SMILES CC1(N)CCCC1(F)F.n1(CC(N2CCC2C2CCC2)=O)cc(C2CCCOC2)nn1 N#CC1(C(N2CCCC(N3CCN(C(C4(F)CCCC4)=O)CC3)C2)=O)CCOC1 C1(C)(CNC(C(C)CSCc2ccccc2)=O)CN(C(=O)COC(F)(F)F)CCO1 N1(C(C2C=CCN(C(CCCC(C)(C)C)=O)C2)=O)CCC2(CNC(=O)N2)C1 C1(CNC(c2nc(C)sc2)=O)CCC2(CN(C(c3ns[nH]c3=O)=O)C2)O1 c1(C(N2C(CNC(C(CSC)O)=O)C=CC2)=O)cn(C2CC2)c(C)cc1=O Cc1cc(NC(=O)C=CC(C)NC(c2c(C)cccc2O)=O)cc(Cl)c1 c1(OC)c(F)ccc(NC(N2CC(O)CC2CN)=O)c1F N1(C(C2N(CC#C)CCC2)=O)CCC(NC(c2c(C)cccc2Cl)=O)CC1C CCCC(C(=O)NCCC1CCC2CC12)NC(C1C=CCC1)=O C(=O)(C(C(C)C)NC(=O)CCCc1cnn[nH]1)NCCC C1(NC(c2c(C)[nH]cc2)=O)CCCN(C(=O)C(C(C)C)NC=O)C1 N1(C(CC(C(C)C)O)=O)CC2(CCCC(CNC(C3CC4C=CC3CC4)=O)O2)C1 N1(C(C(CC=CC)C)=O)C2COCC1CC(NC(C1(C)CCNC1=O)=O)C2 C(=O)(C1=CCCO1)N1C(C(C)(C)CNC(=O)C(C2CC2)C2CC2)CCC1 c1(C(=O)NC(CC)CNC(c2cnn3c2CCC3)=O)cc(F)c(C)cc1Cl C1(CC)(NCC(c2csc(=N)[nH]2)=O)CCCC1 CC(CCc1ccco1)N=c1[nH]c(=N)[nH]c(=NC(CCO)C2CCC2)[nH]1 c1(N2CC(CC(C)NC(C3C(OC)CCC3)=O)C2)ncc([N+](=O)[O-])cc1CO CON(C)CC(O)Cn1cc(-n2cc(C3CC(=O)N(C(C)C)C3)nn2)cn1 C#CCC(C)C(=O)N1CCC(C)(NC(c2ncn(C(C)(C)C)n2)=O)C1 c1(C(=O)NCCN(C)C(C2CCCCC2C(C)(C)C)=O)ccncc1N N1(C(C(COC)C)=O)CCN(C(c2ccnnc2S)=O)CC1CF c1(C(N2CC(CCCNC(CCC(C)SC)=O)OCC2)=O)cc(O)ccc1Cl c1(C(=O)OC)c(=NC(=O)CC2CC2)[nH]n2cccnc12 c1(C(N2CCC(O)(CCNC(c3cn(C)c(O)n3)=O)C2)=O)cc(Cl)c(F)c(Cl)c1 C1(C(N(C)C)=O)(COC(c2cncc(-c3ccoc3)c2)=O)CCCOC1 C1(CNC(CC(CC)C2CCC2)=O)CC2CCC1N(C(C1CC1C#N)=O)C2 c1(C(=O)NC2CC(CNC(C(COC)N(C)C)=O)C2)ccc(C)cc1SC N1(C(=O)NC(C)COc2ccccc2)CC(C2CC2(F)F)C1 C(=O)(CCCCC(F)(F)F)N(C)CC1CN(C(=O)CSCC2CCCO2)CCO1 C1(CNC(C(CC)(C)C)=O)CN(C(C2CN(CC(F)(F)F)C2)=O)CC1(F)F C1(CNC(C(CCC)OCC)=O)CC2CCCC2N1C(c1ccoc1CC)=O N1(C(CCNC(=O)OC)=O)CC(NC(c2cc(C(F)F)nn2C)=O)C(C)C1 N1(C(CC2N(S(CC)(=O)=O)CCC2)=O)CCC(C)(CNC(c2ccsn2)=O)C1 N1(C(C2CC(CC)(CC)C2)=O)CCCC(C)(NC(C2C3CCCCCC23)=O)C1 c1(NC)cc(C(=O)N(C2CCC(NC(C3CN(C)C(=O)N3)=O)CC2)C)cc(Cl)n1 c1(C(N2CCCN(C(C3CCN(C)C3)=O)CCC2)=O)coc2c1C(=O)NCCC2 c1(C(=O)NC2C3CN(C(c4n(COC)ncc4)=O)CC2C3)cnc2[nH]ccc2n1 c1(CC)oc(C(=O)NC2CCC(F)(CNC(C3(O)CCOC3)=O)C2)cc1C c1(NC(=O)NC(CC(=O)OC)c2ccccc2)ccc(S(N)(=O)=O)cn1 c1(C(N2CCC(NC(c3cnc(SC)n3C)=O)C2C)=O)ccc2c(c1)COC2 c1(OCC)ccc(N=c2c([N+](=O)[O-])c[nH]c3ccc(F)cc23)cc1C(F)(F)F N1(C(C(C)(C)CF)=O)CCC(C2CCN(C(=O)Cc3ccco3)CC2)C1 CCCCC(C)(F)C(=O)NC1CCN(CCNC(=O)C(F)=CCCF)CC1 c1(C(NOCC(=O)N(C2CC2)Cc2n(C)cnc2)=O)cnc(Cl)n1C N1(C(COCC(C)C)=O)CCC(C(=O)N(C2CCC(C)C2)C)CC1 N1(C(C2(C#C)CCCC2)=O)C2CCC1C(C)C(NC(C1CC1C)=O)C2 CC(CC(=O)N1CCN(C(=O)C=Cc2ccc(O)cc2)C(CO)C1)C(F)F C1(C(=O)NCCCC(C)NC(C2COCCN2C)=O)Cc2ccncc2N1 C#Cc1cccc(CC(=O)NCC(C(=O)N2CC(O)(COC)C2)SC)c1 Cc1cc(C(=O)NC2CCCC2NC(=O)C(O)c2ccsc2)cn(C)c1=O C(CS(=O)(=O)CC(=O)N1CC(NC(=O)CSc2cnn(C)c2)CC1C)OC CCCCC(C(=O)N(CCCO)CCC)NC(c1ccc(C(N)=O)[nH]1)=O N1(C(CC(CC)SC)=O)C2CCCC1CN(C(=O)Cc1cccc(OC)c1Cl)C2 C(C(=O)N1CCN(C(=O)CC2(C)CCCC2)CC1C)(C(F)(F)F)OC(C)=O C(=O)(CCCC(=O)N(C)CC1CN(c2ncccc2C(C)=O)C1)NC N1(C(CC(=O)NCC#C)=O)CCC(C)C(N(C(=O)C(=O)NCC)C)C1 C(CCCCC(=O)NCCC1(O)CN(C(C2CC2C(=O)NCCO)=O)C1)N(C)C CC1CC(CNC(=O)Cn2cnnc2)CN1C(C1CC(F)(F)CS1)=O N1(C(=O)CSc2ccccn2)CC2=C(C1)CN(C(C1CCCN1CC1CC1)=O)C2 N1(C(C2(CC#N)COC2)=O)CCCC1CNCC1(C2CCCO2)CC1 Cc1cc(C2CCC2)ccc1C(=O)NCC1(O)CN(C(=O)C(C(C)C)N(C)C)C1 C1(CC(F)(F)F)(NCC(=O)NCC2CCCC2)CCCC1 C1(C)(COC)CC(NC(c2ccn(C)c2)=O)CN1C(=O)CC1(C)CCOCC1 N1(C(COC2(C)CN(C(=O)CS(N)(=O)=O)C2)=O)CCN2CCOCC2C1 C1(C(=O)Nc2ncc(C)s2)CC(F)CN(C(c2cc3ccoc3s2)=O)C1 CCC(C)(C#N)C(=O)N1CCC(O)(CCNC(c2nnn(C)c2C(F)F)=O)CC1 C1(NC(C(CC)CC)=O)CCCN(C(=O)Cn2ccccc2=O)C1CC C(=O)(CCS(C)=O)NC(C1(O)CN(C(=O)Cc2ccc(F)cc2)C1)C C1(F)(C(=O)NCC(CC)n2cccn2)CCCN(C(=O)C(CC2CCC2)OC)C1 Cc1cccc(NC(=O)CC2CCN(C(=O)C(O)C(C)C)CC2)c1O C1(F)(CNC(=O)CCC2CC2(F)F)CCC(NC(c2cccnc2O)=O)C1 Cc1cc(F)c(C(=O)NCC(F)CNC(=O)COCCc2ccccc2)c(Cl)c1 N1(C(c2nccc(C)c2)=O)CC2CC(NC(C3CC(=O)N3)=O)C2C1 C(C(N=[N+]=[N-])C(=O)NCC(O)CNC(c1cnc(C2CC2)s1)=O)OCC C(CC(C(=O)NCc1cnc(C)n1C)NC(=O)Cc1ccc(C)cn1)=CC c1(C(C(=O)NC(C)C)N(C(C)C(C)C)CC)ccc(Br)c(F)c1 C1(C(=O)NCC2(NC(C3CN(C(=O)NC)C3)=O)CCOC2)CCCCN1C c1(-n2cc(C(=O)NCCS(N)(=O)=O)nn2)nc(O)c2sccc2n1 C#CC1CCN(C(C2C(NC(C3(SC)CC3)=O)C2(C)C)=O)C1 N1(C(C(CC#C)NC(c2oc(C)cc2C)=O)=O)CCC2(CCCOC2)C1 CCCC(C(=O)NCC12CC1CN(C(c1cc(C)ccc1N)=O)C2)S(N)(=O)=O Cc1cc(CC(=O)NCC2CN(C(C3C=CCC3)=O)CCO2)n(C)n1 C1(CNC(C(F)=CCC)=O)CN(C(C)=O)CC12CCOCC2 c1(OCC=C)ccc(CN(C(=O)Cn2cc(C(O)CC)nn2)C)cc1 N1(C(COCc2cc(C)on2)=O)CC2CCC1C2NC(=O)Cc1nc(C)sc1C Nc1cc(Cl)c(Cl)cc1C(=O)NC12CC(C1)N(C(=O)CSc1n[nH]c(O)n1)C2 N1(C(C2(OC)CCCOC2)=O)CCC(C2(NC(c3ccncc3)=O)CCC2)CC1 N1(C(CCC(C)=O)=O)CCC(C(F)(F)F)CC1CNC(C1CN(C)CCO1)=O c1(CC(=O)NCCC2(OC)CN(C(=O)C(N)=O)C2)cc(F)ccc1O CC(C)(CCCCNC(=O)C(CC(F)(F)F)C(C)(C)C)C(=O)NNC(=O)C1CC1 c1(-c2cccc(C)c2)nc(=NC2CC(NC(C3C=CCCC3)=O)C2)s[nH]1 C1(C)(CNC(c2c(CC)occ2)=O)CC(F)(F)CN1C(=O)COCC1CCCC1 C(S(=O)(=O)CC1CS(=O)(=O)c2ccccc21)c1nc(-c2ccc(OC)cc2)oc1 O=C1CCN(Cc2nnc(C3CCC3)s2)C(=O)N1CCC1=CCCCC1 c1(-c2ccc(C(CC(=O)OCC)NC(=O)C3=CCCC3)cc2)ccc(C=O)cc1 Cc1cc(Cl)cc([N+](=O)[O-])c1C(=O)NC1CC(O)CN(C(=O)C2=COCC2)C1 N1(C(CN2CC(C)(OC)C2)=O)CC(C)N(C(c2cc(C)n(C(C)C)n2)=O)CC1C Cc1c(Cl)cc(C(=O)Nc2ncc(CCNC(c3ccc(I)c(F)c3)=O)s2)cc1Cl N1(C(C(COC)NC(C)=O)=O)CCN(C(=O)C(C)N(CC(F)(F)F)C)CC1 C1(C)(CNC(C2(C(C)C)CC2)=O)CCCN(C(C2NC(=O)OC2C)=O)C1 C(CCC1CCC1)(C(=O)NOC(C)CC)NC(C(CC=CCC)C)=O C1(C(=O)NC(C)CC2CCC2)CCn2ccnc2C1 c1(CNC(CN(C(=O)NCC(C(F)(F)F)OC)C)=O)ccc(F)cc1F N1(C(C(CCCC)C)=O)CC2COCC2(C(=O)N(CC(O)COCC)C)C1 N#Cc1ccc(C(=O)NC2CC23CCC(NC(=O)CC2CC=CC2)CC3)c(F)c1 c1(NC(C)=O)ccc(CC(=O)N(C2CN(C(=O)COC(F)F)C2)C)cc1 C(=O)(C1CCc2nccn21)NCC1CCN(C(CCCOC(C)C)=O)C1 c1(OC)ccc(C(N2CCCC(O)(CNC(=O)CN(C)C3CC3)C2)=O)cc1C Cc1ccc(Br)c(C(N2CCOC(C(=O)Nc3cscn3)C2)=O)c1F Cc1cc(-c2ocnc2C(=O)NCC2CCC2NC(=O)CCC2CCCC2)on1 CN1CCc2cc(C(=O)NC(CNC(=O)CCn3cnnn3)CO)sc2C1 C1(C(=O)NCC(CC)n2cccn2)(OC)CCN(C(=O)CN2CC=CC2)C1 C1(CNC(=NCC)NCCc2coc(C)c2)C2CC3CC(C2)CC1C3 C12(CNC(c3cccnc3CO)=O)CC(CO1)N(C(C1CCCS(=O)(=O)C1)=O)C2 C1(CCNC(CC(CC2CC2)NC(CC2C(CC)C2)=O)=O)CCCC2(CCC2)C1.C C1(NC(CC2CC(OC)C2)=O)CCCN(C(c2ccc(C(F)(F)F)[nH]2)=O)C1C C1(CN(CC(=O)NS(C)(=O)=O)C(=O)C2CC2)CCn2ccnc2C1 N1(C(Cn2ccc(C)c2)=O)CCCC2(C)CCCCC12 C1(C(=O)NC2(CO)CN(C(=O)Cc3ccccc3Cl)C2)(COC)CCC(=O)N1 C1(NC(C2(COC)CCC2)=O)CC2CC(NC(=O)CN(S(C)(=O)=O)C)C1C2 C(=O)(C#CC1CCOCC1)N1CC(NC(COc2cccc(C)c2C)=O)C(C)C1 c1(NC(c2c(C)cccc2)C)ncccc1S(=O)(=O)NCCCn1cnnn1 N1(C(C(CC)CC)=O)CC2CCC(N=c3cc(Cl)nc(C4CC4)[nH]3)CC2C1 C1(CCN(C(C)(C)C(=O)NC2CC2)C)CSCCN1C(C1CCOC1C1CC1)=O C(C(C)C)(C(O)C(=O)NCc1ccc(C(=O)NOCC(N)=O)nc1)OC N#Cc1cn(OC2CN(C(=O)C(F)(F)F)C2)c(=O)n(C(=O)c2ccccc2Cl)c1=O CCC(CNC(=O)Cc1c[nH]nc1C)(CC)C(=O)N(CCS(N)(=O)=O)C Cc1nn(C)c(C)c1NC(C1CCC(CNC(C2(CC(C)C)CC2)=O)C1)=O c1(OCC(=C)Cl)ccc(N(C)Cc2snnc2CC)cc1 CC1CN(C(=O)CC2CC2)CC1CNC(c1c[nH]nc1C1CCOCC1)=O C1(NC(CC#C)=O)CCN(Cc2nccc(OC)n2)CC1O N1(C(=O)Nc2ccc(SC)cc2)CC(NC(C2(C)CCCNC2=O)=O)C(C#N)C1 C=CCC(C)(C)CC(=O)N1CC2CC(NC(=O)CC3CCCNC(=O)C3)C2C1 C1(NC(CCCc2onc(C(C)C)n2)=O)CC2C1CCN2C(=O)CC(C)C(C)C c1(C(=O)NCC2N(C(C=COCC)=O)CCC2)c(C)cc(O)cc1C N1(C(C2(NC(C)=O)CCC2)=O)CCC2CC2(C(=O)NC2CN(C)CC2(C)C)CC1 C1(C(=O)NC2CC(CNC(c3csc(COC)n3)=O)C2)CC2CCCCCCC12 N1(C(C)=O)CC2CC(C)N(C(C3CCNC4(CCC4)C3)=O)C2C1 C1(CC)CCN(C(=O)C(COC(C)(C)C)N(C)C)C1C(=O)N(C1CCOCC1)CC c1(CC(N2CCC(C#N)(c3cc(F)cc(F)c3)CC2)=O)csc2ccc(Cl)cc12 CC1C(NC(=O)CCC[N+](=O)[O-])CC2CCC1N2C(c1cnoc1C1CC1)=O C(=O)(C1=CCC(F)(F)CC1)NC12CC(CNC(C3(OC)CCSC3)=O)(OC1)C2 c1(CC(=O)NCC2C3CN(C(=O)C=CCO)CC23)c(F)cc(Br)cc1F C1(NC(c2cc(Br)cnc2S)=O)CN(C(c2ccsn2)=O)CC12CC2 C(CC1CCC1)(C(=O)N=c1cc(C)n(CCO)[nH]1)NC(c1ccc(OC)s1)=O C1(OC)(CNCC(=O)Nc2ccc(=O)n(CC(F)(F)F)c2)CC(C)CC(C)C1 c1(C(=O)NCC(CC)(CC)NC(C(CCC)OC)=O)nc(N)cc2ccccc12 C1(C(=O)NCC(CNC(c2ccc(C)n2C)=O)O)CC=C(C(C)C)CC1 c1(CNC(c2ccc(C(C)=O)[nH]2)=O)ncc(C(=O)N(C2CC2(C)C)C)cn1 C1(NC(CCCCC)c2nnnn2C2CCOCC2)CCc2nncn2C1 C1(N(CCCNC(=O)Cn2cc(-c3cncs3)nn2)C)CCC(F)(F)CC1 N1(C(C(CC)(C)O)=O)CCN(C(=O)Cc2nc(-c3ccsc3)no2)C(C(C)C)C1 Cc1cc(C(=O)NC2CCCC(CNC(c3ocnc3C(C)C)=O)C2)nn1C C1(C(=O)NCC=CCCC)COCCC1NC(=O)CC1C=NN(C)C1=O c1(CC(=O)N(CC(C)O)CCNC(C2(F)CC2C)=O)nccn1C C1(CC(=O)N(CC#C)CC)CN(C(=O)C(C)N(C)C(C)=O)CCC1C Cc1cc(N2CCC(C3(NC(c4cnc(O)nc4O)=O)CC3)C2)nc(C)c1C#N C#Cc1cn(C)nc1C(N1C2CCC1C(NC(=O)CCn1cc(C)cn1)C2)=O c1(C(N(CCN(C(CC(C(C)C)OCC)=O)C)C)=O)cc(Cl)c(F)cc1O CCCCC(C(=O)N1CC(NC(=O)C(F)(F)F)C(c2ccccc2)C1)OC N1(C(C(CC)OC2CCCC2)=O)CC2CC2(CNC(c2cccnc2S)=O)C1 C1(COC)(CNC(C2CCCC2O)=O)CCCN1C(=O)COCC1CC1 C(=O)(C(C)CC(F)(F)F)NC1(O)CC(C(N(C2(C(=O)OC)CC2)C)=O)C1 c1(C(=O)NCCN(C(=O)C(O)Cc2cc(Cl)cc(Cl)c2)C)coc(S(C)(=O)=O)c1 C(=O)(CCCCC(F)(F)F)N1CC(C2CN(C(C3(OC)CCCC(C)C3)=O)C2)C1 Cc1cnn(C)c1CC(=O)NC1CCCC1NC(=O)CCOCc1ccccc1 c1(C(N2CCC(C)(CC(=O)NCCN3CCC3)C2)=O)ccc([N+](=O)[O-])o1 c1(C(N(C2CCN(C(c3csc(C)c3)=O)C2)CCC)=O)cncc(F)c1 Cc1cc(C(=O)NCCC2(CNC(=O)CC3COC(=O)N3)CC2)c(C)nc1C N1(C(c2nc(C)n(C)c2C)=O)CCC2(CC(NC(=O)COCC(C)(C)C)CO2)C1 CCCC(C(F)(F)F)NC(C1(CC)CCN(C(C23COCC2C3)=O)C1)=O C1(CNC(C(C)Cn2cccn2)=O)CCC(C(=O)NCCC(O)CO)CC1 c1(C(=O)NC2C(C(NOCCOC)=O)COCC2)ccnc2cc[nH]c12 C1(C(N(C(c2ccc(OC)cc2)C(=O)O)C)=O)Cc2cc(C)ccc2S1 c1(C(N2CCC(NC(C3CCCCC3O)=O)(CO)CC2)=O)cncc2nc[nH]c12 c1(C(=O)NCC2(O)CN(C(C(C)NC(COC)=O)=O)C2)csc2c1CCC(C)C2 c1(NC(c2csc(C(N3CCCC3c3nn[nH]n3)=O)n2)=O)ccn2ncnc2c1 CCC(CC)C(CNC(N1CCC(CCO)(CO)CC1)=O)OC O=C(CCC(F)(F)F)NCC=CCNC(C1CCCS1(=O)=O)=O C1(CNC(CCC(C)(C)OC)=O)CCN(C(=O)CCC(C)(C)C#N)CCC1(F)F C(C1=NOC2CCCC12)NC(C1N(C(c2c(C)c[nH]c2)=O)CCC1)=O CC(C1CCCCC1)=CC(=O)NCC(C1CC1)NC(=O)C1=CCCCO1 Cc1cc(=O)c(C(=O)NCCCCN(C)C(c2cn3cccnc3n2)=O)cn1C N1(C(c2ccc(NC(C)(C)C)cc2)=O)CCC2(NC(C3CC3F)=O)CCCC12 C1(C)(CNC(C=C(COC)C)=O)COCCN(C(=O)CC(=O)NC2CC2)C1 CN1Cc2cc(-c3ccc(CNS(=O)(=O)c4ccccc4)cn3)ccc2C1=O C1(NC(CCCC=C)=O)CCN(C(C2(CCN(C)C)CC2)=O)CC(C)(C)C1 N1(C(Cc2c(C)nsc2)=O)CC2CN(C(=O)CNC(=O)Cn3cncn3)CCC12 N1(C(C(C=C)O)=O)CCC(NC(=O)CCCN(C)C(C)C)C(CO)C1 CCC(C)CC(C)N.c1(CS)cncc(-n2nc(C)cc2CO)n1 C1(NC(CSC(C)C)=O)CCCC(NC(C2COCCOC2)=O)C1 C1(=CC(=O)NC2CC(NC(C3C(C)(C)C3)=O)C2)CN2CCC1CC2 CC1(C)CC(NC(=O)CCc2ncc[nH]2)CCN(C(C2(C#N)CCOC2)=O)C1 c1(OC)ccnc(CCNC(C2CC3CCCC23)=O)c1OC CCC(CC(=O)NC1(CCOC)CCN(C(c2snc(O)c2Cl)=O)C1)C(F)F C(=O)(C(C(C)C)n1ccc(C)c1)NC(C1(OCC)CCC1)c1nn[nH]n1 c1(CN(C2CCCN(C(=O)CC(O)c3ccccc3)C2)C)ccc(F)c(I)c1 C(=O)(C(C)(C(=O)NC(=O)OC(C)(C)C)N)NCC(CO)NC(CC)=O.OC CC(C)(C)C(C#N)C(=O)NC1CCCC1C(=O)NC(c1ccco1)CO C1(NC(=O)CCOCC(F)F)COC2(CCN(C(=O)CSC(F)F)CC2)C1 c1(C(=O)NC2CC(C)N(C(c3c[nH]c(=O)cn3)=O)CC2)ccc(F)c(F)c1F C(=O)(C1=Cc2ccccc2C1)NC(C(N1C(C)CCSCC1)=O)CCF N1(C(c2ccc3ncn(C)c3c2)=O)CCCC2C(CCCN2C(=O)C2CC2)C1 CC1=C(C(=O)N2CC(O)CC2C(=O)NCC=C2CCSCC2)CCCO1 c1(OC)cc(C(N2CC(F)(F)C2c2ccccc2)=O)ncc1-c1cnoc1 CC(C)(O)CCCC(=O)N1CC(CNC(c2cncc(O)c2)=O)C1 c1(CSC)cccc(C(=O)NCC(C)N(C)C(c2cc(C(C)(F)F)n[nH]2)=O)c1 N1(C(C(Cn2ccc(C)n2)C)=O)CCN(CCNC(=O)C(C)(C)CC2CC2)CC1 N1(C(C2C(C(=O)OC)C2)=O)CCCCC1CN(C(=O)CC1CC2(CCC2)C1)C N1(c2snc(C(=O)OCC)n2)CCCC(OCCOC(C)C)C1 C12(C(N3CC(CN(C(c4c(C)scn4)=O)C)OCC3)=O)CCCC1CC(=O)CC2 c1(CSC)ccc(C=CC(=O)NC2(CO)CN(C(C3CC3C)=O)C2)cc1 C(C)(CC(C)NC(=O)CC(C)O)NC1CN(C(C)=O)C1 N(C1CCc2cc(CNC(=O)C(=O)Nc3ncc[nH]3)ccc21)C(CCC(C)C)=O c1(OC(c2cn(C3COCC3=O)nn2)CCC)coc(S(C)(=O)=O)c1 c1(OCCC(=O)NCC2(CC)N(C(C(CC)OC)=O)CCC2)cccc(F)c1 N1(C(CC2C=NN(C)C2=O)=O)CCCC2(CCN(C(=O)CC(C)(F)F)CC2)C1 Cc1cc(O)cc(=O)n1CC(N1CCC(C)C(NC(C2CC3(CSC3)C2)=O)C1)=O C1(NC(c2c(CC(C)C)noc2)=O)CN(C(=O)CNC(C2CCC2)=O)CC1C c1(CNC(CN(C(=O)CCC=CC(C)C)CCOC)=O)ccc(OC)nc1 CCCC(C(O)C(=O)NC1CCOCC1O)NC(=O)CCOC c1(CNC(CC2(N(C(c3cnc(C(C)C)o3)=O)C)CC2)=O)cccc(F)c1O c1(C(=O)NCCC2C=CCC2)ccoc1CNC(C1CC1(F)F)=O C1(CN(C)C(C2CCC(C(C)(C)C)CC2)=O)CN(C(=O)C(C)(Cl)Cl)CCO1 C(C(O)CC(F)(F)F)NC(CC1CCC(NC(C2(C)CC2(F)F)=O)CC1)=O C=CCCCCC(=O)NCC(N1CCN(C(C2CC2C2CC2)=O)CC1)=O C#CC1(C(=O)NC(c2ccco2)C2CC2)CN(C(=O)C(C2(O)CCCC2)F)C1 c1(C(=O)NC(C2(O)CCN(C(=O)CCc3ccn(C)c3)C2)C)cccc(CO)c1 c1(CNCc2ccc(C)nc2)cc2cccc(Cl)c2s1 N1(C(C(C2CCOCC2)OC)=O)CCC(N(CCO)C(C2CC(F)(F)C2)=O)CC1 C12(C(N3CC(CN(C)C(C4CCCC(=O)O4)=O)OCC3)=O)CCC(CO)(CC1)C2 C(N=c1[nH]c2ccc(Br)cc2s1)C1CC(C)N(C(=O)Cc2ccccn2)C1 CC1CCCCC1(CO)NC(=O)Cn1cc(CC2CCNC2=O)nn1 c1(C(=O)NC(C2(O)CCN(C(COC(CC)(C)C)=O)C2)C)cc(OC)ccc1F FC1(F)CCCCC1NC(=NCC1CCC1)NCC(F)C(F)(F)F c1(COC(C(=O)NCC(CNC(c2cc(CCC)[nH]n2)=O)C)C)ccccc1C C1(CCNC(c2c(CC)cco2)=O)CCN(C(C2CC(N(C)C)C2)=O)C(C)C1 C12(CNC(c3c(CC(C)C)nc(C)s3)=O)CCC1CN(C(C1CCSC1)=O)C2 N1(Cc2c(Br)cn(C)n2)CC=C(CNC(c2cc(C(C)(C)C)no2)=O)CC1 Cc1c(C(N2CCC3CCC23c2cnn(C)c2)=O)c2ccccc2n(C)c1=O c1(SC(C)C(=O)NC2(CCNC(C3CC4CC4C3)=O)CCCC2)ccc(Cl)cc1 C1(NC(C(CC)C(C)C)=O)CC2CCCC(C1)N2C(c1nnsc1C)=O N1(C(C2C=C(C)CS2)=O)CCCC(C)(C)C1C(=O)NCC(O)C(F)F C1(CO)CC2CCC1N(c1cc(NCC3CCC4CCCC4O3)ncn1)C2 C(CCCCC(=O)NCC1(C)CCC(NC(=O)COC2CC=CC2)CC1)N(C)C c1(C(N2C(CNC(c3csc(C)c3C)=O)C=CC2)=O)nc2c(s1)CN(C)CC2 Cc1nn(C)c(C(N2CCCC(CCNC(=O)CC3COCCO3)C2)=O)c1Cl c1(C(=O)NC2CN(c3ccc(OC)cc3)C(=O)C2)ccc(F)c(Cl)c1 C(=O)(C(C(C)NC(=O)COCCN(C)C)C(C)C)NCCCNC(C(C)C)=O Cc1nn(C(C)C)cc1C(=O)NC1CCCC(NC(=O)Cc2ncn(C)c2C)C1 C#CC1(C(=O)NC(CCCCC)C2CC2)CCN(C(=O)CC(CC)SC)C1 N1(C(C(C=CCCC)O)=O)CC2(C1)CN(C(=O)Cn1cc(CC)cn1)CCO2 C1(CC(=O)NC(CC)C(N)=O)CN(C(C2CC(=O)CC(=O)N2)=O)CC12CC2 c1(NC2C3(C(=O)OC)CC3CC2)cc(C)ccc1[N+](=O)[O-] C(=O)(C(C(C)C)N1CCC(C)CC1)NCC1(F)CN(C(Cc2nnc(C)o2)=O)C1 c1(N2CC(C)(CCO)OCC2)nc(N2CCOC3(CCCC3)C2)nc2sccc12 c1(C(=O)NC2CC(NC(=O)CC(O)CC3CC3)C2)cnc(O)c2c1NCCC2 N1(C(C(CC(C)C)ONC(CN(C(C)=O)C)=O)=O)CC2C3C=CC(C3)C2C1 C1(C(=O)NC2C(NC(CC3CCN(C(C)=O)CC3)=O)CC2)CN2CCC1(C)CC2 CC(C)(CC(F)F)C(=O)N1CCC(O)C(NC(C2CCC=CCCC2)=O)C1 C1(NC(COC)=O)CCC(CNC(c2conc2-c2ccccc2)=O)CC1 c1(C(=O)NCCCCCC=C)ccc2cc(C)oc2c1 C1(NC(C2CC3C=CC2C3)=O)CN(C(=O)C2=CCCCO2)CC12CCOCC2 Cn1cc(C=CC(=O)NCc2cc[nH]c2C(=O)NCC(C)(C)CO)cn1 Cc1nc(S(C)(=O)=O)ccc1N(C1CCNCC12CC2)C(=O)C(C)CN c1(C(N2CCC(c3c(-c4cc(C)sc4)cccc3)CC2)=O)c(F)cc(F)cc1F c1(C(N(CCNC(=O)CCCc2cc(C)no2)CC)=O)n[nH]c2c1CCC2 N1(C(COC(CC)C)=O)CC2(C1)CN(C(=O)CC1CC(COC)C1)CCO2 C12CCCN(CC1)C(=O)N(C)C2.c1(O)ccc(OC)cc1.CCCOC CN1CC=C(C(=O)NCCC2CCC(NC(=O)Cc3ccc(Cl)cn3)C2)C1 C(=O)(C(C(CC)CC)OC)N1CC(C=C)(C(N2CCCC(C)C2CO)=O)C1 C(=O)(C1=CC2CCCC12)N1CCC(O)(C(C)NC(c2cncc(C)n2)=O)CC1 CS(=O)(=O)c1cc([N+](=O)[O-])ccc1NC1CCCOC1 C12(O)CCCN(C1)C(=O)NC2.C1(NC(=O)C=CCN2CCCC2)(CO)CCOC1 N1(C(=O)CCC2CCC2)CCCC12CCCN(C(=O)Cn1ccc(C3CC3)n1)C2 C(=O)(C1CCCc2sccc21)N1CC2CCC(NC(C=C(CC)C)=O)(C1)C2 c1(CNC(CC)CNS(C)(=O)=O)csc2ccc(Nc3ccccc3)cc12 CCCCC(CNC(C1COC(C)(C)C1)=O)NC(=O)C(C)CN1CCOCC1 N1(C(c2n(C)nnc2)=O)CC(C)(C)C1Cn1cc(CS(C)(=O)=O)nn1 N1(C(C(C2(O)CCCCC2)CC)=O)CCN(C(=O)C(C)CF)C2(CCC2)C1 c1(SCC)ccc(C(=O)NC2CCCC2NC(C2CCOC2C2CC2)=O)cn1 c1(C(N2CCC(CC=C)(C(=O)NC(CO)C3CC3)C2)=O)ccc(=O)n(C)n1 c1(C(=O)NCC2C(C)CCN(C(=O)CCC(N)=O)C2)cc(S(N)(=O)=O)co1 C(=O)(CC1CCCc2ccccc21)NCCOCCOCCNC(C(C)CF)=O N1(C(CCN(C(=O)CCC2CCCOC2)CCCO)=O)CCOCC2(CC2)C1 C1(C(N2CCC(NC(C(CC)(F)C(=O)OC)=O)CC2)=O)Cc2ccc(F)cc2C1 C(=O)(CCCCCCCCC1CC1)N1CCN(C(c2c(C)cncc2C)=O)CC1 c1(C(=O)NCC(C)(C)CNC(c2occc2C2CC2)=O)c[nH]c2nc(Cl)ccc12 c1(CC(=O)NC(CNC(C2C(C=C)C2)=O)(C)C2CC2)cc(Cl)c2c(c1)OCCO2 C1(C(=O)NC(c2cccnc2)c2nn[nH]n2)CCc2ccccc2C1 C#CCC(C(=O)N(C)Cc1cc(C)ccn1)NC(c1cc(CC)on1)=O C1(OC)CC(NC(C23CC(F)C2C3)=O)CN(C(=O)Cc2ccc(Br)nc2)C1 Cc1cc(Cl)c(C(=O)NC(C)CCCNC(c2cc(C(N)=O)[nH]n2)=O)cc1C C=C(C)C(CC(=O)NC1CC1NC(=O)CNS(C)(=O)=O)OCC C1(NC(c2cnc(C(C)C)s2)=O)CC2CCC(C1C)N2c1cnc(F)cn1 c1(C(=O)NCC2(O)CCN(C(C3C(CC)C3)=O)CC2)ccnc2c1CCO2 CCCC(C(O)C(=O)N1CC(CO)C(C)C1)NC(=O)C(F)=C(C)C N1(C(=O)NC(c2ncc(C)s2)CC)CCCC2(CNC(=O)O2)C1 CC(C)CC(O)CC(=O)N(C1CCN(C(=O)CC(F)(F)Cl)CC1C)C Cc1cccc2cc(C(=O)OCC(c3cccc(C(F)(F)F)n3)=O)sc12 N1(C(C(C)CF)=O)CCCC(CCn2cc(CN3CCCC3CO)nn2)C1 C(CCC)(C(=O)N1CC=CC1CNC(C1CC(C(=O)N(C)C)C1)=O)=CCC N1(C(C2C(NC(C(C)CC3CC3)=O)C=CCC2)=O)CCC(N=[N+]=[N-])C1 CC(CC(C)NC(C1(CO)COC1)=O)NC(=O)C=CCN1CCCC1 C1(N2CCC(c3n(C)c(O)nn3)CC2)CCN2CCCC2C1 NS(=O)(=O)c1csc(C(N2CC(CNC(=O)Cc3cncnc3)C3CC23)=O)c1 C1(NC(c2ccc(CCC)[nH]2)=O)CCCCC1NC(C1(F)CCOC1)=O C1(NC(C2C(=C)CC2)=O)CN(C(c2nnn(C(C)(C)C)n2)=O)CC12CCC2 c1(C(N2CCN(C(=O)CSC3CC3)C3(CC3)C2)=O)ccc2nc(S)oc2c1 Cc1ccc(CCNC(C2(CF)CCN(C(=O)CCc3ccoc3)C2)=O)cn1 CC(CN=c1[nH]c(=NCC2CC3(CC3)C2)[nH]c2c(F)cccc12)n1cccn1 c1(NC(C)=O)cnc(C)c(C(N2CC=CC2CNC(c2ccc(Cl)cc2C)=O)=O)c1 c1(C(N2C(CNC(C3(C(N(C)C)=O)CC3)=O)CCC2)=O)cc(CC2CC2)ccn1 CCCCC(O)CC(=O)NC(CCOCC)C(N1CCC12CCCCC2)=O n1(CC)nc(C2CC2)cc1C(N1CCC(C)C1CNC(c1nc(C)c(C)[nH]1)=O)=O C1(C(=O)NCCN(C(c2cccc3c2CCO3)=O)CC)(OC)CC(C)CC(C)C1 C1(C(=O)NCC2C=CC(NC(C3ON=C(C)C3)=O)C2)CC2CCC1CC2 c1(C(CC)=O)cc(C(N2CCOCC2CCNC(=O)C=CCOC)=O)ccc1F c1(NC(c2c(CNC(c3cccc(NC)c3)=O)c[nH]n2)=O)cc(F)ccc1O c1(OC)ccc2[nH]c(C(=O)NC(CNC(=O)CC3CC3)C3CCC3)cc2c1Cl CCC1=C(C(=O)NCC2CC(CNC(c3oc(CO)nc3C)=O)CO2)CCCO1 C1(NC(c2cc(C)sc2)=O)CN(C(C2CCCN2C(C)C)=O)CC1(C)C N1(C(C2N(C(c3c(C)cco3)=O)CC(F)C2)=O)CCn2ncc(C)c2C1 C1(NC(C(C)OCC)=O)CC2CCC1N2C(=O)CCNC(c1cccc(C)c1)=O Cc1cc(C(N2CCC(N(C)C(c3nn(C)cc3N)=O)C2)=O)cnc1C C(=O)(C1=CC2(CCN(C(C3(C)CC(C)(C)C3)=O)C2)C1)NCCCCCC(C)C c1(C(=O)NCCC(CNC(c2n[nH]c(C)c2F)=O)O)cc(Cl)cc(Cl)c1 C1(C)(C(=O)NCC(CC)NC(c2cc(C3CC3)n(C)n2)=O)CCC12CCC2 CCCCCC(O)C(C)C(=O)NCCN(C)C(c1ccc(C(N)=O)o1)=O c1(C(=O)NCC2N(C(C(CC)(F)F)=O)CCC2)cnc(C)nc1OC C(=O)(CCCCN(C)C(C1CN(C)CCO1)=O)NCC(C(=O)OC)OC C1(CNC(C2N(C)C(=O)CC2)=O)CC2(CCN(C(=O)CC3CCC(O)C3)CC2)C1 N1(C(C2(NC(CSCCC(C)C)=O)CCSC2)=O)CCC2C(O)CC12 Cc1cc(-c2nc(-c3oc(Br)cc3C)n(CCC(C)C)n2)c(C)o1 C1(CNC(c2c(CC)cc(F)cc2)=O)CC2(CCC2)CN1C(=O)CCCC#N C1(C(=O)NC2(C)CC(NC(=O)CCCNC(=O)C3CC3)C2)CC1C1CC(F)(F)C1 C(=O)(CCOCCOCCN(C(=O)CCc1ccc[nH]1)CC)NCCCO O=C(NNC(=O)CCSC(F)(F)F)C(C(F)F)c1ccon1 c1(C(=O)NC2C(C=C)CN(C(=O)C(C)S(C)(=O)=O)C2)nc2cnccc2s1 N1(C(=O)Nc2cccc(CCNC(=O)OC(C)(C)C)n2)CCC2CCCCC2C1 c1(C(c2n(CC)nnn2)NCCC(C)SC)ccc(-c2cnccn2)cc1 C(=O)(CCC(C)(C)C(=O)N(CC(C)(C)CNC(=O)C(=O)N=S(C)(C)=O)C)OC C1(C(=O)NCCCn2cc(-c3cc(Cl)ccc3Cl)nn2)CC2C(C1)C2(F)F N1(CC)C(=O)CCC1C(N1CC(O)(CCNC(C2CC23CCC3)=O)C1)=O CCC(CN(C(C(C)S(C)(=O)=O)c1cccs1)C(=O)C(O)CC(C)C)(CC)C(=O)O c1(C(=O)NCC2(CNC(C3CC(C)(C)C3)=O)CCCCC2)ccc(Cl)cc1F C1(C(N(C(C)CNC(c2cc[nH]c(=N)c2)=O)C)=O)CCCCS1(=O)=O N1(C(CCC2CCN(C(c3cnc(=N)[nH]c3)=O)CC2)=O)CCCC2CCCC12 N1(C(c2c(C)c[nH]c2)=O)CC(C(=O)N(C2CC(F)(F)C2)C)CC(C)(C)C1 N1(C(C(CSC)OC)=O)CCC2CCCC(C1)N2C(c1cc(N)cc(O)c1)=O C1(O)(CNC(C2C(OC)CCCC2)=O)CCN(C(=O)C2=CCCS2)CC1 C(=O)(C1CCc2c[nH]nc21)NCCCN(C(C12CCC(OC)C1C2)=O)CC CC1CCN(CCN(c2cc(-c3cccs3)on2)C(=O)C(C)OC(F)F)CC1 CN=c1ccc(C(N2CC=CC2(C)C(=O)NCC(O)COC)=O)c[nH]1 N1(C(=O)NCCN(CCCOC)C)CC2(CCC2O)C1 CC(CC(=O)NN(c1cnn(C)c1)C(N1CCC(Cc2ccco2)C1)=O)C1CC1 Cc1nn(C(F)F)c(C)c1CC(=O)NCC(C1CC1)NC(c1nn(C)cc1Cl)=O C1(CC(=O)N(C2CCCN(C(C3CCN(C)C3)=O)C2)C)COc2ccccc2O1 N1(CCCCC=C)C(=O)CN(CCN2CCCOC(C)C2)C1=O C1(CNC(CC2CCCC(C)O2)=O)CCCCCN1C(=O)CCN1CCCC1 CS(=O)(=O)c1cccc(-n2cc(CONC(c3ccc(Br)cn3)=O)nn2)c1 n1(CC)ncc(C(=O)NC2CCCC2NC(=O)COCP(C)(C)=O)c1C(F)(F)F C(=O)(C(C(C)C)OCC(C)C)NC(CC)CNC(c1csc(C)n1)=O c1(OC)ccc(NC(=O)C(c2ccnn2C)N(C)Cc2ccsc2)cc1 N1(C(CC(C)N2CCCC2=O)=O)CC(CNC(c2ccc(Cl)[nH]2)=O)CC1(C)C C1(C(=O)Nc2ccc(CC)nc2)CCN(C(C2CCC(=O)N2)=O)CC1O C(C)(C)(C#CCCCC)NC(C1C(C=CC)CN(C(=O)CC(O)CC)C1)=O C1(CNC(CCCN(C)C)=O)CN(C(c2cc(C3CCC3)no2)=O)CCC1(F)F CC1CC(NC23CCC(C(=O)N(C)C)(CC2)C3)CC(C)S1(=O)=O C(CC(C(C)C)NC(c1ccc(OCOC)cc1)=O)N(C(C1C(=C)CC1)=O)C C=C(Cl)CC(C(=O)N1CCC1C(N)=O)NC(=O)C(n1nccc1C)C c1(C(=O)NCCC2(CNC(=O)C=C(Cl)Cl)CC2)ccnc2[nH]ncc12 N1(C(c2c(CC)n[nH]c2)=O)CCC(C(=O)NC(C)C(F)(F)F)(OC)C1 c1(C(N(CCO)CC)=O)cn2c(n1)CN(C(c1ccc(Br)c(C)n1)=O)CC2 N1(C(=O)C=C2CCCC2)CCN(C(=O)CCc2ccc(O)nc2)C(CCO)C1 Cc1ccc2c(c1)CCC2NC(=O)CCn1cc(C(c2ccccc2)(C)O)nn1 N1(c2ccnc(N(C)CCNc3ccccn3)n2)CCC2(CCSC2)C1 C12(C(N(C(C)CCNC(C3(C(F)(F)F)CC3)=O)C)=O)CCC(CC1)C2(C)C CCC(CCOC)C(=O)NCC1CCN(c2ncc(I)cn2)C12CC2 C1(NC(C=CC=CC)=O)C2CC(O)C1N(C(=O)CC1CCC3(CCC3)O1)C2 Cc1ccc2c(c1C(=O)Nc1ccccc1CN)CCCN2 C1(N)CCC(=O)NC1.C(C(C)(C)C)N(C(=O)CN(C(=O)NOCCC1CC1)CCO)C N1(C(CC(C)C(F)(F)F)=O)CCC2CCN(C(=O)CCCC3CCOCC3)C2C1 C(C(CC(F)(F)F)NC(=O)CCF)NC(C(C1N(C(C(C)C)=O)CCC1)(C)C)=O CN1CC=C(CC(=O)NCCCCC2CCCN(C(=O)CN(C)C)C2)CC1 c1(C(N2CCC(C(N(CCCN3CCCC3)C)=O)C2)=O)cnn(C)c1Cl CN1CCN(C(C2CCC(CNC(=O)Cn3ccnc3)O2)=O)C(CO)C1 C1(CC(=O)NCC(C2CC2)N(C)C(C2CC2[N+](=O)[O-])=O)(OC)CCCC1 OC1CN(Cc2ccc(C3OCCO3)cc2)CCC12CCCNC2 N1(C(c2cc(CNC(C3CCCSC3)=O)ncc2)=O)CC(F)(F)C(F)(F)C1 C1(CNC(=O)NCc2cc(C(F)F)n[nH]2)CCC2CC12 C(CC1=CCN(C(=O)CCc2ccsc2)CC1)NC(C12CCC(C)(C1)CO2)=O CC(C(C(=O)NCc1ccccc1)N(C)CCN1CCCC1=O)C1CCOCC1 C1(C(NOCC(CC)C)=O)CCN(C(=O)Cc2ccc(C)nc2)O1 N1(C(C2C(C)(C)C2)=O)CCCC2CN(C(c3cnnn3C3CC3)=O)CCC12 CCC(CC)C(CNC(c1ccc(C(F)F)c(Cl)c1)=O)OC CC1(C)CC(NC23CC(C(F)(F)F)(CO2)C3)CCN(C(=O)OC(C)(C)C)C1 c1(C(=O)NCC(C)(C)NC(C(CC=CC)C)=O)ccn2cnc(C)c2c1 C1(C)(C(N2CC(COC)(NC(=O)C(C)N(C)C(C)=O)C2)=O)CC(C)=NO1 N1(C(C(CC#C)NC(=O)C=C(C)C(C)(C)C)=O)CC(C2CC2)(CO)C1 N1(C(C2N(CCC)C(=O)CC2)=O)CCC(N=c2cc(C)nc(CSC3CC3)[nH]2)C1 c1(C(=O)OCC(CC(C)C)C)ncc(C(F)F)cc1F CCC(CCOC)C(=O)Nn1cc(-c2ccc(SC)cc2)nn1.C12CC(C1)C2 C(=O)(CC(C)(C)CC(F)(F)F)N1CC2(OCC(NC(C3CC(OCC)C3)=O)C2)C1 c1(-c2nn(CCCS(C)(=O)=O)c(C3CCCCN3C3CC3)n2)cc(F)cc(F)c1 N1(C(C2CC23CC3)=O)CCC2CN(C(c3cc(O)nc(O)n3)=O)C2C1 c1(CC(=O)NCCCNC(=O)C(C2CCCO2)C2CC2)ccnnc1O Nc1cc(C(N2CCC(NC(C3C4COCC34)=O)C(CO)CC2)=O)cc(O)c1Cl N1(C(Cn2ccc(C)c2)=O)CCCCC(N(C)C(c2cc(CCO)on2)=O)C1 C12(C(=O)NC3(C)CC(NC(C4(SCC)CC4)=O)C3)C(=O)C3CCC1C2C3 n1(CC)nnc2c(NCC(C(C)(C)C)NC(c3ccc(=O)n(C)c3)=O)ncnc12 N1(C(c2cn(C(c3n(C)ncc3)C(=O)Nc3ccc4cnnn4c3)nn2)(C)C)CCC2(CC1)CC2CO C(=O)(C#CC1CCOC1)N1CC(C(C(=O)NCC2CN(C3CC3)C2)OC)C1 c1(C(=O)NCC(CO)NC(c2cnc(SC)s2)=O)ccc(C2CC2)nc1 Cc1cc(Cl)ccc1OC(C)C(=O)NC1CCCN(C(=O)CNC(=N)N)C1 c1(C(N(C2CCN(C(=O)C3=CCC3)CC2)CC#C)=O)cc2ccc(C)n2cn1 c1(C(N(C(CCNC(c2cc(C)c(C)o2)=O)C)C)=O)csc2c1CCCC2 c1(C(N(CC(C)NC(C2(COC)CC=CC2)=O)C)=O)cn2ccnc2cn1 c1(CSCC(=O)CNCc2nc(C)sc2)cccc(NC(=O)CC2CC(F)C2)c1 c1(C(C(=O)NC(C)CNC(C2CC2Cc2ccccc2)=O)O)ccc(F)c(F)c1 C1(OC)CC(NC(c2cccnn2)=O)C12CCN(C(C1(C)CC(F)(F)C1)=O)CC2 C(=O)(C1=NOC(C(C)(C)C)C1)NCCCNC(=O)OC(C)(C)C.c1(C)ccccc1 C1(CC)CN(C(c2cnn(CCO)c2)=O)CCC1CNC(C1CCCOC1)=O CC1CN(C(=O)Cc2sc(=N)[nH]c2-c2cccs2)CCN1C(C1CCC2CC2C1)=O c1(SCC)cccc(N(C(=O)C(C)(c2ccccc2)N(C)CCNC)C)c1 C1(c2nnnn2C2CCCC2)(NCCCc2cc[nH]n2)CCN2CCC1C2 c1(C(C)C)ccc(C(CC(=O)O)NC(CCCS(C)=O)=O)cc1 c1(C(N2CC(CN(C(CN(CCCCCC)C)=O)C)C2)=O)cnc(Cl)c(N)c1 Cn1nc(-c2cn(CCC(=O)NC3CCCN(C(C)(C)C)CC3)nn2)n(C)c1=O N1(C(Cc2c(C)n(C)nc2)=O)CCC2(C1)CN(C(c1cc3ccsc3s1)=O)C2 C(CN=c1cc[nH]cc1C)NC(C(N1CC(OCCCCC)C1)=O)=O c1(C(N(CCC2CCN(C(CC(CC)C)=O)CC2)C)=O)ccc(Cl)c(N)c1 Cc1c(C(=O)NC(C)C(CO)NC(=O)C(c2cccnc2)C)cncc1Br N1(C(C2CC2C(=O)NCCNC(=O)OCC)=O)CCC(CCC)CC1.C(N)=O C1(C)(C(=O)NCCCCN(C(C(CC#C)C)=O)C)CCC12CCC2 c1(C(N2CC(CNC(c3cc(C)c(O)nc3)=O)C2)=O)cc2c(C)c(Cl)ccc2[nH]1 N1(C(C(=O)NC(CC)(C)C)C2CC2)CCN(S(C)(=O)=O)C(C)C1 CC1COCCC1C(=O)NCC1CN(C(c2ccc(SC)o2)=O)C1 C(=O)(CCCCC(C)C)NC(c1cn(C)nn1)C(=O)N(CC)CC1CCOC1 C1(CC)C(NC(=O)Cc2cnccn2)CCCN1C(=O)Cc1cc[nH]n1 C1(NC(c2nnc(O)nc2O)=O)CC2CC1CC2C(=O)NCC1CC(CO)CO1 N1(C(CCc2ccn(C)c2)=O)CCC2CCN(C(=O)CC3CC3C(F)(F)F)CC12 c1(C(N(CC(=O)NCC2CCOCC2)CC)C)ccc(F)cc1 C1(NC(c2[nH]cc(C)c2)=O)COC2(CCCN(C(=O)C=C(Cl)Cl)C2)C1 N1(C(CC(C)(C)C)=O)C2CCC1(c1cn(CC(=O)NCC3CCCO3)nn1)CC2 N(C(=NCC(C)(C)CC)NCC1CCOC1)CC(C1CCOCC1)OC c1(CC)ccc(C(N2CC(N(C)C(c3ccc(OC)cn3)=O)C(F)C2)=O)c(C)n1 Cc1ccnc(O)c1C(=O)NC1CCC(NC(C2(C)CCN(C)C2)=O)C1 CC1CC(CC(=O)NCCc2noc(=O)n2C)CN1C(c1cnc[nH]c1=N)=O C1(C(=O)NCCn2cc(C(N(CC(C)O)CC)=O)nn2)CN2CCN1CC2 C#CC(C)(C)C(=O)NCC(=C1CN(C(=O)CSc2ccccn2)C1)F N1(C(c2c(C)sc(Br)n2)=O)CCCC(NC(=O)C=C2CCC2)C1C C1(C(N(C)CC2(C)CCCC2O)=O)CC(NC(C2C(C)(C)C2(C)C)=O)C(O)C1 C=C=C(C)CC(=O)NCCCN(C(=O)CC1NC(=O)NC1=O)C(C)C CN(C)S(=O)(=O)N1CCC(C(=O)NC2CCCC(c3cccc(Cl)c3)C2)CC1 c1(C(N2CCC(NC(CC(COC)(C)O)=O)C2)=O)cc(Cl)cc(C)c1C CCC(CN(C)C)CC(=O)NCC1(NC(=O)COCC2CCCOC2)CCCC1 Cc1ccc(C=CC(N2CC3CC2(C(=O)NC(C2CCOC2)CO)C3)=O)cc1 C(C(O)C(=O)NCCOCCC(=O)NC(C1CCCO1)CC)=CC O=CN1CCCC1C(=O)NC(c1cccnc1)C(=O)NCCC1CC1 C1(NC(CSCc2nc(C)sc2)=O)CCN(C(C2CCOC2=O)=O)C12CCC2 C1(CNC(C2(CCC)CC2)=O)CN(C(=O)C(C)CN(C)C)CCC12CCC2 Cn1cccc1C(=O)C(=O)NC1CC1NC(=O)CCC1CCOCC1 C1(=CCNC(C=CC=CC)=O)CCN(C(=O)Cc2ccc(CCC)cc2)CC1 c1(C(C)OC)nc(CN(C)CCN(C(=O)CC2C=CCC2)C)cs1 N1(CC)CCOCC1C(=O)NCCCC(C)NC(c1cc(-c2ccoc2)[nH]n1)=O C1(C(N2C(Cc3cn(CC(C)C)nn3)CCCC2)=O)CCc2nnc(O)n2C1 N1(C(c2n(CC)ncc2)=O)CC2(CC(C(=O)NC(CC)(CC)CCO)CO2)C1 C1(C(=O)NCC2(O)CC(CNC(CCC=CC(C)C)=O)C2)CC2CCC1O2 Cn1cc(CCC(=O)NC2CCN(C(=O)C(C)(C)C3CCCCO3)C2)cn1 c1(C(N(CCCCCNC(c2cc3cscc3s2)=O)C)=O)cncc2c[nH]nc12 c1(CNC(C(C)=C(C)C)=O)nc(C)c(C(N2CCC(F)CC2)=O)o1 c1(NC(C2CCCCN2C(=O)OCCC(F)(F)F)=O)ncc(Cl)cc1F N1(C(CN2C(C)CCC2)=O)CCC(NC(C2(C)CCCN(C)C2)=O)CC(C)(C)C1 N1(C(CCOCC)=O)C2CCC1C1CC1(NC(=O)C(CC)OCC)C2 c1(-c2ccc(C(=O)NCC3(NC(C(CC)N(C)C)=O)CCC3)o2)ccccc1Cl C(=O)(C(O)CNC(C1(O)CCCC1)=O)N(CC(C)(C)OC)C N1(C(C2C(C=C)C2)=O)CCCC(O)(CNC(c2ccc3ncsc3c2)=O)CC1 C1(NC(CC2(C(=C)F)CCC2)=O)CN(C(c2ccncc2Cl)=O)CCC1O CC1(C(=O)NC2CCN(C(c3cccc(Cl)c3)=O)CC2C(N)=O)CCCCCC1 C1(C(=O)OC(C)(C)C)CC(S(C)(=O)=NC(=O)C2C3CC(=O)OC23c2ccccc2)C1 C=CCCCC(C)(C)C(=O)NCC1CCN1C(c1cnc(C)[nH]c1=N)=O O=C1CCCC(C(=O)N(C2CCN(C(=O)COCC3CCCO3)CC2)CCO)O1 N1(C(CCCCSC)=O)CC2CCC2(CC(=O)NC2CCCN(CCO)C2)C1 c1(C(=O)NCC23CC2CN(C(=O)Cc2cc[nH]n2)C3)cc2c(Cl)cccc2s1 CC1CC(c2nnnn2C2CCOCC2)(NCCc2nc(=O)o[nH]2)CN1C1CC1 N1(C(c2c(C)noc2C)=O)CC(CNC(c2cnc(C3CCC3)o2)=O)C(C)(C)C1 CCC(C)(CC)C(=O)NC(C1CCCC1)CNC(=O)CCCN(C)C CC(C)(C)C#CC(=O)N1CCC(=CCNC(=O)COCC2CCCCO2)CC1 CC1CC(C(=O)NCCCC2CN(C(C3(C#N)CC3)=O)CCO2)=NO1 C1(NC(C(C)(C)O)=O)CCC(NC(C2CCCCC2CC(F)(F)F)=O)CC1 Cc1nccnc1C(N1CCCC1C1CCN(C(=O)CC2CCC(O)C2)C1)=O C1(C(=O)OC)CN(C(=O)Nc2ccc(C(=O)Nc3csc(C)n3)cc2)CCC1O c1(CC(c2nc(C(=O)O)cs2)NCc2ccn(CC)c2)ccccc1F c1(N2CC(c3c(C)nn[nH]3)C2)cc(Cl)cc2c1OCCC2=O N1(C(C(COCC)C)=O)CCN(C(=O)Cc2c[nH]nc2O)C2CCCC12 N1(C(c2c(NC(C)=O)cccn2)=O)CC(CNC(C2C(C)C2C)=O)CC(C)(C)C1 c1(C(N2CC(CNC(C(C)C(F)F)=O)C(O)C2)=O)ccc2cc[nH]c2c1F C1(C)(C(=O)NCC(C(C)C)NC(C2CC(C3CC3)C2)=O)CCN(C)CC1 c1(C(N(CC(C)NC(C2CCC(=C)CC2)=O)CC)=O)cn(C)ccc1=O N1(C(C2CSCC(=O)N2)=O)CCN(C(c2ncnc(O)c2F)=O)C(CO)C1 C1(CCNC(CCSCC(C)C)=O)COCCN1C(C1(C2CCCCO2)CC1)=O c1(CNc2nccc(N3CC4(CC(C(C)C)OC4)C3)n2)cn(C)c2ncccc12 c1(CC)cccc(C(=O)NC2CN(Cc3cc(C(=O)NC)n[nH]3)CC2C)n1 c1(C(N2CC(CC(C)NC(C(C)OCC#C)=O)C2)=O)sccc1C(C)C C1(NC(C2(OCC)CC2)=O)CS(=O)(=O)CC1NC(c1cccc(CC)c1O)=O c1(CC(=O)NCC2(C)CCN(C(CCC(CC)C)=O)CC2)cn2ccccc2n1 C1(NC(c2cnc3ccoc3c2)=O)CN(C(=O)C=C2CC2)C2(CCOCC2)C1 c1(C(=O)NCC(CNC(C(C)C2CC2)=O)CO)cccc(-c2ccccc2)c1O N(C(=S)NNC(=S)N(C)Cc1cccc(C)c1C)CC=C C(=O)(C1CCCc2c1ncn2C)NCC1CCN(C(C2CC(SC)C2)=O)C1 C1(CC(=O)OCCC)(NCCCN(CCCN)C)CC2(CCOCC2)C1 c1(C(=O)NC(CC)CNC(=O)CC2CCCO2)c(OC)ccc2cccnc12 c1(C2(C(=O)NCC(CN(C(=O)C(C)(C)N(C)C)C)O)CC2)ccc(C(F)(F)F)cc1 C1(C)(C(N2CC(OCCNC(C(C3CCC(=O)N3)C)=O)C2)=O)CCCC1 N1(C(c2cc(C(C)C)n(C)n2)C(=O)NCCC2CC2)CCN2CCC1CC2 Cc1cccc(C(=O)NC(C)C(=O)NC2CC(NC(C3CC(C)(C)CO3)=O)C2)c1 C1(C(=O)NCCC2(O)CN(C(CCc3nnc(C)n3C)=O)C2)COCC(C)(C)O1 N1(C(C)C)CCOC(C(=O)NC2(CNC(=O)C(C)C(C)O)CCCCC2)C1 C(=O)(C(C)(C)C(=O)NCc1c(-c2cn(C3(C(F)F)CC3)nn2)cnn1C)N(C)C CN1CCOCC1CC(N1CC(O)(CNC(c2cc(C(C)(C)O)on2)=O)C1)=O c1(-c2nc(-c3ccc(CCN(C)C)cn3)n(CCCO)n2)c[nH]c2ccccc12 c1(C(N2CC(C)(NC(C3CC(C)OCC3)=O)C2)=O)ccc(C(F)(F)F)cc1C#N C(=O)(C1CCc2c[nH]nc21)NC1CCN(C(Cc2cn(CC)nn2)=O)C1 c1(C(N2C(C)CN(C(=O)CSCC3CCCO3)CC2)=O)coc2ccccc12 C1(CC(=O)NC2C(CCOC)C2)CN(C(=O)C(C)n2cccn2)CCO1 CC(C)C(O)C(C)C(=O)N(CCCCCC(=O)NCC1CCCCN1C)C c1(C(N2CC(N(C(C(N3CCN(C)CC3)C)=O)C)C2)=O)ccnc(Cl)c1 N1(C(CC2C(CC)C2)=O)CCC(CSC)C1.c12cc(cs1)CN(C)C2=O.C C1(NC(c2ccc(O)nn2)=O)CCN(C(c2cnc(Cl)[nH]2)=O)CCC1CO N1(C(C)=O)CC(CNC(c2ccc3nn[nH]c3c2)=O)OC2CCCC12 Cc1sc(C)c(CNC2(C)CCC(NS(=O)(=O)c3cccs3)CC2)c1Br CC1(NC(c2ccc(Cl)nc2N)=O)CCN(C(C2COC(C)(C)CO2)=O)CC1 Cc1c(C(=O)Nc2nc(N3CCCC3)cc(N)n2)ccc(Cl)c1Cl C(=O)(C(CNC(C1CCC(CC)CC1)=O)(CC)CC)N1C(C=C)CCC1 c1(C(N(C2CCCCC2C)CC(=O)OCC)=O)c(Cl)cc(Cl)c2ncccc12 CC1CN(C(c2cncc(N)c2)=O)CCCN1C(=O)CCC(C)(C)F c1(COC)cc(C(c2nnnn2C(C)C(=O)OC)NC2(c3cccnc3)CC2)no1 Cn1nc(I)cc1C(=O)NCCc1csc(C2CCS(=O)(=O)C2)n1 c1(CNC(CS(N)(=O)=O)=O)cc(O)nc(CNC(=O)CN2CCCC2=O)n1 c1(C(N(C(C)C)CCNC(C2CCSC2)=O)=O)ccc(CO)c(F)c1 c1(C(N2CC(C)CC(NC(CS(=O)(=O)NC)=O)C2)=O)cc2c(Cl)nccc2o1 c1(CN(CC)CC2CCOC2)ccc(OC)c(Br)c1 CC1CN(C(=O)C2=CCN(C(=O)CCc3nc(=N)[nH][nH]3)CC2)Cc2nncn21 c1(C(=O)NC2CC(CCNC(CC3OCC(C)(C)C3)=O)C2)cc(N)c(F)cc1F c1(OCC)cc(N(CCCNC(c2cncn2C)=O)Cc2ccccc2)ncn1 N1(C(CC(C)SC)=O)CCCC2(CNC(c3cnc4c(c3)CCC4)=O)CCCC12 C1(C)(C(=O)NCC(C)NC(=O)Cn2nccc2-c2ccccc2)CCNC(=O)C1 c1(C(C2CC2)OC)nc(CCc2ccc(C)cc2)n(-c2nc(Br)nn2C)n1 N1(C(CC(CC)C2CCC2)=O)CCN(C(=O)C(C)OCOC)CC(O)C1 C1(CNC(=O)CCC2CC2)CC2CCC(C1)N2C(C1CCCC(F)(F)C1)=O C(=O)(C(C)C(O)C(C)C)N1CCC(NC(CCC=CCC=C)=O)C1(C)C Cc1cccc(C(N2CCN(CC(=O)Nc3ncc(Cl)cc3F)C(=O)C2)=O)c1I O=C1CCC(C(=O)NC2CN(C(=O)C=CC(=O)NC3CC3)CC2C(F)F)CCO1 C(=O)(C#CC1CCCCO1)NC1C(NC(=O)COc2ccc(Cl)cc2F)CCC1 c1(-c2ccc(N(C)C)cc2)n[nH]c(=Nc2cccc(F)c2CO)o1 C1(C(=O)NCCCNC(Cn2cccc(C)c2=O)=O)CCC2CCC(=O)N12 c1(CC(=O)NCC2CC(NC(c3cnco3)=O)CC2O)cc(F)cc(Cl)c1 c1(C(=O)NC2CCN(C(C(CC#C)O)=O)CC(O)C2)cccc2c1OCC2(C)C c1(OC)cc(C(=O)NC2CC(C)(NC(=O)C(C3CCC(=O)N3)C)C2)cc(Cl)n1 c1(NC(=O)C(N2CCCC(C(=O)Nc3ccccc3)C2)=O)cccc(F)c1 c1(CNC(CC(=O)NCC2(OCC(=O)NCC)CC2)=O)ccc(Br)cc1Cl CCC(C)(C)C(C)CC(=O)NC1(C)CCN(C(=O)CC2CCCC3(CC3)C2)CC1 c1(NC(C2CC(NC(c3ccc(O)c(Cl)c3)=O)C2)=O)ncc(O)cc1Cl n1(CC(=O)N(CC(=O)NCCC)C)cc(-c2cnn(C3CC3(F)F)c2)nn1 c1(C(=O)NCCN(C(C=CCC)=O)CCc2ccccc2)cc(OC)nn1C CC1CC(C(=O)NC(C)(C)CNC(c2ccnc(N(C3CCCC3)C)c2)=O)=NO1 c1(C(=O)NC2CC(C)N(C(=O)C=Cc3ncco3)CC2)ccc2ccccc2c1 Cc1ccc(CC(=O)NC2(CNC(C3CC(C)(F)C3)=O)CCOC2)cc1[N+](=O)[O-] N1(C(CCN(C(C)=O)C)=O)CCCC2CCN(C(=O)Cc3ccc(O)cn3)CC12 C1(NC(C2(OC)CCSC2)=O)CCN(C(=O)C=Cc2ccncc2C)CC(O)C1 c1(OC)ncc(C(N2CCCC2CNC(=O)C(=Cc2cnc[nH]2)C)=O)cc1C C(=O)(CC(C)(C)C(F)(F)F)N(C1CCCN(C(CC(C)SC)=O)CC1)C Cc1ccc(C(=O)NCCCC(C)(C)NC(=O)Cn2cc(Cl)cn2)c([N+](=O)[O-])c1 CC(C)C(CCN(C(=O)C(C1CC1)C1CC1)C)NC(c1csc(Cl)n1)=O c1(OCC(=O)NCC(CC)NC(c2cnc(C(=O)NC)nc2)=O)ccc(F)nc1 c1(OC)cnc(Cl)c(C(N2CC(F)(C(=O)Nc3ccc(C(C)=O)cc3Br)C2)=O)c1 C1(NC(CC(C)c2ccccc2)=O)COCCC1NC(C1CNC(=O)C1)=O N1(CCNC(=O)C2=CCC2)CCCN(C(=O)CCn2cccn2)CC1 C1(C)(CNC(CN(C(COC)=O)C)=O)CCN(C(C2CCOCC2(C)C)=O)CC1 Cn1nc([N+](=O)[O-])cc1C(N1CCCC(F)(CNC(c2cc(=O)n(C)o2)=O)C1)=O C1(C)(C(=O)NCCC2CCN(CC(CC)CC)C2)CCC(C)CC1 C1(NC(c2c(C)n(C3CC3)nc2)=O)CN(C(=O)C(N2CCOC2=O)C)C(C)(C)C1 C1(C2CC2)(NC(c2ccc(C)c(C(C)(C)C)c2)=O)CCN(C(c2cnco2)=O)C1 C(CCC(C)C(=O)NCC=CCNC(c1n[nH]c(C)c1O)=O)OC N1(Cc2c(OC)nccc2I)Cc2ccccc2C1C(=O)Nc1cccnc1Cl C=CCCC(F)(F)C(=O)N1CCC(CCNC(c2ccccc2Cl)=O)C1 N1(C(c2ccc(C)nn2)=O)CC2CCC(C1)N2C(c1cnc(C)s1)=O c1(OC)ccccc1OC(F)(F)F.C1(C)C(=O)NCCCN(CCO)C(=O)COO1 C12(C(=O)NC3C(NC(=O)CCc4ccnc(Cl)c4)COC3)COCC1C2(F)F C=Cc1cncc(C(=O)NCC(C)(O)CNC(=O)C(=Cc2ccco2)C)c1 N1(C(C2(C(C)C)CC2)=O)CC(NC(c2cnn3cccnc23)=O)C(N=[N+]=[N-])C1 C=C=CCC(C(=O)NCC(C)Nc1c(C(C)=O)ocn1)NC(=O)OC.C(C)(C)(C)O C(CNC(c1ccn(C2CCOCC2)n1)=O)(CC)(CC)NC(C=CC=CC)=O C(=O)(C1=CC2(CCOC2)C1)NC(CNC(C1=C(C)OCCS1)=O)CC(C)C C1(F)(CNC(c2cc(C)no2)=O)CCN(C(c2ncccc2Br)=O)CC1 Cc1cc(=NCC(C)(C)C2=CCCC2)[nH]c(N2CC(C)OC(C)(C)C2)n1 n1(CCC=C)cc(C(=O)NCCN(C(=O)CC2CC=CCC2)CC2CC2)nn1 CC1(C)CCN(C(=O)CN(C(c2cc(C3CC3)on2)=O)CC2CC2)CC1 N1(C(C2(C3CNCCO3)CC2)=O)CCC(Nc2cc(C(F)F)ncn2)CC1 c1(OC)ccc(C(N2CCOCC2CN(C)C(C2CC2(C)Br)=O)=O)cc1O c1(C(=O)NC(C)C(c2ccccc2)NC(C2CSCCS2)C)cnc(CN)cn1 CC1CN(C(c2cn(C)nc2O)=O)CC(C)CN1C(c1ccnc(S)c1)=O Cc1nccc(CCC(=O)NCC(O)CN(C(=O)Cn2ccc(C(F)F)n2)C)n1 C1(C(C(=O)NCC=C)F)CCN(C(=O)C(c2ccccc2)O)C1 N1(C(c2cc(OC)ns2)=O)CCN(C)CC1C(=O)N(C1CCOC(C)C1)C Cc1cc(C(=O)NC(C2(O)CN(C(c3cccnc3C)=O)C2)C)c(O)nc1C C1(CC)(CNC(c2nnnn2CCSC)(C)CC2CC2)CCCCO1 N1(C(C2C(C)=CCS2)=O)CC(C(=O)NCC2CCCNC2=O)CCC1(C)C c1(NC(C(CC)N(C)CCO)=O)ccc(S(=O)(=O)N(C)C)cc1 C1(CC2CC2)CS(=O)(=O)CCO1.c12ccc(cc1)CN(C)C2=O.c1(O)cccnc1 c1(C(=O)NC2CC(NC(C(=O)OCC)=O)C2)ccc(S(=O)(=O)CC)cc1 n1(CC)ncc(Cl)c1C(=O)NC1(CNC(c2ccn(CC(F)(F)F)n2)=O)CCC1 N1(C(C2C(CCOC)C2)=O)C2CCC(C2)C1C(=O)N(C1CCCC1)C C1(C(=O)NC2CCC(NC(C3(CC)CC3)=O)C2)CCS(=O)CC1 C1(CCC)CN2CC1C2=O.C1(C(N2CC3CC3(CO)C2)=O)COCC(C)O1 Cc1nn(C)cc1CC(=O)NC(C)CCC(=O)NCC1CCCOCC1 C(=O)(C1=CC2CC(C1)CC2O)NCC1(F)CC(CNC(Cc2ccc(C)o2)=O)C1 Cc1cn2nc(N3CCOCC(CNC(=O)CCC4CCCCO4)C3)sc2n1 N1(C(c2c(C)nncc2)=O)CCN(C(=O)C=Cc2cc[nH]n2)C(CC(F)F)C1 C(=O)(C1=CCCOCC1)N(C1CC1)CC1N(C(C2ON=C(C)C2)=O)CCC1 C1(N(CC#C)C(c2csnc2Cl)=O)CCN(C(C2CCC(CN(C)C)O2)=O)CC1 C(=O)(C#CC1(C)CCCO1)NCC1C(C)(C)N(C(C2C3CCC(=O)C23)=O)CC1 N#CC1CN(C(=O)COC2CCCC2)CCN1C(=O)CCn1cncn1 C(C(=O)NCC1(C)CCCC1NC(C1CSCN1CC)=O)(C(C)C)OCCC CCN=C(NCC1(S(=O)(=O)NC(C)(C)C)CCC1)N1CCC(C(=O)N(C)C)C1 N1(C(CSc2n(CCC)c3c(n2)cccc3)=O)CCOC2(CCS(=O)(=O)C2)C1 C1(C(=O)NC2CCCC(NC(=O)CN3CC4CC4C3)C2)Cc2nncn2C1 N1(C(COCC(=O)NC)=O)CCC(O)(CCNC(c2cccc(F)c2C)=O)CC1 c1(C(=O)OCC)ccc(NC(=O)C(C)COC(C)(C)C)cc1Br N1(C(c2c(COC)noc2)=O)CCC(O)(Cn2cc(CCC3CCCC3)nn2)C1 C12(C(=O)NC(C3CCN(C(C(F)=CC)=O)C3)C)CC3CC(C1)CC(O)(C3)C2 CCCC(C)(O)CNC(C1(CC)CCN(C(=O)COC2CC2)C1)=O C1(NC(c2c(O)cccc2F)=O)COCCN(C(=O)Cc2ccc(Cl)c(F)c2)C1 c1(C(=O)NC(CNC(CCC(C)OCC)=O)CO)c(OC)cccc1O CC(CCCCN(C(=O)C(C)(C)F)CC)NC(=O)C(C)Oc1ccccc1.C(CCO)O c1(CCNC(N(C(CC)CC)C)=O)c(OC)ccc2ccccc12 CC1(C(N2CCN(C3CCCN(C(C4C=CCC4)=O)C3)CC2)=O)CCC(F)(F)C1 c1(-c2cnc(CCC(N3CC(C)(NC(=O)CSC4CC4)C3)=O)o2)ccc(F)cc1 Cc1cccc(CC(N2CCC(CN(C)C(c3ccns3)=O)C2)=O)c1 C(=O)(CC(C)C(C)C(C)C)N(CCN(C(C1CC2(C1)CC(OCC)C2)=O)CC)CC CCC(C)C(C(=O)NC1CCCC(NC(=O)C2=COCCO2)C1)SC N1(c2nnc(CC(C)C)s2)CC(NC(=O)C=CCF)C(C)C1 N1(CC)CCCC1CC(=O)NCCCN(C(=O)C(F)OC(F)(F)F)C C1(C(=O)Nc2cnc(OC)nc2)CN(C(C2CC3(C2)CC3(F)F)=O)C2(CCC2)C1 c1(C(N(C2CCN(c3cc(-c4ccccc4)ncn3)C2)C)=O)cc(Cl)cn1C c1(C(N2CCC(CN(C(C(C)OCC)=O)C)C2)=O)cc(Br)cnc1N C(=O)(C(F)(F)C1CCCC1)NCC(C)N(C)C(C1CC(OC(F)(F)F)C1)=O C(=O)(CCC(C)NC(c1ncncc1Cl)=O)NCCCC(C)C N1(CC(=O)NCCOCCNC(C2C(c3n(C)ncc3)C2)=O)CCC(=O)NC1=O c1(C(N2CCC(N(C(C3CC(O)C3)=O)CC)C2)=O)cc(C)c(F)cc1F c1(C2(CNC(C3CCN(C(C4CCNC4=O)C4CC4)C3)=O)CC2)cccc(F)c1 C(C(=O)N1CCC(C(=O)NCCCCS(C)=O)O1)n1ccc(C)n1 c1(CNC(C(C)OC)(C)c2nnnn2C(C)C)cc(F)c(Cl)cc1Cl Cc1cc(C(=O)NCCC(C)NC(c2cccc(F)c2C(C)C)=O)c(N)c(F)c1 C1(CC)CCN(C(c2cncc(O)c2)=O)C1C(=O)NOCC1CCCO1 C1(NC(C2(C)CC2(F)F)=O)CC2CCC1N(C(c1ccc(OCCF)cc1)=O)C2 CCC(O)C(C)C(=O)N1CCC(CO)(NC(=O)Cn2cc(C(F)F)cn2)C1 CC1CCC(NC(c2csc(C(F)(F)F)c2)=O)CN1C(C1CN(C)C(=O)N1)=O C1(CC#C)(C(=O)NCCC2COCCN2C(=O)C(C)n2ccnn2)CCCCC1 Cc1cc(C(=O)NCCCC(O)C(=O)N(C)Cc2ccn(C)n2)ncc1N c1(NC(CN2CCC(C#CC)C2)=O)cc(O)c(C)cc1C C=CC(C)(C)C(=O)NC1CC(C)N(C(=O)C(c2cccc(C)c2)=O)C1 C1(C)(CNC(COCCC(C)C)=O)CCCN(C(C2C=NN(C)C2=O)=O)C1 N1(C(C2CCC(CC)O2)=O)CCC(c2cn(C(C)C(=O)N(C)C)nn2)C1CC Cn1c(C(=O)NC2CC(O)CN(C(=O)C3=CCCC3)C2)cc2c1CCOC2 C1(NC(C(C=C=C)C)=O)CCN(C(C2(Cl)CCCCC2)=O)CC1F C1(N(C(=O)CCc2ccoc2)C)CCCCC1NC(c1coc(Br)n1)=O c1(NC(C(C)n2cnnn2)=O)ccnc(Sc2nncs2)c1 c1(NC(N(CCCN2CCCC2)CC)=O)c(Cl)cccc1[N+](=O)[O-] c1(C(=O)NCC(CCNC(C(=O)NCC(F)F)=O)O)ccc2ccccc2c1F Cc1ccc(Cl)c(O)c1C(=O)NCC(O)CN(C(=O)CC=CC(C)(C)C)C c1(N(C)C)nc2ccc(C(=O)NC3CC(C(=O)Nc4cccc[n+]4[O-])C3)cc2[nH]1 O=c1c2ccnn2cnn1CCc1ncc(C(F)(F)F)cc1Cl N1(C(C2(COC)CCC2)=O)CCCCC(CNC(=O)CCCCCO)C1 c1(C(=O)NC2CC(CNC(CCOCC)=O)C2)cc2c(C)c(C)ccc2[nH]1 c1(C(N2CC(NC(C3(C(F)F)CC(=C)C3)=O)C(O)C2)=O)cnc(C)nc1C C(=O)(CC1=Cc2ccccc2C1)N1CCCC(N(C(=O)CC2(C)CC2(Cl)Cl)C)C1 C=CCC(F)(F)C(=O)NC(C)CCN(C(=O)COc1ccc(C#N)cc1)C c1(C(=O)NC(Cc2cccc(CC=C)c2)C(=O)OC)nc(C)n2c1CCCC2 c1(C(N2CCN(C(C(C)=CC)=O)C(C3CC3)C2)=O)cnn2c1CC(C)CC2 N1(C(C2C(C)CCCC2)=O)CC2CC(C(=O)NCCC3(C)CC3)(C2)C1 c1(C(=O)NCC2CN(C(CCNC(COC)=O)=O)C(C)C2)c(F)cc(F)c(F)c1F N1(C(CC(C)F)=O)CC(C)(C)CC1CNC(C12CCC(CO)(CC1)C2)=O S(=O)(=O)(c1cccc(Cl)c1)N1C(C(=O)Nc2cnc(Cl)c(Br)c2)CC(F)C1 C1(C(N2CC(NC(c3c(OC)nc(Cl)cc3)=O)C2)=O)CCC2CC(C)CN2C1 C(=O)(CC(=O)NCC(O)CN(C)C(C1(SC)CCC1)=O)OCC c1(NC(CC2CC(=O)NC2)=O)nc2c(s1)CC(c1ccccc1)CC2 c1(C(N(C2CCN(C(C(c3cn(C)nc3)O)=O)C2)CCO)=O)ncc(Cl)cc1Cl C1(C(=O)NC(C)C2CC2)CCN(C(C2CC3(CCO2)CC3)=O)C12CCC2 C1(CC(=O)N(CCC(=O)NC)C(C)C)CCC(NC(c2ccc(C3CC3)o2)=O)C1 c1(C(C)C)ncc(C(=O)NCC2CCCC2NC(=O)C(C)CO)s1 c1(OC)ccc2nc(C(=O)NC3CN(C(C4CC4F)=O)CC3(F)F)ccc2c1 C1(C(=O)NCc2cccc(CNC(c3ccc(C)nn3)=O)c2)CC12CC(F)(F)C2 N1(C(CC2ON=C(C)C2)=O)CCC2CCCC12C(=O)NCC1CCOC1C C(CC(=O)N(C)CCN(C(C)C)CC)N(C(=O)CC1CC1C(F)(F)F)CC C1(NC(C2N(Cc3cc(C)[nH]c3C)CC(O)C2)=O)CCc2ccccc2C1 C(C(C(=O)NCCCCc1cnc[nH]1)C(C)C)NC(c1cc(C(C)=O)on1)=O c1(C(N2C(CNC(C(CCC)OCC)=O)CCC2)=O)cnn(C)c1C#N N1(C(C2N3CC(C)N(CC3)C2)=O)CCC2(CC1)CN(C(c1nc(Cl)c(Cl)s1)=O)C2 c1(C(N2CCC(CNC(C3(F)CCCC3)=O)C23CC3)=O)cc(Cl)cc2c1OCC2 C(c1ccc2c(c1)OCO2)=CC(=O)NCC1(N(C(=O)CC2CC=CC2)C2CC2)CCC1 N1(C(c2ccc3nnc(C)n3n2)=O)CC2C(C(F)(F)F)(CCS2(=O)=O)C1 CC1c2c[nH]nc2CCC1C(=O)NC12CC(CNC(=O)CC3CCCOC3)(C1)C2 Cc1ccc(-c2ocnc2C(=O)NC(C)CNC(C2C(C)(C)C2(F)F)=O)cc1 c1(C(=O)NCCC(C(C)C)NC(CC(COC)C)=O)ccc2oncc2c1 Cc1cncc(C(=O)NCC#CC(=O)NC2CCCCC2O)n1 C1(OC)CN(C(=O)CNC(=O)NC2CC2)CC1NC(c1cccc(N)c1)=O N1(C(C(CC)=CC)=O)CCN(C)C(C(=O)NCCN2CC3CCC2C3)C1 C1(NC(C(COC)C)=O)CC2(CCN(C(c3nnccc3C)=O)CC2)C1 CC(C)(C)CC(C)(C)C(=O)N1CCOCC(NC(C2CCC=CCCC2)=O)C1 N1(C(C(C)CC2CC2)=O)CCC(NC(=O)CNC(c2ccco2)=O)C(CO)C1 C(=O)(CC(C)(C)C(C)(F)F)N(C1CCN(C(C(C2CCOCC2)C)=O)C1)CCO C12(NC(=O)Cc3ccsn3)CCN(C(C3(n4cnnn4)CC3)=O)CCC1C2 C1(C(N2CC(CC(C)NC(Cn3c(C)ncc3)=O)C2)=O)CCc2ccccc2C1 C(=O)(CC(O)CCCCC)NCC(CC=C)NC(C1(CC#C)CCCC1)=O C1(C(=O)NCC(C)(CO)NC(c2cccc(CC#N)c2)=O)CCCC(=O)N1 CC(C)(C)C(CNC(=O)C=CC(N)=O)NC(c1c(Cl)nsc1Cl)=O N(C(=NCCS(C)(=O)=O)NCCS(=O)(=O)NC(c1ccccc1)C)C(CC)C C1(C(=O)NCC2(NC(=O)CCC(F)(F)F)CC2)CCC2(CCOC2)O1 Cc1cc(C(=O)NC2C=CCN(C(c3ccc(O)nc3Cl)=O)C2)cc(=O)n1C C1(F)(C(=O)NC(C#C)C)CCCN(C(c2cn(C)cc2C)=O)C1 N1(C(=O)CSc2nc[nH]n2)CCC2(CC1)CC2C(N1CCn2nccc2C1)=O C(=O)(CC(C)(C)CC(=O)N(C1CCN(C(=O)C2=CCCC2)CC1)CC(C)C)OC C1(NC(=O)OC(C)(C)C)CC(S(C)(=O)=NC(=O)C2CSCCS2)C1 Cc1cc(Cl)ccc1OCC(=O)NC1CCCC1CNC(C1CC2(CCC2)C1)=O c1(NC2CC(NC(C(C)C3CCOC3)=O)C2)cc(S(C)(=O)=O)ncn1 N1(C(COc2cc(C)on2)=O)CCCN(C(c2ccnc(C(N)=O)c2)=O)CCC1 C#Cc1cc(F)cnc1NC(C1CC1NC(=O)OCCc1ccccc1NC)=O C(=O)(C1=C(Cl)CCCC1)NC(CC(=O)NC(C)CC(C)(C)C)C(F)F C1(C(=O)NC(C#CC)(C)C)CCN(C(=O)CC(C)CN(C)C)C1C C#CCC(C)(C)C(=O)NC1CCCC(CNC(=O)C(C)(O)CC)C1 C(=O)(C(C)(C)COc1cnn[nH]1)NCC1(NC(c2nc(OCC)oc2)=O)CCC1 C1(C(N2CC3C(CC(=O)N(C4(C)CC(C)=NO4)CC)C3C2)=O)CCCCC(=O)N1 C1(NC(C(CC)O)=O)C=CCCC1C(=O)N(C)Cc1cn(C)nn1 C(c1cncnc1O)=CC(=O)NCC1N(C(C(COC)O)=O)CCOC1 CC(C)C(C(=O)NC(CNC(c1cncc(C2CC2)c1)=O)C1CCC1)N(C)C Cc1nc(C(=O)NCC(C)CN(C(=O)C(C)n2ccnc2)C)cc(O)n1 N1(C(C(F)=CCC)=O)CCN(C(c2nc(C)ccc2F)=O)C(CCO)C1 C12(C(N3CC(CNC(CC4C(C)(C)CCCC4)=O)C3)=O)CC1COC21CCC1 C(=O)(C(O)CCNC(=O)C(Cn1cncn1)NC(=O)C(CO)C1CCCC1)OC c1(C(N2CC(NC(C3CN4CCC3CC4)=O)C3C2C3)=O)cc(F)c(O)c(Cl)c1 CC(C)CCC(CO)NC(=O)CN(C(=O)C(C)CC1CC1)C c1(OC)cc(C2(C(=O)NC3CC3CNC(=O)C3=C(C)OCC3)CCC2)ccc1C c1(C(=O)NCCNC(=O)CC2CC3CC3C2)ccc2c(c1)C(=O)NCC(=O)N2 c1(OCCC(=O)NC2C=CCN(C(=O)C3=CCCS3)C2)ccc(Cl)cc1Cl C12(NC(C3C(C=C)OCC3)=O)CC3CCC(C1C2)N3C(c1ocnc1C)=O C1(NC(CSCC(N)=O)=O)CC(NC(C2CC2CCOC(C)(C)C)=O)C1 C1(C)(CNC(c2scc(OC)c2)=O)CCN(C(=O)Cn2nnc(=O)[nH]2)CC1 C1(C(N(C2CCCN(c3cc(O)nc(O)n3)CC2)C)=O)CC2(C1)CC2(F)F C#CC1(O)CC(C(=O)N(CCNC(=O)CSCC(F)F)CCOC)C1 N1(C(CCNC(C=CCOCCOC)=O)=O)CCC(C)(CN(C)C)C1 N1(C(CCC=CC(C)C)=O)CCC2(CC1)CC2NC(=O)CSCC1CCCO1 N1(C(C2CCCN(CC)C2)=O)CC2=C(C1)CN(C(=O)CCn1ccnc1)C2 C(=O)(C1CCCc2ccccc21)N1C(CN(C)C(c2ccncc2)=O)CCCC1 Cc1ccnc(C(c2nnnn2CC2CCCO2)NCC2(C(N)=O)CC2)c1Br c1(C(=O)NCCOC2CCN(C(C=CCCC(C)C)=O)CC2)ccc(=O)n(C)n1 C1(OC)(CNC(Cc2ccccc2)CO)CCNCC1 Cc1ccc(C(=O)NC2CC2NC(=O)C(C(C)C)c2ccccc2)c2c1CCC2 c1(OC)cc(NN(CCCO)CCCO)cc(C#N)n1.c12ccc([nH]1)C(=O)C(=O)CC2 N1(C(CC(CC)(F)F)=O)CC(NC(=O)Cc2cnccn2)CC12CCCCC2 CCC(C)C(C(=O)NC1CC1)NC(=O)Cc1ccn(C)c1 N1(C(C2CCN(C)CC2)=O)CC2(CC2)CC1C(=O)NC(c1ccc(Cl)cc1)CO C1(CC#C)(C(=O)NC2CCC2NC(C2CC3CC2C3)=O)CC=CCC1 CC(C)(CC(F)F)C(=O)N1CC(CNC(C2CNC(=O)C2)=O)C(O)C1 CCCCC(O)C(=O)NCC1(COC)CCN(C(=O)CNC(N)=O)C1 N(C(O)=C1C=CN=NC1=N)CC(C)(C)NC(C=CCN(CC(F)(F)F)C)=O C1(NC(C2(OCC)CCCC2)=O)CC2CCC1CC2NC(c1cnnc(C)c1)=O c1(C(N2C3CC4(NC(CCC=C)=O)C(C2CC3)C4)=O)ccnc2ccc(O)cc12 N1(C(C2C(=C)C2)=O)CCC(NC(=O)CC(C)(C)c2ccccc2)C(C)C1 C(=O)(CCS(C)(=O)=O)NC(CN(C(=O)CCOc1cccnc1)CC)C CCCC(CC)CCC(=O)NC(CNC(c1cnc2[nH]ncc2c1)=O)CC(C)C N1(C(COC2(C)CN(C(c3cc(C)c(F)nc3)=O)C2)=O)CC(CO)CC(C)(C)C1 N1(C(C2(SC)CCC2)=O)CCOCC(F)(CNC(c2cn3c(n2)COCC3)=O)C1 N1(C(C2CC(=C)C2)=O)CC2CCC1C(CNC(=O)CC1COC3(CCC3)CO1)C2 N1(C(CC2(C=C)CN(C(=O)C(C)(F)C(C)(C)F)C2)=O)CCn2c(C)cnc2C1 C1(CN(C)C(C2CC=CC2)=O)CCCN(C(=O)Cc2cn[nH]c2)C1 C1(OC)CC(C(N2CC(NC(C3CN(C(C)C)C3)=O)CC2C)=O)N(C(C)=O)C1 C12(C(=O)NC(c3ccc(Cl)cc3)C)CCC(C(N3CCCC(O)C3)=O)(CC1)CC2 c1(C(=O)NCC2(NC(CC3CC(SC)C3)=O)CCCC2)nccc(Cl)c1F Cn1cc(C(=O)CN2CC(C(F)(F)F)OC(CO)C2)c2cc(Br)ccc12 N1(C(CC(C)N2CCC(NC3CCC4CC4C3)C2)=O)CCC(O)C(C)(C)C1 O=C1CCC2(C(=O)NCC3CCN(C(=O)COC4CC(F)(F)C4)C3)SCCN12 c1(NC(C2(C)N(C(C(CC)O)=O)CCC2)=O)ncc(Cl)cc1[N+](=O)[O-] N1(C(C2(COC)CCNC2=O)=O)CCC(CC(N)=O)(NC(=O)CS(N)(=O)=O)CC1 Cc1ccc(C(=O)NC2(CNC(c3cc4oc(Br)cc4[nH]3)=O)CC2)c(F)c1Cl C1(C(=O)NCC2(C)CCC(NC(=O)CCCn3ccnn3)C2)CN2CCN1CC2 C=C1Cn2c(C(=O)NCC3CC(NC(c4nc(O)sc4C)=O)C(O)C3)nnc2S1 C(=O)(C#CC(C)(C)CNC(=O)CC1COCCOC1)NC(c1ccn(C)n1)C N1(C(Cc2cc(C)ns2)=O)CCC(O)(C(C)NC(c2oc(CO)cc2C)=O)C1 C(c1ccc(C(N)=O)o1)=CC(=O)NC(CC)CNC(C12CC(O)C1C2)=O C(C(C)N=c1cc(Cl)nc(C2(C)CC2)[nH]1)N(C(CCc1c(C)cccn1)=O)C c1(CNC(C(CNC(=O)Cn2[nH]cnc2=N)OC)=O)cccc(C)c1F Cc1ccnc2nc(C(N3CCC(N(C)C(C4CC(N(C)C)C4)=O)CC3)=O)nn12 c1(C(=O)NC(C2(O)CCN(C(c3cc(C)no3)=O)C2)C)ncn2ccccc12 C1(CN(C(C(C)CN2CCCCC2)=O)C)CCCN(C(=O)C(O)CN(C)C)C1 c1(OC)cnc(C(=O)NCC2CCC(C(=O)NCC(=O)O)CC2)cn1 c1(C2(C(N(CCNC(C(=O)NCC)=O)C)=O)CCC2)ccccc1F C1(N(C(CC(CN(C)C)(C)C)=O)C)CCN(C(=O)C(C)(C)CO)CC12CC2 N1(CCCCCC)CCC(NC(c2nccnc2C(N)=O)=O)C(C)C1 C1(c2nc(CC)on2)CCCN(C(=O)C=Cc2cc(OC)ns2)C1 c1(C(N(CC(C)CNC(=O)CNC(=O)C(C)(C)C)C)=O)ccc2nc(O)[nH]c2c1 Cc1cn2[nH]c(=NCC3CN(C(C4COC(C)(C)C4)=O)C3)sc2n1 N1(C(C(CO)OC)=O)CCN(C(=O)COC2CCCCC2)CC1C1CCCC1 C1(O)(C(C)NC(C2CCC2CF)=O)CN(C(c2ccc(-c3cccnc3)s2)=O)C1 O(NC(=O)C1=CC2C=CC1C2)CC=O.CC(C)(C)Cc1ncco1 C#CC1CCN(C(=O)C(C)CN(C(=O)Cc2ccn(C)c2)C)C1 c1(OC)ccc(C)nc1C(=O)NCC1CN(C)CCN1C(=O)C(CCSC)OC c1(C(=O)NC2C(NC(CC3N(C)CCCC3)=O)C2)cccc2c1OCO2 N1(c2nnc(COC)s2)CC2(CCC2)CC1CNC(C1CC2CCCC(C1)C2)=O C(=O)(C(C)(C)CC)N1CC(c2cn(C(C(=O)OCC)C)nn2)(O)C1 N1(C(c2c(C)cccc2)=O)CCN(C(=O)Cc2ncncc2Cl)C(C2CCC2)C1 N1(C(C(CC)C)=O)CC(NC(C2CC2c2ccc(F)nc2)=O)CC(F)C1 c1(OC)ccc(C(N2CCC(C)C2CNC(=O)C(C)OCC(F)(F)F)=O)cc1Cl C12(C(N(C)Cc3cn(CCCc4ccccc4)nn3)=O)CC1CS(=O)(=O)C2 C1(C(N(CCCCCCNC(C2CCC3CC23)=O)C)=O)Cc2ccccc2O1 N1(C(C(C)(C)SC)=O)CCC(N(C)C(c2ccc(C(C)C)nc2)=O)C(C)C1 C(CC(C(C)(C)C)N(C(C(C=C)CC)=O)C(C)C)NC(=O)COCCCCC CC1CN(C(=O)CCC(C)(C)NC(c2ccn(C)n2)=O)CCC1(F)F C1(C(=O)NCCOCC(C)C)(NC(C2CC(CC)C2)=O)CCN(C)C1 c1(CC)cc(C(N2CCCOCC2C)C(=O)NC2CCC2)ccc1Br c1(CNC(NCC(=C)Cl)=NCCC)ccccc1[N+](=O)[O-] c1(CNC(=O)C2=CCCC2)ccc2c(c1)CCC2NC(C1CC2(CSC2)C1)=O C#CCCC(=O)NC(C)(CNC(c1coc(CO)c1)=O)CC c1(C(=O)NCC(COC)NC(c2cccc[n+]2[O-])=O)cc(=O)c2ccncc2o1 c1(COC)ccc(C(=O)NCC2CC(O)(CNC(c3cnc[nH]3)=O)C2)o1 C1(CNC(C(C=C)OC)=O)CC(C)CCN1C(=O)C(CCSC)OC N1(C(CC2(OC)CC2)=O)CCC2(CC1)CN(C(=O)CCc1cc(F)ccc1F)C2 N1(C(=O)N(c2nc(C)cs2)CC)CCCCC1CCCSc1nnnn1C1CCCC1 C12COCC1NC2=O.N1(C(COCCC#C)=O)CC(OCCCCC)C1 C1(NC(C(CC)C(C)C)=O)CCN(C(=O)C=Cc2cc[nH]n2)CCC1CO c1(C(N2CC(OC(C)(C)C)CC3(C2)CC3)=O)ccc2ccccc2n1 c1(C(N2CCC(CN(C)C(c3sccc3Cl)=O)C2)=O)ncnc(O)c1F C=CCC(C)(C)C(=O)N1CC(O)(C2CCCN2C(C2CCCS2)=O)C1 Nc1cccc(C(N2CCC(OCCNC(=O)CCN(C(=O)CO)CO)C2)=O)c1O c1(C(N(C)CC2CCN(C(C3C(=C)C3)=O)C2)=O)noc(C)c1I c1(SC)ccc(CNC(C2(O)CCN(C(=O)CN3CCOCC3)C2)=O)cc1 N1(C(c2oc(C)c(CO)c2)=O)CCC(C(=O)N(CC(N2CCCC2)C)C)C(C)C1 C(=O)(C(F)CCC(C)C)N(C1CCN(C(CC2(OC)CCOCC2)=O)C1)CCO N1(C(C=CCOC)=O)CCC2(CC1)CC(NC(=O)C(C)CC(C)(F)F)CO2 N1(CCNC(C2C(C)CCCC2)=O)CCC(C(F)(F)F)C(F)(F)C1 C1(CNC(c2c(CC)nn(C)c2)=O)CN(C(C2(C)CCC(=O)N2)=O)CCC1C CCC(C(=O)OC)(c1ccccc1)NCC(C)(C)C1CC1(F)F C1(NC(C(CCC)=CCC)=O)CCCCN(C(c2cc(C)c(CC)o2)=O)C1 c1(C(=O)NC2CCC(CNC(C(CN(C)C)O)=O)CC2)ccc2c(ccn2C)c1 c1(C(N2CCN(C(Cc3cnc(C)[nH]3)=O)CC2C(F)F)=O)ncc(C#N)cc1Cl C(=O)(C#CC1(C)CCCO1)NC1C(NC(c2c(OC)ccc(C(F)F)c2)=O)C1 C(CCCCOC)(C(=O)NCc1cccc(Cl)c1)N(C(C(=O)NCC)C)C C(=O)(C1Cc2ccccc21)N1C(C(=O)NCC(C)(C)F)CCC1 C1(NC(C#CCNC(C2N(C)CCCC2)=O)=O)CCC2(CCCC2)C1 C1(C(=O)NCc2n(CC)cnc2)CCC2CCC1N2C(c1cnnn1C)=O C(=O)(CC(O)(c1ccccc1)C1CC1)N(CC(CNC(CC(=O)NCC)=O)O)C N1(C(C(c2ccc(F)cc2)(C)O)=O)CCN(C(C23CC(CO)(C2)C3)=O)C(CO)C1 c1(CC)n[nH]cc1C(=O)NCC(CC)NC(c1cnc(-c2ccccc2)o1)=O C1(O)(c2cccc(OC)c2)CCN(C(=O)CCCc2ccc(C)nc2O)CC1 c1(NCCNC(=O)NC2C3CCCCCC23)cc(F)ccc1Br C1(CNC(=O)CNC(c2ccoc2)=O)CN(C(C2CCC=CCC2)=O)CC12CC2 c1(C(N2CCC(N(C(=O)CC3CCCCC3O)CC#C)C2)=O)cc(C)nc(O)c1 C(N=c1[nH]c(N2CCC(F)(F)C(F)C2)nc2c(F)cccc12)c1ccc(C)s1 Cc1nc(O)sc1NC(=O)NC(C)C(=O)N(c1ccccc1)C C(=O)(C1=C(C)OCCS1)N1CCCC(C(N2CC(OC)C(O)C2)=O)C1C c1(C(N2CC(C(C(=O)N3CCC3C(C)C)OC)C2)=O)cc(C(N)=O)no1 c1(CC)cc(C(=O)NCCCN(C(=O)CCc2c(C)noc2Cl)C)nn1C c1(OC)cc(C(=O)O)ncc1NC(=O)Cc1nc(Sc2ccccc2)n[nH]1 CCCC(C(O)C(=O)NCC(CO)C(C)(C)C)NC(c1cnn(C)c1)=O C1(CNC(C2CCC(O)CC2)=O)CC2(CCC2)C1 c1(CC(=O)N(CCCN(C(=O)CNc2ncccn2)C)C)ccc(F)cc1 c1(CNC(COCCNC(CCn2ccc(C)n2)=O)=O)ncc(Cl)cn1 c1(C(C)C(=O)N(C)CC2(N3CCOCC3)CCCCC2)cccc([N+](=O)[O-])c1 c1(C(C)=O)cccc(-c2cn(CC(=O)NCC(=O)NC3CCS(=O)(=O)C3)nn2)c1 c1(C(=O)NCCC(C)N(C(=O)C(C)c2ccco2)C)cccc2c1CCC2=O c1(OC)cccc2c(C(=O)NC3CCCN(C(=O)C(Br)=C(C)C)C3)csc12 N1(C(C2(CCC=C)CCCC2)=O)CCCCC(NC(=O)CC2C(=O)NN=C2C)C1 N1(C(CCOC)=O)CCN(C(c2ccc(C3CC3)cc2)=O)CC1CCOC c1(CC)cc(C(=O)NC(CC)(CC)CCNC(c2c[nH]nc2OC)=O)ccc1Cl c1(C(N(CC(CN(C(C(C=C)O)=O)C)O)C)=O)scc2c1CCCC2 c1(C(=O)NC(C(C)NC(=O)Cn2ncnn2)C)conc1C1(C)COC1 N1(C(C#CC(C)C)=O)CCC(CNC(C2CCOC(=O)N2)=O)C(C)C1 C1(NC(CSCC(C)C)=O)CN(C(=O)CCc2cn(C)cn2)C2(CCCOC2)C1 C1(C)(C(=O)NC2CCCN(C(C(C(C)(C)C)=O)=O)C2)CCCNS1(=O)=O C1(NC(COCCN(C)C)=O)CCC2CC1CN2C(C1CCCCC1O)=O c1(C(N2C(CNC(CC3CC(CC)C3)=O)CCC2)=O)cc(C)nc2ccccc12 C1(CCNC(=O)C(C)OCC(C)C)(OC)CN(C(c2ccsc2)=O)C1 Cn1nc2ccccc2c1C(N1CCCC(C2CC2NC(=O)CCC(F)F)C1)=O C#Cc1cn(C)nc1C(=O)N(C)CC1(O)CCN(C(=O)CC2CCCC2C)CC1 C(=O)(CCC(C)N(C)C)NC(CC=C)CNC(C1CCOCC1)=O C12(CCNC(=O)NCc3cc(C)cc(Br)c3)CC3CC(CC(C3)C1)C2 c1(C(N(C2(C(N(CCOC)CC)=O)CCC2)C2CC2)=O)cc[nH]c1C N1(C(C2CC(NC(c3c(C#C)cccc3)=O)C2)=O)CCc2cnccc2C1 C1(O)(CN(C)C(c2conc2C2CCCC2)=O)CCN(C(=O)CSC2CC2)C1 C=CCC(C(=O)OC)NC(C1COC(CNC(=O)Nc2cn(C)nc2C)C1)=O C(C(CC(C)C)C(=O)NC(CC1ON=C(C)C1)C)NC(=O)CCCc1ccc(N)cc1 c1(CC)ccccc1CNC1CC(CN2CCOC(C)C2)C1 c1(C(=O)NC2CC3CC3C2)ccc(CO)nc1.C1(c2ccoc2)C(=O)N1 C1(CCC(N)=O)CC(N=c2[nH]c3c(c(=NCCCc4nccs4)[nH]2)COC3)C1 c1(CC(=O)N(C(C(=O)N(C(C)C(=O)OC)CCC)C)C)ccc2c(c1)CC2 c1(CC(=O)NCC2N(C(COCCC)=O)CC3CC32)cccc2nsnc12 C1(C(=O)NC(C(=O)NC2C(C)(C)C2(C)C)C2CCOC2)CC2(CCO1)CC2 c1(C(=O)NCC(CNC(=O)CC2CCOCC2)F)cnnc(-c2ccccc2)c1 CC1=NOC(CC(=O)NCC(C2CCC2)NC(C2CC(O)C2)=O)C1 c1(C(=O)NC2(C)CCN(C(c3c(COC)cc[nH]3)=O)C2)cccc2nn[nH]c12 C#CC1CCCN(C(=NCc2ccc(OC)nc2C)NCc2ccc(OC)cc2)C1 c1(C(=O)OC)n[nH]c(=NC2Cc3ccc(Br)cc3C2)o1 CCC(C(=O)N1CC(CNC(=O)COC(C)C)C1)n1cccn1 C(=O)(C1=NOC(C2(O)COC2)C1)NC(c1ccccc1)CNC(=O)COC(F)F Cc1cc(N2CCCC(NC(c3ccsc3Cl)=O)C2C)ncc1C#N C1(C(=O)NC)CCOC(C)(CC)C1.C#CCC1C(=O)NC2C(CC2)C(=O)N1 C1(NC(C(N2CCCCCC2)C)=O)(CNC(C2CCOC2=O)=O)CCCCC1 c1(C(=O)NC(C(=O)NC(CC)CCOC)Cc2cc[nH]n2)cc([N+](=O)[O-])n[nH]1 N1(C(c2c(COC)nn[nH]2)=O)CCCC2(C1)CN(C(=O)Cc1csc(Cl)n1)C2 C1(C(C)C(=O)N2CC(CCO)C2)CCN(C(=O)CN(C)C2CC2)C1 C12CN(CCC1O)C(=O)c1ncccc1-c1cn2nn1.C(c1cncc(C)c1)=C.CON CCCC(O)CC(=O)N1CC2C(c3cn(C(c4cc(C)cc(C)c4)C)nn3)C2C1 CCCC(C)(C)CC(=O)N(CCCCCC(=O)NCC(c1ccncc1)O)C C1(NC(CC2CCN(C)C2)=O)CCCCCC1NC(C1SCCCS1)=O N1(C(c2ccc(F)o2)=O)CC2(C1)CN(C(C13CCCC1C3(F)F)=O)C2 [N-]=[N+]=NC1CN(C(c2coc(Cl)n2)=O)CC1NC(=O)C(C1CCOCC1)F C(N=c1[nH]c2c(c(=NCC3C4COCC34)[nH]1)CSC2)c1nc(O)sc1 C1(CNC(C2(NC(=O)Cc3ccoc3)CC2)=O)CS(=O)(=O)CC1c1ccccc1 C(=O)(CCCC(C)(C)CC)N1C2CC(C(=O)NC(CC#C)C(=O)OCC)C1CC2 N1(C(C)C)C2CCC1CC(C(=O)NCCC1(NC(=O)C3=C(Cl)CC3)CC1)C2 N1(C(C=COCC)=O)CC(C)N(C(=O)Cc2nnc(O)s2)CC1C c1(OC)cnc(SC)nc1N(C1CCNCC1F)C(C1CCC(C(C)C)CC1)=O Cc1cc(C)[nH]c(=NCC2(CS(N)(=O)=O)CCC2)n1.c1(CC(C)C)ccc(F)cc1 C(=O)(C1=CCC(C)CC1)NCCN(C(c1cc(OCCC)nc(Cl)c1)=O)C(C)C C#CC1CCCN(C(C2CCC(Cn3cc(CC4CCCN4C)nn3)CC2)=O)C1 C1(C(=O)NC2C(CNC(CCOCCC)=O)COC2)COc2cc(Cl)ccc2C1 Cc1ccc(F)c(C(=O)NCCC2(C)CCN(C(C3CCCC(=O)N3)=O)C2)c1F CCCCCS(=O)(=O)CC(=O)NCC(CCNC(=O)Cn1ccc(C)n1)OC N1(C(CCCSC)=O)CCC(C)C(NC(c2coc(C3CCOCC3)n2)=O)C1 C(C)(C(C)(C)C)CN(C1(C(=O)N(c2ccccc2Cl)C)CCOC1)C.c1(C(C)CC)ccccc1 c1(C(=O)NC2(C(F)F)CC(NC(C=NOC)=O)C2)cccc(Cl)c1 c1(C(=O)NC2CCCCN(Cc3c(C)nn(C)c3)C2)ccc2ncsc2c1 n1(CC)nc2c(c1C(N1CCCC(N(C(=O)C(C)N=[N+]=[N-])C)C1)=O)CCCC2 c1(N2C(C)(Cc3ccc(F)cc3F)CCC2)nc2c(c(=N)[nH]1)CCCC2 N1(C(CS(=O)(=O)NC)=O)CCOC2(CCN(C(C3CC(C(=O)OC)C3)=O)C2)C1 C1(NC(C(C)C2CC2)=O)COC2(CCN(C(=O)C(c3ccc(F)cc3)C)CC2)C1 c1(SC)cccc(-n2nc(-c3cc[nH]n3)nc2C2CC3C=CC2O3)c1 C#Cc1ccc(C(=O)N(CC(=O)NCCCS(C)=O)CCC)cn1 C(CCCC(=O)NC1CCN(C(c2cccc(C)n2)=O)C1C(C)C)OCCC=C C1(CNC(CCC2CCN(C(c3c(CC)cccc3)=O)C2)=O)CC2CC1CC2O C(=O)(C(CNC(=O)C(C)(C1CC1)OC)CC=C)NC(C#C)C1CCC1 N#Cc1ccsc1C(=O)NCC1(F)CC(NC(C2CCCC(C3CC3)O2)=O)C1 C1(COC)CCCN1C(C1(CCl)CN(C(C2CC2c2cccs2)=O)C1)=O CC(C)(C)CCCC(C(=O)Nc1ccccc1)N1CCOC(C)(C2CC2)C1 C12(C(N3C(C)CC(C)(C)C3)=O)CCCC1CN(C(c1ccc(CO)cn1)=O)C2 C1(C(N2CC(CC(C(=O)N(CCO)C(C3CC3)C3CC3)F)C2)=O)CCCC12CCC2 S(=O)(=O)(c1cc(C(=O)OC)c(Br)cc1F)N1CCCN(CCOC)CC1 N1(C(c2c(C)n(C)nc2)=O)CC(C2(NC(=O)CC3CC3C)CC2)C1 C(=O)(CCCCN=[N+]=[N-])NCC1C(C)(C)C1C(=O)NCC1(O)CCCOC1 CC(C)(O)CC(=O)N1CC2C(C(N3CCC(c4cnco4)C3)=O)C2C1 C12(C(=O)NCCC(C)(C)NC(c3n(C=C)ncc3)=O)CCCC(=O)N1CCC2 CCCCC(C)C(=O)NCCC1CN(C(C2CC(CC(F)F)C2)=O)CCCO1 C1(CNC(C(C)N(C(C2(COC)CC=CC2)=O)C2CC2)=O)OCCCC1(C)C c1(CC)nc(C(F)(F)F)oc1C(N1CC(C)(CS(C)=O)C1)=O N1(C(C(CC)F)=O)CC2(CCN(C(C3CCSC3)=O)C2)C1 CC1=C(C(=O)NC(CNC(=O)C(=O)N(C)C)CO)CCC1.C1CS1 CC(C)C(O)C(=O)NCC1C(CO)CCN1C(=O)C=Cc1ccn(C)c1 C1(C(=O)NCc2ncccn2)CC(F)(F)CN1C(=O)CN1CCOCC1 c1(OC)ccc(NC(c2ccc(CCC(=O)NC3CCCCC3)[nH]2)=O)cc1C#N N1(C(C(CC(C)C)C)=O)CCOC2CN(C(c3cnc4n3CCCCC4)=O)CC12 C1(C(N2CC(NC(=O)NCC)C2)=O)C=CCN(C(c2ccn(CCF)n2)=O)C1 N1(C(CCSCC)=O)CCCCC1C(=O)N(C1CCOCC1C)C C(=O)(CCCCCNC(C1CC2(C1)CC2F)=O)NCC(C)CNC(N)=O Cc1occ(C(F)(F)F)c1C(N1CCCC(N(C)Cc2cccc(N)c2)C1)=O CCCCC(CNC(C1CC=C(C)CC1)=O)NC(c1cc(C)c(CC)s1)=O c1(OC)c(C(=O)NC(c2ccccc2F)(C)C)cccc1C#N C(=O)(CCCC(C)(C)NC(=O)C(F)=CC1CC1)NCCC1(C)CCOC1 