCC3CCN3C(=O)C(C)SC(C)C)cc(C)c2n1 c1(N(C)C)ccccc1C(N1CC(OCC(=O)NC2CC(NC(N)=O)C2)C1)=O Cc1cnc2ccc(C(=O)NC3CC(NC(=O)CCC(C)S(C)(=O)=O)C3)cn12 C1(CCC)CCCCN1C(c1n[nH]cc1-c1ccc(C(=O)OCC)cn1)=O N1(C(CC2CCC(=O)C2)=O)CC2CCCC(NC(C34CCC(CC3)OC4)=O)C2C1 N1(C(C(C)SC)=O)CCC(F)(CNC(=O)C(C)NC(=O)C2CC2)C1 c1(SC)cccc(Br)c1CC(=O)NCC(C)(CC(C)C)NC(=O)C(C)O CC1(C)NC(=O)OC12CCN(C(c1cnc(CN)cn1)=O)CC2 CCCCC(O)C(=O)NC1CN(C(c2cc(N)ccc2SC)=O)CC1F c1(CC2CC(C)C2)cccc(Cl)c1.C1(=O)C(C)(C2CC2)N1C(=O)OC(C)(C)C Cc1ccc([N+](=O)[O-])c(C(=O)NCC(CNC(c2cnsc2)=O)CO)c1C CCCCC(C)CCC(=O)N1CCC(C(F)C(=O)N(C2CC(O)C2OC)CC)C1 CC1(C)CC(C)(C(N2CCCCC(F)(F)C2)=O)CN1C(=O)C1=NOCC1 Cc1nccc(C(=O)NC(C)C(C)NC(c2cnc(CC(C)C)[nH]2)=O)n1 C12(C(N3CCN(CCN(C)C(C4(C5CC5)CC4)=O)CC3)=O)CCCN1CC(O)C2 C(C)(CC(C)(C)CO)NC(CC1N(C(C(=Cc2cn[nH]c2)C)=O)CC(O)C1)=O N1(C(c2cc(C)nc(O)n2)=O)CCC2CCCN(C(=O)CCN3CCCC3)C2C1 C(=O)(CCCC(=O)N1CC2CC2(NC(=O)C(C)OCC(F)(F)F)C1)OCC N1(C(c2ccc(C(=O)OC3CCCCC3)cc2)C(=O)NC)CCC2(C1)CC(F)(F)C2 c1(CC)cc(C(N2CCN(C(=O)CC(O)CN(C)C)CC2C)=O)ccc1OC c1(CNc2c(OC)cccc2C(=O)OC)cc(C)c(F)c(F)c1 CCS(=O)c1ccccc1C(=O)NC(CCN(C)C(c1cc(Cl)cs1)=O)C(C)C N1(CCC(=O)N(C2CCN(C(C3CC(CC)(CC)C3)=O)C2)CC)CCCCC1C Cc1nc(Br)c(C(N2CCC(CO)(NC(=O)C(C)C3CC3)C2)=O)s1 N1(C(c2c(OC)oc(C)n2)=O)CCC(O)(CNC(c2cnc(SC)n2C)=O)CC1 CC1CN(C(=O)COCC2CC2)CC(CCNC(c2nn(C)nc2Br)=O)O1 Cc1cnc(F)cc1C(=O)NC(C)CCCCN C(CCCCCC1CC1)NC(=O)CC1CCC(NC(c2csnn2)=O)C1 c1(C(N(CC(=O)NCCCCC2CCCC2)CC)=O)sc(F)cc1C c12ccc(cc1C)[nH]c2=O.CCCCC(=O)NC1(CC(=O)C2CC2)CC1 S(=O)(=O)(c1ccc(NCC2CCC3(CCCC3)C2)c2cnccc12)NCC(=C)Br C=CC1CC(N=c2[nH]c3ccc(S(=O)(=O)N4CCC(F)(CSC)CC4)cc3s2)C1 C1(NC(c2cc(OC)ncn2)=O)CCN(C(=O)CSCC(=O)N(C)C)C1(C)C C=CC1CN(C(C2CCC(NC(c3coc(CO)c3)=O)CC2)=O)CC1O c1(C(N2CCC(O)(CNC(C3C(OCC)C3)=O)C2)=O)cc(-n2cccc2)ccn1 c1(SC)ccc2cc(C(=O)NCC3CC3CNC(c3csc(C#N)c3)=O)[nH]c2c1 CCC(C)C(O)C(C)C(=O)NCC1(CNC(c2cc(C)n(CC)n2)=O)CCC1 Cc1cccn(CC(N2CCC(NC(c3ccc(C(C)C)o3)=O)C(O)C2)=O)c1=O c1(C(C(=O)NCC=C)N(CC)Cc2cc(C)ccn2)ccc(Br)cc1OC CC#CCCCC(C(=O)Nc1ccccc1)N1CCCC1c1cc(C)cs1 c1(C(N2C(C3CCN(C(C(CC)SC)=O)CC3)CCCC2)=O)cc(Cl)c(C)cn1 c1(C(=O)NC(CC)(C)CNC(=O)CN2CCCC2)cccc(C(=O)OC)c1C CC(C)CCCCC(=O)N1CC(CC(=O)NC2C3CCCOC23)C(C)C1 c1(CC(=O)NCC(c2ccc(CC)c(O)c2)=O)cc(F)cc(F)c1Br C(CNC(c1cccnc1C)=O)(C(C)C(C)C)NC(CCn1ncc(C)c1)=O N1(C(CC2CC(=O)NC2=O)=O)C2CCC1C(CNC(c1cc(F)c[nH]1)=O)C2 c1(C(=O)NC(c2ccccc2)C(C)NC(=O)CNC=O)sccc1C#N CC1C(NC(c2cncc(N=[N+]=[N-])c2)=O)CC2CCC1N2C(c1nccn1C)=O C(=O)(CC(CNC(=O)CC(C)n1ccnc1)C1CCC1)N1CC(C)(CC)C1 C1(C(N2CC(C)C(C(N3CCOCC(O)C3)=O)C2)=O)CC2CC(=O)C1O2 N1(C(CC=C)=O)CC(NC(=O)C(C)CC)C(O)C1 c1(CC)ncc(Cl)c(C(=O)NC2CCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)CC2O)n1 C1(C(=O)NC(CNC(c2n(CC)nc(C)c2)=O)C(C)(C)C)CC2(C1)CC(C)C2 c1(CNC(Cc2ccc(C)cc2C)=O)ccc2c(c1)CN(C(=O)C=CS(C)=O)C2 C=CCN=c1[nH]cc(C(=O)NC2CN(C(=O)CSCC(N)=O)CC2C)s1 C1(C(N(CCCCNC(C(C)OCC2CC2)=O)C)=O)CCC(=O)N1C c1(OCC)nc(CNc2ccc(CCC(N3CCOCC3C)=O)[nH]2)ncc1C CCC(Cc1ccccc1)CC(=O)NC1CCN(CC2COC(C)(C)CO2)CC1 C1(C(N(CCCCNC(CSCC=C)=O)C)=O)CCCN(C(C2CCC2)=O)C1 C1(C(N2CCCC(CNC(CCc3cn(C)nc3)=O)C2)=O)CCCN2CCCC12 C(=O)(CCCC(C)(F)F)N1C(C(C)C)CN(C(C2CC=CCC2)=O)CC1 C1(NC(C(CC)(O)c2ccccc2)=O)CCN(C(=O)C2=COCC2)CC1(C)C C1(C)(C(N(CC(C)(C)CNC(c2csc3cncn23)=O)C)=O)CCCNS1(=O)=O C1(CNC(CCNS(CC)(=O)=O)=O)CN(C(c2cncc(COC)c2)=O)C2CC12 c1(C(N2CC(CNC(C(=O)NCC)=O)CC23CCC3)=O)cccc2ncc(C)n12 N1(C(C2N(C(CN3CCC(=O)CC3)=O)CCCCCC2)=O)CCOCC(C2CC2)C1 C=CCCC(F)(F)C(=O)NCC(C(=O)NC(CC1CC1)CC1CC1)N(C)C c1(C(=O)NC2(COC)CCN(C(=O)CC(C)SC)C2)ccc(Cl)c(Br)c1 C=CC1(NC(=O)C(CNC(c2cnoc2C(C)C)=O)N(C)C)CCC1 C1(NC(C(=O)N(CC)CC2COC(C)(C)OC2)=O)CS(=O)(=O)CC1C C1(N(C(=O)C(=O)NCC2CC2)CC)CCCN(C(=O)Cn2ncn(C)c2=O)C1 C12(C(=O)NCC3N(C(C(N4CCSCC4)C)=O)CC3)CCCC1(C(N)=O)C2 N1(C(C(CO)NC(C(C)C)=O)=O)CCC(CO)(CNC(=O)CCS(C)=O)CC1 c1(OCC)ccc(C(=O)NCCNC(c2cncc(C(N)=O)c2)=O)cc1Cl Cn1c(C(=O)NCC(C2CCCCC2)NC(=O)C(F)C2CC2)cc(Cl)c1Cl N1(C(c2nnc(C3CCOCC3)o2)=O)CC2CC(C1)C1CCCCN1C2 C1(C(C)C)CN(C(=O)CCF)CCC1NC(c1nocc1Cl)=O C1(NC(=O)CC2CCNC2=O)CCCCC1NC(C1(CCF)CC1)=O n1(CCC)nc(C)c(C(=O)NCCCN(C)C(c2nnn(C)c2C(F)F)=O)c1C N1(CCc2nc(-c3c(CCC)[nH]cc3)n(CCC(C)(C)C)n2)CC(C)CC(C)C1 c1(NC(C(c2cn(C)nc2)NC(C2CCCCC2)=O)=O)sccc1C#N c1(C(=O)NC2CCC(N(C(CCC(=O)N(C)C)=O)C)CC2)c(F)ccc(Cl)c1N c1(CNC(=O)C(O)C2CN(C(=O)CC3CCCSC3)C2)ncccn1 C1(CCNC(c2ccsc2)=O)CCCN(C(=O)COC2CCCC2)CC1 C(CCN=C(NC1CC(N(C)C)C1)NC1CCCC(C(C)C)C1)OCC C(=O)(C1CNC(=O)c2ccnn21)NCC1(O)CCCN(C(C(N)=O)=O)CC1 N1(C(C(c2cnn(C)c2)C)=O)CC2CC(O)C1C2NC(c1snc(O)c1Cl)=O CCCC(C)CC(=O)N1CCCC(N(C(=O)CCOCC)CC2CC2)C1 N1(C(c2cnc(C)nc2)=O)CC2(C1)CN(C(C1CC1(C)Br)=O)C2 O=C(C1=COCCC1)NC1CC(F)CN(C(c2cc(O)ncc2Br)=O)C1 N1(C(C=CC)=O)CC(NC(=O)C(C(C)C)OCC(C)C)C2(CC2)C1 c1(CCC)nc(C)c(NC(C2CCCC(C)C2)=O)o1 N(C(=NCCF)NCc1cc(F)cc(Cl)c1)CC1CC(CC)C1 Cc1c(Cl)cnn1CC(=O)NC1CC1CNC(=O)CCCc1cncs1 N1(C(C(CC(=C)C)OC)=O)CC2CC(C(=O)NC(CO)C(C)(C)C)C(C2)C1 C1(CNC(C2CCC(N(C)C)CC2)=O)COCCN(C(C2(C)CCNC2=O)=O)C1 c1(C(C(=O)NC(CSCC)C)N(C)C(C)=O)cn(C)nn1.C(C)(C)(C)O C1(OC)CC(NC(c2c[nH]nc2C2CCCO2)=O)CN(C(c2occc2C)=O)C1 C(=O)(C1=CC2CCCCCC12)NC1(CN(C(CSCCCC)=O)C)CC1 C(=O)(C(CN)C(C)(C)C)NC(C(=O)OC)CCSC(C)(C)C c1(C(N(CC(=O)NCC=C(C)C)C(C)C)=O)cc2ccccc2[nH]1 N1(C(COCCOC)=O)CCN(Cc2c(OC)ccnc2Cl)C(CO)C1 N1(C(C(C(=O)OC)OC)=O)CCc2ccccc2C1CNC(c1cscc1F)=O c1(C(=O)NC(C(=O)NCCc2n(CC)cnn2)Cc2cn[nH]c2)cncc(F)c1 c1(C(N2CC(NC(C(CSC)O)=O)C(C)(C)C2)=O)cc(N)c(C)c([N+](=O)[O-])c1 C=CCCCCC(=O)N1CCCC1(C(N1CCC(CC(N)=O)C1)=O)CC N1(CCC(=O)NCC#CCNC(C2C3CCC(=O)C23)=O)CCCCC1=O CCS(=O)(=O)c1cccc(CC(N2CCNCC2c2cccc(Cl)c2)=O)c1 C(=O)(C(O)CC(N)=O)N1C(C(=O)NC2C(OC)C(O)C2)CC1 N1(CC(C(C)NC(=O)OC(C)(C)C)O)CCCC2(CC=CCO2)C1 c1(C(N2CCC(C(C)NC(C3(N(C)C)CCC3)=O)CC2)=O)ccc([N+](=O)[O-])cc1F N1(C(CC(C=C)C)=O)CCN(C(=O)CN2CCCCCC2)CC(C)(C)C1 C(=O)(CCC(C)(C)O)NCC(C1CCCC1)NC(C(C=C)O)=O c1(C(=O)NC2C(NC(C(CC(C)(C)C)OC)=O)CC2)cccc2nn(C)cc12 c1(CC(=O)N(CCN(C(=O)CCc2cccn2C)CC)CC)cc(F)ccc1Cl c1(C(=O)NC(CNC(CC=CCCCCC)=O)CCOC)cc(O)ncc1F CCCCC(C)C(=O)NCC1(C)CCN(C(c2cnc(C3CC3)nc2O)=O)CC1 c1(C(=O)NCCC2N(C(C3CCC(=O)NC3)=O)CCC2)c(F)cc(F)cc1Cl C=CCC(CNC(c1nonc1N)=O)C(=O)N(C)Cc1ccns1 CN1C(=O)CCc2cc(CN3CCCC(NC4CCCCC4)C3)ccc21 CCC(CCCC(=O)N1CCC(CCOC(C)(C)C)C1)NC(=O)CC(=O)OC c1(CCSCC(=O)NC2(CN)CS(=O)(=O)C2)ccc(Cl)cc1Cl N1(C(C(CC=C)C)=O)CCC(C2CC2)(CNC(C23CCCN2CC(OC)C3)=O)C1 C1(NC(Cn2ncc(CC)c2)=O)CCN(C(=O)CCc2ccsc2)CC1CC O=C1Cc2ccc(C(=O)NC3CC4CCC(C3)N4)cc2N1 CCCCCCCCCC(=O)N1CCN(C(=O)C(O)CF)CC1CCC CC1CC(C(=O)NC(C)(C)CNC(c2cc(-c3cnn(C)c3)[nH]n2)=O)=NO1 c1(C(N2CCC(NC(=N)Cc3nc[nH]n3)C2)C(=O)NCC)ccc(CC)nc1 c1(C(N2CC(F)CC(NC(CC3CCN(C)C3)=O)C2)=O)cnn2ccccc12 c1(C(=O)NCCN(C2CC2)CC2CC2)cscc1C(=O)O N1(C(c2c(CC)ccs2)=O)CC2CN(C(C3(F)CCC(=O)CC3)=O)CC2C1 c1(C(C(=O)NCCCN(C)C(C2CCCC2CF)=O)(C)C)ccc(Cl)cn1 c1(C(=O)NC(=O)C(C)Cn2cccn2)cn(CCCCNC(CCOC)=O)nn1 C(=O)(CC(C(F)(F)F)NC(=O)C=Cc1cncs1)NCCC(C)N1CCCC1 Cc1nc2c(F)cccc2cc1C(=O)NC1(C2CN(C(C3CCCO3)=O)C2)CC1 N1(C(C2(CC#C)CCCC2)=O)CCCCC(CNC(=O)CC2CC=CCC2)C1 Cc1ccn2ncc(C(N3CC4=C(C3)CN(C(=O)C(C)C3CCOC3)C4)=O)c2n1 c1(CC)cc(C(=O)NCCN(C(=O)CCC2CCC(O)CC2)C)nn1C C(=O)(C1=NOC(CC2(O)COC2)C1)N1C2(CNC(C#CC(C)C)=O)CC(C1)C2 c1(CN(CCC(C)F)CC(=O)O)ccc(CCC(C)N)cc1 CC(C)(C)C(CC(=O)NCC1OC(=O)NC1(C)C)NC(c1c[nH]c(C(N)=O)c1)=O N1(C(c2c(=O)ccn(C)c2)=O)CC(CNC(C2CC3CCC2C3)=O)CC12CCC2 CCC(C)C(CC(=O)NCCN1CCC(CO)C1)NC(c1ccnc(CO)c1)=O c1(COC)cc(C(N2CCCCC2CCNC(c2ccnnc2O)=O)=O)n(C)c1 c1(CNC(CC(CC)NC(c2ccc(Cl)s2)=O)=O)cc(F)ccc1F C(N=c1[nH]cnc(Cl)c1COCCO)C1OCCCN(C(C#CC2(C)CC2)=O)C1 c1(C(=O)NCC2C3CN(C(C(CCC)C)=O)CC32)cc(O)cc(Br)c1 CN1N=C(C(=O)N2CCC(F)(CNC(c3cccc4c3OCC4)=O)C2)CCC1=O CS(C)(=O)=NCC(=O)NCC(C1CCCC1)Nc1nc(CC2CC2)ns1 O=C(N=c1cc[nH]cc1O)C1CN(C(c2cc(F)c[nH]2)=O)CCC1O C1(NC(CC(CC)C2CCC2)=O)C2CC1CN(C(=O)CC1(C)CCS(=O)(=O)N1)C2 c1(C(=O)NCC2CC(O)(CNC(C(CC)=CC)=O)C2)cccc(NC(C)C)c1 c1(CC)ncc(C(=O)NCC(c2ccccc2)CNC(=O)C(O)CSC)o1 Cc1c(C(N2CC(CNC(c3ccc(C(N)=O)cn3)=O)C(C)C2)=O)nnn1C c1(CCC(N2CCC(F)(CNC(C3(N(C)C)CC3)=O)C2)=O)ccc(Cl)c(F)c1 CC(C(C)C(=O)N(C)Cc1nccs1)NC(=O)CCC1CCCOC1 CCCCCC(C)CC(=O)NCC1(O)CC(NC(=O)CCCCC(=O)OC)C1 C12(NC(Cc3nc(C)[nH]n3)=O)CCN(C(c3ccc(F)cc3Cl)=O)CCC1C2 Cc1cc(O)ccc1N(C(=O)CC=CCNC(=O)C=CC(C)(C)C)C CC1CCc2[nH]nc(CNC(=O)NC3(CO)CCN(C(=O)OC(C)(C)C)C3)c2C1 N1(C(c2cc(C(C)=O)oc2)=O)CCOC(CNC(C2(CN(C)C)CCCO2)=O)C1 C1(CC)CCCCC1OCC(=O)NC(C)(C)CNC(c1coc(C)n1)=O N1(C(C=C)=O)CCC2CCC(NC(c3cc(C(F)F)cc(Cl)c3)=O)C1C2 N1(C(C2(CC=C)CCCC2)=O)CC2CN(C(c3cc(Br)ccc3F)=O)CC2C1 C(F)(F)(C(F)(F)F)c1scc(C(c2n(CCOC)nnn2)NCCC(C)(C)C)c1 c1(CC(=O)N(C(C)CCNC(=O)C#CC2CCC2)C)cc2ccccc2oc1=O N1(C(C2CC(SC)C2)=O)CCCC(C)C1CNC(c1cc(C)ccc1C)=O c1(C(=O)NC(CNC(CC2(C=C)CC2)=O)(C)C2CC2)cnn(C(C)C)n1 N1(C(C2(OC)CCC2)=O)CC(N(C(=O)C=Cc2ccc(SC)cc2)C)C(C)(C)C1 c1(C(N2CCC(C(=O)Nc3c(OC)c(F)ccc3)C2)=O)cc(C)cc2[nH]ccc12 C1(NC(Cc2cccc(C)c2Cl)=O)COC2(C1)CN(C(C1CC3C=CC1O3)=O)C2 c1(C(=O)O)cc(CN2CCC(O)CC23CCC3)c2sc3ccccc3n12 C12(NC(C(C)C3CC3)=O)CCCN(C(c3ccccn3)=O)C1C2 c1(CSC)ccc(C(=O)N(C)CCNC(c2cnccc2C(F)F)=O)cc1 c1(C2(N(S(C)(=O)=O)C(CC(C)C)=O)CC2)ccc(Br)cn1.C12(O)CN(C1)C2=O c1(C(=O)NCCCCCN(C(CC2CCC(C)C2)=O)C)ccc2[nH]c(=N)[nH]c2c1 C1(C(N(CCNC(C(C)OCC#C)=O)CCOCCO)=O)CCC(C(F)(F)F)CC1 c1(C(=O)NCC(CC)NC(=O)C(CC(C)C)OC)[nH]c2cc(F)ccc2c1C N1(C(C2(N(C(C(CC)CN(C)C)=O)C)CC2)=O)CCn2nccc2C1 CC1CCN(C(c2c(F)cccc2Cl)=O)CC1CNC(C1CC(C(F)(F)F)C1)=O C1(C(=O)NC(C)C=CC(=O)NC2(CO)CCC2)CNC(=O)CC12CCC2 C1(CNC(CCN(C(C)=O)C)=O)CC2CC2N1C(c1ccsc1C)=O CN1CCC(C(=O)NCC2CCCN(C(=O)C(C)(C)F)C2)S1(=O)=O C1(C)(NC(C(N2CCC(O)CC2)C)=O)CCN(C(=O)CCc2cncn2C)CC1 N1(C(C(C=C)O)=O)CC2CC1C2C(=O)NC(CO)CCC1CC1 C(C)(CNC(C1CCCN1C(=O)CCCON)=O)(CO)OC c1(C(=O)NC2(CC)CCCN(C(c3coc(Br)c3)=O)C2)cccc2nncn12 N1(C(=O)OC(C)C)CCC(C2CC2(F)F)C1.c12cc(ncn1)NC1CCN2CC1 c1(C(=O)NC2C(Cn3cc(CSC)nn3)CCC2)ccc(Cn2cccc2)cc1 C1(CNC(c2cncc(N)c2)=O)CC2(CCN(C(C3CC3Cl)=O)CC2)CO1 C(=O)(C1=C(C)OCCS1)NCCCC(C)NC(C(C)OCCC=C)=O c1(CC)nc(C)c(C(=O)NCCCN(C(=O)CN2CC3CC3C2)CCSC)o1 N1(C(c2ccc(CC)s2)=O)CC(C2CCN(C(C3(c4ccsc4)CC3)=O)CC2)C1 N1(c2ncnc(NCCCn3ncc(C)c3)c2C)CCc2nccc(N)c2C1 c1(C(=O)NC(C)(C)CNC(C2(O)CCCCCC2)=O)ccc(P(C)(C)=O)s1 C(=O)(CCCCC(=O)OC(C)(C)C)N1CC(NC(c2ccc(C(C)=O)cc2)=O)C1 c1(NC(C(C(=O)OCC)(CC)CC)=O)cc(S(N)(=O)=O)c(Cl)cc1Cl C1(NC(c2ccc(F)o2)=O)CCN(C(c2cnc(S)n2C2CC2)=O)CC1F c1(SC(C(=O)NCCCNC(CCc2ccc(CC)s2)=O)C)ccc(F)cc1 Cc1cc(CNC(=O)C(C2CCCCC2)O)oc1C(=O)NC1(CCF)CCC1 c1(C(=O)NC(C)CN(C)C(C2CCC(=O)C2)=O)cc(F)cc2ccncc12 C(=O)(CC(O)C(C)C)N1CC(OCC)C(NC(C2(Sc3ccoc3)CCC2)=O)C1 N1(C2CCCC(CC)CC2)CCC2(CC1)OCC(O)C2O c1(C(=O)NC(CCCCNC(C2CC(SC)C2)=O)C)cncc2ncn(C)c12 N1(C(C(c2cn(C)nc2)=O)=O)CCC2(CC(C(=O)N)C2)C1.N1(CC)CCC(O)C1 N1(C(=O)CC2CC(=C3CC3)C2)CC2CCN(C(C3COCCC3(F)F)=O)CC2C1 C1(NC(c2ccc(CCC)[nH]2)=O)CN(C(=O)C(C)(O)CCC)CCC12CCC2 N1(C(c2c(C)nccc2Cl)=O)CCCN(C(=O)Cc2csc(=N)[nH]2)C(CO)C1 Cc1ccc(S(=O)(=O)Nc2cccc(NCCC(=O)Nc3nccs3)c2)c(F)c1 CC1(CNC(C2CCCS(=O)(=O)C2)=O)COCCN(C(c2cccnc2N)=O)C1 c1(C(=O)NCC2(O)CCN(C(C(C)c3cccs3)=O)C2)ccc(Cl)c(Cl)n1 C1(CNC(=O)CC2CCC(=O)O2)CC2CCC1N(C(c1c[nH]cc1Br)=O)C2 CN1CCCC1CCNC(c1n[nH]cc1CNC(c1scnc1Cl)=O)=O N1(C(C(C(=O)OC)C)=O)CCCC(O)(C(=O)NCCC2(COC)CCC2)C1 O=C(C1=CCOCC1)NC1COCC1CNC(c1ccc(Cl)c(Cl)c1)=O C(=O)(C(CC(C)SC)N1CCCC(C)(CC)C1)NCC(=C)C C(=O)(C(F)(CNC(=O)C1=CCCCCC1)C(C)C)N(C)Cc1onc(CC)n1 c1(C(=O)NCC2(NC(C(CC#C)O)=O)CC2)cc2c(s1)CCC(C)C2 c1(CC(C(=O)NC2C(CNC(COCC(C)C)=O)COC2)O)ccc(F)cc1 C1(COC(C2(C(C)=O)CC2)=O)CCCC2(CCC2)O1 C1(F)(CNC(c2cnc(SC)[nH]2)=O)CCC(NC(C2CCCCS2)=O)C1 C(=O)(C1(C)CCn2ccnc21)NC(COC)CC(=O)N1CCC1CF C(C)(N=c1nc2sccc2c(N2CCC(C(F)F)CC2)[nH]1)c1c(C)cccc1 N1(C(CC2(OC)CCC2)=O)CCCC(NC(c2cc(C(C)=O)[nH]n2)=O)CC1 CC1CSCCN1C(=O)NCCC1OCCC1(C)C N1(C(C2(OCC)CCC2)=O)CCCC(O)(CN(C)C(c2cccc(N)c2F)=O)C1 C(=O)(CCC(N)=O)NC(c1cccc(Cl)c1)CNC(c1c(OC)n[nH]c1)=O CC1(C#CC(=O)NCCC2(C)CCN(C(c3cccc(F)c3O)=O)C2)CCCO1 C(=O)(C(C)C(=O)N(C)CC1CCN(C(=O)CCN(CC(C)C(C)C)C)CC1)OC C1(C(=O)NC(C#C)CO)CCn2cncc2C1 c1(CC(=O)NCC2CN(C(CC(=C)Br)=O)C(C)C2)ccccc1[N+](=O)[O-] C=C(Cl)CCC(=O)N1CC2CC1C2NC(=O)Cc1csc(C2CC2)n1 c1(C(N2CCc3cccc(Cl)c32)C(=O)N)csc2ccc(Cl)cc12.C1(C2C3CCCCCCC3C2)CCC1 c1(C(=O)NCC2N(C(C(C)NC(C)=O)=O)CC3(CC3)C2)c(Cl)cccc1[N+](=O)[O-] C1(N(C(CCCC)C)C)CCN(C(=O)CCC2CCOC2)CC1C Cc1cc(N)cc(C(N2CCC(NCCO)CC2)=O)c1F c1(CC(N2C(CC)CN(C(=O)C3CC3)CC2)=O)[nH]nc2c(Cl)cccc12 N1(C(CCCn2cc(C3N(C)CCC3)nn2)=O)CCC12CCN(C)C2 C(C1=CCN(C(c2c(CO)n[nH]c2C)=O)CC1)NC(C(C(C)C)SC)=O N1(C(CC)=O)CCCC1CNC(C12CC(C)C1C2)=O C(=O)(C1=COCCC1)NCC1CC(NC(=O)CSC2CCCCO2)C1 c1(C(N2CC(CCCNC(COCC)=O)OCC2)=O)cnc2[nH]c(C)nc2c1 C(CC(CNC(c1cccn1C)=O)NC(=O)CCOC1CCOC1)OC C1(NC(c2ccc(C(N)=O)cn2)=O)CCCCN(C(c2ccnn2C2CC2)=O)C1 N1(C(Cc2c(C)scc2)=O)CCC(NC(=O)C(O)Cc2cnc[nH]2)C(C)C1 C1(OC)CCCC(NC(c2c(Cl)cn(CCC)n2)=O)(OC)C1 C1(NC(c2cn(CC)nn2)=O)CC2CC(NC(c3ccc(CC4CC4)cn3)=O)CC12 CN=S(C)(=O)c1ccc(C(=O)NCC(C)N(C)C(c2ocnc2C)=O)cc1 C1(CNC(CCN(C)C)=O)CCCCN(C(=O)C(C)(C)CC2CC2)C1 c1(OC)ccc(F)nc1NC(C1CC(OC)CN1c1nc(C#N)cs1)=O C1(COC)(NC(c2ccn(CO)c2C)=O)CCCN(C(=O)CN2CC3CC3C2)C1 N1(C(c2c(OCC)ccs2)=O)CC2C(C(=O)Nc3cncnc3O)C2C1 C1(C)(CC(=O)NCCc2nc(C)[nH]n2)CCCN1C(=O)CC1CCCCC1 Cc1nc(C(=O)N(C(C)CNC(c2c(-c3ccccn3)noc2C)=O)C)c(C)o1 C1(NC(CSC)=O)CCSC12CN(C(=O)C(C)Cc1ccc(F)cc1)C2 C=CCCC(C(=O)OC)NC(=O)C(CC)NC(c1nscc1C)=O c1(C(=O)NCCC2OCCN(C(C3C(C)(C)CCC3)=O)C2)cc(Cl)cc(Cl)c1F FC1(F)CCN(C(=NCCc2ccccn2)NCC2CCCSC2)C1 N1(Cc2c(C)cc(C)[nH]2)Cc2ccc(O)cc2CC1C(N1CCC(F)C1)=O c1(OC)c(Cl)cc(NC(=O)Nc2cn(C)nc2C(F)(F)F)cc1Cl c1(COC)cc(NC(=O)NC(C)Cc2cccc(O)c2)ccc1F c1(OC)ccc(C(=O)NCC2(OC)CCN(C(=O)CC3CC(C)(C)C3)C2)c(Cl)c1 N1(C(C(C)CC2CCC2)=O)CC2(CCCC2)C1C(N1CCN(CCO)C(=O)C1)=O C(C(O)C(=O)NCC1CC1CO)NC(c1cc(Cl)ns1)=O C1(CNC(c2c(C)ccnn2)=O)CN(C(c2coc(C(F)(F)F)c2)=O)CCC1C C1(NCC(c2c(C)n(C(C)C)cc2)=O)CCCC(F)(F)C1O C1(C(N2CCC(OCC#C)C2)=O)CCCN(C(C2(C)CSC2)=O)CC1 c1(CC(=O)NCCC2(O)CN(C(CCC(C)OC)=O)C2)coc2ccc(C)cc12 c1(NC(c2cncc(Nc3cc(OC)ncn3)c2)=O)c(Cl)nc(SC)nc1Cl C1(C(N2C(C(=O)NCC(N(C)C)C3CC3)CCC2)=O)CCCC(=O)C1 N1(C(C2CCC=CCC2)=O)CCN(C(=O)CC2C=CCC2)C(CCO)C1 Cc1csc(CC(=O)C(CC2C3CCOC3C(=O)N(C)C2)=O)c1.c1(CCN)cc(C)on1 N1(C(C=CC=CC)=O)CC2CCN(C(c3ccc(Br)c(OC)c3)=O)CC2C1 CCC(O)C(F)(F)C(=O)N1CC(CNC(c2cc(Br)nn2C)=O)C(O)C1 N1(C(c2cc(Cl)nn2C)C(=O)NCCOC)CCN(C)C2CC12 N1(C(C2CCN(C(c3c(C)nns3)=O)C(C)C2)=O)CCC12CCOCC2 N1(C(CC2CC(=C)C2)=O)CC(C)(C)CC1C(N1CC(CO)(OC)C1)=O N1(C(C2C(COC)CC2)=O)CCC2CC12C(=O)NCC1CCOC1C CCC(CNC(C1CC1(F)Cl)=O)(CC)NC(c1cncn1C)=O C1(C(=O)Nc2cc(C(C)(C)C)no2)CC12CCN(C(C1CC1(F)F)=O)CC2 c1(NC(=O)NC(C)CCCOc2cccnc2)cnc2ccnn2c1 Cn1cc(SC=CC(=O)N2CC(NC(C3CN(C(=O)OC(C)(C)C)C3)=O)C2)cn1 CC(C)(CC(=O)NC1CCC1NC(c1c[nH]nc1C(C)(F)F)=O)CC(F)F C=C(C)CC(C)C(=O)N1CCCC(CNC(=O)CCCOc2ccccc2F)C1 c1(CN2CC(C(=O)Nc3cnc(I)cn3)C(O)CC2)c(O)ccc2ccccc12 C1(C(C)(C)C)CC(CNC(=O)CP(C)(C)=O)CN(C(c2cncn2C)=O)C1 c1(C(N(CC(C)NC(c2c[nH]nc2C(F)F)=O)C)=O)cc(CO)ccc1Cl N1(C(c2cccc(OC)c2)=O)CCCC(F)(CNC(=O)CN(C)S(N)(=O)=O)C1 c1(OCC)c(OC)cc(C(=O)NCCC(C)NC(C23CC(C)(C2)C3)=O)cc1Cl C(C(C)(C)C(=O)NC1CCOCC1NC(=O)CC1CNC(=O)O1)SC N1(C(c2c(COC)n(C)nc2)=O)CC2CCN(C(=O)Cc3cc(C)no3)C2C1 CCN=C(NCC12CC(C1)C(C)O2)NC1CC1(c1ccccc1)F N1(C(c2c(C)nsc2)=O)CCC(O)(CNC(=O)CC2CCC(=O)N2)C1 c1(Cn2c(C(CC)(COC)NC(C(C)C)c3cncs3)nnn2)ccc(C#N)cc1 C1(CNC(c2c(C)scc2)=O)CC2CCC1N(C(=O)CNC(=O)NC1CC1)C2 c1(C(N2CCC(O)(C(C)C)C2)C(=O)NC2COC2)cccc2sccc12 c1(C(=O)NCC(CN(C(CC(=O)OCC)=O)C)C)cc2n(n1)CCN(C)C2 C1(NC(CN(C(C=C(C)C(C)(C)C)=O)CCN(C)C2CC2)=O)CCCCC1C C(=O)(C(C)(CNC(=O)C(C)SC(C)C)CC)NC(CCC)CO C(c1ccncc1)=CC(=O)NC(CC(=O)NCC1(O)CN(C)C1)C1CC1 c1(CNCC2N(C(c3cncs3)=O)CCOC2)ccc2c(c1)Cc1ccccc1-2 C(=O)(CCCCCCNC(C1CC1CCOC)=O)N(CC(=O)NCCC)C Cc1cn(CC(=O)NC2CCN(C(c3cnc(S)[nH]3)=O)C2(C)C)c2ccccc12 c1(C(=O)NCCCCN(C)C(C2CC=CCC2)=O)cncnc1-c1ccccc1 C1(NC(c2c(COC)ccs2)=O)CCN(C(=O)C(=Cc2c[nH]cn2)F)C1(C)C C(=O)(C1=CCC(C)CC1)NCCOCCCNC(c1c(C)cccc1)=O c1(C(=O)NCC(CNC(C2CC2CF)=O)OC)c[nH]nc1-c1ccoc1 c1(OC)cc(C(=O)NCC2(NC(C3CCC(=O)N3)=O)CCCC2)ccc1F Cc1c(N(C(=O)COC(C2(C#N)CCOC2)=O)C2CC2)cccc1Cl N1(C(C=CC(=O)OC(C)(C)C)=O)CCC(NC(C2CC2(C)C)=O)C(C)(C)C1 CCCC(Cl)C(=O)N1CCC(CC(=O)NCCc2cnn(C)c2)CC1 C1(S(C)(=O)=O)(C(N2CC(C(C)NC(C(CC=C)N(C)C)=O)OCC2)=O)CCC1 Nc1nc(C(=O)NC2CC(NC(=O)CC3CCCOCC3)C2)ccc1O N1(N2CCC3C(C)(CO)C3C2)CC2(CC(CO)CO2)C1.c1(C=O)ccccc1C N1(C(c2cc(CCC)[nH]n2)=O)CCC(C)C1CNC(c1coc(C)c1)=O Cc1ccnc(C(=O)NC2CCC2CNC(c2c(C)c[nH]c2CC(N)=O)=O)n1 c1(C(N2CC(C)C(NC(C3(c4cccnc4)CCC3)=O)C2)=O)cnc2n1CCC2 C1(CC(=O)NCC(CC)(CC)NC(C(CC)F)=O)CCCCC1(F)F Cc1cc(F)c(NC(=O)C(=O)NCC(C)CSc2ccccc2)c(I)c1 CCC1=NOC(CC(N2CCN(C3CN(C(=O)Cn4nnc(=N)[nH]4)C3)CC2)=O)C1 C1(C#N)(CC(=O)NCCC(C)N(CCC)C)CCOCC1 Cc1c(NC(C2CC2c2cccnc2)=O)n[nH]c1C1CC1 C1(C(=O)Nc2c(C)c(F)ccc2)COC2(CCN(C(C3(F)CCC3)=O)CC2)C1 C(=O)(CC1=NN(C)C(=O)C1)NC1C(C=C)CN(C(C2(c3cccnc3)CC2)=O)C1 CC#CCCC(=O)NCC(C1CCCN(C(c2cc(Cl)no2)=O)C1)(C)O C#CCCCCCCC(=O)NCCCC(O)C(=O)NCC1(OC(C)C)CCC1 C1(NC(c2[nH]nc(OC)c2Cl)=O)CCN(C(c2ncsc2C(C)C)=O)C(C)C1 C1(C(F)(F)F)(C(=O)NC2CN(C(c3cnc[nH]3)=O)CC2O)CC2CCC1C2 Cc1ccc(F)nc1NC(=O)N(C)Cc1nc(-c2ccco2)n[nH]1 N1(C(=O)CC2CCCCCCC2)CCC2CCN(C(=O)CCc3nncs3)C2C1 C(=O)(CS(=O)(=O)CC(C)C)N1CCC(OCCNC(c2n[nH]c(C)c2C)=O)C1 Cc1csc2c(C(N3CC(C)(NC(=O)CC4CCCC45CC5)C3)=O)ncnc12 C1(NC(=O)CC2CC2)CCN(C(c2cnc(C3CC3)nc2O)=O)CCC1CO Cc1cc(C)c(C(N2CCC(NC(c3nncn3C)=O)C(F)C2)=O)c(=O)o1 C(=O)(C(O)C(F)(F)F)NCCN(CCOC)C(c1cc(C(F)(F)F)n[nH]1)=O N1(C(=O)Cc2cccnc2Cl)CC(CNC(=O)C(O)CC2CC2)C2(CC2)C1 c1(OC)ccccc1C(N1CCC(C)(NC(C2CC2(Cl)Cl)=O)C1)=O N1(C(C(C)C2CCCO2)=O)CCC2(CC1)CCN(Cc1ccn(C)n1)C2 N1(C(CCCC)=O)CCN(C(C2(N3CCCC3)CCC2)=O)CC1COC Cc1nc(N)cnc1C(=O)NCC1CCCCN1C(c1cc(C(C)C)n(C)n1)=O c1(SC)cc(C(=O)NCC(C(C)C)NC(C2CC3(CC3)CO2)=O)c(Cl)cc1Cl CCC(CC(=O)NCCN1CCN(C(C2CCCCNC2=O)=O)CC1)C(C)C N1(C(CC2CN(C(CCC(C)OCC)=O)CC23CC3)=O)CCN2CCCCC1C2 CC1(C)CC(CNC(c2ccc[n+]([O-])c2)=O)CN1C(c1cnn2c1SCC2)=O Cc1ccc(C(N2CCCC2C2CCN(C(c3csc(Cl)c3)=O)C2)=O)nc1 C1(CC(N2CCC(CCNC(C3(C4CCC4)CC3)=O)C2)=O)CCC2(CC1)CC2 c1(C(N2CCC(C(C)NC(c3n[nH]cc3Cl)=O)C2)=O)ncsc1S(N)(=O)=O n1(CC(C)CO)nc(-c2cccc(OC(C)(C)C)n2)nc1C(C)CO c1(C(N(C2CC(NC(Cc3ccc(C)o3)=O)C2)C)=O)cnn(C)c1N C1(C(=O)NCCC2(O)CCN(C(c3n(CC#N)ncc3)=O)C2)CCC(F)(F)CC1 CN1N=CC(CC(=O)NCC(C)(C)C(=O)NCC2CC(C)(O)C2)C1=O C(=O)(CCCCCN1CC(C(=O)OC)CC1=O)NC(CC)CNc1cc(C)ncn1 C1(NC(CCC=CC)=O)CS(=O)(=O)CC1NC(c1cccc(Cl)c1)=O c1(C(=O)NCc2cc(C(=O)NCC3(OC)CCCC3)sc2)ccc(OC)nn1 c1(C(=O)NC2C(NC(CNS(N)(=O)=O)=O)CCC2)ncn2ccccc12 Cc1cc(Cl)ccc1C(=O)NC1CN(C(c2cc(Cl)on2)=O)CCC1C c1(C(=O)NC2CCN(C(C(CSC)(C)C)=O)CC2C(N)=O)cccc2c1OCC2 C(CNC(C1CCCC(O)C1)=O)(C(C)(C)C)NC(c1[nH]cc(C(C)=O)c1)=O C(=O)(CN=c1[nH]c2c(c(=NCCc3cncc(Br)c3)[nH]1)CCCCC2)N(C)C C(=O)(C1CCCc2nncn21)N(C)CC1CN(C(=O)CCn2cnnn2)CCO1 c1(NC(=O)NC(C2CCN(C(=O)CC(=O)OC(C)(C)C)C2)C)ccc(F)cc1Cl CON1CCC(C(N2CCC(O)(C(C)NC(=O)C(=CC3CCCC3)C)C2)=O)CC1 Cc1cc(C=CC(=O)NC(C)CN(C)C(C2CCC3(CC2)CC3)=O)c[nH]c1=N c1(OC)cc(=O)n(C)cc1C(=O)N(C)CC1CCCN(C(=O)C(C)=C(C)C)C1 N1(C(c2c(NC(C)=O)c[nH]c2C)=O)CC2CN(C(=O)CC(C)(C)O)CC2(C)C1 C(C)(C)(CC(=O)NCc1nc(CNC(=O)CC2CC(OC)C2)cs1)OC c1(NC(CC)CNC(=O)C=Cc2cnc[nH]2)nc(Cl)nc2c1ncn2CC C1(NC(C2C(OC)CC2)=O)CC2CCC(C1)N2C(=O)CCSc1cccc(C)c1 CC(O)(CNC(c1coc(CNC(=O)C(F)OC(F)(F)F)n1)=O)C(F)F c1(C(=O)NC2C3CN(C(CCc4ccn(C)c4)=O)C2C3)ccc(F)c(CO)c1 C1(C(=O)Nc2[nH]c(=N)sc2)CCCOC1C1CCN(C(=O)COc2ccon2)C1 C12(C(=O)NCc3cc(C)cc(O)c3)CCCC1CN(C(c1cnc(C)n1C)=O)C2 Cc1cccnc1C(N)C(N1CCOC(CF)C1)=O c1(OC)cc(C)c(COC(=O)Nc2ccc3n[nH]cc3c2)cc1OC C=C(Cl)C(C)(C)C(=O)N1CCCC(NC(=O)C(F)(F)C(C)O)C1 c12cc(Cl)ccc1O2.C1(C(N(C(=O)COC(F)F)CC)C)CCCOC1 C1(N2CCN(c3c(SC)cccc3)CC2)CCC2CN(C)CC12 Cc1ccc(C(=O)NCCOC2CCN(C(C3CC(=O)CO3)=O)C2)n1C c1(C(=O)NCCN(C(CC=C)=O)CCCN(C)C)cc(Cl)cc([N+](=O)[O-])c1O c1(OCC(=O)NCCCN(C(c2c(C(C)C)cnn2C)=O)C)nc(O)nc(O)n1 C1(NC(CCC#C)=O)CC2CC(C1)N(C(=O)C(CC(F)F)c1ccccc1)C2 Cc1cc(C#N)cnc1C(N1CCC(C2CCCN2C(=O)C=C2CCC2)CC1)=O N1(C(C2CCC(CC)O2)=O)CCCC(C)C1CCNc1ncc(F)cn1 CC(CS(C)=O)C(=O)NCCCC1(NC(=O)CCc2ccccc2)CC1 Cc1nc(C2CCOC2)sc1C(=O)NC1CCN(C(=O)CC#N)C1 c1(C(=O)NCC2C3CN(C(C4(C)CCCCC4)=O)CC32)cnn2c1CCC2 N1(C(C)C(=O)NC(CC(=O)Nc2cccs2)C2CC2)CCC(O)CC1 c1(C(c2nnnn2C)NCCNC(C(C)C)=O)cccc(C(F)(F)F)c1F c1(C(N2C(CNC(c3c(C(=O)OCC)cco3)=O)CC2)=O)ccc2c[nH]nc2c1 N1(C(C(C)Oc2ccc(Cl)nc2)=O)CCCC(NC(=O)CCS(N)(=O)=O)CCC1 CN1C(=O)CCC1C(=O)NCC1(F)CC(CNC(=O)Cc2ccccc2Cl)C1 C(CC(C)CCCC(C)C)NC(c1c(SCC)cc(Cl)cc1)=O C(C(CC(C)C)C(=O)NCC12CC(C)(CCO1)C2)NC(C(C)=C1CCCC1)=O C1(CC(=O)N(CCC(C)NC(=O)Cc2cccc(Cl)c2)C)CCCCCO1 C12(NC(CC=C)=O)CCCC1(F)CN(C(c1cc(OC)cc(OC)c1N)=O)C2 Cc1occc1CC(=O)NC1CCN(C(=O)C(C2CCOCC2)O)C1 C(=O)(C(C(C)C)NC(=O)CC(C)NC(=O)CCC1CC1C)NCC c1(NC(N2CCCOC(c3ccccc3)C2)=O)ccc2cnccc2c1[N+](=O)[O-] c1(C(N2CCCC(NC(C(CC)C(C)(F)F)=O)C2)=O)nc2sc(C)cn2c1C CC1(NC(C2CC2c2ccncc2F)=O)CCC(NC(c2nn[nH]c2Cl)=O)CC1 Cc1c(F)cc(C(N2CC=CC2C(N2CCC(O)C2)=O)=O)c(F)c1F C1(C(=O)NCCc2c(C)nc[nH]2)CSCCN1C(=O)C(C)n1ccnn1 N1(C(C(C)NS(CC)(=O)=O)=O)CCC(O)(CN(C)C(c2cc(C(C)C)on2)=O)C1 C1(C(=O)NC(C2CCCN2C(=O)CCn2ccnc2C(C)C)C)CC(F)C(=O)N1 c1(C(N2C3C(NC(CSCCOC)=O)C(CC3)C2)=O)c[nH]c2cc(F)c(F)cc12 N1(C(C=CCOC)=O)CCC2(NC(=O)Cc3cc(F)c(C)cc3F)CCCCCC12 c1(C(=O)NCc2ccc(N(CCCC)C)cc2)cc(C)c(CC)nc1O C(=O)(C1CCCn2ccnc21)N1C(C(=O)Nc2nccc(C(N)=O)c2)CCCC1 c1(C(=O)NC(C)CCCCNC(c2snc(O)c2Cl)=O)ncnc2c1CCC2 N1(C(C=CCCC)=O)CCOC(CCNC(=O)C(C)(C)c2cnn(C)c2)C1 c1(C(C)C)cccc(CNC(=O)NCC(C2CC(F)(F)C2)O)n1 C1(C(=O)OC)C2CCC(CC2)C1NC(C1CCN(Cc2ccccn2)CC1)=O Cc1ccc(F)cc1C(N1CCC(O)C(NC(=O)CC2CN3CCC2CC3)C1)=O c1(SC)cc(C(N2CC(O)(CNC(=O)CC3CCCC3C)C2)=O)ccc1[N+](=O)[O-] C(CCC(C)C)(C(=O)N1CCNC(=O)CC1C)NC(Cc1cc(C)n(C)n1)=O C(CCC(O)C(=O)NCC(C)Cn1ccnc1)NC(CC)=O C(CC1=CCCCC1)NC(C1CC(=O)NCC1)c1nnnn1C1CCCC1 C(=O)(CCS(C)(=O)=O)N1CCC(C(=O)NC(c2ccncn2)C)C1C Cc1cnc2n1CCC(C(=O)NC1CN(C(=O)CN(C)C(N)=O)CC1C)C2 c1(C(=O)NC(CCNC(C(c2scc(C)n2)C)=O)C)cccc(-n2cccc2)c1 C1(C)(CNC(c2c(CC(C)C)onc2)=O)CCN(C(c2ccc[nH]2)=O)C1 N1(C(c2[nH]cc(CC)c2)=O)CCN(C)CC1CNC(C1CCCCC12CC2)=O C1(NC(CCN(C(CC)CC)C)=O)CN(C(c2cc(=O)cc[nH]2)=O)CC1C N1(C(C(C2CCC2)OC)=O)CCC(C(C)(C)NC(C2(OC)CCCOC2)=O)CC1 C1(C(=O)NCCN(C(=O)C(C)CC2CC2)CC(C)O)CC(O)(c2ccccc2)C1 c1(C(N(CCC(C(C)(C)C)NC(C2C(=C)C2)=O)C)=O)cc(Br)c(F)cc1O C#CC1CCN1C(C1C(CNC(c2conc2CC)=O)C1(C)C)=O c1(NC)cnc(NC(=O)NCC2(C)CCC(C(=O)OC(C)(C)C)C2)cn1 N1(C(C2C(CCC)C2)=O)CC(NC(c2ccc(-c3cc[nH]n3)cc2)=O)CCC1C Cc1noc(C)c1CC(C)NS(=O)(=O)CCCC1CC1 c1(CCCC)noc(CCC(=O)N(C2CCN(C(=O)CCSCC)C2)CC)n1 N1(C(CC(CC)CC)=O)CC(C)CN(C(=O)CSc2ccc(C)c(C)c2)CC1C C1(C)(C(NOCC(=O)N(C)CC2CCN(CC)C2)=O)CNC(=O)N1 c1(C(=O)NC2C=CCN(C(c3c(CC)nccc3)=O)C2)ccc2c(c1)N(C)CC2 C1(CCCCNC(C=C(CC)C)=O)CCN(C(c2cnn(C3CC3)c2C)=O)CC1 C1(C(=O)NCC(C)N(C)C(C2CC2(Cl)Cl)=O)CC12CCc1ccccc12 c1(C(=O)NCC2C(OCC)CN(C(C3CC3F)=O)C2)cccc2c1CC(C)(C)C2 c1(C(N2CCC(C(N(CC(=O)N(C)C)CC)=O)C2)=O)cnc(O)c(C)c1 c1(C(=O)NC2CCN(C(c3c(CC)c[nH]c3)=O)CC2CC)cc(C)c(F)cc1Cl c1(C(=O)NCC2CC(NC(Cn3c(C)ccn3)=O)C2)ccc2cccc(O)c2c1 N1(C(c2ccn(CC)n2)=O)CC2CC1C2NC(c1nc(-c2cccs2)oc1C)=O C(=O)(C(C)(C)CNC(c1ccns1)=O)NC(C)C1CC1 C(=O)(C(C)(C)C(F)(F)CC)NCCCC(C)NC(CCC(=O)NCC)=O c1(C(N2C(C)(CC)CC(NC(=O)CCC3CCC3)C2)=O)cc(=O)c(OC)cn1C C1(C(=O)NC(c2ncn(C)n2)C)CCCCCCN1C(=O)CC(F)(F)C(F)F c1(C(N2CCC2C(=O)NCC2CC(Sc3ccccc3)C2)=O)cnn(C(F)F)c1 N1(C(COCCC=C)=O)CCCC(C(=O)NCc2cnc(C(C)C)[nH]2)C1CC C1(C(=O)NCCCC(=C)Cl)CC2CC1CN(C(c1ncc(F)cn1)=O)C2 c1(C(=O)O)cccc(Cn2cc(CN3CCC(CCCl)CC3)nn2)c1 C1(C(=O)NC(CCOC)C(C)C)CC12CCN(C(=O)C1=CC3C=CC1C3)CC2 c1(C(N2CCN(CC3CN(C(CC(C)F)=O)C3)CC2)=O)cc(C2CC2)nc(O)c1 N1(C(C(CC)F)=O)CCCCC1C1(CNC(=O)C(C)OC)CCC1 C12(NC(CCC=CCC=C)=O)CC1CN(C(=O)CCOc1ccccc1O)C2 CCCC(C)CCCC(=O)N1CCN(C(=O)C2=CCOCC2)CC1 C(CC1=CCN(C(C2CC(C)(C)C2)=O)CC1)NC(C12CC(CCC)(C1)C2)=O N1(CCCC2C(C)C2)C(=O)CN(CC23COC(C(F)(F)F)(C2)C3)C1=O CC1=C(C(=O)NC2CCC2CNC(C23CCC2C3)=O)CCO1 C1(C(=O)Nc2cn(CC(C)C)nc2)CC2(CCN(C(=O)C(F)C(C)(F)F)C2)C1 C1(N(c2cc(C(=O)OCC)sc2)C(=O)C(C)CC)CCNCC12CC2 N1(C(C2CN(C)C2)=O)CC(CC(=O)NCCC(C)(O)C2CC2)C2(CC2)C1 C=C(Cl)CC(C(=O)NCCC1(COC)CC1)NC(=O)CCc1nc(C)no1 CC1CCN(C(c2cc[nH]c2)=O)CCN1C(=O)CCN1C(=O)NC(C)(C)C1=O N1(C(COC(C)C)=O)CCC2(C1)CN(C(c1ccnc(P(C)(C)=O)c1)=O)CCO2 C1(CNC(C(SC)SC)=O)CCN(C(c2cc3c(s2)CCC3)=O)C12CCC2 c1(C(=O)OC)cc(Br)c(NC(C23CC2CN(C(c2cc(C)[nH]n2)=O)C3)=O)c(I)c1 C(=O)(CC(=O)Nc1nccs1)NC(C)CCN(C(=O)CNC(=O)C1CC1)C N1(C(C=C(C)C)=O)CCC2(CC1)CC(C)N(C(c1ncoc1C)=O)C2 N1(C(C2N(C(C)C)CCC2)=O)CCC(N(C)C(c2cc(O)nn2C)=O)C(C)C1 Cc1nc2nccc(NCC3(O)CN(C(c4cc(C)oc4C)=O)C3)n2n1 C(CC(O)CC(=O)NCC(C)CNC(c1cc(-c2ccn(C)c2)[nH]n1)=O)SC C1(NC(C2(OC)CCOCC2)=O)CC2CN(C(=O)Cc3ccon3)CC12 S(=O)(=O)(c1ccc(Oc2ccccc2)cc1C)N1CC(OC)C2(C1)CC2 N1(C(C2(CCOC)CC2)=O)CCC2(CCC(NC(=O)Cc3cncs3)CC2)C1 Cc1ccc2cc(C(N3CC(C)(NC(=O)CN(C)C(=O)C4CC4)C3)=O)ccc2c1 N1(C(C(C)Cc2cnc[nH]2)=O)CC=CC(NC(=O)C(C)(C)CC2CC2)C1 C(=O)(C(=O)N=S(C)(C)=O)N1C(CN(C(Cc2c(C)cco2)=O)C)COCC1 c1(C(=O)OC)ccncc1S(=O)(=O)NC1(c2ccc(Cl)cc2)CCCC1 C1(CC(=O)NCC(CC)NC(c2c(C)nn(C)c2F)=O)CCCC(C)(C)C1 c1(C(=O)NCC(CC(=O)N(C(C)CS(C)=O)C)(C)C)cncc2[nH]ccc12 Cc1ccc(Br)nc1C(N1CCN(CC(C)F)CC1)C(=O)NCCCN(C)C c1(Sc2ccc(NC(C3CCN(Cc4ccccn4)CC3)=O)s2)cccc(Cl)c1 C1(NC(=O)C(C2CCOCC2)O)CC2CCC1CC2NC(C1(c2nc[nH]n2)CC1)=O C(=O)(C(CC(C)(C)C)NC(C1CC1(C)C)=O)Nc1c(OC)ncc(C)c1 C1(C(N(CCn2ncc(C)c2)C)=O)C2CCC(C2)C1NC(=O)C=CC(=O)N(C)C N(C1CC2CCCc3cccc1c32)C(C(C)OC(C)(C)C)=O CCCCC(CC(=O)NCCCC(C)(C)CO)NC(=O)CCOCCCOC C1(CC)C(C(=O)NC2CC(CNC(=O)CC(C)C)C2)CCN1C(=O)OC(C)(C)C c1(C(N2CC(N(C)C(C34CC3CCC4(F)F)=O)C2)=O)nccc2[nH]ccc12 C1(C(=O)NCCOCCCC)CCCC(NC(=O)C(C)CC(=O)OC)CC1 C1(C2CC2)(NC(C2CCC(NC(c3c(C)[nH]cc3)=O)CC2)=O)CCOC1 N1(C(C(CC#N)NC(=O)OC(C)(C)C)=O)CCC2(CC(C(F)F)=NO2)C1 C1(C(=O)NC2C(C(N3CC(C(C)O)C3)=O)CCOC2)CCC(=O)N(C)C1 c1(C(N2CCC(C(C)NC(c3cnsn3)=O)C2)=O)ccc(S(C)(=O)=O)o1 c1(OC)ccnc(CN2CC(c3cccc(C)c3)(O)C2)n1 N1(C(C=C(CCC)C)=O)CCCCC1CN(C(=O)CCc1ccon1)C CC(C)CC(C)C(=O)NC1CCCC1CNC(c1cc(C(F)(F)F)c(F)cn1)=O C1(CNC(C(CC)CO)=O)CN(C)CCN1C(c1cnnc(O)c1)=O N1(C(C(C)N(C)C)=O)CCC2(CNC(=O)C(C)(C)c3ccno3)CCCC12 c1(C(NNC(=O)Nc2c(OC)ccc(F)n2)=O)nc2ccccc2[nH]1 C(=O)(C(=O)C(C)CC)N1CCN(CC(N2CCC(CN(CC=C)C)C2)=O)CC1 C1(C(=O)NC2(C)CC(F)C2)CCCCCC1NC(=O)CCCCC1CC1 n1(CC(=O)NCC#CCNC(CN(C(C)=O)C)=O)nnc(C)n1 C1(NC(=O)CSC(F)F)CC2CCC1CN2C(C1CCCC2(CC2)C1)=O Cc1cncc(C=CC(=O)NC2CN(C(=O)CC(C)c3ccncc3)CC2C)c1 C1(NC2(c3onc(C)n3)COC2)CC(NC(=O)OC(C)(C)C)C(O)C1 c1(OC)cccc2cc(C(=O)NC3CC(O)CC3O)c(=O)oc12 Cc1cc(=O)n(C)cc1C(N1CCC(N2CCN(C(=O)C(F)F)CC2=O)CC1)=O CS(=O)(=O)CCCCCCCC(=O)N(c1ccc(Cl)c(C(F)(F)F)c1)CC1CC1 c1(C(=O)NC2CN(C(=O)NC3CC3)C2)c(Cl)oc2ccccc12 c1(C(=O)NC(CC#C)C(=O)NCCCN2CCOCC2)ccnc(C)c1N N1(C(C(C=C=C)C)=O)CC(C2CCCN(C(=O)C=Cc3cccc(Cl)c3Cl)C2)C1 C1(NC(c2cc(N)cc(O)c2)=O)CC2CC1CN(C(=O)CC1=CCOCC1)C2 C12(NC(C3CCN(CC(C)C)C3)=O)CC(CNC(=O)C(F)F)(C1)OC2(C)C N#Cc1cccc(-c2cc(CN3CCC(CC(=O)O)C3)ccc2OC(F)F)c1 N1(C(C(COC)C)=O)CC2CC2(NC(c2ccc(Br)s2)=O)C1 CCC(C)(C)C(C)CC(=O)N1CC2(C1)CN(C(c1cnnc(C3CC3)c1)=O)C2 C#CC1CCCC(NC(C2CCN(C(c3ncnc(O)c3F)=O)C2C(C)C)=O)C1 C1(C(NOCC(=C)C)=O)CN(C(C23CC(C#N)(C2)C3)=O)CC1(F)F CC(C)(Cc1ccsc1)C(=O)NC1CC(NC(=O)CNC(c2cccnc2)=O)C1 c1(NC)cncc(C(N2CC(C(N3CCC(CCO)CC3)=O)(SC)C2)=O)c1 c1(C(=O)NC2CCC(CNC(c3cc(C#N)no3)=O)C2)cnc2ccccc2n1 N1(C(C(COC)NC(CCCOCC=C)=O)=O)CCC(COC)C(C)C1 c1(C(=O)NCC2C(NC(CCc3ccn(C)c3)=O)C2)c(C2CC2)cccc1F c1(OCCOC)cncc(C(N2CC(CNC(C3CCC(C)C3)=O)C2)=O)c1.OCC Cn1nnc(CNC(C2CC2Cl)=O)c1C(=O)NC1CNC(=O)C1 c1(C(C(=O)NCC2C3CN(C(C4N(CC)CC4)=O)CC32)=O)ccc(F)cc1F c1(C(=O)NCC(CNC(Cc2c(C)nc[nH]2)=O)C)ccc(CO)cn1 Cc1c(F)ccn2c(CNC(=O)CC(c3ccc(C(F)(F)F)cc3)C)cnc12 CC(CC(=O)NCC1COCC1NC(c1ccc(NC(C)C)nc1)=O)P(C)(C)=O C(=O)(C(F)(F)CNC(C1(NC(C2C=CCCC2)=O)CCCCC1)=O)OC c1(C(N2C3CN(C(CC4(C#N)CC4)=O)C(CC3)C2)=O)ccn2c(O)nnc2c1 N1(C(C2C(NC(c3nn(CC)c(O)c3)=O)CCOC2)=O)CCC2(CCCO2)CC1 C1(NC(C(C)CC2CCCC2)=O)CCCC(CNC(=O)CSc2ccccn2)C1 CC(C)CCN=C(NCc1ccc(C(C)O)cc1)NCC1CN(C(C)C)CCO1 N1(n2c(C(=O)NC(CSC)(C)CO)ccc2)C(=O)c2ccccc2C1=O C(=O)(C1=CCC(C)CC1)NCC1OCCCN(C(C2(COC)CC2)=O)C1 C1(F)(CNC(C(C)(C)c2ccc(Cl)s2)=O)CCCN(C(c2ncccn2)=O)C1 CC1CCC(C)N(C(C23CC(CN(C(C4(C(C)(C)O)CC4)=O)C2)C3)=O)C1 C1(c2cc(C)no2)(NC(C2(C3(C(=O)O)CCCCC3)CC2)=O)CCOCC1 N1(C(C(C)(C)OC(C)=O)=O)CCC(CNC(=O)CN2CC(=O)N(C)C2=O)C(C)C1 CC1CCC2(CC1)CCN2C(=O)CCC1CCN(C(C2(CO)CCC2)=O)C1 c1(CN2C(C(=O)Nc3ncc(F)cc3Br)CC2)ccc(Br)cc1[N+](=O)[O-] c1(OC)ccc(C(C(=O)NC2(C)CC2)N(C)Cc2nncs2)cc1C N1(C(C2CCN(C(C3C(C)(C)C3)=O)CC2O)=O)CCC2(CC1)COC(=O)N2 Cc1cc(C#N)cc(C(=O)NC2CC3CC(C2)N(C(c2cccnc2O)=O)C3)n1 CC1C(NC(=O)CCc2ccncc2)CC2CCC1N2C(c1ccnc(Cl)c1)=O N1(C(c2c(C(C)C)noc2)=O)CC2CCCC2(CNC(=O)CSCC(F)(F)F)C1 c1(OC(C)C)ccccc1CC(=O)NC1CN(C(=O)CC2(C)CC2)CC1C N1(C(=O)C(Cl)=CCl)CC2(C1)CN(C(C1(C(F)F)CCCC1)=O)CCO2 CC1(O)CCCN(C(=O)C2=CCN(C(=O)CCc3ccco3)CC2)CC1 c1(C(N(CC(C)(C)NC(c2ccc(CN(C)C)o2)=O)C)=O)cnc2n1CCOC2 c1(C(=O)NC(c2cn(C(c3cccnc3)C)nn2)(C)C)cc2scc(Cl)c2[nH]1 N1(C(C2(Oc3ccccc3)CC2)=O)CCC(O)C(c2ccccc2)C1 N1(CC(=O)NCC(C2CCCCC2)NC(CC#N)=O)Cc2ccccc2C1 C1(C(N2CCCC(N(C(=O)CCN3CCCCC3)C)CC2)=O)CCCCCS1(=O)=O n1(CC(C)C)cc(S(=O)(=O)NCc2nc3cnccc3s2)cn1 Cc1ccccc1C(C)CC(=O)NCCN(C(=O)C(c1cccnc1)O)C1CC1 c1(NC(C(=O)NCC2(CC)CCOC2)=O)ccccc1C c1(CCOCC)nc(C(=O)NCCCN(C)C(C2CCCN2C(N)=O)=O)co1 CCCCC(O)C(=O)N1CCCC(N(C)C(c2ccc(O)cc2F)=O)CC1 C1(CC(=O)NC(c2ccccc2)CNC(C(C)SCCCC)=O)CCCC1(F)F CCC(C)C(O)CC(=O)NC(COC)CC(=O)NC1CCC(=O)NC1(C)C N1(C(CC2CN(C)C2)=O)CCC(CO)C(NC(c2ncccc2NC(N)=O)=O)C1 c1(C(=O)NCCCN(C)Cc2nn(CC)nc2C)nc[nH]c2nccc1-2 Cc1cc(C)c2nc(N3CCC(NC(c4ccnn4CCF)=O)C(F)C3)sc2c1 CC(C)CC(C)(C)C(=O)N1CCC(C)C(NC(c2ccccn2)=O)C1 Cc1cccc(N(C)C(C23CC(CN2C(=O)Cc2cccnc2)C3)=O)c1C c1(C(=O)Nc2nc(C#C)c(C)cn2)c(Br)cc2ccccc2c1F Cc1cc(C(N2CCOC(CC(=O)NC3CC3c3ccn(C)n3)C2)=O)ccn1 C1(C(=O)NCCN(C(C(C2CCOCC2)OC)=O)CC(C)O)(CF)CCOCC1 N1(C(C=CCN(C(C(CCCC)=O)=O)C)=O)CCCC2NC(=O)CC12 C(c1ccccc1)=C(CC)C(=O)NCC(C)NC(=O)CCc1ncc(F)cn1 N1(C(c2ncc(N)nc2)=O)CCOCC(CNC(C2CC2C(N)=O)=O)C1 c1(C(C(=O)NC(CN(C(C2CC3(CC3)C2)=O)CC)C)C)ccc(C)s1 C(C(CC(C)C)NC(C12CCCC1C2)=O)NC(c1cc(C)on1)=O c1(C(CC(=O)N2CC(CC(=O)N(C3CC(O)C3)C)C2)N)ccc(F)c(F)c1 CC(C)C(CNC(C1(Br)CC1)=O)NC(=O)COc1cn[nH]c1 O(NC(=O)C(CCSC)NC(c1cc(C)c(C)o1)=O)CCCC#C C1(CC)CCC(C(N2CCC(CNC(=O)CCCC3CCCCC3)C2)=O)O1 c1(OC)cccc(CNC(C2C(N)C3CCCCC23)=O)c1Br Cc1cnc(C(=O)NCC2C3CC2N(C(c2ccc(C(F)F)cn2)=O)C3)c(F)c1 Cc1cccc(CC(=O)NCC(CC(C)C)NC(C2COC(=O)O2)=O)c1 N1(Cc2cc(OC)ns2)CCC(C2(NC(=O)C(=O)Nc3ncc[nH]3)CC2)CC1 c1(C(=O)NC2CN(Cc3cccc(Cl)c3)CC2F)ccc2cccc(Cl)c2n1 CC(C)C(CNC(C1CCN1C)=O)N=c1nc(Cl)[nH]c(C)c1C#N N1(C(c2c(Cl)cn(CC)n2)=O)CC2CCC1CC2NC(=O)C(C)CN(C)C CC1CN(C)C(C)CN1C(C1CN(CC#N)CCC1(F)F)=O Cc1cc(NC(C2(C)CN(C(=O)CCN3CCOCC3)C2)=O)c([N+](=O)[O-])cc1C c1(OCC(=O)NCC(CN(C)C(C2COCCO2)=O)O)ccc(C#N)cc1Cl n1(CCCC)nnnc1C(C)(CC1CC=CCC1)NCCC1CC1.c1(C)ccccc1 C12(NC(CC)=O)CC3CCC(C1C2)N3C(c1nn(-c2ccccc2)cc1OC)=O c1(C(C(N2CC(N(C(CC3(OC)CCC3)=O)C)C2)=O)O)ccc(Br)cc1F c1(C(C)C)ccccc1CC(=O)NCC1(O)CN(C(c2c[nH]cc2C2CC2)=O)C1 N1(C(C(CO)NC(C(C)C)=O)=O)CC2CCCC2(NC(C2COCC2(C)C)=O)C1 c1(C2(C(=O)OC)CC(NC(C3CCCN(C(=O)C(C)(C)C)C3)=O)C2)ccc(C)cc1 C1(NC(=O)NC(C(O)C(F)(F)F)C2CC2)CCC2(CCOCC2)C1 N1(C(CC(=C=C)C)=O)CC(C)CN(C(c2cnc3ncc(Cl)cn23)=O)C(C)C1 N1(C(c2c(C)cnnc2)=O)CC(N=c2ncc3ccccc3[nH]2)C1 Cc1c(C(=O)NC(C)CC(C)NC(C23CC(F)(C2)C3)=O)[nH]c2c(C)cccc12 C(CC(=O)NCCCCC1CN(C(=O)COC2COC2)C1)NC(C1C(C)C1)=O CC(C)CCCCCC(=O)N(CCC(N1CCCC1C(O)CO)=O)C c1(C(N(C2CN(C(=O)C(C3CCC(O)CC3)(C)C)C2)C)=O)cc(O)cc(F)c1F Cc1ccncc1C(c1nnnn1C)N(C(Cn1cc(C(C)N(C)C)nn1)=O)C C1(C(N(CCCCN(C)C)C)=O)(NC(C2COCOC2)=O)CCSC1 N1(C(C(C)(C)CC2CC2)=O)CCC2CN(C(=O)CC(F)(F)Br)CC2C1 C1(CNC(CC2(OCC)CCC2)=O)CC2CCC1N(C(=O)CC#N)C2 CC1CCC(CO)N(N(CCN2CCN(C)CC2)CCO)C1 c1(C(N(CCCN(C(CSCCC)=O)C)C)=O)cc2c(=O)n(C)c(=O)n(C)c2s1 N1(c2n(CCC#C)c(-c3cccn3C)nn2)Cc2ncnc(O)c2C1 CON(CCC(=O)N1CCN(C)C(=O)C1C)C(=O)Cc1cc(C)n(C)n1 Cc1ccc2snc(C(=O)NCC(C3CC3)NC(C3CC(N(C)C)C3)=O)c2c1 N1(C(C(CC=CCC)C)=O)CCCC2C(NC(c3cc(C)sc3N)=O)C(C)(C)C12 C=CCC(C(=O)OCC)NC(=O)C(COC)NC(c1ccn(C)c1C)=O C(=O)(C(O)CC(C)(C)C)N1CC(CC(C)NC(=O)CCNC(=O)C(C)(C)C)C1 N1(C(C2(C#N)CCOCC2)=O)CCC=C(C(=O)Nn2cncn2)C1 c1(C(=O)NC2C3CN(C(c4n(C)nc(CC)c4Cl)=O)C2C3)coc2c1CCCC2 C12(CC(=O)N(CC(CC)NC(c3cc(C(F)(F)F)no3)=O)C)CCC(C)(C1)OC2 n1(C(C)C)cc(C(c2nnnn2C(C)(C)C)NCCC2CCCC2)cn1 N1(C(CC(C=C)C)=O)CCN(C(c2cc(Cl)n[nH]c2=N)=O)C2CCC12 c1(C(=O)NCC(C)NC(C2C(OCC)C2)=O)c[nH]c2cc(C)ccc12 N1(CC(N2CCCC(C)(CNC(C3CC(O)C3)=O)C2)=O)CCc2sccc2C1 CCCCS(=O)(=O)NCC(=O)N(CCCCCNC(C1CCC(O)CC1)=O)C N1(C(c2coc(Cl)c2)=O)CCN(C(=O)Cc2sc(O)nc2O)C(CCO)C1 c1(C(=O)NCCOCCN(C(c2cccc(C)c2)=O)C)cccc(Cl)c1Cl C1(=C2CC=CCC2)N=C(c2cc3c(s2)CCC3)NC1c1ccc2c(c1F)OCCO2 C(=O)(C(C)(O)CC(F)(F)F)N(CCCNC(C(C1CC1)OC)=O)C1CC1 c1(C(=O)NCC2C(C)CCN(C(=O)CS(C)(=O)=O)C2)cnc2c(Cl)cccn12 Nc1cc(C(=O)NCC2CCN2C(C23COCC2C3)=O)ccc1-n1cncn1 Cc1cncc([N+](=O)[O-])c1N(C)C(C1CN(c2ncnc3sc(C(C)C)cc23)C1)=O N1(C(CC(C)C)=O)CC2CC1C2NC(=O)C(C)Oc1ccccc1F C(=O)(CC(C)CC(F)(F)F)NCC(C(C)C)NC(=O)Cc1cnnn1C n1(CC(=O)NC2CCN(C(COCCCCC)=O)C2C(C)C)cc(F)ccc1=O CC(F)(F)CCC(=O)N1CCN(C(c2cnn(CCF)c2)=O)C(C(F)F)C1 c1(C(N2CCC(N(C(C(CC)NC(N)=O)=O)C)C2)=O)nnc(C)cc1O C(CO)(C(=O)NCc1cnn[nH]1)NC(C(c1ccn(C)c1)C)=O n1(CC(=O)NCC(CC)(CC)NC(=O)C(C)NS(C)(=O)=O)ccc(=O)cc1C c1(C(=O)NCCOC)cc(CNC(=O)C(c2ccc(O)cc2)=O)ccn1 c1(C(CNC(=O)C(F)=C(C)C)NC(c2nnc(CC)s2)=O)ccccc1OC N1(C(COCC(=O)OC(C)(C)C)=O)CCCC(CCNC(c2cc(F)cs2)=O)C1 N1(C(C)=O)CCc2cccc(C(=O)NC3(c4ccc(Br)c(Cl)c4)CCC3)c2C1 C1(C(=O)NCc2cc(SCC)c(C)s2)CC(C2CC2)=NO1.C1CO1 c1(C(=O)NC2CCCCN(C(c3cncc(C)c3C)=O)C2)cc2ccncc2[nH]1 C(c1cccc(Br)c1)=CC(=O)NC(CNC(C=COCC)=O)CO CC1(C)COC1C(=O)NC(CNC(c1occc1Br)=O)C1CC1 Cc1cc(CCC(=O)N(CC(C)CNC(C2CCCCC2)=O)C)c(C)s1 N1(C(C2C(C)N(C(c3nc(=N)cc[nH]3)=O)CC2)=O)Cc2cccnc2C1 c1(C(=O)NC23CC(NC(CSC)=O)(C2)C3)ccc(Br)cc1O c1(C(=O)Nc2scc(C3C(C(=O)OC)C3)n2)c(Br)cnn1C C(=O)(C#CC1CCCC1)N1C(C)CC(CNC(C2(c3ccno3)CC2)=O)CC1 C1(CN(C)C(c2ccncc2)=O)CN(C(c2cn(C3CC3)nn2)=O)CCO1.O c1(CC(=O)NC2(CCNC(CNC=O)=O)CCC2)cnc(C2CC2)[nH]1 c1(NC(C(N2C(NC(=O)OC(C)(C)C)CC2)=O)=O)cn(C(F)F)c2ccccc12 C1(CNC(=O)NCC2CC2c2ccco2)CCCCN1Cc1ccco1 C1(OC)CN(C(c2cnc(C(N)=O)cn2)=O)CC1NC(c1cc[nH]n1)=O N1(C(c2c(C)[nH]cc2)=O)CCC(C2CCCN(C(c3cnnc(O)c3)=O)C2)C1 Cc1ccc(C(=O)NCC2(F)CC(NC(C3(CCN(C)C)CC3)=O)C2)cc1C C1(NC(c2ccc(C)o2)=O)CCN(C(=O)Cc2ccccc2SC(C)C)CC1C c1(C(N2CC(NC(CC(=C)C)=O)C(C)C2)=O)cn2c(n1)CC(C)CC2 C1(C2CC2)(CNC(C(C=C)(C)CC)=O)CCN(C(=O)COCC(C)C)C1 CC1CN(C(=O)CCS(C)(=O)=O)CCN1C(=O)COc1cc(F)cc(F)c1 C1(C(=O)NC2CN(C(=O)Cc3ccc(O)cc3)C2)CCCN(c2ccncc2)C1 C(C(CC)CC)(c1onc(CCC(=O)OCCCC)n1)N.c1ccccc1 N1(C(C(C(CC)CC)F)=O)CCC2CN(C(=O)C(C)C(CC)CC)CCC2C1 CCC(C#N)(CC)C(=O)N1CCCC(CN(C(=O)CCc2ncccc2C)C)C1 c1(C(=O)Nc2nc(C3CC3(Cl)Cl)cs2)ccc(S(=O)(=O)Cc2ccc(Br)cc2)cc1 Cc1ccc(NC(C2CC(F)CN2C(=O)CCc2ccccc2F)=O)c(C)c1C C1(CNC(c2c(C)onc2C2CC2)=O)N(C(c2cncs2)=O)CCC1(C)C c1(OCC)cccc(C(=O)NCC2(CO)CCN(C(C3CNC(=O)N3)=O)C2)c1N S(=O)(=O)(c1ccc(NCCCN2CCN(C)CC2)cc1Cl)N1CC(C)=C(C)C1 N1(C(CC(CC)(F)F)=O)CC2(CCC2)CC1C(=O)NC1CN(C)CC1C C(CCO)(C(F)(F)F)NC(N1CCN(c2cc(N3CCOCC3)ncn2)CC1)=O c1(OC)ccc(Cl)cc1C=CC(=O)NCC=CCNC(C1CCOC(=O)CC1)=O C(c1c(Cl)cccc1Cl)=CCNC(CCCCNC(=O)OC(C)(C)C)=O N1(C(COCc2c(C)cccc2)=O)CC(C)N(C(=O)CCC2(C)CC2)CC1C c1(C(N2CCC(NC(CC(c3ccc(CC)cc3)C)=O)C2)=O)cc(=O)cc(Cl)[nH]1 C(CCc1cn[nH]c1)(C(=O)NCC(O)CF)NC(=O)OC(C)(C)C C1(NC(c2n(C)nc(C(F)F)c2)=O)CCC2CCN(C(=O)C3=CCCSC3)C12 c1(C(=O)NCCC23CCC2CN(C(=O)C(Cl)=CCl)C3)cc2ccccn2n1 CC(C)(C)CC(O)C(=O)N1CC(O)CC1CC(=O)NCC1(O)CCSC1 N1(C(c2cccc(OC)c2)=O)CCC2(NC(=O)CCC3CC3(C)C)CCCC12 Cc1nc(C(=O)NC(C23CCC(CC2)C3)CNC(=O)Cc2c[nH]nc2C)c(C)s1 C(=O)(C(C)(C)C(N)=O)NC(CCOC)CNC(=O)C(c1ccccc1)SC CC1(C)CC(CC(=O)NC2C3CCCC23)N(C(c2ncncc2Cl)=O)C1 CC1(C(=O)NCC2CCN2C(=O)Cc2csc(Cl)n2)CCc2ccccc2C1 C1(C(N2C(CNC(CCCCCSC)=O)CCC2)=O)Cc2ccncc2C1 c1(C(=O)NC(CNC(C(CC#C)(C)C)=O)C2CCC2)ncnc2c1OCCO2 c1(C(=O)NC2CC(NC(C3CCN(C)C3)=O)C2)c[nH]c2cccnc12 C1(NC(c2c(CCNC(C(C)(C)N=[N+]=[N-])=O)n[nH]c2)=O)CCc2nncn2C1 c1(C(=O)OC)ccncc1C(=O)NC1CC(NS(=O)(=O)CCCOC)C1 N1(C(c2cc(OC)cc(Cl)c2)=O)CC2CN(C(C3CCCC34CC4)=O)CC2C1 C12(CNC(CCCNC(N)=O)=O)CCC(CC1)N2C(c1cc2n(c1)CCC2)=O C(CCC1CC1)(C(=O)N1CCC(O)C1)NC(C(CC)C1CCC(=O)N1)=O C(=O)(CS(=O)(=O)CCO)NC(C1CCCCC1)CNC(c1n(CC)nnc1C)=O N1(C(c2nc(COC)oc2)=O)CCCC(NC(C2CCCC2C(F)F)=O)C1 N1(C(C2(NC(C(CCC)F)=O)CCCC2)=O)CC2C3C=CC(O3)C2C1 c1(C(=O)NCC(CCCC)NC(=O)C(C)(C)CN(C)C)cc(O)ccc1C C1(CC=C)(NC(c2[nH]nnc2C)=O)CCN(C(c2nnc(C)s2)=O)C1 c1(C(=O)NC2CCCC(CNC(C(C)(C)SC)=O)C2)ccc(O)c(CO)c1 C1(C)(NC(CCOCC)=O)CCCN(C(c2cccc(C)c2O)=O)C1 c1(CC(N2CCC(C(C(=O)N(CC(C)N(C)CC)CCO)C)C2)=O)cccc(F)c1 c1(SCC(N2CC(O)(CNC(C3(C(C)C)CCCO3)=O)C2)=O)cc(F)ccc1F n1(CCN(CC)CC)nc(-c2cc[nH]n2)nc1C(C)Sc1nccn1C N1(C(Cc2c(C)noc2Cl)=O)CCCC2(NC(=O)Cc3cccs3)CC2C1 C1(C#N)(C(=O)NC2CC3(CN(C(C4N(CC)CCC4)=O)C3)C2)CC2CCC1CC2 N1(C(C2(C#N)CC2)=O)CC(C(=O)NCCC2CCCC23CC3)C2(CCC2)C1 Cc1cc(=NCC(C)CNC(=O)Cc2c[nH]c3cc(F)ccc23)[nH]c(CO)n1 N1(C(c2cc(COC)[nH]n2)=O)CC(C2CCN(C(=O)C(C)=C3CCCC3)CC2)C1 C1(C(N(CC(C)CNC(c2cc[nH]c2)=O)C)=O)CCC(=O)C1 c1(C(=O)NCC2(O)CN(C(c3nc(CCC)sc3)=O)C2)cc(C)c2[nH]nnc2c1 Cc1[nH]nc(C(=O)NC2(C(N3CC(n4cnnc4)C3)=O)CC2(C)C)c1Cl C1(CN(C(=O)C(C)SC)CC)CCN(C(=O)C=C(C)C2CC2)CC1 CCS(=O)(=O)CC(=O)N1CCCC1CCN(C(C1CCN(C(C)=O)CC1)=O)CC C=Cn1nccc1C(=O)NC1CCCN(C(c2ccccc2C(C)(C)C)=O)C1 n1(CC)cc(C(=O)NC2CCC(CCNC(=O)CNC(C)=O)C2)c(C2CC2)n1 c1(SCC)cnc(O)c(C(=O)NCCC(C)(C)NC(c2nc(O)c(C)s2)=O)c1 c1(CCC(N2C(CNC(C(COC)O)=O)CC3(CC3)C2)=O)csc2ccccc12 CC(C)CCSCCNC(C1(NC(c2cncs2)=O)CCC1)=O C(=O)(C1=NN(C)C(=O)CC1)N1CC2C(CNC(CC(C)N(C)C)=O)(C2)C1 N1(CCNC(C(C(C)OC)O)=O)CCCN(C(c2nonc2N)=O)CC1 Cc1ncc(C(=O)NC2CCCCN(C(c3ccnc(O)c3)=O)C2)c(C(C)C)n1 N1(C(C(=O)NCC(F)F)=O)CC(C(=O)NOCC2CCCC2)CC12CCC2 c1(OC)cccc(CNC2(c3nnnn3CC)CCSC2C)c1 N1(C(CC(=O)NCC#C)=O)CCC(C)C1CNC(=O)CSc1ccc(C)cc1 c1(C(N(CCC(C(C)C)NC(C2CCN(C)C2)=O)C)=O)ccnc2ccsc12 C(=O)(C(F)(F)C(O)C1CC1)NCC1(C)CCCN1C(=O)CSc1nc[nH]n1 N1(C(c2c(C)ncc(N)c2)=O)C2CCC1CC(N(C)C(C1CCCC(C)C1)=O)C2 c1(C(N(CCCNC(C2CC3CC2C3)=O)C(C)C)=O)cc2n(n1)CCCO2 Cn1ncc2cc(C(=O)NCC3C4CN(C(C5CCS(=O)(=O)N5)=O)CC34)cnc12 Cc1c(C(N2CC(NC(C3(C)CNC(=O)C3)=O)C(F)C2)=O)ccc(F)c1F c1(C(N(C2C(N(C(c3c(C)ccnn3)=O)C)CCCC2)C)=O)ccccc1C#N C12(C(=O)OCC)CCC(C(=O)NCCN(C(=O)C(C)CCOC)C)(CC1)CC2 Cc1cc(C(N2CCC(C)(CNC(=O)CC(O)C3CCCC3)C2)=O)nn1C1CC1 C1(C(CNC(CN(S(CC)(=O)=O)C)=O)C)CCN(C(C2C(C)C2C)=O)CC1 CC1CC(N=c2[nH]c(N3CCC(C(F)(F)F)CC3)nc3c(F)cccc23)CCO1 c1(COC)ncc(C(=O)NCC(C2CC2)NC(c2cc(-c3ccco3)c[nH]2)=O)s1 c1(OC)ccc(CN2CCCC(NC(=O)CCC3CCC3)C2)c(Br)c1OC CCCCC(O)C(=O)N1CCCC(O)(CNC(=O)C=C2CCC2)C1 Cc1nc(O)nc(O)c1CC(=O)NC(C)CCN(C(=O)C(C(C)(C)C)N(C)C)C N1(C(Cc2c(C)ocn2)=O)CCCC12CCN(C(C1C(C)(C)C1(F)F)=O)C2 C1(C2CC2)(CNC(CNC(CC)=O)=O)CCN(C(c2cc(CO)[nH]n2)=O)C1 N1(C(CC(CC)(F)F)=O)CC2OCCN(C(c3cnc4[nH]nnc4c3)=O)C2C1 C1(CNC(C2CC=C(C)CC2)=O)CC2(CC(NC(C3(C)CCOC3)=O)C2)C1 N1(C(CCCOCC)=O)CC2CC(NC(c3cc4cnn(C)c4s3)=O)CC2C1 C(=O)(C(F)C(C)CNC(c1cnc(O)cc1C)=O)NCc1cn(CC)nc1 C(=O)(C(CC)CC(F)(F)F)NCC1(F)CCN(C(c2c(CC)occ2)=O)C1 CN1C(=O)OCC1C(=O)NCCCCCCc1cn(CCOCCO)nn1 C1(CNC(c2c(OC)cnnc2)=O)(CO)CCCN(C(C2(C)CCCCC2)=O)C1 c1(CC(=O)NCCN(C)C(c2ncccc2C(F)(F)F)=O)c(F)cccc1C#N N1(C(c2n(C(C)C)ccn2)=O)CC(C(=O)NC2CCC3(CCC3)C2)CC(C)(C)C1 C1(OC)CCC(C)(C(=O)NC2CCCN(C(C3CCCN3C)=O)C2C)CC1 c1(C(C(=O)NCc2ccccc2Cl)N(C2CC2)CC)ccc(F)cc1F c1(OC)cccc(C(C)(C)CNS(=O)(=O)CCN(C)C)c1 N=c1[nH]ccc(C(=O)NCC2CC(NC(c3conc3C3CC3)=O)C2)c1[N+](=O)[O-] C1(C(=O)O)CC2CCCCC2N(C(=O)CCn2ccnc2)C1 c1(NC(=O)CN(C)CCOCCO)ccc(C(=O)NCC#CCNC(C)=O)o1 CCC(C)CCCC(=O)N(C(C(N1CC2(C1)CN(C)C2)=O)C1CC1)C CCCS(=O)(=O)CC(=O)NC12CCC(CN(C(c3ccncc3Cl)=O)C1)C2 C12(C(N3CCC(C(C)NC(c4cc(=O)cc[nH]4)=O)C3)=O)CCCCC1OCC2 C(=O)(C#CC1CCCOC1)N1CCCCC(NC(c2ccc([N+](=O)[O-])o2)=O)C1 c1(-c2n(CC=C)c(N3CCNC(=O)C3)nn2)ncc(C)cc1F c1(C(N(CC(O)CN(C)C(c2cc(C(F)F)no2)=O)C)=O)n[nH]c2c1CCOC2 N1(C(C2C(C)C2C)=O)CCN(C(=O)CCC(=O)c2ccccc2)CC(C)(C)C1 c1(CCC(=O)NCC#CCNC(=O)C2=CCSC2)cc(F)cc(Br)c1 C1(CC)CCCCC1C(=O)NC1(CO)CN(C(c2cc(C3(O)COC3)on2)=O)C1 C1(CNC(Cc2cnc(C)s2)=O)(CO)CCN(C(c2sccc2C)=O)C1 c1(C(=O)NC2C(C(=O)Nc3ncc(C)nc3)C2)ncc(Cl)cc1C c1(C(N(CCNC(=O)CCc2ccon2)CC)=O)c[nH]c2ccc(F)cc2c1=O C1(CNC(COC2CCN(C)CC2)=O)CCCCCN1C(=O)CCc1cccs1 N1(C(c2c(C)onc2)=O)CCCC2(C1)CN(C(C1CCCN1C=O)=O)CCO2 C(CCCCCNC(=O)C(C)(C)C1CC1)NC(c1c(CC)occ1)=O O=C1NCC(NC(C2(F)CN(C(c3cccc(F)c3)=O)C2)=O)CO1 c1(NC)ccc(C(N2CCC(C(=O)NCC34CCC(CO3)C4)C2C(C)C)=O)cc1 c1(OC)cc(OC)nc(Sc2nc(F)ccc2Br)n1 c1(CC)ccc(F)c(C(=O)NC2(CF)CCN(C(=O)CCCNC(=O)OC)C2)c1 CCCC(C(O)C(=O)NCC(C)(F)C(C)C)NC(=O)C=CC1CCOC1 c1(N2CC(CN(C(c3c(C)cn(C)n3)=O)C)OCC2)cc(C(N)=O)nc(Cl)n1 C1(CC)CCCC(N=c2[nH]c3c(c(=NCc4nnc(C(C)C)n4C)[nH]2)SCC3)C1 C(=O)(C1=NOC(C)C1)N1CCC(C)(CC(=O)NCc2nnc(C)n2C)C1 N1(C(c2c(C(C)C)occ2)=O)CC2C(NC(C3C4CN(C)CC34)=O)C2C1 CS(=O)(=O)C1CC(C(=O)NCCCNC(C2CCCN2N=O)=O)C1 c1(C(=O)NC2CN(C3CN(C(CC4C(C)(C)C4)=O)C3)C(=O)C2)cc(Cl)ccc1F c1(CNC(C(C)N(C(COCC(=O)OC)=O)C2CC2)=O)cccc(F)c1F CC(C)CS(=O)(=O)CC(=O)NC1CS(=O)(=O)CC1NC(C1CCCC1)=O CC(C)(C)C(CNC(c1csc(O)n1)=O)C(=O)NCC12CCC(CO1)C2 N=c1ccc(C(N2CCCC2CCCNC(C2CC3C=CC2CC3)=O)=O)c(Cl)[nH]1 C(N=c1nc(N2CCC(OCCO)C2)c2c([nH]1)CCCCC2)c1nnn(C)n1 CCCC(C)(O)C(=O)N1CCC(C(=O)NCCc2cccc(O)n2)C1 c1(C(=O)NCCCNC(C2CC(c3ccc(F)cc3)C2)=O)nnn2c1CSCC2 C(=O)(CCCC(=O)OC)NCC1C(NC(CN(CC)CC)=O)CCCC1 C1(NC(=O)CCc2cccs2)CC2(C1)CN(C(=O)Cn1ccc(C3CC3)n1)C2 c1(C(=O)NC2CC(N(C(C(CC)O)=O)C)C2)cc(OC)cc2c1CCC2 C1(C#N)(C(N(CC(C)NC(C2CCC(C)C2)=O)C)=O)CC1C(F)(F)F c1(-n2c(CC3CCC(O)C3)nc(CC(C)C)n2)nc2ccccc2[nH]1 c1(C(=O)NC2CCCC2CNC(C2(c3ccno3)CCC2)=O)cc[n+]([O-])cc1 c1(C(=O)NCC(c2ccccc2)N(C(C=C(CC)C)=O)C)ncc[nH]c1=O N1(C(c2ccc(OC)cc2)C(=O)NC2CC(F)(F)C2)CCCC(C)(O)CC1 N1(C(Cc2onc(C)n2)=O)CCCC(N(C(=O)CC2CC2(C)C)C)CC1 C1(F)(CNC(C=C(CCC)C)=O)CCC(NC(c2cc[nH]c2CC)=O)C1 N1(C(C(C)n2cncn2)=O)CCN(C(COc2ccccc2)=O)C(C)CC1C(=O)O N1(C(C(CC=CC)NC(=O)CN(C)C(=O)C2CC2)=O)CCOC(C)(CC)C1 c1(C(=O)NCc2ccc(CNC(C(C)(C)SC)=O)cc2)cncc(Cl)c1C c1(OC)ccc(C(=O)NC(C2CCN(C(c3cccnn3)=O)C2)C)nc1Cl C1(NC(c2c(C)cco2)=O)CCC2CCN(C(C3CCCC34CC4)=O)C1C2 N1(C(C2C3(CC(NC(COCC=C)=O)C3)C2)=O)CCC2(CC1)CC2CO C1(NC(C2COC(C)(C)O2)=O)CCC2CN(c3cnc4ccccc4n3)CC2C1 C(C(C)(C(=O)NC1CCC(C(=O)N(C)CC2CCCC2(C)C)C1)OC)OC N1(C(c2c(C)noc2N)=O)CC(CNC(=O)C(C)OC2CCCC2)CC(C)(C)C1 Cc1nc2ccnn2c(C)c1CCC(=O)NCC1CN(C(=O)CN(C)C(N)=O)C1 C(=O)(C(F)(F)C(C)(C)O)N1CCC(C)C(NC(=O)C(O)Cc2cnn(C)c2)C1 c1(C(=O)NC(C)Cc2ccccn2)c(CNC(C2(C)CS(=O)(=O)C2)=O)nnn1C C#CC1CCN(C(=O)Cn2cc(CCNC(=O)OC(C)(C)C)nn2)CC1 c1(C(N2CCC(C)C(C(=O)NCCSCC(F)(F)F)C2)=O)cnn2ccncc12 Cc1oc(-c2cccs2)nc1CC(=O)NCC1CN(C(C2CCOC2(C)C)=O)C1 C1(NC(C(C=C)(C)C)=O)CC(C(=O)NCCNS(N)(=O)=O)=CC1O N1(CCC(C)C)CCCC1C(=O)NC1CCC1CNC(c1ncnn1C1CC1)=O O(N(C)C(=O)CN=c1nc2c(cnn2C)c(NC2CC3CCC2O3)[nH]1)CC N1(C(CC[SH](C)(=O)C2CC(C3CCc4cncn4C3)C2)C)CCC(C)C(C)(C)C1 N1(C(c2ccc(C)c(C)c2)C(=O)NCCCOC)CC(C)Cc2ccccc21 CC1CCC(CC(=O)N(CC(=O)NCc2ccnn2CC(F)F)C)O1 N1(C(c2c(CC)nn(C)c2)=O)CC2CCC2(CC(N2CC3C(C)C3C2)=O)C1 c1(NC(C2(C)CCN(C(Cn3ncn(C)c3=O)=O)C2)=O)ccc(O)c(F)c1 N1(C(CC=C=C)=O)CC(NC(C2SCCCS2)=O)CC2(CC2)C1 C=C1CC2(C1)CC(C(=O)NCCCOCCNC(=O)C(C1CCOCC1)C)C2 C1(C2CCN(C(=O)Cc3ccc(Cl)cc3)C2)(NC(C2CCC2(F)F)=O)CC1 C1(C(=O)NCC2C(C(NOCCC=C)=O)C2)CC=C(C)CC1 C1(NC(CCc2c(C(=O)OC)nco2)=O)CCN(C)C(=O)C1 CCCCC(O)C(=O)NCC1CC(O)CN1C(=O)COc1ccc(Cl)c(CC)c1 c1(C(N2CCC(C)(CNC(C3(CF)COC3)=O)C2)=O)cccc(Br)c1F C(=O)(C1CCCn2cnnc21)NCC(C)CNC(=O)Cc1cccnc1Cl c1(CC(=O)NC2CC(C)(NC(CCOC)=O)C2)cnc(Cl)cc1C C1(NC(CCC(=O)NCCC)=O)CCCCCC1NC(=O)C(CC)CCOC Cc1c(CNC(C2CC(C)(F)C2)=O)sc2cncn12 N1(CCOC)C(=O)NC(c2ccc(C)nc2F)C2=C1CN(C(C)(C)C)C2=O C1(C(F)(F)F)(C(=O)NCC2N(C(=O)Cc3ccns3)CC=C2)CC=CCO1 O=[N+]([O-])c1cnn(C2CC(NCCc3cnccc3F)C2)c1 c1(C(N2C(C)(C(N3CC(C(=O)OC)OCC3)=O)CC2)=O)cc(Cl)nc(Cl)c1 c1(C(=O)OC)ncc(NC(C23CCC2CN(S(=O)(=O)CCCCl)C3)=O)cc1Cl C1(C)(CN(C(CN(CC(=O)NC(C(CCC=C)C)C)C)=O)C)CCS(=O)(=O)CC1 c1(NCC2(OCC)CCOC2)[nH]c(=NCC(C)c2ccsc2)nc2c1cnn2C C1(NC(c2scc(COC)c2)=O)CCC2CCC1OC2 c1(NC(c2c(NC(c3c(C)cn(C)n3)=O)cccc2)=O)ccc(O)c(C(C)C)c1 C(c1ccccc1Cl)=C(C)C(=O)NCC1CCN(C(=O)CCc2ccn(C)c2)C1 C(CCCC(C)(C)C(=O)NNC(=O)c1ccc(C)s1)NC(C(CC)C)=O C(C#Cc1cn(Cc2nccc(F)c2Cl)nn1)NC(C(CC(C)C)=O)=O N1(C(C(C)C2(O)CCC2)=O)CCC=C(CNC(c2ccon2)=O)C1 N1(C(CC(CC)(C)C)=O)CC2CC1CCN2C(c1cnc(C(C)C)s1)=O N1(C(C(N2CCOCC2)C)=O)C2CCC1CC(CNC(=O)CC1CC(F)(F)C1)C2 C1(CNC(c2c(CC(=O)OC)scc2)=O)CN(C(=O)CCC(C)SC)CCO1 C(CS(=O)(=O)CC(=O)OCc1cccc(C)c1)OC.c12ccc(C)c(c1)NC2=O N1(C(c2n(C=C)ncc2)=O)CC(C)(C)OC2(C1)CN(C(=O)CCC(C)OC)C2 Cc1nc2cc(C(=O)NC3CC3c3cn(Cc4csc(Br)n4)nn3)c(F)cc2[nH]1 Cc1cc(N)n(CC(=O)NC2(CNC(C3CC4C=CC3C4)=O)CC2)n1 Cc1scc(C(=O)NCC(CC(C)C)NC(=O)C(N2CCOC2=O)C)c1C C(=O)(C1=CC2(CCOCC2)C1)N1C(CC)CN(C(=O)C(C2CCCC2)OC)CC1 C1(C(=O)NCCCCNC(CCC(C)(C)OC)=O)CC2CCCCN2C1 c1(OC)cnc(CNC(c2ccccc2-c2cccnc2O)CC(=O)O)nc1 N1(C(C2(S(N)(=O)=O)CCC2)=O)CCCC(C2(NC(c3cc(O)no3)=O)CC2)C1 c1(OC)c(N(C2CCN(C(=O)Cc3ccc(Cl)nc3C)C2)C)ncnc1C Cc1nn(C)c(N)c1C(=O)NCC1CCN1C(=O)C(C)CO c1(C(=O)NCC(CO)NC(c2c(C(C)C)onc2)=O)ccc2c(c1)OCC(=O)N2 N1(C(C2(C)CCCN(C(C3CCCCC3(F)F)=O)C2)=O)CCC2(C1)CC2(F)F C#Cc1cc(C(=O)NCC2CN(C(=O)Cn3ccccc3=O)CCO2)ccc1C C1(C)(C(N2CCN(CCN(C(=O)C(=O)C(C)(C)C)C)CC2)=O)CCCNS1(=O)=O CCC(CC)(CC)C(=O)N1CCC(N2CCC(NC(=O)C(C)C(C)C)CC2)C1 C1(c2cn(C3(C(=O)O)CN(C(C4(CO)CCOC4)=O)C3)nn2)CC2(CC(=O)C2)C1 C#CCC(CC(F)F)C(=O)N1CCC2(CC1)CC2NC(=O)CCC1CCCCO1 Cc1ccc(NC(=O)COC(c2cccc(-n3ccc(C)n3)c2)=O)cc1 C1(CC)(NC(c2nocc2Cl)=O)CCCN(C(=O)COC2CCCCCC2)C1 S(=O)(=O)(c1cnc2ccccc2c1)N1CCC(c2ccc(C)cc2)(C)C1 c1(C(=O)NCC(C)CNC(=O)CC(C)n2cccn2)ccc(Cn2cccn2)o1 CC1C(NC(c2cnn(C3CC3)c2)=O)CCN1C(C1CCCSC1)=O C1(F)(C(=O)NC2CC(CNC(c3c(OC)nsc3)=O)C2)C2CCCCC12 N1(C(C(CSC)C)=O)CC=CC1(C)C(N1CCC(CC2CC2)CC1)=O C1(C(=O)NC23CC(CNC(CC4C(C)OCC4)=O)(C2)C3)CN2CCC1CC2 Cc1cc(NC(C2CCC(=O)N(C(=O)C(F)C(C)(C)O)CC2)=O)cc(C)c1C C1(C(C)C)(NC(=O)C(C2(O)CN(C(=O)COC3CCC3)C2)F)CCCC1 C1(C(N(C2CC(NC(c3n[nH]cc3C3CC3)=O)C2)C)=O)Cc2ccc(F)cc2O1 CC(CCNC(C1(CCNC(=O)CC2CC3(CC3)CO2)CCCC1)=O)C(F)(F)F C1(C)(C(=O)NCCC(CNC(c2cc(CO)oc2C)=O)OC)CCC(C)=C(C)C1 N1(C(C(C=CC)O)=O)CC2(CC(NC(C3CCCC(F)(F)C3)=O)CO2)C1 CC1(NC(c2cnc[nH]2)=O)CCCN(C(c2c[nH]c(C#N)c2)=O)C1 c1(C(=O)NCC2N(C(c3cc(C(C)=O)cn3C)=O)CC=C2)cc2n(n1)CC(F)C2 C(=O)(C1=NOC2COCC12)N1CC2(CCN(C(CCCN(C(=O)OC)C)=O)C2)C1 C1(N(C)C(c2nn(C)cc2Cl)=O)CCCC2CN(C(C34CC(F)(C3)C4)=O)CC12 c1(CCNC(C(C)(C)C(C)C)=O)ccc([N+](=O)[O-])cc1Br CCC(C)C(C(=O)NC(C)CN(c1ccnc(C(F)(F)F)n1)C)N(C)C c1(C(N2C3C(NC(C4C(C(=O)OC)C4)=O)C(CC3)C2)=O)ccc(=O)n(C(C)C)c1 C1(CNC(CC(=C=C)C)=O)CC(C)(C)CN1C(c1cnc(C(F)F)s1)=O C1(C(CNC(C(F)=CC)=O)C)CCN(C(c2csc(-c3cccnc3)n2)=O)CC1 C=CC(C)CC(=O)N(C(C)C(=O)NC1CC(N(C)C)C1)C C1(NC(c2cnc(OCC)nc2)=O)CN(C(C23CC(CC(C)O2)C3)=O)CC1(C)C c1(CNC(CONC(c2cc(CCC)[nH]n2)=O)=O)c(C)cccc1Br C1(NC(CC2CC(C)(C)C2)=O)C2CC1N(C(c1ccccc1F)=O)C2 CCC(C)C(O)CC(=O)NC1CC(C(=O)NCC2(C)CCN(C)C2)=CC1O C=CCC(C(=O)NC1CCN(C(=O)Cc2cncs2)C1CC)C(C)C c1(CC(=O)NC2CC(NC(CN(C)C3CC3)=O)C2)cc(C(F)(F)F)ccc1Cl c1(C(=O)NC2CCC(C)N(C(c3ccc(Cl)s3)=O)C2)ncc2c(F)cccn12 c1(NCC2(NC(CSC(C)C)=O)CCOCC2)nnc2c(c1C#N)CCCC2 c1(OC)ccc(-c2nc(C3CCCN(C(C)=O)C3)n(CCS(C)(=O)=O)n2)nc1 c1(C(N2CCC(c3nncn3C)C2)C(=O)NC(C(=O)OC)C)ccc(F)cc1 c1(OCC(N2CCC(NC(=O)C(c3ccc(F)nc3)(F)F)C2)=O)ccc(F)cn1 C1(C(=O)NC(C2N(C(C3N(C(C)=O)CCC3)=O)CCC2)(C)C)CC12CCCCC2 c1(NC)nn(C)cc1C(=O)NCCNC(c1cc(C(=O)OC)no1)=O CC1CCCCC1C(=O)NC(C)(C)CN1CCN(C(=O)C=C2CC2)CC1 Cc1nc(Cl)[nH]c(=NC2CCC3CN(C(c4ncc(F)cn4)=O)CC23)c1[N+](=O)[O-] c1(C(C(=O)N(CC)Cc2nnc(C(C)C)o2)F)ccc(C)cc1 N1(C(c2cnc(SC)n2C)=O)CCN(C(c2coc(C(N)=O)c2)=O)C(C)C1C C(CC1CC1)(C(=O)NCC1(NC(C)=O)CC1)NC(C1(CSC)CCC1)=O N(S(=O)(=O)N1CCC(C)(C)CC1)CC(CCN(C)C)(C)O C(=O)(C(F)C(F)(F)F)NCC1C(NC(c2cnc(=N)[nH]c2)=O)CC1 c1(C(C(=O)NCC=CCNC(CNC(C(CC)C)=O)=O)C)ccc(F)cc1 C(C(=O)NOC1CCOCC1)(c1ccoc1)NC(=O)C(O)CC1CCCC1 c1(CC(=O)OC)ccc([N+](=O)[O-])cc1Br.C1(=O)C(=O)CCO1 c1(CC(=O)NCCNC(C2(C#C)CCCC2)=O)ccc(OC)cc1OC N1(c2nc(-c3ccccc3)cc(C)n2)CC(F)C(N=c2ncnc3[nH][nH]c(I)c2-3)C1 c1(C(C)(C)C)ccc(C(=O)NC2CCC(CNC(c3c[nH]c(=N)o3)=O)CC2)nc1 N1(C(CC(c2scc(C)c2)O)=O)CCC(CNC(C2CC(O)C2)=O)CC1 C1(C(N2C(C3(NC(C(C)CC4CCC4)=O)CC3)CCCC2)=O)CC(S(C)(=O)=O)C1 C(C(=O)NC(c1nc(C(=O)NC2CCCN(O)C2=O)co1)C)(C(C)(C)C)OC C=CCCC(C)(C)C(=O)N1CC(CN(C)C(c2csc(C(C)=O)n2)=O)C2(CC2)C1 C1(C(N(CC(O)CN(C)C(C2CCC3(CCC3)O2)=O)C)=O)CCN2CCCC2C1 c1(CC)ccc(NC(c2cc(OC)ccn2)=O)cc1.C12(F)CN(C1)C2=O C(=O)(CCS(=O)(=O)N(C)C)N(C)CC1CCCN(C(C2(C(N)=O)CC2)=O)C1 c1(C(=O)NCC2C(C)CN(C(C3CCCS3)=O)C2)ncnc(O)c1Br C(=O)(CCCCCNC(C1(n2cnnn2)CC1)=O)NCc1ccc(C)o1 c1(C(N2CCN(C(CN(C(CSC)=O)C)=O)CC2)=O)ccc(O)c(F)c1 N1(C(C2CCC(=O)N2)=O)CCOC2(CCN(C(=O)Cn3ncnn3)C2)C1 c1(CN2C(C(=O)NCc3cccc(CC)c3)CC3CC32)cc(F)c(CO)c(F)c1 c1(CNC(c2cc(-c3ccccc3)cs2)=O)cccc2c1CNC2 N1(C(c2ccc(NC)cn2)=O)CCC(C2CCN(C(c3snc(Cl)c3Cl)=O)C2)C1 c1(C(=O)NC)ccc(Oc2ccccc2NC(c2ccn(C)n2)=O)cc1 C1(C(N(CC(C(C)C)OC)C)=O)(OC)CCN(C(=O)C(C)Cn2ccnc2)C1 C(=O)(C1CCCCc2ccccc21)N1CC(C(C)NC(=O)C2=CCCCC2C)C1 C1(C2CCN(C(=O)C(F)C3=CCCCC3)C2)(NC(C=C(C)C(C)(C)C)=O)CC1 C1(C(F)(F)F)(C(=O)OC)CN(C2CCC(Oc3ccncc3)C2)CCO1 N1(C(C(C(C)C)CO)=O)CCC2(CC1)CCN(C(=O)CCc1ccc(F)nc1)C2 N1(C(CC(CCC)NC(=O)C=Cc2cscn2)=O)CCN2CCC1CC2 Cc1sncc1C(N1CCC(N(C)C(c2cc(C3CC3)no2)=O)C1)=O C1(NC(c2cccc3c2CCCN3)=O)CC1C1CCN(C(=O)CC2CCC2)CC1 N1(C(c2cc(C(C)=O)cn2C)=O)CCCC(O)(CNC(c2ccc(F)s2)=O)C1 c12ccc(F)c(n1)C(=O)N2.c1(OC)nc(CC(C)C)co1 c1(C(N2CC(CNC(C=C(C)C)=O)C3C2C3)=O)cc2ncccc2[nH]1 C1(NC(C(F)=CC)=O)CCCN(C(c2ccc(C)c(N)c2)=O)C1C c1(C(=O)NCc2cccc(C(=O)NC(C#C)CC3CCC3)n2)c(C)cnnc1O N1(CC(=O)NC2(C3N(C(CNC(=O)NC)=O)CCC3)CC2)CCCC(OC)C1=O C12COCC3(CCN(CC3)N(C3CC3)C(=O)CS1)O2.CC(C)CC(C)(C)C c1(C(N2CC3(CN(C(C(C)OCC#C)=O)C3)C2)=O)cnn2c(C)ccnc12 C1(NC(CCOCC)=O)COC2(CCN(C(=O)CSc3cccc(C)c3)C2)C1 C1(C(N2CC(C)(C(=O)NCc3c(C)nsc3)C2)=O)(CO)CCCCO1 CC(CCCCNC(C1CCCN1C)=O)NC(c1c[nH]c(C(N)=O)c1)=O c1(OC)ccccc1NC(=O)C(N1CCCC1CC(N)=O)C1CC1(C)Br C(C(=O)O)(C1=CCC=CC1)C(NNC(Cc1c(OC)cc(Br)cc1)=O)=O Cc1ccc(C#N)cc1NC(C1C2CCC(C2)C1NC(C1CCCCC1)=O)=O c1(C(=O)NCC(C)(C)NC(c2cncc(-c3cc[nH]n3)c2)=O)cc(F)cnc1O C12(CNC(c3ccc(C)nc3N)=O)CCC(CC1)N(C(C1CSCCS1)=O)C2 c1(C(=O)NC(C2(CNC(C(C)NC(CC)=O)=O)CC2)C)cc(C)ns1 Cc1cccc2ncc(C(c3nnnn3C)NCCCC3CCCC3)n12 Cc1[nH]nc2c1CCC(C(N1CCN(C(c3ccc4c(c3)OCC4)=O)CC1)=O)C2 C1(O)(CNC(=O)COCC2CCCC2)CCCN(C(C2CC3CC2CO3)=O)CC1 c1(C(=O)NC2C(CNC(COCC(=O)OC)=O)C2)cccc2nc(C)cnc12 N1(C(c2cc(CC)[nH]n2)=O)CCC(O)(C(C)CNC(c2ocnc2C)=O)C1 C1(CC(=O)NCCn2cccnc2=O)CC2(CC2)CN1C(c1cnn2c1OCC2)=O N1(C(C(C)N2CCC2)=O)CCC(NC(=O)CC(C)(C)CN(C)C)C(F)(F)CC1 Cc1cc(O)ccc1CN(CCc1nn[nH]n1)C(C)C N1(C(=O)OC)CCC(N(C(=O)NC(C)(C)C)CCO)CC1.c1nscc1C c1(CC(N2C(C)(C)CC(C(=O)O)CC2)=O)cc(F)cc([N+](=O)[O-])c1 N1(C(c2n(CC(C)C)ncc2)=O)CCN(C(=O)C(C)O)C(CC(F)(F)F)C1 C(=O)(CC(F)(F)C(F)(F)F)NC(CC=C)CNC(c1cccc(C)c1N)=O CN1CCC(C)(C(=O)NCC(C(C)(C)C)NC(=O)CCc2cnc[nH]2)CC1 CC1CN(C(=O)C(F)(F)c2csc(Cl)n2)CC1NC(=O)C(C)(C)F N1(C(c2c(C)cnnc2)=O)CC(F)(F)CC1(C)CNC(=O)C(c1ccnn1C)O Cc1cc(C(F)(F)C(=O)N(CC(C)N(C(=O)C(C)N(C)C)C)C)cnc1Cl N1(CCC(N2CC(O)(CNC(C(C)c3ccsc3)=O)C2)=O)C(=O)NC(C)(C)C1=O c1(CC)cnccc1NC(=O)NCC=CCOC N1(C(C(F)=CC)=O)CCC(C(C)(O)CNC(c2ccnc(C(F)F)c2)=O)CC1 CCCC(C(O)C(=O)N1CCC1COC)NC(c1cc(C)c(F)cn1)=O c1(C(=O)OC)sc(=NCC2(O)CCCN(C(C3CN(CC(C)C)C3)=O)C2)[nH]c1Cl C(CN=c1[nH]c(=NCCC2CC2)[nH]c2cc[nH]c12)=CCOC c1(C(=O)NCCNC(C23OC(C)C(CC2)C3)=O)cc2nnn(C)c2s1 C12(NC(c3nc(C(C)(C)C)oc3)=O)CCC(CN(C(c3nocc3Cl)=O)C1)C2 N1(C(CC(C)C2CC2)=O)CC2(CCC(NC(C3CCC(C)(C)O3)=O)CC2)C1 O=C(CN=c1cc[nH]cc1)N1CC2CCCC12C(=O)NC1CC(O)(CO)C1 c1(OC)cccc2c1OC(c1nc(C(C)N)no1)C2 c1(C(=O)NC(C(=O)NC2CC(n3cccn3)C2)C2(C)CC2)cc(CO)[nH]n1 c1(C(=O)NC2C(NC(Cc3onc(C)n3)=O)CC2)cccn(CCN(C)C)c1=O Cc1nc(C(=O)N(C(C)CN(C)C(c2cc(C(F)F)on2)=O)C)c(C)o1 C#CC1(C(=O)NC2CCCC2CN=c2ccnc(CO)[nH]2)CCCCCC1 CC1CCN(C(c2cn(C)nc2C2CC2)=O)CC1C Cc1ccnc(C(N2CCOC(CC(=O)NCC(C)C(C)O)C2)=O)c1F C1(NC(=O)CCCF)CCC2(CC1)CCN(C(C13CC1COC31CCC1)=O)CC2 c1(C(N(C2CN(C(C(C(C)C)SC)=O)C2)C)=O)cc2ccc(Cl)cc2c(=O)o1 C1(C(=O)NC(CNC(C2CC(=C)C2)=O)(C)C)(C(=O)OC)C2CCC12 c1(CC(=O)NCC2CCN(C(C3(C)CCOCC3)=O)CC2)cc(Cl)ccc1O n1(CC)nc(C(=O)NCC2(F)CC(CNC(c3c[nH]nc3C)=O)C2)cc1O N1(C(C2CC3(CC(NC(C=C4CCC(C)CC4)=O)C3)C2)=O)CCCC(N=[N+]=[N-])C1 CCCCCC(O)C(=O)NCC(C)CNC(=O)CCCC(C)C N1(C(C2N(C(C(C(C)C)C)=O)CC3CC32)=O)CCS(=N)(=O)CC1 C1(O)(CN(C(CNC(CC(C)C)=O)=O)C)CCN(C(C2CC2(Cl)Cl)=O)C1 N1(C(C(N2CCC(C)(N)CC2)=O)=O)CCCc2cc(OC(F)F)ccc21 N1(C(Cc2c(C)n[nH]c2)=O)CCC=CC1C(=O)N(C)CCn1ccnc1C c1(NC(C=CC(C)NC(=O)C(=O)N(C)C)=O)cc(F)ccc1N1CCOCC1 CCCC(C)CC(=O)NC1CC1CNC(c1cccc(NC(N)=O)c1)=O c1(C2C(C(N(C3CCC(NC(=O)COC4CC=CC4)C3)C)=O)C2)ccccc1F CCCCC(CC)CCC(=O)NCC(C1CCCC1)NC(=O)CCn1ccnn1 O=C(CCCCCNC(c1cccnc1S)=O)NCc1ccc(O)cc1F c1(C(N2CC(NC(c3cc(C(C)(C)C)ncc3)=O)C2)=O)cc2ccc(Cl)cc2s1 c1(C(C)NC(CN(c2ccccc2)C(C=C)C)=O)snnc1C C1(CNC(=O)Nc2c(C(=O)OC)ncc(Br)c2)CCCCC(F)(F)C1 CC1(C)CC(C(N2CCC(NC(=O)CC3=CCOCC3)C(O)C2)=O)CC(C)(C)O1 c1(C(C(=O)NC(CC)C)N2CCC2C2CCCC2)ccc(C(C)C)c(Br)c1 C1(NC(CC(C)c2ccco2)=O)CN(C(=O)CC2CC=CC2)CC12CC2 CCC(C)(C(=O)N1C(C)C2CC1C2NC(c1csc2nnsc12)=O)C(N)=O CC1C(C(=O)NCCC(C)(C)F)CCCN1C(=O)C1=CCCOC1 Cc1c(NCCCNC(=O)N(C)C)ncnc1N1CCN(C)C(c2ccccc2)C1 C(N=c1[nH]c(=NCC2CCOCC2(C)C)c2[nH]ccc2[nH]1)c1c(C)ccnc1 N1(C(c2c(C(C)C)nc(Br)s2)=O)CCC(C2CCCC2C(=O)O)CC1 c1(NC(C2C3CC2N(C(c2cc4sccn4c2)=O)C3)=O)cc2ccccc2[nH]1 C1(NC(C2CCN(C(CC)=O)C2)=O)CCC2(CC1)CC2NC(=O)COC1CCC1 O=C(C1=NOC2(CCN(C(c3ncon3)=O)C2)C1)NCCc1ccc(F)nc1 C1(NC(CCC)=O)(CC)CCCN(C(=O)CC2CCC(F)(F)CO2)C1 C1(C(=O)NCC2C(C)(C)CCN2C(=O)C=CC2CCC2)CCC2(CC1)CC2(F)F c1(C(N(C)CC2N(C(CCc3ccc(C)o3)=O)CCC2)=O)nnc2n1CCCC2 CCCC(CCCNC(=O)C(C1CCCC1)OC)N=c1[nH]nc(CC)o1 C1(CC(=O)NCc2cc(C(C)C)no2)CC(NC(=O)C(F)C2CCCC2)C1(C)C C1(NC(C2(CC)CCC2)=O)CC2CC1CN(C(C1(C(=O)N(C)C)CC1)=O)C2 N1(C(=O)NCC2CC(CO)CO2)CCC2(CCCNC2=O)CC1 N1(C(C2(C(=O)OC)CCCC2)=O)CC(CNC(C2(c3ncco3)CC2)=O)C(C)C1 S(=O)(=O)(c1cc(C(C)C)[nH]n1)NC(COC(CC)C)=O CCC(CC)(CCNC(c1cnc(C(F)(F)F)s1)=O)NC(=O)C(CO)NC(N)=O Cc1ccc(F)cc1C(=O)NC1CC2CCC1N2C(c1cc(N)c(Cl)cn1)=O c1(CN(C(=O)C(O)C2CCC2)C=O)cc(Br)cc(I)c1 C1(NC(=O)C=CC2CCOCC2)CC1C1CCCN(C(C2CCCSS2)=O)C1 c1(CN(C(C(=O)N2CC(OC)C2)C2CCCO2)C(CC)=O)ccc(Cl)c(C)c1 C(c1nc(C)c(C)[nH]1)=CC(=O)NCC1(O)CCN(C(C2C(C=C)CC2)=O)C1 C(=O)(C1=CC(O)C(NC(=O)CCCC2CCCC2)C1)NCC1CCC(=O)NC1 C1(c2nnnn2CCC2(C)CC2)(NCC2CC(C(C)(C)C)C2)CCSC1 C1(NC(c2c(OC)c[nH]n2)=O)CCCN(C(=O)Cc2ccsc2C)CC1 C1(C(N(CCNC(c2cccc(CF)c2)=O)CC)=O)CCC2C(C1)C2(F)F C1(C(=O)NCC(C)(O)C2CCCC2)CCCCN(C(=O)CCCCC2CC2)C1 c1(SCC(=O)NC(CC)CN(C)C(C2CC(C)(F)C2)=O)ccc(Cl)cc1 c1(C(N2CC(O)(CNC(c3cnc(CC)[nH]3)=O)C2)=O)ccc2nn[nH]c2n1 C(=O)(CCCCCNC(C1CC2CC1CC2O)=O)NCc1nc(C)c(C)o1 C1(C(=O)NC(C2(OC)CCC2)C)C2CCN(C(c3cc(O)cc(F)c3)=O)CC12 C1(OCCCNC(C(CC)n2ccnc2)=O)CCN(C(C2(C)C=CCC2)=O)CC1 c1(C(=O)NCC(C)NC(C(F)=CCC)=O)cccc2c1CCC2 C1(OC)CN(C(c2ccc(C)n2C)=O)CC1NC(=O)C(C)NC(N)=O C(CC(=O)N1CCN(C(=O)CNS(=O)(=O)C2CC2)C(C2CC2)C1)(C(F)(F)F)OC C1(CC(=O)NC2CC(OCC(=O)NCCCOCCC)C2)CSCCO1 C1(NC(C2C(C=C)C2)=O)CCC(N(C(=O)CSCCC)C)C1 c1(C(N(CCC)CCNC(=O)C(CC)CC)=O)cc(CNC(N)=O)ccc1Cl O=S(=O)(c1ccc(NC2COCC2O)cc1)Nc1cccc2c1COC2=O c1(CCNC(NC(C#C)CCC)=NCC)c[nH]c2cc(Cl)cc(Cl)c12 c1(NC(C2C(OC)CCN(C(=O)OC(C)(C)C)C2)=O)cc(I)c(F)cc1F CCCC(C#N)C(=O)N1CC2CC2(CNC(c2cc(Br)ncc2OC)=O)C1 N1(C(CCOCCC)=O)C2CCC1CN(C(C1CC=CCO1)=O)CC2 c1(C(=O)NCC(CN(C(=O)Cc2ccon2)C)O)ccc(OC(F)(F)F)cc1F N1(C(c2c(C)con2)=O)CCCN(C(c2cccc(CN(C)C)c2)=O)CC1C N1(C(CCc2ccc(C)nc2)=O)CC2(CC(NC(c3ccsc3C#N)=O)C2)C1 C1(O)(C(=O)NCC2CCN(C(=O)CCc3nccs3)C2)CN2CCC1CC2 Cc1ccc(O)c(CN2CCC(F)(C(=O)NCc3cccc(F)c3)C2)c1 CC1=C(C(=O)NCc2nc(C(=O)NCC3(CO)CCCCC3)c(C)o2)COCC1 C1(C(=O)NC(c2c(C)cccn2)C)CC2(CCC2)CN1C(=O)CCS(N)(=O)=O c1(CNC(C(C=C)O)=O)ccc(CC(C)NC(c2csc(CO)n2)=O)cc1 C1(NC(C2(OC)CCSC2)=O)CC(F)CN(C(=O)CC2CCCC(F)(F)C2)C1 c1(N2CCC(CNC(=O)C(c3ccc(Cl)c(Cl)c3)CO)CC2)nc(Cl)ncc1Cl Cc1nc(C(=O)NCCCN(CCCNC(c2cnc(C(C)C)[nH]2)=O)C)c(C)o1 C(=O)(C1CCCc2ccnn21)N1CC(CNC(Cc2n(C)ccn2)=O)OCCC1 c1(NC(C(N2CC(CC)OC(C)C2)=O)=O)ccc(S(C)(=O)=O)nc1 C1(C(N(CC(CC)NC(=O)C(S(C)(=O)=O)C2CC2)CC)=O)CCC(O)CN1C Cc1nn(CC(=O)NCC2(C)CCCN(C(C34C=CC(CC3)C4)=O)C2)c(C)c1C C1(C(=O)NCC(CC(C)C)NC(C23COC(CCO2)C3)=O)C2(CCC2)C12CCC2 C1(NC(C(COC)C)=O)CN(C(c2cc(Cl)cc(Cl)c2O)=O)C2(CCOCC2)C1 N#Cc1ccc(Cc2noc(C3CC(OC(F)F)C3)n2)cc1 C1(CC(=O)N(C(C2CCCC2)C)C)CCCN1C(=O)CCc1cnn(C)c1 c1(C(N(CC(O)CNC(=O)CCC2CC2CC2CC2)C)=O)ncn2ccccc12 CC(C)(C(=O)NC1CCC1NC(C1COC(=O)N1)=O)c1ccsc1 C(CCS(C)(=O)=O)(C(=O)NC(C)(C)CN(C)C(C1CC1C(C)(F)F)=O)OC N1(C(c2c(C)nc(CC)o2)=O)CCCC(C(N2CCCC(CCO)CC2)=O)C1C C1(NC(C(C)O)=O)CS(=O)(=O)C12CCN(C(C1Cc3cncn3C(=O)N1)=O)CC2 c1(C(CC(C)NC(=O)NCC2(F)CC(C(=O)OC)C2)=O)ccc(F)cc1 N1(C(COC2CN(C(COCCCN(C)C)=O)C2)=O)CC2(CO)CC2(CO)C1 C1(c2n(CCCOC)nnn2)(NCc2cccc(C)c2CO)CCC1C1CCC1 CC1(C)CC(CC(=O)NC2(C)CC3(CC3)C2)N(C(=O)C2=COCCC2)C1 c1(C(N2CCC(N(C)C(c3cc4sccc4[nH]3)=O)C2)=O)ccc([N+](=O)[O-])cc1F C(=O)(C(F)CC(C)(C)NC(c1cnc(=N)[nH]c1)=O)N(C)Cc1cc[nH]n1 C1(NC2CC(C(=O)OCC)CC2O)CCC2C3C=CC(C3)C12 C(CC(C)C)(C(=O)NC1CN(C)CCC1O)NC(c1ccc(OC)o1)=O C1(NCCc2nc(CC)on2)CCCCN(NC(c2cnn(C)n2)=O)C1 c1(C(=O)NCC(c2c(OC)cccc2)O)ccc(Br)c(C)c1C C1(c2scc(CC(=O)OCC)n2)CCCN(C(=O)NC(C)C)C1 C(=O)(CS(N)(=O)=O)N(C(C)CNC(=O)C(c1cscn1)N(C)C)C c1(CC)nc[nH]c1C(N1CC(F)(CNC(=O)C(C)Cc2cnc[nH]2)C1)=O c1(C(=O)NC(CC=C)CNC(=O)Cc2occc2C)cc(C)ccc1 C1(NC(C2CCCN(C)C2)=O)CC2CCC1N(C(=O)CC1CCC(F)(F)C1)C2 c1(C(=O)NC2CCCC(NC(Cn3nc(C)oc3=O)=O)C2)cc([N+](=O)[O-])oc1C CCC(C)C(O)C(C)C(=O)NC(CC(=O)N(C(C)CCO)C)C(F)F CC(C)C(C(=O)NCc1ccc(C#N)o1)C(C)NC(C1CS(=O)C1)=O Cc1ccc(NC(=O)C(=O)N(c2cn(C)nc2O)Cc2ccccc2)c(F)c1Cl n1(CC)nc(C(=O)NC2CCOC(C(=O)NCc3cc[nH]n3)C2)cc1O Cc1cccc(N(C)C(=O)Nc2cn(C(C)(C)C)nc2C)c1C Cc1cc(NC(=O)C(CC2CCOCC2)NC(=O)CC2CSCCO2)cnc1Cl c1(C(=O)NCC2(F)CN(C(C(C(C)(C)C)=O)=O)C2)ncccc1S(C)(=O)=O Cc1ccc(N2CCN(C(=O)C(=O)NC3CCCC3(F)F)CC2)cc1N N1(C(C(=O)NCC23CC(F)(CO2)C3)=O)CCC(C2CC2)C1 c1(C(=O)NCC(CN(C(=O)CC2(C)CCCO2)C)O)cc([N+](=O)[O-])c[nH]1 Cc1cc(C)n(CC(=O)N(C2CNCC(C)(C)C2)c2ccc(F)cc2)c(=O)n1 CCCCCCCC(=O)N(CC(CC)NC(c1c(F)ccc(F)c1Cl)=O)C C(=O)(C#CC1(CC)COC1)N1CC(C(C(=O)NC(CCC=C)CO)O)C1 C1(C(N(C(CNC(c2c(C)onc2)=O)C)C)=O)OCC2CCCC12 C1(NC(c2cc(C(C)=O)on2)=O)CCCN(C(=O)CCC(=O)N(C)C(C)C)CC1 N1(S(CC2(COC)CCOCC2)(=O)=O)CCC12CCOC(C)(C)C2 C1(NC(C(c2cn(C)nn2)NC(c2csc(O)n2)=O)=O)COCC1(C)C CCCC(O)CC(=O)NCCCC(C)NC(c1ccc(C#N)o1)=O c1(C(=O)OC)ccc(Br)nc1NC(c1ccc(-c2ccsc2)nc1)=O C1(C(N(C2CCN(C(=O)C=C(C)C)C2)CCC)=O)CC2(CCCCO2)C1 Cc1cnc(N)c(C(=O)NCC2CCN(C(c3cnc(C4CC4)s3)=O)CC2C)c1 C(=O)(C1CCCc2nnn(C)c21)NC(C)CNC(C1(c2ccccc2)CC1)=O C(=O)(CC(C(F)F)NC(=O)C(F)C(C)(F)F)NC(C(=O)N(CC)CC)C N1(C(C(CC)C#N)=O)CCC2(CC1)CC(CNC(C1(OCC)CCCC1)=O)C2 S(=O)(=O)(c1c[nH]ccc1=NCC1CC2(CC2)C1)NCCCCCC=C CC1CC(NC(C2(C)CCOCC2)=O)CN1C(c1ncncc1F)=O N1(C(C2(CC)CCCC2O)=O)CCCN(C(=O)C(=O)Nc2ccc(C)cc2)CC1 c1(C(N(CCC(=O)NCCCCCN(C)C(C)C)C(C)C)=O)cc(F)ccc1O C(=O)(CC(O)C(C)CC)NCC(=C)CCNC(c1ccccc1CO)=O c1(-c2[nH]c(C)c(C(=O)O)c2C(=O)N=c2cc(C)n(C)[nH]2)ncnc2cccc(F)c12 c1(C(=O)NC(CC)CNC(=O)C(O)COCc2ccccc2)cc(Cl)c(Cl)s1 c1(C(=O)NCC(CO)NC(CCCC(=C)C)=O)cc2ccc(O)nc2s1 c1(NC2CC(C)N(Cc3ccccc3)CC2)cccc2cccc(Br)c12 c1(C(C(=O)NCCCN(C(C(C2CC2)OCC)=O)C)C)ccc([N+](=O)[O-])cc1F C(=O)(CCN1CCCCO1)N1CC2C(CN=c3n(CCOC)[nH]nn3)CC(C2)C1 N1(C(CC(CC)C(F)F)=O)CCCC2(C1)CN(C(=O)C=Cc1cc[nH]n1)CCO2 C1(NC(C(C)OCC)=O)CN(C(=O)C(c2ccc(OC)cc2)(C)C)CCC1F N1(C(COCCSC)=O)CCC(C(C)(C)CNC(C2CNC(=O)C2)=O)CC1 S(=O)(=O)(c1ccc(Br)c([N+](=O)[O-])c1)NCc1ncn(C)n1 C1(CC)CCCN(C(c2cnccn2)=O)C1C(=O)NCCOc1ccccc1 C=CCC(CC)C(=O)NC12CCC(C1)N(C(C1CN(C(=O)CCCCO)C1)=O)C2 O=C(C#CC1CCC1)N1CCN(C(=O)CCc2ccc[nH]2)C(C(F)F)C1 c1(C(=O)NC(CN(C(CNC(CCCCC)=O)=O)C)C)nc(OC)ccc1OC CCC(CC(=O)OC(C)(C)C)NC(c1ccnc(-n2cccn2)c1)=O C1(NC(C(C)=CC(C)(C)C)=O)C=CCCC1C(=O)NCCC=CCCC Cc1ncc(Br)c(C(=O)NC(C)C(C)NC(=O)Cn2cn[nH]c2=N)n1 CCC(C)CC(=O)NC1CCC1CNC(C1CC(CC(C)(C)C)C1)=O C1(CNC(Cn2nnc(C)n2)=O)CC(C(F)(F)F)CN1C(C1CCNC1=O)=O C12(NC(c3c(C)con3)=O)COCCC1CN(C(=O)CNc1ncccn1)C2 N1(C(C=C(C)C(F)F)=O)CC(NC(c2coc(O)n2)=O)CC12CCOC2 C1(C(N2C(C)CN(C(=O)CN3CCS(=O)(=O)CC3)CC2)=O)CC2C=CCC(C1)C2 C(c1cncc(F)c1)=CC(=O)NC1(C)CN(C(Cn2c(C)ccc2C)=O)C1 C1(c2n(CC)c(N(C)CC3(OC)CCC3)nn2)CNC(=O)CC12CCC2 C(=O)(C(C)CC(C)C)N1C(C2CCN(C(c3c(Cl)cc(C)s3)=O)C2)CCC1 C1(NC(CCSC)=O)CCN(CCNC(c2csc(-c3nc[nH]n3)n2)=O)CC1 C1(O)(C(=O)NCC2(CNC(=O)C(O)c3ccco3)CCOCC2)CCCCCC1 N1(C(CCC=C(C)C)=O)CC2CC1CN(C(=O)CCC(C)O)C2 c1(OCC)ccc(CNC(c2ncc(Cl)n2C)C2CCCCC2)cc1 C(=O)(C1CCCc2nn[nH]c21)NC1C=CCN(C(c2cc(CC)no2)=O)C1 c1(C(=O)NC(C)CNC(c2cnc3ccsc3c2)=O)ccc2c(c1)C(=O)NC2=O C(C(C)(C)CCNC(C1(CCNC(c2ccco2)=O)CC1)=O)N(C)C N1(C(C2CCC(C)(CC)O2)=O)CCCC(NC(c2cc(Br)co2)=O)CC1 c1(SC)ccc(Cl)c(C(N2CC=CC(NC(C3CC(C(F)F)C3)=O)C2)=O)c1 CCC(CC)C(C)C(=O)NCC1(C(=O)NC2CC(n3cncn3)C2)CCC1 C=CCC(C(=O)NC(C)(C)C(C)NC(c1csc(S)n1)=O)c1ccccc1 Cc1ccc2cccc(C(=O)NCCC3CC(NC(c4sncc4C)=O)C3)c2n1 C(CCCC)(C(=O)N(CCF)CCOC)NC(C1C(=C)C1)=O CC(N=c1[nH]c(=NCC(C)c2cccc(O)n2)c2cccc(F)c2[nH]1)c1cccs1 N1(C(c2occ(C)c2)=O)CC2(CCC2NC(c2cc(-c3ccc(Cl)s3)on2)=O)C1 C(=O)(C1CCc2cccc(OC)c21)NC(CCN(C(CC(=C)C)=O)C)C(C)(C)C c1(C(N(C(C)CCNC(=O)CC2C=CCCC2)C)=O)ccc(N)c(O)c1 c1(C(N2CCC(C)C(C(=O)OC)C2C)=O)ccc(Br)c2cn[nH]c12 C#CC1(C(=O)NCC2CC(C(C)C)C2)CN(C(=O)Cc2cn(C)cn2)C1 c1(C(=O)NCc2ccc(CNC(C(C)SCCCC)=O)cc2)ncc(F)cc1C C1(NC(c2c(COC)nn(C)c2)=O)C2CC3CN(C(=O)C(C4CC4)SC)C1C3C2 c1(C(=O)NC(C)(C)CNC(c2ccc(Cl)o2)=O)nnn2c1CCCC2 N1(C(C(F)=CC)=O)CCCC(O)(CCNC(C2(OC)CCCCC2)=O)C1 c1(C(=O)NCC(CC)NC(=O)C(c2cccc(OC)c2)OC)cncn(C)c1=O CCCC(C)(C)C(=O)NC1CC1CNC(c1ccnc(OC(F)(F)F)c1)=O c1(CCC(=O)NCC(CCCCC)CO)nc(O)c2ccccc2n1 c1(CN2CC(NC(c3cc(Cl)nc(Cl)c3)=O)C(F)C2)cccc2cc[nH]c12 N1(C(C(Cn2ccc(C)n2)C)=O)CC(NC(c2csnc2C)=O)CC(C)C1 c1(SCC2(C(N)=O)CN(C(C3(C(=O)NC)CCC3)=O)C2)ccc(Cl)cc1 Cc1nc2cc(C(=O)NCC(O)CNC(=O)CC3CCSCC3)cc(O)c2o1 c1(NC(C(C(C)C)NC(c2cocn2)=O)=O)ccc2c(c1)CCO2 C12(C(N3CC(NC(c4cc(C(N)=O)cc(C)c4)=O)C3)=O)CCOC1CCOC2 N1(C(CCCCSC)=O)CCCC1C1CCCCN1C(=O)Cc1cc(C)on1 C12(C(N(CC(CC)(C)OC)C)=O)CCN(C(c3c(Cl)cnn3C)=O)CCC1C2 C1(NC(Cc2c(C)ccc(C)c2)=O)CCC(O)CN(C(C2CC(C)(C)CO2)=O)C1 c1(OC)cc(F)cc(C=CC(=O)N(CCNC(c2cc(C#N)on2)=O)C(C)C)c1 Cc1nnc2n1CCCC2C(=O)N1CCC(NC(=O)C2=COCCO2)C12CC2 N1(C(C(C)SCC)=O)CCN(C(=O)CCc2ccoc2)CC1C1CCC1 c1(C(N2CCC(NC(C3CCSC3)=O)C(O)C2)=O)ccc2c(O)nnc(O)c2c1 Cc1nccc(CCC(=O)N(CCCN(C)Cc2cn(C)nc2C(F)F)C)n1 c1(CC(N2CCC(CNC(C(CCC)OCC)=O)C2)=O)cccc(F)c1O c1(NC(CCNC(c2nc(C)nc(O)c2)=O)C)ncc([N+](=O)[O-])cc1C#N c1(C(=O)NC2(CNC(CCCCC=C)=O)CC2)ccc(N=S(C)(C)=O)s1 CC(F)(C(=O)NC1CCCC(CNC(c2cnc(Cl)c(N)c2)=O)C1)C(F)(F)F N1(C(=O)C=Cc2cnco2)CCC2(CCCN(C(c3[nH]cc4c3CCC4)=O)C2)C1 N1(C(C=CC(C)(C)SC)=O)CCCC2CN(C(C3(C)C(C)(C)C3(C)C)=O)CCC12 N1(C(c2nn(CC)c(C)c2)=O)CC2CCC2(CNC(=O)CCC(=O)NC)C1 C(=O)(C(C)C(=O)c1ccc(Cl)cc1)Oc1nnc(-c2c(C)ocn2)o1 C1(C)(C(N2CC(NC(C3(C#N)CC(C)C3)=O)C(C(F)F)C2)=O)C(C)(C)C1(C)C Cc1nc2cc(C(=O)NCCC(C)N(C(=O)CC3CCCO3)C)ccc2n1C CC1(C)CCC(C(N2C3CCC2C(CNC(C2CCCSC2)=O)C3)=O)CO1 N1(C(C(C=CC)O)=O)CC(NC(c2cnn(CCC(C)C)c2C)=O)CC(F)C1 c1(C(=O)NCC(C)N(c2nnc(C3CCCC3)s2)C)csc(C(N)=O)n1 Nc1c(C(=O)NCCCCNC(C23CC(O)C2C3)=O)nnn1-c1ccccc1 N1(C(=O)C(O)Cc2ccc(Cl)cc2)CC2CCCC2(NC(C23CC(F)(C2)C3)=O)C1 C(=O)(C1CCc2c[nH]nc21)NC(C(C)C)CCNC(c1cc2c(ncn2C)s1)=O CCCCC(CC)NC(=O)CC(CNC(c1ncsc1NC)=O)OC C1(O)(C(C(=O)N(C(CSCC)C)C)F)CN(C(=O)COC(C)=O)C1 C1(C(N2CCC(C)(NC(c3cnc(Cl)s3)=O)C2)=O)CC2CCCCCC12 c1(SCC#C)cccc(C(=O)NC(C)CCCCNC(=O)CC2(C)CC2)c1 CC(C(=O)NCCN1CCC(NC(=O)CCS(C)=O)CC1)C(C)(C)O C(=O)(C1Cc2ccccc21)N(CCN(C(C)C)C(C1CC2(CCC2O)C1)=O)C Cc1cc(C)c(C)c(C(=O)NC(CNC(C2(C)CCCCCC2)=O)C2CC2)c1C c1(SC)nc(C(N2CCC(F)(CNC(=O)C=CC3CCC3)C2)=O)c2ccccn12 c1(C(N2CC(NC)(COC)C2)=O)sc2cccc(F)c2c1COC CC(C)(C)C(CNC(C1(n2ccnn2)CC1)=O)NC(C1(C)CNC(=O)C1)=O c1(C(C(=O)NC(CC)C)N(C)CNC2(CO)CCC2)cnc(OC)cc1OC CC1(C)CC(NC(C2CCS(=O)(=O)C2)=O)CCN(C(=O)COCCCF)C1 N1(C(C(CC)F)=O)CC(NC(c2cnoc2-c2ccccc2)=O)CC12CCC2 c1(CC(=O)NCCC(C)(C)CO)c(C(F)(F)F)cccc1C(F)(F)F c1(OCCC(=O)NCC2(F)CC(NC(C3CCC(C)O3)=O)C2)ccc(F)cc1Cl CC1(C(=O)NC2CC2CNC(=O)COc2ccc([N+](=O)[O-])cc2)CCS(=O)(=O)CC1 c1(C(N(CCCNC(=O)C(O)c2ccco2)C(C)C)=O)ccc2c(c1F)NCC2 C(C#Cc1ccc(F)cc1)N1C2C(NC(c3ccc(C)n3C)=O)(CCC2)CC1 N1(C(C2CCC(C(N)=O)C2)=O)CCCC(C)C1CNC(c1[nH]c(=NC)sc1)=O C1(C(=O)NCCOCC(N2CCC(C(C#C)C)CC2)=O)CCCC(C#N)C1 N1(C(C=C(C)c2cccnc2)=O)CCC2(CC1)CC2NC(C1CC1(C)C(F)F)=O c1(SC)cc(F)ccc1C(=O)NC(C)CCCCNC(C1CN(C)C(=O)N1)=O CC12CSCC1CN(C(c1ccc(CNC(c3cc[nH]n3)=O)cc1)=O)C2 C1(C(=O)NC2C(CNC(c3c(C)nco3)=O)CC2)CCCCN1N=O Nc1ncc(F)cc1S(=O)(=O)NCC1(CF)CCNC1 C(C)(CCC(=O)NCC1CCCN(C(=O)C(c2cccc(C)c2)C2CC2)C1)OC C12(CNC(c3c(C)nn(C)c3)=O)CCCC1CCN2C(c1nccn1C)=O c1(C2(C(N3CC(NC(c4csnn4)=O)(CO)C3)=O)CCC2)ccccc1F N1(CC(N2C(C(=O)NCCNC(=O)OCC)CSCC2)=O)CC(=O)CCC1=O Cn1cc(Cl)cc1-c1nnc(N2CCCC(CF)C2)n1CC1CC1 CCCCC(C(=O)NC1(CNC(=O)C(F)=CC2CC2)CCC1)C(C)C Cn1ccc(S(=O)(=O)N2CC3CCN(C(=O)Cc4ccccc4Br)C3C2)n1 Cc1ncc(C(=O)N(C)CC2CCCN2C(C23CCCC2C3(F)F)=O)cc1C#N C(=O)(CCCC(=O)OC)NCCCNC(C(C(=O)NC)C)=O C1(NC(c2nc(CCC)oc2)=O)CN(C(=O)C(CC)SC)CC12CC2 S(=O)(=O)(c1cc(C(F)(F)F)cc(O)c1)N1CC(c2nc(C(C)C)on2)OCC1 Cc1cc(Cl)c(C(=O)N(C2CCC(NC(=O)Cc3nccs3)CC2)C)s1 CC1(NC(=O)C(C2CCOCC2)F)CC(C(=O)NCC(N2CCCC2)=O)C1 CCC(CO)C(=O)NC(C)CC1CCN(C(C23CCC(C2)OC3)=O)CC1 c1(C(C)NC(c2nnnn2C)C2CC(OCOC)C2)cccc(F)c1C N1(C(CCNC(=O)NC)=O)CCC(NC(=O)Cc2cccs2)C1C(C)(C)C N1(C(CN(C)C)=O)CC(NC(c2cc(Cl)nc(Cl)c2)=O)CC2(CC2)C1 N1(C(c2ccc(COC)[nH]2)=O)CCC(C)(C)C(CNC(=O)CC2(C)CC2(F)Cl)C1 c1(C(=O)NCCC2(CNC(C3(CC)COC3)=O)CC2)cc([N+](=O)[O-])cc(C)n1 CCCC(O)C(=O)N1CCC(N(C(c2ccc(C(C)(C)C)cc2)=O)CC)C1 C1(NC(c2c(OC)nn(C)c2)=O)CCN(CCOCC(C)(C)CCO)CC1C C1(C)(CNC(c2c(C)coc2C(C)C)=O)CC(F)(F)CN1C(=O)CC1CCCC1 c1(SCC)ccc(CC(=O)NC(CN(C)C(c2cc(Cl)no2)=O)CC)cc1 Cn1cc(C(=O)NC(COC(=N)O)Cc2ccccc2)c(C(F)(F)F)n1 CN1CCCCC1CC(N1CC(C)(NC(=O)CC(c2cccc(F)c2)O)C1)=O C1(CC(=O)NCCCC(=C)C)C2CCCC2N1C(=O)C(C1CCOC1)OCC c1(C(=O)NCC(CC)NC(=O)Cc2csnn2)cccc(OC)c1 N1(C(c2ccc(CC)s2)=O)CC(C)N(C(=O)C(C)CC(N)=O)CC1C Cc1occc1NC(=O)NCCCN(C(C)C(O)Cc1ccccc1)CCO N1(C(C=COCC)=O)CC2CCCC2(NC(c2c[nH]c(=N)cc2C)=O)C1 Cc1ccc(CO)c(NC(c2cc(C)nn2C2CCOC2)=O)c1 C1(C(=O)NC(CNC(C(=Cc2cnc[nH]2)C)=O)(C)C2CC2)CC(C(C)C)=NO1 N1(C(c2cnc(C(C)C)s2)=O)CCC(NC(=O)C2CC2)C(C)C1 c1(CN2CCC(CNC(c3cccc(CCC)c3)=O)C2)c[nH]c2cc(C)ccc12 C1(C(=O)NCc2scc(C)c2)CCN(C(=O)Cc2ccn(C)c2)C12CC2 N1(C(CSCC#C)=O)CCCC2(CCC(NC(=O)C(C)(C)C3CCCCC3)C2)C1 C1(CNC(c2cc(OC)ns2)=O)CCC(C)CN1C(=O)CCSC1CCCC1 c1(C(N2CC3(N(C(C(C)CO)=O)CC3)C2)=O)ccc(S(=O)(=O)NC(C)(C)C)cc1 c1(C(N(C2C3CC(NC(=O)C(O)CN4CCCC4)CC23)C)=O)cccc(O)n1 c1(C(=O)NCC2N(C(C(F)OC)=O)CCC2)cncc2c1CCNC2=O c1(C2N(C(C(=Cc3ccccn3)C)=O)CCC2)nnc2n1CCOC2 c1(C(N2CCC(CNC(C3CC=CC3)=O)C2)=O)cccc2c1OCCO2 CC1CC(C(=O)NC2CC(CCNC(=O)CC3(O)CCCCC3)C2)CC(C)O1 c1(OCC)ncc(NC(C2(CCNC(c3cnc(Cl)n3C)=O)CC2)=O)cn1 N1(Cc2ncc(OC)nc2)CCC2(CC2C(=O)Nc2ccnn2CCO)C1 c1(SC)cccnc1Cl.C1C(C)C(=O)N2CC(O)(C2)CN1C(c1cccnc1)=O Cc1ccc(CN=C(NC(C)C)NCC2CCCC2NS(C)(=O)=O)c(C)c1 c1(C(=O)NCC(=O)NCC(=O)N(C2(C(=O)OC)CC2)C)cc(C)n(C)n1 C1(F)(C(N(C2(CCO)CC2)C)=O)CCCN(C(=O)C(F)=CC2CC2)C1 CC(C)(CC(=O)NC1(CNC(=O)C(c2cc(F)cc(F)c2)O)CCC1)C(F)(F)F c1(OCc2c(C)nc(CC)s2)nc(N2CCOCC2)ncc1Cl CCC(C)CC(=O)C(=O)NC(C(=O)NC1(c2cc[nH]n2)CC1)C1CCC1 N1(C(c2c(C)n(C)cc2)=O)CCC2(CC2)CC1C(=O)NC1(C(N)=O)CC1 c1(NCC=CCNC(CCCC)=O)c(C(=O)OCC)cc([N+](=O)[O-])cc1F C(=O)(C(C)S(N)(=O)=O)N1C(CN(C(CS(CC)=O)=O)C2CC2)CCC1 N1(C(c2cc(CC)on2)=O)CCc2ccccc2C(NC(=O)C(C)C2CCC2)C1 N1(C(CC2CCN(OC)CC2)=O)CC2CC(C)N(C(=O)Cc3csc(S)n3)C2C1 CC(O)C(=O)NNC(=O)N(C1C(C)(C)C1(C)C)C(c1cn(C2(n3cccn3)CC2)nn1)C C(=O)(CC1CCOc2ccccc21)NCCCN(C(C1C(C)C1)=O)CCO N1(C(c2cnc(C(F)F)nc2)=O)CCC2CN(CC3CCC4(CC3)CC4)CC12 C1(CNC(CSCCC)=O)CCCN(C(c2nc(C)ncc2Cl)=O)CC1 c1(OC)cc(C)sc1C(N1CC(CCCCNC(=O)C(C)=CC2CC2)C1)=O N1(C(CC(CCC)CC)=O)CCCC2CN(C(C3CC4(CCOC4)C3)=O)CC12 C12(NC(CC(CC)(C)C)=O)CCN(C(c3cc[nH]c4nccc3-4)=O)CCC1C2 c1(C(N(C(CNC(c2cc(OC)c(F)cc2)=O)C)C)=O)ccc2c(c1O)CCC2 C1(C(=O)NCCOC2CCN(C(CSCCN(C)C)=O)C2)OCC2CCCC1C2 N1(S(C)(=O)=O)CCCC(NCc2cnc(C3CCNCC3)[nH]2)C1 N1(C(CCCCC(C)C)=O)CCCCC12CC(NC(C1CCCCC1(C)C)=O)C2 N1(C(C=C(CC)C)=O)CC(NC(c2cnoc2-c2ccccc2)=O)C(O)C1 C#CCC(CC(F)F)C(=O)NC1CCCCC1NC(=O)C(N1CCOCC1)C CC1OCCN(C(=O)CCN2CCC2)C1C(N1CCCC(C)CC1)=O Cc1ccc2c(c1)C(NC1C(C(F)(F)F)C1C(F)(F)F)CCC2 C1(NC(=O)CCCc2cccc(Cl)n2)CN(C(c2cnc[nH]2)=O)CCC12CCC2 C1(C)(C(=O)NC)CCN(CC(=O)NC(CC(C)C)C(N)=O)CC1 c1(OC)cc(C(N2CC(C(=O)NCC3CCCOC3)C(F)C2)=O)ncn1 C1(CNC(c2cc(CC)ncc2)=O)CCCC2CN(C(=O)C(C)(C)C#N)CC12 c1(C(N2CC3(N(C(C4(CC)CC4)=O)CC3)C2)=O)[nH]nc2ccncc12 Cc1cc(C(=O)NC2CN(C(c3ccccn3)=O)CCC2F)cc(Cl)c1 S(=O)(=O)(c1ccc(NC(CO)C2(C)CC2)c(C#N)c1)NCC(C1CCCCC1)C c1(C2C(C(=O)NCCCCNC(=O)CC3(N4CCCC4)CC3)C2)ccc(F)nc1 S(=O)(=O)(c1c[nH]c(=NCCCN(c2ccc(Br)cn2)C)cc1C)N(CCOC)C N1(C(C(C)(C)CCC#N)=O)CCOC2CN(C(C3CC4C=CC3C4)=O)CC12 C1(F)(C(N(CCCNC(CN(C(=O)OC)C)=O)CC2CCCC2)=O)C2CCCCC12 C1(CNC(C=C2CCC(C)C2)=O)CN(C(=O)Cc2cc(Cl)n(C)n2)CCC1(F)F C1(NC(c2cnc(O)o2)=O)CC2(C1)CC(CNC(C1CC3CCC1O3)=O)C2 C1(CCOC)(NC(c2cc(C)sc2C)=O)CCN(C(=O)Cc2csc(C)n2)C1 c1(NC(C)=O)cccc(F)c1C(=O)NCC(O)CNC(=O)C(C)n1ccnc1 C1(C(N2CC(n3cc(SCc4cc(OCC)n[nH]4)nn3)C2)=O)CC(C)CC(C)C1 C(=O)(CC(C)CC(C)C)N(C1CC(C#N)C1)CC(=O)NC(CCCC)(C)C C(=O)(CC1COc2ccccc21)NC1CC(NC(C(C)C#N)=O)C1 N1(C(C2CCN(C)CC2)=O)CCOC(C)(CNC(C2(S(N)(=O)=O)CCC2)=O)C1 C1(C(=O)NC(CC)CN(C)C(C2CCCCN2C)=O)CCC([N+](=O)[O-])CC1 c1(C(=O)NC(C2CCN(C(c3c(CC)scc3)=O)C2)C)cnc([N+](=O)[O-])n1C c1(OCC(=O)NC2(CNC(=O)C(O)CF)CCOC2)ccc(Cl)cc1Cl N1(Cc2cnc(C)o2)CC2CCN(C(C34CC5CC(C(=O)N3)C4C5)=O)CCC2C1 C#CC1(C(N2CCCN(C(C3CC=CC3)=O)CC2)=O)CCCCC1 N1(C(CC=CC=C)=O)CCC2(CC1)CC2C(N1CCC(C)C1(C)C)=O NS(=O)(=O)C1(C(=O)NC2CCC2NC(C2(Oc3ccccc3)CC2)=O)CCC1 CSC1=C(C(=O)N2CCC3(NC(=O)CN4CCCCCC4)CC3C2)CCCC1 C1(NC(c2c(F)cccc2F)=O)CN(C(C2CC(C(F)F)C2)=O)CCC1CO c1(CC(=O)NCC2(CCNC(CC3CC(=C)C3)=O)CC2)coc2cc(C)ccc12 C1(C(N(C)CC2(NC(c3csc(=N)[nH]3)=O)CC2)=O)CCC(C(C)(C)C)CC1 c1(C(=O)NCCOC2CCN(C(C(C)N(C(C)=O)C)=O)C2)nn(C)c2c1CCC2 C1(CNC(C(c2cnn(C)c2)OC)=O)CCN(Cc2ccc(Br)s2)C1 N1(C(CC2(CNC(C)=O)CC2)=O)CC2CC1CS2=O.C(CC(=O)N)N C1CN=C2NCC(=CC=NN(C(F)(F)F)C3C(N2)C(CC)CC3)C(=O)CCC1=O c1(COC)n[nH]c(=NCC2(F)CCN(C(=O)CC3CS(=O)(=O)C3)CC2)s1 c1(C(C(=O)NCC)N(C)C(C2CCCCC2)C)ccccc1OCC c1(C(=O)NC2(C)CC(NC(=O)CCCn3cncn3)C2)ncn2ccccc12 Cc1cn2c(n1)CC(C(=O)N(C1CCCCC1N(C(=O)C(O)CN(C)C)C)C)C2 c1(C(=O)NCC(CNC(Cc2cc(C)nn2C)=O)O)cc2cccnc2cc1F N1(C(c2ccc(OC)c(N)c2)=O)CC2CCC1C1CN(C(C3CC3C)=O)CC21 C1(C(N(CCC)C)=O)CCC2(CCN(C(C3CCc4nc[nH]c4C3)=O)CC2)O1 N1(C(c2cc(CSCC)on2)=O)CCC(NC(c2ccnc(CC)n2)=O)CC1 C(C)(C(CO)NC(c1cc(C2CC2)on1)=O)NC(C=CC(=O)OCC)=O CCC(C)CC(C(=O)NC1CC(O)C1OC)NC(c1nnc(S)n1C)=O Cc1c(C(=O)NC(C)C(C)NC(c2ccn(CC#N)n2)=O)c(C(F)F)nn1C c1(C(=O)NC2(C)CC(C(=O)NCC(c3cccnc3)C)C2)ccc(F)cn1 c1(CC)n[nH]c(CC)c1CC(=O)NC1CC1NC(=O)Cc1cc(C)[nH]n1 n1(CC(=O)NCC(CNC(c2ccc(O)cn2)=O)OC)nc(C)ccc1=O N1(C2CCC(NC(C3(CC)CC3)=O)C2)CCN(C(=O)C=Cc2ccoc2)CC1 C1(NC(C(F)=CC)=O)(CNC(c2cc(SC)c(C)o2)=O)CCCCC1C c1(NC(=O)NCC2CCCC(C#C)C2)c(Br)cc(Cl)c2occc12 C1(NC(C(C)C)=O)(CO)CCN(C(c2cccc(Oc3cccc(F)c3)c2)=O)C1 C1(C)(C(=O)NCC(C)C(=O)NCCN2CCC(C)C2)CCN(C)CC1 N1(CC)CCCCC1C(=O)NC(COC(C)C)C(=O)NCC1(C(N)=O)CC1.COC C1(NC(C(C2CCCC2)OC)=O)COC2CN(C(c3c[nH]c(=N)nc3C)=O)CC12 N1(C(c2cnc(C)s2)=O)CC(C(=O)NC(C(O)CO)C2CC2)C(C2CC2)C1 N1(C(CC(CC)O)=O)CC2C(C1C(=O)Nc1c(Cl)cnc(Cl)c1Cl)C2(C)C CCCCC(C(=O)OC)N1CCC(C(=O)NC2CC(F)(F)C2)(OCC)CC1 c1(C(=O)NCCOCCCNC(C2(COC)CCOC2)=O)ccc2n[nH]cc2n1 C(=O)(CS(=O)(=O)CC)N1CCC(N(C(=O)COCC(C)(C)C)CC#C)CC1 Cc1cc(C(N2CC3CC(C2)N3C(C2CC=CC(O)C2)=O)=O)cc(Cl)c1 c1(C(N2CC(C)(CNC(c3c(C)nc(C)s3)=O)OCC2)=O)cc(C#N)ccc1O c1(CN2CC3N(C(c4ccc(OC)nn4)=O)C3C2)ccc(Br)c(C)c1 c1(CCNC(=NC)NCC(n2cc(C(F)(F)F)cn2)(C)C)ccc(F)cc1 n1(CC)ncc2cc(C(=O)N(CC(C)(C)NC(=O)C(C)C(C)(C)C)C)c(C)nc12 C1(C(N2CC(C)C(NC(=O)CCc3ccc(Cl)nc3)C2)=O)CC12CCOCC2 c1(OC)cc(C#N)c(NC(C2CC2NC(c2ccc(Cl)c(F)c2)=O)=O)cc1OC CC(C)C(C(=O)NC1CC1)NC(=O)CNC(=O)COCCC1CCCC1 C1(CNC(CC)=O)CCC(NC(=O)CC2CC(OCC)C2)CC1.C(C)(C)(C)O c1(C(=O)NC2CC(N(C(C(C)Cc3cccnc3)=O)C)C2)nccnc1C(N)=O C(=O)(C(O)CCS(C)=O)N1CCN(C(c2c(OC)n[nH]c2)=O)CC1 C1(C)(CNC(CCCCOC)=O)CC(F)(F)CN1C(=O)CCC(C)OC C#CCC(C)C(=O)N(CCCCN(C)C(c1cn(C)nc1C(C)C)=O)C CCC(CC)(C(=O)N1CC(CNC(C2CCN(OC)CC2)=O)C(F)(CO)C1)OC CC1CN(C(c2coc(C(N)=O)c2)=O)CC(CCNC(c2cnc(S)n2C)=O)O1 N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CC2CC2(NC(=O)CC2CNC(=O)O2)C1 N1(C(C(C(C)(C)C)O)=O)CCc2c(NC(=O)C3=CC(O)CCC3)cccc2C1 N1(C(c2cnc(CSC)s2)=O)CCC2(C1)CN(C(c1ccc(CO)c(F)c1)=O)C2 C1(C)(C(=O)NC(C2CCOC2C)C)CCCN1C(=O)CCc1cnco1 C1(C)(C(=O)Nc2cn(CC(=O)N(C)C)nc2)CC(F)(F)CN1 Cc1ccc2nsnc2c1C(=O)NCCC(C)CCNC(=O)C(=O)NC1CC1 C1(C(=O)NC(CNC(c2cc(C)cc(C)c2)=O)CO)CC2CCC1C21CC1 Cc1cnc(Cl)cc1NC(C1CCN1Cc1ccc(-n2cccn2)cc1)=O C1(OC)CN(C(=O)COOCc2ccccc2)CCC1CC(=O)C(O)CC(C)C.N N1(Cc2cccc(C)c2)CCC(O)(C(=O)NCc2ccc(C)c(F)c2)CC1 C1(CNC(c2scc(C(=O)OC)c2)=O)CN(C(C23CC(C#N)(C2)C3)=O)CCC1C C1(C)(NC(N(C(CC)C(=O)NCCn2ccnc2CC)C)=O)CC(C)=NO1 C1(C)(NC(C(C)Cc2cnc[nH]2)=O)CCCN(C(C23CCCC2C3(F)F)=O)C1 C1(C(=O)NCC2CCN(C(C3CSCCS3)=O)CC2)CCCCCS1(=O)=O c1(C(N(CCCN(C(=O)C(F)(F)C(F)F)C)C)=O)ccc2nc(CO)[nH]c2c1 c1(CC2CN(C(=O)NCC(O)CCc3ccccc3)C2)ccc(Cl)cc1 c1(C(C(=O)NCCCNC(C(C2CCOC2)OCC)=O)=O)ccc(Cl)s1 N1(C(COCCC)=O)CCC(C)CC1C(=O)NCCSC C1(NC(c2cncc(Cl)c2Cl)=O)CC(C(F)(F)F)CN(C(c2ccccc2)=O)C1 C1(CNC(=O)C2=NOCC2)CCN(C(=O)CN2C(=O)CNC2=O)CCC1(F)F c1(OC)ccccc1OC(C)C(=O)NC1(C)CC(NC(c2ccc(Cl)cc2)=O)C1 Cc1cc(C(=O)NCC2(F)CC(NC(c3ncccc3Cl)=O)C2)cc(F)c1 CN1CCC(C)(C(=O)NC2CCN(C(c3csc(=N)[nH]3)=O)CC2O)CC1 C(=O)(CCS(=O)(=O)NC)NC(C(C(C)C)NC(C=CCCC)=O)C1CCCCC1 CCCCC(CC)C(=O)N1CCC(CO)C(NC(=O)CCOC)C1 N1(C(c2ccc(S(C)=O)cc2)=O)CC(C2CCCN(C(=O)C3=CCOCC3)C2)C1 c1(NC(C(=O)NC(CN(C(c2cc(C(C)=O)on2)=O)C)C)=O)ccc(F)cc1 c1(C(N2C(C(N(CC(C3CC3)OC)C)=O)CCCC2)=O)cnc2n1CCC2 c1(N)cnccc1Br.C12CSCCN1NC2=O.C1(C)CCCN1Cc1ccccc1 C(CCCCCCO)NC(C1N(C(Cc2cccc(C)c2)=O)CSC1)=O N1(C(C(C)OCCOCC)=O)C2CCC1C(F)C(NC(c1[nH]nnc1CC)=O)C2 C(=O)(C1COc2ccccc21)N(CCC(C)(C)NC(c1cccc(C)c1F)=O)C C1(NC(C(CC(N)=O)NC(C2CCC(O)C2)=O)=O)CC2CC1CC21CC1 CC1CC(CNC(c2cnc(Cl)s2)=O)CN(C(=O)CC2CC(=O)NC2=O)C1 c1(NC(C(CCSC)NC(=O)Cc2ccn(C)c2)=O)cccc(Cl)c1O c1(N(C2CCN(C(C)=O)C2)C)nc(=NCC2C=CCC2)[nH]c2c1CCCCC2 C1(C(N2CCCC(C(N)=O)C2)=O)(CC)CCN(C(C2CCC3(CC3)C2)=O)C1 c1(NCCCCCC)ccc(S(=O)(=O)NCC(O)CC=CC)cc1 c1(C(=O)NC(C2CC2C(=O)NCC2C3COCC23)C)cccc(CC2CC2)c1 C1(C(N2CCC(CNC(c3c(CCC)occ3)=O)C2)=O)Cc2cc(C)ccc2S1 N1(C(C2C(=C)C2)=O)CCC2CN(C(c3cc(F)ccc3C3CC3)=O)CC2C1 c1(C(=O)OC)cccc(-c2nnc(NC3(C(F)F)CCOC3)s2)c1 c1(C2C(C(N3CCCC(CN)C3)=O)C2)ccc(-c2ccsc2)nc1 C(CCSC)(C(=O)N1CCCC1CNC(N)=O)NC(c1c(CCC)nco1)=O C1(NC(c2ccc(CC)c(F)c2)=O)CC1C1CCN(C(=O)C(C)(O)C2CC2)CC1 CC1CCN(C(C2CC(CF)C2)=O)C1c1cn(CC(F)(F)F)nn1 C#CCC(C)(C)C(=O)N1CCN(CC(=O)NC(C2(O)CCCCC2)C)CC1 CCCC(C)C(=O)NCCC(C)CCNC(c1onc(Br)c1C)=O N1(C(C(C(C)C)NC(COC)=O)=O)CCC2(CC1)CC(C)N(C(=O)C(C)O)C2 CC1CCCn2c(C(N3CC(CNC(c4cccc(F)c4)=O)C(C)C3)=O)cnc21 c1(OC)cc(C(C(=O)NCC2CCCO2)N(CCN=[N+]=[N-])C)cc(C(F)(F)F)c1 C123CC(C1)(C2)C(=O)NCC3.C(CC(=O)NCC1CCC1OCC)SCC#C C1(O)(C(=O)NCCCCC(=O)NCC(CC)(C)CC)CC2CCC1C2 c1(CC(C)C)nc(C(=O)NC2CC(C)(NC(c3cnn(CCO)c3)=O)C2)cs1 C(CC1CC1)(CC(=O)N1CCOC(CCF)C1)NC(C(CC)=CC)=O N1(C(C(C)C)=O)CCC2(CC1)CC2CO.c1(CC)ccc(C(=O)NC2CCOC2)o1 c1(C(C(=O)NC(CC(N)=O)c2ccccc2)NC)cccc(F)c1 Cc1ccc(C)c(NC(C2CC2C(=O)NCC2(F)CCOCC2)=O)n1 C1(CNC(CN(C)C)=O)CN(C(=O)CSc2nnnn2C2CC2)CCC1CO C1(C2CN(C(=O)C=CC(=O)NC3CC3)C2)(NC(C(CC=C)C)=O)CC1 C1(OC)CC2CC(c3nnnn3C3(C)CC3)(NCc3cc(Cl)ccn3)C(C2)C1 C1(CNC(C(=CC2CCCC2)C)=O)CC2CCC1N2C(=O)Cn1ncc(Br)c1C CCC(C)(C)C(O)C(=O)N1CCCC(C(=O)NCc2ccc3c(c2)CC3)CC1 C=Cc1cnn(C)c1C(=O)N(CCCNC(=O)CCc1cnn(C)c1C)C1CC1 c1(C(C(=O)NCCC2CC(NC(CN(C)C3CC3)=O)C2)(C)C)cccc(F)c1 C(=O)(C(C)C(O)CCCCC)N1C2(CCN(C(C(C=CC)O)=O)C2)CCC1 C1(C(N2CCC(CNC(CCC=CC(C)C)=O)C2)=O)CCS(=O)(=O)C1(C)C C1(O)(C(C)NC(=O)C(F)=CCCF)CN(C(c2coc(C3CCC3)n2)=O)C1 CC1CCN(C(=O)Cc2ccc(O)nc2)C(C(=O)N(CCC(C)(C)C)C)C1 N1(C(C2(CO)CCN(C(CC(CC)SC)=O)C2)=O)CCC(C2(C)CC2)CC1 Cc1cnc2cccc(C(N3CCC3(C)CCO)=O)c2c1 CCCCCC(O)CC(=O)NC(C)(CNC(=O)CCCS(N)(=O)=O)CO N1(C(C(=O)NCCCC2CC2)C2CCCC2)CCC(c2ncccn2)CC1 C#CCCCCCC(=O)NCc1cccc(CNC(=O)CC2CCCCC2O)c1 N1(C(C2C(CNC(c3cnc(C)nc3)=O)OCC2)=O)CCCCN(C)CC1 C(=O)(C(CCC(C)(C)C)NC(=O)C(C12CCC(CC1)CC2)F)OCC N1(C(c2cc(C)c(C)nc2)=O)CCN(C(=O)CC2CCCCC2O)CCC1C CC(O)CCCCCC(=O)N1CC(C)(NC(c2ccc(NC(N)=O)cc2)=O)C1 C1(NC(C2=NNC(=O)C2)=O)COC2(CCN(C(c3cncc4nc[nH]c34)=O)C2)C1 N(C1c2ccccc2CC1NC(=O)C=C(C)Cl)C(C(CC=C)(F)F)=O C1(CCNC(COC(CC)C)=O)CN(C(c2cccc(C(C)(F)F)n2)=O)CCO1 c1(OC)nn(C)cc1C(=O)NC(C)CC(C)NC(C1CC(=O)N(C(C)(C)C)C1)=O C1(CCN)CCCCN1C(=O)N(c1cccc(C2COC2)c1)C1CCCC1 c1(C(=O)NC2C(OC)CN(Cc3ccc(F)cc3O)CC2)nc2ncccn2n1 c1(CCOC(C)C)nc(-c2cnn(C)c2)n(-c2ccnc(Cl)c2)n1 CC1(C)OCCc2cc(C(=O)Nc3ccc(Oc4ccncc4)cc3)ccc21 N1(C(C=Cc2ncc(C)[nH]2)=O)CCC(N(C(=O)COCC2CC2)C)C(C)C1 Cc1cc(C(N2CC(C)(C(=O)NCC(C3CC3)N(C)C)C2)=O)nc(O)n1 C1(C(=O)NCC(CCCC)O)N(C(=O)C(F)n2ccnc2)CCC1(C)C c1(C(=O)NCCOCC(=O)N(C(CCC)C)C)cccc(CC#N)c1 S(=O)(=O)(c1ccc(N2CCC3(CCCC(C(=O)O)O3)CC2)c([N+](=O)[O-])c1)N(C)C C1(C(N2CC(C)(CCC(=O)NC3(CCC)CC3)C2)=O)CC2(C1)CC(C)C2 N1(C(C2CCN(C(C=CC(=O)NCC=C)=O)C2)=O)CCCC(C)(O)C1 O=C1COc2ccc(S(=O)(=O)NC3CCC(NC(c4ccno4)=O)C3)cc2N1 O=C1CC(=O)CC(C(=O)NC2CCCCC2CC(=O)NCCC2CCCCC2)C1 CCCCC(CNC(=O)CN(C)C(c1ccsc1C)=O)CCC C1(C(=O)OCCC(=O)NC(CC)C)CC(=O)N(C)C1c1cnn(C)c1C c1(C(N(C(CNC(C2C(C=C)C2)=O)C)C)=O)csc(C2CCCCC2)n1 C(CC(=O)N1CC(C)CC1CC)(C(F)F)NC(CCC=CCC=C)=O Cc1cc(N)cnc1C(N1CCC1(C)CC(=O)Nc1ccc(O)cc1)=O c1(C(=O)NCC(CC=C)NC(C2(C)CCCS2(=O)=O)=O)nccc2ccncc12 C12(C(=O)NCC3C(C)(C)N(C(C4CS(=O)(=O)C4)=O)CC3)CCC(F)(CC1)CC2 c1(C(=O)NCC2N(C(CC(CC)OC)=O)CC(C)(C)C2)cc2c(=O)cc[nH]c2s1 C(=O)(C1CCCc2nn[nH]c21)NC1(CC)CCN(C(C2(CC#C)CCC2)=O)CC1 N1(CC(=O)NCC=CCC(=O)N(CCOC)C2CC2)CC(=O)NC1=O Cc1cc(C(N2CC(NC(C3CCCCS3)=O)CC2CO)=O)cc(N)c1O C12(C(N(c3ccccc3SCC)CC)=O)C3C4C1C1C2C3C41CO C(=O)(C(C)(C)NC(C12CC(C1)C2)=O)N(C)CCNC(=O)COCC(F)(F)F N1(C(c2c(CC)oc(C)c2)=O)CCN(C(=O)Cn2ccc(C)cc2=O)C(CF)C1 c1(OC)cccc(C(N2CCCC2(C)CNC(=O)CC2CSCCS2)=O)c1 C(=O)(C(C)C(O)C(C)CC)NCC1(C(N2CCC(C(=O)NC)CC2)=O)CC1(C)C C#Cc1c[nH]nc1C(=O)NCc1cncc(C(=O)NCC(N2CCCC2)C)c1 Cc1cc(-n2nc(CSC3CCCCC3)nc2C23CC(C)(C2)C3)cc(C)c1 C1(C(NNC(=O)C(=O)N2CCNCC2)=O)Cc2cc(Br)ccc2O1 c1(C(=O)OC)cncc(C(=O)NCC2CCC2NC(c2sc(SC)nc2Cl)=O)c1 C1(N(C(C(C)OCC2CC2)=O)C)CCCCN(C(=O)C=Cc2ccccc2)C1 Cc1ccc(C(=O)NC2CC(C(=O)Nc3nn(C)cc3C(N)=O)C2)cc1Cl N1(C(CC2C(C)CCC2)=O)Cc2occ(C(N3CCC3CC3CCCC3)=O)c2C1 C(c1cccc(Cl)c1Cl)=CC(N1CCC(CC=C)(NC(C2CCCCS2)=O)C1)=O c1(C(=O)NCCC2CC(NC(CCc3nc(C)sc3)=O)C2)ccccc1C(C)C N1(C(CCCC2C(C)C2)=O)CCC2(CC2)CC1C(N1CC2CCOC2C1)=O CC(C)C(CO)C(=O)NCCOCCN(C(=O)C(C)CCc1cccc(F)c1)C C(=O)(CCCC(F)(F)F)N(C1CCCN(C(=O)CC2CCCOCC2)C1)CC c1(OC)cccc(Cl)c1C(N1CCOC(CC(N2CCC(Br)CC2)=O)C1)=O C#CCC(C)(CC)C(=O)NCC1CCC1NC(c1nc(C)sc1C)=O C1(CNC(c2cnc(OC)c(C)c2)=O)CN(C(C2CN(C)C2)=O)C2CCCC2O1 CC1(C)CC(NC(=O)C(C)(O)C2CCCCC2)CN1C(=O)CCNS(C)(=O)=O C#CC1CN(C(C2CCC(=O)N(C)C2)=O)CCN1C(=O)C=Cc1ncc[nH]1 N1(C(C2CC(OC)C2)=O)CC(NC(C2CCCN2N=O)=O)CC12CCCCC2 C1(C(=O)NCCN(C(=O)Cc2cncnc2O)C)OCC2CCCC12 N1(C(CC(CC)C2CC2)=O)CCCC(N(C)C(C2(F)CCCCC2)=O)CC1 c1(OC)cc(C(=O)NC2CCN(C(=O)CCC3CC3(C)C)C2)cc([N+](=O)[O-])c1N N1(C(C(C)(C2CCC2)NC(C2C(C(C)C)CCO2)=O)=O)CCS(=O)CC1C N1(C(Cc2n(C)ccc2)=O)CC2ON=C(CNC(=O)Cc3ccc(Cl)cc3)C2C1 c1(C(N2CC(NC(CC(CC)SC)=O)C(C)C2)=O)c(N)sc(C)c1C c1(OC)cc(C(N2CCC(CNC(c3cnsc3)=O)(OC)C2)=O)ccc1[N+](=O)[O-] C(=O)(C1=CCCCO1)N(C)CC1CCN(C(Cc2cnc(C)[nH]2)=O)C1 N1(C(C2C(C)=C2)=O)CCC2(CC1)CN(C(C1CC1F)=O)CC2CO N1(C(C=CCOC)=O)CC(NC(c2cccc(-n3cncn3)n2)=O)C2(CCC2)C1 c1(CC(N2C(CN(c3cc(O)nc(C)n3)CC)CCC2)=O)nnc2n1CCCC2 Cc1ccc(C(=O)NCC2(C)CN(C(=O)Cc3cncn3C)CC2C)c(N)n1 CC1=CC(NC(=O)C(CC2CCOCC2)NC(=O)C(C)CC2CCCC2)CCC1 c1(OC)cc(C(=O)NC2CC3CN(C(c4ccc(C#N)[nH]4)=O)CC23)cnc1O C1(CNC(N2CC(C(=O)NC)C2)=O)(Cc2ccccc2)CCOCC1 S(=O)(=O)(c1ccc(Cl)cc1)N1CCC(NC2CCS(=O)(=O)C2)CC1 N1(C(=O)CCc2ccoc2)CCN(CC2CN(C(C3(O)COC3)=O)C2)CC1 c1(-c2cc(C(=O)N(CC3N(C(CCC=CC)=O)CCC3)CC)on2)ccc(F)cc1 C(CO)(C(=O)NCCNC(C1CN(C(c2cn(C3CC3)nn2)=O)C1)=O)N(C)C c1(NC(C2C(C(=O)NN3CCOCC3)C2)=O)cccc([N+](=O)[O-])c1Cl C(=O)(C(O)(C(F)(F)F)c1ccccc1)NCC1CCCCN(C(CCC=C)=O)C1 N1(C(c2oc(CC)c(C)c2)=O)CCCC(C(=O)NC2CN(CC(F)F)C2)CC1 C(C(C)C(F)C(=O)N(C(CCO)C(F)F)C)NC(CCC=C=C)=O N1(C(CN(CCOC)C)=O)CCC2CCN(C(=O)C(=O)NC(C)C)C2C1 CCC(CNC(=O)C(C)C(C)c1ccc(F)cc1)(CC)NC(=O)CCc1cnoc1 c1(C=O)cc(C2CC2)nn1C.c1(C2C(C(N(C3CN(N(C)C)C3)C)=O)C2)cccnc1 c1(C(=O)NCC(CC=C)NC(C2(C(=O)NC)CC2)=O)ccc2cc(Cl)ccc2n1 N1(C(c2ccc(N)c(F)c2)=O)CCCC(O)(CNC(c2ccoc2)=O)CC1 CC1(CO)CN(C(c2cccc3ccncc23)=O)c2ccccc2O1 N1(C(c2nccc(C3(C)CC3)n2)=O)CCCC2(CCOC2)C1 c1(C(=O)NC(CCNC(c2c(C)cccc2C)=O)C)ccc(C#N)cc1O O=C1NCC2(CCN(C(C3CC4CCC(C3)N4C(=O)C3=COCC3)=O)C2)O1 C1(C(=O)OC(C)=O)CN(C(=O)NC(C(=O)OCC)(C)C)CC(C)(C)C1 C=C(Cl)CC(C(=O)NC(C)C(C)SC)NC(c1ccsc1C#N)=O CN1CCN(c2cc(C(=O)NCC3(SC)CC(F)(F)C3)ccn2)CC1 CC#CCCCC(=O)N1CCC(NC(c2ccncc2SCC)=O)C(CO)C1 N1(C(C)C)CC(CNC(N2CCC(O)(Cc3cccc(F)c3)C2)=O)CC1=O c1(C(=O)NCC(CN(C(C2(C(=O)NC)CCC2)=O)C)C)ccc2cc[nH]c2n1 C1(NC(=O)CCNCC(F)(F)F)CC2(CCN(C(=O)OC(C)(C)C)CC2)CO1 Cc1[nH]c(C)c(C(=O)NCC2(O)CC(C(=O)NCC3(O)CCC3)C2)c1C c1(C(=O)Nc2cccc(NC(c3cccc(C#C)c3)=O)c2)ccc(F)c(C)c1Cl C1(C(=O)NCC2(OC)CCN(C(C3CCC3)=O)C2)CCn2c(C)cnc2C1 N1(C(=O)COCCF)CCN(C(c2ccc(Cc3ccccc3)s2)=O)C2CC12 C(=O)(C(C)(C)CC(=O)N1CCC2C(C1)CN2C(=O)C1=COCCO1)OC C(=O)(C1=C(C(C)(C)C)N(C2CC2)C(=S)NC1c1nnc2n1CCC2)OC Cc1sc(C(=O)NCCCCCNC(c2cnn(C)c2CC(C)C)=O)nc1O c1(OCC(=O)NC2C(NC(c3cc(C)no3)=O)C2)c(F)cccc1F N1(C(c2cc(C(N)=O)oc2)=O)CC(NC(=O)CN2CCSCC2)CC(F)(F)C1 C1(N(C(C(C)OCC=C)=O)CC2CC2)CCCN(C(c2cnsn2)=O)C1 CC(C)C(O)C(=O)NC1CC(CCC(N2CCC(n3cnnn3)C2)=O)C1 N1(C(C2CN(CC)C(=O)CC2)=O)CCN(C(=O)C2=CCCC2)C2CS(=O)(=O)CC12 C1(C(N2CCC(N(C)C(c3cccc(CS(N)(=O)=O)c3)=O)C2)=O)Cc2nccn2C1 C1(O)(CNC(CC(C=C)C)=O)CCCN(C(=O)Cc2ccccc2Br)CC1 N1(Cc2cc(OC)ns2)CC2(CCC(C(=O)Nc3cc(F)c(F)cc3OC)O2)C1 CC1(C(=O)NCC(O)CNC(=O)CCCn2c(O)nnc2O)CC=CCC1 N1(C(c2nn(C)c(O)c2)=O)CCCC2C(NC(c3ncccc3Cl)=O)C(C)(C)C12 c1(-n2cc(C3(C)CN(C(C(F)(F)C4(C)N=N4)=O)C3)nn2)cccc(C#N)n1 N1(C(COC(CC)(C)C)=O)CCN(C(=O)CN(C)C(=O)OC(C)(C)C)C(CO)C1 N(C1CC(C)n2ccnc21)C(COCc1c(C)cccc1)=O c1(OCC(=O)NCC(C)(C)N(C(c2cc(CC(C)C)c[nH]2)=O)CC#N)cccnc1 CC1CC(C)N(C(c2cn[nH]c2)=O)CCN1C(=O)C=C1CCSCC1 C=CC(C)C(=O)NC1CCN(CCCNC(=O)CCCn2cccn2)C1 N#Cc1ccc(N2CCCC2C(N2CCC(C(=O)NCCCO)C2)=O)cc1 C1(CNC(COC(C)=O)=O)CC(F)CN1C(c1cc(C)n(C(C)C)n1)=O C1(C(F)F)(CNC(=O)C=CC2CCOCC2)CCN(C(c2ccc(F)cn2)=O)C1 N1(C(c2n(C)c(Cl)nc2)=O)CC(C2CN(C(=O)C(C3CCCCC3)O)C2)C1 C(=O)(C1=NOC2COCC12)NC1C(C(=O)NC2CC(C)(C)C2)COC1 C1(CNC(C2(P(C)(C)=O)CC2)=O)CC2CCC1N(C(=O)CN1CCCC1=O)C2 C1(C(=O)NC2C(NC(=O)C=Cc3ccccc3)COC2)CCn2c(O)nnc2C1 CC1(F)CN(C(=O)C(c2ccc(Cl)c(Cl)c2)O)CCN(C(C2CC(O)C2)=O)C1 c1(COC(C2CCCN(Cc3ccccc3)C2)=O)ccc(C(F)(F)F)cn1 C1(NC(=O)OCC)CCN(C(=NCc2ccccc2)NC2C(C)(C)C2(C)C)C1 N1(C(=O)CSc2ccc([N+](=O)[O-])cc2)CCC2(CC1)COCCO2 N1(C(CCN2C(C)CCCC2)=O)CCN(C(=O)C(O)CC(F)F)C(CO)C1 Cc1ccc(C(=O)NC2CC3CC(NC(=O)CCn4ccnn4)CC23)c(O)n1 C#CCC(C(=O)NCC(C)(F)CNC(c1sc(C(C)C)nc1C)=O)C1CC1 C(=O)(C1=CCN(C(=O)CCNC(=O)C(C)(C)C)C1)N(CC(CC)O)C CC1CN(C(=O)CCCc2ccccc2Cl)CCC1NC(=O)C(F)F Oc1cc(Cl)ccc1-c1ccc(CN2CCC(Cc3nccs3)C2)cc1 O=C1NC(CNC(=O)C(=O)NC(C2CCCCC2)C2CCC2)CO1 CCC(CC(C)C)C(=O)N1CCC(F)(C(=O)NCc2cnco2)C1 Cc1ccc(CN(C)Cc2ccc(-c3cnc(N4CCCC4)nc3)cc2)c(Cl)c1 c1(C(=O)NCCCCNC(C2CCC(F)C2)=O)ccc2nnn(O)c2c1 N1(C(c2ccc(C#N)[nH]2)=O)CCN(C(c2csc(CO)n2)=O)C2CCCCC12 N1(C(C(C)(C)C2CCOC2)=O)CCC(C2CCN(C(=O)Cc3cc[nH]c3)CC2)C1 N=c1[nH]ccc(C(=O)NC2CCCC2NC(C2CC3CCC2C3)=O)c1[N+](=O)[O-] C1(NC(c2ccc3cc[nH]c3n2)=O)COC2(CCN(C(=O)COCCCF)C2)C1 CC12CN(C(c3cscn3)=O)CC1CN(C(C1CCCCC13OCCO3)=O)C2 C(=O)(CCCCCN=[N+]=[N-])N1CC(C)C(CNC(C2CN(C)C2)=O)CC1 C1(CNC(CCC#C)=O)CCCN(C(c2cccc(-n3cc(Br)cn3)c2)=O)C1 c1(C(=O)NC2(C)CC(NC(=O)CN3CC4CCC3C4)C2)cccc(O)c1Cl C1(CNC(CCN(C)CCO)=O)CC2(C1)CN(C(=O)C(F)C1CCOC1)C2 c1(C(=O)NCCOCCN(C(=O)CC2COC(=O)N2)C)ccc(Cl)c(O)c1 N1(C(C(C)CO)=O)C2CCCC1CN(C(C1(C(=O)NC3CC3)CC1)=O)C2 C1(NC(c2n(C=C)nnc2)=O)CCSC12CN(C(=O)C=Cc1ncc[nH]1)C2 c1(C(=O)NCCSCC(=O)NCCC2CCCC3CC23)cc(O)cc(F)c1 c1(CC)nnc2cc(N3CC(NC(C4CC4(C)Br)=O)CC4(CCC4)C3)ncn12 N1(C(C2CCC(C(C)C)CC2)=O)CC2CCC(C1)N2C(=O)Cc1cncn1C c1(C(=O)NC(CCCCNC(CC)=O)CO)cc2c(ccc3ccccc23)[nH]1 CC1CC(Nc2ccc(-c3cncn3C)cc2)C(C)O1 CCCC(C)(O)CC(=O)N1CC(CCC(=O)NOCCO)(C)C1 C(=O)(C1(C)OC(=O)c2ccccc21)NCC1(c2cn(CC(CC)O)nn2)CCC1 C(CC(C(=O)Nc1ccc(CCF)cc1)NC(=O)CC1CCC1)=CC C1(=CC(=O)NCC2(O)CN(C(C(OC)OC)=O)C2)CCC(C(C)(C)C)CC1 CC1OC2(C(=O)NCC=CCNC(c3cnccc3Cl)=O)CCC1C2 C=CCC(CC=C)C(=O)NCC1(C)CN(C(C2(C)CC=C(C)CC2)=O)CCO1 N(C1CN(C(=O)Cc2cnn(C)c2)Cc2ccccc21)C(C(CCCC)F)=O n1(CC(=O)NC2CN(C(c3n(CC)nnc3C)=O)CC2O)ncc2cccnc12 c1(C(=O)NC2(CC=C)CN(C(=O)C(F)(F)c3ccccc3)C2)cc(C)ccc1F C1(NC(c2cc(-c3cccs3)on2)=O)CC2(C1)CN(Cc1csc(Br)c1)C2 c1(C(=O)NC2CC(C)N(C(=O)CCC3CC(F)(F)C3)C2)ncc(C#N)cc1Cl N1(C(CC(CC(=O)OC)C)=O)CCC2C1CCCN2C(c1cc(Cl)ccn1)=O c1(CC(=O)N(CCCN(C(C(C2CC2)OC)=O)C)C)ccc(Cl)cc1Cl Cc1ccnc(C(N2CCC(NC(c3cnc(-c4ccsc4)s3)=O)C2)=O)c1 c1(NC(c2cc(C)nc(-c3cnccn3)n2)=O)cc(C)ccc1SC1CC1 N1(C(CNC(=O)Cc2ccc(F)cc2)=O)CCC2CCN(C(=O)CC(F)F)C2C1 c1(C2(C(N(CCCNC(=O)CCc3nc[nH]n3)CC)=O)CC2)ccc(O)cc1 CC(O)C(C(=O)NCCCNC(=O)CC1CCC1C)NC(=O)OC(C)(C)C C(=O)(C1=CCCN(C(C2CC2(F)F)=O)C1)NC(C)C(C)F C1(C(=O)NCC(=C)Br)CNC(=O)CN1C(C1COCC(C)O1)=O N1(C(C2CCC(C(=O)OC)CC2)=O)C2CCCC1CC(NC(c1ccoc1)=O)C2 N1(C(C(CC)CNC(=O)OC(C)(C)C)=O)CCCC(C)(NC(=O)C=CBr)C1 N1(C(C(C)(C)C(N)=O)=O)CC2C3CCC(C2C1)N(C(c1ccnnc1)=O)C3 N1(C(c2cc(C)n(C)c2)=O)CCN(C(=O)COc2ccc(F)cn2)C2CC12 c1(-c2nc(C(C)O)nn2-c2ccnc3cccnc23)cc2cc(Cl)ccc2o1 C(=O)(CC(C(F)F)C(C)(C)C)N(CCNC(C1N(C(CCC)=O)CCC1)=O)CC C1(C(=O)OC)N(C(c2cc(C(F)(F)F)ccc2F)=O)CC12CCC2 CC1CC(n2nc(C3CCCO3)nc2-c2cc(-c3ccoc3)[nH]n2)CCO1 c1(C(N(CC(CC)O)C)=O)cn2c(n1)CCN(C(c1cccc(F)c1C)=O)CC2 CC(C)(C)CCC(=O)NCC1(F)CC(NC(=O)CC2CCC3(CCC3)O2)C1 c1(OC)cc(Cl)ccc1CNC1CC(C(=O)Nc2c(F)cccc2Br)C1 N1(C(c2cc(C(=O)OC)sn2)=O)CCC2(NC(c3cccc(SC)c3)=O)CC2C1 c1(C(=O)NC2(C)CN(C(C34CCC(CO)(CC3)C4)=O)C2)ccc(Cl)c(O)c1N c1(C(=O)NC2CN(C(C3CCO3)=O)CC2F)c[nH]c2c(Cl)cccc12 CC(CN=c1[nH]c2cccc(Br)c2o1)NC(c1cnc2ncccn12)=O C(=O)(C(C)(C)C1=CCSCC1)NCC(C(C)C)NC(CN(C(COC)=O)C)=O C1(NC(COCCCC)=O)CCN(C(c2cnc(CC)s2)=O)C1C1CC1 C1(CC(=O)NC2CCN(C(c3cnn(C(F)F)c3)=O)CC2)CCCOCC1 CC1CCN(C(C2(NC(=O)CC3CCC(=O)C3)CC2)=O)CC1C c1(N(C)C)cncc(C(=O)NCC(CO)NC(C2CCCN2C(N)=O)=O)c1 c1(C(N2CCC(N(C(=O)C(C)n3ccnc3)CC)C2)=O)cc(N)nc(Cl)c1 C(C(F)(F)C(=O)NC1(CNC(=O)C(C)OC2CCCC2)CCCCC1)OC Cn1cnnc1C1CCCC1C(=O)NCCN1CCC(NC(C2(CF)CC2)=O)C1 c1(C(=O)NCCC2(O)CN(C(C(C)(C)SC)=O)C2)ccc2cnc(C)n2c1 CC1(C)CCC(C(N2CC(C)(CCC(=O)NCC(F)C(C)(C)O)C2)=O)C1 c1(C(=O)NCCCC(C)NC(=O)CN(C)CCO)c(F)ccc(F)c1F CC1=C(C(=O)NCC2CC3(CC3)CN2C(=O)C(C)Cn2ccnc2)CCS1(=O)=O c1(COC)cc(C(=O)OC)cc(S(=O)(=O)NC(C)(CC)C2=CCCC2)c1 c1(OC)ccc(CC(=O)NCC2CN(C(=O)Cc3ccc(C)s3)C3CC23)cn1 C=CC1(C(=O)NC2(C)CCC2)CCN(C(c2c[nH][nH]c2=N)=O)C1 C(=O)(C(CCF)NC(C1CC(C(C)C)C1)=O)NC1C(CCOCC)C1 c1(C(=O)NC2CCC(CNC(CC3CC(=C)C3)=O)C2)c[nH]c(=O)c2ccncc12 N1(C(c2cc(OC)ns2)=O)CCN(C(c2ncc(C(F)F)cc2F)=O)C(CO)C1 C1(C(N2CC3C(NC(=O)Cc4ccns4)(CCC3)C2)=O)CC12CCC(F)(F)CC2 C1(OC)(CNC(=O)CCC2(C)CC2)CCN(C(c2cnn(C)c2Cl)=O)C1 C1(NCC2CC(NC(C(C(CC)C)NC(C)=O)=O)C2)CCCCCCC1O N1(C(c2ccc(CC(C)C)s2)=O)CC2CC1CCC2NC(c1cccnc1O)=O CC1CCC(NCCOc2cccc(Cl)c2)CS1(=O)=O c1(C(=O)NCC(COC)NC(=O)C(C)CN(C)C)cc(C)c[nH]1 c1(N(C)CC2CC3CC3C2)cc(NCCCO)nc(C(F)(F)F)n1 C1(NC(=O)OCC)CCCN(C(=O)CC(=O)N(c2nc(C)nn2C)C)C1 N1(C(C(C2(O)CCC2)NC(C(C(C)C)C#N)=O)=O)CCC2CN(C)CC2C1 c1(SCCCC(=O)NC2CCCOC2)ccc(F)cc1.O=C1C(c2ccoc2)O1 c1(C(N2CCC(C)N(C(=O)CC3CCCC3)CC2)=O)cncc2c(F)cccc12 C1(NC(Cc2c(C)n(C)nc2)=O)CN(C(c2nc(=O)n(C)[nH]2)=O)CC(F)(F)C1 n1(CCSC)nnnc1C(c1csc(-c2ccsc2)n1)NCC(C)OC(F)F C(=O)(C1Cc2c(Cl)cccc21)NC1CCN(C(c2c(CN(C)C)cco2)=O)C1 CC1(C)CN(C(=O)CCCc2cccnc2)C(CNC(=O)CC2C=CCC2)CO1 C1(CNC(C(C)=CC)=O)COCC1n1cc(CNC(=O)CC2(C)CCCC2)nn1 C1(C(=O)NC(CCNC(C(C2CCCCC2)OC)=O)C)CN(S(N)(=O)=O)C1 C12(CNC(C(CSC)(C)C)=O)CCC(CC1)N2C(c1c(C)cccc1Cl)=O c1(-n2c(SC)ncc2)ccc(C(=O)NCCNC(=O)Cc2nccn2C)cc1 C(=O)(C(C)(C)COC(C12CCCC1(C(N)=O)C2)=O)OC N1(C(CCCC)=O)CCC2CC2(NC(c2sc(C3CC3)nc2C)=O)CC1 c1(CC(=O)NCC2CCC(NC(CCC(C)OC)=O)C2)cccc2cn[nH]c12 C(=O)(CCC(C)NC(=O)C=CC(C)(C)C)NCC(CC1CC1)OC N1(C(C2CC3CCC3C2)=O)CCC2OCCN(C(=O)Cc3cn[nH]c3)C2C1 c1(C(C)C)cccc(NC(=O)C(C2CCCC2)NC(=O)C#CC2CC2)c1 N1(C(C)=O)CCCc2cc(NC(C3(Cl)CC3(F)F)=O)ccc21 C1(NC(=O)C(N2CCC(C(F)F)C2)=O)CCC(CF)CC1 N1(C(C(C2(C)CC2)NC(c2cc(C)c(F)cn2)=O)=O)CCN(C)CC(C)C1 C1(C)(N(C)C)CCN(C(C2(CNC(=O)CC3CCN(C)C3=O)CCC2)=O)CC1 C(=O)(C(C)CC(N)=O)N1CC(CC=C)(C(=O)NC(c2ncccn2)CC)C1 C(=O)(C(CNC(c1cc(C)c(C)s1)=O)(CC)CC)NCC(=O)NCC=C C1(C(=O)OCC)C2COC(C(=O)N(CCCN(C)C(C3(SC)CC3)=O)C)CC12 CC1CC(=O)CCC1C(=O)NC1CC(CC(=O)NCc2cnccc2Cl)C1 C1(C(=O)NCC2N(C(CCOCCOCC)=O)CC3CC32)CCC=CCCC1 c1(OC)ccc(C(=O)NC2CCCCC2CNC(=O)C=CC(C)C)cc1N Nc1ccc(C(=O)NCC2CC3CC2CN3C(=O)C(F)=C2CCCC2)nc1N C1(NC(CC2(NC=O)CCC2)=O)COCC1C(N1CCC(c2nn[nH]n2)C1)=O Cc1cnc(C(N2CCCC(NC(=O)C=C3CCCCC3(C)C)C2C)=O)c(F)c1 C1(n2cc(CC3CC(C)(C)O3)nn2)CCCN(C(c2cc(C#N)cs2)=O)C1 Cc1cc(C(=O)NCC2CN(C(c3nn[nH]c3Cl)=O)C3(CCC3)C2)cc(=O)n1C Cc1c(C(=O)NCC2CN(C(=O)Cc3ccc(F)cc3)CC2C)cccc1C#N N1(C(c2cnc(OC)nc2C)=O)CC2(CCN(C(=O)CCCC(F)F)C2)C1 c1(C(=O)NCCSCC(=O)NC2C(C)SCC2)cnn(C)c1C#N c1(C(=O)NCC2CCN2C(=O)CCOc2ccccc2)ncccc1Br C=CCC(C(=O)NCC(C1CCN(C(=O)C(C)O)CC1)O)NC(C)=O C1(C(=O)NCCOC(C)(C)CNC(c2nc(C3CC3)cs2)=O)OC2CCC1C2 N1(C(C(C)NC(C)=O)=O)CC(F)(F)CC1(C)CNC(c1cc(S(N)(=O)=O)c[nH]1)=O c1(OC)ccc(Br)c(F)c1C(=O)N(CCCNC(=O)C(CO)N(C)C)C N1(C(CC(=C)C)=O)CCC2(CO)CN(C(c3cnn[nH]3)=O)CC2C1 N1(CCNC(C(n2ncc(C)c2)C)=O)CCN(C(=O)C(C)(C)n2cnnn2)CC1 CC(C)C(C)(O)C(=O)N1CC(CNC(c2ccc(Cl)cn2)=O)C(F)(F)C1 CC(CCO)N(C(=O)CC1(NC(=O)CSC2CC2)CCC1)C C1(C(=O)Nc2cccc(NC(c3cc(C)ns3)=O)c2)(CC)CCC(O)CC1 C(=O)(C(C)(C)CCNC(=O)C=Cc1ccncn1)NCC1CC(=C)C1 NC(=O)CCCCC(=O)NC1CCCCN(C(=O)C=CC=C(Cl)Cl)C1 CC1(CNC(C2CC3(CC3)C2)=O)CN(C(c2ccnc(Cl)c2N)=O)CCO1 CC(C)CC(C)C(=O)NCC1CN(C(C2CSCC(=O)N2)=O)CCN1C CC#CCCC(=O)NCC1CCCC(NC(C2CCCN2CCC(C)C)=O)C1 N#CCS(=O)c1ccc(C(=O)NC(C(N)C(=O)O)c2ccccc2)cc1 Cc1ccc(O)c(NC(=O)CC2CCN2C(c2ccc(=N)[nH]n2)=O)c1 C1(OCC)CC2CN(C(=O)CC3CC(C)N(C(=O)C(F)=CC4CC4)C3)CC12 CCC(CO)(C(=O)N1CC(C(O)C(=O)NCC2(CC)CCCCC2)C1)OC C1(NC(c2ccoc2I)=O)COC2(CCN(C(=O)Cc3ccccc3F)C2)C1 c1(C(=O)NCC2N(C(c3c(CC)occ3)=O)CCC2)cc2c(cc1N)OCO2 Cc1cnccc1-n1nc(CO)nc1CCN(C)C c1(OCC(=O)NCCNC(C2COCCO2)=O)cnc(Cl)cn1 C(C)(C(=O)N(CC(C)N(C(=O)CSC(C)C)C)C)(C1CC1)OC N1(C(c2n(CCOC)ncc2)=O)CCC2(CCCN2C(C2CCN(C)C2)=O)C1 c1(C(=O)NCCC(=O)NCC(O)CCNC(C2CCCO2)=O)cccc(F)c1F C1(CCC)(C(N2CC(O)(C(C)NC(c3cncc(F)c3)=O)C2)=O)CCNC1=O c1(OC)ccc(F)c(C(=O)N(CCNC(C2(F)CC2(Cl)Cl)=O)C(C)C)c1F C1(COC2CCN(C(=O)C=C3CCC3)C2)CCN(C(=O)CC2CCOCC2)CC1 CC(CC1CC1)C(=O)NCC1(C(=O)NCCSC(F)F)CCCO1 C(=O)(N=S1(=O)CCNC(C)CC1)N1C(C)c2n(cc(C(C)C)n2)CC1 N1(C(C(C)(C)NC(=O)OC)=O)CCC2(C1)CN(C(c1csc(C(F)(F)F)n1)=O)C2 C1(C(=O)NCCN(CCOC)C(c2cscc2C(N)=O)=O)CS(=O)(=O)C1 c1(CNC(C2(OC)CCC2)=O)n[nH]cc1C(=O)N(C(C)CO)CC C#CCC(CC(=O)N(CCCCO)C)NC(c1cc(C)c(N)cn1)=O Cc1cnnc(O)c1C(=O)NCC1CC(F)CN1C(C1CC2(C1)CC(F)C2)=O CN1N=C(C(=O)N2CC(NC(=O)Cn3ncc4cccnc34)C(O)C2)CCC1=O c1(C(=O)NCC(C)(C2CC2)NC(=O)C=Cc2cccs2)cc(O)ccc1F N1(C(C=C(CCC)C)=O)CCCCC1CCNC(=O)C(c1ccccc1)C1CC1 c1(C(=O)NCC2(C(=O)NC3CCC(C(N)=O)C3)CC2)ccc(O)nc1 N1(CC)CC(C)N(C(=O)CCN(C(=O)Cn2cccnc2=O)C)CC1C c1(CC)ncc(Cl)c(C(N2CC(F)(CNC(=O)C=CC(C)CC)C2)=O)n1 c1(OC)nc2ccc(C(N3CC(NC(c4cc(CO)ccc4Cl)=O)C3)=O)cc2[nH]1 c1(C(=O)NC(CC)CNC(c2csc(C(=O)OC)c2)=O)[nH]cnc1C#N c1(C(C)CNC(c2ncsc2C(=O)O)=O)cccc(Br)n1 c1(C(=O)OCC2(C)CNC(=O)C2)ccc2cccc(F)c2n1 N1(C(c2n(C(C)C)ncc2)=O)Cc2ccccc2C1C(=O)N1CC2CC2C1 C(=O)(CC(C(F)(F)F)n1ccnc1)NCC1(C)CCN(C(C=CSC)=O)C1 Cc1cccnc1CC(=O)NCCC1CCN(C(C2CCC(O)C2)=O)CC1 c1(N2C(CNC(CC3C(C)=NOC3=O)=O)CCC2)nc(C)cc(C)c1C#N N1(C(C2(CC)CCN(C(c3cccnn3)=O)C2)=O)CC2CCC(C1)O2 n1(CC)nnc(C)c1CNC(=O)C(C)=CCNC(C1(O)CCCC1)=O C(C(=O)NCC(O)C(C)C)(C(C)C)NC(C1(CC=C)CC=CC1)=O N1(C(CC2CC(=O)NCC2)=O)CCC(F)C(NC(c2ccc(C(F)(F)F)s2)=O)C1 N1(C(Cc2scc(C)c2)=O)CCN(C(c2nnc(O)cc2O)=O)CC1CC(F)F c1(C(=O)NC(C2CN(C(c3cc(Cl)c(Cl)[nH]3)=O)C2)C)cn(C)c(=O)n1C Cc1sc2ccccc2c1NC(=O)NC1(C)CN2CCC1CC2 c1(C(C)=O)ccc(C(N2CCOCC(CNC(C3(F)CC=CC3)=O)C2)=O)cc1F C1(C(N2CCCC(CNC(Cc3cc(C)[nH]n3)=O)C2)=O)CCCS(=O)(=O)C1 N1(C(CN(C(Cc2n(C)ccn2)=O)CC2CC2)=O)CCC(NC(=O)C2CC2)CC1 N1(C(CCC=CC)=O)CCN(C(=O)CC(C)NC(N)=O)CC2(CC2)C1 CC(C)CCCCC(=O)NC1CC2(C1)CC2C(=O)NCC1CCCN1C c1(C(=O)NC2CC3N(C(C4CC(OC)C4)=O)C(CC3)C2)cnn2c1C(C)CCC2 C(=O)(CC(C)(C(F)(F)F)N(C)C)N(CC(O)CNC(=O)CN1C(=O)CCC1=O)C C1(C(=O)NCc2cncc(C)n2)C2CCC(C2)N1C(=O)C(c1ccccc1Cl)O C1(NC(C2CC3C=CC2O3)=O)CCN(C(c2ccc(Br)s2)=O)C12CC2 C1(NC(C2C(C)CCO2)=O)CCCC(C(=O)NC2CC3CCC2C3)C1 C1(CNC(C(C)O)=O)CCCCCN1C(=O)C(c1ccccc1)=O.C1(=O)CN1 c1(C(=O)NC(CC2CCN(C(c3ccn(CC)n3)=O)CC2)C)cc(Cl)ccc1N CCCCCC(CC)C(=O)N1CCC2(COC(CNC(=O)CCC(=O)NC)C2)C1 c1(CN2CC3(CCC(C(=O)N(S(CC=C)(=O)=O)C)O3)C2)sc2ccccc2c1Cl CCCC(C)CC(=O)NCC1CCN(C(=O)Cc2cc(F)ccc2O)C1 C1(CC=C)(C(=O)NC(CSC)CC)CCN(C(c2csc(F)c2)=O)C1 c1(C(=O)NC2(CNC(CCCOCC)=O)CCOC2)cc(Cl)c(Cl)[nH]1 N1(C(C2CCC(CC)O2)=O)CCC(NC(c2ccc(CO)s2)=O)C(CO)CC1 C1(CNC(C23CCC(OC)C2C3)=O)CN(C(c2cnn(C)c2N)=O)C2(CCC2)C1 c1(C(=O)NC2CCC(CCNC(CC(=C)C)=O)C2)c[nH]c2cc(OC)ccc12 Cc1cc(C(=O)N(C2CC(C#N)C2)CC(=O)NC(c2ncc[nH]2)C)ccc1O O=C1NCCCCC1C(=O)NC(C(N1CCC12CCC2)=O)C1CCCC1 CC1CC(CCNC(C2(C(N)=O)CC2)=O)CCN1C(c1ccc(Cl)o1)=O c1(C(=O)NCC2(F)CCN(C(C(CC)COC)=O)C2)coc2cc(OC)ccc12 CCS(=O)(=O)CC(=O)N1CCC(N(C(C2CCCN2C(C)C)=O)CC2CC2)C1 Cc1cccc(C(=O)NCC2CC(NC(c3cccn3Cc3cccs3)=O)C2)n1 c1(CC(=O)NC2C=CCN(C(c3ccsc3Cl)=O)C2)cccc(C(F)F)c1 CC1CN(C(C2CCS(=O)CC2)=O)CC1CNC(C1CN(S(C)(=O)=O)C1)=O C=CC1(C(=O)NC(C)C(=O)NC(C)C)CCN(C(c2cc(O)nc(O)n2)=O)CC1 C(=O)(C1=C(Cl)CCOC1)NC1C(C(=O)NCCC=CC=C)C2CCC1C2 CCCC(CC(C)C)C(=O)NC(C)(C)CCCNC(=O)COCC(F)(F)F N1(C(c2ccc(SC)s2)=O)CC2CC2(CNC(C2CC(F)(CO)C2)=O)C1 c1(SC2CC(C(=O)OC)C2)cnn(CCN(C(=O)CCN(C)CCO)CC)c1.CCC C1(C(=O)NC(CC)C(N)=O)CCC2(CCN(C(=O)CCc3cccnc3)CC2)C1 c1(CC(C(=O)NCc2conc2C2CC2)NC(N)=O)ccc(O)cc1 O=C(CCCC(F)(F)CO)NCC1(O)CCCN(C(=O)CCC2CCCC2)C1 N1(C(c2cc(Br)ncc2F)C(=O)NC)CCc2cc(OC)cc(OC)c2C1 c1(CC(=O)NCCN(C(C2(C(=O)OCC)CC2C(F)(F)F)=O)C)cncnc1O c1(CC(=O)OC)ccc(CNC(=O)N(C2CCCN(C)C2)c2cnn(C)c2)cc1 CCCCCC(=O)NC1CC(NC(=O)COCP(C)(C)=O)C(O)C1 CN1C(=O)C(O)C(C(=O)Nc2ccc(Cl)cc2C(=O)O)C1c1ccccc1 C1(CC(C)C)(C(=O)NCC(O)CCNC(c2sccc2C#N)=O)CCNC1=O Cc1cc(C(=O)NC2CCN(C(c3cnc(O)n3C)=O)C2)nn1C1CCOCC1 C(=O)(C(C)N=c1cncc[nH]1)N1CC2CCN(C(CCOCC)=O)CC2C1 c1(N(CC)CC2CCN(C(c3csc(O)n3)=O)CC2)ncc([N+](=O)[O-])cc1C#N S(=O)(=O)(c1cncc(Br)c1)N1CC(NC(c2cc(Br)c(Cl)cc2F)=O)C2(C1)CC2 c1(CC)[nH]nc(C(=O)NCC=CCNC(=O)C(C)Cc2ccco2)c1[N+](=O)[O-] O=C(CC1OCc2cc(Cl)ccc21)NC1CC(CNC(C23CC(CO2)C3)=O)C1 N1(C(c2ccc(COC)o2)=O)CC(NC(c2cc(C#N)oc2C)=O)CC12CCC2 c1(C(=O)OCC)cccc(NC(=O)NC2(C3CCCO3)CC2)c1C c1(C(C(=O)NC(CNC(CCCCC=CC)=O)(C)C)C)ccccc1S(N)(=O)=O N1(CC)CCOC(C(=O)N(CCC(=O)NCC(N2CCCC2)C)C(C)C)C1 N1(C(c2cnc(OC)c(Cl)c2)=O)CC2(CCCN(C(=O)C(C)C3CC3)C2)C1 C1(C(=O)N(C)CC2CN(C(=O)C(C)(C)OC)CCO2)(OC)CCOCC1 CC(C)CC(CC(C)C)C(=O)NC1CC2(C1)CN(C(=O)CN1CC3CC3C1)C2 CC(C)C(C(=O)OC(C)(C)C)C(=O)N1CCCC(N(C)C(c2coc(Cl)c2)=O)C1 c1(N2C(C)CC(NC(C3CCC(=O)N3C)=O)CC2)nc2cccnc2s1 N1(C(c2cn(C)nc2-c2ccc(F)cc2)=O)CCC2CCNC2C1 C(CC)(C(=O)NCC(CNC(=O)Cc1c[nH]nc1C)OC)OCC c1(C(C)NC(C(COCC)NC(=O)Cc2nccn2C)=O)cccc(C)c1 c1(C(N2CCOCC(C3CC3)C2)C(=O)NCC(=C)C)noc2ccc(Br)cc12 CC1(C)C(CNC(=O)CC2CCC(O)C2)CCN1C(=O)Cc1ccc(O)c(Cl)c1 C1(C(=O)NCC(C)N(C)C(c2ncoc2-c2ccco2)=O)CC12CC(C)(C)C2 C(=O)(C1=C(Cl)CCOC1)NCC1N(C(c2ccc(C#C)cc2)=O)CCC1CC N1(C(c2c(OC)scc2)=O)CC2CC1CN(C(=O)C(CC)OC)C2 N1(C(COCCSC)=O)CCC(C=C)(C(=O)N(C2CCCC(C)(C)C2)C)C1 c1(OCCC)ccc(-c2ccc(CNC(=O)NC3(Br)CC3)nc2)cc1F C(C)(CO)(C(=O)N1CC(N(C)CCO)C1)NC(C(C)=CC=C)=O c1(N2CCN(C(CNC(CCCC)=O)=O)CC2)ccnc2nc(C)nn12 C1(NC(c2cc(OC)no2)=O)CCN(C(=O)C(C)OC2CCCC2)C12CCC2 C(=O)(C(C(C)C)n1cc(Br)cn1)N1CC(CC)(CC)C1 Cc1nc(O)ccc1C(=O)N(C)CCN(C(=O)C(CO)c1ccccc1)C c1(OC)ccc(C(N)=O)cc1C(=O)N(C1CN(C(C2CCN(OC)CC2)=O)C1)C C1(C(=O)NC2CN(C(CCOC)=O)CC2C(F)(F)F)CC(c2cnn(C)c2)=NO1 Cc1cc(NC(C2CN(Cc3ccc(Cl)nc3)CCC2O)=O)ncc1Cl N1(C(c2c(CC)noc2)=O)CC2CC(NC(c3cnn(C(C)C)c3C)=O)C2C1 C1(CNC(=O)NCc2ccc(OC(C)=O)cc2)CC(C)SC(C)C1 Cc1ncc(C(N2CCC(CNC(c3cc(C(F)F)cs3)=O)C(C)C2)=O)c(C)n1 C(=O)(C(C(=O)OC)C(C)NC(=O)C(=O)NCc1ccc(C(C)=O)cc1)OC C(C(CC(C)C)C(=O)NCC(C)CC(=O)N1CC(c2ccccc2)C1)OC Nc1ccc(Cl)c(C(=O)NCC2CN(C(=O)CCC(F)F)C2)c1 n1(CC)cc(C(=O)NC2(CN(C)C(c3cscc3OC)=O)CC2)c(C)n1 CCC(C)CCCC(=O)N(CCCNC(C1CC2CCCC(C1)C2)=O)C1CC1 N1(C(c2ncn(CC)n2)=O)CC(F)(F)CC1CNC(C1COCCN1C)=O S(=O)(=O)(c1cnc(NCCNC(=O)C(C)(C)C)c(Cl)c1)N(CC(O)CF)C.C(CO)N CCS(=O)(=O)c1cccnc1CNC(=O)C(C)NC(C1CCC1)=O C1(NC(c2cc(C)c(O)cc2)=O)COC2C(NC(C3COC(=O)N3)=O)COC12 N1(C(c2cc(F)ccc2F)=O)CCN(N2CC(O)CC2Cc2ccccc2)CC1 Cc1cc(C(N2CC(c3cn(CCCF)nn3)C(C)C2)=O)c(C)o1 C1(C(=O)NCC(N(C)C(c2cc(Cl)c(Cl)s2)=O)C2CC2)CCN2CCOCC12 c1(OC)ncc(Cl)cc1C(=O)NC(c1ccc(Br)nc1)(C)C N1(c2cc(C(C)C)ncn2)CCC(NC(c2ccc(OC(F)F)nc2)=O)C(C)C1 C1(C(N(CC(C)N(C(CC(C)C)=O)C)C)=O)CCC(F)CC1 N1(C(CSCC(C)C)=O)CCC(C(C)CNC(=O)CN2CC=CC2)CC1 C(=O)(CC(F)(F)C(F)F)NC(C1CCN(C(C(C(=O)OCC)OC)=O)C1)C c1(C(=O)NCC2C(NC(c3n(CC)nnc3)=O)CCC2)cn2nc(C)cc2[nH]c1=O C1(CC)(NC(=O)C=CSC)CCCN(C(=O)C(c2cncnc2)C)C1 C1(C=O)CCCCC1O.C(C(=O)N(CC(O)CO)C)(C1CC1)OC c1(NC(c2cncc(NC(c3cncc(O)c3)=O)c2)=O)cc(Br)c(O)c(Br)c1 c1(C(Cn2cc(-c3cc(C)on3)nn2)C)cccc(Cl)c1F Cc1cncc(C(=O)N(C2CCCN(C(=O)COC3CCCCC3)CC2)C)c1C N1(C(c2nc(C)sc2)=O)C2CCC(C2)C1C(=O)NC1(C2CC2)CCC1 CCCCCC(CC)C(=O)NCC(C(=O)NCCOC1CC1)C(C)C CC#CCCCC(=O)NC12CCN(C(=O)COc3ccccc3Cl)CC1C2 N1(C(c2nc(CCC)oc2)=O)CCC(NC(c2cc(C)c(C)[nH]2)=O)C(F)C1 N1(C(CN(C(=O)CCc2nccs2)C)=O)CCN(C(=O)CC(F)(F)F)CC1 N1(C(C=CCN(C)CC)=O)C2CCC1C1CC1(NC(=O)CCc1ccccc1)C2 C#Cc1cccc(C(=O)N(C2CCC(NC(=O)CC3=CCOCC3)C2)C)c1C CCC(CC(=O)N(C)CCc1cnc[nH]1)NC(c1ccc(NC)cc1)=O N1(C(C(C)CNC(C2CCCC2)=O)=O)CC(=O)NC(=O)C1C Cc1nn(C)c(NC(C23CC2CN(C(c2ccsc2)=O)C3)=O)c1C(N)=O N1(C(C=C(CCC)C)=O)CCCN(C(c2ccc(CCC)s2)=O)C(C)C1 CCC(C(=O)N(C)CC1CN(C(C2CC23CC3)=O)C1)c1cccnc1 N1(C(c2c(C#N)ccs2)=O)CC2(CCCC2)C1C(=O)NCC(=O)NC(N)=O c1(OC2CCN(C(=O)NCC(CC=C)C)CC2)cc(Cl)ccc1Cl S(=O)(=O)(c1c[nH]c(C(N2CCN(C(=O)C(O)P(C)(C)=O)CC2CC)=O)c1)NCC C12(NC(C(c3ccc(OC)cc3)CC)=O)CC(C1)N(C(c1ccnnc1O)=O)C2 CCCC(C(O)C(=O)N1CCC(F)(C#N)C1)NC(=O)CC(C)CC N1(C(CC(C)OC)=O)CCCC(C(N2CCC(c3ncn(C)n3)CC2)=O)CC1 C1(C)(NC(CNS(CCOCC)(=O)=O)=O)CCCN(C(c2[nH]cnc2C)=O)C1 c1(C(=O)NC2CC(CNC(C(C)SC(C)C)=O)CC2O)ncsc1S(N)(=O)=O OC1CCC2(CCCN(Cc3ccc(Br)cc3Cl)C2)CC1 Cc1c(Cl)ccc(Cl)c1NC(=O)CN1CCN(C(=O)C(=O)C2CC2)CC1=O c1(NCC(CC)(C)CC)cc(Br)ccc1S(=O)(=O)N1CCn2nc(C)cc2C1 N1(C(CC=C=C)=O)CC(NC(c2cc(O)cc(Cl)c2)=O)C2CC2C1 C(c1ccnn1C)=CC(=O)N(C)CC1CCN(C(COCC(=O)NC)=O)C1 c1(C(N2CC(NC(CCCCCSC)=O)C(C)C2)=O)cc(F)cc2cnccc12 C#Cc1ccc(C(=O)NC2CCOC(C3CCN(C(=O)CC(=C)C)CC3)C2)nc1 C1(C(=O)NCC(C)(C2CC2)NC(c2coc(Br)n2)=O)CC12CCOC2 C(=O)(C1=C(C)CCC1)N1CC(C(=O)NCC(C(CC)C)C)OCC1 C12(NC(=O)Cc3ccc(Cl)cc3Br)CCC(CN(C(=O)CC3CC3)C1)C2 CC(C)CCCCC(=O)N1CC2CCC(C1)N2C(=O)Cn1ncn(C)c1=O Cc1cnc(N2CC3(CCC(C(=O)Nc4ccccc4)O3)C2)c([N+](=O)[O-])c1 N1(C(c2c(C(C)C)[nH]cc2)=O)CCC(C2CCCN(C(=O)C3=C(Cl)CC3)C2)CC1 C1(NC(c2n(CCC)ccc2)=O)CCCCCN(C(C2CCCNS2(=O)=O)=O)C1 c1(C(N(C(C2CCCCC2)C(=O)O)C)=O)cc(SCc2ccccc2)ccc1F C(=O)(C(CC)CC)NC1C(C(N(CCC#C)CCO)=O)CC1 Cc1cnc2n1CCC(C(=O)NCC1(O)CCN(C(c3cc(=O)cc[nH]3)=O)C1)C2 C1(NC(CCC(=O)NCC)=O)CC1C1CCCN(C(c2c[nH]nc2C)=O)C1 C12(NC(C=CC(C)C)=O)CC(CNC(C3CC3c3ccsc3)=O)(C1)C2 N1(C(CC2N(C)CCC2)=O)CCC2(CC(NC(=O)CCCc3cccnc3)C2)C1 C1(C(C)(C)C)(Cc2ccccc2)CCN(CCOCC(N)=O)C1 C12(CN(C3CCN(c4ncc(C(F)(F)F)cc4Cl)C3)CCC)CC=CC(C1)OC2 Cc1cnc(C(=O)NCC2CCC(NC(C3(C(F)F)CCCO3)=O)C2)[nH]1 N1(C(C2(OC)CCSC2)=O)CC2CCC(C1)C2NC(c1ccnc2ccnn12)=O CC(C)C1=NOC(C(=O)N(C)CCNC(=O)C(C(C)(C)C)OC(C)(C)C)C1 N1(C(c2n(C)ncc2)=O)CC(NC(=O)Cc2csc(-c3ccco3)n2)C(F)C1 C#CC1(C(N2CCC(OCCCCC)C2)=O)CCCC1 C1(NC(CNC(c2cc(C)nn2C)=O)=O)CCC(C)(C)CC1CNCC1(F)CC1 c1(OC)cccc(C(=O)NCC(C)NC(=O)CCc2nccn2C)c1N Cc1cc(F)cc([N+](=O)[O-])c1NC(c1nc(NC(C2CCCS2)=O)cn1C)=O CN(CCCC(=O)N1CCC(C(C)(C)NC(=O)C#CC2CCOC2)C1)N=O c1(C(=O)NC)cccc(C(N2CCC(O)(CNC(=O)CCC3CCOC3)C2)=O)c1 C(N=c1nc(O)c(Br)c[nH]1)C1(O)CCCN(C(c2ccc(C)nc2O)=O)C1 c1(OC(C(c2cn(CC)nn2)N2CCCC2c2ccsc2)=O)cccc(F)c1 CC(C)(CCNC(=O)CC1CCC(C2CC2)O1)N=c1[nH]nc(C2CC2)s1 c1(CNC(=O)CC(Cl)Cl)cccc(C(N2CC(c3nc(=O)o[nH]3)C2)=O)n1 c1(C(=O)NC2C(C)CCN(C(C3(CO)CCC3)=O)C2)ccc(N)c(F)c1F Cc1nn(CC(=O)N(C(C)CCNC(C2(C)CNC(=O)C2)=O)C)c(C)c1Cl Cc1cc(F)c(Br)cc1C(=O)N(C(C)CNC(=O)CC(O)C(C)C)C CC1CN(C(C2CCCC(O)C2)=O)CC1NC(c1cc(-c2ccccc2)co1)=O CC(=O)CCCC(=O)N1CCC(O)(CCNC(C2CN3CCN2CC3)=O)C1 N1(C(c2c(C(C)C)occ2)=O)CC2CC1CC2NC(c1nnc(S)n1C)=O c1(CC(C(=O)O)ONC(c2cn(C3CCCNCC3)nn2)=O)cccc(Cl)c1 Cc1n[nH]c(C)c1CN(C(C)C)Cc1ccccc1-c1ccccc1 N1(C(c2cc(COC)cn2C)=O)CCC2CCN(C(c3cccnc3N)=O)CC12 C1(C(=O)NCCCOCCCNC(CC2CC2)=O)CC2CC2C1.CS CS(=O)(=O)c1ccc(CNC(C2CCN(C(=O)CC(O)C3CC3)CC2O)=O)cc1 C1(NC(C(C=C=C)C)=O)CCC(C)(CNC(=O)CN2CCCS2(=O)=O)CC1 C12(C(N(CC(C)NC(c3ccccc3CC#N)=O)C)=O)CC(C1)C(C)(C)O2 c1(OC)cc(C)ccc1C(=O)NC1CCN(C(=O)CCCC(C)=O)C1C c1(C(=O)NCC2CCCN(C(CC(CC)SC)=O)C2)cccn2c(CO)nnc12 c1(C(=O)NCC(=O)NC(C)CNC(c2coc(Cl)n2)=O)ccccc1CC#N C1(NC(c2scc(C)c2C)=O)CCN(C(=O)C(C(C)(C)C)NC(N)=O)CC1O c1(C(=O)NC(C(C)C)CCNC(c2nc(Cl)c(Cl)s2)=O)ccc(O)c(Cl)c1 C1(C(N(C)CCOCCNC(C2CCCC(=O)N2)=O)=O)Cc2ccccc2O1 Cc1nn[nH]c1NC(=O)NCc1cc[nH]n1 c1(C(N(CCN(C(=O)C=Cc2cncs2)C(C)C)C)=O)cc(CF)on1 N1(C(c2nc(OC)oc2)=O)CCCC12CCN(C(=O)CSc1nncn1C1CC1)C2 N1(C(CCC(=O)NCC)=O)CC(NC(C2CS(=O)(=O)CC(=O)N2)=O)CC2(CC2)C1 N1(C(C(CC)C(C)O)=O)CC2CC(NC(=O)C(F)CC3CC3)CC2C1 Cc1cnc(C(N2CCOCC2CC(=O)N(C2CC(F)(F)C2)C)=O)c(C)c1 c1(C(=O)NCC2(CCNC(C3C(C)(C(C)C)C3)=O)CC2)ccc(C(C)(C)C)[nH]1 C1(CCCC)CCCC1NCc1cc(-c2ccccc2)on1 C1(C(=O)NCC(C)CN(C(=O)Cc2ccc(O)cn2)C)CC1C1CC1C N1(C(C(CNC(CC2COCC(C)O2)=O)N(C)C)=O)CCC(C2CC2)C1 c1(C(C(=O)NCCCF)N(C)Cc2ccncc2)ccc(C#N)cc1F N1(C(c2c(NC(c3c(Br)ccc(F)c3F)=O)ccs2)=O)CCC2(CCOCC2)C1 c1(C(N2CC(F)(C(=O)NC(C3CCOC3)C)C2)=O)cc(C#N)ccc1Br N1(C(Cc2c(C)n[nH]c2C)=O)CCCCC(N(C)C(c2ccncc2Br)=O)C1 N1(C(C2CC(C)N(C)C2)=O)CCC2(C=C(C(=O)N3CC(NC(N)=O)C3)C2)C1 N1(C(C2(C)CC(C)C2)=O)CC2CCN(C(=O)C=Cc3ccc(Cl)cc3)C(C2)C1 CN1CC(C(N2CC(C3CN(C(C4CCC5(CC5)C4)=O)CCO3)C2)=O)CCC1=O c1(C(N(CCNC(COC2(C)CCC2)=O)CCOC)=O)cc(F)cnc1O c1(C(=O)OCC)c(NC(C2CCCN2C(c2ccc(OC)s2)=O)=O)ncn1C S(=O)(=O)(c1cccc(F)c1)NCC(N1CCN(C(c2ncn(C)n2)=O)C2C1C2)=O N1(CC(=O)NC(CCCCC)C)CC2(CC(NC(=O)CCn3ccnc3)CO2)C1 C(=O)(C#CC1CCCCO1)NCC(C1CC1)NC(c1cc(CSC)c(C)s1)=O C(=O)(C1CCc2c(Br)cccc21)NC(c1cccnc1)C(C)C CC(C)C(CO)CCNC(=O)CC1CC(C)N(C(=O)COC2CCCC2)C1 N1(C(=O)Cc2ccc(O)c(O)c2)CCC2CN(c3ncnc4cc[nH]c34)CCC12 C12(C(=O)NCC3(CCNC(C4CCC(=O)NC4)=O)CC3)CCC(CC1=O)C2 C1(C)(C(=O)NCC(C)(C)NC(C(CC)n2ccnc2)=O)CCC(=O)N(C)C1 N1(C(C(COC(C)C)NC(C)=O)=O)CC=CC(NC(C2(C)CS(=O)(=O)C2)=O)C1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC1CC(F)(CNC(C2CC(C)C2)=O)C1 N1(C(C2CN(C(C)C)C(=O)C2)=O)CCCN(C(C2CC(CF)C2)=O)C(C)C1 c1(CNCc2cc(C(=O)OCc3c(OCC)ccs3)no2)cc2nc[nH]c2cn1 c1(CCNC(C(C2CCN(C(c3c(COC)ncs3)=O)C2)C)=O)c(C)noc1C c1(C(N2C(C(=O)NCC3(OC)CCC3)COCC2)=O)cc(C)c2ccccc2n1 C1(C(=O)NCC(C)CN(C(=O)Cn2ncn(C)c2=O)C)CCC2(CCC2)CC1 C(=O)(C(C)CC(N)=O)N1CCC(CN(C(C(=O)NC)C)C)C1 C1(C(N2CC(C(CC)C)C2)=O)CSCCN1C(c1ccc(Cl)o1)=O CC1(C)COC(CC(=O)N(CCCNC(=O)CC2(CO)CC2)CCO)C1 N1(C(c2c(COC)noc2)=O)CC(C)C(NC(c2cc(O)ccc2F)=O)C(C)C1 C(=O)(C(C)(C)C(O)C(C)C)NC1(CC=C)CCN(C(=O)C(C)CS(C)=O)CC1 c1(C(C)C)cc(F)ccc1NC(=O)NC(C)CN=[N+]=[N-] CC(C)C(CCN(C)C(c1nccnc1N)=O)NC(=O)C(c1cccn1C)=O N#Cc1cccc(C(N2CC3C(NC(=O)CC45COC(C4)C5)C3C2)=O)c1 Cc1coc2c(C(N3CCCC(CCNC(=O)C(C)CC(F)F)C3)=O)cccc12 C1(C(N(CCN(C(=O)CC2OCCC2C)C(C)C)C)=O)OCCC1C N1(C(C(C)(C)C)=O)CCN(C(C2CCC(=O)O2)=O)C(CC(F)F)C1 CCC(CC(=O)N1CCCC1(C)C(=O)N(C)Cc1ncc(C)o1)CC(C)C c1(C(=O)NCCCN(C(C2ON=C(C)C2)=O)C2CC2)cccnc1-n1ccnc1 c1(C(=O)OC(N2C(CCOC)COCC2)=O)cccn(C2CCSC2)c1=O N1(C(c2ccc(CC)cc2)=O)CCN(C(=O)C2=NNC(=O)C2)CC1CC(F)(F)F C(=O)(C(C)N1CC(C)C1)NCC(=O)NCC(=O)N(C(CC)C)C C12(CNC(C3CCN3C3CCCCC3c3ccc(F)cc3)=O)C(=O)C3CC1C2C3 C1(O)(C(=O)NCC(C)NC(=O)Cn2cnnc2O)CC(F)(F)C1 C1(NC(C=C(CCC)C)=O)CC2(C1)CC2NC(c1ccc(C2CC2)nc1)=O C12(C(=O)NCC(C(C)C)NC(c3ccnc(Cl)c3Cl)=O)COC(CCO1)C2 N1(C(c2cc(CC)c(C)s2)=O)CCC(O)(CNC(=O)C(F)CC2CC2)CC1 c1(C(=O)NCC(C)(C)NC(c2ccncc2)=O)csc(-c2ncccn2)n1 CC1CN(CCN2CC(=O)N(CC3CCC3)C2=O)CC(C)O1 C(=O)(C(C(C)C)NC(C)=O)NCC(CCC)NC(c1ccsc1)=O N1(C(c2c(C)nns2)=O)CCC2C(CCN2C(C2CC3(C2)CC3(F)F)=O)C1 N1(C(c2c(C)noc2)=O)CCN(C(C)CNC(=O)C=CCO)CC1 c1(C(=O)NCCNC(c2cc(C(CC)C)no2)=O)cc(S(N)(=O)=O)c(C)o1 C1(CCCC)CN(C(c2ccc(Cl)[nH]2)=O)CCN1C(c1cncc(N)c1C)=O c1(CNC(C2(CC)CCCC2)c2nnnn2C2CC2)ccc(C(F)(F)F)nc1C c1(C(C)C)ccc(CC(=O)NCC2CCC(NC(=O)CC(F)(F)F)C2)cc1 c1(CN2CC(C(=O)NC3C(=O)NCC3)(CC3CC(O)C(O)C3)C2)cc([N+](=O)[O-])n[nH]1 c1(N2C(CCNC(C(C)(C)C)=O)CCCC2)ncnc2c(Br)c[nH]c12 CC(C)CC(C)CNC(=O)NC(C(F)(F)F)C1CCC1 c1(NC(C2C(C(=O)Nc3c(C(=O)NC)cccc3)C2)=O)cnc(O)nc1O Cc1ccc(C(=O)NCC2CC(NC(c3ccc(O)nc3Cl)=O)CC2O)c(F)c1 CN1CCC(C)(C(N2CCC(C(N3CC(C)(CF)C3)=O)C2)=O)C1 CC1CCC(CC(=O)NCC(O)CN(C(=O)C(F)=CCCF)C)OC1 N1(C(=O)CC2CCN(C(C3CC34CC4(F)F)=O)C2)CCCC(CN2CCOCC2)C1 C1(NC(CCC#C)=O)CN(C(c2c(OC)nsc2OC)=O)CC(F)(F)C1 O=C(NN=Cc1ccc(Br)c(Cl)c1)c1ccccn1 N1(C(=O)NCc2cn(CC(F)(F)F)nc2Br)CCC(CO)C(F)(F)C1 CC1(C#N)CCN(C(=O)C(CC2CCCC2)NC(C2C3CCC(F)C23)=O)C1 N1(C(C2(C#N)CCOC2)=O)C2CCCC1CN(C(C1CCn3nnnc3C1)=O)C2 C=CC(CC)C(=O)NCC1(OC)CN(C(c2cc(C3CC3)cs2)=O)C1 Cc1nn(CC(=O)NC(C)C(C)NC(=O)CC(C)C)c(=O)c2ccccc12 C1(CNC(c2n(CC)nnn2)c2ccc(-c3cc[nH]n3)o2)CC2(C1)CC(F)(F)C2 n1(CC)cnc2nc(N3CC4COCC(C4)C3)nc(N(CCCC(F)(F)F)C)c12 C1(NC(C(CC)C)=O)CCN(C(=O)COc2ccc(F)c(Br)c2)C12CC2 c1(NC(C2(C3N(C(C(C)OCCCC)=O)CCC3)CC2)=O)ccc2nc[nH]c2c1 c1(OC)ccc(-c2noc(COC(=O)C3CC3)n2)cc1NC1CCCCC1C c1(C(N2CCN(C3CC(C)(C)OC3=O)CC2)=O)cnc2c(c1)CCCO2 C1(CNC(C=CC(N)=O)=O)CC(O)CN1C(c1cc(-c2cccs2)on1)=O Cc1ncc(Br)cc1NC(C1CCC(NS(=O)(=O)Cc2ccccc2)CC1)=O c1(C(=O)NCC2C(NC(C(c3cscn3)N(C)C)=O)CC2)ccc2nonc2c1 C(=O)(C(CC(C)(C)C)OC)NC(CN(CC(=O)N(C1CCCC1)CC)CC)C C1(CNC(C2CCC(COC)C2)=O)CC2(C1)CN(C(=O)C=C(C)Cl)C2 N1(CC(=O)N(CCC)CCC)CC(NC(c2c(C)cccc2F)=O)CCC1C c1ccc(N2CCC2c2nnnn2C2(NCC3CCOCC3)CCCC2)cc1 N1(C(C=CS(C)(=O)=O)=O)CC(NC(=O)Cc2ccc(Cl)s2)CC2(CC2)C1 CC(C)(C(=O)NCC(=C1CN(C(=O)COc2ccon2)C1)F)N1CCCCC1 N1(C(CC2CCC(=O)N2)=O)CC(C(N2CC(CO)(CO)C2)=O)C(C2CC2)C1 C1(S(N)(=O)=O)(C(=O)NCC(CNC(C(Cc2ccc(OC)cc2)C)=O)O)CCC1 N1(C(C2CCN(C(c3cc(CC)[nH]n3)=O)C2)=O)CCC(C)(CCO)CC1 c1(C(N2CC34COCC3(C2)C4)C(=O)NC)ccc2ccccc2c1 N1(C(C(CCCCC)O)=O)CCn2ncc(CNC(=O)CC(C)C(F)F)c2C1 