C(=O)(NNC(=O)N(C)CC)NC(CC)Cc1nn[nH]n1 N1(C(C2C(OCC)C2)=O)CCC2(CC1)CC(C)N(C(=O)CC1CC(OC)C1)C2 C(=O)(CCC1CCc2ccccc21)NC1C(C)CN(c2nc(Cl)ncc2Cl)C1 c1(C(=O)NCC2CC(NC(=O)Cn3cnnc3O)C2)cc2c(o1)CCCC2 C1(CC)(NC(=O)CCN2CCOCC2=O)CCCN(C(=O)CC2(O)CCOC2)C1 c1(CC(=O)NCC(CCOC)NC(c2nnn(C)c2N)=O)n[nH]c2c1CCCC2 N1(C(c2c(C)nn(C(C)C)c2C)=O)C2CCC1CN(C(c1ccncc1N)=O)C2 N1(COCC)CCCC(C)(NC(C2(C(=O)NC3CC3c3ccc(C)s3)CC2)=O)C1 C(=O)(C1CCc2ccccc21)N1CCCCC(C(N(c2cnn(C)c2Cl)C)=O)C1 N1(C(Cc2cc(C)sc2)=O)CCC(F)(C(=O)NCCCC(O)CO)C1 N1(C(C(C)C(C)O)=O)CCN(C(c2ccc(C(F)F)cc2F)=O)C(CCO)C1 Cc1nc2cc(C(=O)NCC3CC(F)(CNC(=O)C(C)CN(C)C)C3)ccc2s1 c1(CC)nc(C)c(C(=O)NCCCCC2CCCN(C(C3(C)CCCO3)=O)C2)s1 c1(C(=O)NCC(C)CN(C)C(C2(CCN(C)C)CC2)=O)ccc(Cl)s1 c1(NC(=O)CN2CCCCC2)ccnc2c1CCCC2O Cc1cc(O)ncc1C(=O)NC1CC=CCC1C(N1CCCC1CN(C)C)=O C(=O)(CC(C(F)F)C(C)(C)C)N(CC(C)(C)NC(C(C(C)C)(C)C)=O)C c1(OC(C)C(=O)NC2CCC2NC(c2cc(C(N)=O)c[nH]2)=O)cc(Cl)cc(Cl)c1 C(=O)(C(F)(F)CCn1cccn1)NC1CCCN(C(c2nn(C)c(O)c2)=O)C1 C1(NC(C(OC)OC)=O)CCCC(CC(=O)NCc2cn(C3CC3)nn2)C1 c1(C(=O)NC(CN(C(C2(CC=C)CCCC2)=O)C)C)ccc(-c2cscn2)cc1 N#Cc1cc(S(=O)(=O)N(C2CNC2)Cc2ccc(-c3ccccc3)s2)ccc1F Cc1cc(NC2CCOCC2)cc(C)c1OCC(F)(F)F c1(C(=O)NC(C)(CNC(C2CCCN2N=O)=O)CO)noc2ncccc12 c1(C(N(CC(=O)Oc2cccc(C=C)c2)C(CC=C)=O)=O)c[nH]c(=N)nc1C C1(C(=O)NC2(C(=O)NCC(C)(O)C3CCC3)CCCCC2)CC(=O)NC(=O)N1 C1(F)(CNC(CSCCCC)=O)CC(CNC(=O)Cc2cc(C)cs2)C1 Cc1noc(C)c1C(C)C(=O)NCC(C)CN(C)C(C1CC(F)C1)=O N1(C(c2cnc(C)o2)=O)CC(NC(=O)Cc2cc(O)nc(O)n2)CC2(CC2)C1 Cc1cccc(F)c1C(=O)NCC1(F)CC(NC(c2ncc(C(F)F)s2)=O)C1 C1(O)(CN(C)C)CCN(C(C2CC(O)CN2C(=O)C=Cc2cn(C)cn2)=O)C1 C=CCCCC(C1CC1)NC(c1[nH]ccc1CNC(C1(SC)CC(C)(C)C1)=O)=O C1(C)(C(=O)NC(C2CC2C(=O)NCC2(F)CCOC2)C)CNC(=O)N1 N1(C(CN(CCC)C)=O)CCCCC1CN(C)C(c1ccn(CC)c1C)=O FC(F)(F)CCCc1nc(-c2nccs2)nn1CCOCCS N1(C(c2cnc(C(C)=O)s2)=O)CCC2CCC(C1)N2C(C1CCC1C)=O O=C(C#CC1CC1)NCCN(C1CCCC1)C(C1CC1c1occc1Br)=O C1(CNC(Cn2c(C)cnc2)=O)CCN(C(=O)C(CO)N(C)C)CC1O c1(N2C(C)CNC(=O)C2)ncnc2[nH]c(=N)ccc12 c1(C(=O)NCCC2CCCN(C(CCC(C)O)=O)C2)cccc(C#N)c1 C(=O)(C(C)CC(C)(F)F)N(C1CCCN(C(=O)C=Cc2ccsc2)C1)CC C1(C)(C(N2CCCC(NC(c3ccc(C(C)(C)C)s3)=O)C2)=O)CCCC1(F)F N1(C(C2CCCO2)=O)C2CCC1CC(CC(C)Oc1ccc(OCC)cc1)C2 N1(C(Cn2c(C)c(Cl)cn2)=O)CCC2(CCC2)C(NC(C2CCCC(F)C2)=O)C1 N1(C(c2c(Br)ccc(C#N)c2)=O)CCC2(CC1)CC(NC(C1(CO)CC1)=O)C2 O=S(=O)(c1cc(C(=O)O)sc1Br)N1CCC=C1Cl C(=O)(C(O)CN1CCCC1)NCC1(CC(=O)NCC(C2CCOCC2)O)CC1 Cc1cn2c(n1)CCC(N=c1ccc(Oc3ccccc3)n[nH]1)C2 C(=O)(C1CN(C)C(=O)c2ccccc21)N1CCC2CN(C(CCOC)=O)CC21 C1(CNC(=O)C(F)n2cccn2)CCCCCN1C(c1ccccc1)=O c1(C(N(CCNC(=O)C(C)Cc2ccccc2F)CC)=O)c(C)cccc1F Cc1ccc2c(=NC3CCC3C)[nH]c(=NCCc3ccccc3Cl)[nH]c2c1 c1(C(N2CCN(C(C(C)(C)NC(=O)NCC)=O)CC2C)=O)cc(F)c(F)cc1F CC12CC(C1)C(CN1CCCC(c3cccc(F)c3)C1)CO2 N1(C(c2c(C)con2)=O)CCC(NC(c2cc(Cl)cc(C)c2N)=O)C(F)(F)CC1 c1(OCC)ccc(C)nc1C(=O)N(CCCOCCNC(=O)C=C(CC)CC)C CC(C)(CNC(C1CCn2ccnc2C1)=O)CS(N)(=O)=O C1(C(=O)OC(c2ccc(Cl)cn2)C)CCC(C)(C)O1 Cc1cc(N)ccc1C(=O)NC1CCCCC1NC(C1CC1c1ccn(C)n1)=O c1(C(N2CC(COC)N(C(c3ccno3)=O)CC2)=O)c(Br)ccc2c1OCO2 c1(NCC)cccc(C(=O)NC2(C)CN(C(=O)CNC(C3CC3C)=O)C2)c1 N#Cc1ccc(=NCC2(F)CCN(C(C3CCOC3)=O)CC2)[nH]c1 c1(C(N2CCN(Cc3ccc(F)cc3O)C3CC23)=O)ccc2cccnc2c1O N1(C(C(c2cccc(Br)c2)C)=O)CCCC(C)(CNC(=O)C(C)(C)F)C1 N1(C(C(C)NC(N)=O)=O)CCC(CNC(=O)C(C)(C)CCCF)C(C2CC2)C1 Cc1cc(C)c(NC(=O)C(N2CCCC(C)(CO)C2)c2nc(Br)sc2C)c(C)c1 N1(C(CC2(C)CCCO2)=O)CC2CCN(C(c3coc(Br)c3)=O)C2C1 c1(CC)ccc(C(N2CC3CC3(CNC(=O)CCCOC(C)C)C2)=O)nc1 c1(C(N2C(CCNC(C3(CC)CC3)=O)C(C)CCC2)=O)cc([N+](=O)[O-])cc(C)n1 C1(NC(CNC(CC(C)C)=O)=O)CCN(C(c2ccc(CN(C)C)[nH]2)=O)C12CC2 C1(COC)CN(C(=O)Cn2ccc(C)n2)CCN1C(C1CCC(C)CC1)=O c1(CC(=O)NCCC(CC)(C)NC(c2ocnc2C)=O)ccc(O)c(F)c1 c1(C2(C)CC2)cc(C(=O)NCCC2CSCCN2C(=O)C(C)(F)F)n(C)n1 N1(C(C2(C=C)CC2)=O)CCC(NC(=O)Cc2cc(F)cc(Cl)c2)C(O)C1 N1(C(c2c(NC(CN3CCC(C)CC3)=O)cco2)=O)CC(C)OCC1C c1(OC)ncnc(OC)c1C(=O)NCC1CCC1NC(c1ccc(F)c(O)c1)=O c1(CC)cc(C(N2CC=CC(NC(c3cc(O)nc(OC)n3)=O)C2)=O)cc(F)c1 c1(CC)ncccc1C(N1CCCC1C(C)(C)C(=O)N1CCC1CC1CCCC1)=O c1(NCCC(CC)OC)cc(=NC(C)C(C)CC)[nH]c(C(C)C)n1 C(CC(=O)N1CCCOC(C)C1)(C(F)(F)F)NC(C1(CSC)CC1)=O N#Cc1cccc(C(N2CCCC2CCNC(c2cnn(C(F)(F)F)c2)=O)=O)c1 c1(C(=O)NCC(F)N)cccc2cncn12.N1(C(C(=O)CO)=O)CCN(C2CC2)CC1 c1(C(=O)NCC2(NC(C34CCC3C4)=O)CCC2)sc2cc(F)ccc2c1Cl c1(C(N2CC(NC(c3ccc(C)cc3Cl)=O)C(F)C2)=O)ccc(C#N)c(F)c1F Cc1cc(C(=O)NC2CCN(C(=O)CCC3CCOC3)C2C2CC2)cc(C)n1 CC(C)CC(CNC(c1cccc(CC#N)c1)=O)NC(=O)CCCN(C)C c1(C(=O)NCC2(OCC)CN(C)C2)cnc(C)cc1C C(=O)(CCC(CC)CCC)N(CCC(N1C(C#C)CC1)=O)CCCO c1(NC(N2CCC(c3cn(CC4CCC4)nn3)C2)=O)cc(=O)n2ccccc2n1 Cn1cnc2c1CCCC2C(=O)N1CCCC(CNc2c([N+](=O)[O-])cnn2C)C1 c1(C(N2CC(CCCCC)C2)=O)c[nH]nc1CCNC(=O)C(C)(C)OCC c1(C(=O)NC2CC(CC(=O)NCC3C(OCC)CC3)C2(C)C)cccc(O)c1F CCC(C#N)C(=O)NC(C(=O)N1CC(F)(C#N)C1)C(C)OC c1(C(N2CC3(CN(C(C4CC(=O)OC4)=O)C3)C2)=O)cnc2ncnc(O)c2c1 c1(CC(=O)NC2CC(OC)CN(C(=O)CCF)C2)ccc2c(c1)OC(F)(F)O2 c1(CC(C)NC(C2CC3CCC2N3C(=O)CCC(C)(C)C)=O)c(F)cccc1F N1(C(C(C(C)C)OC)=O)CCN(C(c2ccc(OC(C)C)nc2)=O)CC(C)(C)C1 C1(C(CN(CC(=O)N(O)Cc2cn(C3COCC3O)nn2)C)=O)CCC(=O)CC1C Nc1cccc2cc(S(=O)(=O)NC3CCCC3)ccc12 Cn1c(C(N2CC3CN(C(=O)C4=CCOC4)CC3C2)=O)cc2ccccc12 N1(C(CCC(C)OCC)=O)CCC(O)(CNC(=O)CSc2ccc(F)cc2)CC1 C(=O)(C(=O)N=S(C)(C)=O)N1CC(C)C(NC(=O)Cc2cn3ccsc3n2)C1 c1(OCC)nn(C)cc1NC(=O)C#CCNC(C1CCC(C)C1)=O CCC(C(=O)NC(CNC(c1c(C)coc1C)=O)CC(F)(F)F)C(C)(F)F Cc1oc(C(=O)N(CCNC(C2CC2(C)Br)=O)CCOC)cc1CO Cc1nc(O)[nH]c1C(=O)NCC(Cc1ccccc1)NC(C1(F)CCCOC1)=O N1(C(C2N(C(CCCC)=O)CC3CC32)=O)CCC(O)CC(C)(C)C1 C1(NC(CC(CC)OC)=O)CC2CCC(C1F)N2C(=O)CCNC(N)=O N1(C(C2(OCC)CCOC2)=O)Cc2ccc(CNC(C3CC3(F)Cl)=O)cc2C1 c1(C(N(CC(C)O)CCNC(c2c(C)nn(C)c2F)=O)=O)ccn2nccc2c1 C(=O)(C1CCCc2cccnc21)NCC(C(C)C)NC(=O)CCN(S(C)(=O)=O)C CCC(C)C(O)C(C)C(=O)N1CCCC(CC)C1C(N1CC(OCCOC)C1)=O c1(CN2C(C)CN(C(=O)Nc3cc([N+](=O)[O-])nn3C)C2)cc2ccc(F)cc2[nH]1 C(=O)(C1OC(=O)c2ccccc21)N(C)CC1CCN(C(C2C(C)C2)=O)CC1 N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CCN(C(=O)CCCN=[N+]=[N-])C2COCC12 c1(C(N(CC(CNC(C2C(C)=C2)=O)(C)C)C)=O)cc(C)c(Cl)c(C)c1 c1(NC(C)=O)cnc(O)c(C(=O)NCC2CC2CNC(=O)Cc2nc(C)no2)c1 N1(CC(=O)NC(C)CNC(c2cocn2)=O)CCOCC1=O N1(C(C(C)(C)O)=O)CCCC2(CC(NC(c3nccc(Cl)c3F)=O)CO2)C1 N1(C(CCC(C)OC)=O)CCCCC(NC(c2c(C(F)(F)F)coc2C)=O)C1 CCCC(C)(C)CC(=O)NC1CCN(C(=O)Cc2ccnc(F)c2F)C(C)C1 N1(C(C2N=C(C)SC2)=O)CC2(CCCC2NC(=O)CCOc2ccccc2C)C1 c1(NC(c2n(CC=C)nnn2)c2ccc(COC)s2)cccc2c1OCC2 N1(C(C2CC(OCC)C2)=O)CCN(C(=O)CC(C)(C)O)CC1CC(C)(C)C N#Cc1ccccc1CCC(=O)NCC1(O)CCCN(C(C2(O)CC2)=O)C1 CC(C)(CNC1CCC(NC(=O)OC(C)(C)C)C1)C1=CCOCC1 N1(C(c2cnc(CC(C)C)[nH]2)=O)CCC2CCN(C(=O)Cc3cncnc3)C2C1 CCC(CC(=O)NC1CC(C(=O)NC(CO)CC(F)(F)F)C1)C(F)F C(=O)(C(C)(O)C(F)(F)F)NCC1C(NC(c2cn(C(C)C)nn2)=O)C1 N1(C(CCCC(C)=O)=O)CCCC(C)(C)C1C(=O)Nc1ccc(N=[N+]=[N-])cc1 CCC(C)C(O)C(=O)N(CCCN(C(=O)CC1CC2CCC1CC2)C)C CCC(C)(O)C(=O)NCCC(C)(C)NC(=O)Cc1ccno1 N1(C(C=C(CCC)CCC)=O)C2CCC1CN(C(C1CC13CCC3)=O)C2 C(=O)(C1=CCC(F)(F)CC1)N(CC)CC.C1(=O)CCC(=O)NCC(C)N1 n1(C(C)C)cncc1C(=O)N(CCNC(c1cnn(C)c1)=O)Cc1ccccc1 C1(N(C)C(c2cnn(C)c2)=O)CCN(C(C23CCCC2CC3)=O)CC1 Cc1cc(=NC2CCC(S(C)(=O)=O)C2)[nH]c(=NCC(C)(C)c2ncccc2F)[nH]1 Cc1ocnc1CC(=O)N(C)CCN(C)C(C1(c2cncnc2)CCCC1)=O C1(CNC(C(C)OCCOCC)=O)C(CNCCC(=O)NC)C1(F)F c1(C(=O)OC)ccc(NC(=O)NC2CCN(c3cccc(Br)c3I)C2)c(OC)c1 C#CCCC(=O)NC(C)CNC(c1nnn(-c2ccccc2)n1)=O c1(C(N2CC(NC(C3(CC#C)CC3)=O)CC2(C)C)=O)cc(O)cc(F)c1F C12(C(=O)OC)CCCC1(C(N1CC(C)(NC(=O)CCC3CC3(F)F)C1)=O)C2 C1(NC(CC(CNC(c2nocc2C)=O)OC)=O)CCc2c[nH]nc2C1 c1(CC(=O)NCCN(C(c2cccc(OCCC)c2)=O)C)c(C)nc(O)nc1O C(CC(=O)N1CCC(CCCNC(=O)CC(C)C(C)(C)C)CC1)(C(F)(F)F)OC C1(C(N)=O)COCC1C(=O)NC1CC(O)C1CC(=O)NC1CCCN1CC1CC1 c1(C(N(C(CCNC(c2c(C)cncc2)=O)C)C)=O)ncc(N)cc1Cl c1(C(=O)NC(C(C)C)CNC(=O)C(C)P(C)(C)=O)cc2ccncc2s1 c1(C(=O)NCC(CNC(c2[nH]nnc2C)=O)OC)ncc2c(F)cccn12 c1(C(=O)NC2CN(C(CSc3n(C)nnn3)=O)CC(O)C2)[nH]nc2ncccc12 C(=O)(C1=Cc2ccccc2OC1)N1CCC2(NC(CN(C)S(N)(=O)=O)=O)C(C1)C2 C#CCCC(O)C(=O)NC1CN(C(c2ncncc2Cl)=O)CC1O c1(C(C)C)cc(CC(=O)NCC2CC2NC(c2ncsc2Br)=O)on1 C1(COC)(NC(c2ncc(C(F)F)s2)=O)CCN(C(c2sc(C)cc2C)=O)C1 C1(C(=O)NCCNC(C(C)C)=O)CC(O)CN1C(=O)CC(C)C1CC1 c1(C(N(CCC)CCNC(C2CSC2)=O)=O)cncc(C(C)(C)C)c1 c1(C(N2C(C(C)NC(c3c(C)cccn3)=O)CCC2)=O)nc2c(s1)CN(C)CC2 C(=O)(CC(C)C(=O)N(C(C)C(=O)NCC(O)C(C)O)C1CC1)OC C1(c2n(CC=C)nnn2)(NCc2ncc(CCCCCC)[nH]2)CCCCC1CC c1(C(C(=O)NCCSC)N(C2(C#N)CC2)C)ccc(-n2ccnn2)cc1 c1(C(=O)OCC)c(NC(=O)C(C)CC)sc2c1CCC(C)C2 C1(NC(CC2CC(OCC)C2)=O)CN(C(C2C=CCS2)=O)CC1SC CC(N=c1nc(Br)[nH]s1)C1CC2(CCC2)C1 C(=O)(C1=CCCC(C)(C)C1)N(CCCNC(c1ncccc1Cl)=O)C1CC1 c1(C(N2CC(CN(C)C(C3CC4CC3C4)=O)OCC2)=O)cnc2[nH]cncc1-2 c1(C(=O)NCC(COC)NC(C2COC(=O)N2)=O)cc(Cl)cn1C Cc1ccc(C=CC(=O)NCC2(C(N)=O)CN(C(c3cncn3C)=O)C2)nc1 N1(C(C(C)OCCC=C)=O)CC(C2CN(C(c3cccc(OC(C)C)n3)=O)C2)C1 C1(OCCNC(C(CC)OC)=O)CCN(C(c2cc(Cl)cs2)=O)CC1 N1(C(CN(C(C)=O)C)=O)CC(NC(c2cc[nH]c2C2CCCC2)=O)C(C2CC2)C1 CC1CN(C(c2cnc(C(C)(C)C)o2)=O)CC1NC(=O)CC1COCC1O C1(CNC(=O)Cc2ccco2)CN(C(c2cncc(C3CCCC3)c2)=O)C2CC12 c1(NC(c2ccco2)=O)ccc2c(c1)CN(C(C1(O)CCOCC1)=O)C2 N1(C(CCNC(=O)NC)=O)CCOC(CN(C(=O)C(O)C2CCC2)C)C1 C(C)(C(=O)N=c1cc(C)n(C2CC2)[nH]1)N(C(c1cc(COC)[nH]n1)=O)CC N1(C(C(OC)OC)=O)CCOC(CCC2CCCN2C(C2CCOC2)=O)C1 N1(C(c2cc(C)ns2)=O)CCC2C(CCN2C(c2[nH]cnc2C#N)=O)C1 C1(COC)CCN(C(=O)CC2CCN2C(C2(OC(C)=O)CCOC2)=O)C1 C(C)(C(C(=O)NC(c1nocc1C(=O)N(CCCN=[N+]=[N-])C)C)N(C)C)OC N1(C(CN(CC#C)C(c2ccc(OC)s2)=O)=O)CC2CC(C)C2C1 C12(CNC(=O)OC(C)(C)C)COCC(CN3CCCC3C#N)(C1)C2 C1(NC(C(C=CC)O)=O)CCC12CN(C(c1cnc(Cl)[nH]1)=O)C2 C1(C(=O)NCCCN(c2nc(C)c(Br)cn2)C)CC2CC(O)CC(C1)C2 C1(N(C(c2cccc(C(=O)NC)n2)=O)C)CCCCN(C(=O)C(C)C2CC2)C1 N1(C(c2ccc(CC)cc2OC)=O)CCN(C(=O)C(C)(O)C(C)(C)C)CCC1C Cc1ccc(OCC(=O)N(C2CN(C(C3(O)CCSC3)=O)C2)C)cc1 c1(NC(CCC=CC)=O)ccc(NC(c2cc(Cl)cnc2O)=O)cc1C c1(C(=O)NC2CCN(C(c3cc[nH]c3)=O)CC2O)ccc2cc(Cl)ccc2n1 c1(C(=O)NCC(CC=C)NC(C2(CO)CCCO2)=O)cc(S(C)(=O)=O)cs1 c1(C)ccc(C)cc1.c1(CC(N2CC(NC(=O)CO)(CO)C2)=O)cccc(Cl)c1 C(=O)(CCCC(=O)NC1CCC(C)N(C(c2ccc(F)cc2)=O)C1)NCC C1(N(C(c2c(C)snn2)=O)C)CCN(C(c2ccc(O)nc2Cl)=O)CC1C N1(C(C2C(OC(C)=O)C2)=O)CC2CC1CN2C(=O)C(C)=C1CC1 CC1CCN(C(C2CC3CCC2O3)=O)C1CNC(c1cc(C(C)(C)C)ccn1)=O C(=O)(CCCC(=O)N(C)C)NCC(CC)NC(c1c(C)nnn1CC)=O N1(C(c2cncc(Br)c2)=O)CCCC2(CCN(S(=O)(=O)c3ccc(Br)cn3)C2)C1 c1(C(N2C3C(NC(C4(COC)CC=CC4)=O)CC(C3)C2)=O)cc2n(c1)CCOC2 C12(CC)CC(C(=O)NCC3(C)CCN(C(=O)C(C)(C)CC4CC4)C3)(CO1)C2 N1(C(C2CS(=O)(=O)C2)=O)CCC2(CCN(C(C3(C4(O)CCC4)CC3)=O)C2)C1 N1(C(CCCOC)=O)CCN(C(c2ccnnc2)=O)CC1C(C)(C)C c1(C(=O)NC2CCCC2NC(C2(F)CC3(CCC3)C2)=O)c(OC(F)F)cccc1Cl C1(CNC(CC=CCC)=O)CN(C(c2cnn(CC)n2)=O)C2(CCOCC2)C1 Cc1cc(C(=O)NC2CC(O)(CNC(c3cccc(OCCF)c3)=O)C2)cn1C c1(CC(=O)N(C2CCN(CCCCC=C)C2)CCC)ccc2cccnc2c1 CC12CC(C(=O)NC3(C4CCCN4C(c4cc(CO)on4)=O)CC3)(C1)C2 S1(=O)(=O)c2ccc(c(Cl)c2)C(=O)NCCC(C)N1.C(C(C)C)NC(=O)OC N1(C(c2cc(OC)ccn2)C(=O)NCC)CCC2(CC(CO)C2)C1 c1(C(=O)NC2(C(=O)NC(c3nc(C)on3)C)CCN(C)C2)ccc(F)c(O)c1 Cc1cc(N)n2ncc(C(N3CC4(NC(C5CCCC5)=O)CCC3C4)=O)c2n1 N1(C(C2C(C)=CCC=C2)=O)CC2(CCCC2NC(=O)C=Cc2cccs2)C1 C1(C(N(C)CCNC(=O)Cc2cccnc2)=O)CC(C)(C)C1C(F)(F)F C(CC(F)(F)F)(C(=O)O)NC(c1csc(C2CCCCC2)n1)=O N#Cc1cncc(NC2CCCCN(C(C34CC5CC3C4C5O)=O)C2)n1 N1(C(C(C)N(CC)CC)=O)CCC(C2CC2)(NC(c2cc(C(F)F)n(C)n2)=O)C1 N1(C(Cc2ccc(C)s2)=O)CC(CC(N2CCN(C(C)C)CC2)=O)CC1(C)C C(=O)(CS(=O)(=O)c1ccccc1Cl)N1C(C)CCN(C(COCCC)=O)CC1 S(=O)(=O)(c1ccncc1)N1CC(CC)N(C(=O)C(C)CC(N)=O)CC1 Oc1c(CN2CCCC(Cc3ccc(Br)cn3)C2)cccc1Br C12(C(N3CC(OC)C(NC(=O)C=C4CCCC4)C3)=O)CCCC1OCC2 c1(N(CCOC)C)cc(N2CCOC(c3ccccc3Cl)C2)nc(C)n1 C1(NC(C2(SC)CC2)=O)CCCCC1NC(c1cc(C(C)C)nn1C)=O Cc1[nH]nc2ncc(NC(C3CC4(CC4)CN3Cc3cc(Cl)ccc3F)=O)cc12 CC1CCC(O)(C(=O)N(C2CCN(C(C3OC4CCC3C4)=O)CC2)C)CC1 N1(C(CC(C)(C)n2cc(CN(CC)CC)nn2)=O)CCn2cc(C)nc2C1 c1(C(=O)NCc2c(CNC(=O)CC34CCCC3C4)cccn2)cc(Cl)ccc1O N1(C(Cn2c(C)ncc2)=O)CC(NC(=O)CSc2ccccc2)C(F)(F)C1 n1(CC)nnc(C(=O)NCCN(C2CCCCC2)C(=O)CC2CCC(=O)N2)c1C N1(C(c2c(C)n(C)nc2)=O)CCc2cccc(O)c21 Cc1nc(N2CCC(CC(=O)N(C)CC3(O)CCCCC3)C2)n(C)n1 Cc1nccc(N2CCC(OCc3nc(C4CCC4)no3)C2)n1 C1(NC(C(CC=CC)NC(C2CCC2C(C)(C)C)=O)=O)CN(C)C2(CCC2)C1 CC(Cn1ccnc1)C(=O)N(CCCCCNC(c1ccc(Cl)o1)=O)C(C)C n1(CC(=O)NCC(CNC(c2cncc(OC)n2)=O)O)ccc([N+](=O)[O-])n1 C#CCC(O)C(=O)NCC(C(C)C)NC(=O)CCSCc1ccccc1 CCC(CC)C(C)C(=O)NCC1CN(C(c2cc(C(C)C)n(C)n2)=O)CCCO1 C1(NC(C(CSC)NC(CC=CCCCCC)=O)=O)CCc2n[nH]cc2C1 N1(C(C(CC=C)(C)N(C)C)=O)CCC2CCN(C(C3(C)CC=CC3)=O)CC2C1 C(C(N=c1cc(Cl)nc(C)[nH]1)C1CC1)NC(c1ccc(CNC(CC)=O)cc1)=O c1(OC)ccc(O)cc1C(=O)N(CCCCN(C(=O)C(C)(C)SC)C)C Cc1cc(C(=O)NCCCCNC(c2ccsc2Br)=O)ncc1CO N1(C(CN(CC)Cc2ccccc2)=O)CC2(CC(NC(=O)C(C)C3CC3)C2)C1 N1(C(c2c(C)oc(Cl)n2)=O)C(CC(N2CCC(O)CC2C)=O)C2CCCC12 C12(C(N3CCCC(CNC(C4CC(=O)NCC4)=O)C3)=O)CC(C1)S(=O)(=O)C2 C1=CCONC1=O.C(C(=O)N(C1(C(O)CO)CC1)C)SCC#C N1(C(CCc2cn(C)nc2)=O)C2CCC1CN(C(C13CCCCC1C3Br)=O)C2 N1(C(c2cn(C(C)C)nc2)=O)CCC2(NC(=O)C(=O)NCC(F)F)CCCC12 c1(NC(C2CC(C(=O)N)C2)=O)ncccc1C.c1(CC)ccc(C(=O)O)[nH]1 c1(OC)cnc(CNC(=O)C(O)CCNC(=O)C(F)(F)CO)cn1 Cc1ccc(N)c(C(=O)NCC2CCCC(CNC(=O)C(O)CC(C)C)C2)c1 C1(C(=O)NCC(C)N(C(=O)COCC2CCC2)C)CC(O)C1 c1(COC(=O)Nc2ccccc2)ccc(C(=O)NCCSC(F)(F)F)cc1 C1(CNC(c2csc(C(F)F)n2)=O)CC2(CCC2)CN1C(C1(O)CCSCC1)=O N1(c2ccc(-n3ccc(C)n3)nn2)CC2(CN(CCc3ccc(F)cc3)C2)C1 c1(CC)ccc2c(c1)C(CC(=O)N1CC(F)CC1CNC(=O)CC(C)O)C(=O)N2 C12(NC(=O)Cn3cc(C(F)F)cn3)CN(C(=O)C=CC(F)(F)F)CC1CS(=O)(=O)C2 C1(C(C)C)CN(C(=O)C2=NOC(C)C2)CCN1C(=O)Cc1cc(C(F)(F)F)n[nH]1 C(=O)(CCCn1cc(C2CC=CC2)nn1)NC1(CC=C)CC1 Cn1cnc2ccc(C(=O)NC3(CO)CN(c4nnc(C5CC5)o4)C3)nc12 c1(CN(C2CNC2)C(c2cscc2Cl)=O)ccc(N2CCOCC2)c([N+](=O)[O-])c1 CCCCC(CNC(=O)COCCOC)NC(c1csc(Br)c1)=O CC1CCCC(C(=O)NCC(C)(F)CNC(=O)CN2CCCCC2=O)CC1 C1(C)(C(N2CCC(CN(C)Cc3nnc(-c4ccco4)o3)C2)=O)CC(C)(C)C1 Cc1cc(C(=O)Nc2cccc(C(F)(F)F)c2)c(C)n1Cc1ccncc1 c1(C(N2C(C(=O)NC(c3cnc[nH]3)C)CC3(CC3)C2)=O)n[nH]c2cccc(F)c12 c1(OCC)cccc2c1OCC(C(=O)NCCN(CCOC)C(c1ccon1)=O)=C2 c1(C(N2CCC(CN(C)C(C3(C)CNC(=O)C3)=O)C2)=O)ccc(CC#N)cc1 N1(C(c2ccc3sncc3c2)=O)CCCCC2(CCN(c3ncc(Br)cn3)C2)C1 C(=O)(CC1=NNC(=O)C1)NC1CCN(C(CCCCOCCC=C)=O)C(CC)C1 Cc1c(C(=O)NC(C)(CNC(=O)C(C)CC(F)F)C2CCC2)cccc1F C1(COC)CN(C(=O)Cc2ccccc2Cl)CCN1C(=O)CC(C)C1CC1 N1(C(c2c(C)scn2)=O)CCC(NC(C23COC(CF)(C2)C3)=O)C(F)C1 C(=O)(C1=C(Cl)CCCC1)NCCC1(C(=O)NC2C(CCOC)C2)CCC1 C(=O)(C(O)CC(N)=O)C(=O)CC1(N)CCC1.CC1(OCCN)CCOCC1 C1(CCNC(COCCCOC)=O)CCCN(C(c2c(C)ccnc2C)=O)CC1 Cc1[nH]nc(CO)c1C(=O)NCC1C2CN(C(c3cnc(N(C)C)cn3)=O)CC12 c1(C(=O)NC(CNC(C2(CC=C)CC=CC2)=O)(C)C)cccc2c1oc(=O)n2C c1(C(=O)NCCC2(NC(CS(=O)(=O)NC)=O)CCC2)nccn2nccc12 c1(C(=O)NC2CCCN(C(c3ccn(CCF)n3)=O)C2)cc(Cl)ncc1F C#Cc1cccc(CC(=O)NCCOC(C)(C)CNC(C2SCCC2C)=O)c1 C1(CNC(C=CC=CCC)=O)CN(C(c2ccncc2C)=O)CCC12CCOC2 C1(N(C)C(c2cscc2C(F)F)=O)CCCN(C(=O)C(c2cnn(C)c2)=O)C1 c1(N(CC=C)C)nc2cc[nH]c2c(=NC2CCC(=O)N(CC)C2)[nH]1 c1(C(CC)(C)C)ccccc1NC(=O)NCC1(C(=O)OC)CCOCC1 CC(CS(C)(=O)=O)C(=O)NCC1(C)CCCC1NC(c1ccc([N+](=O)[O-])cc1)=O N1(C(C(C)(C)NC(CCc2n(C)ncn2)=O)=O)CC2CC3CC2C1C3 O=CCS(=O)(=O)CC(F)(F)F.C1(COC)COCCN1C(=O)C(F)CC1CCCC1 N1(C(CCC(=O)NCC)=O)CCN(C(=O)C(CO)OC)CC1c1ccccn1 c1(C(N2CC(NC(C(c3ccc(C)s3)C)=O)C(C)C2)=O)ccc2n[nH]cc2c1C n1(CC)ncc2cc(C(=O)NCC3CC(CNC(C4(Cl)CC4)=O)CO3)cnc12 Cc1cc(O)c(C(N2CC(NC(=O)C(C(C)C)OCC(C)C)C2)=O)cc1F C1(C)(COC(C2C(OC(C)(C)C)C2)=O)CCS(=O)(=O)CC1.C12CCCCN(C1)C2=O C1(NC(C(CC=CC)C)=O)CCN(C(=O)COc2cccc(C)c2)CC1(C)C c1(C(=O)NCC(C)CN(C)C(c2cc(O)nc(O)n2)=O)ccnc2ccncc12 c1(C(=O)NC2C(NC(C(C)C)=O)CCC2)cccc(-c2cc(O)ns2)c1 C1(O)(C(=O)OCC)CCN(C(=O)CCC2CC2)CC1.c1(CCC)nc[nH]n1 c1(OC)cnc(Cl)[nH]c1=NC1CCCCC1NC(C12CC1COC2(C)C)=O Cc1cc(C(=O)NCC23CC(CO2)N(C(C2CC(O)C2)=O)C3)cnc1C(F)(F)F c1(C(=O)NC2CCN(C(C3C(OC)C3)=O)C2)cc(O)nc(Br)c1 C1(CNC(C(C)SCC)=O)CC2(CO1)CN(C(C1(C)CS(=O)(=O)C1)=O)C2 Cc1scnc1C(N1CC(OCCC(=O)NC2(n3ccnn3)CC2)C1)=O N1(C(c2c(CC)non2)=O)CCCCC1CCNC(C1CC2CCC1C2)=O C12(CCNC(C(C)(C)SC)=O)CCC1CN(C(=O)C(C)(C)n1ccnn1)C2 CN1CCOCC12COCCN(N1CC(n3cnc4c3CCCC4)C1)C2 C1(CCC(=O)OC)(CN(C2CC2)Cc2nccs2)CC1(F)F c1(C(N(C(C)CN(C(=O)C(CCO)N(C)C)C)C)=O)cc2cc[nH]c2cn1 N1(C(C)C)CCOC(C(=O)NC2CC(NC(=O)CCN3CCOC3=O)C2)C1 c1(-c2n(C)ccn2)ccc(NC(C2CC2C2CCC2)=O)nc1 c1(C(N2CCC(CNC(C3(C)CC(=C)C3)=O)(OC)C2)=O)c(Cl)cncc1Cl N(C1c2ccccc2CC1O)C(N1CC(c2ccccc2)C1)=O N1(C(C(CC)=CCCC)=O)CCC2(CC2C(=O)NCCc2cc[nH]n2)C1 C1(NC(C2CC=C(C)CC2)=O)CC2CCC(C1)N2C(C1(C)CC(C(F)(F)F)C1)=O c1(C(C)C)n[nH]cc1C(=O)NCC(C)(C)NC(=O)Cc1csc(Cl)n1 C1(F)(C(=O)NCC2(O)CN(C(c3c(C(C)C)ocn3)=O)C2)CCOCC1 Cc1c(C(N2CCCC(O)(CCNC(C3CCCO3)=O)C2)=O)[nH]c2ccccc12 Cc1ncc2c(n1)CC1CCC2NC(=O)C(=O)N(C)CC1CCCNC N1(C(C2C(COC)CC2)=O)CCN(C(=O)CNC(=O)CCSC2CCCC2)CC1 c1(C(=O)NCCOCCCN(C)C(C2(C)CCOC2)=O)cccc2ccn(C)c12 C1(N(N2CCCCOC2=O)C(C)=O)C2CCCOC2C1(C)C.c12cccc(c1)OC2=O C1(C(=O)NCC2CC(C(=O)NCC(C)OCCO)CO2)(CC)CC=CC1 N1(C(Cc2c(C)nccc2)=O)CC(NC(=O)CC2(N3CCCC3)CC2)CC(O)C1 S(=O)(=O)(c1ccccc1C#N)NC1CC(C(=O)Nc2cc(C(=O)NCC)sc2)C1 CC(C)C(F)(CNC(=O)CCc1ccccn1)C(=O)N1CCC(C(F)F)C1 c1(OC)ccnc(C(=O)N(C(C)CNC(c2cnc(C(C)O)s2)=O)C)c1OC C(c1ccncn1)=CC(=O)NC1CC(CC(=O)NCC2(CO)CCOC2)C1 CC1Cc2cc(C(N(C3CN(C(=O)CC45CCC(CC4)OC5)C3)C)=O)ccc2O1 c1(C(N2CC(C(N3CC4C(NC(C)=O)C4C3)=O)C2)=O)ccc(C)c(F)c1F C1(C2CCN(C(=O)C(CO)C(C)C)CC2)(CNC(CNC(C)=O)=O)CCOCC1 Cc1cccc(C(=O)NC2COCC2NC(c2ccc(CO)o2)=O)n1 C(C)(C)(CCC(=O)N1CCCC(O)(CCNC(=O)C2=CCCC2)C1)OC N(C(=NCc1cn(C)cn1)N1CC=C(c2c(F)cccc2F)CC1)C(C=C)C c1(CC(=O)NC2CCCC(NC(c3nnn(C)n3)=O)C2)cc(Cl)ccc1Cl c1(CC)ncccc1C(=O)NC(C)CCC(=O)NCCNC(C)=O C(=O)(C1=CC2(CCOCC2)C1)N1CCN(C(CCc2cc(C)on2)=O)C(C)C1 c1(CC)ccc(N(C(c2n[nH]c(C)n2)C(=O)NCCCF)CC)cc1 c1(C(N(CC(=O)O)Cc2scc(C)n2)=O)cccc2cc(Cl)ccc12 N1(C(C(=O)NCc2cc(Oc3ccc(F)cc3)ccn2)=O)CC2CCC(CC2)C1 Cc1cc(F)ccc1C(O)C(=O)NC1CN(C(c2nc(Cl)ccc2N)=O)CC1F C1(C(=O)NCCCn2cc(Cn3ncc(C)c3)nn2)(N(C)C)CCCOC1 C1(NC(CC(=C)I)=O)CCN(C(=O)CNC(=O)COC)C1C1CC1 N1(C(C2(C)CCC2)=O)CCC(F)(CNC(=O)CC23CCCC2C3)C1 c1(N2CCC(CC)C2)nc(NCC2CCCC2O)cc(C)n1 C(C(C)(C)CC(=O)N1CCN(C(c2sc(C3CC3)nc2C)=O)CC1CF)OC CC1CCCC(C(N2CC(CCNC(c3cnnn3C)=O)C2)=O)CC1 C1(CCC)CCCC1C(=O)N(CCC(=O)NCc1ncc(C)o1)CC c1(CC(N2CC(C)C(NC(C3CCC(C(F)(F)F)C3)=O)C2)=O)ccc(O)c(F)c1 C(N=c1[nH]c2c(c(=NCc3cnc4n3CCC4)[nH]1)CCC2)c1cc(CC)[nH]n1 Cc1cc(C)c(CC(=O)NC(C)C(C)NC(=O)CC2COCCOC2)c(C)c1 c1(C(=O)NCC#CCNC(C(C)C2CCOC2)=O)cc2n(c1)CCCC2 c1(C(=O)NC2CCN(C(Cc3cc(C)[nH]n3)=O)CC2C)ncc2n1CCCC2 C1(C(=O)NCC(=C)CCNC(C2CCCS2(=O)=O)=O)CCOCC12CCCC2 c1(NC(N)=O)ccc(C(=O)NCC2(NC(C34CSCC3C4)=O)CC2)cc1 C1(NC(CCNC(COC)=O)=O)CC(NC(=O)CN(C)C)C(O)C1 N1(Cc2nc(OC)cc(NC3CC3C(=O)OC)n2)CCC2(CCCN(C)C2)C1 C1(CNC(C2(COC)CC=CC2)=O)CN(C(C2C=CCCC2)=O)CCCO1 c1(C(=O)NC(CNC(c2n(CC)nnc2)=O)CO)cnn(CCO)c1C(C)C O=C1OC2CC(C(=O)NC3CCC(NC(C4(CCF)CCC4)=O)C3)CC2O1 Cc1cc(C(=O)NC(C)CCCC(=O)NCC(C)(C)CCO)c[nH]c1=N C1(F)(C(N(OC)Cc2ccccc2)=O)CCCN(C(c2cnc(C)cc2C)=O)C1 C=CCCC(O)CNC(C1(F)CCN(C(=O)CCNC(=O)COC)C1)=O C(=O)(C(C)CC(=O)c1cccc(F)c1)N(CC(CNC(C#CC(C)C)=O)C)C C#CC1(F)CCN(C(C2CC(C)CN(C(c3nc(C)ccc3F)=O)C2)=O)CC1 c1(C(=O)NC(CC)CN2CCCC2)conc1C(C)NC(=O)C=CC1CCC1 N1(C(CN(C)CC)=O)CCCC(C)(C)C1CNC(=O)C(C)Cn1cccn1 C1(C(=O)NCCN(C(c2ccc(C(C)=O)[nH]2)=O)C)CCC2(CC1)CC2 C(=O)(C1=C(C)CCOC1)NCC1N(C(CC=C)=O)CCC1 CCC(C)C(CNC(=O)CCN(C(=O)Cc1cn(C)cn1)C1CC1)OC C1(C(N(C2CCN(C(c3cnc(C)s3)=O)C2)C)=O)CCC(=O)N1CCC(F)(F)F N1(C(C(CC)F)=O)CCN(C(c2cccc(=O)o2)=O)CC1c1ccc(F)cc1 Cc1[nH]c(C)c(C(=O)NCCN2CCN(C(=O)CC3OCCC3(C)C)CC2)c1C c1(C(=O)NCC(C)(C)CO)cc2cc(-c3cccc4c3OCCO4)cnc2[nH]1 c1(C(C(N)=O)NC(=O)NC23CCC2C3)cccnc1 C1(O)(C(C)NC(c2n[nH]cc2Cl)=O)CCN(C(=O)Cc2ccc(Cl)cc2)C1 C1(NC(C2N(C(COCC(=O)OC)=O)CC3(CC3)C2)=O)CC2CC1OC(=O)N2 c1(C(=O)NC2(CNC(C3C(OCC)C3)=O)CCCC2)cccn2nnnc12 CCCS(=O)(=O)CC(=O)NCC(C)N(C)C(C1CC=CCC1)=O c1(CC(=O)NC(CN(C(c2cn(CC=C)nc2)=O)C)C)ccc2c(c1)CCCO2 Cc1cccc(NC(=O)C(n2cc(Cl)cn2)C)c1S(C)(=O)=O C(=O)(CC(CC)CC)NCC(=C)CCNC(=O)CCc1cccc(OC)n1 CC1OC2(C)CC1(C(N1CCC1CNC(C1CC(F)C1)=O)=O)C2 C1(C(=O)NC2CC(NC(C(c3cnn(C)c3)C)=O)C2)C2COCC12 N1(S(c2c(C)onc2)(=O)=O)CCCC2(CCN(C(=O)CC(C)(O)CC(=O)O)C2)C1 c1(N(C(=O)CCNC(c2ccc(C)cn2)CO)CCC#N)cc(Cl)ccc1Cl CN1CCCC(C(N2CCN(C3CN(C(=O)CC4CCSC4)C3)CC2)=O)C1 C1(CNC(C(C)NS(C)(=O)=O)=O)COCCN1C(c1cccnc1N)=O c1(C(=O)NCC2(O)CC(CNC(=O)Cn3ccnn3)C2)ccc(Cl)cc1 N1(C(c2n(CC)ccn2)=O)CC2CC1(CNC(=O)C(C1CCOCC1)OC)C2 C(C(C(=O)NCC(C)(C)C(F)F)C(C)(C)C)NC(COCC(=O)NC)=O C1(C(=O)NC2CCC2O)(CC)CN(C(c2c[nH]cc2CC)=O)C1 CCCCCCCCC(=O)N1CCC2CN(C(c3scc(OC)c3OC)=O)CC12 N1(C(c2cccc(OC)c2F)=O)CC2CCC(C1)N2Cc1cn(C(C)(C)C)nn1 c1(OC)nc(C(=O)NC(C)(C)CNC(c2cn(C3COC3)nn2)=O)ncc1F c1(C(=O)NCC(CN(C(C2(CC(C)C)CC2)=O)C)C)cc2occc2s1 C1(NC(C(CC)OCC)=O)CCCCN(C(=O)CNC(=O)OC(C)(C)C)CC1 C(=O)(C1=NNC(=O)CC1)NC(CCNC(c1cc(C)n(-c2ccccc2)n1)=O)C c1(C(N2C3C(NC(C4C5CC6C(C5)C46)=O)CC(C3)C2)=O)cc2c(s1)CCOC2 C(CC(=O)OCCCOCC(=O)NCC)SC.CCCNCCNC(C)C C(CCCCCNC(c1nnnn1C1(C)CC1)(C)C)NC(CN(C)CCO)=O Cn1ccc(C(C)(C)C(=O)NC2CN(C(=O)CC3CC3c3ccccc3)C2)n1 c1(C(=O)NCCN(C(c2ccc(O)nc2C)=O)CC)ccc(C)cc1[N+](=O)[O-] N1(C(C(CC=C)C)=O)CC2(CCCN(C(=O)CN(C)C(c3ccccc3)=O)C2)C1 N1(C(Cn2nc(C)n(C)c2=O)=O)CCCC2(NC(c3cn(C)nn3)=O)CC2C1 Cc1nc(-c2nn[nH]n2)ccc1NC(C1CCCN(c2nccs2)C1)=O Cc1cncc(C(=O)NC2CCN(C(c3cc[nH]c3C3CC3)=O)C2C(C)C)c1C C1(CNC(c2cc(SC)oc2)=O)C(C)CCCN1C(c1cc(=O)c(OC)c[nH]1)=O N1(C(c2c(C)oc(Cl)n2)=O)CC(NC(=O)C(C)(C)C2CC2)CC12CCOC2 c1(C(N)C(N2CCCC2c2noc(N)n2)=O)ccc(F)nc1F c1ccc(F)cn1.CC1(c2cn(CC(F)(F)F)nn2)CN(N2CCC(C=O)C2)C1 c1(N2CCCC(CC)C2)nc(=NCC23CCCCC2CC(=O)N3)[nH]c2c1CSC2 c1(C(=O)NCC2(C)CC(NC(c3ccoc3CC(N)=O)=O)C2)ccc(F)cc1F c1(CNCC2OC(C)=C(C(=O)OC)C2)nc2ccc(Cl)cc2n1C C1(OC)(OC)CC(NC(=O)N(C(c2ccccc2F)CO)C)C1(C)C C1(NC(C2(CC=C)CN(C(c3cc(C(C)C)no3)=O)C2)=O)CCc2nn[nH]c2C1 Cc1cc(C(=O)NC(c2cnn(CC3CCC3)c2)C)n(C(F)F)n1 CCCC(C)(C)CC(=O)NC1CCCCN(C(c2snnc2C2CC2)=O)C1 C(CCCC(=O)OC)NCCOCC.C1(=O)C(OC)CNC(=O)CCN1 N1(C(C(C)CO)=O)CCCC2(C1)CN(C(=O)Cc1cc3nc[nH]c3cc1Br)C2 c1(C(=O)NC2CCC(NC(c3cc(COC)[nH]n3)=O)C2)ccc2[nH]c(=N)oc2c1 c1(NC(CC)CNC(=O)C2CC2)ccccc1SC(C1(C(F)F)CCOCC1)=O C(c1ccc2[nH]ccc2c1)=CC(N1C2CN(C(C(C(C)(C)O)F)=O)C(C2)C1)=O C1(NC(c2ccnnc2O)=O)CN(C(c2ncccn2)=O)CC1F Cc1ccc(-c2nnc(C(C)OC3CC3c3ccc(Br)s3)o2)c(C)c1 C1(O)(CNC(c2cc(Br)ccc2O)=O)CCCN(C(=O)CC2CCCCO2)C1 CC(C)C#CC(=O)N1CCC1Cn1cc(C2CCC(C(=O)O)C2)nn1 C(=O)(C(C(=O)OOC(F)(F)F)OC)NCC1CN(C(CCSCCCOC)=O)C1 c1(OC)ccc(OC)c(C(=O)NC2CC(NC(=O)C=CC3(C)COC3)C2)n1 N1(C(C(CN(CC)CC)F)=O)CCC(COC)(NC(c2ccnn2CC)=O)C1 n1(CC(=O)NCC(C)N(C(=O)Cc2ccc(Cl)cc2Cl)C)cc(F)ccc1=O c1(NC(C2C3(CCN(Cc4nc(C)oc4)CC3)C2)=O)cc2c(cc1Br)OCCO2 C1(C(=O)NC(C2CCCN(C(c3ccco3)=O)C2)C)CCC2CC1C2(C)C N1(C(c2cc(Cl)c[nH]2)=O)CC2=C(C1)CN(Cn1nnc3c1CCCC3)C2 C=CC(C)C(C)C(=O)NCC1(F)CN(C(=O)C(F)(F)C2CCCC2)C1 c1(C(C(=O)NC2CN(C(C3(C)CCC3)=O)CC2O)O)ccc(F)cc1Br c1(C(=O)Nc2n(CC)ncc2)nc2ccc(-c3cc4ccccc4[nH]3)cc2s1 c1(C(=O)NC2(CC)CN(C(c3cnc(OC)c(C)c3)=O)C2)cc(C)c(C)nn1 Cn1cc(C=CC(=O)NC(CO)C(=O)NCC(=O)NC(=O)NC2CC2)nn1 c1(NC(C(CCF)NC(C(C(=O)OC)OC)=O)=O)cnc2ncnn2c1 c1(C(=O)NCC(C)(C)NC(=O)Cc2ccco2)ncc[nH]c1=O C(=O)(CC(F)(F)F)NCC(C)(C1CCC1)NC(CCNC(C1C(C)C1)=O)=O Cc1cc(CC(N2CCC(C(C)NC(=O)COc3ccon3)C2)=O)cc(C)c1 c1(-n2cc(C(CC)(C)NC(=O)CNc3ccccc3)nn2)ccccc1CO O=C(CC1OCCc2ccsc21)NCCNC(c1c[nH]c2cc(Cl)ccc12)=O N1(C(C(=O)NCC)=O)CC(NC(c2cnc(OC)s2)=O)CC12CCCC2 c1(OC)nc(C(N2CCCC2CNC(=O)C2=CC(C)(C)C2)=O)cc(O)n1 N1(C(C(CN(C(COC(C)C)=O)C)C)=O)CCC2(C1)CN(C)C2 c1(C(=O)NCC2(F)CCN(C(C3CCCOC3)=O)C2)cc(F)cc([N+](=O)[O-])c1 N1(C(CCS(C)(=O)=O)=O)CCC2(C1)CN(C(C1CCC(N=[N+]=[N-])C1)=O)C2 N1(C(C(C=C)CC)=O)CCC(C)(C)C(CNC(=O)CC(C)(C)N(C)C)C1 C(=O)(CC(CCC)NC(=O)C(c1ccn(C)n1)C)N(C1(C#C)CC1)C1CC1 C1(CNC(c2cc(C)c(C(F)F)cn2)=O)CC2CCC(C1)N2C(=O)C=CC1CC1 C1(NC(CCCc2[nH]c(=N)sc2)=O)CC2CC(NC(=O)Cc3ccoc3)C1C2 n1(CC(=O)NCC2CCC(NC(C(C)CCO)=O)C2)c(=O)oc2ccccc12 Cc1cnc(C(=O)NCC2(C)CCN(C(c3cscc3C(F)F)=O)C2)cc1C#N Cc1oc([N+](=O)[O-])cc1C(=O)NCC1CC(O)(CNC(C2C3COCC23)=O)C1 c1(C(N(CCN(C(c2c(C)nsc2)=O)C)C(C)C)=O)n[nH]c(C2CC2)c1C N1(C(CC2CC(=O)OC2)=O)CC(C(=O)NCc2cn(C3CC3)nn2)C2(CC2)C1 C(CCC(C(=O)NC(c1ccccc1)C)NC(c1c[nH]nc1Cl)=O)OC C1(CCC(N2CC(CCNC(C=NOC)=O)C2)=O)CCC(=O)NC1 CCC(C)CCCC(=O)NC1(CCC(=O)NC2(CCCCO)CC2)CCC1 c1(-n2c(C=O)cnn2)c(Cl)cccc1Cl.C1(C(=O)OC)CN(CC)CC1C(C)C c1(C(N2CC(O)(CCNC(C3CC(C)OC3)=O)C2)=O)cccc2c1CCS2(=O)=O Cc1onc(Br)c1C(=O)NC(C)CCCNC(c1ccccc1F)=O c1(C(N2CC(OOCCC(C)C)C2)=O)ccc(OC(F)F)nc1.C1C(=O)NCC1 C1(CC#C)(C(=O)NC(CSC)CC)CCN(C(c2scnc2Cl)=O)C1 C1(CC(=O)N(C(c2ccc(Cl)c(Cl)c2)C)C)CC2CNCC2(c2ccccc2)C1 C1(C(N2C(c3nc(C)c(C)s3)CCC2)=O)COC2(CO)CC1C2 Cc1nc(C(N2CC(CNC(c3csc(CO)n3)=O)C(C)C2)=O)c2ccccn12 CCC(CC(C)CO)NC(=O)CCCCN(C(=O)CCC1(C)CC1)C Cc1ccc2c(c1)N(C(c1coc(CNC(=O)COCC3CCOC3)n1)=O)CC2 N1(C(c2ccc(C(CC)C)cc2)=O)CCCC2CN(C(=O)CCC(C)OC)CC12 C1C(CC)(CC)SCC(=O)N1.C(=O)(C(O)C(C)c1ccccc1)NS(NC)(=O)=O CS(=O)(=O)c1ccc(F)c(C(=O)NCc2cc3n(c2)CCNC3)c1 CC(C)(CC(=O)NCc1cccc(NC(=O)CCC2CCCC(O)C2)c1)C(F)F N(C(=NCCCF)NCc1ccoc1)CC(C1CCC1)OCC c1(C(=O)OCC)cccc(-n2cc(C3CCN(C(=O)C(C)=CCO)CC3)nn2)c1 N1(C(C(C)(C)OCC)=O)CCN(C(=O)C(=Cc2cccnc2)F)CC(C)(F)C1 C(=O)(C(C)(C)C(=O)NCCN(CCCN(C)C)C(c1ccccn1)=O)NC C=CCC(C)(O)C(=O)NCC(O)C(=O)Nc1cnc(F)nc1 N1(C(Cn2ccc(C)cc2=O)=O)CCC2C(NC(C3(C)CC=CC3)=O)C2CC1 S(=O)(=O)(c1cnc(NC2CC=CCC2)c(Cl)c1)N(C(c1c(OC)cccc1)C)C C1(C(=O)NCC(CNC(C2CCS2(=O)=O)=O)O)SC2C=CC1CC2 Cn1cnnc1S(=O)(=O)NC1CCCC(C(=O)NCCO)C1 c1(C(=O)NC(C)CF)cc(F)ncc1NC(c1ccc(C(F)(F)F)c(F)c1)=O CCC(CC)C(=O)N1CCN(C2CCC(NC(C3CC3C)=O)CC2)CC1 C1(CC)CCC(N(C)CC2CC3CCC2O3)CN1 N1(C(C2(c3c(C)c[nH]n3)CC2)=O)CC(CNC(C2C(F)(F)C23CC3)=O)C(O)C1 N1(C(C23CCC(OC)C2C3)=O)CCC2(C1)CN(C(=O)Cc1cc(F)ccc1Cl)C2 c1(C(=O)NC2(C(N(C)Cc3ncc(C)o3)=O)CCC2)cnccc1C C1(C(F)(F)F)(NC(C)=O)CCN(C(c2csc(I)c2)=O)CC1 C(=O)(CC(C)CC(C)C)N(CC(=O)NCCCCC#C)C1CC1 C(=O)(C#CC1(C)COC1)N1CCN(C(C2(CO)CCSCC2)=O)CC1CO.CCO Cc1cc(O)ccc1C(=O)NCCCCNC(=O)C(C)(C)C1CCCCO1 N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCC(C)(NC(c2ccc(C)cc2)=O)C1 CC1(C)CC(CNC(=O)Cc2ccc(O)nc2)N(C(C2COCCC2(F)F)=O)C1 c1(CCNC(COCCNC(=O)CCSC2CC2)=O)cccc(O)n1 C12(CCc3cc(Br)ccc3C1)N(C(=O)COC)C2.CCC(C)OC1CC1 c1(CC)ncc(Cl)c(C(=O)NC(C2CCN(C(c3sc(C)nc3C)=O)C2)(C)C)n1 c1(OC)ccc(C(C)(C)CN2CCCC(C)(CN(C)C)C2)cc1OC N1(C(C(CSC)(C)C)=O)CC2CCOC2(CNC(c2n[nH]c3c2CCCC3)=O)C1 C(=O)(C=CS(C)(=O)=O)NCC1N(C(CCC(=C)Cl)=O)CCC1C N1(C(c2n(CCC)ncc2)=O)CCC2(CCN(C(=O)C(C)NC(N)=O)C2)C1 C(=O)(CCCCCn1cc(C(C)(C)N(C)C)nn1)NCCc1ccn(C)n1 C1(COC(COc2cccc(C(C)=O)c2)=O)CCc2nc(C)[nH]c2C1 c1(C(C(=O)N(C)OC)C)ccccc1Cl.n1(CC)cc(C(CN)(OCC)O)nn1 C1(NC(CN(C(=O)CCc2cnn[nH]2)C2CCC2)=O)CCCSC1 c1(CC)ccnc(C(=O)NC2CCCC(C(=O)N(C)CCC3CC3)C2)c1 O=C(C#CC1CC1)NC(CNC(=O)Cc1ccccc1OC(F)F)C1CC1 c1(C(=O)NCC2(F)CN(C(C3C4CCC(=O)C34)=O)C2)ccc(C2CC2)cc1F O=C1CN(C(CCC2CCCO2)C(=O)NCC2CCOC2)CCCN1 CC(C)CC(F)(F)C(=O)NCC1(C)CCCN1C(=O)C(N1CCOCC1=O)C c1(NC(C2CCN(C(=O)OC)C2)=O)ccc(NC(=O)Cc2ccsc2)nc1 c1(C(=O)NC(C)CNC(=O)CNC(c2ccncc2)=O)[nH]cc2c1CCC2 C1(C(=O)OC)CCCN1S(=O)(=O)NCc1cc(OC)ccc1O CC1=C(C(=O)N(CCC(C(C)C)NC(=O)CCCc2ccc(C)s2)C)SCCO1 CC1Cc2ccccc2C1Nc1nccc(=NCC2(C)CCOC2)[nH]1 C1(C(N(CCCN(C(C(=Cc2cccs2)C)=O)C)C)=O)CC(C)(C)OC1(C)C c1(SC(CC)(C)C)nnc(CC)n1C1CCCC(C(F)(F)F)C1 c1(C(=O)NCCCNC(CC(C)C2CCCO2)=O)cc(Cl)c(F)cc1Cl c1(C(=O)NC2CCCN(C(COCCC(C)C)=O)C2)cc2cscc2s1 c1(COCC)nc(N2CCCCC(CNC(C3C(C)OC(C)C3C)=O)C2)cc(C)n1 C=C(Cl)C(C)(C)C(=O)N1CCOC(CNC(=O)Cn2cc(C3CCOC3)cn2)C1 N1(C(C(=O)NCC2CC2)=O)CCCC1CN(C(C1(Cl)CC1(F)F)=O)C1CC1 C1(NC(c2cncc(-n3c(C)c(C(=O)O)cn3)c2)=O)CCS(=O)(=O)C(C)C1 C1(NC(C2C(C)(C)C(=O)NC2)=O)CC2(CCN(C(c3cc(C4CC4)no3)=O)C2)C1 N#CC12CC(C(=O)NCCC3CN(C(C4CC5CC5C4)=O)CCO3)(C1)C2 c1(CCC(=O)NC2C(NC(C(CN(C)C)O)=O)C2)ccc2ccccc2n1 C1(NC(C(c2scc(C)n2)C)=O)CCOCC1NC(c1cn(C)nn1)=O Cc1ccc(C(=O)NCC=CCC(=O)NCC2CCC(C(N)=O)O2)c(C)n1 c1(CC)noc2ncc(C(N3CC(CNC(C4CCCC4C)=O)C(O)C3)=O)cc12 CC1C(NC(c2cccc(C(C)(C)C)c2)=O)CCN1C(=O)C(C#N)CC1CC1 CC(C)CC(C(=O)N(C)C)N(C(=O)CC1CCN(CC#N)C1)C Cc1ccc(C(=O)NC(CC2CC2)C(=O)NC2CC(CC(N)=O)C2)c(C)n1 N1(C(CCC(=C)C)=O)CC(NC(c2cnc(C)nc2C2CC2)=O)CCC(O)C1 c1(C(=O)NC(C(N2C(C)(CCC)CC2)=O)CO)ccncc1F C1(C(N(CCCNC(c2ccc(C(=O)CO)cc2)=O)C2CC2)=O)CCCS1(=O)=O C(=O)(CC(C1CC1)NC(C1COCCO1)=O)N(C1CCOC1=O)C N1(C(c2c(C)onc2)=O)CCC(O)(CCNC(=O)Cc2ccsc2Cl)CC1 CC1CC2(CC(C(N3CC(NC(=O)C(C)C4(O)CCC4)C(C(F)(F)F)C3)=O)C2)C1 CC1(C)CC(NC(C2CCC3CC2CO3)=O)CN1C(c1c[nH]c(=N)o1)=O C1(CNC(C(CCC)C#N)=O)CC2CCCC2N1C(=O)C(c1nc(C)cs1)C C=CCCC(F)(F)C(=O)N1CC(CNC(C2CCCCCC2)=O)C(F)(F)C1 N1(S(C(C)C)(=O)=O)CCC12CCN(C(=O)CSc1ccncc1)CC2 C1(NC(c2n(CCC)nc(C)c2)=O)CCC12CCN(C(=O)CC(CC)CC)CC2 c1(C(N(CC(C)(C)NC(c2c(C)cno2)=O)C)=O)cc2scnc2[nH]1 c1(N2CCC(NC(c3c(C)cncc3)=O)(CF)C2)nc2ccc(Br)cc2o1 C(=O)(C(C)(C)CO)NCCN(C(C)C)C(c1cnn(C(C)(C)C)c1)=O C12(CC(F)C1)C(=O)N2.CC(C(=O)NCCCCn1ccnc1)N1CCCC1 C1(NC(c2c(C(C)NC(=O)CCCCNC(N)=O)noc2)=O)C(=O)NCCC1C CC1CN(C(c2cc(C(F)F)ccn2)=O)CC1CNC(c1c[nH]nc1Cl)=O C1(C(=O)NC(C)CN(C)C(c2cc(C3CC3)nn2C)=O)CCn2c(O)nnc2C1 c1(COC)nc(N2CCC(C)(CO)C2)cc(NCCN(C)CCO)n1 N1(C(c2ccc(CC)s2)=O)CC(CC(=O)NCC(c2ccccc2)O)CC1(C)C N1(C(C(CO)NC(N)=O)=O)CC(NC(c2cc(Cl)cnn2)=O)CC12CCCC2 CC(CCC(C)(C)C)C(=O)NCCCN(C(=O)COc1ccc(F)c(Cl)c1)CCO C1(N(C(=O)COCc2ccnn2C)C)CC2CC1N(C(C1(C#N)CC1)=O)C2 N1(C(CC2(C)CC2)=O)CCN(C(=O)COc2ccc(F)cc2)CC(O)C1 C1(C(N2CC3CC3C2)=O)Cc2nccnc2CN1C(C1CC1(F)F)=O Cc1cc(C(=O)NC2CCCC2NC(=O)C2=CCCC2C)cc2nn[nH]c12 c1(C(=O)Nc2c(C)nc(NCc3cc(C)ncc3)s2)cc(C(C)C)ccc1C c1(C(=O)NC2CN(c3ncnc4c3CCC4)CC2F)c[nH]c2c(Br)cccc12 CC1(CNc2ncc(I)cn2)CCCN(C(c2nccnc2N)=O)C1 C(CC(=O)NCc1ncc(CO)[nH]1)(C(F)F)NC(C1CCC(C)(C)C1)=O C(C)(CC(=O)NCCOCCNC(=O)CCc1nccs1)(C(F)F)N(C)C C1(NC(c2cnc(C)s2)=O)CCN(C(=O)CSCC(F)F)C1C(C)C CCC1=NOC(CC(N2CCN(CCNC(N3CCCC(CC)C3)=O)CC2)=O)C1 c1(OCC)ccsc1C(=O)N(CC(CC)NC(c1cnc(O)o1)=O)CC C1(C(N2C(CNC(CC3COCC(C)(C)O3)=O)CCC2)=O)CCC2CCCCN12 C(C)(CCCC(=O)NC1CCCCC1C#N)NC(C1(C#C)CC1)=O n1(CC)cnc(C(=O)NC(C)C(C)NC(C2(c3ccsc3)CC2)=O)c1 C(C(CC(F)(F)F)C(=O)NCC1COCCOC1)NC(c1nccc(CC)c1)=O N1(C(C2CCN(OC)CC2)=O)CCCC2(CCCCC2NC(=O)C(C)N(C)C)C1 C(=O)(C1=CCCCC1C)N(CCNC(c1ccc(-n2ccccc2=O)cc1)=O)CC C1(OC)CN(C(=O)C(C)Oc2cccnc2)CC1NC(=O)CC(C1CC1)C1CC1 N1(C2C3C(CCCC2)C(=O)CN(CC#C)C3=O)CC(O)CC1C(N)=O N1(C(c2ccc(OC)cc2C)=O)CC2CCC(C1)N(C(c1cn(C)c(O)n1)=O)C2 C(CC(CC)C(=O)N1CC(NC(=O)CCc2c(C)noc2C)C(CO)C1)=CC N1(C(C)C)CCN(C(C2CCCCC2CNC(c2csc(Cl)c2)=O)=O)CC1=O CCCC(C(=O)NCCNC(=O)C(C)CC)NC(c1ccccc1C(C)(F)F)=O N1(CC(=O)NCCCN(C(=O)CC2CC(F)C2)C)CCCC1 N1(C(C23CC(CCC)(C2)C3)=O)C2CCC1CN(C(=O)C1=CC(O)CCC1)C2 C1(O)(CNC(C2C(NC(C3(OC)CC3)=O)C2)=O)CCCN(C(C)=O)CC1 C1(C)(C(N2CC(C(C(=O)NCC(COC)C)O)C2)=O)CC(F)C1 c1(-c2nc(-c3nc(SCC)c(-c4ccccc4)o3)on2)ccc(C=CCOC)cc1 CC(CC(=O)NC1CCCN(C(c2ccsc2C#N)=O)C1C)P(C)(C)=O C1(NC(c2cnc(C(F)(F)F)s2)=O)CN(CC=Cc2cn[nH]c2)CC2CC12 C1(C(=O)NC2(C)C(NC(Cc3c(C)nc[nH]3)=O)CCC2)CC2(C1)CC(O)C2 C1(C(N2CCCC(CCNC(C(CSC)(C)C)=O)C2)=O)CC(F)(F)CCC1(C)C c1(C(=O)NCCCN(C(Cc2ccc(C)o2)=O)C)cnc(O)c2ncccc12 N1(C(CC(=O)OCC)=O)CC(=O)CC1C(=O)NCc1cc(C(C)C)no1 Cn1ncc(C(=O)NC2CCCC(NC(c3csc(Br)c3)=O)C2)c1F c1(C(N2CC(CC=C)(NC(c3cncc(C)n3)=O)C2)=O)cn2c(n1)CC(C)CC2 C1(NC(C(C)(C)c2ccccc2)=O)(CO)CCN(C(c2ccccc2Cl)=O)C1 Cc1ccc(C(=O)NC2(CC(=O)N(C)CCOCc3cncn3C)CC2)c(F)c1 c1(C(N(C2CCN(c3ncns3)C2)C)=O)coc(Br)c1 C1(OC)COCCC1CC(N1CC(CNC(=O)CSSC)C1)=O C(=O)(C(F)C1=CCCCC1)NC1CCC(N(C(Cc2c(C)n(C)nc2)=O)C)CC1 N1(C(=O)NCC23CCC(F)(CC2)C3)CCc2ccc(F)cc2C1 C1(C)(C(=O)NC(C)CCCNC(c2ncn(C(C)(C)C)n2)=O)CCC(F)(F)CC1 C12(CNC(C3C(CNC(C4(C#N)CC=CC4)=O)CCO3)=O)CCCC1CCO2 c1(C(=O)NC(C(C)NC(CN(C(C(C)C)=O)C)=O)C)cnc(N2CCOCC2)nc1 C(CN=c1[nH]cc(C#N)cc1C)NC(c1c(F)cc(C)c(F)c1)=O C(C)(C)(CC(C)N1CCC(C(N2CCCC23CC3)=O)CC1)SC c1(C(c2nnnn2-c2ccccc2)NCC(=C)C)cnc2n1CCC2 N1(C(C(CC(=C)C)C)=O)CCC(F)(F)C(CNC(=O)CNC(C2CCC2)=O)C1 c1(C(N2CC(NC(=O)Cn3ccccc3=O)C(O)C2)=O)ccc(Cl)c(Cl)c1O N1(C(C23N(C(Cc4c(C)ccnc4)=O)CCC2C3)=O)CC2CC(O)CC2C1 N1(C(CC2(C)OCCO2)=O)C(C(=O)NCCN2CCNC2=O)CCC1C1CC1 C(=O)(C1=NN(C)C(=O)CC1)NC(COC)C(=O)NC1(CO)CC1.C(C)(=O)OC C12(NC(CCOC)=O)CCC(C1)N(C(c1ccc(Br)c(F)c1)=O)C2 C1(NC(COCC(C)(C)C)=O)CCN(C(=O)CNC(=O)NC2CC2)C2CC12 C(CCC1CCC1)(C(=O)Nc1cncc(F)c1)NC(C(C)=O)=O O=C1Nc2ccc(NC(C3CCCCCS3(=O)=O)=O)cc2C1=O C12(NC(C)=O)CCN(C(c3cn(-c4ccc(Cl)cc4C(F)(F)F)nn3)=O)CC1C2 Cc1nc(C(=O)N(CC(O)CNC(c2nc(Cl)c(Cl)s2)=O)C)ccc1[N+](=O)[O-] Cc1ccc(C(=O)NC(C(=O)NC2CCCCC2(C)C)C2CC2)cc1O C1(C(=O)NCc2scc(CNC(Cn3ncn(C)c3=O)=O)n2)CCC(C)(C)OC1 C1(CN(C(c2nc(CC)[nH]n2)C)C)CCCCN1C(c1csc(CC)n1)=O c1(CN(C2CCN(c3c(OC)cccc3)C2=O)CCN(C)C)nn(C)c(Cl)c1I C1(NC(C(C(C)O)NC(c2c(CC)ncnc2)=O)=O)CCCCC12CC2 C1(C(=O)NC(C)CNC(C2Cc3cscc3C2)=O)CC2(CO1)CC(F)(F)C2 C#Cc1ccc(C(N2CC(OC)CC2CNC(c2nn(C)cc2C)=O)=O)cc1C C1(C(=O)NC(CNC(c2cccc(C(C)=O)c2)=O)C(C)(C)C)CCCCC1(F)F N1(NC(C2C(C=CC)CN(C(=O)CC(=O)NC)C2)=O)CCCC12CCOC2 N1(C(c2nc(CCCC)sc2)=O)CCC(C)C(NC(=O)CO)C1 C(c1cccc([N+](=O)[O-])c1)=CC(=O)NCCN(C(C(C(COC)C)C)=O)C n1(COC)c(N2CCCC(C(N)=O)C2)nnc1Cc1ccc(C)cc1 Cc1[nH]c2ccccc2c1C(N1CCC1CNC(=O)CCc1cn[nH]c1)=O C(=O)(C(C(C)C)NC(N)=O)NCC1CC(NC(Cc2cc(OC)no2)=O)C1 N1(C(C2CN(C)C(=O)N2)=O)CC2CCN(C(c3cnn(C4CC4)c3)=O)CC2C1 c1(NC(CC2C3CN(C(CNC(N)=O)=O)CC32)=O)ccc2nncn2c1 CC1C(NC(c2ccc(C(N)=O)cc2)=O)CCCN1c1ncc(Cl)c(O)n1 c1(C(=O)NCC2CCC(NC(C(C)C3CC3)=O)CC2)n[nH]c2ccc(Cl)cc12 CCCCCCCCCCC(=O)N1CCCC(C)(C)C1CNC(=O)CC(=O)OC N1(C(CC2CCC(NC(C3CCCOCC3)=O)C2)=O)CCc2nn[nH]c2C1 C1(NC(C(C2CC2)OC)=O)CN(C(=O)C(C)(C)Cc2ccc(Cl)cc2)CC1CO Cc1nc(CC(=O)NC2(C)CC(NC(C3CCCN3C(C)C)=O)C2)cs1 N1(C(c2ccc(OC)c(F)c2)=O)CCCN(C(C2NC(=O)CC2C)=O)CCC1 CCC(CC)CCCC(=O)N1CCCCCC1C(=O)NC(Cc1cnc[nH]1)CO C1(CNC(CSC)=O)CC2CCC1N2C(=O)CN(C1CC1)CC c1(C(N2CCN(C(CC(C=C)C)=O)C(CF)C2)=O)sc2cc(C)cc(C)c2c1Cl C(=O)(C(C)(O)C(F)(F)F)N1CC(CNC(CN(C(C)C)C)=O)OCC1 c1(NC(C2C(CNC(C(COC(C)C)(C)C)=O)CCO2)=O)ccc2occc2c1 N1(C(CSCCN(C)C)=O)CCN(C(=O)C=Cc2cnccn2)C(C(C)(C)C)C1 c1(OCC(=O)NCC2C(NC(C3(C4CCCC4)CC3)=O)C2)ccc(F)cc1 C1(CNC(C(C)(C)CF)=O)CN(C(c2ccc(Br)c(N)c2)=O)CC12CC2 CC1(O)CCCN(C(C23CCN(C(=O)Cc4cccc(Br)c4)CC2C3)=O)CC1 C(=O)(CC(F)(F)C(F)(F)F)N1CCC(NC(c2ccc(C)nn2)=O)CC1C CC1CN(C(C2(NC(=O)Cc3ccc(F)cc3)CC(CO)C2)=O)C(C)C1C C1(NC(CC(C)(C)SC)=O)CC2CN(C(C34CCCN(CCC3)C4)=O)CC2C1 C1(n2cc(COC(=O)OC)nn2)CN(N2CCN(C3CCOCC3)CC2C)C1 C1(C(=O)NCC(CC)(CC)CO)CC12CCN(C(C1(Cl)CC1)=O)CC2 N1(C(C2CN(C(c3cc(I)ccc3Cl)=O)CCO2)=O)CCCC2(CCNC2=O)C1 C1(CC(=O)NC(C(C)NC(C(C)NC(=O)NC)=O)CO)CCN(C(C)=O)CC1 C(=O)(C(C)(C)C1=CCSCC1)N(CC(C)NC(c1cnc(OC)nc1)=O)CC N1(C(C(CC=C)CC=C)=O)CC2(C1)CN(C(C1CC1OCC)=O)CC2CO c1(C(=O)NCCCCNC(C2CC2c2ccco2)=O)cc2cccnc2[nH]1 C1(CCCC)CN(C(=O)C(C)n2ccnc2)CCN1C(=O)CSc1cn[nH]c1 C12(NC(c3occc3C3CC3)=O)CCCC1N(C(=O)CCNSC(F)F)CC2 C1(NC(c2c(C)nn[nH]2)=O)CCSC12CN(C(=O)C(C)C(F)F)C2 Cc1ccc(CNC(c2cscc2Cl)c2nnnn2CC(F)F)c(C)c1 C1(NC(c2c(C)con2)=O)CC(C)N(C(c2cccc(NC(C)(C)C)c2)=O)C1 C1(C(=O)NC(C(=O)NC)CC2CC2)CC(C)CN(C(c2ccc(O)nc2)=O)C1 CC1NC(=O)OC12CN(C(C1(CNC(c3csnn3)=O)CCCO1)=O)C2 c1(C(N2CCC(C(C(=O)NC(CC=C)C3CC3)(C)C)C2)=O)cccc2ccnn12 Cc1cn2cc(C(N3CC4(CCC4NC(c4cnccn4)=O)C3)=O)sc2n1 C1(C(NOCC(=O)OC)=O)N(C(=O)Cc2cccc(C)c2)CC12CCCC2 Cc1nn(C)c2c(NC3CCC(C)C3)nc(N(C)CC34CCCN3CCC4)nc12 c1(C(N2CCCCC(NC(C3CC3C(F)F)=O)C2)=O)cc2ccccc2nc1O c1(NC(C2CCCN(C(c3cc(Br)ncc3Cl)=O)C2)=O)cc2nccn2cn1 N1(C(C(CSC)C)=O)CC(N(C(=O)C2=CCCCO2)C)C(C)(C)C1 N1(C(COC)=O)CCC2CN(C(c3ncnc4sccc34)=O)C2C1 Cc1nc(C(N2CCCC2c2ccccc2)=O)sc1-c1ccccc1 Cc1coc(C(C)(C)C)c1C(N1CCCC(CNC(=O)Cc2n[nH]c(=N)s2)C1)=O Cc1cc(C(=O)NCCC2CCN(C(C3CCS(=O)(=O)N3)=O)C2)c(O)nn1 c1(C(c2ccnn2C2CCC2)N(CC(C)(C)N(C)C)CCO)nnnn1CC(F)F N1(C(CN(CCC)C)=O)CC2COCCC2(NC(c2cnc3cccnn23)=O)C1 C(=O)(C(CCN(C)C)NC(N)=O)NCCC1(NC(CCC=C(C)C)=O)CCC1 C(C(C)(O)CC(=O)N1CC(NC(c2cccnc2C)=O)C(n2cccn2)C1)OC Cc1nnc2n1CCC(CNC(N1CCC(OC(F)(F)F)CC1)=O)C2 Cc1cc(C(c2nnnn2C2(C)CC2)NCC2(CO)COC2)cc(C)n1 N1(C(C(C)OC(=O)OCC)=O)CC2CCCC(CNC(=O)C(C)S(N)(=O)=O)C2C1 c1(N2CCC(C)(NC(=O)C=Cc3ccc(Cl)s3)C2)ncnc2ccc(Cl)cc12 c1(CN(c2nnc(COC)s2)C)ccc(CNC(C2CC2C2CC2C)=O)cc1 CCC(O)C(C)C(=O)N1CCN(C(=O)CC(C)(C)N(C)C)C(COC)C1 CC1CN2CCN1C(C(=O)NC1CCC(CCNC(=O)Cc3cnc[nH]3)C1)C2 CCCC(CNC(c1ccn(CCC)n1)=O)C(=O)NCc1noc(C2CC2)n1 C12(NC(C3CN(C)C(=O)C3)=O)CCCC1N(C(=O)CCC1CCC(=O)N1)CCC2 C#CCCCCCC(=O)N1CC2CCC1C(NC(c1cn(C)nc1CC)=O)C2 CCCCCCCCC(C)C(=O)N1CC2COCC(C1)C2NC(=O)C1=NOCC1 C1(C(=O)NCC2CCN(C(c3c(C)n(C(C)C)nc3)=O)C2)Cc2ccccc2N1 C1(CCNC(C2CCN(C3CC3)C2=O)=O)CCN(C(=O)C=CCF)CC1 c1(C(C(=O)NCC(CC=C)NC(c2scnc2Cl)=O)(C)OC)cc(F)cc(F)c1 c1(C(=O)NCC2CN(C(c3c(C)con3)=O)CC2O)cccc2ncsc12 c1(CNC(C(CCC)N(C)C)=O)nnc2n1CC(C(F)(F)F)CC2 Cc1cc(C(=O)N(C(C)CNC(=O)CCCCCF)C)cc(C)c1 N1(C(c2ccnn2C2CC2)=O)CC2CCCC2(C(N2CCC23CCOCC3)=O)C1 C12(C(N3C4(CN(C(C(C(C)C)NC(N)=O)=O)C4)CC3)=O)CCC(C#N)(CC1)CC2 C(=O)(CC(O)C(C)(C)C)NCCCCCCN(C)C(c1cccc(C(N)=O)n1)=O c1(OC)ccc2ncc(C#N)c-2nc1C(=O)NC1CC(OC)(OC(C)=O)C1 N1(C(c2cnc(CC)s2)=O)CCC2C(NC(c3c(C)nn(C)c3F)=O)CC12 C1(CC(=O)NCC2CCCN(C(C3C=CC=CC=C3)=O)C2)COCCOC1 C1(CNC(C2CN(C)C(=O)N2)=O)C2CCC(C2)N1C(c1ccc(C(F)(F)F)s1)=O Cc1cccc(C(=O)NCC2CCC(C)CN2C(=O)CC23CCC(CC2)C3)c1O C(=O)(CC(C)(C)N(C)C(C1SCC=C1C)=O)N1CCC(C(=O)NC)C1 N1(C(C(C)OCC)=O)Cc2n[nH]cc2C1C(=O)N1CC(C)CCC1CC C1(CNC(c2c(N(C)C)cccn2)=O)CN(C(=O)CCC2OCCO2)CC(C)(C)C1 C=CCC(C(=O)NC1(CCOC)CCN(C(C2CN(CC)CCO2)=O)C1)N(C)C C(=O)(C(CCC(C)C)NC(=O)C(F)C(CC)CC)NCCCCCCC=C c1(CC(N2CCC(CCNC(C3(SCC)CC3)=O)C2)=O)ccccc1S(C)=O c1(CC)cc(CNC(c2conc2C(C)NC(=O)CC2CCCN2C)=O)no1 Cc1cc(Cl)cc(C)c1C(=O)NCC1CC(F)CN1C(C1COC(C)C1)=O c1(N2CC(O)(C(C)NC(c3cnc(C)s3)=O)C2)nc2cccc(Br)c2o1 c1(NC(C(C)NC(=O)CC2CCOC2=O)=O)cnccc1C1OCCO1 C#CCCCC(C(=O)NC1COC1)N(C1CCC1)C CS(C)(=O)=Nc1ccc(C(=O)NCC2OCCC2C(F)(F)F)s1 C1(c2n(CCCOC)nnn2)(NC(c2ccsc2)C)CCC(=O)N(C)C1 c1(N2CC(NS(C)(=O)=O)C2)ccc(S(=O)(=O)NCc2cnoc2)cc1Cl N1(C(CCOCCOCC)=O)CC(O)(C(C)NC(=O)C(N2CCSCC2)C)C1 C(CC1=CCN(C(=O)C(C)O)CC1)NC(c1cc(C)c(C(F)F)cc1)=O Cc1cnc(C(=O)NC2CN(Cc3ncccn3)CC2O)cc1Br C(=O)(CC(c1cccs1)N(C)C)N(CC(C)CNC(=O)Cn1ncnn1)C c1(C(=O)NC2CC3CN(C(c4nnn(CC)c4C)=O)CC32)snc2ccccc12 c1(C(C)(C)C)ncc(CN2CCC(C(O)C(F)(F)F)C2)s1 c1(C(=O)NCC2CN(C(Cc3cccc(C(N)=O)c3)=O)C2)cc(Cl)c(F)cc1Cl CCC(CC(=O)NCCCCCN1CCN(C(=O)CC(C)(O)C2CC2)CC1)OC C1(C(N2C(CN(C(C(CC)OC)=O)C)COCC2)=O)CCC=CCCC1 C1(C(N(C2(COC)CC2)C)=O)CCCC(NC(=O)C(c2ccccc2)O)C1 c1(CCC(=O)NC(C(C)NC(=O)CS(C)(=O)=O)C)cc2ccccc2o1 C(=O)(C(C(C)C)NC(=O)C(C)(C)C)NC(CNC(COC(C)=O)=O)C CCC(CC(=O)NC(CN(C)C)C(=O)N(C1CC2CCC1O2)C)C(F)F C12(NC(C(CC=CC)C)=O)CC3CCC(C1C2)N3C(c1cccc(C2CC2)c1)=O c1(CNC(C(N2C(=O)CCC2=O)CC)=O)cc2n(n1)CCN(C(=O)CCF)C2 C1(C(=O)NCC2(C(N)=O)CN(C(C(C)OCCCC)=O)C2)Cc2nnc(C)n2C1 c1(C(=O)NCC2CC3(CN(C(c4[nH]c(=N)sc4)=O)C3)C2)cnc2c(c1)CCCO2 C1(CCOC)(NC(=O)Cc2nc[nH]n2)CCN(C(=O)C(C(C)O)N(C)C)C1 C(N=C(NCC(C)(C)C)N1CCC(OC(F)F)C1)c1c(OC)cc(C#N)cc1 C#Cc1ccc(C(=O)NCC2CN(C(=O)C(CC)CC)C2)c(F)c1Cl c1(C(N2CC(NC(c3c(CC)n(C)nc3)=O)C(OC)C2)=O)nc(C)c(C)[nH]c1=O C(=O)(C(CCC(N)=O)N(C)C)NCCCCN(C(C(Cn1ccc(C)n1)C)=O)C CCCC(O)(CCC)CC(=O)NC(C)C(C)NC(c1cccc(O)c1Cl)=O Cc1cn2cc(CC(N3CC(CNC(=O)C=Cc4cnc[nH]4)CC3C)=O)nc2s1 c12cccc(c1)NC(=O)CC2.C1(CCC#C)CCCN1C(C)=O N1(C(C=C(C)C2CC2)=O)CCC2CCN(C(=O)CSCc3ccccc3Cl)CC12 C1(C(N(C2CCN(C(c3cnc(O)o3)=O)C2)CC)=O)CCCCC1(C)C c1(COC)ccc(C(=O)NC(CNC(=O)CCC2CC2(F)F)C(C)C)o1 Cc1cc(NC(CNC(c2cnoc2-c2ccco2)=O)C(C)(C)C)ncn1 O=C(CCCCCBr)NC1CCCN(C(=O)CCc2cccc(OC(F)F)c2)CC1 c1(C(C)(C)C)nccc(=NC(=O)C2CCC(CC(=O)Nc3n[nH]cc3I)CC2)[nH]1 Cc1ccc(SCC(N2CC(CNC(=O)Cn3ccnc3C)C(C)C2)=O)cc1 c1(C(=O)NC(CC)C(=O)N2CC(CC(C)NC(=O)C=CCF)C2)cccc(C)c1C C#Cc1ccc(OCC(=O)NC2CC(O)(CNC(c3cnoc3C)=O)C2)cc1 C1(N(c2cccc(C(=O)OC)c2)C(C(C)NS(CC)(=O)=O)=O)CCNCCC1C c1(C(=O)NC23CCN(C(C=COCC)=O)CC2C3)cnc2onc(C3CC3)c2c1 N1(C(c2n(CC)ccn2)=O)CC(NC(C2CN(CC3CCCCC3)C2)=O)C2CC12 c1(OCC(=O)N(CC(C)(C)NC(C2CCC2)=O)C)cc(Br)ccc1F C1(F)(N(CC(C)(C)C)C)CCC(=O)NC1=O C1(CNC(CC(CNC(CCOCCOCC)=O)OC)=O)CCC=CCCC1 CC(O)CCCC(=O)N(C(C)CCNC(=O)C(C)(C)Cc1cnn[nH]1)C C(=O)(C1=C(C)N2CCN=C2S1)OCC(CC)(CC)CC c1(CNC(c2n(CC)nnn2)c2ccsc2Br)cccc(CC(=O)OC)c1 C=CCC(CC(C)C)C(=O)NCCOC1CN(C(=O)CCC(C)CN(C)C)C1 CC(C)CCC(=O)C(=O)N1CCN(C(=O)Cc2ccc(C(F)F)cc2)CC1C N1(C(C(C)(C)SC)=O)CC2CC(C(=O)N(C)CCc3cccs3)C(C2)C1 c1(C(=O)NC2CC(C)(NC(c3n(CCC)ccc3)=O)C2)cnn(CCO)c1N C1(C(C(=O)C=CC2CCN(C(=O)CN3CC4CC4C3)CC2)=O)CC2(C1)CC(CO)C2 C1(N(C(CC=CC)=O)C)CN(C(C2CC2F)=O)CC1(C)C n1(CC)cc(CC(=O)NCCC2CCCN2C(c2cn(C(C)C)cn2)=O)cn1 C1(COC)CN(C(=O)COCCF)CCN1C(c1cn(C(C)C)cc1C)=O c1(CN2CCCC(C(N3CC(C)C(=O)CC3)=O)CC2)cc(F)c(Cl)c(Cl)c1 C(=O)(CCCCC#N)NCC(C)NC(=O)C=CC(c1cnn(C)c1)=O c1(CC(C(=O)NCCC2C(C)CN(C(c3ccco3)=O)C2)O)c(F)cccc1Cl N1(C(C2(C(C)(C)OC)CC2)=O)CCC(C(C)(C)NC(=O)CCCSC)C1 C(C(CO)(CO)NC(=O)CN(C1CCC1)C)N(C(=O)CCc1nc(O)n[nH]1)C CC1(C)CCN(CCNC(=O)C(c2cccnc2)NC(=O)C(F)=CC2CC2)C1 c1(C(N2C(CNC(C3CC4CCC3C4)=O)CCC2)=O)cc2n(n1)CCO2 CCC(C)(O)C(=O)N1CCC(NC(=O)C(CCSC2CCCC2)N(C)C)C1 C1(C(=O)NCCC(C)(C)NC(C(C)=C(C)C)=O)Cc2n[nH]cc2C(=O)N1 CC(O)CC(C)(C)CNC(=O)C(CCN(C)C)NC(c1ccc(O)c(F)c1)=O N1(C(CC(C(C)C)c2ccccc2)=O)CC2CCN(C(=O)C(C)(C)C#N)CC2C1 C1(C(=O)NC(CNC(c2cnc(CC)[nH]2)=O)(C)C)CCC(=O)N(CC)C1 C1(N(CCOC)C)CCCCC1CNC(C1C=CCN1C(=O)OC(C)(C)C)=O CC1CCCCC1(CNC(C1CCCN1C=O)=O)NC(=O)CC(C)n1ccnc1 Cc1cn2cc(C(=O)NC(C)C(C)(C)NC(c3ccc(C(C)C)o3)=O)ccc2n1 CCCC(C)(O)C(=O)NC1CC(C)CN(C(C2(CO)CC2)=O)C1 N1(C(CN(C(=O)OC)C)=O)CCCC2(CCCCC2NC(c2cc(C)cs2)=O)C1 C(=O)(CCC(=O)c1ccccn1)N(CCCNC(c1cc(C)sn1)=O)CC C1(NC(CC(=C=C)C)=O)CN(C(=O)C(C)OCC(C)C)CC12CCOCC2 C=CC1COCCN1C(=O)CC(C)NC(c1oc(C)nc1C)=O C1(C(=O)NCC2(F)CCN(C(=O)Cc3ccsn3)CC2)CC2C=CCC(C1)C2 c1(C(N2CCC(NC(C(N)=O)=O)C(CO)CC2)=O)ccc2c(c1)CCCS2(=O)=O CN1CCC(=CC(=O)NCC(F)CNC(=O)Cc2cnc(C(C)(C)C)[nH]2)CC1 c1(C(N2CC(NC(COC)=O)C2)=O)coc(CNC(=O)CC2CCOC2C)n1 N1(S(CC)(=O)=O)CCc2ccc(CNc3cccc(C(=O)N(C)C)n3)cc2C1 c1(C(=O)NCC2CCCN(C(C=CC)=O)C2)cccc2c1CCCC2=O N1(C(c2c(C(C)C)con2)=O)CCC2(CO)CN(C(c3cnc(S)[nH]3)=O)CC2C1 N1(C(C2CC(C)(C(=O)OC)C2)=O)CCCC(O)(CNC(c2ccccn2)=O)C1 N1(C(c2c(C)csn2)=O)CC(CC(=O)NCc2cnc(O)c(F)c2)CC1(C)C C12(CNC(COCC(C)C)=O)CCCC1N(C(c1ccc(C#N)cn1)=O)CCC2 N1(C(c2c(C)scn2)C(=O)NCCC2CC2)CCC2(CC1)COCC(=O)N2 Cc1ccc(O)c(C(=O)NC2(CNC(C34CCCC3C4)=O)CCOC2)n1 c1(NCCC2C(C)CCCN2C(=O)C2=CCCCO2)ncnc2cccnc12 C1(=CCNC(C2C(C)OCC2)=O)CCN(C(=O)C(F)(F)CO)CC1 N1(C(=O)NCC(c2ccncc2)(C)C)CCN(C2CC2)c2c(F)cccc21 C1(C(=O)NCCCc2n(C)ncc2)CC1C1CN(C(=O)CN2CC=CC2)C1 C12(NC(c3ccc(CC)[nH]3)=O)CCCC1N(C(c1snc(Cl)c1Cl)=O)CCC2 C1(C(=O)NC2CCC(NC(C3(CO)CCCCC3)=O)C2)CC12CCSCC2 C(=O)(C1=CNC2=NCCCN12)N1C(CCNC(C2CC(OC)C2)=O)CSCC1 C(=O)(C(O)CC(F)(F)F)N1CCC(OCCNC(C2(N(C)C)CCC2)=O)C1 C1(CNC(=O)CCCCO)CCN(C(C2CCCCC2O)=O)C12CC2 C1(CC)CN(C(=O)C(CCC2CCC2)NC(c2cc(C)nnc2O)=O)CCCO1 C=C(C)C(C)(O)C(=O)NCC(C)(C(C)C)NC(c1cc2sccc2s1)=O Cc1nc2ccnn2c(C)c1C(=O)NCC(C)(C)NC(=O)Cc1ccon1 c1(-n2ncc(NC(=O)NCCn3c(C)cc(C(F)(F)F)n3)c2)ncc(Cl)cc1Cl CN1N=C(CC(=O)NCc2cccc(CNc3ccnc4ncnn34)c2)CC1=O N1(C(CN(c2cnn(C)c2)OC(CCSCC)=O)=O)CCC(NC)CC1 c1(OC)ccc(Cl)cc1CC(=O)NCC(O)CN(C(=O)CC1COCCOC1)C C1(C(=O)NCCN(C(C)C)C)CCC(CNC(=O)CSC(F)(F)F)C1 C(=O)(C1=C2CCN=C2NC=C1)NC1CCC(NC(CN2CCC(=O)NC2=O)=O)C1 N1(C(c2cccc(C)n2)=O)CCN(C(c2ccn(CCF)n2)=O)CC1CO N1(C(C(COC)(F)F)=O)Cc2ccccc2C(NC(=O)CN(C)C)C1 C(=O)(C(F)CC(CC)CC)NCCC(C)(CC)NC(CC(CC=C)(C)C)=O Cc1nc(-c2ccccn2)sc1C(=O)NCC(O)CN(C)C(C1(C)CC1)=O C(c1cc(C)no1)=CC(=O)NC(C(=O)NCc1nc(COC)on1)C C=CC1(C(=O)NCC2=NOC(C)C2)CCN(C(C2CC23CCCC3)=O)C1 C1(C(=O)Nc2c(C(=O)OC)cc[nH]2)CCC(C)N(C(C2CC2C(F)F)=O)C1 C1(C(=O)NC2(CC)CN(C(=O)CC(C)OC)C2)CC12CCCC2 c1(CC)nn(C)c(CC)c1C(N1CCCC1CN(C)C(c1nc(=O)n(C)[nH]1)=O)=O c1(C(=O)NC(CC)CN(C(c2cn(C)c(O)n2)=O)CC)ncc([N+](=O)[O-])n1C N1(S(CC)(=O)=O)CCCN(C(=O)Cc2ccc(Br)cc2F)C(C)C1 C12=CC(=NC3CCN(CC3)C1)NC(CC)=N2.c1(C(=O)NC)cc(C)ccc1OC c1cnc2c(=NCCn3ccccc3=O)[nH]c(N3CC4COCC(C4)C3)nc2c1 S(=O)(=O)(c1c[nH]c(=NCCCS(=O)(=O)CC)cc1C)NCC(CC)N1CCCC1 N1(C(C2C(C)(CC)C2)=O)CC2(CCC(NC(c3nc(C)c(C)[nH]3)=O)CC2)C1 C(C)(CCC(=O)N1CCN(C2CN(C(=O)CCCOC(C)C)C2)CC1)OCC C(=O)(C(C)(C)O)N(C1CCN(C(c2cc(-c3ccccc3)cs2)=O)C1)CC c1(C(N2CC(C(=O)NCCNC(C(C)(C)C3CC3)=O)C2)=O)cc(S(N)(=O)=O)c[nH]1 N1(C(c2ncccc2F)C(=O)NCCSC)CCC2(CCCC2)C1 c1(C(=O)NC2CCC2NC(=O)C(F)(F)c2ncccn2)ccc2c[nH]nc2n1 C(=O)(CS(=O)(=O)CC)NC(C(=O)NCC(CCCC)O)Cn1cccn1 N1(C(C(C(C)O)C)=O)CCCC(C)(C)C1CNC(C1CC=CCO1)=O C1(CC(=O)NCC(CC)N(C(=O)CCC=CC(C)C)C)C=CCCC1 c1(CNC(CC=CC)=O)cccc2c1CN(C(C1(C)CCC3CC3C1)=O)C2 c1(C(N2CC(C(C)(C)O)(CNC(COC(C)C)=O)C2)=O)cccc2c1ccn2C N1(CCN(C(=O)Cc2cnn(C)c2C(F)F)C)CCN(C(C2(F)CC2)=O)CC1 c1(NC)ccc(C(=O)NCC2CC(F)CN2C(=O)CCCc2nc(C)no2)cc1 N1(C(C(COC(C)C)NC(C2C(OC)CC2)=O)=O)CCCC(NC(N)=O)C1 CC1(C)CCC(C(=O)NCC2(F)CCOCC2)CN1C(C12CCN(CC1)C2)=O c1(C(=O)NC(C(C)NC(Cc2cc(C)on2)=O)C)cccc2ncnn12 CC1CN(C(=O)C(O)CC2CCCC2)CCC1NC(C1CN(C(N)=O)C1)=O c1(CC)ncccc1C(=O)N(C)CC1(NC(=O)CNC=O)CC1 Cc1ccc(C)c(CN(C2(CO)CCCNC2)C)c1.C12(S(C)(=O)=O)CN(C1)C2 C1(C(=O)NCC(COC)(F)F)(CF)CCN(C(c2ccccc2CC#N)=O)C1 C(CC(C)C(=O)NCC(C)(C(C)C)NC(c1cc(C)c(C)[nH]1)=O)=CC N1(C(c2cnc(C)[nH]2)=O)CCCC(NC(C2CCC(N(C)C)CC2)=O)CC1 C(=O)(C1=CC2C=CC(C1)C2)NC1C(CNC(c2c(Cl)ccc(OC)n2)=O)CC1 c1(CC)nc(C(=O)NCCC2(C(=O)NC(C)CCCO)CCC2)cs1 Cn1c(C(=O)NC2CC(NC(c3cn(Cc4ccccc4)nn3)=O)C2)cnc1O CN1CC2CN(C(C3CCCCC3NC(C34C=CC(CC3)C4)=O)=O)CC2(C)C1 C(C(C(=O)N1CCC(O)(CO)C1)C(C)(C)C)NC(Cc1cc(C)no1)=O Cc1cc(C(=O)NC(C)CCCNC(=O)Cc2cnccc2Cl)n(C2CC2)n1 C1(N(C(Cc2cccc(OCC)c2)=O)C)CC2CC1N(C(=O)CC1OCCO1)C2 C1(CC(=O)NC(CC(=O)OCC)C)CC(C)N(C(c2nnn(C)c2C)=O)C1 c1(C(N2CCC3(CN(C(C(C=C)(C)CC)=O)C3)C2)=O)c(C)nn2cccnc12 CCC(CNC(c1nn(CC)nc1C)c1nnnn1C(C)C)(CC)C(F)(F)F C12(NC(c3ccc(F)cn3)=O)CCC(NC(C3CN4CCC3C4)=O)(CC1)C2 c1(C(N2C(C3CCN(C(CCC(=C)C)=O)C3)CCC2)=O)ccc2c(c1C)CCC2 c1(OC)cccc(C(N2CC3C(C2)C3(F)F)C(=O)NCC2CCCO2)c1C c1(CC)ccc(C(=O)NC23COC(CNC(C4CCOCC4)=O)(C2)C3)cc1Cl C1(C(=O)OC)CCC(NC(C2CN(Cc3cc(C)n(C)n3)C2)=O)CC1 C(CN=c1cc(C)nc(Cc2cccc(C)n2)[nH]1)SCC(=O)NC n1(CC(=O)NC(CC(C)NC(C(COC)CC(C)C)=O)C)cc([N+](=O)[O-])nc1C C1(C(N2C(C)CCCC2)=O)CCN(C(c2ccnnc2)=O)C(C)(C)C1 C1(OC)CN(C(=O)C(C)=CCO)CC1NC(c1[nH]c(O)nc1C)=O C12(NC(c3c(CC)ccc(C)c3)=O)CCCC1CN(C(=O)C=CSC)C2 C1(CN(CC(c2cc(F)ccc2F)=O)CC)CC2(CO1)CC(F)(F)C2 N1(C(CC2C(C)C(=O)CC2)=O)CCC(NC(=O)Cc2cc(C3CC3)on2)C1(C)C C1(CC(N2C(CN(C(C3(C)CC(=C)C3)=O)C)CCC2)=O)CCS(=O)(=O)C1 c1(OC)cccc(-c2nc(CC3CCSC3)n(C(C3CCC3)C)n2)n1 N1(C2CCN(C(C3CC34CCC4)=O)C2)CCN(CCC(N2CCCCC2)=O)CC1 c1(OC)nc(C)ncc1C(=O)NC1CCCCN(C(C2CCCC2C)=O)C1 CCCCC(CCCC)C(=O)NCCCC1(NC(=O)CC2(CC(=O)OC)CC2)CC1 CCS(=O)CC(=O)N1CCCCC1CNC(=O)Cc1coc(C)n1 C=CCCCCCCC(=O)N1CC(OC)C(NC(C2(O)CCCC(C)(C)C2)=O)C1 C(=O)(C(C)(C)C1=CCN(C(c2cccnn2)=O)C1)NC(CC(C)(C)C)CO C(CN=C(NCCN(C)C)NCC1(COCC(C)N(S(CC)(=O)=O)C)CC1)SC C1(NC(c2c(NC(C)=O)cccn2)=O)CN(C(c2n[nH]c(C)c2O)=O)CCC1C C=CC(C)(O)CC(=O)N1CCC(NC(=O)C(C)NC(=O)NC(C)C)CC1 Cn1ncc2cc(C(N3CCCC3CCNC(C34CCCN3CCC4)=O)=O)sc12 C1(C(=O)NC(C=C)C)CC2(CC(NC(c3ccc(Br)c(OC(C)C)c3)=O)C2)C1 CC(C)(Cc1cnn[nH]1)C(=O)NCC1CN(C(C2(C3CC3)CCCO2)=O)CCO1 C(CCN(C(=O)CCCN(C)C(C)C)C)(C(C)C)NC(c1nc(COC)sc1)=O c1(C(=O)NC2CCCC(CNC(C(C)SCC)=O)C2)ccc(C)nc1O c1(-c2cc(C)c(F)cc2)ccc2sc(C(=O)Nc3c(C#N)cnn3C)cc2c1 c1(NC(CCOCCNC)=O)cc(Cl)cc(Cl)c1F N1(C(CC(COC)COC)=O)C(C)CC2CN(C(c3cc(N)cc(F)c3)=O)CC12 C(=O)(CCCC(C)(F)F)NCC(C(C)C(C)C)NC(Cc1cccc(C)c1F)=O C1(CNC(c2cnc3n2CCC3)=O)CN(C(=O)C(F)CC2CCC2)C2(CCC2)C1 CCC(CC)(CCNC(=O)C(C)CC1CCCC1)NC(=O)C=CSC c1(OC(CC)C)cc(CN2CCC(C)(C(=O)NC3CC(F)(F)C3)C2)cc(Cl)c1 Cc1ccoc1C(=O)NC(CC1CC1)C(=O)NCC(O)Cn1cccn1 C(=O)(C(C)(C)C(=O)OC)NCC(CC=C)NC(=O)CCc1nc(C2CC2)no1 CC1CN2CCN1CC2C(N1CCC(NC(c2cc[nH]n2)=O)CC1)=O C(=O)(C1CCCc2nncn21)NC(C1(O)CN(C(c2ccc(C#C)cc2)=O)C1)C C1(CC(N2CC(NC(c3ccc(O)cc3F)=O)C(F)C2)=O)Cc2ccccc2C1 c1(C(=O)NCCCC(C)NC(c2c(NCC)scn2)=O)c(Cl)c([N+](=O)[O-])nn1C N1(CCc2c(OC)cccc2OC)C(=O)NC2(CCc3ccccc3C2)C1=O C1(CCCNC(C(CN(C)C)O)=O)CN(C(=O)CC2(C)CC2)CCO1 C(C)(C(C(=O)NC(c1ncc(C)s1)C)NC(C1COCCC1C)=O)OC N1(C(C#CCNC(C(C(=O)OC)(C)C)=O)=O)CC2COCC(C2)C1 Cc1cn2cc(C(=O)NC3CN(C(=O)CCC4CCC(C)O4)C3)cc(C)c2n1 c1(C(=O)NCC(CNC(C2(COC)CCC2)=O)OC)cccn(CC2CC2)c1=O CC(C(=O)N(CC(C)(C)NC(c1cnc(C2CC2)nc1O)=O)C)C(F)(F)C(F)F CN(C)NC(=O)CCC(=O)N1CC(CNC(C2(O)CC2)=O)N2CCC1C2 c1(C(N2CC(CCCCNC(C3N(CC)CCC3)=O)C2)=O)cc(C#N)n(C)n1 CC1(NC(C2OCCC2C(F)(F)F)=O)CCN(C(=O)C=CCN2CCOCC2)C1 c1(OC)cc(C(=O)NCC2CCCC2NC(=O)CC(O)CC2CC2)ncn1 C(=O)(C(=O)N=S(C)(C)=O)NC1C(C)CN(C(=O)CNc2ccccc2)C1 Cc1cccc2cc(C(=O)NC3(C)CN(C(=O)C=C4CCCC4)C3)cnc12 CC(F)(F)C(F)C(=O)NC1CCCC1CC(=O)NCCC(O)C1CCCC1 c1(CC(N2C3C(NC(=O)CC4CCCOC4)C(C3)C2)=O)ccc2cnccc2c1 c1(CN2C(CC)CN(C(c3ccon3)=O)CC2)ccc(C#N)cc1S(C)(=O)=O C1(N(C(=O)C=CC2CCOCC2)C)CN(C(=O)C(F)OC(F)(F)F)CC12CC2 Cc1ccc(CCC(=O)NC2CC(NC(=O)C(Cl)=CCl)C2)c(Br)c1 c1(NC(C2N(C(CC(C(C)C)O)=O)CCCC2)C)cccc(F)c1C#N c1(NCCC(=O)NCCC2CN(C(C(C)(C3(C)CC3)OC)=O)C2)ccccc1C C1(C(=O)NCC(CC=C)NC(c2cnnn2C)=O)CCN(S(N)(=O)=O)CC1 C(=O)(C#CC(C)(C)C)NCC1CCC(C(N(C)Cc2ccc(O)cc2)=O)O1 c1(CC(=O)NCC2CC(NC(c3ccc(C)cn3)=O)C(O)C2)ccc(F)cc1Cl C=CCCN=C(NCCC1CC2(CCC2)CO1)N1CCC(F)(C#N)C1 C(N=c1[nH]c(Cl)ncc1CC)C1N(C(c2n(C=C)ncc2)=O)CCCC1C c1(CC)ccc(C(N2CC(NC(c3ccc(C#N)[nH]3)=O)CCC2C)=O)c(C)n1 C(=O)(C(=O)N=S(C)(C)=O)NC1C(NC(C2(C)CN(C)C(=O)C2)=O)CC1 N1(C(C2CN(C(=O)C3CC3)CC2C2CC2)=O)CCc2c(O)noc2C1 N1(C(C2(c3ccc(C)nc3)CC2)=O)CCCC2(NC(=O)C#CC(C)C)CC2C1 c1(CC(=O)NC2C(C(N(CCCO)CC)=O)CCC2)cccnc1O C1(C2CCCN(C(=O)C(C)(C)n3ccnn3)C2)(NC(C2CC(C)C2)=O)CC1 N1(C(CCCN(C)C)=O)CC2CC2(CNC(=O)COCC2CCCO2)C1 CC(C)(CC1CC1)C(=O)N1CCCC1C(N1CC(O)(C(N)=O)C1)=O N1(C(=O)Cc2coc(C(F)F)n2)CCCC2C1CCN2C(=O)Cc1ccco1 N#Cc1cc(N2CCC3C(O)CC3C2)ccc1C(F)(F)F c1(CC(=O)NCCCCC(C)NC(C2(C)CC2)=O)cc(Br)ccc1F N1(C(C=CCCC)=O)CCC(NC(=O)CC2CCOC2(C)C)C12CC2 c1(CC(=O)NCC2C(NC(CC=C(C)C)=O)CCC2)cnc2ncccn12 C(C(C)C)(C(O)C(=O)N1CC=CC(C(=O)NCC2CC23CCC3)C1)OC C(N=c1[nH]c(C)cc(=NCC(C)(C)SCCO)[nH]1)c1ccn(CCC)n1 N1(C(C2(C(C)C)CCC2)=O)CCC(NC(=O)C(C)Oc2ccccn2)CC1 c1(CNC(C=C(C)C(C)C)=O)ccc(C(=O)N(C)C(C2CCCO2)C)cc1 C1(CNC(C2C(NC(C(C(C)C)OC)=O)C2(C)C)=O)CCCN(C)C1=O N1(CC)CCCC(NC(=O)CC(C2CC2)NC(c2ccoc2C)=O)C1 C1(NC(c2n(CC(=C)C)nnn2)c2ncc(CN(C)C)s2)CCCC=C1Br N1(C(CCCN(C(C)C)C)=O)CCC2(CC2C(N2CCC3C(C(N)=O)C3C2)=O)C1 N1(C(C2CCSC2)=O)CC=C(CCNC(C23CC4CC2C3C4)=O)CC1 c1(CN2CC3(CCN(C(C(C)(F)F)=O)C3)C2)cc(C(=O)O)cc([N+](=O)[O-])c1 CC(C)(C)C(CC(=O)NC1CN(C(=O)CCF)CC1(C)C)C(F)F C#CCC(C)(C(=O)NCCCOC1CC1)NC(=O)C1=CCCC1 C1(NC(C2C(C(C)C)C2)=O)CC2CCC(C1)N2C(=O)Cc1cnns1 N1(C(c2c(CC)ncs2)=O)Cc2occ(C(=O)NC3CCC(F)(F)C3)c2C1 N1(C(C2C(CCC)C2)=O)CCN(C(=O)Cc2coc(C)n2)C(c2ccncc2)C1 O=C(CCCC(=O)c1ccccc1)N1CC(CC(N2CCCCC2)=O)C1 c1(CN(C2N(C(C(C=C)(C)C)=O)CCCC2)C)cc(OC)c(OC)cc1F c1(C(=O)NC2CC(OCCN(C)C)C2)ncsc1S(N)(=O)=O.c12cn(nn1)C2 c1(OC)cccc(C(N2CCCC2CNS(=O)(=O)CCCCl)=O)c1Br C#CC1(C(=O)NCc2ccnn2C)CCN(C(=O)C(C)OC)C1 C1(C)(C(=O)OC)CCC1(C)C(=O)NCC(C)(C)CN(C(=O)C(F)C1CC1)C C(C1=CCN(C(c2cc([N+](=O)[O-])n[nH]2)=O)CC1)NC(C(n1ccc(C)n1)(C)C)=O N1(C(CN(C(COCC)=O)C)=O)CCCC(Cn2cc(CCCO)nn2)C1 Cc1nnccc1C(=O)NC(CCF)C(=O)NCC1CC1c1ccco1 c1(C(=O)OC(c2onc(C(C)C)n2)C)cc2c(Br)cccc2[nH]1 c1(C(N(CCNC(CSCC#C)=O)CC2CC2)=O)oc2ccccc2c1Cl c1(C(N2CCC(F)(CNC(C(COC)(C)O)=O)CC2)=O)cc(=O)n2nccc2[nH]1 c1(NC(C(N2CC(C(=O)OC)C(C(F)(F)F)C2)=O)=O)c(Br)nc2n1CCOC2 c1(C(=O)NC2CCC(NC(C(C)OCCC#C)=O)C2)cc(F)cc2c1CCC2 C1(NC(C(SC)SC)=O)CCN(C(=O)OC(C)(C)C)CC1O N1(C(C2(CC#C)CCC2)=O)CCCC(O)(CN(C)C(C2COC(=O)N2)=O)C1 Cc1ccn(CCC(=O)NC2CC(C(C)NC(=O)CCCn3cccn3)C2)n1 c1(CNC(C(CCOCCO)NC(=O)C#CC2CC2)=O)ncc(F)cc1F C1(CNC(CCCCNC(C)=O)=O)COC(C)(C)CN1C(=O)C(C)c1ccsc1 N1(C(CCCc2c(C)ccs2)=O)CC2(CCC2NC(=O)C(C)OCCN(C)C)C1 CCCC(C(=O)NCC(CO)NC(c1nn(CC)cc1Cl)=O)C(C)C c1(CC(C(=O)NC2CCN(C(C3C(C=C)C3)=O)CC2)C)ccc(F)c(F)c1 c1(CN2CCC(N(C)C(c3ccc4[nH]ccc4n3)=O)C2)ccc2ccn(C)c2c1 N1(C(Cc2c(C)nsc2)=O)CCCC(C)(NC(C2CC=CCO2)=O)C1 C(=O)(C(CO)NC(N)=O)N(C1CCN(C(c2csc(-c3ccoc3)n2)=O)C1)CC C1(NC(=O)CCC2CC2(F)F)CN(C(c2cccc(-n3cccc3)n2)=O)CC1O c1(CNC(=O)CC2CCCN2CCOC2CCCCC2)ccc(Cl)nn1 c1(C(=O)NCC2CC(NC(C3(C)CCNC3=O)=O)C2)cccc2cc(O)ccc12 C1(C(=O)NC2CC(NC(c3cc(F)cs3)=O)C2)CCc2ccnn2C1 C(CCCCC(=O)N(CC(C)(C)CNC(c1ccccc1N(C)C)=O)C)SC C1(NC(c2ncn(CC)c2)=O)CC(O)CN(C(c2cc(C3CCC3)[nH]n2)=O)C1 C1(C(=O)N(CC)CC)(NC(COC(CC)CC)=O)CC(F)C1 C(=O)(C1=CCCCO1)N1CC=CC(NC(C(C)(C)CF)=O)C1 C1(C(=O)NC2C(OC)CN(C(=O)CC3(C)CC3)C2)(OC)CCCCCC1 c1(OCC(N2CC(N(C)C(c3c[nH]nc3C3CC3)=O)C2)=O)ccc([N+](=O)[O-])cc1 c1(CC)c(C(=O)NC2(C)CCN(C(=O)CC(O)C3CCCC3)CC2)cccc1C Cc1ccc(C(=O)N(C)CCNC(=O)CN(S(C)(=O)=O)C)c2ccccc12 C1(CNC(=O)C=CBr)CCCCC1Nc1scc(C(=O)NOCC2CC2)n1 c1(OC)cccc(C(C)CC(=O)N2CC(NC(=O)C(C)C)C2)c1 n1(CC)nc(C(=O)NCC2COCCN(C(C3CCO3)=O)C2)c2c1CCOC2 C1(C(=O)NCC2CCCN(C(C(C)(C)OC)=O)CC2)Cc2ccccc2N1C C1(Cn2cc(CN(C)C(c3c(C4CCC4)cnn3C)=O)nn2)CC2CC(O)C2C1 CC1CCN(C(c2ncc(Cl)s2)=O)C1CNC(C1CC(O)C1)=O C(=O)(CCN=c1[nH]ccs1)N(C1CCN(C(c2csnc2C)=O)CC1)CCOC CC(C)C(CCNC(C1(NC(C)=O)CC1)=O)N(C(=O)C(C)(Cl)Cl)CCCl c1(C(=O)NC2(C)CC(NC(=O)C=C3CCSCC3)C2)cnc2sccn2c1=O c1(CC(C)C)ccc(C#N)c(N2CC3C(NC(=O)C(C)CC(N)=O)C3C2)n1 C1(C(=O)NCCC(C)NC(=O)CCCc2n[nH]c(=N)s2)CCC(=C2CCC2)CC1 c1(C(=O)NCCC2CCN(C(CCC(C)(C)F)=O)CC2)cc2ccccn2c1 CC(C(=O)NCCCN(C)C(C1CCSC1)=O)N(C)C(=O)OC(C)(C)C C1(NC(COCC)=O)CN(c2ccccc2)C(C)(CC)C1.C12CCC1CNC2=O C(N=c1[nH]c(N2CCC(c3cc[nH]n3)C2)nc2c1COCC2)c1nc(C)sn1 c1(SC)cc(Br)ccc1CNC1CC1C(=O)Nc1ccc(OC(F)F)cc1Cl CC(C)C(C)(O)C(=O)NCC(C)(C)OCCNC(c1ccc(SCCO)cc1)=O c1(C(N2CC(CNC(C3(CCCC)CCC3)=O)(OC)C2)=O)c(C)cc(C)nc1O CC(C)CC(C)CC(=O)N1CCCC(CN(C)C(c2cnc3[nH]cncc2-3)=O)C1 Cc1c(CC(=O)NCCC(C)NC(c2cnc(C#N)s2)=O)c(O)nc2[nH]nc(O)c12 c1(COC)ccc(C(=O)NCC(O)CCNC(=O)C(N2CCOC2=O)C)o1 O=C1CCN(C(=O)Cc2cscn2)C2CCN(C(c3ccc(Cl)o3)=O)CC2N1 c1(C(=O)NCCNC(c2cccc(C)c2F)=O)c(C2CC2)nc2sccn12 C(CC(=O)N1CC(NC(C2(C)CCCC2(F)F)=O)C1)(C1=CCCC1)OCC CC1=C(C(=O)N2CCC(NC(=O)C(C)C(=O)N3CCOCC3)C(F)C2)CCO1 N1(C(C(C)NC(C)=O)=O)CC2CCCC2(CNC(C2CC3(CCOCC3)C2)=O)C1 C1(CC(=O)NC(C(=O)NCCC=C=C)CC2CCCC2)CCCC12CC2 Cc1ccc(CC(N2CCOCC(CNC(c3cnccc3C)=O)C2)=O)cc1C C1(CCC)CN(C(C2CCN(C(c3cn(CC)cn3)=O)CC2)=O)CCO1 C1(CCNC)CCN(C(=O)C(COC)C2CCOCC2)CC1 C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCC2CN(C(CCCCCOC)=O)CC21 N1(C(C(C)(C)F)=O)CCC2(CC1)CC(NC(=O)Cc1csc(Br)c1)C2 CN1CCN(C(=O)C=C2CCCCC2)C(C(N2CCC=C(F)C2)=O)C1 Cc1c(C(N2CCC(C)(N3CCOCC3)C2)C(=O)NCC2CC2)cccc1Br c1(C(=O)NC2(C)CN(C(C(C)CC3CCCO3)=O)C2)cc2ccsc2c(O)n1 c1(NC(=O)Nc2cccc(CC)c2)cc(F)ccc1Oc1cncc(CO)c1 C1(N(C(CC2C(CC)C2)=O)C)CN(C(=O)CCC2CCC(=O)N2)CCC1C N1(C(c2scc(C(N)=O)c2)=O)CCC(NC(c2ccsn2)=O)C1c1ccccc1 N1(C(C(CC(C)(C)C)OC)=O)CC(NC(c2ncccn2)=O)CC12CCCCC2 Cc1ccc(OCCC(=O)NC2(CNC(c3cnc(C)cn3)=O)CCOC2)cc1 C1(NC(C2C(C(=O)OCC)C2)=O)CC(C)CN(C(c2cc(OC)n(C)n2)=O)C1 C1(C(N(CC)CC)=O)C2CCC(CC2(F)F)N1C(c1cccc2ncsc12)=O C(=O)(C(C(=O)N(CCCNC(c1ccc(C)nn1)=O)Cc1ccccc1)OC)OC C1(C(=O)NC2CCCC(CC(=O)N(CC(O)CF)CC)C2)CC2C(C1)C2(F)F c1(C(N(C2CN(C(=O)CSCc3ccc(F)cc3)C2)C)=O)cn(C)c(=O)nc1O Cc1cccc(C(=O)NCC2CC(O)CN2C(c2ccc(Br)c(O)n2)=O)c1C C1(c2cn(CCC(=O)OC)nn2)N(C(=O)CC2CC(=O)NC2=O)CC12CCC2 C(C(C)C(=O)NCCC12CC(CO1)C2)NC(C(C)N(C(C)=O)C)=O c1(C(=O)NCCCCCNC(C2C(SC)CCC2)=O)cc(C)nn1C(C)(C)C c1(OC)cc(Cl)c(Cl)cc1C(N1CC(NC(=O)C(O)Cn2cncn2)C(O)C1)=O Cc1nc(C(=O)NCc2cccc(C(N3CC(C)CC3CO)=O)n2)cc(O)n1 C(=O)(CN1C(=O)Cc2ccccc21)NC(CN(C(c1cnccc1Cl)=O)CC)C CC(C)(C)C(=O)C(=O)N1CC2(CC2)CC1CNC(C1CC(CC(F)F)C1)=O c1(C(N2CC(NC(=O)CC3COCC4(CCC4)O3)C2)=O)cc2cc(Cl)ccc2s1 c1(C(=O)NC2CC(CNC(=O)C(O)Cn3cncn3)C2)[nH]c2ccccc2c1Cl C1(NC(C2CCC(F)CC2)=O)CC1C1CCCN(C(=O)CCn2cnnn2)C1 C1(N=c2nc[nH]s2)(c2ccccc2)CCN(c2ncc3[nH]ncc3n2)CC1 N1(C(C23CCC(OC)C2C3)=O)CCC2CCCC12C(=O)NCCC(=O)N(C)C C1(CC)CC(O)CCN1C(=O)CC1CC(F)CN1C(c1ccc(OC)nn1)=O Nc1cc(C(=O)NC2CCCC(NC(=O)Cn3ncccc3=O)C2)c(F)cc1F C1(OC)CC(CC(=O)NCC2CC2NC(C2(CF)CC2)=O)C1 C1(O)(C(C(=O)NCC(CSC)OC)F)CN(C(=O)CCN(C)CCO)C1 c1(CC)[nH]nc(C(N2CC3C(C2)N3Cc2cccc(C(F)(F)F)c2)=O)c1F c1(CNC(C2CC3CC3N2C(c2coc(Cl)n2)=O)=O)ncccc1F C1(C(N2C(CNC(=O)CCCc3cccs3)CC(OC)C2)=O)CC(C(C)C)=NO1 CC(C)C(C(=O)NCC(C)N(C(=O)C(C)Sc1ccccc1)C)NC(N)=O Cc1c(C(c2nnnn2C2CCCC2)Nc2ccc(OCF)cc2)ccnc1F c1(OC)ccc(OCC(=O)NCCNC(=O)CCCCOC)cc1 CCCCC(CC)C(=O)NC(C1(CNC(=O)CCSc2ccccn2)CC1)C C1(C(N(C)CC2CCN(C(CSCC#C)=O)CC2)=O)CC2CCCC2C1 c1(CC(C(N2CCC(C(N)=O)(OCC)CC2)=O)N)ccc2c(c1)CCO2 CC(C)(C)CCCC(=O)O.C1(=O)C(SC)CCN1.S(C)(=O)(=O)C(F)(F)F C(=O)(CCCCN=c1cc[nH]cc1C#N)OC O=C(C1COc2ccccc21)NC1CCN(C(=O)CCCCCF)C12CCC2 C1(CNC(C(CCC)NC(C2CCCSC2C)=O)=O)CCCC12CCC2 CCC(CNC(=O)CC1CC(O)C1(C)C)(CC)NC(=O)C(C)Oc1ccccc1 N1(C(c2c(CC)non2)=O)C(CNC(c2cnn(C(C)C)c2)=O)CC2COCC12 N1(C(C(c2ccc(C)o2)C)=O)CCC2(CC1)CC2NC(C1CC(F)(CF)C1)=O Cc1cc(C)c(C2NC(=O)N(Cc3cccc(Br)n3)C2=O)c(C)c1 C=C(C)CN=C(NCC1CCCOC1)NCC(c1ccc(OC)cc1)OC c1(NC(C(=Cc2cscn2)C)=O)cccc(NC(=O)C=CBr)c1 c1(C(CC(=O)NC2CC(CSC)C2)NC(C#C)=O)ccc(F)cc1 N1(C(C2C(C)OCCC2)=O)CC=C(CCNC(c2cn(C)c(=O)nc2O)=O)CC1 C1(C(=O)NCC#C)CC2(CCN1C(=O)C(C)N1CC(C)C1)CC2 c1(C(=O)NCC2CCCN2C(C2CCCSC2)=O)cc2occc2s1 C(=O)(C1c2ccccc2CN1C(=O)CSc1nc[nH]n1)Nc1cnn(C)c1Cl c1(CC(=O)NCC2(NC(C=C(C)Cl)=O)CC2)cc(C)cc(C)c1 N1(C(=O)Nc2ccc(CC(=O)NCC)cc2)CCCC2(C1)NC(=O)N(C)C2=O N1(C(C)C)CCCC(C(=O)NCC2CCCCN2Cc2cnc[nH]2)C1 Cc1cccc(C(=O)NC2(CO)CCN(Cc3ccccc3)C2)c1CO C1(C(=O)NCCOC2CCN(C(c3cc(CC)nn3C)=O)C2)NC(=O)C2CCC12 Cc1[nH]c2ccc(NC(N3CCN(CCC(C)C)CC3)=O)cc2c1C C1(C(N2CCC(=CCNC(C3CC3F)=O)CC2)=O)CC2CCC(C1)C2F CN1CC(C(=O)NC2CCCC2NC(C2(c3ccnn3C)CC2)=O)NC1=O N1(C(=O)NC(CCNS(CC)(=O)=O)C)CCN(C(C)=O)C(c2cccc(Cl)c2)C1 Cc1ccc(C(N2CCC(CO)C(NC(=O)CC(C)(C)F)C2)=O)cc1[N+](=O)[O-] C1(NCCN2C(C)COCC2)CCCN1N1CCN(CCOC)CC1C N1(C(CN(C(C)=O)C)=O)CCN(C(=O)CC2CC3(CCC3)CO2)CC(C)C1 C1(C#N)(C(=O)NCC2(C)CCN(C(c3c[nH]nc3F)=O)C2)CC2(CCC2)C1 C1(O)(CC(C(=O)N(CC(C)CO)C)NC(C=C(CCC)C)=O)CCCCC1 c1(OC)ccc(C(C)C(=O)NCC2CN(C(C3(F)CC3C)=O)C2)cc1 C(=O)(CCCn1cccn1)NC(CC)CNC(=O)C(C)n1cncn1 C(CCN=C(NCc1ccccc1C(C)C)N(C)Cc1ncnn1C)SC C(CN=c1[nH]c2ccccc2s1)NC(N(CC(C)C)CC1CCCC(C)C1)=O N1(C(c2c(CC)ocn2)=O)CCN(C(=O)Cc2ncoc2C)C(C2CCCC2)C1 N1(C(c2ncc(C)c(C)c2)=O)CC2(C1)CN(C(C1CCC(F)C1)=O)CC2CO C(CC(F)F)(C(=O)N1CCC1C(N)=O)N(C(C=C1CCC(C)CC1)=O)C C1(C(N2CCC(O)(CNC(C(CC)N(C)C)=O)C2)=O)CC(C)(C)C(C)(C)C1 C(=O)(C(C)CCOC)N(CCC(=O)NC(c1nccn1C)C)CC=C c1(C(=O)NCCNC(C2N(C)C(=O)NC2)=O)cnc2ccc(F)cn12 c1(C(N2C(CNC(C(C)SC(C)C)=O)CC(O)C2)=O)csc2c1CCCC2 N1(C(c2n[nH]c(C)c2Cl)=O)CCC2CN(C(C3CCCN3N=O)=O)CC2C1 Cc1cc(=NCC2CCN(C(c3cc4c(s3)CCC4)=O)CC2C)[nH]c(C)n1 C(=O)(C1CCCn2ncnc21)Nc1c2cnn(C(C)(C)C)c2ncn1 c1(OCC)cc(Cl)n[nH]c1=NCCN1CCC(OC)CC1 c1(CCNC(C(C)N(C(=O)C(C)NC(C)(C)CC)CC)=O)nccc(C)n1 c1(SC)ncc(C)c(N2CCC(CC(=O)NCc3nc(C)no3)C2)n1 C#CCC(CC#C)C(=O)NC1(c2cccc(Cl)c2)CCC1 CCCCCC(O)C(C)C(=O)N1CCCC1C(C)NC(c1ccn(C(C)C)n1)=O N1(C(C(=O)NCCCF)CC2CCCC2)CCCCC1c1ncccn1 N1(C(C(CC)C)=O)CC(C2CCN(C(=O)Cc3ccc(CC(C)C)cc3)CC2)C1 N1(C(c2c(C)cc[nH]2)=O)CC(NC(=O)C(C)(C)c2cc[nH]n2)C(N=[N+]=[N-])C1 C12(CC)CC(C(=O)NCC3(NC(=O)C(C)CSC(F)(F)F)CCCC3)(CO1)C2 C1(NC(c2nc(C)oc2)=O)CC2CCC(C1)N2C(C1CCCC(C#N)C1)=O C1(C(N2CCC(N3CCN(C(C4(O)CC4)=O)CC3)C2)=O)CCCNS1(=O)=O CC(CC(=O)NC12CCC(CC1)CC2)C(C)(C)NC(c1cc2ccncc2[nH]1)=O N1(CCC)CCC=C(c2ccc3[nH]cc(CC(N4CCCCC4CO)=O)c3c2)C1 N1(C(c2cccc(C)c2Cl)=O)CC2=C(C1)CN(C(=O)CN1C(C)CCC1C)C2 S(=O)(=O)(c1csc2ccccc12)N1CCN(C(=O)Cc2ccc(O)cn2)C2C1C2 C1(NC(=O)NCCOCCNC(CSCC=C)=O)CN2CCCC1CC2 c1(CCC(=O)NCC2(NC(=O)C(O)CN3CCCC3)CCOCC2)cccc(Cl)c1 C(C)(C(=O)NCC1CCCCN1C(c1n[nH]c(C)c1C)=O)(C(C)C)NC(C)=O N1(C(C(CC)C)=O)CCN(c2cc(OCc3ccccc3)ncn2)CC1CC#N c1(C(=O)NCC(CNC(CSC)=O)F)cc(Cl)c(Cl)cc1C c1(C(=O)NCC(c2ccccc2)NC(C2CCC(=O)NC2)=O)ccc([N+](=O)[O-])[nH]1 C1(C(F)(F)F)(NC2CCC(CNC(=O)OC(C)(C)C)C2)CC=CCO1 CCCC(CNC(=O)C(O)CCN(C)C)C(=O)NCC1(F)CN(C)C1 C1(NC(C2C(=C)C2C(=O)OC)=O)C2CCC1CN(C(=O)C(C(C)C)OC)C2 c1(NC(=O)OC(C)(C)C)cc(=NC(=O)C(C)C(C)(C)c2ccc(Cl)cc2)[nH]n1C C1(C)(C(=O)NCC(CC(C)C)NC(=O)C(C)S(C)(=O)=O)CCCS1(=O)=O c1(NC(C2(F)CCN(Cc3ccc(COC)o3)C2)=O)nc2cc(Cl)ccc2s1 C(CS(=O)(=O)CC(=O)NC1CN(C(=O)CC2COCCOC2)CC12CC2)OC C1(CNC(C(=O)NCC)=O)N(C(c2cnn3c2CCC3)=O)CCCC1(C)C CC1CCN(C(=O)CCn2cccn2)CCN1C(=O)CCOCc1ccccc1 C1(O)(CCNC(c2ccc(CCC)[nH]2)=O)CCN(C(=O)CCc2ccsc2)CC1 c1(C(C(=O)N(CC(O)CNC(=O)CSCC2CCCO2)C)(F)F)ccc(F)cn1 C(CC(C)C)(C(=O)Nc1cn(C2CC2)nc1C)ONC(CN(CC)CC)=O n1(C(C)C)ccnc1CNC(=O)C(Cn1cccn1)NC(=O)C(F)C1CCCC1 C1(CCC)CN(C(=O)CNc2ccccn2)CCN1C(=O)CC1(CO)CCC1 N1(C(C(CC)(C)O)=O)CC(CNC(c2cc(Br)ccn2)=O)OC2(CCC2)C1 CN1CCCC(O)(CC(=O)NCC(C(C)(C)C)NC(c2ccncc2O)=O)C1 Cc1cnc(C(N2CC(NC(C3CCSC3)=O)C(O)C2)=O)cn1 CCC(C)(C)C(=O)C(=O)N1CC(C(O)C(=O)NCCOC2CC2)C1 C(=O)(CC(C)CC(=O)OC)NCC(CC)N(C(=O)Cn1nnc(C)n1)C C1(C(=O)N(CCO)CCO)C2CCCC1CN(S(=O)(=O)c1nccs1)C2 N1(C(CC(C)CF)=O)CCN(C(c2ccccc2CN(C)C)=O)CC1C1CCC1 Cc1ccc2[nH]c3c(c2c1)CC(NC(C1C(CN)C1(C)C)=O)CC3 N1(C(c2c(C)cno2)=O)CCC2(CC1)CC2NC(c1nc(Cl)c(Cl)s1)=O C(CC(C)(C)CC(=O)N1CCCC1c1cn(C2COC3(CCC3)C2O)nn1)OCC C1(C(=O)NC(CC)(C)CNC(=O)Cc2nc([N+](=O)[O-])n[nH]2)CCC2(CCCC2)C1 c1(C(=O)NCC(CNC(C2CCC(COC)C2)=O)(C)O)cccc2oc(=N)[nH]c12 c1(C(C)(C)C)cc(C(=O)NCCOC2CCN(C(C3(C#N)CCC3)=O)C2)on1 CCCCCCC(=O)NCCCN1CCC(C2OCCO2)C1 N1(C(Cn2nc(C)oc2=O)=O)CC2CC(NC(=O)Cn3nnc(C4CC4)n3)C2C1 C1(F)(CNC(CN(C)C(=O)C2CC2)=O)CCCN(C(C2CCCCC(=O)N2)=O)C1 c1(OC)cnnc(C(=O)NC2CC(CNC(=O)CCOc3ccc(C)cc3)C2)c1 N1(C(C=Cc2cn(C)nn2)=O)CCC2(CCC2NC(C2COCC2(C)C)=O)CC1 CCC(C)(C#N)C(=O)N1CC(N(C)C(c2cc(C3CC3)[nH]c2C2CC2)=O)C1 c1(N(C(C)=O)C)ccc(C(=O)OCC(N2C(C(C3CC3)CN)CCC2)=O)cc1 C1(C(=O)NCCCCNC(c2ccn(C)c(=O)c2)=O)CCCCC(F)(F)C1 C1(C(=O)NCC2C(CCC)CCC2)(C(=O)O)CCSCC1 CC(c1cccs1)=CC(=O)N(C1CCN(C(=O)C(=Cc2cccnc2)F)C1)C Cc1ccc(Br)c2nc(NC(C3CCN(c4ncccn4)CC3)=O)ncc12 N1(C(c2cnc(SC)nc2)=O)CC(NC(c2ncc(Br)cc2C)=O)C(C#N)C1 c1(C(N(C(c2ccccn2)C)C)=O)cc(F)cc(F)c1 c1(CCCC)cc(C(C(=O)NCC(=O)OCC)N(CC(C)(C)COC)C)n[nH]1 C1(NS(CCOC)(=O)=O)CCC12CCN(Cc1ccc(-c3cn[nH]c3)cc1)CC2 C(=O)(CC1=CCCCC1)NCC1(CNC(C2CCC(OC)CC2)=O)CC1 C1(OC)CC(NC(=O)CC(C)n2ccnc2)CN(C(=O)CC2CS(=O)(=O)C2)C1 c1(OCC(=O)NCC(N(C)C(C2CC3CC3C2)=O)C2CC2)ccc(F)cc1O N1(C(C=C(CC)CC)=O)CC2CC1C2NC(c1ccc(C2CCCCC2)o1)=O c1(-c2nc(C(C)C)nn2CCOCCc2ccccc2)cc2oc(Cl)cc2[nH]1 C12(CNC(C(COC)(C)C)=O)CN(C(=O)Cc3nn(C)cc3Cl)CC1CCO2 C1(C#N)(C(N(CCC)CCNC(=O)Cc2csnc2C)=O)CCOCC1 CCC(C)(CNC(C1(CCF)CC1)=O)NC(=O)C=CBr c1(CC(=O)N(C(CNC(CCC(=O)NCCC)=O)C)C)ccc(OCC)c(F)c1 CC(C)CC(C)(C)C(=O)NC1CCC(NC(C23CCCC(CO2)C3)=O)CC1 CN1CC(NC(=O)C(C2CCN(C(=O)CC3CCSC3)C2)F)C2(CC2)C1=O N1(C(C=C(CC)C)=O)CC2ON=C(CNC(c3ccc4n[nH]cc4c3)=O)C2C1 c1(-c2c(OC)snn2)nc(C(C)(C)C)nn1Cc1ccc(Br)cc1 N1(C(C)C)CCC(C(=O)N(C2CCC(NC(c3cnn(C4CC4)c3)=O)C2)C)CC1 CCCCCC(O)C(=O)N(C1CCCC1)CCCNC(=O)CCCC(C)=O N1(C(c2cncc(C)c2Cl)=O)CCN(C(c2nonc2N)=O)C(C)CC1C c1(C2(C(=O)NCCCCCN(C(CC3C(CC)C3)=O)C)CC2)cccc(C)c1 C(CC(C(=O)N1CCC(SC)C1)NC(=O)CCc1cnccn1)OC C(=O)(C(CC(C)CC)NC(=O)Cc1cccc(F)c1)NC1C(C#C)CCC1 C1(C(=O)NC(CNC(c2cnc(CCCC)s2)=O)CO)CCc2nccn2C1 c1(CNC(C(CCOCC)NC(=O)CCc2ccccn2)=O)cc(C)cc(F)c1 CCC1CCCc2sc(N(C(c3ccccc3)=O)Cc3ccccc3OC)nc21 C1(C(=O)NCCCNC(c2cnn[nH]2)=O)(CO)CC12CCC2 C1(C(N(CC(CC)NC(C(C)=CC)=O)C)=O)CCCCN1S(=O)(=O)CCCC C(=O)(CCCC(C)(C)C)NCCC(CC)(CC)NC(=O)Cn1ccc(Br)n1 C(=O)(CC(CNC(c1cc(C)sc1C)=O)C1CCC1)N(C(C(CC)C)C)C1CC1 c1(NC(N2C(CCNC(=O)OC(C)(C)C)CCC2)=O)cc(O)c2ccoc2c1 N1(C(Cc2cc(C)on2)=O)CC2CCC1CN2C(c1coc(C(F)F)n1)=O c1(C(N2CC(C)C(NC(C3(F)CCCC3)=O)C2)=O)[nH]cc2c1CCS2(=O)=O c1(Cc2nc(C3Cn4c(nc(C)n4)C3)on2)ccc2c(O)n[nH]c2c1 C1(OC)CC(C(=O)N(CC(N2CCCC2)C)C)N(C(=O)CCc2ccn(C)c2)C1 Cc1cc(C)c2c(N)c(C(=O)Nc3cc(O)nc(C)n3)sc2n1 N1(C(CCC(=C)C)=O)CC2CC1CC2NC(c1ccc2c(c1)CC2)=O N1(C(C=CC)=O)Cc2ccccc2CC1CNC(C1OCCC1C(F)(F)F)=O N1(C(C2CCC(C#C)CC2)=O)CCC2CCN(C(C3CCCCC3OC)=O)C2C1 C#CCCCC(C)C(=O)N1CCCC1C(=O)NCC1CC2CCC2C1 C=CCC(CC)C(=O)N1CCC(C(N2CC=CC2(C)CO)=O)C1 c1(C(=O)NCCC2CCC(NC(c3ccc(OC)cc3)=O)C2)ncnc(O)c1F CCC(C)CC(CO)NC(=O)C=CC1CCCC1.C1(=O)CC=CCN1 C1(C(=O)NC(CN(C(=O)C(O)Cc2cn(C)cn2)C)(C)C)CCS(=O)(=O)C1(C)C Cc1c(C(N2CCN(C(c3cc4n(c3)CCC4)=O)CC2)=O)cncc1Br c1(COC)nc(NCc2ccc3nsnc3c2)cc(=NC(C)Cn2cncn2)[nH]1 Cc1c(Cl)sc(Cl)c1C(=O)NC(C)CN(C)C(C1CC1c1nccn1C)=O CCN=c1[nH]cc(C(N2CC(NC(C3(C)CCCO3)=O)CC2C)=O)s1 C12(CNC(=O)C(F)CC3CCC3)CCC(NC(c3cc(Cl)cnc3O)=O)(CO1)C2 c1(C(=O)NCCC2(CNC(c3nc(OCC)oc3)=O)CC2)ccc([N+](=O)[O-])s1 C(C(CNC(C1CC12CCCCC2)=O)S(C)(=O)=O)NC(C(C(C)C)F)=O CCC(CC)(CCNC(c1nc(C)ccc1F)=O)NC(=O)CC1(OC)CCCC1 C1(CNC(C2CCC(C)O2)=O)C(C2CC2)CCN1C(C1CCCCC1O)=O C1(C(=O)NCc2ccn(C)n2)CN(Cc2ccc(Cl)cc2O)CC(F)(F)C1 C1(NS(CC(OC)OC)(=O)=O)CC2(CO1)CN(C(=O)OC(C)(C)C)C2 CC(C)CCC(=O)C(=O)NCC(C)(C1CC1)NC(=O)CC1CN(C)C1 c1(CNC(C(C)N2CCCC2)=O)cc(C(=O)NC2(CC3CCC3)CC2)no1 C(=O)(CCCc1ncco1)NCCOCCNC(C(SC)SC)=O C1(CC)CCC(C(N2CC(O)(C3CCCN3C(=O)CNC(=O)C3CC3)C2)=O)CC1 c1(C(=O)NCC(CC=C)NC(C2(C)CC2)=O)ccc2c(c1)nc(C)c(=O)n2C N1(C(C(C)SCC)=O)CCN(C(=O)CCC2CC2(Cl)Cl)CC(O)C1 N1(C(C(CSC)OC)=O)CCN(C(C2(OC)CCC(C)(C)C2)=O)CC12CCC2 c1(OC)c(CC(=O)NCC2C3CCC(C3)N2C(=O)C(O)C2CCC2)cccc1F c1(N(C)C2CC2)[nH]c(=NCC(F)(F)c2ccc(F)cc2)nc2scnc12 c1(CN2C(C(=O)Nc3c(CO)ccc(OC)c3)C=CC2)ccc(Cl)c([N+](=O)[O-])c1 C12(C(=O)NC(CNC(CCOCC#C)=O)(CC)CC)CC(CO)(C1)OC2C C1(COC)CC(N=c2[nH]c(=NCCCc3cnn[nH]3)c3cccc(F)c3[nH]2)C1 c1(CC)c(C(=O)N(CCCCN(C(=O)C(N2C(C)CCC2C)C)C)C)ccn1C N1(Cc2[nH]cc(C#N)c2)CC2CC(C(=O)NC3CN(CC(F)(F)F)C3)CC2C1 C1(NC(CCc2c(C)nn(C)c2)=O)CN(C(c2cccn2C)=O)CCC1CO Cc1nc(Cl)cc(Cl)c1C(=O)NC1CCCN(C(=O)CC2NC(=O)NC2=O)C1 c1(OC)ccc(Cl)c(C)c1C(=O)NCCCCN(C(=O)C1=CCCCC1)C c1(C(N2C(C3(C(=O)OC)CC3)CCC2)=O)ccc(C#N)[nH]1.C12(CC1)C(=O)NC2 c1(SC(C)Cc2ccc(Cl)s2)cccc(-c2noc(-c3ccoc3)n2)c1 C(=O)(CCCCC(N)=O)NCC1CC(NC(C2CCCN(C(C(C)C)=O)C2)=O)C1 c1(C(CNC(C2(N(C(COCC#C)=O)C)CC2)=O)O)ccco1 C1(C(N(CC(CC)O)Cc2ccco2)=O)CCCN(Cc2nccn2C)CC1 c1(C(=O)NC2CCC(N(C(CCN(CC)CC)=O)C)C2)c(C)oc(C)c1Br C12(NC(C=C(C)C(C)C)=O)CCC1CN(C(=O)Cn1ncc(Cl)c1C)C2 C1(NC(=O)NCC(c2ccccn2)C)CCN(C)CC1c1cnn(C)c1 N1(C(CC=CC)=O)CCC2CCN(C(c3ccc(Br)cc3F)=O)C2C1 N1(C(CC(=O)OC)=O)CC2CC2(CNC(=O)CC(C)=C(C)C)C1 N1(C(c2cnc(C)s2)=O)CC(CNC(=O)CC(C)c2ccco2)CC1(C)C c1(CC(N2CC3C(NC(c4c(CC)ccs4)=O)(C3)C2)=O)ccc2ccccc2c1 c1(OC)ccc2oc(C(N3CC(NC(=O)C(CCSC)N(C)C)C3)=O)c(C)c2c1 N1(C(c2cnn(CC(F)(F)F)c2C)C(=O)NCCOC)CCC2CCC(C2)C1 C1(CCC#C)CCCN(C(C2(CNC(c3oc(CO)cc3C)=O)CC(=C)C2)=O)C1 Cc1cnn(C)c1C(=O)NCC(C)(C1CCC1)NC(=O)CCC(=O)c1cccs1 C12(C(N3CC(C)C(NC(c4n[nH]cc4[N+](=O)[O-])=O)CC3)=O)CCC(F)(CC1)CC2 S(=O)(=O)(C(C(C)C)c1ccccc1)NCCCCC(=O)OCC C12(NC(C3C(CCC)CCC3)=O)CCC(NC(=O)CCOC3CCCC3)(CC1)C2 C(=O)(C1=NNC(=O)C1)NCc1cccc(CN(C(C2C(OC)CCC2)=O)C)c1 C1(CC)(CC)CC(NC(c2cccc(O)n2)=O)CN1C(c1cnc[nH]1)=O C1(NC(CN(C)C(N)=O)=O)CC(C2CCN(C(c3ccc(N)c(F)c3)=O)C2)C1 C1(C(C)NC(C(C)COc2ccccc2)=O)CCN(C(=O)C=C2CCC2)CC1 C(C(C)C)(C(O)C(=O)NCC(C)CC(=O)NCC(CO)C1CC1)OC c1(C(=O)NC(C(=O)OCC)(C)C)cnc(CNC(C2CNC(=O)O2)=O)nc1 c1(C(N(CCN(C(=O)Cc2cscn2)CC)CC)=O)ccc2cnn(C)c2c1 C#Cc1ccc(F)cc1C(=O)N(C1CCN(C(c2cscc2SC)=O)C1)C O=C(CC(C(F)(F)F)NC(C12C=CC(CC1)C2)=O)NC1CC(O)CC1O c1(C(=O)NCCCNc2ccc(F)cc2F)ccc2ncsc2c1 C1(COCCNC(C2(C#C)CC2)=O)CCN(C(=O)C(C)NC(C2CCCC2)=O)C1 N1(C(c2cncn(C)c2=O)=O)CC2CN(C(c3ccnc(O)c3)=O)CCC12 Cc1cc(C(N2CC(O)(CN(C)C(c3c(O)cccc3F)=O)C2)=O)ncc1CO C=CCC(C)(CC)C(=O)N1CC2(CC(CC#N)C2)C1 Cn1ncc(CCC(=O)NCCC2CCN(C(C3(O)CCC3)=O)C2)n1 c1(CCNC(c2cncc(C(C)(F)F)c2)=O)noc2cc(F)ccc12 c1(C(=O)NC(CC)CNC(c2ccn(C)c2)=O)ccccc1OCC(N)=O C12(C(N3C(C)CN(C(c4nncs4)=O)CC3)=O)CCCCC1OCC2 C(=O)(C1=Cc2ccccc2OC1)N1CC(C(C)Nc2c(C)c(Cl)ncn2)OCC1 CCCCCCCCNC(C12CC(NC(=O)CC3CCCO3)(C1)C2)=O C1(NC(C(CC)CO)=O)CC2(CCCN(C(c3cc(C)n(C(C)C4CC4)n3)=O)C2)C1 N1(C(CCC#C)=O)CC(F)(F)CC1(C)CNC(=O)CC(C)P(C)(C)=O c1(CSCC(C)C)ccc(C(=O)NC2CCCC2NC(c2cnsn2)=O)o1 CC(CCCCCO)NC(C1CCCCC1CNC(=O)CC1OCCC1(C)C)=O C1(C(=O)NCCN(CCCCCC)C(c2cnns2)=O)CCCC(C(N)=O)C1 C1(C(=O)NCCSCC(=O)NC(C2CC2C(C)(F)F)=O)(CC)CCCCO1 N1(C(CC2N(C(c3c(C)ocn3)=O)CCC2(C)C)=O)CCc2n[nH]cc2C1 N1(C(c2ccn(C(CC)CC)n2)=O)CC2CCC(NC(=O)C=C(C)C)(C2)C1 c1(C(=O)NC2CC(C)(CNC(C(C)n3ccnc3)=O)C2)ccnc(N2CCCC2)c1 CC1CCCN(C(c2cnn(CCO)c2)=O)C1CNC(=O)CN1CCC(O)CC1 C(C(C)(C(=O)NCCCC(=O)NCCC1(O)CCOC1)OC)OC C1(CN(C(C2(Cc3ccccc3)CC2)=O)CC)CCN(C(C2CC2F)=O)CC1 C12(NC(CCCCSC)=O)CCCCCC1N(C(=O)CCc1cn(C)nn1)CC2 c1(CC)c(C(=O)N(c2ccc(N3CCCCC3)nc2)C(C)=O)[nH]c(C)c1C(C)=O Cc1cc(C(N2CCC(F)(C(=O)NCc3c(F)cccc3F)C2)=O)cc(C)c1O c1(C(CNC(C(C2CCN(Cc3ncnn3C)CC2)C)=O)O)cccc(Br)c1 C(=O)(CS(=O)(=O)CC)N(CCNC(c1nc(COCC)sc1)=O)C1CC1 c1(C(=O)NC2CC3(CN(C(C4CN(CC(C)C)C4)=O)C3)C2)ccc(N)c(Cl)c1O Cc1nc(O)nc(O)c1CC(=O)NC1CC(F)(F)CC1NC(C1CC=CCC1)=O CC(C)CSCC(=O)N(CCCN(C(=O)CO)C(C)C)C C1(C(=O)NCC(CC)(C)Cl)CN(C(c2cc(C#N)cs2)=O)CCN1C C1(C(=O)O)CC(C(F)(F)C(F)(F)F)CN(C(=O)CCC2CCCOC2)C1 C1(NC(C(C)NC(C)(C)C)=O)CN(C(C2CC3C=CC2CC3)=O)CCC1C C(=O)(C(CNC(c1nc(O)sc1C)=O)CC1CCCC1)NC(c1nc(C)[nH]n1)C C1(C(N(C2CCCOC2)CC)=O)CC2CCC1N2C(C1C2CC(=O)CC12)=O O=C1CCN(C(c2ccn(-c3ccccc3)n2)=O)C(C(=O)O)C1 C1(NC(c2c(C)cc(F)s2)=O)CCC2(CCN(C(C3(N=[N+]=[N-])CC3)=O)CC2)C1 C1(NC(C(F)=CC)=O)CC12CC(NC(c1cnn(-c3cccc(O)c3)c1)=O)C2 Cc1ccc(C=CC(=O)NCc2cc(C(=O)NCC(O)(CO)CO)no2)cc1 C(CNC(=O)CCc1cn[nH]c1)(C(=O)NC(C)(CO)C1CCC1)N(C)C C1(CNC(C(C2CC2)OC)=O)CN(C(c2cccc(F)c2)=O)CC1C(F)(F)F N1(C(C(C)OCCOC)=O)CCC(C)CC1CNC(=O)C(C(C)C)NS(C)(=O)=O c1(OCC(=O)NCC(CO)NC(C2CCCC(C(=O)OC)C2)=O)cc(F)cc(F)c1 C1(C(C)C)CCCC1C(N1CCCC1CNC(=O)CCc1ccccn1)=O C1(C(=O)NC(C)(CC)CC)(CC)CCN(C(c2nccn2C)=O)C1 C1(C(=O)NCCc2c(CNC(C(CC)F)=O)nco2)CC12CCCCCC2 C1(NC(C2(CC#C)CCCC2)=O)CCN(C(c2cnc[nH]2)=O)CC1(C)C C=CCC(CC=C)C(=O)N1CCC1(C)CC(=O)NC(c1ncc(C)[nH]1)CC c1(C(N2CC(CNC(c3cc(OC)ncn3)=O)C2)=O)cc(F)cc(F)c1O C(c1ccncc1)=CC(=O)NC1(C(=O)NC(c2nc(C)[nH]n2)C)CSC1 S(=O)(=O)(C=Cc1ccccc1)N1CCN(CC(C)(C)NC)CC1 C1(C(=O)NC2(CCCC)CC2)COCCC1NC(c1occc1COC)=O c1(C(N2CCN(C)C(CNC(C3CCC(C)(C)C3)=O)C2)=O)ccc2cc[nH]c2c1 c1(C(=O)NC(C(C)NC(COc2cccc(C#C)c2)=O)C)ccc(C)c(F)c1F c1(C(=O)NC2C(CNC(C=C(CCN(C)C)Cl)=O)CCC2)ccc2c(c1)CC2 CC1CN(C(=O)CN(C)CCO)CC(C)N(C(=O)CC2CCOC2)C1 c1(C(N2CC(CNC(CCC3CC(OC)C3)=O)C2)=O)nn(C)c2ccc(F)cc12 CC(CCNC(C1CCCCN(C(=O)Cc2cnns2)C1)=O)C(C)(C)C N1(C(=O)CC2CC2)CC2CC(C1)CN(C(C1CCC=CCCC1)=O)C2 N1(C(c2c(CNC(=O)C=Cc3cncs3)ocn2)=O)CCC(O)CC1C1CC1 N1(C(c2cn(CC=C)nc2)=O)CCC(NC(=O)C(C)CCCC)CC1C c1(C(=O)NC(CC)CCO)cccc(C#N)c1N c1(C(=O)NC2CC(CNC(c3ccoc3Cl)=O)C2)ccc2cnccc2c1 c1(OC)ccc2c(c1)CC(C(c1nnnn1C)Nc1ccc3nc(C)sc3c1)CC2 Cc1ccc(C(=O)NCC2CN(C(=O)Cc3ccc(C)s3)CCC2C)c(C)c1 c1(SC)cccc(C)c1C(=O)NC1CC1NC(=O)CCc1c(Cl)cccc1Cl C1(C(=O)NC2CC(CNC(C3CCC(C)(C)CO3)=O)C2)CCC(N=[N+]=[N-])CC1 C=C=CCN=c1[nH]c2c(c(=NCC3(C)CCOCC3)[nH]1)CCCC2 C12(CC(O)C1)C(=O)N2.c1(C(N2CC(C(C(=O)OC)O)C2)=O)[nH]ccc1C C12CC3(CCCN3C1=O)C2.N1(N(C(=O)C(C)C)CC)CC(C(=O)OC(C)(C)C)C1 C(c1cccc([N+](=O)[O-])c1)=CC(N1CCN(C(C(CCCC)C)=O)CC1C)=O C1(F)(C(=O)NCCSCC)CCN(Cc2cscc2Br)C1 C1(F)(C(=O)NC2CN(C(C=C(C)c3ccco3)=O)CC2F)CC2(CCC2)C1 CCCC(C#N)C(=O)NCC1CCC1C(N1CCC2CCC12)=O N1C(=NCCC(=O)NS(C)(=O)=O)NC1OC.C1(F)(COC)CC(C(=O)OC)C1 C1(C2CCC(=O)NC2)(NC2CC(C)(C)CN(C(=O)OC(C)(C)C)CC2)CCC1 c1(CNC(C(c2ccccc2Cl)NC)=O)ccc(OC(F)F)c(C)c1 c1(C(C(C2(CNC(C)(C)C)CC2)C2CCC2)C(=O)OC)nnnn1C1(OC)CC1 c1(OCCC(=O)NC(C)CCCNC(=O)CC2CCCC2)ccccc1F C(=O)(C1=CCS(=O)(=O)C1)NC1CC(NC(c2ccc(N)cc2F)=O)C12CCC2 c1(C(N2CCC(NC(C(C(C)C)n3cnnn3)=O)C2)=O)ccc2ncccn12 CCC(C)C(C)C(=O)NCCSCC(=O)NCCCn1ccnn1 C1(NC(C(CCC)F)=O)CC(NC(c2ncnn2CC)=O)C12CCC2 c1(C(N2CC(NC(C3(OCC)CCSCC3)=O)C(C)C2)=O)ncn2c1CCC2 C1(NCC)CCN(C(C2CC3CC3C2)=O)C1 C(=O)(C(C)(C)CC#N)N1CC(C(=O)NCCc2ccn(C)n2)OCC1 C12(NC(C3CC(OCC)C3)=O)CCCC(NC(=O)CCn3ccnn3)(C1)C2 C1(C)(C(N(CCCNC(=O)Cc2csc(Cl)c2)C)=O)CCNC(=O)C1 C1(C(=O)NCC2CC(C(N3CCC(F)(C(N)=O)C3)=O)C2)CC(=O)NC(=O)C1 N1(C(CCCSC)=O)CCC(CCCCNC(C2CCOC2C(C)C)=O)CC1 c1(C(=O)NC(C(C)NC(=O)C=CS(C)=O)CO)ccc(C(C)(C)C)c([N+](=O)[O-])c1 N(C(=NCCCCOc1ccc(Cl)cc1)NC1CCC1)Cc1c(C)noc1C C=CCCCC(C)(C)C(=O)N(C)CC1CCN(C(=O)C(O)CC2CCOCC2)C1 c1(C(N(C2CCCN(C(C(C)NC(C)=O)=O)CC2)C)=O)cc(F)c2c(c1)CCC2 N1(C(C23C(CN(C(CC4CCC(=O)CC4)=O)C2)C3)=O)CCC2(CCC2)C(O)C1 C(C(CC(C)C)C(=O)NC1(C(C)(F)F)CC1)NC(C(C)=CC(C)(C)C)=O c1(C(=O)NCC2CC(OC)CN2C(C2COCCO2)=O)cn(C)c(=O)n1C N1(C(=O)Oc2ccc(F)cc2)CC2CCC(F)(F)C2C1 c1(C(=O)NC(C2(O)CCN(C(C(COC)OC)=O)CC2)C)ccc2cncn2c1 c1(NC(c2ccn(-c3ccc(Cl)cc3)n2)=O)nccc(F)n1 C12(C(=O)NCC(C(=O)NC(C3CCOCC3)CC)O)CC(C)(CCO1)C2 c1(C(=O)NC2C3OCC(NC(COCC#C)=O)(C3)C2)ccc2c(c1)C=CCC2 c1(C(=O)NC(CN(C(=O)CCOC)CC)C)nsnc1O CC(=Cn1ccnn1)C(=O)N(CC(C)CNC(=O)CCCn1ccnc1)C CC1CC(NC(c2cnc(O)c(Cl)c2)=O)CN(C(c2ccco2)=O)C1 C1(NC(c2nc(OCC)sn2)=O)CCN(C(c2cncc(Cl)c2)=O)CC1(C)C C(CC(=O)N1CCOCC(CO)C1)(C(F)F)NC(c1n(CCC)ccc1)=O C1(C(=O)NCC2CN(C(=O)CC(F)F)CC23CC3)(OC)CCS(=O)(=O)C1 CC(CC1CC(F)(F)C1)C(C(=O)NCCC1CC1)N(C1CCN(C)C(=O)C1)C C1(CN(C(=O)C(c2cccc(OC(F)(F)F)c2)O)C)CCCN(C(=O)C2CC2)C1 C1(CN(C(C2(C)C(C)C2)=O)C)CCCN(C(=O)C(C)(C)CC2CCC2)C1 N1(C(c2c(C)cc(C)s2)=O)CCC2CN(C(c3ncc(F)cc3F)=O)CCC2C1 c1(C(=O)NC(C2CCCCC2)CNC(=O)CCC(F)(F)F)cccn2cnnc12 N1(C(C2CC(C)NC(=O)C2)=O)CCC2(CCC(NC(=O)C3=NOC(C)(C)C3)C2)C1 CC1CC(NC(c2ncncc2Cl)=O)CN(C(c2cc(Br)cn2C)=O)C1 N1(C(CN(C)C2CC2)=O)C2CCC1CC(NC(C1CC(=O)N(C)C(=O)N1)=O)C2 C1(CNC(c2c(C)n[nH]c2)=O)CCC(CNC(C2CCCCC2C)=O)CC1 N(C1CCc2cccnc21)C(C1C(C)(C)CCN(C(=O)C2=NOCC2)C1)=O C1(C(N(C(C)CN(C)C(c2cn(C(C)(C)C)nn2)=O)C)=O)COCCN1C c1(C(N(C2CCCN(C(C3(C)CC4CCC3C4)=O)CC2)C)=O)ccc(F)cc1Cl C=CCC(CC(C)C)C(=O)N1CC2(CCC(NC(=O)C(O)C(F)F)CC2)C1 C(=O)(C#CC(C)(C)C)N(C)CCOCCC(N1CCCCC1CN(C)C)=O C12(C(=O)NCC(C)NC(c3cn(C(F)(F)F)cn3)=O)CC3CC(C1)CC(O)(C3)C2 c1(C(C(=O)NC2(C(=O)NCC3(C#N)CC3)CCC2)F)ccccc1 Cc1cc(C(=O)NCC(C(N2CCN(C3CC3)C(=O)C2)=O)N(C)C)cnc1C CCC(O)C(C)C(=O)N1CCCC(CNC(=O)CC2CCC2)C1 c1(C(=O)NC(C)CCNC(C2(C(N)=O)CCC2)=O)cc2c(Br)coc2cn1 CC1CCCC(C(=O)NC2CC(CNC(C3(CC(F)F)CCC3)=O)C2)CC1 N1(CCC(=O)N(C(C)C)CCNC(=O)CC2CC(=O)C2)CCCCC1C CCC(C)(C(=O)N1CCCC(NC(c2ccnn2CC#N)=O)C1)C(N)=O C=CCCC(C1CC1)NC(=O)CN(C(=O)COC1CC(NC(=O)C(C)C)C1)C c1(CN(C(C(C)CC2CCC2)=O)C)ccc(CNC(C2(C)CC2C)=O)cc1 C1(CC=C)(NC(=O)CC(O)CC)CCN(C(c2cnn(C(C)(C)C)c2N)=O)C1 N1(C(c2oncc2C2CC2)=O)CCC(O)(CCNC(C2(CF)CC2)=O)C1 c1(NC)ccc(-n2cnc(C(=O)N(CC(C)O)CC3CC3)c2)cc1 c1(C(N2CC(CNC(COCCC)=O)C3C2C3)=O)cc(OC)cc(F)c1 n1(CC)ncc(C(=O)NCC(C(C)C)NC(C2(C)CC=CCC2)=O)c1Br c1(CC2CCCO2)ncc(CNC(=NC)NN(c2ccccc2)C)s1.CC C#CCC(CC(=O)NC(c1snnc1C)C)NC(=O)C(C)(C)COC Cc1ccc(C(=O)NC(=O)C(C)NCc2ccnn2-c2ccccc2)cc1 N1(C(C(C)OCCC=C)=O)CCN(C(=O)C(C(C)C)n2cnnc2)CC(O)C1 C12(CNC(=O)CSc3ccc(F)cc3)CC(CC1C(=O)O)C2 Cc1cc(CNC(C2(C)CCN(C(=O)CCC(C)(F)F)C2)=O)cnc1F c1(CN(C(C(CC)C2CCC(=O)N2)=O)C)ccc(Cn2ccnc2)cc1 N1(C(CCCOC(C)=O)=O)CC2OCCN(C(c3cc(=O)n(C)o3)=O)C2C1 C1(C)(C(=O)NCCNC(C2(CSC)CC2)=O)COCCO1 c1(C(=O)NC(C2CCN(Cc3ncccn3)CC2)C(F)F)cc(F)c(F)cc1Cl c1(OC)cc(NC(c2csc(C(N3CC(O)C3)=O)n2)=O)cc(OC)n1 C1(NC(C(C)NC(CC)(C)C)=O)COC2(CCN(C(=O)CS(=O)(=O)CC)CC2)C1 Cc1cc(C(=O)NC2CCC(C)N(C(=O)CCOC3CCCC3)C2)c(N)c(Cl)c1 N1(C(CC2(C)CC2(Cl)Cl)=O)CC2CC2(CNC(C2(C3CCC3)CC2)=O)C1 c1(C(=O)NC(C(C)NC(C=CC(C)C)=O)(C)C)ccc(C#N)n1C CCCCCC(C)CC(=O)N1CCC(N(C(C2CC(CCO)C2)=O)CC)CC1 N1(C(C(C)OCC(F)(F)F)=O)CCOC(CN(C(=O)C(=O)NCC2CC2)C)C1 c1(CCNC(N2C(c3ccn(C)n3)COCC2)=O)cc(Br)ccc1I c1(OC(C)C(=O)NCC23CC(CN2C(c2ccoc2)=O)C3)ccc(Cl)cc1 N1(C(C)=O)CCOC(C(N2CCCC2C2(NC(C3CC=CCO3)=O)CC2)=O)C1 N1(C(C2C(C)OCCO2)=O)CCC(C(=O)NCCCC2(C)CC2)CC1C N1(C(C(c2ccc(F)cc2)C)=O)CC2CCN(C(c3cnc(Cl)[nH]3)=O)C2C1 Cc1cc(C(=O)NC2C=CCN(C(=O)C(C)CO)C2)nn1C(C)C Cc1nc(C(N2CC(CC(=O)N(C34CC(C3)C4)C)C(C)C2)=O)cn1C C=CCN=C(NCc1ccsc1C(F)(F)F)NCC(C1CCOC1)OCC C1(NC(=O)C=C(Cl)Cl)(CO)CCCN(C(=O)C(O)C(F)(F)F)C1 c1(C(=O)NCC(C)CNC(c2cc(-c3ccncc3)on2)=O)nnn(C)c1N Cc1ccc(C(=O)NC(C2CCN(c3ncnc(C(C)C)n3)C2)C)cc1 c1(C(N2CCC3(CN(C(CCNS(C)(=O)=O)=O)C3)C2)=O)cccc2nc(O)[nH]c12 O=C(C1=C(Cl)CCOC1)NCCC(O)CNC(C1(CC(F)F)CC1)=O c1(C(=O)NC(c2cn(CCCO)nn2)C)nn(C)c2c1CCCC2 c1(C(=O)OCC(C2(CS(C)(=O)=O)COC2)=O)nc(Cl)cs1 C1(CNC(CC2(C)CCOC2)=O)CN(C(=O)CCOCCN(C)C)C(C)(C)C1 Cc1occ(C(F)(F)F)c1CC(=O)NC1COCCC1NC(=O)C(C)C(F)F C(N=c1[nH]c(=NCC2OCc3ccccc32)[nH]c2c1CSC2)c1n(C)ccn1 CC(C)(CCCCC(=O)NC1CC1(F)F)C(=O)NNC(=O)COCc1nncs1 C(C)(CCCCNC(c1ccc(C(C)(F)F)cn1)=O)NC(C(C)OCC(C)C)=O C(CC(O)CC(=O)N1CCOC(CCNC(=O)Cn2nnc(C)n2)C1)SC Cc1cc(C(C)C)nc(=NCCCCNC(=O)Cc2cc(C3CC3)nn2C)[nH]1 C1(CNC(C2CC(=O)N(O)C2)=O)CC12CCN(C(=O)CCOCC1CCC1)CC2 c1(CN2CCC(C(F)(F)F)(C(=O)NC)C2)cc(Br)ncc1Br C(C)(C(CC(=O)NCC(C1CC1)C1CC1)NC(c1c[n+]([O-])c(C)cn1)=O)OC C1(CCCNC(C=CC=CC)=O)CN(C(C23CC(OC)(C2)C3)=O)CCO1 C1(N(C)C)(CC)CCCN(CC(=O)Nc2cccc(C#N)c2)C1 N1(C(C(C)(C)C#N)=O)CC2CCC(NC(=O)CC3(O)CCOC3)CC2C1 N1(C(CC(CC)C)=O)CCC(C(N2CCC(N(CC)CC)CC2)=O)C(C)(C)C1 c1(OC)ccc(F)c(C(C)C)c1.C12CCN(C1)C(=O)C(=O)N2 C=CCC(CC=C)C(=O)NCC1CCN(C(C2CCC2(C)C)=O)CC1C NC(=O)CCCCC(=O)N1CC(CNC(=O)CCC2CC2)OC(C(F)(F)F)C1 C1(CNC(=O)CC2CCCO2)CCN(C(=O)Cn2ncccc2=O)CC1(F)F C(CCC(=O)N1CC(C)(CC(=O)NCC2CNC(=O)C2)C1)OC(C)(C)C Cc1ncccc1CC(=O)NCCC(O)CNC(c1ccns1)=O CC1CC2(C1)CC(N=c1nc(N3CC4CC3CS4=O)c3c([nH]1)CCOC3)C2 N1(C(C2CN(C)CC(C)O2)=O)C2CCC(C(=O)NC3(C)CCCC3(C)C)C1CC2 N1(C(CSCC#C)=O)CCC(F)(C(=O)NCCC2CCC(C)O2)CC1 Cc1cc(-c2ccc(C(=O)Nc3ccno3)nc2C)cc(C)c1 C#CC1(C(=O)NC2CCCC2NC(=O)CCc2ccc(Cl)nc2)CCOCC1 CS(=O)c1cccc(NC(c2ncccc2C(F)(F)F)c2nnnn2C2CC2)c1 S1(=O)(=O)c2cccnc2N1.Cc1nc(C(C)C)ccc1CNNC1COC(C)(C)C1 c1(C(=O)NCCCCN(C(CCN(CC(C(C)C)C)C)=O)C)occ2c1CCC2 Nc1cc(C(=O)NCC(CO)NC(=O)CCc2ccoc2)ccc1Br c1(-c2cn(C(C)C(C(=O)CCCC3CCCC(=O)N3)=O)nn2)cc(C#N)ccn1.N c1(OC)cc(F)c(C(N2CCC3(C2)CN(C(=O)CSCCN(C)C)C3)=O)c(Cl)c1 C1(C(=O)NC23CC(CNC(=O)CS(=O)(=O)N4CCCC4)(C2)C3)CC12CCSCC2 C1(NC(C(CCOC)(C)C)=O)CCN(C(=O)C(C)(C)c2ccc(Cl)s2)CC(O)C1 c1(C(=O)NC(CC(C)C)CNC(=O)CCCC2CC2)sc([N+](=O)[O-])cc1Cl C12(C(=O)NC3CN(C(c4cccc5nc[nH]c45)=O)C3)CCCCC1CC(F)(F)C2 CCC(CNC(C1(Cl)CC1C(=O)OC)=O)(CC)NC(c1cc(COC)oc1C)=O c1(C(C)C)nc(NC(CC2CC2)C2CC2)cc(N2CCCC(N(C)C)CC2)n1 c1(C(N2CC(C)(C)C(CNC(=O)CC3CC34CC4)C2)=O)ccc2c(c1)COCC2 CCCC(C)(CC)C(=O)N1CCN(CC(C)NC(c2cc(C3CC3)ns2)=O)CC1 CC1(C)CCCC(C(=O)NC(Cn2cncn2)C(=O)NCC2(Cl)CCC2)C1 c1(C(=O)NCC2(O)CCN(C(C(c3c(C)cncc3)C)=O)C2)ccnc(Cl)c1O c1(C(=O)NC2CC(C)(CNC(C(CC)CC)=O)C2)ccc(C=NOC)cc1 Cc1oc2ccccc2c1C(N1CCC(O)(CNC(=O)C(C)(C)F)CC1)=O Cc1nnc(CCC(=O)NCC2(F)CC(CNC(C3CCCC3C)=O)C2)n1C c1(CC(=O)NC(C)CNC(=O)CN2CCCC2CO)cnn2ccccc12 N1(C(CC2CCCN(C(C(C)C3CC3)=O)C2)=O)CC2(C1)CC(C)(F)C2 CCCC(C)(C)NC(=O)NCc1ccc(-c2sccc2C)s1 Cc1nc(CC(=O)N(CCCN(C)C(C2CC(C(N)=O)C2)=O)C)c(C)s1 C=CC12CCN(CC1)C2=O.c1(NC(C2COC(C(C)C)C2)=O)cccc(CO)n1 c1(NC(N2CCN(c3ncccn3)CC2)=O)ccc(C(N2CCCC2)=O)c(Cl)c1 c1(C(=O)NC(COC)CNC(c2cocn2)=O)cccc(N(C)C)c1 O=C1CCc2cc(S(=O)(=O)N3CC(C(F)F)C4(CC4)C3)cc(F)c2N1 CCCC(CC)CCC(=O)NCCC(CNC(=O)Cc1cnc(C2CC2)[nH]1)OC C#Cc1cc(F)ccc1CN1CCC(C(=O)NCc2cncnc2)C1 C1(NC(C=C(COC)C)=O)CCC(C)(CNC(=O)C(F)=C(C)C2CC2)C1 C(=O)(CC(O)C(C)CC)NC1(C(=O)NCc2ncc(CC)[nH]2)CCSC1 c1(CC)ccc(C(N2CC(NC(=O)COC3(C)CCCC3)CCC2C)=O)cc1F C1(C(N2CC(NC(C(C)CC3CCC3)=O)C(O)C2)=O)CCc2ccccc2CC1 c1(NC(c2n(CCC)nnn2)c2cn(C3CCC3)nn2)ccc(Cl)c(C(F)F)c1 C1(CC(=O)NCCCN(C(C2CCN(C(=O)OC)CC2)=O)CC)CCCC(O)C1 C=CCCC(CC(C)C)C(=O)N1C(CNC(c2coc(Br)c2)=O)CC2COCC12 C1(CC(C)NC(C2CC(CF)C2)=O)CCN(C(=O)COC2CCCOC2)CC1 C1(CCNC(CC2(OCC)CC2)=O)CN(C(=O)C(C)OC2CCOC2)C1 C#CC1(O)CCCN(C(C23CCCC2CN(C(=O)CC(O)CC(C)C)C3)=O)C1 C1(NC(=O)Cn2cccn2)CN(C(C23CSC(C2)C3)=O)C2CCCCC12 c1(C(=O)NCC2C=CCN2C(c2cocn2)=O)ccc(OC(F)(F)F)cc1Cl N1(C(c2c(C)nccn2)=O)CCC2(NC(c3[nH]nc([N+](=O)[O-])c3Cl)=O)CCCC12 C(CCCC(c1nnnn1C1CCOCC1)NCC1(C)CCCS1)(OC)OC O=S(=O)(c1ccc2occc2c1)NCc1ccc2c(c1)CCCC2 C1(CF)CCCN(C(=O)C(=O)N(C)NC(c2ccco2)COC)C1 N(C(=NCCSC)N1CC2C(CF)C2C1)C(c1ccc(S(=O)(=O)NC)cc1)C N1(C(C(C=C)(C)CC)=O)CC2CCN(C(=O)CSc3n[nH]c(O)n3)CC2C1 CN1CCN(C(=O)C(CC(F)F)N(C(=O)CC2CC=CCC2)C)CC1=O N1(C(c2c(COC)noc2)=O)CCC2(CCN(C(=O)C(C)(O)COC)CC2)C1 C1(NC(Cc2ccc(C)s2)=O)CN(C(c2sccc2NC(C)C)=O)CCC1CO C1(C(=O)NC2CN(C(=O)C(F)CC3CCOC3)C2)OCC2CCCC1C2 c1(C(=O)NCC2(C)OCCN(C(Cc3cn(C)nn3)=O)C2)onc2ccccc12 C(C(C)(F)CNC(c1ccc(CO)s1)=O)NC(C=CCN(C)CC)=O n1(CCC(N2CCCCCC(NC(C=NOC)=O)C2)=O)cnc2c(N)ncnc12 C1(NC(C(C)(C)n2cnnn2)=O)C(C)(C)C(NC(C2CCCOCC2)=O)C1(C)C N1(C(CC)=O)CCC(NC(c2cnc(C)nc2COC)=O)CC(C)(C)C1 C1(CCC)(NC(=O)CN(S(=O)(=O)CC)C)CCCN(C(C2(C)CCNC2=O)=O)C1 CCC(C)(CNC(c1cnccc1OC)=O)C(=O)NC1CCCCC1C#N N1(C(CCC#C)=O)CCC(C)C(NC(=O)CC(C)(C)c2ccccc2)C1 N1(C(CSCC(C)C)=O)CC2(CCN(C(C3CC3F)=O)CC2)CC1C C1(NC(CCS(=O)(=O)N(C)C)=O)CCCC12CN(C(c1ccc(F)o1)=O)C2 N1(C(Cn2c(CC)ncc2)=O)CCC2(NC(=O)CNC(=O)C3=CCC3)CCCC12 c1(NCC2(N(C)C)CCC2)ccc(S(=O)(=O)NCC2(Cl)CC2(F)F)cc1Br N1(C(C2OCCC(C)(C)C2)=O)CCC(C(=O)NCCOC2CCCC2)CC1(C)C C1(C)(CNC(C(C)NC(C)=O)=O)CCCN(C(=O)CCS(N)(=O)=O)C1 C1(C(=O)OC)(C(C)C)CC1CNC(C)C(=O)NCC(F)(F)F CCC(CC)C(F)C(=O)N(C(C)CNC(=O)C(n1cc(C)cn1)C)CC N1(C(C(C(C(C)C)O)C)=O)CC(C(C)(C)C)Nc2ccccc21 Cc1ccccc1CC(=O)NCCC(C)NC(=O)C(=O)NCC1CC1 C1(CCNC(CC2C(C)CCC2)=O)CCCCN1C(c1cnc(S)n1C)=O C1(CC(=O)NCC(C)(CO)NC(=O)C2=C(Cl)CC2)CCCCCCC1 N1(C(C2C(C(C)OC)OCC2)=O)CC(CNC(=O)C=CSc2nc[nH]n2)CC(C)C1 N1(C(C(C)SC)=O)CCC(OCCNC(c2sccc2-n2cccc2)=O)C1 C1(CN(C(c2c(CC)scc2)=O)C)CN(C(=O)C(=O)N(C)C)CCO1 CCS(=O)CC(=O)N1CCC(C)C1CNC(=O)Cn1ccnn1 c1(NC(C(=O)NCCc2cc(C3CC3)no2)=O)ccc(S(=O)(=O)CC2CC2)cc1 C=CCCC(O)CN(C)C(c1sccc1CNC(=O)CC1CC1(C)C)=O Cc1ccc(-c2nnnn2CSC2(C)CSC2)cc1NCCCN1CCOCC1 C=C=C(C)CC(=O)N(C)CC1CCN(C(c2ccc(C3CCCO3)nn2)=O)C1 N1(C(C(C)Br)=O)CCCC2(CCCN2C(=O)C(C)Oc2ccccc2)C1 C=CC(CC)C(=O)NC1CCOC(CNC(=O)CCc2nccn2CC)C1 C(C(C)C(C)C(=O)N1CC2CC1(CNC(c1c(Cl)nsc1Cl)=O)C2)OC C(=O)(C1CCCc2cncn21)NC1(C2CCCN(C(C3CC(C)(O)C3)=O)C2)CC1 C(=O)(C(CCC(C)NC(C)CC(=O)NC(C(C)C)C1CC1)C(=O)OC)OC Cc1cc(F)ccc1NC(C1(C)CCN(C(C2CC2C(C)C)=O)CC1)=O N1(C(c2cnc(N(C)C)o2)=O)CC(O)CC1CNC(C1CC2C=CC1C2)=O Cc1cnn(C)c1C(=O)NCC1(O)CC(CNC(=O)CCS(C)=O)C1 c1(C(=O)NCC(=C)CCNC(=O)CCC2CCCC2)ccc(SCCCO)cc1 C1(C(N2C(CN(C(CCOC)=O)C)CCC2)=O)CCCCS1(=O)=O C1(CCCC)CN(C(=O)C(C)(C)C(C)C)CCN1C(c1nn(CC)nc1C)=O c1(C(=O)NC2C(OC)CN(C(C34CC(F)(C3)C4)=O)C2)cnc2n1CCC(C)C2 c1(SC)ccc(F)c(-c2cc(NC(C3CCC(CCN(C)C)CC3)=O)cs2)c1 C1(C(F)(F)F)(NC(=O)NC(CC#C)CC(F)F)CCC(C)c2ccccc21 c1(OC)ccc(C(N2CC(CNC(=O)Cc3ncc(C(C)C)[nH]3)C2)=O)cc1 N1(C(Cc2nn(C)c(Cl)c2)=O)CCN(C(C2(C)COCCO2)=O)CC1C1CC1 N1(C(C=CC(C)(C)SC)=O)C(C(N2CCSCC2CO)=O)CCC1C1CC1 N1(C(C(CC)CC)=O)CC(C)CN(C(C2NC(=O)CC2C)=O)CC1C c1(CC(F)F)cccc(NC(c2ccn(C3CC3)n2)c2nnnn2CC2CC2)c1 c1(C(=O)NC2CCCC2C(=O)OC)cc(C)c(C)[nH]1.C=C1CC2(C1)C(=O)NC2 N1(C(COCCCC)=O)C2CCC1C(C(=O)NCc1nccc(O)n1)C2 CC(C)(F)CCC(=O)N1CCC(C(C)(C)C)(CNC(c2cccnc2)=O)C1 N1(C(C=CCNC(c2c(CC)nco2)=O)=O)CCC(OC)C(F)C1 C(c1cnn(C)c1)=CC(N1CC(C(N)=O)(CNC(C2CC23CCOC3)=O)C1)=O N1(C(C2(CC=C)CN(C(=O)C=Cc3ccncc3)C2)=O)CCOC2CC12 N1(C(c2n(C)ncc2I)C(=O)NCc2ccccc2)CCC2CCCCCC2C1 c1(Cn2c(NC(C(=O)NCC(c3ccccc3F)C)=O)ccn2)ccc(Br)cc1 C(=O)(C(C)CC(C)(C)C)N(CCC(C(C)C)NC(C1CCC(C)O1)=O)C C(CCCCC(=O)NC1C=CCCC1C(=O)NC1CCOC1C1CC1)N(C)C C(=O)(C(CNC(C1C2CC(=O)CC12)=O)CC(C)C)NCCc1ncc(C)o1 C(=O)(CS(=O)(=O)c1ncc[nH]1)N1C(C)C(O)CCC1.c12cccc(c1)OC2 C1(C)(C(=O)NCC2(NC(C(C)N(C(C)=O)C)=O)CCCCC2)CCCCCC1 C(=O)(C1=CCSC1)NC(CC)(C)CNC(c1cc(-c2ccc(Cl)s2)on1)=O Cc1cnc(F)cc1C(c1nnnn1CC1CCC1)NCCc1ccns1 c1(CC(C(N2CC(F)(C(=O)OCC)C2)=O)F)ccc(OC)cc1 N1(C(C2CCN(C)C2)=O)CC2CC1C2NC(=O)C(c1cccnc1)O n1(CC)cnnc1C(=O)NCC1CC1COC.N12CC(CO)(C1)CC(=O)NC2=O Cc1cccc(C=CC(=O)NC(CC(=O)NCC(C)CN(C)C)C(F)F)c1 Cc1cc(C(N2CC(=C(F)CNC(=O)CN(C)C(N)=O)C2)=O)nn1C(C)C1CC1 CN1CCN(C(C2C3CCCCC23)=O)C(CNC(c2cnn(C)c2C(F)F)=O)C1 c1(C(=O)OCC(=O)CC2CC3CCC2C3)c[nH]c2cnccc12 c1(C(N2CC3C(C2)C3(F)F)=O)nc2ccc(-c3ccc(C4COC4)cc3)cc2o1 c1(CC)ccc(CNC(=O)NCC2(O)CCCC2(C)C)c(OC)c1 c1(C(=O)NCCC(C)NC(c2ccc(=O)oc2)=O)occ2c1CCOC2 N1(C(C2CCN(C(C(C(C)C)OCC)=O)C2)=O)CCC(C)(C)C1C(=O)NC C1(C(N2CCN(CC=C)CC2)=O)CCN(C(c2occc2C)=O)C(C)C1 C#Cc1cnc(C(=O)N(C2CCCC2)CCNC(=O)CC2CCC2)c(C)c1 N1(C(=O)NC(c2ccccc2)=O)CC2CN(Cc3sc(C=O)c(Br)c3Br)CC2C1 C1(N(C)C(C2CCCN(C(=O)C(=O)NCC(F)(F)F)C2)=O)CCOC(C)(C)C1 Cc1ncnc(NC(CCNC(=O)CC(=O)N(C)C)C(C)C)c1F c1(C(=O)NCCC2(OC)CN(C(CC=C)=O)C2)cc(C(F)(F)F)cn1C C(C(C)C(F)C(=O)NCC1CCOCC1)NC(CN(C1CC1)CC)=O C(=O)(C1=NOC(C)C1C)N1CC(C(=O)NC(CC#C)CO)C(CCC)C1 N1(CCNC(c2c(C)onc2Cl)=O)CCCN(C(C2CC2C2(C)COC2)=O)CC1 C(C1=CCN(C(=O)C2=NOC(C)C2)CC1)NC(CC(c1ccc(F)c(F)c1)C)=O N1(C(CN(CCCCCC)C)=O)CCC(N(C(c2[nH]c(C)cc2C)=O)CC)CC1 N1(C(C2CCOCC2)C(=O)NCCCOC)Cc2cccc(F)c2C1 C1(CSC)CC2(C1)CC(C)N(C(=O)NCc1nnc(C(=O)OC(C)(C)C)o1)C2 c1(OCC=C)ccc(C(=O)NCCCN(C(=O)C=CC)C)cc1OC1CC1 N12CSCC1C(=O)NCCNC(=O)C21CC1.c1(OCC(=O)OCC)cn(C)cn1 C1(C)(CNC(CCC(=C)C)=O)CN(C(c2nncn2CC)=O)C(C)(C)C1 C1(NC(C2=C(C)CCCC2)=O)CN(C(=O)Cn2cccc2)C2(CCOCC2)C1 N1(C(c2c(CC)nccn2)=O)CCN(C(c2ccnn2CC(F)(F)F)=O)CC1C c1(C(N(CCN(C(C(F)=CC)=O)C(C)C)C)=O)ccc(O)c(Cl)c1 C1(NC(C(C)OCC2CC2)=O)CCCN(C(c2cnc(Br)s2)=O)C1 c1(CN2C(C(=O)NCCc3ccc(Br)s3)CC(O)C2)cnc2[nH]ncc2c1 N1(C(c2ncsc2C)C(=O)NCC(=C)C)CCC2(CC1)CC2C(=O)OCC c1(C(N2CCC(NC(c3ccn(CCOC)n3)=O)(CF)C2)=O)cc([N+](=O)[O-])sn1 N1(C(CC2CC(OC)C2(C)C)=O)CC2CCC1CN2C(=O)CC1CCCCCC1 C1(O)(CNC(c2c(SCC)cncc2)=O)CCN(C(=O)C(F)OC)CC1 N1(C(C2(C=C)CCC2)=O)CCOC(CNC(=O)C(O)CC2CCOCC2)C1 C(CS(=O)(=O)C1CCCCC1)N1CC(C)C(C)(CO)C1 C1(c2nc(CS(=O)(=O)NC(C)C(F)(F)F)[nH]n2)COC(C)(C)C1 N1(C(c2cc(C)n(C)n2)=O)CCC2(CC1)CC2CNC(C1CC(F)C1)=O N1(C(COCCC=C)=O)CCCCCC(NC(=O)C(C)Cc2ccccc2Cl)C1 C1(C)(OC)CCCN(C(c2conc2C(C)C)C(=O)Nc2ccccc2)C1 Cc1ccc(NC(c2cncc(C(=O)NC3CC3C3CCCC3)c2)=O)cc1C#N C1(NC(c2cc(CF)on2)=O)CC2CCC1C1CN(C(=O)C=C(Cl)Cl)CC21 CCCC(CC1CCCC1)C(=O)N1CCC(CO)(NC(=O)Cc2ccoc2)CC1 CCC(C)CCC(=O)NCCCCN(CCCNC(C1(C)CC(C#N)C1)=O)C N1(C(c2c(CC)onc2)=O)CCC2(CC1)CC2C(=O)Nc1cc(C)nc(OC)n1 S(=O)(=O)(c1ccc(N2CCCC(C(=O)OC)C2)c(F)c1)N(CCOC)C Cc1ccc(C(=O)N(CC(O)CN(C(=O)CCC2CCCCO2)C)C)cc1CO C1(CC(=O)NC(C)CCC2CCCCO2)CC(O)CN1C(=O)OC(C)(C)C N1(C(=O)OC)CC2CC1C2C(N1CC(NC(c2cn(C3CC3)nn2)=O)C(O)C1)=O C1(C(C(C)C)NC(c2ccn(C)n2)=O)CCN(C(C2C(C#N)C2(C)C)=O)CC1 c1(-c2cnc(C(N(CC(F)(F)F)CC)=O)nc2)ccc2c(c1)CCC2=O Cc1nccnc1C(=O)N(C(C)(C)CC(=O)NCC1(O)CCOC1)C CC(C)C(C(C)NC(=O)Cc1cnsc1)NC(=O)CCc1cncc(F)c1 CC(C)C(C)C(C)CC(=O)N1CCC(NC(C2Cc3nccnc3C2)=O)C1C N1(C(c2cnc(OCC)nc2)=O)CC2(CC2)CC1C(=O)NC(C)C1CC1 Cn1nc(C(=O)NCC2COCC2NC(C2(C)COCCO2)=O)cc1C(F)(F)F N1(C(CC2ON=C(CC)C2)=O)CCC2(CC(NC(=O)CCOC3CCCC3)C2)C1 CCC(C)(COC)C(=O)NCC(C(=O)N1CC(C)(CO)C1)N(C)C Cc1nn(CC(=O)NC(C)(CNC(=O)C(C)C2CCCC2)C(C)C)c(=O)o1 C1(C)(C(=O)NCc2cc(C(N3CC(C(C)OC)C3)=O)n(C)n2)CCC(=O)NC1 C(=O)(CC(C)CC(C)C)NCC(C1N(C(COC(C)=O)=O)CCC1)(C)C c1(C(=O)NCC(CC)(C)NC(C2CN3CCCC3CO2)=O)cnc2[nH]cncc1-2 C(c1ccc(F)cc1)=C(C(=O)NCCCN(C(c1cnc(CC)s1)=O)C)C N1(C(C2C(O)CCN(C(c3ncc(Br)nn3)=O)C2)=O)CCOc2ccccc2C1 CC(CN(C)C)CCC(=O)N1C2CCC1C(CNC(c1cc([N+](=O)[O-])n[nH]1)=O)C2 c1(C(N2CC3CCC3(NC(C3CC(O)C3)=O)C2)=O)nc2c(Br)cccn2n1 Cc1c(Cl)cnc(N2CC(c3cc(O)no3)C2)c1C#N O=C(C1=C(Cl)CCCC1)NC1CCC(O)CN(C(C2CCC(CO)CC2)=O)C1 CC1CN(C(=O)CC(F)F)CC1NC(c1cncc(-c2ccccc2)c1)=O C(=O)(CC(CNC(C12CC(F)(C1)C2)=O)C1CCC1)N1CCC(C(N)=O)C1 CC1CCN(C(c2csc(Cl)n2)=O)C1C(=O)NCC1(CO)CC(C)C1 c1(C(N2CC3C(CNC(C(C4CCC4)OC)=O)C3C2)=O)cncc2ncn(C)c12 N1(C(=O)Cn2ccnn2)CC2(C=C(C(=O)N3CC4C=CCC(C4)C3)CO2)C1 C1(N(C(C(CCOC)NC(=O)C(C)=CC(C)(C)C)=O)C)CC2CCC1CC2 c1(C(N2CC(CNC(CCN(CCC)C)=O)C(C)CC2)=O)cc2n(n1)CCOC2 N1(C(c2nccc(CNC(CCCOCCC)=O)c2)=O)CCCC(C)(C#N)C1 c1(CNC(CC2(CSC)CC2)=O)cc(C(=O)NCC2(N(C)C)CC2)cs1 Cc1cn2cc(CC(=O)N(CCNC(C3(CO)CCCO3)=O)CC3CC3)nc2s1 c1(C(=O)NC(C)CC2CN(C(C3CCC3(C)C)=O)C2)ccc(F)c2cnccc12 CC(O)CCCCCC(=O)NC1CC2(C1)CC2NC(c1ccn(C(F)F)n1)=O C(=O)(C1CCOc2ccc(Cl)cc21)N1CCN(CCNC(C(C)C)=O)CC1 C1(C)(CNC(CCSCC)=O)CN(C(c2ccc(C(=O)OC)o2)=O)C(C)(C)C1 CC(=Cn1ccnn1)C(=O)N(C1CCC(NC(=O)C(O)Cc2ccccc2)C1)C C1(CNC(c2cnccn2)=O)CCN(C(c2ccc3cc[nH]c3c2)=O)CC1(F)F n1(CC)nnnc1C(C1CCCO1)(C)NCC(C)COC(C)C c1(C(C)NC(=O)C(c2cccs2)NC(c2cc[nH]c2)=O)cccc(O)c1 N1(C(C2=CC(C)(C)C2)=O)CCCC2(CCN(C(C34CCCC(C)(C3)OC4)=O)C2)C1 C1(C(=O)NCC2=C(C)CCC2)C2CC(O)C(C2)N1C(c1ccc(C)cc1F)=O N1(C(C(CCSC)NC(N)=O)=O)CCN(C(c2nccn2C(C)C)=O)CC1C C(=O)(CC1OCCc2sccc21)NCCN(C(=O)Cc1ccnc(Br)c1)C C1(C(C(=O)N(CCCC)CCOC)C)CCn2cncc2C1 c1(C(=O)NCC(C)(CC2CCC2)OC)c(C)cccc1F C1(C(N2C(CCC(=O)NC(C)CSC(F)F)CCC2)=O)CC(=O)N(C)C1 S(=O)(=O)(c1cccnc1Cl)N1CC2(CC(NC(=O)Cn3nccn3)C2)C1 N1(C(c2n(CC)ncc2)=O)CC(NC(=O)CNC(=O)CNC(C)=O)C2(CCC2)C1 C(=O)(CCCC(C)(C)C#N)NC(C(N1CC(O)(CN(C)C)C1)=O)CN(C)C N1(C(C(C)SC(C)C)=O)CCCC(F)(CNC(c2n[nH]c3cccnc23)=O)CC1 C1(NC(CSCCC)=O)CC(NC(=O)C(=O)NC(C)(C)CC)C12CCOCC2 N1(Cc2cn(C(CC(C)(C)CO)Cc3cccc(Cl)c3)nn2)CC(=O)CCC1=O C12(CNC(c3cccc(OCC)c3)=O)CCC(C1)N(C(=O)C(O)CC(C)C)C2 c1(NC)ccc(C(=O)N(Cc2cn(CC3CC3)nn2)CC2CCCO2)cc1F N1(C(c2c(OC)cccn2)C(=O)NC2CCOC2)CCc2c(Cl)cccc21 N1(C(COCP(C)(C)=O)=O)CCN(C(c2nccnc2N)=O)C2CCC12 C1(C(=O)NCc2n[nH]c(C)n2)(CC)CCCN1C(=O)C(C)OCC(C)C c1(C(=O)NC(C(C)C)CCNC(C2CC(=O)N(C3CC3)C2)=O)ccc(O)c(O)c1 C1(OCCNC(C(C)n2ccnc2)=O)CCN(C(C2C(C(C)=O)C2(C)C)=O)C1 CC(C)C(CC(=O)N=c1ccn(CCCO)[nH]1)NC(C1CCSC1)=O CCC(C)(CNC(C12CC(C)(CCO1)C2)=O)C(=O)NCCn1nc(C)nc1C C1(CCNC(C2(Cl)CC2)=O)CCCN(C(=O)CC2=CCCC2)CC1 CC1(C(N2CC(OCC(=O)NC3CCNC(=O)CC3)C2)=O)CCC(=O)NC1 C1(C2CC2)(COC)CN(C(=O)CN(C(=O)CC2CCC(C)O2)CC2CC2)C1 N1(C(C(C)(C)CCC#N)=O)C2CCCC1CN(C(=O)CC1CCCCC1(F)F)C2 C(=O)(C(C(C)C)NC(c1cccnc1CNC(C1C=CCCC1)=O)=O)OC C1(=O)C(F)C(C)CN1.C(=O)(C(C)(C)NCC=C)NC(=O)C=CCCC(C)C c1(COC)ccc(C(=O)NCC2(F)CC(NC(C3CC3C)=O)C2)s1 N1(C(c2ccc(CC)cn2)=O)C(C(=O)N(C2CC(O)C2)C)CCC12CC2 N1(C(C2(CC=C)CN(C(=O)CNC(C3CC3C)=O)C2)=O)CCC(C(C)C)(CO)C1 N1(C(c2ccc[nH]2)=O)CCC2C(C1)CN2C(c1ccc(F)c(C(F)F)n1)=O C(=O)(C(C#N)C(C)(C)C)NC(CC)CN(C(c1cncc(COC)c1)=O)CC C(=O)(C(F)(CNC(=O)C(C)=C1CCCC1)C(C)C)N(CCCN(C)C)CC c1(OCCC(=O)N(CC(CC)NC(=O)C(C)(C)CO)C)ccc(C)cc1OC C1(CC)C(C(=O)NCCCCN2CCCC2)CCN1C(=O)CC1CCCC2CC12 C1(OC)CCC(C(=O)NCCCCCN(C)C(c2coc(CO)c2)=O)C1 CCCS(=O)(=O)C(C)C(=O)N1CC2CN(C(C3(C)CC(C#N)C3)=O)CC2(C)C1 CCC(CC(=O)N1CCCC1CCC(=O)Nc1ccc2ccoc2c1)C(C)(C)C C1(C(N2CC(C)(NC(c3ccoc3Cl)=O)C2)=O)CCC2CC1CO2 N1(C(c2cccc(C#C)c2)=O)CCC2CCN(C(=O)C=C(C)C#N)CC2C1 n1(CC=C)cc(C(=O)NCC2CCCN2C(=O)C(C)SC)c2ccccc12 C(=O)(C(C)(C)C(O)C(C)C)NC(CCCNC(c1c(CC)nco1)=O)(C)C C(c1cccc(Cl)c1)=C(C)C(=O)NCC1(NC(=O)CCC#CC)CCOC1 C(=O)(C1=C(Cl)CCC1)N(CC(C)NC(=O)Cc1cc(C)ccc1OC)CC Cc1ccc2cc(CN3CCC(O)CC3C(N3CCC(CO)C(O)C3)=O)sc2c1 N1(C(C(C=C)C)=O)CCC(C)(C)C1C(N1CCCC(C)C1CO)=O Cc1ccc(CS(N2CC(C)(F)C2)(=O)=O)c(F)c1 O(S(=O)(=O)c1ccc(I)cc1Br)c1ccc2c(c1)OC(CC)CC2 c1(C(=O)NCC2(C(F)F)CCN(C(c3n(C)ccc3)=O)C2)cccc([N+](=O)[O-])c1 C(CC(=O)N(CCCCN(C(=O)Cn1ccnn1)C)C)N(C(C)=O)C CC1CN(C(=O)CSCc2ccc(F)cc2)CCN1C(c1ccc(O)nn1)=O C(=O)(C1CNc2ccccc21)NCC(C)N(C(CC(CC)C)=O)C c1(C(C(=O)NC(CNC(CCNC(COC)=O)=O)C2CC2)O)cc(Cl)ccc1F C(=O)(CC1COCc2ccccc21)N(CC(C)(C)NC(C1CCN(C)C1)=O)C C=CCC(CO)CN=C(NCC(C)(C)C)NC1CCOCC1 CC1CC(NC(=O)CCNC(C2CC(F)(F)C2)=O)CCN1C(c1ccccc1)=O CC(C)CC(O)C(=O)NCc1ncoc1C1CN(C(=O)CC(C)CF)C1 c1(C(=O)NC(CC(C)NC(c2nonc2N)=O)C)cc(S(=O)(=O)N(C)C)cn1C c1(NC(=O)NCC(CN(C(C)C)CC)O)nc(CN(C)CC2CC2)cs1 C1(NC(c2ccoc2Br)=O)CCN(C(c2cnns2)=O)CC12CCC2 C(C(C)C(F)C(=O)NCCCc1ccnn1C)NC(Cn1c(C)nnn1)=O C1(C2(C(=O)NCC(CNC(=O)CCC3OCCO3)F)CC2)CCCCO1 C12(C(=O)NC3C(CNC(C4CCCSC4)=O)CCC3)CC(C(F)F)(CO1)C2 Cn1cc2cccc(C(N3CC4CN(Cc5scnc5Cl)C4C3)=O)c2n1 Cc1cncc(C(=O)NCC2(C(C)NC(=O)C(n3cc(Cl)cn3)C)CC2)c1C c1(C(C(=O)NC2CCC2)N(C(C)C2CC2)C)nn(C)cc1Br Cc1ccn(CC(N2CCCC(NC(=O)CNC(=O)CN(C)C)C2)=O)c(=O)c1 c1(OC)ncccc1NC(=O)C(c1ccnn1C)NC(C1CCC(CO)CC1)=O c1(C(=O)NC(C2CN(C(C3CCC(F)CC3)=O)C2)C)c(Br)nc2n1CCCC2 C1(NC(C(CO)N(C)C)=O)CN(C(=O)CCc2nnc(S)n2C)CC1N=[N+]=[N-] c1(C(=O)NC23CC(CNC(C(C)C#N)=O)(C2)C3)cccc(Cl)c1OC(F)(F)F N1(C(c2c(C)[nH][nH]c2=N)=O)CCC2(CCCCC2NC(C23CC(F)(C2)C3)=O)C1 C(C(C)CC(=O)NCCCn1cnnc1)NC(C=CC(C)(C)SC)=O CC1CN(C=O)CCN1C(=O)C(C)C(F)F.C12CCN(CC1)CC2.CC(F)(F)F N1(C(C(CC=CC)NC(=O)C(F)CCCCC)=O)CCC2CN(C)CCC12 c1(C(=O)NC(C2CCN(C(CCC(C)(C)OC)=O)C2)C)ccc2nnn(O)c2c1 c1(CCC(=O)OC)nc(-c2cccs2)no1.N1(CCO)CC1 c1(C(C)(C)C)ncc(C(=O)NCC(C2CCC2)NC(c2n[nH]cc2Cl)=O)cn1 C1(NC(N(C)C)=O)CCN(Cc2cn(CCOCC3CCOC3)nn2)C1 c1(C(N2CCC(CCNC(C3C(C#C)C3)=O)CC2)=O)c(F)cc(C)cc1Cl C1(C(N(C2(C)CC2)C)=O)CC(C)(C)CN1C(C1OCCC1(C)C)=O N1(C(C(CC#C)O)=O)CC2C3CCC(C(NC(c4cncc(CC)c4)=O)C3)C2C1 C1(CNC(c2n(CC)nnc2)=O)CCCCN(C(C23CC(CC(C)O2)C3)=O)C1 c1(C(N2CC(C(C)C)C2)=O)cncc(CNC(=O)C(c2cncnc2)C)c1 C1(C(=O)OC)CN(Cc2cccc(NCc3cccnc3)c2)CC1c1cccs1 C12(NC(c3cc(CC4CC4)cs3)=O)CCCC1CN(C(C1CC3CCC3C1)=O)C2 C(=O)(C(C)CCCOC)N(CCCNC(C1(C=C)CC1)=O)C1CC1 N1(C(C2(OC)CC(C)C2)=O)CCCC(CC(N2CCCC(N(C)C)C2)=O)CC1 C1(C(=O)NCCC(CNC(C(CCCC)C)=O)(C)C)CCc2c(ncn2C)C1 C1(NCCCCCC=C)CON(C(=O)OC(C)(C)C)C1 C1(F)(CNC(C2(C(C)C)CC2)=O)CCC(CNC(=O)CCCc2ccccn2)C1 c1(CC(=O)N(CC(C)N(C)C(c2cccc(CC#N)c2)=O)C)ccc(F)c(Cl)c1 CC(N=c1nc(N(C)CC2CC2(F)F)c2c([nH]1)COC2)c1ccoc1 N1(C(C(OCC)OCC)=O)CCC(C)(NC(c2ccn(C(C)(C)C)n2)=O)CC1 C1(OCCNC(C2CCN2C(=O)CCc2ccoc2)=O)CC1(F)F Cc1cc(F)c(F)cc1NC(=O)CN1CCN(C(c2cnc(Br)o2)=O)CC1 C1(C(=O)OCC)CCCC12CCN(C(c1ccc(OC)cc1)C(=O)NC(C)C)C2 c1(NCCCN(C(CC(C)CC(C)(C)C)=O)C)nc(Cl)nc2cnn(C)c12 CN1CCN(C(=O)Nc2sccc2I)CC1c1ncc[nH]1 N1(C(CCN(C(C)C)C)=O)CCC2(CC2C(=O)NCCNC(N2CCCC2)=O)C1 C12(CNC(CNS(N)(=O)=O)=O)CCC(NC(C3CC3C(N)=O)=O)(CO1)C2 C1(C)(NC(C2C(=C)C2)=O)CCN(C(c2oc(CO)cc2C)=O)CC1 N1(CC2CC(C)SCC2)C(=O)CN(CC2C(c3ccccc3)C2(C)C)C1=O c1(CN2CCN(S(=O)(=O)CC3CCC3)C3C2C3)c(F)cc(I)cc1F Cc1cnc2n1CCC(NC(C1(n3cccn3)CN(C(=O)CN)C1)=O)C2 CCCC(C(=O)N1CCCC1CNC(=O)CC1CC2CC2C1)N(C)C c1(C(N2C3CN(C(c4nccc(Cl)c4O)=O)C(C3)C2)=O)ccc2c(c1)CCO2 CC1=NOC(C(=O)NC2CCN(C(c3[nH]nnc3C)=O)C2)C1 C1(CNC(C2=NNC(=O)C2)=O)CCC2CN(C(=O)CC3CS(=O)(=O)C3)CCC2C1 C(CC(=O)N1Cc2ccccc2CO1)NC(C1(C)CCCO1)=O c1(C(C)C)ccc(C=CC(=O)N(C2CCN(C(C3CCCN3C=O)=O)C2)C)cc1 Cn1ncc(CNC(C2CC2(F)F)=O)c1C(=O)NCCOCC(C)(C)O Cc1cc(C(=O)NCC(C)(C(C)C)NC(=O)Cc2ccc(Cl)cc2Cl)nnc1C C1(COC)(CNC(C2CCSC2)=O)CCN(C(c2cnn(C3CCCC3)c2)=O)C1 c1(N2C(=O)CC(C(=O)NC(C(=O)OC)CCN(C)C)C2)ccc(OC)c(Cl)c1 c1(C(=O)NC2CC(NC(C3CN(CC)C(=O)N3)=O)C2)cc(C)c(O)c([N+](=O)[O-])c1 c1(C(=O)NC(C)CCNC(=O)CSc2nc[nH]n2)c(O)cc(Cl)cc1F Cn1c(C(N2CCCC2CC(=O)NCCc2nn[nH]n2)=O)cc2ccccc12 c1(N2CCCC(C)(N(C)C)C2)[nH]c(=NCc2nc(CO)cs2)nc2sccc12 CCC(C)C(C(=O)NC12CC1CN(C(=O)COCCF)C2)N(C)C c1(C(=O)NC2CCN(C(C3CCCC4CC34)=O)CC2F)cc2ncccc2[nH]1 C1(CNC(C2CC2(F)Cl)=O)CCN(C(=O)CCOC2CC2)CC1C1CC1 C#CC12CCC(C(N3CC4CCC3C4NC(=O)CCCCCC=C)=O)(CC1)CC2 C1(CC(=O)NCCN(C(C)C)C)CCCC1NC(=O)CSCCC#N C(=O)(C(C)CC(=O)OC)NCC1(F)CCC(NC(CCC#CC)=O)C1 C1(CNC(CC(CC)C)=O)CN(C(=O)Cc2cc(C(=O)OC)cs2)CC1(C)C c1(C(N2CC(C)C(NC(C3CC(N(C)C)C3)=O)C2)=O)c[nH]c2c(Cl)cccc12 c1(OC)ccc(C(N2CCN(C(=O)Cn3ccc(Br)n3)C3CC23)=O)c(O)c1 CC1CCCC=C1C(=O)N(C)CC1(O)CN(C(=O)COc2ccccc2)C1 N1(C(c2c(C)cccc2)=O)CC(C2CCCCN(C(C3CCCS3)=O)C2)C1 N1(C(=O)NC(c2cscn2)C)CCn2cnc(C(=O)O)c2C1 C(C)(C)(CC(=O)NCCCCC1CN(C(=O)C(c2cccc(F)c2)C)C1)SC C(=O)(C(CNC(=O)CCc1ccncn1)CC1CC1)NC(c1cncnc1)C S(=O)(=O)(c1cnccc1N1CCCC(C#N)C1)N1CCCC(CC(=O)NC)C1 Cc1ccc(C(=O)NC2CN(C)C2)c(-n2cc(C(c3ccc(Cl)cc3)O)nn2)c1 C1(C(=O)NCc2ccc(CC)s2)CCCN(C(=O)Cc2sccc2Cl)C1 c1(CNc2cccc(C(=O)NC(C)CO)c2)ccc(O)c2ccccc12 CC1(C)CN(CCC(F)C(=O)O)CC2(CN(C(=O)OC(C)(C)C)C2)O1 C1(C)(C(N2C(C(=O)NCC(C)NC(=O)OC)CCC2)=O)CNC(=O)C1 Cc1cc(C(N2CCC(OCc3ccc(C)o3)C2)=O)n(Cc2ccccc2)n1 c1(OC)ccnc(C(=O)NCC(O)CNC(c2coc(SC)c2)=O)c1N c1(C(N2C(CNC(CC3C(C(=O)OC)CC3)=O)COCC2)=O)ncc(C)cc1C N1(C(C(C2CCC2)OC)=O)CCN(C(C2(C)CC2)=O)CC1 C(=O)(C1=CCCC1(C)C)N1CCC(NC(c2cnc(OC)nc2)=O)C12CC2 CC(C)(C#N)CCC(=O)N1CCC(CCNC(C2(C)CC2c2ccccc2)=O)C1 c1(NC(c2ncncc2Cl)=O)ccc(N2CC(OCCO)CC2)nn1 N1(C(CC2C(CC)C2)=O)CCOC(C(=O)NCCC2=CCOCC2)CC1 CC1(C)CCN(C(=O)C(O)c2cnc[nH]2)CC1NC(=O)CCOCC(F)F CCC(C)(CNC(C1(F)CN(C(C2CCC(F)CC2)=O)C1)=O)C(N)=O C1(C)(CNC(C(C)SC)=O)CCCN(C(=O)Cn2cc(C)ccc2=O)C1 N1(C2(C(N(CCN(C(C3CC(OC)C3)=O)C)C)=O)CC2)CCOCC1 c1(C(=O)NCC(C)NC(=O)C(C)(O)CC(F)(F)F)ccc2cccc(Cl)c2n1 C1(C)(C(N(C)CC2(N(C)C)CC2)=O)CCN(C(=O)CC2CCCC3CC23)C1 c1(C(=O)NCC(C)NC(c2cncc(C)n2)=O)sccc1S(=O)(=O)N1CCCC1 c1(C(N2CCC(N(C(C=CCOC)=O)C)C2)=O)ccc(NC2CC2)nc1 C(CC(C(=O)NCC=CCNC(=O)Cn1nnc(=N)[nH]1)OC)OC n1(CCCC)nc(C(=O)NCC2CC2NC(=O)CC(=O)NC2CC2)ccc1=O C1(C(=O)NCC(CN(C)C(c2csc(C(F)F)n2)=O)O)Cc2cc(Cl)ccc2O1 N1(C(c2ccc(CN(C)C)cc2)=O)CCN(C(=O)Cc2ccn(C)n2)C(CO)C1 C#Cc1cccc(C(N2CCCC(C(=O)NCC(C)C(F)F)CC2)=O)c1 c1(OC)cc(C(=O)NC(CNC(c2nc(C)oc2C)=O)CO)ccc1[N+](=O)[O-] C1(NC(C2(C)CC(=C)C2)=O)CC(C(=O)N2CCSC(C)C2C)=CC1O C1(CN(C(C(F)=CC)=O)C)CCCN(C(C2CCCCS2)=O)C1 N1(C(Cc2ccc(C)s2)=O)CC(CNC(C2CCCS2)=O)CC(C)C1 C(=O)(CCCCCNC(=O)CCC1CC1)N(CC(CCC=C)O)C c1(NCC(CNC(c2cc(SC)ncc2)=O)C)nc(C(F)(F)F)ccc1C#N c1(C(N2C(C)C(NC(C3CCC=CCC3)=O)CC2)=O)c2c(c[nH]c1=N)CCC2 c1(C(=O)NC(CNC(=O)CNC(N2CCCC2)=O)C2CCC2)cnnc(O)c1 C1(C2C(CC(=O)N(CCNC(C3CC(CC)C3)=O)C)C2)CCCCO1 c1(N2CCN(Cc3ccc(C#N)nc3)C3C2C3)ncc2ccc(F)cc2n1 N1(C(CSCCN(OCC)CC)=O)CCC2CN(CC(=O)NC3CCCC3)CC12 N1(C(C(C)O)=O)CCC2C(CCCN2C(=O)C(c2ccccn2)O)C1 C(=O)(C1=CCCOC1)N1CC(F)(CNC(=O)CCCn2cncn2)C1 c1(C(=O)NC2CC(N(C(C(C)OCCOC)=O)C)C2)sccc1C C12(C(N(CCCNC(C(CC(C)C)F)=O)C3CC3)=O)CCCCCC1OCC2 C1(CC(N2CCC(N(C(CCNC(C)=O)=O)CCOC)C2)=O)C=NN(C)C1=O c1(C(C)C)cc(C(N2CC(CCNC(=O)CC(C)(F)F)C(C)C2)=O)ccc1F N(C(=NCCC=C)NC1CCC12CCC2)C1(CC=C)CC1 c1(C(N2CCC(CCNC(C(C(C)(C)C)SC)=O)C2)=O)ccc2nc(C)cn2c1 N1(C(c2c(C)sc(Br)c2)=O)CC2(CCN(C(C3(NC(N)=O)CC3)=O)C2)C1 Cc1nc(C)n(CC(=O)NC(C(=O)NC(c2ccco2)CO)C2CCCO2)n1 C(=O)(CCCCCC1CC1)NC(C1CCCN1C(c1cn(CCN(C)C)nn1)=O)C N1(C(C2(C(=O)OCC)CC2)=O)C2CCC1CN(C(=O)CC1CCC13CCC3)CC2 Cc1cc(N(C)CC2CCOCC2)nc(=NCC(C)c2ccc(Cl)cc2)[nH]1 c1(C(N2CCCC(CC(=O)NCC(C)OC(F)F)C2)=O)cncc2[nH]ccc12 C1(C)(C(N2CCC(NC(Cc3c(C)ocn3)=O)(CO)C2)=O)CCCCNC1=O N1(C(C23CC(NC(C(n4c(C)ncc4)C)=O)(C2)C3)=O)CC2(CNC(=O)C2)C1 C1(C(N(C)CCN2CCCC2=O)=O)CCN(C(=O)Cc2cccnc2O)CC1 C1(CC=C)(NC(C2(CNC(=O)C(O)C=CCCC)CCCC2)=O)CCCCCC1 c1(C(=O)NCc2sc(C(=O)OC)c(C)c2)n[nH]c2ccc(-c3nn[nH]n3)cc12 c1(C(=O)NC(C(C)C)CNC(=O)CC2CC2(C)C)cc(F)cc(Br)c1O C(CC(C)C(=O)NCC(O)CNC(c1onc(C)c1C)=O)=CCC N1(C(C2(C)CCCC2)=O)CCCC(C2CCN(C(=O)CC3CCCOCC3)C2)C1 CN(C1CCc2cc(F)ccc21)C(=O)CC1CC(=O)C1 N1(C(c2ccc(C(C)C)s2)=O)CCC2CN(C(c3cccn3C)=O)CCC2C1 Cc1ccc2c(c1)C(C(=O)N1CC(C(C)(C)O)(CNC(C3CC(F)(F)C3)=O)C1)C2 C=CC(C)(C)C(=O)NC1CC(NC(c2cnn(C(C)CC)c2C2CC2)=O)C1 C1(NC(c2ccc(Cl)o2)=O)CCCCCCC1NC(c1ncnc2cc[nH]c12)=O Cn1cc(C(=O)NCCN2CCN(C(C3CCC(C)(C)C3)=O)CC2)cc1Br CCCS(=O)(=O)CC(=O)N1CCC(NC(=O)CC2CC3(CC3)C2)C(SC)CC1 N1(C(C2(CC#C)CC2)=O)CCN(C(=O)C(C2(O)CCCC2)F)CC(O)C1 c1(C(N(C2CN(C(CSCc3ccc(C)cc3)=O)C2)C)=O)ccc2c(c1)COC2 c1(C(=O)NCc2ccc(CNC(C3C(C)CCS3)=O)cc2)cccc2cncn12 C12(Nc3nc(C)nc(C(F)(F)F)c3)CCCC1CN(C(c1cn(C)cn1)=O)C2 c1(CC(C(=O)NCC(CC)(C)NC(c2cc(C3CC3)[nH]n2)=O)O)ccc(Cl)cc1 C1(C(=O)NC2(CC=C)CCN(C(=O)Cc3cnns3)C2)CCn2ccnc2C1 C12(NC(C(N3C(CC)CCC3)=O)=O)CCC1CN(C(=O)Cc1ccc(F)cn1)C2 N1(C(C(CC)O)=O)CCC2(CC1)CN(C(=O)CS(=O)(=O)CCO)CC2CO c1(OC)ncc(F)c(N2CCCC(C(N3CCC(C(F)F)CC3)=O)CC2)n1 C1(NC(CS(CC)=O)=O)(CO)CCCN(C(c2cc(SC)c(C)o2)=O)C1 c1(CC(C(=O)N(CC(C)NC(COCCC=C)=O)C)O)c(F)cccc1Cl O=C(CCCCCO)N1CC2(CC2C(=O)NCC(F)CO)C1 C1(C(N(C(C)CCNC(=O)CSC(=N)N)C)=O)Cc2ccccc2CO1 C1(CC(=O)NC2(CNC(c3cc(OC)c(O)nc3)=O)CC2)CCCC2(CCC2)O1 Cc1cc(=O)n(CCC(=O)NCC2CCC(F)(CNC(=O)C(C)(C)CO)C2)cn1 c1(CCNC(c2ccncc2Cl)=O)ccc(CNC(C23CCC(C2)C3)=O)cc1 c1(C2(C(=O)NCCC3(O)CN(C(=O)C=C4CCC4)C3)CC2)ccc(F)cc1F CCC(C)C(C(=O)NCCc1cn(C)nn1)NC(=O)C(CSC)OC c1(C(N(CCN(C(C2C(C)C2)=O)C)C(C)C)=O)cccc(-c2cccc(Cl)c2)c1 c1(C2CN(Cc3c(C)nn(C4CCC4)c3)C2)cc(F)cc(Br)c1 c1(C(N2C(CNC(C3CC(F)(CO)C3)=O)CC(OC)C2)=O)cc2cccnc2o1 c1(C(N(CCCOCCOC)C)=O)cc2nc(C)cc(C(F)(F)F)n2n1 c1(C(=O)NCCC2(C)CCN(C(C)=O)C2)ccccc1S(=O)C(F)(F)F C1(N(c2cc[nH]n2)C(c2cccnn2)=O)CCC12CCNCC2 c1(OC)ccc(C)c(C(=O)NCC(C)(C)CNC(=O)Cn2cc(C)ccc2=O)n1 c1(C(N2CC(NC(C(C)(C)OC)=O)C2)=O)c(I)cnn1CCF C=CCCCC(C(=O)NCCC(F)(F)Cl)NC(C1CCCCC1(C)C)=O CC1C(NC(=O)CS(=O)(=O)N(C)C)CCCN1C(c1nc(Cl)ccc1N)=O N1(C(=O)CCOC2CC2)CCC2(C1)CN(C(c1cc[nH]c1)=O)C2 S(=O)(=O)(c1ccc(N2Cc3ccncc3C2)cc1Cl)NC(c1cn(C)cn1)C c1(C(C(=O)NC(C2(O)CN(C(C(C)OCCN(C)C)=O)C2)C)O)cccc(F)c1 C(=O)(CCCC(C)(C)NC(=O)C(C1CC1)SC)NC(CC#CC)C C(=O)(CC(C)C(=O)NCCOC1CCN(c2ccnc(C(C)(C)C)n2)C1)OC c1(C(N(CC(=O)OC(C)C)CC(=O)NC2CC2)=O)cnn2c1CN(C)CC2 c1(C(=O)NC2CCCC(NC(CC3C(C)CCC3)=O)C2)ccc(O)c(F)c1 C1(C(N2CC(OC)C(OC)C2)=O)CCC(N=c2nc(N(C)C)c3nc[nH]c3[nH]2)CC1 c1(C(=O)NCC)ccc(NC2CCCC2CNC(=O)CCCCC2CC2)c(C)c1 Cc1ccn(C(C)C(=O)NC2CC(C(=O)NCC3(CC(N)=O)CC3)C2)n1 c1(CC(=O)NCC(COC)C)cc(Cl)ccc1C C(=O)(C1=C(C)OCCS1)NC1(CC=CC(=O)NC2C=CC(CC)C2)CCC1 C1(CNC(CCC=C)=O)(CO)CCCN(C(=O)C(C2CC2)OCC)C1 C(N=c1[nH]cnc2[nH]ccc12)C1CCC(NC(=O)CC2CCCCC2O)C1 C1(C(N(C)CC2(CC3CC3)CC2)=O)CCCC12CCN(C(C1(C)CCC1)=O)C2 C1(C(C(N2CC(C(=O)OC)(SC)C2)=O)C)CCCN(C(c2csnn2)=O)C1 N1(C(C2(CC)CCCC2)=O)CCC(F)(F)C(C(=O)NC)C1.c12nccc(n1)CN2 C(=O)(CCCS(C)(=O)=O)N1CC(CC(CNC(C2CN(C(C)=O)C2)=O)(C)C)C1 N1(C(c2cn(CC)nn2)=O)CC2CC(C(=O)NCCCc3cnccn3)CC2C1 C(=O)(C1CCc2ccccc21)N1C(CN(C(c2ns[nH]c2=O)=O)CC)CCC1 C1(O)(CN(C(c2cnc(CC)s2)=O)C)CCN(C(=O)C=C2CCC2)C1 c1(C(N(CCC(C(C)C)NC(=O)C#CC(=O)N(C)C)C)=O)cccn2ncnc12 N1(C(C(C)(CO)NC(C(CCCC#C)C)=O)=O)CC2(CCC(O)CC2)C1 N1(C(CC=C)=O)CC2CC1CN(C(=O)C=CC1CCOCC1)C2 c1(N(C)C)ccc(C(=O)NCCC2(CNC(=O)C=CC3CC3)CC2)cc1 CC(C)(CO)C(=O)NCC(CO)NC(c1csc(-c2ncccn2)n1)=O C(=O)(C(C#N)(CC)CC)NC(CCC)CNC(c1csnc1Cl)=O c1(N2CC3C(C)C3C2)[nH]c(=NCCC2CCCCO2)nc2scnc12 C1(CNC(CN(C)S(N)(=O)=O)=O)CCCCCN1C(c1cc(=O)cc(Cl)[nH]1)=O c1(C(=O)NCCOCCn2cc(-c3c(C)ccs3)nn2)ccc(C(C)F)cc1 O=C(C1=CCCOC1)NC1CC(CNC(c2cnn(C3CC3)c2Cl)=O)C12CCC2 C1(C(=O)NCc2cnc(C)o2)CCN(C(=O)C2CCC3(CCC3)C2)O1 C1(CNC(=O)C(=CC2CCCCC2)F)C2CCC(C2)N1C(c1cc(CO)on1)=O C1(C#CC(=O)NCC(C)CN(C(=O)C=Cc2ccc(Cl)cc2)C)(CC)CC1 N1(CCC(=O)NC2CN(C(=O)C(O)C3CCC3)C2)CCCCC1=O CC#CCC(C(=O)NCC(C)C(C)CC)NC(c1n[nH]c(C)c1Cl)=O N1(C(C=C2CCC(C)C2)=O)CCCC2(NC(=O)CSc3n[nH]c(O)n3)CCCC12 c12ccc(Br)cc1C(=O)O2.N1(CCSC2(OC(C)C)CCCC2)CCN(C)CC1 CC(C)C(C)C(C)CC(=O)N1CC2CC1C2NC(C1CCN(C)C1=O)=O C1(NC(C=Cc2nnc(C(C)C)o2)=O)CCN(C(=O)CSC2CC2)CC1O C#CC1CN(C(C2CCC(=O)N2)=O)CCN1C(=O)CCC1CC1(F)F c1(C(N2CC(C=C)C(NC(C3CNC(=O)N3)=O)C2)=O)nnc2ccccc2c1N C1(CNC(CC=C=C)=O)CN(C(=O)C(C)Cc2cnc[nH]2)CCCO1 