c1(CC(=O)NCC2C(NC(C3(C)ON=C(C)C3)=O)COC2)cccc2nsnc12 c1(C(N2CC(OCCNC(=O)CCCCC3CC3)C2)=O)cc[nH]c2nccc1-2 C1(N(C)C(C2CCCOC2C(C)(C)C)=O)C=CCCC1Cc1ccccc1Cl N1(C(CCC(C)(C)OC)=O)CC(C)N(C(=O)CC(C)C2CC2)CC1C N1(C(c2cc(CC)oc2C)=O)CC2CCN(C(C3CC34CCOC4)=O)CCC2C1 c1(C(=O)NC2(CC=C)CCN(C(C3CCCC(CF)C3)=O)C2)cc(O)nc(C)n1 CCC(CC)C(C(=O)NCC(CC1CC1)C(=O)NCC1CC(F)C1)OC CCCCC(O)CC(=O)NC1CCCC1CNC(c1ccc(CO)c(F)c1)=O C1(CC(=O)NCC2CCCN(C(C3(CNC(C)=O)CC3)=O)C2)CCCC(C)(C)O1 c1(C(=O)NCc2nc(C)c(C(=O)N(CCCN(C)C)C)o2)cn(C)c(=O)cn1 C(CC(=O)NCc1c(F)cccc1F)(C(F)(F)F)NC(=O)C=CC1CCCC1 CCCC(O)(CCC)CC(=O)NCCCN(C(=O)CC1CCC(=O)N1C)CCO N1(C(C(C2CCC(=O)N2)C)=O)CCCN(C(=O)C(N)=O)CCC1 C=C=CCCC(=O)NCC(C)(C)CNC(c1nocc1CC)=O c1(C(=O)NCC(CC)NC(=O)CC2CCN(C)CC2)ccc(C)nc1C(C)C C(=O)(C1CCCc2scnc21)N1CCOCC(CNC(C=CSC)=O)C1 C(CC(=O)Nn1cncn1)N(C(C1(C)CCC1)=O)C(=O)OC(C)(C)C c1(C(N(CCN(C(C(c2ccc(C)o2)C)=O)C)C)=O)scc(C)c1Cl Cc1ccc(C=CC(=O)NC(CNC(=O)CCC(=O)c2ccc(Cl)cn2)CO)s1 C1(C(N2CC(NC(c3coc(C(N)=O)c3)=O)C(O)C2)=O)CCOCC12CCCCC2 N1(C(C(C)NC(=O)CC(C)(C)C)=O)CCC2C1CCCN2C(C1CC(O)C1)=O C(=O)(C(C)CNC(=O)C(Cn1cccn1)NC(=O)CCC1CC(C)C1)OC C1(C(=O)NCC(CNC(c2c[nH]nc2-c2ccco2)=O)O)CCCCC12CCC2 C#Cc1c[nH]nc1C(=O)NCC1CC(CCC(N2CC(C#N)C2)=O)C1 c1(-c2cn(CC(=O)N(C(CC(C)=O)C)C3CC3)nn2)ccc(OC(F)(F)F)cc1F c1(C(=O)NC2C(C(C)C)CN(C(=O)Cc3cnns3)CC2)cccc2cncn12 N1(SCCNCCCC(C(=O)OCC)O)C(=O)NC(C)(C)C1=O Cc1cc(Cl)cc(C(C)NCC(C(C)(F)F)c2ccccc2)c1O C#CC1CCCN(C(=O)CC2CC(NC(C3CCC(C4CC4)C3)=O)C2)C1 Cc1cccc(Br)c1CNC1CCOC(C(=O)NC(C)(C)C)C1.n12ccc(c1)C2 C(=O)(CN=c1cc[nH]cc1)NC1(C)CCCN(C(=O)CCOCC2CCC2)C1 N1(C(C2(C(C)NC(=O)CC3CCC3)CC2)=O)CCN(C)C(C2CC2)C1 C(=O)(C(C)CCC(C)(C)C)NC(C)CCNC(c1nnn(C)c1N)=O Cc1nc2ccc(C(N3CC(C)(C(=O)NC4CS(=O)(=O)C4)C3)=O)cc2[nH]1 c1(C(=O)NC(C)(C)CNC(=O)C=Cc2cnc[nH]2)c[nH]c2ccncc12 C(=O)(C(CNC(=O)CSc1cn[nH]c1)CCC)NC(C#C)C(C)OC C1(CNC(C(c2ccc(F)cc2)C)=O)CN(c2ccnc(Cl)n2)CC(C)(C)O1 Cc1ccc(C(=O)C(=O)NC(C)CC(C)NC(=O)CC2CC2C)cc1 c1(C(N(C(C)CNC(c2ccc(Cl)nc2O)=O)C)=O)ccc2oc(O)nc2n1 N1(C(C(C)CF)=O)CCC2(CC1)CC2NC(c1ccc(C(F)(F)C(F)F)cn1)=O c1(C(N(CC(C)NC(C2CC2C2CC2)=O)C)=O)cc2ccc(F)cc2o1 C1(O)(CNC(C(C)(Cl)Cl)=O)CCCN(C(=O)C(O)c2ccco2)C1 C1(CC(=O)NCCCOCCNC(c2c(CC)nc[nH]2)=O)CC2CCC1O2 C(c1ccc(Cl)cc1)=CCN1CC(O)(CC(=O)N(CCCCCCN(C)C)C)C1 c1(C(N2CCC(C(C)NC(=O)Cc3cccs3)C2)=O)cn(C)c(=O)nc1O N1(C(C(C=C)O)=O)CCCC(CCC)(NC(=O)Cc2ccc(CCC)cc2)C1 C(CC1=CCN(C(c2csc(-c3cccs3)n2)=O)CC1)NC(C(C)CC(N)=O)=O c1(OC)cc(C(=O)N(C2CN(C(=O)C(F)(F)COC)C2)C)cnc1O c1(OC)ccc(F)c(F)c1C(N1CCC1NC(N1CCN(CCCO)CC1)=O)=O c1(NCC2C(C)N(C(=O)OC(C)(C)C)CCC2)ncc(Br)cc1C#N CC(C)C(C(=O)N1CC(O)C(O)C1)NC(c1cnco1)=O C1(C(N2CC3(CC(NC(C4OCCC(=O)C4)=O)C3)C2)=O)CCc2nccn2C1 N1(C(=O)COc2cccc(F)c2)CC2CCN(C(=O)COC3CCOCC3)C2C1 C1(CC)(NC(C2COC3(CCC3)C2)=O)CCCN(C(=O)CCNC(C)=O)C1 Cc1ccc(C(=O)NCC2CC3(CC3)CN2C(=O)C2=COCC2)cc1C CCC(O)C(C)(C)C(=O)N1CCN(CC2(NC(=O)C(C)c3ccco3)CC2)CC1 c1(C(C(=O)N(C)CC2CCN(C(CC(C=C)(C)C)=O)C2)C)ccc2c(c1)OCO2 N1(C(=O)C=Cc2cnccn2)CC2(C(N3CC(O)(C4CC4)C3)=O)CC1CCO2 C=CCCCC(C(=O)NC(C)C(F)(F)F)NC(=O)Cc1csc2nc(C)cn12 c1(OC)cc(OC)c(C(c2nnnn2C)Nc2ccnc(CO)c2)c(OC)c1 c1(CC)cccc(C)c1-n1nc(CO)nc1-c1n[nH]c(-c2ccccc2)c1C c1(C(N(CC(CNC(C(c2cccnc2)OC)=O)O)C)=O)nccnc1N c1(C(=O)NC(CN(C(=O)CCC2CCOCC2)CC)C)coc2cc(C)ccc12 c1(C(N2C(CC)CN(C(=O)C(C)CC#N)CC2)=O)ccc2cnc(C)n2c1 S(=O)(=O)(c1ccc(NCC(C)(C)C#N)c(C#N)c1)NCc1ccc(OC)c(F)c1 c1(CC(=O)NCCC(CCNC(CC(C)C(F)F)=O)C)ccc2c(c1)CCCO2 N1(C(c2n(CC)ncc2)=O)CC2CCCC2(C(=O)NCC(c2ccccn2)O)C1 C1(CNC(C2N(C)C(=O)CC2)=O)CC2(C1)CN(C(c1cc(Cl)sc1Cl)=O)C2 C1(C(=O)NCC2C(NC(c3cc4cscc4s3)=O)C2)COc2ccc(F)cc2C1 C1(C(=O)NCC#CCNC(=O)Cc2ccc(Cl)s2)CC2CCCCN2C1 N1(C(CC(=C)C)=O)Cc2ccnn2CC(NC(c2nc(C(C)(F)F)cs2)=O)C1 C1(NC(C2N(C(c3cccc(CC)n3)=O)CC2C)=O)CCCCCC1CO S(=O)(=O)(c1cnc2ccsc2c1)NC(c1n(C)nc2c1CS(=O)(=O)CC2)=O C1(NC(C(C)SC(C)C)=O)C=CCN(C(C2(c3ccc(F)cn3)CC2)=O)C1 c1(N(CC(C)(C)C(=O)NC2CCN(Cc3ccccc3)C2)C)cnn(C)c1C#N c1(N2CCCC(CCC)CC2)nc(=N)[nH]c(=NC2CCC(C)(C)C2)[nH]1 CCCC(C#N)C(=O)N1CC(CNC(c2csc(C)c2OC)=O)(OC)C1 C1(C(C)NC(c2ccc(CSC)o2)=O)CCN(C(=O)CC2CCCN2C)CC1 N1(C(C2(CC#C)CCOC2)=O)CCCCC1CNC(c1cncnc1)=O CCC(C)CC(C)(c1nnnn1C1CCC1)NCCc1ccc(C(F)F)cc1 C(=O)(C(F)C(C)(C)O)N1CC(CNC(C(c2ccnn2C)C)=O)OCC1 N1(C(c2c(N)n(-c3ccccn3)nc2)=O)CCCCCC1CNC(C1CC1F)=O N1(C(c2cnc(CC)o2)=O)CCN(C(=O)CC(F)(F)F)CC1C1CCC1 Cc1ccc2cc(C(N3CCNCC3c3ccncc3)=O)nn2c1 Cc1cnc(C(=O)NCC(CNC(c2cc(=O)cc[nH]2)=O)CO)c(F)c1 N1(C(C2CC(C)(C)N(C(c3cccs3)=O)C2)=O)CCCC2OCCC2C1 N1(C(C(C(CC)C)NC(=O)C(=O)C2CCCC2)=O)CCn2nc(C)cc2C1 C(=O)(C(C)(C)CC(C)(C)C)NC(CC(C)C)CNC(c1n[nH]cc1Br)=O c1(CC)occ(C)c1C(=O)NCC(CC)OC(C1CCOC(C)C1)=O c1(CC(=O)NCC2CCCN2C(=O)C(C2CC2)C2CC2)cccc(Br)c1 Cc1c(C(=O)NC2CCCC(NC(=O)C(C)(C)c3ccsc3)C2)sc2nccn12 c1(C(N2CC3CCC(C2)N3C(=O)CCN2CCC2)=O)cn2cc[nH]c(=O)c2n1 Cc1cc2c(cc1C)N(C(C13CCOCC1C3(F)F)=O)CC2 CC1(C)C(NC(c2ccoc2CN2CCCC2)=O)C2CCCOC12 CCCCC(C(=O)NC(C)C(C)NC(C1(CSC)CC1)=O)ON=C(C)C C1(C(=O)NCC2CCN(CCc3n(C)ncc3)C2)CCC([N+](=O)[O-])CC1 c1(C(=O)NCC2CN(C(C(C)NC(C)=O)=O)CC2C)c(C)cnnc1O N1(C(c2n(C)nc(C)c2Cl)=O)CCCC(C2CCN(C(=O)Cc3nc[nH]n3)C2)C1 c1(NC(C(N2CCCCC2CO)CC)=O)ccccc1C(C)C C12(OCC)CC(CO1)N(C(=O)Cn1cc(C)cn1)C2.C12CN(C1)C2=O c1(N(CC(C)CNC(=O)C(C)CC(N)=O)C)ncnc2c1nnn2C1CC1 S(=O)(=O)(c1ccc(NCCCCCF)c(F)c1)N(C)CC1COC(C)(C)O1 c1(OC)c(C(C(=O)NC2COC2)N(C2CCCCC2C)C)cccc1C(F)F N1(CCNC(c2cc(CNC(C3CC(=C4CC4)C3)=O)on2)=O)CCCCCC1 CC(C)C#CC(=O)NC1COCC1NC(c1cccnc1N(C)C)=O c1(OCCCN(C(=O)C(C)(C)NCCC#N)C)ccc(F)cc1 c1(C(N2CCC(NC(C(CC)N(C)C)=O)CC2)=O)ccc(Cl)c2c1OCCO2 N1(C(C2(CCNC(C=CCC)=O)CC2)=O)CCS(=O)C(C)C1 C1(OC)(CNC(C2CCCN2C(c2cc(Cl)no2)=O)=O)CCC(C)C1 C(=O)(C1SCCc2sccc21)N1CCN(C(C2(F)CCCCC2)=O)CC(C)(F)C1 N1(C(c2nnn(CC)c2C)=O)CCc2sc(CNC(=O)CCCC(C)C)nc2C1 C1(NC(c2cncnc2)=O)CN(C(=O)Cn2cccn2)CCC1CO C(=O)(C(CC)c1cccnc1)N1CC(C(C)NC(CN(C2CC2)CC)=O)C1 c1(N2C(COC)(CNC(=O)C=Cc3cnc[nH]3)CCC2)nc2ccccc2o1 Cc1cc(O)ncc1NC(=O)C(CNC(c1cccc(O)n1)=O)CC1CC1 Cc1c(C(=O)NCCOCC(=O)N(C2CC2)CC2CCCCO2)cncc1F CC(C)(C)CC(O)C(=O)NC1CCCN(C(=O)Cc2ccc3c(c2)COC3)CC1 c1(C(c2nnnn2CCCF)NCCC2(C)COCCO2)cc(S(C)(=O)=O)co1 n1(CC)cc(Cl)c(C(=O)NCCNC(C2CN(C)C2)=O)n1 C1(CNC(c2n(C)cc(Cl)c2)=O)CN(C(=O)C2=C(Cl)CC2)CCC1(F)F C(=O)(CCC(F)(F)CN=[N+]=[N-])N1C(C)(C)CC(NC(=O)COCC(F)(F)F)C1 C(=O)(C(C)S(=O)(=O)C(C)C)NC(CCCNC(C(C)(C)OC(C)=O)=O)(C)C CC(C)(C)C(C(=O)NC1CC(CNC(C2CC2(C)C)=O)C1)NC(=O)OC(C)(C)C N1(C(c2cc(Cl)ccn2)C(=O)NCC)CCC(C#N)(C(C)C)CC1 C(=O)(CC(N(C(C1CC1(F)Cl)=O)C1CC1)C1CC1)NC1(C(N)=O)CCC1 C1(NC(CN2CCC(OC)C2)=O)CCN(C(=O)Cn2nccc2C)CC1F c1(NC2CN(C(C(CC)CC(C)C)=O)CC2C)ncc([N+](=O)[O-])cc1Br N1(C(c2scc(C)c2)=O)CCC2CCN(C(=O)CS(=O)(=O)NC(C)(C)C)C2C1 N1(C(c2c(C)nc(O)cc2)=O)CC(C)CN(C(C2CC(F)(CO)C2)=O)CC1C C(=O)(CC(CC)N(C(=O)CCN1CCOC1=O)C)N(CC(CCC)O)C c1(C(N2C(C)CC(NC(CCC(C)=O)=O)C2)=O)ccc(C)c(-c2cnn(C)c2)c1 N1(C(CCCCCNC(C)=O)=O)CC2CCOC2(CNC(c2ccncc2)=O)C1 N1(C(c2c(-c3cn(C)nc3)ocn2)=O)CCCC1C1CCCN1C(=O)COCCF C1(F)(C(=O)NCC2(O)CC(C(=O)NCC3(OCC)CCC3)C2)CCCCCC1 CCCC(C(=O)OC)C(=O)NC(C)(C)CNC(=O)C(c1cccc(Cl)c1F)(F)F Cc1cnc(Cn2cc(C3CCN(C(C4CCS4(=O)=O)=O)C3)nn2)cn1 S(=O)(=O)(c1ccccc1C(=O)NC(C)CNC(=O)C(C)N)N(CCC)C.C(C)(=O)O N1(CC(=O)NCCC2CC(NC(C(F)OC)=O)C2)CC2CC2C1 C1(CNC(C2CC3CCC2O3)=O)CN(C(=O)Cc2cccc(Cl)c2F)CCCO1 C(=O)(CCS(N)(=O)=O)NC1(CC(=O)NC(Cc2cc(C)[nH]n2)C)CCCCC1 C=CCC(CC=C)C(=O)N1CCCN(C(=O)Cc2nnc(O)s2)C(C)C1 C(CC(C)C)(C(=O)N1CCOCC(NC(=O)CCCc2cc[nH]n2)C1)OC C(=O)(C1=CCCN(C(=O)CC(CC)C(F)F)C1)N1CCC(OCC=C)CC1 C(=O)(CC(O)CC(C)(C)C)NC12C(CN(C(c3cccc(C)c3Br)=O)C1)C2 C1(CC(=O)N(CCCNC(c2cccc(=O)o2)=O)CC)CC(O)C12CCC2 C1(C(=O)NC2CC(NC(c3c(C)nn[nH]3)=O)C2)CC(=O)N(c2ccccc2)C1 Fc1ccc(C2CN(CC=CCOc3ccccc3)CCO2)cc1 c1(C(=O)NCC(C2CCN(C(C3CC34CC4)=O)CC2)(C)O)cnc2ccnn2c1 CC1(C(=O)NCC(C)(CO)NC(=O)COc2ccc(C(N)=O)cc2)CC=CCC1 N1(C(CC2(C)CC2)=O)CCC2CCCC12CNC(c1nc[nH]c2ncnc1-2)=O N1(C(C(C)(C)OC)=O)CCN(C(C2CCC(C)CC2)=O)C(CC(C)(C)C)C1 N1(C(C)=O)CCN(NC(C2CC2NCc2ccccc2I)=O)CC1 C(C(C)C(F)(F)F)N(C)CC=CC(N1CC(C)(C(F)(F)F)C1)=O CCC(CC)C(C(=O)NC1CC(C)CN(C(c2ccccc2O)=O)C1)OC C(CCC(C)(C)NC(C1CCCCN1CC(F)F)=O)NC(c1nc(C)oc1)=O C#CC1(NC(C2(C(C)NC(C3CCN(OC)CC3)=O)CC2)=O)CCCOC1 Cc1cc(CCC(=O)NC23COC(CNC(C4CCC(C)C4)=O)(C2)C3)c(C)s1 C1(c2n(CC(=C)C)nnn2)(NC(c2ccccc2Br)CF)CCCSCC1 C1(C(=O)NC(CCC)(C)CC)CN(C(C2CC2CC)=O)C2(CCC2)C1 c1(CNC(C=CC(CC)=CC)=O)cc(C(=O)Nc2cccc(C(C)C)c2)ccn1 N1(C(C(CNC(C2CC3(CSC3)C2)=O)O)=O)CCC2(CCC2)CC1 c1(CS(=O)(=O)N(C)CC2(C(F)(F)F)CC2)cccc(Cl)c1 C1(NC(=O)CCF)CCCCC1NC(c1csc(C2CCCO2)n1)=O c1(CN(C(=O)C(c2ccccc2)c2cccs2)c2nn[nH]n2)ccccc1I Cc1ccnc(C)c1C(N1CCCC(CNCc2nccnc2CC(C)C)C1)=O Cc1occ(C(F)(F)F)c1CC(=O)NC1CCN(C(=O)C(O)CF)C1 N1(C(CCC)=O)CCC(C(=O)N(C2CN(C(c3sccc3Cl)=O)C2)C)CC1 C1(NC(Cc2cccc(OC)c2)=O)C2CC3CN(C(C4CCCN4C)=O)C1C3C2 C(=O)(C1CCc2cccnc21)N(CCCNC(c1n[nH]c(C)c1O)=O)C1CC1 CCC(C)(CNC(=O)CCc1ncccn1)NC(=O)COC1CCC1 n1(CCOC)cnc(=NC(=O)N(C2CC2)Cc2cc(C)cc(C)c2)[nH]1 C(=O)(CCCC(C)=O)N1CC(CCC=C)(C(=O)NC(C)CC(N)=O)C1 c1(OC)c(C(=O)NC2CC2)c(C)nn1C.N12CCN(CC1)CC(=O)N1CCC2C1 C(=O)(C1=CCCC(C)(C)C1)NC(C(C)C)CCCC(C(=O)N)(Cl)Cl.C(=O)(C#CC1(C)COC1)O c1(CC(=O)OCC2N(CC)CCCC2)ccc(C#N)cc1.C1(C)CC(F)(CO)C1 N1(C(c2ccn(C(C)C)n2)=O)CC(C(=O)NC(c2ccccn2)(C)C)CC(C)C1 c1(C(=O)NC(C(C)NC(CC=CC)=O)CO)nn(C)cc1S(N)(=O)=O CC(C)(C)C(=O)NCC(=O)NCCNC(=O)CC1CSC1 O=C(C1=CS(=O)CCC1)NCC1CCCC1NC(c1ccnnc1Cl)=O C1(O)(C(N2CCN(C(=O)CC3CCCOC3)C(CF)C2)=O)CCCCCC1 c1(COC)nc(C)c(C(N2CCC(COC)(NC(C3CCCOC3C)=O)C2)=O)s1 c1(C(=O)NC2CCCN(C(C=CCC)=O)C2)ccc(Cl)c(OC(F)(F)F)c1 CC1CCC(Cl)=C(C(=O)NC2(CNC(c3nccc(C(F)(F)F)n3)=O)CCC2)C1 CC1CCN(C(c2ncccc2C(F)(F)F)=O)CC1NC(=O)CCSCC(N)=O N1(C(C2C(C)C2)=O)CC(CNC(c2cnn(-c3ccccc3)c2)=O)C(C)C1 c1(CN(C2CCCN(C(c3c(SC)cccc3)=O)C2)C)ccncc1[N+](=O)[O-] C1(NC(c2c(F)ccc(OC)c2)=O)CCCCN(C(=O)CCCC2CC2)CC1 C1(NC(CCC=C)=O)CCCCC12CCCN(C(=O)C(C)n1cnnn1)C2 C=CCCCCCCC(=O)N1CC(F)(CNC(c2c(C)nc3sc(C)nn23)=O)C1 C1(CC=C)(C(=O)NCC2(CC)CCOC2)CCCN1C(=O)CN1CCCNC1=O CC(CC(F)F)C(=O)N1CC=CC1(C)C(=O)NCCN1CCOCC1 c1(OCC(N2CCC(N(C)C(C3CC34CCC4)=O)C2)=O)ccc(F)c(F)c1 Cc1ncc(N)cc1C(N1CC=CC1CNC(=O)CCc1ccoc1)=O Cc1ccnc2nc(C(=O)NC3CC(C)N(c4nnc(O)s4)C3)nn12 N1(C(C2(Cl)C(C(C)=O)C2)=O)CC(C(=O)N(CCCCO)C2CCCC2)C2(CC2)C1 C1(C(NOC(CC)C)=O)(NC(c2cnsc2)=O)CC(CO)C1 N1(C(C2CCN(C(C(CCC)N(C)C)=O)C2)=O)CCC2(COC(C)C2)C1 C(C(CO)(CO)NC(=O)COCP(C)(C)=O)N(C)C(c1cncc(CNC)c1)=O CN1N=C(C(=O)N2CCOC(C(=O)NCCc3cccc(Cl)c3)C2)CCC1=O CCC(C)C(CC(=O)N1CCCC1CNC(=O)C(O)CCC(C)C)NC(N)=O c1(C(C)(C)C)n[nH]c(=NCC2CC(NC(C34CC3COC4(C)C)=O)C2)o1 C(=O)(C1Cc2ccc(F)cc21)N1CCOCC(F)(CNC(c2c(C)c[nH]n2)=O)C1 N1(C(C2=C(C)CCC2)=O)CCC(C2CC2)(NC(=O)C=C(C)CN2CCOCC2)C1 c1(OC)cccc(C(=O)NC2(C)CCN(C(=O)CCc3ccc(C)o3)C2)c1 C(CC(C)(C)C)(C(=O)NC(C1CCN(C(C2(C(C)C)CCC2)=O)C1)(C)C)OC c1(N2CCCN(C)CCC2)nc(=NCC2CC3CCC3C2)[nH]c2ccccc12 c1(OCC)ccc(OCC(N2CCC2C(=O)NC2CCC(N(C)C)C2)=O)cc1 C1(NC(C2C(C)(C)OCC2)=O)C2CC3C(C2)C13C(=O)NOCC1(F)CCC1 C12(NC(=O)NC(C(=O)N(CCN(C(C)=O)C)C)(C)CO)CCC(C)(C1)OC2 CCC(O)C(C)(C)C(=O)NC1CCC1CNC(=O)CCc1cnco1 N1(C(C=C(CC)C)=O)CC(C)(C(=O)NC2CN(C(=O)OC)C2)C1 c1(OC)ccc2c(c1)CC(C(=O)NC1CC3(C1)CN(C(=O)CC1(OC)CC1)C3)O2 c1(C(N2CC3C(NC(CCC)=O)C3C2)=O)sc2ccccc2c1CC c1(CN2C(CNC(C(C)(C)C)=O)CCC2)c(F)c(F)cc(F)c1F O=C(CCCCCNC(C1(CO)CCOC1)=O)NCC1=CCCCCC1 C1(C#CC(=O)N(C(C)CCNC(=O)C(c2cccc(F)c2)C)C)(CC)CC1 c1(C2c3n(nnn3)CCN2)cc(Br)c(Cl)s1.CC(C)(C)OC(CC=CBr)=O C(=O)(CCCCC(C)C)N(CCC1CC(C)(C)NC1=O)CC c1(C(=O)NCC2(C(C)NC(c3c(C)cno3)=O)CC2)ccc(OC(F)F)cc1 C1(N(C(CN(CC(C)(C)C)C)=O)C)CCCC(NC(c2nnn(C)n2)=O)C1 C1(NC(C(n2nnnc2C(C)(C)C)C)=O)CC12CCN(C(=O)CC1CSC1)CC2 CCCCCCN(C(=O)CC1SCCS1)CCNC(C1CC1C(C)(C)C)=O C(CC(C)(C)C(=O)N1CC(C)(NC(=O)CNC(=O)OCc2ccccc2)C1)SC C(=O)(C(O)C(C)c1ccccc1F)N(CCOCCOCCOC)C CCC(CC(=O)ON1CC(C)C1c1ccc(C)cc1)C(C)(C)C CS(C)(=O)=Nc1cccc(C(=O)NC2CC3(C2)CS(=O)(=O)C3)c1 C1(NC(CC=C)=O)CC2CCC1N2C(C1CC(=O)N(c2ccc(Br)cc2)C1)=O c1(C(N2C(C)CC(NC(Cn3c(C)ccn3)=O)C2)=O)c[nH]c(C#N)c1C c1(C(N(C)CC2CCCC(NC(=O)Cc3cn[nH]c3)C2)=O)cc2cn[nH]c2cn1 C#CCCCCCCC(=O)N1CCC(N(CC#C)C(c2conc2CC)=O)C1 Cc1cn(C)c2nc(N3CCC4(CCCC4Nc4ncncc4Br)C3)ncc12 c1(OC)ccc2nc(N3C4CCC3CC(O)(C(Cl)(Cl)Cl)C4)sc2n1 C1(NC(CCCNC(CN(CC(F)(F)F)C)=O)=O)CCCC(F)C1 N=c1[nH][nH]c(C(=O)NCC2CCN(C(=O)C=Cc3ccccn3)C2)c1Br Cc1cc(OC2CCN(CC3CCCCN3)C2)ccc1N(C)C C1(C(N2C(C)CC(CC(=O)NCCCN3CC=CC3)C2)=O)CN(C)CCN1C c1(OC)ccc(F)cc1C(=O)NCC1(O)CCN(C(c2cc(C)cc(C)c2)=O)C1 c1(C(=O)NCC2N(C(C(C)NC(C)=O)=O)CCC2)cc2nccc(Cl)c2s1 C1(NC(c2nc(C)sc2)=O)COC2(CCN(C(=O)C(C)n3cncn3)C2)C1 CCCC(C)C(C(=O)Nc1cc(OC)cc(C(F)F)c1Cl)OC C1(C(=O)NC2C3CN(C(COC(C)C)=O)C2C3)CC2(CCC(F)(F)CC2)CO1 n1(CC)c(N2CCN(CC(=O)NCC3CC3)CC2)nnc1C1CC1C(=O)O c1(C(N2CCCN(C(C=CC)=O)CC2C)=O)cc(F)cc2nc(S)[nH]c12 c1(C(=O)NC2CC(N(C(=O)CCCN3CCCC3)C)C2)occc1F c1(N)ccc(C)c(Cl)c1Cl.C(C(=O)NCCC1(CNC(=O)C2CC2)CC1)OCCOC N1(C(c2n(C)ncc2)=O)CC2CS(=O)(=O)CC2(NC(=O)CCC2(C)CC2)C1 C(=O)(C1CCCc2c[nH]nc21)NCC1C(NC(=O)CC2NC(=O)NC2=O)CCC1 c1(C(C)=O)cccc(C(=O)N(C)CC2(O)CN(C(=O)C(C(C)C)NC(N)=O)C2)c1 N1(C(C2CC(SC)C2)=O)CC(NC(=O)C(c2ccc(F)c(Cl)c2)(C)C)CC(C)C1 C(N=c1[nH]c(C)nc(C)c1F)C1(F)CC(NC(C2(COC)CC=CCC2)=O)C1 C#Cc1cncc(C(N2CCN(C(=O)CCn3cc(C)cn3)CC2C(C)C)=O)c1 CON=CC(=O)N1CCC(N(C(=O)CCN2CCOCC2)C)C1 C(C)(C(=O)N(CC(O)CN(C)C(C1CC(C(C)C)C1)=O)C)NC(CC)=O c1(C(=O)NCCCN(C(=O)C=Cc2ccccc2F)C(C)C)cc2n(n1)CCC2 C1(C(=O)NCC(C)C(C)O)(SC)CN(C(=O)CCc2ccc[nH]2)C1 n1(CCC(=O)NC2CC3(C2)CC3NC(C23CC(O)C2C3)=O)cnc2ccccc12 c1(C(N2CCCCC2C2CCCNC2)=O)ccc(OC(F)(F)F)cc1Cl c1(C(=O)NC2(CCNC(CC(C)CN(C)C)=O)CC2)ccc(F)c(F)c1 N1(C(c2cccc(SC)c2)=O)CCCCC1C1CCCN1C(C1(C)OCCO1)=O N1(C(CS(=O)(=O)NC)=O)CC2CCCC2(C(=O)NOCC)C1 C(=O)(C(C)(C#N)CC)NCC1CC(NC(CC2ON=C(CC)C2)=O)C1 c1(C(=O)NCC(C)NC(C2(CCF)CCC2)=O)ccc(C(C)(F)F)nc1 C1(CC#C)CN(C(=O)CN(C(=O)C(C)COC)C(C)C)CCO1 N1(C(c2c(CC)nco2)=O)CCC2(CCC2)C(NC(c2cc(CO)n(C)n2)=O)C1 N1(C(N(CC)CC)=O)CC(C2(NC(=O)C(C)C(C)CC)CC2)C1.c12ccc(o1)C2 C1(CNC(=O)Cc2ccc(F)cc2)CC2(CCN(c3ncc(F)cn3)CC2)CO1 C1(C)(C(N(CCC(C)NC(=O)CCc2ccn(C)n2)C)=O)CCOC1 N1(C(C(C)SCCCC)=O)CC2CCCC(CNC(c3sc(O)nc3C)=O)C2C1 N1(C(C(CC)OCC)=O)CC2(CCN(C(=O)CC3CCC4(CCC4)CO3)CC2)C1 C1(NC(C2CCSC2)=O)CCC12CCN(C(C1CC1c1ccccc1)=O)CC2 C(=O)(C(C)(C)C(=O)NC1CCCN(C(c2ccc(O)nn2)=O)C1)NC c1(CNC(c2c(C)nns2)=O)ccc2c(c1)CN(C(=O)C(C)O)C2 CC(C)(C#N)C(=O)NCC1CCCC1NC(c1sccc1C(C)(C)C)=O c1(C(N2CCC(CF)C2)=O)cnc(-c2ccncc2)cn1 CC1CN(C(C2CC2C2CCC2)=O)CCN1C(=O)CC(F)(F)F Cc1ccc(Cl)c(C(=O)NC2CC2NC(=O)Cc2ccc(C(=O)N(C)C)nc2)c1 N1(C(CC2ON=C(CC)C2)=O)CCOCC(F)(CNC(c2ccc(C)o2)=O)C1 CCC(CC)C(F)C(=O)N(CC(O)CNC(C1CCC(O)CC1)=O)C c1(C(CNC(c2cnc[nH]2)=O)NC(c2cc(Br)n[nH]2)=O)ccccc1F c1(C(=O)NC2(c3nn[nH]n3)C(C)C2)cnc(O)[nH]1 N1(C(c2c(C)nc(C)o2)=O)CCC(NC(=O)C(C)(C)C2CCOC2)CC1C C12(C(=O)NC(CC=C)C(=O)Nc3cnc(F)nc3)CCCC1CCC2 C1(N(C)C(C2CCN(C)CC2)=O)CN(C(=O)C(c2cccn2C)=O)CCC1O Cc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)CCCCCc1cccs1 C=CCC(C(=O)N1CCCC1CNC(C1(S(C)(=O)=O)CCOCC1)=O)C(C)(C)C c1(C(N2C(CNC(CN(CCC)C)=O)CC2)=O)csc(-c2cccs2)n1 c1(OC)cc(Cl)c(C)cc1C(=O)NCC1(CNC(c2nc(C)n(C)c2C)=O)CC1 c1(C(=O)NC2C(OC)CN(C(=O)C(C(C)C)SC)C2)c(C)nn(CCO)c1C c1(C(=O)NCC(CNC(c2cccc(CCC)c2)=O)O)cccc2nc(Cl)cn12 Cc1cc(C(N2CCC(NC(=O)CSC(F)(F)F)CC=C(Cl)C2)=O)cc(N)c1Cl c1(C(=O)OC)ccc2c(c1)C(C(=O)N(C(C)CNC(c1cnc(Cl)s1)=O)C)CO2 C1(C(=O)OCCC2CC(C)OCC2)CC(C)(C)CCN1C(=O)OC(C)(C)C c1(CC(=O)NCC(CNC(c2nnn(C(C)(C)C)n2)=O)F)ccc(F)cc1F C1(NC(C(CCC)N(C)C)=O)CC2C1CCN2C(=O)CC(=O)N(C)C C#CCC(C)(C)C(=O)NC(C)CNC(C1C=CCCC1)=O N1(C(C(CC)(C)CNC(c2nocc2Cl)=O)=O)CC2(CCCCC2)C1 Cc1cc(N(C)C)ccc1CNC(=O)C(CO)c1ccccc1.N12CC(C1)C2=O C1(NC(C=C(C)C)=O)Cc2ccccc2C1NC(c1cnc2c(n1)CCCC2)=O C(C(F)(F)CNC(c1ccccc1-n1cccn1)=O)(C1CC1)OC c1(C(=O)NC(C(C)NC(=O)C(O)c2ccco2)CO)cc(F)c(F)c(F)c1 C(=O)(C1=CCCOC1)N(CC(=O)N)C1CC1.C1(C2CC2)CNC(=O)OC1 N1(C(c2n(CC)nnc2)=O)CCC2(CCOC2)C(CNC(c2cc[nH]n2)=O)C1 CC(C)C(C(=O)NC1CCN(C(=O)C=Cc2cccs2)CC1)c1ccc(Cl)cc1 C1(C(=O)NCC(CNC(c2cnccc2C(F)F)=O)O)CCCC1C1CC1 N1(C(C2CN(C(CC3CC(=C)C3)=O)CC2(C)C)=O)CCCC2(CCCC2)C1 CC1(C)CCN(C(=O)Cc2ccon2)C(C(=O)NC2CCN3CCC2C3)C1 c1(SC)ccc(Cl)c(C(N2CC3CCC3(CNC(=O)CC3CCCN3C)C2)=O)c1 C1(C(N2CC(NC(c3cccc(N)n3)=O)(CF)C2)=O)CN2CCC1CC2 C1(C(=O)NC2C(O)C3CCOC23)CN(C(C2(CCCF)CC2)=O)CC12CC2 N1(C(CC=CC)=O)CCN(C(c2nc(C)sc2Br)=O)CC1C c1(C(N(CC(C)NC(=O)C(O)C(F)F)CC)=O)cc(S(C)(=O)=O)cnc1O C1(C(=O)OC)C2CCCN1C(=O)OC(=O)C(C)N(C)CC(=O)N2.C(C)(C)(C)OC C12(NC(CCC3CC(OC)C3)=O)COC(CNC(C3CCC(C)C3)=O)(C1)C2 c1(OC)ccc(OC(=O)COc2cccc(F)c2)c(C)n1 C1(CNC(C2C(CC)C2)=O)CCN1C(=O)C(C)n1cncn1 c1(CN2C(C(=O)N=c3[nH][nH]cc3Br)CC3CC32)cccc2ccncc12 C(=O)(C#CC(C)(C)O)NC(CNC(CCCCSC)=O)(C)C1CCC1 C1(CN(C)C(c2cnc[nH]2)=O)CCCCN1C(C1(C)CCC1)=O Cc1cc2c(cc(C(=O)NCC(C)(C)CNC(c3ccoc3)=O)n2CC2CC2)s1 C1(CC=C)(NC(=O)C(C)c2cccs2)CCN(c2nc(C(C)C)ns2)CC1 C(C)(CNC(c1cc(Cl)cs1)=O)(CO)NC(CSCC(C)C)=O C(C)(C)(CC(F)C(=O)N1CCC(OCC(N)=O)C1)NC(c1c(C)nc(C)o1)=O c1(N2CC(O)(C(C)NC(c3nc(CC)sc3)=O)C2)ccc([N+](=O)[O-])c(C)c1 c1(C(N)CC(=O)NCCn2cc(C3(O)COC3)nn2)cc(F)c(F)c(F)c1 C1(CC)CN(C(=O)Cc2ccccc2Cl)CCN1C(=O)CCN(C)C(C)=O c1(C(=O)NCC(C)N(C(c2c(C)cc[nH]2)=O)C)c(C)nc2ccccn12 C1(CNC(c2coc3c2COC3)=O)CC2COCC2N1C(=O)Cn1cnnc1 c1(CC)c(C(N2CC=CC(NC(=O)CNC(=O)CC(F)(F)F)C2)=O)nnn1CC C(=O)(CCS(=O)(=O)C1CCCC1)N1C2C(NC(=O)C=Cc3ccoc3)CC(C2)C1 C1(C(=O)NCC2CCC(N(C)C(C3(C)CCCCO3)=O)CC2)CCC2(CCC2)C1 C1(CNC(CC=C=C)=O)CCC2(CO1)CC(NC(=O)Cn1cc(C)cn1)C2 C1(C(C)(C)C)OCCC1CNCC1(F)CCNC1 CC1CCN(C(=O)C(C(C)C)NC(C2CCCN2C=O)=O)C(C)C1 N1(C(C(CCSC)O)=O)CC(C)CN(C(C2CC2(F)F)=O)C(C)C1 N1(C(CCc2onc(C)n2)=O)CCCCC(C(=O)NCCCCC(C)(F)F)C1 Cc1nn(CC(=O)N(CC(C)(C)CNC(C2SCCC2C)=O)C)c(C)c1C Cc1noc(C)c1C=CC(N1CCCCC1CCN(C(=O)CC1C=CCC1)C)=O Cn1cccc(C(=O)NCC(CC2CC2)C(=O)NCC2CCCC2(C)C)c1=O C12(C(N3C(COC)C=CCC3)=O)CCN(C(=O)C=Cc3cncn3C)CCC1C2 n1(CC)nc(C(=O)NC(C)C(C)NC(c2coc(CS(C)(=O)=O)n2)=O)cc1O c1(N(C(=O)NCCN(CCCC)Cc2cccc(Br)n2)C)ccc(F)cc1 Cc1cc(C)c(CC(N2CCC(N(C(=O)C(F)=CCCF)C3CCC3)CC2)=O)s1 CC(C)(CC(F)F)C(=O)N1CCC(F)(CNC(C2CC(OC(F)F)C2)=O)CC1 c1(C(=O)NCC(CO)NC(CCC2CCCN(C)C2)=O)c(O)ccc(Cl)c1F CC1CC(NC(=O)C=CC2CCCO2)CCN1C(C1CC2CCC1C2)=O N1(C(CN(C)CC)=O)CCC2(C1)CN(C(=O)CCC(C)c1ccccc1)CCO2 Cc1cncc(C)c1C(=O)NCCCCCC(=O)N1CCC(F)(CF)C1 N1(C(CCC(C)OC)=O)CC(NC(=O)CCCc2cccnc2)C2CCCCC12 CC(C)CC(C)OCCC(=O)NCCCC1CCCN1C(C1(CC2CC2)CC1)=O N1(C(c2ccc(OC)s2)=O)CCCCC1C(N1CCOC(C2CC2)C1)=O Cc1nn(C)c(C)c1C(=O)NC(C)(C)C(=O)N(C)CC1COCCO1 C1(NC(=O)CSC2CC2)CCCCC1N=c1cc(Cl)nc(-c2ccccn2)[nH]1 c1(C(=O)OCC)ncc(F)cc1NC(C1C2CC1N(C(=O)CC1CCCC1)C2)=O c1(C(C)=O)ccc(C(=O)NCCN(C(C2CCCCN2C(C)C)=O)CC)c(F)c1 C1(C(N(C2CCN(C(COCCCC#C)=O)CC2)C)=O)C2CCCCCCC12 CC(C)CC(O)C(=O)N1CCCC(CNC(=O)CC2OCCC2(C)C)CC1 C1(CC(C)NC(C2CC3(CC3)CO2)=O)CCN(C(C2CC3C=CC2O3)=O)CC1 Cc1cn2c(CC(=O)NCC(CO)NC(c3c[nH]cc(Cl)c3=O)=O)csc2n1 c1(OC)c(-c2nc(CN=[N+]=[N-])no2)ccc(C)c1F N1(C(C(c2ccccc2)OC)=O)CCC(NC(C2CC2[N+](=O)[O-])=O)C(F)(F)CC1 c1(C(=O)NCC2CCN2C(C2CCOC2=O)=O)cccc2c1CCOC2 C(=O)(CC(O)CNC(C1CCCCC1O)=O)NCc1c(CC)nns1 S(=O)(=O)(c1ccc(NCC2(CO)CC(C)C2)cc1Br)N(C1CC(=C)C1)C C1(C(N(C(C)C(C)(C)C)C)=O)CC2CC1CC2NC(=O)COCC(C)(C)C C(=O)(C1=CC2C=CC(C1)C2)NC(CC#C)C(=O)NC1CC(OCC)C1 C1(NC(CN(C(=O)Cc2cn[nH]c2)CCOC)=O)CC(=O)NC1=O C1(C(=O)NCC2(CC(=O)NC(C3CCOCC3)C#C)CC2)CC2CC1CC2=O N1(C(c2c(C3CC3)[nH]c(=N)s2)=O)CC2CC(NC(c3ccc(Cl)nc3)=O)CC2C1 c1(C(=O)NC2CC(NC(C3C4CCC(F)C34)=O)C2)ccc(-c2ccccc2)nn1 c1(CC(=O)NC2(CN(C(=O)CCS(C)(=O)=O)C)CC2)cccs1 C1(NC(CCN(C(C(CC)(C)OC)=O)C)=O)CC2COCC2C1 N1(C(CC=C(C)C)=O)CC=CC1CNC(C1CCC(Cc2ccccc2)O1)=O CC1(C)C(C(N2CC=CC2CNC(=O)CCCc2nccs2)=O)C1C(F)F C1(C(=O)NCCCn2ncc(C)c2)(NC(=O)C(F)C(C)C)CCC(C)(C)C1 c1(C(=O)OCC)cnc(Nc2nc(C)ncc2COC)nc1C(F)(F)F c1(COCC)cccc(SCc2nc(C)ns2)c1 c1(CCC(=O)NC(CNC(C2(CCCC)CC2)=O)(C)CO)cccc(OC)c1F c1(C(N2CCC(CNC(c3c(C)ccn3C)=O)C2)=O)nc(C2CC2)ncc1Cl N1(C(C2(OC)CC(C)C2)=O)CCCC(NC(c2nnsc2SC)=O)C1 N1(C(c2c(C)cc(F)s2)=O)CCC(NC(c2cc(C(C)(C)C)ccn2)=O)C12CC2 CC1CN(C(c2cnccn2)=O)CC1NC(=O)CCOCCOCCCO c1(C(=O)NC23CC(CNC(C(C4CCC4)OC)=O)(C2)C3)cc(CO)c(C)o1 Cc1cnncc1C(=O)NCC(CO)NC(=O)CCC1(C#N)CCC1 c1(C(N2CCC(N(C(=O)CC3CCCC(O)C3)CC)C2)=O)cc[nH]c2nccc1-2 CC1OCCC1C(=O)NCCN(C1CCCC1)C(C1CCCC1)=O c1(C(N2C(CCCNC(c3n(C)nnc3)=O)CCC2)=O)cc2ccc(F)cc2[nH]1 C1(C(N2CC(CC)N(C(C34CSCC3C4)=O)CC2)=O)CN=C2N=CNN2C1 C(=O)(CCCCCN(C)C(C1CC1)C1CC1)N(C)Cc1c(C)n[nH]c1C c1(C(N2C(C)CC(NC(c3ccccc3OC(F)F)=O)C2)=O)ccnn(C)c1=O C1(NC(C2CC(F)(F)C2)=O)CN(C(C2CCCS(=O)(=O)C2)=O)C2(CCOC2)C1 c1(C(N2CCC3CCC(NC(C4(C)CC4(F)F)=O)C32)=O)n[nH]c2ccc(F)cc12 C1(CNC(CC2N(C(CC3(N(C)C)CCC3)=O)CC2)=O)CCCC2(CC2)C1 CCC(C)(O)C(=O)NC1C2CN(C(c3ccc(C4CCC4)nc3)=O)CC12 c1(N(CC)CC)ccc(C(=O)NCC2(NC(=O)C(C)C(C)n3cccn3)CC2)cc1 C12(C(N3CC(OCCNC(C(C(C)C)O)=O)C3)=O)C(=O)C3CCC1C2C3 C(=O)(C(C)CC(C)C(C)=O)N1C(CC(=O)Nc2cn(CCC)nc2)CCCC1 C1(CC)CCC(=O)N1C(=O)CCCc1nnc(-c2ccc(C(C)C)cc2)s1 C1(C(=O)NCC(C)N(C(CN(CCC#C)C)=O)C)(CF)CCOCC1 C1(N(CC)Cc2ccoc2C)CCN(C(=O)OC(C)(C)C)C2(CC2)C1 CC1(C#CC(=O)N2CCC(Nc3ncc([N+](=O)[O-])cn3)C(F)(F)CC2)CCCO1 S(=O)(=O)(CCCCCl)OC(c1cccc(Cl)c1)C(=O)OCC1CC(OC(C)(C)C)C1 O=C1CC2(CO1)CN(C(=O)C(Cn1ccnn1)NC(C1CC1Cl)=O)C2 C(=O)(CC(O)CC(C)(C)C)NCCCN(C(c1c(SC(C)C)cccc1)=O)C N1(C(C(C(=O)OC)(C)F)=O)CC2OCC(NC(=O)Cc3ccno3)C2C1 Cc1nc2cncc(C(N3CCC(C)C(CNC(=O)C(C)(F)F)C3)=O)c2[nH]1 c1(OC)cc(C(=O)Nc2c(Cl)ccnc2Br)cnc1-c1cnc(F)c(F)c1 CCCCCC(=O)N1CCN(CC2CCCN(C(C3CCCCO3)=O)C2)CC1 N1(C(c2c(OC)c(C)cs2)=O)CCC2(CCCN2C(=O)Cn2cc(Cl)cn2)C1 N1(C(C(C)n2cccn2)=O)C2CCC1CC(N(C(=O)CCCC1CC1)C)C2 c1(C(=O)NC2CN(C(=O)Cc3csc(Cl)c3)CC2O)cccc2nc(O)ccc12 N1(C(C2CCN(C(CNC(=O)NC)=O)C2C)=O)CCCCCCC1C c1(OC)ccc(S(N)(=O)=O)cc1NC(C1CNC(=O)C1(C)C)=O C(=O)(C(O)C(C)(C)C)NCCC(C)NC(c1cccc(CO)c1)=O.c1(N)ccccn1 c1(C(C(=O)NC2CC(CNC(=O)CCCF)CC2O)=O)cc(Cl)cc(Cl)c1 CC1CN(C(=O)Cc2nc(=N)[nH][nH]2)CC(C)N(C(c2cc(O)ncn2)=O)C1 C1(C(N(C)Cc2cn(CC)nn2)=O)CC(OC)CN1C(c1ccncc1NC)=O c1(OC)cc(C(=O)NCCCN(C)C(c2cnc(S)nc2)=O)sc1Cl N1(C(C(CC(C)(C)C)OC)=O)CCCC12CCCN(C(=O)C=C(C)C(C)(C)C)C2 C1(NC(c2c(OCC)scc2)=O)CN(C(C2CN3CCC2CC3)=O)C(C)(C)C1 c1(CC)cc(Cl)ccc1NC(=O)C(O)C1CN(C(C2(CF)CC2)=O)C1 C1(C(=O)NC(C2(CNC(c3ccc(C=C)cc3)=O)CC2)C)CCCC2(CCC2)O1 c1(CNC(c2c(C)nc(-c3ccc(F)cc3)s2)C)cccc2c[nH]nc12 N1(C(C(C)=C(C)C)=O)CCN(C(=O)CCc2ccoc2)CC1CO C1(C(=O)NCC(CC(C)C)NC(=O)C(c2ccncc2)C)CCCCN1N=O c1(CC)nn(C)c(CC(=O)NC2(CNC(C3(OC)CC3)=O)CCCCC2C)c1Cl C(=O)(C(C1=CCCCC1)N1CCCC(c2noc(CC)n2)C1)NC(C(=C)C)=O C12(NC(=O)CCF)CCCC1N(C(C1CCC(C(F)(F)F)O1)=O)CC2 CC1CCC(C(=O)N(CC(C)CO)C)N1C(C1CCOC1(C)C)=O c1(C(N(C2CC(NC(=O)CCN3CCCC3)C2)C)=O)cc(F)c(Cl)cc1Cl N1(C(C(CC)OCC)=O)C2CCC1C(C)C(NC(=O)Cc1cnccn1)C2 Cn1cc(Cl)cc1C(=O)NCCOCCC(=O)N(CCF)C1CC1 c1(OCC(=O)N(C2CCCN(C(=O)C3CC3)C2)CC)ccc(Br)cc1 C1(NC(Cc2c(C)n(C)cn2)=O)CN(C(c2ncoc2C(C)C)=O)CC1N=[N+]=[N-] Cc1cc(C(=O)NC2C3CC2N(C(c2ccnc(O)c2)=O)C3C)ncc1F c1(C(C)C)ncc(C(=O)NC(CNC(=O)CC(=O)N(C)C)C2CC2)s1 Cn1nncc1C(=O)NCCSCC(=C1CN(C(=O)CCN(C)CCO)C1)F C1(CNC(c2ccc(OC)s2)=O)CC2CC2N1C(=O)Cc1ccccc1Br CC(C)(C)S(=O)(=O)CC(=O)NCC1CC(O)CN1C(c1cccc2c1OCC2)=O c1(C(=O)NC(C)CNC(c2cnn3c2NCCC3)=O)cncc2c(F)cccc12 Cc1sc(C)c(C(=O)NCC2CC(O)CN2C(C2CCCN2C)=O)c1C#N c1(C(N2CC(CCOC)N(C(=O)C=CCO)CC2)=O)cccc2scnc12.C(C)(=O)O C=C(CNC(C1CC1(F)F)=O)CCNC(c1nocc1C)=O S(=O)(=O)(c1ccc(NC2CCC(O)CC2)c(Br)c1)NC(c1ccnn1C)COC c1(C(N(CCN(C(c2cnnn2CC)=O)CC)CC)=O)cccc(C(C)C)c1F C(=O)(C1=CC(O)C(NC(=O)CN(C)C2CC2)C1)N(C)CC1CCCC1O C1(COC)(NC(c2csc(O)n2)=O)CCN(C(C2COC(C)C2)=O)CC1 O=C1CC(C(N2CCC(N(C(=O)Cc3cnoc3)CCO)C2)=O)CC(=O)N1 c1(C(C(=O)NCC(C)C)N(C)Cc2ccc(F)cc2)cccc(OCCCCl)c1 c1(N2CCC(CC)(CO)C2)nc(N2CCCC(CC3CC3)C2)nc2c1ncn2C c1(C(N(C)CC2N(C(C(C)SC(F)(F)F)=O)CCC2)=O)cc(N)c(F)c(F)c1F C1(CC)(CC)C(OC)CC1N(C)C(=O)NC1CCN(C)CC1 Cc1nc(Cl)c(NC(C2CC23CCN(C(c2cc[nH]c2)=O)CC3)=O)cc1Br C1(CNC(C(N2CCN(C(C3(C)CCC(=O)C3)=O)CC2)C)=O)CCC2(CCC2)O1 N1(C(C2(C(=O)OC)CC2)=O)CCC2CN(C(c3cnc(Cl)cc3C)=O)CC2C1 n1(CC(=O)NC(C(=O)N(CC(C)SC)C)Cc2cn[nH]c2)cnc(C#N)n1 C1(CC(=O)NCC2C(NC(C(C)(C)OC)=O)CC2)CCCC(C2CC2)O1 c1(OCC(=O)NCCCN(C(C(C2CCCC2)OC)=O)C)cc(Cl)ccc1C C1(NC(CC=C(C)C)=O)CCCC12CN(C(C1CC3(CCCC3)CO1)=O)C2 C1(NC(CN(C(=O)Cc2cnn(C)c2)CC#C)=O)COC2(CCC2)C1 C1(C)(C(=O)NCC2(C(=O)OC)CCC2)CC(O)CN1C(c1ccc(F)c(O)c1)=O C(CCN=c1[nH]nc(O)s1)N(C(c1c(C)cno1)=O)CC1CCCCC1 C(=O)(C(F)C(F)(F)C(F)(F)F)NC(C)CNC(=O)C=Cc1cnc(C(C)(C)C)s1 c1(NC(c2n(CC)nnn2)c2nscc2Br)ccc(C(=O)NC)c(F)c1 C1(C(=O)NCC2OCCN(C(c3cc(C)ns3)=O)C2)OCC2CCCCC12 C1(C(NOC(C)(C)C)=O)CC(=O)N(C(c2ccc(Cl)cc2)CC)C1.C(C(=O)O)NCC#N N(C(=NCCSC)NCC(c1cccc(Cl)c1)OC)CC1(COC)CC1 C1(C(=O)NC(CC=C)CNC(C2CN(S(=O)(=O)CC)C2)=O)CN(C)C(=O)CCO1 C(=O)(CC(C)P(C)(C)=O)NC1C(C)CN(C(C2(C(C)(C)O)CC2)=O)C1 c1(C2(C(C)NC(C3(C(=O)OC)CCC3)=O)CC2)ccc(Br)cc1 C1(C(N2CCN(C(=O)CCC[N+](=O)[O-])C(CCO)C2)=O)CCN2CCOCC12 c1(C(N2CC=CC(NC(C(C)CC3CCC3)=O)C2)=O)nc(Cl)cc(N)c1Cl C1(CNC(CSCC#C)=O)COCC1NC(=O)CCC1(C#N)CCC1 c1(CC(=O)N(CCNC(C(C(COC)C)C)=O)CCOC)cnc2cccnn12 c1(C(=O)NC2(CC=C)CCNC2)cc(F)c(F)cc1NC(=O)N(C)C N1(C(c2c(C)n(CC(C)C)nc2)=O)CCN(C(=O)CCC2CC2)CC1CO C(=O)(CP(=O)(C(C)C)C(C)C)N(CCC(C(C)C)NC(C(C1CC1)OC)=O)C C(CC(C)(C)C)(C(=O)NC1CCC(OC)CC1)NC(c1n(C=C)ncc1)=O C(=O)(C(C)(C)CCC#N)N1CCCC(C(N2CC(C)C2(C)C)=O)CC1 c1(C(CNC(C2SCCS2)=O)=O)cc(F)ccc1Br c1(CC)csc(CNC(c2cc(CNC(=O)C(C3CCC3)OC)on2)=O)n1 CC(C)(CNC(=O)CC1CC2(C1)CN(C(=O)C1=COCC1)C2)C1=CCCC1 c1(Cc2ccccc2)cn(C2CCCc3cnccc32)nn1 c1(C(=O)NC(c2c(OCC)cccc2)C(C)NC(C)=O)ccc(C)n(C)c1=O C(=O)(C(C)(COC)OC)NC(COC)CNC(=O)CCSCC(C)C C(=O)(C1=CC(C)CC1)NC1C2CN(c3c(C(=O)OC)cccn3)CC21 c1(C(N2CCC(C(N(C)Cc3c(C)n[nH]c3)=O)(CF)C2)=O)ncn2c1CCC2 Cc1ccc(F)c(C(=O)NC(C)CNC(c2ccc(OCC(F)(F)F)o2)=O)c1 CC1(C(=O)NC2CC2NC(c2cnn(CC(=O)NC(C)(C)C)c2)=O)CC1(Cl)Cl C1(NC(CN(CC)CC)=O)CN(C(C2CCCC(C)CC2)=O)CCC1(C)C N1(C(C2(CCCC)CCC2)=O)CCOCC(C(=O)NCCNS(C)(=O)=O)C1 C1(C(=O)NCC2CC2(Cl)Cl)CCCCN(C(=O)C=CC2CCCC2)C1 c1(CC(=O)NC2CCC(N(C(=O)COc3ccon3)C)C2)cncc(O)c1 C1(C(N(CC(=O)OC)C)=O)(CC)CCCN(C(C2(SC)CCOC2)=O)C1 CC1CCC(C(=O)NCC2CC(O)C(O)C2)CN1C(C1CC1(F)Cl)=O N1(C(C(CC)CC)=O)CCN(C)CC1CNC(=O)C(c1ccc(Cl)cc1)CO C1(C(=O)Nc2c(CC)noc2)CC(NC(=O)C(C#N)CC)CCO1 c1(C(=O)NC2CCN(C(C3(OC)CCCC3)=O)C2)cc2cc(F)ccc2s1 C(CCS(=O)(=O)C(C)C)N(CCCNC1CCCN(C(COCCC=C)=O)C1)C N1(CC(c2cc(C(=O)OC)ncc2)=O)CCN(Cc2ccccc2F)CC1C c1(N(C2CC3CC2CN3)C(C2CC(=O)C2)=O)cc(F)c(F)cc1Br C1(C(=O)NC(CC(C)NC(c2ccc(C(F)F)cn2)=O)C)CCS(=O)(=O)N1 c1(SC(C2(C)CC2(F)Cl)=O)ccc(Cc2cn(CCN3CCSCC3)nn2)cc1 Cc1ncccc1C(=O)NCCOCCN(C(=O)C(C)N(C(C)C)C(C)C)C N1(C(COCC(=O)OC)=O)CCCC(O)(CNC(c2nn(C)cc2Cl)=O)CC1 Cc1cc(CC(=O)NC2CCN(C(c3sncc3Br)=O)C2)cc(F)c1 N1(C(C2(CCC)CCC2)=O)CCC(C(F)CNC(=O)Cn2cc(C)cn2)CC1 c1(C(N(C)CC2CCCN(C(C(C)C)=O)C2)=O)c2c(cc3c1CCC3)CCC2 C1(C(=O)NCC2(NC(c3ncsc3Br)=O)CCC2)CC2CCC1O2 N1(C(C(C=CC)O)=O)CCC(OC)C(CO)CC1.n1(CC(=O)N)nc(C)nc1C C=C(C)CC(C(=O)Nc1cnn(C2CC2)c1C)NC(C1CCOC1CC)=O C(=O)(C1=CC(C)(CC)C1)NCCCC1N(C(CC)=O)CCCC1 c1(NCC(c2cccc(C)c2)(C)C)[nH]c(=NC2CCCC2C#N)nc2scnc12 c1(SC)ccc(C(N2CCOCC2CC(N2CCC(C)(C(N)=O)C2)=O)=O)cc1 C=CC(C)(O)CC(=O)NCC1CC(C)CCN1C(=O)Cc1sc(S)nc1C C1(CC(=O)N(C(C)CCNC(c2cnn[nH]2)=O)C)(CO)CCCCC1 c1(CC(=O)NC2CC(N(C)C(c3ncccc3Cl)=O)C2)cnn2c1CCCC2 c1(C(N(C2C(C)CN(C(=O)Cc3cnnn3C)CC2)C)=O)ccc2nnnn2c1 Cc1ccccc1-c1cc(C(=O)N(C)CC2C3CN(C(=O)C=CCF)CC23)no1 N1(C(c2nc(N(C)C)oc2)=O)CCN(C(c2csnn2)=O)C(c2cn[nH]c2)C1 c1(C(N2CC(C(N3CC(O)C(F)C3)=O)(CC)C2)=O)cccc2cncn12 N1(C(CCOC(C)C)=O)CCC(CCNC(c2ccc(=N)[nH]n2)=O)CC1 Cc1cc(C(=O)N(CCC(C)NC(c2ncn(C(C)C)n2)=O)C)n(C)n1 Cc1cccc(-c2cn(C(C)C(=O)NC(c3ccccn3)(C)C)nn2)c1 C(=O)(C1=CCCCO1)N1C(C(=O)NCC(C)C2CC2)CCCC1 N1(C(C(C)CC2CCC2)=O)CCC2(CCC2NC(=O)CC2(C)OCCO2)CC1 c1(C(=O)Nc2cnns2)cccc(-c2cnc(NCc3ccc(Cl)cc3)nc2)c1 N1(C(c2nnn(COCC)c2N)=O)CC(CNC(=O)C(C)CSC)CC12CCC2 c1(C(N2CC3C(CNC(c4ccnc(OC)n4)=O)C3C2)=O)nccc(Cl)c1O c1(C(=O)NCC(C)(NC(COCC)=O)SC)c(C)nsc1NC1CC1 C(CNC(=O)C(c1cnn(C)c1)O)(CCCC)NC(COCCC=C)=O c1(CC(=O)NC2CC(C(N3CCC(c4ccccc4)C3)=O)C2)ccc(O)c(O)c1 C1(CC(=O)NCCCCCN(C)C(c2cn(C3CC3)nn2)=O)CCCCC1(F)F C(CC)(CC(C)O)NC(CCN(C(C(CC)OCC)=O)C1CC1)=O C1(NC(C2CCC(=C)CC2)=O)CN(C(=O)C(C(C)C)NC=O)CC(C)(C)C1 N1(C(C(CC#C)O)=O)CCN(C(c2cnn(C)c2Cl)=O)CC1CCOC c1(C(c2n(CC(=C)C)nnn2)NC2(C(=O)NC(C)C)CC2)ccc2occc2c1 c1(N(C(=O)CC2CC3COCC23)C)cccc2cccnc12 C1(NC(C(C)=C2CCCC2)=O)CN(C(C2CCN(CC(C)C)C2)=O)CC1C c1(CC(=O)NC2C(NC(C3(OCC)CCSC3)=O)COC2)nc(C)sc1C N1(C(COC(C)C)=O)CCCC(C(C)(C)C(=O)NC2(CCO)CCOC2)C1 c1(CC(=O)NC2CN(C(C3C(CCC)C3)=O)CC2O)cc(Cl)ccc1OCC N1(C(C2C=CCC2)=O)CC23CCCCC2(C1)CN(C(C1(C(F)F)CCCO1)=O)C3 C(=O)(C(CN(C)C)N(C)C)NCCN(C(=O)C(F)C1CCCC1)CC CCC(C)(C(=O)NCC1CCC(C)(C)CN1C(c1cc(C)nn1CC)=O)C(N)=O c1(C(C)(C)C)ccc(C=CC(=O)NCC(CO)NC(C2(C)C=CCCC2)=O)cc1 c1(C2N(CC3CC3CNC(C3N(CC)CCC3)=O)CCC2)ccc(OC)cc1Cl N1(C(CCC=CCC=C)=O)CC(NC(=O)C(Cc2ccccc2)OC)CC(F)C1 c1(C(N2CC(C)C(NC(c3cc(CN(C)C)c[nH]3)=O)C2)=O)cc(Cl)c(F)cc1Cl CC1(C)CC(C)(CNC(=O)C2=CCCCO2)CN1C(c1ccc(C(F)(F)F)s1)=O N1(C(c2cccnn2)=O)CCCC2(C1)CN(C(c1cc(Cl)ccc1O)=O)C2 Cc1[nH]c2ncccc2c1C(=O)OCC1CCCO1.C12CC(CCO1)OC2=O C1(NC(CNC(CCOC)=O)=O)CC(NC(=O)CNc2ncccn2)C12CCC2 N#Cc1nnc2ccccc2c1N1CCC(O)(CNC(=O)C2=COCCO2)C1 Cc1nc(C(N2CC=C(CNC(=O)CCS(C)=O)CC2)=O)ccc1Br Cc1ccnc(C(C)(C)C(=O)NCC2CCC(NC(c3cn(C)c(O)n3)=O)C2)c1 C=CCCC(C(=O)NCc1noc(C(N)=O)n1)NC(C1CC1C1(C)COC1)=O c1(C(=O)OC(C)(C)C)coc(C(C)NC(=O)OC(C)(C)C)n1.CC1C(=O)N1 c1(C(N2CCC(CCNC(CN(C)CC)=O)CC2C)=O)ccc(Cl)c(OC)c1F N1(C(c2cc(C)cc(O)c2)=O)CC(C)(C)OCC1CNC(=O)CCC1CCOC1 c1(N(C)Cc2nn(C)cc2Br)nc2cc[nH]c2c(=NCC2CC23CCOCC3)[nH]1 n1(CC)nc(C)c(C(N2CCC(O)(CNC(C3(COC)CC3(F)F)=O)C2)=O)c1C Cc1nc2ccc(C(N3CC4(CCCCN4C(=O)C4=CCC4)C3)=O)cc2s1 c1(COC)cc(C(=O)NCC2CCCN(C3CC3)C2)ccc1OC(C1(F)CC1C)=O c1(C(N2C(CNC(C(CCC)OCC)=O)C(C)(C)CC2)=O)ccc([N+](=O)[O-])cn1 N1(C(C(CCC)NC(N)=O)=O)CC2CC1CCN2C(=O)CCCCCSC N1(C(CCCCN(C(C2CCN(C)C(=O)C2)=O)C)=O)CCCC(C2CCC2)C1 C1(C(=O)NC2CC(C)CN(C(c3csc(O)n3)=O)C2)CC2COCC(C1)C2 N1(C(CCN(C)CC)=O)CCCCC1C1CCN(C(=O)CCC2CCC2)C1 C1(C(=O)NC(C(C)SC)C)CC=CC(NC(=O)CCn2ccnc2)C1 C(C1CCCC1)=CC(=O)NC(C1CC=CCC1)C(=O)NCC1CC(=C)C1 C(=O)(CCC(C)(C)F)NC(C(=O)NC(C)COCC1CC1)CC1CC1 CC(C(=O)NCC(C)(Cn1cccn1)NC(c1n[nH]c(C(C)C)n1)=O)S(C)(=O)=O C(=O)(C1CCCc2ccnn21)N1CC(NC(=O)CCOCC2CC2)C2(C1)CCC2 C1(NC(c2ccc([N+](=O)[O-])cc2)=O)CN(C(c2cnc[nH]2)=O)C2(CCOC2)C1 Fc1ccc(Br)cc1Sc1cccc(I)c1.C12CCCN1CCC2 C(CCCCCF)N(C1(C(=O)O)CCOC1)C C(=O)(C1CCc2cccc(=O)n21)N1CCC(C)(NC(C2CCCC2O)=O)CC1 C1(CNC(c2cc(C)n(C)n2)=O)CC(C)CCN1C(=O)C(C)Cc1ccnn1C c1(NC2C(NC(C(C)N3CCC3)=O)CS(=O)(=O)C2)ncc([N+](=O)[O-])cc1Br c1(OC)ncc(C(=O)NC2CCN(C(=O)CC3CC3)CC2C)cc1C(F)(F)F C1(Cn2cc(C(C)(C)SC)nn2)CCN(C(c2cccc(C)n2)=O)CC1(F)F C1(C(C)(C)O)(CNC(C23CC(CO)(C2)C3)=O)CN(C(=O)C(C)CF)C1 c1(NC(C2(C)CCN(C(CCc3cccc(C)n3)=O)C2)=O)cc(Cl)ccc1I n1(CC(=O)NC(CC(C)NC(c2cn(C(C)C)nc2)=O)C)cccc(N)c1=O C(CC(C)C)(C(=O)NCC(C(C)C)NC(c1cc(Cl)ccc1O)=O)OC C1(C(=O)NCCC(=O)Nc2c(F)cccc2Cl)C2Cc3ccc(Cl)cc3C12 CC1(C)CCCN(C(C2CC(=O)CO2)=O)C1CNC(c1cccn2ncnc12)=O C(C(CC1CC1)C(=O)NCCCC1CCC1)NC(C1N(C(C)(C)C)CC1)=O n1(CC#C)cnnc1C(=O)NCC1(CC(=O)NC2CNC(=O)C2)CC1 N1(C(C(CC)CC)=O)CCC(C(=O)NC2CC(C)(CO)C2)C(O)C1 N1(C(c2ccc(SCC)cc2F)=O)CC2COCC(C1)C2NC(=O)CCOC N1(C(C(C(C)C)N(C)C)=O)CCN(C)CC1C(=O)NCCCN(CCO)CCO C(CCCC(=O)N(C1CCCC12CC2)C1CC1)N(C(CC1ON=C(C)C1)=O)C C(CSC)(C(=O)NC(C)(CNC(c1cc(-c2cccs2)on1)=O)CO)OC C(=O)(C1=Cc2ccccc2C1C)N(C(CNC(CCCNC(C)=O)=O)C1CC1)C C1(C(N2CCC(N(C(=O)CNC=O)CC)C2)=O)CCC(F)(F)CC1(C)C C(=O)(C(CC)CCCC)NC1CC(Cn2cc(C(=C)C)nn2)C1(C)C C1(NC(C(C)(C)F)=O)COC2(CCN(C(c3cc(C#N)cs3)=O)C2)C1 C1(CC(=O)N(C2CCN(C(=O)C=Cc3ccc(C)o3)C2)CCC)CCCCC1O N#Cc1ccc(CNC(=O)C(c2ccco2)NC(=O)CCC2CC2)s1 C(=O)(CCC(C)S(C)(=O)=O)NC(c1ccccc1F)CNC(CCC)=O N1(C(Cc2cccc(N)c2N)=O)CCCC(C2CC2NC(C2CCC(=O)N2)=O)C1 N(C1CCc2ccccc21)(C(CCC=C)C)CCOC1CCOCC1 C#CCCCCCC(=O)NC(C)CN(C)C(C12CCC(CF)(C1)OC2)=O C12(CNC(CCCCSC)=O)CCCCC1N(C(=O)CCCNC(N)=O)CC2 C1(NC(Cn2ncc(C)cc2=O)=O)CCCC12CN(C(c1n[nH]c(C)c1O)=O)C2 C1(C)(NC(C(N2CCCC2=O)C)=O)CCCN(C(c2csc(C3CC3)n2)=O)C1 N1(C(COCCOC)=O)CCC(CCN(C(=O)CNc2cnc(Cl)cn2)C)CC1 C12(C(=O)NC(CN(C(=O)CC3(COC)CC3)CC)C)CC1COC2(C)C c1(C(N2CC(O)(C(C)NC(CS(CC)=O)=O)C2)=O)ccc(OC)c(N)n1 N1(C(C#CC(C)C)=O)CCS(=O)(=O)C(CCNC(=O)C2=CCC(C)CC2)C1 C1(NC(C(CCC)OCC)=O)CC2CCC1N2C(C1(C)CC1)=O c1(OCC)ccccc1OCC(N1CCCC(N(C(=O)Cc2ccon2)C)C1)=O C1(C(N2CC(NS(CC(=O)OCC)(=O)=O)(CF)C2)=O)CCCC12CCC2 C(C(=O)NCCC(Cl)Cl)(C(C)(C)C)NC(CC(C)c1ccco1)=O N1(C(C(C)c2ccco2)=O)CCC(O)(CCNC(=O)Cn2ccc(Br)n2)C1 c1(C(N2CCCC(O)(CNC(c3nccs3)=O)C2)=O)c(F)cc(Br)cc1F c1(CNC(COC(C)(C)CNC(c2cnns2)=O)=O)cccnc1Cl N1(C(COc2ccn(C)n2)=O)CC(CC(=O)NC2CCCCCC2F)CC1(C)C C(C(C)(C)C#CC(=O)NCC1(O)CCOCC1)NC(CC1ON=C(CC)C1)=O N1(C(c2ccn(CCOC)n2)=O)CCC12CN(C(=O)CCC1CCCC1)C2 c1(CC)nc(C)c(C(=O)N(C2CCCCC2N(C)C(C2CCC(C)(C)C2)=O)C)o1 Cc1c(C(=O)NC(C)(CNC(=O)C(C)Sc2ccccc2)CO)cccc1Cl c1(C(=O)NC2CN(C(c3cc(I)ccc3Br)=O)CC2F)ccnc(Cl)c1Cl C(=O)(C(C)C(F)(F)F)N1CC(OC2CCN(C(c3c(C)cc(COC)o3)=O)CC2)C1 Fc1cccc2nc(C(c3nnnn3C3CC3)NC3CC3)cn12 N1(C(c2cc(F)ccc2Cl)=O)CCC(N=c2ccc3nccn3[nH]2)C1 C1(CNC(C2(CCOC)CCCC2)=O)C2CCC(C2)N1C(c1cc(C)[nH]n1)=O C1(C#N)(C(N(CCCCNC(=O)CSC(C)(C)C)C)=O)CCCOC1 c1(SC)ccc(Cl)c(C(=O)N(C(C)CNC(=O)CNC(c2ccncc2)=O)C)c1 C1(CN(C(=O)C(C)(O)C2CCC2)C)CCCN1C(=O)CC1CCNC1=O C1(CNC(C(=O)NCC(n2cc([N+](=O)[O-])cn2)(C)C)=O)CCC(F)(F)C(=O)N1 C(=O)(C1=CCCC1(C)C)NC1CCCN(C(c2c(N)cn(C)n2)=O)CC1 c1(C(=O)NCCC2(CNC(C(C)(C)CO)=O)CC2)cc2ccnn2cn1 N1(CC(=O)NC2(C)CC(C(F)(F)F)C2)CC(C(F)(F)F)CCC1=O Cc1cc(CNC(c2cc(F)c[nH]2)=O)oc1C(=O)N(C)CC1CC1(F)F NC1CCc2cc(OCc3ccn(C4CC4)n3)ccc2C1 CCC(CC(C)C)C(=O)NC1COCC1NC(C1(N2CCOCC2)CC1)=O C1(C2CCN(C(C3CNC(=O)CC3(C)C)=O)C2)(NC(c2c(CC)nco2)=O)CC1 c1(CC)cccc(C)c1NC(=O)C(c1ccc(OC)c(F)c1)N1CC(C)CCC1C Cc1cc(C(N2CCCC2C=CC(N2CC(O)(C(F)(F)F)C2)=O)=O)cc(C)c1 C1(C)(C(=O)NC2CCN(C(c3cc(C(C)=O)on3)=O)C2(C)C)CCCCNC1=O C(=O)(CC(C)C(C)(C)C)N(CCCCCNC(c1ccn(C(C)C)n1)=O)C CC1(C)CCC(C(=O)Nc2cn[nH]c2)C(CNC(=O)CC(F)(F)F)C1 c1(N(C)Cc2n(CCC)ccn2)cc(NCc2cnn(C)c2Br)nc(C)n1 c1(C(N2CC(CCCNC(C3N(CC)CC3)=O)OCC2)=O)cc([N+](=O)[O-])cn1C C#CC1CN(C(c2ccc(OCCOC)cc2)C(=O)NCc2ccco2)CCO1 C(=O)(C1=CC2CCC(C1)C2)NC(CC(=O)NC(CC1CCC1)CO)C(F)F c1(C(=O)NCC2N(C(CC(COC)C)=O)CCC2)cc(F)ccc1O c1(C(=O)NCC2CCC(NC(c3ccc(Cl)nn3)=O)CC2)ccc2sncc2c1 Cc1ccc2c(c1)CN(C(=O)CC13CCC1CN(C(=O)C(O)CCN(C)C)C3)C2 c1(C(N(C)CC2(CNC(c3ccn(CC#N)n3)=O)CC2)=O)cc(O)nn1C c1(CC)cc(C)nc(NC(C)(C)CCNC(C2CCCN2C(C)=O)=O)n1 CC1C(C(=O)Nc2cccc(CN(C(C3(C)CCCN3C)=O)CCO)c2)CCN1C c1(C(N2CC(C(NOCC(=O)OC)=O)OCC2)=O)ccc(C)c(OC)c1 N1(CC2COCCC2(F)F)CCCC2(Cn3cc(CN4C(=O)OCC4)nn3)CCCC12 C1(CC)CC(O)CN1C(C1COCC1NC(=O)Cn1ccc(C)n1)=O c1(C(=O)NC2CC(F)(CNC(C(C(C)(C)C)OC)=O)C2)cncc2nc(O)[nH]c12 Cc1cc(C(=O)NC(C)CC(C)NC(=O)CCc2cnco2)cc(C)c1O Cn1ncc(C(=O)NC2C3CC4CN(C(C5CC(O)C5)=O)C2C4C3)c1S(C)(=O)=O N1(C(C2CCN(C(CC)=O)C2)=O)CC(NC(=O)C(CC)CC)CC1(C)C.C(CN)O C1(C)(CC)CC(NC(=O)C(C)(C)NC(c2cnc(C)o2)=O)C1 C1(NC(C=Cc2ccc(CC)o2)=O)CC(C2CCN(C(c3ccc(C)s3)=O)C2)C1 C=CC1(C(N2CCCC(NC(=O)Cc3nccs3)CC2)=O)CCOCC1 C12(C(=O)NCCN(C(CSCC(=O)OC)=O)C(C)C)CCC(C(F)(F)F)(CC1)C2 Cc1cc(=NCC(C(F)(F)F)n2cncn2)[nH]c(=NCC(C)Cn2ccnc2)[nH]1 c1(OC(C(CC=C)(F)F)=O)ccc2cc(OS(=O)(=O)CCSC)ccc2c1 c1(OC)cc(Br)cc(CN2CCNCC2C(=O)Nc2nc(C)cs2)c1O N1(C(CCCCCSC)=O)CCCN(C(=O)CCNC(=O)CC(C)C)CCC1 c1(NC(C)=O)ccc(C(N2CCCC(NC(c3ccc(C)nc3)=O)C2)=O)c(Cl)c1 c1(C(=O)NC(C(C)NC(CC(CCC)O)=O)(C)C)ccc([N+](=O)[O-])cc1Br CC1(CCS(=O)(=O)c2ccc(I)cc2)CC12NC(=O)N(C1CC1)C2=O N1(C(C(=O)NC(C)C)=O)CC(NC(=O)C(c2ccccc2Cl)N(C)C)C(C)(C)C1 N1(C(C(CC)F)=O)CCN(C(=O)Cc2ccc(F)cc2C)C(c2cn[nH]c2)C1 N1(S(CCCCC)(=O)=O)CCC2(CCC2)CC1C(=O)OC C1(O)(C(=O)NCCC(CCNC(C(CC=C)CC)=O)C)CN2CCC1CC2 Cc1ccc(C(N2CC(C)(C(=O)NCCc3ccncc3F)C2)=O)cc1C#N N1(C(C2OCC(C)C2)=O)CCn2ncc(CNC(C3CCSC(C)C3)=O)c2C1 C1(N(C(c2ccc(C)s2)=O)CC2CC2)CCN(Cc2nccn2C(C)(C)C)CC1 Cc1nc(CCC(N2CCCCC2CN(C(=O)C=CC2(C)COC2)C)=O)[nH]c1C c1(CC(N2CC(C)CC(NC(CN(C)CC)=O)C2)=O)coc2ccc(C)cc12 c1(N(c2c(C(C)=O)cccn2)Cc2ccncc2)ccc(C(=O)OC)c(F)c1 C(=O)(C(F)(F)C(O)CC)N(CCC(N1CCC(N2CC(O)C2)C1)=O)CC=C.C1(O)CC1 C=CCC(CNC(c1cnnc(C)c1C)=O)C(=O)NCC1(CCO)CC1 N=c1nc2c(C(=O)NCC=CCNC(c3cncc([N+](=O)[O-])c3)=O)cccn2[nH]1 c1(C(N2C3CCC2CC(NC(C24CC5CC2C4C5)=O)C3)=O)cccc2occc12 C1(C(=O)OC2CC(C)OC2=O)COC2COCC2O1 C1(CC(=O)NCCCNC(c2cc(C(F)(F)F)n[nH]2)=O)CCCOC1 c1(C(=O)OC)[nH]c2nccnc2c1NC(=O)NC(C)(C)Cc1ccc(C)cn1 CC(C)CC(C)C(=O)OCC1CCC(Nc2ccc(Br)c(F)n2)CC1 CC1C(C(N2CCN(C(c3n[nH]cc3C(C)(C)C)=O)CC2)=O)CCN1C Cc1cn2ccc(C(=O)NCC(C(C)C)NC(=O)CNC(=O)C(F)(F)F)cc2n1 n1(CC(=O)NC(C)CCCCNC(c2cnns2)=O)nnc2ccccc2c1=O c1(-n2ccc(C)n2)ccc(-c2nc(C(C)C)nn2C(C)C(C)C)cc1 Cc1nc(CC(N2CCC2CNC(=O)C(N2CCOC2=O)C)=O)n[nH]1 C1(CCC)(NC(=O)C(CC)N(C)C)CCCN(C(=O)CSCC(F)(F)F)C1 CN(NC(=O)OC(F)F)C(=O)c1coc(C(=O)N(C)C)n1 c1(SC)nc(O)c(C(=O)N(CCNC(c2csc(CO)n2)=O)C2CC2)cc1C#N CC(C)CC(C)CC(=O)NCc1ccc(C(N2CCCNC(=O)C2)=O)o1 C#CC1CN(C(C2CC2C2CCCC2)=O)CCN1C(c1cnn(C)c(=O)c1)=O c1(SCC#C)cccc(C(=O)NC(CNC(=O)C(C)(O)C2CCC2)C(C)(C)C)c1 c1(C(=O)OC)coc(C(=O)NCCCCCN(C(=O)C(C2CC2)SC)C)c1 N1(C(C2CCC(C)(CC)O2)=O)CCC2(CCC2)C(CNC(c2cc(C)c[nH]2)=O)C1 N1(C(C2OCCN(CC)C2)=O)CCN(C(c2c(C)cc(C)oc2=O)=O)CC(O)C1 c1(C(CC(=O)OC)NC(=O)C(C)(C)OC)ccc(OC(F)F)c(OC)c1 C1(CCCC)CN(C(=O)CC2CCCC(C)(C)O2)CCN1C(=O)CCSCC c1(N2C(C(C)C)CN(C(C3CCCC(F)C3)=O)CC2)nccc(S(C)(=O)=O)n1 C(=O)(CCC1=CCCCC1)N(C)CC1(O)CCN(C(CS(=O)(=O)NC)=O)C1 CCC(C)CCCC(=O)NC1CCCC(NC(c2ccn(C3CC3)c2C)=O)C1 c1(C(C(=O)NC(CC=C)CNC(C2(n3ccnn3)CC2)=O)O)ncccc1C n1(CCC)nc(C)cc1C(=O)NCC(C)(C)NC(=O)C(c1cncc(F)c1)C CC1CN(C(=O)C2=CC(C)(C)C2)CC(CCNC(c2cccc(C#N)c2)=O)O1 c1(C(N2CC(CC=C)(NC(=O)CC3(C)CC3)C2)=O)ccc(Cl)cc1Cl CC(C)C(C)(C)C(=O)N1CC2CC(C1)C2NC(c1ccncc1N)=O CCC(F)(F)CC(=O)NCC1CN(C(C2CC(C)OC2C)=O)CC1C CC(C(C)(C)CN(C)C)NC(=O)Nc1ccc(C(=O)NCc2ccco2)nc1 C1(C(=O)NC2CC(CCNC(=O)Cn3cccc3)C2)CC2(C1)OCCO2 Cc1c(C(=O)NC2(C)CC(NC(C3CCC=CCCC3)=O)C2)cccc1O c1(NC(CC2CCN(C(C3C(C)CC3)=O)C2)=O)ccc2ncccc2c1 c1(OCC(N2CC(CNC(C3CC(=C)C3)=O)C(O)C2)=O)cc(Br)ccc1F CC1=C(C)CC(C(=O)NCC(O)CC(=O)NCC2(CO)CCCO2)CC1 C1(CC=C)(NC(c2cc(C3CC3)oc2C2CC2)=O)CCN(C(C2CC2C)=O)CC1 c1(C(N2C(CNC(c3cccc(OC)c3)=O)CCCC2)=O)cc(F)c(C)c(F)c1 c1(CC)ccc(C(=O)NCC(C2CCC2)NC(c2ccnn2CCF)=O)s1 CCC(C)C(O)C(=O)NC1(C(=O)NCC(=O)N2CCCO2)CC(F)(F)C1 C1(NC(c2n[nH]c(C3CC3)c2Cl)=O)CCCN(C(c2cnccn2)=O)C1 N1(C(C(C)N(C)C(c2cccnn2)=O)=O)CC(O)(C(F)F)C1 C(CN=c1[nH]c(N(CC(C)CO)C)nc2c1CSC2)(C(F)(F)F)OC C1(C(N(CCNC(C2(C(CC)=O)CC2)=O)C)=O)CC=CCC1 CS(=O)(=O)C1CC(NC(C2CCC(NC(c3ccncc3O)=O)CC2)=O)C1 C1(NC(=O)CC2CCOCC2)CN(C(=O)CC2CCCC2)CCC12CCC2 c1(C(N2CC(CNC(C3CCCN(CC)C3)=O)C2)=O)ccc(C#CC2CC2)cc1 Cc1cc(C)n(C2CN(C(=O)CC3(NC(=O)CN4CC5CC5C4)CCC3)C2)n1 Cc1cc(C(N2CCN(C3CCN(C(C4CC4C)=O)C3)CC2)=O)oc1Br C1(C(N2CCC(C(F)F)(CNC(C3(Cl)CC3)=O)C2)=O)CCC(F)(F)CC1 c1(C(=O)NC2(C3N(C(C(CC)SC)=O)CCCC3)CC2)cc(N)ccc1C CN1CCOC(C(=O)NCC(CO)NC(=O)CCc2cncnc2)C1 Cc1cc(CO)oc1C(=O)NC1CC(CNC(c2cnccn2)=O)C1 N1(C(C2(C#C)CC2)=O)CCC2CN(C(c3ccc(F)c(SC)c3)=O)C2C1 c1(C(=O)NCC2C(NC(C(CC)NC(N)=O)=O)C2)oc(C)nc1C C(=O)(CC1=CCOCC1)N1CCC(C(=O)NCCOCCC(C)C)C1C C(=O)(C(Cc1cnc[nH]1)NC(=O)CCc1nc(=N)[nH][nH]1)N(C(C)CO)C C1(NC(c2nccc(C)c2N)=O)CN(C(=O)CCC2(C)CC2)CC12CCOCC2 N1(C(CNC(=O)NCC(=O)NCCn2cncn2)=O)CCC2CC12N(C)C c1(NC(C(CCC)OC)=O)ccc(NC(c2ccn(C(C)(C)C)c2)=O)cc1C N1(C(=O)CC2CSC2)CCN(C(c2ccc3c[nH]nc3n2)=O)C2CCCCC2C1 C=C1CCCN(C(CC2CCC3CC23)C(=O)NCCSC)CC1 n1(CC(=O)NC(CCCCNC(COC(C)=O)=O)C)nc(C(F)F)c2c1CCC2 C(=O)(CC(C(C)CC)NC(C1CSC1)=O)NCc1c(C#C)cccc1 C(=O)(C1CCCc2nncn21)N1C(C)(C)C(NC(=O)C(F)=C2CCCC2)CC1 Cc1cccc(C(=O)NCC2CCN(C(c3cc(C)n(C(C)C)n3)=O)C2)c1 C(=O)(C(F)C(C)CNC(C1CC2(CC(=O)C2)C1)=O)NC(CCC)CO Cc1cncc(C)c1C(=O)NC1CCC1NC(=O)Cc1cccc(Cl)c1Cl CCS(=O)(=O)c1ccccc1CC(=O)NC1CCC(CNC(=O)CC#N)C1 CC1(C)CCC(CNC(C2CC=CCC2NC(C2(CO)CC(C)(C)C2)=O)=O)O1 C1(C(=O)NCC2CCN(C(C)C)C2)C(C2CC2)CCN1C(=O)C1=CCCOC1 CCCC(CC)CCC(=O)N1CCC(N=[N+]=[N-])(C(=O)N(C)Cc2ccccc2)C1 c1(CC)ccccc1C1CC1NC(=O)CC(C)(C)C N1(C(c2cc(C)c(Br)s2)=O)CC(F)(F)CC1Cn1cc(-c2ccc(F)cc2C)nn1 N1(Cc2c(N(CC(=CC(=O)NC)C)C)nccc2)CC2CC1CC2N(C)C Cc1cc(Cl)cc2[nH]c(C(N3CCC(N(C(=O)C4=CCCS4)C)C3)=O)cc12 N1(C(c2c(C)nc(C(C)OC)s2)=O)C2CCC1CN(C(c1nc(O)c(C)s1)=O)C2 N1(C(c2c(C)ccc(CC)c2)=O)CC(C2CCCN(C(c3[nH]cnc3C)=O)C2)C1 C1(NC(c2ccc(OC)nn2)=O)CCN(C(C2NC(=O)OC2(C)C)=O)CC1F c1(C(=O)NCCC2(CNC(C3(Cl)C(C)(C)C3)=O)CC2)ncn2c1CCC2 c1(C(C(=O)NCC(C)C)N(C)Cc2csc(C3CC3)n2)cc2c(s1)CCOC2 C1(NC(c2n(CC(=C)C)nnn2)c2cncn2C2CC2)CC2CC3C(C2)C13 C1(NC(Cc2n[nH]c(=NC)s2)=O)CC2(CCC(NC(=O)CN3CCC3C)CC2)C1 CC1(C)CCCCC1CC(=O)NC1CC2C1CCN2C(=O)C=CC1CCC1 C1(CC=C(C)C)CCCN(C(=O)CCC2CCCC2=O)C1 C(=O)(CC(C(C)C)C(C)C)NC1CCN(C(c2n(CC)ccc2)=O)CCC1CO c1(OC)ccc([N+](=O)[O-])c(NC2CN(C(=O)OC(C)(C)C)CC2CC2CC2)c1 C1(NC(c2ccccc2)CC)CCN(c2ccncn2)C1 Cn1cnc(C(N2CCCC(C)(NC(=O)CCC3CCCO3)C2)=O)cc1=O C1(CNC(Cc2c(C)ocn2)=O)CCCC2CN(C(=O)CCCS(C)(=O)=O)CC12 C(=O)(N=c1cc(C2CC2)n(C)[nH]1)C1C=CCN(C(CC(CC)O)=O)C1 c1(NC(=O)NC(c2cccc(OC)c2F)C)nccn2c(C)nnc12 Cc1cc(F)c2cc(C(=O)Nc3cc(C4CC4)cc(F)c3)[nH]c2c1 C1(CCNC(C(C)NC(c2ccnnc2)=O)=O)CCCC2CC12 C(CCCCCC(=O)Nc1ccc2c(c1)COC2)NC(C(C)(C1CC1)OC)=O CCCC(C(=O)N1CCCC1CCN(C)C)NC(=O)C=Cc1ccco1 N1(C(CN(CCOC)C)=O)CC2CCC(NC(c3cc4ncccc4[nH]3)=O)(C2)C1 c1(OCC)cccc2[nH]c(C(N3CCC(C)C(NC(=O)C(O)CC)C3)=O)cc12 N1(CCCC(=O)NCC(CNC(C2(C=C)CCC2)=O)F)Cc2ccccc2C1=O C(=O)(CS(=O)C(F)(F)F)NCC(C)(F)CNC(=O)C1=NOCC1 N1(C(c2c(OC)ccs2)=O)CC2(COC(CNC(=O)CN3CCCS3(=O)=O)C2)C1 c1(OC)ncnc(NC(c2cc(-c3cncc(SC)c3)cnc2Cl)=O)c1OC c1(-c2c(C(N3C(C)CCC3C)=O)cc(Cl)cn2)nc2c(s1)CCC2 N1(C(CCCn2cc(CSC)nn2)=O)CC(C)C(O)C1 NS(=O)(=O)CCCCCC(=O)NC1CN(C(=O)CCCc2cnn[nH]2)C1 c1(C(=O)NCC2C(NC(C(CC)O)=O)CCCC2)csc2ncnc(O)c12 FC1(F)CC1C1CCN(c2ncnc(-n3nc(C)cc3-c3ccccc3)n2)CC1 C(=O)(C(F)(CNC(=O)C(C)(C)C(F)(F)F)C(C)C)N1CC(CC)NC(=O)C1 C(=O)(C(C)(CC)C(F)F)N(C1CCC(CNC(CCCC(=O)OCC)=O)CC1)C c1(COc2ccccc2)ccc(C2CCC(NC(c3n(CC)nnn3)C)C2)cc1 N1(C(c2ccc(C(=O)OC)s2)=O)CCC(NC(c2cnn(C)c2C)=O)C1C c1(CC)ccsc1C(=O)NC1CC1NC(=O)CC(C)C N1(C(c2nc(CCC)sc2)=O)CCCC(CCNC(c2cncc(Cl)n2)=O)C1 CC(CC(C)(C)C)C(=O)NC1CC12CCN(C(c1ccc(Cl)cn1)=O)C2 C(CCCCCCCC1CC1)(c1n(C(CC)(C)C)nnn1)NCCCC(C)(F)F CCCCC(C)C(=O)N1CCOC(CN(C)C(c2sc(C)nc2C(C)(C)C)=O)C1 c1(OC)ccc2ccc(=NCCOCCc3ccccc3)[nH]c2c1 N1(C(c2n(C(C)C)ccc2)=O)CC(NC(=O)Cn2cncn2)CC(O)C1 N1(C(C2(SC)CC2)=O)CC2(CCC(NC(=O)C(N)=O)CC2)C1 CCCCCC(=O)NCC1CCCN1C(=O)C(C)C(=O)OC C1(O)(CNC(C2C3CCC23)=O)CCCN(C(c2ccccn2)=O)C1 c1(OC)ncccc1C(N1CCCC(C(C)C(=O)NOCCCC2CC2)C1)=O N1(C(C2(NC(C(CC)NC(C)=O)=O)CCC2)=O)CC2CC(C1)C2(C)C C=CCC(C(=O)NC1C=CCCC1C(=O)NCC=CCl)NC(C)=O CC1CCCN(CC(=O)NCc2cn(C)nc2-c2ccc(Cl)cc2)CC1 C(=O)(C(C(C)C)C(C)C)NCC(CNC(c1nc(C(=O)OC)sc1)=O)OC Cc1cnccc1C(N1CC2C(CNC(c3cnc[nH]3)=O)C2C1)=O C1(C(N(CCC)CCNC(=O)CC2CCC3(CC3)CO2)=O)CCC2CC1C2(C)C N1(C(C(C(C)C)SC)=O)CC2(CCCC(CNC(=O)C(C)Cc3ccco3)O2)C1 c1(C(N2CCCC(NC(CC(CC)SC)=O)C2)=O)cc(OCCOC)cc(F)c1 c1(OC)ccc(C(N2CCCN(C(C3CCCS3)=O)CC2)=O)cc1[N+](=O)[O-] C1(NC(C=CC(CC)=CC)=O)(COC)CCN(C(C2CCC(=O)N2C)=O)C1 N1(C(CC)=O)CCCC(C(=O)NCC2C3CN(C(c4c(C)ncn4O)=O)CC23)C1 CCC(CC(=O)N(C)CCN(C)C(c1cnn(CC(F)(F)F)n1)=O)CC(C)C N1(C(C(CC#C)O)=O)CC2CC(NC(c3cc(C(N)=O)ccn3)=O)C1C2 c1(OCC(=O)NC(CNC(C2CCC(CC)O2)=O)CC)cccc(C)c1C N1(C(c2noc(CC)c2C)=O)CCN(C(=O)C(c2cccc(F)c2)O)CC1C Cc1cc(F)ccc1C(N1CC(N(C)C(C2CC2C)=O)C(C)(C)C1)=O C(=O)(CCCCCCCC1CC1)NC(C(C)C)(C)CNC(=O)CSCCC#N N1(C(C(C)=CC2CC2)=O)CCCC2(NC(=O)COc3cc(C)ccc3F)CC2C1 CCCCCC(CCCCC)C(=O)NC1CCN(C(=O)CC2=CCN(C)CC2)C1 C1(NC(c2ccc(C#C)o2)=O)CC2(C1)CC(C(=O)NCC1(O)CCC1)C2 C(N=c1cc(C)[nH]c(=NCC2(C)CCOC2)[nH]1)c1c(CC)noc1CC c1(C(C)C)nnc(CCC(=O)NC2(C3CCCN3C(c3cnn[nH]3)=O)CC2)o1 N1(C(C2(C(=O)OC)CC2)=O)C2CCC1CC(NC(c1cc(Cl)sc1Cl)=O)C2 CC1NC(C(=O)NCCCCc2nn[nH]n2)=NN(c2ccccc2)C1=O c1(C(=O)NCC2CN(C(c3c(C)cc(CC)o3)=O)CC2C)cc(C)c(F)c(C)c1 c1(OCCCC(N2CCC(NC(c3c(CCC)nco3)=O)C2)=O)cccc(C)c1 N1(C(C2(F)CN(C(=O)C(O)C3CC3)C2)=O)CCCN(CCO)CC1 N1(CCN(C(=O)CC2CC2)C2CC2)CCCN(C(=O)Cc2cncnc2O)CC1 C1(NC(C23CC(NC(c4cnn(CC)c4C)=O)(C2)C3)=O)CCCC(O)CC1 c1(C(N2CCC(F)(CNC(=O)CC3CNC(=O)C3)C2)=O)cc(F)cc2nc[nH]c12 Cc1nc(C=CC(=O)NCC(CC(C)C)NC(c2ncn(C)c2C)=O)[nH]c1C N1(CCC(=O)NC2CCC2C(=O)NCC(C)NC(=O)OC(C)(C)C)CCOCC1 N1(C(c2ccc(Br)cc2OC(F)(F)F)=O)CC2(CCCN2C(=O)C#CC2CC2)C1 C1(Nc2c(C)c(NC3CCC(C)(C)C3)ncn2)CCN(CP(C)(C)=O)CC1 N1(C(c2cccc(SCCN(CC)CC)c2)=O)CCC(C#N)(C(C)C)CC1 C1(NC(c2nc(Cl)sc2)c2nnnn2Cc2cccs2)CC2CC3C(C2)C13 Cc1ccc(Cl)cc1C(=O)N(C1CN(C(C2(c3ccc(Cl)cc3)CCC2)=O)C1)C CN1CCC(C(=O)NCCc2ocnc2CNC(C2(C(N)=O)CCC2)=O)C1 C1(NC(C2C(C(=O)NCC#C)C2)=O)CCOCC1NC(=O)CC1(C)CCCCC1 Cc1ccc2oc(C(N3CC4(CCN(C(=O)CN5CCCCC5)C4)C3)=O)cc2n1 C(=O)(C(F)(F)C(C)O)NCCc1c(C(NOCC(C)C)=O)c[nH]n1 C1(C(N(CC(O)CNC(C2(c3ccccc3)CCC2)=O)C)=O)CC2C=CC1CC2 c1(C(N2CCCC(NC(COc3cc(C)on3)=O)CC2)=O)c(C)cc(C)nc1S N1(C(c2ccn(CC)c2C)=O)CC2(CC(NC(C3CCS(=O)CC3)=O)CO2)C1 CCN=C(NCC(c1ccco1)N1CCCC1)N1CCC2C(C1)C2(F)F C(=O)(CC(C)C(C)(C)NC(=O)C(O)Cc1cn(Cc2ccccc2)nn1)OCC Cc1cccc(C)c1C1(C(N2CC=CC(NC(=O)CCCCCO)C2)=O)CC1 Cc1cc2sc(C(=O)NCC(C)CN(C(=O)Cc3c(C)cccc3Cl)C)cc2s1 N1(C(c2ccc(OC)cn2)=O)CCN(C(c2cncc(N)n2)=O)C2CCC12 N1(C(C(F)=CC)=O)CC(C)(C)CC1CNC(C1(c2cccc(Cl)c2F)CC1)=O C1(CNC(C(CC)OC)=O)CCN(C(=O)C(c2c(C)nn(C)c2C)=O)C12CCC2 C(=O)(C1=NOC(CC2(O)COC2)C1)NC1CCC(NC(C2(C=C)CCC2)=O)C1 Cc1ccc(Br)c(C(N2CCC(C(N3CCC(CC#N)CC3)=O)C(O)C2)=O)c1F c1(-c2nc(COC)nn2-c2ccccc2)cc2scc(Br)c2[nH]1 N1(C(CCCCCCCSC)=O)CC2CCC(C2)c2ccccc21 C1(C)(CNC(c2c(CC)csc2)=O)CN(C(c2cc(OC)nn2C)=O)C(C)(C)C1 C1(CC)COC(C)(C)CN1S(=O)(=O)Cc1cccc(F)c1 C1(COC)(NC(c2cnncc2C)=O)CCN(C(=O)CNC=O)C1 C(=O)(CCCCC(F)F)N1CC2(CC(NC(c3cn(CCOC)nc3C)=O)C2)C1 c1(N2C(C(=O)NC(C(=O)OC)C(C)O)CCC2)nc(C(F)(F)F)c2sccc2n1 C(=O)(CC(C)CNC(=O)CN(C)C(=O)C1CC1)NC1(CC)CCC1 Cc1ncc2n1CCC(C(=O)NCC1CN(C(c3n[nH]cc3Cl)=O)CC1O)C2 C12(NC(CCc3c(C)ncs3)=O)CCOC(CNC(C3CCCSC3)=O)(C1)C2 Cc1ncncc1C(N1CC(F)CC1CC(=O)N(C)CC1(CO)CC1)=O N1(C(c2c(CCC)[nH]cc2)=O)CCCC(NC(c2cn(C)cn2)=O)C1 C(=O)(C(C(C)C)NC(C1CC(OC)(OC)C1)=O)NC1C(C(=O)OC)CC1 N1(C(c2c(C)snn2)=O)CC2=C(C1)CN(C(C1CCN(CC(F)(F)F)CC1)=O)C2 CC(C)(C)C(CC(=O)N1CCCC2(CNC(c3csnn3)=O)CCCC12)C(F)F c1(C(C(=O)OC)NC(C2C(C(CC)=O)CCCC2)=O)cc(F)c(F)c(F)c1 c1(OC)ccc2ccccc2c1CCNC(c1cc(CN(C)C)on1)=O N1(C(c2cc(CCC)[nH]n2)=O)CCCC(NC(C2CC23CC3(F)F)=O)C1 C1(NC(C(CCC)C)=O)CN(C(c2cnncc2O)=O)CCC12CCOCC2 Cc1cc(CC(=O)NC2CC(CNC(C3CCSCC3)=O)C2)n[nH]1 CC1(C)C2CCC1(C(N1CCC(C)(NC(c3ccn(CC(F)F)n3)=O)C1)=O)CC2 C1(N(C(C2(N3CCCC3C(=O)OC)CC2)=O)CCO)CCCCCC1 c1(C(=O)NC(C2CCN(C(CC(C)O)=O)CC2)C)ccn(CC(F)(F)F)c(=O)c1 c1(C(N2C(CNC(C3CC3(F)F)=O)CC(O)C2)=O)ccnc2cc(F)cnc12 c1(CNC(c2ccc(Cl)c(Cl)c2)c2cn(C)nc2C2CCC2)cc(Cl)cc(Cl)c1 c1(C(=O)NC2CCN(C(CCC(=C)C)=O)CC2CC)c(O)nnc2c1CCCC2 c1(CC(N2CC(CN(C(C=C)=O)C)C2)=O)nc(-c2ccccc2)oc1C C1(F)(C(=O)NC2CC(CCNC(C=CCCC=C(C)C)=O)C2)CC2(CCC2)C1 C1(C(N2CCC(C)(COC)C2)=O)CN(C(c2ccc(C)nn2)=O)CC1C1CC1 N(C(=NCCCCl)NCCc1ccccc1)C1CCCC(CC)C1 Cc1nc2c(C(N3CCOCC3CNC(=O)C(F)(F)CC(C)C)=O)cccc2o1 C(=O)(C(C)CCC(C)(C)C)N1CC(C(N2CCCC23CCC3)=O)(COC)C1 c1(C(N2C(CN(C)C(c3coc(Cl)c3)=O)CCC2)=O)nn(C)cc1Cl N1(C(C)=O)CCC(c2ccccc2)(C(=O)NC2CCSC(C)C2)CC1 C1(CC(=O)NC(C2CCOCC2)C#C)CC(NC(=O)C=CCCC)C1(C)C N1(C(c2c(CC)scc2)=O)CC2CCC1C2NC(=O)C(C)SC(F)(F)F C(C(CC(C)C)C(=O)N1CC(F)(C(=O)NCC2(CO)CCCCC2)C1)OC c1(C(=O)NC2C3CC2N(C(C2C4COCC24)=O)C3)cccc(S(=O)(=O)C(F)F)c1 c1(C(=O)NC(CNC(C2(C(=O)OCC)CC2)=O)C2CC2)ccc(=O)n(C)n1 C1(O)(CNC(C=Cc2ccc(C(N(C)C)=O)cc2)=O)CCC(F)(F)CC1 C1(CC(=O)NC)CCN(C(=O)NCC(O)CN2CCOCC2)C1 N1(C(c2cnc(CCC)s2)=O)CCN(C(C2C=C2C)=O)C2(CCC2)C1 N1(C(c2c(SC)snn2)=O)CCCC(O)(CNC(=O)C(F)C(C)C)C1 c1(C(C(=O)NCCSC)N(C)Cc2nccc(Cl)c2F)cc2cc(Br)ccc2s1 N1(C(CCCC#C)=O)CC(CC(=O)N(C2CCN(C)C2)C)CC1(C)C c1(-c2cc(C(N(C(CNC(C3C(C)C3)=O)C)C)=O)no2)ccccc1Br N1(C(CC(C)(C)C)=O)CC2CCN(C(c3cc(Cl)c[nH]3)=O)C2C1 C1(CC)CN(C(=O)C(=Cc2c[nH]cn2)F)CCN1C(=O)C1=CCN(C)C1 c1(CC)cc(C(N2CCC23CN(C(c2ccc(F)cc2Cl)=O)C3)=O)cc(F)c1 C#CCC(C)(CC)C(=O)N1CC(O)(C(C)(C)CNC(=O)Cc2cccc(C)c2)C1 N1(C(c2ccc(CC)[nH]2)=O)CC2(C=C(C(=O)N3CCC4CC4C3)CO2)C1 N1(C(C(CCN(C)C)O)=O)CCC2CN(C(c3nocc3Cl)=O)CCC12 C1(C(C(=O)O)F)CCCN(C(c2cccc(C(F)F)c2)=O)C1 CC(C)C(CCNC(=O)Cc1csc(CCC(F)(F)F)n1)NC(=O)CC(C)(C)C C1(C(=O)NC(c2c(C)cccc2)C)CN(C(C2CCCC2F)=O)C(C)(C)C1 N1(C(CCCCC)=O)CCN(C(C2CC2c2ccncc2)=O)C(CCC)C1 N1(CC(=O)NCCC)CCC(CC(=O)NCC(c2cnn(C)c2)(C)O)C1 CCCS(=O)(=O)C(C)C(=O)N1CCN(C(=O)C=C(C)C)CC1CC N1(C(c2c(C)cccc2C)=O)CC(CNC(=O)CC(C)C2CC2)C2(CCC2)C1 N1(C(CC)=O)CCc2cc(C(N3CCC3CNC(=O)CC(C)SC)=O)ccc21 C(=O)(C1CCCc2ncccc21)N1C(CNC(C(C)CCO)=O)CC(F)(F)C1 Cc1[nH]nc2c1CCC(C(=O)NCC=C1CCN(C(=O)C(C)(C)C3CC3)CC1)C2 N1(C(C2(C)CCCO2)=O)CCC2(CCN(C(C3CCCC(=O)N3)=O)C2)C1 C1(N(C(C2CC(Cl)(Cl)C2)=O)CC)CCN(C(=O)CC2CCN(C)C2)CC1 CCCS(=O)(=O)CC(=O)NCC1CN(C)CCN1C(=O)CCCS(N)(=O)=O n1(CC(=O)NC(CC)CNC(C2COC(=O)N2)=O)cc(S(N)(=O)=O)cn1 C1(NC(c2[nH]cc(CC)c2)=O)CCC(C)(CNC(=O)C=Cc2sccc2C)CC1 c1(NC(=O)OCC)ccc(C(=O)NC(CNC(=O)CSCC)CC(C)C)c(F)c1 c1(N(C)Cc2csc(C3CC3)n2)nc(N2CC=CC2)c2c(n1)COC2 N1(C(Cc2ccc(C)s2)=O)CC2CC2(NC(c2cnnn2C)=O)C1 c1(C(N(CCNC(C2CCCOC2C)=O)CC)=O)nccc2ncccc12 C(=O)(CC(C(F)(F)F)OC)NCC1CC(NC(C(C=C)OC)=O)CC1O c1(C(N2CC(CNC(CSCC#C)=O)C(O)C2)=O)ccc(N)c(Cl)c1 C1(CC(=O)NC(C2CCCCC2)C)CCCN1C(c1cc(C(F)(F)F)c[nH]1)=O N1(c2nc(OCC)c(C)cn2)CCC2(CCCN(C(c3cnns3)=O)C2)C1 C12CCC(C#N)(CC1)CC2.C(C)(C)(C(=O)OCC(=O)OC(C)(C)C)NC(C)=O CC(C)CCCC(C)C(=O)NCC1(CC(=O)N(C)CC2CC2C)CC1 c1(C(=O)NC2CCCN(c3nc(CC)nc(C)c3)C2C)sc2cncn2c1C C1(CC)CCN(C(=O)CC2CCCNC2=O)C(C(=O)NCc2ccc(OC)nc2)C1 C1(=CC(=O)NCC(C)(CO)NC(c2cncnc2)=O)CN2CCC1CC2 C1(CNC(CCN(CCC)C)=O)CC(C(C)C)CCN1C(=O)C(CC)NC(C)=O O=S(CCNc1nccc(=NCC2OCCO2)[nH]1)CC(F)(F)F c1(COC)nc(CNC(=O)CC2CCCC2O)cs1 CC1(C)CCCOC1C(N1CCCC(CCNC(C2CCC=CCCC2)=O)C1)=O c1(C(N2CCCC(CNC(c3c(C)ocn3)=O)(CO)C2)=O)cc(C#N)ccc1O c1(C(=O)NCC2C(NS(CC(=O)N(C)C)(=O)=O)CCC2)cc2c(F)cccc2[nH]1 C1(C(N2CCC(CC(=O)N(C)CC3CCOC3)CC2)=O)CCC(C2CC2)C1 C12(Sc3cccc(NC(=O)C(=O)NC4CCC(=O)NC4)c3)CCC(CC1)OC2 Cc1coc(C(=O)NCC2CCCN2C(=O)CCc2cccc(N(C)C)c2)c1C N1(C(C(CC)C)=O)CCCC(CCCCNC(=O)Cc2ccc(C(C)=O)cc2)C1 C(=O)(C(O)C(C)OC)NCCCCC1CN(C(C23CC(C(=O)OC)(C2)C3)=O)C1 Cc1cnc(NC2CCC(NC(=O)CC3CCCC3(F)F)CC2)nc1C c1(C(N2CC(O)(C(C(=O)NC(CCC)CC)F)C2)=O)cncc2[nH]ccc12 C(=O)(CC1CC(=O)c2ccccc21)N(C)CC1CCCN(C(C=CCC)=O)C1 c1(N(C2(C#N)CCNC2)C(C=CC(C)C)=O)ncnc2cccc(F)c12 c1(C(=O)NC(C2CCCN(C(=O)CNC(=O)C(C)(C)C)C2)C)cccc(Cl)c1Cl n1(C(C)C)ccnc1C(=O)NC1CCC(NC(C2CC(C(F)F)C2)=O)C1 N1(C(C2CCCN(C(C3CC(O)(CC#C)C3)=O)C2)=O)CCOC(C)(C)C1C N1(C(c2cc(C(C)=O)[nH]n2)=O)CC(O)CCC1C(=O)NCC1(C(=O)N(C)OC)CC1 C1(CNC(C2N(CC)CCC2)=O)CCC(C)(C)CN1C(c1cc(O)cc(O)n1)=O C(=O)(CCCCc1ccccc1)OCCC(=O)NCC(=C)C(=O)OC CCCCN=C(NCC1CC(F)C1)N1CCC2(CC(C(F)F)=NO2)C1 CC(F)(F)CCCCN1CC(C)(CS(C)(=O)=O)C1 N1(C(c2c(C)coc2)=O)CC(NC(C2CC23CC3)=O)C(n2ccnn2)C1 c1(SC(C)C(=O)NCC2(F)CC(NC(=O)C=C3CCN(C)C3)C2)ccccc1 c1(C(=O)NCC2C(CNC(C3(C(=O)NC)CC3)=O)C2)ccc(O)c([N+](=O)[O-])c1 Nc1nc(Br)ccc1C(=O)NCC1CCN(C(=O)CN2CC=CC2)CC1O Cn1ccnc1C(=O)NCc1n[nH]cc1C(=O)NCC1CC(CO)CO1 N1(C(COC2(C#C)COC2)=O)CC2CCC2(CC(N2CC(C(=O)N(C)C)C2)=O)C1 N1(C(C2(CC=C)CCC2)=O)CC(CNC(c2cc(CC)no2)=O)C(C)C1 c1(C(=O)NC2C(CNC(C(C)(C)c3cnsc3)=O)C2)cc(Cl)c(F)cc1Cl c1(OC)ccc(S(=O)(=O)N(C)C)c(NC(C2CC(=O)C2C(C)(C)C)=O)c1 N1(C(C=CC)=O)CC2(CCCCN(C(C3CCOC(C)(C)C3)=O)C2)C1 N1(C(C(C2CCN(C(C3CCCN(C)C3)=O)CC2)C)=O)CCC2COCC2C1 N1(C(C2N(C(CNC(CC(C)C)=O)=O)CC(C)C2)=O)CCC(O)C(O)C1 N1(C(C2N(C(C)=O)CCCC2)=O)CCCC2(NC(C3CCCC(C)O3)=O)CC2C1 c1(N2CCN(C(c3ccc(C)cc3O)=O)C3C2C3)ncc2[nH]ccc2n1 CCC(CC)(C(=O)NC1CN(C(=O)CC(C)(C)C)CC1c1ccccc1F)OC C(=O)(C1CC(=O)Nc2ncn(C)c21)NCCN(C(=O)CCC1CCCN1C)C CN1CC(C(=O)NCCOCCN(C)C(c2cnc(Cl)cn2)=O)C(C(F)(F)F)C1 S(=O)(=O)(c1cc2sc(=NC(C)CC(C)C(F)F)[nH]c2cc1Cl)N1CCC(CC)C1 c1(C(=O)NC2C(C)N(C(C3CCC3(F)F)=O)CC2)cc2c(s1)CCOC2 c1(CN2CCC(CNC(c3ncoc3C3CCCCC3)=O)C2)cncc(F)c1 C1(NC(C(CCC)NC(C)=O)=O)CCN(C(=O)CCN2CCCS2(=O)=O)C1(C)C Cc1nc2cccc(C(=O)NC(C)CC(C)NC(=O)CN3CC(C)(C)C3)n2n1 C1(C(=O)NCC(C)OC(F)F)CCC(C)N(C(=O)C(C)c2ccco2)C1 n1(CC)cc(C(C)NC(=O)C(c2cccs2)NC(C2CCC(=O)O2)=O)cn1 Cc1cc(CCNC(=O)CC=CCNC(=O)C(C)CN2CCCC2)nn1C c1(C(=O)NCCC2CN(C(C3CCC(CC)O3)=O)C2)ccc(C)c2ccccc12 N1(C(C(CCC)(C)O)=O)CCCC2(NC(C3CCc4ccccc4C3)=O)CC2C1 c1(OC)ccnc(C(N2CCC(NC(c3cc(Cl)c(Cl)cn3)=O)CC2)=O)c1OC Cc1cc(C=CC(=O)NC2CNCC(C)C2)c[nH]c1=N CCCC(C)(CC)C(=O)NC1COCCN(C(C2CCCC2O)=O)C1 c1(N2CCC(CCC)C2)cc(C(=O)OC)nc(C)c1 CC1(C)C2CCC1(CS(N1CC3C(C1)N3c1cc(C3CC3)ncn1)(=O)=O)C(=O)C2 c1(C(N(C(CCNC(C2(CCOC)CCC2)=O)C)C)=O)csc(C(F)F)n1 N1(N(C2C(C)OCC2)c2ccncc2)CCc2nnc(-c3ccncc3)cc2C1 C1(CCCNC(N(CCC)C)=O)CNCCO1 N1(C(CC2(CSC)CC2)=O)CC(C)CCC1CNC(=O)Cc1ccc(C)c(F)c1 C(=O)(C(C)(C)C(N)=O)NCC(CC)NC(=O)C(CC(C)C)N(C)C Cc1ncc(C(N2CC3C(C(F)(F)F)C3C2)C(=O)NCCC#N)cn1 Cn1ncc2cc(C(=O)NCC(CNC(=O)COCC3CC3)C(F)(F)F)sc12 c1(C(=O)NC2CC(C(=O)NCC3CCC(C)C3)CC2O)cnn(C)c1C#N C1(C(=O)NCC2(C)CCN(C(C3C(CC)C3)=O)C2)CCCC12CCOCC2 C1(NC(C(C=CCCC)O)=O)C2CC3C1C3C2C(=O)NC1CC(C(=O)NC)C1 C1(C(=O)NC(CC(C)NC(C2CCCOCC2)=O)C)CC2CCC1CC2 c1(C(C)NC(N2CC(c3ccc(C)cc3)(O)C2)=O)ccc(F)c(F)c1 C(=O)(C(CC(C)C)C(C)C)N1CC(CC=C)(C(N2CCC(C3CC3)C2)=O)C1 N1(C(C(c2cncnc2)C)=O)CC2CCC1C(CNC(c1cnc(N)cn1)=O)C2 C1(NC(C2C3CCCCC23)=O)CCCN(C(C2CC23CCCCC3)=O)CC1 N1(CCCc2c(OC(C)C(=O)O)cccc2)CC2CCCC(C(=O)O)(C1)C2(F)F c1(NC(C(CCCC)C)=O)cc(S(C)(=O)=O)ccc1NC(c1ccc(C)o1)=O N1(C(CC2CC(COC)C2)=O)CCC(C)(CC(=O)NC2CCSC2)C1 N1(C(C(CN(C)C)(F)F)=O)CCC2(CCCN2C(=O)CC2CCNC(=O)C2)C1 C(C(CO)(CO)NC(=O)CN1CCCC1C)N(C(c1cn(CC=C)nc1)=O)C Cc1nc(C(N2CCSCC2CCNC(C2OCCC2C(F)(F)F)=O)=O)nn1C c1(CCC(=O)NC2CN(C(C=CCC)=O)CC(O)C2)c[nH]c2cc(C)ccc12 N1(CC(C2CCCC2)OC)CCC(C(=O)NC2CCCCC2)C1 C1(O)(CNC(C2(C#N)CC2)=O)CN(C(=O)Cc2nc(C3CC3)cs2)C1 CC1CC2CN(C(C3CCCCN3C(c3cnn(C)c3)=O)=O)CC2N1S(C)(=O)=O c1(CCNC(C2CCCN2C(N2CCC(O)(CF)C2)=O)=O)ccccc1N.C1CC1 N1(C(C2C(C=C)OCCC2)=O)CC(CNC(=O)CCOCC2CC2)CC(C)(C)C1 N1(C(c2c(C)c(C#N)[nH]c2)=O)CC2(CCCC2)C1C(=O)NCc1cnns1 CC1CCCN1CC(=O)NCC1CN(C(C2CCN2C(=O)OC(C)(C)C)=O)C1 CN1CCC(C(=O)NCC(F)(F)CC2CC2)(NC(c2ccccc2F)=O)C1 n1(CC#C)c(CNC2CCCC(P(C)(C)=O)C2)cc2ccccc12 N1(C(C(C)C#N)=O)CCN(CCNC(c2ccnn2CC2CCC2)=O)CC1 c1(C(=O)NCC(CC)NC(C(CC)C)=O)cc2cc(OC)ccc2n1C N1(C(CSC)=O)CCCC1C1(N(C(=O)C(O)Cc2ccccc2)c2nncs2)CC1 N1(C(CC2CC(NC)C2)=O)CCCCC(C(=O)NCC(N2CC=CC2)=O)C1 CC1(C#CC(=O)NC2C3CCC(C3)C2C(=O)NC(CO)CCF)COC1 C1(CNC(c2cn(CCO)nn2)=O)CCC2CN(C(=O)C=Cc3cc[nH]n3)CC12 CCC(C)(C(=O)NCC1CN(C(=O)Cc2ccn(C(F)F)n2)CCN1C)C(N)=O c1(C(N2CCCCC(CNC(=O)CSC3CC3)C2)=O)nccc2c1CNC2=O C1(NC(CSC)=O)CN(C(c2cccnc2-n2nccn2)=O)CC1N=[N+]=[N-] N1(C(CCC=C)=O)CCN(C(=O)COc2cc(C)ccc2C)C(C)C1C c1(C(N2C(C)CN(C(C3COCCO3)=O)CC2)=O)cccc2nn[nH]c12 C1(CNC(C(C)Sc2nnnn2C2CC2)=O)CC2CCC1N(C(=O)C(C)(C)F)C2 c1(C(N2CCC(CC=C)(NC(=O)C(C)O)C2)=O)nc(Br)c2c(F)cccn12 C1(NC(c2cc(CNC(CN3C(C)CCC3)=O)sc2)=O)CCCCC12CC2 C1(N(C(CCNC(COC)=O)=O)C)CN(C(c2cnc(C(C)C)s2)=O)CC1F N1(C(C(n2ccc(C)n2)(C)C)=O)CC(NC(C2CCC(=O)NC2)=O)C(C(F)F)C1 O=C(CCCCSc1ccccc1Cl)NCc1snc(Cl)c1Cl C1(F)(CNC(CC2CCC(=O)N2)=O)CCCN(C(=O)Cc2ccncc2Cl)C1 N1(C(C2(N)C(C)(C)C2)=O)CCC(C)(O)C(O)C1 Cc1nc(C(C)C)oc1C(=O)NC12COC(CNC(c3coc(Cl)n3)=O)(C1)C2 N1(C(c2c(CC)c[nH]n2)=O)CCN(C(=O)CCCC2CCCC(=O)N2)C(CC)C1 C12(C(=O)NC3CC(N(C)C)C3)CC(n3cc(C4CCCC4O)nn3)C1C2 Cc1cn2ccc(C(=O)NC3(CO)CN(C(C4CC5CCC5C4)=O)C3)cc2n1 c1(CC)onc(C(=O)N(C2CCN(C(c3cc(C4CC4)ccn3)=O)C2)C)c1C c1(CN(C(C=CC(C)NC(c2ncoc2C2CC2)=O)=O)C)cccnc1O c1(C(c2n(CCCC)nnn2)NCc2nc(CO)cs2)ccc2c(n1)CCC2 c1(C(N(C2CN(C(C=Cc3scc(C)n3)=O)CC2F)C)=O)cc(Cl)cc(C)c1C C1(CC(=O)OCC)CCC(C(N2CCC(NCCCN(C)C(C)C)C2)=O)CC1 c1(CNC(C(c2cnn(C)c2)NC(c2c(C)cccc2)C)=O)ncc(F)cc1F c1(C(=O)NC(CNC(CCCOCC=C)=O)CCOC)ccc(C)c([N+](=O)[O-])c1 c1(CCOC)cccc(C(=O)NCCC(C)(C)CNC(=O)COC2CC2)c1 Cc1cccc(C(C)C(=O)NCCOCCN(C)C(c2nc(Cl)c(Cl)s2)=O)c1 C1(C(=O)NC(C=C)C2CCC2)CC1C1CN(C(=O)CN=[N+]=[N-])C1 C(=O)(C1Cc2c(Cl)cccc21)OC.CCC1CC(=O)NC2(CC2)CNC(=O)COC1 c1(C2(C(=O)NCCC(=O)NCC=CCSC)CC2)ccncc1 Cn1nc2c(c1C(=O)NCc1ccc(Br)c(F)n1)CCCC2 CC1CN(C(c2cnccc2C(F)F)=O)CCC1CNC(=O)C=CCN1CCC1 c1(SCCCNC(NCCc2n(C)ncc2)=S)ccc(Cl)cc1 Cc1nn(CC(=O)NCC2(NC(=O)CC(O)C(Cl)(Cl)Cl)CC2)cc1[N+](=O)[O-] Cc1ccc2c[nH]nc2c1NC(C1CCCN(C(=O)Cc2cc(Br)cs2)C1)=O C1(O)(CNC(C2C(C=C)C2)=O)CCCN(C(c2ccc(N)cc2OC)=O)C1 C1(N(C)C(c2ccnn2CC#N)=O)CCC(NC(=O)CN2C(=O)CNC2=O)CC1 C(=O)(C(CC(F)F)Nc1nccnc1N)NCC(C)C CCC(C#N)C(=O)NC1C=CCC(C(=O)NC2(C(C)O)CC2)C1 c1(C(=O)NCCCNC(C(CC(=O)OC)(C)C)=O)cncc2c1CCNC2=O S(=O)(=O)(c1ccc(NC2CCCN(C3CC3)C2)c(Br)c1)NCC(C)F Cc1cc(C(=O)NCC2CCN2CC=C(Cl)Cl)sc1C C1(NC(C(C)=C2CCCC2)=O)CC(F)CN(C(c2cnc(S)n2C)=O)C1 C(C(C(=O)N1CC(F)(CF)C1)n1cc(C2CC2)nn1)OCC.c12cc(no1)OC2 N1(C(COC(C)=O)=O)CC23CCCCC2(C1)CN(C(=O)C(C)(C)C1CCCCO1)C3 c1(CC(=O)NC2CC3(C2)CC3NC(c2cnn(C3CCC3)c2)=O)ncncc1Cl CC(C)CC(C)C(=O)NC1CN(C(=O)C(O)CCc2ccccc2)CC1C N1(C(C)=O)CC(C)CN(C(c2coc(S(C)(=O)=O)c2)=O)C(C)C1 CCC(CCC(=O)NCCC[Si](C)(C)C)NC(C1C2CCC(F)C12)=O Cc1nn(C)cc1CC(C(=O)O)NC(c1ccc(OC(F)(F)CF)cc1)=O c1(C(=O)NC2(CC(=O)NCc3ccc(Cl)o3)CC2)cnc(CO)cn1 CC(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1CCN(C(c2c[nH]nc2C2CC2)=O)CC1 c1(OC)ccc(F)cc1CC(=O)N(CC(O)CNC(C1CCCN1C(C)=O)=O)C c1(C(=O)NC2C(C)CN(S(=O)(=O)CC#N)C2)ccc2occc2c1 c1(C(=O)NC2CN(C(c3ncsc3C(F)(F)F)=O)C2)ncc2n1CCCC2 c1(C(=O)NCC2CN(C(C(C)(C)C3CC3)=O)CC2O)cc(P(C)(C)=O)cs1 c1(CC(=O)NC(CC)CNC(=O)CN2CCC(C)C2)cc[nH]c(=N)c1 c1(OC)cc2c(C(=O)N(CCNC(C34CC(C)C3C4)=O)C3CC3)c[nH]c2cc1Cl Cn1cc(C=CC(=O)NCC(C)(C)C(=O)NCCn2ccnn2)cn1 c1(C(=O)NCCN(C(C(C)=C2CC2)=O)C(C)C)cc(F)cc([N+](=O)[O-])c1Br Cc1sc(C(N2CC3CC2(CNC(C2CC(=O)NC2=O)=O)C3)=O)cc1[N+](=O)[O-] C(=O)(C(C)C(=O)OC)N1CC(CCNC(c2ccc(CN(C)C)o2)=O)(OC)C1 C1(CC)CN(C(c2ncoc2-c2ccon2)=O)CCC1NC(C1COC(C)C1)=O c1(OC)ccccc1C(=O)NCCC1(O)CCN(C(=O)CC2(C)CCOC2)C1 CC1CCN(C(=O)C=CC(C)(C)NC(c2cnc(C3CC3)o2)=O)C1CO C(CC(CC)C(=O)NC1CC(C)(NC(=O)CCN(C)CC)C1)=CC c1(C(N2CCC(C(C)NC(=O)C(F)=CCCF)CC2)=O)ccc(C#N)cc1F N12CC(O)C(O)C1CNC(=O)C1(CCCC1)CC2=O.c1ccsc1C.C=CC C(=O)(C(Cc1ccccc1)C(C)C)NCCC(C)(C)NC(C1ON=C(CC)C1)=O C(N=c1[nH]c(=N)[nH]c(=NCc2nc(CO)n[nH]2)[nH]1)c1ccc(F)c(C)c1F Cc1cncc(C(=O)NC2CCN(C(c3ccsn3)=O)CC2F)c1C C(=O)(CCS(=O)(=O)CC(C)C)N1CC2(CN(C(C(COC)OC)=O)C2)C(CO)C1 Cc1c(C(N2CCN(CCNC(C3CCO3)=O)CC2)=O)cnn1CCC(C)C c1(OC)ccc(CNC(=O)CC2CCCN2Cc2ccc(F)cc2O)c(C)c1C N1(C(C=C(COC)C)=O)CC2(CCC2)OCC1C(=O)O C(=O)(C1CCCc2nccn21)N(CCCCN(C)C(C1(n2nccn2)CC1)=O)C C1(CO)CC2(C1)CC21CC1.C12(F)CN(C1)C(=O)CN1CC(C1)OCC2 Cc1ccc(C(=O)NCC2CCN(CCCN3CCCCC3)C2)cc1 c1(OCC(N2C(CCNC(C(C)C3CC3)=O)CCC2)=O)ccc(CC#N)cc1 c1(CN2CC(C)CC(NC(=O)Nc3cc(C)cc(F)c3)C2)cccc2cc[nH]c12 c1(OC)cc(C(N2CCC(CNC(c3cccc(C)c3)=O)C23CC3)=O)ccc1F c1(C(N2CCC(C)(NC(C(C)SCCCCCC)=O)C2)=O)ccc(C)cc1CC Cc1cc(C(=O)NC(C)CC(C)NC(c2nnn3c2CSCC3)=O)cc(=O)n1C c1(OC)cc(C(=O)NC2CC(C)CN(C(c3ccc(O)c(Br)c3)=O)C2)ccc1Br C#CCCCCCC(=O)NC1CCCC1NC(=O)C(c1ccccc1Cl)(F)F O=C(CC(C(F)F)NC(=O)COCC1(O)CC(O)C1)NC1CCOC1 C(=O)(CCCC(=O)N1CCOCC(CNC(=O)CC2CCCN2C(C)=O)C1)NC C1(CNC(C=CC(C)C)=O)CC2(CC2)CN1C(c1ccc(C2(F)COC2)cc1)=O c1(C(C(=O)NC2CCCN(C(CN(CC)CC)=O)C2C)O)cccc2c1OCC2 c1(C(=O)OC)ccc(CC(N2CC(NC(C3CC3c3cncn3C)=O)C2)=O)cc1 c1(C(=O)NC2CCN(C(CCCOCC=C)=O)CC2)ccc2ccsc2c1 c1(C(=O)NCC(C)(C2CC2)NC(c2n(C)ccc2)=O)cccc(Br)c1N Cn1nc(C(N2CC3CC2CC3NC(c2ccoc2Cl)=O)=O)ccc1=O c1(N(C(CC(C)C)c2nn[nH]n2)C(=O)CN2CCN(C)CC2)ncccc1F CCCCCC(C)(C)C(=O)NCC(CC(C)C)NC(C1CCC(C)(F)CC1)=O c1(C(=O)NCCN(C(c2ccn(CC(C)C)n2)=O)C)ccc2nc[nH]c2c1F c1(C(=O)OCC)oc2ccccc2c1CC(c1cc(Cl)ccc1F)(C)C(=O)O C1(C(CC)C)CCCN1C(=O)CC(C)N(C(=O)CCN1CCOCC1)C c1(OC)ccc2cc(C(=O)NC3CC(NC(C45CC(C)C4C5)=O)C3)ncc2c1 c1(CNC(=O)NC(c2ccc(OCCCC)cc2)C)cc2ccncc2s1 CC1(C)C(C(=O)NCCC2NC(=O)NC2=O)CCN1C(c1n[nH]c(O)n1)=O CC1CCC(CNC(C2CCC(=O)N2C(C)C)=O)N(C(=O)OC(C)(C)C)C1 c1(C(N2CC(C(N)=O)(CNC(=O)C(c3cncn3C)O)C2)=O)cccn(O)c1=O N1(C(C2C(C)CCO2)=O)CCCN(C(c2c[nH]nc2-c2ccccc2F)=O)CC1 c1(NC2CCCN(CCCO)C2)[nH]c(=NCc2ccsc2)nc2sccc12 C1(C(N(CC(C)(C)NC(=O)CCn2cnnn2)C)=O)CCC2(CC2)C1 N1(C(c2cnc(C)n2C)=O)CCN(C(C2C=CCC2)=O)C(C)C1 Cc1ccc(N2CCCC2)c(C(=O)NC(C)CNC(c2ccc(=O)oc2)=O)c1 CCCC(C)(O)C(=O)N1CCC(c2ccccc2)(NC(=O)CSC(F)F)C1 N1(C(C2C(C=C)CC2)=O)CCC(NC(=O)CCCC)C12CCC2 N1(C(c2c[nH]c(=NC)o2)=O)CC(NC(c2ccc(C(O)CF)cc2)=O)CCC1C C(C(F)(F)C(=O)NC(C1CCN(C(=O)C(=C2CCCCC2)F)C1)C)OC c1(C(N2CCC(O)(CNC(=O)Cn3cnnn3)C2)=O)cccc2nc(O)ccc12 c1(NC(C(=O)NC(CCC)C(=O)NC)=O)cc(C)c(Br)cc1Cl c1(C(N2CC(CCCCNC(CCC(=O)NCCC)=O)C2)=O)cnc(F)cc1C c1(COC(C(CNC(C2(CCCCC)CC(F)C2)=O)O)=O)cccc(C)c1 C=CC(C)(CCOC)C(=O)NCC1CN(C(=O)Cc2cccs2)C2(CCC2)C1 C(C)(CNC(c1ncc(Br)cc1F)=O)(CC(C)C)NC(CSC)=O N1(C(c2cn(C)nc2)=O)CC(CC(=O)NCC(C)(O)C(C)(C)C)CC1(C)C CCC(O)C(F)(F)C(=O)NCC1CCCN1C(C1CC1C(N)=O)=O C(=O)(C1=C(C)CCCC1(C)C)NCC1N(C(C(CC)SC)=O)CCCC1C C(=O)(C1CCCc2ccccc21)NC(C1CN(C(C(F)OC)=O)C1)C c1(C(C)C)ccc(C(=O)NCC2CCN(C(C3(C)CCN(C)C3)=O)C2)nc1 N1(C(C(CC#C)C2CC2)=O)CCC2(CC(NC(C3(c4ccno4)CCC3)=O)C2)C1 c1(SCC(=O)NCC2(c3ccccc3)CC(NC(C3C(C)=C3)=O)C2)ccc(C)cc1 c1(CC)c(C(=O)NC2CCCC2NC(=O)CCc2ccc(O)nn2)cnn1CC C1(N(C(c2nnc(C)s2)=O)C)CN(C(c2cc(C(C)C)oc2C(C)C)=O)CC1F CCCC(C)(C)CC(=O)N1CCC(C(F)C(=O)N(c2cccc(CC)c2)C)C1 C(=O)(C1=C(Cl)CCCC1)N1C(CNC(C2(COC)CC(F)(F)C2)=O)CCC1 c1(C(=O)NCCN(C(=O)CCn2ccnc2C(C)C)CC)ncn(C(C)C)n1 C1(OC(C)(C)C)CC(OCC(=O)NC2CC(Cc3ccccc3)C2(C)C)C1(C)C CCCCC(C)C(=O)N1CCC(C(C)NC(c2cc(COC)cs2)=O)C1 C(=O)(C1CCc2cccc(=O)n21)NCCN(C(CC1(C)OCCO1)=O)C1CC1 N1(C(CC(CC)OC)=O)CCC2(NC(c3ccc(SC)cc3Cl)=O)CCCC12 CC1CCc2[nH]c(=NCCCOc3ccccc3F)[nH]c(=NCC(Cl)=CCl)c2C1 CC1(C)CCCc2c1nc(Cl)[nH]c2=NCC1(CNC(=O)CSC(F)F)CCCC1 C1(C(=O)NC(CNC(C2N(C)CCC2)=O)C2CC2)COc2cc(O)ccc2C1 Cc1ncc(Br)cc1C(=O)NC1CCN(C(C2CC(C)(F)C2)=O)CC1C C1(C(=O)NC(C)CCCNC(=O)C(=Cc2c[nH]cn2)F)CC1C1CCOCC1 c1(CN(C)C(=O)NC2CCCC2(C)C)nnc2c(=O)[nH]ccn12 C1(CC=C)CCCN(C(=O)C(C(C)OC)NC(=O)C(C2CC2)SC)C1 n1(CC(=O)NCC(C)(CNC(c2cncc(C)c2)=O)OC)ccccc1=O c1(CC(=O)NCC(C)CNC(=O)Cn2cnc(C#N)n2)ccc(C(F)(F)F)cc1 CC1CC(CNC(c2csc(CO)n2)=O)CN1C(c1nn[nH]c1Cl)=O c1(C(N2C(C(=O)Nc3c(OCC)ncnc3)CC(F)C2)=O)cc(C)ccc1O C1(NC(c2c(C)cncn2)=O)CN(C(c2ccc(C(C)O)cc2)=O)CCC1O c1(-c2n(C(C(C)C)C)nc(CS(C)(=O)=O)n2)cn2c(n1)CCC(C)C2 c1(C(=O)NCC2N(C(c3c(C(C)C)cccc3)=O)CC2)cc2ccccc2n1C Cc1ccc(C#N)cc1C(=O)NCC1CC(NC(C2CC3CCC(C2)C3)=O)C1 CC(C)C(=O)C(=O)N(CC(=O)NCC(O)C1(Cl)CC1)C1CC1 S(=O)(=O)(c1ccc(N2CC3COCC3C2)cc1Cl)NC1CC(CC)OCC1 C=C1CCC(C(N2CC(C(C)NC(=O)CC(C)(C3CCC3)N(C)C)C2)=O)CC1 C#Cc1ccc(CC(=O)NCCC(C)(C)CNC(c2c[nH]ccc2=O)=O)c(F)c1 Cc1cccc2oc(N3CC4CC(NC(C5(S(C)(=O)=O)CCC5)=O)CC4C3)nc12 N1(C(C2CNC(=O)N2)=O)CCCCC(CNC(c2n[nH]cc2C(F)(F)F)=O)C1 O=C1CC(C(=O)N2CC(NC(c3ccccc3Cl)=O)CC2CO)=NN1 C1(C(=O)NCCc2c(C(=O)Nc3cc(C)no3)c[nH]n2)CCCCC(=O)N1 Cc1cc2ccccc2n1CCC(=O)NCC1CC2CCC(C1)N2 C1(C(=O)NCC2N(CC)CC2)(C(C)C)CCCN1C(=O)C=Cc1cscn1 CC1(Cn2cc(CC3CN(C(C4CCCCC4)=O)C3)nn2)CCCC1(F)F N1(C(CNC(CC)=O)=O)CCN(C)C(C(N2CC3(CC3C(=O)OC)C2)=O)C1 c1(OC)cc(C)c(C(=O)NCCN(c2ccnc(C3CC3)n2)CCC)cn1 C1(NC(C(C)OCC=C)=O)CCCC1CNC(=O)CC1CCCN1C(C)C C1(C(N(C(c2ccccn2)C)C2CC2)=O)OCCC1NC(=O)OC(C)(C)C C1(CC)C(C(=O)N(CCCN(C)C)CC)CCCN1C(c1cc(C)ns1)=O CCCCCS(=O)(=O)CC(=O)NC12CCCC1N(C(=O)Cc1cnc(C)s1)CC2 N1(C(c2cc(C)c(C)[nH]2)=O)CCCC(N(C(=O)CC2CC=CCN2C)C)CC1 C(=O)(CS(=O)(=O)CCO)NCCC1(O)CCN(C(CCSC)=O)C1 c1(C(=O)NC(C(=O)Nc2cnc(NCC)nc2)(C)C)cccc2cncn12 c1(OC)cnc(SC)[nH]c1=Nc1c(NC(=O)C=C(C)C)sc2c1CCC(C)CC2 CN1CCC(C(=O)NCC2CN(C(N)=O)C2)(NC(=O)CCC2CCOC2)C1 C1(C(N(CCNC(c2sc(C)cc2Cl)=O)CC)=O)C2CS(=O)(=O)CC12 N1(C(c2nc(-c3cc(OC)ncn3)sc2)=O)CC(OC)CC(c2ccccc2)C1 Cc1c(C(=O)NCCCC2CCCN2C(=O)CC(C)F)sc2ccc(Cl)cc12 c1(C(c2nnnn2C2CC2)NCCCCCC)cnc(OC)c(C)c1 c1(C(=O)NC(C(C)(C)NC(CSCC=C)=O)C)ccc(-c2cccs2)nc1C C12CN(CCO1)C(c1ccc(I)cc1)C(=O)N1CC2C1.CC(=O)NC1CC1 C1(C(N2CCCN(C(C=Cc3c(C)n(C)nc3)=O)CC2)=O)CNC(=O)CC1(C)C C(CCCCCN(C)C(c1ncsc1Br)=O)NC(C1CCC(C)O1)=O Cc1cc(CC(N2CC(=C(F)CNC(=O)Cc3cn[nH]c3)C2)=O)c(O)nc1C C=CC(O)(C(=O)NCC(CNC(c1ccc(Cl)cc1)=O)CO)C(F)(F)F C1(CNC(c2cnc(C(C)(C)C)o2)=O)(CO)CCN(C(=O)CC2CC(F)(F)C2)C1 C1(SC)CCCC1C(=O)NCC(c1ccccc1)NC(c1cnsc1C)=O c1(SC)cccnc1C(=O)NCC(C)(C)CCNC(=O)C(C)(C)C1CCCCO1 c1(C(C(=O)NCC(CN(C(C2SCCS2)=O)CC)(C)C)C)ccccc1OC c1(SCC(N2CCCC(N(C(=O)CN(C)C(C)C)CC)C2)=O)ccc(Cl)c(Cl)c1 S(=O)(=O)(c1nc[nH]n1)Nc1cc(C(C)(C)C)no1 N1(C(C(C)N(C(C)=O)C)=O)C(C(=O)NC(CC(C)C)C(N)=O)CCC12CC2 CC1CCCC1(C(=O)NCC1(C)CC(O)C1)NC(c1ccc(C#N)s1)=O c1(OC)ccc(C(N)C(=O)NCCC2(c3ccccc3)CCCO2)cc1OC c1(C(=O)NC2C(NC(C3C(C=C)OCC3)=O)CCC2)nccc2[nH]ccc12 CC#CC1CCN(CCNC(=O)Cc2scnc2C)CC1 Cc1onc(CC(=O)NC2(C)CN(C(c3ccn(C(C)C)n3)=O)C2)c1C#N Cc1cc(Cl)c(Cl)cc1CN1CC2C(NC(c3cc[nH]n3)=O)C2C1 c1(C(c2nc(=O)n(C3CCN(C(=O)C(=O)N4CCC4)CC3)[nH]2)C)ccc(F)c(C)c1 C=CC(CCC)CC(=O)N(CC)CC1CCCN1C(=O)Cc1cn[nH]c1 C1(CNC(C2(NC(CCOCCCOC)=O)CC2)=O)CC2C=CC1CC2 c1(NCCc2ncn(CC)c2)cc(Cl)c(Br)cc1O CN1C(=O)c2ccccc2C1C(=O)N1CC2CC(NC(c3cnn(C)c3)=O)C1C2 C1(C(=O)NCC2N(C(CC(C(C)C)(F)F)=O)CCC2)CC12CCc1ccccc12 C123CCC(CC1)(C2)C(=O)CNC3=O.c1(C(=O)OCC)n[nH]cc1CCCC1CC1 C1(O)(CC(N2CC(c3ccon3)(NC(C(C)CN(C)C)=O)C2)=O)COC(C)(C)C1 C(C(C(=O)NCc1nnc(C)o1)C(C)(C)C)NC(c1n(CC#C)ccc1)=O CCCCCC(O)C(=O)NCC1CCN(C(c2ccc3c(c2)NCC3)=O)C(C)C1 c1(C(N2CCCC(N(C)C(c3cc4c(s3)CCC4)=O)C2)=O)cc2cccnc2s1 Cc1ccc(C(=O)NC(C2(CNC(C3(CO)CC3)=O)CC2)C)c(O)c1.C1(C=O)CC1 C(CC(O)CNC(=O)CCOCCCNC(C1C(C)C1C)=O)OC C1(OC)CC(C)(C(=O)NC2(C(=O)NC3CC(C)(C)C3)CCC2)C1 S(=O)(=O)(c1c[nH]ccc1=NCC1C(C)(C)C1(F)F)NCc1c(C)occ1 c1(C(N2CC3C(C(=O)NC(C#C)C)(C3)C2)=O)ccc(Br)c(OC)c1F c1(CN2CCCC(CCNC(c3c(C)cc(Br)cn3)=O)C2)cccc([N+](=O)[O-])c1 C1(C(N(C)Cc2ncn(C)n2)=O)CN(C(C23C(=O)C4CC2C3C4)=O)CC1(C)C c1(C(C)(C)N(C(=O)CN2CCC(N3CC=CC3)C2)CC)cc(C)c(C)cc1C C(=O)(CC(C)C(F)F)NCC(CCCC)NC(C1CCCN(CC)C1)=O c1(NC(C2(CCC=C)CN(C(=O)CC3CCC(=O)C3)C2)=O)ccc(OC)cc1C C12(C(=O)NC3CN(C(C(C)CN4CCOCC4)=O)C3)CCCCC1NC(=O)C2 Cc1n[nH]c(C)c1CC(C)C(=O)NC(C)(C)CCNC(=O)C=C1CC1 C(=O)(C(COC)C(F)(F)F)NCCC1CC(NC(C(CCC)O)=O)C1 N1(C(C2(C)CN(C(C=CC3(C)COC3)=O)C2)=O)CCCCC(CC2CC2)C1 Cc1cccc(C(N2CCCC(N(C)C(C3CCCC34CC4)=O)C2)=O)c1F N1(C(CSC(C)C)=O)CCN(C(C2CCCSC2C)=O)CC(C)C1 c1(C(=O)NCC2(CC(=O)OCC)CCCCC2)ccc2c(n1)OCC(=O)N2 c1(C(=O)NC2CC(F)(CNC(C3(C=C)CCCCC3)=O)C2)c(F)ccc(O)c1F C(=O)(CS(=O)(=O)c1ccccc1F)N(CCNC(C(C)C)=O)Cc1ccccc1 c12ccc-1c(F)c2.S(=O)(=O)(CCCc1ccccc1)N.C(=O)(C(Cl)(Cl)Cl)NC(=O)C c1(O)ccc(=NCCOC)[nH]c1.C1(OCC)CCN(CC)CC1O N1(C(c2c(C)nns2)=O)CCC2C(CCCN2C(c2ccnnc2S)=O)C1 C1(C)(CC(=O)NC(C)C(C)NC(c2cnns2)=O)CCCO1 O=C(C1=NOC2(CCC2)C1)NC(CC1CC1)C(N1CCc2nccnc2C1)=O c1(C(=O)NCC2C3CN(C(c4n(C)nc(Cl)c4)=O)CC32)cnn2ccncc12 C(CCNC(C1(C)CCC(=O)C1)=O)(C(=O)NCCNS(C)(=O)=O)OC C1(NC(CC(=O)NCC)=O)CCOC12CCN(C(c1cc(Cl)ncc1F)=O)CC2 C1(CNC(CC(CC)O)=O)CCCCN(C(C2CC2c2ccccc2)=O)C1 c1(C(=O)NCCN(C(C2C(C)(CC)C2)=O)C(C)C)c(Cl)c([N+](=O)[O-])nn1C N1(C(=O)C=Cc2cn[nH]c2)CCC2(CNC(C3(Br)CC3)=O)CCCCC12 N1(c2cccc(CCC)n2)CCCCC1c1nc(C(C)C2CC2)nn1C1CCOC1 C(C(C)(O)CC(=O)N1CCC(C(=O)NC2CCCC2C(C)O)C1C(C)C)OC C1(NC(C2(C#C)CC2)=O)CN(C(c2c(Cl)csc2Cl)=O)CCC1C(F)(F)F CN1CCN(CC(=O)NC2C=CC(CNC(C3CC=CCO3)=O)C2)CC1 c1(C(N2CCC(C(C)NC(C3C(C(=O)OC)C3)=O)CC2)=O)ccc(C)cc1F C12(CNC(C3N(C)CCOC3)=O)CC(C1)C(NC(=O)CN1C(=O)CNC1=O)CO2 Cc1cccn2c(C(N3CCN(C(=O)Cc4cnoc4)CC3C(C)C)=O)cnc12 c1(C(=O)NC2CC(C)(CC)N(C(=O)Cc3cc(C)no3)C2)ccc(F)c(N)c1F C(=O)(C(F)C(C)C(F)(F)F)NCC1(C)CCN(C(C(C)SCC)=O)C1 CN1CCCC(CN(C)C(c2c(CNC(=O)CCn3ccnn3)nnn2C)=O)C1 N1(CCCNC(C(C)NC(C2CCC2)=O)=O)CCN(C(C23CC(F)C2C3)=O)CC1 n1(CC)cnc(C(N2CC(C(C)NC(=O)CCn3ccc(C)n3)C2)=O)n1 C(c1cc(Cl)ccc1Cl)=CC(N1CCCC2(NC(c3c(C)onc3)=O)C1C2)=O C=CCCCCC(=O)NC1(C)CCN(C(C2CC23CCSCC3)=O)C1 C=CCC(C)(C)C(=O)NC(C)CN1CCN(C(c2n[nH]cc2OC)=O)CC1 CCC(C)C(C(=O)NCCCN(C(C12CC(CC(C)O1)C2)=O)C(C)C)NC(C)=O c1(C(N2C(C(C)C)C(NC(=O)C=CCO)CC2)=O)cc(=O)c2ccccc2o1 c1(NC(=O)NCC(=C)C)nc(C)c(CC2CCN(C)C2c2ccccc2)s1 Cc1c(C(N2CC(NC(=O)C(C)CF)C2)=O)cnn1C1CCCC1 c1(C(N(C2CCC(NC(=O)C(C)(O)C3CCC3)CC2)C)=O)cccc(C(F)F)c1 CC(C)C(CNC(C1C(c2ccccc2)C1C)=O)OCCOC(=O)C(C)(C)O C1(C(=O)Nc2cnc(Br)nc2)CN(C(c2cc(O)no2)=O)CC(F)(F)C1 C1(NC(Cc2cc(CC)nn2C)=O)CN(C(C23COCC2C3)=O)CC12CCC2 N1(C(C(CCCC)O)=O)CC2CCC(C1)N2c1cc(C)nc(C(C)CC)n1 C1(c2cn(C)nc2)CCCCN1C(=O)NC(c1ccc(Br)cc1)C1CCC1 C1(NC(CC2CC(C(=O)OC)C2)=O)CCCCN(C(c2cc(C)c[nH]2)=O)C1 c1(C(=O)NC(C)CCCNC(C2CCCC(C)C2)=O)cn(C)c(=O)c2cncn12 C1(CNC(=O)CC2CCSCC2)CC2(CCN(C(C34CC(C3)C4)=O)C2)CO1 c1(CC(N2CCC(N(C)C(C3CCCC3)=O)C2)=O)ccc2c(c1)CCCO2 C(C(C(C)(C)C)NC(=O)C(C1CC1)C1CC1)NC(c1c(C)[nH]cc1)=O Cc1c(C(=O)NC(C)CCN(C)C(c2ncccc2O)=O)[nH]ccc1=O N1(C(C2N(CC)CCC2)=O)CCC2(CC1)CC2C(=O)NCC1(O)CCC1 N1(C(C2N(C(c3c(C)noc3N)=O)C(C)C2)=O)CCN2CCCCC1C2 Cc1[nH]nc2c(C(N3CCC(NC(C4CCCOC4)=O)C(F)C3)=O)cccc12 C(CCCC(=O)NC1(CCNC(=O)CC2COC(C)(C)C2)CCOCC1)N(C)C N(C1CCCc2cccc(C)c21)C(=O)NC(COCC)CO C1(NC(C(CC)N(C)C)=O)CC(C)N(C(c2csc(Cl)c2OC)=O)C1 n1(CCC(=O)NC2CCN(C(COC3(C)CCC3)=O)C2)ccc2cccnc12 n1(CC)ccc2nc(N3CCC(NC(C4(C#N)CC4)=O)C(O)C3)ncc12 CC1(C)CN(C(=O)CCn2ccnc2)CC(CNC(=O)CCCC#N)O1 N1(C(=O)NC(C)C=CCc2ccccc2)CCCN(CC(O)C(F)(F)F)CC1 C(C(=O)NCC1COCCN1C(=O)C(=O)C(C)(C)C)(C(C)(C)C)N(C)C C(=O)(CCCCC(N)=O)N(C1CC2CC1N(C(=O)CCOCC(F)F)C2)C N1(C(C2CC(C)CC(C)C2)=O)CCCC(O)(CNC(=O)CC2(O)CCC2)CC1 C1(CCNC(=O)C=CC2CC2)CN(C(=O)C2=CCCCCC2)CCS1(=O)=O C1(N(C)C)CCN(C(c2cnc(C(C)(C)C#N)s2)C(=O)NC2CC2)CC1 c1(C(=O)NCC2CCN2C(c2cn3ccccc3n2)=O)cnn2ccc(O)nc12 c1(C(N2CCC(NC(c3nc(CC)sc3)=O)C(F)C2)=O)c(C)ccc(C)c1C c1(C(=O)NCC(CC(F)(F)F)NC(C(CSC)C)=O)nc2ccccc2[nH]c1=O C(=O)(CC(O)Cc1ccccc1)N(CC(C)NC(C=CC(C)C)=O)C c1(OC)cc(C(=O)NC(C2CCN(C(c3ccccc3F)=O)C2)C)ccc1Cl C(=O)(CCCCCN=[N+]=[N-])N1CCN(C(C(CCC(C)C)NC(C)=O)=O)CC1 N1(C(CCCCC#C)=O)CCCC12CCN(C(=O)C(CO)c1ccccc1)C2 N1(C(CN(C)CC2CC2c2ccc(Cl)s2)=O)CCN(C(C2CC(F)(F)C2)=O)CC1 c1(C(N(CCNC(c2cc(C)nc(C(C)(F)F)n2)=O)CC)=O)ccc2ccnn2c1 c1(CC)ccc(C(=O)N(C)CCNC(=O)C(Cc2ccccc2)OC)c(C)n1 c1(OC)cc(Br)ccc1CN1CCC2(CC1)CC2.C12CC1CNC2=O c1(C(=O)NCC2CN(C(C3C(C)=CCS3)=O)CC2O)cc(C)n(C2CC2)c1C c1(C(C(=O)NC(C)CCNC(c2csc(CC3CC3)n2)=O)(C)C)cccc(F)c1 C1(C)(CNC(c2c(C(C)NC(CCCC#C)=O)noc2)=O)CCC(=O)N1C C1(NC(=O)C2=CCOC2)CN(C(c2ccnc3ccsc23)=O)C2(CCOCC2)C1 c1(NC(CCC)C2CCCC2)ncccc1S(=O)(=O)NCCc1cc(Br)ccc1C N1(C(c2ccc(Cl)cc2C(F)(F)F)=O)CCCN(C(=O)C2CC2)CCC1 c1(C(=O)NC2CC(CNC(C(C(C)C)(C)O)=O)OCC2)ccc2c(c1)CC(=O)N2 CC(C)CC(C)(CNC(=O)CC1CC2CCC1CC2)NC(C12CC(F)(C1)C2)=O Cc1cn2ccc(C(N3CC(NC(c4cc(Cl)cnc4C)=O)C(C)C3)=O)cc2n1 c1(C(=O)OC)ccc(C(N2CCCC(C(C)NC(=O)CSC(C)=O)C2)=O)c(F)c1 C(CCC(=O)NO)NC(C(C1CCCN(C(=O)CC2NC(=O)NC2=O)C1)C)=O c1(C(C)C(=O)NC2CC(c3ccccc3)CO2)ccc(F)c(F)c1 c1(C(=O)NC(CC)C(=O)NCc2c(COC)cccc2)c(C)noc1CC(=O)O n1(CCC)ncc(C(c2nnnn2CC(F)F)NCC(C)(CC)CC)c1C n1(C(C)C)ccc(=NC(=O)C2(C)CCCN(C(c3ccc4c(c3)CC4)=O)C2)[nH]1 N1(C(C(C)SCC)=O)CCCCC1CCC1CCCN1C(c1n[nH]cc1CC)=O c1(C(N2CCC(NC(C(CCC#C)O)=O)C2)=O)cc(Br)cc(C)c1C c1(C(NOCCC=C)=O)ccc2c(n1)CN(C(C1CCC(OC)CC1)=O)CC2 c1(C(N(CC(C)NC(Cn2c(C)nnn2)=O)C)=O)ccc(O)c(C(C)(C)C)c1 C(=O)(C(O)C(C)(C)C)N(CC)CC1CCCN1C(c1cccc(CCC#N)c1)=O c1(C(C(F)(F)F)OC(C=CCOC)=O)ccccc1F C(CCCCC(=O)NC)NC(C(CCC)NC(=O)C(C)(C)OC)=O C1(NC(CC(CCC)O)=O)CN(C(c2cc(C(N)=O)no2)=O)CCC1(C)C c1(CN2CCC(C(N(C3CC3)CC)=O)C2)c(C)cc(C)nc1O N1(C(COCC)=O)CCC(C2CC2)C1C(=O)Nc1ccc(C)cc1C C1(OC)COCCC1CC(=O)NCC(C(C)C)NC(C1CCC(=O)O1)=O c1(C(N(C2CCN(C(c3nc(C)n(C)n3)=O)C2)CC)=O)cc(SC)c(C)o1 N1(C(c2cc(CC)no2)=O)CCN(C(=O)CN(C(=O)C(CC)CC)CC)CC1 N1(N2CCC(n3ncc(C)c3)C2)CCC(c2ccc(Br)cn2)CC1 CC1CN(C(=O)COc2ccc(Cl)cc2)CC1CNC(C1C=CC=CC=C1)=O N1(C(C(CC#C)CC#C)=O)CCC2CN(C(=O)CCN(C)CC)CC2C1 CN=c1nc(N2CCN(S(C)(=O)=O)CC2)[nH]c(=NCc2c(OC)cccc2F)[nH]1 C1(CNC(c2c(CC(C)C)onc2)=O)COCCN(C(c2ccc(F)s2)=O)C1 Cc1ccc(C(=O)NCCCCC(C)NC(c2nncs2)=O)c(N=[N+]=[N-])c1 CC(CC(=O)NCC1CC1(Cl)Cl)NC(c1csc(O)n1)=O CCCCCCC(F)C(=O)N1CCCC(CO)(NC(=O)CCc2cc(Cl)no2)C1 N1(c2cc(COC)ncn2)CCC(O)(C(=O)N(C)CCC2CCCC2)CC1 c1(C(=O)NC2CCC(C(=O)NCc3cnc(C)nc3)C2)ccc(Br)cc1O c1(C(CC(=O)O)NC(CC)C(=O)NC(N)=O)cccc(Br)c1 CCC(CC(C)C)C(=O)NCC1CCN(C(C23CC(CN2C2CC2)C3)=O)C1(C)C N1(C(C(CCOC)NC(C(CC#C)O)=O)=O)CC2(COC(C)C2)C1 CC(C(CO)NC(=O)CCC1CCCO1)NC(c1cc(-c2ccccn2)no1)=O N1(C(C(C)C2CCC2)=O)CC2CCCC1(CNC(c1ccn(C)c(=O)c1)=O)C2 c1(C(=O)NCC(CNC(C2C(C)CN(C)C2)=O)(C)C)coc2cc(O)ccc12 C(=O)(C1COc2ccc(F)cc21)NCC12CCC(CN(C(C=CCC)=O)C1)C2 C1(N(C(C2CC2(C)C)=O)CC)CCN(C(=O)CCc2ccc(O)nc2)CC1 n1(CC)ncc(I)c1C(=O)NC(c1ccc(Br)cc1)CC(=O)O c1(C(=O)NC23CC(CNC(COC(CC)(C)C)=O)(C2)C3)cnc(O)c(F)c1 C(C(CNC(C1CCC(=O)N(CCOC)C1)=O)C(F)(F)F)NC(C(CC)(F)F)=O N1(C(CSCCCC)=O)CC2CC(NC(c3ccns3)=O)C(C2)C1 c1(C(c2nnnn2C2CCC2)NCCNS(NC)(=O)=O)c(C)n[nH]c1C Cc1ncc(C(=O)N(CCC(C)NC(=O)C(C)C(C)O)C)cc1C#N C1(C(=O)NC2C(C(=O)NCC(N)=O)CCOC2)CCCC12CCC2 C(C)(C(=O)NCC1CCCN1C(c1cn(-c2cccnc2)nn1)=O)(C1CC1)OC C(=O)(C#CC1CCOC1)NC(C)(C)CCCCNC(=O)CC1(C)CCOC1 C1(c2cn(C(C)CNC(=O)C(C(C)C)n3cnnn3)nn2)(COC)CCOCC1 C1(CC)C(NC(=O)COC(F)(F)C(F)(F)F)CCN1C(C1CCC(OC)C1)=O CCC(C)(C)C(=O)NCCCOC1CCN(C(c2cn(CC3CC3)nn2)=O)CC1 CCC(CC(=O)N(C(CNC(C1CCN(C2CC2)C1=O)=O)CC)C)C1CCC1 c1(C(=O)NC2(CO)CN(C(CSCc3ccc(C)cc3)=O)C2)cc(N)c(Cl)cn1 C(=O)(C(C)(C)C(=O)N1CCCC(C2CCCN2C(c2cc(Cl)ccc2Cl)=O)C1)NC CC(CC(C)NC(=O)CSC(F)(F)F)NC(C1(C)CC1(F)F)=O C(=O)(C(=O)N=S(C)(C)=O)NC(CC1CC(C)(C)NC1=O)C1CC1 c1(OC)ccc(C(C)C(=O)N2CCCn3cc(nn3)C2)cc1.C1(CO)CCCC1 Cc1cc(CCC(=O)N(CCCCNC(=O)C(=C2CCCCC2)F)C)cc(C)c1 C(=O)(CCCn1cc(C2(NC(C3(C(F)F)CC(O)C3)=O)CCC2)nn1)OC C1(NC(=O)NC(C)C(=O)NCc2cccs2)CC2(C1)CC2F C#Cc1ccc(C2CC2C(=O)NCC2(O)CN(C(C3(C(=O)NC)CC3)=O)C2)cc1 C1(NC(C(c2cccc(C)c2)C)=O)CC2CN(C(C3COCCN3C)=O)CC2C1 C1(NC(C2CCCC2O)=O)CC1C1CCCN(C(C2CC3CCC(C2)S3)=O)C1 C=CCC(CNC(C1(c2ccccc2)CC1)=O)C(=O)NCC(C)OC C1(C(=O)NC2CCCC2N(C)C)(CC)CCN(C(=O)COCC(C)(C)C)CC1 CC(CC(F)F)CS(=O)(=O)NCc1cn(C(C)(C)C)c(=O)nc1O CC(O)C(F)(F)C(=O)NCCCNC(C1(C#N)CCCO1)=O N1(C(C(=O)Nc2cc(C)c(C)nc2)=O)CC2CC(C1)C(N)C2CO N1(C(c2ccc(OC)cc2)=O)CCC2CC1CN2C(=O)CCCC(C)=O c1(C(=O)NC2CN(C(COCC)=O)CC2(C)C)cc2c(cc1N)CCCC2 C1(CC(=O)NCCCCSCC)CCCN(C(=O)CC(=O)OC(C)(C)C)CC1 C12(CNC(C3(CC=C)CCCN3C(=O)CCCC3CCC3)=O)COC(C1)C(O)C2 CC1(NC(c2cnc(O)o2)=O)CCCCC1C(N1CCC1CF)=O C(C)(C)(CC(C)N=c1[nH]c2c(c(=NCc3csc(O)n3)[nH]1)CSC2)OC C(=O)(C1=CCCS1)N(C1CCCC1)CCCNC(C(C)Sc1ccccn1)=O CCCCC(CC(=O)NCC1(C(=O)OC)CC1)NC(=O)CN(C)C(N)=O C1(CN(C)C(C2CC2C2CC2)=O)CN(C(c2cccc(=O)o2)=O)CCO1 N1(C(COCC(=O)OC)=O)CCCC(O)(CNC(=O)CCc2ccccn2)CC1 c1(OC)ccnc(OC)c1C(N1CCC(NC(C2CCC(C(N)=O)O2)=O)CC1)=O Cc1nc(C#N)ccc1C(N1CCC(NC(C2CC23CC3)=O)C(C)(C)C1)=O c1(CC)cccc(C(=O)NC2CCN(C(C3CN(CC)CCO3)=O)C2CC)c1F Cc1cc(CC(=O)NC(C)(C)CN(C)C(c2ncoc2Br)=O)no1 N1(C(C=CC(=O)NC2CC2)=O)CC2=C(C1)CN(C(=O)CNc1nccs1)C2 c1(C(=O)NCCCCC(C)NC(C2OCCN(C)C2=O)=O)ncn2c1CCCC2 c1(C(N2CCC(C)(CNC(=O)Cn3nnnc3C3CC3)C2)=O)cc(F)ccc1F N1(C(CCC=C)=O)CC(CO)C2(CCN(C(=O)CC3CCCS3(=O)=O)CC2)C1 CCCS(=O)(=O)C(C)C(=O)N1CC=CC1CNC(c1cc2nc(C)ccc2o1)=O CS(=O)(=O)C1CC(C(=O)NC(CNC(=O)CCc2cscn2)CO)C1 C(=O)(C(C)C(C)NC(=O)Cc1ncccc1F)NCc1nnn(CC)n1 C1(ONC(C2C(NC(=O)CC3CCC3)CCC2)=O)CCC(O)C1O C(=O)(C(F)CC(C)(C)C)N(CC(N1CCOC(CCF)C1)=O)CCC c1(CS(=O)Cc2ccccn2)ccc2c(c1)OCC2 N1(C(Cc2c(C)con2)=O)CCN(C(=O)Cc2cc(F)cc(F)c2)C2CCC12 c1(NC(CC2CC(NC(c3nccc(C)c3)=O)C2)=O)cc(F)c(F)c(F)c1Br Cc1cc(=NC(=O)C(=O)NCC2(C)CCN(C(C3CCCC4CC34)=O)C2)[nH]o1 CN=c1nc(N2CC3CC3C2)[nH]c(=NCC(F)F)[nH]1.C1CC(=O)N1C(=O)C(Cl)(Cl)Cl CCCC(C(=O)N1CCC(N(CC(C)C)C(c2ocnc2CC)=O)CC1)C(C)C c1(C(=O)NCC2C(NC(C(C(C)C)F)=O)CCC2)ncc(C(F)(F)F)cc1Cl C12(CNC(c3nc(C)sc3C)=O)CN(C(=O)Cn3cccn3)CC1(C(F)(F)F)C2 C1(N(C(C(CC)n2ccc(C3CC3)n2)=O)CC)CCN(C(c2ccc(C)s2)=O)CC1 C12(C(CNC(c3n[nH]cc3Cl)=O)NC(Cc3ccc(C)s3)=O)CCC(CC1)C2 N1(Cc2cccc(NC(=O)CCOC(F)(F)F)c2)CCS(=O)(=O)CC1 C(=O)(C#CC1CCC1)N1CC(CCNC(=O)C(C)NC(C)=O)(OC)C1 C1(NC(CCC(N)=O)=O)CN(C(c2snc(Cl)c2Cl)=O)CC(F)(F)C1 C1(CNC(C(C)O)=O)CCCCN(C(c2cc(-c3ccc(O)cc3)[nH]n2)=O)C1 C(CC(=O)NCc1cccc(CO)c1)(C(C)OC)NC(C(CC)SC)=O C1(CNC(c2c(COC)noc2)=O)CC(F)(F)CN1C(=O)CCn1cc(C)cn1 c1(C(=O)NCC(CC)NC(=O)CN(C)CC)cccc(-c2cnn(C)c2)n1 c1(C(=O)NC(C2CCCN2C(=O)C=Cc2cccc(Cl)c2)C)nnc(O)nc1O N1(C(COC)=O)CC2CCC1C1CN(Cc3ccccc3[N+](=O)[O-])CC21 C1(NC(C2C(=C)C2)=O)CC2CCC1CN(C(c1c(C(F)(F)F)cc[nH]c1=N)=O)C2 N1(C(CCc2ccc(C)s2)=O)CC(C(=O)O)C2(CCC2)C1 C1(CNC(c2sc(Br)nc2Cl)c2n(CCOC)nnn2)CCS(=O)(=O)C1 c1(C(=O)NCC(C)N(C(=O)CC(C)SC)CC)cnc(O)c(C(C)=NO)c1 c1(CC)cc(-c2nc(C(C)C3CC3)nn2CCC(F)(F)F)ccc1Br c1(C(N(CCCN(C(CC(CC)C)=O)C)C)=O)nc(C)ccc1C c1(OC)ccc(C(C)(C)CNCC(N)=O)cc1.C1(N(C)C)CCCCN1C1CC1 c1(SCC(N2CCN(C(c3cc(OC)no3)=O)CC2)=O)cc(C)ccc1C C1(NC(C(C)Cc2cnc[nH]2)=O)CN(C(c2ccccc2F)=O)CC2(CCC2)C1 O=C(O)C#CC(=O)NC1CCC(C(N2CCCC(CO)C2)=O)CC1 Cc1cc(CNC2CCN(C(c3ccccc3F)=O)C2)c(O)c(Br)c1 N1(C(C2(COC)CN(C(=O)C(C)c3ccco3)C2)=O)CCS(=O)(=O)CC1 N1(C(c2cn(CCCC)nn2)=O)CC(NC(=O)Cc2ccc(C)s2)C(C)C1 n1(CCC(N2CC(C)(NC(c3c(C)cc(C)o3)=O)C2)=O)nc(O)c2c1CCCC2 N1(C2CN(C(Cc3c(C)n[nH]c3)=O)C2)CC(NC(C2CCC(=O)NC2)=O)CC1=O C#Cc1cccc(C(N2CC(NC(=O)Cc3ccsc3)C(CCC)C2)=O)c1F C#Cc1ccc(Br)c(C(=O)NCC2CN(C(=O)C(C)CC(=C)C)C2)c1 c1(C(=O)NC(C)(CNC(=O)CCn2cnnn2)C2CC2)cc2cnc(Cl)cc2s1 c1(C23CC(CC)(C2)C3)nc(CCSC)nn1C1CCSC1 c1(C(=O)NC(CC)CN(C(=O)CCc2c(C)noc2Cl)C)nccc(Cl)c1C c12nnc(n1CCSCCO)N1CCC(CC1)CN2C(C)C.C=CCOC N1(C(C(c2ccccc2F)OC)=O)CC=CC(NC(=O)C=C2CCN(C)CC2)C1 C(=O)(C1=C(F)CN(C(=O)C(C)CCCC(C)C)CC1)NCc1cnc(C)o1 N1(C(C2(CC=C)CCOC2)=O)CC(O)CC1C(=O)NC1CC(C)(CO)C1 Cc1nc(CCC(=O)NCC2(O)CN(C(=O)Cc3c(C)cnn3C)C2)oc1C N1(C(CCC(C)=O)=O)CCCC(F)(CNC(=O)C(C)Sc2ccccn2)C1 N1(C(c2c(C)cn(C)c2)=O)CCN(C(=O)CN2CCOC2=O)CC1C C1(N(C(=O)CC2CS(=O)(=O)C2)C)CCCC(NC(c2coc(C(C)(C)C)n2)=O)C1 CCCS(=O)(=O)C(C)C(=O)N(C)CC1CCN(C(=O)Cc2cc(C)sc2C)C1 N1(C(c2nc(OC)oc2)=O)CCC2(C1)CN(C(c1c(C)n[nH]c1C)=O)CC(C)O2 C(c1cocn1)=CC(N1CC(CC(F)C(=O)C(N2CCC2C2CCCCC2)=O)C1)=O c1(CNC(C2C(C)C(=O)C2)=O)ccccc1CN(C(=O)COC1CCC1)C C1(N(C(C(c2cccs2)SC)=O)C)CCCN(C(=O)CC2(C(F)(F)F)CC2)C1 N1(C(C2CCN(C(CCNC(C)=O)=O)CC2O)=O)CC(C)N(C)C(C)C1 C(=O)(C1=CCCSC1)NC1C(NC(=O)CCOc2ccc(F)c(Cl)c2)C1 N1(CC(=O)OC)CCC(CNC(C2C3CCC(F)C23)=O)CC1 c1(CC)cccc2c(C(N3CCCC(N(CC(C)C)C(C)=O)C3)=O)c[nH]c12 N1(C(C2CN(S(=O)(=O)C(F)F)C2)=O)CC2(CC(NCc3cc(Cl)ccc3O)C2)C1 CCC(C#N)C(=O)NCc1cc(C(=O)NC2CCCCCC2)on1 c1(OC)ccc(F)c(C(C(=O)NC2CCCC2)N(C2CCCCC2)C)n1 Cc1ccc(C=CC(=O)NCc2c[nH]nc2C(=O)NCCc2nccn2C)o1 C1(C)(N(C)CC)CCN(C(=O)CC2CCCN(C(=O)C(C)C3CC3)C2)C1 C1(C(=O)NCCCCCNC(C(C)(C)c2cccs2)=O)CCCC(C2CC2)O1 c1(NC(C(CC#C)(C)NC(C2CC3(CCC3O)C2)=O)=O)ccc2cnccc2c1 C=CC1CN(C(=O)COCCCC(C)C)CC1NC(=O)Cc1ccc(F)cc1Cl CC1CN(C(C2(S(C)(=O)=O)CCC2)=O)CC1(C)CNC(=O)CN(C)C1CC1 C1(NC(C(CN(CC)CC)F)=O)CCN(C(=O)Cn2ncnn2)C(C)C1 C1(CNC(c2ncn(C(C)C)c2)=O)COCCN1C(c1cccc(Br)c1)=O Cc1cc(C(=O)NCC2(NC(C3C(C)(C)C3(C)C)=O)CCCCC2C)nc(O)n1 Nc1cc(C(=O)NCC2CCCC(NC(=O)CCC3CCOCC3)C2)ccc1Cl CC1CC1C1CC1C(=O)COC(=O)C(F)CC1CC(F)(F)C1 N1(C(C2C(C)C2)=O)CCOCC1CNC(C1(C(C)(F)F)CCC1)=O C1(N(C(CCCOC)=O)C)CCN(C(c2cnn(C)n2)=O)CC1C N1(C(C2(SC)CN(C(C3CC4CCC3CC4)=O)C2)=O)CCCC(C(N)=O)(CCC)C1 C1(NC(c2cc(C)ncc2)=O)CCCC(C(=O)NOC2CCN(C)CC2)CC1 CC1CC=C(C(=O)NCCC2(CNC(C3CCSC(C)C3)=O)CC2)CC1 c1(CCC(=O)NCC2(NC(COC(C)C)=O)CCCC2)ccccc1C(F)(F)F CC1CCC(NC(c2coc(C3CC3)n2)=O)CN1C(=O)CC1OCCO1 N1(C(c2c(C)ncc(C)c2)=O)CCOC2(CCN(C(=O)CC3(O)CCC3)CC2)C1 Cc1cc(C(N2CCOCC2CNC(=O)CSCC(C)C)=O)c(N)c(Cl)n1 c1(OC)c(F)ccc(F)c1C(N1CCN(C(C2CC2C2CC2C)=O)C(C)C1)=O c1(CNCCN(C2CCN(C)CC2)C(C2CC(O)CN2C)=O)ccc(C)cc1.CO c1(OC)c(C)cc(C(N2CCC(NC(c3scnc3Cl)=O)C2)=O)cc1C c1(-n2c(CN(C)C)nc(CC(CC)C)n2)ccc2c(=O)[nH]ccc2c1 N1(C(c2cc(CC)sn2)=O)CCCOC(CNC(c2nccnc2C(N)=O)=O)C1 C(=O)(CCCC(F)F)N1C(CN(C(C(n2ccc(C)n2)C)=O)C)CCC1 N1(C(C(CC)OC)=O)CCCC(C)(C)C1CNC(C1CC2C=CC1CC2)=O CC(C)C(CCNC(=O)CC(O)c1cnc[nH]1)NC(=O)CCCC1CC1 c1(C(=O)NC(C(=O)NC(CCC)C2CC2)c2ccco2)cnn2c1CCC2 c1(CSCC)ccccc1CC(=O)N(CC(O)CNC(=O)C(F)n1cccn1)C CCC(CCCC(=O)N1CC(O)C(N=[N+]=[N-])C1)NC(=O)CSC C1(C(N(CCN(C(=O)Cn2cc([N+](=O)[O-])cn2)C)C)=O)C2CCC(C2)S1(=O)=O N1(C(COC2CCN(C(=O)Cn3cccc3)C2)=O)CC(F)(F)C1C1CC1 Cc1c(C(=O)NC2CCCN(C(=O)C3CC3)C2C)cccc1C(F)(F)F C1(C(C)NC(CCN(C)CC)=O)CN(C(=O)C=CCN2CCCC2)CCO1 c1(C(C(N2CCC(NC(CN(CC)CC)=O)C2)=O)C)ccc(F)cc1 C1(NC(C(=C(C)C2CC2)F)=O)CCC(NC(=O)Cc2ccc(C3CC3)cc2)CC1 C1(NC(=O)Cc2ccc(Cl)cn2)CC2CC1CN(C(=O)CC1CCOC1)C2 N1(C(C(F)OC)=O)CC(NC(C2C=CC=CC=C2)=O)CC12CCCC2 c1(C(N(CCNC(C2CN(C(N)=O)C2)=O)CC)=O)cc(Cl)c(F)cc1N c1(C(=O)NC2CC(C)(NC(=O)CC(=O)NCC3CC3)C2)cnn2c1OCC(F)C2 C(CCCCCCO)NC(C(Cn1cccn1)NC(c1cc(OC)ns1)=O)=O S(=O)(=O)(c1[nH]c(=NCCC(N)=O)ccc1Br)C(N1CCC(c2cccc(F)c2)C1)C N1(C(c2c(Cl)cn(C)n2)=O)CCC2(CCCN(C(=O)CCc3ncnn3C)C2)C1 c1(CCC(=O)NCC2OCC(CC(=O)O)C2)ccc(F)c(F)c1F C(=O)(CCN(OC)C(=O)Cc1cccc(C#N)c1)NC1C(OCC)COC1 N1(CC)CCCC(C(=O)NC2(CO)CN(C(=O)CNC(=O)C(F)(F)F)C2)C1 CC(C(C)N(C)C(=O)NCc1ccc(Cl)cc1Br)S(C)(=O)=O c1(C(N2C(C3CCN(C(c4nc(O)n[nH]4)=O)C3)CCC2)=O)c(Cl)nsc1Cl C(=O)(C(C)(O)CC(C)C)NC1CCN(C(C(CCC)N(C)C)=O)CC1OC c1(-n2ncc(CNCC3C(C(=O)OC)CCO3)c2)cccc2ccccc12 Nc1cc(F)c(Cl)cc1C(N1CC2C(NC(C3CCCS3(=O)=O)=O)C2C1)=O C1(C(=O)NCc2ncc[nH]c2=O)CCC(C2CCCCC2)CN1 c1(C(=O)NC2CC3(CN(C(CC(C=C)(C)C)=O)C3)OC2)cc2cc(Cl)cnc2o1 c1(C(=O)NC(C(C(C)C)C)CNC(c2cnsc2)=O)cccc2nc(Cl)cn12 C1(NC(Cc2nc(C)sc2C)=O)CN(C(=O)C(C)n2ccnc2)CCC1O N1(c2nc(C)c(F)cn2)CCC2(CC1)CC(C(=O)N=c1cco[nH]1)CO2 Cc1cc(C(=O)NC(C2(CNC(C3(F)CCCOC3)=O)CC2)C)ccn1 C1(NC(c2cnc(N(C)C)nc2)=O)CN(C(C2CC2(C)C)=O)CCC1CO N1(C(CCC=CC)=O)CC(NC(=O)Cc2ccc3c(c2)CC3)CC(C)(C)C1 N1(C(C(n2ccc(C)n2)C)=O)CCCC(CN(C)C(c2c(Cl)cnn2C)=O)C1 c1(OC)cncc(C(=O)NCC=CCNC(=O)CCCC2CC2C)c1C CCN=C(NCCCCc1cccc(NC(C)=O)c1)NCc1ncc(C)s1 N1(C(Cc2nnc(C)s2)=O)CCCC2(CCCCC2NC(=O)C2=NOC(C)C2)C1 N1(C(C(C)C)=O)CCCCC1C1CCCN1C(c1c[nH]c(=O)c2ccnn12)=O C1(C(=O)NCCNC(c2cc(F)cnc2O)=O)CC2(CCCCO2)C1 C=CC(CC)CC(=O)N1CCCC1CN(c1ncc(F)cn1)C NS(=O)(=O)c1cc(C(=O)Nc2ccc3nonc3c2)c(F)cc1Cl CCC(C)(C)C(O)C(=O)NC(c1ccccc1)CNC(c1ccc(N)cc1C)=O C1(C(=O)NC(C2CCCN2C(c2cc(C3CCC3)[nH]n2)=O)C)CCC(F)(F)C1 c1(C(=O)NC(CNC(CCC(=O)NCCC)=O)C(C)C)cc(C)cc2cn[nH]c12 C1(C#N)(C(=O)NCC(C)NC(C2C(CN=[N+]=[N-])C2(C)C)=O)CCOCC1 C(CC(CC)(CC)NC(C1CN(c2nncs2)C1)=O)NC(C(C=C)O)=O Cc1cn2c(n1)C(C(=O)N1CCC(C)(NC(=O)C(C(C)C)C(C)C)C1)CCC2 c1(C(C)(F)F)ccc(C(N2CCN(C(c3ccnnc3)=O)CC2)=O)cc1 C1(C)(C(=O)NC2C(C)CN(C(c3ccno3)=O)CC2)CC2CCC(C1)S2 c1(C(=O)NCC2(NC(CCCC=C)=O)CCCCC2)cn2c(n1)SCC2 N1(C(c2cnc(OC)s2)=O)CC2CCC2(CCNC(C2(C(N)=O)CC2)=O)C1 c1(C(C(=O)NC2CCCCC2)N(C(c2cc(C)c(C)s2)C)C)cccc(F)c1Br C1(C)(CCNC(C2(CC)CC2)=O)CCN(C(=O)CCOc2ccc(Cl)cc2)C1 C(=O)(CC(C)C1CCCO1)N(CCN(C(=O)Cc1csc(Br)c1)C(C)C)C C(CC)(C(=O)NCCCCCNC(c1sccc1F)=O)OCC CCCCC(O)C(=O)NC(CNC(=O)CCCc1ccc(F)c(F)c1)CCOC N(C(=NCCc1ccc(OC(F)F)cc1)NC1CCCC1)Cc1cccc(C)n1 C=C1Cn2c(C(=O)NC(CN(C)C(C3CC4CCC3C4)=O)(CO)CO)nnc2S1 CC1CCCN(C(=O)C(=O)NCC2(O)CN(C3CN(C)CC3C(F)(F)F)C2)C1 c1(C(=O)NCCC(C)N(C(Cc2c(C)ccc(C)c2)=O)C)ccc(N)c(Cl)c1O C=C1CC2(C1)CC(C(=O)N(CCCOCCNC(c1cnc(O)cc1C)=O)C)C2 N1(C(C2C(C(C)C)OCC2)=O)CC(C(=O)NC(CCO)C(C)(C)C)C2(CCC2)C1 CC1CCN(C(=O)Cc2cc(Br)cs2)CC1CNC(C1OCCO1)=O Cc1cn2cccc(C(=O)N(C)CCN(C(=O)CCNC(=O)CO)C)c2n1 N1(C(C(CCCCC)O)=O)CC2CN(C(c3cc(OC)no3)=O)CC2(C)C1 N1(C(CC(CCC)(C)C)=O)CCC2(CNC(c3ncc(C)cn3)=O)CCCCC12 C1(C(N2C(C(N3CC(O)(CCC)C3)=O)C=CC2)=O)CSCC(=O)N1 CC(C)CC(C(=O)NC(C)C(C)(C)C(=O)NCC1CC(=O)N(C)C1=O)C(C)C CC1CC(NC(=O)OC(C)(C)C)CCN1C(c1cnc(N)c(N)c1)=O Cc1onc(Br)c1C(c1nnnn1CC(F)F)NCCCCOC(=N)O C1(C)(C(N2CCC(C3N(C(CCC#CC)=O)CCC3)C2)=O)CCC(F)(F)CC1 c1(C(=O)NC(C)C(CO)NC(=O)Cc2ccccc2O)cccnc1O c1(C(=O)NCCOCCC(=O)N(C(C)C(C)C)CC)cc(F)c[nH]1 C1(C(N2CC(C)(NC(C3CC3C(F)F)=O)C2)=O)COc2ccc(F)cc2C1 Cc1ccnc(C(N2CCC2(C)CC(=O)NCC(C)(O)CCO)=O)c1N N1(C(c2csc(Cl)c2)C(=O)NCCOCCO)CCC2NC(=O)NCC2C1 c1(C(CN(C(=O)C(CNC(=O)CC2(O)CCCC2)N(C)C)C)O)ccccc1 Cc1ncncc1C(N1CCC(N(C(=O)C(N2CCSCC2)C)CC2CC2)C1)=O c1(C(=O)NC(C)CNC(=O)C(C)S(C)(=O)=O)nc2n(c1Cl)CCCC2 c1([SH](CC(=O)NCC2(OC)CN(C(C(C)OCC)=O)C2)C2CC2)ccc(F)c(F)c1 c1(C(=O)NC2C(NC(C(CC=C)CC=C)=O)C2)cnc2c(c1)CCCC2 n1(CC(N2CCCC(N(C(C(C=C)OC)=O)C)CC2)=O)cc(OC)c(=O)cc1C c1(C(=O)NCC(CC)(CC)NC(c2cc(C)n(CCO)n2)=O)c(C)cccc1Cl N1(C(C(C2CCC(=O)N2)C)=O)CC(C(=O)NOC2CCOC2)C(C2CC2)C1 C1(NC(CC2CC(=C)C2)=O)CCC(O)CN(C(c2ccn3nnnc3c2)=O)C1 CC1(C(=O)NCC2CCN(C(c3ccc(CS(N)(=O)=O)cc3)=O)C2)CCC(=O)C1 N1(C(c2c(CC)cno2)=O)CCN(C(=O)CC2CCCOCC2)CC1CCOC N1(C(C=C(C)C)=O)C2CCC1CN(C(c1nn(-c3ccc(F)cc3)cc1C)=O)C2 c1(C(=O)NC2CC(CNC(C34OC(C)(C)C(C3)C4)=O)C2)ccc(Cl)c(N)c1Cl c1(OCC)cccc(CC(N2CCC(C)(NC(C3CCS3(=O)=O)=O)C2)=O)n1 C1(CC(=O)NCC(C)CNC(C2CNC(=O)O2)=O)CCC(=O)C1C Cc1nc2cc(C(=O)NCCC3CCN(C(C4CCCN4C(C)C)=O)C3)[nH]c2s1 CN1CCN(C(C2CCC(NC(=O)Cn3cnc(C#N)n3)CC2)=O)CC1(C)C N1(C(C(CNC(CCCC=C)=O)N(C)C)=O)CCC(C)(C#N)C1 c1(C(CC)C)cc(C(N2CCC2CNC(c2ccnn2C(F)F)=O)=O)on1 c1(C(C)(C(=O)N2CCC(CNC(c3nc(Cl)cs3)=O)C2)N(C)C)ccccc1Cl N1(C(C=CS(C)=O)=O)CCC2(CCC(CNC(c3coc(CO)c3)=O)CC2)CC1 c1(C(=O)NCC2CCCCN2Cc2cccc(Cl)c2F)nccc2[nH]ccc12 c1(C(c2n(CC=C)nnn2)NCCC2(COC)CC2)ccncc1C Cc1cccc(C)c1C1(C(=O)NC2CN(C(c3cc(C)c(Br)o3)=O)CC2C)CC1 c1(C(N2C(CNC(=O)NC)CCCC2)=O)ccc2occc2n1 N1(Cc2ccc(CN)cc2F)CCCCC2C1CCCN2C1CC1 C1(C(N(CCC(=O)OC)C2CC2)=O)CCCCN1C(=O)C(=Cc1ccco1)C C(=O)(C1=CCCN(Cc2cccc(CC(=O)O)c2)C1)Nc1ccc(OC)cc1C c1(C(=O)OCC)ccc(C(=O)NC2CC2NC(=O)CC2C(=O)NN=C2C)cc1 c1(C(c2nnnn2C)Nc2cc(C)c(Cl)cc2)ncc2ccccn12 C1(CC(=O)NC(C(C)NC(C2(C=C)CCCC2)=O)C)CC(C)(C)C(=O)N1 Cc1ccn2ncc(C(=O)NC3C4CC3N(C(=O)CCCN(C)N=O)C4)c2n1 C#CCCC(C(=O)NCCCCOCC)NC(=O)C=Cc1ccco1 c1(NC(C2CC(OC)CN2C(=O)C(C)Cc2ccco2)=O)cc(Cl)ccc1CO C(CCC(C)CC(=O)N(CCC(C(C)C)NC(C12CC(F)(C1)C2)=O)C)=C(C)C c1(C(N2CCN(C(CP(C)(C)=O)=O)C3(C2)CC3)=O)cnc2nc(Cl)ccc2c1 c1(OCC)cnc(C(=O)N(CC(C)(C)CNC(=O)C(C)OCC)CC)cn1 c1(NC(C2C3(CN(C(CC(C)C)=O)C3)C2)=O)cn2nc(Cl)ccc2n1 C(C(C)C)(C(O)C(=O)NC1C=CC(CC(N2CC(OC)CC23CCC3)=O)C1)OC CC1CCN(C(=O)C(C)Cn2ccnc2)CCN1C(=O)CC1(O)CCOC1 c1(OC)cc(Br)cc(F)c1C(=O)OC1(C(F)(F)F)CN(C(C2CCC(=O)N2)=O)C1 c1(C(=O)NCC2CCC(CCC)CC2)cc(Cl)ccc1Br n1(CCCSC)nnnc1C(c1n[nH]cc1C)NC(C1CCCC1)C N1(C(C(C(=O)OCC)CC)=O)CC2CCC(C1)C(NC(=O)C=CC(F)(F)F)C2 c1(CC)cc(C(=O)NC(c2nocc2C(=O)NC(C)CC2CCCO2)C)no1 c1(C(C)OC)noc(CCC(=O)NCCC2CC(NC(c3ccco3)=O)C2)n1 CC1CCCN(C(=O)C(=O)N(CCn2cc(C(C)(C)F)nn2)CCO)C1 c1(C(=O)NC2CN(C(CC(C)C)=O)CC(F)(F)C2)cc2n[nH]cc2cc1Cl CCCCC(C(=O)N1CCCC1CNC(c1cccc(C)n1)=O)ON=C(C)C C1(C)(CNC(C2N(C(C)=O)CCC2)=O)CCN(C(C23CC(C#N)(C2)C3)=O)C1 N1(C(c2c(C)csn2)=O)CC(C2CCN(C(=O)CC3CCCC34CC4)CC2)C1 CC(CCNC(=O)Cc1cccs1)CCNC(c1cnoc1-c1ccoc1)=O C(CC(C)(C)NC(=O)CCc1ccoc1)=CC(=O)NC1(CSC)CCC1 c1(NC(C2OCCN(C(Cc3cccc(C)n3)=O)C2)=O)cccc(Cl)c1C c1(NC)ccc(Cl)c(C(=O)NC(C2CCOC2)CNC(=O)C#CC2CCC2)c1 C1(C(C)(C)CNC(=O)Cc2cccnc2)CCCCN1C(c1ccnc(O)c1)=O c1(C(=O)NC2CCN(C(CC3CCC(=O)NC3)=O)C2)cc2[nH]ccc2cc1Cl CC1(C(=O)NCC(CO)NC(c2cnc(C3CC3)o2)=O)CCCCC1(F)F C1(C(=O)NCCCN(N2CCCC2CO)C(c2ccsc2)=O)CCC(F)CC1 c1(C(=O)NCCOCCOCCCNC(C(C)CO)=O)ncnc2c1CCCC2 C1(C(=O)NC2C(NC(C(C#C)(C)C)=O)COCC2)CCC=CCCC1 c1(OC)cccc(NC(C2CC2NC(c2cc(Br)cc(F)c2O)=O)=O)c1C#N c1(NC(C2CCCN(C(=O)CC3CCC(F)(F)C3)C2)C)ccc2ncnn2c1 N1(C(C(CC)C#N)=O)CC2OCCN(C(c3cccs3)=O)C2C1 C(=O)(CP(C)(C)=O)N1C(Cc2cn(C(C(C)O)C)nn2)CCC1 O=C(CCCCNC(=O)COc1ccccc1)NCC1CC(F)C1 N1(C(Cn2cc[n+](C)c2)=O)CC(OC)C(NC(c2csc(C(C)(C)C)n2)=O)C1 N1(C(c2cc(C)n(CC#C)c2C)=O)CC2CC1CN(C(c1ccn(CC)n1)=O)C2 C(CCCOC)(C(=O)NCc1cscc1C)NC(C(C(=O)OCC)F)=O C1(C(N(C)CCC2CCN(C(=O)Cc3ccoc3)CC2)=O)CC12CCOCC2 Cc1cc(=NC(C)c2nnc(CO)s2)[nH]c(=NCC2CC(F)(F)C(=O)N2)[nH]1 CCC(C)C(C(=O)N1CCC(O)(C(C)C)C1)N(C(=O)C=CCO)C c1(CC(N2CC(NC(C3C(CC)CCCC3)=O)C2)=O)ccc(Br)c(Cl)c1 N1(C(C(CCOC)OC)=O)CC2(CC(C(=O)NCCS(C)(=N)=O)CO2)C1 C1(C(N(C)CCOc2ccc(Br)cc2)=O)CC12CCN(CCS(C)(=O)=O)CC2 c1(C(C)C(=O)NC2CCCC2NC(C2CC(O)C2)=O)ccccc1[N+](=O)[O-] C1(NC(CC(=C=C)C)=O)CCN(C(=O)CCNC(=O)CC(C)C)CC(C)(C)C1 N1(C(CSC)=O)CCC2(CCC(NC(=O)COC3CCN(C)CC3)C2)CC1 C1(CC(=O)NCCCCC2C(C)C2)CCN(C)CC1.c12csc(n1)COC2=O.C C1(NC(c2c(C)scc2)=O)CS(=O)(=O)CC1NC(=O)CCCSC(C)(C)C CCCC(CC)C(=O)N1CCCC(CC(=O)N(CC(F)(F)Cl)C)C1 C(=O)(C1=CCCC1(C)C)N(C1CCCC(N(C)C(c2ccc(Cl)cc2)=O)C1)C c1(C(N(C2CC(NC(C(COC)NC(C)=O)=O)C2)C)=O)ccc2oc(O)nc2c1 C1(NC)CCN(C(c2cn(-c3cccnc3)nn2)C(=O)Nc2ccccc2)CC1 N1(C(CN(C)C(N)=O)=O)C2CCC1CN(CC(=O)NCCOC1(C)CCCC1)C2 Cc1ccc(F)c(OCCS(=O)(=O)NC2CC2)c1 C(=O)(C(C)CC(=O)NCC1CC1CC(=O)NCC1(CF)CC1)OC N1(C(C(C=C)OC)=O)CC(C2CCCN(C(c3[nH]nnc3C3CC3)=O)C2)C1 C1(C)(C(=O)NCCN(C)C(c2ccc(CO)c(F)c2)=O)CCNC(=O)C1 c1(NC(=O)NCc2ccc(Nc3ccc(F)c(O)c3)cc2)nc(Cl)c(Cl)cc1Cl C1(C(=O)NCC(C)CNC(c2cc(C(F)(F)F)n[nH]2)=O)C(F)(F)C12CC2 N1(C(CCCCC)=O)CC(CN(C(=O)CSCc2cccs2)C)C2(CC2)C1 C1(C(=O)NC2CCN(C(C3CCN(c4ccccc4)C3)=O)C2)CC2(CCC2)C1 c1(C(N2CCC(CC=C)(NC(C3CCSC3)=O)C2)=O)c(C)nc(C2CC2)nc1O c1(C(=O)NC(CC=C)CNC(c2ccc(Br)o2)=O)nc(C2CC2)ncc1Cl N1(C(c2c(CC)nn(C)c2)=O)CCC2CN(C(=O)Cc3cncn3C3CC3)C2C1 CC(C)CCC(=O)C(=O)NC1(C)CC(C(=O)N(C)Cc2cnn[nH]2)C1 C1(CNC(c2c(C)ccnn2)=O)CCCCN(C(c2ccccc2C(N)=O)=O)C1 CC1CN(C(c2cc(Cl)nnc2O)=O)C(C)CN1C(c1csc2ccncc12)=O c1(NC23CC(C(=O)NCc4ccc(OC)nc4)(C2)C3)ccc(C#N)cc1C C1(C(N(CCCNC(CC(C)C)=O)C)=O)CCC(NC(C2CSC2)=O)CC1 c1(C(=O)NCC#CC(=O)NCC2OCC(C)C2)cn(C)ccc1=O N1(C(C(C)N=[N+]=[N-])=O)CCCC12CCN(C(c1c[nH]nc1Cl)=O)CC2 N1(C(C(C(C)C)S)=O)CCc2nc(C(=O)N(CCO)C3CC3)ccc2C1 N1(C(C2(C(C)C)COC2)=O)C2CCC1CN(C(=O)CN1CCC(C)(C)C1)CC2 Cc1cc(C(N2CCC(NC(=O)CC3(N4CCCC4)CC3)C2(C)C)=O)cc(O)c1 C#Cc1cncc(C(=O)NC(C)(C(=O)NCCCOC(F)(F)F)C2CCC2)c1 c1(NC(C2CCN(C(C3(C)CCCO3)=O)C2)C)nc2ccc(O)cc2s1 C(CC(C)C)(C(=O)NCC1(n2ccnn2)CC1)NC(C(C)SC)=O c1(C(=O)NCC(CN(C(=O)CSC2CC2)CC)(C)C)cc(C)c(Cl)s1 n1(CC)ccc(C(=O)NCC2CCN(C(C3C(F)(F)C34CC4)=O)C2)cc1=O N=c1nc(C(F)F)[nH]c(=NC2CCCC(Nc3ncc(C(F)F)cn3)C2)[nH]1 Cc1noc(C)c1-c1cncc(F)c1.c12ccc(cc1)C(=O)COC(=O)CC2 CC(C(C)(C)C(=O)NCC1CCCO1)NC(=O)CNC(=O)NC1CC1 C1(N(C(C(C)SC)=O)C)CC2CCC(C1)N2C(c1c(-c2cccs2)noc1C)=O c1(CNC(c2cc(C)n(C)c2)=O)n[nH]c2c1CN(C(=O)COCC(C)(C)C)CC2 C1(NC(CCCN(C)C(c2cn[nH]c2)=O)=O)CC(C)(C)C12CC2 Cc1cc(C(=O)NCC(O)CCNC(=O)Cn2cccn2)c(F)c(Br)c1 C#Cc1ccccc1NC(C1CCCN1C(c1ccc(OC(F)(F)F)nc1)=O)=O C1(CNC(C2(CC(N3C(COC)CC(O)C3)=O)CCC2)=O)Cc2nccn2C1 C1(C(=O)NC2CC(CCNC(c3cc(C(C)C)on3)=O)C2)CCC(=O)N1C(C)C Cc1cc2ncnc(N3C4CCC3C(C)C(NC(C3(C)CC(C)C3)=O)C4)c2[nH]1 C1(CN(C(C2(CCOC)CCC2)=O)C)CCCN1C(=O)CC1(N(C)C)COC1 C1(C(=O)OCC)C2CC1CN(CC(C#N)C1CCOC1)C2 N1(C(c2cc(Cl)ccc2Sc2ccccc2)=O)CC2CCCN2c2ccccc21 C=CCC(C(=O)NC1(CCC(=O)N2CC(CC(N)=O)C2)CCC1)C(C)C C(=O)(C1=NN(C)C(=O)CC1)N1CC2CCC(NC(C(CCSC)(C)C)=O)(C1)C2 CC1(C(=O)NCC2CC3C=CC2O3)CCN(C(=O)CC2CCCC(=O)N2)C1 c1(C(=O)NCCOCCCNC(C2(C(N)=O)CC2)=O)ccnc(CO)c1 Cc1nn(C)c(C)c1OCC(=O)NCC(O)CCNC(=O)Cc1csc(S)n1 C1(NC(c2cocc2Br)=O)CN(C(=O)CCF)C2(CCCCCC2)C1 C1(C(C)(C)C)CCCN(C(c2cc(Br)co2)C(=O)NCc2ccccc2Cl)CC1 c1(C(N(C(C)CNC(c2ccco2)=O)C)=O)cccc(Cl)c1O C(=O)(NNC(=O)CN1CCCCC1c1ccccc1)c1ccc(C)cc1 C1(C(=O)NCC2CC(NC(=O)CC3NC(=O)NC3=O)C2)CC2CCCC(C1)C2 c1(-c2ccc(N3CCC(C(=O)NC(C=C)C)CC3)cn2)ccc(C#N)cc1OC N1(C(C(C)OCCC2CC2)=O)CCCCC1C1CCN(CCO)C1 Cc1ccc2ncc(C(N3CC(NC(c4cnc(Cl)cc4N)=O)C3)=O)n2c1 C#CC1(NC(C2(C)CCN(C(=O)C(C)n3ccnc3)C2)=O)CCC(C)CC1 C1(CC(=O)NC2CC(N(C(C(c3cccc(Cl)c3)CC)=O)C)C2)CCC(C)(C)C1 C(=O)(CCC(=O)c1ccc[nH]1)NC1C(NC(C(c2ccccc2)N(C)C)=O)CC1 c1(CNC(=O)Cc2sccc2C(F)F)ccc(Cl)cc1 c1(C(N2CCC(O)(CCNC(COCC#C)=O)C2)=O)cc(O)ncc1Br c1(-c2cn(C)nc2)cnn2c1CN(Cc1cc(F)ccc1Cl)CC2 CCCCC(O)C(C)C(=O)NC(C)C(C(=O)N1CCCOC(C)C1)C(C)C c1(C(N2C(CNC(CC(=C)Br)=O)CC2)=O)nnccc1C C1(CNC(C2CC(CNC(COC(CC)C)=O)C2)=O)CC(C)(C)CO1 N1(C(C=C(CCC)C)=O)CCN(C(=O)C(C)(C)COCCOC)CC1CCOC N1(C(C(CC=CCC)C)=O)CCCCCC(NC(=O)CCCC2CCCCC2)C1 C1(O)(C(C(=O)NC2(Cn3cccn3)CC=CC2)O)CCOCC1 C1(C(=O)NCC2CCN2C(=O)Cn2cnnn2)CC2(COCCO2)C1 CC(CC(C)(C)C)C(=O)N1CCCC1CN(c1ncc(I)cn1)C CCCC(C)CCNC(=O)COC1CCN(C(=O)CC2CCCC2)C1 C1(C(F)(F)F)(C(N(CC(O)CNC(=O)C(C)(C)CN(C)C)C)=O)CC2(CCC2)C1 c1(CC)nn(C)cc1C(=O)NCC1(NC(=O)C2=CCCO2)CCCC1 C1(C(N2CC3C(C(=O)NCC(C)(C)F)C3C2)=O)CC(=O)CC(=O)N1 c1(C(N(CCC(=O)N(CCCCC)C)CCO)=O)csc(=N)[nH]1 c1(C(c2n(C)nnn2)(C)NCCC2CC2)ccc(C2CCCCC2)cc1F CC(C(C)C(=O)NC1(C2CC2)CCC1)NC(=O)C=Cc1cn(C)nn1 CC(C)(C)CC(=O)N=c1ccn(-c2ccc(Br)cn2)[nH]1 N1(C(C2(COC)COC2)=O)CCOC(C(=O)N(C2CCCNC2=O)C)CC1 c1(CNC(c2n(CCC)nnn2)C(C)(C2CCCCC2)OC)nnn(C)c1C C1(NC(=O)COCC2CCC2)CCN(C(=O)C=Cc2ccsc2)CC1O C1(NC(=O)Nc2c(C)c(N(C)C)ccc2)C2CCC1(C)C2(C)C CC1(C)CC(NC(=O)Cc2ccno2)CN(C(=O)Cc2ccccc2[N+](=O)[O-])C1 S(=O)(=O)(c1ccsc1C(=O)NC(C)C(C)NC(=O)C1=COCCC1)NC C1(NC(c2cccc(NC(CC)=O)c2)=O)CC2(C1)CN(C(C1CCC(=O)O1)=O)C2 C1(CNC(c2c(CC)occ2)=O)CC(OC)CN1C(=O)CN1CC=CC1 c1(C(N2CC(NC(C(CCC)CC)=O)C(O)C2)=O)ccc2ncn(C3CC3)c2c1 c1(SC)cc(N2CC3CC2CN3C(C2CCCCS2(=O)=O)=O)nc(SC)n1 c1(-c2nc(NC(C(C3CCC3)OC)=O)sc2)ccc(C)cc1 Cc1cc(NC(C2CCC=CCCC2)=O)nc(Br)c1 C1(NC(c2ccc(CCC)[nH]2)=O)CN(C(=O)CCOCC)Cc2nccn2C1 C1(CC(=O)NC(C)(C)CF)CCCN1C(=O)CC1CC1 C(=O)(C1=CC2(CCOCC2)C1)NC(C)(CNC(C1(C2CC2)CCC1)=O)CO c1(N2CCCC(C)C2)cccc(S(=O)(=O)NC2CCC=C2Br)n1 N1(CC)CC(C)N(C(=O)CCNC(C2(OC)CC(C)(C)C2)=O)CC1C N1(C(CC2CCN(C(C)=O)CC2)=O)CCC2C(NC(C3CC34CCC4)=O)C2C1 c12cccc(F)c1C2.N1(c2ncc(C(=O)O)s2)CCOC(C2CCCCC2)C1 C1(NC(C(CCN(C)C)N(C)C)=O)CC2CCC1CN2C(C1CC(F)(CF)C1)=O N1(C(CC(C)OC)=O)CC(OC)C(NC(=O)CSc2nncs2)C1 c1(C(=O)NC(CNC(C(C)(C(C)C)NC(C)=O)=O)CO)oc(S(N)(=O)=O)cc1C c1(C(=O)NC)cc(C)[nH]c(=NCCCC(C)(C)NC(C2CCC(F)CC2)=O)n1 C1(CNC(=O)C=CCO)C2CN(C(c3ccnc(OC4CCC4)c3)=O)CC12 C(=O)(C(CCF)NC(=O)Cc1ccc(F)cc1)N(CC(=O)OC(C)(C)C)CC N1(CC#C)CCCOC(C(=O)NCCOC2CCCCCC2)C1 N1(c2ncc(C)cn2)CC2CC1CN2Cc1cc(C(F)(F)F)ccc1F c1(NC(C(C)c2ccco2)=O)cccc(C(=O)NCCSCc2ccncc2)c1 CCCC(C)CN(C)C(C1(N(C)C(c2cc(C(C)C)[nH]n2)=O)CC1)=O c1(OCC(N2C(C3(NC(C(C(C)C)C)=O)CC3)CCC2)=O)cc(F)ccc1F CCCCCCC(F)C(=O)NC(C)CNC(c1sc(CC)nc1C)=O n1(CC(=O)N(CC(C)CNC(=O)C(F)(F)c2nccs2)C)ncc(C#N)c1N c1(C(=O)NC2C(NC(C3C(NC(=O)OC(C)(C)C)C3)=O)COC2)cnc2sccn12 N#Cc1cccc(F)c1CC(N1CC(NC(C2CCCO2)=O)CC(F)C1)=O n1(CCSC)nnnc1C(c1cnc(Cl)s1)NC1CC(NC(N)=O)C1 S(=O)(=O)(c1ccc(NC2CCCCC2OC(F)(F)F)cc1Cl)NCC(C)C(F)F c1(OC)ccc(OC)c(CC(=O)NC2CCC2NC(C2C3CC4C(C3)C24)=O)c1 Cc1ccc(NC2CCOC(c3ccccc3)C2)nc1 Cc1cc(NC(=O)C(C)(C)C)sc1C(=O)NCC(C)NC(=O)C(C)(C)C1CCC1 C1(NC(C(C)O)=O)CCC2(CCN(C(=O)Cc3cnsc3)CC2)C1 C=C1Cn2c(C(=O)NC3CCCC(NC(=O)CCCn4ccnn4)C3)nnc2S1 C1(C(=O)NC2CCN(C(COCC)=O)C2C(C)(C)C)CC12CCC(C)(C)CC2 C1(C(=O)NCC(c2ccsc2)C)CCC(CN)O1 CCC(CC(=O)N1CCCC1CC1CCCC1)N(C)C(c1cc(C#N)cs1)=O c1(C(=O)NCC2CCCN(C(C3(C(CC)=O)CC3)=O)C2)coc(S(=O)(=O)NC)c1 C1(C(=O)NCC(CC)(CC)NC(c2nc(Cl)ccc2N)=O)CN2CCCN1CC2 N1(C(Cc2c(C)nc[nH]2)=O)CC2CC(NC(=O)CCn3cnnn3)CC1C2 N(C1c2ccccc2CC1C)C(c1ccc(OC)nc1Br)=O C(c1ccccc1F)=CCC(=O)NC(CN(C)C(c1cn(C)nn1)=O)(C)C C1(N(C(CC(=O)NCC#C)=O)CC)CCCN(C(=O)CCC(=O)NC(C)C)CC1 N1(C(Cc2c(C)ccs2)=O)CCN(C(=O)COC2CCOC2)C(C2CC2)C1 C1(NC(=O)CSC2CCOC2=O)CCCCC1NC(c1cnccc1Cl)=O c1(NC(C2CCOCC2F)=O)ccc(C#N)s1.C12CC1C(=O)NC2C Cc1cc(CN(C(C2(CNC(c3[nH]ccc3C)=O)CC2)=O)C)cc(F)c1 C12(C(N)=O)CCCC1(C(N1CC(NC(=O)CSCC3CCCO3)C1)=O)C2 CN1CCCC(CNC(=O)C=CCNC(C2C(C)(C)C2(C)C)=O)C1 Nc1cncnc1C(=O)NCC1(CO)CCN(C(=O)CN2CCNC(=O)C2)C1 c1(C(N2CC(CO)C3(CC3)C2)C(=O)NC(C)(C)C)ccc2ncccc2n1 N1(C(c2ccnn2CC(F)F)C(=O)NCCOC)CCC12CCN(C)C2 CC(C)CC(C(=O)N1CCCCC1CC(N1CC2CCC2(C)C1)=O)N(C)C CN1CCCC1(C)C(N1CC2C(CNC(c3cncc(-n4cccn4)n3)=O)C2C1)=O c1(OC)ncc(C(=O)NCCNC(=O)C(O)CCN(C)C)c(C(F)F)n1 C1(C(N(CCNC(=O)C(F)C2CC2)CC)=O)CC(C(=O)OC(C)(C)C)=NO1 N1(C(CC2(OC)CCOCC2)=O)CCC2CN(C(=O)CCc3cnc(C)o3)C2C1 C1(CC)CCCN(C(=O)CN2CCOCC2)C1C(=O)N(C)Cc1ccccc1C C1(OC)CC(O)CN(C(c2nnc(C)s2)C(=O)NCCCF)C1 Cc1nc(N)cnc1C(=O)NC1CCOCC1NC(=O)CCn1cccn1 CC1CN(C(C2(C#N)CC2)=O)CCCN1C(=O)CNC(=O)C1CC1 c1(CN2CCCC(CC(=O)NCc3ccncc3)C2)cc([N+](=O)[O-])c(O)cc1O c1(CCC(=O)NC(C2CCOC2)CNC(C=C(CC)CC)=O)nc(C2CC2)no1 C(=O)(C(CCOC)NC(=O)CCC1CC1(C)C)NCC1CC(=C)C1 c1(C(N2CCC(COC)(NC(=O)C=C(C)C(F)F)C2)=O)cc(C)n(C)c1C N1(C(C(C=C)OC)=O)CC(NC(C2CCCOCC2)=O)CC(C)C1 CC(N=c1[nH]nc(C(F)(F)F)s1)C1CCCN(C(C2CC2(F)F)=O)C1 C1(NC(CCc2nc(C)c(C)[nH]2)=O)CCC2(CCCN(C(=O)CC3CC3)C2)C1 c1(OCC=C)ccc([N+](=O)[O-])c(COC(=O)NC(CSC)CC)c1 C1(NC(c2c(C)c[nH]c2)=O)C2CC(NC(C3CS(=O)(=O)C3)=O)CC12 c1(C(C)C)ccc(CC(=O)NC2CC(NC(C34CC(C)C3C4)=O)C(O)C2)cc1F C(=O)(C(CCC(C)C)NC(C1CC(=O)C1)=O)NC(CCOCC)C C1(NC(CCC(=O)OC)=O)CN(C(C2CC23CCCCC3)=O)CC(C)(C)C1 C1(CNC(c2nn[nH]c2Cl)=O)CN(C(=O)Cc2cnsc2)CCO1 C1(C(N(CC(COC)C)C)=O)CCN(C(c2cc(OC)cs2)=O)C1(C)C c1(C(=O)NCCN(C(C2C(CC)OCC2)=O)C2CC2)cccc(F)c1F N1(C(c2ncc(-c3n(C)ncc3)nc2)=O)CCc2ccc(F)cc2C1 Cc1cc(F)c(N)cc1C(=O)NC(CO)C(C)NC(c1ccc(Cl)c(F)c1)=O c1(CC)nnc(N(CC(C)CNC(=O)C=CC2CCOC2)C)o1 C1(CNC(C)=O)CCCCN1C(=O)CC1CCCC(C2CC2)O1 C1(C)(NC(CCNC(=O)NC)=O)CCN(C(C2CCCCC2)=O)CC1 c1(C(N2CC(C)(NC(=O)CCc3csc(=N)[nH]3)C2)=O)cccn2nnnc12 N1(Cc2ccc(OCCC)nc2OC)C(=O)NC(C2CCCO2)C1=O c1(SCC)ccc(C(=O)N(CCCN(C(=O)CC2CSC2)C)C)cn1 C(=O)(CC1OCc2ccccc21)NC1CC(CNC(c2n[nH]c(C)c2Cl)=O)C1 Cn1cc(C(=O)NCC2(F)CCN(C(=O)C=Cc3cnc[nH]3)CC2)c(O)nc1=O C(=O)(C(C)(C)C(=O)NC(CC(F)F)C(=O)NC1C2CCCC12)N(C)C C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(NC(C(CSC)OC)=O)C2(C1)CC2 S(=O)(=O)(c1ccc(NCc2cc(Cl)ccn2)nc1)NC(c1n[nH]c(=N)s1)C S(=O)(=O)(c1ccc(F)c(F)c1)N(C1C2CCC1CNC2)Cc1ccc(C)cn1 C12(NC(C(c3cccc(F)n3)C)=O)CCC(C1)N(C(=O)CC1CCOCC1)C2 CCC(C(=O)NCCCCCNC(c1cc(F)ccc1OC)=O)C(C)O c1(C(=O)NCC(C)SC)cc(=NC(=O)CNC(=O)C(C)(C)C)[nH]n1C N1(C(C(C(CC)O)(F)F)=O)Cc2ccccc2C(NC(=O)COC2CCCC2)C1 c1(C(N(CCNC(=O)C(F)(F)C2(O)CCC2)CC)=O)ccc(SC(F)(F)F)nc1 c1(OC)ccc2cc(NC(=O)CN3CCCC3)[nH]c2n1.N12CCCC1C1(CC1)O2 c1(OC)ccc(C(=O)NC2CC(NCc3c(C(F)(F)F)cccc3Cl)C2)c(O)c1 c1(CCNC(C(COC)NC(=O)C(C)CC2CC2)=O)cn(C)nc1C N1(C(C2C3(CC(NC(c4c(C)oc(CO)c4)=O)C3)C2)=O)CCC(C#N)CC1 CC(C)C(C(=O)NC12CC(NC(=O)C(C)CN3CCOCC3)(C1)C2)N(C)C c1(C(=O)NC(CC#C)C(=O)N(C(C)CSC)C)cc(C)ccc1F c1(CC(C(N2C(CNC(C(C)=C(CC)C)=O)CCC2)=O)C)cccc(Cl)c1 C1(C(=O)NCC2N(C(C3C(C)CC3)=O)CCC2)CC(C)(C)CO1 C1(CNC(C(CC)(C)ON=C(C)C)=O)CCCC2CN(C(=O)C3=CC(C)(C)C3)CC12 N1(C(C(C(CC)C)O)=O)CC2CCC1C(NC(c1[nH]ccc1C)=O)C2 CCC(C)CCCCC(=O)NC1CCC(CNC(c2cncc(CO)c2)=O)CC1 CCCC(C(=O)N1CCC(CCNC(=O)C=CC(F)(F)F)C1)NC(C)=O CC1=C(C(=O)N2CCC(NC(C3CCS(=O)CC3)=O)C(C(C)C)C2)CCC1 C=CCCC(C(=O)NCCC(C)F)NC(=O)CCC(CC)OC c1(N2CC=CC(NC(C3(COC)CCCO3)=O)C2)nc(C)nc2c(C)csc12 Cn1cc(C(F)=CC(=O)NCCC(C)(C)NC(=O)C=CS(C)=O)cn1 CC1(C)CN(C(=O)CC(Cl)Cl)CCC1C(N1CCc2ccccc21)=O N1(C(c2cnc(C)s2)=O)CCC(C)C(CC(=O)Nc2c(C)noc2C2CC2)C1 c1(CC(=O)NC2CN(C(CCCOCCC)=O)CC2C)ccc(CC)c(F)c1 N1(C(c2c(C)cc(F)cc2)=O)CC2CCCC2(NC(c2cnn(C)c2N)=O)C1 CC1(C)CC1(C)CNC(c1csc(O)n1)c1nnnn1CCCC1CC1 C1(CNC(COC)=O)CN(C(=O)CCN2CCN(C(C)C)CC2)C2(CCC2)C1 c1(-c2cn(C(COCC)C(N3CCC(C)C3COC)=O)nn2)ncc(F)cn1 N1(C(CC2(C=C)CN(C(=O)CC(Cl)Cl)C2)=O)CCOCC(O)C1 c1(C(N2C(C)CN(C(CCCC#C)=O)C(C)C2)=O)c[nH]c2cccc(F)c12 C1(NC(CCCOC(C)=O)=O)CC2CCC1(NC(c1cc(C)n(CCO)n1)=O)C2 N1(c2n(CC(=C)C)c(-c3ccoc3C)nn2)CC(C)OC2(CCCOC2)C1 CS(C)(=O)=Nc1ccc(C(N2CCCC(NC(=O)CCOC3COC3)C2)=O)cc1 c1(C(N(CCCNC(C2(C)CCC(C)C2)=O)CCO)=O)ccc(P(C)(C)=O)cc1 c1(C(N(CC(C)NC(=O)C(O)C(C)c2ccccc2F)C)=O)ccc(F)cc1N N1(C(c2cccc(Cl)c2C)CC)CC2CCC(C1)N2Cc1ccccc1F C(=O)(C(C)(C)CCCNC(=O)C(C1CC1)OCC)NC(CC#C)CO c1(C(=O)NC(CCOC)CNC(C2CCSC2)=O)cnc2sc(C)cn12 Cn1cc([N+](=O)[O-])cc1C(N1CC2CCC(C1)C2NC(c1cscn1)=O)=O c1(C(=O)NC(COCC)(C)C)ccc(CNC(c2ccc(SC)o2)=O)s1 C(CC(C)CC)(C(=O)N(C)CC1(O)CCCCC1)NC(C=CC)=O c1(C(N2C(CC(=O)OCC)CCC2)C(=O)OCC)c(Cl)c(C)nn1C Cc1ccc(NC(C2CCOC2CNC(c2nonc2N)=O)=O)c(C)c1O CCCC(C)O.CCC(C)(c1nccs1)NC(=O)COC(=O)CSC N1(C(C(C)SCCCC)=O)CCCC(NCCN(C)C(c2coc(CO)c2)=O)C1 Cc1ccc2c(CC(=O)N(C3CCCN(c4ccccc4)C3)C)cc(=O)oc2c1 C(=O)(CC(C)CC(F)(F)F)NC(CCN(C(C1CC(C)(C(=O)OC)C1)=O)C)C C1(N(C(c2sccc2Cl)=O)CC)CCCN(C(c2cc(Cl)cs2)=O)CC1 c1(C(=O)NC2CN(C(C3CC(CC)C3)=O)CC(O)C2)nn2cccnc2c1Cl C=C(Cl)C(C)(C)C(=O)NCC1(COC)CCN(C(c2ccncc2O)=O)CC1 c1(CN(C(=O)C(C)C(=O)O)C(CC)C)nc(O)c2c(C)c(C)sc2n1 N1(C(c2ccc(CSC)cc2)C(=O)NCc2ccco2)CCOCCC1C1CC1 C1(CC)CCC(c2nc(-c3ccc(N)cc3)nn2CCC(C)C)CC1 C1(CNC(=O)C=Cc2cn[nH]c2)CCN(C(=O)CN2CSCC2=O)CC1 C(C)(c1cnn(C)c1)=CC(=O)NCC#CCNC(C(CC)Sc1ccccc1)=O c1(OCC)nccc(C(=O)NCCCN(C(=O)CCc2cnn[nH]2)C(C)C)c1F c1(OC)cccc(C(N2CCN(C(=O)C(CO)C(C)C)CC2C(C)C)=O)c1F CCC(CN(C)C)N=c1cccc(S(=O)(=O)NCC2CCC(F)(F)CC2)[nH]1 C(=O)(C1=C(C)CCCC1)NCc1cn(CC(C)NC(C(CCC)C)=O)nn1 N1(C(c2c(C)cncc2)=O)CCN(C(c2cnn(C3CC3(F)F)c2)=O)C2CCC12 O=S(=O)(c1cccs1)NCC1(O)CCCN(Cc2cc(Cl)ccc2Br)C1 N12CCN(C(c3cccnc3)C1)C(=O)CSCCC2=O.c1(NC(C)=O)cn[nH]c1 c1(C(=O)NCCC(C)NC(=O)Cn2ccc(C(F)(F)F)n2)ccc(S(C)(=O)=O)o1 C1(C)(COC)CN(C(c2sccc2NCC)C(=O)NC(C)C)CC1(C)CO Cc1cc(Br)cc(C)c1CNCC12CC1CN(C(=O)Nc1cccc(Cl)c1Cl)C2 Cc1nc(N2CCCC2CN(C)C(C2CC23CCSCC3)=O)ccc1[N+](=O)[O-] Cc1nnc2n1CCCC2C(=O)Nc1cnc2n1CC(C(F)(F)F)CC2 N1(C(COCCCC#C)=O)CCN(C(C2(C(=O)OCC=O)CC2)=O)CC(O)C1.C N1(C(C2C=CC(NC(c3ccc(COC)o3)=O)C2)=O)CCC(C)C1CO CC1C(NC(c2ccc(-c3ccccn3)nc2)=O)CCN1c1ccccc1 c1(C2(C(=O)NC(C)CCNC(=O)CCSc3nc[nH]n3)CCC2)ccccn1 C(=O)(C1CCc2c[nH]nc21)NCCOC(C)(C)CNC(C1CCOC(C)(C)C1)=O C(=O)(C(C)(C)CN(C(=O)CC(C)n1cccn1)C)NCCc1cc(C)on1 c1(C(=O)NC2CC2CNC(C2(O)CCOC2)=O)cc(Cl)c(Cl)s1 c1(C(N2CC(NC(C(C)SC(C)C)=O)C3(C2)CC3)=O)cccc2c1COC2 c1(CC(=O)OCC(CC(=O)OCC)COC)ccc(C)c(F)c1F c1(C(N2CC(C=C)C(NC(=O)CCc3cnco3)C2)=O)cncc2[nH]ccc12 Cc1cccc(C)c1N(C)C(C1CCCN(C(C23CCCC2OCC3)=O)C1)=O CN1CC2(CCN(C(C3C4CC3N(Cc3ccc(Br)cn3)C4)=O)CC2)C1 C(=O)(CC(C)(C)CC(F)F)N1C2CC(CNC(C(C)OCCCC)=O)C1CC2 C1(NC(c2cnc3ncccn23)=O)CCC2CN(c3nnco3)CC2C1 Cc1cc(C(=O)NCC2(C)CCCN2C(c2cocn2)=O)ncc1C(F)F CC1CCN(C(c2cnn(CCF)c2)=O)CCN1C(=O)C(F)CC(C)(C)C c1(COC)cc(C(=O)N(C2CCN(C(=O)C(C)NS(C)(=O)=O)C2)C)c(C)o1 Nc1c(F)cc(C(=O)NCCOCCCNC(C2CCOC2C2CC2)=O)cc1F C1(C(=O)NCC(C(=O)NCC(C)OCCO)O)CCC(=O)CC1 C1(CC)CCCCC1C(=O)NC(C)CN(C(=O)C=CCOC1CCOCC1)C C1(C2(C)CC2)(C(N(CCCCNC(C(CC2CCC2)OC)=O)C)=O)CC1 c1(C(=O)NC(CNC(C(CC)O)=O)CC)c(C)cc(=O)n(C)c1C c1(C(=O)NCCCN(C(c2coc(-c3ccccc3)n2)=O)CC)cnc(C)[nH]1 C12(NC(=O)C(=CC3CCCCC3)F)CCN(C(=O)Cc3c[nH]nc3O)CCC1C2 C=CC(C)(C)CC(=O)NC1C2CC1CN(C(C13CC(OC)C1C3)=O)C2 CN=c1[nH]cc(C(=O)NCCOC2CCN(C(=O)C3=NOCC3)C2)s1 CCCCS(=O)(=O)CC(=O)NC1CC1CNC(c1cc(OC)n(C)n1)=O C1(NC(CCOC2CN(C(C(C(=O)OC)C)=O)C2)=O)CCC(=O)N(C)C1 c1(C(C)=O)c(C(=O)NCC2CC2c2ccsc2)sc(C)n1 C=CCC(CC=C)C(=O)N1CCC(NC(=O)CCCF)C(CO)C1 C(Cc1cn[nH]c1)(C(=O)NOCCCF)NC(c1ccoc1Cl)=O N1(C(C2CC(C#N)(OC)C2)=O)CCC(C)C(NC(=O)CC2CCS(=O)(=O)C2)C1C Cc1ccc2occ(C(N3CCC4CN(C(C5CNC(=O)N5)=O)CC4C3)=O)c2c1 N1(C2CN(C(CNC34CC(CC(=O)Nc5cccnc5)(C3)C4)=O)C2)CCCC1=O N1(Cc2cccc(NC(c3ccc(F)cc3F)C)c2)CCOCC(N)C1 CC12COC(C(=O)NCC3(O)CN(C(=O)CCCn4cncn4)C3)(C1)C2 c1(NC(C2CC23CCN(C(c2cnc(Br)s2)=O)C3)=O)cccc2c1OCO2 C(=O)(CCS(=O)(=O)N(C)C)NCCC1CC(NC(C=NOC)=O)C1 c1(OC)cc(CN2CCCC2(C)C(=O)O)cc(Br)c1.c12[nH]cnc1CNC2=O c1(OC)cnccc1CN(C(=O)CCC1CCCN(C(C2CCC2)=O)C1)CCCO c1(CC)nccn1C(C)CC(=O)NC1(CNC(=O)C(C)CC2CC2)CCC1 c1(C(N2CC(CC(C)NC(=O)CC(O)C(C)C)C2)=O)ccc2cnccc2n1 CCC(CCCC(=O)NC1C=C(C)CCC1)NC(c1cc(COC)on1)=O c1(C(=O)NC23C(CN(C(c4cncc(CC)c4)=O)C2)C3)cc(F)c(N)cc1OC Cc1nn2cccnc2c1C(=O)NC(CO)C(C)NC(=O)CN1CCCOC1=O C1(CCNC(c2c(C(N)=O)cccc2)=O)CCCN(C(=O)C2=CCCO2)CC1 CC1(C)C(C(N2CCC(CCCO)C2)=O)CCN1C(C1CC2CCC(C1)O2)=O N1(C(=O)COCc2nccs2)CCN(C(c2coc(O)n2)=O)C2(CCC2)C1 Cc1cc(OCCn2nccc2Nc2c(C)cccc2C)cc(C)c1 C1(NCc2scc(C)n2)CCC(=O)NC1C1CCCO1 C1(C(=O)NC2(C)CC(NC(C(Cc3ccc(C)cc3)C)=O)C2)CCOC(=O)CC1 Cc1c(C(N2CC3CC(NC(=O)C(F)C4CCC4)C2C3)=O)[nH]c2cc(F)ccc12 N1(C(c2nc(C)nn2C)=O)CCC2(NC(=O)CN(C)C(N)=O)CCCC12 C(=O)(C1=C(C)OCCC1)N1C(CN(C(CC2CCC(C(C)=O)CC2)=O)C)CCC1 N1(C(CCc2n(C)ccc2)=O)CCC2CCC(C1)N2C(C1(C)CC1(F)Cl)=O c1(NCC23CC(NC(CC(C(=O)OC)(C)C)=O)(C2)C3)cc2cc(F)cc(C)c2[nH]1 C1(NC(C(COC)NC(C)=O)=O)CC(CO)N(C(=O)CSc2ccccn2)C1 c1(NC(C2CC2C(N2CCCCC(O)C2)=O)=O)cc(F)ccc1Br N1(C(C2(SC)CC2)=O)CCC(N(C(=O)Cn2nnc(C3CC3)n2)C)C1 C12(CC=CCC1)C(=O)N1CC(C1)C2.N1(OC)CCN(c2nccs2)CC1 N1(C(CSCC(=O)OC)=O)CCN(C(=O)C(=CC2CCCCC2)F)C(C)CC1C N1(C(c2c(SC)cc(F)cc2)=O)CCC2(CC1)OCCC2NC(c1ccns1)=O C(=O)(C(O)CC(C)(C)C)NCCCCCNC(C(C(C)C)SCC)=O C(C)(CCC(C)(C)O)(c1n(C(CC)(C)C)nnn1)NC1(CCO)CCOC1 C(=O)(CC(C)(C)n1ccnn1)NC(CCN(C(=O)CC1CSC1)CC)C c1(OCCC)cccnc1C(=O)NC1CCC1CNC(=O)CC(=O)OC c1(NC(CNC(CC(C)=O)=O)=O)cccc(Br)c1OC(F)F Cc1cccc(C(O)C(=O)NC2CCCC2NC(c2sccc2F)=O)c1 C(=O)(C(C#N)(CC)CC)NCCC1CN(C(C(c2ccc(OC)cc2)CC)=O)C1 Cc1onc(C2CC2)c1C(=O)NCCC1CN(C(C2(F)CCOCC2)=O)CC1C N1(C(C2(C)COC2)=O)CCCC(CO)(NC(c2cc(O)nc(O)c2)=O)C1 c1(C(C)(C)C(=O)N2CCC(NC(C3CC(=C4CCC4)C3)=O)C2)cccnc1F S(=O)(=O)(c1c[nH]ccc1=NC1CCCOC1)NCc1c(OC)cc2c(c1)OCO2 N1(C(C2N(C(c3cccc(C)c3N)=O)CCOC2C)=O)CCC(=C(F)F)CC1 Cc1ccc(C(C)C(=O)NCCC(C)CCNC(=O)C(C)(C)C2CCC2)cc1 N1(C(CC2(C=C)CN(C(C3(C(N)=O)CC3)=O)C2)=O)CC2CCCCC12C N1(CC(=O)NC2(C)CC(NC(c3c(C)onc3)=O)C2)C(=O)NC(C)(C2CC2)C1=O C1(NC(C(N2CC(C)OC(C(F)(F)F)C2)=O)=O)CC2(C1)CC1CCC(C2)N1 C1(Cn2cc(C(C)=O)nn2)CCCN1C(=O)C(F)C1CN(C(=O)OC(C)(C)C)C1 c1(C(N2CC(CCNC(C(C(C)C)OC)=O)C2)=O)nn(C)c(=O)c2ccccc12 N1(C(C2(C(C)C)CC2)=O)CCC2(CCCN(C(c3nc(Cl)sc3Cl)=O)C2)CC1 C1(NC(C(C)=CC)=O)CCCN(C(c2cc(C(=O)OC)n(C)n2)=O)CCC1 c1(CN2CC3C(C(=O)NCCC(C)(C)O)(C3)C2)c(F)c(F)cc(F)c1F C(=O)(C(O)C(F)(F)F)N1C(CNC(c2ccc(CCC)[nH]2)=O)(COC)CCC1 c1(N2CC(C(C)NC(Cn3c(C(F)F)cc(C)n3)=O)C2)cc2nnc(C)n2cn1 N1(C(c2c(C)coc2C2CC2)=O)CC(NC(C2C(F)(F)C23CCC3)=O)C2(CC2)C1 Cn1cc(C(=O)NC2(C)CC(NC(C3CC4CCC4C3)=O)C2)ncc1=O c1(-c2cc(C(n3ccnc3C3CCCC3)COC)[nH]n2)ccc(OC(F)(F)F)cc1 C1(N2CCCCC2)(CC)CCCCC1.n1(CCCC)nnnc1C(C1CC(C)C1)N Cc1c(-c2noc(Cc3cn(CCCN(C)C)nn3)n2)cc(C#N)n1C C=CCCCCCCC(=O)NCC1CCCC1C(=O)NC(Cc1ccco1)CO CC(C)C(F)C(=O)N1CCC(C(O)CNC(c2ccc(OCCF)cc2)=O)CC1 N1(C(=O)CSC2CC2)CCCC2(CCN(C(c3csnn3)=O)C2)C1 c1(NC(C2(SC)CC(O)C2)=O)ccc2nc(C)[nH]c2n1 N1(C(C(=O)NCC2CCN(C)C2)=O)CCc2cc(C#N)ccc2C1 C1(C(=O)NCC2(O)CCN(C(C3(c4ccsc4)CC3)=O)C2)CC2(C1)CC21CC1 C1(C(=O)NC(C#C)C)CCC(C(=O)Nc2ccncn2)CC1 c1(-c2nc(C)[nH]n2)ccc(C(N2CC(NC(c3ccc(C)n3C)=O)C(O)C2)=O)cc1 N1(C(CC(=O)OCC)=O)CCOC(C(C)NC(c2cn(C(C)C)nc2C)=O)C1 CCC(CC(F)(F)F)C(=O)NCC1CN(C(=O)CCNC(=O)CC(C)C)CC1O c1(C(N2C(CN(C)C(C3CC(C)(C)CN3C)=O)CCC2)=O)cc(S(N)(=O)=O)co1 C1(O)(C(C)NC(C2CC(OC(F)F)C2)=O)CCN(C(=O)CNC(=O)C(C)(C)C)CC1 N1(C(C2C(C)N(C(=O)CCc3cncnc3)CC2)=O)C2CCCC1CN(C)C2 c12cc(ccc1C)NC(=O)N2.c1(C(=O)NC)ccc(NC(C)C)nc1 C(=O)(C(C)C(C)n1cccn1)NC(CNC(COCc1onc(C)n1)=O)(C)C Cc1ccnc(C(=O)NC(C)(C)CNC(=O)CCC2CCC(O)CC2)c1 Cc1cc(C(=O)NC2COCCC2NC(=O)C=Cc2cn[nH]c2)cc(F)c1 CS(=O)(=O)C(CNC(C1(O)CC1)=O)CNC(c1n[nH]c2c1CCC2)=O c1(C(N(C2CN(C(C3(C#N)CC3(C)C)=O)C2)C)=O)ccc(=O)n2c1COCC2 c1(CC(C(=O)N(CC(CNC(CN2CC(CC)C2)=O)C)C)C)c(C)n[nH]c1C Cn1cc([N+](=O)[O-])c(CC(N2CC3CC3(NC(=O)CC3CCCC34CC4)C2)=O)n1 N1(C(c2cccc(C)c2O)=O)CCC(C2CC2)(CNC(C2(C)CC=CCO2)=O)C1 C(=O)(C(CC)CCOC)N(C(CCNC(C1C(CC)CCCC1)=O)C)C N12CCC(F)(C1)NC(=O)CNC2=O.c1(C(=O)NC2(CC3CC3)CC2)ccncc1 c1(N(C)C)nccc2c1CN(C(=O)C(=O)Nc1ccc(S(C)=O)cc1)CC2 n1(CC(=O)NCC2CC(OC)CN2C(c2ccon2)=O)sc2ccccc2c1=O C1(C(N(C(CC)CC(=O)NC2CCCCC2C)C)=O)CC2(C1)CC(C)C2 N1(C(Cc2cc(C)[nH]n2)=O)CCC2(CCCCN(C(C3CCC4CC4C3)=O)C2)C1 c1(CN(C(C2CCCO2)C)Cc2ccccc2Cl)ncc(Cl)c(C(F)(F)F)n1 N1(C(C(C2CCN(C(C(C)(C)SC)=O)C2)C)=O)CCC(O)(CCO)CC1 N1(C(c2c(CC)nc[nH]2)=O)CC2(C1)CN(C(=O)C(F)(F)Cl)C2 O=C(CC(C(F)F)c1cccc(F)c1)NCC1CCCCCN1C(=O)CNC=O c1(CC(N2CC(NC(C=C(COC)C)=O)C(F)CC2)=O)coc2cc(Cl)ccc12 C1(C(=O)NCCC2(C(=O)NC(c3cc(C)on3)C)CCCC2)CC=CC(O)C1 CC1CN(C(=O)CC(C)c2ccncc2)CC1NC(C1(C)SCCCS1)=O C1(C(C(=O)NCC(CNC(c2cc(C)n(C)c2)=O)OC)C)CCCCCC1 c1(CCNC(=O)CC2CCCCCN2)nc2c(o1)CCSC2 C1(N(C(CCN(CCCCC)C)=O)C)CCCN(C(C2CC3CCC3C2)=O)C1 N1(C(C(C)(C)SC)=O)CCC(C2(NC(=O)CSCc3cccc(Cl)c3)CC2)C1 CC1CCC(NC(C2(C3CCC3)CC2)=O)CN1C(c1cc(F)ccc1Br)=O c12c(C)[nH]c(c1C)C2=O.n1(CC2(CC)CCC2)cc(CCCNC(=O)OC)nn1 C(CC1CCOCC1)(C(=O)NCCC=C=C)NC(COCC#C)=O.C(C)(=O)O