c1(C(=O)NCC2(C)CCN(C(C=CCOC)=O)C2)cccc([N+](=O)[O-])c1Br C1(C(NOCCCN(C)C)=O)CCCCC1NC(C1CC(=O)CCO1)=O C=CCCCC(C(=O)N1CC(O)(C(=O)NC(C(=O)C(N)=O)C)C1)NOC c1(OCC=C)ccc(C(N2CCC(O)(CN(C(=O)CCC(=C)C)C)C2)=O)cc1 C1(CC)C(C(=O)NC(COC)C2CC2)CCN1C(c1nnsc1C)=O Cc1ccc2n[nH]cc2c1C(=O)NCC(O)CN(C(=O)C(F)(F)C(C)O)C c1(C(=O)NC2C(NC(c3csc(CO)n3)=O)COC2)c[nH]c2ccncc2c1=O C12OCCC1NC2.C(C(F)(F)F)N(CCNC(C1CC1C(C)(F)F)=O)CC C=CCCC(C)C(C(=O)NCC1CCOC1)N1CC(C)OCC12CCC2 C(CN=C(NCc1cnccc1C(F)(F)F)NCC1CC1(F)F)OCC=C CC(=O)CCCC(=O)N1CCC(c2ccccc2)(CNC(c2cncs2)=O)CC1 C1(OC)CN(C(=O)Cn2ccc(C(F)(F)F)n2)CC1NC(C1CN(C(C)C)C1)=O c1(C(=O)NCC(C)(C)NC(c2n(C)cc([N+](=O)[O-])c2)=O)ccn2c(O)nnc2c1 N1(C(Cn2ccc(C)cc2=O)=O)CCC2CCC(C1)N2CC1CCS(=O)(=O)CC1 c1(OC)ccc(C(=O)N(C2CCCC2)CCNC(=O)C2=CCCC2C)cc1F c1(CC)cccc(C(N2CC(CO)(NC(=O)C=Cc3ccc(Cl)cc3)C2)=O)c1N c1(C(=O)NC(CCOC)CNC(=O)CCCc2nccs2)cnc(=N)[nH]c1 C1(CC(N2CCC(N(C)C(c3ccoc3C(F)(F)F)=O)C2)=O)CCC(=O)NC1 C1(C(N2CC(CNC(c3cncc(C(F)F)c3)=O)C(C)C2)=O)(CC)CCOCC1 Cc1ccc(CN2CCC(N(C)C(c3ccc(-c4cc[nH]n4)s3)=O)C2)cc1 N1(C(c2n(CC=C)ccc2)=O)CCCCC1CCNC(C1CC1OC(C)=O)=O c1(C(=O)NC2C(OC)C(O)C2)c(CNC(C23CSCC2C3)=O)nnn1C C1(OCC(=O)NC(C=C)C2CC2)CCN(C(c2csc(O)n2)=O)C1 c1(-c2nc(C3N(CC)CC(C#CC)OC3)on2)cc(CC)cc2ccoc12 c1(OC)cc(CC(=O)NC2CCCN(C(c3nccnc3N)=O)C2C)cc(F)c1 C1(NC(COCCSC)=O)CC2(CCN(C(=O)C(C(C)C)c3ccncc3)C2)C1 C1(CC(=O)NC)(CNC(=O)N(C(C)C)Cc2cncc(C)n2)CCCCC1 N1(C(CCP(C)(C)=O)=O)CCCC12CCN(C(c1cc(CC3CC3)on1)=O)CC2 c1(C(=O)NCC2CC(=C)CN2Cc2cccc(O)c2C)ccc(OC)c(O)c1 C#CCCCCC(=O)NC(CCC)CCCNC(=O)Cc1cccnc1OCC C(=O)(CC(=O)NCC(c1ccccc1)N(C)C(c1[nH]nnc1COC)=O)OCC n1(CC(=O)N(CC(C)O)CCNC(=O)CCCc2ccsc2)cccnc1=O c1(C(N2CCC3(NC(C=CSC)=O)C(C2)C3)=O)sc2ccccc2c1Cl c1(C(C)C)ncc(C(=O)NC(CNC(c2cnnn2C)=O)Cc2ccccc2)s1 C12(C(N3CC(C)C(N(C)C)C3)=O)CC(CO1)N(C(=O)CC1(O)CCCC1)C2 C(=O)(C(CC)C(=O)N(C(C)C(N1CCN(CC(N)=O)CC1)=O)C)OC C1(NC(C2CCC(CNC(CCCNC(=O)OC)=O)CC2)=O)CCC(C)NC1=O c1(C(N(CC(CNC(C(=O)N(C)C)=O)(C)C)C)=O)cc(C(F)(F)F)cc(Cl)c1 C1(C(=O)NCCN(OC)C)CN(C(C23CC(C#N)(C2)C3)=O)CC1C c1(N2CC(CNC(CC(CCC)CC)=O)C(F)(F)CC2)ncc([N+](=O)[O-])cc1F N1(CC(=O)NC(C)CC2(O)CCC2)CCN(C(C2COCCO2)=O)CC1 C#CCC(CC#C)C(=O)N1CC2(CC2)CC1CNC(C1(C2CC2)CC1)=O N1(C(c2nc(CC)oc2)=O)CC(C)(C)OCC1CNC(c1csnn1)=O c1(OC)ccc(CN=c2nc(C3(C)CC3)o[nH]2)cc1C Cc1cc(F)cc(C(N2CCC2CNC(=O)CSc2nncs2)=O)c1C CC1(CC(N2CCOCC(NC(C3CCCCC(=O)N3)=O)C2)=O)CCCCCC1 C1(CNC(c2c(COC)ncs2)=O)C2CN(C(C3(C)CCCCC3)=O)CC12 C1(CCNC(=O)CC2(O)CCC2)CN(C(=O)C(O)CN(C)C)CCO1 C=CCC(C)C(=O)NCCN(CCOCCO)C(c1coc(C2CCCC2)n1)=O CC1=C(CNC(=NCC(C)c2ccc(Cl)cc2)NCC2CCC2)S(=O)(=O)CCO1 N1(C(c2n(CC)ccn2)=O)CCC(C2(NC(=O)CCc3cncc(F)c3)CC2)C1 C(=O)(C(CCCCC1CC1)N(C)Cc1ccc(Cl)s1)NCCOC C(C(C)(C(=O)NC1CN(C)NC1=O)NC(c1cccc(CO)c1)=O)SC Cc1nn(C)c(C)c1CC(N1CCCC1C(=O)Nc1cscn1)=O c1(C(=O)NCC(C)NC(C2(NC(C)=O)CCC2)=O)cc2ncn(C)c2cn1 Cc1cnc2c(C(=O)NCCC3(NC(=O)CC4CCCCN4C)CC3)cnn2c1 N1(CC(=O)N2CC2=O)Cc2c(F)ccc(F)c2C1.C(C)(C)(C)SCCOC CCCC(C#N)C(=O)NC(CC1CC1)C(=O)NCc1ccnc(F)c1 c1(C(=O)NCC(C)(C2CC2)NC(C(C)c2cccs2)=O)nccc2ccncc12 C1(C(=O)NC(C)CCNC(=O)CCSc2ccccc2F)CCOC2(CCC2)C1 c1(C(N2CC(NC(C3C(C(C)C)C3)=O)C(N=[N+]=[N-])C2)=O)c(N)c(F)cc(F)c1F c1(-c2n(-c3ccc(F)c(Cl)c3)nc(C(F)F)n2)ccc2ncccc2c1 c1(C(=O)OC)ccc(C=CC(=O)NCCN(C(=O)CCCCN2CCC2)CC)o1 c1(C(=O)NC2(CNC(C(CC=C)C)=O)CCC2)cc(C)cc2c(C)ccnc12 c1(OCC)ccc(Br)cc1NC(C1CC1CNC(c1cc(OC)ccc1I)=O)=O C1(C(=O)NC2C(CNC(COc3cn(C)nc3)=O)CC2)CC2C=CCC(C1)C2 c1(C(C(=O)NCC=C)N(CC)Cc2cn(C)nn2)ccc(-n2cc(Cl)cn2)cc1 C=CCC(F)(F)C(=O)NCC(C)C(F)C(=O)N1CC(CO)(CF)C1 C1(CN(C(=O)Cc2cccs2)C2CC2)CN(C(=O)CSCC2CCOC2)CC12CC2 N1(C(C2C(CNC(C3N(CC)CCCC3)=O)CC2)=O)CCC2(CNC(=O)C2)C1 C=CCCCCCCC(=O)NC(CNC(c1sc(C)cc1C)=O)C1CCC1 N1(C(C2C(NC(c3c(C)scc3)=O)CCC2)=O)CC2COCC2C1 C(=O)(C(C(C)NC(C1CCN(OC)CC1)=O)C(C)C)N1CCC(O)(CC=C)CC1 C(=O)(C(C(C)C)N(C)C)NCCC(=C)CNC(C1CCN(S(=O)(=O)CC)CC1)=O C#CCCC(O)C(=O)N1CCC(CO)(NC(c2cc(C)ncc2C)=O)CC1 Cc1cccc(C(C)NC(C2(CNC(=O)CCn3cccn3)CC(C)(C)C2)=O)c1 C(C(C(=O)N1CCCCC1CN(C)C)C(C)C)NC(COCC=C)=O Cc1c(C(=O)NCCC(C)NC(c2c[nH]nc2C(F)(F)F)=O)oc2ccccc12 C=CC(F)(F)C(=O)N(C(C)(C)CC(=O)NCCP(C)(C)=O)C c1(C(=O)NC2C(CNC(C(CSC)C)=O)C2)ccc(C)c(C#N)c1 c1(C(=O)NCC2(CCNC(C3CCCC3)=O)CC2)nc(Br)n2ccccc12 C(=O)(C(C)(C)CC(=O)NCCCOCCNC(=O)CC(C)N(C)C)OC C=C=CCCC(=O)N(C)CCNC(=O)CC1CC(=O)NC1=O C1(CNC(C2N(C(C3(OCC)CCC3)=O)CCCC2)=O)CCCC12CCC2 C1(C(N2CCC(C(N3CC(C(=O)OC)C3)=O)C2)=O)CCCN(C(=O)C2CC2)C1 c1(N2CCC(NC(CCn3cc(COCC)nn3)=O)C2)ccc(Br)cc1 C1(NC(c2c(COC)ncs2)=O)CCC(N(C(=O)CC2CN(C)CCO2)C)CC1 C(=O)(CC(O)CC(C)(C)C)N1CC(CN2CC(O)(C(C(=O)OC)F)C2)OCC1 CCCCCCC(=O)NCC1CC(F)(CNC(=O)C(=Cc2ccccc2)CC)C1 Cc1cc(F)cc(C(=O)NCc2cccc(-n3cc(CNS(N)(=O)=O)nn3)c2)c1C c1(NCC(CCC)OCC)[nH]c(=NCC(C)(C)C2CC2)nc2c1cnn2C(C)C C1(c2n(CC3CC(OC)C3(C)C)nnn2)(Nc2ccccn2)CCS(=O)(=O)CC1 c1(CN(CC(N2CCC(C(C)NC(C(C)=C3CC3)=O)C2)=O)C)nnc(C)n1C C1(C(=O)NC(C=C)C2CCC2)C(O)CCN1C(=O)C(C1CC1)OCC C(=O)(C(C)CC(F)(F)F)N1CCC(O)(CN(C(Cc2cn(CC)nc2)=O)C)C1 C=C1CC(C(=O)OC)N(C(C2CCN(C(c3ccc(C)s3)=O)CC2)=O)C1 C1(C(=O)NCc2cn(CC=C)nn2)CC12CCN(C(c1ccc(CF)cc1)=O)C2 N1(C(C2C(C)C2C)=O)CCC(C2(NC(=O)Cc3nncs3)CC2)CC1 n1(CC)ncc2c(NC3CC(NC(C4CCC5CC(C)CN5C4)=O)C3)ncnc12 n1(CCOC)cc(NC(c2conc2CNC(C2CCC(O)C2)=O)=O)cn1 C1(CNC(COCCC(C)C)=O)CCC2CN(C(C3CCCN3C)=O)CCC2C1 C1(N(C(c2ccn(CCC)n2)=O)C)CN(C(c2cn(CCO)nn2)=O)CC1F C1(C(N2CC(NC(CC3C(C)(C)COCC3)=O)(CO)C2)=O)CNC(=O)CC1(C)C C1(NC(c2cnc(CC)o2)=O)CCN(C(c2cccc(SC(C)C)c2)=O)CC1C N1(C(c2nc(CC)[nH]n2)=O)CCCC(C(N2CCC(C(=O)O)CC2)=O)C1 c1(CC(=O)OC)occ(C)c1C(=O)NCCN(C(=O)Cc1nonc1C)C(C)C C1(C(N)=O)Cc2cccc(NC(=O)C(c3cc(Br)ccc3Cl)N)c2C1 N1(C(CC2CC3(CN(C(c4cc[nH]n4)=O)C3)C2)=O)CC2CCCCCCC12 Cc1cc(C(N2CCC(NC(c3cc4c([nH]3)CCC4)=O)C2C)=O)cnc1C(F)F CN1CC(C)(C)CC1C(=O)NC1CC(CNC(=O)CCC2CC2(Cl)Cl)C1 c1(NCC(CNC(C(C)CSC(F)(F)F)=O)O)ncnc2ccc([N+](=O)[O-])cc12 C1(C(N(C)CCc2cccc(C#N)c2)=O)CCCCC1(C)C C12(NCCCN3C(=O)CCC3)CCC(CC1)N(C(=O)CN1CC3CCC1C3)C2 C1(N(C(=O)CCNC(=O)Nc2ccccn2)CC)CCCN(C(=O)CCC(C)C)C1 c1(C(=O)NCc2ccc(OC)cc2Cl)ccc(OC)c(OC)c1Cl N1(C(C(C)(C)C2CC2)=O)CCC(C(F)(F)F)C(CNC(C2(C)CCC(=O)N2)=O)C1 N1(C(C2CN(C)C2)=O)CCCCC(C2CN(C(C3CCCN(C(N)=O)C3)=O)C2)C1 CC1CCc2[nH]c(=NCc3nncs3)[nH]c(=NCCCCN3CCCCCC3)c2C1 C1(CNC(CSc2c(C)n[nH]c2C)=O)CN(C(=O)C=CCN(C)C)CCC1(F)F c1(CC(N2CC(NC(c3coc(CC4CC4)c3)=O)C2)=O)csc2ccccc12 C1(NC(CC(CC)C)=O)CCN(C(c2ccc(CN3CCCC3)o2)=O)CC1(C)C N1(C(Cc2c(C)con2)=O)CCN(C(=O)C(c2c(C)noc2C)C)C(CO)C1 c1(C(=O)NCCC2N(C(COC(CC)CC)=O)CCCC2)ccnc(F)c1OC c1(OCC)ccccc1N(C(c1scnc1Br)C(=O)NC)C C1(C(=O)NCc2ccc(C)s2)CC12CCN(C(=O)Cc1cnn(C)c1C)C2 N1(C(=O)NC2CC(COC)C2)CCC(N2CCNS2(=O)=O)CC1 CCCCCC(CC)C(=O)N1CCCC(C)(NC(c2cn(C)c(C(F)F)n2)=O)C1 C1(C(N(C2CC2)CC2N(C(CC3CC(CC)C3)=O)CCC2)=O)CCC(F)(F)C1O c1(OCC(=O)NCCC(C)NC(C(CC)n2ccnc2)=O)ccccc1C(F)F c1(C(=O)NC(CCC)CNC(C2(N3CCCC3)CC2)=O)ccnc(OC)c1 N1(C(C2(OCC)CC2)=O)CCCN(C(c2[nH]nnc2C(F)F)=O)CC1 c1(C(N(CCC(C(C)C)NC(CC(C=C)CC)=O)C)=O)cc2cnn(C)c2s1 c1(CCNC(N2CC3(CN(CC)C3)C2)=O)c(F)ccc(F)c1F c1(C(=O)NC2CC(C)N(CCn3cccn3)CC2)coc2ccccc12 CC(C)(CC(=O)NCC(CC(F)(F)F)NC(=O)C1CCc2nccn21)C(F)(F)F N1(C(c2c(C)onc2)=O)CCC(C)C(NC(c2cc3sccc3s2)=O)C1C c1(CC(N2CC(CCNC(C(C3CCOC3)OC)=O)C2)=O)ccccc1C CN1CCN(C(=O)OC(C)(C)C)C(CNC(C2CC(Cc3ccccc3)C2)=O)C1 O=C1OCCc2ccc(NC(N3CCC(CO)C3)=O)cc21 N1(C(CN2CCC(=O)NC2=O)=O)CC(NC(c2occ3c2CCC3)=O)CC2(CC2)C1 Cc1nn(C)c(F)c1C(=O)NCC1(C)CCC(NC(C2(C3CC3)CC2)=O)C1 C1(N(CCNC(=O)CCF)C(c2cc(Br)cs2)=O)CCCCCC1 c1(CC(=O)N(C(CCNC(COCCCOC)=O)C)C)ccnc(F)c1 N1(CC)CCOC(C(N2CCC(C)C2CNC(c2cccn2C(C)C)=O)=O)C1 c1(C(N2C(CNC(C3CSCC(=O)N3)=O)CC(OC)C2)=O)coc2c1COC2 c1(C(=O)NCC2CC(NC(=O)CCCF)C2)ccc(S(=O)(=O)NCC2CC2)o1 C=CCCCC(C(=O)NC1CC(CC(=O)OC)C1)NC(c1ccc(F)cc1)=O C1(CNC(C2CCC(OC)C2)=O)CCC2CN(C(=O)COC3CC(F)(F)C3)CC12 N1(C(C(CC)N(C)CC)=O)CCC(C)(CNC(c2sc(COC)nc2C)=O)C1 c1(C(=O)NCC(CC=C)NC(=O)C(O)Cc2ccccc2)ccnnc1C C1(NC(Cc2c(C(C)(C)C)cccc2)=O)CN(C(C2CCOC2=O)=O)C(C)(C)C1 N1(C(CCC=C=C)=O)CCN(C(=O)CC2(O)CCC2)C(CCCC)C1 CC(CCO)C(=O)NC(C1CCN(C(c2cccc(NC(N)=O)c2)=O)CC1)C c1(CN2CCC(C(=O)NCC(F)F)C(O)C2)ccc([N+](=O)[O-])cn1 C(=O)(CCC(F)(F)F)NCCOCCCNC(C1CC1C1CC1)=O N1(C(=O)Cc2nc(C3CC3)cs2)CC2CC1CN2C(=O)Cc1nncs1 N1(C(C(c2ccc(CC)s2)=O)=O)CCN(C(=O)CC2CC2C(F)(F)F)C(C)C1 N#Cc1cc([N+](=O)[O-])ccc1NCCC1CCN(C(=O)CCS(N)(=O)=O)C1 C1(CC)CC(NC(C2CN(C(c3sccc3OC)=O)CC2F)=O)CCO1 C1(C(=O)Nc2ccc(O)nc2)CN(C(c2ccc(Cl)cc2I)=O)CCC1O c1(C(=O)NN(CC(C)O)C(C2C(COC)(CC3CC3)C2)=O)ccc(N(C)C)cc1 N1(CC(C)C)CC(C(=O)NCC2(NC(C3CNC(=O)N3)=O)CCC2)CC1=O CC1C(NC(=O)C2=COCCC2)CC2CCC1N2C(=O)CCC(N)=O CN1CCC2C(CCCN2c2nnc(-c3cc(Br)cnc3Br)n2CC2CC2)C1 CCC(CC)(CC)C(=O)NC1CC(NC(C2CC(O)CN2C(C)=O)=O)C(O)C1 N1(C(C(CC)CN(C)C)=O)CC2CCN(C(=O)C=C(C)Cl)CC2C1 c1(C(=O)NCC(CNC(c2cc([N+](=O)[O-])c[nH]2)=O)OC)ccc(Cl)c(Cl)c1 c1(OC)ccc2cc(C(N3CC4CC3(CNC(=O)C(F)OC)C4)=O)nnc2c1 c1(OC)cnc(Cl)c(NC2CCC(C)(NC(=O)OC(C)(C)C)CC2)c1 c1(C(C(=O)NC2(CO)CN(C(C3N(C(C)=O)CSC3)=O)C2)C)c(C)nn(C)c1C c1(C(=O)NC(CN(C(C2=C(C)OCC2)=O)C)C)nnn2c1CCCCC2 C1(C(N2CC(O)(c3cn(CCCF)nn3)C2)=O)CCNC2C1C2(F)F N1(C(C(=O)N(C(c2ccc(O)cc2)C)CC)=O)CCCCC1C c1(OC)ccc(C)c(CCNCC2(c3ccccc3)CC(O)C2)c1 CC1=C(C(=O)N2CC(C(=O)NC3CC(C(F)F)C3)C(F)C2)CC1 CCCCCC(=O)NC12CC(C(N(C[Si](C)(C)C)Cc3ccccc3)=O)(C1)C2 C1(NC(CCCOCCOCCOC)=O)CN(C(=O)CN2CCCC2)C2CC12 N1(C(C(C2CC2)SC)=O)CC(C(=O)Nc2cc(F)ccc2C)C2(CCC2)C1 C1(C(=O)NCCC(C)N(C(c2cnc(OC)c(C)c2)=O)C)CC2(C1)CC(C)(C)C2 C(=O)(C1=NN(C2CC2)C(=O)CC1)NC1(C)CCN(C(c2cncc(F)c2Cl)=O)C1 CCC(C)(C)CCNC(=O)C(Cc1cn[nH]c1)NC(=O)CC1CNC(=O)O1 C1(CC(=O)N(CC(C)C#N)C)CN(C(C2CNC(=O)N2)=O)C(C)(C)C1 C(=O)(C(CNC(c1ncnc(C)c1C)=O)C(C)(C)C)NCC1(CC(=O)OC)CC1 Cc1cnc(C(=O)N(C)CC2CCN(C(c3ccc(C(C)F)cc3)=O)C2)nc1 c1(C(=O)NC(C(C)OC(C=CC(=O)NC2CC2)=O)CO)ncccc1C(F)(F)F N1(C(C2C(C)CC(C)O2)=O)CCN(C(=O)CCN2CCCCC2=O)C2(CCC2)C1 C(C(C)CC(=O)NC(C(O)CO)C1CC1)NC(C1(COC)CC(=O)C1)=O CC1CN(C(C2C(O)CCN2C(C2CN3CCN2CC3)=O)=O)CCC1CO c1(C(=O)NCC(=O)NCC=C)sc(-c2ccccc2C)nc1C N1(C(C2CCC(CNC(c3n[nH]c(=N)[nH]3)=O)O2)=O)Cc2c[nH]nc2C1 Cc1ccc(CNC2CCN(S(=O)(=O)c3cn[nH]c3)C2)cc1O C1(CNC(CC=C)=O)CN(C(=O)COC2CCC(C)CC2)CC1C C1(C(=O)N(CCNC(c2cc(C3CC3)ns2)=O)C2CC2)(OC)CC(C)C1 Cc1cccc2c(CCC(N3CCC(CNC(C4C(C)C4C)=O)C3)=O)c[nH]c12 N1(C(C2C(OCC)C2C)=O)CCCC(C)(C)C1CNC(c1ccc(C)c(Cl)c1)=O c1(C(N(CCCNC(C2CCSCC2)=O)CC)=O)ccn(C(C)C)c1C c1(OC)ccc(COC(c2ccccc2C(C)=O)=O)cc1F C1(C(N(C(CC)C(=O)N(C)CC2(O)CCC2)C)=O)CC2C(C1)C2(C)C N1(C(CCCOCCC)=O)CCC(C)(NC(C2(C)CC3(CC3)C2)=O)C1 c1(NC)ccc(Cl)c(C(=O)NC2CC(C)N(C(c3cn(C)c(O)n3)=O)C2)c1 N1(C(C(CC)n2ccnc2)=O)CC2CC1(c1cn(CC3CCOC3)nn1)C2 c1(C(=O)NCC)cccc(C2CC2)c1C.c12ccc(nn1)N1CCN(CC1)C2.NCC c1(CCCC=C)ccc(C(=O)NCC2CN(C(C3CCCCS3)=O)CC2C)cc1 N1(C(C2CCN(C(=O)NC(CCC)C)CC2)=O)CCC2(C1)NC(=O)N(C)C2=O CCC(CO)C(=O)NCCC1CCCN(C(c2cccc(C(C)(C)C)c2)=O)C1 C(=O)(C(F)C(C)C(F)(F)F)N(CC(n1cc(C(=O)OC2COC2)nn1)C)C c1(C(C(N)=O)NC(N(CC=C)CCOC)=O)ccccc1 n1(C(C)C)cc(C(=O)NCC2(CNC(=O)CC3CCC(C)C3)CCC2)ccc1=O N1(c2nc(C)c(Br)cn2)CCC2(CCN(C(=O)C(C)(C)CO)C2)C1.N n1(CC(=O)NCC(C)NC(c2cnc(-c3cnn(C)c3)s2)=O)cccc(N)c1=O N1(C(c2ncc(C)cn2)=O)CCC2(CCCN(C(=O)CC3CSC3)C2)CC1 n1(CC)ncc(C(=O)NC2COCCC2NC(=O)CN2CC(C)C2)c1Br Cc1cc(C(N2CCC(CNC(C3CCOC3)=O)CC2)=O)nn1CCO c1(C(=O)NC2C3CN(C(c4nc(CC)sc4)=O)C2C3)cccc2c1OCC2 c1(C(N2CCC(CN(C(CCC(=C)Cl)=O)C)C2)=O)nccc(N)c1Cl c1(C(N(CC(C)NC(c2cc(C)nn2C)=O)C)=O)ccc(Cl)c(F)c1F N1(C(CC2CCN(C)CC2)=O)C2CCC(C(=O)NCCc3ccncc3)C1CC2 c1(C(=O)NCCC(C)NC(=O)C(C)Oc2ccccc2Cl)nc2ccccc2o1 c1(N2CCC(CC=C)(NC(C3CC(F)(CO)C3)=O)C2)ncnc(Cl)c1CC C12(NC(C(C)c3ccco3)=O)CCCN(C(c3cc(Cl)ncc3Cl)=O)CC1C2 C1(NC(C(CC)OCC)=O)CC(C(=O)NCCCOC(F)(F)F)=CC1O n1(CC)cc(C(=O)NCC23CC2CN(C(c2cccc(=O)o2)=O)C3)c(C(C)C)n1 c1(C(=O)NC2CN(C(CNC(CC)=O)=O)CC2C)ccc(C(C)(C)C)cc1C N1(C(c2c(NS(C)(=O)=O)cc(Br)cc2)=O)CCC2(CCC(C(=O)O)NC2)CC1 C=C(C)C1OCCC1C(=O)NCC(CNC(=O)CN1CC(=O)NC1=O)CO CCCCC(C(=O)N1CC(O)CC1CNC(c1n[nH]cc1C1CCC1)=O)C(C)C C(C(C(C)C)NC(C1(OCC)CCOC1)=O)NC(CC1CC(=C)C1)=O N1(C(COC2(C#C)COC2)=O)CC2(CC(NC(c3csc(O)n3)=O)CO2)C1 C12(NC(c3n(CCC)ccc3)=O)CCC(CC1)N(C(c1ccc(CSC)o1)=O)C2 C1(NC(=O)C2CC2)CC2CC1CN(C(c1c[nH]cc1Br)=O)C2 c1(CN2CC3C(C(=O)NCc4ccc(C)nc4)(C3)C2)[nH]nc2ncccc12 CC1(C)C(CN)CCS1(=O)=NC(=O)c1c(Cl)ccc([N+](=O)[O-])c1Cl CCC(C#N)C(=O)NC1(CCNC(c2occc2C(C)C)=O)CC1 C1(CC)CN(C(=O)C(C)(C)c2ccno2)CCN1C(C1CC1(C)C(F)F)=O CCCC(CCCNC(=O)C(COC)N(C)C)NC(=O)C=Cc1cnc(C)s1 O=C(CC(O)CNC(c1ccc[n+]([O-])c1)=O)Nc1ccccc1C1CC1 C1(CC(=O)NCC(=CC(=O)N(CCOCC#C)C)C)CCCN(C)C1 CC(=O)CCC(=O)NC(c1nc(C(=O)NCCCCCC2CC2)co1)C C1(CC(=O)NC(CNC(C=CCN(C)CC)=O)CO)CC2C=CC1C2 Cc1ccc(NC(C2CC(O)CN2C(C2CC3(CCC3)C2)=O)=O)c(C(F)(F)F)c1 c1(OC)ncc(Cl)cc1C(=O)NC1CN(C(c2cn[nH]c2)=O)CC1(F)F N1(C(C(C=C)(C)C)=O)CC(NC(c2cccc(Br)c2Cl)=O)CC(F)(F)C1 N1(C(Cc2cn(C)nc2)=O)CC(NC(=O)C(C)(C)c2ccnn2C)CC(O)C1 Cn1nnc(C(N2CCC(C(C)(C)C(=O)NCCc3csnn3)C2)=O)c1N CC1CC=C(C(=O)NC(C2(CNC(c3cccn4nnnc34)=O)CC2)C)CC1 CC(N=c1cc[nH]cc1C#N)C1CCCCN1C(=O)CCCS(C)(=O)=O C1(CC=C)(NC(=O)CC2CC(C)N(C(c3cnc(C)nc3)=O)C2)CCOCC1 N1(C(c2scc(C(N)=O)c2)=O)CCCC(C2CCN(C(C3(C4CC4)CCC3)=O)C2)C1 C1(CNC(c2c(C)nc[nH]2)=O)CCN(C(=O)C=CC2COC(C)(C)O2)CC1(F)F CC1CN(C(C2(CNC(c3cc(C#N)c[nH]3)=O)CCCO2)=O)CC(C)(C)C1 C1(=O)C(CC2CCCC2)N1CC.c1(NC(c2nc[nH]n2)=O)ccsc1OC.C1CO1 CC1=C(C(=O)NCCCNC(C2CCOC2C(C)C)=O)CC1 c1(C(=O)NC2C3N(C(c4c(NC)cnnc4)=O)C(CC3)C2)ccc(F)c(F)c1F C1(C(N2CCC2C2CCOCC2)=O)(NC(C(C2CN(C(N)=O)C2)O)=O)CCSC1 S(=O)(=O)(c1cnn(C)c1)NC12CC(C(=O)Nc3c(C(C)=O)cc(F)cc3)(C1)C2 Cc1cc(C(=O)NC2CN(C(C3CCCCS3)=O)CC2O)c2cnccc2c1 C(=O)(C1=COCC1)NC(CN(C(c1nc(Cl)cs1)=O)CC)C c1(-n2cc(CNC(C(=O)OCCCC)c3ncc[nH]3)nn2)ccc(Cl)cc1Cl CN1CCN(CC(=O)NCC=C2CCN(C(=O)C(c3ccc(Cl)s3)=O)CC2)CC1 N1(C(CC(=O)OC(C)(C)C)=O)CC2CC(C(=O)NCCc3cccc(F)n3)(C2)C1 N#Cc1c[nH]c(C(=O)NCC(=O)NCCn2ncccc2=O)c1 Cc1nn(CC(N2CCN(C(C)C)C(=O)C2)=O)c(C)c1C n1(CC(=O)Nc2ccc(Oc3ccc(OC)cc3)nc2)ncc2ccccc12 c1(C(=O)Nc2cccc(Br)c2)ncn2cc(-c3cccc(OCCF)c3)sc12 c1(C(N(CC)CC2CCCCN2C(C2CCN2C)=O)=O)ccc(C#N)cc1 C1(CCC)(NC(c2cccc(C)c2C)=O)CCCN(C(=O)COCCCOC)C1 C(=O)(C=CSc1nc[nH]n1)N(CCC)CCNC(c1cnc(C(C)OCC)s1)=O c1(C(N2CCC(NC(C(CCCC)O)=O)C2C)=O)cc(C)nc2onc(C)c12 C(C)(C(C(=O)NCCNC(C1(c2ccccc2)CC(O)C1)=O)N(C)C)OC.C(C)C N1(CC)C(=O)CCC1CC(=O)NC1(C)CN(C(C2CC2F)=O)C1 n1(CC(=O)N(C2CCCN(C(c3cnc(Cl)c(Br)c3)=O)C2)C)nnc2ccccc12 c1(NC(c2cncc(CC)c2)c2nnnn2C2CC2)cc(C#N)cnc1C N1(C(CC(C)(F)F)=O)CCOCC(CNC(C23CCCCC2C3)=O)C1 CC(CN=C(NCc1ccnn1C)N1CCC2(CC(C(F)F)=NO2)C1)C(C)(F)F N1(C(C2CC(=C)C2)=O)CCCC2C1CCCN2C(c1cccc(C2(CO)CC2)n1)=O c1(C(N2CC(C)(NC(C=CC(=O)N(C)C)=O)C2)=O)ccc(-n2cccn2)nc1 N1(C(c2noc(C)c2[N+](=O)[O-])=O)CCC2(CCCN2C(C23COCC2C3)=O)CC1 CC1CN(C(C2(S(N)(=O)=O)CC2)=O)CC1NC(c1coc(C2CCOCC2)n1)=O c1(C(=O)NC(CC)(C)CNC(C2(COC)CC2)=O)cnn2ccnc(C)c12 N1(C(C2C(SC)CCC2)=O)CC2CC(C1)C2NC(C1CC2CC2C1)=O c1(C(CNC(c2cnc(C)o2)=O)NC(C2CCC(C)CC2)=O)ccc(F)cc1F C(CCCCCNC(=O)CC1CC12CC2)N(C(=O)Cc1cncn1C)C CCC(C#N)(CC)C(=O)NC(CCN(C(=O)C(O)CCN(C)C)C)C(C)C c1(C(=O)NCC(CCCC)NC(C2C(=C)C2)=O)ccc(N)c(Cl)c1 N1(C(CCN(CCC)C)=O)C2CCC1CC(NC(=O)C(F)(F)CC)C2 C#Cc1cccc(C(N2CCCC(NC(=O)CC3CCC(=O)NC3=O)C2)=O)c1F c1(C(=O)NC(CCN(C(C2(COC)CC=CC2)=O)C)C)cc(OC(F)F)n(C)n1 N1(C(CCCN(C(C)=O)C)=O)CCC2(CC1)CC2NC(=O)C(F)(F)CC1CC1 CCCC(C)CCNC(=O)CNC(=O)CNC(c1c[nH]c(=N)o1)=O C1(NC(c2nc(C(=O)OCC)sc2)=O)CN(C(c2coc(Cl)n2)=O)CC2CC12 n1(C(C)C)ccnc1C(=O)NCc1ccc(C(=O)NCC2CCC(O)C2)s1 c1(NC(C(C)(N(C(C=CCCC)=O)C)C2CC2)=O)ccn2nccc2c1 CCCC(CNC(=O)CCC1OCCO1)C(=O)NCCC1CCC(C)CC1 Cc1cc(I)ccc1C(=O)NC1CCC(C(=O)Nc2nc(Br)cn2C)C1 c1(C(=O)NCC(CO)NC(C2CC(=O)OC2)=O)nc(Br)[nH]c1C(F)(F)F N1(C(c2c(Cl)c(C)n(C)n2)=O)CCC(NC(C2OCCO2)=O)C(C)(C)C1 CCCC(C)(CCC)C(=O)N1CC(CNC(c2[nH]nnc2C2CC2)=O)C(C)(C)C1 N1(C(C2(C#N)CCC2)=O)CC2CCC2(CCNC(C2(F)CC2)=O)C1 c1(CC)ccc(C(=O)NCCOCCCNC(C2CCCC(C)CC2)=O)cc1N c1(C(N(CCN(C(c2cccn2C)=O)CC)CC)=O)nc(C)ccc1F C1(C(=O)OC)CC=CCN1C(C1CCC(NC(C2CC2C(N)=O)=O)C1)=O C(C)(C)(CCNC(=O)C=CSC)NC(C1(COC)COC1)=O c1(NC)ccc(F)cc1C(=O)NC1CCC(NC(c2cc(C)ncc2C)=O)CC1 C12(C(=O)NCC3CCCCN(C(C(C)SC(C)C)=O)C3)CCCCC(F)(C1)C2 c1(CN2CCCC(O)(C(C(=O)NC)(F)F)C2)nc(C)c(Cl)cc1Cl c1(C(N(CCCN(C)C(c2cnn(C)c2)=O)C)=O)cccc(S(C)=O)c1 C(=O)(C(F)CCC(C)C)N1CC(COC)N(C(=O)C(C)N(C)C(C)=O)CC1 c1(C(=O)NCC(CO)NC(=O)COCC2CCCOC2)c(O)nnc2c1CCC2 C(=O)(C(O)CCCCC)NC(C(=O)NC(CC=C)(C)C(F)F)C CC(CC(C)NC(c1cc(F)n(C)n1)=O)N=c1[nH]nc(C(C)(C)C)s1 Cn1nc(C2CCCN2C(c2cc3cc(Br)cn3cn2)=O)c2ccccc2c1=O c1(C(N2C(C)C(NC(=O)C(O)C3CCCC3)CC2)=O)cn(C)c(=O)cn1 c1(C(=O)NCC(CNC(C2CCC(C(=O)OC)C2)=O)O)nccn2cc(C)nc12 N1(C(C(CCC)N(C)C)=O)CC(C)(C)OCC1CNC(c1cc2[nH]ccc2s1)=O CCC(C(=O)NC(C)CNC(c1c(OC)ccc(Cl)c1F)=O)C(F)(F)F O=C(CCC(=O)N1CCC(O)CC1)NCC1CC1CNC(c1ccc(F)o1)=O C1(C#N)(C(N(CCOCCN(C)C(c2cncs2)=O)C)=O)CCCCC1 C(CCC(=O)NCC1CC1NC(=O)CCCc1cc(C)no1)NC(=O)NCC#C N1(Cc2ccncc2)CC2CC3CC2C1C3O.C1(=O)CNC(=O)C2(CC2)C(C)N1 C1(CNC(C(C=CC)O)=O)CN(C(C2CC2c2ccccc2)=O)CC12CCC2 C#CCC(C(=O)NCC1CCN1C(C)(C)C)NC(c1cnn(C)c1Cl)=O c1(C(=O)NCCOCCNC(Cc2c(C)nccc2)=O)cnn2cccnc12 N1(CCN(CC=C)CC)C(=O)CCN(CC(N2CCCCC2)=O)C1=O C(=O)(C1=CCCCO1)NCc1ccc(C(N2C(C(CCC)C)CCC2)=O)s1 Cc1ccncc1C1CC1C(=O)N(C)CC1CN(C(=O)C(C)C)CCO1 C#CCC(O)C(=O)NC1(CO)CN(C(c2cccc(-c3cscn3)c2)=O)C1 c1(NC2CN(C(c3cc(C)[nH]c3)=O)CC2C)ncc([N+](=O)[O-])cc1Br c1(C(c2n(CCCSCC)nnn2)NCC(CC)OC)cccc(C)c1F C1(NC(C2(COC)CC2(F)F)=O)CCN(C(C2CSCN2C)=O)CCC1CO C1(SC)CCN(C(c2cc(Br)ccn2)=O)CC1.C12CC1CCNC2 O=C1CC(CC(=O)NC2CC3(C2)CC(NC(C24CCC(CC2)CO4)=O)C3)=NN1 N1(C(C(=O)NC2CCCOC2)=O)CCCC1C1CCCC1 Cc1ccc2c(C(=O)NCC3COCCN3C(=O)CCC(N)=O)onc2c1 c1(C(C)NC(C2CC2CNC(=O)C=CCN2CCC2)=O)ccnn1C C1(NC(C(C)NS(CC)(=O)=O)=O)CN(C(=O)C#CC2CC2)CC1C(F)(F)F N1(C(c2c(-c3cn(C)nc3)n[nH]c2)=O)CC2CC(C1)CN(C(=O)C(O)C1CC1)C2 N1(C(c2ccn(C)n2)=O)CCC(C2CC2)C1CNC(C1CS(=O)(=O)CC(=O)N1)=O c1(CN(C(C2COCCN(C)C2)=O)CC2CCCO2)nn(C)c2c1CCC2 c1(C(N(CCCNC(=O)C(C2CC2)SC)CC)=O)nccc(Cl)c1C C1(O)(CCNC(C2CCCCCCC2)=O)CCN(C(C2CC2C(F)F)=O)CC1 C(C(CC(C)C)C(=O)NCCCCCn1cc(CC(C)(C)OC)nn1)OC C1(C)(C(N2C3CC(NC(c4ccc(C)nc4N)=O)(C3)C2)=O)CC(C(C)(C)C)=NO1 c1(CC)cc(Cl)ccc1C(=O)NCc1nc(CNC(=O)C(C)CC2CC2)cs1 c1(OC)cc(Cl)c(C)cc1C(=O)OCc1cn(-c2c(C)cccc2C)nn1 CCC(CCOC)C(=O)NC1COCC1NC(c1cc(O)n(CC)n1)=O CC(CCC(=O)NCCC1(CNC(C2CCCN2C)=O)CC1)N(C)C C(C(CO)(CO)NC(C1CC1F)=O)N(C(c1ccn(COC)n1)=O)C n1(CC)nnc2c1C(C(=O)N1CC3OCC(C)C3C1)CN(C(=O)C(C)COC)C2 N1(C(CCC=CC)=O)CC(NC(=O)C=CCN(CC)CC)CC2(CC2)C1 c1(NC(C2(C)CCN(C(CCC)=O)C2)=O)nc(Cl)c(F)cc1C#N C12(NC(=O)NC3(c4ccc(F)c(F)c4)CCC3)CCCCCC1OCC2 N1(C(c2cccc(NC)n2)=O)CC2CN(C(=O)C(c3cccnc3)C)CC2C1 c1(C(N2CC3CC3C2)=O)cnn2ccc(-c3ccc4cncn4c3)cc12 C1(Cl)(C(=O)NCCCC2(NC(c3n(CC)nnc3)=O)CC2)CC12CCC2 c1(OCC(=O)NCC(CNC(CC2(C=C)CC2)=O)F)ccccc1C(N)=O C1(NC(=O)C=Cc2cc[nH]n2)CC(F)CN(C(c2ccsc2Cl)=O)C1 c1(N2CCCC(CC(C)(C)C)C2)nc(NCC2CC(F)(F)C2)nc2c1CCCC2 c1(C(=O)NCC(CNC(C(C2CCOCC2)C)=O)(C)O)c(Cl)ccc2c[nH]nc12 N1(C(=O)Nc2ccc(C#N)c(-c3ccncc3)c2)CCc2c(F)cccc21 N1(C(C(CSC)OC)=O)CC(CN(C(=O)Cc2cccc(C)c2)C)C(C)(C)C1 c1(C(=O)NCCC(C)NC(=O)Cc2ccccc2Cl)ccc(C(=O)N(C)C)cc1 n1(CCC(=O)N(CC(C)CNC(=O)CC2CCC23CCC3)C)cc([N+](=O)[O-])cn1 c1(C(N2CC(N(C(C)=O)C)C(F)C2)=O)n[nH]c2cccnc12 C1(NC(N2CCN(C(COC)=O)C(C)C2)=O)C2CCCC1CCC2 C(=O)(CC1NC(=O)c2ccccc21)NCCCNC(=O)CC1CCC(F)(F)CC1 c1(CN2C(C)(C(N3CCN(C4CC4)CC3)=O)CC2)c[nH]c2cc(F)c(F)cc12 c1(CC(=O)NCC2C(NC(C3(C)N(C)CCC3)=O)CCC2)cncc2ccccc12 Cc1csc2cc(C(N3CC(NC(C4CCN(C)C4=O)=O)C4(CC4)C3)=O)[nH]c12 C1(OC)CC(CNC(C2CC2F)=O)N(C(=O)Cn2cc(Br)cn2)C1 N=c1ccc(C(=O)NC2(CNC(=O)CN3CCCCC3=O)CCOC2)c[nH]1 N1(C(C(CO)NC(=O)OC(C)(C)C)=O)CCC(N(C2COC2)C(=O)C2CC2)CC1 C(=O)(C1=CCCC1(C)C)NCCN(CCC)C(C1Cc2nncn2C1)=O CC(C)C(C)C(CNC(C12CCC(CC1)O2)=O)NC(c1cc(=O)n(C)cn1)=O C=C=CCC(=O)NC1CCOC1C(=O)NC(c1ccns1)C CCCC(CCC)CC(=O)N1CCC(CO)C(NC(=O)CSCCC(C)C)C1 C(=O)(CS(=O)(=O)C1CC1)NC1C(C)(C)CN(C(c2ccc(N)c(O)c2)=O)C1 c1(C(=O)NC(C(=O)NCC)C)ccc2c(n1)CN(C(c1cnncc1C)=O)CC2 C1(C(N2CC(C)C(C(=O)NCCN3CC=CCC3)C2)=O)CCCC(C)(C)C1 C(=O)(C(C)C(O)CC(C)C)NCC1=CCN(C(c2c(C)c(Cl)cnc2)=O)CC1 c1(C(CC)NCCNC2CCCOC2)ccc(OC)c(OC)c1C c1(-c2cccc(OC)c2F)ccc(S(=O)(=O)N2CCN(CC(C)(C)O)CC2)cc1 c1(C(C)NC(c2cccnc2)CC)cc(C)ccc1C c1(C(N2C(C)CN(C)CC2)=O)cc(O)nc2c1CN(C(=O)CSCC(N)=O)CC2 c1(C(N(CCCC(C)O)C)=O)cc(-c2cn(C(C)(C)S(C)(=O)=O)nn2)cnc1O CCCCC(F)C(=O)NC1CC2CC(NC(c3cccc(C)c3Cl)=O)C1C2 N1(C(c2c(OC)nccc2)=O)CCC(C)C(NC(c2coc3c2COC3)=O)C1C C1(OC)CN(C(c2cnc(C3CC3)s2)=O)CC1NC(c1cnns1)=O CCCCCC(O)CC(=O)N1CC2CCCC2(NC(=O)CC2CNC(=O)O2)C1 Cc1[nH]c(C(=O)NC(C2CCN(C(=O)CN(C)C(C)C)C2)C)c(C)c1[N+](=O)[O-] C1(C(N2CC(OC)C(OC)C2)=O)N(C(c2ccncc2)=O)CCC1(C)C c1(-c2cn(C3CCC(OC)C3)nn2)nc(-c2nc(C)cs2)nn1C(C)C c1(C(N2CCOC(c3ccccc3C)C2)C(=O)NC)ccc(C(F)(F)F)c(Cl)c1 c1(NC(C2CCC(C)N2C(=O)C2=CCCCO2)=O)cccc2cccc(Br)c12 Cc1ccnc(C(=O)NC2CCC2CNC(c2cnc(C(F)(F)F)nc2)=O)n1 Cc1ccc(NC(C2(C)CCN(C(=O)Cn3cc(Br)cn3)C2)=O)c(Br)n1 C(CCC(C(=O)N(C)Cc1ccccn1)NC(=O)C(C)C1CCCC1)OC c1(NC)cnccc1C(=O)NCCc1n[nH]cc1C(N1CCC1C(C)C)=O CC(C)C(F)C(=O)N1CCC(COC2CCN(C(=O)C(C)n3cnnn3)C2)CC1 C1(O)(C(C)NC(CC(CC)C)=O)CCN(C(c2cnc3sccn23)=O)CC1 c1(C(=O)NCC2C(NC(C(N)=O)=O)CCC2)cc2ccc(Br)cc2cn1 c1(C(=O)NC(CNC(C(F)=CC)=O)(C)C2CCC2)ccnc2c(F)cccc12 Cc1nn(C)cc1C(=O)NCC1C=CCN1C(=O)CCc1ccc(Br)cn1 CCC(CC(=O)N1CCOC(N(C)C)C1)N(C(=O)CCn1cncn1)C C1(C(=O)NC(C=CC(=O)NCC2(CC=C)CCCC2)C)CCCN(C)C1 C12(NC(c3c(C)nns3)=O)CCCC(CN(C(C3CCC=CCC3)=O)C1)C2 C=CCN=C(NCCNC(C)=O)NCc1ccc(F)cc1 CCCC(CC)CCC(=O)NC(CN(C)C)C(=O)NCC(C)(C)C(N)=O C1(CNC(C=C(C)C)=O)CCN(C(c2cccc(-c3nnco3)c2)=O)C12CC2 N1(C(C(C(C)C)CO)=O)CCC2(CCC(O)C2)CC1 S(=O)(=O)(c1cnc(N2CC(C3CC3)OC(C)C2)c(Cl)c1)NCc1ncc(CC)s1 N1(C(C2(C)CCNC2=O)=O)CCCC2(C1)CN(C(C1CCCCS1)=O)C2 c1(C(N2CC(C)CC(NC(c3c(CC)[nH]cc3)=O)C2)=O)c([N+](=O)[O-])c(C)nn1C N1(C(c2c(C)occ2)=O)CC(CC(=O)NCCN=[N+]=[N-])C(C)C1 C(CC(C(=O)NC12CC1CN(C)C2)NC(c1cc(C(F)F)[nH]n1)=O)=CC c1(C(=O)Nc2cccc(OCCOC)c2)cnc2ccccc2c1 C1(=O)C(C)(C2CC2)N1.C(C(=O)N(CC(C)NC(C)=O)C)SCC N1(C(C23CC(NC(C(C)NC(=O)C4CC4)=O)(C2)C3)=O)CCCC(C)C1C C1(N(C(=O)C2=C(C)OCC2)c2cc(CC)no2)CCC12CCNCC2 C(=O)(CCCC(=O)NC1CC(C)N(C(=O)C=CC2CCCN2C)C1)NCC N1(C(C=CCOC)=O)CC(F)CC1CN(C(=O)Cn1nnc(C)n1)C C1(C(=O)NCCC(C)NC(C2(C(F)(F)F)CCCC2)=O)CC=CCC1 c1(C(N2CCC3(NC(CCc4n[nH]c(=N)s4)=O)C(C2)C3)=O)cnc2ccoc2c1 C1(C(=O)Nc2c(C)noc2)N(C(C2OCCC2C)=O)CC12CCCC2 N1(C(CC(CC)OC)=O)CC(CNC(C2C3CCCC23)=O)C(F)(F)C1 C1(C(N2CC(C)C(NC(=O)Cc3csc(=N)[nH]3)C2)=O)CCCCC1(C)C c1(C(N(CC(C2CCCC2)NC(=O)C(C)NC(C)=O)CC)=O)cc(CNC)no1 N1(C(C(C(C)(C)C)OC)=O)CC2(NC(=O)CC(C)CN(C)C)CCC1CC2 C(C(C)(O)CC(=O)NCCCN(C(=O)CN1CCC(C)(O)C1)C1CC1)OC N1(C(C=CC)=O)CCC(N(CCC)CC)CC1.c12cccc(n1)NC(=O)CC2 c1(C(=O)OC)cnc(C(=O)NCC2CC(NC(C3(C)C=CCCC3)=O)C2)cn1 C(=O)(C1=C2CCCN=C2NN1)NC1C(C)N(C(C2CC3CCCC3C2)=O)CC1 C1(NC(C2CC(Cl)(Cl)C2)=O)CC2(C1)CC2NC(=O)C(O)CC1CC1 n1(CC)cc(S(C)(=O)=O)cc1C(=O)Nc1ncc(Cc2cc(Cl)cc(Cl)c2)s1 C1(C(=O)NCCN(C(CC=CC=C)=O)CC2CC2)OCCC1C(F)(F)F c1(OC)ccc2c(C(=O)NCC(C)CNC(=O)CCCCC(N)=O)n[nH]c2c1 C1(CN(C(C2C(C#C)C2)=O)C)CCN(C(=O)C(C)C=C)CC1 C1(C(=O)OC)CN(C(C2CC2CNC(C2CCC2C)=O)=O)C(C)(C)C1 C=C=CC(C)C(=O)NC(C)(CSC)C(=O)NC(CC1CC1)C(=O)OC c1(-c2cn(C(C(=O)NCc3c(C)cccn3)C)nn2)cnc(OC(C)C)c(C)c1 CC(C(=O)NCC(N1CCN(C(=O)Cc2csc(=N)[nH]2)CC1)C(F)F)C(F)F c1(C(=O)NCC(CC(=O)NC2CC(OC)C2)OC)cnc(O)c(F)c1 C(=O)(CCCC(N)=O)NC(CCNC(c1cccc(C(=O)NCCC)c1)=O)(C)C C(=O)(CC1=CCCCC1)N1CC(C)(CNC(=O)Cc2nnc(O)s2)OCC1 c1(C(N(C(CNC(C(CC)=CC)=O)C2CC2)C)=O)cnc2c(c1)NC(=O)CN2C C1(NC(c2cc(C)ns2)=O)CN(C(=O)C(C)(C)c2ccnn2C)CC(C)(C)C1 N(C1CCCn2cnnc21)C(C12CC(C(F)(F)F)(C1)C2)=O C1(C(N(CCNC(=O)C(=Cc2cccnc2)F)C2CC2)=O)CCc2c[nH]nc2C1 C(c1ccc(Cl)cc1)=CC(=O)NCC1C2CN(C(=O)CCN3CCOCC3)CC12 C1(CCOC)CN(C(c2cscc2F)=O)CCN1C(C1CN(S(C)(=O)=O)C1)=O N1(C(CN(C)CCO)=O)CC(NC(c2ccn(C(C)(C)C)n2)=O)CC12CCOC2 N1(C(C(C)(C(C)C)OC)=O)CCN(C(=O)C=Cc2ccccc2)CC(O)C1 CS(=O)CCC(O)C(=O)NCC1(NC(c2cnc(=N)[nH]c2)=O)CCC1 N1(C(C(C)C(C)(C)C)=O)CC2(CCN(C(=O)CCF)CC2)CC1C n1(CC(CC)O)cc(C(N2CCC2CNC(c2nccs2)=O)=O)nn1 C(CO)(C(F)(F)F)N.C(CC(=O)NCCS)OC.C1C(=O)N1CC(C)C c1(C(N(CC(C)NC(C2CCC2(C)C)=O)CC)=O)nc(C)ccc1OC C12(CCNC(c3c(CC)nn(C)c3)=O)CCC1CN(C(=O)Cc1cncn1C)C2 N1(C(C2(C)CN(C(=O)C=CCF)C2)=O)CCC2CCCCC2C1 n1(CC(C(=O)OCCSCCCCCC=C)(C)O)c(C)cccc1=O c1(C(=O)NCC(CC)(C)NC(=O)CC2CC(C)C2)cc(Br)c2nccn2c1 c1(C(=O)NC2CC(NC(c3c(C)cn(C)c3)=O)C2)nnc(O)cc1O C1(C(=O)NCC(CC)NC(c2cc(CCC)[nH]n2)=O)CCCC(C(=O)OC)C1 c1(C(=O)NC2C(NC(CCC)=O)COCC2)ccc(C(C)C)cc1C(C)C CC1(C)CC(CNC(c2csc(S)n2)=O)N(C(c2ccnc(C3CC3)c2)=O)C1 c1(C(=O)NCC(CNC(C2ON=C(CC)C2)=O)(C)O)ccc(Cl)nc1OC1CCC1 C1(C(=O)NCC(C)N(C(=O)CC2(COC)CC2)CC)Cc2nnc(C)n2C1 C(=O)(CCCCN(C)C)NC(C1CCN(C(C2C(CCC)C2)=O)C1)C N1(C(=O)OC(C)(C)C)CCC2CN(CC(N)=O)C2C1 C1(C(=O)NOC(C)(C)CO)(CC=C)CCCN1C(=O)CCSC c1(C(C)Oc2cnccc2NC(c2nc(C(F)F)cs2)=O)cc(F)cc(C#N)c1 N1(C(C(CC)n2cncn2)=O)CCN(C(=O)CCN2CCC2)CC1CC c1(CCC(=O)NC2CCC(NC(=O)C=CC=C(Cl)Cl)CC2)nnc(O)nc1O C(=O)(C1=NOC(C)C1C)N1CC(CC(N2CC3C(CC)(C3)C2)=O)OCC1 N1(c2[nH]ccc(=N)n2)CCOC2(CCS(=O)(=NC(=O)c3coc(O)n3)CC2)C1 CC(C)CC(CNC(C1(c2cc[nH]n2)CC1)=O)C(=O)NC1(C)CCCC1C C(=O)(C1CCCc2nc[nH]c21)N(CCCCCNC(C1CCS(=O)(=O)C1)=O)C Cc1nc(NC2(CNC(c3ccc(CF)cc3)=O)CCCC2)ncc1[N+](=O)[O-] N1(C(C(n2ncc(C)c2)C)=O)CC2CC2C1C(=O)N(CC1CC1)CC1CC1 C(C)(C)(CCCC(=O)NC1CC12CCCCCC2)NC(C1CC=C(C)CC1)=O c1(C(N(CCNC(C2CC(=C)C2)=O)CCC)=O)cc2c(OC)cccc2[nH]1 c1(C(N2C(C(C)NC(C(C)OCC)=O)CCC2)=O)cc(F)c(F)cc1O CC1=C(C)CC(C(=O)NCC(=O)NCC(O)CF)CC1 C1(NC(c2sccc2F)=O)CCOCC1C(=O)NCCCN1CCCC1=O C1(n2cc(C(=O)OC)nn2)CCN(C(=O)C(c2cccc(OC)c2)(F)F)CC1 C12(C(=O)NCC3N(C(c4c(C)c(C(F)(F)F)n[nH]4)=O)CC3)CCC(CC1)CC2 CCCC(C)(O)CC(=O)N(C1CCN(C(=O)CCOC(C)=O)C1)CCO c1(SCC(=O)NCCCCN(C)C(c2[nH]ncc2C#N)=O)ccc(Cl)cc1 N1(C(=O)Nc2c(-c3cc(C)sc3)nccc2)CCCC2(CCC2)C1 c1(CC(=O)NC2(CCNC(C3(F)C(C)C3)=O)CCCC2)cccc(F)c1F C(=O)(C(=O)C(C)(C)C)NC(CCOC)C(=O)N(C)CC1(O)CCC1 c1(C(=O)NC(CN(C(C(C)N2CCCC2)=O)C)(C)C)cc(N)cc(O)c1F C1(NC(c2ccc(NC)cc2)=O)CCN(C(=O)Cc2c[nH]nc2C)CC1C c1(OC)cc(C(N2CC(NC(c3cc(CC4CC4)on3)=O)C2)=O)c(C)c(Br)c1 c1(C(=O)NCC2(F)CC(CNC(C(C)Sc3ccccn3)=O)C2)cnccc1Cl C1(C(=O)NC(CC(=O)N(c2ccc(N(C)C)cc2)C)CC2CC2)C2CC3C(C2=O)C13 c1(CN(CC(=O)NS(CC)(=O)=O)CC)ccccc1.C1(=O)C(=O)N(C)CCCN1 N1(C(CCC#CC)=O)CC2CCN(C(=O)CC(C)P(C)(C)=O)CC2C1 c1(CN2CCN(S(CC)(=O)=O)C(CO)C2)cc2ccoc2cn1 Cc1nc(N(CCNC(=O)Cn2ccsc2=N)C2CC2)ccc1[N+](=O)[O-] C1(C)(CC)C=C(C(=O)NCc2cn(C3CN(C(c4cc(C)[nH]n4)=O)C3)nn2)C1 CCCC(C(=O)NCC1(CC)CCC1)NC(=O)C#CC1CC1 CC1OC2(C)CC1(C(=O)NCCN1CCN(c3cc(C(N)=O)nc(Cl)n3)CC1)C2 Cc1ccc(OC(C)C(=O)OCCCn2ncc(NC(N)=O)c2)cc1 c1(C(N2CC3(CN(C(c4cc(C)n(C)n4)=O)C3)C2)=O)cn(C(C)C)c(=O)nc1O c1(OC)cc(CC(=O)NCCC2CCN(C(=O)C(C)C(C)(F)F)C2)ccc1Cl C=C(Cl)CC(C(=O)N(C)Cc1nc(C)no1)NC(C1CC2(CC2)CO1)=O CC(C)C1=NOC(C(=O)NCC2CN(C(C3(CO)CCOC3)=O)CC2(C)C)C1 CCC(O)C(F)(F)C(=O)N1CC(O)(CN(C)C(c2ccc(=N)[nH]c2)=O)C1 c1(NCCNCCc2scc(C)n2)nccc(=NC2CC(=C3CCC3)C2)[nH]1 CC1CN(C(C2(C(N)=O)CC2)=O)CCC1CNC(c1nccs1)=O C(=O)(C(C)(C)CCCF)NC12C(CN(C(C(CCC)NC(C)=O)=O)C1)CC2 Cn1ccc(=O)c(C(=O)NC2CC(CC(=O)NCC3(CC4CCC4)CC3)C2)c1 c1(C(=O)NC2CC3(C(NC(CCC(CC)C)=O)C3)C2)cccc(SC)c1[N+](=O)[O-] N1(C(Cc2nc(C)c(C)s2)=O)CCOC2(C1)CN(C(=O)CC1(C)CC1(F)Cl)C2 CC(C)(C)C#CC(=O)NCc1ncoc1CCNC(C1CC1C1CCCC1)=O c1(CC)c(OC)cccc1C(=O)NC(C)(CNC(=O)C(C)n1cncn1)CC c1(C(=O)OC)ccc(S(=O)(=O)Nc2ccc(I)c(C(=O)OC)c2)cc1C(=O)O N1(C(c2c(C)ccn2C)=O)CCCC(O)(CNC(C2(C)CC2(Cl)Cl)=O)C1 C12(C(=O)NC(CC)C(F)(F)F)CCCOC1CCN(C(=O)C(C)NS(=O)(=O)CC)C2 Cc1cc(C(=O)NCC2CC3CCC2N3C(C2(C)CCCCC2)=O)nc(O)n1 CCC(CC(=O)N(C1CCCC1)CCNC(=O)CC1CCC(C)(C)C1)SC CCCC(CC(=O)N1CCCC1(C)C1CC1)NC(C1CCNC1=O)=O c1(C(N2CC(F)(CNC(C=CC(C)(C)C)=O)C2)=O)cccc(-c2cccs2)n1 C1(F)(C(=O)NC2C(NC(=O)CSC3CC3)COCC2)CCCCCC1 CCCCC(O)C(=O)NC1CCN(C(=O)C(C)Oc2ccccn2)CC1O c1(CN2CC(C(N3CC(C(N)=O)OCC3)=O)OCC2)ccc(Cl)c(O)c1 c1(CC)cc(C(N2CC(OCC(=O)NC3CC(=O)N(C4CC4)C3)C2)=O)n(C)n1 CC(C)C1=NOC(C(=O)NC(CC(=O)NCC(O)CCO)C(F)F)C1 Cc1cc(N2CCC(NC3CCCSC3)CC2)ncc1S(=O)(=O)NC1CCC1 C1(CNC(c2ccc(C(=O)OC)[nH]2)=O)CN(C)CCN1C(=O)CC(C)(F)F c1(OCC(=O)NCC(CCNC(CCc2cc(C)[nH]n2)=O)O)cc(F)cc(F)c1 Cc1ccc(C(N2CC(CCO)(NC(c3cnc(C)[nH]3)=O)C2)=O)cc1 CC1(CNC(c2ccc(Br)o2)=O)CC(NC(C2CN(S(C)(=O)=O)C2)=O)C1 N1(C(c2cc(COC)on2)=O)CCCC(CO)(NC(=O)CCC2CC2(C)C)C1 C(=O)(C(=O)N=c1ccn(Cc2ccccc2)[nH]1)NCc1c(F)c(N)c(Cl)c(F)c1 N1(C(C2N(C(c3c(CC)c[nH]c3)=O)CCN(C)C2)=O)CCCN(C)CC1C C12(C(=O)NC3CCCCN(C(C(=O)N(C)C)=O)C3)CC1COC21CCC1 N1(C(C)=O)CC2(CCN(C(C3CCCN(C(C)C)C3)=O)C2)C1 N1(C(=O)CC2(O)CC2)CCc2sccc2C1.CC1C(=O)NCC2CCC2C(=O)N1 c1(C(=O)NCC2(CNC(C3(CC)CC=CC3)=O)CC2)cc2c(cc1Cl)OCCO2 C(CC(C(C)C)NC(=O)Cc1ncc(C)s1)NC(C(CC)n1ccnc1)=O CC1CC(NC(=O)CSc2ccccn2)CCN1C(=O)C1=C(Cl)CCC1 C1(O)(C(=O)OC(C)(C)C)CCN(C(=O)C(N)Cc2cccnc2)C1 n1(CC)ccc(C(=O)NCCCOCCC(=O)NCC2(C)CC3CC3C2)c1C CC1(C)CN(C(=O)CN(C(=O)C=C2CCC2)CC2CCC2)CCC1O c1(CCC)ncoc1C(=O)NCC1(NC(C2CC=CCO2)=O)CCOC1 C1(O)(CNC(c2ccc(F)s2)=O)CCCN(C(=O)Cc2ccc(Cl)c(F)c2)C1 C(=O)(C(F)(CC)C(=O)OC)N(C)CC1CCCN(C(c2nc(CC)oc2)=O)C1 c1(C(N2CCC(C(C)OC)CC2)C(=O)NCC=C)scc(C(=O)OC)c1Cl c1(C(=O)NCCOCCNC(C2(n3cccn3)CC2)=O)cc2n(n1)CCO2 CS(=O)(=O)c1cccnc1N1CCC(NC(c2cccn3nccc23)=O)C(F)C1 c12ccccc1C(=O)NC2.C1(C)(OCC(=O)N(CCCN(C)C)C)CCCC1 N1(C(C(CSC)O)=O)CCC2(CCCN(C(=O)C(c3cc(C)oc3C)C)C2)C1 c1(N2CC(C)CC(C)C2)ncc(S(=O)(=O)NCCNC(=O)N(C)C)cc1Cl Cc1nc(C2CC2)oc1C(=O)NC1CCC(CNC(c2cc(F)c[nH]2)=O)C1 C1(NC(=O)OC(C)(C)C)CCCC(N(C(=O)CCc2cn[nH]c2)CCC#N)CC1 C1(CNC(C(CC)OCC)=O)CC(C(=O)NCC(C)(C)OC)=NO1 c1(C(N2CC(C(C)NC(C=C(COC)C)=O)OCC2)=O)nc(C)c(C)nc1O c1(C(N2CC3C(CNC(c4ccn(C)n4)=O)C3C2)=O)cc(F)c(Br)cc1F c1(C(N(CCC(C)NC(CCNC(C)=O)=O)C)=O)csc2c(F)cccc12 N1(C(c2c(C)c[nH]n2)=O)CCCCC(CNC(C2CC(N3CCCC3)C2)=O)C1 C(=O)(C1CCCc2nn[nH]c21)NCCCNC(C1C2(CC(C)(C)C2)C1)=O C1(CC(=O)NCCOCCNC(c2ccc(OCCO)cc2)=O)CCC2(CC2)CO1 Cc1ccc(S(=O)(=O)N2CC(O)CC2C(=O)N(C)Cc2c[nH]nc2C)cc1 S(=O)(=O)(c1cnc(NC(C)Cc2cccs2)c(Cl)c1)N(C(CCSC)C)C [N-]=[N+]=NC1CCN(C(=O)C(C2(O)CCCCC2)NC(=O)C(F)=CC2CC2)C1 c1(NC(C2CCN(C(=O)OC(C)(C)C)C2)C(=O)O)ccc(S(=O)(=O)NC(N)=O)cc1 C1(C(=O)NC2CN(C(C)C)C(=O)C2)CC12CCN(C(C1CS(=O)C1)=O)C2 C(=O)(CCCCCF)NC1C(NC(c2c(C)n(-c3ccn(C)n3)nn2)=O)CC1 c1(C(=O)NC(C(C)NC(=O)CCS(C)(=O)=O)(C)C)cncc2nnn(C)c12 C(=O)(CCCCCCCC)NC(c1cccc(C)c1)CNC(CSCC=C)=O c1(C(=O)NC2CCC(NC(C(COC)O)=O)C2)ccc2ncccc2c1 C1(OC)CN(C)C(C)(C(=O)NCCC2(O)CN(C(c3cc(C)ccc3F)=O)C2)C1 Cc1nnc2cnc(C(N3CC4CC3C4CNC(=O)CCC3CCCC3)=O)cn12 n1(C2CCN(C(=O)NC(c3cc(C)cc(C)c3)C)CC2)c(O)nc2ccccc12 c1(OC)cc(CC(=O)OC(=O)C(C)N2CC(OCCC3CC3)C2)cc(Cl)c1OC C(=O)(C#CC(C)(C)O)N1C(C)C(C(=O)NC2CC(F)C2)CC1 N1(C(c2cc(CCC)[nH]n2)=O)CCCCC(NC(C23CC(CCO2)C3)=O)C1 C(=O)(C(C)CCCC(C)C)NC1CCN(C(CCOCC=C)=O)CC1CO C1(C(=O)Nc2c(CC)onc2C)CN(C(=O)C(O)C(F)(F)F)CCN1C Cc1c(C(N2CCC(O)(C(C)CNC(C3CC(F)(CO)C3)=O)C2)=O)cccc1N C1(C)(C(=O)NCCC(C)(C)NC(C(C)OCC=C)=O)CC=C(C)CC1 Cc1cccc(C(=O)NC2CCC(NC(=O)CSCc3ccncc3)CC2)c1N N1(C(C(CC)OC)=O)CC2(CNC(=O)C(C)C(O)CC)CC1CO2 Cc1nc(C)c(C(N2CCCC2(C)CNC(c2c(C)noc2C)=O)=O)s1 C1(C(=O)NC2(C)CCN(C(c3cccc(C(N)=O)c3F)=O)C2)CC12CCSCC2 CN(C)NC(=O)CCC(=O)N1CCC2C(C(N3CC(O)CC(O)C3)=O)C2C1 Fc1cc(F)c2cccc(-c3nc(C(c4ccc(C(F)(F)F)cc4)F)no3)c2n1 C1(NC(c2cccc3c2OCO3)=O)CC2CCC1N(C(C1CCCNC1=O)=O)C2 CC1=CCC(C(N2CCC(NC(=O)CS(=O)(=O)N(C)C)C2C(C)C)=O)CC1 C(=O)(C(C)C(=O)N1CCC(C)(CNC(=O)Cn2nc(C)nc2C)C1)OC c1(C(C)=O)cn(C)nc1C(=O)NCC(C1CC1)NC(c1cc(C(C)C)no1)=O C1(C(N(C(C(=O)NCC2C(CCC)C2)C)C)=O)OCCC1CC c1(CC)c(C(=O)NCCC2(O)CN(C(=O)CC(C3CC3)C3CC3)C2)nnn1C CCC(C)C(=O)NC(CN(C)C)C(=O)NC1(CCCF)CC1 C#Cc1ccc(C(N2CCN(C(C3CCC4CC4CC3)=O)CC2)=O)cc1C N(C(=NCC(C)N1CCCCC1)NCC1CCCCC1)Cc1scc(C)c1 CC(C)C(C(=O)N1CCOCC1)OCc1cn(CC2CSCCS2)nn1 C1(c2ccccc2)(CNC(C2C(C)CC2)=O)CC(NC(c2cnc[nH]2)=O)C1 N1(C(CC(C)O)=O)CCc2nc(C(N3CCC(C#N)(CO)C3)=O)cn2CC1 C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(CNC(CC(C)n1ccnc1)=O)C(F)(F)F CCC(CC(=O)NCCCCCNC(=O)Cc1ncn(C)c1C)SC Cc1cc(O)c(C(=O)N(C)CC2CCCN(C(=O)C(C3CC3)C3CC3)C2)nn1 c1(C(=O)NCC2N(C(CNC(C)=O)=O)CCCC2C)cc(O)ccc1[N+](=O)[O-] CCCCC(CNC(=O)CC(C)(C)C1CC1)N1CCOCC1 N1(C(CSCCCC)=O)CC(NC(c2cc(C)n(C(F)F)n2)=O)C(N=[N+]=[N-])C1 CCS(=O)(=O)CC(=O)N(C1CCN(C(=O)CN2CCCC2CO)C1)C c1(-c2cn(C3CC(C(N(C4CCC4)CC)=O)C3)nn2)ccc(F)cc1 CCCCC(O)CCC(=O)N1CCC1CNC(C1(O)CCCCC1)=O c1(C(N2C(CC)C(NC(c3cc(C(C)C)no3)=O)CC2)=O)ccc2sccc2c1 C1(NC(C2(CC#C)CCOC2)=O)CCN(c2cc(OC)ncn2)CC1C c1(CNCC(CNC(COCCC)=O)F)cc(OC)c(OCCC)c(Cl)c1 N1(CC(N2CC(F)(CNC(CN(C3CC3)CC)=O)C2)=O)CCCCC(O)C1=O NS(=O)(=O)C1CC(C(N2CCN(C(c3ccc(O)cc3)=O)C(C3CC3)C2)=O)C1 C#Cc1cnn(C)c1C(=O)NCCC(C)NC(=O)C=Cc1ccc(CC)cc1 c1(C(N(CC(C)NC(=O)CN2C(=O)CNC2=O)CC)=O)ccc(=O)n(C(C)C)c1 Cc1cnn(CC(=O)NCC2(O)CC(NC(=O)CC(C)O)C2)c1 c1(CCSC)cc(C)c(C(=O)CN2CCC(c3ccc(F)cc3C)CC2)cc1C c1(CCC(=O)NCC(C)(C)NC(CC(C(CC)C)O)=O)ccc2cnn(C)c2c1 CC(C)C(C)(C)C(=O)N(CC)Cc1ccc(Cl)nc1.C1(C=O)CCC(N(C)C)C1 N1(C(=O)OC)CCCC(C(=O)NC2CC(CNC(C3CCOCC3)=O)C2)C1 c1(C(=O)NCC2CC(F)CN2C(=O)Cc2ccncc2)c(Br)cccc1[N+](=O)[O-] N1(Cc2cnc(SC)nc2)CCN(C(c2ccc(I)cc2O)=O)C2CC12 N1(C(C(C2CC2)SC)=O)CCN(C(=O)C(N2CCCC2)C2CC2)CC1C c1(OCC#C)ccc(C(N2CC(CNC(c3sccc3C(F)F)=O)C2)=O)cc1 C1(CNC(=O)C=Cc2ccncc2)CCCCN1C(=O)CCCc1ccncc1 N1(C(CC=CC=C)=O)CC(C(N2CCCC(C#N)C2)=O)C2(CCC2)C1 C1(C)(CC(=O)NC(c2ccccc2)C(=O)NCc2cc(CC)on2)CCOCC1 Cc1cc(=NC(C)C2CCCC2)[nH]c(=NCCSCCC(F)(F)F)[nH]1 C1(NC(C2(CN(C)C)CC2)=O)CCCC1CNC(=O)C(C)(C)C1CC1 CC(C)C(O)C(C)(C)C(=O)NC1CCCC1NC(c1cc(O)cc(O)n1)=O O=C1CC(C(=O)NC2COCC2NC(c2ccnc(N3CCCCC3)c2)=O)=NN1 c1(CC(=O)N(CCNC(=O)CCF)Cc2ccccc2)ccc(F)cc1F CCCC(O)CC(=O)NCC12CC(NC(=O)CCNC(=O)C=CCl)(CO1)C2 c1(CC(=O)NC)csc(CCNC(=O)NCCOC)n1 CC(C)C(C(=O)N(CCC(C(C)C)NC(C1(C(N)=O)CC1)=O)C)n1cnnc1 C1(NC(C(CC)(C)O)=O)CCC(C)N(C(c2cnc(OC)c(C)c2)=O)C1 c1(C(=O)NC(C2CCN(C(CC3N(C)CC=CC3)=O)C2)(C)C)ccc(N)c(N)c1 CC1(C)C(NC(C2CC(=O)N2)=O)CCN1C(c1cccc(N(C)C)n1)=O S(=O)(=O)(c1ccc(F)c(F)c1)N1CC2C(NC(c3cc4n(n3)CCC4)=O)C2C1 c1(C(=O)NCC(CNC(c2ccnc(C)c2C)=O)C)ccc(S(C)(=O)=O)cn1 CC(CCC(C)(C)C)C(=O)N1CCCC(N(C)C(c2ccnn2C2CC2)=O)C1 N1(C(CC2CC(NC(CC3N(C)CCCC3)=O)C2)=O)CC2(CCNC(=O)O2)C1 C=CCCCC(C(=O)NC1CN(C)CC12CC2)NC(c1cocn1)=O c1(CNC(C2N(CC)CCCC2)=O)cc(O)nc(CNC(=O)CN(C)C2CC2)n1 C(=O)(C(O)CC(F)(F)F)NC1(CC=C)CN(C(c2ccc(O)c(Cl)n2)=O)C1 C1(C(=O)OC)(NC(CN(C(=O)C(C)N(C)CC)CC=C)=O)CCCCCC1 c1(C(N(CC(=O)Nc2ccc(CC)nc2)C2CC2)=O)cccc2ccnn12 C1(CNC(C2(CC(C)C)CCC2)=O)CC(O)CN1C(c1cnc(Br)s1)=O c1(C(N(C)Cc2ccccn2)=O)cc(NCc2cnn(C)c2)cc(Br)c1 N1(C(c2cc(C(C)=O)sc2)=O)Cc2ccccc2C(CNC(=O)C(C)C(C)C)C1 N1(C(c2csc(CO)n2)=O)CCC2C(CCN2Cc2ccc3c(c2)CCO3)C1 C(=O)(CC1=CCOCC1)N1C(CN(C(=O)C=Cc2ccsc2)C)CC(F)C1 C1(CC)C(C(=O)NCCC2CCC(C)(C)C2)CCN1C(=O)CC1CC(=O)C1 c1(-c2n(C3C(C)OCC3)nc(-c3cccnc3)n2)cc2n(c1)CCS(=O)(=O)C2 C1(CNC(CCCC(N)=O)=O)CCN(C(=O)CC2CCC23CCC3)CC1(F)F c1(C(=O)NCC2(C)CC(NC(=O)CCSC(F)(F)F)C2)cnc2ccccn12 c1(C(N2CC(CCNC(c3ccon3)=O)(OC)C2)=O)sc(C(F)(F)F)cc1C C(=O)(CCCCc1ccccc1)NCC1(OC)CCN(C(=O)COC(C)(C)C)C1 c1(C(=O)NC2C(CNC(c3c(C)c[nH]n3)=O)C2)cc2ccc(Br)cn2n1 C(=O)(C1=CCCC1)NCC(C(C)C)NC(c1cnoc1-c1cccs1)=O C1(C(=O)NCC2N(C(CN(CCC#C)C)=O)C3CCC2C3)CN(CP(C)(C)=O)C1 C1(NC(c2c(C#C)cn(C)n2)=O)CN(C(c2sccc2COC)=O)CC1C1CC1 Cc1cc(C(=O)NCC2CCC2NC(=O)C(F)(F)c2ccncc2)co1 N1(C(c2cc(OC)ncc2)=O)CCC2(CC2NC(C2(N(C)C)CCC2)=O)C1 N1(C(c2ccc(OCC)nc2)=O)CC(F)(F)CC1CNC(C1CC(=O)N(C)C1)=O C1(NC(C(CC=C)C)=O)CC(F)CN(C(c2ccccc2Br)=O)C1 c1(CC)ccc(C(=O)NCc2csc(CNC(C3CC3c3ccccc3)=O)n2)[nH]1 C=CC(C)C(=O)NC(C)(CNC(=O)C(C)(C)C1CCCC1)Cn1cccn1 c1(CC(C)C(N2CC3C(NCc4nc(Br)cs4)C3C2)=O)cccc(Br)c1 c1(C(=O)NC2C(NC(C(F)=CCC)=O)CC2)cnnc(C)c1 c1(C(=O)NCC2CC(NC(C3(CCF)CC3)=O)C(O)C2)c(F)cc(F)cc1Cl N1(C(c2nc(CC)sc2)=O)CC(NC(=O)C(C)CC(N)=O)C2CCCC12 CC1C(NC(c2cccnn2)=O)CCN1C(C1CC2CCCC12)=O c1(C(C(=O)NC2C(O)CC2O)O)ccccc1C(F)(F)F C(C(=O)NC1CCC1C(=O)NC(C)(CO)C1CCCC1)(C(C)(C)C)OC CCC(CC(F)(F)F)NC(c1cn(CCNC(c2ccc([N+](=O)[O-])o2)=O)nn1)=O CCC(CC(=O)N1CC(CNC(C2CC2(F)F)=O)(OC)C1)C1CC1 C(=O)(C1=CCC(C)(C)CC1)NC(CC(=C)C)C(=O)NC1CC(C)N(C)CC1C N1(C(C(COC)C)=O)CC2CC2(NC(c2ccc(-c3nccs3)cc2)=O)C1 C1(CNC(C(OC)OC)=O)CCCCN1C(=O)CC1CCCOCC1 C=CCC(C)(C)CCNC(C1(NC(C2CC(=O)C2(C)C)=O)CCSC1)=O C#CCN=S(C)(=O)NCCCC(F)(F)Br.CC=O C1(NC(C2CCS(=O)(=O)C2)=O)CCOCC1NC(=O)CCOCC1CCCO1 C1(C(N2CC(CNC(=O)C(C3CC3)C3CC3)C2)=O)CCCCS1(=O)=O c1(CCC)c(C(=O)NCC(c2ccccc2)Nc2nccc(SC)n2)cnn1C Cc1cc(Cl)cnc1NC(N1CC(CC(=O)N(C)C)C1)=O c1(C(=O)NCC2(C(=O)NC3CC4(CCC4)C3O)CC=CC2)cccc2cncn12 C(=O)(CCCCC(N)=O)NC1CCCN(Cc2c(CC)nn(C)c2CC)C1 C1(CNC(c2c(C)cno2)=O)CCC2CN(C(=O)C=CC(C)(C)N(C)C)CC12 C1(S(C)(=O)=O)(C(=O)NCC(N2CC(CN(C(=O)CNC(N)=O)C)C2)=O)CC1 C1(CNC(=O)Cc2ccns2)CC(O)CN1C(=O)CSc1nncs1 C1(O)(C(=O)NCCCC(C)NC(c2cc(=N)[nH]c(=N)[nH]2)=O)CCCCCC1 c1(C(N2CC3(C(NC(C(C)O)=O)CCC3)C2)=O)ncnc2c1cnn2C C1(NC(CC(CC)CC)=O)CCC2(CC1)CC(NC(=O)C(C(C)O)N(C)C)C2 CC1CC(O)CCN(C(C23COCC2CN(C(=O)OC(C)(C)C)C3)=O)C1 CC(CC(=O)NCc1cnn(C)c1C(N1CCCC(N=[N+]=[N-])C1)=O)CC(C)(C)C C1(NC(CC(CC)C)=O)CC2(CCCN(c3ncc(Br)c(C)n3)C2)C1 c1(C(N2C(C)CC(CNC(COCCSC)=O)C2)=O)cc(Cl)nnc1O CC(C)CCCOCC(N1CCC1(C)CC(=O)NCC1CC(C(C)C)C1)=O CCCC(CC1CCCC1)C(=O)N1CCCCC(NC(c2c(C)ncn2C)=O)C1 c1(C(C(=O)N(CCN(C(=O)Cc2cccc(O)c2)CC)CC)C)ccc(F)cc1 N(C1COc2c(F)cccc21)C(C(=O)N(C)CC1CCN(c2ccccc2)C1)=O c1(CC(=O)NCC(CO)NC(C2Cc3ccccc3O2)=O)ccc2[nH]ccc2c1 N1(C(C(C)SCC)=O)CCN(C(c2cc(O)cc(O)n2)=O)CC12CCC2 C1(C(=O)NCCCC2(NC(c3nc(COC)sc3)=O)CC2)CC(C)(C)OC1(C)C C1(F)(C(N(C2CN(C(=O)Cc3ccc(Br)cc3)C2)C)=O)CCOCC1 c1(C(=O)NCCN(C(c2c(C)cnn2C)=O)C2CC2)cc2cccnc2cc1F N1(C(c2csc(-c3ncccn3)n2)=O)CCC2C(C1)CN2C(c1sccc1F)=O c1(C(N2CC(NC(C(C)SC(F)(F)F)=O)C(C)C2)=O)cc2c(O)ccc(F)c2[nH]1 C#CCC(O)C(=O)N1CCC(CN(C(=O)COCC(=O)OC)C)C1 c1(C(N2CC(NC(C(C(C)C)C)=O)C(O)C2)=O)cc([N+](=O)[O-])cnc1O c1(C(=O)NCC2(CCNC(C3C(C)(Br)C3)=O)CC2)ccc(OCF)cc1 C1(NC(C(CC#C)C)=O)CCN(C(c2nc(CC)ncc2Cl)=O)CC1F c1(NN(C(=O)NC(CC)C)C)ccc(S(=O)(=O)NC2CC2)cn1 C1(C)(CNC(C(CC2CC2)OC)=O)CC(F)(F)CN1C(=O)C(C)OC c1(C(N2CC(NC(C(C)n3cnnn3)=O)(CO)C2)=O)oc2ccccc2c1CO N1(C(CCNC(COC)=O)=O)CC2OCC(NC(c3cc(C4CC4)[nH]n3)=O)C2C1 Cc1cn2c(n1)CCC(NC(C)Cc1c(C)nn(-c3ccccc3)c1C)C2 N1(C(CCc2ncc(C)[nH]2)=O)CCN(C(c2c(C)cncc2C)=O)CC1C(C)C CCCC(C)CCN=c1[nH]c2c(c(=NCCC3(CSC)CC3)[nH]1)COC2 C(=O)(CS(=O)(=O)C1CCCC1)NCC1(O)CN(C(=O)CC2CCCC(C(F)F)O2)C1 C1(CC)COC(C)(C)CN1C(=O)CCN(C)C(C1(O)CCCCC1)=O C1(NC(C(C)CC2CC2)=O)CC2CC1N(C(c1ccnc(OC(F)F)c1)=O)C2 Cc1c(Br)ccnc1N1CCN(C(=O)C(N2CCCC(O)C2C)=O)CC1 C1(C(N2CCC(CCNC(=O)CCc3cc(C)[nH]n3)C2)=O)(COC)CCCC1 N1(C(C=C(C)C(F)F)=O)CCC2(CCC(NC(=O)CCN3CCOCC3)CC2)C1 c1(C(=O)NC(CC(C)NC(CCCC)=O)C)c(OCCCOC)cccc1Cl c1(CNC(C(C)N(C)C)=O)cc(C(=O)NC(c2ccccn2)CO)cs1 Cc1cc(CC(=O)NC2(CCNC(=O)CC3CC4CC4C3)CCCC2)ccc1O C(CCS(=O)(=O)c1ccccc1)NC(C1(N)CC(F)(F)C1)=O C(=O)(C1=CC2CCC1C2)N1CCN(C(COCc2onc(CC)n2)=O)CC1CO c1(OCC)cccc(CC(N2CCCC(CCNC(c3cnns3)=O)C2)=O)n1 N1(C(C(COC)C)=O)CCC2C1CCCN2C(=O)COCP(C)(C)=O c1(NC(C)CCNC(c2ccc(Cl)nc2Cl)=O)nc2c(cc1C#N)CCC2 C12(NC(=O)Cc3cc[nH]n3)CCN(C(c3ccc(O)c(F)c3)=O)CCC1C2 C(CC(=O)NC1COC(C(C)C)C1)(C(F)(F)F)NC(c1c(OC)scc1)=O c1(-n2ccc(C(=O)NCC(C)NC(C(C)=CC)=O)n2)c(F)cccc1F N1(C(C(c2ccccc2F)(C)C)=O)CC2(CCC2NC(C2C=CCC2)=O)C1 c1(C(=O)NCC2N(C(CCCOCCOCC)=O)CC2)ccc(Cl)c(S(C)(=O)=O)c1 C1(C#N)(C(=O)NC(CNC(c2c(C)scn2)=O)C(C)(C)C)CC2CC2C1 N1(C(c2c(C)onc2)=O)CCN(C(=O)CCCC(F)(F)F)CC12CCC2 C1(CNC(CC2C(C)C2(F)F)=O)CN(C(c2cnn(CC3CC3)c2)=O)CCCO1 c1(NC(C)=O)cnccc1C(=O)N(C)CC1CCN(C(=O)CC2(C)CCCO2)C1 N1(C(Cc2ccc(C)o2)=O)CCOCC(CNC(c2cc(C(F)(F)F)cs2)=O)C1 CC1CC(C(N2CCC2CNC(C2(F)CCC2)=O)=O)CCO1 CCCCC(F)C(=O)N(C)CC1CCC(NC(C2CCCN(C)C2)=O)CC1 C(=O)(NN1CCCC(C(=O)O)C1)C1(N)CCCN(C(C)=O)C1 N1(C(c2cocn2)=O)CCCCC2(CCN(C(C3CCC4(CCC4)O3)=O)C2)C1 N1(C(CC(CC)OC)=O)CCCC(C2CCN(C(=O)CCc3cnc(C)o3)C2)C1 c1(C(=O)NCCN(C(=O)C(C)Cc2cnc[nH]2)CC)cc(C)cc(Br)c1 c1(C(=O)NC(CCNC(CCOCCOCC)=O)C)cnc(C)s1 c1(CC(=O)NCC2(NC(c3ccc[nH]3)=O)CCC2)noc2ccccc12 C(=O)(C(C)CC(=O)NCC1CCCN1C(=O)COCc1ccnn1C)OC N1(C(c2cnn(C(C)(C)C)c2N)=O)CCC(CO)C(NC(c2ccccn2)=O)C1 N1(C(CC(CC)C)=O)CC2(CNC(c3cn(C(C)(C)C)nn3)=O)CC1CO2 N1(c2ncc(C(=O)OCC)cn2)CC2CCCN(C(=O)C(F)CC)C2C1 c1(C(=O)NC(C)CCN(C(=O)Cc2ccn(C)n2)C)ccccc1C1CCC1 Cc1ccc(C(N2CC(NC(=O)Cc3cc(Br)ccc3Br)C(C)C2)=O)cc1F C(CC(=O)NCCN(C(c1cnn(C(F)F)c1)=O)CC)(C1=CCCC1)OCC C(=O)(C(C)(C)C1=CCSCC1)NCCC1CCC(NC(CC2(C)CC2)=O)C1 N1(C(C2(OCC)CCCC2)=O)CC(NC(=O)CN2CC(=O)N(C)C2=O)CC(C)C1 Cc1ccc(I)cc1NC(C1CCCN(C(=O)Cc2cccs2)C1)=O C=CC1CN(C(=O)C(C)SCC)CC1NC(c1ccc(F)s1)=O CC(CNC(c1ccc(Cl)o1)=O)CC(=O)NC1CC12CC(O)C2 C1(CNC(C(CCC)(C)C)=O)C2CCCC1N(C(c1cc(=N)[nH]c(Cl)n1)=O)C2 Cn1ccnc(Nc2cccc(NC(c3cnn(CCN)n3)=O)c2)c1=O C1(NC(c2nc(CCC)oc2)=O)CC2CCC1N2C(=O)CC(C)c1ccco1 N1(C(c2c(CC)nn(C)c2)=O)CCC2C1CCCN2C(=O)CCC1CC1(C)C c1(NC(=O)NC(CC)C2CC2)ccc2nc3n(c(=O)c2c1)CCC3 C(=O)(CN=c1cc[nH]cc1)N1CCC(CC=C)(C(N(C)CP(C)(C)=O)=O)C1 C1(O)(CNC(C(C)NC(c2c(C)occ2)=O)=O)CCCN(Cc2ccccc2)C1 CC1Cc2sc(C(N3CC(NC(c4cccc(F)c4Cl)=O)C3)=O)cc2C(C)C1 N1(C(c2cc(OC)nn2C)=O)CCN(C(C2CCC(=O)N2)=O)CC1c1ncc[nH]1 CC(C)(C(=O)NCCCC1CCOCC1)NC(=O)CC1COCCO1 C1(NC(CCC(=C)Br)=O)CCC2(CC1)CN(C(C1CCC1)=O)CCO2 c1(C(N(C(C)CCNC(c2c[nH][nH]c2=N)=O)C)=O)ccc2c(O)n[nH]c2c1 c1(SC)ccc(C)c(C(=O)NC2(CCCNC(=O)C(O)C(C)C)CC2)c1 Cc1cc(C)c2cc(C(N3CCC3CNC(=O)C3=CCCOCC3)=O)[nH]c2c1 CCCC(C#N)C(=O)N1CC2(CC(NC(=O)C(C)OCCC(C)C)C2)C1 C(=O)(CN=S(C)(C)=O)NC1C(NC(C(CC)Sc2nc(=N)[nH][nH]2)=O)CCCC1 C1(CNC(C=CC=CC)=O)CCCC(CNC(c2cc(CC)ncn2)=O)C1 Cn1cc(CCC(=O)NCC(O)CNC(C2(CO)CCCC2)=O)nn1 C(=O)(C1=NOC2(CCOC2)C1)N1C(CNC(c2ccn(CCF)n2)=O)COCC1 CCC(O)C(C)C(=O)NCC1(NC(c2cn(C)nc2Cl)=O)CCOC1 N(C1C(=O)Nc2c(Br)cccc21)C(c1cccc(-n2cccc2)c1)=O C(N=c1[nH]c(=NCc2cccs2)c2ccccc2[nH]1)C1C(CCC)CCC1 C1(O)(CCNC(c2csnn2)=O)CCN(C(c2ccc(O)c(F)c2)=O)CC1 c1(C(=O)NC(C=C)CO)cn2c(C)ccc(-c3cccc4c3OC(F)(F)O4)c2n1 c1(OC)cc(C(=O)NC2CC2CNC(c2csc(CO)n2)=O)ccc1NC1CC1 c1(N(CCCCCCC)C)nc(=NC(C)c2nnc(COC)s2)[nH]c2c1CCC2 c1(CC)nc(C)oc1C(=O)N(C1CN(C(=O)C(CC2CC2)OC)CC1O)C C1(C(=O)NCC(CNC(=O)CCCN(C)C)OC)(OC)CCC12CCC2 N1(C(C2C(C)C2)=O)CC2(CCC(NC(=O)Cn3ccnn3)CC2)C1 c1(N(C)C)ccc(C(=O)NCCOC2CCN(C(=O)C(C)(O)C3CC3)CC2)cc1 c1(CN2CCC(NC(C3CCN(CC)C3)=O)C(O)C2)cc2c(OC)cccc2[nH]1 Cc1csc(NC(C2CC(F)CN2C(C2CC2F)=O)=O)c1C#N C1(CNC(C(F)OC)=O)CCN(C(c2ccc(C)nc2O)=O)C12CC2 N1(C(C2CN(C)C2)=O)CC2(CO)CC1(C(N1CCC=C(F)C1)=O)C2 c1(C(N(CCNC(C2N(C=O)CCC2)=O)CC2CC2)=O)cc2sccc2[nH]1 C#Cc1cc(C(N2CCC(CNC(C3(c4ccn(C)n4)CC3)=O)C2)=O)cc(Cl)c1 N(C1CCCc2ccc(F)cc21)C(N1CCC2(CCCNC2)C1)=O C1(CCC)CN(C(=O)CCCNC(N)=O)CC1C(=O)NCCN1CCCC(O)C1 N1(C(C(CCC)OCC)=O)CCC2(CCC2)C(NC(c2oc(C)nc2C)=O)C1 C1(C(C)C)CN(C(C2(F)CCN(C(=O)CC3(C)CCOCC3)CC2)=O)CCCO1 c1(CC)ncc(C(c2nnnn2C2CCCCC2)NC(c2cccs2)CC)[nH]1 c1(OCC(=O)NCCCCN(C)C(C2CCC3CC23)=O)cccc(F)c1F C1(C(N(C(CCNC(C2ON=C(CC)C2)=O)C)C)=O)CC2CCC1CC2 c1(OCCCC)ccc(C2(C(=O)NC3CC(NC(=O)C(F)(F)C4CC4)C3)CC2)cc1 C(=O)(C(C)CC(N)=O)N(CC(N1CCN(C(CC=CCC)=O)CC1)=O)C c1(CCNC(C2CC2Cl)=O)c[nH]c2ccc([N+](=O)[O-])cc12 c1(C(N2CC(C)C(NCc3ccc(Cl)s3)C2)=O)cccc(O)c1[N+](=O)[O-] N(C(=NCC(=O)NCc1nnnn1C1CC1)NC1CC1)CC(C)(C)C N1(C(c2ccc(CC)nc2)=O)CCC(O)C(C(=O)Nc2ncc(O)cc2Cl)C1 c1(C(N2CC(OC)(CNC(c3scnc3C(C)C)=O)C2)=O)cc(F)cc(C)c1N N1(C(C(C)N2CCC2)=O)CCOCC(F)(CNC(=O)CCc2cn[nH]c2)C1 c1(OC)ccc2[nH]c(=NCCc3ccnn3C)nc(N3CCSC(C)(C)C3)c2c1 CCC(CC(=O)N1CCCC(C(N2CC[Si](C)(C)C2)=O)(CC)C1)C(F)F Cc1cnc(CN2C(C(N3CC4CC4C3)=O)CC3CC23)c(F)c1 c1(C(N2CCC(C3N(C(C(F)OC)=O)CCC3)C2)=O)nc(Cl)sc1Cl c1(C(N2C3C(NC(CCC(=C)C)=O)C(CC3)C2)=O)c(C2CC2)nc2sccn12 Cc1ccc(CCCn2cc(CN(O)C(=O)N(C)CC3CCCC3)nn2)o1 C(=O)(C(C)(C)C(C)(F)F)NC(C1CC(NC(c2c(C)occ2)=O)C1)C C1(NC(c2c(C)[nH]nc2C(C)C)=O)CCN(C(=O)C(=O)N(C)C)C(C2CC2)C1 C1(C(=O)NC(C)CCNC(=O)CC2CC2(Cl)Cl)CCOC2(CCCCC2)C1 C1(OC)(OC)C(C(N2CCC(C(=O)OC)CC2(C)OC)=O)CC1(F)F Cc1ncc2cc(C(=O)NCC3CCCN3C(=O)CC(C)CC(C)C)ccn12 CCCC(CC)C(c1nnnn1CC(F)F)NCCc1cnccc1C CC(C)(COC1CCCC1)C(=O)NC1CCOCC1NC(=O)Cc1cnsc1 C1(NC(Cn2c(CC)nnc2S)=O)CCCC(NC(c2cc(C)nc(C)n2)=O)CC1 CC1(C)CC(CNC(=O)C(CCF)NC(C2CC3(CCC3)C2)=O)CCO1 C(=O)(CCCCC(F)F)NCC1CC(O)(CNC(=O)Cc2nnc(O)s2)C1 c1(C(N2CC(O)CC(NC(CCC(C)N(C)C)=O)C2)=O)ccc(F)c(Cl)c1F c1(C(=O)NCC(CC)NC(C2CC3CCC2O3)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NC(CNC(c2nc(C)sc2)=O)(C)CO)cccc2occc12 C(=O)(CN=c1cc[nH]cc1)N1C(CNC(c2ccccc2Cl)=O)CC(O)C1 C(CCC(=O)N=c1ccn(C2CCC2)[nH]1)NC(=O)CC=Cc1ccccc1 CC(C(F)C(=O)NC(C)CC1CN(C(c2sccc2C2CC2)=O)C1)C(F)(F)F c1(C(=O)NCC(C(C)(C)C)NC(c2cn(C)c(=O)cc2)=O)cccn2cncc12 C1(C(N2C(C)(CCC)CC2)=O)CC(C)CCN1C(c1cc(O)nn1C)=O C1(CNC(C(=O)N(CCC)Cc2ccc(Br)cc2F)=O)CC12CCOCC2 c1(C(=O)OC)cc(C)c(C(N2CCC2CNC(c2cnn(C3CC3)c2)=O)=O)o1 c1(C(N2C(CCCNC(c3cc(CC)no3)=O)CCC2)=O)cccc(=O)n1C c1(OC)cccn2ncc(CNC(c3nc(COC)no3)c3ccccc3)c12 CC(=O)CCCC(=O)NC(C(=O)NCc1cc(=O)cc[nH]1)C(C)C c1(C(=O)NCC(CC)N(C(=O)CC2CNC(=O)O2)C)ccc(C)c(C)c1F N1(C(c2c(C)nc(C3CC3)o2)=O)CCCCCC1CNC(c1ccc(C2CC2)o1)=O c1(C(N2C3CCC2CC(N2CCCC(CCO)C2)C3)=O)cnn2cccc(F)c12 CC(CS(=O)(=O)Nc1ccc(N2CC(C)(O)C2)cc1)C(C)(F)F c1(CNC2CC(NC(c3c(C)ncs3)=O)C2)cc([N+](=O)[O-])c(Cl)cc1F N#Cc1c(Cl)nc[nH]c1=NCC(CNC(=O)C=Cc1ccccn1)C(F)(F)F N1(C(C(=Cc2cn[nH]c2)C)=O)CC(CNC(C2CC2(F)Cl)=O)CC1(C)C N1(C(c2c(C)nn(C)c2)=O)CCCC(O)(CCNC(C2C(C)C2(F)F)=O)C1 c1(C(=O)NCC2CCCCN(C(CCC(C)(C)F)=O)C2)cc2n(n1)CC(F)C2 c1(C(=O)Nc2n(C)nc(CO)c2)c(-c2ccc(F)nc2F)ccc2c1OCO2 C1(NC(c2n(C)ccn2)=O)CN(C(=O)C(C)(C)C(N)=O)CC12CCC2 C(=O)(C1=NOC(CNC(C2CNC(=O)N2)=O)C1)N1C(C)(CC(=O)NC)CCC1 C(=O)(N1CCC(C(=O)NCC2CCC2CO)O1)C1CN(C)C1 CCC(CC(F)(F)F)OC(c1cnn(C2CC2(F)F)c1)=O C12(NC(c3c(C)nc(CC)s3)=O)CC(CNC(=O)C=C(C)C(C)(C)C)(C1)OC2C CC1(C)CCCC(C(N2CCC(C(F)F)C2)=O)C1 N1(C(c2sccc2F)=O)CCN(C2CN(C(c3[nH]nnc3C3CC3)=O)C2)CC1 C1(C(=O)NCC(CC)NC(=O)C=C2CCC(C)C2)(OCC)CCCCCC1 CC(C)(CCCNC(C1CC(C)(C)C1)=O)NC(C1CC1C(F)(F)F)=O c1(NC(N)=O)ccc(Cl)c(C(N2CC(NC(C3CCCCNC3=O)=O)C2)=O)c1 C1(C(=O)NC2C(NC(c3ccc(-c4ccccn4)s3)=O)CC2)CCC=CCCC1 CC1C=C(C(=O)NCc2ncoc2C2CN(C(=O)C3=COCCO3)C2)CC1 C12(CNC(CC3(C)CCCO3)=O)CCC(CC1)N(C(c1ccnn1C(F)F)=O)C2 Cc1ccc(OCC(=O)NC(CNC(c2ccc(=O)n(C)c2)=O)C2CC2)c(Cl)c1 N1(C(C(F)OC)=O)CC(CNC(C2(CCF)CCOCC2)=O)C2(CCOCC2)C1 N1(C(C(=O)NC(C)C)=O)CCCCC1CC(=O)NCC(C)C1CC1 n1(CC(=O)NCC2C(NC(CC(CC)SC)=O)CCC2)nc(C)ccc1=O C1(C)(C(=O)NCC(CC)(CC)NC(=O)C(F)CN(C2CC2)CC)CC2CCC1C2 N1(C(CCCCCCC)=O)CC2COCC(C1)C2NC(c1coc(CC)n1)=O C(=O)(N=c1ccn(CCCO)[nH]1)C1(CC=C)CCN(C(=O)C=C(C)COC)C1 CCCC(CCC)=CC(=O)NCC1CC(C(N2CC(F)(CC)C2)=O)C1 c1(C(=O)NC(CC)CC2CC2)ccc(C(F)(F)F)nc1C(F)(F)F N1(C(C(C2CCN(C(c3c(OC)n(C)nc3)=O)CC2)C)=O)CCC(CO)CC1C C=CC(C)(CC)C(=O)N(CCCNC(=O)CCCn1c(C)csc1=O)C N1(C(c2c(SC)csc2)=O)CCC(CN(C(=O)CC(C)F)C)CC1 C(=O)(C1=CCCN(Cc2cc(F)cc(Br)c2F)C1)NC(CC=C)CO CC1(NC(c2ccc(CO)cn2)=O)CCN(C(=O)C=CC(N)=O)C1 C(=O)(C(C#N)C(C)(C)C)N1C(C(=O)Nc2cccc(C)c2F)C(C)(C)CC1 c1(CC)cnc(Cl)[nH]c1=NC1CCCN(C(=O)Cn2nc(C)cc2C)CC1 C(=O)(C(C)(CO)NC(c1ccoc1)=O)N(C(CC)CC)C C1(NC(c2c(CC)oc(C)n2)=O)CC12CCC(NC(=O)CCNC(=O)OC)CC2 c1(CC)ncccc1C(=O)NC(Cc1cnc[nH]1)C(=O)N(CC(C)CO)C c1(NC(C2CCN(C(c3c(C)oc(Cl)n3)=O)C2C)=O)ccc(O)c(Cl)c1 CC1CN(C(C2(C)CN(C(=O)CC3CCCN(C)C3)C2)=O)CCCO1 Cn1ncnc1CCCNC(=O)C=CCC1(N(C(=O)CSC(F)F)CC)CCC1 C(CC(=O)NNC(=O)c1cc2ccccc2[nH]1)(C(F)(F)F)OC(C)(C)C O=C1N=C2NNC(=C2C(=O)C=Cc2csc(Br)c2)C1=O.c1(S)ccccc1 c1(C(N(CC(=O)N(C)CC2CCOCC2)C2CC2)=O)ccncn1 c1(C(N2CCCC(C(=O)NC3CCS(=O)(=O)C3)CC2)=O)c(O)cc(O)cc1O c1(C(N2CCC(CC#C)(C(=O)NCC(C)OC)C2)=O)ccc(O)c(CO)c1 c1(C(=O)NC)ccnc(O)c1-c1csc(C(=O)Nc2ncccc2NC(C)=O)c1 C1(C(N2CC(O)(C(C(=O)NCc3scc(C)n3)F)C2)=O)CCC(=O)NC1 Cc1ccc(F)cc1-c1cn(C2CN(C(C3CS(=O)C3)=O)CC2C)nn1 c1(C(=O)NC2C=CCN(C(C3(CC)CCC(O)CC3)=O)C2)ccn2ncnc2c1 c1(C(CN2CCC(c3ccc(OC)c(SC(C)C)c3)C2)=O)ccccc1S(C)=O C12(C(=O)NC3CCN(C(CC4(CC=C)CCCC4)=O)CC3)CCC(F)(CC1)CC2 c1(CC(N2CC(NC(c3ccc(C=C)cc3)=O)C3C2C3)=O)ccc2occc2c1 C=Cc1ccc(C(=O)NC2CC3(C2)CC(Nc2ncncc2I)C3)cc1 CCCCC(CC(=O)N1CCCCC1CF)NC(C1C(C)C1C)=O N1(C(C=CC(CC)C)=O)CC(CNC(=O)CCCC2CCC2)(OC)C1 c1(C(N2CC(C)CC(NC(C(C)NC(N)=O)=O)C2)=O)cncc(P(C)(C)=O)c1 CC1CN(c2nc(=N)nc(N3CC4CC4(CO)C3)[nH]2)CCC1(F)F c1(C(N2CCN(C(C3N(CC)CC3)=O)C(CO)C2)=O)cc2c(NC)cccc2s1 N1(C(CC(C)O)=O)CCCC(NC(c2nnc(S)n2C)=O)C1C CCCC(C(=O)Nc1ccnn1-c1ccccc1OC)NCC(c1ccccc1)=O C(N=c1cc(CC(C)C)nc[nH]1)C1CCN(C(CCc2ncc(C)[nH]2)=O)CC1C Cc1cc(N)cnc1C(=O)NCCCCC(C)NC(C1(C(C)C)CCCO1)=O C(=O)(CC1OCCc2ccsc21)NCCOCCNC(C(c1ccnn1C)C)=O N1(C(C2C(=C)C2)=O)CC(NC(=O)CC2CCS(=O)(=O)C2)CC1C c1(C(C)C)cc(CC(=O)NCC(C)(F)CNC(C2(CF)CC(=O)C2)=O)on1 C(=O)(CC(CN(C)C)C(F)F)N(C1CC(NC(c2c(C)cccn2)=O)C1)C C1(C(N)=O)(C2CC2)CN(C(=O)COCCSCC#N)C1.C1(C2CC2)CC(=O)N1 Cc1nc(N(C2CC23CCNCC3)C(c2cc[nH]c2)=O)c2sccc2n1 c1(C(=O)NCC2N(C(CC(=O)OC)=O)CCOC2)c(Cl)c([N+](=O)[O-])nn1C C1(CC(N2CCC(NC(CC3CC(CC)C3)=O)(CF)C2)=O)CCCCC1(C)C C(CO)(C(C)NC(=O)C(CO)NC(N)=O)NC(C1(CCC)CCC1)=O c1(C(=O)NCC2N(C(c3cc(CC)oc3C)=O)CCC2)cc2nc[nH]c2cc1F N1(C(c2c(C)nc(C)[nH]2)=O)CC(CNC(C2CCCS2)=O)CC12CCOCC2 CCC(C)CC(=O)N(CCCCN(C)C(c1nn(CC(C)C)cc1C(F)F)=O)C c1(CC(=O)NCc2cc(OC)c(O)cc2)cnc2ccccc2c1 CC1CCC(CNC(c2cccc(O)c2F)=O)CN1C(c1cnns1)=O c1(C(=O)NC(C)(CNC(=O)CCCn2ccnn2)CO)coc2ccc(Cl)cc12 C1(NC(c2ccnc(N3CCCC3)c2)=O)CCC2(CC1)CC2NC(C1CCO1)=O C(=O)(CCCCC(F)(F)F)N1CC2C(NC(c3cccc(C)c3N)=O)(CCC2)C1 N1(C(c2c(COC)ncs2)=O)CCCC2CN(C(=O)C(C)(O)C(C)C)CCC12 CC(C)C(F)(CN)C(=O)Nc1cc(CN)cc(F)c1 Cc1cc(F)cc(C(=O)NC2CC(NC(=O)Cc3ncn4c3CCCC4)C2)c1N C#CCCC(O)C(=O)NCC1(CNC(c2cnc(C)nc2C)=O)CC1 c1(C(N2CC3C(NC(c4cn5c(n4)CCC5)=O)(C3)C2)=O)ccc2c(c1)CNC2=O O=C1Cc2cc(C(=O)NC3CC(NC(C4CCCS(=O)(=O)N4)=O)C3)ccc2N1 c1(C(=O)NC2CC(CNC(=O)C=CC3CCCC3)C2)cc(CO)ccc1Cl C1(CC)CCCN1C(=O)CC1(N(C)C(C2(C3CCCO3)CCC2)=O)CC1 c1(C(=O)NCCCN(C(=O)C(C)SC(F)(F)F)CC)occ2c1CCCC2 N1(C(COCCCC)=O)C2CCC1CN(C(c1ccno1)=O)CC2 C1(C(=O)NC2CC(N(C)C(c3ccc(CN4CCCC4)o3)=O)C2)CC(F)C(=O)N1 c1(C(N2CCN(C(CC=C)=O)C3C2CC3)=O)cc2c(Br)cccc2cn1 c1(CC(=O)NCC(C)N(C(c2c(CC)con2)=O)C)cnccc1C CC(CC1CC1)C(=O)N1CC(C(N)=O)(CNC(=O)COc2ccon2)C1 CC1CN(C(=O)C(C2CCCC2)NC(C2CC2(C)C)=O)CCC1O C1(C(N(C(C(CC)C)C)C2CC2)=O)CN(C(c2cc(C)oc2C)=O)CC1(F)F C1(NC(c2c(C)snn2)=O)CC2(CCN(C(=O)C(C)SC(C)C)CC2)C1 CC1(C)CCCCC1CC(=O)NC1(C)CCN(C(c2cc(O)cc(O)n2)=O)C1 C12(C(N3CCCC(C)C3CO)=O)CCC(CC1)N(C(=O)C(O)C1CCCC1)C2 N1(C(c2ccc(N(C)C)cc2)=O)CC(CNC(=O)CCC(F)(F)F)OC(C)(C)C1 C12(CNC(C(CC)CC)=O)CC(COC)(CN1C(c1cc(C3CC3)nn1C)=O)C2 C(CNC(=O)C1=CCCC1)(CC(=O)N(C)CCc1cccnc1)OC CC1(C)CC(S(=O)(=O)C(N2CCN(c3ncc[nH]3)CC2)=O)CCO1 C1(CNC(C(C)N(C)C)=O)CN(C(=O)CC2CC2C)CCC12CCOCC2 Cc1ncnc(C)c1CC(=O)NC(C)C(C)NC(=O)COc1ccc(O)cc1 c1(CC(C(=O)O)OCCN(C)CC2CC2)cccc(OC(F)(F)F)c1 C#Cc1cnc(NC2CCN(C(c3ccc(C(C)C)cn3)=O)C(C)C2)nc1 N1(C(c2cnco2)=O)CC2CN(C(c3c(O)cccc3Cl)=O)CC2C1 Cc1ncnc(C)c1CC(=O)NCC(CO)NC(=O)C(c1cccnc1)O C1(CC)CN(C(=O)C(O)CN(C)C)CC1C(=O)NC(c1cccnc1)CC c1(NC(c2cn(C3CCC(=O)NC3)nc2)=O)ccc2nc(O)[nH]c2c1 N1(C(C2N(C(CC3CC(CC)C3)=O)CCC2O)=O)CC2(C1)OC(=O)NC2C C1(C(=O)NC2C3(CC(NC(c4ccn(CCCC)n4)=O)C3)C2)CCC2CCC1O2 C=CCC(CCCCC)C(=O)NCC(CC)N(C)C(C12COCC1C2)=O C1(C(N2CCC(C(=O)NCCCCCO)C2)=O)CCc2ccccc2C1O c1(CC(C)C)ccc(C#N)c(NC(C2CCCCN2C(C2CC=CCC2)=O)C)n1 Cc1ccccc1-n1cc(CNC(=O)CN(C2CCC2)C(c2ncc[nH]2)=O)nn1 C12(C(=O)OC(C)(C)C)CCN(CC1)C2=O.N1(OC)C2CCC1C(CO)C2 C(=O)(CCCC(N)=O)NC1CCN(CCNC(c2ncc(C)nc2)=O)CC1 c1(C(=O)NCC2CC(C(=O)NC(c3ccco3)CO)CO2)cnn2c1OCC2 C12(C(=O)NCC(CN(C(c3snc(C)c3N)=O)C)C)CC1Cc1c[nH]nc12 Cc1nc2cc(O)nn2c(C)c1CC(=O)NCC1(O)CN(C(=O)COCCF)C1 Cc1cc(C)c(C(=O)NC2COCC2NC(C2(F)CCCN(C)C2)=O)c(C)n1 C(=O)(CS(=O)(=O)C(C)(C)C)NCC(C)CN(C(=O)CC1CC1C1CC1)C N1(C(Cc2cnc(C)s2)=O)CC2CC1CN2C(c1snc(C)c1N)=O N1(CC)C(=O)CCC1CC(N1CCCCC1CNC(=O)C=CCN1CCCC1)=O N1(C(C)=O)CC(NC(c2nccn2-c2ccccc2)=O)C(c2ccccc2)C1 C(CC(C)(C)CC(=O)N1CC(CC(=O)Nc2cc(C)c(F)c(C)c2)(OC)C1)OC C1(C(=O)NCCCN(C(=O)C(C)=C(C)C)CC)CCC(=O)CC1C C1(NC(C(C(CNC(C2(C(C)C)COC2)=O)C)F)=O)CC2C(O)C(O)CC12 C1(OC)CCCC(CC(=O)NCC(C)=CC(=O)NC)C1.C1C(=O)N1C1CC1 C1(CNC(c2ccc(OCCC)cc2C)=O)CCOCC12CCC2 C1(CC(=O)OC)(CC(=O)NCCNC(=O)C(C)OCc2cccnc2)CCCC1 C1(C(=O)NC2C(C)(C)C(C(N3CC(c4nc(=O)o[nH]4)C3)=O)C2)CC(=O)NC(=O)C1 c1(C(=O)NCC(C)NC(C(c2ccc(C)cc2)C(C)C)=O)nc2ncccn2n1 c1(OCC(N2C3CN(C(c4cccnc4)=O)CC32)=O)ccc(Br)c2ncccc12 c1(C(=O)NCCCCCN(C(CCN(CCC)C)=O)C)sc2ncccc2c1N c1(CNCC2(C(=O)NCc3cc(C)no3)CC2)cncc(C#N)c1 c1(COC)ccc(NC(C2CCN(C(c3nc(C4CCC4)co3)=O)C2)=O)cc1 Cc1cccc(Cl)c1CC(=O)NCC(C(C)C)NC(=O)CCCCF N1(C(C(C(CC)O)C)=O)CCOC2(CCN(C(c3ccnc(Cl)c3N)=O)C2)C1 C1(F)(CNC(C2CC(=C)C2)=O)CCC(CNC(c2nc(Cl)c(CC)[nH]2)=O)CC1 CCC(CC(=O)N1CCN(C(=O)Cn2cc(Cl)cn2)C(C)C1C)CC(C)C N1(C(C)=O)C2CCC1CC(NC(=O)C(c1ccc(Cl)c(Br)c1)(F)F)C2 CCC(CNC(c1cc(OC)ccn1)=O)N=c1cc(C2CC2)nc(Cl)[nH]1 c1(C(N2CC(C(C)NC(=O)CC3C=CCCC3)C2)=O)n[nH]c2cc(OC)ccc12 c1(N(CC(C)C)C)ccc(C(=O)NC2CCCC2NC(=O)Cn2cncn2)cn1 C1(C(C)NC(CCNS(CC)(=O)=O)=O)CCN(C(=O)CC2(O)CCCOC2)CC1 c1(C)cc([N+](=O)[O-])ccc1F.c1(O)cncnc1N(C(C1CCCNC1)C)CC C1(NC(c2c(CC)ocn2)=O)CC(F)CN(C(=O)CCCc2ccccc2)C1 C(=O)(C(C(C)C)NC(=O)C(CNC(=O)C(=O)NCC1CC1)CSC)OC C1(NC(C2CCCN(c3nccs3)C2)=O)CN(C(=O)C2=CCC2)CC12CC2 C(=O)(C(F)(F)C(F)(F)F)NCC1(F)CCN(C(c2ccc(OC)c(N)n2)=O)C1 N1(C(Cc2c(C)oc(C(F)(F)F)n2)=O)CCN(C(C2(C3CC3)CC2)=O)CCC1C c1(CCC)noc(CCCC(=O)NCC(CO)NC(c2cc[nH]c2)=O)n1 C1(C)(C(N2CCCC(NC(CNC(=O)OCC)=O)C2)=O)CC(C(C)C)=NO1 c1(C(N(C(CN(C(C(C)C2CC2)=O)C)C)C)=O)ccccc1C(F)(F)F C(=O)(C1=CCCCC1C)NC(CC=C)CC(=O)NC(c1nc(C)no1)C CC1CCCCN1CCC(=O)NCCNC(C1CCC(=O)NC1)=O N1(C(CCCN(C(=O)OC)C)=O)CCC(CC(N)=O)(NC(C2CCSC2)=O)CC1 N1(C(CCC=C)=O)CCC(O)(CCNC(C2(COC)CCCO2)=O)C1 C(=O)(CCC(C)CN(C)C)NC(C)CCNC(c1cnn(-c2ccccc2)c1F)=O N1(CC(=O)N(CC(C)NC(C2(CCF)CCC2)=O)C)CCCC(C(F)(F)F)C1=O CC1CN(C(c2csc(=NCc3ccn(C)n3)[nH]2)=O)CC(=O)N1 C#CCC(CC(=O)N1CCOC2CC12)NC(=O)C(=O)C(C)CC Cc1cccc(C(=O)NC2CN(Cc3cccnc3)CC2F)c1C c1(C(N2CC(C(C)NC(c3ccns3)=O)C2)=O)cc(C(F)F)no1 N1(C(C(CCCC)C)=O)CCC(C)(C)C(CNC(c2cnn3ccn(C)c23)=O)C1 c1(C(=O)NCCCCCCn2cc(C(C)(C)SC)nn2)cccc2ccn(C)c12 C1(CCC)(NC(=O)COCC)CCN(C(=O)CCCC2CC(C)=NO2)CC1 c1(-c2scc(-c3nc(CCCC)nn3CCCO)n2)ccc2c(c1)OCO2 N1(C(CCCOCCC)=O)CCC(CC(N2CCC(C)(C)C2C)=O)C1(C)C C1(CC)COCCN(C(=O)C(C)Oc2ccc(C3CC3)cc2)C1 N1(C(CCCSCC)=O)CC2(CCNC(=O)CNC(=O)C(C)(C)C)CCC1CC2 C1(N(C(C(CC)SC)=O)C)CCN(C)C1(C)C.C12CCC1C(=O)NC2 c1(C(N2CC3(CCN(C(C(C4CC4)OC)=O)C3)C2)=O)cnc2ncnn2c1N C12(NC(c3c(COC)cccc3)=O)CCN(C(c3cn4c(n3)SCC4)=O)CC1C2 N1(C(CCc2n(C)ccn2)=O)CCC(F)(CNC(=O)Cn2cnnc2O)C1 c1(C(N2C(CCC)(C(=O)OC)CCC2)=O)cc2nc(C)cc(C(F)(F)F)n2n1 CC1CCN(C(C2CC3(CSC3)C2)=O)CC1NC(c1ccnc(CO)c1)=O N1(C(CCCNC(C)=O)=O)CCC2CC2(NC(C2(C(=O)N(C)C(C)C)CC2)=O)CC1 N1(C(C2CCC(=O)N2)=O)CC2(CC(NC(c3ncccc3Br)=O)CO2)C1 Cc1ccc2c(c1)CC(C(=O)NCC(C)N(C(=O)C1=NOC(C)C1)C)S2 c1(OC)nc(C)ccc1C(C(=O)NC1CC(F)(F)C1)N(C)Cc1cnc(C)s1 CCCCC(C(=O)NC(c1cn(C)nn1)C(=O)NC1CN(C)CC1O)N(C)C C1(C(=O)NCCc2ccncc2)CC2OCCC2N1C(=O)CCc1ccccc1 c1(C(C)NC(=O)CSc2nccn2-c2ccc(Br)cc2)cccc(Cl)c1Br c1(OC)cc(C(N2CC3CC(CNC(C4CC4CF)=O)C3C2)=O)cc(N)c1OC C(=O)(C1OCCc2ccccc21)N(C(C)CNC(C12CC(C)(C1)OC2(C)C)=O)C c1(CC2CCN2C(C2CCC2)=O)cnc(O)cc1OC.c1(C(C=C)(C)O)cn(C)nn1 N1(C(c2nc(SCCC)sc2)=O)CCC(C2(C)CC2)CC1 c1(SC2(C(C)NC(C(C)OC)=O)CCOCC2)cccc(C(F)(F)F)c1 Cc1c(F)ccc(C(=O)NCC2(CO)CCN(C(=O)CCNC(N)=O)C2)c1N N1(C(C=C(COC)C)=O)CCN(C(c2cc(-c3ccoc3)[nH]n2)=O)C2CCC12 c1(C(=O)NCC(CNC(CN(C(C)C)C)=O)CO)c(Cl)ccc(F)c1N c1(CC)cc(NC2CC(c3ncc[nH]3)C2)nc2ccccc12 N1(C(=O)NCCCl)CC2CCN(Cc3ccc(I)cc3O)CC2C1 CC(C)(CC(F)C(=O)NC1CC2C=CC1C2)NC(=O)CCCN=[N+]=[N-] C1(CNC(C(C(C)C)C#N)=O)COC(C)(C)CN1C(=O)Cc1csc(Cl)c1 C1(Nc2nc(NC(C(CC)(C)OC)C3CC3)nc(C)c2)CCc2cnn(C)c2C1 C1(NC(C#CC2(C)CC2)=O)CCC2(CC1)CCN(C(C1CCS(=O)(=O)CC1)=O)C2 C(=O)(C1CCc2cccc(O)c21)NC1CN(C(C(C)OCCC(C)C)=O)C(C)C1 c1(C(N2CC(C)CC(NC(CN(CC)CC)=O)C2)=O)cc2cccc(F)c2s1 CN1CCCC2(CCN(C(=O)NCC(F)C(C)(C)O)C2)C1=O c1(C(CO)N(C(C(=O)NC2CC(C#C)C2)=O)C)cccc(F)c1 C(=O)(CCCC(C)(F)F)NC1C(N(C)C(c2cc(O)cc(O)n2)=O)CCCC1 N(C(=NCC(F)(F)C1(O)CCOCC1)NCC(C)(C)C)C(C=C)C C1(NC(CSCC#C)=O)(CNC(C2CCCOCC2)=O)CCCCCC1 C1(C(N(OCC)CC)=O)CCC(C)(C)N(C(C2CC23CCCCC3)=O)C1 C1(NC(CCC#CC)=O)C2CC3CN(C(=O)Cc4cc(C)cc(F)c4)C1C3C2 C1(NC(CC2(OC)CCC2)=O)CN(c2ncccc2[N+](=O)[O-])CCC1(F)F CC(C)C(C(=O)N1CC(C)(NC(=O)Cc2cnnn2C)C1)c1cnn(C)c1 C1(CC(=O)NCCn2cc(C(=O)NC(c3nnnn3C)C)nc2)CCOC1(C)C N1(C(C(C)SCC)=O)CCN(C(c2ccc(O)cc2C(F)F)=O)CC1CO n1(CC(=O)NC(c2ccccc2)C2CCC2)cc(Br)cc(Cl)c1=O N1(C(C=Cc2occ(C)n2)=O)CC(C2CN(C(c3ncc4[nH]ncc4n3)=O)C2)C1 c1(C(=O)OC)c(C)sc2cc(C(=O)NC(CO)C(C)NC(=O)CC(C)C)[nH]c12 C(=O)(CCCC1CC1)NCC(C)CN(C)C(C1(F)CC1c1ccccc1)=O C1(C(N2CC=CC(NC(CN(C(COC)=O)C)=O)C2)=O)CCCN(S(N)(=O)=O)C1 C(=O)(CC1COc2cc(O)ccc21)NC1(CNC(C2C(C)C2(F)F)=O)CCC1 c1(C(=O)NCC2CCCCN(c3nnc(COC)s3)C2)ccnc2nccnc12 c1(C(=O)NC2(C)CCC(NC(c3c(C)noc3)=O)CC2)ccc2[nH]nc(O)c2c1 C(=O)(C(COC)CC)NCCN(C(c1c(CC)cc[nH]1)=O)CC1CC1 C1(C(=O)NCC=C2CCN(C(c3ccncc3F)=O)CC2)CCc2cncn2C1 C#Cc1cc(C(N2CC(CNC(=O)CC(F)F)C(O)C2)=O)ccc1Cl c1(C2(C(=O)NCC(CC=C)NC(=O)CC(C)C3CC3)CC2)ccnc(Cl)c1 C1(C(N(C)CC2(NC(=O)C=CSc3ccccc3)CC2)=O)CC2CCC1C2 Cc1cc(C(=O)NCC2(C)CCCN2C(=O)COc2ccc(Cl)cc2)cc(O)n1 C1(NC(C2C(C)=CCS2)=O)CCN(CCNC(=O)Cc2nc[nH]n2)CC1 C(C(=O)NC1(c2cccnc2)CC1)(C(C)(C)O)NC(CC1(SC)CC1)=O N1(C(c2cc(C)sc2)=O)CCC2(CCC2)C(CNC(c2cc(F)cc(F)c2)=O)C1 c1(C(=O)NCCC2CCN(C(C3C(C)C3C)=O)CC2)cc2cccnc2[nH]1 c1(OC(CC)C)ccc(COC(=O)NCC(C)(C)CC2CCCCC2)cc1 C1(C#N)(CNC(CC2C(C(=O)NC3(CC#C)CCOC3)CCC2)=O)CCOCC1 C(C(CC(C)C)C(=O)NCCCCNC(C1(C(C)(C)C)CCCCC1)=O)OC c1(C(=O)NC2(CO)CCN(C(C(C)C3CCC3)=O)C2)cccn(C2CC2)c1=O C=CCC(CC)C(=O)N(CC(C)CNC(=O)CSc1ccccc1C)C N1(C(c2ccn(C)n2)=O)CCC2(CCCN2C(c2csc(=NC3CC3)[nH]2)=O)CC1 N1(C(C2CC(OC)C2)=O)CCN(C(C2CCC(=O)NC2)=O)CC1c1nccn1C N1(C(C2CNC(=O)N2)=O)CCC(CO)(NC(=O)CCC2NC(=O)NC2=O)CC1 CCCC(CCC)C(=O)NC1CCCC12CN(C(=O)C(CC)c1ccccc1)C2 N1(C(C=COCC)=O)CCCCC1C(C)NC(c1cccc(C)c1)=O CCC(CN(C)C)CC(=O)N1CC(CO)(NC(c2cccc(CO)c2C)=O)C1 c1(NC(C(Cn2ccc(C)c2)N(C)C)=O)ccc(OC)c(O)c1.c1(CO)ccccc1 CS(=O)(=O)c1ccc(CNC(=O)NCC(c2ccccc2)CO)cc1Cl N1(C(CCC(=O)NC)=O)CCCCCC1C(=O)NC1CCC2CCC12 CCC(CCC(=O)N(C1CC2CCC1O2)C)NC(=O)C=Cc1nccs1 C1(C(=O)NC2(c3ccc(F)cc3)CCN(C(=O)CO)CC2)Cc2cccnc2C1 N1(C(N(C)Cc2c(OC)cccc2)=O)CCN(c2ccc(F)cn2)CC1C c1(C(=O)NC2C=CC(CNC(c3cscc3Br)=O)C2)cc2n(n1)CCCC2 C(=O)(C(C)CCCC(C)=O)N1C(C#C)CN(C(=O)C(C)n2ccnn2)CC1 C#CCC(C)(C)C(=O)NCC1(CNC(c2c[nH]nc2CC)=O)CC12CCC2 c1(C(N2CCC(NC(CC(C(C)C)O)=O)C2)=O)cnc2[nH]nc(O)c2c1 C1(NC(C(C)N(C(C2C3CCC(C3)C2C)=O)CC)=O)CN(C)C(=O)C12CC2 C(=O)(C(F)CC(C)(C)NC(=O)C#CC1CCOC1)NCC1CC(C(=O)OC)C1 C1(NC(C2CN(CC)C(=O)C2)=O)CCN(Cc2cncs2)CC1O C1(C)(C(=O)NC2CC(C)(NC(C(C)N(C(C)=O)C)=O)C2)CCOC(C)C1 c1(CCCSCC)cn(C2CCN(C(=O)C(C)(C)C)C2)nn1 C1(C(=O)NCC(N(C(=O)CC2(C#N)CC2)C)C2CC2)CC(F)(F)CS1 C(C(CC(C)C)C(=O)N1CCCCC1CN(C(=O)CC1CN(C(C)=O)C1)C)OC Cc1cccc(F)c1C(=O)NCC1CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)CCO1 C1(CC(C)C)(C(=O)N(C)CCN(C)C(C2CCCN2C(C)C)=O)CCNC1=O Cc1nc(O)ccc1C(=O)NCC(CC1CC1)C(=O)N(C(C)C(=O)N(C)C)C N1(C(CC(c2ccc(Cl)cc2)C)=O)CCOC2CNCCC12 Cc1cnc(C(C)NC(c2cc(C3CC3)ns2)c2nnnn2CC2CC2)s1 c1(CC(N2CCC(O)(CNC(C3(CC)CC3)=O)C2)=O)cc(F)c(C)cc1F CCCCC(C)CCC(=O)NC1C2CC(NC(c3csc(C4CC4)n3)=O)CC12 c1(C(N2CCC(NC(c3occ4c3CCC4)=O)C2)=O)ccc(Cl)c2cccnc12 c1(C(=O)NCCC(C)N(C(=O)CC2CC2)C)nccc2c1[nH]c1ccccc21 C1(NC(c2c(CN(C)C)cccc2)=O)CN(C(C2(C)CCCS2)=O)CC(F)(F)C1 C1(C(=O)NC(C(=O)OCCC)C)CN(C(C2(F)CCC2)=O)CCO1 c1(OCC)cnc(C(=O)NCCN(C(c2sc(OC)nc2Cl)=O)CC2CC2)c(Cl)c1 n1(CC)nc(C(N2CCCCC2CNC(=O)C(F)(F)CC2CC2)=O)cc1C C=C1CC2CCCC(C1)N2C(=O)CC(C1CC1)NC(c1ccnn1C1CC1)=O N1(CC2CCC(C)(C)C2)C(=O)CN(CCP(C)(C)=O)C1=O C(=O)(C1CCCc2sc(=N)[nH]c21)NCCNC(C1(C)CC1(F)F)=O CC1CCN(C(=O)Cc2cncnc2)C1CNC(c1ccc(C2CC2)s1)=O N1(C(c2cccc(OCC)c2)=O)CCC(NC(=O)C2=CCCS2)C12CCC2 c1(OCC=C)cccnc1C(N1CCCC1CNC(=O)CCNS(C)(=O)=O)=O C1(CCOC)CN(C(c2nnc(Cl)cc2N)=O)CCN1C(C1CN(C)CCO1)=O CC(C)(C)C(CNC(=O)Cc1ccon1)NC(c1ccn(C2CCCCC2)n1)=O Cc1nc2cc(C(=O)NCC3(C)CC(NC(C4CC=CCC4)=O)C3)cnc2s1 C1(CNC(CN(C(C(C)C)=O)C)=O)CCCCN(C(C23CSCC2C3)=O)C1 c1(C(C(N2CCC(N(C(=O)Cc3cscn3)CC)C2)=O)(F)F)ccc(C)cc1 C1(C(C(=O)NCC(CC)CO)(C)C)CCCN(C(=O)C(O)CCSC)C1 CCCCCCCC(F)C(=O)NC(C)(CNC(c1conc1C)=O)CO N1(C(C(C)NC(=O)CCNC(=O)CO)=O)CCC2(CCSC2)C1 N1(C(CN(c2ccccc2)C)=O)CCCCC(N=c2[nH]c(Cl)nc3c2CCC3)C1 N1(C(c2n[nH]c(C)c2F)=O)CCC2(CCCN(C(=O)CN3CCN(C)CC3)C2)C1 N1(C(CN(C)S(N)(=O)=O)=O)CCC(CCNC(=O)C2=CCCCO2)C(F)(F)C1 N1(C(c2c(C)nc(O)cc2)=O)CCCC(C)(C)C1CNC(C1(C(N)=O)CCC1)=O c1(OCC)cccc(C(=O)NCC(C)(C)NC(C2CC2COC)=O)c1 c1(NC(CN2C3CC(C(=O)NCC)C2CC3)=O)nc2ccc(OC(C)C)nc2s1 c1(C(=O)NC(CN(C(CC2N(CC)CCC2)=O)C)C)ccc(F)cc1C1CC1 C1(CNC(C2CC2F)=O)CCCC12CCN(C(=O)CC1CSCCS1)CC2 Cc1ccc2c(c1)SC(C(=O)NC1CC(NC(c3coc(O)n3)=O)CC1O)C2 C(=O)(CC(C)CC(C)C)NC1CC(N(C(c2c(OC)c(C(F)F)ccc2)=O)C)C1 N1(C(C(C)SCC)=O)CC(C(=O)NC2(CC(=O)NC3CC3)CC2)(SC)C1 N1(C(C(CC)(C)CNC(=O)C(F)F)=O)CCC2CC1C(=O)O2 N1(C(C2CCC(CC)O2)=O)CCCC12CCN(C(=O)CCC(=O)OC)C2 c1(CC(N2CC(Cn3cc(CCO)nn3)C2)=O)cccc(Br)c1 S(=O)(=O)(c1ccc(NCC(F)C2CCC2)c(C#N)c1)NCc1c(CC)nn(C)c1 c1(CC(=O)NCCC2(OC)CN(C(c3sc(CO)nc3C)=O)C2)ccc(C)cc1 N1(C(c2n(C)c(S)nc2)=O)CCC(C2(NC(=O)CC3CC=CCC3)CC2)CC1 Cc1ncn(C)c1C(=O)NC(C)C(C(C)C)NC(c1cnn(C2CC2)c1C)=O N1(C(c2cc(C)ns2)=O)CC(CNC(=O)CSCc2csc(=N)[nH]2)CCC1C N1(C(Cc2c(C)n[nH]c2C)=O)CCC2(CC2NC(C2CC2F)=O)C1 C1(CNC(C(c2cccc(Cl)c2)C)=O)CN(C(c2coc(C(N)=O)c2)=O)CC1O C1(NC(c2ccn(CCNC(C(CC=C)C)=O)c2)=O)CCc2nncn2C1 C(=O)(C(C)CC(C)C(C)=O)NC1C(CC)N(C(c2cn(C)nc2OC)=O)CCC1 c1(C(N(CCN(C)C(C2CSCCS2)=O)C)=O)cnc(N(C)C)s1 N1(C(C2(C)ON=C(C)C2)=O)CC2(CC(C(=O)NC3(C)CC3)CO2)C1 C1(NC(C2(C)ON=C(C)C2)=O)CC(C(=O)N(C(CO)C(C)C)C)=CC1O C1(NC(CSC)=O)CC=CCC1C(=O)NCCn1cnc(CO)c1 C(=O)(C(CC)N(C(=O)Cn1cc(COC)cn1)C)NCC(=O)N(C)CC c1(-c2cc(F)c(NC(C)=O)c(F)c2)cc2c(s1)CCN(Cc1cccc(C)n1)C2 c1(SC)cccnc1Cn1ccnc1Cc1ccccc1 N1(CCC)CCN(C(C2CCC(c3cccc(Cl)c3)C2)=O)CC1 C(=O)(CC(O)CNC(=O)CC1CC(C)=NO1)NC(C(=O)NCC)C C1(CNC(c2cn(CC)nc2)=O)CCC(C(N2CCC2C(C)C)=O)CC1 c1(C(=O)NCCCNC(c2c(N)ccc(C(C)=O)c2)=O)cc(S(N)(=O)=O)sc1C c1(OC)cc(OC)c(NC(C2CN(C(=O)CCc3ccc(C)s3)CCN2)=O)cn1 C(C(C)(C)C(C)(C)C)ONC(C(COC)C(=O)OC(=O)CC(C)(C)C1CC1)=O.OC c1(C(=O)NCCC(C)NC(c2c(COC)cccn2)=O)oc2ccccc2c1C Cn1nnnc1SCC(=O)NC1(CCNC(C2CC2C(F)F)=O)CC1 c1(C(N(CCN(C(C(CC=C)NC(C)=O)=O)C)C(C)C)=O)ccc(OC)nc1C CCCCC(CC)C(=O)NCCCOCCN(C)C(C1CSCCS1)=O C(CS(=O)(=O)CC(=O)N1CCN(C(c2cnn(C)c(=O)c2)=O)CC1C(C)C)OC c1(C(=O)NC2CC(N(C)C(c3ccnn3C)=O)C2)cc(Cl)cc(F)c1N c1(C(=O)NC2CC(C)N(C(c3cncn3C)=O)C2)cc2c(Cl)cccc2s1 N1(C(C2CCCC(=O)O2)=O)CCC2(CCC2)C(CNC(c2sccc2Cl)=O)C1 C#Cc1ccc(Cl)c(C(=O)NC(C)C(C)NC(c2cc(C(C)(C)C)nn2C)=O)c1 Cc1cc(F)ncc1C(=O)NC(C1CCN(C(=O)CCc2cccs2)C1)C c1(C(C)C)sc(Cl)nc1C(N1CCN(C2CN(C(=O)C(C)(C)OC(C)C)C2)CC1)=O C(C(F)(F)C(F)(F)F)OCCC(=O)NCC1(C(C)NC(C(CC)SC)=O)CC1 Cc1cc(Cl)cc(N)c1C(=O)NC1CN(C(=O)CN2CCC2C)C(C)(C)C1 C1(NC(=O)CC(O)C2CCCC2)CC2CN(C(=O)CCCCc3cnn[nH]3)CC12 Cc1ccc(C(F)(F)C(=O)NC2CCC2NC(c2cc(C)ncn2)=O)nc1 c1(C(N2CCC(C)C(NC(C3(F)CCCC3)=O)C2)=O)cc2ccccc2o1 C(CNC(c1c[nH]c(C(N)=O)c1)=O)(CO)(CO)N(C(=O)Cc1cn(CC)nn1)C C1(NC(=O)NC(C(F)(F)CO)C2CC2)CCn2nncc2C1 C1(NC(C(C)CC(F)(F)F)=O)CCCCC12CCN(C(C1CC3CCC1O3)=O)C2 C1(CN(C(C=CC)=O)C)CN(C(c2cccc(C3CC3)c2)=O)CCO1 Cc1cccc(Br)c1C(N1CCC(=CCNC(c2cccnc2Cl)=O)CC1)=O C1(CNC(c2ccc(F)s2)=O)CC2(CCN(C(c3cc[nH]c3C3CC3)=O)C2)CO1 N1(C(c2ccc(F)c(CO)c2)=O)CC2CCCN(C(C3C4CCC3CC4)=O)C2C1 C(=O)(C1CCCn2nccc21)N1CCCCC(N(C(=O)C2=C(Cl)CC2)C)C1 c1(C(=O)NCC2C3CN(C(c4ccccc4O)=O)CC32)c(O)ncc2c1CCC2 C1(NC(c2ccc(C)cc2Cl)=O)CN(C(=O)CC2CCOCC2)CCC1(C)C c1(C(=O)NC(CC)CNC(c2cncc(F)c2Cl)=O)ccn(C)c(=O)c1O Cc1ccnnc1C(=O)N(C1CCN(C(=O)Cc2ccccc2F)C1)C N1(CC(=O)OCCCF)CCCC(CC(F)F)C1 c1(C(N2CCN(C3CCN(C(=O)COC4CCC4)C3)CC2)=O)cc([N+](=O)[O-])c[nH]1 c1(N(C)C)ccc2cc(C(N3CCN(Cc4cncs4)CC3)=O)ccc2c1 CCCCC(O)C(=O)NCC(O)CN(C(=O)C(C)(C)COCC(F)F)C C1(NC(=O)CCC2CCC2)CC2CCC1CC2NC(C1CC2CCCCC2O1)=O c1(NC(C)=O)ccc(Cl)c(CC(=O)NC2CCN(C(=O)C(C)C(F)F)C(C)C2)c1 c1(CC(=O)NCC(CNC(CCCOC)=O)F)c[nH]c2cccnc12 c1(C(=O)NCC2CCC(C(=O)NCc3cc(CC)no3)C2)cc(C)n(C)c1 c1(NCc2ccc(C)cc2Br)ccc(S(=O)(=O)NCc2ccn(C)n2)cc1Cl Cc1cc(NC(=O)C(=O)NC2CC(CNC3CC4(CC4)CO3)CO2)ccc1N n1(CC(=O)OC)cnc(C)c1C(=O)NC1C=CC(CNC(c2oc(C)nc2C)=O)C1 CCCC(C(O)C(=O)NCc1cncc(F)c1)NC(=O)C(C)CCOC C(=O)(C(O)C(C)C)NCCOCCNC(c1n(CCC)ccc1)=O N1(C(CCNC(C)=O)=O)CCC(C(N2CCN(CCCO)CC2)=O)C(O)C1 CC(CO)(CO)C(=O)NC1CCC(C(=O)Nc2cc(F)cnc2Cl)C1 O=C1OCc2c(C(=O)NCCC(=O)NC3CCCCC3)cccc21 N1(CC(=O)N(C2COC(C)(C)OC2)C(C)C)CCCC(C)C1C(=O)OC CN1CCOCC1C(=O)NC1CCC(C(=O)NOCC2(F)CCC2)C1 Cc1nc(C)c(C(=O)N(CCCCCNC(=O)CC2(C(F)(F)F)CCC2)C)[nH]1 c1(C(N2CCC(NC(CC3ON=C(C)C3)=O)(CF)C2)=O)ccc(Cl)c(C)c1N CCC(O)C(F)(F)C(=O)NC1CCN(C(=O)C=Cc2ccccc2)C(C)C1 c1(OC)ccncc1CNC(=O)C(Cc1ccoc1)NC(=O)CN1CC(C)(C)C1 C1(F)(CNC(C2C=CCC2)=O)COCCN(C(=O)CC2CCCCC2)C1 c1(C(N(CCN(C)C(c2cc(Cl)n(C)n2)=O)C)=O)cc(O)nc2ccc(Cl)cc12 C(=O)(C(CC#CC)NC(c1ccc(C)cc1O)=O)NC(CCC=C)(C)C C1(C(=O)NCC(C)O)COCCN(CC(O)CN2CCOCC2)C1 CC1(C)OC(=O)CC1C(N1CCOCCC1C(=O)NC1CCS(=O)CC1)=O c1(C(N2CC(OCCNC(C(C(C)C)C)=O)C2)=O)cc2cccnn2n1 C1(NC(C2(SCC)CC2)=O)COC2(CCN(C(=O)CCC3CCC3)C2)C1 c1(C(=O)NC2C(CNC(c3ccc(CCC)cc3)=O)C2)cccc2c(C)[nH]nc12 N1(C(C2(NC(C3C(C)(C)C3(C)C)=O)CC(F)(F)C2)=O)CCOCC(CO)C1 Cc1cnc2c(C(=O)NCC3CCN(C(C4Cc5nccn5C4)=O)C3)cnn2c1 C=CCC(CC)C(=O)NC(c1cccnc1)C(=O)Nc1cnccc1OC c1(C(=O)NC(CCCNC(C2CC(O)(CC#C)C2)=O)(C)C)cc(C#N)[nH]c1C Cc1c(C(=O)N(CC(C)O)CCNC(c2coc(Cl)n2)=O)oc2ccc(Cl)cc12 c1(C(=O)NCC(CNC(CCCCOC)=O)O)ccc(=O)n(C(C)C)c1 C1(C(=O)NC(CN(C(c2c(C(C)C)[nH]cc2)=O)C)C)CC2(C1)CC1(CC1)C2 C(=O)(C1=NOC(C)C1)NC(C(=O)NCC1ON=C(CC)C1)Cc1ccoc1 N1(CC(c2n(C(COC)C)nc(-c3ccccn3)n2)C)CCc2ccccc21 S(=O)(=O)(c1[nH]c(=NCC2CCCNC2=O)ccc1Br)OC.C12CC3(C1)CC3N2 C(=O)(C1CCc2ccc(Cl)nc21)NC1C(CNC(C2=C(C)OCC2)=O)COC1 Cc1sc(O)nc1C(=O)NC1CC=CCC1C(=O)NCC(=O)NC1CCCCC1 Cn1cc2c(C(=O)NCC3C4CN(C(c5ns[nH]c5=O)=O)CC34)cccc2n1 c1(C(=O)NC2CN(Cc3cc(OC)cc(O)c3)CC2(F)F)cc(Cl)cc(Cl)c1O C1(C(=O)NC(CC#C)CO)CC(C)CN1C(=O)COC1CCOCC1 C(CCC)(C(=O)NC1(CCC(=O)NCCCc2ccncc2)CCC1)=CCC c1(C(=O)NC(CN(C(=O)CCC2C(=O)NN=C2C)CC)C)ccc2c(n1)CCC2 C1(C(=O)NCCCNC(N)=O)CC2C=CC1N(C(c1cc(F)ccc1O)=O)C2 c1(NC(Cn2c(-c3ccccc3)cc(=N)[nH]2)=O)c(F)ccc([N+](=O)[O-])c1F C1(CC(N2CCC(C(C(=O)N(C)CCn3cncn3)(C)C)C2)=O)CCCNC1=O CC1(C(N2CCC2)=O)CCCN(C(=O)CCCC2CCC(C(=O)O)O2)C1 C#Cc1cc(C(=O)NCC(CO)NC(c2ccc(O)nc2)=O)cc(F)c1 N1(C(c2nc(CC)oc2)=O)CCC(NC(c2cc(CC)cnc2OC)=O)C(F)C1 CC(C)CCC(O)C(=O)NCC12CCC(NC(C3SCCCS3)=O)(CO1)C2 N1(C(C(CC=C)(C)N(C)C)=O)CC2CCC1CN2C(=O)C(CC)OC N1(S(=O)(=O)C2CC3CC2C3)CC(O)CC2CCCCC12 C1(C(=O)NC(C(=O)NC2CCC(C)(C)C2)(C)C)CCOCC1(C)C O=C(N1CCC(O)CO1)C1CC2CC(O)C(C1)C2 c1(C(=O)NCCC2OCCCN(C(CC(C)C)=O)C2)cnc2cnccc2c1 C1(NC(c2cccc(C(C)C)c2)=O)CCN(C(=O)C(F)CC2CCC2)C1(C)C Cc1cc2ccc(CNC(=O)NC3CC(c4ccc(F)cc4)C3)cc2[nH]1 c1(N(CC(C)CNC(c2ccsc2)=O)C)cc(-c2ccccc2)ncn1 c1(C(=O)NCC(C2(O)CCN(C(CCC)=O)C2)C)cc2c(s1)CCC2 c1(OC)ccc(Cl)c(C(=O)NCCCCCCN(C)C(c2ccns2)=O)n1 CCC(CC(C)C)C(=O)N1CCC(CN(c2nccc(C#N)n2)C)C1 c1(C(=O)NC2CCCC(C(=O)NC3(C)C(C)(C)C3)C2)cnc2cccnn12 n1(CC(=O)NCC2CN(C(C3C4COCC34)=O)CCO2)cnc2sccc2c1=O C1(NC(=O)CCC)CC(C(=O)OCC)CCN1C(=O)CC1CCC(C)(C)C1 C1(CNC(CC)=O)CCCN(C(c2cccc(-c3ccccc3Br)c2)=O)C1 CC1CN(C(=O)CC(=O)NC2CC2)CCN1C(=O)Cc1cn(C)nc1Cl c1(OC)cc(C)sc1C(=O)NCC1CC(NC(=O)COC2CCOC2)CCO1 N1(C(CCNC(N)=O)=O)CCN(C(=O)CC(F)(F)Cl)CC1CC(F)(F)F C#Cc1cc(NC(=O)CN2CCN(C(c3ccco3)=O)CC2)ccc1C C1(C2CCN(C(c3nc(C(C)(F)F)cs3)=O)C2)(NC(c2ccc(C)nc2)=O)CC1 c1(N2CC(C)=C(C)C2)nc(N2CCCC(C(N)=O)C2)nc2cccnc12 CC1CCC(C(=O)NCC=CCl)CN1C(=O)Cc1cccnc1O C1(NC(C2CSCCS2)=O)CN(C(c2ncncc2Cl)=O)CCC1CO C(=O)(C(CC(C)C)OC)N1CC(CCC=C)(C(=O)NCCC=CC=C)C1 N1(C(c2cc(OCC)n[nH]2)=O)CC2CC1CCN2C(=O)CC1=CCCCC1 C1(C)(CC)C=C(C(=O)N(CCNC(c2ccc[n+]([O-])c2)=O)C2CC2)C1 C1(C(N2CCN(C(CC=C)=O)C(CS(C)(=O)=O)C2)=O)CC2(C1)NC(=O)NC2=O Cc1cc(NC(=O)CCC2CCCN2C(=O)C(C)S(N)(=O)=O)cc(C)c1F C1(N(C(C2N(C(C)=O)CCC2)=O)C)CCCC(NC(=O)CNC=O)C1 N1(C(CN(C(C)=O)C)=O)CCCCC(N(C(=O)C=C(C2CC2)C2CC2)C)C1 C(C(CNC1(c2ccsc2)CC1)CC1CCCC1)NC(=O)OC(C)(C)C C1(NC(C2(CCC)CC2)=O)CCCC(NC(c2ccccc2SCCO)=O)C1 C(=O)(CC(F)(F)C(F)F)N1CC(C(=O)NCc2sccc2-n2ccnn2)C(F)C1 C1(NC(C2(CC)CC2)=O)CCCCCN(C(c2cc(F)c(Br)cc2N)=O)C1 c1(OC)cc(F)cc2[nH]c(C(N3CC(O)CC3C3CCCOC3)=O)cc12 n1(C(C)C)ncc(C(=O)NC2CCCC(CNC(=O)CCC(=O)N(C)C)C2)c1F c1(C(N2CC(NC(CC3(C)CCC3)=O)C2)=O)cccn2nncc12 S(=O)(=O)(c1cncc(Cl)c1)Nc1c(C#N)nc(Cl)cc1 c1(CC(=O)OC)cnc2ccc(CN3CCCC(C)(OC(C)(C)C)C3)cn12 S(=O)(=O)(c1cc(Cl)c(F)cc1F)N1CC(C)OC(C(F)(F)F)C1(C)C N1(C(c2c(C)oc(CO)c2)=O)CC2CCCC2(CNC(=O)CCC=CC(C)C)C1 CCCC(O)C(=O)N1CC(C(=O)NCC#CC2CC2)(COC)C1 c1(C(N2C(CCCNC(c3c(C)cn(C)n3)=O)CCC2)=O)cc(O)ccc1N c1(-c2c(C(=O)NC(C)CF)n[nH]c2)ccc2c(c1)OCC(=O)N2 c1(CC)cc(C(=O)NCCC2CN(C(C3CC34CCOC4)=O)C2)nn1C C(=O)(N=c1ccn(C(C)(C)C)[nH]1)C1(C(C)NC(c2[nH]nnc2C(F)F)=O)CC1 CN(C)S(C)(=O)=NC(=O)CN1CCCC(c2nccs2)C1 N1(C(C(C)SCC)=O)CCN(C)C(CNC(=O)C=Cc2cc(OC)ns2)C1 C(N=c1[nH]cnc(C)c1OC)C1C(NC(c2ccc(OCC)cc2)=O)CCC1 C(CC(O)CC(=O)NC12CC1CN(C(c1oc(C(F)F)cc1C)=O)C2)SC c1(C(N(CCC(F)(F)F)C)=O)ncn2c1CCC2 N1(C(c2cnn(C)n2)=O)CC(C)(C)OCC1CNC(c1ccc(F)c(F)c1F)=O N1(C(CCNC(C)C)=O)CCN2CCN(C(C3CN(S(C)(=O)=O)C3)=O)CC2C1 N1(C(c2c(CNC(C(CCC)OC)=O)noc2)=O)CCOC(C)C1CO c1(CC(=O)NC2CN(C(CCOCC)=O)C2)ccc(F)cc1F n1(CC)ncc(C(=O)Nc2cccc(NC(=O)C(C)(C3CC3)OC)c2)c1C1CC1 c1cc(-n2cc(C3CNCCOC3)nn2)c2c(c1)CCOC2 c1(NC(N(CCS(C)(=O)=O)CC)=O)ccc(OC(=O)COC(C)(C)C)cc1 N1(C(C(CCC)C)=O)CCN(C(=O)COc2c(C)cccc2Cl)C(CCO)C1 C(=O)(C1=CC2CCC(C1)C2)N1CC(C)CC(C(=O)NCc2c(C)non2)C1 N1(CCC)CC2CC(NC(=O)C(C)OCc3ncccn3)CC1C2 c1(C(=O)NCCN(C(C2CCN(C3CCCCC3)C2)=O)C2CC2)ccc[n+]([O-])c1 CC(CC(=O)NC1CCCC1NC(=O)CCCc1ccc(O)c(F)c1)C(F)(F)F C1(C(=O)NCC2C(NC(C)=O)CCC2)COCCN1Cc1ccccc1 C#CCCCCCNC(=O)CC1(C)CCN(C(=O)C(C)(C)N(C)C)C1 C12(C(N(C(C)C(=O)NCCCP(C)(C)=O)CCC)=O)CCC(C1)C2(C)C C1(C(N2CCC(C(=O)NCC(C(=O)NC)C)C2)=O)COCC(C)O1 Cc1cccc(C(N2CCCC2CC2CCCCN2C(=O)ON(C)C)=O)c1 N1(C(c2c(OC)csc2)=O)CCN(C(c2cc(CO)n(C)n2)=O)C(C(C)C)C1 c1(CNC(C(C)N(C(C2CC23CCOCC3)=O)C2CC2)=O)cccc(F)c1O C(=O)(C1=CC2CC=CCC12)N1CCN(C2CCN(C(CC(=O)OC)=O)CC2)CC1 C#Cc1ccc(F)cc1C(=O)NCC1CN(C(C2(SC)CCC2)=O)CCCO1 C(=O)(CCC(F)(F)C(F)F)NC(c1ccc(C)cc1)CNC(=O)Cn1cncn1 C(=O)(CCC(=O)N(C)CC1(O)CCN(C(=O)CCN2CCCC2=O)C1)NC C1(C(=O)NCC2OCCN(C(c3cccc(SC)n3)=O)C2)CCCCNC1=O N1(C(COCC)=O)C2CCC1C(C)C(NC(=O)CC1CCCC(OC)C1)C2 C1(C(N2C(c3ncc(C)s3)CCCC2)=O)CC(O)C(N=[N+]=[N-])C1 N1(C(c2cc(CSC)c(C)o2)=O)CCC12CN(C(c1cc(Cl)c(C)cn1)=O)C2 C1(CC#C)(CNC(=O)CN(C(=O)C(F)CCC)C)CCCCO1 Cc1cc(Cl)ncc1CC(=O)N(C1CCN(C(C2CSCC(=O)N2)=O)C1)C C(=O)(C(C)C(C)(C)C)NCc1occ(C(=O)NC2C(C)COCC2)c1 c1(C(N(CCN(CC#CC)CCCO)C(=O)OC(C)(C)C)=O)ccccc1C c1(CNC(C2CC(O)(CNC(C(C)=C3CCC3)=O)C2)=O)cc(C)cc(F)c1 N1(C(=O)NC(C)CCc2ccc(Br)cc2)CCSCC1(C)C c1(OC)c(C(N2CC(CNC(=O)C(C)(C)CO)C(C)C2)=O)oc2ccccc12 N1(C(C(C(C)OC)NC(=O)CC2CCCN2C)=O)CCN(C)CC(O)C1 C1(CC(=O)N(C2CCN(C(C3(C)CC3(F)F)=O)CC2)CC#C)CCOCC1(C)C c1(CNC(N(C(C)CN(C)C)CCOC)=O)ncnn1-c1ccccc1 N1(C(c2c(CC)ccs2)=O)CCC(C)(CCNC(=O)CC(C)C2CCCC2)CC1 C1(O)(CC)CCN(C(=O)CCCC(C)NC(c2cnc(O)o2)=O)CC1 C(=O)(C(F)(F)C(O)C1CC1)N(C1CC(NC(c2ncn(CC)c2)=O)C1)C C1(C(=O)NC(CCCCC)C2CC2)N(C(C23CCCC2C3(F)F)=O)CCC1(C)C CCCCC(CC(=O)N1CCCC1CC1CC1)NC(C1CN2CCC1C2)=O c1(NCC(C)CN(C(=O)C=CCN2CCCC2)C)snc(Cl)c1C#N CC(C(C)(C)C)=CC(=O)NCC(O)CN(C)C(c1cc(C2CC2)sn1)=O C(CC)(C(=O)NCCCCc1cnc[nH]1)N(C(C(C)NC(CC)=O)=O)C c1(CC(=O)NC(CC)(CNC(=O)Cn2cc(Cl)cn2)CC)cc(F)ccc1O CCC(O)C(F)(F)C(=O)N1CC=C(C(=O)NCc2ccc(CO)cc2)CC1 c1(C(N2CC=CC(NC(c3cc(C)c(C)nn3)=O)C2)=O)cc2ccc(F)cc2s1 C1(C(=O)NCC2C(NC(c3cn(C(C)(C)C)nn3)=O)CCC2)CC2(C1)CC2(F)F C1(CNC(C(C=C)(F)F)=O)CC2CCCC2N1C(=O)Cc1cncnc1 C1(NC(c2nc(C)c(C)s2)=O)CC(C(=O)NCC2CCOC2(C)C)C12CCC2 N1(C(C2(C#C)CCC2)=O)CCN(C(c2[nH]ccc2CC)=O)C(CO)C1 CC#CCC(C(=O)N(C1CCOC(C)C1)C)NC(C1CNC(=O)C1)=O c1(C(N(C2CCC(NC(c3cnn[nH]3)=O)C2)C)=O)noc2ccc(Cl)cc12 C1(C(=O)NC(C2CN(C(=O)C(c3ccc(F)cc3)(C)F)C2)C)CCc2nn[nH]c2C1 C1(C(CC)CC)CN(c2cc(N(C)Cc3cccnn3)ncn2)CCO1 n1(C(C)NC(=O)C(Cn2cncn2)NC(=O)OC(C)(C)C)cnc2ccsc2c1=O c1(CC)[nH]c(=N)sc1C(N1CCC(N(C)C(c2c[nH]nc2C)=O)C1)=O c1(CNC(CN(CC#C)C(c2cnsc2C)=O)=O)cn(C)nn1 C1(C(N2C(CCNC(CC)=O)CCC2)=O)CCN(C(C2(C)CC2(F)F)=O)CC1 C1(NC(C(C)SC(C)C)=O)C2CCCN(C(c3ccns3)=O)C2C1(C)C C(=O)(C(CCC(N)=O)n1cc(-c2cscn2)nn1)NC(c1ncc[nH]1)CC C(C(C)(O)C(=O)NCCC1CCCN(C(C2CNC(=O)N2C)=O)C1)OC c1(NC(C2C(O)CCN(Cc3c(C)c(Br)cnc3)C2)=O)cc(C#N)ccc1F c1(C(=O)NC2C(NC(C=CC(CC)C)=O)C2)cccc(OCc2cscn2)c1 N1(C(CNC(=O)NC)=O)CCC(N(C)C(c2ccnc(OC)n2)=O)C(C)C1 N1(C(C2CC(C)C2)=O)CCN(C(=O)C=Cc2ccsc2)C(c2ncc[nH]2)C1 C(CC(C(N)=O)NC(c1coc(C(C)NC(=O)CC2CN(C(C)=O)C2)n1)=O)OC N1(C(C2CC3CC2C3)=O)CCCC(C2CCN(c3ncc4ncnc-4[nH]3)C2)C1 C12(NC(c3c(CC)scc3)=O)CCCCC1CN(C(=O)C(C)(Cl)Cl)C2 n1(CC)nnc2c1C(C(=O)Nc1ncccn1)CN(C(C1(C)CC1)=O)C2 C(CC(O)C(=O)NCC(C1CC1)NC(=O)CCN1CCC(N(C)C)CC1)N(C)C CC(C)CN(Cc1ccccc1F)N(C)Cc1ccc(CO)c(F)c1 C1(CC)CN(C(c2cnco2)=O)CCN1C(=O)C(COC(C)C)NC(C)=O CCCC(CC)C(=O)NCc1ccc(C(=O)NC2(C)CC(F)C2)nc1 N1(C(C(CC(=O)OCC)C)=O)CCC2(CCC(NC(=O)CN(C)C(C)C)C2)CC1 Cc1cn2ccnc(C(N3CC(NC(=O)C(F)CC4CCCC4)C(F)C3)=O)c2n1 C1(C)(C(=O)NC2CC(CNC(C(CCC)N(C)C)=O)C2)COC(C)(C)OC1 c1(C(N2CCCC(O)(CCNC(CCC#C)=O)C2)=O)cccc2sccc12 N1(C(CCCC#N)=O)C2CCC1CN(C(=O)CC13CC(c4ccccc4)(C1)C3)C2 N(C1CCC(=O)c2ccccc21)C(=O)C1=NOC2COCC12 Cc1nc(C(=O)NCCOCCCN(C)C(C2CC(C)(O)C2)=O)c(C)n1C1CC1 C1(C(=O)NCCC(CC)CO)CC2CC1CC2NC(c1cccc(Cl)c1)=O Cc1cc(CC(=O)NCC(C2CCC2)NC(=O)C(C)OCC(C)C)ccc1F C#Cc1ccc(C(=O)NC2C3CN(C(=O)C(c4ccc(F)cc4)CC)CC23)nc1 c1(CC)cnccc1C#N.C12(C(=O)NCCCC3CCCC3O)CCCN1C2=O c1(C(=O)NC(C2CCCC2)CNC(C(C2CCC2)OCC)=O)cscc1C(N)=O C1(C(=O)NC(C(N2CC(CC)(OC)C2)=O)COC)COCC1(C)C N1(C(c2nc(NC(C)=O)sc2)=O)CCC(NC(=O)C(C)CCO)C(CO)CC1 N1(C(C(CCSC)O)=O)CC(=O)N2CCOCC2(CNC(C2CCCN2C)=O)C1 C(C#CCN=c1nc2c(ncn2C)c(NCCC(C)O)[nH]1)OC N1(C(C(F)OC)=O)CC(NC(c2ccccc2O)=O)C(C(F)F)C1 C(C)(C)(CCCC(=O)NCCC(C)SC)NC(C1CCC(OC)CC1)=O c1(C(N2CC(NC(C(C)(O)C3CCOCC3)=O)C2)=O)ccccc1F C1(N(C(CCCc2ccc(C)s2)=O)C)CCCN(C(c2c[nH]cc2C(C)C)=O)C1 C1(C(=O)OC)CCC(NC(=O)C(C)(C2CCC2)NC(c2csc(O)n2)=O)C1 c1(CCC(=O)NCCC(OC)OC)ccccc1[N+](=O)[O-] c1(-n2cc(CCNC(COc3ccc(OCC)cc3)=O)nn2)cc(C)ccc1C C1(C(=O)NCCC(C)NC(c2ccc(C(F)(F)F)o2)=O)(CO)CCCO1 C1(CC)CN(C(=O)CC2(OC)CN(C(=O)C(C)n3cccc3)C2)CCO1 N1(C(C2(c3cccc(Cl)c3)CC2)=O)CC2CC2(CNC(=O)Cc2cnsc2)C1 CC1(C)CC(CNC(c2cccnc2-n2cncn2)=O)CN1C(=O)C=C1CCCC1 c1(CSCCC(N2CC(C(C)NC(C3CC3(Cl)Cl)=O)C2)=O)ccccc1 c1(C(=O)NC(C)CCNC(C2CC2F)=O)cc(F)cc(S(N)(=O)=O)c1 C1(C(N2CCC2COCc2ccccc2)=O)CCN(C(C2(C3CC3)CC2)=O)CC1 c1(CC)sc(C(N2CCC(C(C)NC(=O)CS(=O)CC)CC2)=O)cc1C N1(C(=O)COCCC2CCCC2)CCCN(C(c2cnn(CCO)c2)=O)CCC1 c1(C(=O)NCC2(NC(c3ncc(Cl)s3)=O)CCOC2)ccc(O)cc1 N1(C(CC(C)CC(C)(C)C)=O)CCC2(CCCC2NC(=O)C2=CCOCC2)CC1 c1(C(=O)NCCC=C=C)ccccc1C(=O)N(CC=C)Cc1ccccc1 N1(C(c2n(CC)cnn2)=O)CC2CCC1C(CNC(=O)C=CC=C(Cl)Cl)C2 C1(C(=O)NCCSCC#C)CN(C(=O)C(=O)NCC(F)F)CC12CCC2 c1(C(N(C)CCC2CCCCN2C(C2(F)CC2)=O)=O)cc2n(n1)CC1(CC1)C2 C(=O)(C(CC(C)CC)NC(=O)Cc1cnn(CC)c1)NC(CCC)C1CC1 N1(C(c2c(C)nn(CC)c2C)=O)CCC(Nc2ncncc2Cl)C2(CCC2)C1 N1(C(CSCc2nnc(C)s2)=O)CCCCCC1COC(C1CC2CC2C1)=O c1(OC(C(CCC)F)=O)ccc(=O)n(C2(C(=O)OCC)CCCCC2)c1 N(C(=NCC(C)C)NCC1CC(=O)N(c2ccccc2)C1)C(C#C)CC1CC1 c1(C(=O)NCC(C)N(C(C(C)Nc2scc(C)n2)=O)C)ccc(C2CCC2)nc1 Cc1cc(C)c(C(=O)CN(C(=O)CN(C=O)Cc2cc(F)cc(I)c2)C)cc1C N1(Cc2ccc(COCC)o2)CCC=C(C(=O)Nc2cnc(C(F)(F)F)nc2)C1 C12(C(=O)NCC3(CCOCC)CC3)CC(CO1)N(C(=O)CNc1ncccn1)C2 C(C(=O)N(C)CCNC(c1c(C)c[nH]c1CCO)=O)(C(C)(C)C)c1ccc(C)s1 c1(OC)ccc(C(N2CCCC(NC(C3CC(=C(F)F)C3)=O)C2)=O)cc1Cl C1(C(=O)NC2CN(C(C3ON=C(CC)C3)=O)C(C)C2)CCc2nnn(C)c2C1 n1(C(C)C)nc(C2CC2)cc1NC(=O)CCCc1ccc(Br)cc1 N1(C(C=C(CC)C)=O)CCC(C2(NC(=O)CN3CCS(=O)CC3)CC2)C1 N1(C(C=NOC)=O)CCN(C(c2ncccc2F)=O)CC1c1ccccc1Cl c1(C(N(c2nc(C)c(Br)cn2)C2CCCCNC2)=O)ccc2ncccc2c1 c1(C(=O)NCCN(C(=O)CCc2cnn(-c3ccccc3)c2)CC)ccncc1 C(CC(O)C(F)(F)F)NC(CCN(C(C(COCC)C)=O)CCO)=O c1(OC)cccc(OC2(CC(=O)OCC3CCCC(=O)O3)CCC2)c1 C(=O)(C1=C(C)CCOC1)NC1C(NC(CCN(C)CC)=O)COCC1 N12CCC(C(OC)C1)NC(=O)C2c1cc(Cl)nn1C.C(COC)OC.CCOC C1(C(C)C)COCCN(C(C2CCC(NC(c3cncc(O)c3)=O)CC2)=O)C1 N1(C(CC2ON=C(C)C2)=O)CCCC1(C)CNC(=O)COCC(C)(C)C N1(C(c2c(C)n(C3CCC3)nc2)=O)CCCN(C(C2CC(C)(F)C2)=O)C(C)C1 c1(CC)ncnc(CC)c1C(N1CCOC(CS(=O)(=O)NCC)C1)=O C=CCC(C)(CC)C(=O)N1CCC(NC(=O)CCCC2CCCCC2)C(O)C1 N1(CCC#C)CCC(C(=O)NC2(CCNC(=O)C(C)C3CCC3)CCC2)CC1 C#CCC(CC#C)C(=O)N1CCC(CF)(NC(=O)Cn2nnnc2C(C)C)C1 C1(CC=C)(NC(=O)C(F)OC)CCN(C(c2cc(C)c[nH]2)=O)C1 C(=O)(CC(C)(C)CC(F)(F)F)NCC1CC(NC(C2CC(CC)OCC2)=O)C1 C(=O)(C1CCCc2n[nH]cc21)NC(CCNC(c1n(C(C)C)nnc1)=O)C C(=O)(C(F)CCC(C)(C)C)NCC(C)N(C(c1ccc(C)c(O)n1)=O)C N1(C(C2CC(=C)C2)=O)CC(C2CCCN(C(C3CC3(F)F)=O)C2)C1 c1(OC)ccc2cc(CC(N3CCN(C(C4CC4Cl)=O)CC34CCC4)=O)ccc2c1 c1(C(=O)NC(C(C)C)CNC(C2OCC2(C)C)=O)cnn2c(C)cccc12 S(=O)(=O)(CCS(=O)(=O)C(F)(F)F)C(CCc1onc(C)n1)=O.C12(N)CNCC(C)(C1)C2 N1(C(C(C)NC(CC)=O)=O)C2CCC1CN(C(C1CN3CCN1CC3)=O)C2 n1(CC(N2CC(CN(C(CC=CC=C)=O)CC)C2)=O)nc(-c2cccs2)oc1=O C1(C(N2CCC(CCNC(C3CSC3)=O)CC2)=O)CSc2ccccc2O1 C1(NC(COC(CC)(C)C)=O)CCCCC1CNC(=O)C(n1ccc(C)n1)C C(C(=O)N1CCCO1)NC(C(C1CC(C#N)C1)NC(C1OC2CCC1C2)=O)=O C1(CC(=O)NCCc2cn(C3CCC(C(=O)O)C3)nn2)Cc2cccc(Cl)c2O1 O=S(=O)(c1ccc2nc(N3CCC(=C(F)F)CC3)sc2c1)NC1CCCC1O c1(C(N(CC(O)CNC(=O)CCn2ccnn2)C)=O)ccc(CC2CC2)s1 C12(C(N(C)C3CC3)=O)CCN(C(c3cnc(Cl)s3)=O)CC1C2 C(=O)(CC(CCC)NC(c1conc1C)=O)N1CC(=C)C1 C1(C(=O)NCC2CC(NC(Cc3nnc(C)s3)=O)C2)CCS(=O)(=O)N1C CC1CN(C(=O)CCCS(N)(=O)=O)CC(C)N(C(=O)Cn2ncccc2=O)C1 O=C(C(F)CC1CN(C(C2C=CCS2)=O)C1)Nc1cnn(CCF)c1 C(=O)(CCCC(=O)NCC1CN(C(=O)C(C)N2CC(OC)C2)C(C)(C)C1)OCC c1(C(N(C2CCN(C(=O)COC(C)C)C2)CC)=O)cnn2c(C)cccc12 c1(C(=O)NCC2CC(NC(C3(OC)CCCC3)=O)C2)cnc2occc2c1 C(=O)(CC(C)CC(F)(F)F)N(CC(C)NC(Cc1nnc(C)o1)=O)C c1(CNC(C)(CCBr)c2nnnn2C2CCC2)cccc2ccsc12 C1(C(N2CCC(OCCNC(=O)CC3CCC(O)C3)C2)=O)CC2C=CCC(C1)C2 C(C(=O)NCCC1CCN(C(=O)C(F)n2cccn2)CC1)(C(C)(C)C)SC Cc1cnc(N)c(C(N2CC(CNC(=O)CCOC(C)C)CC2(C)C)=O)c1 c1(C(=O)NC2CCN(C(CC3(C=C)CC3)=O)C2C)cc(Br)cn2ccnc12 c1(C(=O)NC2CN(C(c3cnc(SC)n3C)=O)CC2F)cccc(Cl)c1C C(C)(C)(CCCC(=O)N(C)CC1CC1)NC(C(COCC)C)=O Cc1cc(C(=O)N(C2CCN(C(C3(F)CCOC3)=O)CC2)C)ccc1C1CC1 c12ccc(cn1)CNC2=O.N1(C(C)(C)C)CCC1C(=O)NC1CC(NC2CC2)C1 N1(C(C(C(C)C)O)=O)CCCOC(CNC(=O)CCNC(=O)C=CCl)C1 N1(C(CC2CCN(CC3CC(C)OC3)C2)=O)CCOc2ccccc21 C1(C(=O)NC2(CNC(CC(C)n3cccc3)=O)CC2)COC2(CCC2)C1 C(=O)(C(C)(C)C1=CCN(C(=O)C=C2CCC2)C1)NCC1CCN(CCC)C1 c1(C(=O)NCC2C(C)CCCN2C(c2cncc(F)c2)=O)cc([N+](=O)[O-])nn1C O=C(C1=CCCN(C(C2C3CCC(=O)C23)=O)C1)N1CCCC1CF C1(NC(CCCCOC)=O)CN(C(=O)CCc2cc(C)no2)C2CCCCC12 c1(C(=O)NC2C(C)CN(C(C3CCCC3O)=O)C2)coc2c1C(O)CCC2 CC(C)C(CCO)NC(=O)CC1(N(C)C(c2ccc[nH]2)=O)CC1 Cc1ccc2nc(C(=O)NC3CC(C)CN(C(c4cc(C)ns4)=O)C3)cn2c1 C1(CCC#C)CCCCN1C(=O)CC1CCCN(C(=O)CC=CCC)C1 Fc1ccc(N=c2scc(-c3ccc(Br)cc3)n2CC2CC3C(C2)C3(F)F)cc1 c1(C(N2CCN(C(Cc3nc(=N)[nH][nH]3)=O)CC(O)C2)=O)coc2c(F)cccc12 C(=O)(CN=c1cc[nH]cc1)NCC(=O)Nc1n(C)ccn1 C1(C(N(CC(C)N(C(CCCN(C(C)=O)C)=O)C)C)=O)CCC(NC(N)=O)CC1 N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CC(NC(=O)C(CC)N(C)C)C(C)C1 N1(C(c2cc(C(C)C)cc(C(F)(F)F)c2)=O)C2CCC1C(O)CCC2O C=CCC(C)(C(=O)N1CC2(CC2)CC1CNC(=O)CC(C)COC)N(C)C C1(CC)CN(C(c2sc(O)nc2C)=O)CCN1C(c1cc(Cl)ccn1)=O C(CC(C(=O)NCC(O)CNC(=O)CC1CCNC(=O)C1)NC(C)=O)SC N1(C(C(CC)OC)=O)CC2CC(NC(c3c(OC)nsc3OC)=O)C(C2)C1 CCC(CC)C(F)C(=O)N1CCC(C(C)(C)C(N2CC[Si](C)(C)C2)=O)C1 c1(C(=O)NC2CCCC(NC(c3ccc(C)nc3)=O)CC2)ccc2occc2n1 C(c1ccc(CN2CCC(C(=O)NC3(CO)CC3)CC2)o1)=CC(=O)OC C1(CNC(c2cc(OC)no2)=O)CCC(CN(C)C(c2ccccc2Cl)=O)CC1 c1(-c2cc(C(=O)NCC3CCN(C)C3)sc2)cccc2c1CCCC2 c1(NC(C2C(C)C2C)=O)ccccc1C(=O)OC.c1ccccc1 c1(NS(=O)(=O)CCOCC2CC2)nccc(N2CCC(CCCO)C2)n1 N1(C(C2C(CC)OCC2)=O)C2CCCC1CN(C(=O)C1=CC3CCC(C1)C3)C2 N1(C(C(C)NC(C)(C)C)=O)CCC2(CCC(CNC(c3ccoc3)=O)CC2)CC1 CCCCC(C(=O)N1CCN(C(c2cc(OC)n[nH]2)=O)CC1)N(C)C c1(C(=O)NCC(CO)NC(c2c(C(C)(C)C)cccn2)=O)ccc2nonc2c1 c1(CC(N2CCCC(NC(C3(C=C)CC3)=O)C2)=O)ccc(C)c([N+](=O)[O-])c1 C(=O)(CCS(C)(=O)=O)NC1(c2ccccc2)CN(c2nccc(SC)n2)C1 c1(C(NOCCCCC)=O)cccc2nc[nH]c12 C(=O)(CC(O)CC(C)(C)C)N1CCC(NC(CCCC#CC)=O)C(C(N)=O)C1 c1(C(=O)NCC2C(C(=O)NC3CN(C)C(CO)C3)CC2)n[nH]c2c1CCC2 c1(CCC=C)ccc(C(=O)NC2(C)CC(NC(C3CCSC(C)C3)=O)C2)cc1 C(=O)(CCCS(N)(=O)=O)N1C(C(CNC(c2c(C)n(CO)nc2)=O)(C)C)CCC1 C1(OC)CC(CNC(c2cnn(C)c2C2CC2)=O)N(C(=O)CCn2ccnn2)C1 c1(C(N(CCC(=O)N(C)CC2CC2C)CC)=O)ccncc1O c1(SC(C)C)ccccc1C(=O)NCC1COCC1NC(c1coc(O)n1)=O Cc1[nH]nc2c(C(=O)NCCC3CN(C(=O)CC(C)(C)O)CC(C)O3)cccc12 c1(N(C(C(CC)C)=O)OC(C2CCCCN2)=O)cnc([N+](=O)[O-])n1C C(=O)(CCCCc1ccccc1)NC1(C)CC(NC(C2CC23CC3(F)F)=O)C1 CCCCC(O)C(=O)NCC1(CNC(=O)C(C)(C#N)CC)CCC1 Cn1cc(C(N2CC(C(O)C(=O)NOC3CCC(O)C3O)C2)=O)cn1 C(=O)(CCCC(=O)N1CC2(CNC(c3c(C)cccc3F)=O)CC1CO2)NC c1(N2CCC(CC(CNC(=O)OC(C)(C)C)OC)CC2)cc(O)nc(C)n1 n1(CC(N2CC(CCCCNC(CC3(C)CCC3)=O)C2)=O)ncccc1=O N1(C(c2ncc(C(C)=O)s2)C(=O)NCCC2(C)CC2)CCCC(CC2CC2)C1 C1(C(=O)NC2(CC#C)CCCO2)CN(C(c2cnn(C)c2CCC)=O)CC1OC c1(C(=O)OC)cc2c(cc1NCCSc1cc(OC)c(C)cc1OC)CCCC2 c1(CN(C)C(c2c(Cl)cnn2C)=O)ccc(CNC(=O)CC2CCC3CC23)cc1 C(=O)(C(CC)CC(C)C)NC(CC#CC)C(=O)NCc1ccc(C#N)cc1 c1(C(c2n(CCCC)nnn2)NCC2CC23CC3)cc2ccccn2n1 N1(C(C2CC(C(C)C)C2)=O)CC2CC(NC(=O)COCC3CCOCC3)C1C2 C#CC1(C(=O)NCC2(C)CCN(C(=O)C(c3cnccn3)C)CC2)CCOCC1 C(CNC(c1cnsc1)=O)(CO)NC(=O)COCC1CCCO1 Cc1cc(Cl)cc(C)c1C(=O)NCC1C(C)CCCN1C(C1CCS(=O)(=O)N1)=O N1(C(CNS(CCOCC)(=O)=O)=O)CCN(C(c2ncn(CC)n2)=O)C(C)C1 C(=O)(C(C)C(O)CC(C)C)NC(CC=CC(=O)NC(CCCC=C)C1CC1)(C)C CC1CN(C(=O)COc2ccccc2Cl)CCC1CNC(=O)CC(=O)N(C)C c1(C(N2C3CC(NC(c4cn(CC)nc4)=O)(C3)C2)=O)c(Cl)c(CC)nn1C c1(C(N2CCCC(NC(c3ccc(CO)s3)=O)C2)=O)cnc(=NCCF)[nH]c1 c1(OC)cc(CN2CCC(O)C(C(=O)NCCCS(C)(=O)=O)C2)ccc1I c1(C(N2CC(NC(c3c[nH]c4ncc(Cl)cc34)=O)C2)=O)cc(F)c(F)c(Cl)c1F CC(C)(O)C(C(=O)NC1CCCC1C(C)(C)C)NC(=O)C(=O)NCC(F)F c1(CNC(C2CC(NCc3c(C(=O)OC)ccs3)C2)=O)cn(C)nc1C C(CCCCC(=O)NC1CC(NC(=O)C(C)Oc2ccccc2)C1)OC CCCCC(C(=O)NC1CC=CCC1C(=O)NCC(c1cnc[nH]1)C)N(C)C c1(CC(=O)NC2CCC2CNC(=O)Cc2ccc(Cl)s2)csc(Cl)n1 N#Cc1ccc(C(=O)NCCCN(C(=O)COC2CCCOC2)CCO)cc1 c1(C(=O)NCC2N(C(C(C3CCCC3)OC)=O)CC2)ccccc1C1(C#N)CC1 N1(C(C(C)CF)=O)CCC2(CCCC(CNC(=O)CC3(CS(C)(=O)=O)CC3)O2)CC1 C1(C#N)(OC)CC(C(N2CCC(n3cc(C4CCCC(O)C4)nn3)C2)=O)C1 n1(CC)nc(C2CC2)cc1C(=O)NC1CC(NC(=O)C(C)NS(C)(=O)=O)C1 C(=O)(C(C)CC(N)=O)NC(CNC(C1(C)ON=C(C)C1)=O)(C)C1CC1 CC(CCNC(=O)CNC(=O)CN)n1ccnc1 c1(C(=O)NC2CC(NC(c3ccc(C)c(C#N)c3)=O)C2)ccc(S(N)(=O)=O)cc1 c1(C(=O)NC(CC(C)C)(C)CNC(=O)CC2CC(=O)C2)cc2ccccc2[nH]1 N1(CCCOC(C)C)CCC(CNC(c2cscc2C(F)F)=O)C1 C1(C(=O)NC2C=CCN(C(=O)CCC3CCCCC3)C2)CC12CCOCC2 c1(C(N2CC(C3(NC(C45CCC(C4)OC5)=O)CC3)C2)=O)noc2c1CCCC2 N1(C(c2cn(CC=C)nn2)=O)CCC(C)(NC(=O)Cc2c(Cl)cccc2Cl)CC1 c1(C(N2CCCC2c2cnn(C)c2)C(=O)NC2C(C)=C2)cnc2cc(C)nn2c1 C12(NC(C=C(C)C)=O)CCN(C(=O)CCc3ccc(F)nc3)CCC1C2 C(C(CCC)C(=O)N(C)C)NC.n12cccc(c1=O)C(=O)Nc1ccc-2nc1 c1(SC)ccc(CNC(C2(Cl)CC2CNC(=O)CSc2nc[nH]n2)=O)o1 N1(C(C(C)NC(C=C)=O)=O)CC2OCC(C(=O)NC)C2C1 Cc1cnc(C(N2CCN(C(c3nccc(Cl)c3F)=O)CC2C)=O)c(F)c1 N1(C(C(C)OCC)=O)CCC2CCN(C(C3CCc4n[nH]c(C)c4C3)=O)CC2C1 c1(NCCCN(C)C(c2cnn(C3CCOC3)n2)=O)ncn(C)c(=O)c1Br N1(C(c2n(C(CC)CC)nc(C)c2)=O)CCOC2CCN(C(C3CC3F)=O)CC12 C1(C(C)C)CN(C(c2ccccn2)=O)CCN1C(=O)C=Cc1csc(Br)c1 c1(N(C(C)CCNC(c2ccc(Cl)cn2)=O)C)cc(O)nc(O)n1 C1(C(=O)NCCOCC#C)CCCCCCN1C(c1conc1CC)=O C1(C)(C(=O)NCC2(C(=O)NC(C=C)C3CC3)CCCC2)CCCCCC1 C1(C(N(CCNC(C(C)(C)NS(C)(=O)=O)=O)C2CC2)=O)CCCC12CCOCC2 N1(C(C(C)Cc2ccco2)=O)CCCC(C2CCN(C(C34CC(F)(C3)C4)=O)C2)C1 c1(C(=O)NCCN(C(C2CC(n3ccnn3)C2)=O)C2CC2)cnccc1Cl c1(COC)ccc(C(=O)NCC(C)N(C)C(c2cncc(C(N)=O)c2)=O)cc1F N1(CC)CCCC(c2nnnn2C2CCC2)(NC(c2cc(Cl)cc(Cl)c2)C)C1 N1(C(Cn2c(C)ncc2)=O)CC(NC(c2nn(C)cc2Cl)=O)CCC1C Cc1ccc(Nc2ccc(C(C)NC(=O)CCc3cnccn3)cc2)cc1C C(C(=O)NCC1(C)NC(=O)NC1=O)(C(C)(C)O)NC(c1nc(OCC)oc1)=O c1(C(=O)NCCCCCN(C(CC2(C=C)CC2)=O)C)nccc(Cl)c1Cl N1(C(c2ccc(OC)nn2)=O)CC(NC(c2nc(C)nn2C)=O)CC1(C)C c1(CC(=O)NC(C)C(C)NC(=O)CNC(=O)Cc2ccccc2)cncnc1 c1(C(N(C)CC2CCCN2C(c2cncc(Cl)c2)=O)=O)c(N)cccc1F n1(CCCC(=O)NCC2CCCC2NC(C2CC(CC3CC3)C2)=O)ccccc1=O CC1(C)CN(c2nc(Cl)c(C(F)(F)F)nc2N)CC(C(F)(F)F)O1 n1(CC)cc(NC(=O)C(CC(F)F)NC(=O)CC2=CCCC2)ccc1=O c1(C(c2cnsc2)NCC(=C)C)nnnn1C1CCOC1 C(=O)(C(O)Cc1cn(C)cn1)NC(CNC(C1(C(=O)NC)CC1)=O)C c1(SC)cnn(C)c1C(=O)NCC12CC1CN(C(=O)C(C)C1(O)CCC1)C2 S(=O)(=O)(c1ccc(NC2CCOC(C(F)F)C2)cc1Cl)N(CCN(C)CCO)C C1(CC(=O)NCCC2CN(C(C)=O)CCO2)(CNC(C)=O)CCCCC1 N1(C(c2ccc(CN=[N+]=[N-])o2)=O)CC(F)(F)CC1CNC(C1CCC=CO1)=O N1(C(c2cccc(C(C)C(F)(F)F)c2)=O)CCC(O)C(C(N2CCOCC2)=O)C1 c1(NC(C23C(CN(C(c4cc(O)cc(F)c4)=O)C2)C3)=O)cccn2ncnc12 c1(C(=O)NCCC2N(C(c3cnc(C)o3)=O)CCOC2)cccc2nnn(C)c12 C(=O)(C(O)CC(C)(C)C)N1CC(CNC(Cc2n(C)ncc2Cl)=O)C(C)(C)C1 C1(CC(F)F)(CNC(=O)NCCNC(=O)OC)CCCO1 N1(C(=O)CSc2ccncc2)CCC2(NC(C3(F)CCOC3)=O)CCCCCC12 CC(C)(C)C(CC(=O)NC1CCC(NC(=O)C2Cc3ccc(F)cc32)C1)C(F)F CC(CCCNC(c1cncs1)=O)NC(=O)C(c1ccccc1)NC(N)=O c1(C(=O)NC(C2(NC(=O)COCCF)CC2)C)ncc(F)cc1F C(CCCCCNC(c1cnn(-c2ccccc2)c1)=O)N(C(=O)C(CO)N(C)C)C N1(C(C(C2CCC2)OC)=O)CCC2(CCOC2)C(CNC(=O)CN(C)C)C1 C(=O)(C1=CC(C)(C)C1)N(C1CCC(N(C)C(C2C3CCCCC23)=O)CC1)CCO c1(OC)ccc2c(C(=O)NC3CC4CN(C(c5cc[nH]n5)=O)CC4C3)cnn2c1 c1(COCC(N2CCC2C)=O)cn(CCO)nn1.C1CCSCC1 CCCCCC(CC)(c1nnnn1CCC1(C)CC1)NC(COCC)CCO c1(CC)cc(Cl)ccc1C(=O)NC(C)C(C)NC(=O)C(C)(C)NS(C)(=O)=O c1(C(N(CCC(C)NC(c2cncc(-c3cc[nH]n3)c2)=O)C)=O)ccc(=O)oc1 N=c1nc2c(c[nH]1)CC(C(=O)NC1(CNC(c3cc4c([nH]3)CCC4)=O)CC1)CC2 C12(C(N(C3CN(C(=O)CC4CCC(F)(F)C4)CC3O)C)=O)CCC(F)(CC1)C2 O=[N+]([O-])c1cc(F)c(CNCCCOCC2CCOC2)c(F)c1 Cn1nc(CNC(C2CCCN2Cc2ccc(Br)cc2)=O)n(C)c1=O N=c1[nH]cnc2cc(C(N3C4CCC3C(CNC(=O)COC=CCl)C4)=O)ccc12 C1(NC(C2C3C(NC(C(C)=C4CC4)=O)C4C(C3)C42)=O)CC(C)(C)C12CCC2 Cc1cc(=NC(=O)C2CCCN(C(=O)N3OC4CCC3CC4)C2)[nH]n1C c1(CC)cccc(NC(C2CCCN2C(c2ccc(C(C)O)cc2)=O)=O)c1 C1(NC(c2cc(Br)sn2)=O)CCCN(C(=O)CN(CCO)CCO)C1 C=CC(C(F)(F)F)NC(=O)C(CCC1CCC1)NC(=O)CCCn1ccnc1 CC(=O)CCCC(=O)N1CCN(C(=O)Cc2ccc(C)cc2Cl)C(CC2CC2)C1 c1(C(N(CC(CC)NC(c2ccc(C(N)=O)o2)=O)C)=O)ccc2occc2c1 O=S(=O)(c1ccc(NCC2CCCCO2)cc1Cl)NCCc1ncccn1 N1(C(c2ccc(F)c(C)c2)C(=O)NC)CC2(COC(=O)C2)C1 S(=O)(=O)(c1ccc(Br)cc1Nn1cccn1)N1CCCC(NC(N(C)C)=O)C1 C(=O)(C1=CCCOCC1)NC1C(CC)CN(C(c2occc2C2CC2)=O)CC1 c1(C(=O)NC2C(C)(C)CN(C(=O)C3=CCS(=O)(=O)C3)CC2)cccc2ncccc12 Cc1nc2ncccn2c1C(N1CC2CC1CN2C(=O)C(C)S)=O C(=O)(C#CC1CCCCC1)N1CC(C)(CNC(C2CSCC(=O)N2)=O)OCC1 C1(CC)C(C(N2CC(c3ccn(C)n3)C2)=O)CCCN1C(=O)Cn1cccn1 C1(NC(c2cc(OC)no2)=O)CC2CC(NC(=O)C=C(C)C(C)(C)C)C2C1 c1(NC(CC2C(NC(C=CCOCCOC)=O)CC2O)=O)cc(C)c(F)cc1O C(=O)(C1CCOc2ccccc21)N1CC(CC=C)(NC(=O)C(C)CC)C1 C(=O)(C1SCc2cccnc21)NC(C1(CNC(C(C(C)C)(C)C)=O)CC1)C C1(CCNC(c2nnnn2C2CC2)COC(C)(C)C)CCS(=O)(=O)CC1 O=C1CCN(C(C2CC3(CC3)CN2C(=O)CC2CC3CCC2O3)=O)CCN1 CCC(C(=O)NC1CCC(CNC(=O)C(F)(F)c2cnn(C)c2)C1)n1cccn1 c1(C(N2CCN(C(c3scc(C)c3)=O)CC2)=O)cc2c(nc1O)CCCC2O N1(C(CCN(S(CC)(=O)=O)C)=O)CC(CN(C(=O)C(C)N(C)C)C)C2(CC2)C1 N1(C(Cc2c(C)n(C)nc2)=O)CC2CC(NC(C3CC(=C4CCC4)C3)=O)CC1C2 C1(C)(NC(NCC(N2CCCCC2)C)=NCCc2ncccn2)CCS(=O)(=O)CC1 CC(C)(C)C(C)(C)C(=O)NCC(O)CCNC(c1ccc2occc2c1)=O c1(C(=O)NC2CCC(C(=O)NCC(=O)NC)CC2)cc(F)cc(I)c1 N1(C(c2c(N)c(F)ncc2)=O)CC(NC(c2ccc(CO)o2)=O)CC12CCC2 N1(C(Cc2cn(C)nc2)=O)C2CCC(C2)C1CNC(c1cc(F)c[nH]1)=O N1(C(CC2CCCC(C)(C)C2)=O)CCC2(CC1)CC2CNC(=O)CSCC(N)=O c1(C(N2CC(NC(=O)OC(C)(C)C)C2)=O)ccc([N+](=O)[O-])cc1Cl.CC1C(=O)N1 CC1(C)CC(N=c2ccnc(C3CC3)[nH]2)CN(C(c2ccn(CC(F)F)n2)=O)C1 N1(C(COC2CC(OCC)OC2)=O)CC(O)(Cn2cc(-c3cccs3)nn2)C1.C1CC1 C1(C(=O)NCc2cc(OC)ns2)C2CCC(C2)N1C(C1CC2(CC2)C1)=O C#CCCCC(=O)NC(C)C(C)(C)NC(=O)C(C)OCOC Cc1cc2cc[nH]c2cc1C(N1CCOCC1CNCc1cc(C#N)ccn1)=O C1(F)(CNC(COCC=C)=O)CCN(C(c2sc(C#N)cc2C)=O)CC1 CN1CC(C)(C)CC1C(=O)NC1(C(=O)NCC2(CO)CCCO2)CC(F)C1 C1(C(=O)NC2C=CCN(C(=O)C=CC3CCCC3)C2)Cc2ccccc2S1 N1(C(C(CC=C)CC)=O)CCC2(CCCN2C(c2cc(C)c(C)[nH]2)=O)C1 C=CCCC(C(=O)N1CCC(O)C(C)C1)NC(=O)C(C1CCCCC1)C c1(C(N2C3C(NC(c4coc(CO)c4)=O)C(CC3)C2)=O)ccnc2ccccc12 C1(O)(CNC(C(C)CC2CCC2)=O)CCN(C(C2CCC(O)CN2C)=O)CC1 CC1(C)CCCN(C(c2cnsn2)=O)C1C(=O)NCCC1(O)CCOC1 C(CCCC(=O)N1CCCCC1CCO)NC(CCc1cc(C)no1)=O N1(SCCCNC(=O)C(O)C2CCCC2)C(=O)CCC1C(=O)N(C)CCOCC C(CCC(O)C(=O)NCCOC1CCCC1)NC(c1nn(C)c(CO)c1)=O Cc1cc(CCN2CCC(NC(=O)CCCc3ccccc3)C(O)C2)ccc1F C(=O)(CC(C)C(C)(C)NC(c1c[nH]c(=S)cn1)=O)NCC(c1nccs1)C C1(C(=O)NC2(C(=O)NCC(c3nncn3C)C)CC2(C)C)CC(=O)OC1(C)C c1(C(N2C(CNC(C(C)OCC)=O)COCC2)=O)coc2cc(F)ccc12 CC1CN(C(=O)C(c2ccc(Cl)cc2)C)CC1Nc1cc(C(C)(C)C)ncn1 c1(COC)nc2n(n1)CCCC2NC(=O)C(n1cc(C2CC(F)(F)C2)nn1)C c1(C(N2CC(O)(CCNC(c3c(C)cn(C)c3)=O)C2)=O)c[nH]c2cccc(F)c12 C1(NC(c2ncn(C(C)C)n2)=O)CCN(c2ccc(C(F)(F)F)nn2)CC1O c1(OC)ccc(C(=O)NCC2(CNC(C3CCC(C#N)C3)=O)CCC2)c(Cl)n1 c1(C(=O)NCC2CC(C)N(C(C3C4CCCC34)=O)CC2)ccc(F)c(F)c1F C1(O)(C(C)NC(CC2(COC)CCCC2)=O)CCN(C(C2CCSCC2)=O)CC1 C1(C(N(CC(C2CC2)OC)C)=O)(C(C)C)CCCN1C(=O)CC1(C)CCC1 CN1CCN(C2(C(=O)NC3CC(NC(=O)CC4CC5COCC45)C3)CC2)CC1 C1(NC(c2sccc2C2CC2)=O)CCN(C(C23CCC2C3)=O)CC1O C1(NC(Cc2c(C)cco2)=O)CN(C(c2nc(Br)c(C)s2)=O)CC1C C1(C(N(CCCN(C)C)CCC)=O)CCCCN1C(C1CCCOC1)=O c1(N2CCC(C)(NC(C3CCCS3)=O)C2)ccc([N+](=O)[O-])cc1-n1cnnn1 c1(OCC(=O)OCc2ncc(-c3ccc(Cl)cc3)s2)cccc2cccnc12 N1(C(CCCCC=CC)=O)CCCC(C)(C)C1CNC(=O)Cn1nccc1C S(=O)(=O)(c1cnc(NCC2CCCSC2)c(Cl)c1)NC(c1nncn1C)C N1(C(C(C=C)O)=O)CC2(COC(CNC(=O)CCCn3nc(C)cc3C)C2)C1 c1(C(N(CC(C)CNC(c2nc(C(C)(C)C)no2)=O)C)=O)ccc(C2CC2)cc1 c1(C(=O)NC2C(C)(C)CN(C(C3(Br)CC3)=O)C2)ccc2ncccn12 c1(C(N2C(C(N(C3CCCC3)CC)=O)CCCC2)=O)ccc(COC(C)=O)nc1 C1(NC(C(C)c2cncs2)=O)CCC2(CCN(C(=O)C(C)(C)C3CCOC3)C2)C1 C1(C(N2CCC(N(C)C(c3sccc3C3CC3)=O)C2)=O)CC2C=CC1C2 C1(CC)(NC(=O)C=C(C)C)CCCN(C(C2(c3ccc(F)cc3)CC2)=O)C1 c1(C(=O)NC(C)CNC(C23CC(CF)(CO2)C3)=O)c(Cl)cncc1Cl C(CCCCC(=O)N1C2CCC1COC2)NC(C(C)CCN(C)C)=O N1(C(CCCOCC)=O)CCC(C2CCCN(C(c3ccncn3)=O)C2)C1 C(=O)(CCCC(=O)c1ccccc1)NC(C1CN(C(=O)CC2CSC2)CCO1)C Cc1[nH]c(=NCc2ccc3c(c2)CCO3)sc1C(=O)Nc1ccc2c(n1)CCC2 C(C)(C(=O)N(CCN1C(=O)CC1)CCN(C)CCO)O.C=CCCCCC.CCC C1(NC(c2n(CC)ccc2)=O)CCCCC1N(C(=O)C(N1CCC(C)C1)=O)C c1(C(=O)NC(CCCCNC(CCc2nnc(C)o2)=O)C)cc2sccc2s1 N1(C(C2CC(OC)C2)=O)CC2=C(C1)CN(C(C1CCCC1C1CC1)=O)C2 C(=O)(C1=CCCN(C(=O)Cc2cc(Br)ccc2C)C1)Nc1cccc(CCC)c1 c1(C(=O)NC2CCC23CN(C(c2ccc(O)cc2F)=O)C3)nccc2n[nH]cc12 c1(C(=O)NCC2C(NC(Cc3c(C)n(C)cn3)=O)CC2)cc2c(cc1O)OCO2 C(C)(CCC(=O)N(CCCCCNC(=O)CCC(=O)c1ccc(C)s1)C)OCC Cc1[nH]c(C)c(C(=O)NCc2cc(C(N3CC(CC(C)(C)C)C3)=O)no2)c1C C(CC(C)N=c1[nH]c(=NCCc2c(F)cncc2F)c2cccc(F)c2[nH]1)SC C(=O)(CCCCC(F)F)NCCNC(C(c1cn(C)nc1)=O)=O C1(CNC(CC(C)(C)F)=O)CCN(C(=O)C=CC2CCOCC2)CC1(F)F C12(CNC(C=C(COC)C)=O)CCC(CC1)CN2C(c1csnc1Cl)=O c1(CC)ccc(C(=O)NCC(O)CNC(c2cnn(C)c2C(F)(F)F)=O)cc1N Cc1ccc(N)cc1C(=O)NC1CCCCC1N(C)C(C12CCC(C)(C1)OC2)=O N1(C(c2c(CC)onc2)=O)CCOCC1CN(C(=O)CCNC(N)=O)C c1(OC)cncc(C(N2CCC(NC(=O)CCSC3CC3)C(CO)C2)=O)c1C c1(OC)ccc(O)c(C(N2CCCCC(NC(=O)Cc3cnc(C)s3)C2)=O)c1 c1(C(N2CC3C(CNC(C4CC4C(F)F)=O)C3C2)=O)n[nH]c2c1CCC2 C#CC1(C(N2CCC(OCCNC(=O)C(C)c3cc[nH]n3)CC2)=O)CCCC1 N1(C(c2cccc3c[nH]nc23)=O)CCOC2(C1)CN(C(C13CCCC1CC3)=O)C2 c1(C(=O)NC(C)CNC(C23CC(C)(CCO2)C3)=O)cc(F)cc(F)c1N C(=O)(C(O)CCCNC(C1(C(C)(C)O)CC1)=O)N(CCn1c(C)ncc1)C N1(C(c2scc(OC)c2)=O)CCC(NC(c2csc(Cl)c2Cl)=O)C(OC)C1 CC(C(=O)NCC1CC2(CC2)CN1C(c1ccc(O)nc1Cl)=O)S(C)(=O)=O CCCCCCC(CC)(CC)C(=O)NC(CNC(=O)CC1CCC(C)(C)C1)CC C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCC(C)(C)NC(=O)CC1OCCO1 CCC(CC)CC(=O)N1CCCC(C2CCCCN2C(=O)CC2CCC2)C1 C1(C(=O)NC(Cn2ncc(C)c2)C)C2CCC1CN(C(c1ccccc1)=O)C2 C(=O)(CC(C(F)(F)F)NC(=O)CCc1cn(C)cn1)NC1C(OC)COC1 C#Cc1ccc(C(=O)N(CCN(C(=O)C=CSC)C)C(C)C)cc1F c1(C(N(CCN(C(=O)CC2CCCOC2)C)C)=O)ccccc1F C1(C(=O)NC(CNC(c2ccc(C(C)C)s2)=O)C(C)C)OC2CCC1CC2 C1(C2CCN(C(=O)CC3(C(F)(F)F)CC3)CC2)(NC(CCS(C)(=O)=O)=O)CCC1 C1(C(=O)NC(C)(C)CCNC(C2CC(O)C2)=O)COCC1(C)C C1(CNC(CCCCC)=O)CCN(C(=O)CCc2ccc(Br)s2)CC1C c1(OC)ccsc1C(=O)NCC(O)C(=O)NCC(C)OCCO C=CCC(CC)C(=O)NC1(C2CN(C(=O)C(=Cc3cnn(C)c3)C)C2)CC1 CCCCC(C)C(=O)NCCOCCNC(C1(c2ccccc2)CC12CCC2)=O N1(C(C(=O)N(C)CCOc2ccccc2)=O)C2CC2C2CC12 C1(CNC(CC=CCC)=O)CC2(CCN(C(=O)CCSC)C2)CO1 CCC(C(=O)N(C(C)C(=O)NCC1CCOC(C)(C)C1)C)C(C)(C)CC C1(C)(CC)CC(NC(=O)Cc2ccc(C)nc2)CN1C(=O)C=Cc1ccc(C)o1 N1(C(C(CN(C)C)NC(CC2C(C)=NNC2=O)=O)=O)CCn2c(C)cnc2C1 CCC(C(=O)NCCC1(NC(c2cc(C3CC3)ccn2)=O)CCC1)C(C)(F)F N1(C(C2CC3(CC(NC(c4ccnc(C)n4)=O)C3)C2)=O)CCc2cnccc2C1 Cc1nc(C)c(C(N2CCC3CN(C(=O)CNC(C4CCC4)=O)C3C2)=O)c(C)n1 c1(C(=O)NCC(C(C)C)NC(C2CC=CCO2)=O)nn2ccccc2c1Br N1(C(c2nncc(CCC)c2)=O)CCC=C(CNC(=O)CCCC(C)C)C1 N1(C(C(CCC)(C)C)=O)CC=C(CCNC(C2CCC23CCCO3)=O)CC1 C=C(C)C1OCCC1C(=O)N(CC(CC)NC(C1CC(=O)CCO1)=O)C c1(-c2cnc(OC)s2)nc(C2OCCc3ccccc32)nn1CC(C)C N1(C(c2c(C)nn(C)c2)=O)CC2CCOCC2(NC(c2cc[nH]c2C2CC2)=O)C1 c1(CC)ncsc1C(=O)NCC(C(C)C)NC(=O)C(c1cncnc1)C c1(C(C)C)ncc(C(N2CCCC2C(C)NC(=O)CNC(=O)NC2CC2)=O)s1 C1(C(=O)NCCC(=C)CNC(c2cncc(Cl)c2C)=O)C2CCCCCC12 CC1CCCN(C(C2CC(CNC(C3CC4CCC4C3)=O)C2)=O)C1 c1(C(C)=O)ccc(C(=O)NCC2(CNC(c3cncn3C(C)C)=O)CC2)s1 N1(C(=O)C=CC2CCCO2)CC2(CCCN2C(c2cccc3scnc23)=O)C1 c1(CC(=O)NC2(C(N3CCC(CC)C3)=O)CCC2)ccc(F)cc1 c1(CC)ccc(C(=O)N(CC(C)CNC(=O)C(C)N(C)C)C)cc1[N+](=O)[O-] C1(NC(=O)CCOc2ccccc2F)CCCC2CN(C(C3CC(O)C3)=O)CC12 C1(CCC)(NC(c2coc(Cl)c2)=O)CCN(C(=O)C(=O)NCC2CC2)CC1 C1(NC=O)CCCC1COC(C1(NC(C2(CCCC)CCC2)=O)CC1)=O.SC C1(CCC)C2CN(C(=O)C(=O)NCc3csc(-c4ccc(C)o4)n3)CC12 N#Cc1cc([N+](=O)[O-])cnc1N1CC2CN(C(=O)CCn3cccn3)CC2C1 C#CCCC(=O)NCCOC1CCN(C(=O)CC2CC2C(F)(F)F)C1 C1(NC(C(OC)OC)=O)C2CC(O)C1N(C(c1cccc3nn[nH]c13)=O)C2 Cc1ccc(C2CC2C(=O)NC(C)(C)C(C)NC(=O)CCc2nncs2)s1 C(=O)(C(C)C(=O)N1CCCCC1CC(=O)NCC12CCC(CC1)C2)OC N1(C(C2(CC=C)CCCC2)=O)CCCC(O)(CNC(c2sccc2COC)=O)C1 C(=O)(CCCC(F)(F)CO)N1CCC(C)(C)C(CNC(=O)CSC(F)F)C1 C1(C(=O)NCc2ccoc2C(=O)NCc2nncs2)CC2(CCC2)C1 CCC(CCC(=O)N1CC(N2CC(F)C2)C1)NC(c1cc[nH]c(=NC)c1)=O c1(OCC)c(Cl)cc(C)nc1C(=O)NCC1(O)CN(C(=O)C=Cc2cccs2)C1 C(=O)(C1=NOC(C)C1)NCC(C1CCCCC1)NC(CC1(CSC)CC1)=O c1(NC(C2C3(c4ccc(OC)cc4)COC2C3)=O)c([N+](=O)[O-])ccc(Cl)c1Cl CC(C)C(C)C(C)CC(=O)N1CCN(C)C(CF)C1 N1(C(C(CN(C)C)O)=O)CCC(C(=O)NCc2ccc(F)cc2F)C1(C)C CCCC(CC)(c1nnnn1CCOC)NC1(C)CC1(C)C S(=O)(=O)(c1ccc(Br)cc1Br)N1CC(OCCCCC)C1 N1(C(CN(CCCCCC)C)=O)CCCC(CNC(C2CCC(=O)N2)=O)CC1 C1(C(N(CC(C)NC(c2ccnn2CC#N)=O)C)=O)CCC(=O)C1 c1(C(=O)NC2CC(N(C(CC(C)C(F)F)=O)C)C2)ncnc2c1CCCC2 N1(C(CCc2cn(C)nc2)=O)CC(C(F)(F)F)CC1CNC(C1C(C#N)C1(C)C)=O c1(C(N2CC(C#N)C(NC(=O)Cn3cccn3)C2)=O)cccc2[nH]ccc12 C(=O)(C(C)(O)CC)NCC(CO)NC(c1c(C)nns1)=O.C(C)(C)(C)OC(C)=O c1(-c2n(CC(N3CC(CC(=O)OC)C(=O)CC3)=O)c(=O)on2)cccc(O)c1F C(CCS(=O)(=O)c1ccc(NS(=O)(=O)c2sc(Br)cc2OC)cc1)OC c1(OC)ncc(C(N2CCN(C(=O)CC(C)N(C)C)C(CC(F)F)C2)=O)cc1Cl c1(C(C2(C(=O)NCC(C)N(C(CCCCC)=O)C)CC2)=O)cnc(OC)cc1C c1(NC(c2ccncc2)CNC2CCCCO2)cc(N2CCOCC2)ncn1 N1(C(C(F)=CCC)=O)CCC(NC(c2ccc(F)c(C(C)(C)F)c2)=O)C(F)C1 Cc1ccc(C(N2CCC(C)C2CNC(c2ccn(C3CC3)n2)=O)=O)cc1CO c1(CC(=O)NC2CCN(C(=O)CNc3nccs3)CC2F)ccccc1[N+](=O)[O-] N1(C(C2(C)CCN(C(Cc3cc(C)[nH]n3)=O)C2)=O)CCSCCC1C c1(C(=O)NCC(C)N(C(C(CC)=CC)=O)C)cnc(C(F)(F)F)cn1 CC(C)C(C#N)C(=O)N1CCCC(N(C)C(c2ccc(N(C)C)cn2)=O)CC1 CN=c1[nH]cc(C(=O)NCC2CN(C(C3(O)CC3)=O)CCO2)s1 C(=O)(C(C)(F)C(F)(F)F)NCCC1(O)CN(C(C2(C(C)C)CNC(=O)C2)=O)C1 CC1(C(=O)NCC2CC2CNC(=O)C(c2cccc(N)c2)O)CCNC1=O C(=O)(CS(=O)CCC(F)(F)F)NCCCCCn1cc(CCOC(C)=O)nn1 C(c1ccc(Cl)cc1F)=CC(=O)NCC(CNC(C1CC2CC2C1)=O)OC C1(NC(=O)Cc2ccn(C3CCCC3)n2)CC2CC1N(C(c1n[nH]cc1Cl)=O)C2 CCC(Cc1ccccc1C)C(=O)N1CCC1CNC(C1(C(=O)NCC)CC1)=O c1(OC)ncc[nH]c1=NNC(=O)CC(N)C(C)(C)C C#CCC(CC(F)F)NC(C1(F)CN(C(C2CCC(F)C2)=O)C1)=O C1(NC(C2OCCC(C)(C)C2)=O)CCC2(CCN(C(C3(CO)CCOC3)=O)C2)C1 CC1(C2(C(=O)NC3CN(C(=O)CN=[N+]=[N-])CC3CO)CC2)CC1 C(C(C)(C)C#CC(=O)NCCC1(C)CC1)NC(C(C)(C)NC(C)=O)=O C1(F)(CNC(C=CCOC)=O)CCCN(C(=O)C(C)(C)Oc2ccccc2)C1 C1(NC(CN(C)CCO)=O)CCC2(CC1)CC2NC(c1ccc(C#N)c(F)c1)=O C1(NC(=O)C2=NOCC2)CC2(CCN(C(c3cc4c(cn3)CCCC4)=O)CC2)C1 N1(C(CC(C)(C)O)=O)CC2(C1)CN(C(=O)CCCC1CCC1)CCO2 C1(NC(c2c(C)cco2)=O)CN(C(=O)CC(c2ccccc2)N(C)C)CC2CC12 c1(CC)cc(C(=O)NCC2=CCN(C(=O)CN(C)CC)CC2)ccc1Br Cc1cc(C(=O)Nc2ccc(OC(F)(F)F)c(F)c2)n2nc(C)cc2n1 c1(OCC)cccc(CC(=O)NC2(CCNC(C3CCOC(C)C3)=O)CC2)c1 N1(C(C2C(C)(COC)C2)=O)CCN(C(c2cccc3[nH]ccc23)=O)CC(C)(C)C1 CC1(F)CCN(C(=O)C(c2cccnc2)NC(=O)C(F)OC(F)(F)F)CC1 Cc1cccc(N(NC(=NCC2CC2Cl)NCC(C)(C)c2cccs2)C)c1 c1(C(C)N(C(=O)C(=O)NC2CC2)C)ccccc1F.c1(N)ccccc1 Cc1cc(=NC(=O)C2C3CC4C(C3NC(=O)C(c3cccn3C)=O)C24)[nH]n1C N1(C(C(C)NC(C)=O)=O)Cc2ccccc2C(CNC(=O)C=C(C)C(C)(C)C)C1 Cc1ccc(CN(CC(C)C)C(c2ccnn2C2CC2(F)F)=O)cc1 N1(C(C2N(C(c3cc(C(C)=O)[nH]n3)=O)CC(F)C2)=O)C2CCC1CN(C)C2 C(CC(C(C)(C)C)NC(c1cc(CO)n(C)n1)=O)N(C(C1CC(C#C)(O)C1)=O)C Cc1cc(C(N2CCCCC2c2ocnc2C(=O)O)=O)cc(F)c1 N(C)(C1=NS(=O)(=O)c2ccccc21)Cc1n(CC(=O)OCC)nc(C)n1 CCCCCCC(CC)NC(=O)NS(=O)(=O)CCOC c1(C(=O)NCC2(F)CCC(NC(c3c(C)ccs3)=O)C2)cc(O)cc(Cl)c1Cl c1(OCCC(=O)NC2(CF)CCN(C(C(CCC)O)=O)C2)ccc(Cl)c(F)c1 C(=O)(CC1OCc2cc(Cl)ccc21)NCc1scc(CNC(CCC(C)C)=O)n1 n1(CC)ccc(C(N2CC(CF)(NC(=O)C=Cc3cccnc3)C2)=O)c1C N1(C(c2cc(C)oc2C)=O)CC2CCCC2(NC(C2Cc3nnc(C)n3C2)=O)C1 N1(C(c2cccc(C)c2)=O)CC(CNC(=O)C=C2CCN(C)CC2)CC12CCC2 N1(C(C=CCC(C)(C)NC(C2C(OC)(OC)CC2)=O)=O)CCC(C)C(C)C1 C1(CNC(C2(C)N(C)CCC2)=O)CC(C)(C)CN1C(c1ocnc1C1CC1)=O c1(N2CC(C)(C)C(CO)C2)ccc(S(=O)(=O)N2CCc3ccccc3C2)cn1 C(=O)(C1=CCSC1)N(C(C(=O)NC(c1cnn(C)c1)C)(C)C1CC1)C Cc1cnc(C(=O)NCC(C2CCCC2)NC(=O)CN2CCCC2)cc1C#N C1(CN(C(c2nc(CO)no2)=O)CC)CCCN1C(=O)C(C)Sc1nncn1C CC(C)C(F)(F)CC(=O)N1CCCC1CNC(=O)CCC(=O)c1ccc(O)cc1 C(=O)(C1COc2ccccc21)N1CC(CCCCNC(C2CCC(C)C2)=O)C1 C12(C(=O)NCCSCC(C)C)CC(CN(C(=O)CC3CCC(C)O3)C1)C2 c1(C(=O)NC2CCN(C(c3cc(C)sc3)=O)CC2O)cc2sc(C)cc2s1 CN1CCOC(C(N2CC(C(=O)NCCNC(C3(O)CCN(C)C3)=O)C2)=O)C1 N1(C(CCC=C)=O)CC2(NC(c3cnc(C(C)(C)C)nc3)=O)CCC1C2 CN1CCN(C(c2occ3c2CCC3)=O)C(C(=O)NC2CCC(F)CC2)C1 C=CCC(CC=C)C(=O)N1CCCC1C(=O)Nc1ccc(F)c(CO)c1 C(CNC(=O)CCc1cnn[nH]1)(CNC(=O)CCOCCN(C)C)OC C1(C(=O)NC(C#C)CC2CCC2)(CNC(=O)C(F)C(=O)OC)CC2(CC2)C1 C1(C(N2CCC(CC(=O)NC(COC)(C)C3CC3)C2)=O)CCCCC1(C)C c1(SCC)ccccc1CC(=O)NC1CCCCC1NC(=O)CC1CC=CCC1 C(=O)(C1=C(Cl)CCOC1)NC1CC(NC(=O)CC(C(F)F)c2ccc(F)cc2)C1 c1(CCCC)cc(C(N2CCCC(NC(=O)CCCNC(C)=O)C2)=O)c(C)o1 N1(C(CCOCC#C)=O)CC(NC(=O)CS(N)(=O)=O)CCC1C C(C(c1ccccc1)NC(c1onc(C)c1C)=O)(C(C)C)NC(COCC)=O C1(C(=O)NCC2(C=C)CCC2)(NC(C2CCOC2C(C)C)=O)CCCCC1 N1(C(=O)CN2CCC2)CCCCC(C2CN(C(c3cnsn3)=O)C2)C1 C(=O)(CCCCN=c1[nH]c(=NC2CC(CC#N)C2)[nH]c2c1CCCC2)NC C1(N(C(c2cn(-c3cccnc3)nn2)C(=O)NCC(=C)C)C)CCC(C)CC1 c1(NC2N(C(C3CCCN(C(CC(=O)O)=O)C3)=O)CCC2)ccc2c(c1)OCO2 c1(C(=O)NCC23N(C(c4nc(C)sc4)=O)CC(C2)C3)cc2ccc(F)cc2s1 O=C(CCNC(c1ccccc1Br)=O)NNC(=O)Cc1ccccc1 c12nc(C)c(o1)C(=O)NC2.C1(C)(NC(CC2CC(CC)C2)=O)CCC(C)C1 N1(C(C(CCSC)O)=O)CCC(N(C(=O)CCc2ccsc2)C)C2(CC2)C1 CCCCCC(O)CC(=O)NC1CC(NC(c2ncccc2OC)=O)C1 O=C1CC(C(=O)NC(C(F)(F)F)C2CCCOC2)c2cccnc2N1 N1(C(C(C(C)(C)C)CO)=O)CC2(C1)CN(C(c1coc(S(N)(=O)=O)c1)=O)CCO2 C(CC(C)C)(C(=O)NCCCc1nc[nH]n1)NC(C(CCSC)O)=O N1(C(c2[nH]nc(OC)c2Cl)=O)CCN(C(C2CC3CCC2O3)=O)CC(O)C1 c1(C(=O)NCC(CO)NC(C(CCC)C)=O)cnc2c(c1)NCC2 N1(C(c2sc(C)c(I)c2)=O)CCC(C(=O)O)C(C(=O)O)C1 N1(c2cc(NCc3nnc(CC)s3)nc(C)n2)CCC(C2CNC(=O)C2)C1 Cc1ccc(Cl)cc1OCC(=O)N(C1CCN(C(c2c(C)nn(C)c2Cl)=O)C1)C C1(C(=O)NCCOCCCNC(c2cc(Br)ccn2)=O)COCCC1(F)F Cc1cc(F)ccc1C(O)C(=O)NCC1CC1NC(=O)CN(C)C(N)=O c1(C(=O)NCC(CNC(c2cnc(C(C)C)s2)=O)C)cnc2c(c1)CCOC2 CC(Cc1ccco1)C(=O)NCC1(CNC(=O)CCNS(C)(=O)=O)CC1 C=CCC(C(=O)N1CCC(C(=O)N(C)CCN(C)CCO)C1)C(C)C C(c1ccc2c(c1)OCO2)=CC(N1CCN(C(C2CCS(=O)CC2)=O)C2CC12)=O C1(C(=O)NC(CN(C(c2ccc(CSCCC)o2)=O)CC)C)CC(C2CC2)C1 c1(C(=O)NC2CC(CNC(CCOCCOCC)=O)C2)cc(C)c(C)c(F)c1 N1(C(c2cnn(CC)c2C)=O)CCC2CN(C(=O)CCc3ccncc3)C2C1 N1(C(c2[nH]c(=NCC)sc2)=O)CC2CCC1CN2C(=O)C=Cc1ccc(Cl)cc1 C(CC(O)C(=O)N(C)Cc1ccc(CNC(=O)C(O)c2cnc[nH]2)cc1)SC c1(CC(N2CC3(CCC3)C2)=O)n[nH]c2cc(-c3cncc(O)c3)ccc12 C1(NC(c2cnn(C(F)(F)F)c2)=O)CN(C(=O)C=CC2CCOCC2)CC12CC2 Cc1c(C(N2CCC(CNC(=O)C(C)C)C(F)(F)C2)=O)cc(Br)cc1N N1(C(CCC)=O)CCC2(CCN(C(=O)Cc3sc(SCCN(C)C)nc3C)C2)C1 C(CCCCC(=O)NC(C(=O)N(C)CC1CCCC1O)C1CC1)=CC Cc1nc(C(N2CCC(O)(CNC(C3CC(C)OC3C)=O)CC2)=O)ccc1C#N CC1CC(c2nnnn2C2CCC2)(NCCCSC(C)(C)C)C1 c1(C(=O)NCC2CCC2C(=O)NCc2cscn2)coc2ccccc12 C(=O)(CCCCCCNC(C1C(C#N)C1(C)C)=O)NC(C)C(C)(C)O c1(CSC)cncc(C(=O)NC2(C)CCN(C(c3ncccc3C3CC3)=O)C2)c1 C1(CC(N)=O)CN(C(C2(C)CCCN2C(c2ccc(CO)o2)=O)=O)CCO1 CCCCC(F)C(=O)NC(c1ccccc1)C(N1CCCC1CC(N)=O)=O C1(CCNC(CSCCC)=O)C(C)CCCN1C(=O)Cc1nc([N+](=O)[O-])n[nH]1 c1(CC(C)C)cc(C(=O)NCCCNC(C2CC(C)(C)C2)=O)no1 C1(CNC(C2CC(C)CN2C(=O)CNC=O)=O)CC(C(N)=O)=NO1 CCC(CC(F)(F)F)C(=O)NCC(CCOC)NC(c1c(C)cc(O)cc1C)=O C1(C(=O)OC)C2CCC1N(c1nnc(-c3ccc(Cl)cc3C(F)(F)F)o1)C2 CC(CN=c1ccnc(Cl)[nH]1)N(C(=O)CCC1CC1(F)F)C C#Cc1cncc(C(=O)NC2CN(C(C3CN(S(N)(=O)=O)C3)=O)CCC2O)c1 N1(C(c2c(CC)con2)=O)C2CCC1CN(C(=O)CC(C)c1ccccc1)C2 c1(C(=O)NCCCN(C(c2cnc(NC)cn2)=O)CC)cc(Cl)ccc1Br N1(C(CCOC(C)C)=O)CCC2OCCN(C(=O)C3=NOC(C)C3)C2C1 c1(NC(CCc2c(C)[nH]n(-c3cccnc3)c2=O)=O)cc2cccc(Br)c2s1 C(c1ccccn1)=CC(=O)NCC1C=CC(NC(c2c(C(C)C)ncs2)=O)C1 C1(NC(COC(C)=O)=O)CCN(C(=O)Cc2csnn2)CCC1(F)F C#Cc1cc(C(=O)N(CC)CC2CC3CC3N2C(=O)C(CC)OCC)ccc1C Cc1cc2c(cc1Br)N(C(=O)COCC1CCCOC1)CC(C)O2 CCC(CC)C(=O)NCC(C1CCN(C(c2cc(C)n(C)n2)=O)CC1)F Cc1cnc(C(=O)N(CC(C)(C)CNC(c2ccc(C(C)(C)C)cc2)=O)C)nc1 C1(CC)C(NC(=O)C(CO)NC(N)=O)CCN1C(C1(N(C)C)CC1)=O C(C(C(=O)N1CC(CNC(c2cc(OC)no2)=O)C(C)C1)C(C)(C)C)OCC=C C1(C(N2CCC(NC(C3(CC(=O)OCC)CC3)=O)C2)=O)CCC2(CC1)CC(O)C2 Cc1csc2cc(C(=O)NCCC(C)(C)CNC(=O)CC3C=CCC3)[nH]c12 c1(C2C(C(=O)OCC)C23CC3(F)F)ccc(C#N)c(C)n1 C(=O)(C(CCC1CCC1)NC(=O)COC1CCOCC1)NC(C(C)C)C1CC1 CCCC(C(=O)N(C)OCC(F)(F)F)NC(C1CCOCC1(C)C)=O C12(NC(C(CSC)C)=O)CC(C)(C1)OC21CCN(C(=O)CCC[N+](=O)[O-])CC1 N1(C(C2C(CCC)CCC2)=O)CCCC(N(C)Cc2cccnc2C)C1 c1(C(=O)NCCC(=O)OCC)c(C)[nH]c(C(=O)Nc2ncccc2F)c1C C1(NC(c2n(C)ncc2)=O)CC(CNC(c2n[nH]cc2F)=O)C12CCC2 N1(C(=O)C=Cc2ccc[nH]2)CCCC2(CCN(C(C3CC4C(C3)C4(F)F)=O)C2)C1 CCCC(C(=O)NC1CCCCC1CNC(=O)C=C1CCCCC1)NC(N)=O N1(C(CCSCCC)=O)CCC2C(C(=O)NCC(C)C)C2C1.C(COC)S N1(C(c2n(CC)c(O)nc2)=O)CC(C2CC2C(=O)NCC2(C)CC2(F)F)C1 