C1(C(=O)OCc2cc(C)sn2)CCC(=O)C(C)C1(C)C c1(C(N2CCC(C)C2CNC(=O)C=CC2CCC2)=O)cc2ccc(Br)cn2c1 C=CCC(CNC(c1ncccc1CC)=O)C(=O)NCC(CO)C1CC1 C1(C(=O)NCC(C)NC(COCCCOCC)=O)CC(n2cnnc2)C1 c1(C(=O)NCCC(C)N(C(=O)Cc2cccc(Cl)c2Cl)C)cnc2[nH]cncc1-2 CN=S(C)(=O)c1ccc(C(=O)NCCN(C(=O)CC2COCC(C)(C)O2)C)cc1 N1(C(CC2(CS(C)(=O)=O)CC2)=O)CC(F)(CNC(=O)C(F)C2CCOC2)C1 c1(C(N2CCC(CNC(CCCC#C)=O)CC2C)=O)cccc2c1NCC2 S(=O)(=O)(CC(=O)NCC1CCCCC1NC(=O)CC(C)(F)F)NC(C)(C)C N1(C(C2C(OC)CN(C(C3CN4CCN3CC4)=O)C2)=O)CCC2(COC(=O)N2)C1 CC(CN(C(=O)Cc1nccn1C)C)C(=O)NC1(C2CCCO2)CCC1 N1(C(C(C)NC(C)(C)C)=O)CC(C)(C)C(NC(=O)C=CC(=O)N(C)C)C(C)(C)C1 Cc1nc(C(N2CC(OCCNC(c3ccc(=O)oc3)=O)C2)=O)c(C)o1 N12CC(CC1C(N1CC3C(N(C)C)C3C1)=O)OCCC2=O.CCCOC Cc1c(C(N2CCC(C)(NC(c3ccc(OCF)cc3)=O)CC2)=O)cncc1F c1(OC)cc(C(=O)NCCC2CCN(C(=O)C#CC(C)(C)C)C(C)C2)ccc1F Cc1cc(N)cnc1C(=O)NCC(C)N(C)C(c1ccc(C(C)(C)C)s1)=O C12(NC(c3c(Cl)c(C)n(C)n3)=O)COCCC1CN(C(=O)C1=CCCCC1)C2 C1(CC(=O)N(C(CC)CO)CC)CC(c2ccccc2)=NO1 Cc1ccc(Cl)c(OC(C)C(=O)NCC(C(C)(C)C)NC(=O)C=CC(F)(F)F)c1 c1(OC)ccc(C(N2CCC(C)(NC(=O)CN(C)S(N)(=O)=O)C2)=O)c(C)c1OC c1(CN2C(C(=O)OC)CC(C(C)(C)C)CC2)cn2c(n1)CCCC2 N1(C(CCC(=O)NC)=O)CCC2(NC(=O)CP(C)(C)=O)CCCC12 C(=O)(C(C)C(C)(C)c1ccccc1)N1C(CNC(Cc2c(C)nc[nH]2)=O)C=CC1 c1(C(CNC(c2cccc(Oc3ccccn3)c2)=O)F)ccc(F)cc1F N1(C(c2n[nH]c(C)c2Cl)=O)CC(NC(C2C(F)(F)C23CC3)=O)CC(C)(C)C1 c1(C(=O)NCCC2CN(C(C(C)OCCN(C)C)=O)C2)cc2occc2s1 c1(OCCC(=O)NCCC(C)NC(=O)CC2CC3(CC3)CO2)ccc(F)c(Cl)c1 C(=O)(C(F)(F)CCn1cccn1)NC1C2CN(C(c3c(OC)n[nH]c3)=O)C1C2 c1(OC)cc([N+](=O)[O-])c(-c2nc(CC3CCCCC3)no2)cc1OCCC(C)C N1(C(c2cc(C)ns2)=O)CCCC(NC(C2CCC(C)(C)OC2)=O)C1C C1(CC)CN(C(=O)COc2ccc(F)cc2)CCC1NC(C1C=CCC1)=O c1(C(C(=O)NCC2CCN(C(C(C(C)SC)O)=O)CC2)=O)ccc(F)c(F)c1F N1(C(=O)CSCc2ncc[nH]2)CCCC2C1CCCN2C(c1c[nH]ccc1=O)=O N1(C(c2ccc(Cl)cc2)=O)CCn2ncc(-c3cnn4c3CCC4)c2C1 CC1(C(=O)NCC(O)CCNC(=O)C(c2ccccc2Cl)O)CCCCCC1 CCCCC(C(=O)N(C1CN(C(=O)C(C)CC2CCCC2)CCC1O)C)C(C)C c1(C(N(C2CCN(C(=O)CCc3cccn3C)C2)CC#C)=O)cnn(CCO)c1 N1(C(C(CC)F)=O)CC(NC(c2ccc(OC(F)F)cc2F)=O)CC(C)(C)C1 c1(C(C)C(=O)N2CCC2CNC(=O)NC23CCCC2C3)cccc(C(F)(F)F)c1 N1(C(C2C=CC(NC(=O)CCCC3CCCC3)C2)=O)CC2CCC(O)C(O)C12 N1(CC(N2CCCC(C(C)NC(C(OC)OC)=O)C2)=O)Cc2ccccc2C1=O Nc1cncc(C(=O)NCC2C3CN(C(C4CCCC(O)C4)=O)CC23)c1 C(C(C(C)(C)C)NC(c1c(Cl)n[nH]c1C)=O)NC(CCCOCCOCC)=O CCN=c1[nH]c(C(=O)NCC2CC(F)(CNC(C3CCN(CC)C3)=O)C2)cs1 c1(CC(=O)NC2(CNC(c3c(CC)c[nH]n3)=O)CCOC2)c[nH]c2ncccc12 N1(C(C(C)NC(COC)=O)=O)CC2N(C(=O)C(C(C)(C)C)SC)CCC2(C)C1 c1(C(C(=O)NCC(CC)N(C(=O)CC2CCCOC2)C)O)ccnn1C C1(NC(CCC#CC)=O)CCN(C(=O)C#CC(C)C)C12CC2 c1(CN2C(C(=O)Nc3c(C(=O)OC)nsc3)CC2)cc(Cl)nc(Cl)c1 C#CC1(O)CC(C(N2CCCCC2CNC(c2oc(SC)cc2C)=O)=O)C1 c1(NC2C(NC(C(C)CF)=O)CCC2)cccc(F)c1C#N C(=O)(C(CC(C)C)C(C)C)NCCC1CCN(C(C(C(=C)C)(C)C)=O)CC1(F)F CN1N=CC(CC(=O)NCC(CC2CC2)C(=O)NCC2(CO)CCC2)C1=O CC1(C)CCCCC1=CC(N1CCOC(C)(CNC(=O)CN2CC3CC3C2)C1)=O C1(CNC(C(CO)OC)=O)CN(C(c2cnn(C(C)C)c2N)=O)CCCO1 C(=O)(CCCCC(N)=O)NC(C)C(C)NC(C1(S(N)(=O)=O)CCCC1)=O Cc1nocc1CC(=O)NC(C)CN(C(=O)C(NC(C)=O)=Cc1cccs1)C c1(C(=O)NC(CC=C)CNC(C2CC2CC)=O)cc([N+](=O)[O-])ncc1Br c1(C(N2CCC(CNC(CC(CC)O)=O)C2(C)C)=O)cc2c(nc1O)CCCC2 O=C(CCCCO)O.C1C#CCNC(=O)C1.C(=O)(C(O)c1ccsc1)NC n1(C(C)(C)C)ncnc1C(=O)NCC1CCCN1C(=O)CC1(n2cccn2)CC1 N1(C(C(CC)SC)=O)CC2(C(=O)NCC3(C)CCCO3)CCC1CC2 C1(C(=O)NCC2CN3CCC2C3)(CC)CCN(C(=O)CC(C)(C)O)CC1 Cc1nocc1C(=O)NCC1(O)CN(C(=O)C(C)N(CC(F)(F)F)C)C1 C1(C(N2C(C(C(=O)NC(C(=O)OC)C)(C)C)CCC2)=O)C2CCC(C2)C1C c1(NC(CCC)CCCNC(=O)CCOCCOCC)ncc2ncnc-2[nH]1 O=S(=O)(c1c[nH]ccc1=NC1COC2(CCC2)C1)NCC1C2CCCC12 C(=O)(C(C)C(O)C(C)C)N1CCN(C(Cc2cc(C)nn2C)=O)C(C(C)C)C1 N1(C(c2c(CC)nc[nH]2)=O)CCc2sccc2C1CNC(=O)C(F)CC(C)C c1(OC)ncc(CNc2cn(C)c(C(=O)Nc3ccc(C)nc3O)n2)cc1Br C(=O)(N1CCCc2nncn21)C1(NC(c2cccn(C)c2=O)=O)CCCOC1 N1(C(CSCCN(C)C)=O)CCC(CNC(c2cc(C3CC3)on2)=O)C12CCC2 Cc1ccc2nc(C)c(C(=O)NC3CN(C(c4cccc(Br)c4)=O)C3)n2c1 n1(CCC(=O)NCCC2CN(C(C(COCC)C)=O)C2)cnc2ccccc12 CCCC(CCC)C(=O)N1CCC(O)(C(C)NC(c2cc(C(F)F)ncn2)=O)C1 Cn1cc(C(=O)NC(C)(CNC(c2cc(C(N)=O)cs2)=O)C2CCC2)ccc1=O c1(C(=O)NCC2(C)CCN(C(C3(C4CC4)CC=CC3)=O)C2)cc(Br)ccc1N c1(C(CN2CCCCCC2)=O)cc(N)cc(C(F)(F)F)n1.CC1CN1 C1(NC(c2cccc(OC)n2)=O)CCOC12CCN(C(=O)C(O)P(C)(C)=O)CC2 c1(C(C)C)cnn(C)c1C(=O)NC(CNC(=O)CC(O)Cc1ccccc1)CO Cc1cc(O)ncc1NC(=O)CCN(C(c1cc[nH]c(=N)n1)=O)C1CC1 CC(C)CC(C(=O)NCC1(C)CC(NC(c2ccc(Cl)c(F)c2F)=O)C1)C(N)=O c1(C(N2CC(NC(COCCOC)=O)CC2(C)C)=O)cnc2c(C)cccc2c1 c1(C(COC(C2C(C)(C)CCO2)=O)=O)cnc2n1CCC2 Cc1ccc(C(=O)NC(CNC(C23CSC(C2)C3)=O)C(C)(C)C)n1C CC(C)C(C(=O)N1CCC(C(=O)NCc2ncccc2F)O1)C1CCC1 c1(N2C(C(=O)NCCC(F)(F)F)CCC2)nccc(Br)n1 C1(C2CC2)(N(C(=O)C(O)C2CN(C(=O)CC3CC(=O)C3)C2)C)CC1 c1(C(N2CC=C(CNC(C(C)CO)=O)CC2)=O)n[nH]c2c1CC(C)(C)C2 Cc1cn(C)cc1C(=O)NCC(C)(C)CNC(C1CC(C)(c2ccccc2)C1)=O CCCCC(=O)N1CSCC1C(=O)NCCCNC(=O)COc1ccsn1 C1(C(=O)OC)CCC(C(=O)NC(C)CN(C(=O)CCCOC2CCOCC2)C)C1 C(=O)(N=c1[nH]cc(C#N)cc1C)c1nccc(-c2c(C)nc(C)s2)c1 C(=O)(CC1=CCOCC1)NCC1C(C(N(C(CF)CF)C)=O)C1 c1(C(N2CC(C(C)NC(c3cscc3F)=O)OCC2)=O)cc2c(ncn2C)s1 C(=O)(C1=C(C)OCCS1)NCC(CC=C)C(=O)NC1COC(C(F)F)C1 c1(C(=O)NCCNC(CC2C(NC(=O)C=C(Cl)Cl)C2(F)F)=O)ccc(F)cc1 C=CC1COCC1NC(=O)CC1CC1C=O.c1(C(=O)NC)cccc(CO)c1 Cc1cccc(C(=O)NCC(C2CCN(C(c3cc(C)n(C)n3)=O)CC2)F)c1C C1(CNC(c2nncs2)=O)CCN(C(C23CC2C3)=O)CC1 C(=O)(C(C)(C(C)C)NC(=O)OC)NCC1(OC)CN(C(=O)CSc2ccoc2)C1 C(C(C)CC(=O)NCC1CCN(C(=O)CNC(c2ccco2)=O)CC1)OC C1(C(N2CCCC(N(C(=O)COc3cnn(C)c3)CC)C2)=O)CC(=O)OC1(C)C CC(F)(C(=O)N1CC(NC(=O)CNC(N)=O)C1)C1CC1 C1(C(=O)NC2(CC)CCOC2)C2CC2CN1C(=O)CC1C(C)(C)C1(C)C C1(F)(CNC(CN(C)CC)=O)CCCN(C(C2(C(F)(F)F)CC2)=O)C1 c1(CNc2cnn(-c3c(OC)cccc3)c2C)nn(C)c2ccccc12 C1(CC(=O)N(CC)CC2CC2)CN(C(C2CCC(C3CC3)C2)=O)C(C)(C)C1 c1(C(=O)NC(CC)CNC(C2CCC2C(F)(F)F)=O)cscc1C(F)F N1(C(COCCCOC)=O)CC(C)CN(C(=O)CCCc2ccccn2)CC1C O=C(C1Cc2ccccc21)NC1CCN(C(=O)C(c2ccccc2Cl)O)CC1O c1(C(=O)NC2C(NC(C3C(=C)C3)=O)C2)cnc(OC)c(Br)c1 c1(CC)sc(C(N2CCCC2CCCNC(c2csc(O)n2)=O)=O)cc1C CCCCC(C(=O)NC1(C)CC(NC(=O)Cc2cc3ccccc3o2)C1)C(C)C C(=O)(C1CCc2c[nH]nc21)NC1CCN(C(c2n(COC)ncc2)=O)CC(O)C1 c1(C(N2CC(C)(NC(c3cn(C(C)C)nn3)=O)C2)=O)ccc2c(c1)C(C)C(C)O2 C(C(C)NC(=O)CCN(C)C(C)=O)(C(C)C)NC(CN(C(=O)OC)C)=O c1(C(=O)NCC2C3CN(C(C(C)(C)F)=O)C2C3)ccc2n[nH]cc2n1 C=CCCCC(C1CC1)NC(C1CC1CNC(c1ccc(F)cn1)=O)=O N1(C(c2cc(COC(C3CN(C(C)=O)C3)=O)sc2)=O)CCOCC1C1(CO)CC1 c1(NC(=O)CCC2CCN(C(c3ccc([N+](=O)[O-])o3)=O)C2)cccc2c1CCO2 N1(C(C=CC(=O)OCCCC)=O)CCC(O)(CNC(c2cnccc2OC)=O)CC1 c1(OC(C)C(=O)NC2CC(NC(=O)CC3CCOCC3)C2)ncccn1 c1(OC)ncc(C)cc1NC(C1(NC(C2(C)CC3C=CC2C3)=O)CCC1)=O N1(C(c2cccc(CC)c2O)=O)CC2(CC(NC(=O)C(C)=CC3CC3)CO2)C1 Cc1cc(C)c(C(=O)NC2CCCC2n2cc(CCS(N)(=O)=O)nn2)cn1 n1(CC(=O)NCC2C(NC(CCCc3ncc(C)o3)=O)C2)nc([N+](=O)[O-])cc1C N1(C(C2C(CCC)CCC2)=O)CCC2CCC(NC(=O)CCCCN(C)C)C12 CC12C3C4C1C1C2C3C41C(=O)NC1CCN(CCCNC(=O)Cc2ccco2)C1 C1(C(=O)NC2C(CNC(C=C(C)C3CC3)=O)CC2)CCCc2ccccc2C1 n1(C(C)C)ncc2c1CCCC2NC(=O)Cc1cccc2nsnc12 C1(CNC(C2CC(CNC(=O)COC(=O)CO)C2)=O)Cc2nccn2C1 c1(CC)cnccc1C(N1CCC(CC)C1CNC(C1CC(C)=NO1)=O)=O C1(CC(F)F)C(=O)N1.C(C(=O)NC1CC1)N(C(=O)COC1CCC1)C Cc1ncn(C)c1C(=O)NCc1cn(C2CCN(C(C)(C)C)CC2)nn1 c1(C(=O)NCc2cn(CCOC)nn2)oc(CN2CCSCC2)cc1C C1(C(=O)NC2CCC(NC(Cc3c(C)n[nH]c3)=O)C2)CC1C1(C)COC1 N1(C(C(C(C)C)O)=O)CC2COCCC2(NC(c2ccc(O)c(C(N)=O)c2)=O)C1 C(CC1=CCCCC1)N(C(C1(CC=C)CN(C(C2CC(C3CC3)C2)=O)C1)=O)C c1(OC)ccc(F)cc1CCC(=O)NCC(CO)NC(C12CC(C1)C(C)(C)O2)=O Cc1nc(C(=O)N(CCCOCCN(C)C(c2sccc2Cl)=O)C)sc1C c1(C(C)CC(=O)N(CCN(C)C(C2CCCSS2)=O)C(C)C)ccc(F)cc1 C1(N(C)C)CN(C(=O)C(O)CCNC(c2cccc(O)c2)=O)CC1F C#Cc1ccc(C(=O)NC2CC3(CCOCC3)C2)cc1Cl C1(N(C)C)CCCCC1C(N1CC(NC(C2CC(NS(C)(=O)=O)C2)=O)C1)=O C1(CC=C)(NC(=O)CCn2cncn2)CCN(C(C2CCS(=O)(=O)CC2)=O)CC1 C(C(C)(C)CC(=O)NCC1CC1CC(=O)N(CCO)Cc1ccccc1)OC N1(C(CC2N(C(c3cc(C)ncn3)=O)CCCC2)=O)CCCC2(C1)N=N2 c1(C(=O)OC)ccc(CN2CCCC2CNC(C2(c3ccccc3)COC2)=O)s1 c1(C(=O)OC)c(C)[nH]c(C(=O)NC2CN(C(C3CC(OC)C3)=O)CC23CC3)c1C N1(C(CCC#C)=O)CC2(CNC(=O)C=CCCC(C)C)CC1CCO2 S(=O)(=O)(c1ccc(F)c(F)c1F)NC(C1CN(Cc2c(O)cccc2F)C1)C c1(CN2CCC(C(=O)Nc3onc(C)c3Br)C2)cc(Cl)cc(Cl)c1Cl C(=O)(C1=C(C)OCCS1)N(C1(C2CCCN2C(=O)C(C)C#N)CC1)CC C12(CNC(c3c(CC)c[nH]n3)=O)CC1CN(C(C1CC=CCC1C(F)(F)F)=O)C2 c1(C(=O)NC(CC=C)CNC(=O)Cc2cncn2C)cnc(CC)cn1 C=C(C)CC(C)C(=O)NCCCCN(C(=O)C(C)(C)C1CCCCO1)C CS(=O)(=O)c1cscc1C(N1CCC(F)(F)C(CNC(=O)Cn2ccnn2)C1)=O C(=O)(C(C)C1CC1)NCCN(CCOCC)Cc1nncs1 N1(C(C(F)=CCC)=O)CCCC(CC)C1C(=O)Nc1ccc(OC)nc1 c1(C(=O)NC(C(=O)OC)Cc2cc(Cl)sc2Cl)ccc(OC(F)(F)F)cc1F C1(C(=O)NCCN(C(=O)Cc2csc(C)n2)CC)CCCCC(C)(C)C1 C12(CNC(c3cc(F)ccc3F)=O)CCC(CC1)N(C(=O)C(F)=CCCF)C2 N1(Cc2cn(CC)nc2)CCC2(CCN(C(=O)Cn3ccc(C)cc3=O)CC2)C1 C(=O)(CCCC(C)(F)F)NC1C(N(C(C(=O)N2CCCC2)C2CC2)C)CCCCC1 c1(OC)c(C(N2CCOC(CNC(c3ccc(C(F)F)s3)=O)C2)=O)cccc1F N1(C(C2(CCCC)CCCCC2)=O)CC(NC(=O)CSCC(C)C)CC(F)C1 N1(C(CC)=O)CCC(C)(CNC(=O)CCc2scnc2C)C1 c1(C(N2CCC(C=C)(C(=O)NC(C#C)CC)C2)=O)cc(C#N)ccc1C N(C(=NCCCCl)NC1CCC(=O)NC1)CC1(NC(=O)OC(C)(C)C)CC1 N1(c2cc(OC)nc(C)n2)CC2(CCC(NC(=O)CCN3C(=O)C=CC3=O)C2)C1 CCCC(CC)C(=O)NC(c1ccccc1F)CNC(c1cnc(S)[nH]1)=O C(=O)(C#CC1CCOC1)NCC1C(NC(C=CC(=O)OC(C)(C)C)=O)C1 C1(C(=O)NCC(NOC)=O)CN(C(=O)C=Cc2nccs2)CC12CCC2 N1(CC(=O)NCCC)CC2CCC(NC(c3ccc4c(c3)OCCO4)=O)CC2C1 c1(C(=O)NCCSCC)sccc1CNC(=O)C(C)CN(C)C C1(CC(=O)NC2CCN(C(C=C3CCC(C)CC3)=O)C2)CCOCC1(C)C C(=O)(C(CO)C(F)(F)F)N(CCCC(=O)OC)Cc1cscc1NC(C)=O c1(CN2CCN(C(C)CC3(C(F)(F)F)CC3)C3C2C3)c2cc(Br)ccc2nn1C N1(C(C2CC=CC2)=O)CCCC(C2CCCN2C(C2(O)CCOCC2)=O)C1 c1(C(N2CC(NC(c3c(OC)c(F)ncc3)=O)C(O)C2)=O)cc(F)c(F)cc1N C1(NC(COC2CN(C(C(C)(F)F)=O)C2)=O)CC2OCCCC12 CC(C)CC(O)C(C)C(=O)N1CC(O)(CCNC(=O)Cc2ccc(O)c(Cl)c2)C1 c1(OC)ccc(C(N2CC(C)(C)C2CO)=O)c(C(F)(F)F)c1 CC(C)(C)C(O)C(=O)NC1CC(CCNC(=O)CCCc2ncco2)C1 C(CCCCNC(c1[nH]nnc1C1CC1)=O)NC(=O)COC1CCCOC1 C(=O)(C(CO)C(F)(F)F)NC1(CC=C)CCN(C(C2CC3(C2)CC(C)(C)C3)=O)C1 C1(CC)CCCCC1C(=O)N(CCCNC(=O)C(C)(C)c1ccncc1)C C1(C(=O)NC(C)C(CO)NC(c2ccc(O)nn2)=O)CCN(C2CC2)S1(=O)=O C(=O)(C(C)CCCc1ccccc1)N1CCC(C)(CNC(C=CCCC)=O)C1 C(C(CCN=c1[nH]c(=NC(C)CCSC)[nH]c2ccccc12)C(C)C)OC C(c1cc(Br)ccc1C(C)O)=Cc1ccc(CC)s1 CCCCS(=O)(=O)CC(=O)NC1C2CC1N(C(=O)Cn1cc(C(F)(F)F)nn1)C2 c1(NC(C2N(Cc3cccc(OC)c3F)C3C(C2)C3)=O)ccc2nc(O)[nH]c2c1 c1(C(N2CCC(CCOC)(NC(=O)CN(C)C)C2)=O)coc2ccc(Br)cc12 N1(C(COCC#C)=O)CCCC(C)(CNC(c2ncccc2C)=O)C1 C(=O)(CCCN(C)C)NCCC(C)NC(c1cccnn1)=O N1(C(COCCCC#C)=O)CCOC(C(=O)NCC2(C)C=CCCC2)CC1 Cn1cc(C(C(=O)Nc2cccnc2)NC(c2ccc(I)s2)=O)cn1 N1(C(c2scc(C)c2)=O)CC(CCNC(=O)C=CC(=O)NC2CC2)C(C)C1 c1(N(C2CCN(C(C3(C)CC(=C)C3)=O)CC2)CC=CC)nc2cccnc2s1 C1(C(=O)NCC2(C)N(C(C#CC(C)C)=O)CCC2)CCc2cncn2C1 c1(CC)ccc(C)c(NC(=O)C(Cn2cncn2)NC(C2CC(=O)C2(C)C)=O)c1 C1(C#N)(C(=O)NC(CCNC(c2cccc(OCCC)c2)=O)C)CC2(CC2)C1 C1(F)(C(N(C)CC2N(C(c3c(C)cns3)=O)CCC2)=O)CCS(=O)(=O)C1 C1(NC(C(C)NS(C)(=O)=O)=O)CCC(NC(c2ncc[nH]2)=O)CC1 N1(C(C(=O)N(c2cc(Br)cs2)C)=O)CCC(c2cn(C(C)(C)C)nn2)CC1C CC1CN(C(C2CC(C)(C)C2)=O)CC2(CCN(C(=O)C(F)(F)c3nccs3)C2)O1 CS(=O)CCCC(C=CC(=O)N)CCC CC1(C)CC(NC(C2(C)CCCNC2=O)=O)CCN(C(=O)COC2CCCC2)C1 CC(=O)CCN=C(NCCC1SCCS1)N1CCN(c2nnc(C)c(C)n2)CC1 CC(=O)CCCC(=O)NCCC1CC(NC(c2cn3c(n2)SCC3)=O)C1 C1(N(C(c2cc(CCC)oc2C)=O)C)CN(C(C2CC(F)C(=O)N2)=O)CC12CC2 N1(C(c2c(C#C)c[nH]n2)=O)CCN(C(=O)C2=C(Cl)CC2)CC1CC(F)F N1(C(c2coc(Cl)c2)=O)CCN(C(=O)Cc2cncnc2O)C2CCCCC2C1 N1(C(C(C)C)=O)CC(NC(C23CC(CN2C2CC2)C3)=O)CC12CCCCC2 N1(C(CC2(C)N(C(CC(CC(C)C)C)=O)CC2)=O)CC2(CCC2)C12CCC2 C(=O)(C(C)(CN(C)C(=O)OC(C)(C)C)C(C)C)OCC1N(CC)CC1 N1(C(c2ccc(C#C)c(F)c2)=O)CCCC2CN(C(c3scnc3C)=O)CCC12 N1(CC(COCC)OC(=O)CC(O)CCSCC)CCc2sccc2C1 N1(C(CC(CC=C)(C)C)=O)CC2CC3CC2C1C3NC(c1scc(C)c1C)=O c1(C(=O)NC(C(C)NC(C2CC(=C)C2)=O)C(C)C)cnn2c1NCCC2 c1(N2CC3CN(c4ncc(SCC)cn4)CC3C2)nc2c(cc1C#N)CCOC2 CC1OC2(C(N3CC4CC4(NC(c4ccc5c[nH]nc5n4)=O)C3)=O)CCC1CC2 N1(C(C2CC(NC(C=CCCC(C)C)=O)C2)=O)CC(C)OC(C)(C)C1C Cc1ccc2nc(C(N3CCN(C(=O)Cc4occc4C)C(CO)C3)=O)cn2c1 C1(OC)CCC(C(=O)NCCCCCCNC(c2coc(N(C)C)n2)=O)CC1 c1(C(=O)NCC(CCCC)NC(C2(S(C)(=O)=O)CCC2)=O)cc(C)c(O)c(N)c1 C1(N(C(=O)NC2CC2c2ccccc2C)CC)CCC2COC1O2 c1(CC)ncc(Cl)c(C(=O)NC2C=CCN(C(c3ncnc(C)c3C)=O)C2)n1 c1(C(N2CC(CC(N3C(NC(N)=O)CC3)=O)C2)=O)cccc(CCO)c1 CC1CCCCCCN1C(C1CC2CCC1N2C(C1(CCF)CCC1)=O)=O C1(C)(CC2N(C(CN(C(=O)COc3ccsc3)C)=O)CC2)CC=CCC1 C1(NC(C2CCC(=C)CC2)=O)CCN(CCc2scnc2C)CC1C c1(C(N(CC)CC2CCN(C(=O)CC3C=CCCC3)CC2)=O)cnc(O)c(F)c1 Cc1cc(C#N)nc(Nc2cnc(Cl)cc2C(N2CCC(CO)C2)=O)n1 N1(C(c2sc(C(=O)OC)c(C)c2)=O)CCCC2CN(C(C3CC(O)C3)=O)CCC12 C1(C#CC(=O)NCCOC2CN(C(c3cc(C(F)F)[nH]n3)=O)C2)(CC)CC1 C1(CNC(c2cncc(OCC)c2)=O)CN(C(=O)C(C)OCCOC)CCCO1 c1(C(=O)NC2(CCO)CN(C(C(CCCC)C)=O)C2)cccc2scnc12 N1(C(C(c2ccc(Br)cc2F)C)=O)CC2(CCCC2NC(=O)CNC(=N)N)C1 c1(C(N2CC(C(C)NC(c3cccc(SCCC)c3)=O)C2)=O)cc(F)cc(F)c1 N1(C(C(CSC)OC)=O)CCC(CNC(c2cccnc2N(C)C)=O)C(F)(F)C1 C#CC1CN(C(C2CCN(C(c3cc(C)sc3C)=O)C2)=O)CCO1 c1(CC(=O)NCC2CN(C(=O)C(F)=CC3CC3)C2)cc(Cl)ccc1O c1(OC)ccc(O)c(CN2CCN(C(=O)Nc3ccc(C4CC4)cc3)CC2)c1 C1(CNC(c2cnn(C(F)F)c2)=O)CN(C(c2cc(F)c[nH]2)=O)CCC1(F)F CC1CC(C(N2CC=CC(C(=O)NCCC3C=CCC3)C2)=O)CN1C CC1(C)OCCC1NC(C1CC(CCNC(=O)CCN2CCCC2)C1)=O C1(C(=O)NC)CCCN(CC(=O)Nc2ccccc2Oc2ccccc2)C1 O=C1NCC(C(=O)N(C2(C(=O)NC3CC3C(F)F)CCC2)C2CC2)N1 C=C(C)CCCC(=O)N1CC(CC(N2CCC(OC)C2(C)C)=O)C2(CC2)C1 N1(c2ccnc(C(C)C)n2)CCC(NC(=O)C(C(C)O)NC(=O)C2CC2)C(C)C1 C1(CNCc2cn(C(C)(C)C)nc2)COCC(C)(C)O1.N12CC(C)(C1)CC2=O C(=O)(C(F)(CNC(=O)C(c1cnn(C)c1)=O)C(C)C)NCC(=C)Cl C(=O)(CCCN=[N+]=[N-])N(C1CCC(NC(=O)C(C)(C)N(C)C)CC1)C Cc1cccc(COC(C)C(=O)NCc2nc(COC(=O)CC(C)C)cs2)c1 CC1(C)CN(S(C)(=O)=O)CCN1C(c1ccc(NNC(=O)C2CCC2)s1)=O c1(CC(=O)N(C(CNC(C2N(CC)CCCC2)=O)C)C)cc(F)ccc1Cl CSC1=C(C(=O)N(C)CCN2CCN(C(C3CCSC(C)C3)=O)CC2)CCCC1 C1(C(N(CC=CC(=O)NCC2(C)ON=C(C)C2)C)=O)CCCCC1(C)C CC1CN(C(C2CCC=CCC2)=O)CCN1C(C12CCC(F)(CC1)C2)=O N(C(=NCC1CCC2(CC2)C1)NC1CCOCC1)CC(C=C)(F)F Cc1ccc(C=CC(N2CCN(C(=O)CC(C)(C)F)C(C3CC3)C2)=O)cc1 NS(=O)(=O)c1ccc(C(=O)NC2CCC23CN(C(=O)CCc2cnc(O)[nH]2)C3)s1 C(=O)(C(C(C)(C)C)OC)NCC(C(=O)NCc1c(OC)cccc1)O C1(CNC(C2(OC)CCOCC2)=O)CCCC2(CN(C(=O)Cn3cccc3)C2)O1 c1(CNC(C2CC(F)CN(C(c3sccc3Cl)=O)C2)=O)ccc(CO)cc1F N1(C(C(=O)Nc2c(NC(N)=O)cccc2)=O)CCCC(O)(C(F)(F)F)CC1 c1(C(=O)NCCN(C(=O)C(C)N(C2CCC2)C)CC)ccc(Cl)c(O)c1 CC1(C)CCCN(C(C2CCC2C(C)(C)C)=O)C1C(=O)NC1(C)CCCC1(F)F C1(C(=O)NC(C(=O)OCC)C)CCC(C(C)C)N1C(c1ccc(C)n1C)=O CC(C)C(CNC(C1CCCCCC1)=O)C(=O)NCCN1CCCC1 CCC(C)(CNC(c1cc(OC)ns1)=O)C(=O)NCCN(C)C1CC1 N1(C(CC2CCCN(C(C3(C#C)CC3)=O)CC2)=O)CCCCC(C)(C)C1 CC1CC2CN(C(=O)CCc3nccn3C)CC2N1C(C1CC2C=CC1CC2)=O N1(C(C(=O)NCC(CC)NC(=O)OC(C)(C)C)=O)CC(C)(C)OC2CCCC12 C(=O)(C(C)CS(C)(=O)=O)NCC12N(C(C3(COC)CC3(F)F)=O)C(CC1)CC2 N1(C(C2C(=C)C2C(=O)OC)=O)CCC(CCC(=O)N(CC(C)C)CC(C)C)C1 C1(NC(C2CC3(C2)CC3(F)F)=O)CCCN(C(c2cccnc2C(F)F)=O)CC1 N1(C(C(CC=C)(C)O)=O)CC2(C=C(C(=O)NCC(C)CC(F)(F)F)CO2)C1 C1(C)(C(=O)NCC2CCN(C(CC)=O)C2)CCN(C(c2cnc(C)o2)=O)C1 O=C1NCCN(C(C2C(O)CCN2C(=O)Cn2cccc2)=O)C1CCO Cc1snc2sc(C(N3CC(C)(NC(C4CCCC4C)=O)C3)=O)cc12 C1(CNCC2(C)OCCO2)CN(Cc2cc(C(F)(F)F)cc(Cl)c2)CCC1O c1(CNC(C2C(CC)OCC2)=O)cccc(C(=O)NCC2=NOC(C)C2)n1 N1(C(CC(C(=O)OC)C)=O)CC(n2cc(C(C)(C)N(C)C)nn2)C(S(C)(=O)=O)C1 c1(C(=O)NCCC2CCC(NC(=O)C=CBr)C2)cc2n(n1)CCO2 c1(C(N2C(CNC(C(CC)=CC)=O)CC2)=O)ccc(F)c(C(F)(F)F)c1 C1(N(C)C(c2cncn2C)=O)CCC2(CC1)CN(C(=O)CSCc1ncc[nH]1)C2 C=CC1(C(=O)NCC2C3CN(c4nnc(C(F)F)s4)CC23)CCCCC1 c1(C(=O)NC2CC(NC(C3(C)CC3(F)F)=O)C2)ccc(-c2cncnc2)cc1F C1(C(=O)NC(C)C(N2CCN(C)CC2)=O)CC(=O)N(C)C1c1cccs1 C=CC(CCC)CC(=O)NCC12CC(NC(=O)CCNC(=O)C=CCl)(C1)C(C)O2 O=C(C1=CCCOCC1)NCC(C1CCOC1)NC(=O)CC1(CO)CC1 C(C(C)(C)CCO)NC(C(C1CN(C(C2OCCC2C)=O)C1)OC)=O CN1CC(NC(=O)C(C2CC2)NC(=O)CC2CSCCO2)C2(CC2)C1 C1(NC(C2CC(SC)C2)=O)CN(C(=O)CCCC2CCC2)CC1OC c1(C(N2CC3(CN(C(c4cncc(SC)c4)=O)C3)C2)=O)cc2ccccc2[nH]1 C1(C(=O)NCC(CC2CC2)CO)(CC)CCN(C(c2cscc2C)=O)CC1 c1(C(N2CCC(N(C(C3C(C=C)CC3)=O)C)CC2)=O)ccc(C)c(F)c1 N1(C(C(CCN(C)C)O)=O)CC(NC(=O)CCc2cnco2)CC(O)C1 C1(C(N2CC(OC)C(C(=O)NC34CCCC3C4)C2)=O)CC(C2CC2)=NO1 C=C(Cl)CC(C(=O)NCC(c1cnn(C)c1)O)NC(=O)CC=CC(C)(C)C c1(C(=O)OC)cc(CN2CCOCC2C(N2CC3CC3C2)=O)ccc1O C1(CNC(c2c(C)csc2)=O)CC(NC(=O)CCc2ccc(=N)[nH]c2)CC1O N1(C(C2CN(C(C)=O)C2)=O)CCC2(CCN(C(c3cc(O)cnc3N)=O)C2)C1 C(=O)(C1COc2ccccc21)NC1(C)CCN(C(c2ccnc3[nH]cnc23)=O)C1 c1(N(C(=O)NCC(C)Oc2ccccc2Br)C)cccc(Br)c1Cl CCC(C)CC(C(=O)NC(CO)C(=O)N(C)C)NC(c1cnn(C)c1C)=O c1(C(=O)NCC2C(NC(C=CSC)=O)C2)ccc(C(F)(F)F)nc1N Cn1nccc1C=CC(=O)NCC1CCCN(C(=O)CCc2ccc(Cl)nc2)C1 Cc1[nH]c2ccc(C(=O)NCCN(C3CC3C)C(c3ccccc3)=O)cc2c1C c1(C(N2CC(SC)C(NC(C3CC3[N+](=O)[O-])=O)C2)=O)cnc2cc(O)ccc2c1 C12(C(=O)NCC3CC(NC(c4cocn4)=O)C3)CCC(CO)(CC1)C2 c1(OC)ccc2cc(C(=O)NCCCC(C)NC(=O)C(O)CN(C)C)[nH]c2n1 N1(C(c2nncn2C)C(=O)NCCOC)CCC2(CC1)OCC(O)C2O c1(N(C)C)ccc(C(=O)NCC2(NC(=O)CN3CC4CC4C3)CCOC2)cc1 C=C(C)CC(C(=O)N1CCN(C(=O)C(c2cnn(C)c2)C)C(CC2CC2)C1)OC C1(CCNC(C(C)=CC)=O)(OC)CN(C(c2cnc(-c3ccncc3)s2)=O)C1 C1(N(C(COCCC)=O)C)CCCN(Cc2cc[nH]n2)CC1 Cc1c(C(=O)NC2CC(NC(=O)CC3CC3C)C2)oc2cc(Cl)ccc12 c1(C(=O)NCC(CN(C)C(C2CCCN2C)=O)O)ccc([N+](=O)[O-])c(Cl)c1 c1(C(=O)NC(C2CCN(C(c3c(C)cncc3)=O)CC2)C)ccnc2[nH]cnc12 N1(CC(c2ccccc2)OC)CC2CCCN(C(c3csc4cncn34)=O)C2C1 N1(C(C(CCC#C)NC(c2coc3c2COC3)=O)=O)CCCC2(CCCO2)C1 N1(C(c2c(CC)c[nH]n2)=O)CCC(NC(=O)CN2CCC(CO)CC2)CC1C C1(NC(c2n(CCC)nnn2)CCCOC)COc2ccc(F)cc2C1 c1(C(=O)NC2CN(C(CN(C(C)=O)C)=O)CC(C)C2)cnn2ccn(C)c12 C1(COC)CCC(C(=O)NCCN(C)C(=O)C2CC2)C1 c1(C(=O)NC(CC(C)C)c2ccccc2)cnc2c(c1)CNCC2 c1(SC)cccc(N2CC3CC(NC(C4(S(N)(=O)=O)CC4)=O)CC3C2)c1[N+](=O)[O-] C1(CNC(C(C)OCC)=O)CCCC2CN(C(=O)Cc3nc(C)no3)CC12 Cn1cncc(C(=O)NCC2CN(C(=O)C(O)C(C)(C)C)CC2(C)C)c1=O CC(C)(CC(=O)NCCN1CCCN(C(C2CCC23CCCO3)=O)CC1)C(F)F C=CCC(C)C(=O)N(CCCN(C)C(c1cccc(OC(C)C)n1)=O)C c1(C(N2CCC(O)(CNC(C(C)C)=O)C2)=O)cc(C2CC2)nc2c1cnn2C C(=O)(CCCCCCCCCO)NC(C)CNC(C12CCC1C2)=O CCCCC(F)C(=O)N1CCN(C(=O)CN(C)C(c2cc(SC)c(C)o2)=O)CC1 C(=O)(CC(C)C(=O)NCC1CCCC1C(N1CC(C)(C)C1C(=O)O)=O)OCC c1(C(C)CC(=O)NCC2(NC(=O)CN3CCC(C)C3)CCCC2)ccc(F)cc1 O=C(CCCC(F)(F)CO)NC1CCCN(C(c2cc3c(cc2Cl)NCC3)=O)C1 c1(C(N(C(CNC(=O)CCC(=O)N(C)C)C2CC2)C)=O)cccc(F)c1 c1(C(N2CCC(C(N(C3CCC(O)CC3)C)=O)(CF)C2)=O)cnn2cccc2c1 N1(C(COCCCCC)=O)CCN(C(C2(OC)CCC2)=O)CC1CC1CC1 Cc1cc(=NC(=O)C2CC(F)CN(C(c3ccc4cnc(C)n4c3)=O)C2)[nH]n1C C(=O)(C(C)(C)F)N(CCN(C(C(C)OCCC=C)=O)C)C(C)C Cc1cc(=NC2CCN(C(c3cn(C)nc3C(C)(C)C)=O)CC2C)[nH]c(CO)n1 C1(F)(CNC(=O)C(O)C2CC2)CC(N=c2ccnc(Sc3ccccc3)[nH]2)C1 Cc1cc(C(C)Nc2cc(NCC(c3ccccc3F)(F)F)ncn2)cc(C)c1 N1(C(CN(CCOC)C)=O)CC2CC(NC(=O)CC3(OCN)CCC3)CC1C2 C1(C(=O)OC)CN(C(=O)C(C)(C)C)CC1c1cccc(Br)c1 CC1CCc2c(C(=O)NC3(C)CN(C(C4CC4c4ccsc4)=O)C3)csc2C1 C=CC(C)(CC)C(=O)NCCCC(C)NC(c1ccccc1SCC(F)(F)F)=O C1(NC(=O)CCC2CC2)CCOC12CCN(C(=O)C(=Cc1cccnc1)F)CC2 C(=O)(CC(=O)N(C1CCN(C(c2snnc2C(C)C)=O)C1)CCO)OC C1(C(=O)NCCC2(O)CN(C(C34CC(CO3)C4)=O)C2)(OCC)CCOCC1 C(=O)(NNC(=O)C(=O)OCC)c1nc(-c2cncc(C(=O)OCC)c2)sc1 CCCCC(C)(F)C(=O)NC1CCCCC1NC(=O)CN=S(C)(C)=O C1(C(C)C)CCC(C(=O)NCC(C2(O)CN(C(C3CC(C)CO3)=O)C2)(C)C)CC1 c1(C(=O)NC(C(=O)NCCS(=O)(=O)NC)C2(C)CC2)cccc(C)n1 C(=O)(CCS(N)(=O)=O)NC1CCN(C(c2c(OC)c(C)sc2)=O)C1 C1(C(=O)OC)CCCC(C(=O)NCC2CCCN2C(=O)C(C2CCCC2)OC)C1 CC(C)(C#N)CCCC(=O)NC1CN(C(C23C=CC(CC2)C3)=O)CC1C1CC1 c1(C(=O)NC2CCCN(C(CC3(C)CC3(Cl)Cl)=O)CC2)ccc(C#N)cc1O C(=O)(C#CC1(C)CCCO1)NCCC(C(C)C)NC(c1ccc(CC)c(Cl)c1)=O c1(CN2CC(C(=O)Nc3nnco3)SCC2)cc(Br)cc(F)c1F C1(CCNC(c2n(CC)cnc2)=O)CCCN(C(c2c(C)ncn2O)=O)CC1 C1(NC(C(CC2CCCCC2)OC)=O)CN(C(=O)C(N)=O)CC1C c1(OCC(C(=O)N(CCO)CCNC(C(CC)N(C)C)=O)(C)C)cccc(C#N)c1 c1(C(=O)NC2C3CN(C(C(C)N4CCC4)=O)CC32)cc2nc[nH]c2cn1 C1(CN(C(c2c(CC)ncs2)=O)C)CCCN(C(=O)C(C)N=[N+]=[N-])C1 N1(C(c2n(CC)cnn2)C(=O)NCCOC)CCC(C#N)CC1 CC1(C)C(C)(C(N2C3CC2CN(C(c2cc([N+](=O)[O-])sn2)=O)C3)=O)C1(C)C c1(OC)ccc(N)c(C(=O)NCC2CN(C(C3CC4(CSC4)C3)=O)CC2C)c1 C(=O)(C1Cc2ccc(F)cc21)N(C1CCCN(C(c2c(CC)nc(C)s2)=O)C1)C c1(C(=O)NCC2CC2NC(C2(c3ccsc3)CC2)=O)ccc2sncc2c1 Cn1cnc(C(N2CCC(CNC(c3c(C(F)F)cnn3C)=O)C2)=O)cc1=O C1(CNC(c2ncn(C(C)(C)C)n2)=O)CC(C2CC2)C1 Cc1nn2c(c1CNC(=O)C(O)CC(F)(F)F)CN(C(=O)C(C)S(N)(=O)=O)CC2 c12nc(Cl)ccc1NC2.c1(CCOC)nnc(CCCNC(=O)C2CC2)n1CC C1(NC(C2C(NC(C(C=C)OC)=O)CC2)=O)CCOCC1(C)C C(C)(C)(CCC(=O)NCc1ccccc1O)NC(c1ccc(CC)cc1)=O c1(NC(C(CC)C)(C)c2nnnn2Cc2ccc(OC)cc2)c(C)cccc1F c1(NC(C(CO)NC(Cc2c(C)n(C)cn2)=O)=O)ccc(O)cc1F c1(OC)cnc(C(=O)NCC(=O)NC2CCN(CC(F)F)C2)cn1 N1(C(C2CCN(CC)C2)=O)CCC2(CC2C(=O)NC2(C)CC3CCC2C3)C1 C1(CNC(CN(CCOC)C(C2OCCC2C)=O)=O)CCCC1C(C)C C1(NC(C(=O)NCCC(N)=O)=O)CN(C(=O)CC2CC3CCC2C3)CC12CC2 c1(C(=O)NCCCCCNC(Cc2n(C)cnc2)=O)cc(C#N)n(C)n1 N1(C(c2ncc[nH]c2=O)=O)CCN(C(=O)COc2ccc(Cl)cc2Cl)CC(O)C1 C(C1c2ccccc2CCN1C(c1cccn1C)=O)NC(CSCCN(C)C)=O C12(NC(CCCC)=O)CCN(C(C3CCN(c4ccncn4)CC3)=O)CC1C2 N1(C(c2ccc(CC)s2)=O)CC(OC)C(NC(c2ccc(Br)cn2)=O)C1 Cc1cc2ccc(C(=O)NC3CCCCC3N(C(=O)C(=O)NC(C)C)C)cn2c1 CC1Oc2c(C(=O)NCCNC(c3ccnc(C(C)(C)C)n3)=O)cccc2C1C C1(NC(C(CCCC)O)=O)CC2CN(C(=O)CC(O)c3ccccc3)CC2C1 C1(C(=O)NC2CCN(C(c3ccc(C(C)C)o3)=O)C2)C2CCN1CC2 c1(C(N2C(C)(CNC(C(CC#C)C)=O)CCC2)=O)cc(OC)ccc1[N+](=O)[O-] C(C)(C)(CCC(=O)NC1CC2(C1)CN(C(C1CN(C(C)=O)C1)=O)C2)OC c1(C(=O)NC2CCCCN(C(CC(C=C)CC)=O)C2)ccsc1S(N)(=O)=O c1(C(=O)OC)cncc(C(N2CC(F)(CNC(=O)C(C)Cc3ccco3)C2)=O)c1 C(=O)(CC(C)C(C)C)NCC1(O)CCN(C(c2n(CCOC)ncc2)=O)C1 N1(C(c2ccc(OC)s2)=O)CCN(C(c2cc(F)cc(F)c2)=O)CC1C#N C1(NC(C(C)(C)OC(CCC)=O)=O)CCN(C(C2COCC2C(N)=O)=O)CC1 C1(NC(c2cc(C)nc(C)c2)=O)C(C)CN(C(c2cnc[nH]2)=O)CC1C c1(C(=O)NC2CCCN(C(C=NOC)=O)C2)ccc2nc(CO)[nH]c2c1 C(=O)(CCCC(F)(F)Br)N1CCC(n2cc(C(N3CCCCC3=O)N(C)C)nn2)C1 c1(C(=O)NC(CC)(C)CCNC(=O)C(CN(C)C)C(C)C)cn2ccnc2cn1 CC#CCCCC(=O)NCCN(CCCCCC)C(C1CCC=CCCC1)=O C1(CNC(c2onc(CC)n2)=O)CCN(C(C23CC2COC3(C)C)=O)C1(C)C C1(OC)(CNC(=O)CC2CC(N(C)C)C2)CCN(C(C2(C(N)=O)CCC2)=O)C1 C1(C(C)=O)CC(=O)N(CC(=O)NCC2(CNC(=O)C(C)C3CCCO3)CC2)C1 C(=O)(C(C)(CC)C(N)=O)N1CCN(C(c2nc(COCC)sc2)=O)C(CF)C1 N1(C(c2ccnc(OC)n2)=O)CC(NC(=O)CCc2ccn(C)n2)CCC1C c1(C(=O)NC2CC2)ccccc1C(=O)NCC1CCCN1C(c1ccon1)=O C1(CNC(C2(OC)CCSC2)=O)COCCN(C(=O)Cc2c(Cl)cnn2C)C1 C12(CNC(=O)CCCCO)CC(CO1)N(C(c1cc(C(F)F)on1)=O)C2 C1(C)(C(N2C(CC)(CC)CCC2)=O)CC=C(C)CC1 Cc1cc(C(=O)N(C)CCOCCNC(=O)CC2OCCN(C)C2=O)cc(O)n1 N1(C(c2cccc(CC)c2)=O)CCC2(NC(=O)Cc3ncoc3C)CC2C1 C1(CC(=O)N(CCC(=O)N2CC(O)C2)CC#C)CC(CC)=NO1 CN1C(=O)CN(CC(=O)NCC2CCN(C(=O)Cc3ccns3)C2)C1=O C(=O)(C(O)CC(F)(F)F)NCCOC1CCN(C(C(C(C)C)NC(N)=O)=O)CC1 c1(NC(C)C(=O)NN(CCN2CCOCC2)C(C2CCCCC2)=O)cccnc1 C(=O)(C1=CCCCCC1)N1CCC(NC(=O)Cc2n[nH]cc2Br)C(O)C1 C(=O)(C(O)C(C)(C)C)NCC1(CNC(C2(OC)CCCC2)=O)CCOCC1 C=CCC(C)(C)CC(c1nnnn1C)NCC1CC1c1c(F)cccc1Cl c1(C(N2CC(N(C(=O)OC(C)(C)C)CC)C2)=O)nc2c(s1)CC(C)(C)CC2 N(C1c2ccccc2CC1NC(=O)CCCC1CC1)C(C(C(C)O)N(C)C)=O Cc1cc(C(=O)NCC2C3CC2N(C(=O)Cc2cnn(C(C)C)c2)C3)nc(C)c1 C1(C(=O)NC(CCC)C2CCCC2)CN(C(c2sc(C)nc2C)=O)CCO1 C(C(CC(C)C)C(=O)NC1CCCC1N=[N+]=[N-])NC(C(C(C)C)SC)=O Cc1nc(C(F)(F)F)oc1C(N1CCOC(CNC(c2cc(Cl)c[nH]2)=O)C1)=O N(C1c2ccccc2CC1NC(C1CCCC12CC2)=O)C(C(CCC)N(C)C)=O c1(CC)nc(C)cn2cc(-c3cccnc3OC(F)F)cc12 c1(SCC)cc(C(=O)NCC2CC2CNC(C2CCCC3(CC3)C2)=O)ccc1C N1(N2C(CC)CCCC2)CCN(C(=O)Cn2cnc(C=O)c2)CC(C)(F)C1.C(C)=O Cc1oc(C(C)(C)C)cc1C(=O)NC1CN(C(C2CC2OC(C)(C)C)=O)CC1F c1(C(=O)NCC2CC2CNC(c2cscc2C2CC2)=O)cc(C(F)F)cc(F)c1 c1(C(N2CCSCC2)=O)ccc(C(N2CCCC2c2ccc(F)cc2)=O)nc1 CC1CC(C(F)(F)F)(NCc2ccccn2)CC(C)O1 C1(C)(C(=O)NCC(C)C)CC12CCN(C(C)CC1CCCCCN1)CC2 c1(CCC(=O)N(C2CCCCC2)CCNC(C2C(C#N)C2)=O)ccccc1F Cc1cccc(CC(C(=O)N(C(CNC(=O)CC(F)(F)F)C2CC2)C)N(C)C)c1 N1(C(c2c(CC)n(C)nc2)=O)CCC2CN(C(=O)C(O)CCSC)CC2C1 Cc1ccc(C(N2CCCCC2C(C)NC(=O)Cc2ccccc2C)=O)cc1C C(=O)(C1=CC2CCCC12)NCCC1CCCN(C(C2(C(C)C)COC2)=O)C1 N1(C(CCSCC)=O)CCN(C(=O)CN(c2ccccc2)C)C(CCOC)C1 C1(N)CCC(C)CC1.CC(C)(CCNC(c1ccc(NC=O)o1)=O)CNC(=O)C1CC1 C12CC3(CCCN(C3)C1=O)C2.c1(SC2(NC(c3cnco3)=O)CC2)ccccc1 c1(CC)cc(C(N2CCOC(CNC(C3CC(OC(F)(F)F)C3)=O)C2)=O)nn1C c1(C(=O)NC2CCCC(NC(c3cc(C)ncn3)=O)C2)cc(F)c2cn[nH]c2c1 CC1(C)CN(C(=O)C(O)C(F)F)CCC1NC(c1ncn(-c2ccccc2)n1)=O CCC(F)(F)C(C)(C)C(=O)NCC(C)CNC(c1cnn2cc(C)cnc12)=O N1(C(CCCC=C)=O)CC2CCC(CNC(c3ccn(CC)n3)=O)C2C1 c1(C(=O)NC(CCOC)CNC(C2C(Cl)(Cl)C23CC3)=O)c(F)ccc(C)c1Cl N1(C(Cc2c(C)nc(S)s2)=O)CCCN(C(C2CCCCS2(=O)=O)=O)C(C)C1 N1(C(CCOCC#C)=O)CCC2(CCCN2C(c2ccnn2CCCC)=O)C1 C=CCCN=C(NCc1cc(C)nc(C)c1)NCC1CCC(C)O1 CN1C2CCCC1CN(C(C1NCC3CCC1C3)=O)C2 c1(C(N2CC(NC(C(CC)SC)=O)C(C)C2)=O)csc(=NC2CC2)[nH]1 N1(C(c2sccc2CO)=O)CC2CCC(C1)N2C(c1c(O)cccc1F)=O C1(C2CCN(c3cnc(F)cn3)CC2)(NC(C2CCN(OC)CC2)=O)CC1 C1(NC(c2cc(C)c(C)nn2)=O)CCC2CC1CN2C(C1(C2CCC2)CC1)=O CCC(C)(CO)NC(=O)CC1C(NC(c2cocn2)=O)CC1O N#Cc1cncc(CC(=O)NCC2CN(C(=O)CC3CC=CC3)C2)c1 c1(OCC(=O)NCC(CNC(c2nn[nH]c2Cl)=O)CO)ccccc1O N1(c2c(F)cnc(C)n2)CCC2(CCCCC2NC(c2n[nH]c3c2CCC3)=O)C1 N1(C(C2C(C)(C)C2(F)F)=O)CC(NC(=O)CCn2cc(Br)cn2)CC1(C)C c1(CC)nnc2n1CCN(N(C)Cc1nnc3ccccn13)C2 C#Cc1c[nH]ccc1=NC(=O)N(c1ccc(F)cc1)CCCCC CC(C(C)(C)C)=CC(=O)N(C(C)CCNC(C1CC(CN(C)C)C1)=O)C C(CC(=O)N1CC(CO)(OC)C1)(N(C1CCCCC1)C(C(=O)NC)=O)C1CC1 CC(C)C(C(C)NC(C1(CC(=O)N(C)C)CCC1)=O)NC(=O)CSc1cccs1 N1(C(c2ccc(CC)o2)=O)CC(NC(=O)CC2CCCN2C(C)=O)CCC1C Cc1cc(NC(=O)C(F)C(C)CNC(=O)Cc2cc[nH]n2)cnc1O C1(CCNC(c2cccc(OC)n2)=O)CC(F)(F)CN1C(C1C=CC=CC=C1)=O CC(C)CC(CNC(c1cccc(N(C)C)c1)=O)NC(C1CCCCC1O)=O N1(C(C(C)OCCOC)=O)CCC(F)(C(=O)NCCCCCCN(C)C)CC1 N1(C(C2CCCC2)=O)CC(O)(C2CCN(C(C3OCCOC34CCC4)=O)CC2)C1 C(CC(O)CC(=O)N1CCOC(CCNC(=O)C=Cc2cc[nH]n2)C1)SC C(c1ccc2c(c1)OCO2)=CC(N1CC(CC=C)(NC(=O)C2=CCCO2)C1)=O c1(OC)ccc(C(N2CCCC(N(C)C(C3CC3CF)=O)CC2)=O)cc1Cl C(=O)(C(C)(C)CC(F)F)NCC(CC(=O)NCc1c(CC)nn(C)c1)C1CCC1 C1(C(N(C(CN(C(c2ncn(C(C)C)n2)=O)C)C)C)=O)CCC2(CCC2)C1 C1(CNC(CCN(c2ccccc2)C)=O)CCCN1C(=O)CSC(F)F Cc1nc2c(o1)CCCC2CC(=O)N1CCN(c2ncnn3cccc23)CC1C N1(C(=O)OC(C)C)CC2(C1)CN(C(C1CC=CCO1)=O)C2.N12CCCCC1C2=O c1(N(C)CCF)nc2ccc(Cl)cc2c(=NC2COc3ccc(F)cc32)[nH]1 C(C(=O)N(C)CCNC(C1CCCN1C(=O)C(C)(C)C)=O)(C(C)C)NC(=O)OC C(=O)(C(F)C(C)(C)O)NCCC1(NC(C(C)NC(C2CCCCC2)=O)=O)CC1 N1(C(C2N(C)C(=O)OC2)=O)CC=C(CCNC(=O)CC2CCCOC2)CC1 C1(C(=O)NCC(C)(COC)CC)(CC)CCCN(C(C2CCC2)=O)C1 C(=O)(C#CC1CCCO1)N1CC(CNC(c2ccc(CSC)cc2)=O)C(C)C1 N1(c2ccc(C#N)cn2)CC(NC(C2(C3CCC3)CCC2)=O)C2CCCCC12 N1(CC(C)C)C(=O)c2ccc(C(=O)Nc3ccc(S(=O)C(F)F)cc3)cc2C1=O C(=O)(N=c1cc2ccccn2[nH]1)C1CN(C(CC(C)OC)=O)CC(C)(C)C1 c1(C(N)=O)cc(C(=O)NC2CCN(C(C3CN(C4COC4)C3)=O)C2)n[nH]1 C(C(C)(C(N)=O)NC(=O)NC1(c2ccccc2Br)CC1)OC c1(C(=O)NCC2N(C(C=CC=CCC)=O)CC(O)C2)cccc2nccn12 C(=O)(C(C)CC(F)F)N1CC(C)C(NC(=O)COC(C)(C)C)C1 C(=O)(C1CCc2c[nH]nc21)NC(CCC(N1CCN(C(=O)NC)CC1)=O)C c1(SCC)oc(C)cc1C(=O)NC1CCCC1NC(=O)CN(CC(=O)NCC)C Cc1nc(C(F)(F)F)ccc1CN=c1[nH]nc(C2CC2)s1 N1(C(c2scc(C)c2)=O)CCCC(NC(=O)CC2CCCO2)C1C c1(NCC2(F)CC(NC(c3cc(CCC)oc3C)=O)C2)ccc(C#N)nc1 C#CCC(C(=O)NC)NC(c1cnc(CNC(C2(C#N)CC=CC2)=O)nc1)=O c1(CCC)cc(C(=O)NCC2(OC)CN(C(=O)C(C(C)C)SC)C2)ccn1 c1(OC)ccc(C)c(NC(c2c(CNC(c3cccn3C)=O)nnn2C)=O)c1 c1(OC)ccc(Cl)cc1C(=O)NCC1CCC1NC(=O)C1=CCCS1 C1(C(C)C)CN(C(c2ccncc2F)=O)CCC1NC(c1cnn(CCF)c1)=O N=c1nc(O)c(CC(N2CCCC(CCNC(=O)CC3=CCCC3)CC2)=O)c[nH]1 N1(C(C(C)(O)c2ccccc2)=O)CC2CC2(NC(=O)Cn2ncnn2)C1 N1(C(CC(C)n2cccn2)=O)CC2(CCNC(C3CCCN3C)=O)CCC1CC2 C(=O)(CCCCC(=O)NCC1(C)CCC(NC(=O)CCCC(F)(F)F)CC1)OC N1(C(C2CC(CC)C2)=O)CCCCCC(NC(=O)Cn2nc(C)oc2=O)C1 C(=O)(C#CC1CCOCC1)N1C2CC(CC(NC(CC3C(C)CC3)=O)C2)C1 c1(C(=O)NCC23CC(NC(C4CC(OCC)C4)=O)(C2)C3)c(C)n[nH]c1C C(=O)(CC(F)(F)C(C)C)NC1CCCN(C(c2c(C)nc(=N)[nH]c2)=O)C1 c1(OC)ccc2nc(N3CC(CN(C)C(c4coc(Cl)n4)=O)C3)c(C#N)cc2c1 c1(OC)cccc(C(=O)NC2CC2NC(=O)CNc2ccc(C)cc2)c1F CCS(=O)(=O)CC(=O)N1CC(CNC(c2cc(C3CC3)no2)=O)C(C(F)(F)F)C1 c1(OC)cccc(C(C(=O)NCC(=C2CN(C(=O)C(C)CF)C2)F)OC)c1 Cc1cc(C(=O)NCC23CC(CN2C(=O)COC(F)(F)F)C3)nnc1C Cc1oc(C#N)cc1C(=O)NCC1CC1CNC(=O)CN1CCS(=O)(=O)CC1 C1(CC(=O)N(CCCNC(C2(C(=O)OC)CC2)=O)C)OCCCC1(C)C c1(C(N2CCC(CNC(CCC#C)=O)CC2)=O)cc(F)ccc1F Cc1c(Cl)ccnc1C(=O)N(C)CC1(NC(=O)COc2cccc(F)c2F)CC1 c1(C(N2C3C(C(N4CC(C)OCC4C)=O)C(C3)C2)=O)c[nH]c2cccc(Cl)c12 Cc1cc(O)ncc1C(c1nnnn1Cc1ccccc1)NC1(C)CC1(C)C CC1(C)CC(C(=O)NC2(c3cccc(F)c3)CCN(C(C3CCC3)=O)C2)CCO1 C1(CCOC)(NC(c2cn(C3CCC3)nn2)=O)CCN(C(=O)COC)CC1 N1(C(c2ccc(SC)o2)=O)CC(NC(=O)Cn2cc(C)cn2)C2CC12 C(C)(CN=c1[nH]cnc(=N)[nH]1)N(C(C=COCC)=O)Cc1ccccc1 C1(CC(=O)NCc2n(C(C)C)ncn2)CN(C(C2CC(=C3CC3)C2)=O)CC12CC2 C(C(CCCC)NC(C1(OCC)CCSCC1)=O)NC(c1cn(CC=C)nn1)=O C(CCN=C(NCC1CCC2(COC2)O1)NC(C)COC(F)F)SC c1(C(=O)NCCOC2CN(C(CC#N)=O)C2)c(O)nnc2c1COCC2 c1(N(CC(C)(C)C)Cc2ccccc2)cnn(C(C)C2CC2)c1 C(CN=C(NC(C1CCCO1)C)NC1CC(=O)N(CC2CCCCC2)C1)SC CCC(C(=O)NCC(O)CNC(c1ocnc1C)=O)OC1CCCCC1 C12(C(=O)NC(CCOC)CNC(=O)C(O)CSC)C3CCC(CC13)C2(F)F Cc1cc(N)c(C(=O)NCCC2CCC(NC(=O)C3=C(Cl)CC3)C2)cc1C C#Cc1cnc(C(N2CCCCC2C(N2CC(O)(c3cnn[nH]3)C2)=O)=O)c(C)c1 Cn1cc2ccc(NC(C3CC(O)CCN3Cc3ccnc(O)c3)=O)cc2n1 N1(C(c2n[nH]cc2Br)C(=O)NCCSC)CCC(S(=O)(=O)c2ccccc2)CC1 C(=O)(CC(C)(C)C(=O)NCC1CCN(C(=O)CNC(N)=O)CC1C)OCC C(=O)(CS(=O)CC)N(CCC(=O)NCCc1ncnn1C)CC=C N1(C(Cc2c(C)ncs2)=O)CCC2(CO)CN(C(=O)CCc3cn[nH]c3)CC2C1 c1(NCc2nnc(C(F)F)o2)nccc(=NCc2cnc(C(F)(F)F)s2)[nH]1 c1(OC)ccc(Cn2cc(C(=O)NCCn3ccnc3C)cn2)cc1 c1(C(=O)NCC(CC=C)NC(c2cc(C(F)F)cc(F)c2)=O)ccc(N)c(F)n1 C(CC(CC)C(=O)N1CCC(N(C(=O)CN(C)S(N)(=O)=O)CCO)CC1)=CC c1(OCC)cc(C(=O)NC2(C)CCN(C(=O)COC3CCC3)C2)cc(Cl)c1O c1(N(CC(N2CC=CC2)C)CC)ccc(C(=O)OC(=O)CSCC(C)(C)C)cc1 Cc1nnc(CC(=O)NCCC2CCC(NC(=O)Cc3nncn3C)C2)o1 c1(C(N2CCC(OC(C)C)C2)C(=O)NCCCSCC)csc(C#N)c1 C1(OC)CCCCN(CC(=O)NCC(C)(Cc2ccccc2)CO)C1=O C1(NC(C2C3CCC(F)(F)C23)=O)CN(C(C2SCCS2)=O)CC12CC2 c1(OC)cccc2cc(C(N3CCCC3CCCNC(C3CC3(F)F)=O)=O)[nH]c12 C1(CNC(CC(C)C2CC2)=O)CN(C(=O)CNS(N)(=O)=O)CCCO1 CC1CCCN(C(C2CCCN(C(C(=O)O)c3ccsc3)C2)=O)C1 C1(NC(c2nn(C)c(O)c2)=O)CC2CCC1CN2C(=O)C(O)Cc1cnc[nH]1 Cc1ccc(C)c(CNC(C2(C)CCCN2C(=O)C=CC(F)F)=O)n1 C12(NC(C(CC)C)=O)COC(C1)C(NC(c1ccc(F)cc1OC(F)F)=O)C2 N1(C(C2C(NC(=O)C(C3CCCCC3)O)CC2)=O)CCC(N2CCC2)CC1 c1(C(=O)NC2CC(C)(CNC(c3c(CC)nn[nH]3)=O)C2)cccc(N)c1C CCC(C)CCCCC(=O)N1CCC(Nc2ccc(C(=O)OC)c(C)n2)C1C c1(C(=O)NCC#CCNC(c2ncccc2C(F)(F)F)=O)cnc2n1CCC2 N1(C(CCN(C(C2CCC(=O)N2)=O)CC)=O)CCC(C(F)F)CC1 C(=O)(C(C)S(N)(=O)=O)NCC(CC(=O)NC1CC(CC(=O)OC)C1)C c1(C(=O)NC2CC(NC(C=CCC)=O)C2)cccnc1-c1nncn1C c1(OC)cc(=NC(=O)C=CCC(C)(C)NC(=O)C(O)C2CC2)[nH]n1C c1(C(=O)NCC2(NC(C(=O)NCC3CC3)=O)CC2)cnc(-c2cccnc2)s1 C(C(CC)(CC)C(N)=O)NC(C1CC(CC)N(C(C2CCCN2CC)=O)CC1)=O CCC(C(=O)N(C(C)(C(=O)NCCC1CCC(=O)N1)C1CC1)C)C(C)(C)CC C1(NC(C(CSC)O)=O)CC2(CCN(C(c3cccc(SC)c3)=O)CC2)C1 C1(C(=O)NCc2cnc(C(C)OC)s2)COCCN1CC(F)(F)F C1(NC(Cc2ccc(C)cc2)=O)CCCC12CCN(C(c1scnc1Cl)=O)CC2 C1(C(N2CC(NC(c3ccc(CO)nc3)=O)C2)=O)C2CCCCC12 c1(OC)cc(N)cc(C(=O)NCC(C)(C)CNC(C2CC2CC(C)C)=O)c1OC c1(C(=O)OC)ccc(C(=O)N(C(C)CCNC(=O)C#CC2CCC2)C)c(OC)c1 c1(C(=O)NCC(CCCC)NC(=O)CC2(OCC)CC2)cc(N)ccc1CC Cc1csc(=NCC(=O)NCC(C2CC2)NC(C2CCCSS2)=O)[nH]1 C1(NC(c2ccc(OC(C)=O)cc2)=O)CCCCN(Cc2cccc(Br)n2)C1 CS(=O)(=O)C1CCC(C(N2CCC(NC(=O)CC(F)(F)C(F)F)C(O)C2)=O)CC1 C1(CNC(c2c(COC)ccs2)=O)CCCN(C(C2(c3ccnn3C)CC2)=O)C1 c1(C(N2CCC(=CCNC(c3nncc(OC)c3)=O)CC2)=O)nnc(O)nc1O C1(N(C)C(c2ccn(CCF)n2)=O)CCCC(NC(=O)CC2CC2)C1 c1(C(N2CCC3C(NC(c4cc(CC)c(C)s4)=O)C32)=O)cc(N)cnc1Cl c1(C(N2CCC(OCCNC(C(C)OC)=O)C2)=O)ccc(CO)nc1 c1(OC)ccc(C(C)NC(c2ccc(OC)cc2)c2nnnn2C2(C)CC2)cc1 Cn1cc(C(=O)NCCn2ccc(C(N3CCC(CCO)C3)=O)c2)nn1 c1(C(=O)NCCC2CN(C(C3N(C=O)CCC3)=O)C2)cc2ccccc2oc1=O c1(CNC(CC2N(C(c3n(CC)ccc3)=O)CC2)=O)ccccc1F c1(CC)ccc(F)c(C(=O)NCC2CCCC(NC(c3[nH]nnc3C)=O)C2)c1F Cc1cc(C(=O)NCc2ccc(C(=O)NCCCC3CCCC3O)cc2)c(C)s1 c1(C(=O)NCC23CC(NC(C4CCC5CCC4O5)=O)(C2)C3)cccc2c1OCO2 C1(CNC(CCCCC#C)=O)CN(C(=O)CCCCOCC)CC(C)(C)O1 N1(C(c2ccc(SC)o2)=O)CCC2CCC(NC(=O)C(C3(O)CCCC3)F)C1C2 N1(C(C(C)CC2CCOCC2)C(=O)NC2CCC2)CCC(S(=O)(=O)C(F)F)CC1 c1(OC)cnc(F)c(C(=O)NC2CC(F)CN(C(c3ccc(CSC)o3)=O)C2)c1 CN1CCN(C(=O)Cn2ncccc2=O)C(CNC(=O)CC2(O)CCCC2)C1 N1(C(CNC(=O)OC)=O)CCC(C2CC2)C1CNC(=O)C(C)S(C)(=O)=O N1(C(C2(C)SCCCS2)=O)CC(C2CN(C(C3COCCC3(F)F)=O)C2)C1 C1(NC(CCCOCCC)=O)CN(C(=O)Cn2cnc(C#N)n2)CCC1C CCCCC(C(=O)NCC1(C)CCCCO1)N(C(=O)C(c1ccccc1)C)CC C1(C(=O)NCC(CC)NC(c2c(Cl)nn(C)c2Cl)=O)CCCNS1(=O)=O c1(OC)ccc2c(C(=O)NCC3CCN3C(=O)C3=CCSC3)ccnc2c1 Nc1ccc(Cl)cc1C(=O)NCC12CC(NC(c3c[nH]nc3C3CC3)=O)(C1)C2 C1(NC(CCC(CC)OC)=O)CCN(C(c2ccc3sccc3c2)=O)CC1(C)C N1(C(C2(OC)CC2)=O)CC2CC2(NC(c2ccc(O)cc2)=O)C1 c1(C(=O)NC(C(C)NC(c2ccc(CC)o2)=O)C)cc2c(Cl)c(OC)ccc2[nH]1 c1(C(c2n(CCC)nnn2)NC2CCCS(=O)(=O)C2)cc2cccnc2o1 c1(SC)ccc2sc(CN(C)CCCCCN)nc2c1 C1(C(C(=O)NCCN(C(c2c(SCC)cccn2)=O)CC)O)CCCCCCC1 Cc1cc(C#N)cnc1C(=O)NC1(C(=O)Nc2cn(C)nc2C)CCC(C)(C)C1 CC#CCC(C(=O)NCCN(C)CCOc1cccnc1)NC(=O)OC(C)(C)C c1(C(=O)Nc2nc(C)cc(C)n2)ncn2cc(-c3cccc(O)c3)sc12 C1(F)(C(N2CC(NCc3cn(C)nc3)OCC2)=O)CCCCC1(F)F CC1(CNC(=O)Nc2ccnc(OC(F)F)c2)CCCCCC1 Cc1c(C(=O)NC(C)CNC(=O)COCc2cccnc2)cccc1O c1(C(N2CC(COC)(NC(=O)C(F)CC3CCC3)C2)=O)nc(C(C)C)ncc1Cl c1(C(=O)NCCCN(C)C(c2cnn[nH]2)=O)ccc2nc(O)cc(O)c2c1 C1(OC)CC(CNC(C2C=C(C)CS2)=O)N(C(=O)CN(C2CCCC2)C)C1 N1(C(COC2(C)CCCC2)=O)CCC(C)(CCNC(=O)CSS(C)(=O)=O)C1 C1(F)(C(N2CC(F)(CNC(c3cc(SC)ncc3)=O)C2)=O)C(C)(C)C1(C)C c1(C(C)NCCCCCCCl)cc(Cl)ccc1Cl C1(C(=O)NC(CC=C)(C)C)CCC(C)(C)N(C(=O)CC2C=CCC2)C1 N1(C(C)=O)CCC(CC(=O)NCC(C)CN(C(=O)CCC2(C)CC2)C)CC1 c1(C(N2CC(NC(C#CC(C)(C)C)=O)C(F)CC2)=O)ccc2cncn2c1 c1(C(N(CCCNC(=O)CSC)CC)=O)cn(CC(=O)N(C)C)nn1 C1(N(C(COCCCC)=O)CCO)CCCN(C(=O)CNC(=O)NC)C1 C1(CCOC)(NC(c2c[nH]nc2F)=O)CCN(C(=O)C(n2nccc2C)C)C1 c1(C(N2CCC(=CCNC(C3C(C)(C)CO3)=O)CC2)=O)cc(O)nc(C2CC2)n1 c1(OCC(=O)N(C2CCCC2O)CCNC(CC)=O)ccsc1Cl C1(NC(c2c(SC)scc2)=O)CC2CCC1N2C(=O)C(C)OC1CCCC1 C1(C(=O)NC(C=C)C2CC2)CC(N=[N+]=[N-])CN1C(c1c[nH]c(C)c1)=O N1(C(C(C)OCCOC)=O)CCC2(CC2)CC1C(N1CC(C)(C#N)C1)=O CC(CC(=O)N1CCCC1C(C)(C)CNC(c1ccccc1C(C)C)=O)C(F)F C1(CC)CCC(C)N(C(C2CC(O)(CNC(=O)CNC(C)=O)C2)=O)C1 C1(C)(C(=O)NC(CC)CNC(=O)C(C)CC2CCC2)CCC(F)(F)C1 n1(CCNC(C2C=CC(NCc3ccc(O)cc3Br)C2)=O)nnc2ccccc12 Cc1ccc(C(C)C(=O)NC2CCC2CNC(c2ccsc2C(F)(F)F)=O)cc1 C(=O)(C1=CC2(CCOCC2)C1)N1C(C)(CC)CC(NC(=O)C(C)(F)F)C1 CCC(CC)(CCNC(C1CCCC(=O)N1)=O)NC(C1OCCCC1(C)C)=O C(C)(N=c1[nH]c(N2CCC(C3CCC3)C2)nc2cc[nH]c12)c1c(C)nc(C)[nH]1 C1(C(=O)NC(C(=O)NCC(=O)NCCC)CC)OCCC1NC Cc1oc(C(=O)NC2CC(CCNC(=O)CCC3CCCO3)C2)cc1CO n1(CC(N2CCC(C(CNC(CCCOC)=O)O)CC2)=O)cnc([N+](=O)[O-])n1 CN1CC(C(=O)N(C)CCN(C)C(c2ccc[n+]([O-])c2)=O)C(C(F)(F)F)C1 N12CC(C(O)C1)N(C)CC1(CC1)CC2=O.C(=O)(CCCc1ccncc1)OC CC#CCCCC(=O)NCCOCCN(C(=O)C(c1ccc(F)cc1)C1CC1)C c1(N2CCC(=CNC(c3cnn[nH]3)=O)CC2)ccncc1[N+](=O)[O-] c1(C(N2C(C)CC(NC(C3(C4CCC4)CC3)=O)CC2)=O)cc2n(n1)CCCO2 CC(C)(C)C(O)C(=O)N1CC2(CC(NC(=O)CN3CCC(O)CC3)C2)C1 CC1CC1C1CC1C(N1CCC(CCNC(C23CC(C)(CO2)C3)=O)CC1)=O N1(C(c2cc(Cl)c(Cl)c(Cl)c2)=O)CCC2C1CCCN2C(C12CC(C1)C2)=O Cc1cc(O)ncc1C(=O)NCCN(C(=O)CC1COC2CC1C2)CC1CC1 n1(CC(=O)NC2CN(C(C3(CN(C)C)CC3)=O)CC2F)cnc([N+](=O)[O-])n1 C1(CNC(CN(C)C)Cc2ccccc2)COC2(CCOCC2)O1 CC1(C)CC2(CC(C(=O)NC3CC(CNC(c4cccn4C4CC4)=O)C3)C2)C1 N1(C(C(C)(C)C2CCC2)=O)CCCCC1C1CCCN1C(C1CC2C=CC1C2)=O Cc1cccc(C)c1C(O)C(N1CCC(C2CCCN2C(=O)CC2CC2)CC1)=O C1(NC(c2c(C)cncc2C)=O)CN(C(=O)Cn2ccccc2=O)C2(CCC2)C1 c1(C(=O)NC(CCNC(C(CCC)C(C)C)=O)(C)C)ccc2c(c1)CCC2(C)C N1(C(C=CC(=O)OC(C)(C)C)=O)CC2CC2(NC(=O)CC(O)c2ccccc2)C1 c1(C(F)(F)F)[nH]c(=NC2COC3(CCOCC3)C2)ccc1Br C1(CNC(C=NOC)=O)CC2(CCOCC2)CN1C(=O)C(C)OC1CCCC1 N1(C(c2cnc(CC)s2)=O)CC(CNC(c2cnc(=N)[nH]c2)=O)C(C)C1 N1(C(CC(=O)OC(C)(C)C)=O)CC2(CC(S(C)(=O)=NC(=O)Cc3ccn(C)n3)C2)C1 C1(NC(COCCOCC)=O)CCCC12CCN(C(c1nnn(C)c1N)=O)CC2 Cc1ccc(COCC(=O)NC(c2ccnn2C)C(=O)NCc2nc[nH]n2)cc1 C(=O)(NNCC(F)F)NCC1(COC)CCCO1 C1(NC(C2(CCOC)CC2)=O)CCC2CC1CN2C(=O)C=Cc1nc(C)cs1 C1(NC(C(C(C)C)C)=O)CC(F)CN(C(c2ccc(CC(N)=O)cc2)=O)C1 C(=O)(C1=NNC(C(F)(F)F)C1)NCc1cn(C)nc1 c1(NC2CN(C(=O)CC3CCS(=O)(=O)C3)C2)ncnc2c1CCC2 S(=O)(=O)(c1ccc(Br)cc1NCc1nc2ccccc2n1C)NC(CC)CO N1(C(CS(=O)(=O)NC)=O)CCC2CCN(c3ncc(C)c(C)n3)CC2C1 c1(C(=O)NCC=C2CCN(C(CC(C=C)(C)O)=O)CC2)cn2nccc2nc1C c1(NC2(CNC(C(CSC)C)=O)CC2)ncnc2c1cnn2C C=CC1(CC(=O)NC2(CC3CCC3)CC2)CN(C(=O)CC2CC2)C1 N1(C(C=NOC)=O)CCCCC1C1CCN(C(=O)C(C)Cc2c(C)noc2C)C1 N1(C(C(C)NC(N)=O)=O)CCOCC1CNC(c1ccc(C(F)(F)F)s1)=O Cc1[nH][nH]c(=NC(=O)C23CC2CN(C(=O)Cc2cccc(O)c2)C3)c1Cl C1(OC)(OC)CC2(CN(C(=O)NCC(C)(C)C3CCCO3)C2C(C)C)C1 c1(C(N2CC(NC(C(c3ccccc3)SC)=O)C(O)C2)=O)cc(C)cc(F)c1N N1(CC(=O)NCCCN(C(=O)Cc2cccc(Br)n2)C)CCC(C)(O)C1 c1(C(C(=O)NCC(CNC(c2cncc(C)n2)=O)C)O)ccc(O)c([N+](=O)[O-])c1 CC1(C(=O)NC2CCC(NC(=O)CCSC(F)(F)F)CC2)CCC12CCC2 C1(C(=O)NC(C(C)NC(=O)CCN2CCC(F)C2)(C)C)CC2CC(=O)C1C2 Cc1nc(C(=O)NC(CNC(=O)C(C)Oc2ccccn2)C2CCC2)cs1 C(C(=O)N1CCCC(C)(CNC(=O)C(O)CC2CC2)C1)(c1ccccc1)=C(C)C N1(C(COCCCC)=O)CC(O)(C2CCCN2C(=O)CCc2ccsc2)C1 N1(C(CC2(NC(C)=O)CC2)=O)CCN(C(=O)CC(C)(C)SC)CC1c1cn[nH]c1 CC(F)CCN=C(NC(C)Cc1ccccc1)N1CCC(CC(=O)N(C)C)CC1 Cc1c(NC(=O)CC2(C)CN(C(=O)COC3CCCC3)C2)ccc(Br)c1Cl N1(C(CC(C=C)CC)=O)CC(NC(C2CCC(=O)N(C)C2)=O)CC12CCOCC2 c1(C(=O)OC)cc(CC(=O)N(CCCNC(=O)C(C)n2ccnc2)C2CC2)[nH]n1 Cc1c(C(=O)NCCC2CCN(C(c3cc4occc4s3)=O)C2)cccc1N Cn1cnc2cccc(C(N3CC(NC(c4cccnc4S)=O)C4CC34)=O)c12 C12(C(N(CC(C)(C)NC(c3cn(CC)nc3C)=O)C)=O)CCC(F)(CC1)C2 N1(C(=O)NC(c2ccccc2)C)CCCC2(CCN2C(c2cc(Cl)ccn2)=O)C1 C1(C(=O)O)CN(C(=O)CCBr)CC12CN(C(c1cnsn1)=O)C2 CC(C)C(F)(CNC(C1C2CCCCC12)=O)C(=O)NC1(C2CCCC2)CC1 C(CC(F)F)(C(=O)NC(c1ccncc1)C)N(C(CCC(C)OCC)=O)C N1(C(C2CC(NC(C3(F)CC3C)=O)C2)=O)CCC(C(=O)OC)CC1 Cn1cc(C(=O)N2CC(=O)N2)c(C(N)=O)n1.c12ccc(cc1)s2 C1(NC(C(C=C)OC)=O)CCCCC12CCN(C(c1[nH]ccc(=O)c1C)=O)CC2 N1(C(c2cccc(N(C)C)c2)=O)CCCC(F)(CNC(C2CCCN2C=O)=O)C1 C12(C(=O)NC3(CC=C)CCCC3)CC(CO)(CN1C(c1ccns1)=O)C2 C#Cc1ccc(C(=O)Nc2c(C)cnn2CC2CCC(C)CC2)cc1C c1(N(C2CCCC2)CCCC)ccc(C)c(OC(c2cccc(SC)c2)=O)c1.OC c1(C(=O)NC2(C3CN(C(=O)C4=COCC4)C3)CC2)cncc2n[nH]cc12 c1(CN(CC)Cc2ccnn2CC2CCCO2)ocnc1C1CCC1 c1(CC(=O)NCC(CCOC)NC(C2CCC(=O)NC2)=O)cc(C(C)C)n(C)n1 C=CCCC(C(=O)O)NC(=O)Nc1ccc(CO)c(COC)c1 C1(NC(c2cc(CCC)ncc2)=O)CCCN(C(c2cc(CC)[nH]n2)=O)CC1 c1(C(N2CC(CN(C(=O)C(C)(C)C(F)F)C)OCC2)=O)c(O)cc(F)cc1F Cc1ncnc(C)c1C(=O)NCCC(C)NC(=O)CC1(CO)CCCC1 C1(N(C(c2c(CCC)nns2)=O)C)CC2CC1N(C(C1CN3CCC1CC3)=O)C2 c1(NC(N2C3CCC2CC(N2CC(F)C(F)C2)C3)=O)ncc2cncnc2n1 N1(CC(=O)NCCN(C(CC2C(C)=NNC2=O)=O)C(C)C)CCc2sccc2C1 c1(N(C)C(=O)NC(CC)=O)ccc(S(=O)(=O)N2CCCC(C)(COC)C2)cc1F CC1(C)CC(=O)NCC1C(N1CC(O)(CCNC(=O)CC2(O)CCCCC2)C1)=O c1(CN2CCC(C#N)(NC(CCN(C)C)=O)C2)ccc2cc(O)ccc2c1 c1(CCC(=O)NC(C(C)NC(c2c(C)ccnn2)=O)CO)cc2ccccc2o1 c1(C(=O)NCC2N(C(C(=O)Nc3c(OC)cccc3)=O)CC2)sc(C)c(C)c1C N1(C(C2C(CC)CCN2C(=O)C=CCN2CCC2)=O)CCc2nc[nH]c2C1 CC1CN(C(=O)Cc2cc(F)cc(F)c2)CCCN1C(C1OCCN(C)C1=O)=O N1(C(c2ccc(C)cc2C)C(=O)NC(C(=O)OC)C)C2CCCC1CC(F)(F)C2 C=CCC(CC(F)F)C(=O)NCC1CCC(C)(C)CN1C(=O)CC1CCC(=O)N1 C1(C(N2CC=CC(NC(C=Cc3ncn(C)c3)=O)C2)=O)CCCC(F)(F)CC1 C(=O)(CCC(CC)CCC)N1CCC(N(C(CC(=C)Br)=O)CCO)CC1 c1(C(=O)NCC(c2ccccc2)CNC(C=C=C(C)C)=O)cn2cccnc2n1 c1(C(C)=O)ccc(COC(C2(C(F)(F)F)CCCS2)=O)cc1 C#CCCCCC(=O)NC(CNC(c1cn(-c2cnn(C)c2)cn1)=O)CCOC CCCCCCC(O)CCC(=O)N(CC(O)CN(C(=O)C=CC=C(Cl)Cl)C)C N1(C(c2nc(C)sc2C)=O)CCOCC(C(=O)NC(c2nc(=O)o[nH]2)C)C1 n1(C(N2CC3C(Nc4nc(CC)nc(Cl)c4F)C3C2)=O)c(C)nc2ccccc12 N#CCCCCC(=O)NC(CCOCCO)C(=O)NCC1(CO)CC=CC1 C1(CNC(CSCC(=O)OC(C)(C)C)=O)CN(C(c2ccsc2)=O)CC1C(F)F c1(OC)ncc(C)cc1CNC(=O)NC(C(F)(F)F)C1CCOCC1 C1(C(=O)NCC(C(C)C)=O)CCCN(C(c2cccc(CN)c2)=O)C1 N1(C(C=COCC)=O)CCCC2CCN(C(=O)Cc3ccc(Cl)s3)CC12 N1(C(C2CC(CCC)C2)=O)CCC1(C)CC(=O)N(C1CCOC1)CCF C1(CC(=O)NCCSCC(=O)NCCN(C)C)CCC2CC12 c1(SC)cc(C(N2CCC(C(C)(C)NC(=O)C=CC3CCOC3)C2)=O)co1 O=C(C(O)C(F)(F)F)NCC1CC2CCC1N2C(c1ccnc(CO)c1)=O N1(C(COC(C)C)=O)CCC(CNC(c2cnc(C(N)=O)s2)=O)CC1C c1(C(=O)Nc2ccccc2Br)cc2ccc(-c3cc4ccccc4o3)nc2[nH]1 C1(O)(CNC(C(C)Cc2cnco2)=O)CCN(C(C2CC3(CCC3O)C2)=O)CC1 c1(C(N(C2CCN(C(C3(C)CCCOC3)=O)C2)C)=O)cc(OC(F)F)nc(Cl)c1 n1(C2CCCN(C(C=C(C)c3ccsc3)=O)C2)cc2ccccc2n1 C1(NC(CC(CCC)O)=O)CN(c2ncc(I)cn2)CC12CCOCC2 N1(CCC(N2CC(O)CC(NC(COC)=O)C2)=O)CCCc2ccccc21 c1(OC)c(F)cc(Br)cc1Br.c12ccc(cn1)-c1cncnc1C(=O)N2 C12(CNC(CCC#C)=O)CCCCC1CN(C(=O)C(C)(C)C1CCC1)C2 Cc1nc2sccn2c1C(=O)NC1CC(CNC(c2ccc3cncn3c2)=O)C1 C(C(CC(F)(F)F)NC(=O)C(C1CCC1)C1CCC1)NC(C(C)O)=O C1(NC(c2cncc(C)c2C)=O)CC2(CCN(C(=O)C=Cc3ccn(C)c3)C2)C1 N1(CC(C)C)CCN(CC(=O)N(CCCc2ccccc2)C)CC1=O c1(COC(C)C)ccccc1CC(N1CCCC1CNC(=O)C(C)CN(C)C)=O N1(C(c2c(NC)scn2)=O)CCC2(CCCN(C(c3c(C)noc3C)=O)C2)C1 CC1=NOC(C)(C(=O)NC2CN(C(c3ccc(N(C)C)cc3)=O)CC2C)C1 CCC(O)C(C)C(=O)NCCC1(NC(=O)CNC(c2ccc(Cl)cc2)=O)CC1 C(=O)(C#CC(C)(C)CNC(=O)CC1(N(C)C)CC1)NCCCC1CC(C)C1 N#Cc1cncc(C(=O)NC(CC(=O)NC23CCC(CC2)C3)C2CC2)c1 c1(C(=O)NCC2OCC(CNC(C(=O)N(C)C)=O)C2)cccc(N)c1 C(=O)(C(CC1CC1)NC(=O)CC(C)N(C)C)N(CC(C1CC1)OC)C c1(NC(C2COCCN2c2ncc(C(F)(F)F)cn2)=O)nc(Cl)ccc1F c12cccnc1COC2=O.C1(C(=O)NCC2(CC3CCC3)CC2)CCCC(OC)C1 C=C(C)CCC(C)NC(=O)CCCCNC(=O)CCC(=O)C1CC1 C(=O)(CCC(C)(C)F)NCCC(C)CCNC(=O)CNC(c1ccnn1C)=O Cc1c(Br)noc1C(=O)NC1CCCC1NC(=O)C(N1CCNC1=O)C C12(C(=O)Nc3ccc(NC(CC(=O)N(C)C)=O)cc3)CCC(CC1F)C2 c1(C(=O)Nc2ccc(OC)nc2)ccc2c(C(=O)Nc3cnc(O)[nH]3)n[nH]c2c1 CCC1=NOC(C(=O)NCC2CCN(C(=O)NCc3ccco3)CC2)C1 C(C1=NOC2CN(C(c3cc(CO)[nH]n3)=O)CC12)NC(C(C)=C1CC1)=O C#CCCCCC(=O)N(C)CC1CC(F)CN1C(C1(CCOC)CCCC1)=O N1(C(C=C(C)C2CC2)=O)CCC(C(=O)NCC2CC(C)(C)CO2)CC1 c1(NCC)ccc(S(=O)(=O)N2CCN(CCNC(C)=O)C(C)(C)C2)c2ccncc12 c1(C(=O)NC(C(C)NC(CCC#C)=O)C)oc2c(Cl)cc(Br)cc2c1C C1(NC(c2n(CC=C)ccn2)=O)CCN(C(c2ccsc2Cl)=O)C1C C1(O)(C(C(=O)N(CCC(=O)OC)CC=C)F)CN(C(=O)C(C)CC2CC2)C1 C1(CC)CN(C(C2OCC3CCCC23)=O)CCN1C(=O)C(O)C(C)C C(Cc1ccsc1)(C(=O)NCCCN(C(=O)Cc1ccc(C)o1)C1CC1)NC=O C1(CNC(C(CCC)CC)=O)CCCC12CCN(C(C1(C#N)CCCC1)=O)CC2 CC1CN(C(=O)C(C)(C)C2(O)CCNC2)CCC(c2ccccc2)O1 c1(CN(CCCOC)CCO)nc(-c2ccc(C)o2)no1 N12CC(C1)C(OC)C(=O)NCC(=O)NCC2=O.C1(COCC)CCCC1 CCC(O)C(C)(C)C(=O)NCC1(OC)CN(C(c2cc(Cl)ccc2F)=O)C1 N1(C(N(S(=O)(=O)CC)CCC)=O)CCC2(CCC(C(=O)NC)C2)CC1 N1(C(Cn2c(C(C)C)ncc2)=O)CC2C(CN(C(=O)CN(C)CCO)C)C2C1 c1(C(=O)OC)cncc(C(=O)NC2CC2CNC(c2ccc(C)c(N)c2)=O)c1C Cc1cc(N)c(C)nc1C(N1CCC(O)(C(C)NC(c2ccn(C)n2)=O)C1)=O N1(C(c2ccc(OCC=C)cc2)=O)CCN(C(=O)C(F)C2CCC2)CC1C c1(C(=O)NCC2CN(c3ncnc(C(F)(F)F)c3Br)C2)cnc2[nH]ncc2c1 N1(C(COCCCC)=O)CCCC1(C)C(=O)NCC1OCCC1C c1(OC)ncnc(OC)c1C(=O)N(CCCCNC(=O)CN(C)C)C C1(NC(CC(C)SC)=O)COCCN(C(c2ccc(OC(C)(C)C)cn2)=O)C1 CCCCCC(C)CC(=O)NCC(C)CNC(c1cc(-c2ccncc2)no1)=O CN=c1cc(C(=O)NCC2(CNC(C3CCSC3)=O)CC23CCC3)cc[nH]1 Cc1c[nH]c(C(N2CCCC2(C)C(=O)NCCN2CCOCC2)=O)c1C Cc1ncc2n1CC(C(N1CCC(CF)(NC(C3CC3C)=O)C1)=O)CC2 Cc1ncc(C(N2CC=CC2CNC(c2cn(C(C)(C)C)nn2)=O)=O)cn1 c1(C(=O)OC)cnoc1-c1cn(C(C)C(=O)N2CCC2C2CCOCC2)nn1 N1(C(CCC#C)=O)CC2CCC1CN2C(C1CCCN1c1ccccc1)=O C(=O)(C1CN(C2CC2)c2ccccc21)NCCCNC(C1CN(S(C)(=O)=O)C1)=O N1(C(C(C2CC2)OCC)=O)CC=C(C(=O)Nc2ccc(C)c(O)c2)CC1 CC(C(=O)NC1CN(C(c2cc3ccsc3s2)=O)CC12CC2)S(N)(=O)=O CC(CC(=O)N1CC2CC(NC(C3(n4cncn4)CC3)=O)C2C1)CC(C)(C)C N1(C(=O)NCC(C)OCC=C)CCC(c2ccnn2C)C1 Cc1c[nH][nH]c1=NC(=O)C1CC(NC(C2(C)CC2(F)F)=O)C1 C(CN=C(NCC1CCC1)NCC1CC2CCC1CC2)C1CCC(OC)CC1 c1(OC)ccc(CCC(N2CCN(c3nc(O)cs3)CC2)=O)cc1Br C(=O)(C(C)CNC(C1CCCC1OC)=O)N(CC)Cc1ccoc1 CCCC(CC)C(=O)NC1CC2CC1N(C(=O)C1=COCCC1)C2 C(=O)(CCCC(F)(F)F)NC(c1ccc(C(C)C)cc1)CNC(C(CC)O)=O N1(C(C(C)=CC)=O)CCC(NC(=O)CCCCCc2ccccc2)CC(C)(C)C1 CCCCC(CNC(=O)C(C)NS(C)(=O)=O)NC(=O)Cc1sc(C)nc1C N1(C(c2c(C)cno2)=O)C2CCC(C2)C1CNC(c1ncsc1C(C)C)=O C(=O)(C(F)C(C)(C)O)NC(c1ccc(F)cc1)CNC(C=C(CC)C)=O c1(C(=O)NC2CCCN(C(CC3CN(C)C3)=O)C2)ccc2nn[nH]c2n1 c1(C(=O)OC)c(C)sc(C)c1NCC1CC(F)(F)C12CC2 N1(C(C2CCC(CC)O2)=O)CCCCC1C1(NC(c2nc(O)sc2C)=O)CC1 c1(C(N(CC(C)(C)NC(c2ccc(C)c(O)c2)=O)C)=O)cn2cccc(Cl)c2n1 Cc1ccc(CCC(N2CCC(CN(C(=O)CCC(C)(C)F)C)C2)=O)cc1C C1(NC(C2CC3(C2)CC3F)=O)CC2CN(C(C34CCC(O)(CC3)CC4)=O)CC2C1 CC(C)CCCC(=O)NC1(C)CCN(C(c2cnn(C(C)(C)C)c2Br)=O)C1 c1(C(=O)NCC2CC(C)(C)CN2C(=O)CC(F)F)cc(Cl)c(F)cc1[N+](=O)[O-] C1(C(=O)NC(c2cn(C)nn2)C(=O)N(CC(C)C#N)CC)CCCC(C)(C)C1 C1(CC=C)(NC(c2csc(C(F)F)n2)=O)CCN(C(c2nn(C)cc2C)=O)CC1 C(CC(C)(C)C(=O)N(CCCNC(c1sccc1SC)=O)C1CC1)OCC c1(C2C(CC)CCC2)nc(-c2cccc(Cl)c2)nn1CCN(C)C N1(C(c2c(C)nc(C3CC3)o2)=O)CCN(C(=O)CCCCC2CC2)C2CCC12 c1(C(=O)NC(C(C)NC(C(C)C(F)F)=O)(C)C)cccc2nc(C(F)F)sc12 N1(C(CCSCC)=O)CCc2ccccc2C1CCNC(=O)CCS(N)(=O)=O c1(C(N2CCCC(N(C(CNC(CC)=O)=O)CC)CC2)=O)nccc2nn[nH]c12 C(CCSC)(C(=O)NCC1(F)CCN(C(C2CN(C(C)C)C2)=O)C1)OC C(=O)(C(C)(C)C(=O)N1CC=CC(NC(=O)Cn2cc(Cl)cn2)C1)NC N1(C(c2ccc(-c3ccccc3)cc2I)=O)CC(S(=O)(=O)C2COC2)C1 C1(CNC(CCN(CC)CC)=O)CCCN(C(=O)C(C)(C#N)CC)CC1 C(=O)(C(CCC(C)(C)C)N(C)Cc1ccc(C(C)C)cc1)NCC c1(C(=O)NCC2N(C(C3C(CC)CCC3)=O)CCCC2)cc(Cl)ccc1N C(=O)(C1=CCN(C(C2CC3C(C2)C3(F)F)=O)CC1)NC1(C(N(OC)C)=O)CC1 CC(C(=O)N1C(C(=O)NCC(O)CC2CCCC2)CCC12CC2)S(C)(=O)=O N1(C(c2cc(C)ns2)C(=O)NCCC2CC2)CC(F)(F)CCC1C c1(OC)cc(C(N2CC(CNC(=O)Cc3ccno3)CCC2C)=O)cc(F)c1F CP(C)(=O)C1CCC(C(=O)NCC(N)CC2CCCC2)C1 c1(C(N2CCC(C)(CNC(C3(CC#C)CC=CCC3)=O)C2)=O)n[nH]cc1[N+](=O)[O-] C#CCCCC(C)C(=O)NCC(C(C)(C)C)NC(c1cc(C)n(C(F)F)n1)=O C1(c2nnnn2C)(C(c2ccc(Cl)cc2)C)CNC(=O)Cc2ccccc2CC1 C1(CC)CCCCN1C(C1CC(NC(C2(CC)CC2)=O)C(O)C1)=O c1(NC(c2nc(C)oc2)=O)ccc(NCc2ccc(CO)cc2)nc1 C1(C(N2CCCCC(NC(CN(C)S(N)(=O)=O)=O)C2)=O)CCn2nncc2C1 C12(C(N(CCCN(C(c3ccc(NC)nc3)=O)C)C)=O)CCC(CC1=O)C2(C)C c1(C(=O)OC)ncccc1NC(=O)N(C1CCCC1)Cc1ccc(COC)o1 C(=O)(C(CNC(=O)C(C)C(C)(C)C)CC(C)C)NC(CCC)C(=O)NC C(c1ccccn1)=CC(=O)NC1(C)CC(NC(=O)Cc2cc[nH]n2)C1 C=C(F)C1(CC(=O)NC2CC(C(=O)NCC(=O)N(C)OC)C2(C)C)CCC1 c1(C(=O)NC(CCC)C(=O)NC2CCC(C3CC3)C2)cccc(F)c1C O=C(CCCn1cccc1)NCC(C1CC1)NC(=O)CCN1CCC(F)C1 C(=O)(C(C(=O)NC1CC(N(N2CCN(CC(C)O)CC2)C)C1)OC)OC.C=O c1(C(=O)NC2(CO)CCN(C(CCCOC)=O)C2)cn2c(n1)CCCC2C O=C(C#CC1CCCCO1)NCC1CCN1C(=O)COc1ccc2c(c1)OCO2 N1(C(c2ccc(COC)s2)=O)CC(O)CC1CNC(C1(C)CCCCC1)=O C1(C(N(CCC(=O)O)CC=C)=O)CCc2cc(C)ccc2O1 C(=O)(C#CC1CCC1)NC(C1CC=CCC1)C(=O)NCCCNC(=O)OC c1(C(=O)NCCCCNC(C=CC=CCC)=O)ccnn1C(C)C N1(C(CN2C(C)CCC2)=O)CCC(C(=O)NCCCC2(O)CC2)C12CCC2 C1(CC=C)(NC(C2CC2C2CC2)=O)CCN(C(c2cc(OC)ncn2)=O)CC1 N1(C(C(C)(C2CC2)NC(Cc2cn(CC)nc2)=O)=O)Cc2ccc(C#N)cc2C1 Cc1cc(Br)ccc1C(N1CCCC(N(C)C(c2cn(C)cn2)=O)C1)=O C1(NC(C(CC=C)C)=O)CS(=O)(=O)C2CN(C(=O)C#CC3CC(F)(F)C3)CC12 c1(C(=O)NC(CC)CN(C(=O)CC2C=CCC2)C)cnc(S)nc1 C(CCC(=O)NC(c1ccccc1)CNC(=O)C(c1cccnc1)C)=CC(C)C c1(C(N2CCCC(CC=C)(NC(c3cc[nH]c3)=O)C2)=O)ccc2cccnc2c1 Cc1ccc(C(F)(F)F)cc1CN1CC(O)C(O)C1C(=O)O CCC(CC(F)(F)F)C(=O)NCCN(C)C(c1cccn2nncc12)=O C1(CNC(C(CCCC)C)=O)CC2(CCC2)CN1C(c1ccc(N)cc1Cl)=O c1(-c2nnc(-c3c(OC(F)F)ccc(C)c3)o2)cc2n(c1)CCS(=O)(=O)C2 c1(C(N2C(CNC(CC(=O)OC)=O)CC(O)C2)=O)cn(C)c(=O)c2ccccc12 Cc1ccc(C(C2CCCN2C(=O)OC(C)(C)C)NS(=O)(=O)CC(F)F)cc1 c1(C(N(CC=CC(=O)N(C2CCN(CC)C2)C)C)=O)csc(C)c1N c1(C(=O)NC2CCN(C(C3CNC(=O)N3)=O)CC2O)n[nH]c2c1CCOC2 N1(C(c2ccc(CC)[nH]2)=O)CCC(C)C(NC(C2(C(F)(F)F)CCCC2)=O)C1 CC(C)C(C)CC(=O)N1CCN(C(c2cc(O)nc(O)n2)=O)C(CF)C1 N1(C(C(CC=C)C)=O)CCC(COC)(NC(=O)CC2CN(C(C)=O)C2)CC1 N1(C(C23COCC2C3)=O)CCCCC1CN(C(=O)CSCC(F)F)CC1CC1 CC(CNC(c1coc(C2CC2)n1)=O)(CO)NC(c1ccc(Br)o1)=O C1(NC(CCc2onc(C)n2)=O)CCSC12CN(c1nc(Cl)nc(C)c1F)C2 c1(NC(C(=O)Nc2cccc(CC)c2COC)=O)c[nH]c2ccc(Cl)cc12 c1(C(CO)NC(C2C(C)(C)NC2)=O)ccccc1F N1(C(N(C2CCCCC2)CCNC(C)=O)=O)CCCC(C)C1CO CCCC(C(=O)N1CCCC1CNC(C1OCCCO1)=O)S(N)(=O)=O N1(C(Cc2c(C)n[nH]c2C)=O)CCCC2(C1)CN(C(C1CC(C#N)C1)=O)CCO2 C1(CNC(C=CC=CC)=O)CC(C)N(C(c2nnn(-c3ccn(C)n3)c2C)=O)C1 C1(NC(c2c(CC)nco2)=O)CC2CCC1C(NC(=O)CCOC)C2 C(=O)(C1=CCCC1C)NC(c1cccnc1)C(=O)NC(CCCC=C)C1CC1 C1(NC(C2C(C)=C2)=O)CN(C(c2cnc(S)n2C)=O)CC2(CCC2)C1 Fc1ccc2sc(CN3CCN(c4ccc(Br)cn4)CC3)nc2c1 Cc1ccc(CC(=O)NCC(O)CCNC(c2ccc3c(c2)CC3)=O)c(F)c1F C(CN=C1NCC2(CCCC2)N1)c1ccc(OC)cc1OC CC1(C)CN(C(=O)CCc2cnccn2)CC1CNC(C1(CF)CC1(F)F)=O c1(C(=O)NC2C(CC)CN(C(=O)C3=COCCO3)C2)scc2c1CCCC2 c1(C(=O)NCC2CN(C(C(N3CCC(C)CC3)=O)=O)CC2C)n[nH]c2c1COC2 Cc1cc(C)n(Cc2ccc(C(=O)NCCCNC(C3CC3(F)Cl)=O)o2)n1 CC1OCCC1C(=O)NCC1CC(C(=O)NC(C(N)=O)C2CC2)C1 N1(C(c2cc(CNC(C(C)(CO)OC)=O)no2)=O)CC2(CCCO2)C1 C#CCC(CC#C)C(=O)N1CC(NC(=O)CCc2ccc(F)cc2)CC(C)(C)C1 C1(CNC(C2CN(C)C(=O)CC2)=O)CC12CCN(C(C1CN(C3CC3)C1)=O)CC2 O=C1CC(NCCN2CCN(Cc3ccccn3)CC2)CC1(F)F Cc1cc(C(N2CCC2C(=O)NC(C)C)=O)c[nH]c1=N C12(CC(=O)N(CCC(C)NC(CCc3onc(COC)n3)=O)C)COC(C)(C1)C2 C1(C)(CNC(C2ON=C(CC)C2)=O)CCN(C(C23CCCC2C3(F)F)=O)CC1 c1(NC2CCCC(CC)C2)ccc(C(C)C)cc1S(=O)(=O)NCC1CCOCC1 Cc1cccc(N)c1C(=O)N(C)CCC1CCCCN1C(c1ccoc1)=O CC1(NC(=O)C(O)CN2CCCC2)CN(C(=O)C(C)(C)NC(C2CCCC2)=O)C1 C12(C(N3CC(n4cc(C(=O)NCCOC)nn4)C(O)C3)=O)CC1COC2(C)C N1(CCC2N(C)CCC2)CCOCc2ccc(Br)cc21 Cc1cc(C(=O)NCC(C2CCCC2)NC(c2ncccc2F)=O)c(Cl)cc1F C1(CNC(CC(CC)C)=O)CN(C(=O)C(C2CCC(=O)N2)C)CCC1(C)C C1(C(=O)NC(CN(C)C(c2sccc2Br)=O)(C)C)C(C)(C)C1(F)F c1(C(C(=O)NCCCCNC(C(CN(C)C)(C)C)=O)(F)F)cc(Cl)ccc1Cl c1(C(=O)NCCN(C(=O)CN(C)C(N)=O)C(C)C)cn2c(n1)CCC(C)C2 C1(C(=O)NC2CC3(C(C(N(C)CC4CC(F)(F)C4)=O)C3)C2)CCCCCN1C Cc1nn(C)c(N2CC(n3cc(NC(=O)C(O)CC(C)C)cn3)C2)c1Cl Cc1ccc(C(=O)OCC=CCO)c(N(C(=O)CCC(C)C)C(C)(C)C)c1 c1(C(=O)NCCC2CCC(NC(CN(CCC#C)C)=O)C2)ccc2sncc2c1 c1(C(=O)NCC2N(C(c3c(C)n[nH]c3)=O)CC2)cc(Cl)ccc1N C1(NC(C(c2ccccc2)N)=O)CCN(c2ccccn2)CC1 c1(N2CCCC(OC(C)C)C2)nc2c(c(=NCc3nc(O)n[nH]3)[nH]1)COC2 N1(C(C2C(C)CC2C)=O)CCC(N(C)C(C2CC(Cl)(Cl)C2)=O)CC1 c1(Nc2c(N(C(C(=O)OCC)C)C)ncnc2)cccc(C(=O)OC)c1C N1(C(c2cccc(C)c2)=O)CC(C(N2CC(OC(=N)O)C2)=O)CC(C)C1 C1(NC(C(c2cccc(C)c2)N)=O)C2CCC(C2)C1C(=O)NC1CCCOC1 Cc1cc(COC(c2scnc2C2CCCC2)=O)c(O)nn1 C1(C)(C(=O)NCCCN(C(c2cc(CCOC)on2)=O)CC)CCCNS1(=O)=O N1(C(C(c2n(C)ncc2)(F)F)=O)CC2CCN(C(=O)C(O)P(C)(C)=O)CC12 N1(C(c2c(CC)nc(C)[nH]2)=O)CC2CN(C(=O)C(F)CN(CC)CC)CC2C1 N1(C(C=CCCC)=O)CC2(CCNC(C3(C(N)=O)CCC3)=O)CCC1CC2 c1(C(=O)NC(C)CCCNC(=O)Cc2cccc(O)c2)ncnc2c1OCCO2 C1(CCC)CCCC1C(=O)NCC1CC(NC(=O)COc2cn[nH]c2)C1 c1(OC)ccc(Br)cc1CCC(N1CC2C(C(N3CC4(CCC4)C3)=O)C2C1)=O C1(CNC(C2CCCC(C)CC2)=O)C2CCCC1N(C(=O)Cc1ccoc1)C2 C#CC1N(C(c2cccc(NC(=O)Nc3c(F)cccc3F)c2)=O)CC1(C)C C1(C(N(C)C)=O)CN(C(c2cccc(C(=O)NC3CCCC(N)C3)c2)=O)CC12CC2 c1(CN2C(C(=O)NC(C(C)C)CO)CC(C)C2)ccc(N(C)C)c(C(F)(F)F)c1 C1(NC(C(C)O)=O)CN(C(C2CCN(CCF)CC2)=O)CC1n1cccn1 c1(CC(=O)NC2COCCC2NC(C2(n3cnnn3)CC2)=O)ccc(Cl)cc1F N1(C(CN(C)CC)=O)CC2CCCC2(NC(=O)C(c2ccc(Br)cc2)C)C1 c1(CC(N2CCC(NC(C=C(CC)C)=O)C2CC)=O)cnc(Cl)cc1C C(c1cc(Br)ccc1F)=CC(=O)NC(c1nc(C(CC)C)[nH]n1)C C1(CNC(C(CC#C)C)=O)(CO)CC12CCN(C(c1ccccc1CO)=O)CC2 C1(F)(CNC(c2ccn(CCCC)n2)=O)CCN(C(c2oc(C)cc2C)=O)C1 c1(CC)nc(C)oc1C(=O)NC1CCOCC1C(=O)NCCC1(C)CC1 N1(C(C(C)=CC)=O)Cc2ccccc2C(NC(C2(COC)COC2)=O)C1 c1(C(=O)NCC(CCNC(c2c(CC)non2)=O)O)cc([N+](=O)[O-])ccc1C c1(OC)cccc(C)c1C(N1CCN(C(=O)CNC(=O)C(O)C2CC2)CC1)=O Cc1snnc1C(=O)N(C1CC1)CC1CCCN1C(c1ccsn1)=O C1(C(N2CCCC(CCO)C2)=O)CC(O)CN1C(=O)CCc1ccccc1F C1(NC(C=C(C)Cl)=O)C2CC3CN(C(=O)CCc4n[nH]c(=N)s4)C1C3C2 C(C(C)CC(=O)N1CCC1CNC(C1CCS(=O)(=O)C1)=O)OC CC(CC(=O)N1CCC(N(C)CCO)C1)C(C)(C)NC(C1COCC1(C)C)=O N1(C(C(C(C)C)SCC)=O)CCN(C(C2(C)CC2)=O)CC12CC2 N1(C(CCCC2C(C)C2)=O)CCOCC(NC(C2(n3cnnn3)CCOCC2)=O)C1 c1(C2CCN(C(C34C(CN(Cc5nc(C)[nH]n5)C3)C4)=O)C2)cccc([N+](=O)[O-])c1 C#CCC(CC(F)F)C(=O)NC(C(N1CC(F)CC1C)=O)C1CC1 c1(N2CC(C)(C)OC(CNC(c3cnns3)=O)C2)nc(Cl)nc2[nH]cnc12 c1(C(C(=O)NCC(C)NC(=O)CCn2cc(Cl)cn2)O)cc(F)c(F)cc1F Cc1c(C(=O)NCCC2(NC(C3COC4(CCC4)C3)=O)CC2)cccc1F C1(C(=O)NCCC(C)N(C(=O)C=CC2CC2)C)Cc2nccnc2C1 CS(=O)c1cccc(C(=O)NC2CC(NC(c3cc(O)ncc3Br)=O)C2)c1 c1(CC(=O)NCCCCNC(c2c(C)nc(CC(C)C)o2)=O)c(F)cncc1Cl c1(C(=O)NC2CCN(C(c3ccc(COC)s3)=O)C2)n[nH]c2nccc(Cl)c12 c1(C(=O)NCC2N(C(c3n(CC)nnc3)=O)CCCC2)cccc2ncccc12 N1(C(C2(CC)COC2)=O)CC(C2CCCN(C(=O)CC3CC4(CCC4)CO3)C2)C1 C(=O)(C(C)C(O)C(C)CC)NCCN(C(CCc1cccc(NC)c1)=O)C(C)C c1(C(=O)NC(CCOC)CNC(=O)COCC(F)F)cccc2c(C)ccnc12 c1(C(=O)NCC2C(C)CN(C(=O)C(O)C3CCC3)C2)cc2ccncc2s1 CCS(=O)(=O)c1ccccc1C(=O)N(CC(C)(C)NC(C1COC(=O)N1)=O)C C1(CNC(C(F)=C(C)C)=O)CC(C)N(C(C2CC(CF)C2)=O)C1 CC#CCCCC(=O)NCC(CCCC)NC(c1c(C(F)(F)F)coc1CC)=O N1(C(=O)OC(C)(C)C)CCOCC1CCOC(C1CC(=O)N(CCC2CC2)C1)=O c1(C(=O)NCC(C)NC(c2ccc(OCC)nc2)=O)ccc(CC)c(OC)c1 CCCC(C(=O)N1CCCC1CCCNC(=O)C=C1CCCC1)N(C)C c1(CC)nc(C(=O)NCC2(C(=O)NCCC#CCO)CCCCC2)c(C)o1 N1(C(C2(C)C(C)(C)C2)=O)CCC(C2CN(C(C3CC4(CCC4)CO3)=O)C2)CC1 c1(C(=O)NC(Cn2cc(CSC)nn2)C)ccc2ccc(C)nc2n1 C1(C(=O)NC(c2ccc(N(C)C)cc2)C)CN(C(=O)C=C2CC2)CC1CC(C)(C)C c1(NC(C)=O)cccc(CC(=O)NCCCC(C)NC(=O)C(O)C(C)C)c1 C(=O)(C1COc2cc(C)c(C)cc21)NC1(NC(C(CCOC)OC)=O)CC1 c1(NC(C2CC2C(N2CCC2CO)=O)=O)cc(O)c2ccccc2n1 C(=O)(CS(=O)(=O)Cc1cccs1)NC(CCNC(c1c(CC)cncc1)=O)C c1(C(=O)NC2C3CN(c4cc(C(C)C)nc(Cl)n4)CC32)c[nH]nc1S(N)(=O)=O c1(C(N2CCN(C(C(C)C3CCC3)=O)CC(O)C2)=O)cc(S(N)(=O)=O)ccc1O c1(C(C(=O)NC2(c3nnc(C(=O)OCC)s3)CC2(C)C)(F)F)ccc(F)cc1C C12(CNC(CCC3CCCN(C(c4c(C)n[nH]c4)=O)C3)=O)CCC(C1)C(=O)N2 c1(C(=O)O)ccc2nc(C3CC3)oc2c1.C12CCN(CC1)CC(C1CC1)N2 O=C(C1=NOC2(CCCN(S(=O)(=O)C3CCOCC3)C2)C1)N1CCC(F)C1 Cc1cc(C(C)C)ccc1C(N1CCC(NC(c2cc(O)ncn2)=O)C(F)C1)=O CCN=c1ccc(C(N2CCN(C(=O)CC3(CSC)CC3)C3CC23)=O)c[nH]1 Cn1cncc1C(O)C(=O)NCC1(F)CN(C(=O)CCn2ccnc2)C1 CC1CCCCC1(CNC(c1nc[nH]c1C(F)(F)F)=O)NC(=O)C=CCO C(=O)(C1=C(C)OCCS1(=O)=O)NC1CCC(CCNC(c2cc(OC)no2)=O)C1 C(=O)(C(C)(C)C(=O)N1CCCC1)NC1C(NC(CCC=CC)=O)CCCC1 C1(C(N2CC(O)(CN(C(C(C)OCC3CC3)=O)C)C2)=O)CC2(C1)CC(CO)C2 C(=O)(C1=CC2(CCN(C(=O)C=Cc3nccs3)C2)C1)NCC(CC(=O)NC)C Cn1cc(S(C)(=N)=O)c(CNC(c2ccc(Cl)cc2C(F)F)=O)n1 N(C1CCOc2ncccc21)C1CCN(C(=O)OC(C)(C)C)CC1(F)F c1(OC)ccc(C(=O)NC2CN(C(c3cc(C(N)=O)cc(F)c3)=O)C2)c(F)c1F CC(CC(=O)NC1CN(C(c2occ3c2CCC3)=O)CCC1C)CC(F)(F)F C(=O)(CC(C)(C)CC(=O)N1CCCC2CN(C(c3cnc(C)[nH]3)=O)CC12)OC c1(C(N2C(C)(C)C(C(=O)NCC(O)CO)CC2)=O)cnn2ccccc12 Cc1cccnc1C(=O)NCC1CCC(C(=O)NC2CC(N(C)C)C2)C1 C1(C(N2CCCC(N3CCCC3)C2)C(=O)NCCCF)CCCN(CC2CC2)C1 