C(=O)(C1=NOC(C(C)(C)C)C1)NCC(CNC(C1(CO)CC1)=O)OC c1(C(N2C3CC(CNC(CC4N(C)CCC4)=O)C2CC3)=O)ncn2ccccc12 Cc1c(NC(C2CCCN2C(=O)CNCc2cc(Br)ncc2Br)=O)cccc1I N1(C(=O)OC(C)(C)C)CCCC2(NCc3cocc3Br)CCCC12 C1(CC(N2CC(NC(c3c(-c4cn(C)nc4)c[nH]c3)=O)C2)=O)CC2C=CC1C2 c1(C(N(CCCNC(c2c(C)coc2C)=O)CC)=O)cc2c(O)cccc2n1C c1(NC(CC)=O)ccc(NC(=O)CCCCC2CCNCC2)cc1Cl C(C(=O)NCc1ccc(F)cc1)(C1=CCCCCCC1)N1C(CC)CCC1 C1(C(=O)NCc2c(C(N(C)Cc3cc(C)on3)=O)con2)CCCSC1C Cc1ncc(C)c(N2CC(C(N)=O)(CNC(=O)C(C)(C)C)C2)n1 c1(NC(C2(N(C(C(C)SCC)=O)C)CC2)=O)cncc(Cl)c1 N1(C(c2c(C)coc2)=O)CCC(C2(NC(C3CCCC3O)=O)CC2)C1 C(=O)(C1=CC2C=CC1C2)NCC(CC)(C)NC(C1CC2CCCCN2C1)=O C1(C(=O)NC(CC)C(C)CN(C)C)CCc2ncn(C)c2C1 N#Cc1ccc(N2CC3C(NC(C4CCC(F)CC4)=O)C3C2)nc1 Cc1nc(O)c2c(n1)CCN(C(C1C=CCN1C(c1cc(Br)ccn1)=O)=O)C2 c1(OC)cc(C(=O)NCC2CCN(C(=O)CC3CC(SC)C3)C2)ncn1 C1(C(=O)NCCC(C=C)C)COCCN(C(C2(C)CCN(C)C2)=O)C1 N1(C(C2N(C(C)C)CCC2)=O)CCC(C(=O)N(CCO)CCO)C1C(C)C C1(CCNC(c2ccc(CCC)[nH]2)=O)C(C)CCCN1C(=O)CC1CC1 C(=O)(C1=NNC(=O)C1)NCC1(OC)CCN(C(=O)CN(C2CCSC2)C)C1 CCC(CC(=O)NCC#CCNC(c1ccc(OC)cc1)=O)c1ccc(C)cc1 c1(C(N2CCC(CN(C(c3cc(C)[nH]n3)=O)C)C2)=O)ncnc2c1CCC2 C1(CCNC(c2nc(C(C)(F)F)sc2)=O)CN(C(c2c[nH]ccc2=O)=O)CCO1 Nc1c(C(=O)NC2(CNC(c3cccc(Br)c3)=O)CC2)cc(F)cc1F c1(C(=O)NCCOCC)nc(CNC(c2cc(CC)[nH]n2)=O)oc1C C1(NC(CCn2c(C)ncc2)=O)CN(C(C2CCCC3(CC3)C2)=O)CC2(CC2)C1 c1(C(=O)NCCN(CC(C)O)C(C2(C)CC2(F)F)=O)ccccn1 CC1(C)CCC(CNC(=O)CC2CC(F)C2)N(C(=O)CCn2cnccc2=O)C1 CC1(c2nc(-c3ncccc3Cl)no2)Cc2ccc(Br)cc2C(=O)O1 N1(C(CCSC)=O)CC(F)CC1CNC(c1cc(C#N)cs1)=O c1(C(=O)NCCN(C(C2C(C)(C)C2(F)F)=O)CC2CC2)cncc2[nH]ccc12 c1(C(N2CC(CC)N(C(C3CC(O)CN3C)=O)CC2)=O)ccc(F)c2ccoc12 C1(NC(CCc2ccc(CC)cc2)=O)CN(C(=O)CCC#N)CCC1CO C(c1cccc(F)c1)=CC(=O)NCCC(C)CCNC(=O)COC(F)(F)F c1(C(N(C(C)CF)C)=O)cc(C(F)(F)F)ncc1I c1(CC(N2CCN(C3CN(C(C(CC)=CC)=O)C3)CC2)=O)ccc(F)c(Cl)c1F C1(NC(C(C)Cn2cccn2)=O)CN(C(c2cc(Cl)cn2C)=O)CC1C(F)(F)F C1(OC)CCC(N(CCC(C)(C)c2ccccc2)C)C1 C#Cc1ccccc1CC(=O)NC1(C2CCCN2C(=O)C(C)SC)CC1 C(=O)(C1CCSc2ccccc21)N1C(CNC(c2c(F)ccc(C)c2)=O)CC1 Cc1nc(O)ccc1C(=O)NCCN(C(=O)C(F)C1CCCC1)C(C)C N1(C(C2(CCNC(CC(=O)NCC#C)=O)CCC2)=O)CCC(C2CCOC2)C1 C(=O)(CCCNC(N)=O)NC1C(NC(C=C(COC)C)=O)CC1 C(=O)(C(c1cccs1)NC(=O)CC1CCOC1)NCCSCC#C C1(C)(C(=O)NCC23C(CN(C(c4cnc(OC)nc4)=O)C2)C3)CCC(F)(F)C1 c1(C(=O)NC2CCCC(NC(c3c(C)n(C)cn3)=O)C2)ccc(C(F)F)c(F)c1 N1(C(CN(C)C)=O)CC2CC(C1)CN(C(=O)Cc1cccc3ccccc13)C2 C(=O)(C(C)(C)C(O)C(C)C)N1C2CN(C(c3cc(C(C)C)on3)=O)CC1CC2 c1(C2c3nnnn3CCN2)cc(Cl)cnc1O.N1(CC2C(C)(C)C2)CCOCC1 c1(C(=O)NC2CC(N(C(c3nc(OCC)oc3)=O)C)C2)nn(C)cc1COC c1(C(=O)OC)ccc(S(=O)(=O)N2CCC3(CN(Cc4cnn(C)c4C)C3)C2)n1C C(=O)(CCCCC(N)=O)NC(C(=O)NCC1CC(CC)C1)CO N1(C(C(C)OCC)=O)CCCC(C(=O)N(CC(C)C#N)CCOC)CC1 CC1(C)CCC(C(N2CC3C(NC(=O)Cc4ccn(CC(F)(F)F)n4)C3C2)=O)O1 C1(CNC(Cc2c(C)nc(C)s2)=O)C(O)C(O)CN1C(=O)CCc1ccn(C)n1 C1(C(=O)NC2CCC(NC(c3cc[nH]c3C3CCC3)=O)C2)(COC)CCOC1 C1(C(=O)NCCC2(CNC(C3(C(=O)NC)CC3)=O)CC2)CCn2nnnc2C1 Cc1cc2[nH]c(C(=O)NC(CNC(c3ccc(S(C)=O)cc3)=O)C3CC3)cc2s1 C#Cc1cn(C)nc1C(=O)NC(CC(F)F)C(=O)NC1CCCC1OC C1(C(=O)NCCC(=O)NCCC(=O)OC)C2CCC(C2)C1N Cc1csc2cc(C(N3CCN(C(C4(C)COCCO4)=O)CCC3C)=O)[nH]c12 c1(C(=O)NC(CCNC(CC(CCC)C)=O)C)cc2cnn(C(C)C)c2nc1C c1(OC)ccc(Cn2cc(-c3nccc(C)n3)nn2)cc1OCC1CCCO1 Cc1c(C(=O)NCC(O)CNC(=O)Cc2ccc(F)cn2)sc2cccc(F)c12 CCC(CC(=O)NC1CCC(O)CN(C(c2nc(OC)c(C)s2)=O)C1)C(C)(C)C C(=O)(C(C)(C)C(C)(F)F)NCC(C(=O)NC(c1nn[nH]n1)CC)N(C)C N1(C(Cc2c(C)n(C)cn2)=O)C(C)CCC1(C)C.C1(C=O)C2CC3C(C2)C13 N1(C(C2(CC#C)CCCC2)=O)CCC(NC(c2cc(CO)ccn2)=O)C(O)C1 c1(C(N2CCC(N(C(CCOCC)=O)CC)C2)=O)cc(C)ccc1NC(C)(C)C N1(C(C(C)OC2CCCC2)=O)CC2(C1)CN(C(c1cccc(=S)n1O)=O)CCO2 N1(C(CCN(C(C(OC)OC)=O)CCO)=O)CC(CO)(CF)C1 C1(C(=O)NCCC2CCN(C(=O)CCSC(F)(F)F)C2)CC12CC(F)(F)C2 c1(CNC(C(CC#C)O)=O)ccc2c(c1)CN(C(c1cnoc1C)=O)C2 c1(C(=O)NC(C)CNC(=O)C=CC2CCCCC2)cc2sc(Br)cc2[nH]1 c1(N(C(C(C=C)O)=O)C2CCNCC2)ncnc2cccc(OC)c12 c1(C(N(CCC(C)NC(c2c(C)cncc2)=O)C)=O)n[nH]c2c1CC(C)CC2 c1(C(=O)NCCCC2OCCN(C(C3(C)CC3)=O)C2)n[nH]c2c1CCCC2 C12(C(=O)NCC(C)(C)CNC(=O)CC3CCNC3=O)CCC(CC1)C2(C)C O=S1(=O)c2ccc(nc2)N1.C1(NCCCOCC(F)(F)F)C=CCCC1 C#CCC(C)(C)C(=O)NCC1CC1NC(c1cc(Cl)n(C)n1)=O C1(C(=O)NCC(CNC(c2cc(C)c(=O)n(C)c2)=O)C)CCc2n[nH]cc2C1C C1(CC(=O)NCC(C)OCC=C)CN(C(c2ccn(C)c2CC)=O)CCO1 C(=O)(C1=CC2C=CC(C1)C2)N1CCOCC(NC(C(C)OC)=O)C1 C=C(Br)CN=c1nc(N2CCc3nn(C)c(=O)cc3C2)c2c([nH]1)CCC2 C(N=c1[nH]c2c(c(=NCc3n[nH]c(=N)o3)[nH]1)COCC2)c1c(COC)ocn1 C1(NC(=O)C=C2CCSCC2)CCN(C(=O)C=CC2CCOCC2)CC1F N1(C(C(CC(=C)C)C)=O)CC(CNC(=O)CC=C(C)C)OC2CCCC12 N1(C(C2CN(CC)C(=O)C2)=O)CCCC(C)(NC(C2CCOCC2)=O)C1 N1(C(c2c(C)nc[nH]2)=O)CC(C)CCC1CNC(=O)CCCc1ccc(Cl)cc1 CC(C)(O)C#CC(=O)NC(CC1CCC1)C(=O)NC1CC2CC2C1 C(c1ccc(OCC(N2CC=CC2CNC(=O)C(C)N(C)C)=O)c(OC)c1)=CC C(=O)(CCS(=O)(=O)C1CCCC1)N1CCCCC(CNC(C(C)(C)C)=O)C1 CC(C)CC(C(=O)N(CC(C)NC(C12CCC(CO)(CC1)C2)=O)C)C(N)=O Cc1[nH]c(C(C)(C)C)cc1C(=O)NCC1CCCN(C(=O)CC2(O)CCOC2)C1 N1(C(c2cccc(CCC)c2)=O)CC2CC1CN2C(c1cn(C)ccc1=O)=O C12(C(C)C)CCC(N=c3[nH]c(N4CCCCC4C)nc4cccnc34)C1C2 C1(C(C)NC(C2CSCN2C(=O)C(C)(C)C)=O)CN(C(c2cnsc2)=O)CCO1 c1(C(=O)NCC2CC(NC(C=COCC)=O)C2)cc(OC)cc(C)c1N C(=O)(CC(C)(C)C(=O)NCC(C)(CNC(C1CC(C)(C)CO1)=O)OC)OCC c1(C(C)OC)nc(C)c(C(=O)NCCCCCCNC(=O)C(C)OC(C)(C)C)s1 N1(c2nnc(CC)s2)C2CCC1CC(NC(=O)CC1CC1(C)C)C2 CCCCCC(=O)NC(c1ccc(CNC(C2CCCN2C=O)=O)cc1)C c1(CC(=O)NCCOCCNC(c2cncc(NC)c2)=O)c(F)cccc1F N1(C(C(C(C)C)n2cccc2)=O)CCC2(CCN(C(=O)C(F)(F)C(F)F)CC2)C1 N1(CC#C)CCN(C(=O)CC(C)CNC(=O)C(C2CCOCC2)C)CC1=O C1(CC(=O)NCC(N2CCN(C(C3(C)CC(C)C3)=O)CC2)C)CCCC(C)(C)C1 CC1CCn2cc(CNC(=O)NCC34CCC(CF)(C3)OC4)nc2C1 c1(C(N(C)CC2CCCN2C(=O)C(F)C2CCOC2)=O)cccc2c1CNC2=O N1(C(C23N(C(=O)Cn4cccc4)CC(C)(C2)C3)=O)CCCC(C2CC2)CC1 c12ccc(nc1)Nc1cccc(c1)OCCn1c(nnn1)C2NC.C1(OC)CC1 c1(NC(c2n(CCC)nnn2)C2(CC)CCCC2)ccc(CCC(=O)OC)cc1 C(CC(=O)NOCc1ccc(N2CCNC(=O)C2)cc1)OC c1(C(=O)NC2CC(C(NOCCCC=C)=O)C2)c(C)nsc1N c1(C(=O)NC2CC(NC(=O)C=CCF)C23CCC3)ccc2nc(S)oc2c1 C1(C)(NC(C2CCN(C(CC)=O)C2)=O)CCN(C(c2cc(OC)cs2)=O)C1 C(CCC1CCC1)(C(=O)N1CC(N2CC(O)C2)C1)NC(=O)CCc1ccncc1 C1(CNC(=O)CCN(C(C2C=CCC2)=O)C2CC2)CCCCS1 CC(C)(O)C#CC(=O)NCC1CCCC(NC(=O)CCc2ccoc2)C1 N1(C(=O)OC(C)(C)C)CCC(n2nnnc2C(F)(F)F)CC1.N12CCC1COC2=O C1(C(=O)NC2C(CNC(C3C(CC(C)(C)C)C3)=O)CCC2)CCC(C)(C)CO1 C1(NC(c2conc2C2CCCC2)=O)CCC12CCC2 C1(C(=O)NCCN(CCC)C(C2CCCC(=O)O2)=O)CN(CP(C)(C)=O)C1 C(=O)(C(CC(C)(C)C)OC)N1C(C(=O)NC(C#C)C(C)(C)C)C(CC)CC1 C(=O)(C(C)(C)CS(C)(=O)=O)NC1CCC(NC(C(CCC)CC)=O)CC1 c1(C(=O)NC2C(NC(c3cc(C(F)F)[nH]n3)=O)CC2)cc(C(F)(F)F)ccc1F C1(C(=O)NCCOC(C)C)CC2CC2N1Cc1ccc(Br)s1 c1(SC)ccc(CCC(=O)N(CCCNC(C23COC(C2)C3)=O)C)cc1 N1(CCC)CCCC1C(=O)NCCCC1(CNC(C2COC(=O)O2)=O)CCCC1 CC(C)C(CCC(=O)NCC(C)(C)CC(C)O)NC(c1ccsc1Cl)=O CC1(C)CN(C(c2nccnc2C(N)=O)=O)CCC1NC(=O)CN1CC=CC1 C1(NC(CC=CC)=O)CCC(C)N(C(c2cccc(N(C)C)n2)=O)C1 N1(C(c2c(C)non2)=O)CC(C(=O)N(CC2=CCCOC2)C)C(C(C)C)C1 CCC(C)C(O)C(C)C(=O)NC1CCCCN(C(=O)C(c2ccc(C)o2)C)C1 N1(CC)CCC(NC(N2CC(N(C)C)(COC)C2)=O)CC1 C=CC1(C(c2nnnn2-c2cnsc2)NC2CCC(=O)NC2=O)CCOCC1 C1(C(C)=O)CCCN(C(=O)CCC2(NCc3sccc3C)CCC2)C1 c1(NC(=O)NC2(CC=C)CCCC2)cn(C)nc1CC N1(C(C(C)c2ccsc2)=O)CC2N(C(C3C=CCC3)=O)CCC2(C)C1 c1(-c2c(C3CC3)occ2)ccc2[nH]cc(CC(=O)NCC3(C)CCOCC3)c2c1 c1(C(=O)NC2C(CNC(c3cc(C)c(C)nc3)=O)C2)ccnc2ccc(F)cc12 O=C(C1NCCn2nccc21)NC1CC(N2CCCC2)C1 Cc1cc(NCC2CCN(C(c3cc(C4CC4)on3)=O)C2)c(C#N)cc1[N+](=O)[O-] C1(OC)CN(C(c2ncc[nH]c2=O)=O)CC1NC(c1c(Cl)nsc1Cl)=O CCS(=O)(=O)CCCN=c1nc(N2CCOCC2)[nH]c(=NCC(Cl)(Cl)Cl)[nH]1 C(C(=O)N=c1ccn(C(C)(C)C)[nH]1)(c1cccnc1)NC(C(CCCC#C)C)=O C1(NC(CNC(CCC)=O)=O)CC2CC(C1)N(C(c1nnn(C)n1)=O)C2 CC(C)CC(Cc1ccccc1)C(=O)N1CCN(C(c2ccc(CO)s2)=O)CC1 Cc1nc(CN2CCC(CNC(=O)CC(F)(F)F)CC2)c(C)n1C Cc1cnc(C(N2CCCC3(NC(=O)CSC4CC4)CC23)=O)cc1Br C1(C(=O)NCC2(C)CCOCC2)CCN(Cc2cnc(Cl)s2)CC1O N1(C(Cc2c(C)n[nH]c2)=O)CCCN(C(=O)CC(F)(F)Cl)CC1C c1(COC(C2(c3nn[nH]n3)CCC(NC(COCC)=O)C2)=O)cc(Cl)cnc1C C(=O)(CCN=c1[nH]ccs1)N1CC(COC)(CNC(c2ccsc2SC)=O)C1 N1(C(C(C)OCCOCC)=O)CCC2(CCCC2CNC(=O)CC2CCC2)CC1 N1(C(C(CC)COC)=O)C2CCC1C(NC(=O)Cc1cc(F)ccc1Cl)C2 c1(C(=O)NC(CNC(C(CC)(C)COC)=O)(C)C(C)C)cc2ccncc2[nH]1 C1(NC(c2c(C)ccs2)=O)COCCC1NC(=O)C(C)Cc1ccncc1 Cc1cc(F)c(C(N2CCN(C3CCOCC3)CC2)=O)cc1-c1cccnc1C N1(C(C(COC)N(C)C)=O)CCCC(CO)(NC(C2CC(NS(C)(=O)=O)C2)=O)C1 c1(CC)ccc(C(=O)NC2CC(C)(NC(c3nc(CC)ncc3Cl)=O)C2)cc1N C1(CC)CN(C(c2ccc(COCOCC(C)C)cc2)=O)CC(CC)O1 Cc1cc(=NCCn2cnnc2)[nH]c(NC(c2cccnc2)C)n1 Cc1csc(=NCC(=O)N2CCCC(CNC(c3ccc(Cl)cc3F)=O)CC2)[nH]1 CC(C)C(C#N)C(=O)N(C(C)CCNC(C1CCC(C(F)(F)F)CC1)=O)C c1(C(=O)NCCC2CC(NC(C3C(C)(CC)C3)=O)C2)scnc1C n1(CC)nc(C)c(C(=O)NC2CC(O)(CNC(=O)C(=O)NC(C)C)C2)c1Cl c1(C(N2CC(C(C)NC(c3ccoc3C3CC3)=O)C2)=O)cn(C)c2ccccc12 CCCCC(C(=O)NCCC1CCOC(C)C1)NC(=O)CNC(C1CC1C)=O c1(C(N(CC(Cc2ccccc2)NC(C(C)CF)=O)C)=O)ccc(S(N)(=O)=O)s1 N1(C(C2(F)CN(C(C(C)n3ccnc3)=O)C2)=O)C(C)CCC1C n1(CC(N2CCC(CNC(c3c(C)oc(C#N)c3)=O)C2)=O)nc2c(n1)CCCC2 Cc1cc(C(=O)N(CCCNC(C2(C(F)F)CCCC2)=O)C2CC2)nn1C C=CCC(CC(=O)NCC1C(CO)C1(F)F)NC(=O)CCC1CC(C)C1 c1(C(=O)NCC(CC)N(C)C(c2cn(C)cn2)=O)cccc2cnn(C)c12 C(CN=c1cc(C(F)F)nc[nH]1)NC(c1c(Cl)cncc1Cl)=O c1(C(N2CCC(CN(C(=O)CCC(F)(F)F)C)C2)=O)ccc(F)c(F)c1F N1(C(c2ccc(C)cc2)=O)CCN(C(=O)CC2CC(C3CC3)=NO2)C(CCO)C1 C1(CNC(C(C)CN(C)C)=O)CN(C(=O)Cc2nncn2C)C2COCC2O1 c1(CNC(C2CCN(CC(C(C)(C)C)O)CC2)=O)cccc(F)c1F c1(NC(=O)N2CCCC2)ccnn1C1CCCC1.c1(SC2CCOC2)ccccc1 CC(C(C(=O)NCCC1(C)CC1)N(C)CC1CC1)C1CCCOC1 n1(CCC(=O)NCCCNC(CN(C2CCSC2)C)=O)sc2ccccc2c1=O c1(OC)cc(C(N2CCC(C(C)CNC(=O)CC(C)C(C)C)CC2)=O)ccc1Cl c1(C(=O)NC2CCCC(NC(C34CCN(CC3)C4)=O)C2)csc2nnsc12 Cc1ccc(F)cc1C(N1C(CNC(=O)Cc2ccccc2F)CC2CC12)=O c1(CC(N2CCC(NC(C(C)(C)SC)=O)C(F)C2)=O)ccc2c(c1)COCC2 c1(CN(C(=O)NCC(C(C)OC)(C)C)C2CC2)cccc(C#N)c1 C(=O)(CC(C)(C)CC(C)=O)N1C(CCNC(C=C(C)C2CC2)=O)CSCC1 c1(C(=O)NCC(C)CN(C(=O)Cc2cnnn2C)C)cccc(C#CCO)c1 N1(C(C(CCSC)O)=O)CCCC(NC(c2ccc(N)cc2Cl)=O)CC1 C(CCS(=O)(=O)c1cccc(C)c1)CCN(C(C(COC)C)=O)C C1(C(=O)NC2(CCCC)CC2)CC2CCN(C(C3CCC=CO3)=O)CC12 N#Cc1c[nH]c(OCC2N(C(CC3CN(C(=O)O)C3)=O)CC2)c1 N1(C(Cc2c(C)scc2)=O)CCC(C)C(NC(c2c[nH]nc2-c2ccoc2)=O)C1 C1(NC(C2(C#C)CC2)=O)CCC(C)N(C(c2scnc2CC)=O)C1 N1(C(CC)=O)CSCC1C(=O)N(C1CCN(C(C2(Cl)CC2)=O)C1)CCO c1(NC(C2CCCC(NCc3cc(OC)ncc3)C2)=O)cnc(Cl)cc1OC CC1CCN(C(=O)CSc2ccc(F)c(F)c2)CCC1(F)F C(C(C)(COC)C(=O)NC1CCC(CNC(=O)C(F)F)C1)OC C1(C(=O)NC(CC)CCOC)(CC)CCN(C(=O)Cc2cc(C)on2)C1 C1(N(C(CCN(CCCCC)C)=O)C)CCN(C(C23CC(F)(C2)C3)=O)C1 c1(OC)ccc2c(c1)C1(CC1)CN(S(=O)(=O)c1ccc([N+](=O)[O-])c(Br)c1)C2 C1(C(=O)NC(c2c(C)nn(C)c2)C)CCN(C(=O)CCC(C)C)C(C)(C)C1 C12CCN(CC1)CC(=O)NCC2.C(C(F)(F)F)N(C1CCCC1)C Cc1cnncc1C(N1CCCCC1C(C)NC(=O)CSCc1cccs1)=O C1(CCC)CN(C(=O)C(C)N=[N+]=[N-])CC1NC(c1cc(C)sc1C)=O c1(OC)ccnc(C(=O)NC2CC(NC(c3ncoc3C3CCCCC3)=O)C2)c1 c1(C(=O)NC2CCN(C(c3n(C)ccc3)=O)CC2O)cnc2sccn2c1=O N1(C(C2CCN(C)CC2)=O)CCC2CN(CC3CCC3)CC2CC1 C1(CN(C(=O)CCN2CCCCCC2)C)COCCN1C(c1cc(C#N)on1)=O c1(C(N(CCNC(C2CCO2)=O)CC)=O)cc(S(N)(=O)=O)cc([N+](=O)[O-])c1C N1(C(c2ccc(OC)c(F)c2)=O)C2CCC1CN(C(C1CCOC1C)=O)C2 N1(C(=O)NCCC)CCC12CN(C(c1c(C(=O)OC(C)(C)C)cccc1F)=O)C2 c1(C2(C(=O)NC3C(OC)CN(C(=O)CC4(C)CCC4)C3)CC2)ccc(C#N)cc1 c12ccc(cc1)CNC2=O.c1(C2(COC(=O)NCC)CC2)ccc(F)cc1 N1(C(CC(C=C)(C)C)=O)CCC2CN(C(=O)C(C(C)C)NC(=O)OC)C2C1 Cc1nc(N2CCSCC2CCNC(c2sccc2C(F)F)=O)cc(C#N)n1 C1(C(N(C(C)COC)CC=C)=O)CCN(C(=O)c2cccn2C)O1 c1(OCC)oc(C)nc1C(=O)NC(C)CC(C)NC(=O)C(c1c(C)n[nH]c1C)C C1(NC(=O)Cn2cc(CN3CCCC3)nn2)CCC(c2ncc[nH]2)CC1 C1(CC)(CN(c2nccs2)CC(C)C)CCNC1 N(C1CN(C(=O)CCSC2CCCC2)Cc2ccccc21)C(C(CC=CC)C)=O C(=O)(C(C)(C)CC(C)C)NCC(CC)NC(=O)C(N1CCCC1)C1CC1 C1(NC(c2ccon2)=O)CCCC12CN(C(c1cccnc1C1CC1)=O)C2 c1(-n2cc(CN(C(C3C(C(C)C)CCC3)=O)C)nn2)ccc2c(c1)oc(=O)n2C C1(CNC(C(=O)N(CC(c2ccccc2)CC)CC)=O)CCC(=O)N1C N1(C(C(C=C)c2ccccc2)=O)CC2C(CNC(=O)CSS(C)(=O)=O)C2C1 c1(C(C)C)nc(NC(C)(CNC(=O)C2=CC(C)(C)C2)Cn2cccn2)cc(Cl)n1 c1(OC)cc(NC(=O)C(CC(N)=O)NC(c2cnc(O)o2)=O)ccc1C C1(NC(CC2(C=C)CN(C(C3CCSC3)=O)C2)=O)C=CC(C)(C)CC1 Cc1c(C(N2CCC(CN(C(=O)C3=NOC(C)(C)C3)C)C2)=O)cc(O)cc1N C(CCC(F)(F)F)(C(=O)OCC1(C)CCOC12CC2(F)F)OC CCC(C)C(O)C(=O)NCc1cccc(CNC(c2cnc(C(C)C)nc2)=O)c1 Cc1cc(F)c(NC(=O)CC(C(C)C)NC(c2cc(C(C)C)on2)=O)cc1F Cc1c(-c2cnc(NC(c3ccnc(F)c3)=O)s2)cccc1F C1(NC(C(C)OCC)=O)CCCCCC1C(=O)NCC(C)(C)SC C1(C)(C(=O)NCC(C)NC(C2CC=CCC2)=O)CCC(F)(F)C1 Cc1nc(C)c(C(C)NC(=O)CCN(C(c2ncccc2C)=O)CC2CC2)[nH]1 C(=O)(C1CCCc2nn[nH]c21)NCCC(CNC(C(C)SC)=O)(C)C N1(C(C=CCOCCOC)=O)CC2(CCCN(C(c3cnc(C4CC4)[nH]3)=O)C2)C1 c1(C(=O)NC(C2CCCC2)CNC(C(C)NC(N)=O)=O)ccc(F)c2occc12 C1(NC(CC2CC(CC)OCC2)=O)CCN(CC2CCCCO2)C(C)C1 N1(C(C(C)C#N)=O)CCC(C)(C)C(NC(c2cccc(Br)c2F)=O)C1 C(=O)(C1CCCc2c[nH]nc21)N1C(CCNC(C(C)C)=O)CSCC1 n1(CC)ccc(C(=O)NC2CCC2NC(=O)C(C)Oc2ccc(OC)cc2)c1C CC1CN(C(C2CCCN2C(c2cc(Cl)cc(Cl)c2)=O)=O)c2ccc(F)cc2O1 c1(C(=O)NCCC(C(=O)OC)C)c(-n2cc(C(C)(C)SC)nn2)cccc1F C(CC(F)(F)F)NC(CN(C)C1CC1)=O.C1CCC1C(=O)NCC1(N(C)C)CC1 c1(CN(C(=O)NCC2OCCN(C)C2c2ccccc2)C)noc2c1CCCC2 c1(NC(c2ccc(C(N3CC(C(N)=O)(OC)C3)=O)o2)=O)cc(O)ncn1 C1(NC(CC(c2ccc(F)cc2)C)=O)CCC(Nc2cc(F)ncn2)CC1 n1(CC)nnc2c1CCN(C(C1CC(C3CCNCC3)C1)=O)C2 c1(C(=O)NC2CCCC(NC(C=CC)=O)C2)cccc2c(C)[nH]nc12 C(=O)(CCCS(C)(=O)=O)Nc1cnc(Nc2ccc(CC)cc2)nc1 N1(C(c2c(CC)noc2C)=O)CCC(CO)C(NC(=O)Cc2csc(=N)[nH]2)C1 CC1CCN(C(=O)Cc2ccc3c(c2)CC3)CCS1 C1(C)(C(=O)NC2CN(C(C3(C(C)=O)CC3)=O)CC2O)CC2CCC1O2 N1(C(=O)Cc2ccon2)CC2(C(N3CC4C=CC4C3)=O)CC1CCO2 c1(C(N2C(CNC(=O)CC34CCC(CC3)C4)CCCC2)=O)cccc2c1OCC2 CC1(CNC(=O)C=Cc2ccccn2)COCCN(C(c2ccsc2Cl)=O)C1 C1(CC(=O)N(CC(C)NC(=O)C=Cc2cc[nH]n2)C)CC(O)C12CCC2 C1(CCC(=O)NCCNC(C2(CCCC)CCCC2)=O)CCc2cnn(C)c2C1 CC1CCCCC1(CNC(c1cc(F)cnc1O)=O)NC(=O)C=Cc1cocn1 N1(C(C2CC23CCC3)C(=O)NCCCF)CCCC12CCS(=O)(=O)C2 C1(NC(Cn2ncc(C)c2)=O)CC2(C1)CC(NC(C1CCC(F)C1)=O)C2 CC1OC(C)C(C(=O)NCCCC2CCS(=O)(=O)C2)C1C CC(C)C(C(=O)NC(C)CCNC(=O)C=Cc1cocn1)n1cnnc1 c1(CNC(CSCC)=O)ccc(CNC(c2cn(C)nc2C(C)(C)C)=O)c(F)c1 Cc1cc(=O)oc(C)c1C(=O)NCCC(C(C)C)NC(c1ccsc1C(F)F)=O C1(COC)(NC(=O)COCC2CCCC2)CCN(C(=O)Cc2n[nH]c(C)n2)C1 c1(C(=O)NC(C2(CNC(c3cccc(=O)n3C)=O)CC2)C)cn2ccccc2n1 N1(C(c2cn(C(C)C)nc2)=O)CC(CNC(=O)C(C)SCC2CCCO2)CC1C C1(CCNC(=O)Cc2ccno2)COCCN1C(=O)Cc1cscn1 c1(C(=O)NC23CC(CNC(c4c(OC)c(Cl)sc4)=O)(C2)C3)cnc2ccnn2c1 c1(C(N2CC(C#N)C(NC(c3ccc(Br)c(Br)c3)=O)C2)=O)cccc2c1CCC2 Cc1cc(O)cc(=O)n1C(C)C(N1CC2CC1C2NC(C1CC1C(C)(C)C)=O)=O C12(C(=O)NCCN(C)C(c3ccc(Br)o3)=O)CCCCC1CC(F)(F)C2 N1(C(C(C)c2ccco2)=O)CCCC(CNC(c2nn(C)nc2Br)=O)CC1 CC(CCC(C)(C)C)C(=O)NCC1CN(c2nnco2)CCC1(C)C C(CCCC(=O)N(C1C=CCN(C(C2CC2COC(=O)C2CC2)=O)C1)C)OCC N1(C(c2sc(Br)nc2C)C(=O)NCCOCC)CCN(C)CC12CCCCC2 N1(C(C(C)=C2CCCC2)=O)CC(C)C(NC(c2ccc(C)c(C)n2)=O)C(C)C1 C1(C(=O)NCc2n(CCC)cnc2)C(CC)CCN1C(=O)C=Cc1ccccc1 CCC(C)C(C(=O)NC1(COC)CCC1)N(C)CC1CC(C(=O)OC)C1 CC1OC2(C)CC1(C(=O)NCC1(C(N)=O)CN(C(c3cc(C(N)=O)cs3)=O)C1)C2 C1(C2CCC2)(C(=O)NCC2C(NC(c3c(C)cc(F)cc3)=O)COC2)CC1(F)F CC1CC(F)(F)CCN1C(=O)C(CNC(c1cccs1)=O)C(C)(C)C N1(C(c2c(C)con2)=O)CCC(C(C)CNC(c2cccc(CCO)c2)=O)CC1 C(C(=O)NOCC(F)F)(c1cccc(Cl)c1)OC c1(C(N2CCCC(NC(CC(CCC)C)=O)CC2)=O)c(N)ccc(F)c1F C(CCC(=O)NOOCOC)(C(C)C)N(C(C1CCCN(CC)C1)=O)CC C1(CNC(C(c2scc(C)n2)C)=O)(NC(=O)CC2OCCC2C)CCCCC1 C1(OCCCOC)CCN(C(=NCC(C)C#N)NCC2CCCCO2)CC1 Cc1cc(=N)[nH]cc1C(N1CCC(O)(C(C)CNC(c2cnn(C)c2Cl)=O)C1)=O Cc1ccc2c(C(=O)NC3CN(C(=O)CCc4ccn(C)n4)CC3F)n[nH]c2c1 c1(C2(C(N3CC(N(C)C(C4CN(C5CCOC5)C4)=O)C3)=O)CC2)cccc(Cl)c1 C1(NC(C(C#N)C2CC2)=O)CC(CNC(=O)COC2CCCCCC2)C(O)C1 CC(O)CC(C)CN=c1[nH]c(=NCc2csc(O)n2)[nH]c2c1CCCC2 C1(O)(NC(CN(C)C)=O)C2C3CC4C5C3CC2C5C14.O1NC(=O)OCC1 N1(C(CC(=O)NCC)=O)CCN(C(C2(C(F)F)CCCCC2)=O)CC1CC(F)F N1(C(c2ncc(OC)cn2)=O)CCN(C(c2cc(NC)ccc2Cl)=O)C2CC12 C1(C(C)C)COCCN1C(=O)C=CCN(C(=O)CC1CCCC2CC12)C C=CC1CCN1C(C1(N(C(=O)C(F)C2CCC2)C)CC1)=O N1(C(C(C)(c2ccccc2)OC)=O)CCCC(N(C(=O)Cn2nnc(C)n2)C)C1 C(=O)(C1=CC2(CCOC2)C1)NCC(C)(O)CNC(c1ccc2ncsc2c1)=O C(c1ccccc1Cl)=CC(=O)NC(C)CCCCNC(C1CCCN1N=O)=O C(=O)(CCCCCCN=[N+]=[N-])N1CCC(CNC(CC(CCC)O)=O)CC1 c1(C(C(=O)NCCCSCC)N(C2CC2)Cc2cccnc2)cccc(CO)c1 c1(C(=O)NCC2OCCN(C(CCC)=O)C2)nn(C)c(C(F)(F)F)c1Cl C1(CC)CC(C)CN(C(C2(NC(=O)CC3CCSC3)CCOCC2)=O)C1 C1(NC(CCN(C)CC)=O)C(C)(C)CN(C(=O)C2=NOCC2)CC1(C)C c1(C(=O)NCC(C(C)C)Nc2cc(C(C)=O)ncn2)cc(S(C)(=O)=O)co1 c1(C(=O)NC2C(CNC(=O)CC3CC3(Cl)Cl)CC2)cc(Cl)ccn1 c1(C(N2CC(=C(CNC(C3N(C)C(=O)CC3)=O)F)C2)=O)ccc2nnn(O)c2c1 CCC(C(=O)NCC1(C(=O)N(CCCC(C)O)C)CC1)n1cncn1 c1(C(=O)NCC2(NC(c3c(Cl)cnc(C)n3)=O)CCC2)ccc2c(c1)CC(C)O2 C(=O)(CCC(CF)CF)NC1C(CC)CN(C(=O)CCc2cnc(O)[nH]2)CC1 c1(NCC2N(c3nccnc3)CC2)cc(NC2CCCCO2)ncn1 CCCCC(C(=O)NCCCCc1ncc[nH]1)NC(c1cnc(C2CC2)o1)=O c1(C(N(CCCCNC(C(CC)(C)F)=O)C)=O)cnn2c1NCCC2C(F)(F)F c1(CCC(=O)NC2CC(CNC(Cc3cn(CC)nc3)=O)C2)ccc(C)c(C)c1 Cc1cc(C=CC(=O)NCC(O)CNC(C2CC2C(F)F)=O)ccc1OC(C)C C1(C)(NC(c2ncn(C)n2)=O)CCC(NC(c2ccccc2Cl)=O)CC1 c1(C(C(=O)NC(C)CC)N(CC=C)C(C)C)cn(C)c(=O)n(C)c1=O C1(CC(=O)N(CC(C2CCCC2)O)C)CN(C(=O)CSCC(F)F)CCO1 c1(C(=O)NCC(CN(C(C2(CC#C)CCCOC2)=O)C)C)ccc(CC)nc1C C1(NC(C2(CC#C)CCC2)=O)CC2CCC1N(C(c1c(C)ccc(C)c1C)=O)C2 N1(C(C)=O)CCc2cc(C(=O)N(C3CC(NC(=O)C(C)CO)C3)CCO)ccc21 N#Cc1cc(C(=O)NC2CCC3CC23CO)cc(F)c1F N1(c2cc(C)ncn2)CCC2CC(NC(c3scnc3C(C)(C)C)=O)CCC2C1 n1(CC)cc(CCNC(C2C(SCC)C2)=O)nn1.C1(C=O)CCC(N(C)C)C1 C1(N(C(=O)CC23CC(C2)C3)C)CCN(C(C2(C(F)(F)F)CCC2)=O)CC1 C(=O)(C(CC)CCCC)NC(CC1CCN(C(CC=CC)=O)CC1)C c1(C(=O)NC(CN(C(c2ccc(OCC)cc2)=O)C)C)cncc(C)c1Cl N1(C(c2c(C)nc(C3CC3)[nH]2)=O)CC2CN(C(C3C4(CC4)C34CC4)=O)CC2(C)C1 c1(C(N(CC(C)CNC(c2cccc(F)c2)=O)C)=O)ccc2cn(C)nc2c1 CCC(O)CC(=O)NCCN(C(=O)CC(n1nc(C)cc1C)C)Cc1ccccc1 N1(C(=O)Cc2cncnc2O)CC2CCC(C1)N2C(C1CCSC1)=O C(=O)(CC(C)(C)C#N)NCC(CN(C(=O)C(F)C1CCOC1)C)(C)C C(=O)(C(CCCCN)OC)OCCCN(CC)CC N1(C(C(CC)SC)=O)CCC(O)C1C(=O)NCc1ccn(CC)n1 C1(CNC(=O)C2=CCC2)CCC2(CN(C(c3cc4ncccn4n3)=O)C2)O1 c1(C2(C(=O)NCCC3(NC(C(CCCC)O)=O)CC3)CC2)ccc([N+](=O)[O-])cc1 CC1CCCC1N=c1nc(N2CCC3(CC2)C(F)(F)C32CC2)c2cccc(F)c2[nH]1 CC1CCCCN1CCC(=O)NC1CC(C)(NC(=O)Cc2cn[nH]c2)C1 c1(OC(C)C)ccc(C(=O)NCC2(NC(=O)C=CS(C)=O)CC2)c(O)c1 S(=O)(=O)(c1ccc(N2CC(OC)CC(O)C2)c(F)c1)NCC1(COC)CC1 N#Cc1cncc(CC(=O)NC2CC2NC(c2ccccc2-n2cnnn2)=O)c1 CCC(C)C(CNC(=O)CC1CCC(NC(=O)CN(C)C(=O)OCC)C1)CO c1(SC)cc(C(=O)N(C2CC(NC(=O)C(O)Cc3ccccc3)C2)C)ccc1N CC1CN(C(C2(C3CC3)CN(C(=O)C=CC3CCOCC3)C2)=O)CCC1CO c1(-c2cn(CC3CC(CNC(C(COC)C)=O)C3)nn2)ccc(Cl)c(C)c1 CC1C(=O)CC1C(=O)N(CCCN(C)C)CCNC(=O)CC1(C(F)(F)F)CC1 c1(CC(=O)NC(CC)CN(C)C(c2ccon2)=O)ccc2c(c1)CC2 c1(OC)oc(C)nc1C(=O)NCC1CC(NC(C2CCCO2)=O)CC1O C(c1cc2ccccc2o1)=CC(=O)NCC(CNC(C1(C(=O)NC)CC1)=O)(C)OC C1(NC(c2c(CCC)n[nH]c2)=O)(CO)CCN(C(=O)CC2CC(CC)=NO2)C1 c1(COC(C2CN(C(=O)OC(C)(C)C)C3CCN2C3)=O)cc(F)c2ncccc2c1 c1(CC)ccccc1CC(=O)NC(C)CC(C)NC(c1coc(OC)n1)=O c1(NC2(CO)CCCN(C(C(COC)C)=O)C2)ccc([N+](=O)[O-])cc1C c1(C(=O)NC2CCCC2NC(=O)C(F)(F)CO)n[nH]c2c1NCCC2 CC1CN(C(=O)CC2CCCOC2)CCC1NC(=O)CCc1cncc(O)c1 c1(CN2CCN(CCOCC)CC2)cccc2cncc(F)c12 CCC1=C(C(=O)NCC2CCCN2C(c2cc3c(C)cccn3c2)=O)CCCO1 C1(C(N(C2CN(C(C3COC(C)(C)CO3)=O)C2)C)=O)COC2(CCC2)C1 c1(NCC(C)SC(F)F)nc(Cl)nc2c(-c3ccccc3)scc12 C1(C(N2CC(CN(C(=O)C(C3CCOCC3)F)C)C2)=O)C2CCCOC12 N1(C(c2cc(OC)n[nH]2)=O)CCOC2(C1)CN(C(c1ccc3nc[nH]c3c1)=O)C2 C=C(C)C(CC(=O)N1CCC(CNC(c2cnc(OC)nc2)=O)C(C)C1)OCC c1(OC)ccc(O)cc1NC(=O)CN(C(C1CCCOC1C)=O)C(C)C N1(C(=O)Cn2cnnn2)CCC2(CC1)CC(Nc1ncc3ncnc-3[nH]1)CO2 N(C(=NCC1CC1)NCC1(CO)CCCCC1)CC1(SC)CC1 C1(CC)CN(C)CCCN1C(c1cn(C)nc1C)C(=O)NCCCF c1(OC)ncccc1CC(=O)NC(C)CCNC(C1C2CCC1CC2)=O Cc1c(C(=O)NC(C)C(=O)NC(C)Cc2ccnn2C)cccc1O c1(C(N2CCC(=CCNC(C3C(C)C3)=O)CC2)=O)cc2cccnc2o1 N1(C(CC(=C=C)C)=O)CC2CCCC(CNC(=O)C(C)(C)CN(C)C)(C2)C1 CCC(CC(N1CCC(n2cc(CCC3CCOCC3)nn2)CC1)=O)(CC)CC c1(CCC(=O)N(C)CC2CCN(C(C(C)C3CCC3)=O)C2)cccnc1F n1(CC(=O)N(CCCNc2c(C(=O)OC)ccc(O)n2)C)cnc2c1CCCC2 c1(CNC(C2CCC(n3cc(Cc4ccccc4)nn3)C2)=O)c(Cl)cccc1Cl c1(C(N2CCC(N(C(CC=C)=O)C)CC2)=O)[nH]c(=N)ccc1C Cc1cc(C)c(C(=O)NCC2CC3COCC3N2C(=O)C2=C(Cl)CC2)c(C)c1 c1(COC)cc(NC2CNCC2C(F)(F)F)ccc1C Cc1ccc(C(=O)NCC2CCC(NC(=O)C=Cc3cn[nH]c3)C2)o1 NC(=O)CCCCC(=O)NC12CC(CNC(c3scnc3C3CC3)=O)(C1)C2 c1(CC(C(N2CC(F)(CNC(COCC=C)=O)C2)=O)O)ccc(Cl)cc1 CCC(CC)CC(=O)N1CCN(C(C2CCCN(C(=O)COCCF)C2)=O)CC1 c1(CC)cc(Br)ccc1C(N1CCCC1CNC(c1ccnn1C(C)C)=O)=O C(=O)(CCC1=CCCCC1)NC(CC(=O)NCC1C=CCC1)C(F)F N1(C(c2cc(C)sn2)=O)CC(NC(=O)C(C)NC(C)(C)C)C(CC(C)(C)C)C1 C1(C(=O)OC)CN(C(C2CC(F)CN2C(c2c(Cl)cncc2Cl)=O)=O)CC(=O)N1 C#CC1(O)CCN(C(C2(CNC(c3ccc(F)cn3)=O)CCC2)=O)CC1 c1(C(N2CCC(NC(CC(C=C)(C)C)=O)C(CC)C2)=O)ccc(F)c(OC)c1F C1(C(=O)NCCC2(O)CCN(C(C=C(C)C(C)(C)C)=O)C2)CC2OC1C1CC21 N1(C(c2n(C(C)C)ncc2)=O)CCC(CNC(C2(C)CCCCO2)=O)C(F)(F)C1 C(CC(CC)C(=O)NC1CCOCC1C(=O)NCc1ccc(C)s1)=CC c1(C(=O)OCC)cc2n(n1)CCN(C(C1CCCCCC1)C(=O)NC(C)CC)C2 C(=O)(C(O)CCc1ccccc1)NC(C)CNC(=O)Cn1cnc(C(F)(F)F)n1 c1(CC)cccc(C(=O)NC(Cc2cc[nH]n2)C(=O)NC2(C(=O)NC)CC2)c1 N1(C(C(C)=C(C)C)=O)CCC2(CC1)CN(C(C1CC3CCCC13)=O)CCO2 N1(C(C2(C)CC(C)C2)=O)CCN(C(C2CC(C)CC(=O)N2)=O)CC1C c1(C(=O)NCC2CCC(NC(CC=C=C)=O)C2)cnccc1C(C)(C)C N1(C(Cc2cn(CC)nn2)=O)CC(NC(c2c[nH]cc2C(C)(C)C)=O)CC(F)C1 N1(C(C(C)n2cncn2)=O)CCC2(NC(=O)CCc3ncccn3)CCCC12 c1(CNC(C2CC3CC3N2Cc2cccc(O)c2F)=O)cccc2ccccc12 C(=O)(C(CCN(C)C)NC(C1CC=CC(O)C1)=O)NC(C)Cn1cccn1 N1(C(C2(C)CC(F)(F)C2)=O)CC2(CO)CC1(C(=O)NCCc1cc[nH]n1)C2 C1(S(=O)(=O)NC(C2CCCC2)C2CCC2)(C(=O)OC)CCC1 c1(C(=O)NCC2CC2CNC(C2CC3(CC3)CO2)=O)cc(O)cc(F)c1F C#CCC(C(=O)N1CC(NC(C2CCC(C)CC2)=O)C1)C1CC1 N1(Cc2cc(OC)cc(Br)c2)CCc2[nH]nc(C(=O)NC3COC(=O)C3)c2C1 N1(C(c2cccc(SC)c2)=O)CCC2CN(C(=O)C=CCF)CCC12 n1(CCN(C(C23CSCC2C3)=O)CC)cc(CCC2CCCCO2)nn1 CCCCCCCCCCN(c1cc(NC(C)CC2CCCO2)nc(C)n1)C c1(OC(C(C)CCc2nnc(C)n2C)=O)ccc(F)c(F)c1 CC(C(=O)N(CC(O)CNC(=O)CCC1OCCO1)C)NC(=O)C1CC1 C1(NC(C=C(C)Cl)=O)CCC2(CCN(C(C3CCC3c3nc(S)n[nH]3)=O)CC2)C1 N1(C(c2ccccn2)C(=O)NCC(C)C)CCCN(c2nnc(C(C)C)o2)CC1 C1(CC)COC(C)(C)CN1CCNC(c1ccc(C)c(Cl)c1)=O c1(NC(CSCCC)=O)ccc(NC(c2ccc(O)c(C)c2)=O)cc1C c1(CC)c(C(=O)NC2(COC)CN(C(c3cc(CC(C)C)c[nH]3)=O)C2)cnn1C c1(C(N2CC3CC3(C(=O)NC3CSC3)C2)=O)ccc(Cl)cc1I C1(c2nnc(C(=O)OC)s2)CCCN(C(=O)CSc2nnc(S)s2)C1 O=[N+]([O-])c1cccc(C(c2nnnn2C2CCCCC2)NC2C=CCC2)c1 c1(C(=O)NCCN(C(CC(CCC)O)=O)C(C)C)ccc2sccc2c1 C(=O)(CCC(=O)NC1CC1NC(=O)CC1C(O)CCC1)OC Cc1cc(C(=O)NC2CC(F)CN(C(C3CCCC34CC4)=O)C2)cnc1O CCCCCC(F)C(=O)NCC1(C(=O)N(C)Cc2cccnc2)CC12CCC2 C1(NC(=O)Cn2cc(Cl)cn2)(CO)CCCN(C(=O)C(=Cc2c[nH]cn2)F)C1 N1(C(C(C)(C)N(C)C)=O)CC2CC(NC(=O)CC3CCN(CC(F)F)CC3)C2C1 N1(CCCc2cn(C)nc2)CC2CC(F)(F)CCC2(C(=O)O)C1 N1(C(CC(COC)C)=O)CC2CCC(NC(=O)CSCc3ccccn3)CC2C1 c1(OC)cc(-c2cccc(C(=O)NCCN3CCN(C)CC3)n2)ccc1[N+](=O)[O-] C(CC(=O)NC1(CO)CN(C(c2cc(=N)[nH]c(Cl)n2)=O)C1)(C(C)C)OCC c1(C(=O)NC2CCN(C(CC3(C=C)CC3)=O)CC2C(C)C)cccc2nc[nH]c12 C1(CNC(=O)CCC2CC2)CC(F)CN1C(=O)CSCc1ccccc1 N1(C(C2CC(N3CCOCC3)C2)=O)CC(NCc2cc(OC)ncn2)CC1(C)C Cn1cc(Cl)cc1CNC(=NCC1CC1)NCC1(C)CCC(=O)N1 CC(C)S(=O)(=NC(=O)c1nn(C)c(Br)c1C)C1CCNC1 c1(CC(=O)N(C(C)CN(C)C(c2cnns2)=O)C)nccn1C c1(OC)cc(OC(F)(F)F)ccc1-c1cccc(C(=O)Nc2cnns2)c1 n1(CCOC)ncc(C(=O)NCCC(O)CNC(C2(COC)CCOC2)=O)c1C C1(C(N(C2CS(=O)(=O)CC2O)C)=O)N(Cc2ccccc2)CCCC1(C)C c1(OC)ccc(C)c(C(=O)NCC(CNC(=O)C(O)C(C)(C)C)CO)n1 N1(C(C2(OC)CCOC2)=O)CCN(C(=O)CCC(C)(F)F)CC1C CC(N=c1[nH]c(=N)[nH]c(=NCC2(N(C)C)CCCOC2)[nH]1)c1nccn1C C1(C2CN(C(C3CCOC3)=O)C2)(NC(=O)C2=C(Cl)CC2)CC1 N1(C(CCN(CC)CC)=O)CCCC1(C(=O)NCc1noc(C(N)=O)n1)CC C(=O)(CC(CC)C(F)F)NCC1(C(=O)Nc2c(CNC)cccc2)CC(C)(C)C1 CC(C)(O)CCCNC(c1ccc(C(N)=O)o1)=O C1(NC(c2ccc(C(CC)C)cc2)=O)CCSC12CN(C(C1(C)CC1Br)=O)C2 c1(C(=O)NC2CC(NC(c3ccc(=O)oc3)=O)C2)cc2cccnc2nc1O CC(C)C(O)CC(=O)NCCCN1CCN(C(C2C(F)(F)C23CC3)=O)CC1 n1(CC(=O)NCn2cc(C3CCC3)nn2)nc(C2CC2)cc1C1CC1 c1(C(=O)NCc2c[nH]nc2C(N2CC(c3ncc[nH]3)C2)=O)ccc(CO)nc1 CC(C)C(O)CC(=O)NCCC1CCN(C(=O)CC(O)CN(C)C)CC1 N#Cc1cc(F)ccc1C(=O)NCC1(O)CCN(C(C2CCCO2)=O)C1 N1(C(c2cc(CNC(c3c(C)cc(C)s3)=O)on2)=O)CC(C)C(C)C1C c1(C(=O)NCC2CCC(F)(CNC(C3CC4CC4C3)=O)C2)nnc(O)cc1O Cc1cc(Br)c(C(=O)N(CC(C)O)CCNC(C2CC2C)=O)cc1Cl C1(NC(C2CC(C#C)(O)C2)=O)C2CC3C(C2)C13C(N1CC(=O)NC(C)C1)=O C1(C(N(C2CCCN(C(=O)CCC(C)CN(C)C)C2)CC)=O)CC2(C1)CC2(F)F c1(C(N(C2CCCN(C(C3C(C)C3)=O)C2)CCO)=O)ccc(S(N)(=O)=O)s1 c1(C(=O)Nc2c(C)n[nH]c2)cc2c3c(ccc2[nH]1)N(C(=O)CCCCCBr)CC3 C1(NC(C2C(C)(C)C2(F)F)=O)CCC(O)CN(C(=O)CCCSC(C)(C)C)C1 C1(C(=O)NCC2CC(C)N(C(=O)CCC(C)(C)C#N)CC2)CN(S(=O)(=O)N(C)C)C1 N1(C(CCSCC(=O)OC)=O)CCC(CNC(C23CCC(CC2)O3)=O)C1(C)C CCC(N=c1[nH]c(=NCC2CC(C)(C)C2)[nH]c2ccsc12)c1cc(C)cc(C)c1 N1(C(C2(CC)CC2)=O)CCCC(C2CCN(C(c3cnc(C)[nH]c3=N)=O)C2)C1 N1(C(Cc2n(C)cnc2)=O)CCCCC(CNC(=O)CC2CCC(F)(F)CC2)C1 N1(C(c2c(C)coc2)=O)CC(C)OC2(CCN(C(c3cncc(C)c3Cl)=O)C2)C1 C(CC)(C(=O)N1CCCC1CCC(=O)NCC(C1CC1)C1CC1)OCC N1(C(c2c(NC)nccc2)=O)CCC2(CC2C(=O)NCC(c2cnc[nH]2)C)C1 N1(C(CCOCC(C)C)=O)CCCCC12CC(NC(c1cnnn1C)=O)C2 N1(C(C(C)CC(N)=O)=O)CC2CCCC2(C(N2CCOC(C)(C)C2)=O)C1 c1(NC(CCNC(c2c(C)oc(CO)c2)=O)(C)C)cnc2ccccc2n1 Cc1nn(CC(C)C)c(C)c1CC(N1CC(N(C)C(c2ccoc2)=O)C1)=O Cc1ccc(CC(=O)NCC23CC(NC(c4ncc[nH]c4=O)=O)(C2)C3)cc1O C=CC(C)C(C)C(=O)N(CCNC(c1ccc(C)c(NC(C)=O)c1)=O)CCNC C(C(N=[N+]=[N-])C(=O)NC1(CSC)CN(C(=O)Cc2cccc(OC)c2)C1)OCC c1(NC(N(C(CCC)C2CC2)CC=C)=O)cc(C)c2n[nH]cc2c1 N12CC3COCCC3(C1)C2=O.S(=O)(=O)(c1cc(C)sc1C)N1CCN(CC)CC1 Cc1cc(C)c(CNC(C2CCOC2CNC(=O)Cc2cccnc2F)=O)cn1 N1(C(C(C)O)=O)CCC(C2(NC(c3cnc(O)c4ccsc34)=O)CC2)CC1 c1(C(N2CC(O)CC(NC(CC3CC(=C)C3)=O)C2)=O)cc2cccc(F)c2o1 C(CC(C(C)(C)C)NC(c1cnn(C(C)C)c1F)=O)N(C(CN(C)CC)=O)C c1(OC)ccc(Br)c(CC(N2CCCC(N3CCCS3(=O)=O)C2)=O)c1 CC1=CCC(NC(C2(C)CCCN2C(C23CSCC2C3)=O)=O)CC1 C1(Nc2oc(C(=O)OCC)c(C(F)(F)F)n2)CCC2C3CCC(C3)C12 c1(-c2c(OC)cccc2O)ccc2c(c1)CCN(Cc1c(F)cc(O)cc1F)C2 NC1(CO)CCN(C(=O)C(N2CCC(Cc3cccc(F)c3)CC2)=O)C1 Nc1ccc2c(c1)CN(C(C1CCC(F)(F)C1O)=O)CCO2 CCCC(CCCNC(c1cc(C)n(C2CC2)c1C)=O)NC(=O)CC(F)F C1(NC(C(C=C=C)C)=O)CC2CC(C1)N(C(=O)CSc1nncs1)C2 C(CCCC(C)NC(C1CC2CC2C1)=O)NC(Cc1c(C)non1)=O Cc1ccc(C(=O)NC(C(=O)N(C(C)C(F)F)C)C2CCCC2)cn1 C12(NC(Cc3cc(C)sc3)=O)CC3CCC(C1C2)N3C(C1CC(=O)NC1(C)C)=O C(CCC(=O)N(C1CCN(C(=O)Cc2csc(NC(=O)C(C)(C)C)n2)C1)C)OC C1(NC(CC2(C=C)CC2)=O)CCC(O)CN(C(C2CCN(C(=O)CC)C2)=O)C1 N1(C(C(CCSC)OC)=O)CCCCC2(C1)CN(C(=O)Cn1ncnn1)C2 C(CC1CC1)(CC(=O)NCC(C)CCCO)NC(c1cc(C(C)=O)[nH]n1)=O c1(-c2cccc(NC(CC)=O)c2)nc(C(N2CCC2CO)=O)n2ccccc12 N1(C(CCC(C)OCC)=O)CCC2(CC1)CC2C(N1CCn2nccc2C1)=O C#Cc1ccc(CNC(C2(C(C)NC(C3CC4CCCC4C3)=O)CC2)=O)cc1 N1(C(CC)=O)CC2(CCOCC2)CC1CNC(c1c[nH]nc1OC)=O Cc1cc(NC(C2CCN(C(=O)C(O)C3CCCC3)CCO2)=O)cc(C)c1F C(C(CC)(CC)C(=O)N(C1CCC2CC12)C)NC(c1c(CC)n[nH]c1)=O C1(NC(C2CC(C)(C)C2C(F)(F)F)=O)CC(F)CN(C(=O)Cc2cc[nH]n2)C1 N1(C(c2cc(C)oc2C)=O)CCN(C(C2CCCCCC2)=O)C2(CC2)C1 c1(C(=O)NC2C(CNC(=O)CSC3CC3)CCC2)ccc([N+](=O)[O-])s1 CCCCCC(C)CC(=O)NCC1CCCN1C(c1cc(NC)nc(Cl)c1)=O c1(NC(N2C(C3(O)CN(C(c4c(C)nsc4)=O)C3)CCC2)=O)occ2c1CCC2 Cc1cc(CC(=O)NC2CC(F)(CNC(C3COC(=O)C3)=O)C2)cc(C)c1 c1(C(=O)NCC(=O)NC(CC)CNC(=O)C(N)=O)ccc(OC)cc1 N1(C(C(c2ccc(CC(=CC(O)C(=O)O)C)c(C)c2)(C)C)=O)CC2(C)CC1CCO2 C(C1CCCN1C)=CC(N1C(C2(NC(CN(CCC#C)C)=O)CC2)CCC1)=O C(=O)(CCCc1csc(C)n1)N(CC(CC)NC(=O)CNC(c1ccoc1)=O)C C(=O)(CC1=CCCC1)N(C1CN(C(=O)COC2CC2)CC12CC2)C CN1CCC(CCn2cc(C3CCCN3C(=O)CC3COC4CC3C4)nn2)OC1=O CC1(CNC(=O)Nc2nc3c(s2)CCCCC3)CC(=O)CC(C)(C)O1 N1(C(CSc2ccc(OCC)cc2)=O)CC2(C1)CN(C(=O)C(CO)OC)CCO2 C(=O)(C(C)=Cn1ccnn1)N1CCCC(N2C(CCC)C2=O)C1.C(N)(=O)OCC N1(C(C2C(C)N(C(=O)CC3CC=CCC3)CC2)=O)CCC(C)(O)C(O)C1 C1(CNC(c2nccc(OC)c2)=O)CCN(C(C2CCCC23CC3)=O)C12CCC2 C(=O)(C1=C(C)CCC1)NCC(=C)CCNC(C1CC(C)N1C(=O)OC(C)(C)C)=O CN1CCCCC1C(=O)NCC=CCC(=O)NCCC(O)C1CC1 C1(C(=O)NC(CC)CC)(CC)CCCN(C(=O)CCCCCOC)C1 N1(C(C2(CC=C)CCCN2C(c2cc(C)oc2C)=O)=O)CCc2nn[nH]c2C1 C(C(CCO)NC(C1CCCC1NC(=O)C=CCO)=O)N(C)C N1(C(C(C)SCC)=O)CCC2C(CCCN2C(c2ccn3c(O)nnc3c2)=O)C1 c1(C(=O)NCC(C)(CNC(C2CCCC2O)=O)OC)ccccc1SC c1(NC(c2nc(COC)oc2)=O)cc(C2CCC2)ccn1.C12CC1CNC2=O N1(C(c2scnc2C)C(=O)NC(CC)(C)C)CCC(O)(c2cc[nH]n2)CC1 C1(C(N(C2CCN(C)C2=O)C)=O)CCCN(C(=O)CC2CCCN2C)CC1 C1(C2CCC(CCCC)CC2)NC(=O)N(CC)C2=C1C(=O)NC2c1ccccc1 C(=O)(C1CCCc2cncn21)N(C1CN(C(c2c(CC)nc[nH]2)=O)CC1(C)C)C c1(C(=O)NC2CCC(CNC(c3c(C)nc(N)cn3)=O)C2)cc(F)c(F)cc1F c1(CC2(C(=O)NCCOC3CN(C(CC=C=C)=O)C3)CC2)ccc(Br)cc1 c1(OC)ccnc(C(=O)NCC(C)(C(C)C)NC(=O)Cc2cn(C)nn2)c1OC CC(C)C(C(=O)N1CCCCCO1)C(C)NC(C1C2CC(=O)CC12)=O C1(CC)CCN(C(c2nocc2C)=O)C1C(N1CC[Si](C)(C)C1)=O C12(C(=O)NC3CC(c4cn(C(CC=C)CC=C)nn4)C3)CCCN(CCC1)C2 C1(C(N(CC(=O)NC(C#C)CC2CC2)C(C)C)=O)CC2CC(=O)C1O2 N1(C(c2c(C#C)c[nH]n2)=O)CCC(C2(NC(c3cc(CO)[nH]n3)=O)CC2)C1 c1(C(c2nnnn2CC)NC(CCCC=C)C2CC2)csc(S(N)(=O)=O)c1 Cc1nc2c([nH]1)C(C(=O)N1CC(C(=O)O)C3(CCC3)C1)CCC2 c1(CC(C)C)ccc(C=CC(N2CCCC(NC(C3(C)CC4CC4C3)=O)C2)=O)cc1 C1(NC(C=NOC)=O)CN(C(=O)C#CC2(C)CCCO2)C2CCCCC12 C1(CNC(C2(C#C)CC2)=O)CCCCC1NC(c1cc(-c2ccncc2)no1)=O C12(C(N3CCCCC(C(=O)NCC45CCC(CC4)OC5)C3)=O)CCN(CC1)CC2 N1(C(=O)CCNC2(CF)CC2)CCOCC1c1cccs1 C12(CNC(COCC)=O)CCC(CNC(c3ccc(C)c(C)n3)=O)(CC1)OC2 c1(C(=O)NCC(C)NC(C2CC(=O)N(C)C2)=O)cc(F)ccc1Cl CCC1=C(C(=O)NCC(C2CC2)NC(=O)CCc2csc(C)n2)SCCO1 CC(CO)CCCNC(=O)CC1(CNC(=O)C(C)(O)C2CC2)CC1 C1(C)(C(=O)NCC(CC)NC(=O)CCC2CCCN(C)C2)CC(=O)N(C)C1 c1(OC)ccc(CC(=O)NCC(C)N(C(=O)CSC(C)C)Cc2nncs2)cc1 c1(C(N(C2CCCN(C(CCOCC(C)C)=O)CC2)C)=O)ccc(Cl)c(F)c1F c1(C=O)cc2cccnc2o1.N12CCC(C1)SCCC2=O.c1(C(=O)N)cnc(O)s1 CCC(CNC(=O)CCc1cccc(C)c1)(CC)NC(=O)CC1CCCC(=O)N1 C1(NC(C2CC3(CCC3O)C2)=O)CCCCCC1C(=O)NC1COCCOC1 C1(C(=O)Nc2c(C(=O)NCc3ccc(C)s3)n[nH]c2)CCC(F)(F)C1 N1(C(c2ccc(SC)o2)=O)CCC2CCN(C(c3ccn4nnnc4c3)=O)CC12 C1(NC(CCc2ccc(CC)cc2)=O)CS(=O)(=O)CC1NC(c1nnn(C)n1)=O C(=O)(C(Cc1ccccc1)N(C)C)NC(C)CCNC(C1(C(C)(F)F)CCC1)=O c1(C(=O)NCC(CC=C)NC(c2n[nH]cc2C(C)C)=O)nn(C)c(=O)cc1C c1(CC)ccccc1N(C(=O)COC1CCN(C(=O)C=CC(F)F)C1)C C=C=C(C)CC(=O)NC1(CNC(C2CC3CC2C3)=O)CCCC1 CC1(C)CCN(C(C2CN3CCC2CC3)=O)C(C(=O)NC2CNC(=O)OC2)C1 CC1CC2(CCN(C(=O)CC3NC(=O)NC3=O)CC2)CN1C(=O)C(Cl)=CCl Cc1cnc2ccc(C(=O)N(C(C)CNC(=O)Cc3ccon3)C)cn12 C=Cn1nccc1C(=O)NCC(C1CCCC1)NC(C1CC(N=[N+]=[N-])C1)=O c1(NC(C2CCN(C(=O)C=CI)C2)C)cnc(C#N)cn1 Cc1cc(C(N2CC3CCC(C2)C3NC(c2cnc(C)[nH]2)=O)=O)c(F)c(F)c1 Cc1nc(CN2CCC(NC(=O)CCN3CCCCC3)C(O)C2)ccc1Br c1(C(N(CCCOCCN(C)C(c2cscn2)=O)C)=O)cnc(N)c([N+](=O)[O-])c1 N1(C(C(C=C)OC)=O)Cc2n[nH]cc2C1C(=O)NCCC1CC=CC1 c1(OCCNC(C2(CCNC(C3C4CCCOC34)=O)CCC2)=O)ccc(F)cc1F c1(C(=O)NCC2CN(CC(N3CCN(C(C)=O)CC3)=O)C2)cccc(F)c1N c1(CC)oc(C)cc1C(N1CC2C(NC(=O)Cc3ncc(C)s3)C2C1)=O C1(C(N(CCCCNC(c2cc(F)cs2)=O)C)=O)CC2(CC2)CN1C N1(C(=O)C=Cc2cccnc2)CCC2CN(C(C3CCC3(F)F)=O)CC12 N1(CC(c2ccc(-c3ccc(CO)cc3F)o2)=O)CCC2(CC1)OCC1CC21 C(c1cccc(O)c1)=CC(N1CCCC(CNC(C2N(C)CCC2)=O)C1)=O C1(c2n(CC=C)nnn2)(NCC2CC(F)C2)CCN(c2ccncc2)CC1 c1(NC(Cc2c(NC(C(CC(C)C)O)=O)ccc(F)c2)=O)ccc2[nH]ccc2n1 C1(CC=C)(NC(=O)C=NOC)CCCN(C(C2CCCCNC2=O)=O)C1 C(=O)(CCCCCC#N)NC(C1(CNC(c2cccnc2)=O)CC1)C C1(C(=O)NCC2N(C(C(C)=C(CC)C)=O)CC2)CC2CC1C1C2C1(F)F C(=O)(CCCCCC)NC1(CCNC(C(C)OCC=C)=O)CCC1 c1(NC(C2CC(NC(Cc3ccc(C(C)(C)C)cc3)=O)C2)=O)c(Cl)ccc(Cl)c1Cl c1(NC(C2(F)CCN(C(CN(C(C)C)C)=O)CC2)=O)c(O)ccc(F)c1F C1(C(N(C)Cc2nc(C)[nH]n2)=O)(NC(=O)C=CC(F)(F)F)CCC(C)(C)C1 c1(CC(=O)NC2C(C)CCN(C(=O)Cc3ccon3)C2)ccc2c(c1)CCCC2 C1(CC(=O)NC(C)CC(F)(F)F)N(C(=O)OC(C)(C)C)CCC1(C)C Cc1ccc2c(c1)SC(C(N1CCC(C3(NC(c4ncn(C)n4)=O)CC3)C1)=O)C2 O=S(=O)(c1cccc(=NC2CC2CC(F)(F)F)[nH]1)N1CCOC2(CCCC2)C1 C1(OCC)CC2CN(C(=O)CC3CC(C)N(C(=O)C(C)C(F)F)C3)CC12 C(CCN(C(=O)CCc1ccc(F)cc1)C)(C(C)C)NC(c1cn(CC)nc1)=O CCCC(CC)NC(C)COCC1CC1.C(COC)O CC1CC(N(C(=O)CN(C2CCC2)C(C2(O)CCOCC2)=O)C)CC(C)C1 CC1(C)CC(Cn2cc(Cc3cccc(CO)c3)nn2)CN1C(C1CC1Cl)=O Cc1cc(C#N)ccc1C(N1CCC(CF)(NC(c2cccc(CF)c2)=O)C1)=O CC1CCCCC1CC(=O)NCCCN(C(c1cccc(N(C)C)c1)=O)C1CC1 C=C(C)CC(C(=O)NC(C(=O)NCC1CCC(=C)CC1)C1CC1)OC c1(C(=O)NC(CNC(CC(C=C)C)=O)CO)cc(S(N)(=O)=O)ccc1Br C1(C(=O)OC)CC2(CC(NC(=O)NC(c3cccc(F)c3OC)C(F)(F)F)C2)C1 c1(CC(N2CC3CC3(NC(C3(C(F)F)CCCO3)=O)C2)=O)cnc(C2CC2)nc1 N1(C(c2c(CCC)n(C)nc2)=O)CCN(C(C2COCC(C)O2)=O)C2(CC2)C1 CCCCC(C)C(=O)NC(C)CNC(c1ccccc1-n1cc(Br)cn1)=O C12(NC(C(CC#C)O)=O)CCCC1(F)CN(C(c1cnc(C3OCCO3)s1)=O)C2 C1(OC)(CNC(C2CC2F)=O)CCN(C(c2oc(CO)nc2C)=O)CC1 c1(C(=O)NCC(C)(CO)NC(C2CC(CC(=O)OC)C2)=O)cc(C(C)C)oc1C CC1(C)CC(S(C)(=O)=O)CN1C(C(=O)NC1CC(F)(F)C1)c1nc[nH]n1 c1(CNC(C2(c3cn(-c4cccc(N)c4)nn3)CCOCC2)=O)ccc(F)c(Br)c1 C12(OC)CCCCC(C(=O)NC3(CNC(C4CCCS4)=O)CCOCC3)(C1)C2 c1(C(=O)NCC(C(C)C)NC(C(C=C)(C)O)=O)ccc(=O)n(CC(=O)N(C)C)c1 c1(C(N2CC=CC(NC(CN(C3CCSC3)C)=O)C2)=O)cc2c(nn1)CCCC2 C(=O)(CC(C)CC(=O)NCC1(C)CCC(NC(=O)Cc2cnc(C)o2)CC1)OC Cc1noc(CNC(=O)CC2CCCN2C(=O)CN(C2CCCC2)C)n1 C1(CNC(C2(C(=O)OCC)CCC2)=O)C(C)CCCN1C(=O)C1=CSCCO1 C1(C(N(CCN(C(c2cnc(C(C)C)[nH]2)=O)CC)CC)=O)CCCN1CC C1(NC(CCC2(C)CC2(F)F)=O)CC(NC(=O)COc2cccnc2)C12CCC2 c1(C(N2CCC(CCC(N3C(COC)CCCC3)=O)C2)=O)cccc2c[nH]nc12 N1(C(CC(C)C(C)(C)NC(C2CCCO2)=O)=O)CCC2(CNC(=O)N2)C1 C1(N(C(CC)=O)CSc2ccccn2)CCCN(C(=O)Cn2ccnc2C)CC1 C(=O)(C(F)(F)C(C)(C)O)NC1CC(C(=O)NC(c2ccccn2)C)C1 C#CCCCC(C)C(=O)NC1CC(C)(NC(=O)CCCc2ccc(O)cc2)C1 C(=O)(C(F)CC(C)(C)NC(=O)COc1ccn(C)n1)NC1CC(C)(CC)C1 C1(NC(=O)CN2CCSCC2)CN(C(=O)Cn2cnnn2)C2(CCCC2)C1 c1(OC)ccc(Cl)cc1N(C(C1CCC=CO1)C(=O)NC(c1ccccc1)C)C c1(OC)c(C(=O)NCC(CNC(=O)CS(N)(=O)=O)OC)csc1Cl c1(CC(C)C)ccc(CC(=O)NC2CC2NC(C2(C#N)CCC2)=O)cc1 c1(CC(=O)NCC(C)N(C(C2CC2(C)CCOCC)=O)CC)cc(O)n(C)n1 C1(CC)CN(C(=O)C(C)(C)F)CC1NC(C1CN(C(=O)N(C)C)C1)=O CC1CC(NC(C2CCN(C)C2C)=O)CCN1C(=O)CSCCC#N Cc1cc(C(=O)O)cc(S(=O)(=O)NC2CCOc3cccc(Cl)c32)c1Cl c1(CC(N2C(CNC(c3cnncc3O)=O)CCCC2)=O)ccc2n[nH]cc2c1 C1(NC(C(CCOC)C)=O)CC(F)(F)CC1NC(c1snnc1C(C)C)=O C1(C(N2CC3C(CNC(C4C(C(=O)OC)C4)=O)(CC3)C2)=O)C2CCC3C(C2)CC13 Cc1ccnc2c(C(N3CC(C(C)NC(=O)Cc4cc[nH]n4)C3)=O)cnn12 CC1(CNC(c2ccsc2)=O)CCN(C(C2CCCN2c2ccccc2)=O)C1 C(N=c1[nH]c(Cl)nc(C)c1Cl)C1(O)CN(C(Cn2c(C(F)F)cc(C)n2)=O)C1 c1(C(=O)NC)ccc(C(N2CCCC2CNC(=O)C=Cc2cc[nH]n2)=O)cc1F c1(C(N2CCC(C)(CNC(C3CC4OC3C3CC43)=O)C2)=O)c(F)cc(Cl)cc1F C1(S(C)(=O)=O)(C(N(CCNC(c2ccc(F)c(CO)c2)=O)CC)=O)CCCCC1 Cc1noc(N)c1C(=O)NC1CCC1NC(c1ccnnc1)=O c1(CC)noc(CCC(N2CCCC2CN(C(=O)C=CI)CC)=O)n1 C1(CNC(CSCCN(C)C)=O)(NC(C2CCCO2)=O)CCOCC1 c1(C(=O)NCC2CN(C(c3scc(OC)c3)=O)C(C)CC2)ccc(F)c(C#N)c1 C#CC(C)(C)C(=O)N(C1CC(NC(c2nccnc2C)=O)C1)C C1(COC(C(C)Sc2ccccc2)=O)CC1C1CCC1 C1(C(=O)NC2C3(CC(NC(=O)COc4ccsn4)C3)C2)CCC([N+](=O)[O-])CC1 C1(CC)CN(C(C2CN(CC(F)(F)F)C2)=O)CCC1NC(c1cc[nH]c(=N)c1)=O C1(C(=O)NCc2c(C)nccn2)CC2C=CC1N(C(c1ocnc1C(C)C)=O)C2 C#Cc1cccc(C(=O)NC2(CNC(c3cncnc3C)=O)CC2)c1F CN1CCOCC1C(=O)NC1CN(C(C2CSC2)=O)CC1CC(C)(C)C C1(CNC(C2CC(CC3CC3)C2)=O)CN(C(C2(C3CCC3)CC2)=O)C2(CCC2)C1 C(=O)(C1=CC2CCC(C1)C2)N1CC(NC(C=COCC)=O)(COC)C1 N1(CC(=O)NCC(CC(F)(F)F)NC(c2ccc(O)cn2)=O)C(=O)CCCC1=O c1(CN2CCC(CC(=O)NC3CC(CO)C(O)C3O)C2)ccc(Br)cc1[N+](=O)[O-] N1(C(C(CCC)NC(N)=O)=O)C2CCC1CN(C(C1CC1(C)CC)=O)CC2 C1(COC)(NC(=O)C2CC2)CCN(C(C2(c3cccc(C#N)c3)CC2)=O)CC1 C1(NC(CC(C)(C)SC)=O)CC2CC1CN2C(=O)Cn1cnnc1O N(C1CCc2c(C(=O)CCC)cc(F)cc21)C(C(CCC)=CCC)=O C1(OC)CCC(CC(=O)NC2CCN(C(C3CN(C4CCOC4)C3)=O)C2C)CC1 N12CCCC(C1C)OC2=O.C(CCS(=O)(=O)NCC)CC c1(C(=O)NCC2C3CN(C(CCCC)=O)CC32)ccc(=NC)[nH]c1 C(=O)(C(F)C(C)C(F)(F)F)N1CCN(C(Cc2ccc(SC)cc2)=O)C(C)C1 C1(C(=O)NC2(CNC(c3nccc(N(C)C)c3)=O)CCC2)CC2(CCCC2)CO1 C1(C(=O)NCC2(O)CCN(C(c3[nH]cc(C#N)c3)=O)C2)CCC=CCCC1 C(Cn1cccn1)(C(=O)NCc1ncon1)NC(=O)CCc1cscn1 c1(C(=O)Nc2cc(C)sc2)cccc(CNC(=O)CCc2c(C)noc2Cl)c1 C1(C(=O)NCC2(F)CN(C(CN(C)C(=O)C3CC3)=O)C2)C2CC3CC(C2)CC1C3 CCC(=O)CCC(=O)N1CC(C)CCC1C(N1CCCC(C(=O)OC)C1)=O Cc1cc(=NC(C)C2CCN(C(c3cn4cc(Cl)cnc4n3)=O)C2)[nH]c(C)n1 N1(C(c2ccc(CC)s2)=O)CCC2(CCN(C(C3CCN3C3CCCC3)=O)C2)C1 c1(NC(C)=O)nc(CNC(CC2N(C(C3CC3C3CC3)=O)CCC2)=O)cs1 N1(C(c2c(CC)n(C)nn2)=O)CC(NC(=O)C(C)OCC(C)C)CC1(CC)CC C1(CNC(c2c(C)nc(O)[nH]2)=O)CCN(C(=O)Cn2cnc(C#N)n2)CC1(F)F Cc1nc(NC(C)CC(C)NC(c2csc(S)n2)=O)c(Cl)cc1C#N N1(CC(=O)NCC2CN(C(c3ccc(C)[nH]3)=O)C2)OC(C)(C)CC1=O n1(C(C=C)C)ccc(CNC(=O)C=CC(N2CCSCC2)=O)n1 n1(CC(=O)OC)ccc(=NC(=O)CNC(=O)C(C)N=[N+]=[N-])[nH]1 N1(C(C(C)OCC=C)=O)CCC2(CC(C(=O)Nc3ccc(Br)cc3O)=NO2)C1 c1(C(=O)NCC(C)N(C(c2cccc(CC)n2)=O)CC)cccc2cncn12 N1(C(Cc2ccc(OC)cc2)=O)CC2CC(C1)CN(C(=O)Cc1cncs1)C2 C1(C)C(=O)N(CC)CC(CO)NC(=O)O1.C(C)(=O)OCC CCC(CO)C(=O)NCCN(CCOC)C(c1cc(-c2ccccc2)[nH]c1C)=O c1(C(N(CCCNC(CC(C)C(F)F)=O)C)=O)c(O)ncc2c1CCC2 CC1CN(C(c2cnn[nH]2)=O)CC1CNC(=O)C(c1cccc(Cl)c1)(F)F C(CC(C)C(=O)NC1CN(C(=O)Cc2cnns2)CC1OC)=CCC c1(CN(C(=O)OC)C)ccc(NC(=O)NCC2CC3CC3C2)cc1 O=C(C(O)C(F)F)NCCCCC1CN(C(c2ccc(C3(F)COC3)cc2)=O)C1 N1(C(CC(C(C)OC)NC(C(CC=C)OC)=O)=O)CCN2CCCC2C1 c1(N2C3CN(C(C4C(C)CCCC4)=O)CC2CC3)nc(Cl)nc2cnn(C)c12 C#CCCC(C(=O)O)NC(=O)C(C)OCc1ccccc1Br C1(N(C(=O)C(Cl)=CCl)C)CCC(NC(=O)CN2CCS(=O)CC2)CC1 c1(N(CCCNC(=O)C=CCNC(=O)C(F)CC2CCC2)C)cc(=O)n(C)cn1 c1(OC)ccc(Br)cc1C(N1CC2CC2(CNC(c2cnn[nH]2)=O)C1)=O c1(CC)ncc(C(=O)N(C)Cc2ccccc2C(C)(C)C)c(=O)[nH]1 C(C(=O)N=c1cc2n([nH]1)CC(C)OC2)Oc1c(CC)nc(C)cc1 C1(NC(=O)CCC2CCCCCC2)CN(C(=O)C=C2CCC2)CC12CCC2 CC1CCCC(C(=O)N(CC(=O)N(C2(C3CC3)CC2)C)C)CC1 N1(C(C2(COCC)CC2)=O)CCOC2(CCN(C(=O)CC(C)n3ccnc3)C2)C1 C1(C(N(C2CCN(C(c3cnn(C4CC4)c3)=O)C2)CC)=O)CC2(CCO1)CC2 C(=O)(CS(=O)(=O)C1CCCC1)N1CC(NC(C2CC(=O)N2)=O)CC2(C1)CCC2 C(CC(C(=O)NC1CN(C(N)=O)C1)NC(c1cn(CC)nn1)=O)=CC Cn1cncc1C=CC(N1CCCC(CCNC(C2CC2c2ccsc2)=O)C1)=O N1(C(Cc2c(OC)cccc2)=O)CC2CCC1CN2C(c1cc(=O)cc(Cl)[nH]1)=O C1(C(N2CC3N(C(C4C(CCOC)C4)=O)C(C3)C2)=O)CC2CCCC(C1)C2 C1(C(=O)NCC(C)=CC(=O)NC(c2ccccc2)CO)CCN(C)C(=O)C1 c1(C(=O)NCCC(C)NC(C(COC)(C)OC)=O)[nH]c(C)c(C(C)=O)c1C CC1(C)COCC(C(=O)NCC2(C)CCN(C(C3CC=CCC3)=O)C2)O1 c1(SCC=CCOC(C=COOCC)=O)ccc(C)cc1 c1(Cc2nc(C(CCC)C)nn2-c2cnn(C)c2)cc(C)cc(F)c1 N1(C(CCCC#N)=O)CCC2CN(C(=O)C=Cc3ccc(F)cc3)CCC2C1 CC(CNC(=O)CC1(O)CCOC1)CC(=O)NCC1CC2(CC2)C1 C(CC(C(=O)N1CCCC(C)C1)NC(=O)COCc1nc[nH]n1)=CC N#Cc1cccc2c1CCN(c1nc(C(F)F)ns1)C2 c1(C(=O)NCC(CN(C(CCCC(=O)OC)=O)C)C)cc2nnn(C)c2s1 C(CC1=CCN(C(=O)Cc2cc(F)cc(F)c2)CC1)NC(c1cc(C)ncn1)=O C(=O)(CCCCCCN=[N+]=[N-])NCC1N(C(C2C(C=C)C2)=O)CC=C1 C1(NC(CN(S(C)(=O)=O)C)=O)CCC(NC(=O)C(F)n2cccn2)CC1 c1(C(=O)NCC2CN(C(C(CCSC)(C)C)=O)C2)cc2cc(C)ccc2o1 c1(-c2ccc(C(N(CCOC)CCNC(=O)CN3CC=CC3)=O)s2)cccc(C)c1 N1(C(CC(CC)C2CC2)=O)CC(CNC(=O)C=Cc2ccc(C)s2)C2(CC2)C1 CC(C)C(O)C(=O)NC(CNC(=O)C(C)C1CCCO1)C(C)(C)C C(C(CC(=O)N1CC2CC1C2C(=O)OC)OC)NC(COCC(=O)NC)=O C=CCCCCCC(=O)N1CC(C(=O)NOC(C)C=C)C2(CC2)C1 Cc1nnc2n1CCC2(C)C(=O)NCC(C)(C)CNC(=O)C(C)S(N)(=O)=O Cc1ccc(Cl)cc1C(=O)NC(C)C(C)NC(C1CCN(c2cncs2)CC1)=O N1(C(C2C(c3cccc(C)c3)CCCC2)=O)CCC(SC2CCCC2)C12CCCC2 C1(NC(C(c2cncc(F)c2)C)=O)CN(C(c2cnc(S)[nH]2)=O)CC(C)(C)C1 C1(NC(c2n(CC)ccn2)=O)CCCN(C(C2(COC)CC2(F)F)=O)C1 C1(NC(=O)NC2(CC)CCCC2)CCCN(C(c2cccs2)C)C1 c1(OC)cc(C)c(C(N2CC(NC(c3ccccc3)=O)C(F)(F)C2)=O)cn1 C1(C(N2CCC(NC(=O)Cc3cnn[nH]3)C2)=O)(CO)CCOCC1 Cc1oc(Br)cc1C(=O)NCCC(C)CCNC(c1nn[nH]c1Cl)=O c1(Oc2cncc(CC)c2)nc(CC(=O)OC(F)(F)C(F)F)cc(O)n1 N1(C(c2ccn(CC(C)C)n2)=O)CC(C)CCC1CNC(c1cnc[nH]c1=N)=O C1(C2CCN(C(=O)CCC(C)(C)F)C2)(NC(C2N(C(C)=O)CCC2)=O)CC1 c1(N2C3(CN(C(c4ccc(OCC)nn4)=O)C3)CC2)ncnn2cc(Br)cc12 N(C(=NCC1=CCCC1)NCc1cccs1)C1CCC(NC(C(C)C)=O)CC1 c1(C(=O)NC2CC(N(C(=O)CC3C=CCCC3)C)C2)coc2c1C(=O)NCC2 CC(CCC(=O)NCC(CNC(c1ccnn1C(C)(C)C)=O)CO)N(C)C C(CN=c1[nH]c(C)nc(C)c1C)C1CCCN(C(c2c(COC)noc2)=O)C1 CN1CCN(C(=O)Cc2cc(O)nnc2O)C(CNC(C2CCSC2)=O)C1 C1(C#N)(CC)CCN(C(C2CCC3(CC3)N2C(C23C(=O)C4CC2C3C4)=O)=O)CC1 C12(C(=O)NCC)CCN(C(=O)CCCCNC(N)=O)CCC1C2 c1(C(=O)NCCCC(=O)N(CC(O)CNC(=O)CSC2CC2)C)ccc(O)cc1 C12(NC(c3n[nH]c(C)c3Br)=O)CCC1CN(C(=O)C(O)CCN(C)C)C2 c1(C(N2CCC(N(CC(C)C)CCC)CC2)=O)cnn2ccccc12 S(=O)(=O)(c1ccc2c(c1)CC(C)O2)NC(c1c(C)cccc1)CN1CCOCC1 C1(CCN(C)C)CCN(C(=O)C(c2ccccc2)N2CCOCC2)C1 Cc1cnc2nc(NC(=O)NNC(=O)c3cnn(CCN4CCOCC4)c3)sc2n1 N1(C(C2CC(NC(C(CSC)C)=O)C2)=O)CC2(C)CC1CCO2 C=CC(CC)C(=O)NCCCN(CCCNC(C1C(C(C)=O)C1(C)C)=O)C c1(NC(CC(C(=O)OC)(C)C)=O)cccc2nnn(C)c12 CC1Cc2cc(C(=O)NC(C3CCCN3C(C3(C(F)F)CC3)=O)C)ccc2O1 C1(CC)(NC(c2cc(C)c(C)s2)=O)CCN(C(=O)Cc2conc2C)CC1 C1(NC(CN(C(Cn2ncc(CC)c2)=O)C(C)C)=O)CC2(C1)CC(C)(C)C2 N1(C(C2C(=C)C2)=O)CCc2nc[nH]c2C12CCN(C(C1CNC(=O)CC1C)=O)C2 N1(C(C2CCN(C(c3n(CCC)ncc3)=O)C2CC)=O)CC(O)C2(CCCC2)C1 c1(C(N2CCOCC(CNC(C3C(C)(C)C3)=O)C2)=O)cc2c(O)ncnc2cn1 c1(C(=O)NCC2(C)CCC(NC(c3c(OC)scc3)=O)C2)cnn2cccc2c1 CC(C(=O)N1CCCC(O)(CNC(c2csc(-c3ccco3)n2)=O)C1)C(C)(C)O Cc1ccc(CCC(N2CC(CNC(c3cnsn3)=O)C(C)(C)C2)=O)cc1C C1(CNC(C2(C)CC=CCC2)=O)CN(C(=O)C(F)=C2CCC2)CC12CC2 Cc1ccc(C(=O)NCC(CNC(=O)CNS(N)(=O)=O)C(F)(F)F)cc1[N+](=O)[O-] CC1CN(C(=O)COCC2CCCCO2)CC1CNC(C1CC(C)(F)C1)=O c1(CC)cc(OC)c(NCc2cc(F)c(F)c(F)c2)cc1ONC(=O)c1cccs1 CCC(C(=O)NCc1cc(C)c(C(=O)NCC(C)(C)CCO)o1)C(C)C Cc1ccc(Br)c(CCC(=O)Nc2ccc(Br)c(Br)c2)c1 C1(NC(C=C(CC)CC)=O)C2COCC1CN(C(c1ccc(Cl)c(Cl)c1)=O)C2 C12(C(=O)NC(C(CO)SC)C)C(=O)C3CC1C2C3.C1(=O)C2=NOC(C2)CN1 C1(N(C(=O)C(CCSC)OC)CC)CCCC(c2nn[nH]n2)C1 C1(NCc2ccc(C(=O)NC)o2)CCN(CC(C)CBr)CC1 Cc1c(C(=O)NC(CC2CC2)C(N2CCCCC2CC(C)C)=O)cccc1C#N C1(C)(C(N2C(CCC=C)CCC2)=O)CC(O)CN1C(=O)COc1ccccc1 N1(C(c2cc(CCC)[nH]n2)=O)CCCC(CCNC(=O)C2=C(C)CCC2)CC1 S(=O)(=O)(c1ccc(F)c(C(=O)NCC2COCC3(CNC3)O2)c1)NC(C)(C)C N1(C(c2c(OC)ccs2)=O)CC(C(=O)N(C(C)C(C)(C)C)C)C2(CC2)C1 C1(C(=O)NC2CC(CCNC(C=CC(=O)N(C)C)=O)C2)CS(=O)(=O)CC12CC2 C1(C(=O)NC(CCC=C)C)CC(O)CN1C(=O)CN1CCCCC1C N1(C(c2cc(C)c(CO)cn2)=O)CC2CCC(C1)C2NC(=O)C(C)C(C)(C)C c1(CC(=O)N(CC(CC)NC(c2cc(OC)nn2C)=O)C)c(Cl)cnn1C Cc1ccc(C=CC(=O)NC2CC(C)N(C(=O)Cc3cnns3)C2)cc1 C1(C2CCOCC2)(C(=O)NCCC(C)N(C)C(c2cc(Cl)cn2C)=O)CC1(F)F C1(C(N2CCC(N(C(=O)C(C)(C)c3cccnc3)CC)C2)=O)CCCC(OC)C1 N1(C(C(C)NC(=O)C2CC2)=O)CCOCC1CCNC(C1(C)CCC(=O)N1)=O Cc1sc(C)c(C(=O)NCCC2(NC(c3cc(CO)on3)=O)CCCC2)c1C#N c1(C(N2CCC(CO)(Nc3ncccn3)CC2)=O)ccc2nncn2c1 C1(O)(C(=O)NCC2N(C(C(F)=CC)=O)CC2)CCSCC1 c1(C(N2CC(C)OC(CCNC(=O)C(F)=CCCF)C2)=O)ccc(N)c(F)c1F c1(NC(c2nccc(C(C)C)c2)=O)c(F)ccc(I)c1Br C1(OCC)(CNC(C2CC=CCO2)=O)CN(C(=O)CCNC(=O)COC)C1 Nc1nc(Cl)ccc1C(=O)NCCC1CCN(C(=O)C(C2CCCCC2)O)C1 N#Cc1ccc(=NCC(=O)NCC(C2CCCC2)NC(c2n[nH]cc2Br)=O)[nH]c1 C1(NC2(c3n(C(C(=O)OC)C)nnn3)CCSC2)CCOC(c2ccccn2)C1 Cc1nc(NC(=O)NC(C)(Cc2ccc(F)cc2)CO)nn1-c1cccc(F)c1 c1(N2CCN(C3CCN(C(c4nnn(CC)c4C)=O)C3)CC2)cnc(C#N)cn1 N1(Nc2cncc(C(=O)NCC3(C(=O)NOCC)CC(=C)C3)c2)CCCCC1C n1(CC(=O)NC23CN(C(c4c(COC)nn[nH]4)=O)C(C2)C3)cc(C)ccc1=O C1(CC(=O)NC(CCNC(C(C2CCCC2)OC)=O)C)CCC(C2CC2)CC1 C12(NC(C(C)(C)c3ccccn3)=O)COC(CNC(=O)C=CC(=O)N(C)C)(C1)C2 c1(OCCC)ccc(CC(=O)OC)c(OCC)c1.C12(C)CCN1C2=O c1(C(=O)NCC(C)C(=O)N(C2COCC2(C)C)C)cccnc1S C#CCC(CC(=O)NC(C#C)CC1CC1)NC(C1CCCO1)=O Clc1ccccc1-n1nc(CC2CC2)nc1-c1cccc(N2CCOCC2)n1 C12(CNC(CCC(=C)Br)=O)CCC(CNC(=O)C(=O)N(C)C)(CC1)OC2 C1(CCCNC(c2ccc(C3CC3)cc2F)=O)CN(C(=O)C(F)C2CC2)CCO1 C1(NC(C=CC(C)(C)SC)=O)CC(O)CN(C(=O)CCC(C)C)C1 CC1CC(CN(c2ccccc2)C(=O)CCC2CC2)CN(C(=O)Cc2ccoc2)C1 c1(OC)cnc(Cl)[nH]c1=NC(=O)c1nc(-c2cc(C)c(F)c(C)c2)sc1C C1(C(N2CCN(CCC)CC2)=O)CCC(O)CN1C(c1ccncc1N)=O CC(C)C(O)Cc1cn(CCCN(C)C(c2cn(C)nn2)=O)nn1 c1(OC)cc(C)cc(C(=O)OC(C(N2CCC3(CC2)CC3CO)=O)C(C)C)c1O CC(C)CCC(C(=O)NCC1COCC(C)O1)NC(c1cn[nH]c1)=O N1(C(c2c(C)oc(Cl)n2)=O)CCOCC(C(=O)NC2C=CCCC2CO)C1 N1(C(C2(CNC(C3=C(C)CC3)=O)CCC2)=O)CCCCC(CN(C)C)C1 C1(CNC(CC=C)=O)(CO)CC12CCN(C(c1coc(C(N)=O)c1)=O)CC2 c1(C(=O)NCC(CC)NC(c2c(C)nc(CCC)o2)=O)cncc(F)c1Cl c1(CCC)cc(C(N2CCC(CN(C(=O)C=CC3CCCC3)C)C2)=O)n[nH]1 C(CC1CC1)(CC(=O)NC(C(N)=O)C1CCC1)NC(CN(CC#C)CCC)=O CC1(C)CC=C(C(=O)N2C3CCC2CC(NC(=O)C2=CCCC2)C3)CC1 CC1CN(C(=O)CNC2CCCc3ccccc32)c2cc(F)ccc2C(=O)N1 C=CCC(C)(C)CC(=O)NC1(C(=O)NC(C)C(F)(F)F)CCC1 C12(C(=O)NCC3(NC(c4cc(C(N)=O)[nH]c4)=O)CCCC3)CCCC1CC2 C1(CCOC)(NC(=O)CC(O)CN(C)C)CCN(C(=O)C(C)(C)C#N)CC1 N1(C(C(C)SCC)=O)CCCCCCC1C(=O)NCc1n[nH]cc1C c1(OC)ccc(C(C(=O)NCC(C)C)N(C(C)Cc2nccn2C)C)cc1CO C12(C(=O)NC3CN(C(C=C(COC)C)=O)C3)CCC(F)(CC1)C2 C1(CCn2c(-c3cc(C)ncc3)nc(CCO)n2)CN(C(C)C)CCCO1 N#Cc1cc(Br)ccc1CN1CC2C(C1)N2C(c1cnc2snnc2c1)=O C(C(C)(C(=O)NCC(C)(F)C(C)C)NC(=O)Cn1ncnn1)SC c1(NC(CC(C)NC(=O)CC(F)(F)C(F)F)C)ncnc2cnccc12 C1(NC(C2CCCC(C)C2)=O)CC2(CCN(C(c3ccc(F)c(F)c3)=O)C2)C1 C1(N(C(=O)CS(=O)(=O)N(C)C)CC)CCC(NC(=O)CCc2cn(C)cn2)CC1 C(=O)(CCCCCC#N)NCC(C(C)(C)C)NC(=O)Cc1c[nH]c2ccccc12 N1(C(c2ccc(CNC(C(C)N(CC)CC)=O)cn2)=O)CC(=O)N(C)CC1CC C(C(=O)NC(C)(C)C(F)F)(C(C)C)NC(CC1C(CC)C1)=O Cc1cc(=NCC2CCN2S(C)(=O)=O)[nH]c(-c2cccnc2)n1 C(CC(C(=O)N1CC(C(=O)NCC)C1)NC(=O)C(C(C)C)SC)OCC C1(NC(C(C)(C)C(N)=O)=O)CC(C2CCN(C(c3cccc(O)c3F)=O)C2)C1 C1(CC(=O)NCCCCC(C)NC(c2c(C)scn2)=O)CC2(CCC2)CO1 CC1(CNC(c2ns[nH]c2=O)=O)CC(F)(F)CN1C(=O)C(F)C(F)(F)F c1(C(=O)NC(C2(O)CN(C(c3cnn(C(C)(C)C)c3)=O)C2)C)nccnc1N c1(OCCC(=O)Nc2ccc(C3C(=O)NC(=O)S3)cc2)ccc(Cl)cc1Br C=CCC(C)(C)C(=O)NCCn1cc(C(=O)N(C2CCC2C)C)cn1 CC1(C(=O)NCCN(C(c2cc(Cl)cs2)=O)Cc2ccccc2)CCC2CC2C1 Cc1cccc(-n2nc(CCSC(F)F)nc2CNc2ccc(Cl)cn2)c1 C1(C(N2CCC(C(N(C)C)=O)C2)=O)CCN(C(c2cccnc2O)=O)CC1 C1(CC)CC(CC)CCN1S(=O)(=O)CC(C#N)C1CCN(C(C)=O)CC1 n1(CC)cc(C(=O)N(CCC(N2CCC(C)(C(N)=O)C2)=O)C2CC2)c(C)n1 C1(NC(C(C)(C)OCC)=O)CN(C(C2CC2C)=O)CCC1c1ccc(F)cc1 N1(C(C(CCN(C)C)NC(CC(C)C)=O)=O)CCCCCCC1C C1(C(N(C)CC2(NC(c3ccc(CC)[nH]3)=O)CC2)=O)CC(F)(F)C1(C)C C(C(=O)NC(C)CC1CN(C(c2ccc(C3CC3)cc2)=O)C1)(C(C)C)NC(C)=O N1(C(c2c(CC)nn[nH]2)=O)CC(F)(F)CC1CNC(=O)CCc1ncco1 CC(C)(CC(=O)N1CC(CNC(C2CC3(CCC3)CO2)=O)C(C)(C)C1)C(F)(F)F c1(C(=O)NC2(C(=O)NCC3(Cl)CCC3)CCSC2)cccnc1O C1(CNC(C2CC(CC)OCC2)=O)CCCCCN1C(c1cc2occc2[nH]1)=O N1(C(c2c(CNC(C3CC34CCC4)=O)cc[nH]2)=O)CC2(CC(O)C2)C1 C1(=CC(=O)NCC(CCCC)NC(=O)C(C)c2cccs2)CCC(C)(C)CC1 C1(CNC(C2C(C)CCC2)=O)CN(C(c2ccc(NC(C)C)cc2)=O)CCCO1 Cc1cc(F)ccc1NC(c1cc(C)c(Br)s1)c1nnnn1CCCC1CC1 Cn1cc(C(O)C(=O)NCC2CCCN2C(c2coc(O)n2)=O)cn1 N1(C(c2nc(C)sc2)=O)CCC2(CCN(C(=O)C(C)(C)C(C)(C)O)CC2)C(C)C1 C1(C(=O)NC(CNC(C2CN(C(=O)NC)C2)=O)(C)C)CCC(COC)O1 c1(N(CC=C)C)nnc(CCC2CCCO2)n1CC1CCCCO1 C(=O)(CCCc1nncn1C)N(C(C)C)CCNC(C1(n2cncn2)CC1)=O Cc1nc[nH]c1CC(=O)NCC(C)NC(=O)CNC(=O)NC1CC1 C1(C(=O)NC(C)(CNC(c2cnn(C3CC3)c2)=O)C2CCC2)CN(S(N)(=O)=O)C1 C(CCC(=O)NCCC1(C(=O)N(C2CCSC2)CC)CCC1)OCC c1(C(=O)NCC2C(C)CN(C(=O)COCC(=O)N(C)C)CC2)ccc2c(n1)NCC2 C1(CC(=O)NCCOC2CCN(C(C3(C)ON=C(C)C3)=O)C2)CCCS(=O)(=O)C1 c1(C(N2C3CCC(NC(CCC=CC)=O)(C3)C2)=O)cccc2c1OCC2 Cc1cc(=O)c(C(N2CCC2CNC(=O)C(C)(O)C2CCC2)=O)cn1C N1(C(C=C(CC)C)=O)CCC2(CC1)CC2CNC(C1(CC(C)C)COC1)=O C(=O)(CC(C(C)(C)C)NC(=O)CC1CSCCO1)N1C(CC(C)C)CCC1 C1(C(N2CCC(NC(c3ccc(CC4CC4)s3)=O)C2)=O)OC2CCC1CC2 Cc1nc(CCNC(=O)C(Cc2ccco2)NC(=O)C=CCN2CCCC2)cs1 C1(CN(C)C(c2[nH]nnc2C2CC2)=O)COCCN1C(c1ncccc1Cl)=O C1(N(C(CC=C(C)C)=O)C)CCN(C(C2C3CCCCCC23)=O)CC12CC2 N1(C(C(C(=O)OCC)F)=O)CCCC(C2(NC(c3oc(COC)cc3C)=O)CC2)C1 c1(N2CCC(CCNC(c3ccnn3CCF)=O)C2)cc(C(F)(F)F)nc(Cl)n1 c1(C(N2CCCC2c2cn(C3CC(O)C3)nn2)=O)c(F)ccc2occc12 Cc1nc(N2CC(OCCNC(c3c(Cl)cnn3C)=O)C2)c(C)c(C)n1 C=CCC(C(=O)N(CC(O)CN(C)C(C1CC1C)=O)C)NC(C)=O c1(C(=O)NCCCC2N(C(C(C)OCCOCC)=O)CCC2)cc(F)ccc1C C1(NC(C2CN(C)C2)=O)COC2(C1)CN(C(=O)Cc1cnns1)C2 C1(OC)CC2(CCC(C(N3CC(NC(c4nc5ccccc5o4)=O)C3)=O)CC2)C1 C1(C(N(C2CCCN(C(=O)CN3CCC(F)(F)C3)C2)CC)=O)CC12CC(C)(C)C2 CC(C)CS(=O)(=O)CCC(=O)N1CCC(CF)(NC(=O)CC(O)C(C)C)C1 c1(CC)nccn1C(C)CC(=O)N1CCCC1C(C)(C)NC(C1CCC1OC)=O N1(C(C2C3(CCN(C(c4[nH]cc(C#N)c4)=O)C3)C2)=O)CC2CCC(C1)C2O c1(C(N(CCNC(C(C=C)C)=O)CC)=O)cnn2cccnc12 C(=O)(N1CC=CCO1)C1(C)CCN(C(CC(COC)C)=O)C1 Fc1ccc(I)c(CNC2CN(CC3CCC3)C2)c1 C1(NC(c2cccc(CC=C)c2)=O)CCN(C(C2(COCC)CC2)=O)CC1O CCCCC(O)C(=O)N1CC2CC2(NC(c2ccc(-c3cc(O)ns3)cc2)=O)C1 C(CCN(C)C)(C(=O)N1CCCC1CCO)NC(c1nc(CC)sc1)=O c1(C(=O)NCCC2CCCN2C(c2ccc(Cl)s2)=O)ccnnc1Cl n1(CC(=O)NC(C2CN(C(c3c[nH]nc3F)=O)CCO2)C)cnc([N+](=O)[O-])n1 c1(C(N2CC3COCC3C2)=O)cnn2cc(-c3cc4c(F)cccc4[nH]3)ccc12 CC1(C)C(C(N2CCN(C(c3cncc(N)c3)=O)CC2CF)=O)CCS1(=O)=O c1(NCCCC(CC)O)ncnc(NCCN2CCC(C)(F)C2)c1C C1(COC)(CNC(c2cc3sccc3s2)=O)CCN(Cc2cc(C)no2)CC1 c1(C(=O)NC(C(CO)NC(CC)=O)C)cncc(C(=O)NC2CCC2)c1 C(=O)(C(CCC)CC(C)C)N1CC(CNC(CC=CCC)=O)C2(C1)CC2 N#CC1(C(N2CCOCC(NC(c3c[nH]cc3C(F)(F)F)=O)C2)=O)CC2CC2C1 C1(NC(CC(C)OCC)=O)CCC2(CCN(C(c3ccc(NC)cc3)=O)CC2)C1 C12(NC(=O)NCc3ccc(OC)cc3C)CCC(CC1)C(C)(C)O2 N1(C(c2c(C)n(C)nc2)=O)CCC2CCCN(C(=O)Cc3ccc(F)cn3)C2C1 OC12CCCCC1CN(CC=Cc1ccc3c(c1)OCO3)CC2 C12(CCNC(C(C)OCC)=O)CCC(CC1)N(C(=O)C(CC)c1cccnc1)C2 C1(C(N2CC(C)C(NC(=O)CCCCCNC(N)=O)C2)=O)CC(=O)NC(=O)C1 CC1CCCCCC1NC(c1ccc(F)c(F)c1)=O CCCCCCCC(=O)N(CCNC(C1(C(=O)OC)CC1C)=O)CC c1(CN(C2CCCN(C(CC3C(C)CCO3)=O)C2)CCO)nnc2n1CCCCC2 c1(CC(=O)NCC(CN(C(=O)CC2(c3ccccc3)CC2(C)C)C)O)nc(=N)[nH][nH]1 C1(C(=O)NC2CC=C(C)CC2)CN(C(=O)Cn2ncn(C)c2=O)CC12CCC2 c1(C(N2CC(CC(=O)NC3(CO)CCOC3)(OC)C2)=O)c(F)cccc1F CC1(C)CCC=C(C(=O)NC2(CCNC(=O)Cn3cccn3)CCCC2)C1 O=C(C(O)CC(F)(F)F)NCC1C(C2CC2)CCN1C(c1cc(F)ccc1Cl)=O CCCCS(=O)(=O)NCC(=O)NCC1(OC)CN(C(=O)CC(C)(C)O)C1 C#Cc1cccc(NC(C2CCCN2C(C2CCCC(F)C2)=O)=O)c1 C(C1=NOC2(CCC2)C1)C(N1C(c2cn(CC(CC)O)nn2)C(C)CC1)=O C1(CCN(C)C(C2CC2C#N)=O)CCN(C(=O)C(c2cscn2)N(C)C)CC1 N1(C(c2nccc(C(=O)OC)c2)=O)CC2CCC1C(Nc1ncnc(Cl)c1F)C2 S(=O)(=O)(c1cccc(N2CCCc3[nH]ccc3C2)n1)N(CCCC=C)C c1(N(CC(=O)NCC(CN(C(c2c(C)ocn2)=O)C)C)C)ccc(Cl)cc1C#N CCCC(C(=O)NCC1CN(C(C2CC(CF)C2)=O)CCO1)N(C)C C1(CNC(c2c(C)nn[nH]2)=O)COCCN(C(=O)CCC2CCN(C)CC2)C1 C1(NC(C2CC23CCC3)=O)C2CC3C1C3C2C(=O)NC1CC2CCC(C1)S2 CC(C(F)C(=O)NCC1CCN(C(c2ccc([N+](=O)[O-])c(O)c2)=O)C1)C(F)(F)F c1(OC)cccc2sc(-c3nc(-c4ccsc4)nn3CCN(C)C)cc12 C1(C(=O)NC2CC(C(C)NC(COC(CC)CC)=O)C2)CCC(F)C1 N1(C(CCOCC(C)C)=O)CCN(C(C2CCC2)=O)CC1CC(F)F C(=O)(C1c2ccccc2CN1Cc1ccc(F)c(F)c1)N1CCC(C)CC1 c1(C(=O)NCCC(CNC(C2CC3CCC(C2)C3)=O)OC)cn2ccccc2n1 C1(C(=O)NCc2cc(C(=O)NCC(C)(O)C3CCC3)n[nH]2)C2CCC(=O)C12 C=CC1CCCCN1Cc1c(C(=O)OC(C)(C)C)cccc1 C1(C(N(C)Cc2nc(C)[nH]n2)=O)C2CCCC2CN1C(=O)C(Cl)Cl C1(CNC(C(C)C23CC2C3)=O)CCCN(C(=O)Cn2nnc(-c3cccs3)n2)C1 c1(OC)cc(Br)ccc1C(N1CC=CC(NC(=O)CN2CCCC2=O)C1)=O c1(CC)cc(C(=O)NCC2CCN2C(C2CC2c2cnc[nH]2)=O)cc(O)n1 C1(C(=O)NC(CC)C(=O)NC)C=CCN(C(=O)C(C)c2ccco2)C1 C1(C)(CNC(c2nc(C(C)C)oc2)=O)CCCN1C(c1n[nH]c(C(C)(C)C)n1)=O N1(C(CNS(C)(=O)=O)=O)CCCOC(CNC(c2ncoc2C2CC2)=O)C1 Cc1sncc1C(=O)NCC(C1CCCCC1)NC(=O)CCn1cc(Cl)cn1 Cn1ncc(Br)c1C(N1CCC1CNC(C1(C(F)(F)F)CC=CC1)=O)=O C(=O)(CC(C)(C)C(F)F)N1C(CN(C(COCC#C)=O)CC)CCCC1 C=CCC(C)(C)CC(=O)NCC1CN(C(c2ccc(F)c(N)c2)=O)CCC1C N1(C(c2cc(C)[nH]n2)=O)CC2CC(NC(=O)CC3CC4(CC4)CO3)C1C2 C(=O)(CC(C(F)(F)F)OC)NCC(C1CCC1)NC(Cc1cc(CC)nn1C)=O c1(C2(C(=O)NC3C(NC(CN(CCOC)C)=O)CCC3)CC2)ccc(F)c(Cl)c1 C1(CCC)CN(C(=O)Cc2ccco2)CCN1C(=O)CC1COCCN1C c12cc(F)ccc1S(=O)(=O)NC(=O)NCC2N1CCCC1.N1(CC)CCC(C)CC1 C1(Cn2cc(-c3ccc(OC)cn3)nn2)COCCN(C(C2CC2(Br)Br)=O)C1 C1(SC)CCCC(NC(=NCc2ncccn2)NCc2ccnn2C)C1 c1(OC)ccc(C)c(OC)c1C(N1CC(NC(c2ncncc2Cl)=O)C1)=O N1(C(C(CCC)(C)C)=O)CCC2(CCC(CNC(=O)C(C)CC3CC3)OC2)CC1 c1(C(N2CCC(CNC(C3(C)C(C)C3)=O)C2)=O)c(N)cc(F)cc1Cl c1(-c2n(C(COC)C)nc(C3CC3)n2)ccc2c(c1)nnn2Cc1ccccc1 N1(Cc2cccc(OC)c2C)CCC(NC(=O)C(c2ccccc2)F)C(C)(C)C1 c1(SC)cc(C(=O)NCCC(C)N(C)C(c2sc(CO)nc2C)=O)c(C)o1 C1(NC(CC=CC=C)=O)CC2CCCC(C1)N2C(C1COC(C)(C)C1)=O Cc1cnc(N)c(S(=O)(=O)N)c1.C1(C2(O)CCC2)(NCC(C)C(F)(F)F)CC1 Cc1cc(C(N2CCC(O)(C(N3CCCC3(C)C(F)(F)F)=O)C2)=O)c(C)n1C CCCCN=C(NCCC1CC1(Cl)Cl)NCCn1cncn1 C=CC(CCC)CC(=O)NCC(CCC)C(=O)N(C1CCCCC1(C)O)C CC1CCc2nc(C(=O)NC3CNCCC3CO)cn2C1 N1(C(C2CSCN2C(C2CN3CCC2C3)=O)=O)CCC(=C(F)F)CC1 C(=O)(C(C)CC(F)(F)F)NC1(COC)CCN(C(c2c(CC)sc(=N)[nH]2)=O)CC1 C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NCCC(CCNC(C(CC)OC)=O)C Cc1cn(CC(N2CC(F)(C(=O)NCCC(=O)NC(C)(C)C)C2)=O)c(=O)nc1O CC(O)C(C(=O)N1CCC(O)(CCNC(=O)CCc2ccccc2)C1)N(C)C c1(C(N2CC(CNC(C(CC)n3ccnc3)=O)C2)=O)cn2ccnc2cn1 C(C(C)(C)C(=O)N=c1ccn(CCF)[nH]1)N(C(C1Cc2nccn2C1)=O)CC CCC(C#N)(CC)C(=O)N1CC=CC(NC(=O)C=CSc2nc[nH]n2)C1 c1(C(=O)NCCC2CN(C(c3c(C)nccn3)=O)C2)ccc2ccnc(Cl)c2n1 c1(C(N(C2CCN(C(C3CC=CCC3)=O)CC2)C)=O)cn(C)c(=O)cn1 c1(CC)c(C(N2CC3CC3(NC(=O)CSc3ccc(F)cc3)C2)=O)nnn1C C1(CCOC)(NC(=O)C(c2ccc(C)cc2)C)CCN(C(=O)CNS(N)(=O)=O)C1 c1(C(=O)NC2CN(C(C(CCSC)NC(N)=O)=O)CC2O)cnc2sccn12 C1(C(=O)NCC2(CCNC(c3cc(Cl)cnn3)=O)CC2)OCCOC12CCC2 C1(CNC(C2CCC(O)C2)=O)CC2CCC1N(C(c1cncc(Br)c1)=O)C2 c1(CCC)cc(NC(=O)C(C)(c2ccccc2)NC(=O)NC)c(C)o1 CC1CN(CCO)CCN1N1CCC(CN2CCN(C)CC2)CC1 c1(C(C)(C(=O)O)OC(C)=O)cccc(Cl)c1.N1(C(CC2(CC(=O)OC)CC2)=O)CCCC1 Cc1[nH]c(C(C)(C)C)cc1C(=O)NC1(C)CCN(C(=O)CCc2ccsc2)C1 N1(C(CC2C(C)(C)OCCO2)=O)CCN(C(c2cccc(N)c2F)=O)CC(O)C1 Cc1cc(C(N2CCC(F)(C(N3CCOC(CCF)C3)=O)CC2)=O)cc(C)n1 C(=O)(C(C(C)CCCC)N1CCCC(OC(C)(C)C)C1)NCCOC Cc1ccc(C=CC(=O)NCC(C(C)C(C)C)NC(c2cnc(O)o2)=O)cc1Cl c1(C(=O)NCc2cn(CC(=O)NCC(CC)O)nn2)cc(F)cnc1O CCC(C#N)C(=O)N(O)Cc1cn(C(C)C(=O)NCc2ccc(C(F)F)o2)nn1 C1(NC(CN(C2CCSC2)C)=O)CCN(C(c2cnnn2C2CC2)=O)CC1C N1(C(c2c(C)oc(C)c2C)=O)CC(O)(C2(CNC(=O)C(C)(O)C(C)(C)C)CC2)C1 C(=O)(C1CCc2c(Cl)cccc21)NC1C(NC(c2cc(CC3CC3)on2)=O)CC1 C1(CNC(Cc2cn(C)nn2)=O)(CO)CCN(C(=O)CCCc2cc[nH]n2)CC1 C1(C(N2CCC(NC(C(CC)(C)C)=O)C(CO)C2)=O)CCCc2ccccc2C1 C1(C(N(CC(CC)NC(=O)C(c2cccc(C)c2)O)C)=O)CCN(OC)CC1 c1(OC)ccc(C(N2CCC(NC(=O)Cc3scnc3C)C(F)C2)=O)c(Cl)c1 C=CCC(CNC(c1cc(C2CC2)[nH]n1)=O)C(=O)N1CCCC(F)CC1 N1(C(C=CC(C)NC(C(C)CCN(C)C)=O)=O)C2CCC1CC(F)C2 CC1(C(=O)NCC2(CNC(C3CCCCC3(F)F)=O)CC2)CCCCCC1 c1(NC(C(CC)C)c2nnnn2-c2cccs2)ccc(-n2cccc2)c(Cl)c1 N1(C(c2cc(C(C)=O)[nH]n2)=O)CCCC1(C)C(=O)NC(c1cccc(C)c1)CO c1(C(=O)OCC2CC2(Br)Br)n[nH]c2ccc(I)cc12 Cc1ccc(CC(=O)NC(C)(C)CCCNC(=O)CCCCC#N)cc1O N1(C(C2(CC)CCCC2)=O)CC(O)(C2CCN(C(C3CC4CCC4C3)=O)CC2)C1 Cc1cc(C(=O)NCC2CCCC2NC(=O)CC2COC(=O)C2)cc(O)n1 c1(C(N2CCC(C(C)NC(c3c(C)cco3)=O)CC2)=O)c(C)nn2ccccc12 C1(F)(CNC(c2n(CC)ncn2)=O)CCCN(C(=O)CCS(N)(=O)=O)C1 CC12CC(CO)(C1)C(CNC(c1csc(C3CCCCO3)n1)=O)O2 c1(CCN)ccc(-c2nc(-c3ccc(Br)cc3)n[nH]2)cc1 C(CCF)(C(=O)NCC1(O)CCC(C)C1)NC(C1C=C(C)CS1)=O C(=O)(CCCC(=O)N1CC(NC(c2c(C)noc2C(C)C)=O)CC1C)NCC Cc1ccc(C(=O)NC(Cc2cc[nH]n2)C(=O)NC(C(C)(C)O)C2CC2)c(F)c1 CC1CC(NC(=O)Cc2nc[nH]n2)CN(C(c2nnc(O)cc2O)=O)C1 C1(NC(C=CC=CC)=O)CCN(C(=O)C(O)Cc2ccccc2)C1C(C)C c1(C(CSC2CCOC2)NC(=O)Nc2c(CCC)onc2C)c(C)cccc1Br C(C1=CCN(C(C2CCCC(=O)O2)=O)CC1)NC(CC=C(C)C)=O CC1CCc2cc(C#N)c(N3CC(C)(NC(c4cc(Br)co4)=O)C3)nc2C1 c1(C(=O)NCC(C2CC2)NC(C(C)OCC)=O)ccc2c(c1)C(=O)N(C)C2=O N1(C(C(C)(C2CCC2)NC(c2c(CCC)nco2)=O)=O)CCOC(C)(C)C1C C1(CC(=O)NC2(CN(C(c3c(OC)nsc3)=O)C)CC2)CCC(=O)NC1 CCC(C(=O)NC1CCC(CCC(=O)Nc2conc2CC)C1)SC c1(C(N(C2CCN(C(=O)CCF)CC2)CCOC)=O)ccc2c(c1)CCC2 N1(CC(=O)NCCCN(C(c2cnc(-c3ccco3)s2)=O)CC)C(=O)CNC1=O N1(C(C2N(C(C)=O)CC(O)C2)=O)CCCC(C(=O)Nc2ncc(Br)nn2)CC1 C1(NC(c2conc2C2CCCC2)=O)Cc2cscc2C1 c1(NC(=O)Cc2cc(C3(C4CCCC4)CC3)on2)ccccc1Br c1(-c2n(Cc3ccc(OC)cc3)nc(C3CC3)n2)cc2cc(F)c(F)cc2[nH]1 c1(C(=O)NCC2C(NC(CC(C)CN(C)C)=O)C2)ccc2cc(F)ccc2n1 C(=O)(C(O)CC(C)(C)C)NC1CC(O)(CNC(c2c(C)n[nH]c2C)=O)C1 c1(C(=O)NC(CNC(=O)C=CCn2cncn2)C2CC2)cc(F)cc2c1NCCC2 N1(C(C(C2CCC2)OC)=O)CCC(C2CC2)(NC(c2ccns2)=O)C1 c1(C(=O)NCC2C(NC(c3cnc(O)s3)=O)C2)ncccc1N1CCOCC1 C1(NC(c2c(CC)occ2)=O)CCN(C(=O)CSCC(=O)OC(C)(C)C)C(C)C1 N1(C(C2N(C)CCCC2)=O)CCC(C(=O)NCC2(CC(N)=O)CC2)C(C)(C)C1 c1(C(=O)NCCCNC(c2ccc(C)c(C(F)(F)F)c2)=O)cc2c(cn1)OCO2 Cc1ccc(C(N2CC(NC(c3c(O)cccc3F)=O)CC(C)C2)=O)c(F)c1F n1(CC)nc(C(=O)NC(C)(C)CNC(C23CCC(CC2)O3)=O)cc1C(F)(F)F N1(C(c2cc3c(s2)CCOC3)C(=O)NCc2ccco2)Cc2ccc(O)cc2C1 C1(NC(C(CC)C)=O)C=CCN(C(c2cc(-c3ccc(Cl)cc3)no2)=O)C1 C=CCC(C(=O)NCC1CC(C)(C)CN1C(=O)CC(=O)N(C)C)C(C)C C1(C(=O)NCc2cc(C)ncc2)CN(C(c2cc(Cl)cs2)=O)C(C)(C)C1 C1(NC(CCC(=O)NC)=O)CN(C(c2cc(N)c(F)cn2)=O)C2(CCOCC2)C1 N1(C(CN)C(F)F)CCN(C(N(c2cc(O)cs2)C2CC2C2CC2)=O)CC1.C Cc1cc2ncc(C(=O)NCC3CCN3C(=O)CC3CC4CC4C3)c(C)n2n1 CC1=NOC(C)(C(=O)N(C)CCN(C(=O)CC2(C)CC2(F)Cl)C)C1 C(=O)(CN=c1[nH]c(C)cs1)NCCOC1CCN(C(C2CC3(CC(=C)C3)C2)=O)C1 C1(C)(CC)CCCN(C(C2CC(CNC(c3cncc(C)n3)=O)C2)=O)C1 C1(C(N2CCC(C)C2)=O)CCC(NC(=O)NC(c2ccccc2)=O)CO1 c1(C(=O)NCC(C2CC2)Nc2ccc(C(=O)OC)cn2)cnc2cc(C)nn2c1 C(C(CC(F)(F)F)NC(C1CCCOC1c1ncc[nH]1)=O)NC(C=C(COC)C)=O Cc1c(C(=O)NC2(C)CCN(C(=O)CCC(C)O)CC2)oc2c(F)cccc12 c1(C(=O)NCC(CC2CN(C(C3C(CC)OCC3)=O)C2)(C)C)cn2ccnc2cn1 c1(C(C(=O)NC(CC)(C)C)N(C2CCCCC2(C)C)C)n[nH]c2c(Cl)cccc12 Cc1cn2cc(C(=O)NCC3(C)CC(F)(F)CN3c3ccnc(C)n3)sc2n1 C1(NC(=O)CNC(=O)C2CC2)CCOCC1NC(c1cn(C2CCC2)nn1)=O c1(C(=O)NC(CC)C(=O)NC2CC(=C(C)C)C2)ccn(CC)c1C N1(C(CC=CCCCCC)=O)CCN(C(c2cc(C)sc2N)=O)CC1 N1(C(c2ccc(COC(C)=O)cc2)=O)CCOCC(CNC(=O)CCC2CC2C)C1 c1(C(=O)NCC2(F)CC(NC(CCC#C)=O)C2)ccccc1CS(C)(=O)=O N1(C(C2C(C)C2)=O)CCC2CCC(NC(=O)C=Cc3ccn(C)c3)C12 CN1CCN(C(C2CC3COCC3C2)=O)C(CNC(c2n[nH]cc2Br)=O)C1 n1(CCC2(C)CC2)cc(C#CC(C)(C)NC(=O)Cc2cccc(Br)c2)nn1 c1(C(=O)NCC2N(C(COCCC)=O)CCC2C2CC2)cc(F)c2c(c1)CCC2 CCCC(O)CC(=O)NCC1(CNC(C2CCN(c3ncccn3)CC2)=O)CC1 c1(C(=O)NCC(C)(C)NC(C=CC)=O)ccc(=O)n(CCO)c1 CC(C)CC(C)(O)C(=O)N1CC2=C(C1)CN(C(=O)CCc1ncco1)C2 CCC(C)(C)C(=O)NCC1(F)CC(NC(C2CC(CC(F)F)C2)=O)C1 CCCCC(CC)CC(=O)NCC1CC(F)CN1C(C1CC(OC(C)(C)C)C1)=O CCCCCC(O)C(=O)N1CC(NC(c2nnc(C)cc2O)=O)CC(C)(C)C1 C1(C(N(C2CCCOC2)CC)=O)CCCN(C(=O)CCc2cscn2)C1 Cc1oc(C(C)(C)C)cc1C(=O)NCC1CCCN1C(N)=O N1(C(C2CC(C#N)C2)=O)CCCC(C2CC2NC(c2ncccc2CO)=O)C1 C1(CN(C2CCOC(C)C2)C(CC(C)C)=O)CCC(NC(=O)C(C)(C)C)CC1 C1(C(=O)NCC2N(C(c3cnc(CC)[nH]3)=O)CC(O)C2)CCC2(CCC2)C1 Cn1cc(C(N2CC3CC3(CNC(C3(CO)CCCO3)=O)C2)=O)ncc1=O c1(CSC(C)C(N2CCN(c3ccncc3F)CC2)=O)ccccc1C(F)(F)F c1(C(=O)NC(CC=C)CNC(c2nccn2C)=O)[nH]c2cc(F)cc(F)c2c1C C(=O)(C(O)CC(C)(C)C)NC(CCCC)CNC(c1ccc(C(C)C)c(F)c1)=O C(c1ccc(F)c2ccccc12)=CCNC1(c2ccc(F)cc2)CC(CC(=O)O)O1 c1(NC(C=CC(=O)N(C)Cc2nc(-c3cccs3)n[nH]2)=O)ccc(F)cc1 C(=O)(CC(C(=O)N1CCC(NC(=O)C(C(C)C)SC)C1)N(C)C)OC CC1CCC=C1C(=O)NCCC1CC(NC(c2ccc(SC3CC3)cc2)=O)C1 N(C1COc2cc(Br)cc(F)c21)C(N1CCCC(F)(CO)C1)=O c1(C(=O)Nc2nc(Cl)ccc2I)ccc2c(C(=O)N=c3cco[nH]3)n[nH]c2c1 N1(C(c2cnc(Cl)[nH]2)=O)CCCC2(CCN(C(=O)C3COc4ccccc43)C2)C1 C1(NC(C2(C)CC=CCC2)=O)CC2(CCCCN2C(=O)CCC2CC2(F)F)C1 C(C(C(=O)NC(C)C(=O)NCC(C)C)C(C)C)NC(c1n(CC)nnc1)=O C=CC(CCC)CC(=O)NC1CCCCC1NC(c1cnn2ncccc12)=O C=CCC(CNC(c1ccc(C2CC2)o1)=O)C(=O)NC1C=C(C)CCC1 CC1=C(C(=O)NCC2CCN(C(=O)C(c3c(C)n[nH]c3C)C)CC2)CCO1 c1(SC)cc(C(=O)N(CCCNC(=O)CC2C=CCCC2)CCO)oc1C n1(CC(=O)NCCN2CCN(C(C(C)OCC3CC3)=O)CC2)cc(F)ccc1=O c1(C(N(CCOCCNC(c2n[nH]c(C)c2N)=O)C)=O)cc2cscc2s1 c1(C(N2CC(N(C(=O)CCC3CCCN3C)C)C2)=O)coc2c1C(O)CCC2 c1(C(COC)N(C(CCC)C(=O)Nc2cccs2)CC)ccc(Cl)cc1Cl c1(C(C)OC(=O)COCCC2CC2(Cl)Cl)ccc2c(c1)CCC2 C1(c2ccc(CC)cc2)CN(C(=O)CSC(C)C)CCN1C(=O)CCCC(C)C C1(C(=O)NCCC(=C)CSC)CC2CCC(C1)N2C(=O)C(C)Cn1ccnc1 Cc1nn(CC(N2CC(CNC(C3CC3CF)=O)C(O)C2)=O)cc1Br c1(C(=O)NC(C2(C(N(CCSC)CC)=O)CC2)C)ccc(C)c(F)c1 C1(C(N(C2CCN(c3snc(COC)n3)C2)C)=O)(CCF)CCOCC1 c1(CNC(C(C=CC)O)=O)cc(C(=O)NCc2nnnn2CCC)ncn1 c1(C(=O)NC2CCN(C(C=COC)=O)CCC2CO)cnc(O)c2ccccc12 C1(C(=O)NCC(CCNC(C2(CC)CCCO2)=O)O)CC(=O)N(O)C1 C1(C(N(CCCNC(c2c(CC)n[nH]c2)=O)CCO)=O)CC2CCC2C1 N1(C(C(C)NC(c2ccc(NC)cc2)=O)=O)CC2CCN(C(=O)CC(C)(F)F)C2C1 C1(C(=O)NCC2N(C(C(C)C3CCC3)=O)CC2)CC2CC1C1C2C1(F)F c1(N(CC(C)CNC(=O)C(C)(C)C)C)nccc(CO)n1 c1(C(N2CC3C(NC(CCc4ccc(CC)cc4)=O)C3C2)=O)ccc(Cl)c(O)c1 C(=O)(CCC1=CCCCC1)NC1CCC(NC(C(CCC)OCC)=O)C1 Cc1ccc(C=CC(=O)NC(C)CC2CN(C(=O)CC(F)F)C2)s1 N1(C(CC(C)n2cccn2)=O)CCC(C2CC2)C1CNC(C1(O)CCSCC1)=O N1(C(C=CCCC)=O)CCN(C(C2CC2(C)C)=O)CC2(C)CCCC12 c1(C(C(=O)NCC(=C)C)N(CC(C)(C)COC)C)ccc(C(F)F)cc1Cl c1(C(C)NC(=O)C=CCC(C)(C)NC(=O)CCC2CCC(=O)C2)nn(C)cc1O C(=O)(C#CC(C)(C)O)N1C(C(N(CC(CC)(O)CC)C2CC2)=O)CC(O)C1 c1(CC)c[nH]cc1C(=O)N(CCNC(=O)Cc1csc(C2CCCC2)n1)CC Cc1ccc(C(N2CCC(CCNC(=O)C(O)C(C)C)CC2)=O)c(Br)c1F CCC(CCC(=O)NC(C)CCF)NC(c1ccc(C(C)=O)o1)=O C1(C(N2C(C3CCN(C(c4ocnc4C4CC4)=O)C3)CCC2)=O)CCS(=O)(=O)CC1 CCCCC(CNC(=O)CCCOC(C)(C)C)NC(c1nccn1CC)=O NS(=O)(=O)c1cnn(CC(N2CCCC2CNC(c2cccs2)=O)=O)c1 c1(C(=O)NCC2CCN(Cc3onc(C(C)C)n3)C2)cnn2ccn(C)c12 c1(N(C)C)cnc(C(=O)N(C2CCCCC2)CCNC(C2CC2(F)F)=O)cn1 N1(C(CCC2CC(OC)C2)=O)CCC(CNC(=O)CC2CSCCO2)C1(C)C C(=O)(CC(F)(F)C(F)F)NCC12CCN(CC1)CC2.CC12CCN(C1)C(=O)C2 c1(OC)cccc(-c2cn(CC(=O)NCCCCCCC3CCCCC3)nn2)c1 n1(CC(=O)NCC(CNC(=O)C#CC2CC2)CO)c(=O)oc2ccccc12 C1(c2ccccn2)CCCN(CC(=O)N)C1.C(COCCOCCOCCO)OC c12ccc(F)c(c1)C2.c1(CNc2cccnc2)ncsc1Br.O=C1C(C2CC2)N1 n1(C(C)C)ncnc1C(=O)NCC1CC(F)(NC(=O)COCC2CCC2)C1.C1CC1 c1(C(=O)NC(CC)CNC(=O)Cc2cn[nH]c2)oc(P(C)(C)=O)cc1C c1(C(N2CC(OCCNC(C(C)NC3CC3)=O)C2)=O)cnnn1C1CCCCC1 c1(C(N(CCC(=O)NC(COC)C2CC2)C2CCC2)=O)cccc(O)n1 CCC(CC(=O)N1CC(C(=O)N(CC(C)O)C(C)C)C(C(C)C)C1)C(F)F N1(C(C#CC(C)C)=O)CCC2(CCCC2NC(c2cc(O)cc(F)c2)=O)C1 N1(C(=O)CN2CCOCC2)CCN(C(C2CCCC3CC23)=O)CC1 c1(CNC(C2CCC(C)N2C(=O)COc2ccsn2)=O)ccnc(F)c1F c1(C(N2CC(CNC(C3CC4(CCC4)C3)=O)OCC2)=O)ccc2ncsc2c1 Cc1cccc2cc(C(=O)NC(CO)CCCCNC(=O)CCC#N)sc12 C1(C(c2cnsc2)NC(=O)Cc2cccc(Cl)c2)CCS(=O)(=O)C1 C(=O)(C(C1CC1)N(C(=O)CCn1cnnn1)C)N(CCCC)CCCO N1(C(c2nc(C)sc2)=O)CCC2CCCN(C(c3ccc4oncc4c3)=O)C2C1 C(CCO)(C(=O)NCC1CCN(C(c2cnccc2SC2CCCC2)=O)C1)N(C)C Cc1ccc2c(N(c3cnccc3C)CCC(C)C)ncnc2c1 c1(CNC(C2(OC)CCC2)=O)ccccc1CNC(c1n[nH]c(C)n1)=O c1(C(C)(C)C)cccc(C(=O)NCC2C=CC(NC(C3CCCN3N=O)=O)C2)n1 N1(C(C(c2c(C)cccc2)(F)F)=O)CC(NC(c2sccc2F)=O)C2CC2C1 c1(C(N2CC(CC)C(NC(=O)C(C)(CC)OC)CC2)=O)ccc2c(ccn2C)c1 c1(NC(CCCC)C)ccc(S(=O)(=O)N(C2CC=CCC2)C)cn1 C#CCC(CC#C)C(=O)NCC(CC=C)NC(=O)COc1ccc(F)cc1F C1(O)(CNC(c2c(C)cncc2)=O)CCCN(C(C2CC23CC(C)(C)C3)=O)CC1 CC(C(CO)NC(C1CC1c1ccccc1)=O)NC(=O)C(C)(C)N(C)C C1(C)(CCNC(C2(OC)CCSC2)=O)CCN(C(c2cccnc2)=O)C1 N1(C(CCCOC(C)C)=O)CC(NC(=O)CC2=CCOCC2)C2CCCC12 C#CCC(C)(C(=O)NCc1cc(F)ccc1C)NC(=O)C=CCOC C1(NC(CC2C(=O)NC(=N)S2)=O)COC2(C1)CN(C(C1CCS(=O)(=O)N1)=O)C2 C#CCCC(C(=O)Nc1cccc(C)c1)NC(C1C(C)(C)C1(F)F)=O N1(C(c2c(C)snn2)=O)CCC(CCNC(c2ccsc2C#N)=O)CC1C Cc1ncccc1C(N1CC(NC(=O)C(c2cccnc2)C)C1)=O C(=O)(CC(CN(C)C)C(F)F)NC(c1ccccc1)CNC(C(COC)OC)=O C1(C(=O)NC(CCC)C2CCC2)CCCN(C(=O)CNC(=O)OC)CC1 C(CCC(=O)NC(C)CCNC(C1(C(C)(C)C)CCCC1)=O)OC(C)C C1(CNC(CCOC(C)=O)=O)CN(C(=O)COc2ccc(C#N)cc2)CCC1C N1(C(C(c2cccs2)SC)=O)CCN(C(C2(C)CCCCC2)=O)C2(CC2)C1 C1(NC(c2cn(-c3ncccn3)cn2)=O)CCN(C(=O)Cc2ccc(Cl)s2)C1 c1(CCC)cc(C(=O)NC(C)(C)CNC(=O)Cc2ccc(Cl)cn2)ccn1 CN1CCn2nc(C(=O)NCC(F)CNC(C3(n4cccn4)CC3)=O)cc2C1 c1(C(N2CCC(NC(C3CN(C)C(=O)C3)=O)C(F)C2)=O)nnc2n1CCCC2 N1(C(c2c(C(C)C)cnn2C)=O)CCC(NC(=O)Cc2ccsn2)CC(C)(C)C1 CC(C)C(C)(C)C(=O)NCCN(C(=O)C=Cc1cn[nH]c1)C c1(C(=O)NCC(CNC(C2(C(C)C)CC2)=O)F)ccc2occc2c1 C1(C(N2C(CNC(CC3(C)CC3)=O)CC3(CC3)C2)=O)CC2CCCC(C1)C2 N1(C(C(C)OCCN(C)C)=O)CCOC(CCNC(C2CCC3CC23)=O)C1 c1(C(=O)NC2CN(C(CCCC(CC)(C)C)=O)CC2C)cc2ccc(Cl)cc2s1 C(=O)(CCCCC1CC1)NC(C1CC=CCC1)C(=O)NCC1(OC)CCC1.C1CC1 C(=O)(C(O)C(F)(F)F)NC(C1CC=CCC1)C(=O)N(CCC(C)O)C CC(C)CC(CN=c1[nH]c2ccc(Cl)cc2s1)NC(=O)CCN1CCCCCC1 C1C(C)(C)C(=O)N1.C12(C(=O)NCC(CO)NC(=O)OC(C)(C)C)CCC(CC1)O2 Cc1c(C(N2CCC(NC(c3cccc(F)c3)=O)C(F)C2)=O)ccc2c1CCC2 c1(C(=O)NCCOCCNC(C2CCC(N=[N+]=[N-])C2)=O)cc2c(cn1)CCCC2 C1C(CC(F)(F)F)NC(=O)N1.C1(C2CC2)(COC(C(C)C)=O)CCCO1.C(C)(C)(C)O Cc1cccc(C(N2CC(CC(C)NC(=O)C(C)CN(C)C)C2)=O)c1C#N C1(CNC(CC=CCCCCC)=O)CCCN(C2CCN(CCCC)C2=O)C1 C#Cc1ccc(F)c(C(=O)NC2CN(C(C3(C(N)=O)CC3)=O)CC2O)c1 C=CC(CC)CC(=O)NC1(CCOC)CCN(C(C2CCN(C)C2C)=O)CC1 C1(CNC2(C)CC2(F)F)CCCCC1n1cc(Cn2ccsc2=O)nn1 N1(C(C(C#C)(C)C)=O)CCCC2(CCC(NC(c3cncn3C3CC3)=O)C2)C1 c1(COC(CNC(C2C(c3n(CC)ccn3)OCC2)=O)=O)cc(SC)ccc1O CCCCC(CC)C(=O)NC(CNC(=O)C=CCOC)C1CCC1 c1(CC(=O)NCC2CCCN(C(=O)CCc3nccs3)C2)coc2ccccc12 CCCCC(CC(=O)NC1CCC(=O)NC1)NC(=O)Cn1ccc(C)c1 c1(SC)ccc(C=CC(N2CC(NC(=O)CC(C)(C)C)CC(F)C2)=O)cc1 C1(OC)CCN(C(C2C3CCCC3CN2C(c2cc(C)nn2C)=O)=O)CC1(C)C CC1CN(C)CC1NC(=O)NCc1cccc(C2COC2)c1 c1(C(N2CCC(C)(CNC(c3n(CC)ncn3)=O)C2)=O)cc(C(C)C)nc(O)c1 CC(C)(CC(=O)NCC1(C2CC2)CCN(C(C2(F)CCC2)=O)C1)C(F)(F)F C1(NC(CC2N(C)CC=CC2)=O)CC=C(C(=O)NCCn2cccn2)C1 C1(C(N2CC(O)(CCNC(=O)C(F)n3ccnc3)C2)=O)CC2C(C1)C2(F)F c1(OC)ccc(CS(C)(=O)=O)cc1C(N1CCCC(C(C)O)C1)=O CCC(CC(C)C)C(=O)NC1(C2CN(C(c3cc(C)n(C4CC4)c3C)=O)C2)CC1 C=C(C)CC(C(=O)OCC)NC(=O)CN1CCN(C(C2CCCO2)=O)CC1 N1(C(C2C(C)C2)=O)CCC(C2CCN(C(c3ccc([N+](=O)[O-])n3C)=O)C2)CC1 CCC(C(=O)N1CCC(NC(=O)Cc2c(C)n[nH]c2C)C(CO)C1)C(C)(F)F C(CC(C(=O)N1CC(N2CCOC2=O)C1)NC(=O)C1=NOCC1)N(C)C c1(C(=O)OC)ccc2nc(NC(CC3CCOC3)CO)cn2c1 c1(C(=O)NC2CCCC(N(C(CSCC=C)=O)C)C2)c(C)cc(OC)cc1F C=CC(C)(CCOC)C(=O)N(C(CNC(=O)CCCCO)Cc1ccccc1)C C1(CC(=O)NCC2N(C(CCc3scc(C)n3)=O)CCCC2)CCn2cncc2C1 C(C(F)C(=O)NC1(C)CN(C(N)=O)C1)C1CN(C(C(N2CCCCC2)C)=O)C1 N1(C(CC(CCC)(C)C)=O)CCN(C(C2CC2(C)C)=O)C2CCCC12 c1(NCc2ncc(C)c(OCC)c2C)ncc2c(n1)CCC(C(=O)O)C2 C(=O)(C1COc2ccccc21)N(CCNC(c1ncoc1C(F)F)=O)CC1CC1 C#CCC(C(=O)NCCC(O)CCO)NC(c1cnncc1O)=O N1(C(c2cc(C(C)(C)C)sc2)=O)CC(F)CC1C(N1CCC(C(N)=O)C1)=O C1(OCCNC(c2nccs2)=O)CCN(C(=O)CNC2(c3ccno3)CC2)CC1 N1(C(C)=O)CCCC(C(N2CCOCC2c2cccs2)=O)C1 c1(-c2nc(C(CC)C)nn2C(C)C(C)C)ccc(Cl)cc1OC C1(C(NC(C(=O)Nc2scc(C3(C#N)CC3)n2)=O)C2CC2)CC2(CCNCC2)C(=O)O1 CCC1=NOC(CC(=O)c2nnnn2CC)C1.C1(NC(=O)CC(Cl)Cl)CC12CC(N)C2 Cc1cc(C(=O)NC(C2CN(C(C3CC(CF)C3)=O)C2)C)cc(C)c1 N1(C(CC(C)(C2CCC2)N(C)C)=O)CCC(NC(c2cc(=O)n(C)o2)=O)C(O)C1 c1(C(N2CC3C(NC(c4c(C)snn4)=O)(CC3)C2)=O)cccc(F)c1C#N c1(C(c2nnnn2C2CCOC2)NCC(CC)(CC)CC)cc2ccccc2o1 c1(OC)cc(Br)c(CNCc2ccsc2Cl)cc1OC C(=O)(C(N)C[Si](C)(C)C)NC(C1CCN(C(C)C)C1)=O c1(C(=O)NC2CCC(c3cn(CCS(CC)(=O)=O)nn3)CC2)csc2nccn12 C(=O)(C1CCc2ccc(OC)cc21)NCC1(NC(C(CC=CC)C)=O)CCCC1 S(=O)(=O)(c1ccc(=NCCOC)[nH]c1)N(CCOC)CC1(F)CC(NC(C)=O)C1 C(c1ccc(F)cc1)=CC(C1N(CC(c2ncn(C)c2)=O)CCC1)=O N1(c2c(C(=O)OC)cc(C)cn2)CCC(F)(F)C(NC(=O)CCCC2CCC2)C1 c1(CCNC(=O)NC(C)(C)CNC(=O)OC(C)(C)C)c(F)cc(Cl)cc1F Cc1cc2cc(C(=O)NC3CCCN(C(C4CC5(CC5)CO4)=O)C3)ccc2cn1 Cc1nc(C2CCCOC2)sc1C(=O)NCC1CC2CC2N1C(=O)CC1CCC1 Cc1ccc(NCC2CCC(NC(c3cn(C(C)C)cn3)=O)CC2)c([N+](=O)[O-])c1 c1(OC(CN(CCC)CCC#N)=O)cc(OC)cc(C(F)(F)F)c1 N1(C(CN(CCCCCC)C)=O)CCCCC1C(=O)Nc1ccccc1C c1(C(C(=O)N(CCN(C(C(CSC)C)=O)C)C)C)cccc(Br)n1 C(COC(C)C)(C(=O)NC(CNC(C12CC(CO1)C2)=O)CO)NC(C)=O c1(C(=O)NCC2(NC(COCC(=C)C)=O)CCCC2)cc(Cl)c2n[nH]cc2c1 C1(C2C(NC(CCC=C)=O)CCO2)CCN(C(C2CC2c2cnn(C)c2)=O)CC1 c1(C(N2CC(CO)CC(OCCOC)C2)=O)ccc2cc[nH]c2c1F c1(C2C(C(N3CCC(F)(CNC(C(CCC)C)=O)C3)=O)C2)ccc(C#N)cc1 c1(C(=O)NC2CN(C(CN(C)CC)=O)CC2F)cc2cc(Cl)ccc2[nH]1 c1(C(=O)NCC(C)CNC(=O)C(F)CC2CC2)nc[nH]c2nccc1-2 CCC(CC1CCCC1)C(=O)NCC(=O)N(CCn1cccn1)Cc1ccccc1 C1(SC)CC(C)(C)CCO1.c1(C2(C)CN2)nnnn1C1CCC1.C(C)OCCOC N1(C(=O)CSCC2CCCO2)CC2(CCC2)CC1CNC(C1CCC=CCC1)=O C1(C(N2CCC(C(CO)NC(=O)COCC(F)(F)F)CC2)=O)CC2(CCC2)CO1 c1(OC)ccc(Cl)c(CNCC23CC2CN(C(c2cc(O)ccc2F)=O)C3)c1 C1(CNC(C(C)NC=O)=O)CN(C(=O)Cc2cnnn2C)CC1N(C)C C(CCC(C)NC(=O)C(C)C#N)NC(C1C(C)C1C)=O CN1N=C(CC(=O)NC2(CNC(C3CCCN3C(=O)C(F)(F)F)=O)CC2)CC1=O C1(C(C)NC(CSCCC=C)=O)CCCCN1C(=O)CNC(c1ccncc1)=O c1(CC)ccc(F)c(C(=O)NCCCCCNC(C2CCCC(O)C2)=O)c1F C1(CCNC(c2cnc[nH]2)=O)COCCN1C(=O)COC1CC(F)(F)C1 C(=O)(C1=CCC(C)(C)CC1)NC(C1CCN(C(C2CCCC2)=O)CC1)C CC1(C)CC(C(=O)NCC(CC(F)(F)F)NC(c2ncccn2)=O)CC(C)(C)C1 N1(C(c2cc(C)ns2)=O)CCC2CC(C1)CN(C(C1CC1C1CC1)=O)C2 CC1(CCCc2ncn(-c3ccccc3)n2)CCN(C(=O)NC23CCC(C2)C3)C1 C(=O)(C1=NOCC1)NC1CCC(NC(c2c(OCC)scc2)=O)C1 CCCCCCC(=O)NCCOC1CN(C(c2cc(C)ccc2Cl)=O)C1 C1(NC(C2(C)CCCCC2)=O)C2CCN(C(c3ccc(Cl)c(C#N)c3)=O)CCC12 CC1CC=C(C(=O)NCC2C(CNC(c3cccc4nc[nH]c34)=O)C2(F)F)CC1 C(C(C)(CCO)NC(c1ccc(CNC(=O)Cn2cc(CO)nn2)cn1)=O)OC CCC(C)(C)C(O)C(=O)NC1CN(C(=O)CCc2csc(Br)c2)CC1C C(=O)(C(F)(F)C(C)(C)O)NCCOCCN(C)C(C1CC2CCC1O2)=O c1(C(=O)NC2C(CCC)CN(C(=O)C#CC3CC3)C2)nc[nH]c2ncnc1-2 C(=O)(N=c1cc(Cl)nc(O)[nH]1)c1c(CC)nc(-c2ccccc2)[nH]1 c1(OC)nccnc1C(=O)NCC1CC(C(N2CCC(C(C)OC)C2)=O)C1 c1(C(N2CCOCC(NC(C3C(C)=CCS3)=O)C2)=O)ccc(C)c2ncccc12 c1(CNC(=O)NCC2(c3cccs3)CC2)ccc(C2CCC23CCC3)cc1 C1(C(=O)NCc2ocnc2C(N2CCC3CCC23)=O)(OC)CC(C)(C)C1 CCC(C)(CNC(C1CC(C)(F)C1)=O)C(=O)Nc1cncnc1OC O=S1CCOC(CSc2cnn(Cc3ccccc3)c2)C1 c1(C(N2C(CC(=O)NC(C)CC3CCCCC3)CCC2)=O)ccc(O)nn1 C1(C(C)NC(C2(c3ccccc3F)CCC2)=O)CN(C(=O)OC(C)(C)C)CCO1 c1(C(=O)NC(C2CC(NC(C3CC4(CCCO4)C3)=O)C2)C)cnn2c1CCC2 c1(NC(C2N(C(CC)=O)CC(F)C2)=O)ccc(O)cc1C(F)(F)F N1(CC(Cn2c(C)ncc2)C)CC(N2CCN(C(=O)OC(C)(C)C)CC2)C(C)C1 N1(CC(=O)NC2C3(CN(C(C(C)N4CCC4)=O)C3)SCC2)C(=O)CC(C)(C)C1=O CCCCC(C(=O)N1CCC1CNC(C1CCC2(CCC2)C1)=O)NC(N)=O S(=O)(=O)(c1ccc(NCC2=CCCC2)cc1Br)NCc1cc(OC)c(F)nc1 C1(c2n(C3C(F)(F)CCC3)nnn2)(NC2COC2)CCC(C(F)F)CC1 C12(CNC(C(C)SCCCC)=O)CC(CN1C(c1ccn(C(C)C)n1)=O)C2 C1(NC(COCCC(C)C)=O)CCC2(CCCN(C(=O)CC(F)(F)C(C)C)C2)C1 C(=O)(C(C)(C)N=[N+]=[N-])OC(C1CCCC(CN=[N+]=[N-])C1)C C1(C)(C(N(CCCCCNC(C2(CC)CC2)=O)C)=O)CCSCC1 CN1N=CC(CC(N2CC(NC(=O)Cn3ncc(Br)n3)C(O)C2)=O)C1=O C(=O)(C1=Cc2cc(F)ccc2OC1)N(CC(C)NC(C(CC)C(C)O)=O)C Cc1onc(CC(N2CCCC2(C)CNC(=O)CSCC(C)C)=O)c1C#N C1(C)(CC(=O)NCCC(C)NC(=O)C(n2cc(Cl)cn2)C)CCOCC1 C1(C(=O)NCCCN(C(=O)CC2(C3CC3)CC2)C)CCN(c2ncccn2)C1 C12(CNC(CN(C)S(N)(=O)=O)=O)CCC(NC(=O)CC3CN4CCC3CC4)(CO1)C2 CC1CN(C(=O)CCC2CCN(C)C2)CC1NC(C1CN(CC(F)(F)F)C1)=O CCC(CC)C(F)C(=O)NCC(CCOC)NC(=O)CSCC(F)F c1(NCC(COC)C)nccc(=NCC(OC)c2ccccc2)[nH]1 N1(c2ccc(NC(=O)OC)cc2C(N)=O)CC(C(=O)OC(C)(C)C)C(C)CC1C C1(C)(CNC(Cc2scc(C)c2)=O)CN(C(=O)CCSC2CCCC2)C(C)(C)C1 Cc1nc(COC(C2CC2Cc2ccccc2)=O)sc1C c1(C(N2C(C(=O)NCc3ccccc3)CCCC2)=O)ccc2cc(Cl)ccc2n1 CCC(C)CC(=O)NC1CC(CCNC(c2cn(CCO)nc2C)=O)C1 Cn1ccc(C=CC(N2CC(OCC(=O)NCC(C)(C)CCO)C2)=O)c1 c1(C(=O)Nc2ccc(C(=O)NC(C)C)cc2)n[nH]c2c(-c3cnoc3)cccc12 C1(C(N(CCOCCN(C(=O)CNC=O)C)C)=O)CCCC2(CC2)C1 C1(NC(c2c(SC)cc(C)cc2)=O)CC2CCC(C1)N2C(=O)C(C)CCN(C)C N1(C(=O)Cc2cc(F)c(Cl)cc2Br)CC2CC(C2)c2ccc(Br)cc21 N1(C(c2n(CC)ccn2)=O)CCC2CCC12CNC(=O)CCCCC#N Cc1cc(C=CC(=O)NC2(N3CCNC3=O)CC2)ccc1Br c1(C(=O)NCC2(F)CC(NC(c3c(CC)cccn3)=O)C2)cc(Cl)ccc1O Cc1ccc(NC(C2CC3CC3N2Cc2cc(C(C)C)no2)=O)c(C(F)(F)F)c1 c1(CNC(=O)Nc2c(C)nc(C(=O)OCC#C)s2)cccc(OC(C)(C)C)c1 N1(C(C(C(CC)C)C)=O)CC(O)(C2(CNC(=O)Cc3cc(OC)ccc3Cl)CC2)C1 C1(CNC(C(C)OC2COC2)=O)CC(O)C(O)CC1C(=O)NCCCOC(=N)O C1(C(=O)NC(CNC(c2nc(C(=O)OC)oc2)=O)C2CC2)CCC(CO)CC1 Cc1ccc(CC(N2CCN(C(C3CCCCCC3)=O)C3CC23)=O)cc1[N+](=O)[O-] c1(SC)ccccc1C(=O)NC1(C)CN(C(=O)CN(CC(C)(C)C)C)C1 Cc1nn(C)cc1C(=O)NCC(C)(C)CNC(=O)C(F)CC1CCOC1 N1(C(=O)CC2CCCCS2)CCCC2C1CCN2C(=O)CN1CCC(F)CC1 CN1CCC(CC(N2CC(O)CC2C(N2CCC(CF)C2)=O)=O)CC1 Nc1cc(C(=O)NC2CCC(CNC(C3CCCC4CC34)=O)CC2)ccc1Cl N1(C(CC(C)(C)C2CC2)=O)CC2(CC2)CC1CNC(=O)CN1CCCCS1(=O)=O C1(CC(N2CC(CC(C)NC(=O)Cc3cncn3C3CC3)C2)=O)CCC=CCC1 C1(NC(=O)COc2cncc(Cl)n2)CN(C(C2CC(F)(F)C2)=O)C2(CCCC2)C1 N1(CC(=O)NC2CN(C(CNS(N)(=O)=O)=O)CC2O)CC(=O)Nc2ccccc21 c1(C(N2CC(C)C(NC(C3(S(N)(=O)=O)CCC3)=O)C2)=O)ccc2ccccc2n1 N1(C(CCNC(=O)OCC)=O)CC(C)CCC1C(=O)N(C1CCCC1C)C C1(F)(C(N(C(C)CCO)C)=O)CCCN(C(=O)CC#N)C1 c1(C(N2CCC(C)(CNC(CC=C=C)=O)C2)=O)ncc(N)cc1Cl C1(c2cc(CNC(C=NOC)=O)on2)CCN(C(c2ncccc2OC)=O)CC1 CCC(CCC(=O)N1CCC(C)(CCO)CC1)NC(=O)Cc1cscn1 c1(NC(c2csc(I)c2)=O)c(F)ccc(Cl)c1CO c1(C(N2CCC3(NC(c4ccc(Br)s4)=O)C(C2)C3)=O)ccc2c(n1)CCC2 c1(CC(=O)NCC2(F)CC(CNC(C(C)NC=O)=O)C2)ccccc1Cl C(=O)(CC(C(F)F)n1ccnc1)NC1CC(C)(NC(c2c(C)nn[nH]2)=O)C1 c1(N2CCC(C(C)=O)CC2)ccnc2cc(I)ccc12 Cc1cc(C(=O)NCC(CNC(c2csc(Cl)c2)=O)C(F)(F)F)ncc1C#N CC1Cc2ccc(Br)cc2CN1C(=O)Nc1c[nH]c2cccc(Br)c12 CC1CCN(C(c2cc(Cl)ns2)=O)CC1CNC(c1ccns1)=O C1(CNC(c2cnn(C)c2C(F)(F)F)=O)CC2CCC1N2C(=O)CCCC#N N1(C(C2(NC(C)=O)CCSC2)=O)C2CCC(C2)C1C(N1CCN(C(C)C)CC1)=O c1(C(N2CCC(C)C(NC(=O)CNS(C)(=O)=O)C2)=O)cc(C#N)c(F)cc1F N1(C(CC(CC)OC)=O)CC(C(=O)NCc2cc(C)cnc2O)CCC1C C#CCC(C)(C)C(=O)NN1C(C)CC(CC(=O)NCCSc2cc(C)nn2C)C1 N1(CC(=O)NC2(COC)CCN(C(C(CCC)OC)=O)C2)C(=O)CC(C)(C)C1=O C1(OCC)(CNC(C2(F)CC(C(=O)OC)C2)=O)CN(C(C2(C)CCCO2)=O)C1 C12(C(N(C(CN(C(C(C)N(N3CCCC3)C)=O)C)C)C)=O)COCC1C2 c1(C(N(CC(C)C)CC#C)=O)cncc(CNC(c2scnc2Cl)=O)c1 c1(NC(CSC)Cc2cccs2)cc(=O)n(CC(=O)O)nc1Cl CC(=O)CCCC(=O)N1CCC(C(=O)NC2CC(CF)C2)(C(C)C)C1 C(=O)(C(CCO)N(C)C)NCCn1cc(CNC(C(C)(C)OC)=O)nn1 C(=O)(CC(C)CC(C)C)N1CCC(O)(C(C)NC(C(Br)=C(C)C)=O)CC1 C(=O)(CC(C)P(C)(C)=O)NC1(CCNC(C2CC(C)=C(C)CC2)=O)CCCC1 C=CCC(F)(F)C(=O)NCCCC(C)NC(=O)Cc1csc(C(C)C)n1 c1(NC(CCOCCOCC)=O)cnc(F)cc1C(=O)Nc1cc(Cl)nc(C)n1 C1(NC(=O)CC2CC3(CCC3)C2)CCN(C(c2ncccc2Cl)=O)CC1F c1(C(=O)NCC2CN(C(c3cc(C)c(C)[nH]3)=O)C(C)C2)c(C)nc(C)n1O C(c1ccc(F)cc1)=CCC(=O)NC(CNC(c1cn(CC)nc1)=O)CC(C)C N(C1CN(C(=O)CCCC2CC2)Cc2ccccc21)C(C(C1CC1)OCC)=O Cc1cc(CNC(=O)CCCC2(N(C)C)CC2)ccc1F.C12CC(C)(C1)NC2=O N1(C(C(C)(C)C)=O)CCCCC1C(N1CCC(CNC(c2cnc(O)s2)=O)C1)=O N1(C(C(CC)OC2CCCC2)=O)CC2CCN(C(=O)CCC(=O)OC)CC12 c1(CCNC(=O)NCC2CCN(S(=O)(=O)C(F)F)C2)cccnc1 c1(C(N2CCCN(C(C(CCC)(C)C)=O)CCC2)=O)ccc2nc(=N)[nH]n2c1 C1(CC(=O)NC(c2cccs2)CC)CCN(C(c2cccc(COC)c2)=O)CC1 C1(C(=O)Nc2ccccc2)C2CCC(C2)N1C(c1cccc(F)n1)=O C1(CNC(C2(C#N)CC2)=O)CC2(CCN(C(=O)COc3ccccn3)CC2)CO1 c1(C(C)C)cc(C(=O)NC23CC(NC(=O)CC#N)(C2)C3)n[nH]1 c1(C(=O)NCC2CC(Cn3cc(C(CC(C)C)O)nn3)C2)ccc(Cl)c(F)c1 C=C=C(C)CC(=O)N1CC2CC2(NC(c2sc(Cl)cc2Cl)=O)C1 c1(N2CCC(N(C(C(C=C)O)=O)C)C2)nc(C)cc(C(F)(F)F)c1C#N c1(CNC(C2CCC(C)N(C(=O)Cc3cncn3C)C2)=O)cnc2cc[nH]c2c1 CCCCCCCCNC(=O)C(CNC(=O)C(C)COC(C)=O)OC C1(C(=O)NC2CC2)CSCN1C(=O)C(c1ccccc1)F Cc1c(F)ccc(C(=O)NC2CCN(C(c3ncccc3Cl)=O)C2C)c1C C=CC1(NC(c2ccn3ccsc23)=O)CCN(C(=O)OC(C)(C)C)C1 c1(C(N(C(CNC(C=CC=CC)=O)C)C)=O)cn(C(C)C)cc1C c1(CC(N2CCC(N(C(C3CCCCS3)=O)CC)CC2)=O)noc(C)c1C#N C(=O)(C(F)C(F)(F)F)NCC(CC)(C)NC(=O)CNC(C1CCC1)=O c1(CC)c(C(=O)NC23CC(C2)N(C(=O)Cc2sc(S)nc2C)C3)cnn1CC C1(NC(C(c2cccc(C)c2)C)=O)CCN(C(c2n[nH]c3c2COC3)=O)C12CC2 C1(C(N(CC=C)CCOC)=O)CC(=O)N(Cc2ccccn2)C1 c12ccc(nc1)CNC2=O.c1(NCC)ccc(OCC(F)(F)F)nn1 C12(C(=O)NCC(C)NC(C3(C4CCCCO4)CC3)=O)CCCN(CC1)C2 C1(CC(=O)NCC(C)OC)CC(NC(=O)CNc2cn[nH]c2)C1 N1(C(C(C(C)C)(C)C)=O)CC2CC(NC(=O)CC(C)(O)C3CC3)CC2C1 C1(C(=O)NCCCN(C(c2ccc(C3CC3)cn2)=O)CC)CCS(=O)(=O)N1 N1(C(C2C3CN(C4CC(COC)NCC4)CC32)=O)CCS(=O)C(C)C1 CC(C)C(CC(=O)N1CC(NC(=O)C(=O)N(C)C)C1)C(C)C Cc1ncc2n1CCC(C(=O)NC1CC(CNC(C3CC3C3CCCC3)=O)C1)C2 CC1CC(=O)NCC1C(=O)N(C1(C(=O)NCCC2CC(F)(F)C2)CCC1)C1CC1 C12(NC(c3csc(Cl)c3)=O)CCN(C(=O)CCCCc3ccccc3)CCC1C2 N(C1CCCc2n[nH]cc21)C(C(C(C)OC)NC(=O)C(C)CN(C)C)=O c1(CC)cc(C(N2CCOCC2C2CCOC2)C(=O)NC2CCOC2)cc(C)c1 C12COCCN1N(C)C2.C1(O)(C=O)CCOCC1.c1ccncn1 c1(C(N2CC(C)C(NC(=O)CC3CC3)C2)=O)nn(C)c(=O)c2ccccc12 C1(NC(CCc2n(C)ncc2)=O)CC2CC1N(C(C1CCC(C(F)(F)F)O1)=O)C2 N1(C(c2cnn(C(C)C)c2N)=O)CC(C)CN(C(=O)CCc2cnc[nH]2)CC1C C(=O)(C1=NOC(CN(C(c2nccs2)=O)C2CC2)C1)N1CC(N(CCOC)C)C1 c1(CC(=O)NCC2(F)CCN(C(COC)=O)C2)cccc2c(C)csc12 c1(C(=O)NC2(CO)CCN(C(c3[nH]c(CC)c(Cl)n3)=O)C2)nccc2[nH]ccc12 N1(C(CC2(C)CCN(C(C(CC=C)NC(C)=O)=O)C2)=O)CC2CC3CC2C1C3 C1(C(N2CCN(C(C3(C#N)CC(C)C3)=O)CC2)=O)(CC)CCNC1=O c1(NC(C)=O)ccccc1C(=O)NCC(N1CC(NC(=O)C(Cl)=CCl)C2CC12)=O C=C1CCC(C(=O)N(CCNC(C2CC2SCc2ccccc2)=O)CC)CC1 C1(C(=O)NCC2(CC(N)=O)CC2)(SC)CN(C(=O)CNC(C)=O)C1 c1(NC(N(CCC)Cc2ccccc2)=O)ccc(-n2cc(CO)nn2)cc1 C1(C(=O)NC2(c3ccccc3)CCOC2)(CNC(C2CC(OC)C2)=O)C=CCC1 c1(OC)cccc(CNC(=O)CNC(=S)Nc2cccc(F)c2)c1 c1(COC)ccccc1C(=O)NC1CCCCC1CNC(c1nc(O)c(C)s1)=O N1(C(c2cc(CC)c(C)s2)=O)CC(C)(CNC(C2(C)CCNC2=O)=O)CC1(C)C Cc1cc(C(=O)NC(C2CCN(C(=O)CSc3nccn3C)CC2)C)nc(O)n1 C1(NC(Cn2ncc(C)c2)=O)C(C)CN(C(c2cc3cnccc3o2)=O)CC1C Cn1ccc(CC(=O)N(C(=O)CCC2CCC(=O)C2)CCCN(C2CC(=O)C2)C)c1 C(=O)(C1c2c[nH]nc2CN1C(c1ccn(C2CC2)n1)=O)NCC(COCC)C CC1(CNC(=O)CSc2nnnn2C2CCCC2)CC(NC(C2COC(=O)C2)=O)C1 c1(C(=O)NCCCCCNC(C(CC)SC)=O)cc(F)c2ncccc2c1 C(=O)(C(C)(C)C(=O)NCCC1CC(NC(=O)Cc2nc[nH]n2)C1)NC C(=O)(CC1=NNC(=O)C1)N1CC(C2OCCN(C(CCn3ncn(C)c3=O)=O)C2)C1 c1(CC(=O)NCC(C)CN(C)C(C2CC(C)OC2C)=O)cccnc1Cl n1(CCC)cc(-c2cscc2CN(CC(C)C)C)cn1 N1(CC(=O)N(C(C)C(=O)NCC2CCCC2)CC)CCNC1=O N1(C(C2N(C(C3(C)CNC(=O)C3)=O)CC=C2)=O)CCNC(=O)CC1 c1(C(=O)NC2C(CNC(C(CSC)O)=O)CCC2)cc2ccccc2cn1 C#CCC(CC#C)C(=O)N1CCC(C)(CNC(c2cc(C)c(CC)s2)=O)C1 C1(NC(c2ccccc2Cl)CCOC)CCN(C(c2ccsc2C)=O)CC1 Cc1ccc(N)c(C(=O)NC2C=CC(CNC(c3cc4n(n3)CCO4)=O)C2)c1F C1(NC(c2c[nH]nc2[N+](=O)[O-])=O)CN(C(c2nc(Cl)cs2)=O)C2(CCOCC2)C1 c1(C(=O)NC(C(C)NC(C(CC)n2ccnc2)=O)C)c(Cl)ccc(F)c1F CC1CN(C(c2cc(Cl)cn2C)=O)CC(C)N(C(=O)CN2CCC(CO)CC2)C1 N1(CC(N2CCC(N(CCC)C(c3cnc(Cl)s3)=O)C2)=O)C(=O)CC(C)(C)C1=O O=C1CCC2CN(C(C3CC(=O)N(C(C4CC4)C4CC4)C3)=O)CC2N1 c1(COC)ccnc(C(N2CCC2CNC(=O)CN(C)C(c2cccs2)=O)=O)c1 CP(C)(=O)CN1CC(C(=O)NCCNC(=O)CCC(=O)NC(=O)NC2CC2)C1 c1(C(N(c2cncc(Cl)c2)CCN(C)C)=O)ccc(C#N)cc1F CC(C)CCCCC(=O)NCCCOCCN(C(=O)CCC1(C)CCC(=O)N1)C c1(NCC(n2ccnn2)C)ncccc1S(=O)(=O)NC(CC1CCCC1)CO C1(N(C(c2ccc(C#C)cc2)=O)CC)CC12CCN(C(=O)Cc1nc[nH]n1)CC2 c1(C(=O)NC23CC(CNC(c4ncc(F)cn4)=O)(C2)C3)cnc2nccn2c1 c1(OCC(=O)NC(C)CCN(C(=O)C(C2(O)CCCC2)F)C)cccnc1 CN1CCN(C(C2CCC(O)CN2C)=O)CC1CNC(c1ccc(F)cc1F)=O CCC(CC)CCC(=O)N1CCCC(C(C)(C)C(=O)NCC2=NOC(C)C2)C1 Cc1cc(C(=O)NCC(C)N(C)C(c2cc[nH]c2)=O)cc(Br)c1C C(=O)(C1=CCS(=O)(=O)C1)NC1CN(C(CC2CN(C)C2)=O)CC12CC2 C1(NC(=O)C=Cc2cnc[nH]2)COC2(C1)CN(C(=O)COc1ccc(Cl)cc1)C2 c1(C(=O)NC2C(C)N(C(c3cc(F)ccc3Cl)=O)CCC2)ccc2nccn2c1 c1(C(=O)NC2CC(N(C(C3C(CC)C3)=O)C)C2)cc(-c2cccs2)on1 c1(CC(N2C(C(=O)NC(COC)CO)CC2)=O)csnc1C c1(CC)nn(C)cc1C(=O)NCC(C(=O)N1CCC(OC)C1)OC.C(COC)OC C12(C(=O)NCCC3(O)CCN(C(c4nn(C)c(O)c4)=O)C3)CCC(C1)C(C)(C)O2 N12CCC(C)CC(C1)NC(=O)c1ccc(s1)CNCC2=O.C(=O)(C1CC1)OCC Cc1ncc(C(=O)NC(CCNC(C2CCCC23CCC3)=O)C(C)C)cc1C#N O=C(N=c1[nH]nc(O)s1)C1=NN(c2cccc(C(F)(F)F)c2)C2(CCC2)C1 C(=O)(C(C)(C)C(F)(F)F)NCC(CC(C)C)NC(C1CCn2nnnc2C1)=O CC1CCSCCN1C(C1CCN(C(c2cc(O)cc(=O)o2)=O)CC1O)=O N1(C(CCCN(C(=O)OC)C)=O)CCN(C(=O)CC2CN(C)CC2O)CC1CO c1(C(N(CC(F)(F)F)CC=C)=O)cn(C(F)F)nc1C(F)F C1(NC(COCCC)=O)CCN(C(=O)C(C)Cn2cccn2)C12CC2 Cc1ccc2cc(C(N3CCC(CNC(C4(C)CC4)=O)C3(C)C)=O)[nH]c2c1 N1(C(CN(C)CC)=O)CCN(C(c2cc(Cl)no2)=O)CC1c1ccccc1OC Cc1cc(O)ncc1C(N1CCC(C(=O)NC2COC3(CCC3)C2)(CO)C1)=O c1(CCC(=O)NCCC2CC(NC(C3C(C=C)CC3)=O)C2)ccc(SCC)cc1 CCCC(CCC)C(=O)NC1CC2CCC1N2C(=O)CC(C)(C)COC(C)=O c1(OC)nn(C)cc1C(=O)NC1CCC1NC(c1cncc(N)c1)=O C1(NC(c2cc(=O)cc(Cl)[nH]2)=O)CCN(C(=O)Cc2ccsn2)CC(O)C1 C=C(C)CC(C)C(=O)N(C)CC1CCCN(C(C2(C(N)=O)CC2)=O)C1 C1(CNC(CC=C(C)C)=O)OCCC1C(=O)NC(C1CCC1)C1CC1 C#CCCCCC(=O)N1CCC(F)(C(=O)NC(c2cccs2)C)CC1 N1(C(c2c(C)nc(C3CCC3)o2)=O)CCCC2CN(C(=O)C(C)CN(C)C)CC12 c1(NC(CC(C)(C)N(C(C(CC#C)C2CC2)=O)C)=O)cc(O)ccc1C C1(C(=O)NC(c2ccncc2)CC)CCN(C(c2cccn2C2CC2)=O)C1 C1(C)(CNC(CCCC(C)O)=O)CC(F)(F)CN1C(c1ncc(Cl)n1C)=O c1(C(=O)NCCCN(C(c2cc(N(C)C)ccn2)=O)CC)nc(O)c(C)s1 c1(NC(C2C(CNC(C(CCC)C#N)=O)OCC2)=O)ccn2nccc2c1 CCC(C)(C(=O)NCCN(C(=O)Cc1ccc(Cl)cc1)CC1CC1)C(F)F c1(NCC2(COC)CCNCC2)cnc2n1CCCC2 C(c1ccc(F)nc1)=CC(N1C(C)CC(NC(=O)CCc2ccc(Cl)nc2)C1)=O N1(C(COC(CC(C)(C)CC2CCCCC2)=O)=O)Cc2ccccc2C1 Cc1cnc(NC(c2ccccc2)=O)nc1.c12cccc(c1)NCC2=O c1(CCNC(C(C2CC=CCC2)NC(CC(C)C)=O)=O)cccnc1O C1(CNC(c2cc(C)c(C)o2)=O)N(C(c2cncc(Cl)c2)=O)CCC1(C)C c1(C(=O)NCCC2(NC(c3ccn(CCCC)n3)=O)CC2)ccnc(OC)c1 C12(C(=O)N(C(C)C3CC3)C)C(NC(C3CCC3C#N)=O)C3CC1C2C3 N1(C(C2C(C)(C)C2)=O)CCCC2(CCN(C(=O)CN3CCS(=O)CC3)CC2)C1 C(=O)(C(C(C)O)NC(C1CCCC1CNC(C1CCCC(=O)C1)=O)=O)OC O(S(=O)(=O)c1c(C)nn2cccnc12)c1cc(C)c(Br)cc1 n1(CC)ccc(CC(=O)N(C)CCNC(=O)C(COCc2ccccc2)OC)n1 c1(OC)ccc(-c2nc(C)c(-c3nccn3Cc3cccc(F)c3)s2)cc1OC C1(NC(c2cc(-c3ccc(Cl)cc3)[nH]n2)=O)CC12CCN(C(C1CC1F)=O)CC2 C1(N(CCC)CC2CCCS2)CC(NC(=O)CCCc2ccccc2)C(O)C1 N1(C(C2(C(C)=O)CC2)=O)CCc2ccccc2C(NC(c2ccn(C)c2C)=O)C1 c1(C(N2C(CNC(C=C(C)C)=O)CCC2)=O)cc([N+](=O)[O-])ccc1Cl N1(C(C(C2CCCC2)OCC)=O)CCC2(CCCN2C(c2ccc(C#N)o2)=O)C1 N1(C(c2cc(CC)sn2)=O)CCCC(C)(C)C1CNC(c1cc(C)on1)=O c1(CN2C(CNC(C3C(C)OCCC3)=O)CCC2)ccc2c(c1)CCC2 c1(C(=O)NC2C(C)(C)CN(C(=O)C(O)P(C)(C)=O)CC2)cccc2cnccc12 c12cncc(c1)CNC(=O)N2.N1(C(CC)C)CCC(Cn2ccnn2)C1 C1(NC(C(N2CCNC2=O)C)=O)CCOC12CCN(C(c1ccc(Cl)s1)=O)CC2 C(=O)(CS(=O)(=O)c1ccc(C(=O)NCCCNC(C2CCOCC2)=O)cc1)NC C1(NC(CCCc2ccc(C)cc2)=O)CN(C(C2CC2CF)=O)CC2(CCC2)C1 CC1N(C(c2conc2CNC(=O)C=Cc2ccsc2)=O)CCOC1(C)C C1(C(=O)NCCCC)CCC(CNC(=O)COC2CCCC2)C1 N1(C(c2ccc(C)cc2Cl)=O)C2CCC1CN(C(c1ccn(CCO)c1C)=O)C2 C1(C(=C)F)(CC(=O)NC)CCC1.C(CCN1C(=O)CN(C)CC1)OC=C c1(CC(=O)NCC2(OCC)CN(C(CS(CC)=O)=O)C2)ccc(Cl)c(C)c1 c1(OC)ccc(CC(=O)NCC2CCCCN2C(c2cccnn2)=O)c(OC)c1 c1(C(=O)NCC2(CCNC(C(C)OCC#C)=O)CC2)c(F)ccc(OC)c1N C1(CNC(c2csc(Br)n2)=O)CC2CN(C(C3COC4(CCC4)C3)=O)CC12 N1(C(CCN(C)CC)=O)CCCN(C(c2cc(N3CCCC3)ccn2)=O)CC1C c1(C(=O)NCC(C)(C)CNC(=O)C2=CCCOC2)c(C(F)F)nc2ccccn12 CCC(C)(C)C(=O)C(=O)N1CC(F)(F)CC1(C)CNC(=O)Cn1ccnc1C C1(NC(CCC2C(C)C2)=O)C2CC1CN(C(C1(O)CCOCC1)=O)C2 C(N=c1[nH]c(Cl)nc2c1SCC2)C1CC(NC(=O)CS(=O)(=O)C2CC2)C1 C1(COC)CN(C(C2CCC(C)C2)C(=O)NCC2CCCO2)CCO1 CC(C)(CF)C(=O)N1CCC(N2CCN(C(c3cnc(=N)[nH]c3)=O)CC2)C1 c1(C(N(C)CC2N(C(CC(C)F)=O)CCC2)=O)cnnc(O)c1 CS(=O)(=O)CCNCC(N1CCCC1CO)=O N1(C(C(=O)NCCOC)=O)CC2CC2(NC(=O)Cc2csc(CCC(F)(F)F)n2)C1 C1(C2CCOCC2)(NC(C2N(C(C(C(=O)OC)C)=O)CSC2)=O)CC1 C1(NC(=O)C2CC2)CC2(CCN(C(C3C(C4CC4)C3(F)F)=O)CC2)C1 Cc1cc(N2CCN(CCCNC(c3csc(C4CC4)n3)=O)CC2)nc(CO)n1 c1(CC#N)ccc(OCC(N2CC(N3CCN(C(=O)CCF)CC3)C2)=O)cc1 c1(OCC)ccc(CCC(=O)NCC(C2CC2)NC(C2(C3CCC3)CC2)=O)cc1 Cc1nc(-c2ccccc2)oc1C(=O)NC(c1cccnc1)CN1CCCC1 c1(C(N2CC(OCCNC(c3csc(CO)c3)=O)C2)=O)csc(-c2nc[nH]n2)n1 c1(-c2nnc(N(C3CCCC3)CC)n2C2C(C)CCCC2C)cc2cnccc2o1 C=CCC(C)(C)C(=O)N1CC(C(C)(C)O)(CNC(C2CCC(=O)N2C2CC2)=O)C1 C12(Nc3snc(CCOC)n3)CCCC1CN(C(C1CCC(=O)N1)=O)C2 C(=O)(C1CCc2cc(F)ccc21)NCCCN(C(c1cnc(CCCC)s1)=O)C C#Cc1cncc(C(N2CC(C)CC(O)C2)C(=O)NC2CCOC2)c1 CC1(C)CC2CC(C)(CN2C(C(=O)NCCC2CC2)c2cnc[nH]2)C1 c1(C(=O)NC2CC(C)(CC)C2)cncc(C(=O)NC(C2CN(C(=O)NC)C2)=O)c1 N1(C(CSCCOC)=O)CC(NC(c2nccn3nccc23)=O)CC2(CCC2)C1 Cc1cc(C)n(C(C)C(N2CC(NC(c3ccnc(C4CC4)n3)=O)C(O)C2)=O)n1 Cc1oc(CO)cc1C(=O)NCc1cnn(C)c1C(=O)NCCC1CC1C C(CCCCNC(=O)C(N)=O)N(C(=O)COC1(c2ccccc2)CC1)C c1(C(=O)NC(CN(C(C(C)(CO)OC)=O)C)C)cc2c(nc1O)CC(C)(C)CC2 C(C(C)C(=O)NC(C)(CNC(=O)C=CC(=O)NC1CC1)CC)OCC N1(c2ncc(OC)cn2)CCC(F)(F)C(NS(=O)(=O)CCN2CCCCC2)C1 C(=O)(C(F)(F)c1csc(Cl)n1)NC(C)C(C1CCCCC1)NC(=O)C=CC1CC1 c1(CC)ccc2c(c1)OCO2.C(C(=O)OC(C)(C)C)(c1nccs1)N(C)C=O c1(C(C(=O)NCCCC)N(CC(F)(F)F)CC2CC2C)ccc(C(=O)OC)s1 CC(C)(CS(C)(=O)=O)C(=O)NCC1CCC1NC(c1ccnc2ncnn12)=O C1(NC(C(C)c2ccco2)=O)CC2(CCN(C(=O)CC(C)(C)F)CC2)C1 CCCC(CC)C(=O)NC(Cn1cncn1)C(=O)NCCN1CCCC1=O C1(C(=O)Nc2c(CC)nn(C)c2)CCN(C(=O)CC2=CCN(C)CC2)O1 C1(NC(c2c(F)ncc(OC)c2)=O)CCC2(CC1)CN(C(=O)CC(C)F)CCO2 CCCCCCCCCCC(=O)NC1(C)CCN(C(C2CC(C)CO2)=O)CC1 N#Cc1cnc(NC(C2CC3CC3N2C(c2c(Cl)cccc2I)=O)=O)c(Cl)c1 N1(C(CCOCCOC)=O)CCC2(CCN(C(=O)C(CC)C(=O)OC)C2)C1 c1(C(=O)NC2CC3N(C(CC(=O)OC)=O)C(CC3)C2)ccc(Br)c([N+](=O)[O-])c1 c1(CC(=O)NCC2(OC)CN(C(=O)CC3CCC(C#N)C3)C2)cccc(Br)c1 c1(NC(c2c(C)nsc2)c2nnnn2CC(F)F)cc(C)c2nccn2c1 C1(C)(C(N(C)CC2CCCN(C)C2)=O)CC12CCN(C(c1cc[nH]n1)=O)CC2 C1(C(=O)NCCOCCOCC)CCCC1NC(c1csc(C2CC2)n1)=O N1(C(COCC=C)=O)CCCC(C)C1CNC(=O)CCc1cn(C)nn1 c1(C(=O)NCC2CCCN(C(C(CCSC)O)=O)CC2)n[nH]c2c1CCSC2 C1(OC)CCC(c2nnnn2C2CC2)(NCC2(c3cc(F)ccc3F)CC2)CC1 C1(CNC(CC2C(C)=NOC2=O)=O)CN(C(=O)CC(=O)NC2CC2)CCC1(C)C c1(CN(C(c2c(C)nc[nH]2)C(=O)NC2CCOCC2)C)cccc(C(C)(C)C)c1 N1(C(c2cc(OCC)no2)=O)CCN(C(=O)CC2CC(OC)C2)CC1CO C1(CNC(C(CN(C)C)(C)C)=O)CCC(C)(C)CN1C(C1CC(F)C1)=O CC(C)C1C(=O)N1.c1(C(=O)OCCCCCc2ccccc2)ccc(N)cc1 C1(NC(C(CCC)OCC)=O)CCC2CC1CN2C(c1nncn1C)=O c1(C(N2CC(C)C(CNC(C3(C)CCCCO3)=O)C2)=O)ccc2c(c1)CCCC2 c1(NC(=O)NC(C)C(=O)OC(C)C)ccn2c1CNCC2 N1(C(C2CCCC23CCC3)=O)CC2CN(C(C3CCOC3)=O)CC2C1 N1(C(C=CC=CC)=O)CC=CC(NC(=O)CNC(=O)C(F)(F)F)C1 Cc1ccc(F)c(S(=O)(=O)N2CC3CCC(C2)C3C(=O)Nc2cc(F)ccn2)c1 N1(C(c2c(CC)occ2)=O)CCN(C(c2cnn(C3COC3)c2)=O)CC12CC2 CN(CC1CCCN(CC(C)(C)O)C1)N1CC(S(C)(=O)=O)CCC1(C)C c1(C(=O)NC(CC2CN(C(C(=O)NCC)=O)C2)C)cnc(CC2CC2)nc1 C1(NC(C(c2scc(C)n2)C)=O)CCCC12CN(C(=O)Cc1cnc(C)[nH]1)C2 Cn1nc(C(F)(F)F)cc1C(=O)NCC1CN(C(=O)CCOC2CCC2)CCO1 c1(C(=O)NC2(CCNC(=O)CSC3CC3)CCCC2)ccc(F)c(C(F)F)c1 N1(C(C(C)(C)C2CC2)=O)CCC2CC(NC(c3cccc[n+]3[O-])=O)CCC2C1 CC1(C)OCCOC1CC(=O)NC1CC(F)CN(C(=O)C2=CCCC2)C1 c1(OC)cc(CC(=O)N(CCC(C)NC(=O)C(C)NC(=O)C(C)(C)C)C)ccn1 c1(C(N(C2CCN(C(C(CC3CCC3)NC(C)=O)=O)C2)C)=O)cnc(=N)[nH]c1 C1(CNC(C2CCC2)=O)CN(C(=O)CC2CC3(CC3)C2)CC(C(F)(F)F)O1 c1(OC)ccc(C(O)C(C)N(C(=O)C=CC=C(C)C)C2CC2)cc1 C1(=O)C(C(C)C)C(=O)N1C1(C(C)O)CC1.c1(C2CCCO2)ccncc1 CS(=O)(=O)CCC(=O)NCc1csc(C(=O)NC2CCCC(O)CC2)c1 N1(C(C(CC)=CCCC)=O)CC(N(C(=O)CC=C(Cl)Cl)C)C(C)(C)C1 c1(-c2cc(CSC)[nH]n2)nc(-c2cccc(Br)n2)nn1CCN(C)C N1(C(C2CC=C(C)CC2)=O)CCN(C(C2OCCN(C)C2=O)=O)CC(C)C1 c1(C(=O)NC(C2CCCN(Cc3cccc(C)c3)C2)C)csc2ccccc12 CC(C)CC(CN=c1nc(-c2ccccc2)[nH]s1)NC(=O)C1=CC2CCCC12 c1(C(=O)NC2CCC(CNC(CSCCCC)=O)C2)cc2c(C)n[nH]c2cn1 C(CC(N)=O)(C(=O)NC1CNC(=O)OC1)NC(c1n(CC)ccc1)=O CCCC(C)(O)C(=O)NC1C2CN(C(=O)CC3(n4cncn4)CC3)CC12 C1(NC(CCn2c(C)ncc2)=O)CN(C(C2(F)CCOC2)=O)C2(CCCCC2)C1 Cc1onc(C2CC2)c1C(N1CC2CC1C2CNC(=O)C(C)n1cncn1)=O N1(C(C(C(=O)OC)OC)=O)CCn2ncc(CNC(c3ccccc3)=O)c2C1 C1(OCC)CN(C(=O)C(=O)NCC)CC1NC(=O)C(C)OCC(F)(F)F CC(C)CC(CC(=O)NC1(c2cc[nH]n2)CC1)NC(=O)C(C)(O)C1CCC1 Cc1cc(Cl)cc(C)c1C(=O)NCC1CCCC1NC(=O)C=Cc1ccco1 C(=O)(C(F)(CNC(=O)CC(C)(C)C(C)=O)C(C)C)Nc1cccc(CC)c1 CCC(C)(C)C(C)CC(=O)N1CCC(CCCC(=O)CP(C)(C)=O)CC1 Cc1ccc(C=CC(=O)NCC2CN(C(=O)CCC(F)F)CC2(C)C)c(C)c1 C1(C2CCN(C)CC2)(C(=O)NCC(CNC(C=CC=CCC)=O)O)CC1 N#Cc1ccc2oc(C(=O)Nc3ccnn3C3CCCCC3)cc2c1 C(=O)(CS(=O)CCC(F)(F)F)NCC(CNC(c1nccc(CC)c1)=O)O c1(C(=O)NC2C(CNc3snc(C)c3C#N)CCC2)ccc2c(c1)C(C)C(C)O2 C1(C(N2CC(C(C)OC)C2)=O)CC2CC1CN(C(C1CC(O)C(F)C1)=O)C2 C=C(C)c1cc(C#N)ccc1NC(=O)C(=O)NCc1cc(C)cc(F)c1 Cc1cc(F)cc(C(=O)NCC(O)CN(C)C(c2cnc3[nH]ncc3c2)=O)c1O C1(F)(CNC(CCOCCOC)=O)CCN(C(C2CC(n3ccnc3)C2)=O)C1 N1(C(C2(OC)CC2)=O)CCN(C(c2cncc(C(F)F)c2)=O)C(C(C)C)C1 N1(C(=O)OC(C)(C)C)CC2CC(C(=O)NCCNC(c3nc(Cl)cs3)=O)C2C1 Cc1cccc2c1CCN(C(C1CN(C(c3cc(CO)on3)=O)CCO1)=O)C2 N1(C(CCOCCOC)=O)CCCCC(NC(c2ncc(Cl)cc2Cl)=O)C1 C(CCN=c1[nH]c(=NC2CC3CC4C(C3)C24)[nH]c2c(F)cc(F)cc12)N(C)C c1(NC(CC2CN(C(=O)Nc3ccc(OCC)cc3)C2)=O)cc(Br)c(F)cc1F C=CCC(C(=O)N1CCC(C)(CNC(c2cc(Br)n(C)n2)=O)C1)NC(C)=O Cc1cnnc(O)c1C(N1CC(NC(c2c[nH]nc2C)=O)CC(F)C1)=O N1(C(C2N(C)CC(F)C2)=O)CCCC(O)(CNC(c2ccoc2C2CC2)=O)CC1 C1(NC(c2cnoc2C2CC2)=O)CCN(C(=O)Cc2ccc(O)nc2)CC1CO C(CN=c1[nH]ccc(=NCC2(C)CCCC2O)[nH]1)c1nnc(C)s1 C(CC(O)C(=O)NCC1(c2ccon2)CC1)NC(=O)CC1CCCOC1 C(=O)(C(O)CN(C)C)NCC(=C1CN(C(CC2CN(C)C2)=O)C1)F CCCCCC(CC)C(=O)NC(C)CCNC(c1nn(C)cc1C(F)(F)F)=O C1(C(=O)NC(CC(C)C)CNC(c2c[nH]nc2Cl)=O)CCCCC12CC2 C1(C(=O)NCc2ccc(SC)o2)CCCCN1C(C1(O)CCSCC1)=O C1(C(N2CCC(C)(F)CC2)=O)CC2CCCC2N1C(C1CC1C(F)F)=O N1(C(c2ncc(NC)nc2)=O)CCCC(NC(C2CC(OC)C(OC)C2)=O)C1C Fc1c(N2CCOC(c3ccc(F)c(Cl)c3)C2)ccnc1N1CCOCC1 c1(C(=O)NCCC2CCCN2C(C2CC23CC3)=O)cc2ccccc2cn1 N1(C(CCCN(C(=O)OC)C)=O)CCC(CNC(c2ncsc2C)=O)C12CC2 N1(C(Cn2c(C(C)C)nnn2)=O)CCCCC1CNC(=O)Cc1cccc(O)n1 C1(NC(C2C(c3n(C)cnc3)C2)=O)CCN(C(C2CN3CCC2CC3)=O)CC1O C1(NC(c2ccc[nH]2)=O)COCCC1NC(C1(C(=O)NC2C(CF)C2)CCC1)=O C1(NC(C=CC(CC)C)=O)CCC2(CC1)CN(C(=O)Cc1csnn1)CCO2 Cc1cc2c(cc1C)N(C(C1(C#N)CCCO1)=O)CC2 C1(NC(C2CCC23CCC3)=O)CCCCN(C(=O)CSc2ccc(Br)cc2)C1 C(CCCOC)(C(=O)NCCCSC)N(C1CCN(C)C1)CC N1(C(C(c2cccc(Cl)c2)N(C)C)=O)CC(NC(c2ccc(Cl)cc2)=O)C(O)C1 C1(NC(C(CNC(Cc2cnc(C)s2)=O)C)=O)CCC(C2CC2)C1 c1(C(=O)NCC2(NC(CN3C(C)CC3)=O)CC2)n[nH]cc1Br C1(C)(CN(C(=O)CCN(C(=O)CCCC2CC2C#N)CCCO)C)C(C)(C)C1(C)C C(C)(C1OCCc2sccc21)NC(=O)NC(c1ccccc1N(C)C)C c1(C(=O)NCC(C)NC(C2(C)CC2(F)F)=O)ccccc1C#N c1(N2CC(CN(C)Cc3ccc(F)cc3Br)C2)ncc2cc(Br)cnc2n1 c1(C(N(CC(C)NC(=O)CC2CC2(C)C)C)=O)ccncc1F Cc1ccc2ncc(C(=O)NCC(C)NC(c3cc(CO)n(C)n3)=O)n2c1 C1(C(N2CCC(O)(CCNC(C3(F)CC3)=O)C2)=O)CCc2nn[nH]c2C1 Cc1nc(F)ccc1N(C1CCNCCC1C)C(=O)C(F)F C(=O)(C(C)S(C)(=O)=O)N1CCC(N(CC#C)C(C2CC(OC(F)F)C2)=O)CC1 N1(C(CCN(C(C(CC)N(C)C)=O)C(C)C)=O)CCOC2COCC12 c1(C(N2C3CC(NC(CNC=O)=O)C2CC3)=O)ccc2c(c1)OCCO2 c1(C(N(CCCN(C)C(C2CCCC2(C)C)=O)C)=O)ccc2cncn2c1 CC1CN(C)CC1NC(=O)C(C1CC=CCC1)NC(c1ccnnc1O)=O c1(N2CCCC(CNC(C(CCC)CCC)=O)CC2)cc(C#N)ccc1[N+](=O)[O-] C1(NC(CCCCNC(C23CCC(OC)C2C3)=O)=O)CC(C)N(C)CC1C c1(OC)nc(C)ncc1C(=O)NC1(CO)CCCN(C(C2(S(C)(=O)=O)CC2)=O)C1 S(=O)(=O)(c1ccc(NCc2cc(OC(C)CN(C)C)no2)cc1Br)OC(C)(C)C N1(C(CC)C(=O)NC(C)Cc2ccc(Cl)cc2F)CCc2ccccc2C1 CCC(C)C(O)CNC(c1cnn(-c2ccccc2OC)c1)=O Cc1nc(SCC(=O)NCC(C)CNC(C2(O)CCC2)=O)n[nH]1 C(c1ccccc1)=C(C)C(N1CCC(C(C)(C)NC(=O)COCC2CCC2)C1)=O Cc1nnc2n1C(C(=O)NCC1CN(C(=O)C3CCCc4nc[nH]c43)C1)CC2 C1(NC(C=CSC)=O)CC2CC(C1)N(C(=O)Cc1noc(C)c1C#N)C2 C1(NC(CCc2c(C)noc2)=O)CCCC(C(F)(F)F)C1 c1(OC)cc(-n2nc(Cc3cccc(F)c3)nc2-c2ccc(F)s2)cc(F)c1 CCCC(CCC)CCCC(=O)NCC1CC1CNC(=O)CN1CCSCC1 c1(NC2CC(=CC=CC(=O)N(C(C3(C(=O)NC)CC3)=O)C)C2)nc(C)no1 N1(c2nnc(CN(S(C)(=O)=O)C)n2CC2CCCO2)CCS(=O)(=O)C(CCO)C1 N1(C(C2CC(C(C)C)C2)=O)CCN(C(=O)C=Cc2ncco2)C(CO)C1 C1(N(C(CN(C)CC)=O)C)CCN(C(=O)CSc2ccccc2OC)CC1 C1(CC)CCC(N=c2[nH]c(=NCC3CCOC3)[nH]c3ccccc23)CC1 c1(C(N2CC(=C(CNC(c3cnc(O)o3)=O)F)C2)=O)ncc[nH]c1=O C(CCC(C)(C)NC(C1(CC(C)C)CC(=O)C1)=O)NC(C(C)OC)=O CCCC(C)(CC)C(=O)N1CC(CNC(=O)CCCC2CC2)(OC)C1 C1(C(N2C(C)(CCO)CC2)=O)CCOCCN1C(C1CN2CCC1C2)=O C1(NC(c2ncsc2C2CC2)=O)CCCN(C(c2cc(-c3ccco3)no2)=O)C1 c1(NC(CC)CC)[nH]c(=NC2COc3cc(Cl)ccc32)nc2c1ncn2C CCC(C)N=c1[nH]c(=NC)[nH]c(=NCc2ccc(-c3nc[nH]n3)cc2)[nH]1 C(C)(C)(CCCC(=O)NCC1CC1C(=O)OC)NC(c1nccc(CC)c1)=O C1(NC(CNC(=O)OCC)=O)CN(C(c2cnc(C3CCOCC3)s2)=O)CC1C CC(C)(C)C(O)CN(C(C1(C)CCCC1O)=O)Cc1nc(-c2ccc(Cl)cc2)no1 N1(C(C(c2c(C)cccc2)(C)C)=O)CCC(CNC(=O)C(C)C)C(F)(F)CC1 N1(C(CC(=O)NCC)=O)CCC(NC(c2cc(C(C)C)sn2)=O)C(CC)C1 c1(-c2cn(CC(=O)NCCCNC(=O)NC)nn2)ccc(CCN)cc1 c1(C(=O)NCC2N(C(C3CCC(C)CC3)=O)CCC2)nccc(N)c1Cl N1(C(C(CC)N(C)C)=O)CCC(C(=O)NCc2nc(O)ccc2C)=C(F)C1 CC1CC(NC(c2cccnc2C(F)(F)F)=O)CN1C(=O)CCCc1cncs1 C1(C(=O)Nc2cccc(NC(c3c(C)cn(C)c3)=O)c2)C2CC3CC(C2)CC1C3 CC(CCC(=O)NCC1C=CCOC1)NC(=O)CC(=O)Nc1nccs1 c1(-c2c(NCc3ccc(C(C)(C)C(F)(F)F)cc3)cccc2)ccc2c(c1)CCO2 c1(C(COC)NC(=O)NCC(C2CCC(CC)CC2)(C)O)cc(F)ccc1O Cc1cncc(C(=O)NCC2CCCC(CNC(C3CN(C4COC4)C3)=O)C2)n1 C#CCCCC(C)C(=O)N1CC2CCN(C(=O)CC(C)(C)C=C)C2C1 C1(NC(=O)NC2(c3cn(CCN(CC)CC)nn3)COC2)CCCOCC1 N1(C(C2(F)CN(C(c3nn(CC)c(C)c3)=O)C2)=O)CCC(O)C(O)C1 C1(CNC(CSc2cccc(C)c2)=O)C2CCC(C2)N1C(=O)COCC1CCC1 c1(N2C3CN(C(C)=O)C(C3)C2)ccc(S(=O)(=O)NCC(O)C(C)C)cc1Cl C=CCCC(C(=O)OC)NC(=O)CC(CC1CC1)NC(=O)C1=NOCC1 C(=O)(CCCC(C)(F)F)NCC12CN(C(C3CN(CCC)C(=O)C3)=O)C(CC1)C2 N1(CCOC)CCC(C)C(CO)C1.c12ccccc1OCCCNC(=O)CC2 CC(C)C(F)(F)CC(=O)OCC1(C)CN(C2CCN(C(=O)OC(C)(C)C)CC2)C1=O Cc1ccc(F)cc1C1CC1C(N1CC(NC(=O)C2=CCOCC2)CC(O)C1)=O N1(C(C2CN(C(N(C)C)=O)C2)=O)CCCCC(NC(=O)CC2CCN(C)C2=O)C1 c1(C(N(CCN(C(CCOC)=O)C)C(C)C)=O)csc(-c2ccncc2)n1 c1(N2CC(CNC(C)=O)OCC2)cc2ccc(-c3sc(C)nc3C)cc2cn1 CCCCC(C)C(=O)N1CCN(C(=O)C(O)C(C)CC)C(c2cn[nH]c2)C1 CC(C)(C)C(=O)NCC(C1CCCC1)NC(c1cc(C(F)(F)F)n[nH]1)=O c1(C(=O)NC(CCNC(c2c(C)ccs2)=O)C(C)C)cccc(F)c1F C(CCC(C(=O)NCC1(C)CCC(C)CC1)NC(c1c[nH]ccc1=O)=O)OC CC1CN(C(c2ccc3c(c2)CCC3)C)CCc2ccc(F)cc21 CC(O)C(C(=O)NCC1CCCN1C(=O)C=CSc1nc[nH]n1)N(C)C C1(C(=O)NCC2(NC(C3=C(C)CCCC3)=O)CC2)CCc2nnc(O)n2C1 CC(C)CC(C(=O)N1CCN(C(c2cnc3n2CCC3)=O)CC12CCC2)C(C)C C1(CC(C)NC(=O)C2CC2)CC2CCC(C1)N2C(c1cnc(-c2cccs2)o1)=O CCC(CC(=O)NC1CC2(C1)CC(CNC(=O)CN(S(=O)(=O)CC)C)C2)C(F)F N1(C(c2c(CC)nco2)=O)CCCC2C1CCCN2C(=O)CN1CCCCCC1 c1(SC)cc(C(=O)NCC2(NC(=O)CC3CC3(C)C)CC2)ccc1N n1(C(COC(CC(C)NC(c2ccccc2)=O)=O)=O)nc(O)ccc1=O c1(-c2onc(CC3C(=C)C3)n2)cc2c(cc1OCC)OCO2 N1(C(c2ccccc2)C)CC23CCCC2(CNC3)C1 C1(C(=O)NC(CCC)CNC(C2CC(CC)(CC)C2)=O)CN2CCN1CC2 C1(C(=O)NCCC(C)NC(Cn2c(C)ncc2)=O)CC12CCSCC2 c1(SCC2CC2CO)ccccc1Cl.c12cc(n[nH]1)NC2=O.C12CCCN1NC2 c1(C(=O)NCC(C)N(C)C(c2c[nH]nc2-c2ccccn2)=O)ccnn1C(F)F Cc1ccsc1CC(N1CCCC1C1(O)CN(C(=O)C(=O)NC(C)C)C1)=O C1(C(=O)NCC(C)Oc2cccc(C)c2)CC(N)CCS1(=O)=O N1(C(CSC)=O)CCC(C2(O)CN(C(=O)C(C)(O)C3CCC3)C2)CC1 C(CC(C(=O)NC(c1cnc[nH]1)C)NC(c1cccc(CC)n1)=O)=CC CC(C)(O)C(F)C(=O)NC1CCC(NC(C2(CO)CCCC2)=O)C1 c1(N2CCC(n3nccc3)C2)nc(=NCc2cn[nH]c2)[nH]c2c1CCC2 c1(C(=O)NC(CC)(CNC(C2CC2(F)F)=O)CC)nn(C)c(N)c1C C1(N(C(CSC)=O)Cc2ccccc2)CCC(NC(C2CCNC(=O)C2)=O)CC1 c1(CC)nn(C)c(CC(=O)NC2CCN(C(=O)CCCC#N)C(C)C2)c1Br c1(C(N(C)C)=O)ccc(C(=O)NC2CC(NC(c3ccc(F)s3)=O)C2)s1 c1(C(=O)NCC(CC)NC(c2c(N)cc(F)cc2F)=O)cnc2scc(C)n12 c1(C(=O)NC(c2cn(CC3CCOC3)nn2)C)sccc1F c1(OC)cc(C(=O)NC2CCN(C(=O)C=C(Cl)Cl)C(C)C2)cc([N+](=O)[O-])c1C c1(C(C)NC(c2ccns2)=O)nocc1C(=O)N(c1ccn(C(C)C)n1)C N1(C(c2ccc(SC)o2)=O)CCC2CCC(NC(C3(C)CC(C#N)C3)=O)C12 C1(C(=O)NCC(CC)NC(c2cc(C)ccn2)=O)CC2OC(C)(C)OC2C1 CC(C)(C)C(CNC(C1CC(F)(F)CS1)=O)NC(c1ccc(C(F)F)cn1)=O CC(C)(C)C(CNC(C1CC(=O)CCO1)=O)C(=O)N1CCC(CN=[N+]=[N-])C1 C=C(CC)CN=C(NCC1CCC1)NC1CCN(c2ccc(F)cc2)C1 C1(CNC(C2(C)CN(C(COCCCCC)=O)C2)=O)CC(C)OC(C)C1 C(CC1=CCCCCC1)NC(c1n[nH]c(-c2ccccn2)n1)=O C=CCCC(C(=O)NCCCOC)NC(=O)CN(C)C(=O)C1CC1 N1(C(C2CCC3(CCC3)O2)C(=O)NC2CCOC2)CCCCC1C1CCCO1 C1(C(N(C(C#C)C)CCCC)=O)CN(C(=O)CC2CC(=O)NC2=O)CC1C1CC1 C1(c2nnnn2Cc2ccccc2)(NCCC(CC)(C)C)CC2CC1CC2(F)F C=Cc1cnn(C)c1C(=O)NCCOC(C)(C)CNC(c1cnccn1)=O S(=O)(=O)(c1cccc(OCCN)c1)NC(CCC)C c1(CC2N(CC(C=C)c3cccs3)CC2)cncc(F)c1 c1(OCCC(=O)NC2COCC2NC(C2C=CCC2)=O)ccc(F)c(F)c1 C(=O)(C(C)CC(F)(F)F)N(CC(C)NC(C1CCN(C2CC2)C1=O)=O)C Cc1ccn(CC(=O)NCC2(CNC(c3cc(C(F)(F)F)n[nH]3)=O)CC2)c(=O)c1 c1(CC)ccoc1C(=O)NC(C(=O)NCCN1CCC(O)C1)c1ccoc1 Cc1cccc(C)c1CNC1(c2ccc(C(N3CC(C)(O)C3)=O)cc2)CC1 C1(CNC(Cc2n(C)ccn2)=O)N(C(=O)CCP(C)(C)=O)CCC1(C)C C1(NC(CC=CC=C)=O)CN(C(=O)Cn2nc(C)n(C)c2=O)CCC1C C(=O)(CCC(=O)NN(C)C)NC(C)C(C)NC(c1ccc2nc[nH]c2c1)=O c1(C(=O)NC2CC(CNC(CC3C(OC)CC3)=O)C2)c(C)cc(C)oc1=O C1(C(=O)NCC2CCN(C)C2)COC2(C1)CN(C(c1cc(O)n(C)n1)=O)C2 c1(C(N(C(C)C)CCN(C)C(C2CC(=O)C2(C)C)=O)=O)c2c(nn1C)CCCC2 C1(O)(CNC(CCc2cc(C)[nH]n2)=O)CCN(C(c2cnn(C3CC3)c2C)=O)C1 N1(CCOC)C(=O)NC(c2cc3n(n2)CCC3)C2=C1C(C)CN(C)C2=O CCCCC(CC)CC(=O)N1CCOC(CNC(c2cncc3nc[nH]c23)=O)C1 Cc1ccc(F)c(CC(=O)NCCC2(O)CN(C(C3CCC(C#N)C3)=O)C2)c1 c1(C(=O)NC2CN(C(CC(C=C)CC)=O)CC2C)cccc(S(=O)(=O)NCC)c1 C1(CNC(C2C(C)=CCS2)=O)CN(C(C23CCCC(CO2)C3)=O)CCC12CCC2 N1(C(Cn2c(C)nc(C)n2)=O)CCCC(F)(CNC(=O)COC2CCCCC2)C1 c1(C(=O)NCC2C(CC)CN(C(=O)CC(C)(F)F)CC2)nc2ncccn2n1 c1(C(=O)NCC(CC(C)C)NC(CCCC(C)=O)=O)[nH]nc2c1COC2(C)C c1(CC(N2CCC(OCCNC(C(C)(C)CC3CC3)=O)C2)=O)ccc(O)c(Cl)c1 C=CCCN=C1NCCC(CSC)OC(=O)N2CCC(N1)C2.C(C)(C)(C)OC N(C1CCc2sc(Br)cc21)C(C(=O)NC(c1cccc(Cl)c1)C)C C(=O)(C(O)C1=CCCCC1)N1CC(F)(C(N(C)CC)=O)C1 C1(C(=O)NCC2OCC3(CN(C(CC=CC)=O)C3)C2)CCc2nncn2CC1 C1(C(=O)NC2CC3(C(NC(=O)C=C4CCCCC4)C3)C2)Cc2c(F)cccc2O1 C1(C(=O)NCCC2=CCN(C(C(CC)CC)=O)CC2)COc2ccccc2C1 CC(C)(CC(=O)NC1CCC1CNC(c1ccc(F)c(Br)c1)=O)C(F)F c1(CC)ccc(NC(=O)CCC23CC(CN2C(=O)C(C)(C)COC(C)=O)C3)cc1 N1(CCNC(C2C(NC(COCC(C)C)=O)CC2)=O)CCCOC1=O CCCCCCC(C)CC(=O)N1CC(C(C)NC(c2cscc2Cl)=O)C1 CC(O)C(F)(F)C(=O)NC1(CC(N)=O)CCN(C(C2CCOC2(C)C)=O)CC1 CC(C)CC(C)(CNC(=O)C(C)(F)c1ccccc1)NC(=O)COCCF n1(CC)cnnc1C(=O)NC1CCC(CNC(=O)C(C)Cn2ccc(C)n2)C1 c1(SC)nc(C)c(CC(N2CC(N(C)C(C3(CO)CCCO3)=O)C2)=O)c(O)n1 C1(C(=O)NCCCCNC(COC(C)=O)=O)CCCCC1F c1(C(=O)NC2CC(CNC(C3(SC)CC3)=O)C2)ccc(C)o1 N1(C(C(C)NS(CC)(=O)=O)=O)C2CCCC1CN(C(C1CCO1)=O)C2 c1(NC(=O)CSc2ccccc2)ccc([N+](=O)[O-])cn1 N1(C(c2cccc(C)c2)=O)CC2CCN(C(c3nn(C)cc3N)=O)CC(C2)C1 C#Cc1ccccc1CC(N1CCN(C(C2CCC3(CC3)C2)=O)CC1COC)=O CCCCCC(C(=O)N1CC2CCCC1(CNC(C1(CCC)CC1)=O)C2)C(C)C CCC(C)(C)C(C)CC(=O)N1CC(F)CC1CNC(=O)C(=O)C(C)(C)C c1(OC)ccc(C)c(C(=O)NC2CCC(NC(=O)C(C)(O)C(C)C)C2)c1 n1(CCNC(C=CCN(C(c2cc(CCC)[nH]n2)=O)C)=O)ccccc1=O c1(C(=O)NCC2N(C(c3ccnc(OC)n3)=O)CC=C2)ccc2nc(CO)[nH]c2c1 C1(COCc2ccccc2)C(=O)O1.C1(O)(CCCNC(C)=O)CCC1 c1(N(C)Cc2ccccc2)cnn(C2CN(S(=O)(=O)CCCl)C2)c1 C1(NC(=O)OC(C)(C)C)CC2(CCC2)N1C(N1CCC(n2c(C)cc(C)n2)CC1)=O C1(NC(C2C(C)N(C)CC2)=O)CCN(C(=O)C2=COCC2)C12CC2 N1(C(C(C(=O)OCC)OC)=O)CCC(C(=O)NC(C)CS(N)(=O)=O)C12CCC2 CCC(F)(F)CC(=O)NC(CC(N)=O)C(=O)N(C)CC1CCCC2CC12 Cc1nn(CCF)cc1NC(=O)C(C)(C1CC1)N(C)C(C1C2CC(=O)CC12)=O c1(C(=O)NC(CC)CC(=O)NCc2ncco2)cccn(C)c1=O C(=O)(C(=O)CCC(C)C)N(CCC(N1CCC(N(C)C)C(C)C1)=O)CC=C Cc1nc(C)c(C(=O)NC(CNC(=O)C(C)(C)C2(C)CC2(F)F)CO)o1 c1(CCC(=O)Nc2ccccc2N2CCCC2)ccc(F)c(F)c1 c1(C(N(CCC(=O)NC(c2nc[nH]n2)C2CC2)CC#C)=O)cc(O)ncn1 N1(C(c2cncc(N3CCCC3)n2)=O)CCN(C(=O)C=C2CCC2)C(CCO)C1 C(=O)(C1Cc2ccccc21)NC1C2C(NC(C(CC=C)CC=C)=O)CC(CC2)C1 c1(C(=O)NCC(C)(CO)NC(c2cc(O)ncn2)=O)cnc2n(c1=O)CCS2 c1(CC(N2CC=CC(NC(=O)CSC3CCCCC3)C2)=O)ncnc2ccsc12 N1(C(C2(CC=C)CN(C(=O)CC3CCCNC3=O)C2)=O)CCC2CN(C)CC2C1 O=C(CCCC(F)(F)F)N1CC2CC(C1)N2C(=O)CC1CCCO1 C1(C(=O)NCCC(=C)CNC(=O)C(C)C(C)(F)F)CC(c2ccccc2C)=NO1 N1(C(c2cccc(CC)c2)=O)CC2CC3CC2C1C3NC(=O)C(F)C1CCC1 N1(C(CC2CC(C(=O)OC)C2)=O)CCCC2(CCN(C(c3n[nH]cc3Cl)=O)C2)C1 c1(SC(C(=O)OC)C)cccnc1.C1(=O)CNC(=O)C2(CC2)CCCN1C(C)C N1(C(COC(C)=O)=O)CCN(C(C2CNC(=O)C2)=O)C(C(C)C)C1 c1(C(=O)NCC2CN(C(C3CC(C4CCC4)C3)=O)CCO2)ccc2c(c1)OCO2 C12(O)CCN(C1)C2=O.c1(C(=O)OC)cnoc1NC1CC1c1ccccc1 C1(NC(C(CC)NC(C)=O)=O)Cc2ccccc2C1NC(=O)C(F)=C(C)C1CC1 Cc1nc2ccccn2c1CC(=O)NCC1CCN(C(C2CC(F)C(=O)N2)=O)C1 N1(C(COCCOC)=O)CCC2(CC1)CC(C)N(C(c1cc([N+](=O)[O-])n[nH]1)=O)C2 C(c1cccnc1)=CC(=O)N(C(C(=O)NCC(c1ncc[nH]1)C)C1CC1)C C1(C#N)(C(N2C(C(N(CCOCC#C)C)=O)CCC2C(C)C)=O)CCCCC1 C1(NC(CCC=C(C)C)=O)CN(c2ncc(F)cn2)CC(F)(F)C1 N1(C(C23CC(CC)(C2)C3)=O)CCC(C2CN(C(=O)Cc3ccc(O)cn3)C2)CC1 C1(C(C)NC(c2cn(C(F)F)cn2)=O)CN(C(c2cc(Cl)c[nH]2)=O)CCO1 Cn1c(C(N2CC(C)(NC(C3CCCCS3)=O)C2)=O)ccc1C#N N12CC(CCC1C)C2.c1(N(CCN(C(C)=O)CC)C(C)=O)ccsc1C c1(C(=O)NCC2N(C(C3CC(C)OC(C)C3)=O)CCCC2)cc(C#N)ccc1O C#CCC(CC#C)C(=O)NCCCC(C)NC(C1Cc2ccccc2O1)=O C1(C(=O)NC2C(CC)OCCN2C)CN(C(=O)CC(C(=O)O)N)CCC1O.C(C)C c1(-c2cn(CC(=O)NCc3snc(C)n3)nn2)cnn(C)c1C c1(CC(N2C(CC)C(NC(=O)CN3CCC(F)CC3)CC2)=O)cc(F)cc(F)c1 N1(C(C(C)SCCCC)=O)CC2CC(C1)CN(C(=O)COCC(F)F)C2 CC(O)C(=O)N(CCC(=O)NC1CC(CC(N)=O)C1)CCCO C(=O)(C(C)CCCC(C)C)NCC1N(C(c2c(C)ccnc2)=O)CC(C)(C)C1 C=CCC(C(=O)NC(C)CCCO)NC(c1cnn(CCC)c1)=O c1(C(N2CCOCC2C2CCC2)C(=O)NCCOC)cc(OC)c(Br)c(OC)c1 C#Cc1cc(C(=O)N(CCCNC(=O)C(CC)CC)CCO)cc(F)c1 C1(N(C(C)=O)C)CN(C(c2ccc(C3CCCC(=O)N3)cc2)=O)CC12CC2 Cc1sc(Cl)nc1C(=O)NC(c1ccc(CNC(=O)C=Cc2ccsc2)cc1)C c1(C(=O)OC)cc(OC)cc(C(=O)NC2CN(C(=O)C=CC(C)(C)SC)CC2C)n1 c1(C(N2C(C)CC(CNC(C3C(OCC)C3C)=O)C2)=O)nn(C)c(C)c1N CC(C)C(C)(O)C(=O)NCC1CC2CN(C(=O)Cc3ccc(O)c(Cl)c3)CC12 c1(C(N(C(c2cccc(O)c2)C)C)=O)cc2c(s1)C(C)(C)CCC2 N1(CCNC(C2C(C=C(C)C)C2(C)C)=O)CCCN(C(=O)CNS(N)(=O)=O)CC1 C(=O)(C(F)C(CC)CC)N1CC(C(C(=O)NCc2onc(CC)n2)O)C1 C1(CNC(c2n(CC)ncc2)=O)CC(C)(C)CCC1NC(C1(C)CCC1)=O c1(CC=C(C)C)ccccc1CC(=O)NC1CCCC1CNC(=O)Cc1ccsc1 CC1CN(C(=O)CSC(F)(F)F)CC(C)N1C(=O)CC1CCCOC1 CC(C(=O)OC(C)(C)C)C(=O)N1CC(N(C)C(c2cc(C(C)(C)C)nn2C)=O)C1 C(=O)(C1COc2ccccc21)NC(C)CC(C)NC(c1occ2c1CCOC2)=O C1(CC#C)CN(C(c2cnn(C(C)C)c2)=O)C12CCC2 c1(CC(N2C(CNC(c3cc(CC4CC4)on3)=O)CC2)=O)ccc(Cl)cc1 c1(C(C(=O)NCC(CNC(c2c(C)cco2)=O)O)C)ccc(Br)cc1F CCCC(CNC(=O)C(C)n1ccnn1)C(=O)NCCC(C)(C)C C(=O)(C1CCc2cccnc21)NCCCCNC(CC(C)(O)c1ccccc1)=O C1(CCC2N(C(CCSC)=O)CCC2)CCCCN1C(=O)C=CC1CCCC1 C1(F)(CNC(c2c(C)nn(C)n2)=O)CCN(C(c2cnn(CCO)c2C)=O)CC1 c1(N(CC(C)N(C(C)=O)C)C)ncnc(NCc2cc(-c3ccco3)on2)c1C c1(C(=O)NCCN(C2CCCC2)C(CN2C(C)CC2)=O)c(F)c(F)cc(F)c1F C#Cc1ccc(C(N2CC(NC(=O)Cc3cccs3)CC2C)=O)cc1Cl CCCS(=O)(=O)CC(=O)NC1CN(C(c2cnc(OC)c(Br)c2)=O)CC1C c1(C(=O)NCC2C(NC(C(C)=C(CC)C)=O)COC2)[nH]c2ccccc2c1Cl C1(NC(C(COC)O)=O)CN(C(=O)CC=Cc2ccc(F)cc2)CC12CC2 C(CCC(=O)NC(C)C=CC(=O)NC(CC1CCCC1)CO)OCC CCC(F)(F)C(C)(C)C(=O)N1CCC(C2(NC(c3nc(C4CC4)cs3)=O)CC2)C1 C1(CNC(C2(C(N(C)C)=O)CC2)=O)CN(C(=O)Cc2ncc[nH]2)CC1(C)C c1(OC(CC)CNCc2cc(C3CCC3)[nH]n2)ccc(Cl)cc1C c1(C(=O)NCC2(NC(c3on(C)c(=O)c3)=O)CCOCC2)nc2ccccc2s1 C1(CNC(C(C)OC)=O)C(C)CCCN1C(c1sccc1C)=O Cc1cc(=O)c(C(N2CCOC(C)C2C(=O)NCCCc2ncnn2C)=O)c[nH]1 C=C1COc2c(C(=O)NC3(C)CN(C(=O)Cn4cccc(N)c4=O)C3)cnn2C1 C(=O)(N1OC2CC1C(O)C2O)C1CN(C(=O)C=CC2CCOC2)CC12CCC2 CC(CCC(=O)NC(c1nccs1)C)NC(=O)Cc1ccc(O)cc1 C=CCC(CC(=O)NCC(F)(F)Cl)NC(=O)CC(C)(C)C1CC1 C(=O)(C(=O)CC(C)CC)N(CC(N1CCCC(OCC#C)C1)=O)CCC C1(NC(C(C2CC2)OC)=O)CCSC12CN(C(c1ccc(F)c(C#N)c1)=O)C2 N1(CC)C(=O)CCC(CNC(=NC)NCC=CBr)C1c1cccs1 C1(NC(NC(CC)CC)=NCc2ncoc2C(C)C)Cc2cccc(OC)c2C1 C1(C(N2CCC(N(C(=O)CCN3CCC3)CC)C2)=O)Cc2cc(F)cc(F)c2O1 Cc1ccc(F)cc1C(N1CCC(C(C)NC(=O)CCCC(N)=O)C1)=O CN1CCC(CCNC(=O)CCN(C)C(C2CCCCC2)=O)C1=O CC1CN(Cc2ccc(Cl)c(F)c2)CCC1CCC(=O)O N1(C(CC2CC(=C)C2)=O)CCN(C(=O)CCC23CCC(CC2)C3)CC12CCC2 N1(C(C)C)CC(NC(=O)NCC2(c3nn[nH]n3)CCCCC2)CC1=O CCC(CC(=O)N(C(C)C(=O)N1CCC1C(C)O)C)C(C)(C)C c1(C(N(CCCC(=O)NC(CC)(C)C2CC2)C)=O)cc(Cl)n(C)n1 c1(C(=O)OC)cc(F)cc2c1CCN(C(C)C(=O)Nc1ccccc1C)C2 C(CC(F)F)(C(=O)NCC1COCC1C(N)=O)N(C)C(c1ccc([N+](=O)[O-])o1)=O C1(CNC(CC=CCC)=O)CCN(C(=O)CN2CCCC2=O)CC1C1CC1 C1(CC(=O)NC(C(=O)NCC2(C)N=N2)CC2CC2)OCCC1(C)C C12(NC(=O)OC(C)(C)C)CC(C1)C(CNC(c1ccccc1)CO)O2 C(CC1=CCN(C(=O)CC2CC2C)CC1)NC(c1ccc(C(C)=O)cn1)=O C(=O)(CCC(=O)NC(C)CC(C)NC(C1(C)C=CCC1)=O)OC N1(C(CC=C)=O)CC(OCC)C(CNC(=O)CCc2n[nH]c(=N)s2)C1 Cc1cnc(C(N2CCC(N(C)C(c3cc(CF)on3)=O)C2)=O)c(Br)c1 n1(CC(N2CCC(C)C2CNC(C2CCCC2)=O)=O)nc2ccccn2c1=O C1(CNC(c2ccncc2)=O)CN(C(=O)Cc2csnn2)CC1C(F)(F)F C(=O)(C(CC)C(=O)N1CCC(O)(C(C)NC(c2ncccn2)=O)CC1)OCC N1(C(C=CC(C)C)=O)CC2CN(C(c3ccc(F)cc3Br)=O)CC(C1)O2 C1(C)(CNC(c2cc(SC)oc2)=O)CCCN1c1nnc(C(C)(C)C)s1 c1(C(=O)NC(C)C(C)(C)NC(C2CC23CCC3)=O)cnc2c(c1)NC(=O)CN2C c1(CNC(C(C2CCC2)OCC)=O)cccc(NC(c2nc(=N)cc[nH]2)=O)c1 c1(CC)ccc(C(=O)NCC(C2CC2)N(C(=O)CCSCC(N)=O)C)cc1CC c1(C(=O)NC(CN(C(c2coc(Cl)c2)=O)CC)C)cn(C(F)F)nc1C(F)F N1(C(c2nn(CC)c(C)c2)=O)CCC2(CC2C(=O)Nc2cccc(C3CC3)n2)C1 CCC(C)C(=O)C(=O)N1CCOCC(NC(C2C=CC=CC=C2)=O)C1 Cc1nn(C)cc1-c1ccc(C(=O)N(C(C)CCO)Cc2ccccc2)nc1 C=C(C)CC(C(=O)OC)NC(C1CCCCN1C(c1cnc(O)n1CC)=O)=O c1(NCC(c2ccc(I)s2)C)snc(Cl)c1C#N N#Cc1cc(C(=O)NCC2(O)CC(C(=O)NCCC34CC(CO3)C4)C2)c[nH]1 CCCCCC(C(=O)NCCCC(C)NC(c1ccnn(C)c1=O)=O)C(C)C c1(NC(=O)Nc2cccc(C(C)(F)F)n2)cn2ccc(Br)cc2n1 N1(C(COCC(=O)NC)=O)CCC(C(=O)N(C(COC)CC)C)(C(C)C)C1 CCC(C)C(C(=O)Nc1ccc(F)cc1C)N(CC)Cc1cnn(C)c1 CC(Cc1nc(-c2cccc(Br)n2)nn1CC(F)(F)F)C(F)(F)F c1(C(N2CC(O)(CNC(=O)Cc3ccccc3)C2)=O)ccc(I)cc1Br C1(C(=O)NC(c2cccnc2N2CCCC2)C2CC2)CC2(C1)CC(F)(F)C2 C(CNC(=O)CCc1cncc(F)c1)(C(C)C(C)C)NC(C1(COC)COC1)=O c1(C(=O)NCCC(C)NC(=O)CSCC2CCCCO2)ccc2nc(O)oc2c1 CN1CCCCC1CC(N1CC(C2CCCCN2C(=O)Cn2cc(Cl)cn2)C1)=O Cc1nc(C(=O)NCC2COC(CNC(c3c[nH]c(C(F)(F)F)c3)=O)C2)nn1C C1(CC)(NC(=O)C=C2CCC(C)CC2)CCCN(C(=O)CCc2c[nH]c(=N)[nH]2)C1 