N1(C(c2c(CC)cco2)=O)CC(OC)CC(NC(c2cc(=O)n(C)cn2)=O)C1 Cc1ccc(C(=O)NC2(CNC(=O)C(c3cnn(C)c3)C)CCOC2)cc1C#N N1(C(C(C(C)C)=O)=O)CCC(C)(C(=O)NC2CCC(F)(F)CC2)CC1 C1(NC(CNC(=O)NC)=O)(CO)CCN(C(=O)Cc2cc(Cl)ccc2OC)CC1 C(CC(N)=O)(C(=O)Nc1ccc(C)c(C(N)=O)c1)NC(C1CCC(C)(CC)O1)=O N1(C(C2=NOC(C)C2)=O)CC2(C1)CN(C(c1cc3c(cc1Cl)OCO3)=O)CCO2 Cc1ccccc1CN(C(=O)C(F)C(C1CC1)C1CC1)c1ccccc1 N1(C(C(C)c2ncco2)=O)C2CCC1CN(C(=O)COc1ccc(F)cn1)C2 CC1CN(C(C2CCC(O)CC2)=O)CC2(CCN(C(C3COC(C)(C)C3)=O)C2)O1 Cc1nnc2n1CC(C(N1CC(C)(C)CC1CNC(C1CCOC1)=O)=O)C2 C12(CNC(c3ncn(C(C)(C)C)n3)=O)CCC(CNC(=O)C=CCO)(CC1)CO2 C1(NC(C(CC=C)NC(C)=O)=O)CCC2(CCN(C(=O)CN3CCC(C)C3)C2)C1 N1(C(C(C)C2CCC2)=O)CCC2CN(C(c3cnn4c3OCCC4)=O)CC12 c1(C(=O)OC)cccc(CN2CCN(C(C3(S(N)(=O)=O)CC3)=O)CC2)c1 C(=O)(C1CCCc2scnc21)NC(CCCCNC(CSC)=O)C C1(CC)CN(C(=O)CNc2cccc(Cl)c2)CC1C(=O)NC(=O)COC(F)F Cc1c(C(N2CC(C)(CNC(c3ccc(Cl)c(Br)c3)=O)C2)=O)cccc1O C1(NC(C2CC(OC)C2)=O)CCSC12CN(C(=O)CC(=O)OC(C)(C)C)C2 C1(C(=O)OC)CC2(CNC(c3ccccn3)=O)CC1C2 c1(OCCCCOC(COC(CC)=O)=O)ccc(S(C)(=O)=O)cc1 C1(CC)CC(C(=O)N(C2CC2C2CC2)C)CCN1C(c1ccsc1C#N)=O C1(C(=O)NCC(=C)C)CCCN(Cc2ncccc2Br)C1 C1(CNC(C(CCC)OC)=O)CN(c2nnc(-c3ccccc3C)o2)CCN1C Cc1nc[nH]c1C(=O)NC1COCC1NC(=O)COCC(F)(F)F C1(C(=O)NC(C)C(=O)N(C)Cc2ccccn2)CCN(C)C1 CC1(C)CN(N2CCCC(c3ncc(Br)cn3)C2)CC(CC(F)(F)F)O1 N1(C(CCSCCC)=O)CC(NC(c2ncsc2Br)=O)C(C2CC2)C1 C1(C(=O)NC(c2ccc(F)c(F)c2)(C(=O)OC)C)CSC(c2cccs2)=N1 c1(CC(=O)NC2C(CNC(c3c(C(=O)OC)c[nH]n3)=O)CC2)ccnc(CO)c1 c1(CC)nc2ccccn2c1C(=O)NNC(=O)C1CNC(CC)C1 C(c1ccc(F)c(C)c1)=CC(=O)NCC1(NC(C(CC)SC)=O)CCCC1 c1(NC(C2CCCN2C(=O)Cc2sc(O)nc2O)=O)ccc2ccncc2c1 C12(C(N3CC(NC(C4C(C)(C)CO4)=O)(CO)C3)=O)CCCN(CC1)C2 Cc1c(C(N2CC(NC(=O)C(CO)N(C)C)C(F)C2)=O)nnn1C(C)C c1(C(N(CC(CC)NC(=O)C(C(C)C)N(C)C)C)=O)c[nH]nc1S(N)(=O)=O c1(C(=O)NCCN(C(=O)C(O)c2ccco2)C)csc2cncn12 S(=O)(=O)(c1ccc(O)c(C(=O)O)c1)N1C(C)(CC(C)C)CCC1 c1(SC)ncc(C(=O)NC(C)CN(C(=O)C(C)Sc2nncn2C)C)s1 C12(C(=O)NCC3CN(C(C4C(C)CC4)=O)C(C)(C)C3)CC3CC1C2C3(F)F C1(NC(c2cc(CC(C)C)[nH]n2)=O)(CF)CCN(C(=O)CC=CC(C)(C)C)C1 C1(NC(C2CC3(CC(F)C3)C2)=O)CCN(C(=O)Cn2ncnn2)CC1F CON(Cc1ccccc1)C(=O)C(F)=Cc1cn(CC(C)(C)O)nn1 N1(C(C2(CCC)CCC2)=O)CC2CC(C(=O)NCCC#CCO)(C2)C1 c1(C(=O)NCCCCCCNC(C(CC)C(C)O)=O)c(C)ccc(Cl)c1F C1(C(=O)NCCN(C(C2CCC(N(C)C)CC2)=O)CC)CCC2CCCCN12 C1(OC)CCC2(C(N3CSCC3C(=O)NCCC(C(C)C)OC)=O)CC12 C(=O)(C#CC1CCOC1)NC1C(NC(c2cc(C)c(C)s2)=O)CCOC1 c1(C(=O)O)cc(CN2CCC(F)(C(=O)Nc3c(Br)ccnc3Br)C2)ccc1O C1(NC(C2C(C)CC(=O)N2)=O)CN(C(C2CC(=O)C2)=O)CC2(CC2)C1 c1(NC(c2cc3sccn3c2)=O)nc(Cl)c(Cl)cc1Cl C1(CNC(Cn2cc(CNC(C3CCC(=O)O3)=O)nn2)=O)CCS(=O)(=O)C1 N1(C(c2cncc(C)c2)=O)CCCN(C(c2ccnn2-c2ccccc2)=O)CC1 c1(CC(=O)N(C2CCN(C(COCC#C)=O)C2)CC#C)cc(Cl)cc(Cl)c1 N1(C(CN(C)C)=O)CC(NC(c2cncn2C2CC2)=O)C(C2CC2)C1 S(=O)(=O)(c1ccc(F)cc1)NCCNC(c1scc(C)n1)C c1(C(=O)NC2CCC(NC(c3cccc(CO)c3)=O)C2)cnnc(C2CC2)c1 c1(C(N(C2CCN(C(C3CCC(=O)N3)=O)C2)CC)=O)n[nH]c2c1CCC2 C1(CNC(C2CC(C(=O)OC)C2)=O)(CNC(=O)CC2COC(=O)C2)CCCCC1 Cn1nc(-n2cc(CCC3CCCN3C(=O)C(c3ccccc3)F)nn2)nc1Br c1(C(C)OC)nc(C)c(C(=O)N(CCCCN(C(=O)C2=CCOC2)C)C)s1 C1(NC(C2(COC)CCC2)=O)CCC(C)N(C(=O)C2=COCCO2)C1 n1(CCC)cc(C(=O)NC(C)CC(C)NC(=O)CC(=O)Nc2nccs2)c(C)n1 C(=O)(C1CCc2snnc21)N1CCCCC(CNC(c2ncn(CC)c2)=O)C1 N1(C(C2C(C)=CCC=C2)=O)CCc2cccc(C(=O)NC(C)(C)C#N)c2C1 C(CC(C(C)C)NC(c1ccc(SC(F)(F)F)cc1)=O)N(C(C(COC)O)=O)C C(C(N=[N+]=[N-])C(=O)N1CCC(CCC(=O)N(C)CCO)CC1)OCC CC1(NC(=O)C=CCO)CCC(NC(c2cccc(CO)c2)=O)CC1 C(c1cnc(C)nc1O)=CC(=O)NCCNC(c1ccc(C(CC)(C)C)cc1)=O C1(C(N2CC(O)(CC=C)C2)=O)CC(F)CCN1C(=O)C(C1(O)CCCC1)F C1(NC(CNC(C)=O)=O)CCCN(C(c2ccc(-c3cccnc3)s2)=O)CC1 N1(C(C(CC2CC2)OC)=O)CCN(CC(=O)N(c2ccccc2)C)CC1 C1(C(N2CCN(C(=O)Cc3cnns3)C(CCO)C2)=O)CCCC1C1CC1 c1(NCCCN(CCC)C)ncc(S(=O)(=O)NC2CCN(CC)C2)cc1Cl N1(C(c2c(C)ncnc2)=O)CC2CCC(N(C(=O)C(O)C(F)(F)F)C)C2C1 c1(CC(=O)NC(CN(C(C(N2CC(C)C2)C)=O)C)C)csc(C(F)(F)F)n1 N1(C(CCCC)=O)CC(C)N(C(=O)C=Cc2ccc(C)s2)CC1C C(=O)(C(C(C)(C)C)C1CCC1)NC(CNC(c1cc(C)on1)=O)(C)C c1(SC(C)(C)C)nnc(-c2cccs2)n1NC(=O)Nc1cccc(Cl)c1 c1(C(=O)NC2(CO)CCCN(C(CCC(CC)OC)=O)C2)n[nH]c2c1COCC2 CC(C)(C)CCCCC(=O)N1CC(=O)NCC1C(N1CC(CCO)C1)=O c1(Cn2c(C(C3CC3)NC(C)(C)C)nnn2)cn(-c2ccccc2)nn1 Cc1cccn2ncc(COCC(c3cc4ccc(Br)cc4s3)=O)c12 CC1(NC(C23CSCC2C3)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C1 c1(C(N(CCC)CCNC(c2cc[nH]n2)=O)=O)ccc(CC)cn1 N1(C(C(C)=C(CC)C)=O)CC2(CNC(C3CC3(C)COC)=O)CC1CO2 Cc1cc(F)c(CC(N2CCC(C(C)NC(=O)CC3CC3(Cl)Cl)CC2)=O)cc1F c1(N(CC(CN(C)C(c2cc(CC3CC3)on2)=O)O)C)cc(CO)nc(Cl)n1 c1(OCCCC(=O)N(C)CC2CCN(C(C(CC)(C)O)=O)C2)ccc(O)c(F)c1 N1(C(C(C)OCCC#C)=O)CCC2CN(C(C3CC(n4ccnn4)C3)=O)CC12 C1(NC(C2N(CC)CC2)=O)CCCCC1NC(c1cccc(C(C)C)n1)=O C1(CNC(C(C)(CSC)NC(CC(C)SC)=O)=O)Cc2nccn2C1 CC1CC(c2ccoc2)CN1S(=O)(=O)CC1COC1 Cc1csc(C(=O)NC2CC2NC(=O)CSc2ccc(O)cc2)c1C CCCCC(O)C(C)C(=O)N1CCN(C(=O)C(COCC)N=[N+]=[N-])CC1CO C1(CC)CN(C(=O)C(O)C(C)C)CCN1C(=O)CCCN(C)C(C)=O c1(NC(=O)COCCC(C)C)cccc(C)c1.C(C)(C(=O)N1CC2CC2C1)OC CC1=NNC(=O)C1CC(=O)N(C)CC1CCCN1C(=O)CCC1CC1(F)F c1(C2(C)CC2)nc(N2CCN(C(C3CCCC(C)C3)=O)CC2)cc(Cl)n1 C(=O)(C(C)(C)CNC(=O)C(C1CCN(C(c2c[nH][nH]c2=N)=O)C1)F)NC c1(C(N2CCCN(C(c3ccc(C)nn3)=O)CC2C)=O)sc2nnc(S)n2c1C C(=O)(C1CSc2ccccc21)NC1(CCNC(C(=Cc2cccs2)C)=O)CC1 C1(CC(N2CCC(NC(C3(N=[N+]=[N-])CC3)=O)C(O)C2)=O)CCC2(CCC2)CO1 C12(CCNC(=O)C(C3CCCCC3)O)CCC(CC1)N(C(=O)CN1CCCC1)C2 c1(C(=O)NCC2OCCCN(C(C3C(C#N)C3)=O)C2)cccc2ccoc12 C1(C(N2CC(O)(C(C)NC(c3c(C)sc(Cl)n3)=O)C2)=O)OCC2CCCC12 C1(C(=O)NC(CCCNC(CC(C)C2CCCC2)=O)(C)C)CN=C2N=CNN2C1 C(=O)(C(C(C)(C)O)NC(C)=O)NCC1CC(C(=O)NCC2CC(OC)C2)C1 C(c1nccs1)=CC(=O)NCC(C1CCOC1)NC(c1cc(CCO)on1)=O C1(CNC(c2n(C)ccc2)=O)(CNC(=O)C2=NNC(=O)C2)CC2CCCC2C1 C(CCS(N)(=O)=O)N(C(c1c(C)n[nH]c1)C(=O)Nc1nnn(C)n1)C CCCCCCC(C)CC(=O)N1CCCC(CO)(NC(c2nc(CC)no2)=O)C1 c1(C(=O)NCC2(O)CCN(C(c3cncc(O)c3)=O)C2)cc2c(Cl)cccc2[nH]1 C1(O)(CNC(C(CC)Oc2ccccc2)=O)CCN(C(c2ccnnc2C)=O)C1 N1(C(c2ccc(C)cn2)C(=O)O)CCC(C)C(NS(C)(=O)=O)C1 C#CC1(O)CCCN(Cc2ccc(Sc3cc(C)ccc3F)cc2)C1 C#CC1CCCN1C(=O)C(C)CNC(=O)CCC(=O)C1CC1 Cc1nc2c(s1)CCCC2C(=O)N1CCC(CNC(c2cnsc2)=O)C(F)(F)C1 c1(N(C)CCF)cc(N2CCC(CC(=O)NCC3CCCO3)C2)nc(C(F)(F)F)n1 C1(CC(=O)NCCOC(C)=O)CCCCC1NC(=O)Cc1ccc(C)s1 c1(C(=O)NCC(CNC(c2c(C)ncs2)=O)O)cc2nc(Cl)ccc2s1 N1(C(CC(C=C)(C)C)=O)CC(NC(c2cc(F)c(O)c(Cl)c2)=O)C(C2CC2)C1 C1(C(N2CCC(OC)(CNC(C3CNC(=O)C3)=O)C2)=O)CC2CCC(C1)C2 C(c1c(C)coc1C)=CC(=O)NCC(CNC(=O)CC1(C)CCCCC1)OC C1(C(=O)NC2CC(NC(COc3cn(C)nc3)=O)C2)CN2CC3CC2(CO1)C3 CCCCC(C(=O)N1CCCC1C1CCN(C(c2nocc2Br)=O)CC1)N(C)C Cc1cnc(F)cc1C(=O)NC1CCCCN(C(C23CC2C3)=O)C1 c1(N(CC(CCC)C)C)nc(NC(C)CCn2cncn2)c2c(ncn2CC)n1 c1(OC)ccc(NC(=O)C(=O)Nc2cnns2)c(C#N)c1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CC(C(=O)NCCCS(N)(=O)=O)C(F)C1 C12(C(=O)NCC(C)N(C(=O)Cc3ccccn3)C)CCC(C1)C2(C)C c1(CC)nncn1NC(=O)C1CCCCCN1C(c1cnco1)=O C(=O)(CCCC(=O)NCC1C2CN(C(C3COCCO3)=O)CC12)NC(C)C CC1=C(C)CC(C(=O)NC2CC(O)(CNC(c3[nH]cnc3C)=O)C2)CC1 CC(C(=O)NCC(C1CC1)N(C)C(c1cnnc(O)c1)=O)C(F)F N1(C(CNC(CC)=O)=O)CCC(C(=O)NC2CC(CO)C23CCC3)=C(F)C1 Cc1nn(C)cc1C(C)C(=O)NCC(CNC(C1(P(C)(C)=O)CC1)=O)CO C(CC[Si](C)(C)C)NC(C(N1CCC(CCC(=O)OCC)C1)=O)=O C1(CCOC)(NC(c2ccncc2)=O)CCN(C(c2cc(C)n(C)n2)=O)CC1 CC(C)(C)C(CNC(C1(C#N)CC1)=O)NC(c1cnncc1O)=O C1(C(=O)NCCOCCOCCCSCC)(OC)CC1 C(CC(O)C(F)(F)F)CONC(CCC1N(C(CCc2onc(C)n2)=O)CC1)=O CC1CN(C(C2CCCCCN2C)=O)CCC1CN=c1ccnc[nH]1 N1(C(C(CC)=CC)=O)CC(C)CCC1C(=O)NCC1(C#N)CCCCC1 C1(COCC)CCN(C(=O)CCCNC(C2COCCN2C2CCCC2)=O)CC1 c1(-c2cn(CCN(C(COCP(C)(C)=O)=O)C3CC3)nn2)cccc(O)c1 N1(CC(N2CCC(CCC(=O)NCCC3C(C)C3)C2)=O)CC(=O)NC1=O N1(C(C2(OC)CCC2)=O)CCN(CC2CN(C(c3cnc(O)o3)=O)C2)CC1 C12(C(N(CC(COC)O)C)=O)CC(CN(C(=O)CCS(N)(=O)=O)C1)C2 c1(OC)ccc(CNCc2cnn(CC(C)C)c2C2CC2)c(F)c1Br c1(C(N2CCCC(C(C)NC(=O)C3=CCSC3)C2)=O)c(F)cc(F)cc1F c1(C(N(C2CN(C(COCCC#C)=O)CC2F)C)=O)cc(C)n(CC)c1C N1(C(C(CCC)C)=O)CC2(C1)CN(C(=O)C(C)S)CC2C(=O)O c1(C(=O)NC(CCCCCC=C)C)ccccc1S(=O)(=O)N1CCOCC1 C1(N(C(C(COC)C)=O)C)CCCCN(C(=O)CSC(C)(C)C)C1 N1(C(CCC)=O)CC(NC(=O)C=Cc2ccc(C(N)=O)o2)CC12CCCCC2 C(=O)(C1CCc2nnc(C)n21)C1(C2N(CCc3c(C)cc(O)cc3)CCC2)CC1 Cc1cc(C)c(C(N2CCCC(N(C(=O)Cn3cccn3)C)CC2)=O)c(S)n1 C1(C(=O)NCC2CC(C(N3C(C(C)C)CCC3)=O)C2)CCN(C)C(=O)C1 Cc1ccc(C(N2CC3C(CNC(=O)CCCCC(N)=O)C3C2)=O)c(O)c1C Cc1cn2c(CC(=O)NC3CC(NC(c4ccc(F)cc4F)=O)C3)csc2n1 CN(C)S(=O)(=O)N(C)CC(=O)NCCC1CCN(C(=O)CSc2n[nH]c(O)n2)C1 c1(CC)cccc(NCC2CCC(C(=O)OC)O2)c1 c1(CN2CC3C(C(=O)NC(C=C)C)C3C2)cccc(OC)c1OC(C)C c1(COC(CC2C(OC)COCC2)=O)nc2cc(Cl)ccc2s1 Cc1cc(C#N)cnc1N(C1CCCN(C(C2(F)CCOC2C)=O)C1)C c1(C(N(C2CCCN(C(c3cc(C(C)(C)C)n[nH]3)=O)C2)C)=O)cc2c(s1)CCC2 c1(-n2cc(C3N(C(C(C)CF)=O)CCC3)nn2)cnnc(Br)c1 c1(C(=O)NC2C(CNC(C(N3C(CC)CCC3)=O)=O)CC2)cccc(CO)n1 c1(C(=O)NC(C(C)C)CNC(c2cn(C)ccc2=O)=O)cc(N)c(N)cc1F c1(C2(NC(=O)C(F)=CC3CC3)CN(C(c3cccc(Cl)c3)=O)C2)ccc(F)cc1 C(=O)(C(C#N)C(C)C)NCC#CC(=O)N(CC(COC)C)C c1(CC)ccc(C=CC(N2CCCC2CCNC(=O)C(F)n2ccnc2)=O)cc1 CC#CCCCC(C)(c1nnnn1CCOC)NC(C)Cc1ccc(OC)cc1 c1(C(=O)Nc2c(OC)nc(F)cn2)cc(-c2cccc(F)c2)cc2c[nH]nc12 C1(NC(C(c2cc(C)sc2)(F)F)=O)CC(=O)N(C2CN(C(=O)C(C)C(C)C)C2)C1 C1(CNC(c2ccnc(C)n2)=O)CC2(CC2)CN1C(=O)C(C1CCCCC1)F Cc1nn(CCO)cc1C(=O)NC1CC(C)N(C(=O)COc2ccc(F)cn2)C1 N1(C(CC(C)=C(C)C)=O)CCC2(CC2C(=O)N(C)CC2CC2C)C1 CN1CCOCC1CC(N1CC(n2cc(CNC(=O)CC3CC(F)C3)nn2)C1)=O c1(C(=O)NC2CCN(C(C3(C)C(C)(C)C3)=O)C2)ccc(-n2cnnn2)cc1Cl C(=O)(C(C)(C)C1=CCSCC1)N(CCC(C)NC(C1CC1C(F)(F)F)=O)C C1(NC(c2cnccc2Cl)=O)CCC12CCN(C(=O)CC1CCCCO1)CC2 C1(C(=O)NC2(C)CC(NC(C3C(C)(C)OC(=O)C3)=O)C2)CCCCN1S(N)(=O)=O C1(NC(=O)CC2CN(C(c3cnc(Cl)cc3I)=O)CCO2)CCC(F)(F)CC1 c1(C(N2CCC(NC(C3(CF)CCC3)=O)C(F)C2)=O)cc(Cl)cc(Cl)c1Cl c1(OC)cc(CN2CC(O)CC2C(=O)NCCCc2ccncc2)ccc1Br CC1(CNC(C2CC(F)(F)C2)=O)CCCN1C(c1cn(CC(F)(F)F)cn1)=O c1(C(=O)NCc2c(C)nccn2)ccc2c(n1)CN(C(C1(C)CCOC1)=O)CC2 CC1(C)CC(C(N2CCC(C(CO)CO)C2)=O)CN(C(C2OCCC2(C)C)=O)C1 C1(C(=O)NCCCc2n(C)nnn2)CCCCC1(C)NC(=O)CCn1ccnc1 C1(C(=O)NC2CCCN(C(C)=O)C2)CC(C)(C)CN1C(c1cc(C)oc1C)=O C=C(C)C(C)(C)C(=O)N1CCN(C2CCN(C(=O)C(CC)NC(N)=O)C2)CC1 N1(C(C2(c3ccccc3F)CCC2)=O)CCN(C(C2CC3CC3C2)=O)CC12CC2 C(C(CC(C)C)NC(c1ccc(C(=O)NC)cc1)=O)NC(C(C)N(CC)CC)=O Cc1[nH]nc(C(=O)NC(C(=O)NCCCC(C)O)C2(O)CCC2)c1C C=C=CC(C)C(=O)N(CCC(=O)NCCSCC)CC C1(C(=O)NCC2C(CNC(=O)COC(=O)CO)C2)CC2CCC(C1)C2O c1(OCN2CCC(OC)C2)nccc(C(=O)NCCC(c2ccc(CO)s2)=O)n1 c1(CCC)ccc(NC(=O)CCN(C)C(c2cn(CCOC)nn2)=O)cc1 c1(OCCC)ccc(C(=O)NC(C)Cn2cc(CCSC)nn2)cc1 C(CS(=O)(=O)CC(=O)NCC(C)CN(C)C(C1CCCN1C)=O)OC C1(NC(c2cc(F)c[nH]2)=O)CCCCC12CCN(C(=O)C1=CCCC1)CC2 c1(NC(CC)CNC(C2CCCC2(C)C)=O)ccc(C#N)cc1[N+](=O)[O-] C(CC(=O)NCC1(O)CCCCCC1)(C(F)(F)F)NC(c1nn(C)c(=O)cc1)=O C=C(C)CC(C(=O)N(CC(C)(C)C(=O)NC1CCOCC1C)C)OC c1(-c2cc(C(=O)NCC)ncc2)n[nH]c2c1CN(C(c1cccc(Br)c1F)=O)C2 c1(CCC(=O)NC2C(CNC(CN(C(C)C)C)=O)C2)cnn(-c2ccccc2)c1 C1(CNC(C(C)CO)=O)CC2CCC(C1)N2C(c1cnn(C)c1N)=O c1(C(N2CC(NC(COC)=O)C(C(F)(F)F)CC2)=O)cc2c(C)n[nH]c2cn1 C1(CC(N2CC(CNC(C3CCC(C)(C)CO3)=O)C2)=O)CCc2sccc2C1=O c1(C(N2CC3CN(C(=O)CC45CCCC4C5)CC3C2)=O)ccc2nonc2c1 c1(OC)ccc2[nH]cc(CN3CCC4C3CCCN4C(=O)CC3(O)CCC3)c2c1 O=C(CCC(=O)N1CCOCC1)NCC(CO)NC(c1cn(C2CC2)nn1)=O c1(C(N(C)CCNC(=O)C(c2ncc(Cl)n2C)(F)F)=O)ccc(Cl)cc1C(F)F c1(C(N(C)CC2COCCN2C(=O)CC2(CO)CC2)=O)cc(F)cc(Br)c1 S(=O)(=O)(c1cnn(CCO)c1)N1CC(Nc2cc(OC)cc(OC)c2)N(C)CC1 c1(CNC(C(=O)NC(c2c(C)cnnc2)C)=O)ccc(S(=O)(=O)NC(C)C)cc1 Cc1cn2ccnc(C(N3CCC(NC(=O)CC(C)CC(C)(C)C)C3)=O)c2n1 C(CC(F)F)(C(=O)NC1CCCC1(C)C)N(C(c1nnn(CC)c1C)=O)C N1(C(C(C)OCCOC)=O)CC2CCC(NC(=O)CSCCC#N)CC2C1 c1(C(=O)NCCCC(C)NC(c2nccnc2C(F)(F)F)=O)ccc(F)c(Cl)c1 S(=O)(=O)(c1ccc(NS(C)(=O)=O)cc1)NC(C)CCN1CCOC1=O C1(NC(COCCSC)=O)CCC(CNC(c2ccccc2COC)=O)CC1 Cc1ccc(-n2nc(CCN(C)C)nc2C2CC2c2ccccc2)c(C)c1 c1(C(=O)NC2CC(C)(NC(C=NOC)=O)C2)ccc(C2CC2(Cl)Cl)cc1 N1(C(C=C=C(C)C)=O)CCC(C)(CNC(C2CCN2C)=O)CC1 c1(C(=O)NC(CCOC)CNC(=O)CCC(C)OC)cc([N+](=O)[O-])cnc1C c1(CNC(c2n(C)ncc2-c2cn(C(C)(C)C)nn2)=O)ccc2cccnc2n1 N1(C(C2C(CC)C2)=O)CCC2(CCN(C(=O)C(F)CCC(C)C)CC2)C1 N1(C(C2N(C(C3CCC(C)(C)OC3)=O)CCCCC2)=O)C2CCC1CC1(C2)N=N1 c1(CC)cc(C(N2CCC(F)(CNC(c3ccc(O)nc3)=O)CC2)=O)ccc1F c1ccc(NC(=O)NCC(c2ccccc2C)(C)C)cc1.N(CCO)(CC)CC N1(C(c2cc(C#N)sc2)=O)CCC(F)(CNC(c2ccc(F)c(Cl)c2)=O)CC1 C(N=c1nc(N2CCCCC(SC)C2)c2c([nH]1)CSC2)c1cc(OCC)ncc1 C12(C(=O)NCC(CC)NC(=O)C(F)CC3CCCC3)CCC(O)(CC1)CC2 C1(CC(=O)NCC(C)(C)NC(C(CCC)N(C)C)=O)OC(C)(C)OC1=O c1(C(=O)NCC2(F)CC(NC(CCS(=O)(=O)N(C)C)=O)C2)nccc2[nH]ccc12 N1(C(C(n2ccc(=NCc3ccccc3)[nH]2)C)=O)CC2(CO)CC(C)(C1)C2 C1(C2CN(C(=O)C(C)S(C)(=O)=O)C2)(NC(c2c(SC)cccn2)=O)CC1 Cn1[nH]c(=NC(=O)C2CCN(Cc3c(Br)cc(F)cc3Br)C2)cc1Cl N1(C(CN(C)CC)=O)CCN(C(C23CC2COC3(C)C)=O)C(C)C1 N1(C(C(N)=O)=O)CCOC(CCNC(=O)CCC(=O)c2cccc(F)c2)C1 N1(C(CCOCCC)=O)CCOC(CNC(=O)C#CC2CC2)C1 c1(SC)ccc(C)c(C(=O)NC2CCCC2NC(C2CC23CC(F)(F)C3)=O)c1 N1(C(CC#N)=O)CCC2(C1)CN(C(=O)CNS(=O)(=O)c1ccc(Cl)s1)CCO2 c1(C(N(CC(CN(C(c2c(C)scc2)=O)C)O)C)=O)nccc(Cl)c1F C(CC(=O)N1CCC(O)(C(F)F)C1)(C(F)F)NC(=O)Cn1cc(CO)nn1 c1(C(=O)NCC2CCCCN2C(=O)CCn2ccnc2)ccc2c(c1)CCC=C2 c1(C(N2C3CC(NC(C4CN(C)C4)=O)C(C3)C2)=O)cc2c(cc1Cl)NC(=O)CO2 C1(c2ccc(F)cc2)(C(N2C(CNC(c3ccon3)=O)C=CC2)=O)CCCCC1 C1(CNC(C(C)(C)OC)=O)CCC(CN(C(=O)CN(CC(C)(C)C)C)CC)CC1 c1(CN(C)C(=O)NC2(c3ccncc3F)CC2)ccc(Cl)cc1F C(CC(C(=O)N1CCC(NC(C2CC2[N+](=O)[O-])=O)C1C)OC)OC c1(OCCC(N2CCC(C)(CNC(=O)CCC#N)C2)=O)cccc([N+](=O)[O-])c1 C(C)(C)(C(F)(F)F)OC(C1C(C)CCC1)=O.c1(C(=O)OCC(=O)N)cccn1CO C1(c2ccccc2)C2CC3CN(C(=O)CCCNC(CCC(=C)C)=O)C1C3C2 c1(C(N(C2CCN(C(=O)CN3CCCC3C)CC2)CC)=O)cnc2ccoc2c1 c1(CCC)cc(C(N2CCCC(CCNC(C3CSCC(=O)N3)=O)C2)=O)ccn1 c1(NC2CC(CCNC(C(C)NC(CC)=O)=O)C2)cc2nn[nH]c2cc1[N+](=O)[O-] c1(C(=O)NCCC2CCC(NC(CC=C)=O)C2)nccc2c1[nH]c1ccccc21 C(=O)(C1Cc2ccccc21)NC(CC=CC(=O)NC(CC=CC)CO)(C)C C(CN=c1ccnc(SC#N)[nH]1)c1ccc(C(=O)O)cc1Cl C1(CCOC)CCN(C(=O)C=C(Br)Br)CC1 c1(CC(=O)NC(CNC(C2C(c3ccc(C)s3)C2)=O)(C)C)cccc(Cl)c1F c1(N2CCCC(NC(=O)CCc3ccc(Cl)s3)CC2)nc2cccc(Br)c2o1 N1(C(=O)C=CC2CC2)CCC2CCC(NC(C3(C4CC4)CC3)=O)C1C2 C(CS(=O)(=O)C(F)(F)F)SCC.c12cc3c(cccc3o1)NCCn1nnnc1-2 C(=O)(CC(O)C(C)C)NCC(CCOC)NC(=O)C=CC(=O)NC1CC1 n1(CC)c(C)nn(CC(=O)N(C(C)CNC(=O)C(CCSC)N(C)C)C)c1=O C1(c2n(CC)nnn2)(NCC2(OC)CCCSC2)CCOCC1F C1(C(=O)NCCN(C(=O)Cc2nn(C)cc2Cl)C)CCC(C)(F)CC1 c1(NCC2OCCN(C(=O)C(F)Cc3ccccc3)C2)c(Cl)cccc1[N+](=O)[O-] N1(C(c2scc(C)n2)=O)CC(C)CC1C(=O)Nc1nc(C)cs1 CC(C)CC(O)CC(=O)N1CCN(C(C2CC23CCC3)=O)C(C(C)(C)C)C1 c1(CC(=O)NCc2ccccc2CNC(C2(F)CCCC2)=O)ccc(Cl)cc1Cl Cc1nc2ccc(C(N3CCC(NC(=O)C(C)(C)F)C4(CCC4)C3)=O)cc2s1 C(=O)(CC1OCCc2ccccc21)N1CCC(CN(C(c2cc(C)sn2)=O)C)C1 C(=O)(C(O)CCCCC)NC1CN(C(C(CC=C)NC(C)=O)=O)CC1CCC C1(C(=O)NCCC(C)N(C)C(C2CCCN2C)=O)CC12CCOCC2 c1(C(=O)NC2(CO)CN(C(C(C)CN(C)C)=O)C2)ccc(CC(C)(C)C)cc1 c1(C(=O)NC2CCN(C(CS(CCCC)(=O)=O)=O)C2)ccccc1C#CC1CC1 c1(C(=O)NCCCC(C)NC(CCN(CCCCC)C)=O)cc2c(s1)CCOC2 C1(C(N2CC(F)(CNC(c3cc(C(F)(F)F)c[nH]3)=O)C2)=O)(OC)CCOC1 c1(C(c2n(C)nnn2)NC(c2nnnn2C2CC2)C2CC2)ccc2cccnc2n1 C1(CN(C)C(C2CC2c2ccsc2)=O)CCCN1C(=O)CCc1cncs1 C1(NC(C(CC)C)=O)CCCC1(C)CNC(=O)CCC1CCC1 C12(CNC(C(CCCC)O)=O)CCC(CN(C(C3(C)CCCN3C(C)=O)=O)C1)C2 c1(CC)ccc([N+](=O)[O-])cc1C(=O)NC(C1(O)CCN(C(C2CCCC2)=O)C1)C N1(C(c2ccc(N(C)C)nc2)=O)CC(NC(c2snc(Cl)c2Cl)=O)CC2(CC2)C1 c1(NC(=O)CC2CCCNC2)ccc2c(c1)CN(C(c1csc(Br)c1)=O)CC2 C(=O)(C(O)CC(F)F)N1CCC(C(CNC(c2cc(C(C)(C)C)n[nH]2)=O)F)CC1 N1(C(c2nc(CC)oc2C)=O)CCC2(CC1)CC(NC(c1cc(C)ns1)=O)CO2 C#CC1(C(=O)N(C)CCN2CCCC2=O)CCN(C(=O)CC2CC(C)=NO2)C1 c1(C(C(=O)C=Cc2ccccc2)=O)cc(CO)cc(C(F)(F)F)c1 C1(CNC(CC)=O)CC2(CC2)CN1C(=O)C(c1cccc(C#N)c1)C(C)C c1(C(=O)NCCN(C(=O)C(=O)NCC(F)(F)F)C)ccc2ncn(C)c2n1 C1(CNC(C(C)CN(C)C)=O)CCN(C(c2cnn(C)c2F)=O)C12CC2 Cc1nn2c(C(=O)NCC3COCC3NC(c3sccc3C)=O)c(C)nc2s1 CC(C)C1CNC(=O)c2cc(NCc3cnc4ccc(Br)cn34)ccc21 C1(CS(N2CC3C(C(N)=O)C3C2)(=O)=O)CC2(CCNCC2)CO1 Cc1c(C(=O)NC(C2(O)CN(C(c3ccc(C#N)s3)=O)C2)C)cnn1C1CCC1 c1(C(=O)NC2CCN(C(C3CSCCS3)=O)C23CC3)c[nH]c2cc(Cl)ccc12 C1(NC(CCN(C)CC)=O)CCC2CC1CN2C(=O)C(C)c1cccs1 CCC(C)(CO)C(=O)NCCCCCN(C)C(C1(F)C(C)(C)C1(C)C)=O N1(C(C2(NC(N)=O)CC2)=O)CCC(CCNC(=O)C=Cc2cnc[nH]2)C(F)(F)C1 N#Cc1ccccc1OCC(=O)NC1CC(O)(CNC(=O)CC2CCCCO2)C1 c1(C(=O)NCC2C3CN(C(C4(C(CC)=O)CC4)=O)CC32)nc(Cl)ccc1Cl c1(CC(N2C(CC(=O)NC3CCN(CCC)C3)CCC2)=O)cccnc1C c1(OC)cccc2[nH]cc(CN3CCC(O)C3C(N3C4CCC3COC4)=O)c12 N1(C(CCC(C)c2ccccc2)=O)CC(=O)NCC1C(N1CC2CC1CN2C)=O C1(CC(=O)N(C2COC2)CCO)CCN(C(=O)Cc2ccccc2)C1 N1(C(C(C)Sc2ccccn2)=O)CCCC(C(C)NC(=O)CNC(=O)C2CC2)C1 C(=O)(CCCCCC(C)(C)C)NC(C(C)NC(C1CCN(C(C)C)CC1)=O)CO N1(C(C(F)=CC)=O)CCC2(C1)CN(C(C1(OC)CS(=O)(=O)C1)=O)CCO2 C1(NC(C(CC=CC)CC)=O)CN(C(c2cc(F)c(N)c(F)c2)=O)CC(C)(C)C1 c1(SCC#C)cccc(C(=O)NCC2(NC(=O)C(C)C(F)F)CCOCC2)c1 C1(NC(C2(CC=C)CCC2)=O)CCC(NC(C2CCOCC2C)=O)CC1 c1(OCC)cnncc1C(=O)N(C)CCOCCNC(=O)CNC(N)=O C1(C)(C(=O)NC(CC)CNC(c2csc(-c3ccsc3)n2)=O)CCCOC1 c1(C(=O)NC(CCCNC(C2C(OCC)C2)=O)C)ccc(N2CCCC2)cn1 N1(C(c2cc(C)[nH]n2)=O)CC(F)CC1CN(C)C(C1CCN(S(C)(=O)=O)CC1)=O C(=O)(CC1COCc2ccccc21)NC1(C)CN(C(c2cc(Cl)c(Cl)s2)=O)C1 c1(C(N2CC(NC(c3n(CCC)nc(C)c3)=O)C(C)C2)=O)ccc(F)c(F)c1N N1(C(C(C2CC=CCC2)NC(CC=CC)=O)=O)CCCC2(CC2)C1 CCC(CC(F)F)C(=O)N1CC(O)(C(C)NC(=O)CCn2ccnc2C(C)C)C1 N1(C(c2c(C(C)C)ncs2)=O)CCOCC(NC(C2(n3cnnn3)CC2)=O)C1 c1(C(N(CCNC(C2CCCC2OC)=O)CC)=O)ccc2cccnc2c1O Cc1cc(C(=O)NC2COCCN(Cc3ccc(Cl)nc3Cl)C2)ccc1O CCC(CC)C(C(=O)N1CCCC1C(C)(C)NC(=O)C=Cc1cnccn1)OC Cc1ccc(C)c(C(=O)NCC(CNC(=O)C(C)Cn2ccnc2)S(C)(=O)=O)n1 C1(C2CN(C(C3CC3C(F)(F)F)=O)C2)(NC(C(c2cn(C)nc2)=O)=O)CC1 C(=O)(C1COc2ccc(F)cc21)N1CC2(C(CO)CN(C(C3(C)CC3)=O)C2)C1 O=C(CC1OCc2cc(Cl)ccc21)NCCNC(=O)C(c1cccc(Cl)c1)(F)F C(C(C)(C)NC(=O)C(=O)NC1CC1)NC(C=CC(=O)NC1C(C)C1)=O c1(OC)ccc(C(C)=CC(=O)N(C2CCN(C(=O)C3CC3)CC23CC3)C)cc1 c1(C(=O)NCC2C(NC(=O)CC3CC3(Cl)Cl)C2)cc(C(F)F)cc(F)c1 c1(C(N)=O)ccc(C(N2CCC(N(C(C3CCCCC3O)=O)CC)C2)=O)c(F)c1 C=CC(C)CC(=O)NCCOC(C)(C)CNC(C1CCC(O)C1)=O CS(=O)CCC(=O)N1CCC(CCCCCNC(=O)CCC2CCOCC2)CC1 c1(CC(=O)NC2CCN(C(CC3CC(OCC)C3)=O)C2)ccc(Br)c(O)c1 c1(C(=O)NC2CN(C(C(C)(C)SC)=O)CC2c2ccnn2C)ccnc(F)c1N c1(C(=O)NC(C)CNC(=O)C(C)(C)Oc2ccccc2)cccc2nc(O)oc12 C(=O)(CCC(C)(C)C)N1CCC(CN(C(=O)Cc2cnns2)C)C1 c1(CNC(c2nnnn2C2CC2)C2C(c3ccccc3)C2)cc2ncccc2o1 C1(C(=O)NCCC2ON=C(C)C2)CCCC(NC(c2ccc(CO)cn2)=O)CC1 CCC(C)C(O)C(C)C(=O)NCC(C)CNC(c1c(C)ncnc1C)=O c1(CC)nc(C)[nH]c1C(=O)NCC(F)CNC(=O)C(CCSC)OC c1(-c2c(C(=O)NCC(CC)(C)NC(=O)C3CC3)c[nH]n2)ccccc1Br c1(C(=O)NC(C)CCNC(=O)CC2CCC(=O)N2C)cnc2c(c1)CCOC2 N1(C(C=C(CC)C)=O)CC2COCC(C1)C2NC(=O)CCc1cc[nH]n1 c1(CC)ccc(C(=O)NCCc2n[nH]cc2C(=O)NCC2COCC2O)o1 C(=O)(C(O)CC[S+](C)C)NCC1N(C(c2c(OCC)nccc2)=O)CC2(CC2)C1 c1(C(=O)NCCN(C(c2n(C)cnc2)=O)C2CC2)c[nH]c2cccc(Br)c12 Nc1cc(F)c(CC(N2CC3CCC(C2)N3C(C2CCCC(O)C2)=O)=O)cc1F N1(C(c2ccc(S(C(C)C)(=O)=O)cc2)=O)CC(CO)Oc2cc(F)ccc21 C1(C(N2CCC(c3nc(C)cs3)(NC(C)=O)C2)=O)CC2(CO1)CC(F)(F)C2 c1(CC(N2CC(C3(NC(CC(C=C)(C)O)=O)CC3)C2)=O)ccc([N+](=O)[O-])cc1 C(CN(C)C(C1CN(C)CC1C(F)(F)F)=O)(CO)(CO)NC(CC=C)=O c1(C(N(CCCN(C(CN(C(COC)=O)C)=O)C)C)=O)oc(C)cc1C C1(NC(c2ccn(CC)n2)=O)CCCCC1NC(=O)C=CC(C)(C)C N1(C(c2ccc(COC)o2)=O)CC(C(=O)NC(C)(C)CO)C2(CC2)C1 C(=O)(C1CCCc2c[nH]nc21)NCC(CNC(C(C(CC)C)NC(C)=O)=O)O Cc1ccc(-n2nc(-c3ccc(C)o3)nc2C(=O)NC2CC2)cc1 c1(NC(c2ccc(-c3ccco3)o2)=O)cncc(-c2ccccc2)c1 CS(=O)(=O)c1ccc(C(O)CNC(C2CC3CNCC23)=O)cc1 C1(OC)CC(NC(c2cnn(C(F)F)c2)=O)CN(C(c2cccc[n+]2[O-])=O)C1 C1(C(N(CC(C)NC(c2cc(CO)on2)=O)C)=O)CC1C1(C)COC1 c1(NC(N(C2CC2CNc2ccc(C(F)(F)F)cc2I)C)=O)ccc(C#N)c(O)c1 CC(CCC(=O)N1CC(CC(N)=O)C1)NC(c1c[nH]cc1C1CC1)=O n1(CC(=O)N(C(C)C)CCN(C(=O)CC#N)C)cc(CN2CCC2)nn1 c1(C(=O)NC(C(C)NC(C(CSC)O)=O)CO)c(C2CC2)nn2ccccc12 C(=O)(C1=CCC(C)CC1)NCCC1CCC(NC(c2cc(CC)c(CC)o2)=O)C1 C(=O)(C(C(C)CC)N(C(=O)C1=C(C)CC1)C)NC(CCC=C)CO c1(C(=O)NCC2C(C)CCC2)cc(OC2CCCC2)cc(Br)c1 CS(=O)(=O)c1cncc(C(N2CC3C(C(=O)Nc4ncc(F)s4)C3C2)=O)c1 c1(OCCC(=O)NC2C(NC(CCNC(C)=O)=O)COC2)ccccc1[N+](=O)[O-] c1(C(N(C2CCN(C(C(CCC)C)=O)C2)C)=O)cc2nccnc2cc1F C(=O)(C1=NOC(C)C1C)NCC1(CNC(C(C)c2ccsc2)=O)CC1 CC1c2ccccc2N(C(=O)CN2CCCC3(CCCNC3)C2)C1C C1(C(N(CCOCCCNC(C=CCCC)=O)C)=O)CC2CC2C1 N1(C(c2oc(CC)c(C)c2)=O)CCN(C(c2cnc(C)s2)=O)C2CCCCC12 C1(C(=O)NC2CN(C(CCCCOC)=O)C(C)(C)C2)CC(c2ccccc2)=NO1 CC1CC(O)CCN(C(C2CCCCN2C(c2cccc(=O)n2C)=O)=O)C1 C(C(C)(C)C(=O)NC(c1ccccc1)C(=O)NCCCC(C)(F)F)OCC C1(F)(NC(C(C)CCN(C)C)=O)CCN(C(=O)C(=O)NCC2CC2)CC1 C(=O)(C(C)CC(C)C)NC1(C2N(C(c3ccc(C(C)=O)cn3)=O)CCC2)CC1 C1(C(=O)NCC(C)(CO)NC(CC=CC)=O)CCCCC12CCC2 C1(CC=C)(NC(c2coc(Br)c2)=O)CN(C(c2cnn(Cc3cnn(C)c3)c2)=O)C1 c1(C(N2CCC(C(F)(F)F)C2)=O)c[nH]c2cc(-c3cccnc3)cnc12 S(=O)(=O)(C1CCCC1)N1CC(CN(C(=O)OC(C)(C)C)C2CC2)CC(OC)C1 CC1(C)CC(CNC(=O)CC2CC(F)(F)C2)N(C(c2csnc2Br)=O)C1 C(c1cncn1C)=CC(N1C(C2(NC(CC3(OC)CCC3)=O)CC2)CCC1)=O N1(C(COCCCC(C)C)=O)CC2(CCN2C(=O)CCC2CCCO2)C1 C1(CCOC)CCCCN(C(c2nonc2N)=O)C1 N1(C(C(C(C)C)c2cccnc2)=O)CC(C2(NC(=O)CC(C)C3CC3)CC2)C1 N1(C(CCC(=C)Cl)=O)CCCC2(NC(c3ccnn3C(CC)CC)=O)CC2C1 c1(CC(=O)N(CC(C)NC(=O)CCc2cncs2)C)ccc(C#N)c(F)c1 N1(CCC#C)CCC(C(N2CCC(C)C2CNC(=O)C(F)=C2CCCC2)=O)CC1 N1(C(CONC(=O)OC(C)(C)C)=O)CCC(NC(C2CCC(=O)N2)=O)C(C)(C)C1 c1(NC(CC2N(C(c3cccc(C#C)c3)=O)CCCC2)=O)ccc2nccn2c1 C1(CC=C)(NC(=O)CSc2cccs2)CCCN(C(C2CC2C(N)=O)=O)C1 C(=O)(C(C)C(=O)NCCC(C)(C)NC(=O)CN(C)Cc1ccc(Cl)s1)OC N1(C(c2n(C=C)ncc2)=O)CCN(C(=O)Cc2cncs2)CC1CCO Cc1cnc(NC(C)Cn2cncn2)c(S(=O)(=O)NC2CC=CCC2C)c1 C1(NC(C2(CNC(C3(CC#C)CCOC3)=O)CC2)=O)CCCN(C)C1=O C1(CNC(C(C(C)C)SCC)=O)CN(C(=O)Cn2nc(C)oc2=O)CC(C)(C)O1 n1(CC)cc(CCNC(c2cn(CCNC(C3(C)CCC3)=O)cn2)=O)nn1 c1(C(N(C2CN(C(C3CC(O)C3)=O)CC23CC3)C)=O)cc2ccccc2s1 Cc1ccnc2ccc(C(N3CCN(C(c4cccnc4S)=O)C4CC34)=O)cc12 C1(CNC(C=CC(C)(C)SC)=O)CCC(C(=O)NC2CCOC2C)CC1 c1(OC(C2CCN(Cc3c(Br)cncc3Br)C2)=O)ccc(C(=O)OC)cc1OC c1(C(N2C(CNC(c3cc(C)nc(O)c3)=O)COCC2)=O)cc(F)cc(C)c1C C(=O)(C=C1SCC(=O)N1C)NC1C(NC(CN(C)C)=O)COC1 C1(C)(CC)CC(NC(=O)CCNC(N)=O)CN1C(=O)CCCn1ccnc1C C1(CCNC(c2cc(C(=O)OC)on2)=O)CN(C(C23CCC2C3)=O)CCS1(=O)=O N1(C(CC)=O)CCC(NC(C2CCC3(CC2)CC3)=O)C(CO)C1 C1(CCNC(CCn2ncc(C)c2)=O)CSCCN1C(=O)CSc1n[nH]c(C)n1 c1(OCCC(N2C(CN(C(=O)CC(C)C3CC3)C)CCC2)=O)cc(F)cc(F)c1 C(=O)(C(C(C)C)S(=O)(=O)C1CCCCC1)N(CCC)CCNC(c1cnc[nH]1)=O N1(C(C2C(COC)C2)=O)CCC(CNC(c2ccc(C)cn2)=O)C(C)C1 N1(C(C(CCC)(C)CC)=O)CCCC2(CC(NC(C3CC4CCC3CC4)=O)C2)C1 N1(C(CCC2CCC(C)O2)=O)CCC(C2CN(C(=O)C3=CCCC3)C2)CC1 C(=O)(C(C)(C)C(C)O)N1CCC(N(C(Cn2c(C)cnc2)=O)C)C1 c1(CNC(=O)C(N2CCC(OC(F)F)C2)=O)ccnc(OC(F)F)c1 C1(C)(CC)CC(NC(C2(C)CC2)=O)CN1C(=O)CCc1cc(Br)cs1 CC1(CNC(C2CCS2(=O)=O)=O)CCCN(C(c2ccc3c(c2)CC3)=O)C1 c1(C(N2CC(C)C(NC(=O)CC3CCN(C)CC3)C2)=O)nnc(Cl)cc1N C=CCCCCCNC(=O)C(CO)NC(c1ccoc1CC)=O Cc1cc(C(N2CC(NC(=O)CSc3nnnn3C3CC3)C(C)C2)=O)nnc1C Cc1c(N2CC(C)OC(C)C2)nc2c(F)c(Br)ccc2c1Cl Cc1cc2nc(C(N3CC(C(=O)O)C4(CCOCC4)C3)=O)cc(=O)n2o1 C(=O)(C(O)CC(N)=O)NCC(CNC(=O)CCCN1CCCC1)OC N1(C(C2CCC(C)(C)OC2)=O)CC(CNC(=O)Cc2ccccc2)CC12CCC2 Cc1cc(C(N2CCC23CN(Cc2cc(O)ccc2Cl)C3)=O)cc(O)c1 N1(C(CNC(N)=O)=O)CCC(F)(F)C(CNC(=O)C=Cc2ccccc2)C1 C12(CNC(C3N(C)CCCC3)=O)CCC1CN(C(c1ncoc1C1CCC1)=O)C2 N1(C(C2(COC)COC2)=O)CC2(C1)CN(C(=O)C(c1ccc(C)cc1)C)C2 C(=O)(C(CCS(C)=O)N(C)C)N1CCC(C)(NC(C=C(COC)C)=O)C1 C(C(C)(C)CC(=O)NC1CC(C)(NC(c2cnc(-c3ccccn3)s2)=O)C1)OC C(C(C)(C)C(=O)NC1CCCC(CN(C)C(C23CC(COC)(CO2)C3)=O)C1)OC C1(CNC(C2C(C)C2C)=O)CC(F)CN1C(c1cnn(CCN(C)C)c1)=O c1(C(C(=O)NC(CC)CNC(=O)C#CC2CCC2)O)cc(F)c(F)cc1F N1(CC=CCC)CCC(C(=O)NC2(c3nn[nH]n3)CC2)CC1CC C1(CNC(C2CN(CC)C(=O)C2)=O)CC2(C1)CN(C(=O)C(O)C(F)(F)F)C2 C1(CC(=O)NC(CC=CC)CO)CN(C(=O)CCCCC)CC1C c1(CCC)n[nH]cc1C(N1CC(N(C(=O)C(C)CC2CCC2)C)C1)=O N1(C(C=CCNC(c2c(NC)cncc2)=O)=O)CC(C)OCC(C)(C)C1 C(=O)(CCNC(=O)C=CC(C)(C)C)N(C1CCOC1)CC#CC CCC(C)(CC(=O)O)NC(=O)CCn1cc(-c2cc(OC)cc(Cl)c2)nn1 N1(C(C2(CCOC)CCCC2)=O)CCN(C(C2CC23CCC3)=O)C(CC2CC2)C1 Cc1cc(C(N2CC(NC(c3cccc(Br)c3)=O)C(C)C2)=O)c2c(C)noc2n1 Cc1nc2cc(Cl)ccc2cc1C(=O)NCC1CC(F)CN1C(=O)C1=CCSC1 CCC(CC)(CC(=O)OC)C(=O)N1CC(NC(=O)CCS(C)=O)C2(CC2)C1 c1(C(=O)NC2CCN(C(c3c(C)cnnc3)=O)CC2)c(Cl)cccc1Br Cc1cccc2c1NCCC2C(=O)Nc1ccc2c(C(=O)O)nn(C)c2c1 CC1CCN(C(=O)CCC(=O)NCCC(N)=O)CC1NC(C12CC(CCO1)C2)=O c1(N2CCC(OCC(N3CCCC(C(F)(F)F)C3)=O)C2)cncc(Cl)n1 Cc1cncnc1C(=O)NCC(O)CN(C)C(c1nnc(S)n1C)=O C#CC1CCN(C(=NCCSc2ccc(Cl)cc2)NC(c2ccccc2C)C)C1 c1(C(=O)Nc2cccc(CCC)n2)[nH]c(C)c(C(=O)NC2CSC2)c1C CC(N=c1[nH]c2ccccc2s1)C(=O)N1CC(C(=O)NCc2ccc(F)cc2)C1 C1(C(N2CC(C)C2)=O)(CO)CCCN(C(C2(c3ccccc3)CCC2)=O)C1 C(=O)(C1=CCCC1)N1CCC(CNC(C2C(C)C2)=O)C1 c1(C(N2C(CCNC(C3(C#C)CC3)=O)CCC2)=O)cc2c(C)ccc(F)c2o1 c1(CN(C(=O)CC2CCCO2)C)cnn2c1CN(C(C1(F)CCCCC1)=O)CC2 c1(OC)ncc(C(=O)N(C2CCCN(C(=O)C(=O)NC3CC3)C2)C)nc1C c1(C(=O)NCC2C(OCC)CN(C(=O)CCNC(N)=O)C2)noc2ncccc12 C(CN=c1[nH]c2ccccc2s1)N(C(C1CC2CC2C1)=O)CCOCCC1CC1 Cc1c(NCC(C2CCC2)C2CC2)ncnc1NC1CC1 C1(C(N(C)CCN(c2ccc3nnnn3n2)C)=O)CCc2nnc(O)cc2C1 N1(C(C(c2ccccc2)C)=O)CCCCC1C1CCCN(C(C2(CO)CCC2)=O)C1 N1(C(CC2(C(=O)OC)CC2)=O)CC2=C(C1)CN(C(=O)C=Cc1ccccc1)C2 CC1=CCC(C)(C(=O)NCC2CC(NC(c3cnc(C4CC4)s3)=O)CC2O)CC1 Cc1nn(CC(=O)NC2CCN(CCc3cn(CCCF)nn3)CC2)c(C)c1C CC(COc1ccccn1)N=c1[nH]c(=N)[nH]c(=NC2CC2C2(C)CCOCC2)[nH]1 C(C1CCCc2cccnc21)NC(C1CCNC12CCSCC2)=O C1(CNC(C2CN(CC)C(=O)C2)=O)CC2C=CC1CC2.C12(CCCCC1)C(=O)N2 CC(C)(C)C(CNC(=O)C1=NOCC1)C(=O)NCC1CC2C=CC1O2 C(CN=c1[nH]cncc1Cl)C1(O)CCN(C(c2cccc(C3CC3)n2)=O)CC1 C1(NC(c2n(CC)cc(Br)c2)=O)CC2CC(NC(c3nnn(C)n3)=O)C2C1 c1(OC)cc(=NC(=O)C2=NN(c3nc(C(C)OC)nc(OC)n3)C(=O)C2)[nH]n1C N1(C(C(n2ncc(C)c2)C)=O)CCC2CCN(C(=O)CNC=O)CC12 c1(C(=O)NC2CCN(C(CC3NC(=O)OC3)=O)C23CC3)cncc2cnccc12 C1(C(=O)NCC(CC)CC)CCC(NC(c2coc(COC)n2)=O)CC1 C(=O)(C1CCc2c[nH]nc21)NCC(CC=C)NC(c1cnc(O)n1C)=O C1(NC(C(C)NC(=O)COC(=O)C2CC2)=O)CC(C)(C)OC1(C)C c1(CC)nc(C)[nH]c1C(=O)NC1CCN(C(=O)C(c2cccnc2)N(C)C)CC1 N1(C(c2ccc(CN(C)C)o2)=O)CCCCC(CNC(=O)CCNC(=O)CO)C1 C12(C(=O)OC)CC1CN(C(=O)C(F)CC1CN(C(c3ccc(C(C)=O)o3)=O)C1)C2 c1(C(=O)OC)ccc(C(=O)N(C)C)cc1F.C12C3CN(CC13)C2 N1(CCC(=O)NC2C=CCN(C(CC(CCC)O)=O)C2)CCCc2ccccc21 C1(N(C(CC(CNC(C2C=C(CO)CCC2)=O)OC)=O)C)CC(C)CC(C)C1 c12cc(C)ccc1S2.C1(C(=O)OC)CCC(C(=O)OC)C1.C12CCN(C1)C2 N1(C(c2ccc(C#N)cc2)=O)Cc2ccc(O)cc2CC1C(=O)C1CC1 CCC(C#N)C(=O)N1CCCC1CCNC(=O)CC1(C)CCCC1 c1(CO)cc(F)c2ccc(Cl)cc2c1 C1(CNC2CCN(C(N(c3cccc(F)c3)C)=O)C2)CC2(CCOCC2)CO1 c1(NC(CC(=O)NCc2cccc(Br)c2Br)c2ccccc2)cc(Br)nc(Br)c1 C12C3CC4C1C4C3C(=O)N2.C1(C(=O)NC2(C(C)(F)F)CC2)CN(C(C)C)CCO1 CN1CCC(O)(C2(C(N3CCC(CN(C(=O)C4=CCCCO4)C)C3)=O)CC2)CC1 Cc1nn(C)cc1OCC(N1CCC(O)(C(N2CC(c3ncccn3)C2)=O)C1)=O c1(C(=O)NC2C(NC(CSCC=C)=O)CCCC2)cnc(C)nc1OC c1(CNC(C2N(C(C(CN(C)C)(C)C)=O)CCC2)=O)cc(F)cc([N+](=O)[O-])c1 CC1CN(C(=O)Cn2ncccc2=O)CC(CNC(=O)NC23CC4CC2C3C4)O1 Cc1cccc([N+](=O)[O-])c1NCC1(F)CC(NC(=O)C=Cc2ccccc2F)C1 C=C(Br)CC(C)(C)C(=O)NCC1CCCCN1C(=O)C(C)=C(C)CC c1(C(=O)NCc2ccc(CCNC(C(C)C#N)=O)cc2)ccc2c(n1)CCCC2 c1(C(=O)N(CCN(C)C(C2CC2c2ccnn2C)=O)C2CC2)c(F)cncc1Br Cc1cnc(C(N2CCC(OCCNC(=O)CC3CCCC3(F)F)C2)=O)c(C)c1 c1(C(=O)NCCCOCCNC(CCc2cnc(C)o2)=O)cc(C(C)C)n(C)n1 C1(C(=O)NC2(COC)CCCC2)CC12CCN(C(c1cn[nH]c1)=O)C2 Cc1ncc(CC(N2CC=CC2C(=O)NOCCF)=O)s1 C1(C(N(CCN(C(=O)CC2COCC(C)(C)O2)C)C)=O)CC(F)(F)C1(C)C C1(CCNC(c2ccn(CCF)n2)=O)CSCCN1C(C1CCC1(F)F)=O c1(C(N2CCC(F)(CNC(CCC(C)N(C)C)=O)C2)=O)ccn2ncccc12 CC1CN(C(=O)Cc2ccoc2)CCCN1C(=O)CCc1ccc(C#N)cc1 N#CCCCCCC(=O)NCC1CCN(C(C2CCCS2)=O)C1 C1(NC(c2n(CC)ccc2)=O)CCCCN(C(=O)C(C)OCCC(C)C)C1 N1(C(c2c(CC)n(C)nc2)=O)CCC(C)C(CC(=O)NCC(C)C(C)(F)F)C1 C1(NC(CCN(CC)CC)=O)CCC2(CCN(C(C3(C(=O)NC)CCC3)=O)C2)C1 c1(C(=O)Nc2cccc(CNC(=O)NCC)c2)ncn2c1COCC2 C1(C(N(CC(C)(CO)CO)C)=O)COCCN(C(C2CN(C(N)=O)C2)=O)C1 C(CCC(C)CC(=O)NCC1(NC(=O)CC2CCC3(CC3)CO2)CCC1)=C(C)C c1(C(C)=O)[nH]c(C)c(C(N2C3CCC2(CNC(=O)COCC(F)F)CC3)=O)c1C S(=O)(=O)(c1ccc(NCC2CCC2)c(F)c1)N1CC(CC)OCC1 C1(C(N(C2C(C)CCC2)C)=O)CC2(CC2)CN1C(=O)CCc1cnc[nH]1 C1(CC)CC(CC(=O)N(C)CC2(CNC(c3ccccc3O)=O)CC2)CCO1 C1(N(C(C2CCC(CN(C)C)O2)=O)C)CCCN(C(c2ncncc2Cl)=O)C1 c1(C(=O)OCc2cccc(OC3CCNCC3)c2)cc2ccc(O)cc2oc1=O C1(CC(=O)NCCCCN(C(CNC(CCNC(C)=O)=O)=O)C)CCCC1(F)F C1(NC(CC2C(CC)C2(F)F)=O)CN(C(c2c[nH]nc2OC)=O)CC12CCC2 c1(-c2cn(CC(CNC(C(C)NC=O)=O)(F)F)nn2)cccc(Cl)c1 C1(NC(CSc2cccc(C)c2)=O)CC2(C1)CC(C(=O)NC(C)(C)CF)C2 N1(C(CC2CN(C)C2)=O)CCOCC2(COCCN2C(c2ccc(Cl)nc2)=O)C1 c1(CC(N2CCN(C(CC(CC)C)=O)CC2CC)=O)ccc2c(c1)OC(F)(F)O2 C1(NC(=O)C)CCc2nnc(O)n2C1.c1(C(=O)NCC2(C)CC2)ccc(F)c(Cl)c1 C1(CN(C(=O)Cc2ncc(Br)cn2)C)CCN(C(C2CC2F)=O)CC1 c1(C(N2CCCN(C(CC(C)(C)OC)=O)CC2)=O)ccc([N+](=O)[O-])c(C)c1 c1(C(C)(C)OC)occc1NC(=O)N(CCN(C)C)Cc1cocn1 N1(C(c2c(OC)c[nH]n2)=O)CCN(C(=O)C(c2ccccc2)F)CC1CC(F)F N1(C(CCCc2cn(Cc3c(OC)cccc3)nn2)=O)CCS(=O)CC(C)C1 C(=O)(C(F)C1CCCC1)NCCCN(C(=O)CC1(C(F)(F)F)CC1)C(C)C C1(NC(N2C(CC)CCC2C)=O)COc2cc(CO)nn2C1 n1(CC(=O)OCC(=O)OC)[nH]cnc1=NCc1ccccc1CN=[N+]=[N-] C1(NC(CCCNC(=O)OC)=O)CS(=O)(=O)CC1NC(=O)Cc1ccon1 CC(C)C(C(C)NC(=O)C1=CCCC1)NC(c1csc(Br)n1)=O N1(C(c2cnn(C)c2Cl)=O)CC(NC(=O)Cc2c(F)cccc2F)C(C#N)C1 CCCCCCC(=O)N(C1CCC(NC(=O)COC(C)CC)CC1)C C1(C(=O)NCC(=O)N(CCC#C)C)(CO)CCC1 N1(C(Cc2n(C)cnc2)=O)CC2CCC(NC(C3CC4CCC3C4)=O)CC2C1 CC1=C(C(=O)NC2C=CCN(C(=O)COc3cc(F)cc(F)c3)C2)CCCC1 C1(O)(CC(=O)NC(CC)(CNC(c2ccc(C)nc2)=O)CC)COC(C)(C)C1 CCC(C#N)C(=O)N1CCCCC1c1n[nH]cc1C(=O)NCc1ncc(C)[nH]1 N1(C(c2nc(OCC)oc2)=O)CC(CNC(=O)Cc2csc(C(C)=O)c2)C(C)C1 N1(Cc2cc(OC)c(O)cc2)CCCC2(CCN(C(C3CCC(F)(F)C3)=O)C2)C1 N1(C(C(C)C)=O)CCC2(CCC(C(F)(F)F)N2C(c2cnccc2F)=O)CC1 C(=O)(C(C)(C)C(C)NC(=O)CC1(O)CCC1)N(C)CC1C(C)C1 N1(C(c2c(C)onc2C(F)(F)F)=O)CCCCC(CNC(C2CCNC2=O)=O)C1 c1(OCC)cc(F)ccc1NC(C1OCCC1NC(=O)Cn1ncn(C)c1=O)=O C1(NC(c2c(C)nc(C(C)OC)s2)=O)CN(C(=O)C=CSC)C(C)(C)C1 c1(CN2CCCC(CNC(=O)NCCCl)C2)cc2ccoc2cn1 C1(C(C)O)CN(C(=O)CN(C)C(C2CC23CC3)=O)CCO1 Cc1ccc(SCC(N2CCC(NC(c3[nH]ccc3C)=O)C2)=O)cc1 C1(NC(C(CC=C)C)=O)C2COCC1CN(C(c1cc(C)[nH]n1)=O)C2 C12(CC(=O)NCC(C)CNC(=O)C(C)n3ccnn3)CCCN1CCC2 c1(CNCCOCCC(C)CO)ncccc1O C#CCC(C(=O)NOC(C)(C)C)NC(=O)COCc1ccccc1 c1(C(=O)NC2C(CNC(c3c(CC)onc3)=O)C2)cc(Cl)cc(C)c1C CC(CCNC(=O)CCOC1CN(C(C2CCCCO2)=O)C1)C(C)(C)C N(C(=NCC=CC1CC1)NCc1ccco1)CC1(C)CCCO1 c1(OC)ccc(CC(=O)NC2CCN(C(c3cccnc3N)=O)CC2F)c(F)c1 C(=O)(C(CNC(=O)OC)CSC1(F)CC(c2ccccc2)C1)OC(C)(C)C Cc1ncc(C(N2CC(O)CCC2C(=O)NCC2CC3(CCC3)C2)=O)cc1C#N CC(N=c1[nH]c(=NC(C)CS(C)(=O)=O)[nH]c2c1COC2)C1CCC1 Cc1[nH]nc2c1CC(C(=O)NCCCC(C)(C)NC(=O)C(O)C(F)(F)F)CC2 Cn1ccc(C(=O)NCC2CCC(N(C(=O)C=C3CCSCC3)C)CC2)cc1=O N1(C(CSCC#C)=O)CCN(CC(=O)NCC2CC(CCC)C2)CC1 c1(OC)cccc(C(c2nnnn2C(C)(C)C)NC2(C)CCOC2)c1 N1(c2cc(N(C)C)[nH]c(=N)n2)CCC2CC(C(=O)NCC(C)O)C2C1 c1(CNC(C(C2CC2)OCC)=O)cncc(C(=O)NC2CC(=O)N(C)C2)c1 C(=O)(C(C)CSC)N(CCN(C(CC1C(OCC)CC1)=O)CC)CC.C.NCC c1(C(N2CCN(CC(O)C3CC3)CC2)C(=O)NCC(C)C)ccnc(Cl)c1Br [N-]=[N+]=NCCCC(=O)NC1CCCCCC1NC(=O)Cn1cc(Cl)cn1 C1(NC(CC(CC)SC)=O)CCC2(CCN(C(c3ccnc(Cl)c3O)=O)CC2)C1 C(=O)(C1=NOC(C)C1C)NC(CCC(=O)NC(CCOC)C)(C)C c1(C(=O)NC2(CCO)CN(C(=O)CC3CCOC3)C2)cccc2sncc12 Cc1scc(C(=O)NC2C3CC2N(C(c2cc(C(N)=O)c[nH]2)=O)C3)c1C Cc1ccc(Br)c(C(=O)NC2CC(C)N(C(=O)Cc3nnc(O)s3)C2)c1 C(=O)(C(C)COC)NC1C(CNC(CNC(CCOCCOC)=O)=O)CC1 c1(C(C2CC2)NC(CC=CCC)=O)ccc([N+](=O)[O-])cc1 C(=O)(C(C)CC(F)F)NC1(CC(=O)NC(CCC)CO)CCCCC1 N1(C(C(CC)=C2CCCCC2)C(=O)NCC(F)F)CCc2cc(F)ccc21 c1(C(N(C2CCN(C(C(CSC)O)=O)CC2)CCO)=O)cnc2cccnc2c1 C1(C(N2C(N(CC)CC)C(C)(C)C2)=O)CC2(CC2)CN1C(c1cc(I)ccc1C)=O N1(C(c2c(CC)occ2)=O)CC2(CCN(C(c3ccc(O)cc3Cl)=O)C2)C1 N1(C(c2c(C)onc2CO)=O)C2CCC1CN(C(C1CC(C)(C)CO1)=O)CC2 N1(C(C(=O)NCCC2CC2)C2CCCC2)CCCCC(C2CCOCC2)C1 C1(COC)(NC(=O)NCCCN(C(=O)CC2CC2C)C)CCCCC1 c1(N2CCC(C(C)NC(C3(OC)CCOCC3)=O)C2)nc(C)cc(C)n1 N1(C(C2(C)COC2)=O)CCC2(CC1)CC(NC(C1(C3CC3)CCCO1)=O)CCO2 S(=O)(=O)(c1cncc(Br)c1)N1CC2N(C(=O)CCc3ccc(CO)cc3)C2C1 C1(C(=O)OC)CCN(C(=O)Nc2cccc(C3SCCS3)c2)C2(CC2)C1 C1(CC(=O)N(CC(=O)NCCCc2cnccn2)CCC)C(=O)NN=C1C C=CCC(F)(F)C(=O)N1CC(NC(=O)Cn2ccccc2=O)CC(C)C1 N1(C(c2c(C)cc(Cl)cc2)=O)CC2CN(C(C3CC(C)(C)OC3(C)C)=O)CC2C1 Cc1nc2ccc(C(=O)NC(C)CC3CCN(C(=O)CSC4CC4)CC3)cc2[nH]1 C1(C(N2CCC(CC(C)NC(C3CCCC(O)C3)=O)CC2)=O)CC2(C1)CC(F)C2 N1(C(c2cc(C)c(-n3cncn3)cc2)=O)CCC(CNC(=O)CNC=O)C(F)(F)C1 c1(C(N(CC(C)NC(C2CC(n3cnnc3)C2)=O)C)=O)cc(C#N)on1 CCCCC(CNC(C1CCC(NC(C)=O)CC1)=O)NC(c1cc[nH]n1)=O C1(CNC(CN2CC(C)(OC)C2)=O)CN(C(C2(C)C=CCC2)=O)CC1(F)F c1(C(=O)NCC(CC)NC(c2cnc[nH]2)=O)ccnc(C(C)(F)F)c1 c1(C(N(CC(C)NC(C2(C)CC(C)C2)=O)CC)=O)cnn2c1CCCC2 Clc1cc(-n2cc(C3CCOC3)nn2)cc(Cl)c1Cl O(NC(=O)CN(C(=O)CCOCCCO)CC1CC1)CC(=O)OC CC1CCN(C(c2ncoc2C(F)(F)F)=O)C(C)C1NC(=O)C=Cc1nccs1 CCC(O)(C(=O)N(C(CNC(c1ccc(C)nc1)=O)C1CC1)C)c1ccccc1 O=C(CC(O)CNC(c1cnn(CC2CC2)c1)=O)NCC1CCC(C2CC2)O1 CCCCCCC(=O)NCC1COCCN1C(=O)C=CSC c1(CC(N2CC(CCNC(c3nc(OCC)oc3)=O)C2)=O)ccc(C(N)=O)nc1 C12C3CCC(C3)C1NC(=O)C(=O)N2.c1(C(N(C)C)=O)ccc(COC(C)C)cn1 C1(NC(c2ccc(C)cn2)=O)CC(CNC(=O)Cc2cc(C)[nH]n2)C12CCC2 C1(CC(=O)Nc2cnc(C)s2)CCCCN1C(c1ccccc1-c1nn[nH]n1)=O C(=O)(C(C)(F)C(=O)N1CCC(NC(=O)CS(=O)(=O)C(C)C)C(O)C1)OCC C1(C(C2(CF)CC2)C)CCCCC1C(=O)N.C1(=O)CC2(CC2)CN1.C1(SC)CC1 N1(C(C2(CCNC(c3c(CC)[nH]cc3)=O)CC2)=O)Cc2ccnn2CC1C C1(C(=O)OC)CCCN(C(=O)NCC2(Nc3ccccc3)CCN(C)C2)CC1 c1(C(N2CCCC(NC(C=C(C)Cl)=O)C2)=O)c(N)cc(F)cc1Br C(=O)(C1(C)CCCc2ccccc21)NC1C(NC(c2c(C)ccc(F)c2N)=O)C1 N(C1CCc2sc(Cl)cc21)C(c1c(C)n(-c2cnn(C)c2)nn1)=O C1(C(=O)NC(C(O)CO)C2CC2)CN(C(C2(O)CCCCC2)=O)CC12CCC2 C=CCCN=C(NCc1cccc(C(C)C)n1)NCc1ccnn1C1CC1(F)F S(=O)(=O)(c1ccc(C(=O)NCC2(C)CC(NC(=O)C3=COCCC3)C2)cn1)NC C1(N(C)C(c2cc(C(F)F)no2)=O)CN(C(c2cc(O)nn2C)=O)CC1(C)C S(=O)(=O)(c1ccc2c(c1)C(=O)C(=O)N2)NCC.n12c(C)cc(c1C)C=CC(C)CC2 Cc1c(C(=O)NCC2CCC2NC(C2CCNC2=O)=O)sc2[nH]cnc(=S)c12 C1(NC(CCCCCCSC)=O)CC2CCCC(C1)N2C(c1ncncc1F)=O c1(C(N(CCCCNC(c2ccc(-c3ccncc3)o2)=O)C)=O)cnc(=N)[nH]c1 CCCC(C)CCN=c1cc[nH]cc1S(=O)Cc1ccc(C(C)(C)C)cc1 n1(CCC(=O)NCC2(COC)CCCNC2)cc[nH]c(=O)c1=O C12(CC(F)C1)C(=O)N2.C(=O)(C=CC(C)C)NC1(C(COC)O)CC1 c1(NC(C(CC2CCC2)NC(C(CCCOC)C)=O)=O)cccc([N+](=O)[O-])c1 n1(C(CNC(c2ccc(Br)s2)C)=O)ccc(=NC(=O)OC(C)(C)C)[nH]1 CC(C)C(C(=O)NCCNC(C1CSCCS1)=O)S(=O)(=O)C1CCCCC1 O=C(CC1OCCc2ccsc21)NCC1(CNC(c2ncc(C(F)F)s2)=O)CC1 C(c1ccnn1C)=CC(=O)N(C)CC1(NC(c2c(OC)scc2)=O)CC1 N1(C(c2c(CC)cccc2)=O)CC2CCCC(C1)N2C(C1CC(F)C1)=O CCCCCCC(C)C(=O)NC1(C)CCN(C(c2cnc(OC)cn2)=O)C1 C1(C(=O)NC2CC(CCNC(CCc3n(C)ncc3)=O)C2)CCc2nnnn2C1 C(C(CC(C)C)C(=O)NCC1(n2ccnn2)CC1)NC(C(CC)(F)F)=O S(=O)(=O)(CC(=O)NCC1(F)CC(CNC(=O)C(c2cccc(F)c2)C)C1)NC C1(CNC(CC2CC(C)C2)=O)CCC(N(C)C(c2sccc2C2CC2)=O)CC1 C1(=CC(=O)N(CCC(C)(C)NC(Cc2cc(C)on2)=O)C)CCN(C)CC1 N1(C(CCNC(c2cn(C(C)C)nn2)=O)=O)CCCC(CO)C1 c1(C(=O)NCC2CC(NC(C(C(CC)C)C)=O)C2)cc([N+](=O)[O-])cnc1C c1(C(=O)NCC(C(=O)NC(CN(CCC)CC)C)N(C)C)cc[nH]c(=NC)c1 c1(C(N2C(CNC(CC(C)C(F)F)=O)CC(F)(F)C2)=O)cc2ccc(F)cc2s1 Cc1cnc(Cl)[nH]c1=NC1CC2CN(C(=O)C(C)C(C)C)CC12 CN=S(C)(=O)c1cccc(NC(=O)Cn2cnc3ccsc3c2=O)c1 N1(C(C2CC(CC)C2)C(=O)NCCCF)CCC(C)(O)C(C)(O)C1 Cc1cc(C)c(C(N2CCSCC2C(=O)N(C)CC2CCOC2C)=O)s1 C(C(C)(CC(C)C)NC(c1cn(CC)cn1)=O)NC(C(CC=C)C)=O C(=O)(C=C1SCC(=O)N1C)N(C1CCN(C(=O)C2=NNC(=O)CC2)CC1)CC#C c1(C(N2C3C(NC(C(C(C)C)(C)C)=O)CC(C3)C2)=O)sc([N+](=O)[O-])cc1Cl C=CCC(C(=O)N1CCC(C)(NC(c2ccc(CN(C)C)nc2)=O)C1)NC(C)=O Cc1nc2ncnn2cc1C(N1CC2CCN(C(c3csc(Cl)n3)=O)C2C1)=O c1(N2CCC(COC)C2)nc(N2CCN(C)C(=O)C2)c2ccccc2n1 c1(C(=O)NC2CCN(C(C(N3C(=O)CCC3=O)CC)=O)C2)sccc1S(N)(=O)=O n1(CC)ncc(C(N2CC(NC(=O)COC3CCCCC3)C(CO)C2)=O)c1C N1(C(c2n(C)c(Cc3ccccc3)cc2)=O)CCc2ccc(F)c(Br)c2C1 Cc1cc(Br)c2c(c1)CN(C(C1C3CCOCC13)=O)CC2 c1(C(=O)NCC(C(C)C)NC(=O)C(C)(C)N2CCCC2)cc(CO)ccc1Cl C#CCCCCCC(=O)NCC(=O)N.C(C(C)C(C)(C)C)CNC(COC)=O n1(CC#C)c(C)cc(C(=O)NC2CCC(NC(c3ccc(F)c(O)c3)=O)C2)c1C Cc1c(Br)ccc(S(=O)(=O)N2CCCN(CCS(C)(=O)=O)CC2)c1F c1(C(=O)NCCN(C(C=C(C)C)=O)CC(C)O)cn2c(Br)c(C)nc2s1 Cc1ccc(I)c(NC(C2CN(C(c3cccn3C(C)C)=O)CCS2)=O)c1 c1(COC(C2(Cc3ccc(Cl)cc3Cl)CC2)=O)cc2cc(F)ccc2o1 Cc1nc(N2CCC(C)C(NC(=O)C(C)Oc3cccc(F)c3)C2)c(C)c(Cl)n1 C1(CC(=O)NCC(C)OC(F)F)N(C(=O)C(=O)C(C)(C)C)CCC1(C)C Cc1cccc(CNC(C2CC(F)CN2C(=O)CC2(C)CCCCC2)=O)c1F c1(C(=O)NCC(n2cc(-c3ccn(C)n3)nn2)C)cnnc(Cl)c1 C1(CC(=O)NCc2n(C)ncc2)CCCCN1C(=O)CCn1cccn1 C(=O)(C(CC)(CC)OC)N1C(CN(C(C=CCN(C)CC)=O)C)CCC1 C1(NC(C2(COC)CC(=O)C2)=O)CCN(C(=O)C(Cl)=CCl)CC1C c1(C(C(=O)NCC2C(NC(C(C)(C)OC)=O)CCC2)OC)ccc(OC)cc1 c1(C(=O)NCC(CN(C(CCOCC)=O)C)(C)C)cnc2ccoc2c1 C1(NC(c2c(C)ccn2C)=O)CC2(CCC(NC(C3CC4CCC3C4)=O)CC2)C1 c1(OCC)cccc2c1CCC2NC(=O)C(=O)N(C(C)CC)CC C1(NC(CCC=C)=O)CC(OC)CN(C(c2c(C(F)(F)Cl)n[nH]c2C)=O)C1 C1(C(=O)NC(CC2CCN(C(c3cccc(C)c3)=O)CC2)C)CC2(C1)CC2(F)F C1(NC(CC(CC)O)=O)CN(C(=O)COC(C)CC)CCC1C(F)(F)F CCCC(C(=O)NOC(C)(C)C(=O)OC)NC(c1c(Cl)cnn1C)=O c1(C(=O)NC2C(NC(c3nc(N(C)C)oc3)=O)CC2)cc(Cl)sc1Cl c1(C(=O)NCC2C(NC(C(N3C(=O)CCC3=O)CC)=O)C2)ccc(Br)cn1 c1(C(N2CCOCC(NC(CC=C)=O)C2)=O)c(C)nc(C(C)C)nc1O N1(C(c2c[nH]c(=N)o2)=O)CCN(CCNC(C23CC(F)(C2)C3)=O)CC1 Cc1cc(C(N2CCC(CN(C)C(c3cc[nH]n3)=O)C2)=O)cc([N+](=O)[O-])c1Cl Cc1ccnc(C(=O)NC(CNC(=O)C(C)OCc2ccncc2)C(C)C)n1 C(CNC(c1cc(Br)sc1C)=O)(C(C)(C)C)NC(CNC(=O)OC)=O c1(C(N(C2CCCN(C(C3C(=C)C3)=O)C2)C)=O)cc2c(F)cc(F)cc2o1 C1(NC(C=CCNC(C(C)(C)OC)=O)=O)CCCSCC1 c1(C(=O)NCC(CC(C)C)NC(C2(CC)CCNC2=O)=O)c[nH]cc(F)c1=O N1(C(CCCCCC#C)=O)CC(CNC(=O)C(=O)NCC)CC12CCOCC2 C(=O)(C(O)CCC(F)(F)F)N1CCC(CN(C)C(C2CC3(CCO2)CC3)=O)C1 C(CCCC(C)NC(=O)Cn1nnnc1C(C)C)NC(C1C(C(=O)OC)CC1)=O C(=O)(C(C(C)(C)C)C1CCC(F)(F)CC1)NCCN(C(=O)C(F)C(C)(C)O)CC Cc1cn2c(C(=O)NC(C3(O)CN(C(C4CCC(=O)C(C)C4)=O)C3)C)cnc2s1 N=c1nc2c(c[nH]1)CC(C(N1CCCN(C(c3ccsc3)=O)CC1CO)=O)CC2 N1(CCC)C(=O)CCC1C(=O)N(C)CCN(C)C(C1CC1c1ccc(Cl)cc1)=O c1(SCC(=O)N(CCCNC(C2C(C=C)C2)=O)C(C)C)ccccc1O C(=O)(C#CC(C)(C)CNC(=O)CC1CCC(O)C1)NCCc1c(C)nccn1 c1(C(=O)OCC(CCCC(=O)OCC)=O)cc2n(n1)CCCNC2=O c1(OC)ccc(O)c(C(=O)N(C)CCNC(C2(CF)CC2(F)F)=O)c1 C1(C#N)(C(=O)NCC2C(C)CCN2C(C2CC(=O)NC(=O)N2)=O)CC2C=CC1C2 N1(C(C2(C)CC2F)=O)CCN(Cc2nc[nH]n2)CC1 c1(OC)ncc(Cl)c(C(=O)NCC2CCN(C(c3conc3C)=O)CC2C)c1Cl N1(CCCNC(C2C(C=C)OCC2)=O)CCCNS1(=O)=O N1(C(C(C2CN(C(CC=CCCCCC)=O)C2)O)=O)CC(CO)C(C)C1 C1(NCc2cn(C3CCN(C(CSC(C)C)=O)C3)nn2)CCCC(C(F)(F)F)O1 CC1CCCC(CCN(C(C2CCCN(C(=O)Cc3cnoc3)C2)=O)C2CC2)C1 C1(C)(CC(=O)OC)CCCN1C(=O)NCc1ccccc1-c1cn[nH]c1 S(=O)(=O)(c1ccc(Cl)cc1C(F)F)NC(c1ccc(Cl)c(F)c1)C c1(CC(=O)N(C2(CC=C)CNCCO2)CC)cc(F)c(C)cc1F N1(C(C(C(C)C)c2cccs2)=O)CC2(CCN2C(N)=O)C1 CC1(C)C=CC(NC(c2cc(CNC(=O)CCN3CCCCC3)cs2)=O)CC1 N1(C(C2(CC#C)CCOC2)=O)CC2CC(C1)N2C(=O)C(O)Cn1cncn1 C(=O)(C1CCCn2cnnc21)NC(CNC(Cn1ncc(C#C)c1)=O)C1CC1 N1(C(c2cc(OC)c(Cl)cc2)=O)CCC2(CCCC2C(=O)NCCNC(C)=O)C1 CCC(CC(F)(F)F)C(=O)NCCC1CN(C(=O)CC2CC3(CC3)C2)CC(C)O1 C1(N(C(=O)CCC2CCCN(C)C2)C)CC2CCC(C1)N2CC1CCCC1 CC1OC(C)(C)OC1(C)C(=O)N(C)CCN(C(=O)C=Cc1nnn(C)n1)C CCS(=O)(=O)CC(=O)N1CCCCC(NC(c2cnn(C(C)(C)C)c2C)=O)C1 C1(CNC(CC(CCC)O)=O)CN(C(=O)C=CC=C(Cl)Cl)CC2(CCC2)O1 N#CC1(CNC(=O)C(C2CCOC2)NC(c2cccc[n+]2[O-])=O)CCOCC1 c1(C(N(CC(CC)NC(c2ccncc2)=O)CC)=O)ccnn1C1CCCCC1 C=CC(CCC)CC(=O)N1CCN(C(=O)CC(O)CC(C)C)C(C)C1 N1(C(CNC(CC)=O)=O)CCC(CNC(c2ccc(Br)cc2O)=O)C1(C)C CCCC(C)(C)CC(=O)NC1CCCC(NC(=O)COCCSC)CC1 N1(C(C(C2CCCO2)NC(CC(=O)NCC#C)=O)=O)CCC(C)(C(=O)OC)C1 N1(c2cc(C)nc(C)n2)CCC2(CC1)CC2NC(=O)CC(C)C c1(CCNC(C2C(C)CCCC2)=O)cn2c(n1)CCCC2 N1(C(C2(CC=C)CCCNC2)=O)CCN(Cc2ccc(Cl)cc2)CC(O)C1 C(=O)(CCC(C)S(C)(=O)=O)N(C1CCC2CN(C(COC(CC)(C)C)=O)CC21)C C1(NC(=O)CCOC2CCC2)CC(F)(F)CC1C(=O)Nc1ncc(F)cn1 CC1CCCC(C(N2CCC(C3CCCN3C(=O)CC3C=CCC3)C2)=O)CC1 c1(C(N2C(C(C)NC(CN3C(C)CCC3)=O)CCC2)=O)cccc(O)c1Cl c1(CNC(CCNC(=O)OC)=O)n[nH]cc1C(C)C c1(C(=O)NCC2C(NC(CC(C(C)C)C)=O)CC2)sccc1S(=O)(=O)C(F)F C=CC1(CC(=O)NC2CCN(C(C)=O)C2C)CN(C(=O)COC)C1 c1(-c2c(SC)cc(F)cc2)ccc2c(O)c(C(=O)NC(CO)CC(C)C)sc2c1 C#Cc1cc(C(=O)NC(CNC(=O)C(CC(C)C)OC)C2CCC2)cc(N)c1 c1(C2(C(=O)NCC34N(C(C(C)O)=O)CC(C3)C4)CCC2)ccc(S(N)(=O)=O)cc1 c1(CC(=O)N(C2CCCCC2)CCCNC(CCOC)=O)sc(C)cc1C C1(CC(=O)NCCN(C(=O)CCCc2cnccn2)CC2CC2)COC(=O)N1 C1(CC)(NC(=O)COCC2CCCC2)CCCN(C(=O)C=CSC)C1 C1(C(=O)OCC)CC2(C1)CN(CCCC1CC(C(C)(C)C)C1)C2 C#CC1CCN(C(C2CC(NC(c3ccc(CO)s3)=O)CCO2)=O)C1 C=CCCC(O)CNC(C1(CO)CCN(C(=O)CC2CCC(C)CC2)C1)=O c1(CC(C)C(=O)NCC2(NC(C3CC3F)=O)CCC2)ccc(F)cc1 c1(OC)ccc(OC(C)(C)C)c(NC(=O)N(S(=O)(=O)C2CN(C(C)=O)C2)C)c1 N1(C(C(CCC)NC(=O)Cn2ccc(C)n2)=O)CC2(CC(N(C)C)C2)C1 C1(NC(C=CC(C)(C)C)=O)CN(C(c2ccc(C(O)CF)cc2)=O)CC1(C)C c1(C(C)C)ncc(C(=O)NCC(C2CC2)NC(C2CC(CC3CC3)C2)=O)n1C N1(C(C(=O)NCCOC)=O)CCC(CO)C(NC(c2oc(Br)nc2C)=O)C1 CC(CC(C)(C)C)C(F)C(=O)N1CC(CCNC(=O)C=Cc2cocn2)C1 Cc1ccc(Cl)c(N=c2scc(-c3ccoc3)n2CCC(=O)NCC(C)C)c1Cl c1(CCC(N2CC(CNC(C(C3CCC(=O)C3)(F)F)=O)C2)=O)ccc(O)c(F)c1 c1(C(N2CCC(OCCCF)CC2)C(=O)NCC(F)F)ccc(C2CC2)cc1 C(=O)(C1=Cc2ccccc2C1)N1CC2C(C(N3CCC(CCC)C3)=O)C2C1 C(CC(C(N)=O)NC(=O)CONC(=O)OC(C)(C)C)OC c1(C(=O)NC2C(CNC(=O)COC3CCOCC3)C2)ccc(Br)c(F)c1 C(=O)(CCC(C(C)C)NC(C1C(C)(C)C1(C)C)=O)N(CCSC)C O=C1NC(=O)C(CCNCCC(=O)NC2CN(C(C3CC34CC4)=O)C2)N1 N1(C(COC(C)C)=O)CCC2CN(C(c3ccc(N)c(Cl)c3)=O)C2C1 C(=O)(C(F)C(=O)N1CCSCC1C(=O)Nn1cncn1)OCC C(=O)(C(CC)CCCCC)N1CCN(C(CC(=C)Br)=O)CC1CO CN1CCCC(C(=O)NC(C2CCC(CNn3cc(CCCO)nn3)CC2)=O)C1 N1(C(CCc2c(C)noc2Cl)=O)CCCC2(NC(c3cc(C)n(C)c3)=O)CC2C1 Cc1cc(C(=O)NCc2cc(C(=O)NCCCC(=O)NO)no2)ccc1C#N C12(C(NOCC(N3CCC(C=C)C3)=O)=O)CC(C)(CCO1)C2 N1(C(C(C(C)C)OC2COCCOC2)=O)CCC2CN(CCC(C)C)CC12 c1(OC)ccnc(C(N2CC(NC(C3CCCCS3(=O)=O)=O)CCC2C)=O)c1N CC1=C(C)CC(C)(C(=O)NCCC2CSCCN2C(=O)COC2CCCC2)CC1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCC2CCN(C(=O)Cc3ccnn3C)CC12 C1(NC(=O)CCC2CCCOC2)CN(C(c2ccco2)=O)CC1(F)F N1(C(CC(COC)C)=O)CCC(NC(c2ccc(C)cn2)=O)CC1C C1(NC(CC=CC)=O)CCC(C(=O)NCCN2CCC(O)CC2)CC1 CC(C)(F)CC(=O)N1CCC(CNC(=O)Cn2ccccc2=O)C1 C(=O)(C1CCCn2cnnc21)N1CCC2CN(C(=O)Cc3sc(O)nc3O)CC21 C1(C(N2CCC3CN(C(c4c(C#N)csc4)=O)CC32)=O)CS(=O)(=O)CC12CCC2 N1(C(C2C(NCc3ccc(C(=O)OC)cc3)CC2)=O)CC2(CC(C(=O)O)CO2)C1 c1(C(C(=O)NCCCN(C(c2c(CC)onc2)=O)CC)C)ccc(Cl)c(Cl)c1 O=C(CC(C(F)F)NC(C1CC12CCCC2)=O)NC12CCN(CC1)CC2 Cc1c(C(=O)NCC2(NC(c3ccsn3)=O)CC2)cnc2c(Cl)cccc12 CC1(C)C(C(=O)NCC2(C)CCC(=O)N2)CCN1C(=O)CC1CC=CCC1 c1(C(N2CCN(C(C3C(C)C3C)=O)CC2)=O)nnc(O)cc1O Cc1[nH]nc(C(=O)NCC2CCN(C(C3CCCCC3F)=O)CC2)c1C Nc1c(C(N2CCC(NC(C3CCc4nccn4C3)=O)C2)=O)nc(O)nc1O N1(C(c2sc(CC)c(C)c2)=O)CC2CC(C1)N(C(C1CC(C)CC(=O)N1)=O)C2 C(=O)(C(C)C(C)c1ccc(F)cc1)NCC(C)NC(C1CC1F)=O N1(C(C(=O)Nc2cccc(C)c2OCC(F)(F)F)=O)CCc2ccncc2C1C C12CN(CCS1(=O)=O)CCOCCCC2.Cc1[nH]nc(Cl)c1C(=O)NCC(F)F c1(C(=O)NCC(CC)NC(C2CC(=O)N(C)C2)=O)c(Br)c2ccccc2n1C C1(CNC(c2scc(OC)c2)=O)(CO)CCN(C(C2(C)C=CCCC2)=O)C1 c1(C(=O)NC2CN(C(C3ON=C(CC)C3)=O)CC23CC3)c[nH]c2cccc(C)c12 N1(C(c2nc(C)sc2)=O)CCC(C2(NC(C3CCS(=O)(=O)N3)=O)CC2)CC1 N1(C(c2ccc(C(C)=O)[nH]2)=O)CC(CNC(c2ccc(C)o2)=O)CC(C)(C)C1 C1(CC(=O)N(C(C#C)C)CC)(NC(=O)CCNC(N)=O)CCC1 N1(C(C(C)(C)OC)=O)CCCC(O)(CCNC(=O)C(C2CCOCC2)O)C1 CCS(=O)(=O)C=CC(=O)N1CC(CC(C)NC(c2csc3ccccc23)=O)C1 c1(SCCC)ccc2c(c1)OCO2.C1(C(N2CCC2)=O)CCCS1(=O)=O C(=O)(C(O)Cn1cncn1)NC1CC(OCC(=O)N(C)Cc2ccoc2)C1 C(CC(C(C)C)NC(=O)C(C)NC(=O)C1CC1)N(C(c1c(OC)ccs1)=O)C C1(C(N2CC(OC)(CNC(c3coc(C)n3)=O)C2)=O)CCN(C)C1=O N1(C(C2C(C)(C)CC2)=O)CCOCC2(COCCN2C(c2snc(Cl)c2Cl)=O)C1 c1(NC(CC2N(Cc3c(C)nn(C)c3)CCC2)=O)ccc(S(N)(=O)=O)cc1Cl C1(C(N(C2CC(O)C2)C)=O)CCC(O)CN1C(C12CSCC1C2)=O c1(NCCNC(C(=O)Nc2c(C)cccc2)=O)scc(C(C)(C)C)c1C#N c1(C(N(C2CCCN(C(C3CNC(=O)C3)=O)C2)C)=O)cnc(C(F)(F)F)cn1 c1(NC(C2N(C(=O)NC(C(C)N(C)C)=O)CCC2)=O)cnccc1C(C)(C)C c1(C(C(=O)NCC(CNC(c2c(CC)c[nH]c2)=O)C)C)ccc([N+](=O)[O-])cc1F Cc1nc(O)ccc1C(N1CCC(O)(C(C)CNC(=O)CN(S(C)(=O)=O)C)C1)=O Nc1cc(C(N2CCC3(NC(=O)CCc4ccoc4)CC3C2)=O)ncc1F c1(C(=O)NC2(CCNC(C(C3CCCC3)OCC)=O)CC2)ccc(O)c(C)c1C C(CCCC(=O)NCC1CN(C(=O)C(=O)NCC(F)F)C2CC12)SC N1(C(c2c(C)sc(O)n2)=O)CCCC2C(NC(=O)CC(C)CC(C)C)C(C)(C)C12 N=c1nc2c(c[nH]1)CN(C(=O)C(N1CCC3(CCCCN3C)C1)=O)CC2 C1(O)(CNC(CCN(C(C)=O)C)=O)CCCN(C(C2CC2(C)C(F)(F)F)=O)CC1 N1(C(c2n(C=C)nnc2)=O)CCC2(C=C(C(=O)N3CC(=O)NCC3C(N)=O)C2)C1 N1(C(C(C#C)(C)C)=O)CC2CCC1C1CN(C(c3cccc(N)c3F)=O)CC21 c1(C(N2C(CCOC)CN(C(C3CC(O)C3)=O)CC2)=O)nc2cnccc2s1 C1(C)(CC(N2CCCN(C(COCC=C)=O)C(CO)C2)=O)Oc2ccccc2O1 c1(OCCC(C)(c2nnnn2C2CCOC2)NCCC(N)=O)ccc(F)cc1 C12(NC(CNC(CCC)=O)=O)CCC(CNC(c3cnsc3)=O)(C1)OC2 c1(OC)c(F)ccc(F)c1C(N1C2CN(c3nccc(Br)n3)CC12)=O c1(CC(C(=O)N(CCC(C)NC(c2c(CC)cno2)=O)C)C)ccccc1C C(C(C(C)C(C)C)NC(=O)CCc1nc[nH]n1)NC(C(c1ccc(CC)s1)=O)=O Cc1[nH]nc2ncc(NC(=O)C(C)(O)CCc3ccccc3)cc12 c1(C(N2CCCC(NC(C(C)(C)c3nccs3)=O)C2)=O)ccc(N)c(N)c1 CCC(C)C(=O)C(=O)NC(C1CCOC1)CNC(C1CC=CC1)=O c1(-c2ccc(C#N)nc2)cccc2ccc(C(=O)NCC3CCC(O)CC3)nc12 C1(C(N2CC(C(N(CC(=O)OC)CCOC)=O)C2)=O)CCCC2(CC2)C1 C1(Cc2cn(C3CN(C(Cc4cnc(C)[nH]4)=O)C3)nn2)NC(=O)NC1=O C1(C(=O)NC(c2ccccc2)CC=C)CN(C(C)=O)CCO1 C1(NC(c2c(C)n(CC(F)F)nc2)=O)CCN(C(C2OC(C)CC2C)=O)CC1C CC1CCC(NC(c2cc(O)nc(Cl)c2)=O)CN1C(=O)CC1C(C)(C)C1(C)C C1(COC)(CNC(C2CSCCS2)=O)CCN(C(=O)C(C)(O)COC)C1 C(=O)(CS(=O)(=O)CC(F)(F)F)N1CC(NC(=O)Cc2csc(S)n2)C(O)C1 N1(C(C(CCC)C)=O)CC2CCC1CN2C(c1nc(-c2ccc(Cl)cc2)no1)C C1(CC)(CC)SCCN(Cc2nc(C)ccc2OC)C1C(=O)OC C#C[Si](C)(C)CCCNC(C1CC1NC(C)=O)=O N1(CC)CCOC(C(=O)N(CC)CC2CCS2(=O)=O)C1 C1(C(N2CC(CNC(c3csc(-c4ccccc4)n3)=O)C2)=O)CN2CCN1CC2 C1(C(=O)NC2(C)CC(C(=O)NC(c3cncnc3)C)C2)CN(C)CCN1C CC1CC(CC(=O)NCc2nc[nH]n2)CN1C(c1csc(C#N)c1)=O c1(OCC(N2C3(CNC(CC(C)(F)F)=O)CC(C2)C3)=O)ccc(F)cc1Br Cc1c(Br)ccc(C(=O)NCC(C2CC2)NC(C2CCCOC2C)=O)c1F c1(NC(C2CCCCN2C(c2cncc(Cl)c2)=O)=O)cccc(F)c1F N1(C(Cc2cn(C(C)C)nc2)=O)CC2CCC1C2NC(c1cncc(N)c1)=O CC(CS(=O)Cc1ccn(-c2ccccc2)n1)C1CCCC1c1ccccc1 N(C(=NCC(=O)N1CCCC1)N1CCC(n2cc(Cl)cn2)C1)Cc1n(C)ncc1 C1(NC(C(CC)OCC)=O)CC2CC(C1)N(C(=O)C(C#N)=CC(C)C)C2 N1(c2nnc(C)s2)CC2CCC1C(NC(=O)CC1CCCS1(=O)=O)C2 CCCCC(C)C(=O)N1CC2C(N(C)C(C3CC4CCC(C3)S4)=O)C2C1 c1(C(=O)NCC2C(NC(CC=CC(C)(C)C)=O)CCCC2)ncnc(O)c1Cl C1(N2CC(CCC3CCCO3)C2)CCC(C(=O)N(CCO)NC(C)(C)C)CC1 C(CCCCNC(=O)C(n1ccc(C(F)(F)F)n1)C)N(C(C(C)OCC=C)=O)C O(NC(=O)CC(C)CNC(=O)C=Cc1cnn(C)c1)C(C1CCCCC1)C c1(COC(c2c(C)cc(C)s2)=O)cc(F)nc(F)c1F c1(C(=O)NC(CCN(C(C(C(C)C)N(C)C)=O)C)C)cccc2nncn12 c1(C(=O)NCCC2CC(NC(C(C)n3cncn3)=O)C2)ccccc1C(F)(F)F C(C(C)(O)C(C)(C)C)NC(c1c(CNC(C2C(C(=O)OC)C2)=O)noc1)=O c1(C(N2C(C)CCC(NC(c3c(OC)csc3)=O)C2)=O)cc2oc(C)c(C)c2[nH]1 N1(CC(COC)O)CCC(NC(=O)C(C)(C)c2cccs2)CC(C)(C)C1.C1=CC1 N1(C(C=C(C)C2CC2)=O)CCSCC1C(=O)NC1CC12CC(O)C2 CS(=O)(=O)c1ccc(F)c(-c2nnc(N3CCC(C4CCC4)C3)n2CCC#N)c1 S(=O)(=O)(c1ccc(N(C)Cc2cnnn2C)c(F)c1)NCC(C)O c1(C(N2C(CNC(COC)=O)CC(O)C2)=O)ccc(N2CCCC2)c([N+](=O)[O-])c1 c1(OC)ccc(C(=O)N(C)CCN(C(=O)C(O)P(C)(C)=O)C(C)C)c(Cl)n1 O=C1CCC(C(=O)NC2(CNC(c3ccc(-c4cscn4)cc3)=O)CC2)CN1 C1(C(=O)NCc2occ(C)c2)CCC=CC1NC(c1ccon1)=O C1(NC(C2(SC)CCC2)=O)CCN(C(c2cc(O)ccc2Cl)=O)CC1C C12OCCC1CNC2=O.C1(CC(N2C(C(=O)OC)CC2)=O)CCOC1C C1(C(=O)NC2(C)CN(C(Cc3c(C)noc3C)=O)C2)Cc2ccccc2C(=O)O1 C(=O)(CN=c1cc[nH]cc1)NC1C(C(=O)NC(C2(C)CC2)CO)CC1 c1(NCC(CCCCC)O)ccc(S(=O)(=O)NC2(CCOC)CCCC2)cn1 C=CCC(C(=O)N1CC(NC(C)=O)(CNC(c2cc(C3CCC3)no2)=O)C1)OC c1(C(N(CCCNC(C2CCOC2)=O)CC)=O)ccc(OCC)cc1.C1(=O)CN1 CC(C)C(C)(Cc1ccccc1)C(=O)N(CCCNC(c1cn(C)c(O)n1)=O)C C(=O)(C1=Cc2ccc(Cl)cc2OC1)N1C2CC(NC(CCSCC)=O)C1CC2 c1(C(N2CC3CN(C(CSCC)=O)CC32)=O)c(F)ccc(Br)c1F c1(C(=O)NCC2C(C)CCCN2C(=O)CCC(N)=O)ccc2c(n1)CCC2 C1(C(=O)NCc2nncs2)CCC(O)CN1C(c1cc(Cl)c[nH]1)=O c1(C(N2C3C(C(N4CC(COC)OCC4)=O)C(C3)C2)=O)ccc2c(Cl)ncnc2c1 N1(C(CC)CNC(=O)C(C)C(=O)OC)CCN(C(=O)C(c2cccnc2)OC)CC1 C1(CC(=O)NCCC2CCCN(C(C3C(C#N)C3)=O)C2)CCc2ccccc2C1 c1(CC(=O)NCC2(F)CCN(C(c3nc(C(C)C)oc3)=O)C2)c(O)ncnc1O CCC(C)CCC(=O)NC1CCC12CN(C(=O)COCc1ccc(OC)nc1)C2 c1(CNC(CCOC(=O)COCC2CC2)=O)ccc2c(c1)OCCCO2 C(=O)(C(N=[N+]=[N-])C(C)C)NCC(CC=C)NC(c1cc([N+](=O)[O-])c(C)s1)=O N1(C(C(C(=O)OCC)F)=O)CCC2CCN(C(=O)C(CC)N(CC)CC)CC12 C1(C(=O)NC(CC)CC(=O)NC)(CC)CCCN(C(C2CCCN2C(C)=O)=O)C1 C1(C)(C(=O)NC2CC(CNC(c3c(SC)cccn3)=O)C2)CCN(C)CC1 c1(NC(C2(CC=C)CC2)=O)ccc(NC(C2CCCCS2(=O)=O)=O)cc1C C1(C#N)(C(N2C(COC)(CNC(C3CCN3C(C)(C)C)=O)CCC2)=O)CC2CC2C1 N1(CCCNC(C2C(C(C)C)OCC2)=O)CCN(C(c2cccnc2)=O)CC1 CC(C)(C)C(CNC(=O)CNC(=O)C=CC(F)(F)F)C(=O)NC1CCC(F)(F)C1 c1(C(N2C(CCOC)CN(C(=O)C(C)CSC)CC2)=O)cc2ccccc2nn1 N1(C(C2C(CNC(CN3CCC(C)C3)=O)OCC2)=O)CCC(CN=[N+]=[N-])CC1 c1(OCC)ccc(Cl)nc1C(=O)NCC(C)(O)CNC(C1Cc2nncn2C1)=O N1(C(C=CCOC)=O)CC(C2CCN(C(c3cccc(C(C)(C)C)c3)=O)C2)C1 C1(NC(Cn2c(C)nnn2)=O)CC2(C1)CC(C(=O)NOCC1CC=CCC1)C2 N1(C2CN(C(C3N=C(C)SC3)=O)C2)CCN(C(=O)Cn2cccn2)CC1 c1(CC(C)C)ccc(NC(C2CN(C(C3CC4CCC3C4)=O)CCN2)=O)cc1 c1(C(N(CC(C)NC(COCC(=O)NC)=O)C)=O)ccc2oc(S)nc2c1 C(=O)(CC(C)C(C)C)NCC(Cc1ccccc1)NC(c1oc(CC)c(C)c1)=O C=C(Cl)CC(C(=O)N1CCC(C(=O)N(C)C)C1)NC(=O)CCC1CCCN1C Cn1nc(C(=O)NC2CCC2NC(C2(CC3CCC3)CC2)=O)ccc1=O Cc1ccc(N(C)C(C)C)c(C(=O)NC2CC(CNC(C3CC34CC4)=O)CC2O)c1 CC1CN(C(=O)CC(C)n2cccc2)CCCN1C(=O)Cc1cnsc1 N1(CC)CCCC(C(N2CC3CC3(C(=O)NC3(C)CC(F)(F)C3)C2)=O)C1 C(=O)(C(CCC(=O)NCc1ncc(F)cc1Cl)N(C)C)OC C(c1ccncc1)=CC(=O)N(C1CCCC(NC(=O)CCC2CC(OC)C2)C1)C Cc1ccc2oc(N3CC4CC3CN4C(c3ncccc3C(C)(C)C)=O)nc2c1 C1(NC(C2C3COCC23)=O)CN(C(C2CCCOC2)=O)CC12CCC2 CC1(C(=O)NCC(CO)NC(c2cc[nH]c2C2CCCC2)=O)CCCNC1=O C1(NC(c2ccn(CC)n2)=O)CCC12CN(C(=O)Cc1ccc(COC)cc1)C2 C1(C(N2C(C(C)NC(=O)COCC(F)(F)F)CCC2)=O)CC(=O)NC1(C)C c1(C(N2CC(C(C)(C)O)(CNC(c3cnc(C)[nH]3)=O)C2)=O)c([N+](=O)[O-])cnn1C Cc1cc(C(=O)N(CC(O)CN(C)C(c2cnc(C(C)O)s2)=O)C)ccc1N Cc1ccccc1CCC(=O)NC(c1cccc(Cl)c1)CNC(=O)C(O)C(F)F N1(CC)CCN(CN2CCC(N3CCCC3)C2)C(=O)C1=O N1(C(C(C(CC)C)N(C)C)=O)CCC(C2CC2)(C(=O)NCc2ccncc2F)C1 c1(C(=O)NCC(=O)NCC2N(C(c3c(CC)ocn3)=O)CC2)cc(Cl)cnc1O c1(CNC2CC(NC(c3ncn(-c4ccccc4)n3)=O)C2)ccc(I)c(F)c1F c1(C(N(CCc2scc(C)n2)C)=O)ccc(CNC(=O)C(C)c2cc[nH]n2)cc1 C1(C(=O)NCC(CC)N(C(=O)C2=C(C)CCC2)C)CC12CCC(=O)CC2 c1(C(=O)NCC(CC(C)C)(C)NC(=O)C(O)P(C)(C)=O)cncc2cnccc12 N1(C(CCCCCOCC)=O)CCN(C(=O)CC2CCOCC2)CC(CO)C1 C1(CNC(CCN(C(CC)CC)C)=O)COC(C)(C)CN1C(C1CC2CC2C1)=O c1(CN(C2C(NC(=O)NC(C)CCO)COC2)C)ccccc1Cl CCCC(C)(C)C(=O)N1CC(O)(CCNC(=O)C(C)Oc2cccnc2)C1 c1(C(=O)NC(C2CCCN(C(=O)C(F)(F)c3cscn3)C2)C)cc(O)n(C)n1 C1(CC(=O)NCC2CC(COC)C2)C2CN(C(c3cc(Cl)cn3C)=O)CC12 N1(C(CCOC)=O)CCCC(N(CCO)C(c2sccc2CN(C)C)=O)C1 N1(C(C=CC(C)NC(c2nn(C)cc2Cl)=O)=O)CCC(C)(O)C1 Cc1cccc2[nH]c(C(=O)NC3CCCN(Cc4c[nH]c5ncccc45)C3)cc12 CC(C)(C)C(CNC(C1OCCCC1(C)C)=O)C(=O)NC1(CO)CC(F)C1 n1(CC(C)NC(c2cnn(C3CC3)c2)=O)cc(CNC(C2CC(F)(F)C2)=O)nn1 C(c1ccc(CO)cc1)=CC(=O)NCC1CN(C(C(C)N(C)C)=O)C(C)C1 C(=O)(CCC(N)=O)N(CC(=O)NCCN(C)C)C(C)C Cc1cc([N+](=O)[O-])c(C(=O)NC2CCC(F)(CNC(=O)C(C)O)C2)cc1Cl N(C1CCCc2c1cnn2C)N(C(CCN1CCCC(N(C)C)C1)=O)C C1(C(=O)NC(CCOC)C(=O)NCCc2cn(C)cn2)CC2OC1C1CC21 N1(C(C2OCCN(C(C(F)=C(C)C)=O)C2)=O)CCc2ccc(C)cc21 c1(NC(C2(C)CCCC2)=O)ccc2c(c1)CCN(C(=O)C#CC(=O)O)C2 CCC(CCC(=O)NCc1cc(C)ncn1)NC(=O)C(C)NC(=O)NC N1(C(C2N(C(C(SC)SC)=O)C3C(C2)C3)=O)CCCC(O)(C2CC2)C1 c1(C(N2CC(CC)C(NC(=O)C(C)(C)N=[N+]=[N-])CC2)=O)ccc([N+](=O)[O-])n1C C(=O)(C(CO)C(C)(C)C)N1CCC(COC)(NC(=O)CCOC2CCCC2)C1 C(c1ccc2ncccc2c1)=CC(=O)NC1CCCC1NC(=O)CC1CCOC1 c1(C(=O)NC(CC)CNC(=O)CCCc2ccsc2)cccc(S(C)(=O)=O)c1 C=C(C)CC(C(=O)N1CCC(CC2CCC2)C1)NC(=O)CC1CCC(=O)NC1 N1(C(N2CCN(C3CC3)CC2)=O)CCC(F)(C(=O)NCCO)C1 c1(C2CCCN(C(c3n(CCN)ncc3)=O)C2)cc(F)ccc1F C(C(=O)N1CCCc2nncn21)(C1CC1)NC(C(COC(C)=O)C)=O C(=O)(CC(C)n1cc(Br)cn1)NCC(CC)NC(=O)CCCc1cnn[nH]1 Cc1ccc(S(=O)(=O)C2CCN(C(c3cnc(C(F)F)o3)=O)CC2)cc1 c1(C(=O)NC2COCC2NC(C2(C3CCCO3)CCC2)=O)cc2cccnc2[nH]1 c1(CC)ccc(C=CC(=O)NC(C)CN(C)C(c2ccnn2CC)=O)o1 n1(CC)nc(C)cc1C(N1CCC1CNC(C1(n2ccnn2)CC1)=O)=O c1(C(=O)NCC(C)(CO)NC(c2ccc3c(c2)CCO3)=O)ccc2nn[nH]c2n1 CCC(CNC(=O)COC)(CC)C(=O)NC(c1cc(C)on1)C C#CCCN=C(NCc1ccc(C2CC2)cn1)NC(C)CCS(C)(=O)=O N1(c2n(CC=C)c(C3CN(C(=O)OCC)C3)nn2)CC2CS(=O)(=O)CC2(C)C1 CC1CN(S(=O)(=O)CCNC(=O)N(C)CCc2ccccc2)CC(C)O1 O=C(CS(=O)(=O)C1CC1)N1CCN(C(C2C=CCS2)=O)CC1 CC1CCN(c2nnc(C(F)F)s2)CC1NC(=O)CC1CC2(CC2)C1 c1(C(=O)NCCN(C(=O)C(C)(C)C2CC2)CC)ccc(C(C)C)cn1 C1(CNC(c2c(C)coc2C2CC2)=O)CCN(C(=O)C(O)CC(C)C)C12CC2 N1(C(C=C(C)c2ccccc2)=O)CC2CC(C)N(C(C3CC3F)=O)C2C1 Cc1ccc2c(N(C)Cc3cn(C)cn3)nc(=NC3CCCC(C)C3)[nH]c2c1 C1(NC(c2cnc(C(C)C)[nH]2)=O)CC2(NC(C3CC(C)(C)CO3)=O)COC1C2 S(=O)(=O)(c1ccccc1C#N)N1CC2CCN(C(C#CC)=O)C2CC1 c1(CC)cc(C(N2CCCC(N(C(=O)C=CSC)CCO)C2)=O)ccc1F N1(C(C(C)OC)=O)CC2CC(C1)C2NC(=O)C(CC(C)C)n1ccc(C2CC2)n1 C(=O)(CC(C)(C(F)(F)F)NCCN)NC(C1(c2cc(Cl)ccc2O)CC(C)(C)C1)=O C1(C(=O)NC(CNC(C(CC#C)O)=O)CO)CCCC2(CC2)C1 c1(C(N(CC(CNC(c2cc(COC)[nH]n2)=O)C)C)=O)c(C)ccc(F)c1O c1(C(N2CCCCC(CNC(c3ccsn3)=O)C2)=O)cc2cccnc2o1 C1(C(N(C2CCOCC2)CC)=O)CCC2(CC1)CCN(Cc1ccc(I)o1)CC2 O=C(CC1CC2(C1)CC(O)C2)NN=c1ccn(C2CCOCC2)[nH]1 C12(NC(CCC(C)OC)=O)CCC(C1)N(C(=O)CNC(C1CCCC1)=O)C2 CC1CN(C(=O)CC2CCCCC2NC(c2cnn(C)c2)=O)CCS1=O N1(Cc2ccc(OCCCCCCCN=[N+]=[N-])cc2)CCC(C2CCOC2)C1 c1(C(=O)NCC2C(NC(C(C)Cc3ccccc3Cl)=O)C2)ccn(C)c(=O)c1 C12(NC(CCCOC)=O)CCC(F)(F)CC1CN(C(=O)C(C(C)(C)C)OC)C2 N1(C(C(n2ccc(C)n2)C)=O)CCC(C(N2CCC(C#N)C2)=O)C1C(C)C N1(Cc2cn(CC(CNC(c3cncn3C)=O)OC)nn2)CCCCC1=O N1(C(C(CC(N)=O)O)=O)CCC(CNC(c2nc3cnccc3s2)=O)C(F)(F)C1 c1(C(=O)Nc2c(O)ccc(C)c2)n[nH]c2c1CN(C(=O)CC1CCN(C)CC1)C2 N1(COC)CCC(N(C2CCC2)Cc2oncc2C(=O)NC)CC1 C1(NC(C2N(C(c3c(CC)cns3)=O)CC2)=O)CCCN(O)C1=O c1(CSC)ccc(C(=O)N(C)CC2CCCC2NC(C23CC(F)(C2)C3)=O)o1 CC(C)(C)C(C#N)C(=O)N1CCSCC1C(=O)NCCCCN1CCC1 c1(C(=O)NCC(C)NC(c2cncc(F)n2)=O)cc(C2CC2)cnc1Cl O=C1CCCC(CCCC(=O)NCC2COC(CNC(=O)CNS(C)(=O)=O)C2)N1 C1(NC(CC(C)(C)C)=O)CC(F)CN(C(c2ccc(O)c(F)c2)=O)C1 C12(CNC(C(CC)CC)=O)CCC(NC(C3CC34CCCOC4)=O)(CC1)CO2 N1(C(c2cscc2Br)=O)CCC(CNC(C2(F)CC=CC2)=O)CC1 N#Cc1ccc(C2CC2SC(CCN)C(F)F)cc1 CCS(=O)(=O)CC(=O)NC1COCC1NC(C1CC2CCC2C1)=O c12oc3ccccc3c1NC2=O.C12(CCC1)NC(=O)CN(CC)C2.C1(CO)CC1 N1(C(C=CCCC(C)C)=O)CCC(C)C(N(C(=O)Cc2ccon2)C)C1 C1(C(=O)NCCOCCOCCNC(c2c(C)con2)=O)CC(C)OC(C)C1 N1(CCC(=O)NC2CC(F)(CNC(=O)C(C3CCCO3)C3CC3)C2)CCCCC1 N1(CC#CO)CCN(c2cnccn2)CC1.c1(CCC(C)=O)ccccc1OC(F)(F)F c1(C(=O)NCCOCCOCCNC(c2ccns2)=O)cnc2ncccn12 N1(C(c2ncc(C)s2)=O)CCCCC12CCCN(C(=O)C(Cl)(Cl)Cl)C2 c1(OC)ccc(Cl)cc1CC(=O)N(C(C)CN(C(=O)Cc1cccs1)C)C CC1=C(C)CC(C(=O)NCCC(O)C(N2CC3CC3C3CC23)=O)CC1 Cc1ccccc1C1CC1C(=O)NCC1CCCN1C(=O)CN(C1CCSC1)C C(=O)(CCCCCC#N)N1C(CC(N2C(CC)CN(CC)CC2)=O)C2CCCC21 CCC(CC(=O)NC1COCCN(C(C2CC2F)=O)C1)CC(F)(F)F Cc1ncc(C(=O)NCC(C)(C)CNC(C2CC(CF)C2)=O)cn1 c1(C(N2CCN(C(C(C=C)C)=O)C(C)C2)=O)ccc([N+](=O)[O-])cc1 C1(NC(=O)C=CC2CCCC2)CN(C(=O)CC2CC(F)(F)C2)C2(CCCOC2)C1 C1(NC(CN(C(C)=O)C)=O)CCCC1C(=O)NCC1(N2CCOCC2)CC1 c1(CCC(=O)NCCCC2CCN(C(=O)CC=C(Cl)Cl)CC2)ccc(F)cc1Cl C1(CC)(NC(=O)C(C)O)CN(C(=O)C(C)(F)c2ccccc2)C1 c1(C(N2CC(CNC(C(N3CCOCC3=O)C)=O)C2)=O)ccc2[nH]ccc2c1F N1(C(CNC(=O)OC)=O)CCC(NC(=O)CC(C)C(F)F)C(CO)C1 C1(CC(c2n(C)nnn2)NCc2nnnn2C(C)(C)C)CCCC(C)(C)O1 c1(CNC(COC)=O)ccc(C(=O)NCCC(C)N(C)C)s1 C(=O)(C1=NN(CC)C(=O)CC1)NC(CC)(CNC(C1CC2CCCC2C1)=O)CC c1(C(=O)NC(c2c(C)c(F)ccc2)C)cc([N+](=O)[O-])c2n[nH]cc2c1 c1(CCC)ccccc1C(=O)NC1CCN(C(c2cc(CC)oc2C)=O)C1C C(CCC(C)(C)C(=O)Nc1ccc(NC(c2n[nH]cc2Cl)=O)cc1C)OC N1(CC(=O)NC(C2CCCN(C(c3cnn(C4CC4)n3)=O)C2)C)C(=O)CNC1=O C(=O)(C1CCCc2ccnn21)NC1(CF)CCN(C(C(C)C2CCCC2)=O)C1 C1(CN(C(=O)CCc2nccs2)C)CCCN(C(c2snc(O)c2Cl)=O)C1 CCCC(C)(CC)C(=O)N1CC(CC(C)NC(=O)C(C(C)CC)OC)C1 C=C(Cl)C(C)(C)C(=O)NC(CNC(=O)Cc1csc(C(C)OCC)n1)CC c1(OC)ccc(CC(C)C(=O)NC2CCCN(C(c3nc(Cl)sc3C)=O)C2)cc1 c1(C(N2CC3CCC(CNC(c4c(C)c[nH]c4)=O)(C2)C3)=O)cnc([N+](=O)[O-])cc1C C1(NC(c2cnc(N)c(Br)n2)=O)CC2(C1)CC(O)(C(F)(F)F)C2 CC(C)CC(CNC(c1cc(=N)[nH][nH]1)=O)C(=O)N1CCCC1(C)C(C)(C)C C(c1cc(Cl)c2c(c1)OCCO2)=CC(=O)NCCCOCCN=[N+]=[N-] c1(C(C(N2CCCC(N(CC(=O)OC)C)C2)=O)CN)ccc(OC)c(OC)c1 c1(OC)ccc(C2CCN(C(=O)NCC3CCOC(SC)C3)CC2)cc1 N1(c2nnc(CCC)s2)CCC2(CNC(=O)CCC3(O)CCC3)CCCCC12 N1(C(C(C)SCC)=O)CCN(C(=O)C(c2cccnc2)OC)CC1 Cc1cc(C(=O)N(c2cccc(Cl)c2)CCCO)c([N+](=O)[O-])c(O)n1 N1(C(C2N=C(C)SC2)=O)CC(F)(F)CC1(C)CNC(c1cn(CCO)nn1)=O C(=O)(CCC(C)(C)O)N(C1CN(C(=O)C2=COCCO2)C1)C N1(C(c2c(CC)oc(C)c2)=O)CC(NC(c2cnc(C(C)OC)s2)=O)CC(O)C1 C1(CC(=O)NCC(CNC(C2(CC)CCCCC2)=O)O)COCC(C)(C)O1 CCCCC(CC)C(=O)N(CC(O)CNC(c1cc(-c2csc(=N)[nH]2)c[nH]1)=O)C C1(NC(c2ncn(C)n2)=O)CCSC12CN(C(=O)CC1CCC(C)(C)C1)C2 C(=O)(C(F)(F)CN1CCCC1)NCC#CCNC(c1nc(C(=O)OC)sc1)=O CC(c1ccccc1C)=CC(N1CC(CO)(NC(c2cccnn2)=O)C1)=O N1(CC(C)NC(=O)C(O)Cc2ccccn2)CCN(C(C2(O)CCC2)=O)CC1 Cc1cncc(NC(c2nnnn2CC2CC2)CC2CCCCO2)c1 C1(NC(c2n(C(C)C)ncc2)=O)CCC(N(C(=O)CC2CCN(C)C2)C)CC1 c1(C(C(=O)NCCN(c2c(C(C)C)noc2)C)C2CC2)ccccc1F.CCN N1(C(C2(OCC)CCOC2)=O)CC(CC(=O)Nc2cncc(C#N)c2)C2(CC2)C1 C=CCCC(C(=O)N(C)CCSC)NC(c1cocn1)=O C1(C(=O)Nc2c(O)cccc2Cl)COC2(CCN(C(c3ccnnc3)=O)CC2)C1 CC1CN(C(=O)NC2(CNC3CC(O)C3)CCC2)CCC1(O)C(F)(F)F C1(NC(C(=C(C)C2CC2)F)=O)CCC2(CC1)CN(C(c1n[nH]c3c1CCC3)=O)C2 c1(C(c2nnnn2CC2CCCO2)NCc2cn(CCC)nc2)cn(C)nc1C C(C(=O)NCC1CCCC1C(N1CCC2CCC12)=O)(C(C)C)OC c1(OC)nccc(C(=O)NC2CN(C(=O)C(C)OCC3CCCO3)C2)c1F N1(C(CCCCC#C)=O)CC2OCC(NC(C3C(C(F)F)C3(C)C)=O)C2C1 N1(C(C(CCCC)=O)=O)CCC(C)(C)C(C(=O)NCCC(O)C(F)(F)F)C1 CCC(C)(CNC(c1ccc(O)cc1)=O)C(=O)NCC(C)CC(C)C C1(CC)(CC)CC(C(=O)NC(c2cn(CC(C)O)nn2)C)C1 c1(C(N(C2CCC(NC(COCCC#C)=O)C2)C)=O)ccc(P(C)(C)=O)cn1 n1(CC(=O)NCCNC(=O)C=Cc2ccc(F)nc2)ccc2cc(F)ccc12 Cc1nc(C2CC2)sc1C(N1CC=CC(NC(=O)Cn2ccnn2)C1)=O c1(C(=O)NCC2(CCNC(CN(CCOC)C)=O)CC2)nccc2c1NCCC2 C1(NC(CC2OCC(C)(C)C2)=O)CC2CC(C1)N(c1nnco1)C2 N1(C(CC(=C)C)=O)CCC2(NC(c3cnn4ccsc34)=O)CC2C1 Cc1nc2cc(Cl)cc(C(=O)NC3CN(C(=O)CC4CCC4)CC3C(F)F)c2[nH]1 c1(C(CN(C=O)CCOC)O)cc(O)ccc1C.C12CN(C1)C(=O)N2 Cc1ccn2ncc(C(=O)NC34CCCN(C(c5n[nH]cc5Br)=O)CC3C4)c2c1 C1(C(N(c2ccccc2)C)=O)CCCN(Cc2cccc(I)c2)CC1 c1(C(=O)NCCN(C(c2cn(CC=C)nn2)=O)C)c(OC)ncnc1C C(=O)(C1=NOCC1)NCC(CNC(c1c(CC)nc[nH]1)=O)O Cc1ccc(Cn2ccnn2)cc1.N12CC(C1)NC(=O)C1(CC1)CC1CC1C2=O C1(CC(=O)NCCOCCC(=O)NC(C)Cc2nc[nH]n2)CC=CCC1 C(C(=O)NNC(=O)c1cc(C)oc1C)C1(c2nc(C)cs2)CC(OC)C1 Cc1cc[nH]c(=N)c1C(=O)NC1CC(NC(=O)C(C)Oc2ccc(F)cc2Cl)C1 CCC(C)(O)C(=O)NCC12CC1CN(C(c1ccc(OCOC)cc1)=O)C2 c1(CNC(C2(C#C)CN(C(=O)CCc3cnoc3)C2)=O)cnc(F)c(C)c1 N1(C(C=CC)=O)CCCC2(CNC(c3cc(OC)n(C)n3)=O)CCCC12 Cc1c(Br)cnn1CC(=O)N(C(C)CCNC(c1ccc(N)cn1)=O)C c1(C(C)NC(Cn2cc(-c3scc(C)n3)nn2)=O)ccc(Cl)cc1F c1(CC)[nH]nc(C(=O)NCC(C(C)C)NC(=O)C(C(C)C)SC)c1[N+](=O)[O-] n1(CC)nc(C(N2CCC(NC(c3ncccc3OC)=O)CC2)=O)cc1C1CC1 c1(C(=O)NC2CCC(NC(C3CN(C)C3)=O)CC2)cc(S(N)(=O)=O)co1 C(=O)(C(C)CS(C)(=O)=O)N1C2C(NC(c3c(C)n(CCN(C)C)nc3)=O)CC(C2)C1 c1(C(N2CCC(C(CNC(C(CC)F)=O)C)CC2)=O)nnc2ccccc2c1O Cc1coc(C=CC(=O)NCCN(CC(C)O)C(c2ccc(Cl)o2)=O)n1 N1(C(C2COC3(CO)CC2C3)=O)CCCC(O)(CNC(=O)C(F)(F)C(F)F)CC1 N1(C(C2(COC)CC2)=O)CCCCC(NC(=O)CC(C(F)F)c2ccccc2)C1 CCCS(=O)(=O)CC(=O)OCC(=O)Nc1ccc(Br)cc1F C1(N(CC(C)OC(F)F)C(=O)CC2CCC(C)C2)CC2C=CC1C2 c1(NC(C2(OC)CCN(C(C34CSCC3C4)=O)C2)=O)cc(C)ccc1C C1(C)(CNC(CCC=CCC=C)=O)CCC(NC(C2COCCO2)=O)CC1 C1(NC(C2CC(C(F)(F)F)(OC)C2)=O)CCN(C(C2CC(F)(F)C2)=O)CC1F N1(C(C(=O)NCCCOC)C)CC2CC1CCC2NC(=O)CCC1CCC1 C1(C(C)C)(CO)CCCN(c2cc(Cl)nnc2O)C1 C1(C(=O)NC(CC)CN(C(=O)C=CCN2CCCC2)C)CCC2(CCC2)OC1 C(=O)(C(CC(N)=O)NC(=O)Cc1cc[nH]n1)N(C1CC(=C)C1)C N1(C(C(C)C2CCC2)=O)CCC(NC(C2(S(C)(=O)=O)CC2)=O)C(CO)CC1 CC(C(=O)N1CCCC1CCC(F)(F)F)C(C)(C)C Cc1ncc(Br)cc1NC(C1CC1C(=O)Nc1cnc(C#N)nc1)=O N1(C(C=CC(C)C)=O)C2CCC1CC(NC(=O)C(c1ccc(F)c(F)c1)O)C2 C(C(C(=O)N1CC(O)(C(N)=O)C1)C(C)C)NC(CC(CC)OC)=O c1(C(=O)NC(C(C)NC(C2CCC(N(C)C)C2)=O)C)ccnc2[nH]cnc12 c1(C(=O)NCC2(NC(C3N(C)CCN(C)C3)=O)CCOC2)cc2c(ccn2C)[nH]1 C1(O)(CNC(c2cnns2)=O)CCCN(C(=O)CCCn2ccnc2)C1 N1(C(c2c(C)cc(C)s2)C(=O)NCc2c(C)cccc2C)CCC(O)CC1(C)C C1(CNC(C(C)n2cccn2)=O)CN(C(=O)CC(C)(C)CN(C)C)CC1(C)C CC1=C(C(=O)NCCCN(CCO)C(c2coc(C(F)(F)F)n2)=O)SCCO1 CC(C)(C)S(=O)(=O)CC(=O)NCC1CCC(NC(=O)C=Cc2ccccc2)CC1 c1(C(=O)NCC(C2CCOC2)NC(Cc2nc(C)oc2)=O)oc(C)nc1C(F)F N1(C(C2N(CC)CCC2)=O)CCC2CN(C(c3ccc(N(C)C)cn3)=O)CC2C1 C1(NC(=O)COCC2CCC2)CCN(C(c2ncncc2Cl)=O)CCC1CO CC1OCCC1CC(=O)N(CCNC(=O)C(C)(C)n1ccc(C2CC2)n1)C1CC1 c1(N2CC3(C(=O)OCC)C(C2)CCCOC3)nc2ccc(N)cc2s1 c1(C(=O)NC2C=CC(C(=O)NCC3CC3[N+](=O)[O-])C2)cnc(Cl)s1 N1(C(C(CC=CC)CC)=O)CC2CC(NC(c3n[nH]c(CC)c3Cl)=O)C(C2)C1 c1(OC(C)C)cc(N2C(C(=O)NC3CCCC(O)C3)CC3CC23)ncn1 c1(CCCC(N2C(CN(C(c3ccc(=N)[nH]c3)=O)CC)CCC2)=O)ncc(Cl)cn1 CCC(C)CC(C(=O)N1CC2C(C(=O)OC)C2C1)NC(c1cc(C)[nH]n1)=O c1(C(=O)NC(CN(C)C(c2cc(C3CC3)[nH]n2)=O)(C)C)ccc(N)c(F)n1 c1(OC)cc(OC)c(-c2nc(-c3ccnn3C)nn2C(C2(C)CC2)C)c(OC)c1 c1(CC)ncc(C(=O)NC2CCN(C(c3csc(C)c3N)=O)C2C)c(C)n1 C1(C(=O)NCC(C)(C)NC(C2CC(C)OC(C)C2)=O)Cc2cc(F)ccc2O1 Cc1cccn2cc(C(N3CC4CCCC(C3)N4C(=O)C3=CCCC3C)=O)cc12 Cc1cc(C(=O)NCC2CCC(NC(C3Cc4nccn4C3)=O)C2)cc(N)c1O c1(C(=O)NC2C(C)(C)CN(C(=O)CN3CC(=O)NC3=O)C2)cnc2sccc2c1 C1(C(=O)NCC(CNC(Cc2c(C)nc[nH]2)=O)O)C(C)OC(C)C1C c1(C(=O)NCC(CCOC)NC(c2nc(C)c(C)s2)=O)ncc(C(N)=O)cc1Cl CCCC(C)(C)CN=c1[nH]c(=NC2CCCCC2N2CCCC2)[nH]c2c1SCC2 O=C1CC(CC(=O)N(C2CCCN(C(C3(F)CCCCC3)=O)C2)CCF)CCCN1 c1(C(N(CCCCN(C(C(C)Cn2ccnc2)=O)C)C)=O)cn(C)nc1C(F)F c1(NC(C(CN(C)N(C)C(=O)OC(C)(C)C)=O)=O)nc(CSC2CC2)cs1 N#Cc1cnn2cc(C(=O)NC3CN(C(C4CC4F)=O)C3)cnc12 C1(=CC(=O)NCCC2CN(C(C3CCC=CCCC3)=O)C2)CCCCCC1(F)F c1(NCC(C2CCC2)OC)nccc(=NCC2CCC=CCC2)[nH]1 CC(CSC(F)(F)F)C(=O)NCC1CCCC1NC(=O)C(=O)N(C)C c1(C(=O)NC(C(C)NC(CCCCC#C)=O)CO)cc(F)cc2nn[nH]c12 c1(C(=O)NC2C(NC(C=CC(CC)C)=O)C2)ccc2ccoc2c1 c1(C(=O)NC(CCNC(C2(C(=O)NC)CCC2)=O)C)cc(-c2ccco2)on1 N(C(=NCc1ccc(Cl)nc1)NCC(=O)N(C)OC)C(CC)C.C(CC)SC C1(CNC(CC(C)O)=O)CCCCC1C(=O)NCCNC(C1CCC1)=O n1(CC)cc(C(N2CC(C)(NC(=O)C(O)CC3CC3)C2)=O)c(C(F)(F)F)n1 N1(C(C2CCN(C(CC(CC)O)=O)CC2O)=O)CCN(CC)C(C)(C)C1 C=C(C)CC(C(=O)N1CC(CC(C)NC(=O)C2=CCCSC2)C1)OC N1(C(=O)Cc2csnn2)CCC2C(CCN2C(c2c(F)ccc(F)c2O)=O)C1 C(CCC(=O)NCC1CC1CNC(C1CN(C2CCC2)C1)=O)OC C1(NC(C(C2CCN(C(c3csnn3)=O)CC2)C)=O)CC2CC1CC21CC1 c1(CC(=O)N(CCOCCN(C(=O)Cn2nnc(=N)[nH]2)C)C)ccsc1Br c1(C(=O)NCC23OCC(CNC(c4cnc[nH]4)=O)(C2)C3)c(C2CC2)nc2sccn12 C(=O)(C(C)(C)C(C)(C)O)NCC1C(NC(c2cn(CC)nc2C)=O)CC1 CC(C)C(C(C)NC(c1ncncc1Cl)=O)NC(=O)C=CC(C)(C)C N1(C(C2CC(=O)OC2)=O)CCCC2(CNC(c3cnoc3)=O)CCCC12 CC1(C)CC(CC(=O)NC2(C)CCN(C(c3cn(CC(F)(F)F)nn3)=O)C2)CO1 Cc1cncc(C(=O)NC(CC2CCC2)C(=O)NCCCNC(=O)C(C)C)c1 N1(C(CCC=CC)=O)CC(CC(=O)N(C)Cc2ncn(C)n2)CC1(C)C CCC(CC)C(C)C(=O)N(C)CC1COCCN1C(c1ccc(S(C)(=O)=O)o1)=O C(=O)(CCCCCF)NCc1scc(C(N2C(CC(=O)NC)CC2)=O)c1 CC1(C)COC(CCC(=O)NCCN(C(=O)C(F)=CC2CC2)C2CCCC2)C1 c1(-c2cc(OC)c(Br)cc2)n[nH]c2c1CN(C(=O)C(C)N(C)C)CC2 N(C(=NCCC=C(C)C)NCC(C)C)CC.C1(COCC)(OC)CCCOC1 C(=O)(CCCCCn1cc(C2CCN(C)C2)nn1)N(CC(=O)OC)C(C)C c1(NC(C(=O)NC(c2nnc3n2CCCC3)C)=O)ccc(C)c(S(=O)(=O)N(C)C)c1 C(=O)(CCS(C)(=O)=O)NCCCCC(C)NC(c1nc(C)n(C)n1)=O N1(C(CCOCCOC)=O)CC2CC1C2CNC(=O)C(C)C(F)F n1(CC)nc(C(=O)NC(C)CCNC(=O)C(O)C(C)(C)C)c(Cl)c1Br CC1(C)CCCC(NC(N2CCOCC2c2ncno2)=O)C1 C1(CNC(C(C)SC)=O)CN(C(=O)COCC(C)(C)C)CC(C)(C)O1 N1(C(C2N(C(C3CCCO3)=O)CCC(CC)C2)=O)CCc2nc(C)[nH]c2C1 C1(Nc2ncc(C(C)=O)cn2)CC2CCC(C1)N2C(=O)C(C1CC(C)(C)C1)OC C12(NC(CCCC#C)=O)CCOCC1CN(C(c1noc3ccc(Cl)cc13)=O)C2 CCC(C)CC(=O)NC1CC(NC(=O)CN2CSCCSC2)C1 N1(C(C=C(CC)C)=O)CCC(COC)(NC(=O)C(C)C)C1 Cc1cc(C)n(CC(=O)NC2CC(C)(CNC(C3(F)CCCC3)=O)C2)n1 C1(C(C)NC(CNC(C2C(OCC)CC2)=O)=O)CCN(C(=O)Cc2cc[nH]c2)C1 C1(NC(c2n(CC)nnc2C)=O)CN(C(=O)Cn2nnc(C3CC3)n2)CCC1CO C1(C(=O)NCC2(F)CCN(C(c3c(C)nn(C)c3Cl)=O)C2)CCc2cncn2C1 C12N(CCC1(C)C)C2=O.c1(C(=O)NC(CNC(=O)OC)C)cccc(C)c1 N1(C(C=CC)=O)CCC2CCC(NC(c3ccc(F)cc3[N+](=O)[O-])=O)C1C2 n1(CC(N2CC(NC(C(C(C)OC)O)=O)(CO)C2)=O)cc([N+](=O)[O-])ccc1=O C=CC(CC)CC(=O)NC(c1ccccc1)CNC(=O)CC1(OC)CCCC1 c1(C(=O)NCC2N(C(C(CCSC)NC=O)=O)CC=C2)ccnc2c1CCO2 N1(C(CCC(C)OC)=O)CCC(C2(NC(=O)CCC3CCCOC3)CC2)CC1 O=C(N1CC2COCC2O1)C1CCN(c2ccc(Br)cc2)CC1 c1(CC)nncn1CCNC(=O)CCOCCN(C(=O)C(c1ccn(C)n1)C)C C1(NC(c2ccc(COC)[nH]2)=O)CCC(NC(C2(S(N)(=O)=O)CC2)=O)CC1 c1(C(=O)NC2CN(Cc3cn(C(CC)C)nn3)C2)cccc(C)c1 C1(C(=O)NCCOC(C)=O)CCCCN(C(C2CCC(C)(C)OC2)=O)C1 C1(C(=O)NCCOC2CN(C(C3(CC#C)CCCO3)=O)C2)CCN(C)C1=O C(=O)(NNc1cc(C#N)cc(Cl)n1)NC1C(C)CCN(C)C1=O CON1CC(C(=O)NC(C)(CNC(c2cn(C)nn2)=O)C2CC2)CC1=O c1(C(=O)NCCCCN(C(C(C)CC2CC2)=O)C)ccc(S(C)=O)cc1 C(C)(N=c1[nH]c2c(c(=NCC3(C)CCOC3)[nH]1)CCCCC2)c1scc(CC)n1 C1(C(=O)Nc2ccc(CC)nc2)C(C2CC2)CCN1C(=O)Cc1ncoc1C c1(CC(=O)NCCN2CCN(C(c3c(C)ccs3)=O)CC2)ccccc1S(C)=O Cn1ccc2c(C(=O)NC3CC4CCC3N4C(=O)CN3CSCC3=O)cccc12 c1(CNC(CN(C)C2CC2)=O)cccnc1CNC(c1ccc(NC=O)cc1)=O C1(C(=O)NC2CC(CNC(=O)CCS(C)=O)C2)(OC)CCSCC1 c1(CNC(c2cc(C)nn2C)c2n(CCOC)nnn2)cnc2ncccn12 C(=O)(C1=NNC(=O)CC1)NCC(c1cccs1)N(C(=O)C(c1ccccc1)O)C C1(C(N2CC3(CN(C(C=CCC)=O)C3)C2)=O)CCc2ccc(F)cc2O1 c1(C(N2CC(O)(C(C)NC(=O)COCCN(C)C)C2)=O)sc2cccnc2c1Cl CC1CCN(C(=O)COc2ccc(Br)cc2)CC1NC(C1CCCN1C)=O n1(CC(=O)N(CC(CC)NC(=O)CCCn2ccnc2)C)nc(C)n(C)c1=O c1(CNC(CC2(C)CC2F)=O)ncoc1C1CN(C(=O)CNC=O)C1 C(C(=O)N1CCC(F)(c2cn(CCN(C)CCO)nn2)C1)(C(C)C)NC(C)=O Cc1cccc(C)c1S(=O)(=O)CCN1CCCCCC1c1ccco1 C1(CC)CN(C(=O)COC(F)(F)F)CCN1C(=O)Cc1nccn1C n1(CC)nccc1C=CC(=O)NCCC(C)CCNC(c1cnc(C(C)=O)s1)=O CC1CN(C(C2CCCCS2)=O)CCN1C(=O)COC1CCCOC1 C1(O)(C(=O)NCCN(C(=O)CSc2nccn2C)C)CCOC1 N1(C(C(CC)(C)CC)=O)CC2CCC1C(NC(c1ccc(C)c(N)c1)=O)C2 CC1CC(C)(C(=O)NCC(=O)NCC(=O)NCC2CC23CCC3)C1 Cc1ncc2c(n1)CCCC2NC(c1sccc1Br)c1nnnn1C N1(C(c2cncc(C)n2)=O)CC2(CCCC2)C1C(N1CCC2(CC(F)C2)C1)=O c1(NC(c2cccc(N(C)C)c2)=O)coc2ccccc12.N12CC(CC(F)C1)C2 c1(C(N(CC(CNC(c2nc(CC)oc2)=O)C)C)=O)cc(Cl)c(F)c(Cl)c1 N1(C(C)=O)CC2CCCC(C1)N2C(C1CN(C=O)CCS1)=O.C(C)(C)(C)O c1(C(N2CC(F)(CNC(c3cc(F)ccc3Cl)=O)C2)=O)cc(F)cc2nn[nH]c12 N1(C(C2C(=C)C2)=O)CCC2(CCCN2C(c2cccc(SCCC)c2)=O)C1 n1(CF)cnc2c(NCCN3CC4CCC3C4)nc(N3CC4C(C3)C4(F)F)nc12 C1(C)(C(=O)NC(C)CN(C)C(c2cc(C(F)F)[nH]n2)=O)CCNC1=O C1(OC)CC(CNC(c2cc(Cl)no2)=O)N(C(=O)CCC2CC2(F)F)C1 N1(c2nnc(C(CC)(C)C)o2)CC2CCCC1C2CNC(c1nc(Cl)sc1Cl)=O C1(C2N(C(C(C)C3CCCC3)=O)CCC2)CCN(C(c2c[nH]nc2F)=O)CC1 Cc1cc(N)cnc1C(=O)NCC(C)(C(C)C)NC(=O)CC1OCCC1(C)C C(CCCC(=O)NCc1ncoc1C1CC1)N(C)C(C1(c2ccncc2)CC1)=O c1(C(N2CCCC(NC(C(C)(C)CC3CC3)=O)C2)=O)cn2cc(Cl)cnc2n1 CC1CN(C(=O)CCC2CCCCN2C(=O)C=CC(F)F)CC1O c1(C(N2CCC(COC)C2)=O)cc(N2CCCC2)nc(Cl)c1 c1(N2CC(C)(C)C2)nccc(N2CCOC(C3CCCOC3)C2)n1.C1CC(O)C1 c1(NC(C2CCN(C(COCCOCC#C)=O)CC2O)=O)ccc2ccoc2c1 C1(COC)CN(C(c2cc(C)on2)=O)CCN1C(c1cc(C)ccc1I)=O N1(Cc2cc(N3CCCN(C(C)(C)C)CC3)ncn2)CCCC(S(C)(=O)=O)C1 c1(NC(C(=O)NC2CC(NC(C(COCC)C)=O)C2)C)ccc(C(F)(F)F)cn1 N1(C(C(C)Oc2ccccc2)=O)CCN(C(c2ccc(F)c(CO)c2)=O)C2CC12 N1(C(c2ccn(C)c2)=O)CCCC(CCNC(c2c[nH]c(=O)cn2)=O)CC1 CCCCC(C)(F)C(=O)N(CCCNC(=O)CC(=O)Nc1cccc(C)c1)CC N1(C(C2C(C)(C)C2(C)C)=O)C(CNC(C23CCC(CC2)OC3)=O)CC2CCCC12 C1(CNC(Cc2nnc(C)o2)=O)CN(C(c2sc(Cl)cc2Cl)=O)CCC1C Fc1cc(-c2ccc3c(c2)CN(c2ncc(Br)cn2)C3)c2ncccc2c1 c1(C(=O)NCC2CCCCN(C(=O)C(F)CC3CCC3)C2)cccc([N+](=O)[O-])c1 Cc1cc(C(N2CC=CC2C(=O)NCCCc2ncn(C)n2)=O)cs1 c1(CC(=O)NC2CN(C(c3cc(C)n(C)c3C)=O)CC2O)cccc([N+](=O)[O-])c1 C(CN(C(=O)CC1CSCCS1)CC)(C(C)(C)C)NC(CSCC#C)=O C(=O)(CC(CC(=O)O)C(C)(C)C)N(CCO)C(c1nc(C)cc(C)n1)C(C)(C)C C=CCCCC(C)N=c1[nH]c(N(C)Cc2cccc(C(F)(F)F)c2)nc2ccsc12 C(C(COC)CC(=O)NCCC1CCN(C(=O)Cc2ccsc2C)CC1)OC C(=O)(C(CC)C(F)(F)F)N(C(C(CCC(N)=O)n1cc(CCCC)nn1)=O)CC c1(C(=O)NCCN(C(c2c(C)c(C3CC3)on2)=O)C(C)C)cccc2c1COC2 CC1CC(=O)CCC1C(=O)NC1CC2(C1)CC(C(N1CCCC1CN(C)C)=O)C2 C1(C(=O)OC)CCCCCN1C(C(=O)NC(C)(C)C)C1CC(CC(C)(C)C)C1 C1(C2(O)CN(C(C3CC(F)(CO)C3)=O)C2)(CNC(=O)Cc2ccc(Cl)cn2)CC1 C(=O)(C(C)C(C)C)NC(CN(C(CCNS(CC)(=O)=O)=O)C)(C)C c1(C(=O)NCCNC(C)=O)ccc(-c2ccc(F)c3[nH]ncc23)c2cc[nH]c12 N1(C(C)=O)CCC2(CC1)OC1(C)CC2(NC(=O)CCCc2ccc(C)c(C)c2)C1 C1(C(N2CCCC(CN(C(c3c(COC)nn[nH]3)=O)C)C2)=O)CC2C(C1)C2(C)C N1(C(c2c[nH]c(=NC)s2)=O)CCC(O)(CNC(c2ccnnc2S)=O)CC1 c1(CC)ccc([N+](=O)[O-])cc1C(N1CCCC(C(C)NC(=O)C2=CCC2)C1)=O c1(CCNC(C2C(=C)C2)=O)ccc(CNC(c2sccc2OC)=O)cc1 N1(C(CCC2CCC(C)O2)=O)CCCC(C2CCCCN2C(c2coc(Cl)c2)=O)C1 N1(C(=O)CC2OCCCO2)CCC2C(C(N3CCOC(C4CC4)C3)=O)C2C1 C1(C(N2CC(F)(CNC(Cn3c(C)cnc3)=O)C2)=O)CCn2ccnc2C1 N1(C(C2=C(C)OCC2)=O)CCC(NC(=O)C=CC2(C)CCOCC2)C2(CCC2)C1 C12(CNC(C(C(C)C)NC(C)=O)=O)CCC(CC1)CN2C(=O)CC1CCCC1 C1(NC(c2nccc(SC)n2)=O)C(C)CCN(C(C2CCC(=O)N(C)C2)=O)C1C c1(CC)nc(C)cc(=NC(C)C2CN(C(=O)CSCc3csc(C)n3)CCO2)[nH]1 C1(NC(c2c(C)nc(CC)o2)=O)CN(C(c2[nH]ncc2C#N)=O)CC12CCC2 c1(C(N(CCOCCOC)C)=O)n[nH]c2ccc(C(F)(F)F)cc12 c1(NC(C2C(NC(c3ccc(F)nc3)=O)C2)=O)ccnc(Cl)c1 c1(C(c2nnnn2C2CCOC2)NC(CCCSC)(C)C)cccc2c[nH]nc12 CCC(CCO)N=c1nc2c(ncn2CC)c(NC(CC)CCO)[nH]1 c1(C(=O)NCC2C(NC(COCCCOC)=O)C2)[nH]c(=N)ccc1C c1(C(=O)NCC2N(C(CC(CC)C)=O)CC(O)C2O)cnc2c(ccn2C)c1 O=C(C1=CS(=O)CCC1)NC1(CF)CCN(C(c2cccn3cnnc23)=O)C1 c1(C(=O)NC(CNC(C(C(C)C)OC)=O)CC(C)C)cc2c(F)cc(F)cc2[nH]1 Cc1oc(CO)cc1C(N1CCCCC1C(=O)N(CC(C)CO)C)=O N1(C(c2ccc(C#C)cc2)=O)C2CCC1CC(N(C(=O)C(F)n1cccn1)C)C2 C(CC(O)C(=O)NCc1ncccc1CNC(=O)CCn1cccn1)SC N1(C(CNC(C)=O)=O)CCC(CNC(c2c(C)noc2-c2ccccc2)=O)C12CC2 C1(O)(CNC(c2cn(CC=C)nn2)=O)CCCN(C(C2CCC3(CC2)CC3)=O)C1 C(=O)(CCC1=CCc2ccccc21)NC1CC(NC(C(CCC)C#N)=O)C1 N1(C(Cc2cnc(C)s2)=O)CCN(C(=O)CSCC(N)=O)CC1c1cccnc1 C(=O)(C(C)C(F)(F)F)NC1C=CC(CC(=O)NC2(c3nc(C)on3)CC2)C1 C1(CCNC(C(=O)NCC)=O)CCN(C(C2CC2C(C)(C)C)=O)CCC1(F)F C(=O)(CCN(OC)C(=O)C(C)C1CCOC1)N(C(c1nn[nH]n1)C)C1CC1 c1(C(C)C)cnc(O)c(C(=O)NCCCN(C(=O)C(C)(C)COCC(F)F)C)c1 N1(C(C(CC)SC)=O)CC2=C(C1)CN(C(C1CCCCN1N=O)=O)C2 N1(C(C=CCOC)=O)CC(CNC(c2cccc(C)c2C)=O)CCC1C N1(C(C(F)OC)=O)CC(n2cc(C3CC3c3cccc(N)c3)nn2)C(C)C1 C1(C(=O)NCc2cnc[nH]2)COCCC12CCN(C(C1CCCS1)=O)CC2 N1(C(CNC(=O)OCC=C)=O)CCCC(C)C1CNC(c1ccn2ccsc12)=O Cc1ccc(C(=O)NC(CNC(=O)CC2(C)CCCC2)C(C)C(C)C)c(=O)n1C Cc1ccc(Cl)c(NC(=O)C(=O)NC2CC3C2CCN3C(=O)C2=CCOCC2)c1 C1(CC)CN(C(c2cncc(CO)c2)=O)CC1C(=O)N(C)Cc1nc[nH]n1 C1(C(=O)NC2C(CN(C)C(C3(n4cccn4)CCC3)=O)C2)CCS(=O)(=O)C1(C)C Cc1cc(=NCC2(CNC(C3CCC4CCCCN34)=O)CC2)[nH]c(C(C)C)n1 N1(C(C=CC)=O)CCN(C2CCN(C(c3cncc(N)c3)=O)C2)CC1 Cc1nc(N2CCCC(CNC(=O)C(C)(C)CN(C)C)CC2)[nH]c(=N)n1 C(=O)(CCC(N)=O)N(C1CCN(C(=O)C=Cc2ncc[nH]2)CC1)CC#C c1(C(N2CCC(C3N(C(CC4C(=O)OCC4)=O)CCC3)C2)=O)c[nH]c(=O)cn1 N1(C(CCOC)=O)CCN(C(=O)CC2CCC(OC)CC2)CC1c1nccn1C c1(C(N2CCC(=CCNC(C3(COC)CCCO3)=O)CC2)=O)cc(=O)n(C)cn1 C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCC(NC(CC(CCCC)O)=O)CC1 N1(C(C)C)CC(C(=O)NCCC(C)N(C(=O)Cc2cccn2C)C)CC1=O C1(C(N(CC)CC2CCN(C(=O)C(C)CO)CC2)=O)CC2CC1CC2O C1(NC(C=C(CNC(COCC(=C)C)=O)C)=O)CC=C(C)CC1 c1(CC)cc(C(N2CC3CC3(CNC(c3ncccc3C(F)F)=O)C2)=O)ccn1 CC1OCCC1(C)C(=O)NCC1(CNC(=O)Cc2ccccc2)CCC1 CC1CC(NC(C2CC2(C)C)=O)CCN1C(c1csc(-c2cn[nH]c2)n1)=O N1(C(c2nnn(COCC)c2N)=O)CCCN(C(C2CC2(C)CC)=O)CCC1 N1(C(CCNC(=O)OC)=O)CCC(CNC(C2CCS(=O)CC2)=O)C1(C)C c1(C(=O)NCC2CCN(C(C=CCC)=O)CC2C)cc(Cl)cc(Cl)c1OC C1(C(=O)NC(CCNC(c2nc(C)nn2C)=O)C)CC(c2cnn(C)c2)=NO1 CCC(CC(=O)NCC(O)CCNC(=O)Cc1nncn1C(C)C)C1CC1 Cc1cc(=NC(=O)COCCNC(=O)Cn2cc(C#N)cn2)[nH]n1C C(C(=O)NC1CCC(NC(c2occc2-c2cnn(C)c2)=O)C1)(C(C)C)SC C(=O)(C1=C(Cl)CCC1)N1CC(F)(C(NOCC(C(C)(C)C)O)=O)C1 N1(C(C=CC)=O)CCN(C(=O)CC(F)(F)F)CC1CS(C)(=O)=O c1(C(C)=O)cc2n(n1)CCN(C(C1CCc3cc(Br)ccc3O1)=O)C2 N1(C(CCC#C)=O)CC(C)OC2(CCN(C(c3cc(O)cc(Cl)c3)=O)CC2)C1 C(CCCC(=O)NCCc1ocnc1CNC(=O)C(C1CC1)C1CC1)OC N1(C(C)=O)CCCC(C2CCCCN2C(c2cn(-c3cccnc3)nn2)=O)C1 C1(NC(C2C(C)OCC2)=O)CCC2(CC1)CC2NC(c1nn(C)cc1N)=O c1(C(=O)NCCCN(C(C2CCSC2)=O)C2CC2)[nH]nc2ncccc12 CCC1(C(=O)OC)CNC1=O.N1(C(C(=O)OC)=O)CCCCC(c2ccco2)C1 C1(NC(c2cc(C)no2)=O)CCCN(C(=O)C(C)n2cccc2)C1C S(=O)(=O)(c1cc(F)c(F)cc1F)N1C2CN(C(c3cc(C)cc(C)c3)=O)CC21 c1(C(N(CCNC(C(C)(C)CF)=O)C2CC2)=O)ncc(Cl)cc1Cl C=C(C)CC(C(=O)N1CC2CCC2(NC(=O)C(N2CCCCC2=O)C)C1)OC C(=O)(C(O)CCCCC)NCC(CC=C)NC(=O)CCOc1ccc(C)cc1 C1(NC(CNC(CNC(c2cc(CC)ncn2)=O)=O)=O)CC12CCCCCC2 CCCCCCC(=O)N1CCC(COC)(NC(c2cnc(C(N)=O)cn2)=O)C1 C1(C(=O)NCC(C2CCC2)NC(CC=C(C)C)=O)COC2(CCC2)CO1 Cc1cnn(C(C)C(N2CC(c3ccccc3)(NC(=O)CCC3CCC3)C2)=O)c1 O=C(CC1OCCc2ccccc21)N1CCN(C(=O)COC2CCC2)C(CF)C1 C1(C(=O)NCC2N(C(C3(c4cccc(F)c4)CC3)=O)CCC2)CCCS(=O)(=O)N1 c1(C(=O)NC(CN(C(=O)CSCc2ccno2)C)(C)C)ccc(S(N)(=O)=O)cc1 C1(NC(C2CC3CC3C2)=O)CCCC12CN(C(c1csc(Cl)c1Cl)=O)C2 C1(NC(COCC(=C)C)=O)CCCC(NC(c2cnc(C)nc2C(C)C)=O)CC1 C(=O)(C1CCCc2c[nH]nc21)N1C2C(NC(c3c(COC)cc[nH]3)=O)C(C2)C1 C1(c2onc(C)n2)CCCN(C(=O)Nc2ccccc2C(C)C)C1 N1(C(=O)CSCCNC(C2CC2C(F)(F)F)=O)CCN2C(=O)NCC2C1 CCC1CCCC(=O)NC(C(C)C)C(=O)N1.c1(C(=O)NC)cncn1C(C)C C1(NC(CC(C)n2ccnc2)=O)CCCCN(C(=O)CP(C)(C)=O)CC1 c1(NCc2ncc(CC)s2)cccc2c(CC(=O)OC)c[nH]c12 c1(C(=O)NCC2COC(CNC(C3CN(C4COC4)C3)=O)C2)n[nH]cc1[N+](=O)[O-] CCC(C)(C)C(=O)C(=O)N1CC2CC1CN(C(=O)COC1CCOC1)C2 C(=O)(C1=CCCC1)N(CC1CC1NC(Cc1nc(CC)sc1)=O)Cc1cccnc1 c1(C(N2CCC(C(N3CC(OC(=O)NCC)C3)=O)C2C)=O)cc2cccnc2[nH]1 C1(C(N2CC(CC=C)(NC(=O)CC(C)OC)C2)=O)CCC(NC(C)=O)CC1 C1(CC(=O)NCCCC=CC)CC(C)N(C(c2cnc(C)s2)=O)C1 N1(C(C(C2CCOC2)OC)=O)CC2CCC1CN2C(c1nocc1C(C)C)=O c1(C(=O)NCC(c2ncc[nH]2)C)ccc(CNC(C2CCSC2)=O)nc1 C1(C(c2ccc(F)cc2)NC(c2ccc(-n3ccnc3)cn2)=O)CCCCCC1 N1(C(c2n(CCCC)ncc2)=O)CCCCCC(NC(c2cnoc2C)=O)C1 c1(SCC)ccc(C(N2CCC(CNC(c3ccn(CCOC)n3)=O)C2)=O)cc1 N1(C(c2ccn(CCC)n2)=O)CC(C(=O)NCC2CC23CCCCC3)CC1(C)C C1(C(N(CCCNC(=O)C(O)C2CCCC2)CC)=O)CC12CCSCC2 C1(C(C)(C)C)CCCC(C(=O)NC(C)(CNC(=O)CCc2ccco2)C2CC2)C1 CC1CCC(CC(=O)N(CCCN(C)C(c2cnn(C)n2)=O)C)O1 N1(C2CCN(C(C3C(=C)C3)=O)C2)CCN(C(=O)C(CC)n2ccnc2)CC1 C1(O)(C(N2CCC(C(C)O)C2)=O)CCN(CC=Cc2ccco2)CC1 N1(C(C(C)n2cncn2)=O)CCC(CO)C(NC(=O)CCN2CCN(C)CC2)C1 c1(CN(C2COC2)CC#C)ccc(NC(C2CCN(C(=O)NC)C2)=O)cc1 C=CC(C)CC(=O)N1CCOC(CCCNC(c2ccc(CC)[nH]2)=O)C1 c1(N2CCC(=CCNC(c3c(Cl)nc(N(C)C)s3)=O)CC2)ccc2nnnn2n1 c1(C(=O)NC(CC)CN(C(=O)C=C2CCOCC2)CC)cn(C)c(C)n1 C=C(C)CC(C)C(=O)NCCCC(CCC)NC(c1csc(C(C)(C)C)n1)=O c1(C(N(CCOCCNC(CCC)=O)C)=O)ccsc1Cn1cncn1 c1(C(=O)NCC(C)N(C(=O)CC2CSCCS2)CC)cnc(C)nc1C1CC1 C(CC)(C(=O)NCC(O)CN(C)C(C1(NC(N)=O)CC1)=O)OCC n1(CC)ncc(C(=O)NCC2C(C)CCN2C(c2ccc(C(C)=O)o2)=O)c1C c1(C(=O)NCC2(NC(C(SC)SC)=O)CCOC2)cc(C)c(O)nn1 N1(C(C=COCC)=O)CCC2(CCC2CNC(C2(C)CCN(C)C2)=O)CC1 c1(OC)ccccc1C(C)CC(=O)NC1CCCC1(C)N1CCOCC1 CC1CN(C(c2cnc(O)n2C)=O)CCC1C(=O)NCC1CCC(C)(C)CO1 c1(NC(Cc2c(C)cccc2)C)nccc(=NCCCc2cc(N)ccc2Cl)[nH]1 c1(CC(=O)NCC(CNC(C(C2CC2)SC)=O)C)ccc(C(N)=O)nc1 c1(C(=O)NCC(=O)NC2CC2)cncc(C(F)(F)F)c1 N1(C(c2cnc(C)[nH]2)=O)CCC(F)(F)C(CNC(=O)CN2CCCNC2=O)C1 C1(NC(C(C)=C(CC)C)=O)CCC(C)(CNC(=O)C(C)OCCN(C)C)CC1 n1(CC)ncc(Cl)c1C(=O)N(C)CC1CCN(C(c2cnc(C(N)=O)cn2)=O)C1 CCCC(C)CCCC(=O)N1CCCC1C(C)(C)NC(C1CCS(=O)(=O)CC1)=O c1(C(C)(C)C)nc(C(=O)NCC2CC(O)(CNC(c3ccsc3)=O)C2)cs1 N=c1[nH]c(=NCc2ncccc2N)[nH]c(=NC2CCN(CO)C3(CCCC3)C2)[nH]1 N1(C(c2cc(OC)ns2)=O)C2CCC1CC(NC(C1(N(C)C)CCCOC1)=O)C2 c1(C(=O)NCC(C)(CO)NC(C(CC)n2cncn2)=O)ccc2n[nH]cc2n1 N(C(=NCCN1CCC(C)(C)CC1)NC1CN(C)CC1O)CC(=O)NC(C)C N1(C(CC(C(C)C)O)=O)CCCN(C(c2cc(N)cnc2Cl)=O)C(C)C1 C(=O)(C1NCCc2ccccc21)Nc1c(N2CCC(CC)C2)ccc([N+](=O)[O-])c1 C1(C(=O)NCC(=O)N(C(C)CCO)C2CCCC2)C2CCC1(c1ccn(C)n1)C2 Cc1cc2c(cc1C(N1CCCC(C(C)(O)CNC(C3(O)CC3)=O)C1)=O)OCO2 N1(C(C2C(CC)C2)=O)C(Cn2cc(-c3ncoc3C3CC3)nn2)CC2CCCCC12 CC1CN(C(=O)C(F)n2ccnc2)CC1NC(c1csc(C(N)=O)n1)=O N1(C(C2(SCC)CC2)=O)CC(CNC(=O)CSc2nccn2C)(OC)C1 C1(C(=O)NC2CC(CNC(=O)Cc3cccc(Cl)c3)CC2O)OC2CCC1CC2 N1(C(C(C)O)=O)CC(C)(NC(c2ccoc2I)=O)C1 C(C)(N=c1[nH]c(N2CCCN(C)CCC2)nc2ccsc12)C1CCC(CC)CC1 Cc1ncccc1CNC(c1nnn(C2CC2)c1C(F)(F)F)=O N1(C(c2n(C=C)nnc2)=O)CCC2(CC1)CC2CNC(=O)CCc1cc(C)[nH]n1 c1(C(N(C(CC)CNC(c2cn(CCOC)nn2)=O)C)=O)cnc2ccccn12 C1(CNC(CC(c2ccccc2Cl)C)=O)CCN(C(=O)COC2CC2)CC1C C1(C(=O)NCC(C)(C)C2(O)CCC2)CC12CCC(F)(F)CC2 N1(C(C(CCC)OC)=O)CCCN(C(=O)COc2cccnc2)CC1C(C)C C(N=c1[nH]c(C)cc(=NC2CCC3CC2CO3)[nH]1)C1CCN(CC)C1 C(CCF)(C(=O)OC(C)(C)C)NC(N1CCC(C(F)(F)F)(C(=O)OCC)C1)=O C1(CC)CCCC1(C)C(N1CCN(CCCNC(=O)C2CC2)CC1)=O N1(C(C2CC(C)C2)=O)CCC(C)C(NC(C2(C)CCN(C)CC2)=O)C1 CP(C)(=O)CCC(=O)NCc1cc(C(=O)Nc2ccc(Cl)cc2O)co1 C(=O)(CCCC(=O)C1CC1)N1CCC(N(C(=O)CCC2CC2)CC2CC2)CC1 O=C(CC(C1CC1)NC(c1c[nH]cc1C1CC1)=O)NCC(O)CO C(C(C)(O)CC(=O)N1CCC(C(=O)NCCC(F)(F)CO)(C(C)C)C1)OC C#Cc1cccc(C(=O)NCCCOCCNC(C2(CC3CC3)CCOC2)=O)c1 c1(C(=O)C(c2c(F)cccc2F)(F)F)c(Br)cc(F)c(C(F)(F)F)c1F C1(NC(c2nc(CC)sc2)=O)CN(C(=O)COCC2CCCC2)C2CC12 Cc1nc2c(C(N3CCC(N(C(=O)COCCCF)CCO)C3)=O)cccc2o1 C12(C(=O)NCC(C#C)OC)C(NC(=O)CC3CCOC3)C3CC1C2C3 C(CCCCCC(=O)NCC1CCSC(C)C1)NC(COCCCCC)=O C(Cn1cccn1)(C(=O)Nc1conc1CC)NC(C=C(CC)C)=O c1(C(=O)NC(CN(C(CC(CC)C2CC2)=O)C)C)cc(S(C)(=O)=O)ccc1OC N1(C(c2c(CC)cno2)=O)CCCC(F)(CNC(C2CC(F)(CO)C2)=O)C1 c1(C(N2C(C(C)(C)NC(C(C)C(F)F)=O)CCC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 c1(C(=O)NC2(CC=C)CCN(C(C3CCN(C)C(=O)C3)=O)C2)cnc(Cl)cc1N CC1=C(C(=O)NC(C(=O)NCC(C2CCCCC2)O)C2(C)CC2)SCCO1 N1(CC(=O)NC2CN(C(=O)CN3CCCC3)CCC2F)CCCCS1(=O)=O C1(C(=O)NCC2CC(F)(CNC(c3ccc(C)cn3)=O)C2)CCc2nn[nH]c2C1 c1(C(=O)NC2(CC(=O)N(CCOC)C)CCC2)ccc(C)cc1O C=CC(CC)CC(=O)N1CCCC(NC(=O)COc2ccc(C)cc2)C1CC C1(N2CC(NC(=O)NCCN(C)Cc3ccccc3)C2)CCOCC1 CCCN=C(NCc1ccc(CC(=O)OC)cc1)NCc1ncn(C)n1 C1(NC(C(C=C)CC)=O)CN(C(=O)C(c2ccccc2F)O)CC1C=C N#Cc1cc(S(=O)(=O)N2CCCC(C(=O)Nc3ccsc3)C2)ccc1F CC(C)(C)C(CC(=O)N1CC(CO)(CO)C1)NC(=O)Cc1ccsc1 Cc1ccc(C(=O)NC2CC3CCC2N3C(=O)CC(C)c2cnn(C)c2)nc1C Cc1cccc(C)c1C(N1CC(NC(=O)CCc2ncco2)CC(F)C1)=O c1(C(=O)NC2CN(C(C(N)=O)=O)CC2c2ccccc2)ccnc2ccncc12 C12CC3CN(CC13)C(=O)C1(CCOCC1)OCC(=O)N2.c1csnn1.COC c1(C(=O)NCC2CCC(NC(c3c(CC)nns3)=O)C2)cnc(C2CC2)nc1O c1(C(N2CCN(C(C=CCOC)=O)C(C(C)C)C2)=O)ccn2c(C)ncc2c1 Cc1cc(C)c(C(=O)NC(CC2CCCC2)C(=O)NCCc2ncon2)cn1 O=C(CC1OCc2ncccc21)NCCSCC(O)CO c1(C(=O)NCC2(CNC(Cc3c(C)nc[nH]3)=O)CCC2)csc([N+](=O)[O-])c1 CCC(C#N)C(=O)N1CCC1C(=O)NCCC(=O)N1CCC1 C1(NC(C(=O)Nc2ccc(F)cc2)=O)CCN(C(C2CCCC2CF)=O)CC1O c1(C(=O)NC(C2(O)CCN(C(CCN(CCC)C)=O)C2)C)cccc2nncn12 C(C(O)(C(=O)NCC(CNC(=O)CCCCC(F)(F)F)OC)C(F)(F)F)N(C)C Cc1ccc(SCC(=O)NCC23CC2CN(C(=O)CC(C)(F)F)C3)cc1C N1(C(c2c(Cl)cn(C)n2)=O)CC(C)(C)OCC1CNC(=O)CC1CSCCS1 c1(C(N2CCCC(C(=O)NC(C(=O)OC)C(=O)O)CC2)=O)ccc2cncnc2c1 c1(C(N2CC3C(NC(=O)COCc4ccccc4)(C3)C2)=O)c(F)ccc(F)c1F N1(C(=O)COCC2CCC2)CCC(F)(C(N2CCC2(CO)CO)=O)C1 c1(C(=O)OC)[nH]c(=NC2CC23CC(NC(C2OCC2(C)C)=O)C3)sc1C c1(C(=O)NCC2CCCCN(C(c3cnncc3O)=O)C2)cccn2cncc12 C1(C2CCN(C(=O)CC3CCOCC3)C2)(NC(c2cnnc(O)c2)=O)CC1 C(=O)(CC(C(F)(F)F)N1CCOCC1)NC1(CO)CN(C(CCCC(C)C)=O)C1 N1(c2nc(N3CCN(C)CC3)c(Cl)cn2)CCC2(CC1)CC(N(C)C)CO2 C(=O)(C1=CC2CCCCCC12)NC(C(c1ccc(OC)cc1)OC)C C1(C(N2CC(N(C)C(C3CCC3)=O)C3(C2)CC3)=O)Cc2cc(Cl)ccc2O1 C1(OC)CCC(C(=O)N(C2CCN(C(=O)CCc3cccnc3F)CC2)C)CC1 Cc1csc2c(C(=O)NC3COCCN(C(=O)C(O)C(F)(F)F)C3)cccc12 C1(NC(COCCCC(C)C)=O)CN(C(C2CC(S(C)(=O)=O)C2)=O)CCC1C C1(CC(=O)NC(CC)CNC(=O)CNC(C2CC2C)=O)CCCCC1 C1(OC)CCC(CNC2CCCN2C(=O)COc2ccccc2)CC1 CC(C)(C(=O)NC1CC(CNC(c2cc[nH]c2)=O)C1)C1CCCCO1 N1(C(CCCNC(C(=O)Nc2n(C)ccn2)=O)=O)CCC(N)CC1 N#Cc1c[nH]cnc1=NC1CCC(NC(=O)CN2CCCCCC2=O)C1 c1(CC(=O)NC(C)(CNC(=O)CSC2CC2)CO)cc(F)cc([N+](=O)[O-])c1 C1(C(=O)NCC2CN(C(=O)C3=CCOC3)CC2O)CC2CCC(C1)S2(=O)=O c1(-c2nc(CC(CC)C)nn2CCC(C)C)cc(C)ccc1Br C(C(C)(C)C(C)(C)C)NC(CNC(CNC(c1cc(OC)no1)=O)=O)=O c1(C(C(=O)OCCc2cccc(OC(F)F)c2)=O)cc2ccccc2s1 O=C(C1CCc2cc(O)cc(=O)n21)NC1CC1C(F)F c1(NCC(c2cccc(OC)c2)C)nc[nH]c(=NCC2CC2(C)C)c1C C=C(Cl)C(C)(C)C(=O)NCCC1CCN(C(c2cccc(C(N)=O)n2)=O)C(C)C1 C1(OC)CC2(C1)CN(C(=O)C(C)CNC(C1(C)CCNC1=O)=O)C2 C(C(COC)C(=O)NCCN(C(=O)CC1CCCOCC1)C)OC c1(CC)ccc(C(=O)N(C)Cc2cccc(Br)c2)c(OC)c1 C1(CN(CC)CC)CCCCN1C(=O)Cc1cnn(C)c1C N1(C(C2CN(C(C3(SC)CC(=O)C3)=O)CC2F)=O)CC(C)=CC(C)C1 c1(C2C(NC(=O)CCCC3N=N3)C2)cccc2ccccc12 N1(C(c2c(C)nccc2)=O)CCC2(CC1)CC2C(=O)NC1CCC1(C)C C1(N(C(c2nc(OCC)oc2)=O)C)CCC(NC(=O)CCC(=O)N(C)C)CC1 CCC(CC)CC(F)C(=O)OC1CC(N2CCNC2=O)C1 c1(C(=O)NCC(CO)NC(c2ccc(OC(F)(F)F)nc2)=O)c[nH]cc(F)c1=O C1(C(=O)NCC(C)OCC=C)CC=CCC1NC(=O)COc1ccn(C)n1 C(C)(C(=O)NCCN1CCC(NC(C2CCS2(=O)=O)=O)CC1)(C(C)C)OC c1(C(=O)NC(c2ccsc2)C)ccc2c(c1)CCN(Cc1cc(Cl)ccc1Cl)C2 C(=O)(C(C)CC)N(CCC)Cc1sccc1C CCCC(CNC(C1CCN(C(=O)C=Cc2cc[nH]c2)C1)=O)OC C(=O)(C(O)(C(F)(F)F)C1CC1)NCC(CNC(c1nc(CCC)oc1)=O)F c1(OCC)cc(Cl)ccc1C(N1C2CCC1(CNC(C1CCC1(C)C)=O)CC2)=O c1(OC)nscc1C(N1CCCC1CC(=O)NC1CC1C(F)(F)F)=O N1(C(C)=O)CC(NC(C2CC(NC(=O)COc3ccsc3)C2)=O)C1 N1(C(C(C)(c2cccs2)N(C)C)=O)CCC(F)(CNC(=O)C#CC(C)(C)O)CC1 C1(C(=O)NCc2nnn(C)c2C)(NC(C(C)=C2CCCC2)=O)CCCC1C c1(C(c2n(CC=C)nnn2)NC(C2(C)COC2)C)cnn(CC(C)C)c1C1CC1 C(=O)(C(C)(C)S(C)(=O)=O)NC1CCN(C(C2(CC#C)CC2)=O)CC1F Cc1csc(=O)n1CC(N1CCC(C)(CNC(=O)Cc2cnn(C3CC3)c2)C1)=O C(=O)(C1SCCc2ccccc21)N(CCNC(CC(C=C)CCC)=O)C N1(C(CC)=O)CCc2[nH]nc(CNC(=O)CSc3cc(Cl)cc(Cl)c3)c2C1 C1(C)(C(=O)NC2CCC(CNC(C(C)(C)c3ccno3)=O)C2)CCCNC1=O CCS(=O)(=O)CC(=O)N1CCC(C)(N(C(=O)C(c2ccccn2)C)CC#CC)C1.C CCC(CC)C(F)C(=O)N1CCC2(CC2C(=O)NC(C)(C)CN(C)C)C1 N1(C(C(C)OCCCC)=O)CCC(CNC(c2cn(CCC3CC3)nn2)=O)CC1 c1(CNC(CCSC)=O)n[nH]cc1C(=O)NC(CO)C(C)C N1(C(CC2(C)CCC2)=O)CC=C(C(=O)NC(C(F)(F)F)C2CC2)CC1 c1(C(N2CCCC(NC(C(C)(C)C3CC3)=O)C(F)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(NC(C2(F)CCC2)=O)ccc(C2CCN(Cc3ccnnc3)CC2)cc1 N1(C(CC2(C=C)CC2)=O)CC(NC(=O)C(C)NC(=O)NC)C(C)(C)C1 CC1CC(C(N2CCN(C(c3cn(C4COC4)nn3)=O)CC2)=O)CN1C c1(OC)cc(=NC(=O)C(C)(C2CC2)N(C)C(C2C3CCCOC23)=O)[nH]n1C c1(NC2CC(C)C(C)(C)CC2)ccc(S(=O)(=O)NC2CCCCC2)cn1 CC1(C(N2CCCC2CNC(=O)C(F)(F)c2csc(Cl)c2)=O)CCNC1=O CCCC(C)(C)CC(=O)NCC1CCC2(CN(C(=O)C(CC)(CC)CO)C2)O1 c1(C(=O)OC)cccc(N(C)C(=O)NCCNC(c2ccc(C)cn2)=O)c1 N1(C(c2c(C#N)ccs2)=O)CCC(NC(=O)CC(F)F)C(CO)C1 c1(C(=O)NCC2CCCC(NC(=O)CSC(F)F)C2)ccc2nc[nH]c2c1 C1(NC(C2CCOCC2)=O)COCC1CNC(C1CC1F)=O C1(C(=O)NC(CC#C)C(=O)N2CCC2C2CCOCC2)CC(C)(C)CN1C S(=O)(=O)(c1ccc(-c2cccc(C)c2F)s1)N(C(C#C)C)C c1(CSCC(=O)NCCC2CCN(C(=O)C(=O)NC(=O)CO)C2)cccnc1 c1(CNC(=O)CC2CCCCCN2)ccc(S(=O)(=O)N2CCOCC2)cc1 C(=O)(C1CCc2cccc(O)c21)N1CC(CNC(C=CCOC)=O)C(F)(F)CC1 CCCC(C)C(c1nnnn1CC)NCCCc1noc(C(C)(C)C)n1 C(=O)(C(F)(F)C(F)F)N1C(CN(C(C(c2scc(C)n2)C)=O)C)CCC1 N1(C(C2CCN(C(C)=O)C2)=O)CCC2(CCC(NC(c3csc(Cl)n3)=O)C2)C1 CCC1=C(C(=O)N2CCN(C(=O)C(F)C3CCOC3)CC2CCO)CCCO1 C(CN=c1[nH]nc(C(N)=O)s1)=CCNC(C1=C(C)CCC1)=O c1(CC)ccc(C(=O)NC(C)(CNC(=O)C(C(C)C)NC(N)=O)C(C)C)c(C)n1 CCC(C)(C)CCCC(=O)NC(C1(O)CCN(C(=O)C#CC2(CC)CC2)CC1)OC CC(C)CC(CNC(c1cc(F)n(C)n1)=O)NC(C1CC1C)=O c1(C(N(CCCCN(C(C=CCC)=O)C)C)=O)ccc(C(C)(C)C)cc1N Cc1cccc(Br)c1C(=O)NC(CNC(c1ccc(Cl)s1)=O)C(C)C C1(CNC(c2ccn(C(C)(C)C)c2)=O)CC2(CC2)CN1C(=O)CCC(=O)C1CC1 Cc1c(C(N2CC(C3CN(C(c4ccns4)=O)C3)C2)=O)cnc2ncnn12 c1(CCOCC(=O)NC2(CNC(C=CC=CC)=O)CCOC2)ccc(Cl)cc1 CCC(C)C(C(=O)NCCCCOc1ccc(F)cc1)NC(C)=O C12(NC(C(CNC(C=C(CCC)CCC)=O)C)=O)CC3CC(CC1C3)C2 C1(NC(C=CCC(C)(C)NC(=O)CP(C)(C)=O)=O)CCC(O)CC1 C(CCN=C(NCc1ccc(F)c(F)c1)N1CCC(C)(F)C1)SC c1(OC(C(=O)Nc2nccc(CC)n2)C)ccc(Cl)cc1C C1(CC(=O)NCC2CCC(NC(c3cc(-c4ccoc4)[nH]n3)=O)C2)CC2(CC2)C1 C1(C(=O)NC2(CO)CN(c3ncnc(Cl)c3F)C2)C2Cc3ccccc3C12 c1(C(=O)NCCc2c(CNC(C=C=C(C)C)=O)nco2)cncc2[nH]ccc12 C(C(C)(CO)CO)N(C)C(C1CCOC1CNC(C1COCCN1C1CC1)=O)=O C(CC(C(=O)N1CC=C(C)CC1)NC(=O)CCCN1CCCC1)OC CC(C)CC(C)(CNC1C=CC=CC=C1)NC(=O)C(O)CN(C)C Cc1cc(N)c(C(=O)NC(C)CCNC(C2CC2[N+](=O)[O-])=O)c(F)c1 C1(NC(c2ccc(C(C)=O)s2)=O)CC2CCCC(C1)C2(F)F C(=O)(C1=NN(CCO)C(=O)CC1)NC(C1CCCCN1C(=O)CCCN=[N+]=[N-])C C1(NC(CC(C)OC)=O)CC2CC(C1)N(C(C1CCCN1C=O)=O)C2 N1(C(C2(CC)CCN(C(=O)C=CC3CCOC3)C2)=O)CCOCC(C)(O)C1 c1(C(=O)NCC2(CC(=O)N(CC(CC)O)C)CC2)cncc(NC)c1 C1(C)(CNC(CC(C)=C(C)C)=O)CCN(C(C2(C)CCCCO2)=O)CC1 Cc1cccc(C(C)NC(=O)C(O)CNC(C2(Cl)CC2)=O)n1 C1(C(=O)Nc2ccc(CN(CC)CC)cc2)(OC)CCC(F)(F)CC1 CON1CC(C(N2CC(C)(C(=O)NC3(CCO)CCCC3)C2)=O)CC1=O N(C(=NCCC1CCCC1)NCc1ccco1)CC1C(N(C)C)CCCC1 c1(CNC(c2cccnc2N(C)C)=O)ccc(C(C)NC(CCC)=O)cc1 N1(C(C(CC)COC)=O)CC(NC(C23CC4CC2C3C4)=O)C2CCCCC12 C(C)(C(C)CCC)NC(CCN(C(CCCC)=O)CC1CC1)=O c1(CC)cnc(C(=O)N(C(C)CCNC(=O)C(c2cccnc2)O)C)s1 c1(OC(C)C(=O)NCC=C2CCN(C(C3(C)COC3)=O)CC2)cccc(F)c1 N1(C(C2N(C(C3OCCC(C)C3)=O)C(C3CC3)CC2)=O)CCC2(CCC2)CC1 C1(C(N2C(CN(C(CCCCOCC)=O)C)CCC2)=O)CCc2c(n[nH]c2C)C1 c1(SC)ccc(C(=O)NCc2ccsc2C(N2CC(c3nncn3C)C2)=O)o1 C1(C(N2CCCC(CNC(=O)COC(F)(F)F)C2)=O)(OCC)CCOCC1 C(=O)(C1(C)CCc2ccccc21)N1C(CNC(COC(C)=O)=O)C(C)(C)CCC1 N1(C(C2CC(C(C)(C)C)C2)=O)CCCC(O)(CNC(c2ccoc2)=O)CC1 N1(CC)CCCc2cc(NS(=O)(=O)CC3CC4CCC(C3)C4)ccc21 c1(-c2cccc(OCC)c2C)c[nH]c2ccc(C(N3CC(CO)C(O)C3)=O)cc12 C1(CC(=O)NCCCN(CCC)C(c2cnc[nH]2)=O)CCCC1C c1(C(=O)NCC=CCNC(C(C)OCOC)=O)cnc(C)nc1C Cn1cc2c(n1)CC(C(=O)NC1COCC1CNC(=O)C(=O)NC1CC1)CC2 CCCCCC(F)C(=O)N(CCCN(C(=O)CC(C)(C)N(C)C)C)C c1(OC)ccc(C(C(=O)NCC2CC2)N2CCC2C2CCC2)c(Br)c1O C(=O)(C(O)(C(F)(F)F)c1cn[nH]c1)NCCC(CNC(c1c(C)n(C)nn1)=O)O N1(C(Cc2c(C)con2)=O)CC2(NC(c3ccc(=O)n(CCF)n3)=O)CCC1C2 C(=O)(C1CCCn2ncnc21)N1CC(C(C)NC(C2CC3(C2)CC(O)C3)=O)C1 C1(CNC(=O)Cc2cncnc2)CC2(CCN(C(c3cnccc3Cl)=O)C2)CO1 c1(C(=O)NCCCN(C(c2ncoc2C2CC2)=O)CC)cnn2c1OCC(O)C2 c1(C(=O)NC(C(C)(C)C)CNC(C2OCCO2)=O)n[nH]c2c1CS(=O)(=O)CC2 C1(CNC(CC2C(C)CCC2)=O)COCCN(C(c2ncc(C(F)F)s2)=O)C1 N1(C(C)C)CC(C(=O)N(CCCCN(C)C(C2CNC(=O)N2)=O)C)CCC1=O N(C1CCOc2c(Br)cccc21)CC.c12cc(NC(C)=O)cc(c1)CNC(=O)N2 N1(C(C2CCCCC(=O)C2)=O)CCc2cc(-c3cn[nH]c3)ccc21 O(P1(=O)COCCCO1)C(C)C.c1(-c2ccc(C(=O)OC)o2)cc(Cl)ccc1Cl c1(CC)oc(C(=O)OCC2C3CCCCC23)cc1C C1(NC(c2ccc(-c3nc[nH]n3)nc2)=O)(CO)CCN(C(c2ccc[nH]2)=O)C1 c1(C(N(CC(CC)NC(=O)C(C)(C)O)C)=O)ccc2c(c1)S(=O)(=O)NC=N2 CC(C)(C)C(O)C(=O)NCC1(NC(=O)CSCCN(C)C)CCCCC1 N1(C(C(c2ccn(C)n2)C)=O)CCCC(C(=O)N(CC(C)(O)C2CC2)C)C1 C(=O)(C#CC1(C)CC1)OCC1CCC(CNC(Cc2c(OC)nccc2)=O)CC1 c1(C(=O)NCC(CCCC)NC(=O)C(O)CCN(C)C)cc(N)ccc1SC CS(=O)(=O)C1(C(=O)NC2CC(c3ccccc3)C2)COC(=O)C1 c1(CC(=O)NC2CCCCC2c2nc[nH]n2)ccc(Cl)nc1 C1(CNC(C(CC)OC)=O)Cc2ccccc2CN1C(=O)COC1CCCOC1 c1(CC)cc(C(=O)NC2(CO)CN(C(C3(Sc4ccccc4)CC3)=O)C2)oc1C N1(C(Cc2c(C)con2)=O)CCC(CNC(=O)C(C)C(C)C)C12CCC2 C=CC(C(=O)NC1CCCC1NC(=O)CSCC(N)=O)c1ccccc1 c1(CC)conc1C(=O)NC(CC1CCCC1)C(=O)NC(C)CC1CCC1 C=CCCC(C)(C)CNC(=O)C=CC1CCCN1C(=O)C=C1CCC1 N1(CCn2c(C)cc(C)n2)C2CCC1CN(C(=O)C(=O)C1CCCC1)CC2 C1(N2CCN(c3c(C)nccc3)CC2)CCCCN(C(c2ccn(C)c2)=O)C1 C1(C)(CC)CC(NC(c2cc(C#N)cn2C)=O)CN1C(=O)Cn1cc(C)cn1 C1(NC(CCS(C)=O)=O)CN(C(c2cc(C(N)=O)c[nH]2)=O)CCC1(C)C N1(C(C(C)OCCC=C)=O)CC2CCOC2(CNC(c2cn(C)nc2CC)=O)C1 C(=O)(C(C)(C)CC1CC1)NC(CCN(C(CSc1n(C(C)C)cnn1)=O)C)C C1(CNC(c2c(C)csc2)=O)CC12CCN(C(c1scnc1C)=O)CC2 Cc1ccoc1CNC(=O)N(CC(C)C(C)C)C C1(OC)CCC(c2nnnn2CC2CC2)(NCCCSC)CC1 c1(OC)ccc(C(F)(F)C(=O)NCC2CCCN2C(C2(O)CCCC2)=O)cn1 C(=O)(C(O)C(F)(F)F)N(CC(CNC(c1n[nH]c(C)c1Br)=O)C)C C(CN(C(=O)C(C1CCN(C(=O)CCN2CCCC2=O)C1)C)C)(C(C)C)OC N1(C(=O)Cc2ccc(Cl)nc2)CCN(C(C23CCCC2CC3)=O)CC12CC2 c1ccc2c(-c3ccc(N4CCC(C)C4C4CCCC5CC45)[nH]3)cccc2c1 CC(CC(=O)NC1CC(CO)C1)C(C)(C)NC(C1CC1(F)Cl)=O N1(C(CC(=C=C)C)=O)CCCCCC(NC(c2nnc3ccccn23)=O)C1 c1(CCC(=O)NCC2(C(N)=O)CN(C(C3CCC(OC)C3)=O)C2)ccnc(Cl)c1 C(=O)(C#CC1CCOC1)N(CCCC(=O)NC1CC2(CCCC2)C1)C C(CCCCCNC(c1c(C)nco1)=O)N(C(=O)C(CO)c1ccccc1)CCO C1(CC)CN(C(=O)C(=O)C2CC2)CCC1NC(c1ccc(=O)n(C2CC2)c1)=O c1(C(=O)NC2CCN(C(Cc3nnc(C)s3)=O)CC2C)cc2cccc(F)c2o1 N1(C(C(C)=O)=O)CCN(C2CCN(C(=O)CC(C)C3CCCO3)C2)CC1 c1(C(N(CC(C)NC(C2CCC(=O)C2)=O)C)=O)nc(Cl)cs1 CC1(C)CC(NC(c2ncccc2F)=O)CN1C(C12CCC(F)C1CC2)=O N1(C(C(C2(O)CCC2)NC(c2cn(CCC)nc2)=O)=O)CCN(CC)C(C)C1 N1(C(C2N(C(c3c(COC)cco3)=O)CC(=O)NC2)=O)CCOCC(C)(O)C1 C1(NC(c2ccc(CC)s2)=O)CCN(C(c2ccc(N)cc2C)=O)C(C)C1 N12CCC(C1)CC(=O)OCC2=O.c1(N(C(C)(C)C)C)cc(-c2cnn(C)c2)[nH]n1 C1(CC)CCC(NC(=O)C(CCNC(=O)CCCN(C)C(C)=O)OC)CC1 C12(C(=O)NCC(C3CCN(C(c4n[nH]c(C)c4Cl)=O)CC3)F)CC1COC2(C)C C(C)(C)(C(=O)N1CC(CCO)(NC(=O)C(C)CN(C)C)C1)OC N1(C(c2cn(CCC)nc2C)=O)CCN(C(=O)C(O)COC)C(C)C1 c1(C(=O)NC(c2cn(CCCNC(=O)C(O)c3cnc[nH]3)nn2)C)c(Cl)cnn1C CN(CC1CCN(S(C)(=O)=O)CC1)N1CCOC(c2ccc(C#N)cc2)C1 c1(C(C)(C)C#N)ccc(C(=O)NCC(C)(O)CNC(=O)CSC(F)F)cc1 N1(C(=O)Cc2csc(Br)n2)CCC(CNC(C2(CC3CC3)CCCO2)=O)C1 C1(N(C)C(C2CC(C)(C)CCN2)=O)CCS(=O)(=O)CC1 N1(C(C(C)OCCOCC)=O)CCOCCC1C(N1CCC(CC)C1)=O C1(NC(C(C2CCC2)NC(C(C)NC(CC)=O)=O)=O)CNC(=O)C1(C)C C1(C(=O)NC(CC)COC)(CNC(=O)CSC(C)(C)C)CC2(CC2)C1 C(=O)(CC1=CCN(C(c2cnc(C3CC3)o2)=O)CC1)N(C)Cc1nc(C)[nH]n1 c1(OC)cc(NCc2cc(Br)c(C)cc2OC)ccc1S(C)(=O)=O CC(C)(C(=O)NCC(C)(C)C#CC(=O)NC1(C(C)(F)F)CC1)C(F)(F)F c1(C(N2CC(C(C)(C)O)(CNC(CCc3nc(C)sc3)=O)C2)=O)nc(=O)n(C)[nH]1 C1(OC)CNCCC1CNCc1cnc(N2CCN(C)CC2)n1C C(=O)(C1=CC2CCC1C2)N1CC(NC(c2ccc(C(N)=O)[nH]2)=O)C1 c1(C(=O)NCC2N(CC(=O)NC3CCC4CC34)CCCC2)cccn2cncc12 CN1CCN(c2ncc(Cl)c(O)n2)C(CNC(c2ccc(F)c(C(F)F)c2)=O)C1 c1(C(=O)NCCN(C(CN2C(C)CCC2C)=O)C)cc(Cl)c(F)cc1F C1(N(C(=O)CCc2cc(Cl)cs2)C)CN(C(=O)CC2COCCN2C)CCC1O c1(C(=O)NC2CC(C)CN(C(c3ccoc3)=O)C2)n[nH]c2ccc(C(F)(F)F)cc12 C(=O)(C1CCc2ccc(Cl)nc21)N1CC(F)(CNC(c2ncc(F)cc2F)=O)C1 c1(SCC(N2CCC(CNC(c3cscn3)=O)CC2)=O)ccc2c(c1)CCC2 C(=O)(CCCCCC#N)NC(CNC(COc1c(C)ccc(Cl)c1)=O)C C1(C)(CNC(c2nc(CC)oc2)=O)CCCN1C(=O)C(CO)NC(=O)C(F)(F)F N1(C(CCCCC)=O)CCOC(C)(CNC(C23CSC(C2)C3)=O)C1 Cc1cc(C(=O)N(CC(C)NC(C2(Nc3ccccc3)CC2)=O)C)c(Cl)cc1N c1(C(=O)NC(C)CC(C)NC(C23CC(F)(C2)C3)=O)cc(=O)c(Br)c[nH]1 CCC(CC)(CC)C(=O)NC1CCN(C(=O)C=C(C)C(F)F)CCC1CO C1(C(=O)NCC(CC(N2CCN(C(C)C)C(=O)C2)=O)OC)CC2CCC(C1)C2 C(=O)(C(O)CCC(C)C)NCC12C(CN(C(c3c(C)cn(C)n3)=O)C1)CC2 c1(OC)ccc(C=CC(=O)N(CC(C)(C)CNC(=O)C(C)CS(C)=O)C)nc1 c1(C(=O)NC(COC)C(=O)NCCc2cnc(C)cn2)cc2cccn2cn1 C1(NC(C2(C)CC=CC2)=O)COC2(C1)CN(C(C1CCOC3(CCC3)C1)=O)C2 C(=O)(CC(C)C(F)(F)F)NC(C(=O)NCC1CCCN(CC)C1)C(C)O C(=O)(CCCCC(=O)c1ccccc1)NCC1(C)CCOC1 C1(C)(CCNC(C(c2n(C)ncc2)(F)F)=O)CCN(C(=O)CC2CC(F)(F)C2)C1 CC1OCCN(C(=O)CC2(C#N)CC2)C1C(N1CCCN(C(N)=O)CC1)=O N1(c2cc(CC)nc(Cl)n2)CCCC12CCN(C(=O)COCCN1CCCC1)C2 C1(C(N(C2CCN(C(CC(=C)Br)=O)CC2)CCC)=O)CCn2c(O)nnc2C1 N1(C(C2(CC)CC2(F)F)=O)CCC2CCC(NC(C3CCCCCC3)=O)C1C2 c1(C(N(C2CCCN(C(=O)CCS(=O)(=O)NC)C2)CC)=O)csc2nccn12 C=CC1(CC(=O)NCc2cc(Cl)cs2)CN(C(c2cccnc2OC)=O)C1 c1(C(N2CCC(CNC(C3CN(C(C)C)C(=O)C3)=O)C2)=O)cc2c[nH]nc2s1 C(C(C(=O)N1CC=CCO1)NC(=O)C#CC1CC1)OC c1(C(C)=O)nn(C)cc1C(=O)NCCOCCCNC(C1CCCSC1C)=O N1(C(c2c(CC)nccn2)=O)CCC(C(=O)NC(C)CN2CCOCC2)=C(F)C1 c1(C(=O)OC(C)CF)ccccc1N1CCCS1(=O)=O N1(C(C2(OC)CC2)=O)CCN(C(c2ccc(CC3CC3)s2)=O)C(CF)C1 c1(NC(C2(C)CCN(CCCCCC)C2)=O)ccc(OC)cc1C c1(C(=O)NC(C2CCN(C(C3CCS3(=O)=O)=O)C2)C)ccc2oc(=N)[nH]c2c1 C1(NC(c2nocc2Cl)=O)CC(CO)N(C(=O)C=Cc2ccc(Br)o2)C1 CC(C)CC(C(=O)NCCC(N1CCCC1C1(C)CC1)=O)C(C)C c1(OC)c(C(N2CCC(CNC(=O)CC3CCCCC3)C2)=O)oc2ccccc12 N1(C(CCCOCCOC)=O)CC2CCCC2C1C(=O)NCC(C)O c1(C(N2CCC(C(=O)NCCCC)C2)C(=O)NC2(C)CC2)cc(Cl)c(F)c(Cl)c1 C(CC(C)(C)C)(C(=O)N1CCC(C(C)(C)NC(C2CCCCN2N=O)=O)C1)OC N1(C(c2cc(OCC)no2)=O)CCCC2(NC(=O)C(C)(C)CC)CCCC12 c1(C(=O)NC(C)CC(C)NC(C2(C#N)CCCC2)=O)cc2c(ncn2C)s1 C(C)(CCC(=O)NCc1ccc(C(N2CCC(C3(C)N=N3)C2)=O)cc1)OC c1(C(=O)NCC2N(C(C3CC(C)C(C)CC3)=O)CCC2)ccc2c(c1)CCN2C c1(N(CCC(=O)N(CC)CC)C)nc(N(C)C)nc2c1CC(F)(F)CC2 Cn1ncc2c(C(N3CCOC(C(=O)Nc4nc(Br)cs4)C3)=O)cc(Br)cc12 N1(C(c2c(CC)nn[nH]2)=O)CC(C)(C)CCC1CNC(=O)CNS(=O)(=O)N(C)C C1(OC)CCN(C(=O)C(C)N(C(=O)C(O)C2CC2)C)C1C(C)C Cn1cc(C(N2CCN(c3ncc[nH]3)CC2)=O)c(=O)c2cnn(C)c12 Cc1ccc(C(N2CCN(C(C3CC3F)=O)CC2c2cccnc2)=O)c(=O)n1C C1(CC=C)(NC(C2CC2C2CC2)=O)CC2CCC(C1)N2C(C1(C(C)C)COC1)=O CC(C)CS(=O)(=O)CC(=O)NC1CCN(C(C2CCCS2(=O)=O)=O)C1 N1(C(c2c(C)oc(CO)c2)=O)CC2CC(C1)N(C(=O)Nc1cnc3[nH]ccc3n1)C2 C1(C(=O)OC)CCN(CCO)C(=O)C1.N12CC(C1)N(C)CC=CC2=O c1(OCCCC)ccc(C(=O)NCC(F)CNC(C2(C)CCNC2=O)=O)cc1 c1(COC(C2CCOC(CN3CCN(CC4CC4)CC3)C2)=O)ccc2occc2c1 N1(C(=O)OC(C)(C)C)CCCC(O)(C(F)(F)C(=O)NCC2CCCN2C2CC2)C1 c1(C2CC(C(=O)Nc3nnc(N4CCCOC4=O)s3)C(O)C2)cccc2nncn12 CCC(C(=O)N(C)CCOCCCNC(c1csc(Cl)n1)=O)C(C)C c1(-n2ccc(CS(N3CCC(OC)C3)(=O)=O)n2)ccccc1[N+](=O)[O-] N1(CC(C)S(C)=O)C(=O)CN(CC2(C3CCCO3)CCC2)C1=O c1(C(=O)NCC(CNC(C(CC)n2ccnc2)=O)F)noc(C)c1C(=O)OC CC1=C(C(=O)NC2CCC(CC(=O)NCC3C=CCC3)CC2)CCCO1 C(=O)(C(F)CC(CC)CC)N(CCN(C(C(C1CCCC1)OCC)=O)C)C C=CCCCCC(=O)NC1COCC1C(=O)NC1CCCSCC1 c1(C(=O)NC(CC)(C)CNC(c2cnco2)=O)cnc2cc(Br)ccc2c1 c1(C2C(CC)CCO2)cc(CN2CC(=Cc3cccs3)CC2=O)nn1C C1(C(N2C(COC)(Cc3ccccc3)CCC2)=O)CC(N(C)C)CN(C(C)=O)C1 C1(CC)CC(CC(=O)NC2CCCC2NC(=O)C=CCO)CCO1 C1(C(=O)NCC#CCNC(CNC(=O)OC)=O)CC(CO)C1(C)C C(=O)(C1CCc2cc(Cl)ccc21)NCCNC(C(C)(C)C1CCOC1)=O C(C1CCc2ccc(Br)cc21)NC(c1cc(C)c2n(c1)ccn2)=O C1(F)(CNC(C(C)SCC)=O)CC(CNC(c2c[nH]c(Br)c2)=O)C1 c1(CC2N(CC)CCCC2)ccc(-c2nc(C3C(C)C3C)n(CC3CC3)n2)cc1 c1(C(N2CCN(C(c3cccc(C)c3C)=O)C(CF)C2)=O)cnn2ccccc12 CC1CCN(C(=O)CN2CC(F)(F)C2)CC1CNC(=O)C=CCC1CCCCC1 CC(N=c1[nH]c(N(C(c2ccccc2)CN(C)C)C)nc(=N)[nH]1)c1ncccn1 N1(C(c2ccn(C)c2CC(=O)O)=O)CC2(C1)CN(C(c1ccc(Br)cc1)=O)C2 C1(C(N)=O)CCCN(CC2CCN(CCC3CCOC3)CC2)C1 c1(C(=O)NC2CC(C)N(C(c3cc(N)cnc3Cl)=O)CC2)ccc2cc[nH]c2c1 c1(NC23CC(C(=O)OC)C(C2)C3)ccc(C(C)=O)cc1Br C(C(C)C(C)C(=O)NC1CCC(CNC(C2(CF)COC2)=O)CC1)OC N1(C(CSC(C)=O)=O)CCC2C1CCCN2C(=O)C(O)CC c1(C(C(=O)NCC2CCN(C(C=CC(C)C)=O)C2)O)ccc(O)c([N+](=O)[O-])c1 c1(CC)nc(C)cc(=NC2C3CN(C(=O)C(C)Cc4cccc(Br)c4)CC23)[nH]1 Cc1cnc(O)cc1NC(C1CN(C(c2ccc(S)cc2)=O)CCO1)=O Cc1cc(F)cnc1C(N1CCC(C)C(NC(c2cc[nH]c2C)=O)C1)=O C=CC(C)(C)C(=O)NCC1(O)CCN(C(C2CCC2(F)F)=O)C1 N1(C(C(CCCC)O)=O)C2CCC1C(F)C(NC(c1c(Br)nnn1C)=O)C2 N1(C(COC)=O)CCCC(C(=O)N(C)CCN)C1.C(=O)(C(C(C)C)OCC)CCC#C C1(Cl)(C(=O)NCC(C)(C)CNC(C2CN(CC(F)(F)F)C2)=O)CC12CCOCC2 N1(C(c2c(C)oc(C(C)(C)C)c2)=O)C2CCC1CC(NC(c1n[nH]cc1Cl)=O)C2 C#CCC(C)C(=O)NCCc1ccc(NC(c2cscc2C)=O)cc1 Cc1ccc(-n2ncc(-c3nc(CP(C)(C)=O)no3)c2C)cc1 N1(C(C=Cc2c(C)ccs2)=O)CCN(C(C2CCCN2C)=O)CC2(CC2)C1 c1(C(N2CC(NC(CC(C)F)=O)C3(C2)CC3)=O)cc(F)cc(N)c1F C1(NC(c2n(C=C)nnc2)=O)CN(C(c2cnoc2CC)=O)C2CCCC12 C1(NC(c2c(CC)non2)=O)C(C)CCN(C(=O)Cc2ccc(C)nc2Cl)C1C C1(C(N(C2(C(=O)NC3CCC(C)C3)CCC2)C2CC2)=O)CCN(C)C1=O C1(NC(=O)C(=Cc2cccnc2)F)CC(O)CN(C(c2c[nH]nc2Br)=O)C1 c1(C(=O)NC2C(NC(C(C)OC)=O)CCCC2)cc(F)c(Cl)cc1Cl c1(C(N2CCN(C(C3(CC)COC3)=O)C(C(C)C)C2)=O)cccc([N+](=O)[O-])c1Br c1(OC)cc(CC(=O)NCC2(C)CN(C(c3ccccc3)C)CCO2)cc(Cl)c1 C(C(C)(CO)NC(=O)C(C)CC1CCC1)NC(COCCCN(C)C)=O C(=O)(C(O)C(F)F)NC(C1CCN(C(c2cccc(N)n2)=O)C1)(C)C Cc1ccnc2c(N3CCN(CCOC(=O)CCCc4ccsc4)CC3)cnn12 C12(C(N(CCCCCC)C)=O)C(NC(c3ccccc3OC)=O)C3CC1C2C3 C1(CC(=O)NC2(C(=O)OC)CCCC2)CCC2(CN(CCCC(=O)O)C2)O1 c1(CC)nnc2n1CCN(c1ccncc1C(=O)N(S(C)(=O)=O)C)C2.C1CO1 c1(C(=O)O)cc(=NCc2cccc(Br)c2OC(F)F)[nH]c(Cl)n1 c1(C(N2CCC(NC(c3c(CC)n(C)nc3)=O)CC2)=O)c(F)ccc(Br)c1C c1(NC(C(CCC=C)NC(C2CC(=O)N(OC)C2)=O)=O)cc(C#N)ccc1C C1(CCC)CN(C(C2(COC)CNC(=O)C2)=O)CCN1C(=O)CCS(N)(=O)=O c1(C(=O)NC2CCCC2NC(C2CC(n3ccnn3)C2)=O)coc2c1COC2 C1(F)(CNC(C(CCOC)C)=O)CCCN(C(=O)COC2CCCCC2)C1 CC1CC(NC(c2cnn(CC(F)(F)F)c2)=O)CN(C(C2(n3cnnn3)CC2)=O)C1 Cc1cn2c(n1)C(C(=O)N1CCCC(O)(CNC(=O)CSC3CC3)C1)CCC2 C1(C(=O)NCC2C(C)C2C)CC2CC1CN(C(=O)C#CC1CCC1)C2 C1(C(=O)Nc2c(C)noc2)CCC(C2CC2)N1C(=O)CC1CSCCO1 N1(C(C(C)=CCC)=O)CCCC(CC(=O)NCCCC(F)(F)F)CC1 Cc1noc(C2C(C(=O)NC3CCC3CNC(c3ccsc3)=O)C2(C)C)n1 C(=O)(C1COc2ccc(F)cc21)NCC1(O)CN(C(Cc2nc(=N)[nH][nH]2)=O)C1 c1(CCOC)n[nH]c(=NCCCC(C)NC(=O)C(c2cccc(Cl)c2)C)s1 c1(C(=O)NC2C(CNC(c3cc(-n4cnnc4)ccn3)=O)C2)ccc(F)cc1O N1(C(CNC(=O)COC2CCOCC2)=O)CC(C)(COCCSC)CC1(C)C CC1CN(C(c2cn(C(F)F)nc2C2CC2)=O)CCN1C(=O)CN(NC)CC1CC1 C12(NC(c3c(C)con3)=O)CCCC1N(C(c1cc(Cl)sc1Cl)=O)CC2 CC(C)CC(C(=O)NCCc1ccon1)ONC(C1(C)CC=CCC1)=O N1(C(CCN(C)CC)=O)CC(NC(c2ccc(N3CCCC3=O)cc2)=O)CC1C C(=O)(C(C(=O)N1CCC(C(=O)N(C)CC2CCCC2(C)C)(CC)C1)OC)OCC N1(C(c2c(CC)cc[nH]2)=O)CCOC(C)(CC)C1 c1(C(=O)OC)ccc(CC(=O)NCC2CN(Cc3n[nH]cc3Cl)C2)cc1 C1(OC)CN(C(=O)Cc2cn[nH]c2)CC1NC(c1c(C2CC2)cnn1C)=O Cc1cccc(C(=O)NCCC(=O)NCCC(O)C2CC2)c1 N1(C(CCc2ncn(C)c2)=O)CC=C(C(=O)NC2CC(O)C2(C)C)C1 C(=O)(CCS(N)(=O)=O)NCC(CC)N(C(=O)C=CSC)C N1(C(C(C(C)C)SCC)=O)CC(CO)C2(C1)CN(C(c1nn(C)c(C)c1Cl)=O)C2 C#Cc1cn(C)nc1C(=O)NC1CCN(C(C2(SC)CCOCC2)=O)CC1 C1(CCNC(C(C)NC(COC)=O)=O)CCCCN1C(c1cc(C)c[nH]1)=O C(=O)(C(F)(F)C(C)(C)O)NC1CC(C)CN(C(c2ccnn2C2CC2)=O)C1 Cc1ccc(C(=O)NCCC2C(=O)N3CCC(C3)O2)c(C)n1.C(CN(C)C)OC C1(CNC(C2(c3c(C)ccc(C)c3)CC2)=O)CC2COCC2N1C(=O)CCF c1(SC)nc(Cl)cc(=NC2CCC(NC(=O)CCCC3CCCC(=O)N3)CC2)[nH]1 C1(C(=O)NC(CC#C)C(=O)N2CC3C(C(=O)NC)C3C2)CC2(CCCO2)C1 N1(C(c2cccc(SC)c2)=O)CC2CCC(C1)N2C(c1ccnc(F)c1)=O Cc1cc(C#N)ccc1C(N1CC(C)(CNC(=O)CCCCN(C)C)C1)=O CC(C)(F)C(C)(F)C(=O)N1CC(NC(C23CC(CC(F)F)(C2)C3)=O)CC(O)C1 c1(OC)ccccc1CCC(=O)NC1CN(C(=O)CCc2cn[nH]c2)CC1C N1(C(C2C(CC)CCCC2)=O)C(C(=O)N(CCCO)C2CCC2)C2CCCC12 c1(CCCCC(=O)NC2C(C=C)COC2)cc(OC)c(OC)cc1OC c1(C(=O)NC(C(C)NC(c2cc(F)c[nH]2)=O)CO)cc2c(s1)CN(C)CC2 N1(C(C(=O)NC(C)C)=O)CC2(CCC2NC(=O)C(O)Cc2ccc(F)cc2)C1 C[Si](C)(C)c1cccc(-c2ccc(CNCc3cc(Br)c[nH]3)cc2)c1 c1(C(=O)NC(C)CC(C)NC(c2scnc2Cl)=O)cncc(Cl)c1 c1(C(=O)NCC(CC)(CC)NC(=O)CCc2cnoc2)sc2ncccc2c1N N1(C(c2ccc(CCC)s2)C(=O)NCCOC)CCC(P(C)(C)=O)C1 C(N=c1[nH]c(Cl)ncc1F)c1ccc(CNC(C(C(C)C)F)=O)cc1 C1(CNC(c2cc(OCC)n[nH]2)=O)CCCN(C(=O)C(=Cc2c[nH]cn2)F)CC1 c1(CC(N2CC(NC(=O)Cn3cc(CO)nn3)C(F)C2)=O)ccc2c(c1)CCO2 C(=O)(CC(C)(C)CC(F)F)NC(C1(O)CCN(C(C2CC2C(C)(F)F)=O)CC1)C c1(C(=O)NC(CNC(C(C)c2ncco2)=O)C)sccc1Cl C(=O)(C(CCOCC)NC(=O)CCn1ccnc1)N1CC(C#C)C1 C1(C(=O)NCC2CCCS2)CCN(C(=O)CCOCC2CC2)C1 C1(C(N2CCCC(C(C)(C)NC(c3ccncc3N)=O)C2)=O)CCCC1(C)F Cc1ccc(CCC(=O)N(C(C)CN(C(=O)CC2CCCC2)C)C)s1 N1(C(C(F)=C(C)C)=O)CCC2(CC1)CC(NC(=O)C(F)(F)C(C)O)CCO2 C1(O)(C(=O)NCC(CC)NC(c2c[nH]c(C(F)(F)F)c2)=O)CCCC(C)CC1 c1(C(=O)NCCC2N(C(C=CSC)=O)CCC2)ccc(Br)c(C)n1 C(CC(C(=O)OC(C)(C)C)OC(C1(c2cccc(Cl)c2)CCC1)=O)SC C(=O)(C(F)CC(C)C)NCCN(C(c1ccc(C)nc1O)=O)CC N1(C(CC)CC)C(=S)NC(c2cc(C)cs2)C2=C1CCN(C)C2=O C1(NC(N2CCN(C)C(c3cccs3)C2)=O)CCc2nc(N(C)C)sc2C1 CN1CCC(N(C)C(C2CC2(c2ccccc2Br)F)=O)C1=O c1(-c2n(CCN(C)C)nc(C3CC3(C)C)n2)cc2c(C(F)(F)F)nn(C)c2s1 Cc1cc(C(N2CCCC2c2cc(C)oc(=O)c2)=O)c(C)c(C)c1 c1(C(N(C(C)C(N2CCCC2CCCO)=O)CC)=O)ccnc2cc[nH]c12 NS(=O)(=O)c1cc(C(=O)NCC2C=CCN2C(=O)Cc2cc[nH]c(=N)c2)co1 N1(C(c2cnn(CCO)c2)=O)CCCC(CNC(=O)C(F)(F)c2nccs2)CC1 c1(C(N(C2CCC(NC(C3(C)CC4CC4C3)=O)CC2)C)=O)cccc(=S)n1O c1(C(N2CC(C(=O)NC3(C)CCCOC3)OCC2)=O)cc(O)ncc1F C1(NC(COCC=C)=O)CCN(C(C2CCC(F)(F)CC2)=O)CC1CO Cc1nccnc1C(=O)NCC1CCN1C(=O)C(N1CCCCC1)C C(=O)(C1CCCn2nccc21)NCC1(O)CCN(C(c2ccc(C)cc2F)=O)C1 N1(C(C(C)(C)O)=O)CC2CC1CN2C(C1CCCS(=O)(=O)C1)=O C1(NC(CN(c2ncccn2)C)=O)CCCCN(C(c2cccc(F)c2Cl)=O)C1 CC1CCCCC1(CNC(C1CCC2(CC1)N=N2)=O)NC(c1scnc1Cl)=O N1(C(c2cc(OC)nc(Cl)c2)=O)CC2CCN(C(C3C(C)(C)OC3(C)C)=O)C2C1 C[Si](C)(C)C1(CNC(=O)NC2(C(=O)NC3CCCO3)CC2)CC1 C1(CNC(C2N(C(C)=O)CC(O)C2)=O)CCN(C(c2cc(C)cs2)=O)C12CCC2 c1(C(=O)NC23CC(CNC(c4nc(CCC)sc4)=O)(C2)C3)ccc2sncc2c1 c1(C(=O)NCC2C(NC(C=COCC)=O)CCCC2)cc2ccccc2o1 c1(CCC(N2CC(OCCNC(CN(C3CC3)CC)=O)C2)=O)ncc(C)[nH]1 c1(NC2CC(CC(=O)Nc3n(C)nc4c3CCC4)C2)ncnc2c(F)cccc12 c1(C(N2C(CNC(=O)C3CC3)CCC2)=O)cccc(C2(O)COC2)c1 c1(C(=O)NC2C(CC)CN(C(=O)C=C(C)Cl)CC2)cn(C)c2ccccc12 Cc1noc(C)c1C(C)CC(=O)N(C)CCN(C(=O)CCNc1ccccn1)C C1(C(=O)NCC2N(C(c3cc(C)sc3)=O)CCC2)CCCCCS1(=O)=O N1(C(c2c(C)cco2)=O)CCC2(NC(c3cccc(N(C)C)n3)=O)CCCC12 N1(C(c2cc(=N)[nH]cc2)=O)CCC(CNC(c2scnc2Cl)=O)C12CC2 N1(C(CNC(c2c(C)c(C)cc(C)c2C)=O)=O)CCCC2(CC1)CNC(=O)O2 N1(C(c2c(C)cc(=N)[nH]c2)=O)CC(C)CN(C(=O)CC23COCC(C2)C3)C(C)C1 C1(C(=O)NC(C)(CNC(=O)CCC(F)F)C2CC2)CC2CCC1CC2 C(CCS(C)(=O)=O)NC(C1(NC(Cc2cc(C)no2)=O)CCSC1)=O Cc1oc(CO)cc1C(=O)NCC(C)=CC(=O)NCCOC1CC1 C1(CNC(CCCOCC=C)=O)C(CC)CCN1C(c1ncncc1N)=O C(CCC)(C(=O)N1CCC(N(C(=O)CN2CC3CC3C2)C)C1)=CCC CN1CCN(C(c2ccc(C(N)=O)[nH]2)=O)CC1CNC(=O)CCC1CC(F)(F)C1 C(CO)(C(F)(F)F)NC(C(CC1CCOCC1)NC(c1cc(=N)[nH][nH]1)=O)=O C1(N(C(c2c(CC)ocn2)=O)C)CCCN(C(=O)Cc2ccccc2O)CC1 C(=O)(CC(F)(F)C(F)F)NC(CC(C)NC(C=CCC)=O)C C1(NC(C(C)C2CCCO2)=O)CCC(N(C)C(C2C=CCCC2)=O)CC1 N(C1CCCn2ncnc21)C(c1cc(CNC(C2SCCS2)=O)cs1)=O c1(C(=O)NC2CCN(C(=O)CCC3CCCO3)CC2O)ccc2[nH]nc(O)c2c1 CC(CC(F)(F)F)NC(=O)CCC1CC(NC(C2CCCS2)=O)C1 Cc1[nH]c(=N)nc(N2CCCC(C)(C(=O)NCC3CCCC3)C2)c1C Cc1ncncc1C(N1CCN(CCN(C)C(C2(Cl)CC23CCC3)=O)CC1)=O c1(C(=O)NC2CN(C(COC)=O)C(C)C2)cc(S(=O)(=O)N2CCOCC2)ccc1O C1(=CC(=O)NC2CCC2NC(c2ccc3c(c2)OCC3)=O)CCCCCC1(F)F c1(CC(=O)NCCC(C)NC(CCSCC)=O)ccc(C(=O)OC)cc1Cl c1(CC(=O)N(C)CC2CCN(C(c3n(CCC)ccc3)=O)C2)ccc(Cl)nc1 C(=O)(C(O)C1=CCCCC1)NCC1N(C(C(C=C)(F)F)=O)C2C(C1)C2 c1(COC)nc(C(=O)OC(c2cnn(Cc3ccccc3)c2)=O)n[nH]1 N1(C(C2(OC)CCOC2)=O)CC2(C1)CN(C(c1ccoc1C)=O)C2 N1(C(c2cn(CCC)nn2)=O)CC(CNC(c2cncn2C)=O)CCC1C C(=O)(C1=CCCOCC1)N1C(C(C)NC(c2ccn(C(C)C)n2)=O)CCC1 C(C)(C(C)C(=O)N1CCN(C(C)C)CC1)NC(c1cnc(CC)s1)=O S(=O)(=O)(CCCN=c1[nH]c2c(c(=NCC(C)S(C)=O)[nH]1)COC2)NC C1(C(=O)NC2CC(CCNC(c3cc(C)n(C(F)F)n3)=O)C2)CC(S(N)(=O)=O)C1 c1(C(=O)NCCC(C(C)C)NC(=O)CCCC(N)=O)cc(F)cc2ccncc12 N1(C(c2c(C)nc(C)s2)=O)CCC2CN(C(=O)CC(F)(F)F)CC2C1 c1(C(N2C(C)CC(NC(c3c[nH]c(Br)c3)=O)CC2)=O)cnn2cccc(Cl)c12 c1(CN(C(CCN(C(c2nc(C)oc2)=O)C)=O)C)cccc(O)n1 C1(C(N(C)CC2CCN(C(=O)COc3ccon3)C2)=O)CN(C)C(=O)N1 N1(C(c2ccn(CCC)c2)C(=O)NCC=C)C2CCC1C(C)C(O)C2 N1(c2snc(SC)n2)C2CCC1CC(NC(=O)COC1CCCC(C)C1)C2 C12=CC(=NCCC(=O)N1)NC=N2.C(CN(C)C)(C1CC1)OC C(=O)(C1=CCCN(Cc2cc(F)c(O)c(F)c2)C1)NCc1c(Br)ccc(OC)c1 C1(C)(C(N(CC=C)C)=O)C=CCN1C(c1cnc(C2CC2)o1)=O c1(OCC)ccc(C)cc1NC(C1CC1NCc1nccn1C)=O CC1CCCN(C(=O)C(=O)NC2(C)CCN(C(=O)Cc3cc[nH]n3)C2)C1 CC(C#N)CN=c1nc2sccc2c(NCC2(C)CC2(F)F)[nH]1 C(=O)(C#CC1(C)CCCO1)N1C(CC(=O)NC2C(N(C)C)CCC2)C2CCCC21 c1(OC)cccc(-c2ccnc(N3CCN(C(=O)C=CCBr)CC3)c2)c1 C1(C(N2CCC(CNC(CCCc3c(C)ccs3)=O)C2)=O)(CF)CCOCC1 C1(C(F)(F)F)(CNC(CCC2(C(=O)OC)CC2(F)F)=O)CCC(=O)N1 N1(C(C(CC)O)=O)CCc2sccc2C1CNC(c1ccc[n+]([O-])c1)=O c1(C(N2C(CNC(C(C(CC)O)C)=O)C3CCC2C3)=O)ccnc2[nH]cnc12 CCCC(O)CC(=O)NC1CCN(C(=O)C2CC2)CC1C(=O)NCC c1(SC)cccc(C(=O)NCCC(C)NC(=O)C2=CCC2C)c1[N+](=O)[O-] Cc1cccc2c(C(=O)NCC3C(C)(C)C3(F)F)c[nH]c12 N1(C(C)=O)CC(O)CC1C(=O)NC(C1C=CCS1)=O.c12ncoc1CCN2 c1(C(=O)NCC2(O)CN(C(=O)C=C(Cl)Cl)C2)coc2c1CS(=O)(=O)C2 c1(OC(CC)CNC(=O)NCc2cccc(OCC#N)c2)ccccc1C c1(C(N2C(CNC(c3csnc3C3CC3)=O)CC(OC)C2)=O)ccc(C)cc1C C1(C2CC2)(CNC(C(CC)(C)O)=O)CCN(C(c2cnc(O)nc2O)=O)C1 N1(C(Cn2c(C)ncc2)=O)CCN2CCN(C(c3cc(C(F)F)no3)=O)CC2C1 N1(C(c2c(OC)ccs2)=O)CCN(C(=O)CC(C)(C)C2CC2)CCC1C C12(C(N3CCC(NC(C(C)CC(F)F)=O)C(F)C3)=O)CC3CC(C1)CC(C)(C3)C2 C(=O)(C(C)C(C)(F)F)N1CCCC(C(=O)NCCN2CCC(C)CC2)C1 c1(C(N(CCC(=O)NCCc2cc[nH]n2)CC=C)=O)cncc(OC)n1 c1(C(=O)NC2C(OC)CN(C(C3CC(SC)C3)=O)C2)cnc(O)c2cccnc12 CCCC(CC(C)C)C(=O)N(C1CCC(CNC(=O)C(C)OC)CC1)C CN1CCC(CC(=O)NCC2(C(N3CC4C=CC4C3)=O)CC2)CC1 N1(C(CCN(C)C(C2CCC(N=[N+]=[N-])C2)=O)=O)CCC2(CCOC2)CC1 C1(CNC(c2cn(CCC)nc2C)=O)CC(N=c2[nH]c3c(C)c(C)ccc3s2)C1 C1(O)(CCNC(COCCCCC)=O)CCN(C(=O)C(C)(F)CC)C1 C1(CC(=O)NC2CCC(F)C2)CC2(C1)CN(C(C1CC1c1ccccc1)=O)C2 C(CS(=O)(=O)CC(=O)NCCC1(C(=O)NC(C)Cc2cccn2C)CC1)OC C(=O)(CCCCCCC(=O)O)NC1CC(N(C)C(C)=O)C12CCCC2 C(=O)(C(C)(C=C)CCOC)NCCCC(C)NC(C(C=C)(C)C)=O Cn1cc(C(=O)NCC2CC(F)CN2C(c2csnn2)=O)c2cc(F)ccc12 N1(C(C2CCN(CC)C2)=O)CC(N(C(c2nc(Cl)c(CC)[nH]2)=O)CC)C(O)C1 C(=O)(CC(C(C)(C)C)NC(C1CC1(Cl)Cl)=O)NC(C(=O)OC)C N1(C(CCC(CC)C)=O)Cc2ccc(CNC(=O)C(C)N(C)C(C)=O)cc2C1 c1(OC)cc(C(N2CCC3CCN(C(C4CC4F)=O)CC23)=O)c(C)cc1[N+](=O)[O-] C1(C(=O)NC(CNC(CN(C)CC)=O)(C)CC)CCc2nc(O)[nH]c2C1 CC1(CNC(=O)C(O)Cc2cnc[nH]2)CCCC1NC(c1cccs1)=O C1(CC(N2CC(C)C(NC(C3CC(C4CC4)C3)=O)C2)=O)CCCCC1(F)F N1(C(c2cccc(CC)n2)=O)CC2CCC(N(C)C(c3ccnnc3O)=O)C2C1 c1(CN(C(F)(F)C(F)(F)F)CC(=O)NCCNC(=O)COCC)cccc(C)c1 N1(C(C=Cc2c(C)ccnc2)=O)CC2(CC2)n2nccc21 C(=O)(CC1=C(C)NS(=O)(=O)N=C1C)N1CC(C)CC(NC(C(COCC)C)=O)C1 CCC(O)C(C)(C)C(=O)N1CCC(CO)(NC(c2ccc(O)c(C(N)=O)c2)=O)C1 c1(C(C)(C)C)cccc(C(=O)NCC23CC(NC(=O)CS(C)(=O)=O)(C2)C3)n1 c1(C(n2cc(C3CCCCN3C(=O)C(N)=O)nn2)C)ccc(F)cc1 CCC(C)(F)C(=O)NC1CC(CNC(=O)COCc2cc(C)no2)C1 N1(C(C=NOC)=O)CC(NC(=O)CSCc2ccncc2)CCC1C c1(C(CCC)C)n[nH]c(=NC(=O)N(C2CCCCC2)c2ccccc2)s1 CN1CC2C(C(N3CCC(C4CCCN4C(=O)Cc4cccnc4)CC3)=O)C2C1 C1(C(C(=O)NCC(=C)C)N(C(C)C)CC)CCCC1(C)C Cc1n[nH]c(=NCCC(C)(C)NC(C2CC(OC(F)(F)F)C2)=O)s1 CC(C(C)(C)NC(C1CC1c1ccn(C)c1)=O)NC(=O)Cc1c[nH]nc1O N1(C(C=CCCC)=O)CCC(CC(=O)N(C)C(C2(C)CC2)C)CC1 CC#CCCCC(=O)NCC(CNC(c1ccccc1SCC(N)=O)=O)OC CP1(=O)CCN(CC(N2CC3(C2)CN(C(c2ncccc2Cl)=O)C3)=O)CC1 c1(C(=O)NCC(CC)(C)NC(=O)CCC2CCCN2C)cnn2c1CCC2 c1(CC(=O)N(CC(C)O)CCNC(C(CC2CC2)OC)=O)cc(C)sc1C CC1=C(C(=O)N(CCCNc2ccc(Cl)c(OC(F)(F)F)c2)CCO)CCC1 C1(NC(C(CCOC)C)=O)CCCC2CN(c3cc(C#N)nc(C)n3)CC12 C(c1cccc(OC)c1OC(F)F)=CC(N1CCC(CNC(C(CC)C)=O)C1)=O N1(C(CCC)C)Cc2ccc(NC(=O)N(C)CC3CCC(=O)N3)cc2C1 c1(NC(c2c(-c3ccc(N(CC)CC)cc3)csc2)=O)c(F)c(F)cc(F)c1F C1(C)CCC(F)(F)CC1.c1(SCC)nnc(S)s1.C12CCCN1C2 N1(C(c2c(Cl)cn(CC)n2)=O)CCC2C(CCN2C(=O)C(C)=C(C)C)C1 c1(N(C(C)(C)C)C(c2sccc2C)C)ccc(OCC(=O)N(C)C)cc1[N+](=O)[O-] C1(NC(C2=CCN(C(C(CC=C)(C)O)=O)C2)=O)C2CCC(C2)C1(C)C c1(N2C(NC(=O)OC(C)(C)C)CC3(C2)CC3(F)F)c(N=[N+]=[N-])cnnc1O c1(CC(=O)NCCN(C(C=Cc2occ(C)n2)=O)C2CC2)ccc2ncsc2c1 CS(=O)(=O)c1ccccc1C(N1CC2CC1C2C(=O)Nc1cc(O)ccn1)=O CC(C)(C#N)CCC(=O)NCC1CC(NC(C2CCCCN2C(N)=O)=O)C1 Cn1cnc2nc(N3CCC(c4nncs4)CC3)[nH]c(=NC3CCOCC3F)c12 Cc1cc(C)c([N+](=O)[O-])cc1C(C(=O)NC1CCOC1)N(C)Cc1ccsc1Cl c1(OCC(=O)NC(CNC(CCC(C)Cl)=O)C2CC2)ccccc1C#N c1(C(=O)NCCC2(NC(C3=C(C)OCC3)=O)CCC2)ccc(S(N)(=O)=O)cc1 C1(NC(c2c(C)nncc2)=O)(CO)CCCN(C(C2(C#N)CCOC2)=O)C1 C=CCC(CC(=O)NCC(C)CC(=O)OC)NC(C1(CCC)CC(=O)C1)=O c1(C(C(=O)NC(C2(O)CN(C(C(C(C)C)CO)=O)C2)C)C)cc2ccccc2o1 c1(N(CC(CC)(C)OC)C)nc(=NCC(C(C)C)OCC)[nH]c2cc[nH]c12 c1(OCC(=O)NC2C(NC(C(C)c3cccs3)=O)C2)ccccc1C(F)F c1(NC(C2(C)C(C(=O)OC3CN(C(CC)=O)C3)CC2)=O)c(C)noc1C1CC1 C12(C(=O)NC)COCC1CN(C(=O)CN(C)C(=O)C1CC1)C2.C1CCN1 c1(C(=O)NCC(CC(=O)NCCn2c(C)cc(C)n2)O)cc2n(n1)CCC2 c1(C(C(=O)Nc2ccc(Cl)cc2)N(C)C)n[nH]c2c(F)cccc12 S(=O)(=O)(c1ccccc1Br)NC1CC(NS(CC)(=O)=O)C1 c1(-c2cn(C(C)C(=O)NCC3CN(C)C(=O)O3)nn2)ccc2cc(Br)ccc2c1 CC(C)C(C)(O)C(=O)NC(CNC(c1cc(-c2cccs2)on1)=O)CO c1(C(=O)NC2CC3CN(C(C(C)OC)=O)CC2C3)coc2cc(C(C)C)ccc12 C1(C(N2CC(C)C(CNC(=O)CCn3cccc3)C2)=O)CC2CCC1CC2 N1(CC)CCOCC1C(=O)NCCC(C)N(C)C(c1cnn[nH]1)=O CC1CC2(CC(NC(C3C=CCN3C(C3CC4(CCC4)CO3)=O)=O)C2)C1 Cc1ncc(NC(c2nc(NC(=O)Cc3cccc(Br)c3)cn2C)=O)c(O)n1 c1(C(N2C(CNC(c3c(CC)ncs3)=O)C(C)CC2)=O)cnc2[nH]c(=N)sc2c1 CC1CC2CN(C(C3CCC(C)(C)OC3)=O)CC2N1C(=O)C(F)CC1CCOC1 c1(OC(c2ccco2)=O)ccc(N2CCOC2=O)cc1 N1(C(CCCC(=O)OC)=O)CCC2(C=C(C(=O)NC(C3ON=C(CC)C3)=O)C2)C1 C1(OC)CC(CO)N(C(=O)CC(CNC(=O)CC2CCSC2)C2CCC2)C1 C(CCC(=O)NC(C)CN(C)C(C1CC1(C)C(F)(F)F)=O)OCCC CC1CN(C(=O)Cc2c[nH]nc2O)CCCN1C(C1OC2CCC1CC2)=O c1(NC(CCC=C)C)ncccc1S(=O)(=O)NC(c1cccc(F)c1C)C C1(C(=O)NC2(C(=O)NCCOCCOCF)CC(C)(C)C2)CC2CC1CC2=O N=c1[nH]c(=NCCC2CCC2)[nH]c(=NCCC2CCS(=O)(=O)CC2)[nH]1 C1(C(N(CC(CC)NC(C2CC(O)C2)=O)C)=O)CCCCC1n1cccn1 c1(C(=O)NCCOCCCNC(C2(SCC)CC2)=O)c(C)ccc(F)c1N c1(C(N2C(CNC(C3(COC)CCCO3)=O)CCC2)=O)cc(Cl)c(N)cc1F C1(NC(=O)CCc2cnco2)CC2CC(NC(c3ncnc(O)c3Cl)=O)CC12 N1(C(C(CCCC)O)=O)CCCN(C(=O)Cn2cc(C(F)(F)F)nn2)C(CO)C1 C1(NC(c2nc(Cl)sc2Cl)=O)CC2CC1CN(C(c1coc(CO)c1)=O)C2 N1(C(C2CCCN(C(C)=O)C2C)=O)CC2CCC(C1)C(=O)O2 N#Cc1cnc(NC(=O)Cc2csc(NC(c3ccc(F)nc3)=O)n2)cn1 c1(CC(=O)NC2CC(CNC(C3(C(N)=O)CC3)=O)C(O)C2)nc2ccccc2o1 C(=O)(C(O)CC(C)C)NC(CC#C)C(=O)NCc1sccc1C Cc1ncc(C(N2CC=CC2(C)C(=O)NCCN2CCC(C)(C)C2)=O)n1C Cc1csc(C=CC(=O)NCCC(O)CNC(=O)C(Cc2ccsc2)C2CC2)n1 c1(C(=O)NC2C(NC(CC3N(C)CCC3)=O)COC2)ccn2nccc2n1 N1(C(c2cccc(CC)c2N)=O)CC(C)(C)OCC1CNC(=O)Cn1cnnn1 CCC(O)C(C)C(=O)N1CC(C)C(C)(CNC(=O)CSCc2c(C)noc2C)C1 c1(CC(=O)NCC2C(NC(c3c(CC)cco3)=O)COC2)cccc(O)c1 CC1=NOC2(C1)CC(C(=O)NC1C=CCN(C(=O)CN(c3ccncc3)C)C1)C2 c1(C(=O)OC)nc(NCC(N2CCC(O)CC2)C)cnc1OC c1(C(=O)NC2C(CNC(C=C(CC)CC)=O)CC2)cc(S(N)(=O)=O)c(C)cc1C C1(CCCC)(C(=O)NCC(C)(C)NC(=O)CSCC(=O)OC)CCCC1 c1(N(CCC(=O)O)C(=O)NC(c2ccc(OC)nc2)C)nc(OC)cc(C)n1 c1(C(=O)NC2C(CC)CN(C(c3ccoc3C)=O)CC2)ccc(C)c(F)c1N N1(C(COCc2nc(C)on2)=O)CC(CNC(=O)COCCF)C(O)C1 N1(C(c2ncc(C)nc2)=O)CC2(CNC(c3c[nH]nc3C)=O)CC1CCO2 C(=O)(C(CO)C(C)C)N1C(CN(C(c2ccc(OC)cc2)=O)C)CCC1 N1(C(C(Cc2cn[nH]c2)NC(C2C=CC=CC=C2)=O)=O)CCC(C2CCCC2)C1 c1(C(N2C(CNC(=O)CC3CC3(Cl)Cl)C=CC2)=O)ccc(CN2CCCC2)cc1F C(=O)(CC1=CCN(C(C2(Cl)CC2C(C)=O)=O)CC1)NCC(CC(=O)OC)O Cc1nccc(C(=O)NC2CN(C(c3n[nH]c4c3CCC4)=O)C2)c1C c1(C(=O)OC)ccc(Br)cc1NC(=O)NC1(CC(C)C)CCC1 c1(C(=O)NCCC2N(C(C3CC(=O)NC3)=O)CCC2)cc2c(cn1)COCC2 C1(C(=O)NCC2CCCN(C(COCCCCC)=O)C2)CC2(C1)CC1(CC1)C2 Cc1c(C(=O)NCC2CCCN(C(=O)CCOCC3CCCO3)C2)ncn1C c1(C(=O)NC2CCN(C(=O)Cc3sc(O)nc3O)C2)cc(F)c(C(F)F)c(F)c1 C1(CNC(c2c(COC)cc[nH]2)=O)COCCN1C(=O)CCC1C(=O)NN=C1C C1(N(C)C(C2CCCN2C(=O)C(F)C2CCC2)=O)CCCCCC1.C(C(C)(C)C)N C12(NC(c3c(C)ncnc3)=O)CC(CNC(=O)C(c3ccccc3)C)(C1)OC2C C1(C(N(C(CC#C)C)C)=O)C2CCC(C2)C1NC(c1cnsn1)=O C1(COC)(NC(=O)C2=NOCC2)CCN(C(C2(C)COC2)=O)C1 c1(C(N2CC(CNC(CCSC)=O)C3C2C3)=O)cc(Cl)c2c(c1)OCO2 C1(COCC(=O)N(CC(CN(C(C2(CC(C)C)CC2)=O)C)O)C)CCCCO1 CCC(CC(C)C)C(=O)NC(C)(C)CN(C)C(c1cnnn1CC)=O C(=O)(CC(C)C(=O)c1ccccc1)N1CC(CN(c2ccc(C)s2)CCOC)C1 C1(CNC(c2nc(C(C)C)sc2)=O)CCC12CCN(C(=O)C(F)(F)C(C)O)CC2 C(=O)(C1=C(C2CC2C)N(C)C(=O)N(C)C1c1cc(C)cc(O)c1)OCC CCC(C(=O)NCC1C2CCC(C2)N1C(c1cc(C)cc(N)c1)=O)C(F)(F)F c1(C(N(C(C)CN(C(=O)Cc2ccc(CO)cc2)C)C)=O)cn(C)c(=O)nc1O C1(CNC(=O)C=CC2CCOC2)(CO)CCN(C(c2ccc(O)nc2)=O)C1 N1(C(CCN(C(=O)CN2CCCC2=O)CC)=O)CCC(C)(C2CC2)C1 C1(CC(=O)N(C)CC2CCN(C(C3(C(F)F)CC(O)C3)=O)C2)CN2CCN1CC2 c1(N2CCC(CN(C(c3c(CC)nn[nH]3)=O)C)C2)ccc([N+](=O)[O-])c(OC)c1 C#Cc1cnc(NC(=O)NCC2N(C(=O)OC(C)(C)C)CCOC2(C)C)c(C)c1 Cc1sc2ccccc2c1C(N1CCC(C(C)NC(=O)CN(C)CCO)C1)=O CC1CN(C(=O)C(Cc2cc[nH]n2)NC(c2cc(Cl)ns2)=O)CCC1CO CCN=C(NCCCN(C)CC)NCC1CN(Cc2ccccc2)C(=O)O1 CC1(CNC(=O)C2=CCCO2)CCN(C(c2ccnc(C3CC3)n2)=O)C1 S(=O)(=O)(c1ccccc1S(=O)(=O)N1CC(c2ccc(C#N)nc2)C1)NC N1(C(COC(C)=O)=O)CCCC(C)(C(=O)NCC23CCCC2CCC3)C1 CCC(CCCO)NC(=O)C(N1CCCCC1COCC(C)(C)C)=O N1(C(CCC(=O)NCCC)=O)C2CCC1CN(C(C1CC(=O)N(C3CC3)C1)=O)C2 Cc1nc2ncccc2cc1C(=O)NCC1CC2CN(C(=O)CS(N)(=O)=O)CC12 c1(C(=O)OC)ccc(C(=O)NCC2(O)CC(NC(C3(C#N)CCCO3)=O)C2)cc1 C12(CC(=O)NC(C(C)C)C(C)NC(=O)C(=O)NCC(F)F)CCC(CC1)CC2 c1(C(=O)NCC2(C(=O)NCc3snc(C)n3)CC2)c(C)cncc1C N1(C(C(c2ccnn2C)NC(CCCNC(=O)OC)=O)=O)CCCCCCC1C CCCCC(C(=O)NCC(C)C(=O)NC1CC1)NC(c1ccc(C)cc1)=O c1(C(N2CC(NC(CCCC#C)=O)C2)=O)c[nH]c2cc(OC)c(OC)cc2c1=O CC(CCCc1ccccc1)C(=O)N1CCCC(C)(NC(c2cc(F)cs2)=O)C1 C(c1cnccn1)=CC(=O)OCC(c1nnc(C)s1)=O c1(NC(CC2(O)CCN(C(c3nc(C)oc3)=O)CC2)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NC2CCCN(C(C3CC(OC)C3)=O)C2C)cnn2cc[nH]c(=O)c12 N1(C(c2cc(CNC(C3C(=O)NCC3)=O)sc2)=O)CC2C=CC1CC2 C1(CCCNC(C=C(CC)C)=O)CCCN1C(C1CC1c1ccncc1)=O Cc1ccn2ncc(C(=O)NCC3CCCCC3NC(c3ccn(C)c3)=O)c2c1 CC(C)(O)C(F)CNC(=O)CC1(C)CCN1C(C1CC=CCO1)=O N1(C(CCC2CC(NC(c3ccc(=N)[nH]c3)=O)C2)=O)CCC2CCC(C1)S2 C1(CNC(c2c(C)ccs2)=O)CN(C(=O)CNC(C2CCC2)=O)C2CC12 c1(C(N2CC(NC(=O)Cc3c[nH]nc3O)C(CO)CC2)=O)cc(F)c(F)cc1F N1(C(C(C(C)C)F)=O)CC(C)(C)CC1CC(=O)Nc1cccc(C(N)=O)c1 N1(C(C2(C)CC(=C)C2)=O)CC2(CCC2NC(=O)C(C2CCCCC2)O)C1 C=C(F)C1(CC(=O)NCC(C)N(C)C(c2ccc(CC)cn2)=O)CCC1 c1(NC(c2ccc(O)cc2)=O)ccc(NC(c2cc(Br)c[nH]2)=O)nc1 C1(C(=O)NCC(C(C)C)NC(c2c[nH]c(=NCC)s2)=O)CCc2cncn2C1 CC1=CC(C)CN(C(=O)CC(CC2CC2)NC(=O)Cn2c(O)nnc2O)C1 c1(C(=O)NC(C)(CNC(=O)Cc2ccnc(Br)c2)CO)cc2n(n1)CCC2 c1(CC)nc2sc(C)cn2c1C(=O)NC1CC1CNC(C1CC1C#N)=O C1(OC)CN(C(=O)CCC(N)=O)CCC1NC(=O)CC1(CO)CC1 N1(C(C=C(C)c2ccco2)=O)CC2(CCC2)CC1C(=O)NC1CNC(=O)C12CC2 C1(C(N(CCC)CCC)=O)(CNC(=O)CC2C=NN(C)C2=O)CC(F)(F)C1 N1(C(c2c(C(=O)OC)scc2)=O)CCC(C2CCCN(C(=O)CSC3CC3)C2)C1 Cn1ncc(C(=O)N(C2CC2)CC2CCCN(C(c3ccc(COCO)s3)=O)C2)c1N C12(C(N(CCCCCNC(C3CC34CC(O)C4)=O)C)=O)CCC(CC1)C2(C)C C1(C(=O)NCC2(F)CC(CNC(=O)CCF)C2)CN2CCN1CC2 N1(C(C2C(C)C2)=O)CCC(N(C(=O)CNS(N)(=O)=O)CC2CC2)CC1 C1(NC(c2ccc(C)s2)=O)CC2CCC1(NC(=O)CCc1ccc(C)c(Cl)c1)C2 C=CC(CC)CC(=O)N1CCC(C)C(CNC(C23CC4CC2C3C4)=O)C1 Cc1nc(CC(N2C(C(=O)Nc3ccccc3Br)CC3CC23)=O)c(C)s1 c1(C(=O)NC(CNC(c2cccc(SCC#C)c2)=O)C)cccc(=O)n1C CCC(C(=O)N1CCC(NC(c2cn(C(C)(C)C)nn2)=O)C(F)C1)C(C)C c1(C(CC)C)nc(N2CC3(CN(C(c4cc5sccc5[nH]4)=O)C3)C2)cc(C)n1 N1(C(CC2(C)CCN(C(c3c(C)cnn3C)=O)C2)=O)CCCC(C)C1CO CC(CS(C)=O)C(=O)N1CC2CC1(CNC(=O)CCSCc1ccccc1)C2 c1(C(=O)NC2C(NC(C3(C)CNC(=O)C3)=O)C2)cc([N+](=O)[O-])c(Cl)cc1Cl Cc1c(C)c(C)c(C(=O)NC2CCCC(NC(C3CC3C)=O)C2)c(C)c1C N1(C(C2(CC=C)CC2)=O)CCC(N(C(=O)C=CCn2cncn2)CCO)CC1 C1(CNC(C=CSC)=O)CCCC(CNC(=O)C(C)n2ccnn2)C1 c1(CC(C)C)ncc(C(=O)NC2CC(NC(C3(OC(C)C)CC(CF)C3)=O)C2)[nH]1 C(CC(F)(F)F)SC.C12CC(F)(C1)NC(=O)CN1CC(C1)N(C)C2=O CC1CN(C(C2OCCCO2)=O)CCCN1C(C1CN(C)CCN(C)C1)=O C(C#CC1CCCCC1)OC(C(CC#C)C1CC1)=O CC(CC(=O)NCCOc1ncccn1)N(C)C(C1CC1(Cl)Cl)=O N1(C(C2CC(SC)C2)=O)CCC2(CC1)CC(NC(c1cn(C3CC3)nc1C)=O)C2 C1(OC)(OC)CCC1C(=O)N(C(C)C(=O)NCCCS(C)=O)C1CC1 C1(NC(c2ccc(Cl)c(-n3nnnc3C3CC3)c2)=O)CCCNC12CCC2 C1(C2CCN(C(C=NOC)=O)C2)CCCN(C(=O)CC2(C)CC2)C1 C1(C)(C(N2CCC(CC)C2C)=O)CCCN(C(C2CC3(CSC3)C2)=O)C1 CC(C)C(C)C(=O)NCCC1(CNC(=O)C(C)Oc2cccc(F)c2)CC1 c1(SCC(N2CCC(NC(c3c(C)nns3)=O)C23CC3)=O)nnc2ccccn12 N1(C(CCOCC)=O)CCCC2(CNC(c3cnc4cc[nH]c4c3)=O)CCCC12 Cc1ccc(C(F)F)c(C(=O)NCC(C)N(C)C(C2CCN(C3CC3)C2=O)=O)c1 c1(C(=O)NCC2C(NC(C3N(N=O)CCC3)=O)C2)cnc(C2CC2)nc1O C1(NC(C(CNC(C=Cc2c(C)cccc2)=O)O)=O)CC2(CCCCC2)C1 CC1CCCCC1C(=O)N(C)CC1(O)CN(C(=O)CS(=O)(=O)N(C)C)C1 Cc1nc(C(=O)NCC(C(C)C)NC(C2(O)CC2(C)C)=O)nn1C C(CC(=O)NC(C)C(=O)NC1CC1)N(C(=O)CSCCC#N)C(C)C C=CCCCC(=O)N1CCC(N(CCC)C(c2cnccc2Br)=O)C1 c1(OC)ccc2c(C(=O)NC3(C)CN(C(c4cc(=O)cc[nH]4)=O)C3)ccnc2c1 C(=O)(CC(C(F)(F)F)NC(=O)CC1CCSC1)NCCN(C)CCO C1(C(N2CC(O)(C(C)NC(c3cc(CC)on3)=O)C2)=O)CC(OC)C(OC)C1 c1(OCC)cc(C(=O)NCC2CC2C(=O)N(CC)Cc2cn(C)cn2)[nH]n1 N1(CCC=C)CC2CCN(C(c3ccc(C(C)(C)C)s3)=O)CCC2C1 C(CC(C)(C)C(=O)NC1(CC(=O)NCC2(C)CCCOC2)CC1)OC N1(C(C(C=CC)O)=O)CCC(C(=O)NCC(C)(O)C(C)CC)CC1(C)C C(=O)(CCC(CC)CC)NCC(CCC)NC(=O)C(F)CC1CCOCC1 C1(CC(=O)NC2CCN(C(Cc3cccc(CC)c3)=O)C2C)OCCOC1(C)C CCC(O)C(C)(C)C(=O)NCC1(F)CC(NC(c2cccc(SC)c2)=O)C1 c1(C(N(CCNC(CCn2ncn(C)c2=O)=O)C2CC2)=O)cnc2nccn2c1 N1(C(CCc2onc(C(C)C)n2)=O)CCC(NC(C2CCCC(=O)N2)=O)C(C)C1 N1(C(CCCC)=O)CCC(C(F)CNC(C2(CC)CC(C)(C)C2)=O)CC1 c1(C(=O)NCCN(C(=O)C(C)C(C)C)CC)cncc2n[nH]cc12 C(=O)(CN1C(=O)Cc2ccccc21)NCC(CC=C)NC(C1CC(Cl)(Cl)C1)=O CN1CC2(CC2)CC1C(=O)N(C1CC(C(N2CCC(O)(CO)C2)=O)C1)C c1(OC)ccc(F)c(NC(=O)N(C2CCNCCC2C)c2ccc(F)cc2)c1 c1(NC(C2CCN(Cc3ccc(CO)o3)CC2O)=O)cccc2c(I)n[nH]c12 N1(C(C2(C(C)(C)NCCC#N)CC2)=O)CC(C)C1.CO CC1OCCC1CC(N1CC(C)(NC(CNC(C2CCC2)=O)=O)C1)=O c1(C(c2nnnn2C2CCCCC2)NCCOCCOCC)cnc(C)[nH]1 C#CC1(NC(C23CSCC2C3)=O)CCC(C)(C)CC1 c1(C(N2C(CCN(C(C3C(CC)C3)=O)C)CCCC2)=O)cc2c(=O)[nH]ccn2n1 C1(NC(c2c(C)cnc(F)c2)=O)CN(C(=O)C=CC(N)=O)C2CCCCC12 Cc1nccnc1C(=O)NCCC1CCC(NC(=O)C=Cc2cnc[nH]2)C1 Cc1c(C(=O)NC2CN(C(=O)C=CCOC3CCOCC3)CC2O)nnn1C O(C1CCCc2ccccc21)CC(=O)NC1C(NC(=O)CCc2cnccn2)C1 CC(C)(CF)C(=O)NCCC1CCN(C(c2ncc(C(F)(F)F)s2)=O)C1 C1(C(=O)NCC2(NC(=O)Cc3ccncc3F)CCCCC2)CC2C(C1)C2(F)F c1(C(c2n(CCSC)nnn2)NCCCc2ncccc2C)ccc(Cl)cc1F c1(CNC(CC2OCC(C)(C)OC2)=O)ccc2c(c1)CN(C(=O)C1=CCC1)C2 C12CN(CCO1)C(=O)CNC2=O.c1(C(C)NC(CNC(=O)OCC)=O)cccs1 c1(C(N(C(C)CNC(=O)C(C)(O)C2CCOCC2)C)=O)noc2cc(Cl)ccc12 C(=O)(CCC(=O)c1cccnc1)NCC(CNC(C12CC(C(=O)OC)(C1)C2)=O)F C=C(C)C(CC(=O)NC1CN(C(c2cnc(C)cn2)=O)CCC1C)OCC Cc1cc([N+](=O)[O-])cnc1C(=O)NC1CCC(NC(=O)C(=O)NCC(F)F)CC1 N1(C(C2N(C(C(CC#C)C3CC3)=O)CC2)=O)CCC2CCCC2C1 C1(CC=C)(NC(=O)CN2CC=CC2)CCN(C(c2cccc(C(C)C)n2)=O)C1 N1(C(C2CSCCN2C(=O)C(F)(F)c2ccccc2)=O)CCC2(CC1)COC2 C1(NC(C2C(OC)CCC2)=O)(CNC(C2CC=C(C)CC2)=O)CC2CCC1CC2 n1(CCCC(=O)NCC(C)(C)NC(c2cnc(CC3CC3)s2)=O)c(O)nnc1O N1(C(C(c2ccc(F)cc2)CC)=O)CCc2cc(C(=O)O)ccc2C1C CCC(C)(C(=O)N1CC(O)(C(C)NC(=O)Cn2ncnn2)C1)OC C(c1ccc(F)c(F)c1)=CC(=O)NC(CCC)CCCNC(=O)C(C)(C)CSC C1(C(=O)NCCOC)CC12CC(NC(=O)COC1(C)CC1)C2 CC1CC(C(=O)N2CCC23CN(C(C2COCCN2C)=O)C3)=NO1 CCC(C(=O)N1CCC(C2CCCCN2C(=O)COCC(C)(C)C)CC1)C(C)C C(=O)(C(CCF)NC(=O)C(C)C1CCC1)NCC(=O)OCCCCC C1(CC(=O)N(C2C(OC)COC2)C)N(C(=O)CNc2ccccn2)CCC1(C)C CON(CCC(=O)N1CCC(C2(O)CC2)CC1)C(=O)c1cc(C)oc1C C(=O)(C(C)CC(C)CC)N1CCC(CNC(CC=CCC)=O)C12CC2 c1(C(N(C)CC2CCN(C(CC(C=C)CC)=O)CC2)=O)cc2occc2n1C N1(C(c2c(C)noc2)=O)CCN(C(=O)CCc2cccnc2Cl)CC1C(C)C C#Cc1ccc(C(N2CCC(CC=C)(NC(=O)CC(CC)OC)CC2)=O)cc1 c1(C(=O)N(C(C(C)O)CO)C2(CC=C(C)C)CC(C[Si](C)(C)C)C2)cccnc1O C(=O)(NNc1c(F)cccc1F)N(C(C1CCC1)C)CC c1(C(=O)NCC(C2CCN(C(C(C)C)=O)CC2)F)cccc(C2CC2)c1Cl c1(C(N2CCC(C(C)(C)NC(C3C(CC)CCC3)=O)CC2)=O)ccc(C)cc1F N1(C(c2ccc(OC)s2)=O)CCC2CCC(NC(=O)CC3CCC4CC4C3)C1C2 N1(C(C(CCC)NC(N)=O)=O)CCOC2(CCC(NC(=O)C(F)(F)CO)CC2)C1 C(=O)(C(O)C(C)(C)C)NC1CCN(C(CC(C)SC)=O)C1 C(=O)(CC(C)C(F)F)NCC(CCNC(CNC(c1nccc(OC)n1)=O)=O)O CC1C(=O)CC1C(=O)NCC1CC(NC(=O)CCC2CCCO2)C1 C1(NC(C(CCF)NC(CCCCN(C)C)=O)=O)C(O)C2CCCC12 C(N=c1nc2c(ncn2C)c(N(C)Cc2ncc[nH]2)[nH]1)c1cc(C)nc(C)c1 N#Cc1cnn2ccc(N(C(=O)CCCC(F)(F)F)C3CC4CCC(C3)N4)nc12 Cc1cc(C(N2CC(CNC(=O)C(c3cscn3)N(C)C)C3(CC3)C2)=O)ccc1F N1(C(C(C)N(CCC)C(c2ccn(C)c2CC)=O)=O)CCCC2CC1C2(C)C N1(C(CCc2onc(C)n2)=O)CCC2CCC12CNC(c1cccnc1N)=O c1(C(C(=O)N(CCC(=O)NCCOCCC=C)C)C)ccnn1C C1(O)(C(=O)NCCCC(C)NC(c2ccc(OC)c(Cl)n2)=O)CCCC(C)CC1 C1(CNC(c2cc(OC)nn2C)=O)CC2COCC2N1C(=O)COC(C)=O CC1CCc2ncc(C(=O)NC3CN(C(c4nccn4C)=O)CC3C3CC3)n2C1 N1(C(CCc2n(CC)ccn2)=O)CCCC(C(C)(O)CNC(=O)COCCF)C1 c1(OC(C)C)cccc(C(=O)NCC(O)CNC(=O)C2=CCCOC2)c1F C(=O)(C1=Cc2ccccc2C1O)NC1C(CNC(c2c(COC)ccs2)=O)CC1 FCCN=C(NCC(N1CCCCC1)C1CCOC1)NCC1CC12CC2 CC(C)(CCCF)C(=O)NC12CCC(NC(=O)CC3CC(F)(F)C3)(CC1)C2 N1(C(c2cc(C)c(C(N)=O)cn2)=O)CC2CN(C(c3ccsc3)=O)CC2(C)C1 C1(C(N2CCC(C(C)NC(C)=O)C2)=O)(NC(C(F)=CCC)=O)CCOCC1 CC(C(=O)NC(C(=O)NCCNC(=O)C1CC1)C1CC1)S(N)(=O)=O c1(C(C)(C)C(=O)NCC2(CCNC(=O)Cc3ccon3)CC2)ccc(Cl)nc1 c1(CC)nc(C)c(C(=O)NC(C2(O)CN(C(c3ccc(CN(C)C)o3)=O)C2)C)s1 C(=O)(C1CCCn2nccc21)N1C(COC)CN(C(c2ccc(O)c(O)c2)=O)CC1 C(CC(C(=O)N(CC(CO)(CO)NC(C12CCCCC1C2)=O)C)NC=O)SC N1(C(c2nc(C3CC3)cs2)=O)CCN(C(C2C=CCC2)=O)C(CF)C1 C1(NC(CCCC2(N3CCCC3)CCC2)=O)C2CC3C(C2)C13.N12CCC(C1)C2=O N1(C(CN(C(C=CCCC)=O)CC)=O)CC(CO)C(O)C1 CC1(C)C2CN(C(=NCCCN3CCCC3)NCc3ccn(C4CCC4)n3)CC12 c1(OC)cc(Br)c(CN2CC3(CC(NC(c4cc5sccc5s4)=O)C3)C2)cc1O N1(S(CC)(=O)=O)CCCC(NC(=NCc2cscn2)NCC(C)(C)N(C)C)C1 C#Cc1c[nH]nc1C(N1CCC(OCC(=O)NCCN(C)C2CC2)C1)=O c1(CC)n[nH]c(=NC2CC(CNC(=O)CC3(O)CCCOC3)C2)s1 c1(N(C(Cc2nc(CC)sc2)=O)CCNC(C2CCN2)=O)cnc(C)nc1 C1(C)(CNC(COCC)=O)CCCC1NC(=O)C(C)NC(=O)OC N1(C(c2cc(C)c(C)s2)=O)CC(C)CN(C(=O)CN2CCC(C)C2)CC1C N1(C(C(C)Oc2ccccn2)=O)CCC(NC(=O)C=CC2CCCC2)CC1 C1(C(=O)NC2CCN(CC)C2=O)CCN(C(=O)C=Cc2cc[nH]c2)C(C)C1 C1(NC(=O)C=C2CCC2)CN(C(=O)COc2ccc(F)cc2)CC1n1ccnn1 N1(C(c2nccc(OC)c2)=O)CCN(C(=O)Cc2ccc(F)cc2)CC1C(C)C C1(C(N2CCN(CC)CC2)=O)C2CC3C(C2NC(c2ccc(C#N)n2C)=O)C13 N12CCC(C3CCN(C3)C1=O)C2.CN1CCS(=O)(=O)CC1CSCCOC(C)(C)C N1(C(c2cccnc2OCC2CC2)=O)CCN(C(C2CC2F)=O)C(C2CC2)C1 c1(CC(=O)NC2(CO)CN(C(Cc3cc(C)on3)=O)C2)ccc(C2CCC2)cc1 O=S(=O)(c1ccncc1Cl)NCc1ccc(-c2cccnc2)cc1 c1(CNC(C(C)N(C)C(c2cccn2C2CC2)=O)=O)ncn(C2CC2)n1 CC(C(=O)NCCCN(C)C(c1cn(C)nc1-c1ccccc1)=O)P(C)(C)=O N1(C(C(C)Oc2ccc(F)cc2)=O)CCN(C(=O)CCCF)C(C)C1 N1(C(c2cc(Cl)no2)=O)CCC2C(CCCN2c2ncncc2Cl)C1 C1(O)(CN(C(c2cc(C)nn2C)=O)C)CCN(C(C2CCCCC2F)=O)CC1 N1(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCC2C(CCCN2C(=O)Cc2ccsc2)C1 C1(C(N2C(C#C)CCC2)=O)CC2CC1CC2NC(c1cnc(C)o1)=O S(=O)(=O)(c1cnc(Cl)nc1)N1CC(C)(C(=O)Nc2c(C(=O)OC)cc(I)cn2)C1 c1(C(=O)NCC2CCN(C(CC(CCCC)O)=O)CC2)c(N)nn2ccccc12 c1(C(=O)NCCN(C(=O)CC2OCCC2C)CCOC)nnn2c1CCCC2 C12CCCCC1CNC2=O.C1(NC(C(C)(C)Cl)=O)CCS(=O)CC1 N1(C(C(F)=CC)=O)CC2(CCN(C(=O)CC(C)C(=O)c3ccc(Cl)cc3)C2)C1 c1(N(C)C)ccc(C(N2CC(C(=O)NC(C3(C)CC3)=O)C3CC23)=O)c(F)c1 Cc1cccc(-n2cc(CN3CCN(C(C4CCC(=O)NC4)=O)CC3)nn2)c1O N1(C(Cn2ccc(C)cc2=O)=O)CCN(C(c2cnc(F)cc2C)=O)CCC1C C1(C(N2CC(C=C)C(NC(=O)C(=O)N(C)C)C2)=O)CCc2ccccc2C1 CC1(C)COC(C(=O)NCC(=O)NC2C=CCCC2)C1 C1(CCCNC(C2(CC=C)CC2)=O)CCCN1Cc1nc(CC(C)C)no1 c1(CC(=O)OC)ccc(NCc2ccnc(F)c2)cn1 N1(C(C2CC(CNC(C=C(C)c3ccco3)=O)C2)=O)CC2CCOC2C1 c1(C(=O)NC2CN(C(c3n(CCCC)ncc3)=O)C(C)C2)c(OC)cccc1C c1(C(=O)NC2CC(NC(c3cc(C)cc(CO)c3)=O)C2)c(Br)cc(F)c(Cl)c1F Cn1nc(C(=O)NCC2CCCCCN2C(C2C3CCCOC23)=O)c(Cl)c1Cl C=CCCC(CC(C)C)C(=O)N(C)CCN(C)C(c1cn(C)nc1Br)=O C#Cc1cccc(C(=O)NCC2CC2NC(=O)C=Cc2ccc(Cl)cc2)c1C N1(C(CCCCSC)=O)CC2CC1CN2C(c1c(Cl)ccnc1C)=O C1(C(N2CCC(N(C(=O)CCc3ccc(Cl)s3)C)C2)=O)CCCC12CCC2 CC1=C(C)CC(C)(C(N2CC(CNC(c3n[nH]cc3[N+](=O)[O-])=O)C(C)C2)=O)CC1 C(=O)(C1=CCCCC1)NCC(N(C(=O)C(C1CCOCC1)O)C)NC(=O)COC C1(N(C(C(C)SC)=O)Cc2ccccc2)CN(C(c2cncn2C)=O)CC1O c1(C(N(CCOCCC(=O)NC(CC#C)C)C)=O)ccnc(O)c1 C1(NC(c2cc(CNC(c3ccc(C(C)=O)[nH]3)=O)[nH]n2)=O)CCC(C)CC1 c1(C(=O)NCC2(O)CCN(C(C(C)(C3CC3)NC(C)=O)=O)C2)cccc(F)c1C N#CC1(C(=O)NCCn2cnc(C(=O)NCc3cc(=O)cc[nH]3)c2)CCOC1 c1(N(C)Cc2cccc(CC)c2)nc(=NCC2(C3CC3)CC2)[nH]c2cccnc12 C1(C(=O)NCC(C)N(C)C(c2c(N)cnn2C)=O)CC2C=CC1C2 C1(c2nnnn2C2CC2)(NCc2c(C)cccc2)CCC(C)(C)CC1C N1(C(CC=C(C)C)=O)CCCC2(NC(=O)CN(C)S(N)(=O)=O)CCCC12 C12(C(N(C)CCc3nccs3)=O)CCN(C(c3cc(Cl)ns3)=O)CCC1C2 C=CCC(CN(C(=O)C(O)CSC)C(c1ccccc1)=O)C(=O)OCCC N1(C(C2CCN(CCC)CC2)=O)CCN(C(=O)C2=CCCC2)C(CO)C1 C1(NC(c2c(CC)ccc(F)c2)=O)CCC2(CCCN2C(c2cocn2)=O)CC1 N1(C(CC(C)CF)=O)CCN(C(=O)C=Cc2c(F)ccc(Cl)c2F)CC2(CC2)C1 Cc1cc(C(F)(F)F)c(C#N)c(N2CCC3C(CCN3C(C3CCC3)=O)C2)n1 CC1(C)CCC(C(N2CCC(C)(CNC(C3(C(F)(F)F)CCC3)=O)C2)=O)OC1 N1(C(CCN(CCCO)C(C2C(CC)CC2)=O)=O)CCC(F)(F)C(C)C1 N1(C(c2nc(C)oc2)=O)CCC2(CCCC2C(N2CCOCC2)=O)C1 C1(C(=O)NCCOCCNC(=O)CCC2CC(F)(F)C2)CCCC2CCCN12 c1(C(N2CCC3(NC(c4ncc(N)nc4)=O)C(C2)C3)=O)cccc2ccnn12 C1(NC(COCCC)=O)CCC(N(C)C(c2cc(C3CCCC3)no2)=O)C1 Cn1c(C(=O)NC(CO)C(=O)NCc2cn[nH]c2)cnc1Cl c1(C(=O)NC2C3CN(C(C(C)(C)C(F)F)=O)CC32)csc2ncnc(O)c12 [N-]=[N+]=Nc1ccc(Cl)cc1NC(c1ccc(OCC(F)(F)F)nc1)=O Cc1nn2cc(CC(N3CCCC(CNC(c4oncc4C)=O)CC3)=O)nc2s1 Cc1ccc(F)c(C(N2CCC(N(c3cnc(O)[nH]3)C)CC2)=O)c1Cl C1(C(C)NC(CSCC(C)=O)=O)CCN(C(=O)Cc2nc(O)n[nH]2)C1 N1(C(C(=O)NCC(F)(F)F)=O)CCCC2(CCN(C(=O)Cc3cscc3F)C2)C1 CCC(CC)CC(=O)NCC1CCC(C)N(C(=O)Cc2ccccc2C)C1 CCCC(CCC)CC(=O)N1CC=C(C(=O)N2CC(O)(C(F)(F)F)C2)C1 C1(OC)CN(C(c2cnoc2C2CCC2)=O)CC1NC(C1CCCC1)=O c1(NC(CCNC(C=Cc2cccc(C)c2)=O)C)ncnc2cc(F)c(F)cc12 c1(CCC(N2CCC(Cc3cn(C4CCC4)nn3)C2)=O)cnc2ccccc2c1 N1(C=O)CCN(C(N2CC(c3cnc(C)[nH]3)C2)=O)CC1.C(C)(C)(C)OC=O c1(C(=O)NCC(=O)NC2CC2CNC(=O)CC2CCC2)cccc(Br)n1 C1(CCC(C)C)CCN(C(C2CCCN2C(=O)COCCO)=O)CC1 CCC(CCC(=O)NC1(C2CN(C(C3CCCCCCC3)=O)C2)CC1)OC CC1(NC(=O)C(F)=C2CCCC2)CCN(C(C2CN(S(N)(=O)=O)C2)=O)CC1 c1(C(N2CCC(F)(CNC(c3coc(Cl)c3)=O)C2)=O)coc2ccc(Cl)cc12 C1(C)(OC)CC(NC(=O)C(F)C2CC(NC(C3(O)CCOCC3)=O)C2)C1(C)C C(C(=O)NCCN(C(=O)C(O)Cc1ccccc1)C1CC1)(C(C)C)SC c1(CC(C(=O)NC2CN(C(c3nc(Cl)cs3)=O)C2)O)ccc(F)cc1 c1(NC(C(CCNC(c2ccccc2C)=O)OC)=O)ccc(SC)cc1N N1(c2cc(NCC3(CCO)CC3)nc(C)n2)CCC2(CCC(C)CC2)C1 C(=O)(CCC(F)(F)F)N1C(C(=O)Nc2n(CC)ncc2)CC(C)C1 N1(C(C(COC)C)=O)CCC(C2CCC2)(CNC(=O)Cc2nnc(S)n2C)CC1 N1(C(C(CCC)O)=O)CCN(C(C2(F)CCOCC2)=O)CC1CC#N C(c1nc(CC2CCOC2)no1)=C(COCC)C(F)F N1(C(c2c(C)snc2)=O)CCOC2(CCCN(C(=O)C(F)C(C)C(F)(F)F)C2)C1 Cc1cc(S(N)(=O)=O)sc1C(=O)NCC=CCNC(=O)CCS(C)(=O)=O CP(C)(=O)CCC(=O)NCCn1cc(CNC(C2CC3CCC2O3)=O)nn1 C1(CC(=O)NCCn2cc(CCS(=O)(=O)N(C)C)nn2)CC(O)C1(C)C N1(C(C2C(CC)C2)=O)CCC(CN2CCN(C(=O)C(C)(C3CC3)OC)CC2)CC1 N1(C(c2c(N)n(CCO)nc2)=O)CCN(C(=O)CC=C(Cl)Cl)C2CCCCC2C1 C1(CN(C(=O)CC2CC3C=CC2C3)CC)CCCCN1C(=O)C(C)c1ccco1 C1(OCC)CC2CN(C(=O)C(CC(C)C)NC(=O)CC3CCC(C)(C)O3)CC12 C1(N(C(C2(CCOC)CC2)=O)C)CCN(C(=O)C=C2CCC(C)C2)CC1 C(C(=O)NCC1=CCCOC1)(C(C)C)NC(CC(C)OC)=O c1(C(=O)NCC(C)NC(C2(COC)CCCCO2)=O)cc(C)ccc1O N1(C(c2c(NC)ccc(F)c2)=O)CCC2CC1CN(C(=O)CCC=C(C)C)C2 C1(NC(C(C)SCC)=O)CCC2(CC1)CN(C(c1ccc(C(C)=O)nn1)=O)C2 c1(C(=O)NCCCCCCNC(C2(C(CC)(F)F)CC2)=O)nnc2n1CCOC2 C1(NC(C2N(C(Cn3ncc(C)c3)=O)CC=CC2)=O)CN(C)CCC1O N1(C(c2nc(CS(C)(=O)=O)cs2)C)CCCOC(CNC(N)=O)C1 S(=O)(=O)(CC(=O)NC(F)F)N(CCOCCOCCNC(CC1CCC(C)C1)=O)C C1(C(N2C3C(NC(=O)CC4CCS(=O)(=O)C4)C(C3)C2)=O)CC12CCOCC2 C=CC1CCCCN1C(=O)COC1CC(NC(c2ccccc2CCOC)=O)C1 C=CC(C)C(C)C(=O)N1CC2(NC(=O)Cn3ccccc3=O)CC1(COC)C2 c1(C(N2CC(COC)N(C(c3nccn3C)=O)CC2)=O)ccc2c(c1)COCO2 C(=O)(CC(O)C(C)(C)C)OC(C(=O)N(S(=O)(=O)c1cccs1)CC)C c1(C(=O)NCC(C)(C)CNC(=O)C(CC(F)F)C2CCC2)ccc(N)cc1F CC(F)(F)CCCC(=O)NCC1CC(NC(c2cccnc2O)=O)CC1O C1(CNC(c2cc(CC(C)C)on2)=O)CN(C(=O)CN(C)C(=O)C2CC2)CCO1 O=C(N=c1ccn(C2CN(Cc3ccc(I)c(F)c3)C2)[nH]1)c1c(F)ccnc1Cl c1(CC(=O)N(C)CC2(NC(c3ccnnc3)=O)CC2)nc(F)c(F)cc1F C1(C(=O)NCC23CC(NC(C4CC4(F)F)=O)(C2)C3)C2Cc3ccc(Br)cc3C12 C1(NC(C(c2ccccc2)OCC)=O)CCN(c2ncc(F)cn2)C12CCC2 N1(CC(COc2ccc(OCC)cc2)O)CC2CCC1C(C(=O)O)C2 CS(=O)(=O)c1cccc(C(N2CC(NC(c3ccnc(Cl)c3)=O)CC(F)C2)=O)c1 N1(C(c2nc(C(C)C)oc2)=O)CC(C2CN(C(C3SC4C=CC3C4)=O)C2)C1 CC(C(=O)N1CCC(O)(CNC(C2CCC3(CCC3)C2)=O)CC1)C1=CCCC1 Cc1nn(CC(C)C)c(C)c1S(=O)(=O)NCC1CCC1O C1(CCS(C)(=O)=O)COCCN1C(=O)Nc1ccc(CO)cc1 C1(C(=O)NC2C(NC(c3ccc(F)c(Cl)c3F)=O)C2)CCc2cc(F)ccc2O1 C1(NC(CCCC#C)=O)CCc2nc(NC(c3cc(F)cc(Cl)c3)=O)sc2C1 c1(C(N(CCOC)CCNC(=O)C(C)CF)=O)cccc(C2CCCOC2)c1 CCC(C)(COC)CNC(C12CC1CCN2C(=O)CNC(C1CC1C)=O)=O C1(NC(C2CCC(F)(F)CO2)=O)CC2(C1)CN(C(=O)C=Cc1cncs1)C2 C1(C(N2CC(SC)C(N(C)C)C2)=O)N(C(=O)CN2CCCCC2)CC12CCCC2 c1(CC(=O)N(CCC(C)NC(=O)Cn2ncnn2)C)csc2ccccc12 C1(C(N(CC(=O)N(C)C)CC)=O)CN(C(=O)Cc2cnoc2)CC1(F)F Cn1ncc(C(C)N(C(N2CC(O)(C3CCCCN3)C2)=O)CS(=O)(=O)C(F)F)c1F N1(C(c2c(C)scc2)=O)CCC2CN(C(c3cnc4n3CCS4)=O)C2C1 c1(C(C)C)nc2c([nH]1)CC(C(=O)N(C(C)CNC(=O)CN1CCSCC1)C)CC2 c1(C(=O)NCCC2CCN(C(c3cnc(C)nc3)=O)CC2)scc2c1OCCO2 c1(C(N(C)CCNC(=O)CC2CCCS2(=O)=O)=O)cccc2ncnc(O)c12 CC1(C)CC(NC(C2CC3CC2C2CC32)=O)CN(C(c2ccnc(Cl)c2Cl)=O)C1 c1(CN2CCC(C(=O)NC(C(=O)OCC)CO)C(O)C2)ccc2ccccc2n1 O=C(C1=CCCS1)NC1CCN(C(=O)C(O)CC2CCOCC2)CC1 C(=O)(C1Cc2ccccc21)NCC(C)NC(c1cc(C(=O)OC)no1)=O c1(C(N2C3(COC)CC(NC(C4CC4C)=O)(C2)C3)=O)cc(S(C)(=O)=O)ccc1O c1(C(N2CC(CCNC(=O)CC3CCCC3)(OC)C2)=O)cn(C)c(=O)n1C c1(C(C)Nc2cccc(C(=O)NCCCC(C)C)c2)cccc(Cl)c1Cl C1(CNC(CCSC)=O)C2CCC(C2)N1C(c1ncccc1C(F)F)=O c1(C(=O)NCCCNC(=O)COC(F)F)cc2c(nc1O)CCCCC2 c1(OCC(N2C(CNC(=O)CSCC(F)(F)F)C=CC2)=O)ccc(F)cc1O C1(CC(=O)NC2(C)CN(C(c3c(CC)scn3)=O)C2)CCCC(C(F)(F)F)C1 CC1CC(C(=O)N2CCC(CC(N3CC(n4ccnc4)C3)=O)C2(C)C)=NO1 c1(C(N2CCC(CNC(C(C)(C)CO)=O)C2)=O)cnn2cc[nH]c12 c1(C(N(C(C)CNC(C2(C(F)(F)F)CC=CCO2)=O)C)=O)cc(F)c(F)cc1N C1(C(=O)NC(COC(C)=O)CO)CC(C)CN1C(c1cc(C(C)C)[nH]n1)=O CC1CCN(C(C2(C)CCCO2)=O)CCN1C(c1c[nH]c2cccnc12)=O N1(C(CCC=CC)=O)CC(C)CCC1CNC(c1cc(C)sc1C)=O c1(NC(C2CC(NC(c3c(C)nn(C)c3)=O)C2)=O)cccc(Cl)c1C c1(CC)ccc(-c2nc(CCCS(C)(=O)=O)n(C3CCSCC3)n2)cc1 C1(C(N2CCN(C(CC)=O)CC2)=O)(NC(=O)CC)CC2(CC2)C1 Cc1cc(C(F)F)nn1CC(=O)NC(CNC(c1ccc(C(N)=O)[nH]1)=O)CC(C)C C1(OC)CCCN(C(C2CC3CCC2O3)C(=O)NCC(C)C)CC1 CCC(C(=O)NCC=CC(=O)N(C)CC1(CO)CC1)C(C)C n1(CCC(N2CC(c3onc(C)n3)C2)=O)cnc2ccccc12 c1(C(=O)NCC(C2CC2)NC(C2CN(C(C)C)C2)=O)cnn(C2CC2)c1 O=C(N=c1[nH]nc2[nH]ccnc1-2)C1CCCC(NC(C2CCCS2)=O)C1 C1(CCC(=O)NC2CC(CNC(C3(CS(N)(=O)=O)COC3)=O)C2)CC2CCC1C2 C1(CNC(Cn2c(C)cc(C)n2)=O)CCCCCN1C(=O)C(C)CF N1(C(C2(OC)CCCC2)=O)CC2C(NC(=O)C=C3CCCCC3)C2C1 c1(C(=O)NC(C2CN(C(C=CC=CC)=O)C2)C)nn(C)c(Cl)c1Cl c1(NC=O)nc(CC(=O)N(C2CCN(C(C3CC3C(F)F)=O)C2)CCO)cs1 C#CC1(C(=O)NCCCCC(=O)OC)CCN(OC(C2CC2C2CC2)=O)C1 C1(N(C(=O)CCOC2CCCOC2)C)CCCC(NC(=O)CSc2cccnc2)C1 C=CCC(CNC(c1ccn(CCC)n1)=O)C(=O)NCC(O)CF N1(C(C(C)(C)C#N)=O)Cc2ccc(CNC(=O)C=CSc3nc[nH]n3)cc2C1 CCCCC(C(=O)N1CCCC(CO)CC1)NC(c1cc(=N)[nH][nH]1)=O CN=c1nc(C(N2CCC(O)C(N(C(=O)CC3CCC4CC34)C)C2)=O)cc(C)[nH]1 c1(C(=O)NCC(=O)NCc2cn(CC(=O)OCC)nn2)cnn2cccnc12 c1(CNC(=O)COC(c2csc3ccccc23)=O)cn2cnnc2cn1 c1(C(=O)NC2C(CNC(CCC=CCC=C)=O)C2)ncc2n1CCCC2 C(=O)(CCCCCC#N)NC(C(C)NC(c1cc(C)nc(C)n1)=O)CO Cc1nc(NC2CCN(C(=O)CC3CCCOC3)CC2)sc1C(=O)OCC1CC1 C1(C(=O)NCCn2c(C)cc(C)n2)CC12CCN(CCC13CCCC1C3)C2 N1(C(C2(CC=C)CC2)=O)CCCC(C(N2CCN(C(=O)C(C)SC)CC2)=O)C1 N1(C(C2N(C(C)=O)CCC2)=O)CCN(C(=O)CNC(C2CCC23CCC3)=O)CC1 S(=O)(=O)(c1ccc(-c2ccc(O)cc2)o1)NC.C1(N(C)C)CN2CCC1C2=O C12(C(=O)NC(CC=C)CNC(=O)C(C)Oc3cccc(Cl)c3)CCN(CC1)CC2 O=C(C(F)CC1CN(C(C2CC2c2ccco2)=O)C1)N1CCC2CC12 N1(C(C(CCC)CCC)=O)CCC2(CO)CN(C(=O)C(=O)NC(C)C)CC2C1 C=C(Cl)CCC(=O)NC1(C(=O)N(CCN2CC=CC2)CC)CC(CO)C1 c1(OC)ccc(C)c(C(=O)N(C(CNC(=O)C(C2CC2)C2CC2)C2CC2)C)c1 c1(C(N2C(CCNC(C(=O)NC3CC3)=O)CSCC2)=O)cccc2occc12 CCCCC(CC)CC(=O)NC1CCCN(C(=O)CSCc2ccccn2)CC1 C1(CN(C(C2(C(C)C)CCOC2)=O)C)CN(C(=O)C(F)(F)CN(C)C)CCO1 c1(C(=O)NC(C2(O)CN(C(c3nc(CC)sc3)=O)C2)C)cc(CO)oc1C C12(C(=O)NC3(CN(C)C)CC3)C(NC(=O)CC3CCOC3)C3CC1C2C3 C(N=c1nc(N2CCCC(C)C2)c2sccc2[nH]1)c1cccc(OC)n1 c1(NC(=O)CN2CC3CC2CO3)ccccc1COc1ccccc1 CCCC(C)(O)C(=O)NCCCOCCOCCNC(=O)CSc1cnn(C)c1 C(C(F)(C(=O)N1CCC1C(N)=O)C(C)C)NC(CC1(OC)CCC1)=O C1(NC(c2ncc[nH]2)=O)CCCC2CN(C(c3cnn(C4CCCC4)c3)=O)CC12 Cc1c(Br)cc(C(=O)NCCCCNC(C2(C)CC(C)C2)=O)c(=O)n1C CCCCCCN1CCC(CC(=O)OC)C1.N12CCCC1CC(=O)NCC(C)O2 C(=O)(CC(C)C(C)(C)NC(N1CC(C)C(F)(F)C1)=O)OC N1(C(CCC(C)=O)=O)CCC2(CC1)CN(C(c1cnn(C)n1)=O)CCO2 C(=O)(CS(=O)C(F)(F)F)NCCC1CCN(C(C2C(CC)N(C)CC2)=O)CC1 c1(CNC(CC2C(C)C2)=O)ccc(CNC(C2CCCOCC2)=O)cc1 N1(C(c2n(CC)ncc2Cl)=O)CCCC(O)(CNC(=O)C(O)CSC)C1 N1(C(c2c(C)scc2)=O)CCC12CN(C(C1CNC(=O)CC1C)=O)C2 N1(C(C2(CC)CN(C(=O)CN(C)C(C)C)C2)=O)CC2(CCOC(=O)N2)C1 C(CCC(=O)NC1(C(=O)NOCCF)CCSC1)OCCOC C1(C(N(CCCCNC(Cc2cc(C)no2)=O)C)=O)CCCC(CF)C1 N1(C(C2CC(OC)C2)=O)CCC(O)(C(C)NC(c2cnc3sccn23)=O)CC1 c1(C(N2CCC23CN(C(C2(F)CCCC=C2F)=O)C3)=O)cnc(Cl)cc1Cl c1(C(N2CC(NC(Cc3cc(C)n(C)n3)=O)C(F)C2)=O)ccc2c(n1)NC(=O)CC2 Cc1ccc2ncc(C(N3CCC4CN(C(c5cnn(C)n5)=O)CCC34)=O)n2c1 N1(C(C(CC)c2cccnc2)=O)CC2(CNC(c3ccc(SC)o3)=O)CC1CO2 c1(C(=O)NC2CCC(NC(=O)CSc3ccccc3Cl)C2)cccc2nncn12 CCC(CC)CCC(=O)NC1CCC1NC(C1(Br)CC1)=O Cc1ccc(C(=O)NCC2CCCCC2NC(C2OCCCO2)=O)c(Br)c1 c1(C(=O)NCC2CC(NC(C3CCC=CCCC3)=O)C2)ccc2cnccc2c1 C(=O)(CCC(=O)N(C)CCN(C)C(c1c[nH]nc1Cc1ccccc1)=O)N(C)C c1(CC(=O)NC(CC)CNC(=O)C(F)CC2CC2)cc(C(F)(F)F)n(C)n1 N1(C(c2ccc(OCCC#C)cc2)=O)CCC(N(C)C(c2ccsc2)=O)C(C)C1 N1(C(C2(C(=O)OC(C)(C)C)CCC2)=O)CCCC(NC(=O)C=CBr)C1 C(=O)(CC(C(F)F)NC(=O)C#CC(C)(C)O)NC(CC(C)(C)C)c1cccnc1 C1(C(N2CC(OC)(CNC(=O)C(C)CC(F)F)C2)=O)CC2CCC(C1)C2O c1(C(N2CCC(CCNC(c3c(CC)n(CC)nc3)=O)C2)=O)cc2n(n1)CCO2 c1(C(=O)NC(CC)CNC(C2(C)CCOC2)=O)nc(Br)c2n1CCCC2 C=CCCCCCCCCC(=O)NC(CNC(C1CCCN1N=O)=O)CCCC c1(C(N(CCC)Cc2cccc(C3CC3)c2)=O)cc(C2CC2)ncc1Br N1(C(C(C)CC2CC2)=O)CCN(C(c2cnc(C(C)(C)C)[nH]2)=O)CC1 c1(NC(C2C3CN(C(C(C)(CO)CO)=O)C2C3)=O)cnc2ccc(Br)cc2n1 N1(C(C(C)c2cccs2)=O)CC2CCC1CC2NC(c1ccncc1Cl)=O c1(C(C)=O)cc(C(=O)NCC(C)(C)NC(=O)CC2CC2(Cl)Cl)co1 N1(C(C2CCC(C(C)C)CC2)=O)C2CCC1CN(C(C1(C)CC3CC3C1)=O)CC2 C1(C(=O)NCC2CC(F)(CNC(CCC=CCC=C)=O)C2)COCCN1C C(=O)(C(CCC(C)C)NC(c1ncccc1F)=O)NCc1nc(C)sc1C CC(CC(C)(C)C#N)Nc1c(C(N)=O)c(C(F)(F)F)nn1C C1(CC)CCCC1(C)C(=O)N(C)CC1COCCN1C(=O)CSc1nncs1 N1(C(=O)OCC)CCC(C(N2CCC(CNC(C3(F)CC=CCC3)=O)C2)=O)CC1 c1(C(=O)NCC2CCN(C(c3ncncc3F)=O)C2)c(F)cccc1Br c1(C(=O)NC23C(CN(C(c4nc(CC)sc4N)=O)C2)C3)cccc2nnn(C)c12 c1(-c2onc(C(N3CC(CCNC(C4CC(SC)C4)=O)C3)=O)n2)cccc(F)c1 C1(O)(CN(C)C(C2(F)CCCC2)=O)CN(C(C2CSCCS2)=O)C1 N1(CC)CCOC(C(=O)N(CC(CO)(CO)NC(C2CC(F)C(=O)N2)=O)C)C1 C1(NC(c2c(C)oc(CNC(=O)C(C)CC3CCC3)n2)=O)CCCCC1(C)C C1(C(N2CC(N(C)C(c3cnc(-n4cccn4)o3)=O)C2)=O)CCCC12CC2 N1(C(C2(NC(CCCN(C(C)C)C)=O)CCOCC2)=O)CCOC2CCOCC12 FCCN=C(NCc1cc(Cl)ns1)NCc1nc(C2CCCCC2)no1 c1(OC(F)(F)F)cccc(CC2CCCN2S(=O)(=O)Cc2ccc(F)cc2)c1 Cc1cc(C(=O)NC2(C)CC(NC(=O)CC34CCC(CC3)CC4)C2)nc(C)c1 c1(CNCc2ccc(-c3ccc(C(C)(C)C#N)cc3)nc2)ccc2c[nH]nc2c1 c1(NC(C(CC(C)C)ONC(C2COCC(C)O2)=O)=O)cccc2ccncc12 C12(C(N3CCC(COC)(CNC(c4ccoc4)=O)C3)=O)CCC(C)(CC1)OC2 C1(CC(N2C(c3ccc(C)o3)COCC2)=O)CCC2CNCCC2C1 c1(C(=O)NCC2CCC2NC(c2cnc(C3CC3)[nH]2)=O)ccc(OC(F)F)nc1 CCCC(C(=O)NC12CC(NC(=O)C(C(=O)OC(C)(C)C)N(C)C)(C1)C2)N(C)C c1(C(=O)NCC(C2CCCC2)NC(CC(=C)C)=O)c(S(C)(=O)=O)cnn1C C1(CNC(C2CC2Sc2ccccc2)=O)CN(C(=O)CC2(C)CC2)CCO1 CCC(F)(F)CC(=O)N(C1CCCCC1NC(C1C(Cl)(Cl)C12CC2)=O)C c1(CCC)cc(C(=O)NCC2(CNC(=O)CCC(C)N(C)C)CC2)cc(O)n1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CC(NC(=O)CC2CC2(Cl)Cl)CC2(CCC2)C1 c1(C(N2CCCC(NC(CCC3C(C)(C)C3)=O)CC2)=O)cc2c(s1)CCCCC2 C(C(C)CC(=O)NCc1cc(NC(=O)OC(C)(C)C)cn1C)OC C#Cc1ccc(NC(=O)C=C(C)CNC(c2ccc(C)nc2O)=O)c(C)c1 N1(C(C2OCCN(C)C2)=O)CCC(C)(C)C1C(=O)NOCCC1CC1 N1(CC(N2CC(C(C)NC(=O)C(c3ccc(Cl)nc3)(C)C)C2)=O)CC(=O)NC1=O N1(C(C2(CC)CCOCC2)=O)CCC2(CC(NC(c3sc(C)c(C)c3C)=O)C2)C1 CCCCC(C)CCC(=O)N1CC2CC1CN(C(c1cnn(C(C)C)c1N)=O)C2 C1(NC(C(C)N(C)C)=O)C(C)CCN(C(c2cc3ncccc3[nH]2)=O)C1C c1(OC)cc(OC)cc(C(N2CC(NC(c3ccc(F)o3)=O)C(C)C2)=O)c1 c1(NC(C2CN(C(c3c[nH]nc3C(F)F)=O)CC2F)=O)cc(Cl)cnc1O N1(C(c2c(C)cc(F)s2)=O)CCC(CO)(NC(c2ccc(O)nc2)=O)CC1 N1(C(C2(CC)CC2)=O)CC2CCCC(CNC(C3CC(F)C3)=O)C2C1 c1(N2CC(NC(c3nc(CCC)oc3)=O)C(C)CC2)nc(C)nc2n[nH]cc12 C#Cc1ccc(C(=O)NCC(C(C)(C)C)NC(C2(CC)CC2)=O)o1 C1(C(N2CC(C(C(=O)O)OC)C2)=O)CC(=O)N(c2cccc(C(F)(F)F)c2)C1 C(=O)(CCCCCCCC(=O)NCCCNC(=O)CC1(C)CCCCC1)OC C(=O)(C#CC1(C)CCCO1)NC(C)(C)C.CC12CN(CCO1)Cc1nc[nH]c12 C(=O)(C(=O)C=Cc1cccs1)NCC(C)N(C)C(c1ccnn1C)=O C1(C(N(c2ccccc2)C(C)C)=O)CCC(n2cc(C3CCN(C)C3)nn2)C1 c1(CN(CC(=O)O)C(C)=O)ccccc1Br.c12cn(cn1)C1CN(C1)C2=O C1(CCCC)CN(C(C2CC(C(F)F)(OC)C2)=O)CCN1C(=O)C(C)N(C)C CC1CC(C(N2CCOCC(CNC(C34CCC(C3)OC4)=O)C2)=O)CC(C)C1 C#CCCN=C(NCCN(CCCS(=O)(=O)C1CC1)CC)NC1COC2CC1C2 c1(CC(N2CCC(N(C(=O)C(F)n3cccn3)C)CC2)=O)cnn2c1CCCC2 N#Cc1cc(C(=O)NCC2(F)CCN(S(=O)(=O)C(Cl)(Cl)Cl)CC2)ccc1O c1(C(=O)NCC(CO)NC(CC(CCC)CCC)=O)c(C)ccc2ncccc12 C1(C(=O)NC2CCCC(NC(CCCCOCC)=O)C2)Cc2cc(C)ccc2O1 c1(C(N2CC(CC(=O)NCCC(C)CO)OCC2)=O)ccc(C#N)cn1 CCC(CC(=O)NCC(C)(C)CNC(C1(CC)CCCO1)=O)c1ccccc1 O=C(CCc1ccc(O)cc1)N1CCCc2c(Br)cccc21 C1(CNC(=O)Nc2ccc(SCC(=O)NCCOC)cc2)CNC(=O)C1(C)C c1(-c2cc(C(=O)OC)ncc2)ccc(S(=O)(=O)N(C)CCN(C)C)c(Cl)c1 C(=O)(CC(C)(C)C(=O)N1CC(C)C1C(N1CC2COC(=O)C2C1)=O)OC c1(C(=O)NCCCNC(C2CCC2)=O)cccnc1-c1ccccc1 N=c1[nH]c2ncc(C(=O)NCC#CCNC(c3ccc4sccc4c3)=O)cc2s1 Cc1ccc(OCC(=O)NCC2CN(C(=O)CCC3OCCO3)CC2C)c(F)c1 N1(C(Cc2cc(C)[nH]n2)=O)CCC(NC(=O)C(C)(C)CCF)C(O)C1 C1(CNC(c2c(C)n(C(C)C)cc2)=O)CC2(C1)CN(C(=O)C=CC(F)(F)F)C2 CC1(C)CC2(CN(C(C3CN(C(C4CCC4(F)F)=O)C(C)(C)C3)=O)C2)C1 S(=O)(=O)(c1ccc(N2CCCC(C(N)=O)C2)cc1Br)N1CCC(C)(CC)C1 Cc1c(CC(=O)NCCNC(C2CC3CCC2CC3)=O)nc(Br)n1C Cc1nc2cccc(C(N3CCCCC(N(C(=O)C(C)C(C)O)C)C3)=O)n2n1 c1(CNCCC(C)N(C)C)cc(Br)ccc1Br C1(NC(C=CC)=O)CCC12CCN(C(c1c(F)ccc(Br)c1F)=O)CC2 c1(C(=O)NC23CC(C(=O)Nc4c(C(=O)NC)cccc4)(C2)C3)cc(Cl)ccc1I N#CCCCC(C(=O)Nc1cccc(-c2ccco2)c1)N1CC2CCCCCC12 c1(C(=O)NCCN(C(=O)Cc2cccnc2Br)CC)c[nH]c2cc(C)ccc12 N1(C(CCC=CC(C)C)=O)CCC2(CC1)C(N(C(=O)CC(C)(C)O)C)CS2(=O)=O CC1CN(C(=O)CC2(N(C)C)CCCC2)CCN1C(=O)C(F)CC1CCC1 Cc1cnc(CNC2CCCCC2C(=O)Nc2ncc(Br)cc2C(F)F)cc1Br N1(C(C(CC)(F)F)=O)CCC(CNC(=O)Cc2ccc(C)o2)C(C)C1 N(C(=NCCCCc1ccccc1)NC(c1ccccc1)CC)CCCOCC c1(C(=O)NC2(C)CCN(C(C(CCSC)O)=O)CC2)cnnc2ccccc12 Nc1cccn(CC(N2CCC(OCCNC(c3cccc(F)c3)=O)C2)=O)c1=O Cc1[nH]cc(C(=O)NC2CCCCC2NC(=O)CCC(N)=O)c(=O)c1Cl c1(C2(C(=O)OCCCSC)CC2)ccc(Br)cc1 N1(C(CSCC(=O)OC)=O)CC(C2CCCCN(C(=O)CC3CCCOC3)C2)C1 c1(CC)cc(C)ccc1C(=O)NCC(CNC(c1ccccc1CC#N)=O)OC c1(C(N(CCNC(=O)C(C)(O)C2CC2)CC)=O)snnc1C(C)C c1(C(N(C2CCN(C(=O)C(=O)NOC)CC2)CCCC)=O)cc(C)nc(C)c1 c1(C(c2n(CC(=C)C)nnn2)NCCc2ccc(Cl)s2)ccc(OCCC)nc1 C#CCCN=C(NCc1cc([N+](=O)[O-])ccc1Cl)N1CCC2(CCCN(C)C2)C1 CCC(C)C(CNC(=O)C(F)CC1CN(C(=O)Cn2ncn(C)c2=O)C1)CO c1(OCC)cc(C(N2CSCC2C(=O)NCc2cc(Cl)no2)=O)on1 c1(C(N(C2CC(NC(Cc3c(C)ncs3)=O)C2)C)=O)cnc(C(C)C)nc1 N1(C(COCC(=O)NC)=O)CCN(C(=O)Cc2ccc(SCC)cc2)C(C)C1C c1(-c2cn(C3CCC(C(=O)NCC(C)(C4CC4)OC)C3)nn2)cn(C)nc1CO C1(O)(CNC(c2c(SC)scc2)=O)CCN(C(C2(C)CC(C)C2)=O)C1 c1(CCC(=O)NC(C)CC2CN(C(=O)CCC3CC3(Cl)Cl)C2)cn(C)cn1 c1(C(N2CCC(CNC(C3N(C)CC3)=O)CC2)=O)cc2cnccc2[nH]1 c1(OC)cccc(C(N2CC3C(CNC(c4cc(O)no4)=O)C3C2)=O)c1[N+](=O)[O-] C=CCC(C(=O)N1CC(=C(F)CNC(c2cnc(C(C)(C)C)[nH]2)=O)C1)N(C)C C1(C(N2CC(n3cc(CCC4CCCCO4)nn3)C2)=O)COCCN1CCO Cc1cc(C(=O)NCCc2n[nH]cc2C(=O)NC(C)CCC2CC2)ncc1N CC(C)CC(C)CC(=O)NC1C2CC1N(C(=O)CCc1ccc(Cl)s1)C2C c1(C(N2CCC(NC(C=NOC)=O)C2)=O)ccc(C)c(F)c1 N1(C(c2cn(CCNC(CSC)C(=O)OC)nc2)=O)CCOCC1CC(=O)OC Cc1cccc(O)c1C(N1CC2(CCC2NC(c2cnn(C)c2)=O)C1)=O CC(CCC(=O)N1CCC(c2cc[nH]n2)C1)c1ccccc1.C1(CCC)CC(F)(F)C1 c1(C(=O)NCC(C)Oc2ccccc2Cl)cncc2n[nH]cc12 c1(NC(C)C)ccc(C(=O)NCCCCCNC(=O)CC2(O)CCC2)cn1 n1(CC(N2C(C)C(C)N(C(C3CC3C#N)=O)CC2)=O)ccc(=O)c2ccccc12 c1(OC)ccc(NC(=O)C(c2cccc3c2OCC3)O)cc1S(N)(=O)=O N1(C(C2C(C)OCC2)=O)CC(F)CC1CN(C)C(C12CCC1CC2)=O C1(N(C(c2cc(SC)oc2)=O)C)CCN(C(=O)C(=Cc2cccnc2)F)CC1C c1(C(=O)NC(CC)CN(C(=O)C(C)=C(C)C)C)sc(N2CCOCC2)nc1Cl C=CC(C)(O)C(=O)N(C(C)C(=O)NCCc1ccncc1)C1CC1 C(=O)(CC(CNC(C1CCCN(CC(C)C)C1)=O)CC(C)C)OC(CC)C C1(F)(CNC(=O)CS(=O)(=O)Cc2cccs2)COCCN(C(=O)CC(F)F)C1 N1(C(CN(C(CN(CC(C)(C)O)CC)=O)C)=O)CCOCC1 N1(C(C(C)NC(=O)NC)=O)CC2CC1CN(C(C1CN=C3N=CNN3C1)=O)C2 N1(C(CC2C(C)CCC2)=O)CC(C2CCN(C(C3(O)CCCCC3)=O)CC2)C1 C1(CCNC(CC(C)c2ccco2)=O)CN(C(=O)C(C)(C)O)CCS1(=O)=O N1(C(c2n(CCOC)ncc2)=O)C(CNC(=O)CSC)CC2COCC12 Cc1nn(C)cc1CC(=O)N(CC(=O)NC1CCCC1)C(C)C C1(NC(c2csc(O)n2)=O)CN(C(c2cccc(Cl)c2)=O)CC12CC2 C1(CCC)(NC(c2ncn(C)c2C)=O)CCCN(C(=O)CC2(O)CCCOC2)C1 CC(CC(=O)NCC12CCCC1C2)C(C)(C)NC(C1CCCN1C1CC1)=O c1(OC)ccc(Cl)c(C(=O)N(C2CCCN(C(=O)CC(C)OC)C2)C)c1F Cc1cnn2cc(C(N3CC(NC(C4(O)CCSC4)=O)C(C4CC4)C3)=O)cnc12 C(=O)(N1CCC(C(=O)NC(c2ccncc2F)C)O1)c1c(CC)nn[nH]1 C(CCS(C)(=O)=O)(C(=O)OC(C)(C)C)NC(=O)OCC(CCO)C(F)(F)F c1(OCC(=O)N(C(C)C)CCN(C(=O)CCC#N)C)ccc2c(c1)CCC(=O)N2 C(=O)(CCCC(=O)OC)N1CCC(N(C(=O)C(C)CC2CCCO2)CCC)CC1 c1(CC(=O)NC2CCN(C(=O)C=Cc3cc[nH]c3)C2)nccc2ccccc12 C1(OC)CC2N(C1)CC(=O)NC2.C(=O)(CCCC1CCC1)NCC1CCOCC1 N1(C(C2CC(CCC)C2)=O)CCC2(CC1)CCN(C(=O)C(=O)C(C)C)CC2 C1(NC(C2CC(=C)C2)=O)CC2CCC1C(NC(=O)C(C)Cc1cccc(Cl)c1)C2 c1(C(=O)NCCN(C(COC(CC)CC)=O)C(C)C)cc(C(C)(C)O)on1 C1(C(=O)NCC=CC(=O)NCCC2CCOC2)CCC2CC12 N1(C(c2c(C)cn(C)c2)=O)CCC(C)C(NC(c2ccncc2Cl)=O)C1C c1(OC)nc(C(F)(F)F)c(C(=O)N(C2CCN(C(=O)OC(C)(C)C)C2)C)s1 C(CCCCC(=O)N(C1CCCN(C(C2(C)CC=CC2)=O)CC1)CC)OC N1(C(c2ccc(CN(C)C)nc2)=O)CCC(C2CCN(C(=O)C(N)=O)C2)CC1 Cc1cc2occ(CC(N3CC(O)(C(C)NC(C4CC4(Cl)Cl)=O)C3)=O)c2cc1C Cc1cc2ccccc2cc1C(=O)NC1CN(C(=O)C(C)c2cc[nH]n2)CC1C C(C)(CNC(=O)C(=Cc1ccccc1)C)(C(C)C)NC(CCCNC(C)=O)=O N1(C(CCC(=O)NCCC)=O)CCOCC(C)(CNC(=O)C(C)c2ccsc2)C1 N1(C(C(CNC(C(CC)C(=O)OC)=O)C)=O)CCc2cncnc2C1 Cc1cc(CNC(=O)CC2C=CC2)sc1C(=O)O N1(C(Cc2cc(C)[nH]n2)=O)CC(N(C(=O)CCc2cc[nH]n2)C)C(F)C1 c1(C(N2C3CC(NC(c4cncc(F)c4)=O)C2CC3)=O)nnc2ccccc2n1 C1(C(=O)NCCOC2CN(C(CN(CCC)C)=O)C2)CC2(C1)CC(F)C2 C1(CC(=O)N(C(COC)COC)C)CN(C(c2[nH]ccc2C2CC2)=O)CCC1C C(C)(CCC(=O)OCC)SC.C(C)(C)(C(C)C)NC(=O)COc1cnn(C)c1 C1(CNC(c2ccc(Br)nc2)=O)CN(C(c2cccc(Br)c2)=O)CCO1 C1(CC)(NC(C2OCC2(C)C)=O)CCN(C(C2CCCC(C(=O)OC)C2)=O)CC1 C1(C(N2CCC(CCC(=O)NC(c3cnn(C)c3)CC)C2)=O)CCC(F)CC1 N1(C(=O)Cc2ccon2)CCCN(C(c2cn(CC(F)(F)F)nn2)=O)C(CO)C1 S(=O)(=O)(c1cc(F)cc(F)c1)N1C2CC(C(=O)NCCCOCC)C1CC2 C(=O)(CC(O)CCC)NC1(CC=C)CCN(C(=O)C(=O)Nc2ccccc2F)C1 N1(C(C2CCN(CCC#C)CC2)=O)CCC(C)N(C(=O)Cc2cccnc2)CC1 O(NC(=O)C(C(C)O)NC(=O)CC1(COC)CC1)CC C(N=c1nc(N(C)CC2CCCCO2)c2c([nH]1)c(C)nn2C)c1ncc(C)o1 c1(CNC(C(C)CC(C)(C)C)=O)cccc2c1CN(C(C1CCCC(O)C1)=O)C2 C(=O)(CC(C(F)F)C1CC1)C(=O)C=C1CCSCC1.CC(C=CC(=O)NC)NC C1(CC=C)(NC(C2CCCC2O)=O)CCCN(C(C2CCC3(C2)N=N3)=O)C1 C(=O)(CCCCCNC(C12CCN(CC1)C2)=O)NCC1C(C)(C)CCO1 c1(C(=O)NC(CCCCNC(CCC=C=C)=O)C)ccn(CC)c(=O)c1 C1(C(=O)Nc2c(C)cc(F)cc2Br)CCc2ccccc2N1 c1(C(=O)NCC(CO)NC(C(C=C)O)=O)cc(N(C)C)cc(C#N)c1 C1(CNC(c2c(CC)[nH]nc2Cl)=O)CN(C(c2cccnc2)=O)C2CCCC2O1 c1(C(=O)NC2CCC(NC(CCC3CC(OC)C3)=O)C2)cnc2c(F)cccn12 c1(C2(CC)CC2)ccc(C(=O)NC2CC(NC(C3(C)CS(=O)(=O)C3)=O)C2)cc1 c1(C(C)N(C)C(c2cnc(-c3ccnn3C)cn2)=O)ccccc1F CCCC(C#N)C(=O)NC1CC(CCC(=O)NC2CCCCCC2F)C1 C(CC(=O)NCC(C)(C)C1CCCC1)N(C(=O)C(C)N1CCCC1)CC C1(C(N(C)CC2CCCCCC2)=O)C2CC2CN1C(=O)C=CC(C)(C)C c1(CC)oc2ccccc2c1CC(=O)NCC(C)(C)NC(=O)CC(C)CC c1(C(=O)NC2C(OC)CN(C(C3CCOC(=O)N3)=O)C2)cc(C)cc(F)c1 N1(C(CC2CC(=C)C2)=O)CC(NC(=O)C(=O)NCC(F)(F)F)CC1C c1(C(=O)OC)cnc(N2CCN(C(=O)C(c3cnn(C)c3)O)CC2C)nc1C c1(C(N(CCC2N(C(C(COCC)C)=O)CCCC2)C)=O)n[nH]c2ccccc12 c1(C(=O)NC(CC=C)CNC(c2ccc(C(F)F)s2)=O)ccc2c(c1)OCC2 C1(c2ccc(Cl)cc2)(C(=O)NCCN(C(=O)C(F)C2CCC2)CC)CC(F)(F)C1 N1(C(C(C)Sc2ccccn2)=O)C2CCC1C(NC(=O)CCc1ccc(Cl)s1)C2 N1(C(CCOC)=O)CCN(C(C2CCC(F)(F)C2)=O)C(C2CCC2)C1 Cc1cnc(C)c(C(=O)NCC2CN(C(=O)CCSCC(C)C)CCC2C)c1 C1(C(N2C(CNC(C(C)n3cncn3)=O)CC(O)C2)=O)CC12CCSCC2 Cc1n[nH]c(C)c1CC(=O)NC1(CNC(C2CC23CC3)=O)CCOC1 C1(CNC(c2c(C)n[nH]c2)=O)CCCN(C(C2CCN(C)C2)=O)C1 c1(C(=O)NCC(CNC(c2onc3c2CCCC3)=O)OC)cnc2cc[nH]c2c1 Cc1ccc(F)cc1C(C(=O)O)NC(=O)C=CC(c1cccc(F)c1)=O C(CC(=O)N1CCC(CNC2CCC(C)(C)CO2)CC1)(C(N)=O)NC(C)=O c1(C(N2CCCC(CNC(C3C4CC(=O)CC43)=O)C2)=O)occ2c1CCCC2 CN1C(=O)NCC12CN(C(C1CN(C(C3(C)COCCO3)=O)CC13CCC3)=O)C2 c1(CNC(c2cc(O)cs2)=O)cc[nH]c1C(=O)NCc1cc(Cl)no1 C1(NC(CC)=O)CCOC12CCN(C(c1cncn1-c1cnn(C)c1)=O)CC2 C1(CNC(C(CC)OC)=O)Cc2ccccc2CN1C(c1cn(CC)nn1)=O c1(C(=O)NC2C(C)(C(F)F)C2)ccc(CNC(C2(CO)CCOC2)=O)o1 C1(CC)CN(C(=O)C=CCN(C)CC)CCC1CNC(C1CC(=O)CCO1)=O C1(NC(c2c(Cl)cn(C)n2)=O)CN(C(=O)CC2CCCC2(F)F)CCC1CO C(=O)(C(C(C)(C)C)NS(C)(=O)=O)NCC(C)CNC(=O)C=CC1CCCO1 C#Cc1cnc(C(=O)NC(C)(CNC(=O)Cc2nnc(C)o2)CC)c(C)c1 N1(C(C(CCSC)NC(c2cocc2C)=O)=O)CCCC2(C1)N=N2 Cc1noc(C)c1C(C)(C)C(=O)N(CCCn1ccnc1C)C CC1(C)NC(=O)CC1C(=O)NC1COCC1C(=O)N(C1CCCCC1)CCO c1(NC(C2CN(C(C(F)=CCC)=O)CC2F)=O)ccc2ccncc2c1 c1(OC)nc(C)ncc1C(=O)NCC1C2CC1N(C(C1CCCC(C)(C)C1)=O)C2 N1(C(C2CCC(C)C2)=O)CCCC(N(C(=O)Cc2cnoc2)CCO)C1 N1(C(C2(F)CN(C(CC(C)F)=O)C2)=O)CCC2(CCOCC2)C1 n1(CC)ccc(C(=O)NC2CCC(C)(CNC(=O)Cc3csc(C)c3)C2)c1C c1(CC(=O)NC2(C)CN(C(C(C)C(C)n3cccn3)=O)C2)cc(S(N)(=O)=O)cs1 c1(N2CCC(C)(C(C)C)CC2)nc2ccc(Cl)cc2c(=NCCCOC2CC2)[nH]1 Cc1ccn(CC(N2CC(NC(C3CCCN3C(N)=O)=O)CC2(C)C)=O)c(=O)c1 C1(NC(Cc2c(C)scc2)=O)CC(C(=O)NCC(F)(F)C(C)C)C1(C)C N1(CC(=O)NCCc2cn(C)nc2)CC2CC(C(=O)O)CC2(CO)C1 C12(NC(CNS(NC)(=O)=O)=O)CCOCC1CN(C(c1sccc1C(F)F)=O)C2 N1(C(C(n2cc(CC(O)C(C)(C)C)nn2)C)=O)CCC(C=CC(=O)O)CC1 O(NC(=O)C(CN=[N+]=[N-])NC(=O)CC12CCCC1C2)CC=C Cc1nc2ncnn2cc1C(=O)NCCC(C)NC(c1ncc2ccccn12)=O c1(CC(=O)N(C2CCN(c3nncs3)C2)CCC)ccc(C)nc1Cl c1(-c2cc(C(=O)NCCc3ccc(C)cc3)n[nH]2)ccc2ncnn2c1 N(C(=NCCCc1cccc(F)c1)NCCF)C1CCCN(CC)C1 C(C)(C)(CCCC(=O)Nc1cncc(CO)c1)NC(CN1CCC(C)C1)=O CCCS(=O)(=O)CC(=O)NC1CCN(C(=O)Cc2occc2C(=O)OC)C12CCC2 c1(C(C)NC(CC(C)NC(C2N(CC)CCC2)=O)=O)ccc(F)cc1 n1(C(CC)C)nnnc1C(c1nc(COC)cs1)NCCC1(COC)CC1 C(=O)(C(O)CC(F)(F)F)NC1C(SC)CN(C(c2ccnnc2)=O)C1 C1(N(C(C(CC)F)=O)Cc2cc(-c3cccs3)on2)CCN(CC(C)C)CC1 C1(C(=O)NCC2CC2NC(=O)CC2(C#N)CC2)(CC)CCCCO1 c1(CC)ccnc(NC(c2noc(=O)n2C)c2nnnn2CC2CCCO2)c1 C=CCC(C)(O)C(=O)NC1CCC(NC(C2CCC3CC23)=O)C1 c1(C(C(=O)NCC2CC(NC(c3nc(OCC)oc3)=O)C2)(C)F)ccccc1F N1(C(C23OCC(C(C)C)(C2)C3)=O)CC(NC(C2CC(S(C)(=O)=O)C2)=O)C2(CC2)C1 C1(NC(C(CC)C)=O)CCC(CNC(c2cc(O)ncn2)=O)CC1 C(=O)(C1COc2ccc(Cl)cc21)N(CC(C)(C)NC(C(S(CCC)(=O)=O)C)=O)C N1(C(=O)OCC)CCC(C(=O)NCC2CCCC(OCC(=O)OCC)C2)CC1 c1(NC(CC)CSC)[nH]c(=NC2CC2C(C)C)nc2c1ncn2C(C)C C(=O)(C1=COCC1)NCC(CCOC)NC(=O)CSCc1ccccc1F C1(CNC(CCP(C)(C)=O)=O)CCN(C(c2ccc(CO)nc2)=O)CCC1(F)F c1(C(=O)NC2C3(CN(C(C(C)CN(C)C)=O)C3)CC2)ccc(S(=O)(=O)CF)cc1 O=C(C(O)C1CCc2ccccc21)N1CCOC(C(F)F)CC1 CCCCC(CCC)CN=c1[nH]c(=NC(CC)C2CCC2)[nH]c2c(F)cccc12 N1(C(c2ncn(CC)n2)=O)CC(NC(C2CCCC(OC)C2)=O)C2(CC2)C1 C(C(O)CC(C)(C)CO)N1CCC(Oc2c(OC)cccc2)C1 c1(C(=O)NCC2(O)CC(NC(CC(CC)C3CC3)=O)C2)cnc2cnccc2c1 c1(CNC2C(C(=O)Nc3ncc(C#N)nc3)CCCC2)ccc(O)c([N+](=O)[O-])c1 Cc1nn(C)c(C)c1CC(N1CCC(C)(C(N2CCCC(C#N)C2)=O)C1)=O O(NC(=O)C(C(C)CC)NC(=O)C(CC(C)C)OC)CC=C N1CCC(CN(C)S(N)(=O)=O)C(F)C1.c1(C=O)cccc(Nc2ccccc2)n1 CC1C(NC(C2(CF)CCC2)=O)CCN1C(C1CCN1Cc1ccccc1)=O C(=O)(C1=CC(C)(COC)C1)N1CCC(CC=C)(NC(=O)C=CC(CC)=CC)C1 CCCCC(CO)NC(=O)CCN(C(=O)CC1CCC(=O)C1)C1CC1 c1(C(=O)NC(CC)(CNC(=O)C(C)C(C)COC)CC)ccc2c(c1)NC(=O)C2 N1(C(C(CSC)C)=O)C2CCC1CC(NC(=O)C(F)(F)CC(C)C)C2 c1(C(N(C(CC)CO)C2CC2)=O)coc(CNC(=O)C(O)CN(C)C)c1 C1(CNC(Cn2ncc(C)c2)=O)(NC(c2c(C)cncc2C)=O)CC2CCC1C2 N1(C(CCSCC(C)C)=O)CCC(C)(NC(C2CCC2(F)F)=O)C1 c1(C(C)N(C(=O)NCC(C)(O)Cn2cc(Br)cn2)CC)ccc(Cl)cc1 N1(C(CCCC#CC)=O)CCC2C(CCN2C(c2cc(Cl)n(C)n2)=O)C1 Cc1cc2c(CC(=O)NCC(F)CNC(=O)Cn3cc(C(F)F)cn3)csc2s1 C1(N(C2CC2)NC(C)(C)C)CCN(Cc2cc(C)[nH]n2)C1(C)C C(=O)(C1=NNC(=O)CC1)N1C(C)CC(NC(CCCCN(C(C)=O)C)=O)C1 CC(C)(C(=O)N1CCC1CC(N1CCC1CN=[N+]=[N-])=O)C1CCCC1 C1(NC(=O)NCc2cccc(C(OC)OC)c2)CCOC12CCOC2 C(CCCCNC(C1COC(=O)N1)=O)N(C(=O)CCC1CNC(=O)N1)C c1(C(=O)NCc2cccc3[nH]ccc23)cnc2nc(O)nc(O)c2c1 C(=O)(C(C(C)C)NC(=O)OC(C)(C)C)NCCCNC(c1c(CC)cco1)=O c1(NCCC2(CSC)CC2)ncccc1S(=O)(=O)N1CC(C)C(C)C1 C1(NC(C2CN3CCN2CC3)=O)CN(C(=O)COc2cccnc2)CC12CCC2 c1(NC(N2C(C(=O)OC)C3CC3C2)=O)ccc(OC(F)(F)F)cc1Br c1(C(=O)NCCCN(C(c2csc(CSC)n2)=O)CC)nccc2nn[nH]c12 C1(NC(=O)CCc2ncc[nH]2)CC2CCCC(C1)N2C(c1ncncc1Cl)=O C(=O)(CC(F)(F)Br)NCCOCCN(C(=O)C=CC=C(Cl)Cl)C c1(CCC(=O)NC2C(NC(C(C)(C)NS(C)(=O)=O)=O)CC2)ccc(F)cc1 C1(NC(CCOC)=O)CCC2(CC1)CC2NC(c1cc(-c2csc(=N)[nH]2)c[nH]1)=O N1(C(CC=CC=C)=O)CC=C(CNC(=O)C(C)n2ccnc2)CC1 c1(C(N(CC(C)N(C)C(c2cnc(O)o2)=O)C)=O)n[nH]c2c1CS(=O)(=O)CC2 C1(C)(NC(c2c(COC)noc2)=O)CCN(C(=O)CCCc2ccc(C)cc2)C1 c1(C(=O)NC(C(C)C)C(C2CCCCC2)NC(C2CCC2)=O)ncc(F)cc1F C1(C(=O)NC2CCN(C(C(c3ccc(F)cc3)=O)=O)C2)CCC12CCOCC2 c1(C(=O)NC2CC(F)(CNC(CCOCCN(C)C)=O)C2)c(F)cccc1F N1(C(C(C)SC)=O)CC(F)CC1CNC(=O)C=C(Cl)Cl c1(NC(C2CCN(Cc3c(C)[nH]c(C)c3C)CC2)=O)ccc2c(c1)CCC2 c1(C(N(C)CC2(C)C(NC(c3c(C#C)c[nH]n3)=O)CCC2)=O)cc(C)nc(O)n1 c1(C(=O)NC2C(C)N(C(=O)CC3(C)CC3)CCC2)ccn2c1CCCC2 C1(NC(C(C)N(C)C)=O)CCC(NCC(C)(C)N(C)C)CC1.C(CCOC)N O=C(C1=NOCC1)NC1CN(C(c2cccc(C(F)(F)F)c2)=O)CC1O CC1CN(C(C23CCC(C(=O)O)(CC2)C3)=O)Cc2cccc(Br)c21 CC1CCCn2c(CC(=O)NCCNC(=O)Cc3ccccc3)cnc21 C12(CC(=O)NCC3(NC(CCC(C)N(C)C)=O)CC3)CCCCC1C2(F)F c1(C(=O)Nc2cccc(CS(C(C)C)(=O)=O)c2)cc(F)c(F)cc1I C1(CNC(C(=O)NCC)=O)CCC(C(=O)N(C)CCC)CC1 C1(C(=O)NCCC(CC)(O)CC)CC(N=[N+]=[N-])CN1C(C1CC(C)=NO1)=O C#Cc1ccc(C(N2CCC=CC2C(=O)NOCCCCCC2CC2)=O)cc1 C1(C(=O)NCC(CNC(COc2cn(C)nc2)=O)O)C(F)(F)C12CCC2 C=CC1(C(=O)NCc2c[nH]nc2C2CC2)CCN(C(c2cnc(N)cn2)=O)C1 C1(NCc2ccc(CC(C)C)cc2)CCS(=O)(=O)CC1 Cc1cc(C)c(C(=O)NC2CC2CNC(=O)C(C)Cc2ccco2)s1 C(CO)(CCCCNC(=O)C(C)(O)COC)NC(c1cccc(SCC)c1)=O N1(C(C(C)=CC)=O)CCC(C)(C)C1CNC(=O)Cc1nn(C)cc1Cl C12(C(=O)NCC(CNC(CCn3c(C)ncc3)=O)O)CCOC(C)(C1)C2 c1(C(N2C(C(CC)O)CCC2)=O)oc(CNC(c2[nH]cc(C)c2C)=O)cc1C C(CC(C)C(=O)NCC1C(O)C(O)CN1C(C1(c2cccnc2)CC1)=O)=CC c1(CNCC(CN(CCOC)C)O)ccc(C(=O)O)s1 c1(C(=O)NCC(N(C(C(CC)CC)=O)C)C2CC2)ccc2c(c1)NC(=O)CN2C N1(C(CC(CC2CC2)NC(CCSCCCC)=O)=O)CCCC(C)CC1 N1(C(C=C(C)C(F)F)=O)CC(NC(=O)C(c2cccc(C)c2)C)CC(C)C1 Cc1cc(C(N2CCC(C(C)NC(c3cocn3)=O)CC2)=O)cc(Br)c1C C1(CNC(c2cccc(C)n2)=O)CC(C)(C)CN1c1cc(-c2cccs2)ncn1 C1(NC(c2cc(C)[nH]n2)=O)CC(C(=O)NC2CN(c3ncco3)C2)C12CCC2 CC(=O)CC(C)(C)CC(=O)N1CCC2(CCC(NC(=O)C(F)(F)F)C2)C1 C#CC1CCC(C(N2CCC(NC(=O)C(c3ccc(Br)s3)C)C2)=O)CC1 c1(C(=O)NC2C(NC(COCP(C)(C)=O)=O)COCC2)cnc(O)c2ccccc12 Cc1cnn(C)c1S(=O)(=O)N1CCN(CC(=O)Nc2ncc(Cl)cc2Cl)CC1 c1(C(N2CCNCC2)C)cc(Br)c(O)cc1O.Cc1cccc(F)c1-c1cncc(C(C)N)c1 c1(C(N2CC3C(NC(c4scc(C#N)c4)=O)(CC3)C2)=O)cccc2nn[nH]c12 CC(C)C(CC(=O)NCC12CCC(CC1)N(C(c1cncc(O)c1)=O)C2)C(C)C CCCC(CC)CCC(=O)N1CCCN(C(c2ccc(O)c(Cl)n2)=O)C(C)C1 C1(NC(c2cnc(N3CCN(C)CC3)s2)=O)COC2(C1)CN(C(=O)CC#N)C2 c1(CC(=O)NC2(C)CC(NC(C3CC(F)(CO)C3)=O)C2)ccc(F)c(Br)c1 c1(NC2CCN(C(c3cccs3)=O)CC2)nc(Cl)nc2sccc12 C1(NC(CCCCC)=O)CC2(C1)CC(CNC(C1(C(=O)N(C)C(C)C)CC1)=O)C2 Cc1cccc(C(N2CCC(C)(CC(=O)NC(C)C(C)(C)CO)C2)=O)c1C C(=O)(C(CC)C(=O)NCC1CCC(NC(=O)CCc2cccc(O)n2)C1)OCC Cc1cc(C(=O)NC(CNC(c2cc(CF)on2)=O)C(C)(C)C)[nH]c1C n1(CC(N2C3CC(NC(=O)C#CC4CCC4)C2CC3)=O)ncn2nccc2c1=O CC1CCN(c2ncc(C(N3CC(NC(c4csc(Cl)c4Cl)=O)C3)=O)s2)CC1 N1(C(CC=C=C)=O)CCCC(C(C)(O)CNC(=O)Cc2cn(CC)nc2C)C1 c1(OC)ccc2c(c1)CC(C)N(C(c1csc(Cl)n1)=O)C2 c1(OC(C)C)cc(-c2csc(NC(c3ccc(C(C)(C)C)cc3)=O)n2)c(F)cn1 C(C(C(=O)NCc1ccncn1)NC(=O)Cc1cncn1C)OCC Cc1ccc(C(c2ccccc2)NC(=O)NCC(N)C(F)(F)F)cc1 C(=O)(CS(=O)(=O)C(C)C)NC1CCN(C(Cc2ncc(C)s2)=O)C1(C)C C=CCC(C(=O)N1CC(C)C1C(=O)NC(C)C(C)C)OC C(=O)(C(C(C)(C)C)c1ccccc1)N(CC(c1nn(C)c(F)c1)=O)C(C)(C)C CC1=C(C(=O)NCC2CC2NC(c2ccc(C)c(C)c2)=O)CCCO1 C(=O)(C(CO)C(C)(C)C)NC(CCC)CCCNC(=O)CCc1cc(C)n(C)n1 Cc1nc(N(C)C)sc1C(=O)NCC1(NC(c2cn(C3CC3)cn2)=O)CCOC1 c1(CNCC2(CCOCC)CC2)nc(C)nc(O)c1C c1(C(=O)NCCCC(CCC)NC(=O)C(C)N(C)C)ccc2c(c1)C=CCC2 C(=O)(CCC#Cc1ccccc1)NC(C)CCN(C)C(c1ccccc1CO)=O CC(C)C(CCN(C)C(C1CC1(F)F)=O)NC(c1c(Cl)cnn1C1CCCC1)=O C1(CC(=O)N(C(C(=O)OC)C2CC2)CC(F)(F)F)CC(C)CCC1C(C)C N1(C(C(CC)n2nccc2C)=O)CCCC(C)(NC(c2cc(C(C)C)[nH]n2)=O)C1 NS(=O)(=O)CCC(=O)NC1CN(C(=O)Cn2nnc(-c3ccco3)n2)CC1O C1(=CC(=O)NCC(C)N(C(=O)C2=NNC(C(F)(F)F)C2)C)CC2CCC(C1)N2C c1(C(C)=O)ccsc1C(=O)NC(C)CNC(=O)C(c1ccn(C)n1)C c1(C(=O)NC(CC(C)NC(C2CCC(C)(C)O2)=O)C)cc2ccccc2c(=O)o1 C1(NC(C(COC)C)=O)CCSC12CN(C(=O)C=Cc1ccccc1OC)C2 c1(C(=O)NCCCC2N(C(C=CC=CCC)=O)CCCC2)nc(Cl)ccc1N N1(C(C(C)CC2CC2)=O)CC(F)CC1CNC(=O)Cn1nnc(-c2cccs2)n1 CC1(NC(c2ncc[nH]c2=O)=O)CCC(NC(C23COCC2C3)=O)CC1 C1(C(N2CCC(CN(C(C(CC#C)C)=O)C)C2)=O)CCC2(CC1)CC(O)C2 c1(C(=O)NCCSN)nc[nH]c2ncnc1-2.c1(C(CCCN)=O)ccncc1C(F)F n1(CC(=O)NCCC2CC2)cc(SCCCN(CCCNC(COC)=O)C)nn1 C1(NC(CCC(CC)NC(C2CC=C(C)CC2)=O)=O)CCCCC1N=[N+]=[N-] C1(C(N(CC(C)NC(CSCCC)=O)C)=O)CC2(C1)CC(C)(C)C2 C(=O)(CC(C)CC(=O)NC1(CC(=O)NCc2nccn2C2CC2)CCC1)OC C(N=c1[nH]c(SC)ncc1C)C1OCCN(C(c2c(OC)cc(O)cc2)=O)C1 C(CCCC(C)NC(=O)C(C)CCO)NC(C1(C)CC(=C)C1)=O c1(CCNC(CCN(C(C(COCC)C)=O)C)=O)ccccc1F C12(C(=O)NC3C(C)CN(C(=O)Cc4ccsn4)C3)CCCCN1CCC2 c1(C(=O)NCC(C)C(=O)NCc2ccc(O)nn2)ccnc2cc[nH]c12 N1(C(CN(S(C)(=O)=O)C)=O)CCN(C(=O)C=CC2CCCO2)CC(C)(C)C1 C1(C(=O)NCC2N(C(CC3(OCC)CCCC3)=O)CC2)Cc2cc(C)ccc2O1 N#Cc1ccc(C(=O)Nc2sc(-c3cc(OC(F)(F)F)cc(F)c3)nc2C)cn1 C(=O)(CS(=O)(=O)C1CC1)N1C(CCCNC(c2c(C(N)=O)nccn2)=O)CCC1 c1(C(=O)NCCOCCC(=O)N(C(C(=O)OC)C)C)cnc(N)cn1 c1(C(C(=O)NCC(CO)NC(=O)Cc2ccoc2)NC(N)=O)cc(F)cc(F)c1 c1(C(=O)NCC2CC(NC(C3(C(F)F)CC(=C)C3)=O)C2)cccc(C=C(F)F)c1 N1(C(C(C)c2ccsc2)=O)CCN(C(C2C3CC4C(C3=O)C24)=O)CCC1C C1(CC=C)(C(=O)NCC2CCC(C(=O)N(C)CCNC(C)=O)C2)CCOC1 C(=O)(C#CC1CCCOC1)N1CCCC(NC(c2cc(N)c(F)cn2)=O)(CO)C1 N1(C(CCC(CC)OC)=O)CCCC12CCN(C(c1cnn(C)n1)=O)C2 C1(CS(N)(=O)=O)CCC(N=c2[nH]c(=NCC3CC3C3CC3)[nH]c3c2CCCCC3)C1 N1(c2cc(C)nc(N(CC(C)(F)F)C)n2)C(C)C2CCCCC2C1C N1(C(=O)CN2CCCS2(=O)=O)CC2C3CCC(C2C1)N(CCn1cccn1)C3 C(C(=O)N1CC2C(CN(C(=O)CN3CCOCC3)C)C2C1)(C(C)(C)C)SC C1(C)(NC(CCCOCC)=O)CN(C(C2(SCC)CC2)=O)CC1C c1(N2CCC(C)(NC(C3C4CCCC34)=O)C2)ncc(Cl)c(O)n1 N1(C(C=CC)=O)CCn2c(CNC(C3(C)CNC(=O)C3)=O)nnc2C1 C(=O)(CCS(=O)(=O)C(F)(F)F)NC1(C2CN(C(C3N(C)CCOC3)=O)C2)CC1 C1(CC)(Nc2ccnc(OCCO)c2)CC(F)(F)C1 C1(C(N2C(CNC(CC3CC(C)C3)=O)CC(C)(C)C2)=O)Cc2ccccc2N1C C1(c2nnnn2C2CCOC2)(NC2CCN(c3sncn3)C2)CC2CC2C1 C(C)(C)(CCCC(=O)N(C1CC(CO)C1)C)NC(CC1N(C)CCC1)=O CN=c1cc(C(=O)NC(c2cccc(Cl)c2)CNC(=O)C(C)=C2CC2)cc[nH]1 N1(C(C(CC)C)=O)CC2(CCN(C(C3(c4cccc(C)c4)CC3(F)F)=O)CC2)C1 C1(CC)(NC(=O)CCc2conc2C)CCCN(C(=O)C(C)N2CCC2)C1 c1(CNC(=O)C(=O)NCC2COCCN2Cc2ccccc2)cc(O)cc(Br)c1 C1(C(=O)NC2C(NC(C3(C#N)CCOC3)=O)C2)CCCCCCC1 C(=O)(C#CC1CCOC1)N(CCCCCNC(C12CCC(CC1F)C2)=O)C c1(C(N2CCCCCC(NC(CC=C(C)C)=O)C2)=O)[nH]nc2c1CCCC2(C)C c1(C(N2CC(NC(c3ccc(OC)cc3)=O)C(F)C2)=O)cccc(Cl)c1Br c1(C(=O)NCC2CN(C(C(COCC)(C)C)=O)CC2C)cc(C)cc(Cl)c1N N1(C(=O)C=C2CCCC2)CC2(C1)CN(C(c1ccnnc1O)=O)C2 Cc1cc(F)ccc1C(O)C(=O)NC1CC(C)N(C(C2CCC=CO2)=O)C1 CC1(CNC(C23CSCC2C3)=O)CCCN(C(c2ccc(O)nc2)=O)C1 N1(CCNC(C2CCC3CCC23)=O)CCCN(C(c2cccnc2)=O)CC1 N1(C(Cc2nc(-c3ccc(OC)cc3)sc2)=O)CC2(CCC2NC(=O)CCF)C1 Cc1ccc(C=CC(N2CCCC(C)(C)C2CNC(C2CC23CC3)=O)=O)cc1Cl C(=O)(C1=C(C)OCCC1)N(C1C(N(C(CCCC#C)=O)C)CCCC1)C c1(C(=O)NCC(CC(C)C)NC(C2CC(O)C2)=O)ccc2occc2n1 CCCC(C)(O)CC(=O)N1CCN(C(c2nccnc2CC)=O)CC1CC1CC1 C(=O)(C(F)C(C)(C)O)NCCCOCCN(C(CC(C)N1CCCC1=O)=O)C C1(C)(NC(C(CCNC(c2cncc(O)c2)=O)OC)=O)CCCC1(C)C c1(CC(=O)N(C2CCN(CC)C2)C)nc(C)c(C)[nH]1 N1(C(COCCN(C(=O)CCOC2CCC2)C)=O)CCN(C2(C)CC2)CC1 N1(CCOC)CCC(C(=O)NC(C2CCOC2)CNC(c2nc(Cl)cs2)=O)CC1 C1(CNC(C2CC(C)C2)=O)CN(C)CCN1C(c1cnns1)=O c1(COCC)nc(C(=O)NC2CCC(CCNC(C34CC(C)(C3)C4)=O)C2)cs1 C1(CC)CCC(C)CN1C(=O)CCCN(C(=O)Cc1cccn1C)C c1(C(=O)NC2CC(C)N(C(c3cnc(O)s3)=O)CC2)cccc(S(C)(=O)=O)c1 c1(CC)nnc2n1CCCC2C(=O)N1CC(NC(C2CN(S(N)(=O)=O)C2)=O)C1 c1(C(=O)NC2CCN(C(=O)COCC3CCCO3)C2)c(Cl)cc(F)cc1Br C(=O)(CCC(=C)Cl)NCCCC(C)NC(C1(CC#C)CCOC1)=O C1(C)(NC(=O)Nc2n(C)ccn2)CCCN(C(=O)C(CO)Nc2ccccc2)C1 CCCCCCC(C)C(=O)N1CCCC1CNC(=O)CCNC(c1ccsc1)=O N1(C(C=C(C)CNC(c2cnc(S)nc2)=O)=O)CCC(C)OC(C)C1 N1(C(c2cnc(C)s2)=O)CC2(CNC(=O)C(F)n3ccnc3)CCC1CC2 c1(C2C(n3c(-c4cnn(C)c4Cl)nc(CC(C)(C)C)n3)C2)ccc2ccccc2c1 c1(CS(Oc2c(C#N)cccc2)(=O)=O)ccc2c(c1)OCCO2 Cc1cc(C)c(C(=O)NCC(C)(O)CNC(=O)C(O)CCN(C)C)c(N)c1 C1(CC(=O)NCC(CC)(CC)OC)CC2(C1)CN(C(=O)CCc1ccn(C)c1)C2 n1(Cc2ccc(C)cc2)cc(C#CCNC(c2cc(Cl)cc(Br)c2F)=O)nn1 Cc1ccc(C(=O)NCCc2ccc(C(=O)NCc3ccncc3)cc2)c(O)n1 c1(CC)ccc2occ(C(=O)NC3CCC(NC(=O)CCn4ccnn4)C3)c2c1 N1(C(COCCCOC)=O)CC2CCC1C2NC(=O)Cn1ccc([N+](=O)[O-])n1 c1(C(N(CC(OC)OC)CC(C2CC2)OC)=O)cc(Cl)ccc1C c1(CC(=O)N(CCCCN(C)C(c2cc(Cl)cs2)=O)C)nc(C2CC2)cs1 c1(NC(C2CC2c2cccc(-c3cnn(C4CCC4)c3)c2)=O)cc(F)cc(Cl)c1 c1(C(N2C3CN(Cc4cc(Br)cc(Br)c4F)CC23)=O)cc2n[nH]cc2cc1Cl C1(Oc2ccc(-c3n(CCC)nc(C)n3)cc2)Cc2ccc(Br)cc2C(=O)O1 C1(N(C)C(c2ccn(-c3ccccc3)n2)=O)CCC(NC(c2cc[nH]c2)=O)CC1 C1(C(=O)NC(C#C)C(C)OC)C2CC(O)C(C2)N1C(C1CCC2(CCC2)C1)=O N1(Cc2cc(C(=O)OCC)[nH]c2)CC(C)(C)OC2(CCOC2)C1 C(=O)(CC(C)(C)O)N(CC(=O)NCCOCCCC)C1CC1 O=C1CN(CCCN(S(=O)(=O)CC2CCC(C(=O)O)C2)C2CC2)CCCN1 CC(C(C)(C)C(=O)NCC1CCCOC1)NC(C1COCCC1C)=O N1(C(C(C)OCCOC)=O)C2CCC(C2)C1CC(=O)NCC(C)CC(=O)OC C(c1ccc(OC)cc1)=CC(=O)NC(CCCC)CNC(=O)CC(C)OC C1(NC(c2n(CCC)ncc2)=O)(CNC(c2scc(C)c2C)=O)CC2CCC1C2 C1(n2cc(CN3CCC(N(CCC)CCO)CC(N)C3)nn2)C2CS(=O)(=O)CC12 N1(CC)CC2(CN(C(=O)CC=CCNC(=O)CC3CCCOC3)C2)C1 N1(C(=O)CC2C3CCCC3N2C(=O)CC2CC(F)(F)C2)CCc2n[nH]cc2C1 CC(CC(F)F)C(=O)NCC(c1ccccc1F)NC(c1n[nH]cc1Br)=O c1(OC)c(C(=O)NC(CO)C(C)NC(=O)Cn2ncn(C)c2=O)cc(Cl)cc1Cl CN1CCC(C)(C(=O)NCC2(C(C)(C)C)CCN(C(=O)OC(C)(C)C)C2)C1=O c1(OC)ccnc(C(N2CC(N3CC(CC4CC4)CC3=O)C2)=O)c1O C1(CNC(c2c(Cl)cn(C)n2)=O)CC2(C1)CN(C(=O)COC1CC(F)(F)C1)C2 c1(C(=O)NCC(C)CN(C)C(C23CC(CO)(C2)C3)=O)cnccn1 C(=O)(C1=NOC(C)C1)N1C(C(=O)NC(C(=O)OC)CC2CC2)CC(O)C1 C1(OC)CN(C(=O)C(C)SC(C)C)CCC1NC(c1ccc(C(N)=O)[nH]1)=O C1(NC(c2cnc(OC)s2)=O)CN(C(=O)C(C)(C)C2CC2)CC(C)(C)C1 c1(C(=O)NCC2CCCN(C(CSc3c(C)noc3C)=O)C2)cc2[nH]ccc2s1 C(C(C)CC(C)C)NC(C(COCC)NC(=O)CC1CCSC1)=O CCC1=NOC(CC(=O)NCC2CCCCN2C(c2cc(C(=O)OC)cs2)=O)C1 C(=O)(CC(O)c1ccccc1)NCCC(C)NC(=O)C(c1cscn1)N(C)C c1(C(N(CC(C)NC(=O)C(C)CCCOC)CC)=O)ccc2nc(C)sc2c1 C1(CNC(c2ccc(C)nn2)=O)COCCN(C(C2CN(C3CCOC3)C2)=O)C1 N1(C(=O)OC(C)(C)C)CCC2(COC(COC(c3n[nH]c4c3CCCC4)=O)C2)C1 c1(OC)cc(OC)c(C(=O)NCC2C=CCN2C(C2CC3(C2)CC(O)C3)=O)cn1 C1(NC(c2cc(C)c(C)nn2)=O)COC2(C1)CN(C(c1ccc(Br)o1)=O)C2 C1(C(=O)NCC(=C)CCN)CC(N=[N+]=[N-])C1 C1(NC(C(C)OCC)=O)CN(C(=O)CCC(C)(C)F)CCC12CCC2 Cn1ccc(CCC(=O)NC2CC(NC(=O)C=CC(F)(F)F)C2)c1 N1(C(C2C(OCC)C2)=O)CCCC2CN(C(=O)CSc3nccn3C)CC12 N1(C(C=CC)=O)CCc2ccccc2C1CNC(c1sc(Br)cc1F)=O C(=O)(C1=CCC(C)CC1)N1CC(NC(c2c(C)nc(C(C)(C)C)s2)=O)(CO)C1 N1(C(c2cc(C)cc(F)c2N)=O)CC2CCCC(NC(C3CC34CCC4)=O)C2C1 C1(CNC(Cc2c(C)cc(C)s2)=O)N(C(=O)CC2CC2C2CC2)CCCC1(C)C N(C1c2ccccc2CC12CCC2)C(c1cc(=O)n2ccsc2n1)=O N1(C(CC2(CSC)CC2)=O)CCC2CCC(C1)N2C(=O)C(c1nc(C)cs1)C C1(CCCC)CCC(C(c2ccc(F)cc2)NC(CN)CC)CC1 CC(C(=O)N1CCCC(CNC(=O)C(C)(C)n2cc(Br)cn2)C1)C(F)F C1(C(=O)NCCNC(Cc2c(OC)c(F)ccc2)=O)CCCCC(C)(C)C1 N1(C(c2c(C)con2)=O)CC2CS(=O)(=O)CC2(CNC(=O)C2=CCS(=O)(=O)C2)C1 c1(C(=O)NCCNC(CCC)=O)sc2ccc(Br)cc2c1C N1(C(c2cc(F)c(O)c(F)c2)=O)CCC2(CCCN(C(c3coc(O)n3)=O)C2)C1 C1(N(C(C2(CCNC(C=CC)=O)CC2)=O)CC)C=CCCCC1 C1(N(CCCC)C)CCCN(c2nnc(C3CCOC3)n2CC(OC)OCC)C1 N1(C(CC2C(C)OCC2)=O)CCCN(C(=O)CCCN2CCN(C)CC2)CCC1 c1(NC2CN(C(C(CC)CC3CCCC3)=O)CC2C)[nH]c(=O)n(C)c(=O)c1C#N CCC(C(=O)NCCCN(C(C1(CCO)CC1)=O)C1CC1)C(C)(C)CC c1(OCC)ccc(C(=O)NCCCC(CO)NC(=O)C(O)c2ccsc2)cc1 C1(N(C(=O)Cc2scnc2C)CC)CCCN(C(c2csc(S)n2)=O)C1 N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CCC(O)(CCNC(C2CCC3(CC3)C2)=O)C1 N(C(=NCCC1COC1)NC1CC12CC2)Cc1cn(C)nc1 N1(C(C2(CC)CCCC2)=O)CCC2(CCC2)C(CNC(C2C=CC=CC=C2)=O)C1 c1(OCC)cccc(CC(=O)NC2CCC2NC(c2cc(C)c(C)[nH]2)=O)c1 n1(CC)cnc2c(NC(C)Cn3cccn3)[nH]c(=NC(C)C3CC3)nc12 N1(C(=O)OC(C)(C)C)CCC(O)C(C(=O)NCCNCc2ccc(=O)oc2)C1 Cc1c(C(N2CCN(CCCCCNC(C3(O)COC3)=O)CC2)=O)cccc1Cl c1(C(=O)NC(C(C)(C)NC(C(C)N(C(C)=O)C)=O)C)ccc(S(N)(=O)=O)nc1 CC1c2cccc(F)c2CCN1Cc1sc(Cl)cc1Br C1(CC(=O)NCC(C)OC(F)F)CN(C(=O)COC2CCCCCC2)CC12CC2 c1(CC(=O)NC2CC(CO)N(C(c3ccc(Cl)[nH]3)=O)C2)ccc(F)cc1F C1(C(N2CC3C(NC(C(C)(C)C(N)=O)=O)(C3)C2)=O)CC(c2ccccc2F)=NO1 C(=O)(C(F)CCC(C)(C)C)NCC12CCN(C(COCCN(C)C)=O)C1CCC2 c1(C(=O)NC(CC)C(C)O)cnn2cccc(-c3cc(OC)ccc3O)c12 C(=O)(CC(O)C(C)C)NCC1N(C(CNS(CCCC)(=O)=O)=O)CCC1CC Cc1cc(C(N2CC=C(C(=O)N3CC(n4cc(C)cn4)C3)C2)=O)nc(C)c1 C(=O)(C(CC1CCCC1)NC(=O)CC)N(CC(C)N(C(CSCCC)=O)C)C c1(OC)ccc(CC(=O)NCC2(O)CN(C(C3(C)COC3)=O)C2)cn1 C(=O)(C(C(=O)N(CCNC(c1n[nH]c(C)c1[N+](=O)[O-])=O)CC)C(C)C)OCC c1(CCNC(C(C)NC=O)=O)nc2ccc(Cl)cc2[nH]1 Cn1ncc(C(F)(F)F)c1C(N1CCN(C(=O)Cc2csc(NC=O)n2)CC1)=O N1(C(C(C)C)=O)CCC2CCN(C(c3cnn(C4CC4)c3)=O)CC2C1 c1(OC(C)C)c(-c2cnc(C(=O)NCC3CC3)nc2)ccc(F)c1F C1(NC(C(CC)NC(C)=O)=O)CCCC12CN(c1nc(Cl)ncc1C(N)=O)C2 c1(C(N2CCC(CSC)C2)C(=O)NCC(=C)C)ccc(SC)o1 c1(C(=O)NC2CC3(C(NC(CC(C=C)CCC)=O)C3)C2)cc(F)cc([N+](=O)[O-])c1 N1(C(c2c(SC)ccs2)=O)CCC(F)(CNC(=O)C(F)C2CC2)CC1 c1(CC(N2C(C)C(N3CCCCC3)CC2)=O)cc(F)cc(F)c1F c1(C(C)NC(c2csc(CNC(C3CCNC3=O)=O)c2)=O)c[nH]ccc1=O CC1CCC(NC(=O)C(C2CCCCC2)N(C)C)CN1CC1C2CC3C(C2=O)C13 c1(C(N2CCC(C)C2CNC(=O)CNC(=O)CC(C)(C)C)=O)coc2c1COC2 c1(C(=O)NC(CC)CNC(=O)CN2CCC(C)C2)cc(Cl)c(C)cn1 C1(C(N2CC(O)(CNC(C3CN4CCN3CC4)=O)C2)=O)CCC(F)(F)CC1 Cc1cc(C(=O)NC2CCCC2NC(C2CN3CCC2CC3)=O)ccc1O CCC(C)(CC(=O)N1C2CCCC1CN(C(=O)C=CCCC(C)C)C2)C(=O)OC c1(C(N2CCC(C)(NC(C=CSC)=O)C2)=O)c(Br)cncc1[N+](=O)[O-] N1(Cc2cccc(C(=O)OC)c2F)CCC2(CC1)OCc1ccccc12 c1(N2CCC(C(F)(F)F)(CC)C2)nc(=NCCC2(C)CC2)[nH]c2c1CCCCC2 c1(OCC)cccc(CCc2nnc(C)n2CCCCO)c1 N1(C(C(C2(OC)CCCC2)N)=O)CC(C(F)(F)F)CC(c2ccccc2)C1 C1(NC(CCCCCOC)=O)CC12CCN(C(c1cc([N+](=O)[O-])n(C)n1)=O)CC2 C1(C(C)C)CC(O)CN1N(C)Cc1nncn1CC c1(C(N2CCN(C(c3n[nH]cc3Br)=O)CC2)=O)cccn(CC(F)(F)F)c1=O C1(C(=O)NCC(CO)NC(c2cnc(C(C)(C)C)s2)=O)C(F)(F)C12CCC2 CCC(CC(C)C)C(=O)N1CCCC(C(=O)N(C2CCC2)CCC(F)F)CC1 c1(C(N2CC(CNC(c3c(OC)cc(C)cn3)=O)C2)=O)nccn2nc(C)cc12 C=C1CC2(C1)CC(C(N1CC3CC(NC(=O)C4=CC(C)(C)C4)C1C3)=O)C2 C1(C(=O)NCc2occ(C(=O)NCc3nc(C)oc3)c2)CN(C)CCO1 c1(C(=O)NC(C)CC(C)NC(c2ccco2)=O)cc(Cl)ccc1OC(F)F Cc1cnc(NC(C2C(C(C)C)CCN2C(=O)COCc2nc[nH]n2)=O)nc1 c1(SC)nc2ncnc(N(CC(C)NC(=O)CC3NC(=O)NC3=O)C)c2s1 c1(C(=O)NC(CNC(C(C)OCC)=O)CO)c(C)nc(C)nc1C N1(C(C(C)CC2CC2)=O)CCCOC(CNC(=O)Cc2cc(C(F)(F)F)n[nH]2)C1 N1(C(C2C(NC(C(C)(C)OCC)=O)CC2)=O)CCCC(CC(N)=O)C1 N1(C(CCCCC(=O)NC)=O)CC(C2CCN(C(C3CC3(C)C(F)F)=O)CC2)C1 C1(NC(C=CCN(CC)CC)=O)CN(C(=O)CC2CC(N(C)C)C2)C(C)(C)C1 C1(NC(C(C)(C)C#N)=O)CC(NC(=O)Cn2nnnc2-c2ccsc2)C12CCC2 C12(CNC(C3CCC(CSC4CC4)C3)=O)CC(CO)(C1)OC21COC1 CC1CC=C(C(=O)NC(CO)CCCCNC(c2cn3ccnc3s2)=O)CC1 S(=O)(=O)(c1cc(C(N2CCCC2CN(C(=O)C(F)C(C)C)C)=O)ccc1F)NC c1(N2CCC(N(C(C)=O)C)CC2)nc(NCCCCCF)c2ccsc2n1 N1(C(C(CN(C)C)NC(CCC(C)OCC)=O)=O)CCOC(C#N)C1 C(=O)(C(F)CC(C)(C)C)NCC1OCC(C(=O)NC(C(C)O)C(N)=O)C1 N1(C(c2cc(OC)no2)=O)CCCN(C(=O)CC(c2ccccc2)N(C)C)CC1 S(=O)(=O)(c1cccc(N2CCC(CCO)C2)n1)NCCCCN(C)C c1(CC)cc2c(c(=O)o1)C(c1c(Cl)scc1Cl)NC(=S)N2c1ccccc1Cl C(=O)(C(C(=O)OC(C)(C)C)C(C)C)NC1(CCCNC(c2c(C)ocn2)=O)CC1 N1(C(C(n2ccc(C)n2)C)=O)CCC(C(=O)NCC(C)S(N)(=O)=O)CC1 C(N=c1[nH]c2c(c(=NCC(C(C)(C)C)SC)[nH]1)CCCCC2)c1c(CC)n[nH]c1 C1(NC(CCCC)=O)CN(CC(=O)Nc2ncccn2)CC1(C)C C(CCCCCCO)NC(=O)CCc1ccoc1.C12(CC1)N(C)C(=O)N2 n1(CC)nc(C(=O)NCC2(C)CCC(NC(=O)CN3CCC(F)CC3)C2)cc1C C(=O)(C1=CCCCC1)N1CC(N(C)C(C2CCCCN2C2CCCC2)=O)C(O)C1 N1(C(C(C)SC)=O)CCC(C(C)CNC(c2cc(Cl)nn2C)=O)CC1 c1(C(=O)NC2(C(=O)NCC(C(CC)C)OC)CC2)ncc(C)cc1F C(=O)(CC(CC(C)C)NC(=O)CCCCOC)NC1CCCC(C=C)C1 CC1CCC(O)(C(=O)NCC2CC(O)(CNC(=O)CCCOC(C)C)C2)CC1 N1(Cc2c(Cl)nc(NC(C)=O)s2)C2C=C(c3ccccc3)CC1CC2 C(C)(C)(CCC(F)F)NC(c1cccc(Br)c1)C N1(CC=C)C(=S)NC(c2sc(Cl)nc2Cl)C2=C1CCN(c1ccc(F)cc1)C2=O C(=O)(C(C)CC(C)C)N(CCC(=O)NCCc1ccnn1C)CC#C CCCC(C(=O)N1CCN(C(c2cc(N)c(C)cc2Cl)=O)C(C)C1C)C(C)C c1(NC(C(CC)NC(=O)C=Cc2cscn2)=O)ccc2c(c1)OCO2 CC(C)(CC(=O)N1CCC(C)(CCNC(C23CCN(CC2)C3)=O)C1)CC(F)F C(CNC(c1sccc1C#N)=O)(CC(F)(F)F)NC(CN1CCC(C)CC1)=O c1(CC)onc(C(N2CCCC2C2CCN(C(c3c[nH]c(Br)c3)=O)C2)=O)c1C c1(CNC2CCC(C#N)C2)c(F)ccc(Br)c1F c1(C(N2CC(O)CC(NC(CSCCCC)=O)C2)=O)nc(C)c(C)nc1C c1(C(=O)NCC(CC)(CC)NC(=O)C(C)CO)cncc2ncccc12 Cc1cccc(C(F)(F)C(=O)NC2CC(CNC(=O)Cc3cncc(O)c3)C2)c1 Cc1nc2cc(C(=O)NC3CCC3NC(c3n[nH]c4c3CCC4)=O)ccc2s1 C(=O)(C1=CCCC1)NCC(C(C)C)NC(C(C)NC(=O)NC)=O C1(CCNC(C2(OC)CC2)=O)CCN(C(=O)Cc2cncnc2O)C(C)C1 CC(C)(C)C(CC(=O)NC1CN(C(=O)CC(F)(F)F)CC2CC12)C(F)F Cc1cc(C(=O)NC(C)C(c2ccccc2)NC(c2cccs2)=O)nc(O)n1 C1(N(C(c2cnccn2)=O)CC)CCCN(C(=O)C(C)n2cnnn2)C1 c1(C(C(=O)NCCC)N(c2cnn(C)c2)CC)cccnc1CC Cc1ccn(CC(=O)NC2(CC(=O)NC3CSC3)CCC2)n1 C1(NC(C2C(OCC)CCC2)=O)CC2CC(C1)N(C(c1ccc(F)cc1)C)C2 N1(C(c2c(C)c[nH]n2)=O)CC(NC(c2cc3occc3[nH]2)=O)CC(F)C1 Cn1nccc1C=CC(=O)NC1(C(N2CCC(C(F)(F)F)C2)=O)CCSC1 C(=O)(CC(C)CC(C)C)N(C1CN(C(c2ccc(C)c(C)n2)=O)CC12CC2)C C(C(=O)N(C)Cc1ccncc1)(C(C)(C)O)NC(C(C)=C1CC1)=O c1(C(=O)NC2CC(OC)CN(C(COCCSC)=O)C2)cnc2ncc(Cl)cn12 C1(NC(=O)NCC(=O)OCC)CCC(CC(C)C)CC1.N12CCCC(C1)C2=O N1(C(=O)C=Cc2nccs2)CCCCC1CCNC(C1(c2nccs2)CC1)=O