c1(OC)cc(C(N2CCC(c3ncco3)C2)C(=O)NCCC2CC2)sn1 N1(C(C23CC(NC(C4C(COC)CC4)=O)(C2)C3)=O)CCCNC(=O)CC1 n1(C(C)C)cnc(C(=O)NCC(CO)NC(=O)C(C)(C)c2cccs2)n1 c1(C(=O)NC(C2CCCCN2C(c2ccc(F)cc2)=O)C)cccn2nccc12 c1(N(C(C(=O)NC)C)C)ncc2ccc(-c3ccnc(Cl)c3F)cc2n1 N1(C(CNC(C2C(C)C2)=O)=O)CC(C)(C(N2CC3(CCC3(C)C)C2)=O)CC1(C)C Cc1cccc(C)c1C(=O)NC1C=CC(CC(N2CC3(CCC3O)C2)=O)C1 N1(C(c2ccc(F)s2)=O)CC23CCCC2(C1)CN(c1ncnn2cccc12)C3 C1(C(N2CC3CN(C(CCC(=O)NC)=O)CC3C2)=O)Nc2ccccc2C1(C)C N1(C(CCNS(C)(=O)=O)=O)CCN(C(c2cc(Cl)ccc2F)=O)C(CF)C1 C12(CNC(C=CC(C)C)=O)CC1CN(C(C1(O)CC(C(=O)OC(C)(C)C)C1)=O)C2 C1(NC(c2[nH]cc3c2CCC3)=O)CCN(C(=O)CC2CCCO2)CC1F c1(Nc2ccc(N3CC(C)OC3)cc2)cccc2ncccc12 c1(CN(C2CCN(CCC)C2)C)ccc(C(=O)Nc2nnc(CC)s2)cn1 N1(C(C2CCCCC23OCCO3)C(=O)NCCOC)CCC2(CCCCCC2)C1 c1(C(=O)NCC2C=CC(NC(C(C(C)C)NC=O)=O)C2)noc2ncccc12 c1(C(C)C)c[nH]cc1C(=O)NC(C(=O)NCCN1CCC(C)C1)c1ccco1 C1(C(=O)NCC=CCCOC)CC=CC(NC(C2CCOC2C)=O)C1 C1(NC(CC(C)OC)=O)CC2CC1N(C(C1CCN(OC)CC1)=O)C2 CC1CC(NC(=O)CCn2cnc(=N)[nH]2)CCN1C(=O)Cn1nccn1 C1(NC(C2CC(SC)C2)=O)CCC2(CC1)CC2NC(c1cccc2nccn12)=O Cc1c(I)ccc(NC(=O)CCCc2cccc(Br)c2)c1C CCCCC(CC)CC(=O)N1CCCC(NC(c2nn(CCC)cc2Cl)=O)C1C N1(C(c2ncc(NC)nc2)=O)CC(C)CN(C(c2nc(Cl)ccc2F)=O)C(C)C1 C1(C(N2CCOCC2CC2CC2)=O)CCCCN1C(=O)C(C1CC1)C1CC1 c1(OC)ccc2c(C(=O)NC(C)CCNC(c3cccn3C(C)C)=O)n[nH]c2c1 N1(C(C(C#N)CC2CC2)=O)CC=C(C(=O)N2CCCN(CCO)CC2)C1 C1(C(=O)NCCCC2CC(C)C2)CCCC(NC(=O)CN2CC3CC3C2)C1 C1(C(=O)NCCC=CC=C)(OC)CCN(C(=O)Cc2csc(C)c2)C1 c1(C(=O)NC(CNC(C2CC(C)(C)O2)=O)CO)c(Cl)ccc(Br)c1F c1(OC)cccc(C(CNC(C2CC3CC3N2C(=O)CCCC#N)=O)N(C)C)c1 Cc1oc2ncn(C)c(=O)c2c1C(N1CCOCC(CNC(C2(O)CC2)=O)C1)=O CCC(CO)(CO)C(=O)NCc1c(C(F)(F)F)coc1C C1(C(=O)NCC2CC(C(=O)NCC(CC)(C)OC)C2)CC2(CC2)CO1 c12cc(cnc1OC)C(=O)N2.C1(SC)COCCN1C(=O)NCC1CCCCC1 Cc1cc(C(=O)NCCC(C)N(C)C(C2CC(C)C2)=O)c2c(n1)CCCC2 c1(C(=O)NCCC(CNC(C(C2CC2)OCC)=O)O)cc(C(F)(F)F)cc(O)c1 CC1(CO)CCCN1C(=O)C(C1CCN(C(c2cccc(O)c2)=O)C1)F C12(CNC(C(C3CC3)OCC)=O)CC1CN(C(=O)C=Cc1cc(Br)cs1)C2 C1(CNC(C2(OC)CCSC2)=O)COCCN1C(c1ccn(C2CC2)n1)=O C(=O)(C(C)CCCC(C)=O)NCc1ccc(C(=O)NC(CC)C)cc1 c1(C(=O)NC(C(=O)NCCC2CN(C)C(=O)C2)CCF)cc2cccn2cn1 Cn1ncc(Cl)c1C(=O)NCCC(C)(C)NC(=O)CCC1CCC1 C1(NC(=O)Cc2cc[nH]n2)CCN(C(C2(Cc3cnn[nH]3)CCC2)=O)CC1O c1(C(=O)NCCCN(C(c2nn(C)nc2Br)=O)CC)ccc(Cl)cn1 C1(OCC)(CNCc2sc(C)cc2C)CCCSC1 C1(NC(C(C)(C)C)=O)CN(C(c2cc(-c3ccccc3F)on2)=O)CC1O CCCCCCCCC(=O)NCCCCC(C)NC(=O)C(C)n1ccnc1 C1(C(=O)NCCC2(CNC(C3(O)CCC(C)CC3)=O)CC2)CCCC2(CCC2)C1 CC1(C)C(CNC(C2CC23CCC3)=O)CCN1C(=O)CN1OC(C)(C)CC1=O c1(NCC2(COC)COC2)cc(F)nc(O)c1Cl c1(CC)cnc(O)c(C(=O)NC2(CNC(c3cnn(C)n3)=O)CCCCCC2)c1 C1(NC(c2cccc(CO)c2)=O)CN(C(C2CCSC2)=O)CC(F)(F)C1 c1(C(=O)NC(CN(C(c2cnn(CCF)c2)=O)CC)C)ccn(C)c1C N1(C(c2nc(OC)oc2)=O)CC(CO)C2(C1)CN(C(c1cccn1C1CC1)=O)C2 C(CC(CC)C(=O)N1CC2CC(NC(=O)CC3(c4ccon4)CC3)C1C2)=CC C1(N(C(C2C(OCC)C2)=O)C)CCC(NC(=O)Cc2ccccc2C(N)=O)CC1 c1(CC)cc(C(=O)N(C(C)CNC(=O)CCC2OCCO2)C)nn1C c1(NC(N2CCC(NC(C(C=C)C)=O)C2)=O)sc2c(c1C#N)CCCCC2 N1(C(CCOCC)=O)CCN(C(C2(CC(C)C)CC2)=O)CC12CC2 S(=O)(=O)(c1ccc(F)c(Cl)c1)N1C2C(C(=O)NCCC)C(C2)C1 C1(CNC(C(CC)CCOC)=O)CCCC2(CN(C(=O)Cn3nnnc3C)C2)O1 CCC(C(=O)NCC(O)CNC(=O)Cc1ccc(CO)cc1)C(C)(F)F c1(NC(C2(C)CCCN(C(c3cocn3)=O)C2)=O)ccc(Br)c2ccccc12 N1(C(Cc2c(C(=O)OC)csc2)=O)CC2CCC1CN2C(C1C2CCCC12)=O c1(OCC(=O)NCC2COCCN2C(c2cc(Br)c[nH]2)=O)cncc(Cl)n1 C(C(C(C)C)NC(=O)C(C)(F)F)(c1ccccc1)NC(c1[nH]cc(CC)c1)=O c1(OC)ccc(S(=O)(=O)NC(c2cnn(C3CC(N)C3)c2)=O)s1 N1(C(C=CCCC(C)C)=O)CCSCC1C(=O)N(CCC(C)(C)O)C N#CC1CN(C(c2nc(C(=O)N(c3ccc(Br)cc3CO)CCO)cs2)=O)CCO1 C1(N(C(C2SCC=C2C)=O)CC)CCN(C(C2CN(C(C)C)C2)=O)CC1 C1(C#CC(=O)N2CCCCC2C(C)(C)CNC(=O)CNC(C)=O)(CC)CC1 n1(CC(=O)NCCNC(C2CC3CC3C2)=O)ccc2ccccc2c1=O N12CCCC1C1(CC1)C2=O.n1(CNC(C2CC2CF)=O)cc(CO)nn1 C(CCCCCCO)NC(C1C(CNC(C2CC(CF)C2)=O)CCC1)=O c1(OCC(=O)NCC)ccc(C(N2CC(NC(=O)C(F)OC(F)(F)F)C2)=O)cc1 C1(C2CCOCC2)(C(=O)NCC2C(C)CCN(C(c3c(C)nccn3)=O)C2)CC1 CC1OC2(C(N3CCC(CNC(=O)CCN4CCOCC4)C3)=O)CC1C2 c1(C(N2CCC(COC)(NC(=O)Cn3cncn3)C2)=O)ccc2scnc2c1 CC1=C(C(=O)NC23CC(CNC(C4CCCCN(C)C4)=O)(C2)C3)SCCO1 N1(CC)CCC(C(=O)NCCCCNC(c2csc(-c3cnn(C)c3)n2)=O)C1 c1(C(=O)NC2C(CNC(C(C(C)(C)C)OC)=O)C2)c(Br)ccc(F)c1N c1(C(N2C(C(=O)NC3CC3c3cccc(Br)c3)CC3CC32)=O)cc(I)cnc1Cl c1(C(=O)NC2CC(CNC(Cc3scc(C)c3)=O)CC2O)ccc2cnsc2c1 CC(C)P(=O)(CC(=O)NCC1(O)CCN(C(=O)Cc2c[nH]ccc2=O)C1)C(C)C Cc1cc(C(=O)NC2CC(NC(c3ccccc3)CCO)C2)c(C)[nH]1 C(=O)(C(F)(F)C(F)(F)C(F)F)NCC1CN(C(CNC(=O)NC)=O)C(C)(C)C1 c1(C(C)(C)C)n[nH]cc1S(=O)(=O)NC1CS(=O)(=O)C1(C)C c1(C(=O)NC2C(NC(C3C(C)C(=O)C3)=O)CCC2)cnc2[nH]cncc1-2 c1(C(=O)NCC(C2N(C(C(C(C)C)C)=O)CCCC2)(C)C)cc2n(n1)CCCC2 N1(C(C(C)n2ccnc2)=O)CC(CNC(C2CCN(CC3CC3)CC2)=O)C(O)C1 O=C1CCC2CN(c3cc(N(C)Cc4ccc(C5CC5)cn4)ncn3)CCC2N1 C(=O)(C1=Cc2ccccc2OC1)N1C2CC(NC(=O)C=CC(F)(F)F)CC1CC2 c1(C(=O)NC(C)CCNC(c2cccc(CN=[N+]=[N-])c2)=O)cc(F)c(F)cc1N c1(C(=O)NC2CC(O)(CNC(C(CSC)O)=O)C2)cccc2sncc12 C12(NC(CS(C)(=O)=O)=O)COCCC1CN(C(c1cnc3[nH]cnc3c1)=O)C2 n1(COC)nccc1C(=O)NC1CC1CNC(=O)COC1(C)CCCC1 C12(NC(C(CSC)OC)=O)CCCC1N(C(=O)COc1cccc(F)c1F)CC2 c1(C(=O)NCC2CN(C(Cc3cc(C)sc3C)=O)C(C)C2)cc(C)n(C)c(=O)c1 N1(C(c2c(C(C)=O)ccs2)=O)C2CCC1CC(N(C(=O)Cc1c[nH]nc1C)C)C2 c1(C(=O)NCC2C(CNC(C3(C(=O)NC)CCC3)=O)C2)coc2ccc(Cl)cc12 C(=O)(C(C)(O)CC(C)C)NC(CC)CN(C)C(C1(N(C)C)CCC1)=O N1(CC(=O)NS(CC)(=O)=O)CCS(=O)(=O)C(CCNC(=O)CC(C)(F)F)C1 c1(NC(CCOCC)C)ccc(S(=O)(=O)N2CCC(OC)C2)c(Cl)c1 C1(NC(CCSCCCC)=O)CC2C1CCN2C(c1ccc(N2CCC2)cc1)=O c1(-c2ccc(C)nc2C)ccc2c(c1)COC21CN(Cc2cc(F)cc(Br)c2)C1 Cc1cc(C(=O)NC(C)C(C(C)C)NC(=O)CN(C)C2CC2)n(C(C)(C)C)n1 C1(O)(CN(C)C(c2conc2C2CC2)=O)CCN(C(=O)C(C)(C)CC2CCC2)C1 c1(N(CC(C)C(C)(C)C)C)cccc(S(=O)(=O)NCc2ccc(Cl)o2)n1 O=C(C#CC1CCCCO1)N1CCC2CN(C(c3ccc4c(c3)CC4)=O)C2C1 C=CC(C)(CCOC)C(=O)NC1CCN(C(=O)CNC(C2CCOCC2)=O)C1 N1(C(CCCOC(C)=O)=O)CCCC(c2cn(C(C)C(=O)N3CCCC3)nn2)C1 Cc1cc(C)c(CC(N2CC3(CCN(C(C4CC(=O)N4)=O)C3)C2)=O)c(O)n1 N1(C(C(C)C)=O)CCCCC1C(=O)NCC(C)NC(=O)C(c1cccc(F)c1)O C1(C(=O)NCC(CN(C(C2(OC)CCOC2)=O)C)O)CCCCCCC1 N1(C(CC)=O)CC2(COC)CC1(CNC(=O)CC1(c3ccccc3)CCCO1)C2 c1(C(=O)NC(CC=C)CNC(c2nnn(C(C)(C)C)n2)=O)cnc2sccn12 c1(OC)ccc(C=CC(=O)N(C2CN(C(=O)C(C)CS(C)=O)C2)C)c(C)c1 N1(C(CC(=O)N(C)C)=O)CC(CC(=O)NC(C2CCCCC2)CO)C2(CC2)C1 CCCC(C)(O)CC(=O)NC1CCCCN(C(c2ccc(F)cc2F)=O)C1 N1(C(C2CC(C)N2)=O)CCCC(C#N)C1 c1(C(N2CC(COC)(NC(=O)CCc3cnn[nH]3)C2)=O)nc2ccccc2[nH]1 C1(C)(NC(=O)NCC(c2ccccc2)(C)C)CC(CO)C1 CC(C)C(O)C(F)(F)C(=O)N1CCCN(C(=O)CCCCN2CCCC2)C(C)C1 C(=O)(C1CCc2ccccc21)NC1CN(C(C=CC=CCC)=O)C(C)CC1 C1(OCCOCCOC)CCCC(C(=O)NC(C)(C)CNC(=O)CC2(O)CCC2)C1 C1(CCNC(C23CC(F)(C2)C3)=O)(OC)CN(C(=O)CCC2CC2(Cl)Cl)C1 N1(N(C(c2nc(Br)sc2Cl)=O)CCN2CCOCC2)CCCC(C2CCCCC2)C1 Cn1cc(C(=O)NCC2CCN(C(C3(CO)CCCO3)=O)C2)c(O)nc1=O N1(C(C23OCC(C)(C2)C3)=O)CC2CCC(C1)N2C(C1(C)CC(F)(F)C1)=O C=CC(C)(CCOC)C(=O)NC(CNC(c1csc(CO)n1)=O)CCCC C1(C(=O)NCC23OCC(NC(=O)CCc4nccs4)(C2)C3)COC2COCC12 c1(C(=O)Nc2c(C)cc(O)nc2)cnc2c([N+](=O)[O-])cnn2c1 c1(C(N2CCC(C)(C(=O)NC(C(=O)OCC)C3CC3)C2)=O)cc2ccccc2o1 C1(N(C(=O)COC2CN(C(C)=O)C2)CC)CCN(C(=O)C(Cl)=CCl)CC1 CC1(CNC(c2csc(C3CCCO3)n2)=O)CCCN1C(=O)COC1CC1 c1(CNC(CC2CN(C(C=CC=CC)=O)C2)=O)cc2cc(Br)ccc2s1 c1(C(N(CCC)CCNC(c2nc(C(C)C)oc2C)=O)=O)cc2cnccc2o1 C1(NC(=O)NC2(C3CCC3)CCC2)CCCCC1C1CC1 S(=O)(=O)(c1ccccc1)N1CCN(C(=O)CNC2CNCC23CCCC3)CC1 C=CCCCC(C1CC1)NC(c1cn(CCNC(C2(C)CC(F)(F)C2)=O)cn1)=O c1(C(=O)NCC2(C)C(NC(C(CCC)C)=O)CCC2)c(C(N)=O)cccc1F c1(OC)ccc(CO)cc1C(=O)N(C(CNC(=O)CC1(O)CCCC1)C1CC1)C N1(C(COC(C)C)=O)CCC(C)(NC(=O)Cn2ncnn2)C1 Cc1cc2ccc(C(=O)NC3CN(C(=O)C4=CS(=O)(=O)CCC4)CC3O)cc2o1 c12nc(no1)CN(CCC1CC1)C2C.CCCCOCc1ccco1 N1(C(C2CC(C)(C(C)(C)C)C2)=O)CCC(NC(c2csc3nccn23)=O)C12CC2 N1(C(c2nc(C)sc2)=O)C2CCC1CC(CNC(c1ccnnc1Cl)=O)C2 N1(C(C=COCC)=O)CCC2(CCCC2NC(c2cc(C3CC3)ncn2)=O)C1 C1(NC(c2cccc(OC3CC3)c2)=O)CCC(n2cc(C3CC3C(=O)O)nn2)CC1 C=C(C)C1CCC(C)=CC1CC(N1CCC(C)(NC(=O)CC2CC(C)C2)CC1)=O C1(CC(=O)NCC2CN(C(c3nc(C)sc3)=O)CC2(C)C)CCn2cncc2C1 C1(CC)CN(C(=O)CC2CCCCC2O)CC1NC(C1(CO)CCCO1)=O C(c1ccc(F)cc1)=CC(=O)NC1C(NC(CN(C(C)=O)C)=O)C1 CC(c1ccccc1)=CC(=O)N(CCC(C(C)(C)C)NC(c1sccc1C)=O)C C1(C(N)=O)CN(C(C2CCN(C3CC3)CC2)=O)CCC1NC(c1ccsc1)=O Cc1nc(C=CC(=O)NCC2(NC(=O)COC3CCOC3)CCCCC2)[nH]c1C C1(NC(=O)CC2CCCOC2)CCSC12CN(C(c1ncc3[nH]ncc3n1)=O)C2 Cc1cn2c(n1)CC(C(N1CC(C(C)NC(c3cc(Cl)sc3Cl)=O)C1)=O)CC2 Cc1ncc(NC(=O)C(C2CCN(C(c3ccc(O)c(F)c3)=O)CC2)C)c(Cl)n1 C1(C(N(CC(C)(C)NC(=O)C(F)=C2CCCC2)C)=O)CC(C(F)(F)F)CO1 N1(C(CCCOC(C)=O)=O)CCSCC1C(=O)N(C(C)CCN(C)C)C c1(CC(N2CCC3CC23C(=O)NCCC23CC(CCO2)C3)=O)ccc(F)c(F)c1 C(=O)(C(C(C)O)NC(=O)OC)NC(CC)CNC(c1sccc1F)=O C1(NC(=O)CCc2ccccc2)C2CCN(C(=O)C=C3CCSCC3)CCC12 Cc1coc(C(C)C)c1C(N1CC(NC(C23CCC2C3)=O)C(F)C1)=O c1(C(=O)NCCN(CCC)C(C2(Cl)CC23CCC3)=O)c(Cl)ccc(F)c1F Cc1nn(C)cc1CNC(C1C=CCCN1C(=O)C(F)CC1CCOC1)=O C(C)(C)(CC(C(=O)NCc1ccc(F)cc1)N(CCCF)C1CC1)SC c1(N(C)C)ccc(C(=O)NC2CCCCC2CNC(=O)CCNC(=O)CO)nn1 N1(S(c2cccc(C#N)c2Cl)(=O)=O)CCc2nc(C3=CCC(O)CC3)sc2C1 C(C(=O)NC(C)(C)CCNC(C1CC=CCC1)=O)(C(C)C)NC(CC(C)C)=O c1(N2CCC(N(C(C(COC)O)=O)C)C2)ncnc2ccc(O)cc12 Cc1c(C(=O)NC2CC2NC(=O)Cc2cnc[nH]2)nn2ccccc12 c1(N2CCC(CC(C)NC(C3(CCC)CC3)=O)CC2)c(F)cccc1[N+](=O)[O-] C(=O)(C(=O)CC(C)CC)NC(CCCC)C(=O)N(C)CC1CCCN1CC c1(C(N2CCC(COC)C2(C)C)C(=O)NCCSC)ccc(Br)c(Cl)c1F N1(C(c2cc(CC)nn2C)=O)CCOCC(NC(C2(F)CC=CC2)=O)C1 C1(CNC(C2CN(C(C)=O)C2)=O)CCCN(C(C2NC(=O)OC2C)=O)CC1 c1(C(=O)NC2(CNC(C3C=CC=CC=C3)=O)CC2)cc2n(n1)CCOC2 c1(C(N2CCC(COC(C)=O)C2)C(=O)NCC(C)C)ccc(C(C)C)cc1F c1(C(N(C=O)Cc2cc(Cl)ccn2)C)ccc(Br)c(Cl)c1 CCCC(O)CC(=O)N1CCN(CCN(C)C(C2CC23CCOCC3)=O)CC1 N1(C(CC(C)OC)=O)CCCC(C)(CNC(=O)C=Cc2ccco2)C1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1C2CC(C(N3CCC(F)(F)CC3)=O)C1CC2 C1(NC(C(CCC)C#N)=O)CN(C(=O)CCc2ccc(Cl)cc2)CC2(CCC2)C1 C1(=O)C(CC)(CC)CNC(=O)C2CCN12.c1(CC)n[nH]cc1CC C(c1cccc(Cl)c1)=CC(=O)N(C)CC1COCCN1C(c1cc(F)n[nH]1)=O C#CC1(C=C)COCCN1C(c1n[nH]cc1C(C)(C)C)=O c1(OC)ccc(=NC(=O)CC2CCCCCCC2)[nH]c1C(F)(F)F C1(NC(=O)CCc2ncccn2)C2CN(C(=O)CCc3nc[nH]n3)CC12 N1(C(c2c(C)csc2)=O)CCCC(C)C1CNC(C1(C)CCC(F)(F)C1)=O Cc1ccc(NC(=O)C(N2CCC(NC(F)(F)C(F)(F)F)C(C)C2)=O)c(C)c1 c1(-c2ccc(C#N)nc2)cccc2c1CCN(S(=O)(=O)CC1CCCC1)C2 C1(NC(C(C)(C)NC(=O)NCCC)=O)CN(C(c2cccc(=O)o2)=O)CC1C CCC(O)C(C)C(=O)NCCNC(C1CCCN(C(=O)Cn2ncnn2)C1)=O C1(C(=O)NC2CCC(CNC(c3ncccn3)=O)CC2)CCC=CCCC1 C1(C(C(=O)NCC(C)N(C)C(C2(C(F)(F)F)CC(O)C2)=O)OC)CCCCCC1 c1(C(N(CC(CNC(C(CC)CCOC)=O)O)C)=O)cc2c(s1)CN(C)CC2 C1(COC)CN(C(C2CCC2)=O)CCN1C(=O)C(C1CCCCCC1)C N1(C(c2c(CCC)cccc2)=O)CC2CCOC2(CNC(c2nn[nH]c2Cl)=O)C1 c1(NC(C2C(Nc3c(C(=O)OC)cc(C)s3)C2)=O)ccc(F)c(C2CC2)c1.C(C)=O CN1CCC(F)(C2CC2)C1.C1(C(=O)NC)CC12CC(NC(C1(C=O)CC1)=O)C2 C12(OC)CCC(C(N3CC(NC(=O)C(F)=CC4CC4)C4CCCC34)=O)(CC1)CC2 C(CNC(C=C)CO)(C(=O)OCC)NC(C(=O)NCC)c1nccs1 N1(C(CC(C)C)=O)CCCN(C(C2CC3(C)CC2CO3)=O)CC1c1ccccc1 C1(CN(C)C(c2ccnc(C(F)F)c2)=O)CCCN(C(c2cc(Cl)n[nH]2)=O)C1 C12CCN(C(=O)CN3CCN(C(=O)OCC)CC3)C(C)C1C2.C1C(O)CCN1 c1(C(=O)NCC2(O)CN(C(C34CC(OC)C3C4)=O)C2)cccc2c1CCCC2 C1(n2cc(SCC)nn2)CCCCC1SC.C1(C(=O)NCCSCC)CC1C(=O)O N1(C(C2(CC#C)CCC2)=O)CCCC(NC(=O)CC(C2(OC)CCCC2)C)C1 N1(C(c2nnn(C(C)(C)C)n2)=O)CCC2(CCCCN(C(C3CC3(F)F)=O)C2)C1 c1(CC(=O)NCC(C2CC2)NC(C(OC)OC)=O)cc(Br)cc2c1OCC2 C1(C(N2CCN(C)CC2CNC(=O)CC(F)(F)Cl)=O)CCc2[nH]nc(O)c2C1 C=C(C)CC(C)C(=O)N1CCC(F)(CNC(=O)C(O)CCC)CC1 CC1=C(C(=O)N2CCC2CNC(c2ccc3oc(C)nc3c2)=O)C(=O)OC1(C)C C(=O)(C(C)(C)C(=O)N1CCN(C)C(CNC(c2nc(=O)n(C)[nH]2)=O)C1)N(C)C CCC(CC(=O)NC1CCN(C(=O)C=C(C)c2cccc(Cl)c2)CC1)C(C)(C)C C1(F)(C(=O)NC2C(CNC(CN(C)C(c3ccsc3)=O)=O)CC2)CC2(CCC2)C1 N#Cc1ccnc(C(N2CC3C(CNC(=O)C=CCF)C3C2)=O)c1 Cc1nc(C(=O)NCCC2CCC(NC(=O)C(C)(Cl)Cl)C2)sc1C N1(Cc2ncc(C)s2)CCCC(C2CCCN(C(c3cc(C)nn3C)=O)C2)C1 C1(C(=O)NC(CC=CC)C(=O)N(C2CC2C)C)CCC(O)CN1C C(=O)(CC1CC(O)c2ccccc21)N1CCCCC(CNC(C(C)(C)SC)=O)C1 N1(C(C(C2CCC2)OCC)=O)CCCC1(C)C(N1CCCC(CN=[N+]=[N-])C1)=O Nc1ccc(Br)c(F)c1C(=O)NCCNC(C1C2CCCCCCC12)=O Cc1nn(C)c(C(=O)NCC(C)CN(C)C(C2C(C)C2(F)F)=O)c1Br n1(CC(=O)NCc2occ(C(N(CC(C)C)C(C)C)=O)c2)ncn(C)c1=O C(=O)(C(CP(C)(C)=O)C(F)(F)F)NC(c1ccc(OC)cc1)C1CC1 N1(C(CC(=C)C)=O)CCCC(c2cn(C(c3ccccc3F)C)nn2)C1 CCC(CNC(C1Cc2nccn2C1)=O)(CC)C(=O)N1CCC(N2CC(O)C2)C1 Cc1cccc(CN2CCC(O)C2C(=O)Nc2ccc(Cl)c(F)c2)c1O N1(C(C2(CCC)CC2)=O)CC(NC(=O)C(CO)c2ccccc2)C(N=[N+]=[N-])C1 c1(SC)nccnc1NC(=O)CNC1COCC1NC(=O)CCC(C)N(C)C c1(C(=O)NCC(CC)NC(C2(SC)CCC2)=O)cc(Br)c([N+](=O)[O-])[nH]1 c1(OC)cc(N2CC3(CC3)CC2CNc2ccccc2SC)nc(S(C)(=O)=O)n1 N1(S(CCOC)(=O)=O)CCn2cc(C(N3CC4(CCOC4)C3)=O)nc2C1 CC12CN(C(=O)CCS(C)(=O)=O)CC1CN(C(c1n[nH]c3c1CCC3)=O)C2 N1(C(c2c(C)snn2)=O)CC2CC(C(=O)NC3(C4CC4)CCCC3)(C2)C1 C1(NC(CN(C)C(=O)C2CC2)=O)COCCC1NC(C1(CF)CC1(F)F)=O c1(C(=O)NCC(CNC(c2nc(C)nn2C)=O)S(C)(=O)=O)cc2ccncc2[nH]1 C1(N(C(c2cc(F)ncc2OC)=O)CC)CCCN(C(=O)OC(C)(C)C)C1C Cc1ncc(NCc2nncn2CC(F)(F)F)c(C#N)n1 c1(C(CO)NC(C2C=CC(NCc3ccnc(Br)c3F)C2)=O)ccc(F)cc1F N1(C(CCSCCC)=O)CC(C)CCC1CNC(=O)Cn1ccc(C)cc1=O C(C)(C)(CCCNC(C1(C#N)CC1C(F)(F)F)=O)NC(C1C(CC)C1)=O C1(CC(=O)NCCCc2nc(C)[nH]n2)C2CCCC2N1C(c1sccc1C#N)=O c1(C(=O)NC2CCN(C(CCCC=C)=O)CC2O)ccn2nccc2n1 C(C(CC(F)(F)F)NC(C12CCC(C1)C2)=O)NC(CC1(CC)CCC1)=O N1(C(CCCCSC)=O)CCC(N(C)C(c2ccnc(CO)c2)=O)C(C)C1 c1(OCCOC)ncccc1C(=O)NCC1CCN(C(=O)C(F)C2CCC2)C1 c1(-n2cc(OC)nn2)ccc(C(C2CCN(C(C3(F)CCCCC3)=O)C2)=O)cc1 c1(C(=O)NCCCN2CCC(NC(C(C=C)(C)O)=O)C2)ccc2snnc2c1 c1(NC(=O)NC)ccc(C(=O)NCC2CC2NC(c2ccc[n+]([O-])c2)=O)c(Cl)c1 CC1=CCC(C(N2CCC(C)(NC(=O)CCc3cc(C)[nH]n3)C2)=O)CC1 C12(C(=O)NC(CCN(C(c3cnc(C(=O)OC)s3)=O)C)C)CCCN1CCC2 C(CCC(C(=O)NCC(F)Cl)NC(c1nonc1N)=O)OC Cc1[nH]nc(C(F)(F)F)c1C(=O)N(C(C)C)Cc1ccccc1N1CCCCC1 Cc1ccc(NC(=O)C(C2CC2)N(C(=O)C(C)Nc2cnn(C)c2)C)cc1 N1(C(C2CC(C)(C)OCC2)=O)CCC2(CC1)OCCC2NC(=O)C1=COCCC1 c1(C(=O)NCCC2(NC(C(CCOC)C)=O)CCC2)ccc(OC)cc1F CN1CCC(C(=O)NCC#CC(=O)NC2CCCC2C(N)=O)C1 c1(CC(=O)NC2C(NC(c3c(C)coc3)=O)COC2)ccccc1S(C)=O c1(NC(C2(C)N(Cc3c(OC)ncnc3OC)CC2)=O)nccc2scc(Br)c12 c1(C(=O)NCCC(C)N(C)C(c2cnc(S)[nH]2)=O)cc2c(nc1O)CCCC2=O C1(Cl)(c2onc(C34CC(C#N)(C3)C4)n2)C2CCC(=O)C12 C1(NC(C=COCC)=O)CCN(C(C2CCC(F)(F)C2)=O)C(C)C1 Cc1cc(Cl)ccc1OCC(=O)N(C1CCN(C(C2CC2C#N)=O)CC1)CCO C(C(=O)N1CCCC(C)(NC(=O)CCCC(N)=O)C1)(C(F)(F)F)OC(C)=O C1(CNC(CCC(C)SC)=O)CCCCCN1C(=O)COC(F)(F)C(F)(F)F N1(C(C2(C#C)CC2)=O)Cc2nccn2CC(NC(c2cnc(C(C)(C)C)s2)=O)C1 C1(N(C(C(C)N2CCCC2)=O)C)CCCN(C(c2cnc(C(F)F)s2)=O)C1 N1(C(Cc2nc(C)[nH]n2)=O)CCCCC(CNC(c2cnn(C3CC3)c2C)=O)C1 c1(CC(C)NCC2CC(=O)N(Cc3ccccc3)C2)cc(Br)ccc1F C1(NC(CSC(C)(C)C)=O)CN(C(c2cncn2C2CC2)=O)CC12CC2 C1(CC(N2C(CC(=O)NCCn3ncc(C)c3)CC2)=O)CCOC1(C)C c1(CNC(c2cc(F)cc(F)c2)C(=O)OC)cc(F)cc(I)c1 c1(C(=O)NCC2CCCN(C(C(CC)n3cncn3)=O)C2)cc2ccccn2n1 CC1CCN(C(=O)C(C)(C)C(=O)N(C)C)CC1CNC(=O)C(C)(C)F C1(C(=O)NCCOCCC(=O)N(CC(C)SC)C)CCC(=O)N(C)C1 CCCCCS(=O)(=O)CC(=O)N(C)CC1CCN(C(=O)C(C2CCCCC2)F)C1 c1(C(=O)NC(CC)CNC(=O)C=CS(F)(F)(F)(F)F)cnc2cc(O)ccc2c1 C(=O)(CC(C)(C)C)NC(C)C(=O)NCC#CCNC(C1(C(C)(F)F)CCC1)=O N1(C(C(F)=C(C)C)=O)CC(C(=O)NCc2ccc(C#N)cn2)C(C)(C)C1 CC1CCCC(C(=O)NC(CNC(=O)CC2(N(C)C)CCCCC2)CO)C1 C(=O)(C1CCc2snnc21)NC1(CNC(=O)Cn2ccnn2)CC2CCC1C2 c1(C(=O)NC(C)C(C)NC(c2ccc(N)c(Cl)n2)=O)cc2cccnc2cc1F Cc1c(Br)ccc(NC(C2(O)CCN(C(c3c(F)cc(Br)cc3Br)=O)C2)=O)c1F C(N(O)C(=O)CCc1ccc(Cl)c(Br)c1)c1cn(CC(CC)O)nn1 C1(C2CC2)(C(N(OC)Cc2ccc(C)o2)=O)CN(C(C23COCC2C3)=O)C1 c1(CNC(C2CCCN(c3cc(CO)ccn3)C2)C)nc(C)cc(C)n1 c1(OC)cc(C)cc(CNC(C2CC2c2cc(F)ccc2F)=O)n1 C(=O)(C(C)CC(C)(F)F)NC1CCN(C(c2cccc(NC(C)=O)n2)=O)C1C C12(NC(C=CC=CC)=O)CCCCC1CN(C(C1CC3(CCC3)CO1)=O)C2 O=C1CCN(Cc2nc(C(F)(F)F)cs2)C(=O)N1CC12CCCC(CO1)C2 N1(C(C(c2cncnc2)C)=O)CC2CC1C2NC(=O)Cn1cc(Br)cn1 Cc1ccc(CN(C(C2CC2NC(c2ccccc2)=O)=O)Cc2ccccc2)nc1 c1(OC)ccc2c(c1)C(C(=O)N1CCN(C(c3ccnc(CO)c3)=O)CC1)CC2 c1(OC)cc(F)ccc1-n1cc(CC2CCCN(C(c3sncc3C)=O)C2)nn1 Nc1cccc(C(=O)NCC2(O)CC(CNC(=O)C(C3CCCCCC3)O)C2)n1 c1(C(N2C(CN(C)C(c3cc(CN(C)C)c[nH]3)=O)CCC2)=O)cc2n(n1)CCO2 C1(NC(C(=Cc2cccnc2)C)=O)CN(C(=O)Cc2nc(=N)[nH][nH]2)CCC1(C)C c1(C(N2CC(C)C(NC(=O)CC3CCC4CC34)C2)=O)c(Cl)nn(C)c1Cl C1(C(=O)NC(C2CCOC2)CNC(C2CC3C=CC2CC3)=O)CC2CCC1CC2 C1(N(C(CNC(N(CC(=O)OC(C)(C)C)CC)=O)=O)CC2CC2)CCCSC1 c1(C(N2CCN(c3nc(SC)nc(C)c3)CC2)=O)ccc(F)c(Br)c1F N1(C(=O)OC(C)(C)C)CCC2CC1CN(C(=O)CCC(N)=O)C2.c12csc(n1)S2 CCN=c1ccc(C(N2CC(O)(CNC(=O)CCn3cccn3)C2)=O)c[nH]1 C=C(C)C1OCCC1C(N1CCN(C(c2cc(O)ncn2)=O)C(c2cn[nH]c2)C1)=O C(CC#CC(C)(C)C)NC(C1(C#C)CN(C(C2CC2CCC)=O)C1)=O c1(C(=O)NCC2(NC(CC(C)n3cccc3)=O)CCOC2)cc2ccncc2s1 C(=O)(CC1=CCCC1)NCC(C)C(=O)NCC1(C(N)=O)CC1 CC(C)(CCC(=O)NC1CCCCN(c2ncns2)C1)[N+](=O)[O-] c1(CS(=O)(=O)NC)cc(OC)ccc1NC(C1CCN(c2ccncc2)C1)=O CC1CC(C(F)(F)F)N(C(=O)COc2cccc(Cl)c2)CC1C N1(C(C(C)OC(F)F)=O)CC(C)CN(C(=O)CCOc2cccc(Cl)c2)CC1C N1(C(C(=O)N(C)C)=O)CC2(CCNC(c3cc(Cl)cc(F)c3N)=O)CCC1CC2 N1(C(c2cc(C3CC3)[nH]n2)=O)CCC(CCNC(C23CCC2C3)=O)CC1 N1(C(CCC#C)=O)CCC(CC)C1C(=O)NC(c1cscn1)CO C1(CNC(=O)NCCC=CC)C2CC3C(C2)C13 N1(C(C2C(C)N(C(C3CCOCC3)=O)CC2)=O)CC(C2CCCC2)C1 C1(CC=C)(C(=O)N(C(C)C(=O)OCC)C)CCCN1C(=O)C(N)=O c1(C(N2C(CNC(c3cccc(OC)c3F)=O)CCC2)=O)cnc2cccnn12 c1(NCC(C)N(C(c2cccc(COC)c2)=O)C)ncnc2c1cnn2C(C)C C(CCC(C)C)(C(=O)NCCC(C)N(C(=O)COC(C)=O)C)NC(C)=O C1(C(N2CC(C)N(C(=O)COCCF)CC2)=O)CC2CCCCCC12 CC(C)CC(C)C(=O)NCCCN(C)C(C12CCC(C(F)F)(CC1)C2)=O C1(O)(CC(=O)Nc2cncc(Br)c2)CCN(C(c2cnc(Cl)s2)=O)C1 c1(CC)ncc(NC(c2cccnc2C(F)(F)F)c2nnnn2C)cn1 CCCCCC(O)C(=O)NC1CC(F)(F)CC1CNC(=O)C1=C(C)OCCS1 O=C(C1SCCc2ccccc21)NCC1CCN1C(=O)CC=Cc1ccccc1 CCCC(C)CC(=O)N(CCNC(C1CCC(C(N)=O)O1)=O)CCOC c1(CN(C(C)=O)Cc2ccccc2)nc(C)c(NC(C)=O)s1.n1(CC2CCCC2)cccn1 C1(CC)CCCN(CC(=O)NCc2cccc(NC(=O)Cc3ccccc3)c2)C1 C1(CCCC)CN(C(=O)C(C)SC(C)C)CCN1C(=O)CCCCC1CC1 C(CCCC(F)(F)F)NC(C(c1cn(C)nc1)NC(c1coc(CO)c1)=O)=O CC1=C(C)CC(C(N2CCC(OCC(=O)NCc3cc(C)sc3C)C2)=O)CC1 C1(C(=O)NCCC2(NC(=O)Cc3cc[nH]c3)CCC2)Cc2c[nH]cc2S1(=O)=O CC(CN(C)C)CCC(=O)NC(c1cccc(Cl)c1)CNC(=O)CCS(C)(=O)=O c1(CNC(C2N(C(c3c(C)c(I)ccc3)=O)CCOC2)=O)cc(Cl)c(F)c(Cl)c1 C1(CNC(c2n(CC)nnc2)=O)CC(O)CN1C(c1cc(C)[nH]n1)=O c1(C(C)NC2CCC(OCC(N3CCCC3)=O)C2)cc(Cl)sc1Cl c1(CNC2(C(N3CCC(n4cccn4)CC3)=O)CC2)cc(F)c(Br)cc1[N+](=O)[O-] c1(N(CCC)C)ccc(C(=O)N(C2(C)CN(C(C3CCC(=O)C3)=O)C2)CC)cn1 C1(C#N)(C(=O)NCC(CC)NC(=O)C(C)COC)CCS(=O)(=O)CC1 Cc1cnn2c1CN(C(c1ncc(I)s1)C(=O)Nc1cccc(Cl)c1C)CC2 C(=O)(C1COCc2ccccc21)NCC(CNC(=O)Cc1nc[nH]n1)O C(N=c1[nH]c(=NCC2CC3CCC3C2)[nH]c2cc[nH]c12)C1(c2ccc(Cl)cc2)CC1 c1(NC(c2ccc(Cl)cc2)C(N2C(C(=O)OC)CCC2)=O)cccnc1N(C)C N1(C(C(C)N(C)C)=O)CCC2CC(CNC(C3CC(C)(F)C3)=O)CCC2C1 c1(CC)cc(Cl)ccc1C(=O)NC1C=CCN(C(=O)CCNS(C)(=O)=O)C1 c1(CC(=O)NCCC(C)NC(=O)CC(C2CC2)C2CC2)nn(C)cc1Cl C1(C(N(C(C#C)C)C)=O)CC2(CC2)C12CCC2 CCCCCC(C)CC(=O)NC1CCN(C(=O)CC2CN(C(C)=O)C2)CC(O)C1 N1(C(C2(C(N(C)C)=O)CC2)=O)C2CCC1CN(C(=O)C(c1ccc(Cl)cc1)=O)C2 C1(C(=O)NC2CC(OC(C)C)C2)N(C(C2CCCCC(=O)N2)=O)CCCC1(C)C C(=O)(C1=C(C)OCCS1(=O)=O)NC1CC(CNC(C(=Cc2ccco2)C)=O)C1 c1(C(=O)NC2C3CN(C(C4CS(=O)(=O)CCO4)=O)CC23)cnn2cccnc12 C1(CC(=O)N(C2CC2)CC2(NC(c3cc(Cl)c[nH]3)=O)CCC2)COC(C(F)F)C1 c1(CC(=O)NCCN(C(CC(=C=C)C)=O)C2CC2)ccc(F)cc1C N1(C(CCC(C)NC(C23CC(C#N)(C2)C3)=O)=O)CC2(COC(=O)N2C)C1 c1(C(=O)NCCC(C)NC(C2CC(C#N)C2)=O)cc(C2(C)CC2)n[nH]1 C1(C(=O)NCC(CO)OC)CC(C)CN1C(c1[nH]nnc1C)=O c1(C(=O)NCCNC(C(CCC)O)=O)cnc(C)c(Cl)c1Br C1(CNC(C(C)(C)OC)=O)CCN(C(c2cc3ccccc3[nH]2)=O)C12CCC2 c1(C(N2CCCC(CCNC(C3(C)CCOC3)=O)C2)=O)ccc(P(C)(C)=O)o1 C1(CC)CCc2nc(O)c(C(N3CCC(C)(NC(=O)CC(F)(F)F)C3)=O)cc2C1 N1(C(C(C(C)CC)NC(C(C2CCC2)OCC)=O)=O)CCC(C2(C)CC2)C1 c1(C(=O)NCCCCC(C)NC(C2(NC(N)=O)CCC2)=O)cc(Br)ccc1F N1(C(C(c2cccc(F)c2)C)=O)CCCCC1CCN(C(=O)CO)C Cc1cc(C(=O)NC2CCC(NC(C3(C)CCCOC3)=O)CC2)cc(C)c1Cl c1(CC)cccc(C(N2CC=CC2CNC(c2cc(C3CCC3)no2)=O)=O)n1 N1(C(CN(C)C)=O)CC(F)CC1CNC(C1CC1c1ccco1)=O C(=O)(C1=C(CC)OCCC1)N1CC(NC(c2c(Cl)ccc(C#C)c2)=O)C(C)C1 CN1C(=O)CC(C(=O)Nc2nnc(CC(F)(F)F)s2)NC1=O c1(C(=O)NCCN(CC(C)O)C(c2cnc(C(C)C)[nH]2)=O)cnc(Cl)c(F)c1N c1(OC)cccc(CC(=O)OC(C)(CC(=O)O)c2cccc(F)c2)c1F C=C1C(C(=O)OC)C1C(=O)NC(C)C=CC(=O)NC(C)(C)CC1CCOC1 c1(C(=O)NC(CNC(C2CC(C(C)(C)C)C2)=O)CO)ccnn1CC(F)F N1(C(Cc2cccc(CC)c2)=O)CCC2CC1CN2C(c1csc(=N)[nH]1)=O N1(C(c2cc(C#N)[nH]c2)=O)CCC2(C1)CN(C(=O)C(F)=CCCF)CCO2 c1(-c2c(OC)cccc2F)ccc2[nH]c(C(=O)NCC3(C)CC3)nc2c1 N1(C(C(CC=C)C)=O)C2CC1CN(C(=O)Cc1ccccc1CC)C2 CC(C(=O)NOCCOCC(=O)Nc1ccc(F)cc1)C(C)c1ccc(Cl)cc1 N1(C(C(C(C)C)C#N)=O)CCCC(C)(C)C1C(=O)N(C)CC1CC(F)C1 C1(C(C)C)CN(C(C23CC(C)(CO2)C3)=O)CCN1C(=O)CCc1ccsc1Cl N1(C(c2n(CC)nnc2)=O)CC(C2CCCN(C(C3C4CCCOC34)=O)C2)C1 CC(C(=O)NCc1cn[nH]c1)(C1CCC1)NC(=O)CCc1ccccn1 N1(Cc2ccc3c(c2)OC(C)(CC)O3)CCCCC1C1CCCN1C(C)=O C1(N(C(=O)CCc2ccncn2)C)CCCCC1NC(C1(C)CNC(=O)C1)=O C(=O)(CCC(=O)OC)NC(C(=O)N(CC#C)CC1CC1)C Cc1cc(F)c(N)cc1C(=O)NCCC(O)CNC(=O)C1=CCCOC1 C1(C)(C(=O)NC2C(NC(c3c(CC)ncs3)=O)CC2)CCCCNC1=O c1(C(=O)NC2CC(F)(CNC(=O)CCC3CCCC3)C2)ncccc1C(F)(F)F CN1CCN(C(c2cc(N)cc(O)n2)=O)C(CNC(=O)CC2CCCCC2O)C1 C(CCC(C)(C)C(=O)N1CC(C)(C)C1C(=O)OC)NC(C(CC=C)OC)=O C1(CCNC(C2(Br)CC2)=O)CN(c2ccnc(-c3ccccc3)n2)CCS1(=O)=O C#Cc1cccc(C(=O)NCC2(F)CC(NC(=O)CCc3cc(C)n(C)n3)C2)c1 CCCCC(CC(=O)N1CCCCC1C1(O)CC1)NC(c1ccc(C#N)[nH]1)=O c1(C(N2CCC(C)(C(=O)NC3CCN(C4CC4)CC3)C2)=O)cc(F)ccc1F C1(C(N(C(c2cccnc2)C)C)=O)CN(C(c2ccsc2)=O)CC1(F)F c1(CSC)nc(-c2csc(COc3ccccc3)n2)n(-c2cccc(C)c2)n1 C1(NC(CN(CC(C2C(C)CCCC2)=O)C)=O)CC2CCCC1N2C CC1(C)CCC(C(=O)NCC(C2CCCC2)NC(=O)C(C)(C)c2cc[nH]n2)C1 C1(NC(C2(C)CN(C(C3C4CCCCCC34)=O)C2)=O)CCCN2CCCC12 Cn1cc(C(N2CCC(NC(c3ccncc3Br)=O)C2C2CC2)=O)ccc1=O N1(CC(N2CCC(O)(CNC(C(C)C3(O)CCC3)=O)C2)=O)CCP(C)(=O)CC1 c1(C(C(=O)NCC2C(CNC(CCC#N)=O)C2)O)ccccc1Br C1(N(CC(C)C)CC#C)(CNCC(=O)Nc2cnoc2C)CCCCC1 S(=O)(=O)(c1cc(C#N)ccc1F)Nc1nc(-c2ncc3[nH]nc(C)c3c2)n(C)n1 C1(C#N)(C(=O)NCCC(C)N(C(=O)CCC2CC2)C)CCOC1 C(CC(CC)C(=O)NCC(C)(CC)C(=O)NCCCCCCO)=CC N1(C(C2C(C)C2)=O)CCN(C2CN(C(=O)CN(C)C3CC3)C2)CC1 c1(C(=O)NC2C=CCN(C(C3N(CC)CCOC3)=O)C2)cc(O)ncc1Br Cc1ncc(Cl)cc1C(=O)N(C1CCN(C(=O)Cn2nccn2)CC1C)C c1(OC(C)C(=O)NCCN(C2CCCC2)C(c2cc(F)n[nH]2)=O)ccccc1F c1(C(=O)NC2CCCCC2NC(C2C=CCC2)=O)cnc2ccccn2c1=O c1(CCC(=O)NCC2(CNC(c3c(C)c[nH]n3)=O)CC2)c(C)nc(O)nc1C.C1CC1 c1(C(=O)NC2CC(O)CN(C(c3scnc3C3CC3)=O)C2)cc2cnccc2[nH]1 CCC(CO)C(=O)NC1CN(C(C2(c3ccc(C)nc3)CC2)=O)CC1C N1(C(C(C)(C)C2CCOC2)=O)CCOCC(C(=O)NCCN2CC=CCC2)C1 C1(OC)CCCC(C(=O)NC2CCCC2CNC(c2cnccc2Cl)=O)C1 C1(C)(CNC(c2c(OC)ccnc2O)=O)CN(C(=O)CCCC(N)=O)C(C)(C)C1 c1(C(=O)NC2(C)CCN(C(=O)C=C3CCCCC3)CC2)ccc2ncccc2n1 C(=O)(C1=CC2(CCN(C(=O)C=CC3CCCCC3)C2)C1)N(C1CCCC1)CC=C CC1(C)OCC2(CCN(C(=O)C(=O)NC3CCC(C)(C)CC3)C2)CO1 C12(NC(COCCCCCC)=O)CCN(C(=O)Cc3csc(C(C)C)n3)CC1C2 C1(NC(c2c(C)ncs2)=O)COCCN(C(C2(C#N)CC3CC3C2)=O)C1 C1(NC(c2ccsc2S(N)(=O)=O)=O)CCC2CC1CN2C(C12CC3CC1C2C3)=O C(=O)(C1CCc2c[nH]nc21)NC1C=CCC(C(N(C2CCCCC2)CC)=O)C1 N1(Cc2nc(C)c(C)s2)CCC12CCCC(C)(C)C2 c1(OC)nc(C(N2CCCC(OCc3ncc(C)[nH]3)C2)=O)cc2ccccc12 c1(N2C(C)CCC(C)(C)C2)cc2ccncc2cn1 c1(CC)ccc(C)c(NC(=O)CC2(OCC)CN(C(C3CCCC(=O)C3)=O)C2)c1 c1(C(=O)NCCC(CNC(c2c(CC)onc2C)=O)O)cccc(O)c1F C(=O)(CCC(=O)c1cccc(F)c1)N(CCCCNC(C1CC(Cl)(Cl)C1)=O)C c1(N(CC(C)C)CC)nnc(C2CCC2)n1CC1CCSC1(C)C N1(C(C(C)C2CC2)=O)CC(C(=O)NCCc2ccccc2O)CCC1(C)C N1(C(CCC(=C)Cl)=O)CCC2(CCCN(C(=O)CCSc3nccn3C)C2)C1 C(C)(C)(CCC(=O)NCC1(c2ccccc2)CC(NC(c2cnc[nH]2)=O)C1)OC N1(C(c2c(SC)ccs2)=O)CCC(NC(=O)C(C)Cn2ccc(C)n2)C12CC2 C1(NC(C2NC3CC2C3)=O)CCC(OCCF)CC1 Cc1nc2cc(C(=O)NCCC3CC(NC(=O)CCc4cnc[nH]4)C3)ccc2s1 N#Cc1ccc(N2CCCN(c3cnc(F)cn3)CC2)c(F)c1 c1(C(N2CCC(O)(C(C)NC(=O)C=CC3CCC3)C2)=O)c(Cl)ccc(Cl)c1O N1(C(C=CC(=O)OCC)=O)CC(NC(C2CCC(F)CC2)=O)C(C)C1 C1(NC(c2ccc3cccnn23)=O)COC2CN(C(=O)C(O)O)CC12 C=CCCN=C(NCC1CC=CCO1)NC(C)C1CC1 c1(-c2n(CCOC)nc(-c3cccc(OC)c3)n2)ccc(Br)c(Cl)c1 CCCC(CC)C(=O)N1CCOCC1(C)c1cn(Cc2ccco2)nn1 C(C1=CCN(C(=O)CC2CC23CC3)CC1)NC(=O)Cc1cc(Cl)sc1Cl c1(CC(=O)NC2(COC)CN(C(C3N(CC)CCC3)=O)C2)nn(C)cc1Cl Cc1cc(C(=O)NCC2CC(C)N(C(c3ccco3)=O)C2)cc(C)c1 Cc1cc(C(N2CC(F)(F)CC2CNC(=O)C(C)(C)C(C)C)=O)c(Cl)cc1N C(C(C)(C)C(=O)NCCC1CCC(C)(C)O1)N(C(=O)CCC1CCCOC1)C N1(C(N(C2CCCCC2O)C)=O)CCCCCC1c1ncon1 C(CC(C(=O)N=c1ccn(C(F)F)[nH]1)NC(=O)C(C)C1CC1)OCC C12(NC(CCC)=O)CC(C)(C1)OC21CN(C(C2CNC(=O)N2)=O)C1 C1(C(=O)NCC23CCN(CC2)C3)(COC)CCN(C(=O)C(C)SC(C)C)C1 c1(C(=O)NCC2CCC(C(=O)NC(CC#N)c3ccccc3)C2)ccc(Cl)cc1 C1(CC)CCCCC1OCC(N1CCC(NC(=O)C=Cc2sccc2C)C1)=O Cc1cc(Br)ccc1C(N1CC(CNC(C2CCC(C(N)=O)CC2)=O)C(C)C1)=O c1(C(N2CCC(C(C)NC(c3c(C)nncc3)=O)C2)=O)ccc2c(ccn2C)c1 CC1=NOC(C)(C(=O)NC2(C(=O)NCC(C)(C)C#N)CC2C)C1 CC1Cc2cc(CN3CCC(Nc4nc(Cl)nc(C5CC5)c4F)CC3)ccc2O1 c1(NC(C2(O)CCN(C(c3ccc(C(C)C)cc3)=O)C2)=O)cccc2nccn12 N1(CC(=C)Cl)CCC(C2CCN(C(c3csc(O)n3)=O)CC2)C1 C1(CCNC(CN(CC(C)(C)C)C)=O)CC(NC(=O)CC2(C#N)CC2)C1 c1(C2(C(N3C(CNC(c4sccc4Br)=O)CCC3)=O)CCCC2)ccc(Br)cc1 C(=O)(C(C)(C)C(=O)NC1CC2CC1N(C(c1csc(C(C)C)n1)=O)C2)NC N1(C(C2(C(CC)=O)CC2)=O)CCC(C(=O)NCC2CCC(C)C2)=C(F)C1 N1(C(C(C)SC(C)C)=O)CCOC2(CCN(C(=O)CCn3ccnc3)C2)C1 C1(c2cc(C(=O)OCC)no2)CCCCN1C(C1CCS(=O)(=O)N1)=O CN=c1[nH]c(=NCC2CCCSCC2)[nH]c(=NC2CCSc3c(F)cccc32)[nH]1 C1(C(=O)O)CCN(C)C1.n1(C2(C(=O)NC(=O)CC3(C4CC4)CC3)CC2)cc(Cl)cn1 N1(C(CCCOCCC)=O)CCCC(CNC(=O)C(c2cccc(C)c2)OC)C1 C1(C)(C(=O)NC(COC(C)=O)CO)CN(C(=O)C(C)C#N)C1 C1(NC(C2CC3(C2)CC3F)=O)CCN(Cc2cn(CC3CC4CC4C3)nn2)CC1 N1(C(C(CC)(C)O)=O)C2CCC1CC(N(C)C(c1csc(COC)n1)=O)C2 CC(Cc1ccco1)N=c1nc(N2CC(F)C(F)C2)c2[nH]ccc2[nH]1 CCCC(C)CC(=O)N1CC2C(CNC(c3c[nH]nc3-c3cccs3)=O)C2C1 C1(NC(CC2CC(=O)NC2)=O)CCCC(NC(=O)CC2COCCOC2)C1 c1(C(=O)NC2CC(F)C2)[nH]c2ccccc2c1-c1cccnc1OCC(F)(F)F N(C1CCc2ccc(Cl)cc21)C(C12CC1CN(C(=O)CC1COCCO1)C2)=O c1(C(=O)NCCN(C(C2COC(C)C2)=O)CC)cc2n(c1)CCSC2 c1(C(=O)NC(C2CCCC2)CNC(c2cnco2)=O)nocc1Br C(=O)(C(C)CN(C(=O)CN1CC(C)(OC)C1)C)N1C(CC)CC1 N1(C(C=COCC)=O)CCC(CN(C(C2CCN(C(C)=O)C2)=O)CC)CC1 N1(C(C=Cc2n(C)ccc2)=O)CCC2C(C1)CN2C(=O)C(C1CCOCC1)F C=CC(C)(C)C(=O)N(C)CCNC(c1ccccc1SCc1cccs1)=O C(c1cc(Cl)cc(Cl)c1)=CC(=O)NC(CC(=O)OC)Cc1ccc(C)cc1 C1(CCC(=O)NC2(C3CC3)CCC2)CCCN(C(C23CCCC2C3)=O)C1 CC(C)CC(C(=O)N(C(C)C(C)C)C)N(C)C(c1cccc(=O)o1)=O N1(C(CNC(N)=O)=O)CCC2CC12C(N1CC(N2CCCCC2)C1)=O c1(OC)cn(CC(N2CCOCC2CNC(=O)C(C)P(C)(C)=O)=O)c(C)cc1=O Cc1cc(N2CC(O)CC2C(=O)NCCOc2ccccc2Br)ncn1 C(CNC(=O)CN1CCC(C)CC1)(C(=O)NOC(CC)CC)OC CC(O)(CC(=O)NCC1CCCC1NC(C1(CC2CC2)CC1)=O)C(F)(F)F C1(CNC(c2scnc2Cl)=O)CCC2CN(C(=O)Cn3cnnc3O)CCC2C1 N1(C(c2c(CC)ncs2)=O)CCOCC1CC(=O)NCCCc1nc(C)no1 Cc1nc(C(=O)O)ccc1C(=O)NC(c1cn(Cc2ncccn2)nn1)C CCC(C)(C)C(=O)C(=O)N1CCN(C(C23CC(CC)(C2)C3)=O)CC12CC2 C=C(C)CC(C(=O)N1CCCC1CN(C)C(c1nccc(C)n1)=O)OC CC(C)(C)CC(C)(C)C(=O)NC(CNC(c1n[nH]c2c1CC1CC21)=O)C1CCC1 N1(C(=O)OC(C)(C)C)CCCC(C)(NC(N2CC(CCO)(CO)C2)=O)C1 C1(C(=O)NC2C(CC=C)CCC2)N(C(=O)CC2CCCN(C)C2)CC12CCCC2 C1(CN(C(C2(CNC(CN(CC)CC)=O)CCC2)=O)C2CC2)CCCOCC1 Cc1cc(C(N2CC3CC3(CNC(C3(C)CC4CC4C3)=O)C2)=O)nc(C)c1 C(=O)(C#CC1CCCO1)N(C)CC1(NC(C2CC2(F)F)=O)CC1 c1(C(=O)NCCCN(C(C(C=C)(C)C)=O)C)cccc2ncnn12 N#Cc1cc(F)ccc1C(N1CCC2(CC(NC(C3CCCS3(=O)=O)=O)C2)C1)=O CC(C)(N=[N+]=[N-])C(=O)N1CCCCC(CCC(=O)NCc2cc(O)cc(F)c2)C1 c1(C(=O)OCC(=O)NCC2CCC3CC23)nsc2cc(Br)ccc12 N(C(=NCCC1(O)CCC1)NCCN1CCCC1)CC(c1ccc(C)cn1)(C)C N1(C(C(=Cc2ccco2)C)=O)CCC(C)(C(=O)NC2CN3CCC2C3)CC1 N1(C(CCCC(C)O)=O)CCCC(C2CCN(C(c3nn(C)cc3Cl)=O)CC2)C1 C1(NC(CCC(N)=O)=O)CN(C(=O)COCC2CCCC2)CC2(CC2)C1 O=C1CCC(CC(=O)NCCc2n[nH]cc2C(=O)NCCC2CCCO2)CC1 C1(CC)CN(C(=O)CC(C)(C)N(C)C)CCN1C(=O)CC1(C)CCCC1 C1(CCNC(c2nccc(C)c2)=O)CCN(C(C2(C)CNC(=O)N2)=O)CC1(F)F C=CC(F)(F)C(=O)NC(CN(C(=O)C(C)Cn1ccc(C)n1)CC)CC C(=O)(C(C(=O)OCC)NC(=O)NC1(CC(=O)OC)CCC1)OCC CC(C)(CNC(=O)Cc1cncc(O)c1)CCNC(c1cncc(Br)c1)=O C=CCCN=C(NCC1COC(C)(C)C1)NCC1CCC2(CCCC2)O1 c1(C(=O)NC(C(CO)NC(c2c(OC)nsc2)=O)C)cc2sccc2cn1 C#Cc1cn(C)nc1C(=O)N(CCNC(C1(CCN(C)C(C)C)CC1)=O)C(C)C Cc1cccc(C(O)C(=O)NCCC(C)NC(c2ccsc2C)=O)c1F C1(C(N(CCC(C)C)CCC#N)=O)Cc2ccccc2CN1C(C1(C)CC1)=O C(=O)(CC(F)(F)CC(=O)NC1COCC1NC(C1COCCN1C)=O)OC CC1CN(c2ccc(CN(C)CCN3CCOCC3=O)cn2)CCO1 c1(CCC(=O)N(CCN(C(=O)CCNC(=O)NC)CC)CC)ncccc1F N1(C(c2cncc(OCC)c2)=O)CCN(C(c2c(CO)n[nH]c2C)=O)CC1C N1(CCNC(CCCOC)=O)CCCN(C(=O)C(C)Sc2ccccc2)CC1 CCCCCS(=O)(=O)CC(=O)NCCCC(C)(C)NC(=O)CC(CC)OC N1(C(C=CC)=O)CCC(c2ccccc2)(NC(c2cc(C)co2)=O)C1 C1(NC(COc2cn(C)nc2)=O)CCN(C(c2ccoc2)=O)CC1 c1(C(=O)NCCCC(C)NC(c2ccc(NC)cc2)=O)cc2n(n1)CCCC2=O C1(C(=O)NCC(Cc2ccccc2)NC(C(F)OC)=O)CCCCC1O C1(CN(C(c2ccc(CC)s2)=O)C)COCCN1C(C1CCCN1CC)=O CC1CN(C(C2OCC2(C)C)=O)CC1CNC(c1ccnc(CN(C)C)c1)=O C1(C(C(C)C)NC(c2cc(Cl)ns2)=O)CCN(C(C2CNC(=O)C2)=O)CC1 c1(C(C(=O)N(C)CC2CCCCN2C(C23CC(C2)C3)=O)O)cc(Cl)cc(Cl)c1 Cc1nocc1C(=O)NC1CC(O)(CNC(c2cccs2)=O)C1 C1(O)(CNC(c2ccc(OC)cc2C(=O)O)=O)CCCC12CCOCC2 N1(C(CC(c2cccc(F)c2)C)=O)CCN(C(c2cnc(Cl)s2)=O)CC(O)C1 C(C(CNC(=O)CCN1CCCCC1)C(F)(F)F)NC(=O)CC1CCOC1 c1(C(=O)NC2(CNC(C(C)C3CCCO3)=O)CCCCC2)cncc(O)c1Cl C1(c2cc(C)sc2)CCN(C(=NCC(C)C)NCCN(S(C)(=O)=O)C)C1 C1(CNC(C2CC=CCO2)=O)CCN(C(=O)CCc2sccc2Br)CC1 N1(C(CSCC(N)=O)=O)CCC(NC(=O)CC2(Sc3ccccc3)CC2)C(F)C1 c1(SC)cccc(C(N2CC(NC(=O)CN(C)C(=O)C3CC3)C(C)C2)=O)c1 C#CCCCCCCC(=O)NC1CCC(CCC(N2CCCC(CC)CC2)=O)C1 C#CCC(C)C(=O)NCC(F)CNC(=O)CCc1ccc(C(F)F)cc1 c1(C(N2CC(NC(c3cc(CC)[nH]n3)=O)C(F)CC2)=O)cnc2snnc2c1 C1(OC)CCC12CC(C(=O)NCCN(C(C1CCc3nccn3C1)=O)C(C)C)C2 C(CCCCC(=O)N1CCSC2CCC12)NC(c1cc(CCC)[nH]n1)=O n1(CC(=O)NC2CC(NC(CC)=O)C23CCC3)cc(C)c(O)nc1=O CCCCCC(CC)C(=O)NC1CC(CCNC(c2ncccc2F)=O)C1 c1(-c2cc(OCC)c(F)nc2)ccc2sc(C(=O)Nc3c(C)csc3C)cc2c1 N1(C(c2c(NC)cnnc2)=O)CCN(C(=O)C(=Cc2ccc(F)cc2)C)C2CC12 Cc1[nH]nc(C(N2CCC(O)(CN(C)C(c3cn[nH]c3)=O)C2)=O)c1Cl C1(C(=O)NCC2(OCCNC(C3CC3Cl)=O)CCOCC2)CC2(C1)CC(F)(F)C2 c1(CC(C(=O)NC2(CC=C)CN(C(=O)C(C)(CO)OC)C2)O)ccc(O)cc1 c1(C(=O)NC2CC(NC(=O)C(F)F)C2)ccc(-c2ccc(Cl)cc2)cc1 c1(C(C)C)nccn1CCN1CCC(N(C(=O)CC(C)c2ccco2)C)C1 CCCC(C(=O)N1CC(NC(c2cc(S(N)(=O)=O)cs2)=O)C2(CC2)C1)C(C)C C(=O)(CC(C)(C)C(C)(F)F)N1CCC(N(C)C(c2ccc3cncn3c2)=O)CC1 N1(C(c2c(C)cns2)=O)Cc2ccccc2CC1CNC(C1CCCOC1)=O c1(N2CC3(C(NC(c4c(C#N)cn[nH]4)=O)CCS3)C2)ccc([N+](=O)[O-])cc1[N+](=O)[O-] CCCC(O)CC(=O)NCc1ccccc1CNC(C1(F)CC=CC1)=O C#CCC(C(=O)N1CC=C(C)C1)NC(C1CC2CC2C1)=O C#Cc1cnn(CC(=O)NCC2CCN(C(=O)CC3CC(O)CN3C(C)=O)C2)c1 C1(O)(CNC(c2c(Cl)nsc2Cl)=O)CCCN(C(=O)Cc2ccc(Cl)cn2)C1 C1(CC(=O)NC(C2CC(F)(F)C2)C)C2CCC(C2)N1C(=O)CN1CC2CC2C1 c1(OC)ccc(C)c(C(=O)NCCC2CN(C(C3(C4CCC4)CC3)=O)CC2C)c1 N1(C(C)=O)CCN(C(C2(C)CN(C(c3ccc(C)c(F)c3)=O)C2)=O)C(C)C1 C(=O)(CCN(OC)C(=O)C1CCC(C)O1)N1CC(C#C)N(C)CC1 n1(CCOC)ccc(C(=O)NCC2CC(CNC(C3C(C)C3C)=O)C2)n1 C1(N(C)C(C2CCC3CC3C2)=O)CCC2CC1CN2C(=O)CC1CCC(=O)N1 N1(C(C2(NC(=O)OC(C)(C)C)C(C)C2)=O)CCS(=O)C(C)(C)CC1 c1(C(C)NC(C=CC(C)NC(=O)C(Cl)=CCl)=O)cccnc1O N1(C(c2ncn(CC)c2)=O)CCC2CN(C(c3cc4n(n3)CC(F)C4)=O)CC2C1 C1(CN(C(c2ccccc2Br)C)C)CCN(C(=O)CC2CCOC2)CC1 c1(C(N2CCC(c3ncccc3Cl)CC2)C(=O)NCCOC)nc(Br)ccc1F C1(c2nnc(N3C(c4ccoc4)CCCCC3)n2CC2CC2)CC2CCCCN2C1 CC12CC(CC(N3CCCC(C4CCCCN4C(c4ccsc4)=O)C3)=O)(CO1)C2 Cc1ccc([N+](=O)[O-])cc1C(N1CCCC(C)(NC(C2CCCCC2)=O)C1)=O C(c1ccc(O)cc1)=CC(=O)N(C(C)CNC(C1CN(S(=O)(=O)CC)C1)=O)CC c1(C(=O)NCC(C(C)C)NC(C(CCC)C#N)=O)nc2ncc(C)cn2n1 CCC(Cc1ccccc1)CC(=O)NC1CC(C)(NC(C2CN(C)C2)=O)C1 N(C1CCCc2[nH]ccc21)C(c1c(C)cc(Cl)c(Cl)c1)=O C1(CNC(c2cnc(CC)[nH]2)=O)C2CCC(C2)N1C(c1ccc(C#N)o1)=O N1(C(CCc2onc(C)n2)C)CCOCC(C(=O)NCc2noc(C(C)C)n2)C1 c1(C(N2CC3C(NC(=O)Cc4ccsn4)(C3)C2)=O)ccc2cccnc2c1F CC1CN(C(=O)CN2CC(C)(C)C2)CC1(C)C(=O)N(C)CC1(C)CCCO1 c1(N2CCC(CC)(CO)CC2)ncc(S(=O)(=O)N(C)CC2CCOCC2)cc1Cl c1(C(=O)NCC2C=CC(NC(C(CCCC)O)=O)C2)ccc2c(c1)CCN2C=O C(=O)(C1CCCc2c(O)cccc21)N1CCCN(C(C2(C)CC2)=O)CC1CO c1(C(C(=O)O)N(Cc2ccc(OC)cc2)Cc2cccnc2)cccc([N+](=O)[O-])c1 N1(C(CC2C(C)(C)C(O)C2)=O)CC2CC(NC(c3cc(Cl)c[nH]3)=O)CC1C2 C1(NC(c2cc(C)nn2C)=O)CCN(C(C2CCC(=O)C(C)C2)=O)CC12CCC2 c1(C(=O)NC2CC2)ccncn1.C1(C(N2CCCC2)(C)C)CCCN1C(=O)C=CCF C1(=CC(=O)NCC2(C)N(C(CCSCC(C)C)=O)CCC2)CN2CCC1CC2 Cc1cc(CNC(C2(NC(=O)C(c3ccccc3)F)CCSC2)=O)cc(C)c1 CCC(CC(C)C)C(=O)NC12CC1CN(C(=O)C=Cc1nc(C)c(C)[nH]1)C2 C(=O)(CCCC(=O)NC1CN(C(=O)CCCn2cccn2)C(C)(CC)C1)NCC N1(C(=O)Cc2ccc(Br)cn2)CC2CN(Cc3ccccc3I)CC2C1 c1(NC(N2CC(F)(c3ccccc3)C2)=O)ccc(-c2cncnc2)cc1F n1(CC#C)cnnc1C(=O)NC1(CCC(=O)N(C)Cc2cncs2)CCCC1 C1(NC(c2c(C(C)(C)C)[nH]cn2)=O)CC(N=c2nc[nH]s2)C1 C1(CCNC(c2cocc2C)=O)(NC(C(C2CC2)SC)=O)CCOCC1 C(=O)(C(C(C)C1CC1)N1CCC(CSC)C1)NCCSC C1(C(=O)NCCCNC(c2ccccc2-c2nc[nH]n2)=O)CCc2ccnn2C1 C12(CNC(=O)CSCCC3CCCCO3)CC1CN(C(C13CC(F)(C1)C3)=O)C2.N CS(=O)CCC(=O)NC1C=CCN(C(c2cc(COC(C)(C)C)on2)=O)C1 C1(C(N2C(CNC(CCCNC(C)=O)=O)CCC2)=O)CCS(=O)(=O)N1C C1(N(C(c2cc(CC)[nH]n2)=O)CC2CCCCO2)C2CCC1CNC2 C1(NC(C2CCOC2C(F)(F)F)=O)CN(C(c2c[nH]ccc2=O)=O)CC2(CC2)C1 C=Cc1ccc(C(=O)NCCOC2CN(C(c3cnn4cc[nH]c34)=O)C2)cc1 N1(C(C)=O)CCN(C(=O)C(C)(C2CC2)N(C(=O)CC(C)C)C)CC1 c1(C(=O)NCC(CN(C(C(C)OCCC#C)=O)C)C)oc(C2CCC2)nc1C C(=O)(C1=CCCCCC1)NCC1N(C(C(C)=CC2CC2)=O)CC(F)(F)C1 N1(CC)C2CCC1CN(C(=O)CNC(C)=O)C2.c12nn(C)c(c1Br)NC2=O N1(C(C2CC(CN(C)C)C2)=O)CC2CC(C1)N2C(=O)C(C)(Cl)Cl C1(C(N2CCC2C(C)C)CC)CCN(Cc2[nH]nnc2C)C1 c1(CNC(c2nnnn2CCN2CCOCC2)C2CC(=C)C2)cnc(C(C)C)o1 C(=O)(C1CCc2ccccc21)N(C(C)C(N1CCN2CCCCC2C1)=O)CC c1(SCC(=O)NC(C2CCN(C(C3(CO)CCCCO3)=O)C2)CC)ccccc1Cl c1(CC)ccc(F)cc1NC(=O)CCCCCNC(c1ccnn1C)=O c1(COC)nc(C)c(C(=O)NC2COCCC2NC(=O)C(O)CC2CC2)s1 Cc1cncc(F)c1C(=O)NC1CC(CNC(=O)CN2CCCC(N(C)C)C2)C1 c1(C(C)=O)c(C)[nH]c(C(=O)NC(C)CNC(=O)CCSc2cccc(C)c2)c1C c1(C(=O)NCCC2CN(C(=O)CCN3CCOCC3=O)C2)cc(F)c(F)cc1O N1(C(C2CCCN(c3cc(C)[nH]n3)C2)=O)CCC(O)CC(C)(C)C1 N1(C(Cc2ccc(C)s2)=O)CC2(COC(CNC(C3(C)CCC3)=O)C2)C1 Cc1cc(C(=O)N(CC(C)NC(c2cn(CCF)nn2)=O)C)c(C)c(C)c1 c1(C(=O)NCC(CNC(C(C)=CC)=O)F)csc(CCC)n1 C(CNC(=O)CSCCC(C)C)(CC(C)C)NC(c1cnc(OC)s1)=O CC(CCNC(c1ccc(-c2cccnc2)cn1)=O)CCNC(=O)C1=CCOC1 c1(-n2ncc(C(=O)NCCOCC(C)(C)C)c2)ccc(Cl)c(Cl)c1 CC1(C)NC(=O)CC1C(N1CCCC(O)(CCNC(C2(S(C)(=O)=O)CC2)=O)C1)=O C1(C(=O)NC2CC(OCC(=O)NC3C(C=C)COC3)C2)CCCC(C)(C)C1 c1(C(=O)NC=O)cc(C(N)=O)cc(F)c1.CC1(O)CNC(=O)C2CN(C2)C(=O)NC1 C(=O)(CC(C)(C(F)(F)F)Nc1cc(OC)c(Cl)cc1I)OC C(CCCC(=O)NC(C)CCC1CCCC1)NC(C(C1CC1)SC)=O C1(CNC(CC(=C)C)=O)CCC2(CCN(C(=O)C(CC(C)(C)C)OC)CC2)O1 CC(C)CCC(C(=O)Nc1cccc(N(C)C)c1)NC(=O)C(C)C1(O)CCC1 c1(-c2cn(CC)nc2)cnc2ncc(C(=O)NC(c3ccno3)C)n2c1 c1(NC(c2ccns2)=O)nnc2ccc(-c3cnccn3)cn12 S(=O)(=O)(c1cccc(-c2c[nH]nc2C(=O)NCc2nc(CSC)no2)c1)NCC N1(C(C(C)(C)OCCC)=O)CC2(C)CC1(C(=O)NCc1ncc(C)cn1)C2 N1(C(C(=O)NC(CC)(C)C)CCC2(C)CC2)CCCC(C(=O)OC)(OC)C1 C(c1ccc(C)cn1)=CC(=O)NCC(CCNC(C1C(COC)C1)=O)O N1(C(c2ccc(CCC)s2)=O)CCCC2(NC(C34COC(CCO3)C4)=O)CC2C1 C1(N(C(C)=O)CCc2noc(=O)n2C)CCN(C(C23CC(F)(C2)C3)=O)C12CCC2 CCCC(CC)C(=O)N1CCC=C(CNC(=O)C2=NOC(C)C2)C1 c1(C(N2C(CNC(c3ccc(CF)cc3)=O)CC2)=O)ccc2c(c1)OCC2 c1(NC(C(N2C(CNC(c3c(CC)nn[nH]3)=O)CC2)=O)C)ccc(Cl)cc1Cl c1(C(=O)NC2(C)CCN(C(CCC(=C)Cl)=O)C2)cc(F)ccc1O c1(C(=O)NCC2N(C)CCN(C(C3CC(SC)C3)=O)C2)cccc2c1CNC2=O c1(CC(N2CCC3CN(C(=O)C(F)(F)C4CC4)CC23)=O)ccc([N+](=O)[O-])cc1Cl C1(NC(C(C)=CC)=O)CC2(C1)CN(C(=O)C(C)SCC1CCCO1)C2 N(C1c2ccccc2CC1C)C(=O)NCc1cc2cc(C)ncc2cc1 C(=O)(C1=CC2CCCCC12)N1CCC(NC(CN(C(C)C)C)=O)C(O)C1 N1(C(c2ncn(C)c2)=O)CCCC(CO)(NC(=O)COC2CCCCC2)C1 Cc1c(Br)ccc(NC2CC(CNC(=O)CCc3ccc(F)cc3)C2)c1[N+](=O)[O-] c1(C(C(=O)NC(CC)(C)C)N(N2CCCC2)C)ccc(OCC(N)=O)cc1 c1(-c2cc(C(=O)NCC3C(NC(C(CSC)O)=O)CC3)n[nH]2)ccc(C)cc1 c1(N2CC(C)C(F)C2)cccc(S(=O)(=O)NCC(c2ccnn2C)N(C)C)n1 N1(C(C2(CCCC)CCC2)=O)CCCC(CNC(c2cc[n+]([O-])cc2)=O)CC1 c1(C(=O)NCCCN(C(=O)CC2CCCC2C)CC)cccnn1 Cc1cc(Cl)ccc1C(N1CC(CNC(=O)COCc2nccn2C)C(C)C1)=O S(=O)(=O)(c1c(Cl)ccc(F)c1F)N.c1(C(=O)OC)cc(SC)n(C(C)(C)C)n1 CC1(C)CC(NC(c2cnn[nH]2)=O)CN(C(=O)C(=Cc2c[nH]cn2)F)C1 c1(NC2C=CCC(C(F)(F)F)C2)ncnc2cc(C3CC3)nn12 C(=O)(CC(C)C(C)(C)NC(=O)C(C)c1cc[nH]n1)Nc1c(CC)nc(C)cc1 N1(C(C2N(C(C)=O)CC(O)C2)=O)CCN(C(=O)CC(C)C)C(C#N)C1 N1(C(C(CNC(CCOC)=O)(F)C(C)C)=O)CCCC2C(=O)NCC12 C1(C(=O)NC(C2CCCN(C(C(C)O)=O)C2)C)CNc2ccccc2O1 O=C(CCCOC)NCC1(CCNC(=O)CNC(c2cccnc2)=O)CC1 CC1(C)CC(C(N2CCCC(F)(CNC(C3CCC3)=O)C2)=O)CC(C)(C)C1 N1(C(C2N(C)CCCC2)=O)CCC(F)(F)C(N=c2nc[nH]cc2C#N)C1 N=c1ncc(C(=O)NCC2CN(C(=O)CC3CCCCCO3)CCO2)c[nH]1 N1(C(C2(C)C(C)CN(C(=O)C(C3CCCCC3)F)C2)=O)Cc2cccnc2C1 C(=O)(C1=CCCSC1)NC(C(=O)NC1CCN(CC)CC1)Cn1cncn1 c1(C(=O)NC2CCN(C(C(CC)(C#N)CC)=O)CC2O)cccc(P(C)(C)=O)c1 C1(C)(C(=O)NC(C(=O)OC)CO)CCCN(Cc2ccc(N)c(Cl)c2)C1 c1(C(=O)NC2CC(CNC(C(C)=C(CC)C)=O)C2)cc(COC)oc1C c1(C(N2C3CC(NC(C(c4ccccc4)C)=O)C3CC2)=O)cc(Cl)c(F)c(Cl)c1 N1(C(Cn2c(C)ccn2)=O)CCC2(NC(=O)CN3CCSCC3)CC2C1 C#CCCCC(C)C(=O)N1CCN(C(=O)Cc2cccc(C#N)c2)CC1COC CC(C)(C)CCC(=O)N1CCCC(CCCCNC(c2n[nH]cc2F)=O)C1 CC(C)C(C)(CNC(=O)C#CC1CC1)NC(=O)Cc1ccc(-n2ccnc2)cc1 C(=O)(C(C)(O)C(F)(F)F)N1C(CC(=O)NCC(c2ccccc2)(C)O)CCC1 c1(OC)ccc(CN2CC3CC2C3C(N2CCC(N(C)C)CC2)=O)c(F)c1F C=CCC(C)C(=O)N(C1CC(C#N)C1)CC(=O)N(C)CC1(C(=O)OC)CC1 CC1CCC(CNC(=O)CCc2cn(C)nn2)N(C(c2cnc(C(C)C)[nH]2)=O)C1 N1(C(C(CCC)N(C)C)=O)C(C(=O)NCCNC(=O)NC)C2CC(O)C1C2 CC1(C)CC(O)CCN(C(=O)C(F)CC(C)(C)NC(=O)CC2CCCO2)C1 C1(C(=O)NCC(CN(C(c2c(C)nc(C)s2)=O)C)C)C(C)OC(C)C1C c1(C(=O)NCC(F)CNC(=O)C(F)CC2CCC2)noc2c1CCCC2 c1(C(N2C(CCNC(C3(C)C(C)C3)=O)CSCC2)=O)cc2ccc(Cl)cn2c1 C1(C(=O)NCC(CC)C)CC(N=[N+]=[N-])CN1C(c1cc2occc2[nH]1)=O c1(C(=O)NCC2CC2C(=O)NC2(CCO)CCC2)ccnc(-n2cccc2)c1 c1(C(=O)NC2C(CNC(=O)C=CC=C(Cl)Cl)CC2)cc2nc[nH]c2cc1F c1(-c2cn(CCNC(C(C)NC(c3ccc(C)o3)=O)CO)nn2)ccc(=O)oc1 C1(OC)CC(C(=O)NC2CC(CNC(C3CC4(CCC4)C3)=O)C2)C12CCC2 C(CS(=O)(=O)CC(=O)NCC(C1CCCC1)NC(=O)C(C)O)OC C(CCN(C(=O)C(C(C)C)NS(N)(=O)=O)C)(C(C)C)NC(Cc1nc(C)sc1)=O C1(CNC(C(=O)NC(c2ncnn2C)C)=O)CCC2(CCCC2)O1 CCS(=O)(=O)NC(C)C(=O)N(CC(O)CN(C(=O)CCOCCN(C)C)C)C n1(CC(N2C(CNC(COC)=O)C=CC2)=O)c(C(C)C)nc2ccccc12 CC1CCCN(C(=O)C(c2cccs2)NC(c2ncn3c2CCC3)=O)CC1 c1(OC)nc(C)ncc1C(=O)NCCC1CN(C(=O)CCc2cn(C)nn2)C1 c1(C2OCCN(c3n(CC=C)c(-c4ccoc4C)nn3)C2)ccc([N+](=O)[O-])cc1 c1(CN2CCCC2c2cn(NC(CC3(SC)CC3)=O)nn2)c(C(C)=O)c[nH]c1C N1(C(CC)=O)CCC(C(F)CNC(C2CCCN2C)=O)CC1 C1(OC)C2CN(C(=O)Cn3cc(C(c4ccc(F)cc4)O)nn3)CC12 c1(CCNC(=O)NCC2CCCC23CC3)ccccc1-c1cncnc1 CC1CCC(F)(C(=O)NCc2ccccc2CN(C)C(c2c[nH]c(=N)s2)=O)CC1 C1(CC)(CC)CC(NC(=O)CC2CCOCC2)CN1C(=O)C(C1CCC1)OC CC1C(=O)NC(=O)CN1C(=O)CC1(N(C)C(C23CCN(CC2)C3)=O)CC1 C1(C(N(C)CC2(O)CCOC2)=O)CN(C(=O)CCS(C)(=O)=O)CC(C)(C)C1 c1(NCC=CCNC(CC2(CSC)CC2)=O)ncnc2sc3c(c12)CCC(C)C3 N1(C(C2C(NC(C3N(C)CC4(CC4)C3)=O)CC2)=O)CCC12CCSCC2 c1(C(=O)OC)ccc(C(N2CCC(N(C(=O)C(C)N(C)C)C)C2)=O)c(F)c1 CC1CN(C(=O)C(C2CCOCC2)O)CCN1C(=O)C=CC1CCCN1C n1(CC(=O)NC(C2CCCC2)CNC(C(n2ncc(C)c2)C)=O)ncn(C)c1=O c1(C(=O)NCC(C2CCC2)NC(=O)CNC(c2ccco2)=O)ncc(Cl)cc1F C(c1ccc(C)cc1C)=CC(=O)NCCC(C)NC(Cc1cccc(C#C)c1)=O C1(NC(C2(C)CCC(C)CC2)=O)CCC2CC1CN2C(c1ncnc(O)c1F)=O C12CC(C13CCC3)NC(=O)C2.c1(CN(C)C(C2CN(C(N)=O)C2)=O)nc[nH]n1 c1(CC)cccc(C(=O)NCC(C)CN(C)C(C2CN3CCC2CC3)=O)c1F c1(C(C)C)cccc(C(N2CCC(CNC(=O)C(C)(C)c3cncnc3)C2)=O)c1 Cn1ncc2cc(C(N3CC=CC(NC(c4cnccn4)=O)C3)=O)sc12 c1(C(=O)NCC2C(C(N3CC(NC(N)=O)C3)=O)CCO2)ccc(F)cc1F C(CCS(C)=O)(C(=O)NCC1CCC1NC(=O)C=Cc1ccccc1F)N(C)C N1(C(C2(CCOCC)CCC2)=O)CC(Nc2nccc(CO)n2)C(C)C1 CC(C(=O)N1CCCC(CN(C(=O)Cn2nnnc2C2CC2)C)C1)P(C)(C)=O C1(NC(C2C3CCN(C(C4CCOCC4)=O)C23)=O)CC(C2CCCC2)C1 c1(C(N2CCC(C)(CNC(C3(CO)CC3)=O)CC2)=O)c(F)ccc2n[nH]cc12 C1(C(=O)NC(C)CCc2cn[nH]c2)CN(C(=O)COC(N)=O)CCC1(C)C C1(C)(C(N2CC3C(NC(c4c(COC)cc[nH]4)=O)C3C2)=O)CCC2CC2C1 C#Cc1ccc(C(=O)NCCCN(C(C2CCCSC2)=O)C(C)C)nc1 N1(C(C2C3CN(C(c4ccc(SCC)cc4)=O)C2C3)=O)CC2C(C1)C2(C)C C=CC1(CC(=O)NCCC2CCCCN2C(C2CCCC2(F)F)=O)CCCCC1 C1(CN(C(c2coc(C(F)F)n2)=O)CC)CCCN1C(C1CCC(C)O1)=O c1(OCCC)ccc(CCC(=O)NCC2CCN2C(C2CC(F)C2)=O)cc1 c1(CNC(C2(CNC(C(C)n3cncn3)=O)CCC2)=O)ccc(F)cn1 N1(C(C2(C)CC(O)CN2C(C2CCC2C#N)=O)=O)CCC2(CNC(=O)C2)C1 N1(C(C(C)(C)n2cnnn2)=O)CCC(C(=O)NC2C(C(=O)OC(C)(C)C)C2)=C(F)C1 Cc1ncc(C(N2CC(C(=O)NC(c3nccc(O)n3)C)C(F)C2)=O)c(C)n1 c1(C(N2CC(NC(C(C)CO)=O)C(c3nccn3C)C2)=O)ccn2ccnc2n1 C#CCCCCCC(=O)N1CCCC(CC(N2CCSCC2C2CC2)=O)CC1 c1(OCC)ncc(C(=O)N(CC(C)(C)CNC(=O)CC#N)C)cn1 Cc1ccc(S(=O)(=O)N2CCC(C(N3CC(N(C)C(C)C)C3)=O)CC2)cc1C CN1CCN(C(=O)CC2CCOC2(C)C)C(CNC(=O)CSCC(N)=O)C1 c1(C(N2CCC(C(C)(C)C)(CNC(CC(=C)C)=O)C2)=O)cc2sccc2n1C CC1(O)CC(C(=O)NC(C2CCCCC2)CNC(=O)C2CC2)C1 N1(C(Cc2cc(C)cc(F)c2)=O)CCC2CN(C(c3n[nH]cc3C)=O)CC12 C(=O)(CCC(F)(F)F)NC1(C(N(C)CCc2cccnc2)=O)CCC1 N1(C(c2cn(C)nc2C(C)(C)C)=O)C2CCC1C(NC(=O)C1CC1)C2 c1(-c2cn(CCNC(C3C(F)(C(=O)OC)C3)=O)nn2)cc2ccccc2s1 Cc1cnn(C(C)C)c1C(=O)NCC1CN(C(C2CC(C)(F)C2)=O)CC1O Cc1nn(C)c(C)c1C(=O)NCC1COCC1NC(=O)Cc1cc(F)ccc1O n1(CC)cnc2[nH]c(=NCCNS(C)(=O)=O)nc(N3CCC4(C)C(C3)C4(Cl)Cl)c12 c1(C(=O)NCC2CN(C(CCc3cc(C)no3)=O)C(C)C2)ccc(Cl)c(N)c1 C1(C(NNC(c2cc(C)n(C3CC3)n2)=O)=O)CC(C2CCC2)C1 C1(NC(c2ccc(C)s2)=O)(CO)CCCN(C(=O)Cn2cccc(N)c2=O)C1 c1(CCCCCN2C(=O)C2)nc(O)n[nH]1.CC(C(=O)N1CCCC1)SCC1CCCO1 c1(OC)cc(C(=O)NC(CNC(=O)C(N2CCC(C)C2)=O)C2CCC2)cc(C)n1 C=CCCCC(C)(C)C(=O)NCCN(C)C(c1ccc(OC2CC2)cc1OC)=O c1(C(=O)NC2(CC)CN(C(c3csnc3OC)=O)C2)cc(C)c(F)c(C)c1 Cc1cc(C)c(COC(=O)C(C)N2CC(C)C2)cn1 C1(CNC(c2n(CCOC)nnn2)c2cnc(Cl)s2)CC2CC1CC2O C1(NC(C=CCC)=O)CC2CC1CN2C(c1c(C)nn(-c2ccccc2)c1Cl)=O N1(c2n(Cc3cc(C)on3)c(C3CCOC3)nn2)CC2CC(F)(F)C2C1 C1(c2nnnn2CCCSC)(NCc2cnc(CC)o2)CCOCC1C C1(CC)CN(C(=O)CC2OCCO2)CC1C(=O)NCC(C)(O)C(F)F CCCC(O)C(=O)NC1(COC)CCN(C(c2ccnc(-c3ncc[nH]3)c2)=O)C1 CCCC(CNC(c1ccsn1)=O)NC(=O)Cc1cnc(C)[nH]1 CC1CCc2nc(NC(=O)C(=O)Nc3nnc4n3CCNC4=O)c(C#N)cc2C1 S(=O)(=O)(c1cc(Br)ccc1Cl)NC1CCC(CC(N2CC(O)C(F)C2)=O)CC1 C1(NC(c2c(OC)nccn2)=O)CN(C(C2CC2(C)C)=O)CC(F)(F)C1 C#CCC(C)(C(=O)NC1COCC1N=[N+]=[N-])NC(=O)CCOCC(F)F N1(C(c2c(CC)onc2)=O)CC2CN(Cc3ccc(OC)cc3)CC2C1 C1(NCC)CCCC1C(=O)NCC1(NC(=O)C2CC2)CCC1 CCC(CC(=O)N1CCN(C(C2OCCC2(C)C)=O)C(CC)C1)C(F)F c1(C(=O)NCCCOCCC(N2C(C)(C)C(O)CC2)=O)c[nH]c2cnccc12 C=CC1CCCN(C(=O)CCC(C)NC(C2(N3CCCC3)CC2)=O)C1 C1(C(=O)NCC(C)N(C(COCCC=C)=O)CC)CCCOC1 N1(C(C2(CC#C)CC2)=O)C2CCC1CC(NC(c1csc(C)c1C)=O)C2 C1(NC(CC2CC(SC)C2)=O)CC2(C1)CC2NC(c1cc(C)no1)=O Cc1cnn(C)c1CC(=O)NC1CN(C(c2coc(C(C)(C)C)n2)=O)CC1O N1(C(C(C(C)C)NC(C)=O)=O)CCN(C(=O)CCc2ccc(Cl)nc2)CC1C N1(C(COC(C)=O)=O)CCCC(CO)(CNC(c2cc(Cl)n[nH]2)=O)C1 c1(NCC(C2CC2)OC)ncc(C)cc1Br CC1CCc2ccccc2N1CCNC(N1CCN(C(N)=O)c2ccccc21)=O C12(C(=O)NCC(C)N(C(=O)C(c3cccn3C)=O)CC)CCCC1OCC2 C1(NC(COC)=O)CN(C(c2cccc(-c3cccc(C)c3)c2)=O)CC1(C)C C1(O)(CC(=O)NC(CNC(CSCCC)=O)C2CC2)CCC1 C(=O)(C1=CCc2ccccc21)NCCN(C(CCC(C)N(C)C)=O)C c1(NC)cnc(C(=O)NCC2(C(=O)NC3CCCC3CCO)CCC2)cn1 C1(C(N2CC(OCCNC(c3coc(O)n3)=O)C2)=O)CCC2(CCC2)C1 c1(CC)[nH]nc(Cl)c1C(=O)NCC(O)CN(C(=O)C(CC1CCCCC1)OC)C c1(CC(=O)N(C)CC2N(C(C(C(C)C)SC)=O)CCCC2)cccc2c1OCO2 CC1(C)CC(=O)CCC1C(=O)NC1(C(=O)N(C)C)CCCCC1 S(=O)(=O)(c1c[nH]c(-c2ncco2)c1)NC(C1CCN(c2ccccc2Cl)C1)=O c1(C(N2CC(NC(C3CCCCC3(F)F)=O)(CO)C2)=O)n[nH]c2c(F)cccc12 N1(C(c2scc(C(C)=O)c2)=O)CCCC(CO)(NC(=O)CC2CCCC2O)C1 C1(CC(=O)NCCCOCCNC(=O)C(F)(F)c2ncccn2)CCCCC1 C1(CC(=O)NCCCN(C(=O)CC(C)n2cccn2)C(C)C)CCCCC(=O)N1 C1(CNC(Cc2cc(C)on2)=O)CCN(C(c2cc(Br)c(C)o2)=O)CC1 C(=O)(C1=NOC(C)C1C)NCc1scc(C(=O)NC(C)C)n1 C1(CC)CCC(C)CN1C(C1(CNC(=O)Cc2cc[nH]c2)CC(C)(C)C1)=O C(=O)(CCCCC1CC1)N(C(C)C(=O)N(C(C)C(C)C)C)CC C1(O)(C(N(C(CC(N2CCC(N(C)CC)C2)=O)C)C)=O)CCCCC1 C=CCCCC(C)(C)C(=O)N1CC(C2(NC(=O)CN(C)C(=O)C3CC3)CC2)C1 C(=O)(C(F)CC(C)C)N1CCC(CCNC(CCN2CCN(CC)CC2)=O)C1 C1(NC(CNS(N)(=O)=O)=O)CN(C(C2CCOCC2)=O)CCC1CO C1(CC(=O)NCC2CC(NC(c3cc(C)sc3)=O)C2)CC(=O)NC1=O Cc1onc(C(=O)NCCCNC(C2(F)CC2C)=O)c1I C(=O)(C(C(C)(C)C)N(C)C)N1C(CCNC(c2c(C(C)C)cco2)=O)CCC1 N1(C(C(c2cc(OC)ncc2)(F)F)=O)CCN(C(C2CCC(O)CC2)=O)C(C)C1 CC(C)C(O)C(C)(C)C(=O)NC1CN(C(=O)C=CCN2CCCCC2)CC1C C(=O)(C1COc2ccc(F)cc21)N1CC(O)(C(C)(C)CNC(=O)C(O)C2CC2)C1 c1(CC(=O)NCCN(C(=O)CC2CCC2(C)C)CC)ccccc1C N1(C(CSC(C)(C)C)=O)CCC(O)(CNC(=O)CC2CC=CCC2)C1 Cc1ccc(CN(C2CCNCC23CC3)C(c2cn(C)cn2)=O)c(C)n1 CCC(C)C(C(=O)N1CC(O)(CCNC(c2sccc2NC)=O)C1)NS(C)(=O)=O Cc1cc(C(=O)NC23CCCC2CN(C(=O)C2=CCN(C)C2)C3)c(C)c(C)c1 c1(SCC)cc(C(=O)NC2CSC(C)C2)ccn1 CCC(O)C(F)(F)C(=O)N1CCCC(CC(=O)NC2CCN(C(C)C)CC2)CC1 Cc1nnc2ccc(C(=O)NC3CCCC(NC(=O)CCC4CC4)CC3)cn12 Cc1ccc(OC(C)C(=O)NCCNC(c2[nH]nnc2CN(C)C)=O)c(C)c1 C1(C(C(=O)OCCC2(C(F)(F)F)CCC2)F)CCOCC1 c1(CC)cc(C(N2CCCCC2C2CCN(C(=O)C(C)(C)CO)CC2)=O)ccn1 CC1OCCN(C(C2CCCN2C(=O)C2CC2)=O)C1C(=O)O C1(C(=O)NCC2(O)CCC2)(NC(=O)Cc2ccc[nH]2)CC(CO)C1 Cc1cc(C(N2CCC(N(C)C(C3COC3)=O)CC2)=O)ccc1-c1ccccc1 N1(C(C2N(C(c3c(CCC)[nH]cc3)=O)C(C3CC3)CC2)=O)CC2CC(O)CC2C1 Cc1cc(CCN2CCC(C)(c3ccc(F)cc3)C2)ccn1 c1(CC)ccc(CCC(=O)NC(C2CN(C(=O)C(C)CSC(F)(F)F)C2)C)cc1 C(=O)(CC(C)C(C)(C)NC(=O)CN(C)C(=O)OC)N1CCC(O)(CCC)CC1 c1(C(=O)NCC(C)CN(C(=O)CC2(O)CCCC2)C)ccc(P(C)(C)=O)s1 C12(CNC(=O)CC3CCC3)COC(CNC(c3cccc(CC(F)(F)F)c3)=O)(C1)C2 c1(C(N2C(C)CCC(NC(=O)C(F)(F)CC3CC3)C2)=O)ccc2oc(O)nc2n1 CC1CCCCC1C(N1CCC(C(C)(C)CNC(=O)C(F)=CCCF)CC1)=O CCC(C)(C(=O)NCc1cc(C(=O)NC(C)CCCCO)co1)OC Cc1ncn(C)c(=O)c1C(=O)NCCNC(C1CC(C)(C)OC1c1ccccc1)=O C1(CNC(C2C3CC3CN2C(c2cc(Cl)n[nH]2)=O)=O)(CO)CC2CC2C1 CC(C)CC(O)C(=O)NC1CCCC1N1CCN(C(c2cscc2SC)=O)CC1 CC(C)C(C#N)C(=O)NCC=CC(=O)NC(c1ccco1)C N1(C(CCC)=O)CCCC(C)(NC(c2ccnc(OC)c2)=O)C1 C(c1cc(F)c(F)c(F)c1)=CC(=O)NCC1CC(CNC(c2cnco2)=O)CO1 C1(CNC(CCCOC)=O)CC(NC(=O)CCn2nc(C)nc2C)C1(C)C C(C1CCCCCC1)=CC(=O)NC1(CC)CN(C(=O)CC2CCCC23CC3)C1 C1(C(=O)NCC2CC(NC(c3sccc3C(F)F)=O)C2)COCCO1 C(=O)(C(CC)CC(F)(F)F)NC(CC)CNC(=O)C(C)Cc1ccccc1Cl CN(S(=O)(=O)N=S(C)(=O)C(C)(C)C)Cc1cccs1 N1(C(CCc2n(C)ncc2)=O)CCC(NC(=O)C=CCO)CC1C1CC1 c1(C(=O)NC(C2CCCN(C(CNC(=O)NC)=O)C2)C)ccc2n[nH]c(C)c2c1 c1(CCC(=O)NC23C(CN(C(C(C)OC)=O)C2)C3)cc(F)cc(F)c1 c1(CN2CCN(CCCNC(CC(C)(C)C)=O)CC2)c[nH]c2cccc(Cl)c12 c1(CC(=O)N(C2CCN(C(=O)Cc3cnn(CCF)c3)C2)CC)scnc1C C1(C(N(CCOCC)C)=O)CC(C)CCN1C(c1cc(C)[nH]c1C)=O N1(C(C2CN(C)C2)=O)CC2(CNC(c3ccc(F)c(F)c3N)=O)CC1CCO2 N1(C(c2c(C)con2)=O)CCOCC(CNC(C2CCCCN2S(C)(=O)=O)=O)C1 C1(C(=O)NCCCNC(C(C(C)C)Cc2ccccc2)=O)COCC2(CCC2)O1 C(=O)(C(O)C(F)(F)F)NC(C(=O)NCCCCC1CCCC1)CC1CCCC1 c1(C(N2CCC(C(C)C(=O)NC3CC4(CCC4)C3)C2)=O)ccc2ccoc2c1 C(CO)(C(C)(C)CO)NC(C(C)(N(C)C(C1CC12CC2)=O)C1CC1)=O C1(C(=O)NCCC2CC(NC(C(C)=C(CC)C)=O)C2)CCCCC1F c1(C(=O)NC23CC2CN(C(=O)COCCCF)C3)ccc2ncsc2c1 C1(C(=O)NCCCC(CCC)NC(=O)CCCC(F)F)CCS(=O)(=O)C1(C)C CC1(C)C(C(N2CC(F)CC2CNC(C2(O)CCOCC2)=O)=O)CCS1(=O)=O C=CCC(CC(C)C)C(=O)NC1CCCC1NC(c1cnc(C(=O)OC)s1)=O C1(NC(CC(=C)C)=O)CN(C(C2CC23CCOCC3)=O)C2(CCCCCC2)C1 c1(C(N(CCCCNC(C(CC)(C)C)=O)C)=O)ccc2cc([N+](=O)[O-])ccc2n1 C(=O)(CC(F)(F)C(F)F)NC(CNC(c1ccc(CC)cc1N)=O)(C)CC(C)C n1(CC(N2CCC(NC(Cc3c(C)non3)=O)C2)=O)c(=O)oc2ccccc12 C1(CC(=O)NCCC(C)NC(=O)C(C)N(C)C)SC(=N)NC1=O C(=O)(CC1=CCOCC1)NCCC(C)(CC)NC(CC(C=C)(C)C)=O C1(CNC(CCc2c(C)noc2C)=O)N(C(=O)CC2CCC(=O)O2)CCC1(C)C c1(C(N2CCCC(NC(c3ncc(NC)nc3)=O)C2)=O)c(F)cccc1Br c1(CN(C2CCN(C(c3csc(Br)n3)=O)C2)C(C2C(=C)C2)=O)ccccc1 Cc1csc2cc(C(=O)NCC3(O)CCN(C(c4ccc(F)cc4F)=O)C3)[nH]c12 c1(NC(C2CS(=O)C2)=O)cc(C2CC2)[nH]n1 C1(NC(C(C)CC2CCCCC2)=O)CC2CCC1N(C(=O)CCCC(C)(C)C)C2 c1(C(N(C2CCN(C(=O)CCC#N)C2)C)=O)ccc(C2CC2)c(Cl)c1 N1(C(C=C(C)C(C)(C)C)=O)CCC(C)C(N(C)C(C2CCC3(CCC3)O2)=O)C1 c1(C(N(C(C)CNC(=O)Cc2cnccc2Cl)C)=O)cc2n(n1)CCN(C)C2 C1(OC)CC(NC(=O)C(F)(F)C(F)F)CN(C(=O)CC(O)c2ccccc2)C1 Cc1cc(-c2cccnc2F)c(C)cc1C(=O)Nc1ccccc1NS(C)(=O)=O C(=O)(CC(O)CN(C)C)NC(C)(C)CNC(=O)CC1(C)CCCO1 Cc1ccc(C(=O)NCC2CN(C(=O)CSCC(N)=O)CCO2)c(N)c1 c1(CC(=O)N(C2CCN(C(CNC(CC(C)C)=O)=O)C2)C)ccc(Cl)cc1Cl O=C1CCCCC(C(=O)NCCC2CN(C(c3ccncc3)=O)C2)N1 C(=O)(CS(=O)(=O)NC(C)(C)C)NCC(C)NC(=O)C(N1CCOCC1)C S(=O)(=O)(c1ccc(Br)s1)N1CCN(CC(=O)N(C2CC2)Cc2cccnc2)CC1 C(C)(CCCCCO)NC(C1(CNC(=O)COC2CCCC2)CC(=C)C1)=O c1(CN(CC(=O)N(C)CCN(C(=O)C#CC2CC2)C)CC#C)ccc(OC)cc1 N1(C(C#CC(C)C)=O)C(CNC(c2c[nH]c(C(N)=O)c2)=O)CC2CCCC12 Cn1c(C(=O)NC2(CF)CCN(C(c3csc4cncn34)=O)C2)cc2sccc12 N1(C(Cn2c(=N)[nH]nc2)=O)CC(NC(C2CCN(CC3CC3)CC2)=O)C(CO)C1 c1(C(N(CC)CC2CCCN(C(=O)C(C)C3CCCC3)C2)=O)nn(C)c(N)c1C C1(C(N(C2CCN(C(c3sccc3-n3ccnn3)=O)C2)C)=O)CCC(O)C1 c1(CC)c[nH]c(=NCCc2ccc(C(=O)OCCOC)cc2)o1 Cn1nnc2cncc(C(N3CC(C)(NC(C4CCC5CCCCN45)=O)C3)=O)c12 C1(c2nnnn2CC(F)F)(NC(CC)C2CCC2)CC(C)SC(C)C1 c1(C(N2CCC(N(C(C34CC(C)C3C4)=O)CCO)C2)=O)cccc2sncc12 N1(C(CC(=O)N(C)C)=O)CCN(C(=O)CCc2nc[nH]n2)C2CCCCC12 c1(N(C(C2CCCN(C(CCCC#C)=O)C2)=O)C(=O)N(C)C)ccc(F)cc1C Cc1cc(Cl)nc(NC(c2cccn2Cc2cccnc2)=O)n1 c1(OC)cncc(C(=O)NCC2CCCCCN2C(c2n[nH]c(C)c2Cl)=O)c1C c1(C(C)C)ccc(C(=O)NCCC(O)CNC(C2CCC(C)O2)=O)c(O)n1 C(C)(C(=O)NCCOc1ccncc1)(N(C(C=CC(=O)N(C)C)=O)C)C1CC1.OCN c1(C(=O)NC(COCC)C)coc(CNC(c2ccc(C(N)=O)[nH]2)=O)c1 C1(CNC(C(C(C)(C)C)O)=O)CC2(CCN(C(c3cc(Cl)no3)=O)CC2)CO1 N1(C(C2(CC=C)CCCC2)=O)CCCC(N(CCO)C(c2ccc(C)s2)=O)C1 Cc1cccc(C(=O)NC(C)(C)C(C)NC(c2ccc(Cl)s2)=O)c1F N1(C(CCc2ccc(C)nc2)=O)CCN(C(c2cc(C)no2)=O)C2CCC12 N1(C(c2c(C)cn(C)c2)=O)CCC(C2CCN(C(C34CC(C)C3C4)=O)CC2)CC1 S(=O)(=O)(c1cnn2ccc(=NCCC(F)F)[nH]c12)N1CCC(C(C)C)C1 c1(C(C)C)ccc(C(=O)NC2CC(O)C2CC(=O)N(C)CCc2cnc[nH]2)o1 Cc1ccc(C(C)C(=O)NCC2CC(NC(=O)CN(C3CCSC3)C)C2)s1 C(=O)(C1CCc2nccn21)NC(C(=O)Nc1cc(CC)c(C)nc1)C(C)C N1(C(CCC(C)SC)=O)CC(C)OC2(CCN(C(c3cc(C(C)C)no3)=O)C2)C1 c1(N2CCCC(n3c(O)ncc3)C2)nccc(=NCC#CC2CC2)[nH]1 c1(CN2CCCC2)c(F)cccc1F.c12nnc(o1)CC1N(CC1)C2C CCC(C)(C#N)C(=O)NCCC1CCCN(C(c2csc(COC)n2)=O)C1 Cc1c(CC(N2CCCC2C2(NC(C(C(=O)C3CC3)C)(C)C)CC2)=O)cnn1C Cn1cc(C(=O)NCCCS(=O)(=O)N2CCCC2)c(Br)n1 c1(C(=O)NCCN(C(C2C(C)(Br)C2)=O)CC2CC2)ncoc1-c1ccccc1 C1(C(=O)NCCN(CC(C)C)CC)CCOCC1NC(c1cccc(=O)o1)=O N1(C(C2(OC)CCSCC2)=O)CCC2(C1)CN(C(C1CC(C)OC1=O)=O)C2 c1(OC)ccc(C)c(OC)c1C(N1CC(NC(c2cc(F)c[nH]2)=O)CC(F)C1)=O C(=O)(C(CC(C)CC)NC(C1C=CC=CC=C1)=O)NCCCCC#CC C12(CNC(COC)C(=O)NCC(C(C)C)N(C)C)CCCC(CO1)C2 C1(CS(C)(=O)=O)CN(C(c2ccccc2F)=O)CCN1C(C1COCCO1)=O c1(OC)ccsc1S(=O)(=O)NC(=O)C(C)Oc1ccc(Cl)cc1Cl CC1(C)CC(NC(=O)C(=O)NCC2(O)CCSCC2)C(C)(C)O1 C1(CC(=O)N(C2CCCNC2)C2CC2)CNC2CCCCC12 C(=O)(C1=CCCS1)N1C(CN(C(=O)CCOC2COC2)C2CC2)CCC1 C1(C(=O)NCC(N2CCCCC2)=O)CN(C(=O)Cc2cncnc2)CCO1 c1(C(=O)OCC=C)c(OC)sc(C)c1C.c12cccc(c1)NC(=O)N2 CC(CN(C)C)CCC(=O)NC1CC1CNC(c1ccncc1)=O C(=O)(N1CCC(C(N2CC(N(C)CC)C2)=O)O1)c1n(C=C)nnc1 C1(C(=O)NCCc2ccc(Br)s2)COCCN1Cc1cccc(O)c1 N1(C(C(N2CCNC2=O)C)=O)CCC(CCNC(C2CNC(=O)O2)=O)CC1 CC1(C)CCCCCN1C(=O)CN1CCN(CC(=O)Nc2ccccc2)CC1 c1(N2C(CNC(CNC(C=C(C)C)=O)=O)CCCC2)ncnc2occc12 C1(C(=O)NCCN(C(C=C(C)C(F)F)=O)C(C)C)CCCS(=O)(=O)C1 N1(C(C(COCC)NC(=O)Cn2nccn2)=O)CCCC(C)(COC)C1 C1(CC)C(C(=O)NCC(C(C)(C)C)NC(=O)CSc2nncn2C)CCN1C N12CCC3(CC(=NO3)C(=O)NCCNC1=O)C2.c1(NS(C)(=O)=O)ccccc1 CCC(C)CC(C)CC(C)C(=O)N1CC(c2ccc(Br)cn2)(O)C1 c1(C(C(=O)N2CC(CCNC(=O)C(C)n3cccn3)C2)SC)ccccc1 CC1(C(=O)NCC#CCNC(C23CC2COC3(C)C)=O)CCC(F)(F)CC1 C=CC(C)(CC)C(=O)NC1CN(C(=O)C(c2ccccc2)OCC)CCC1C c1(C(N(CCCC(N2C(COC)COCC2)=O)C)=O)cc(C)c(N)cn1 c1(C(N(C2CC2)Cc2ccc(-c3ccc(CC)s3)cc2)=O)nccn2ccnc12 C(=O)(CC(C)C(C)(C)C)N1C(C)CCC(NC(CCCCC#C)=O)C1 c1(C(=O)NC2(CCNC(c3cnccc3Cl)=O)CC2)ccc(O)c([N+](=O)[O-])c1 c1(CNCC(C(C)C)Nc2ccccc2)ccc2oncc2c1 C1(C(N2CCC(N(C(C(CCC)OC)=O)CCO)CC2)=O)OCC2CCCCC12 Cc1cccc(C(=O)NCC2CCC2C(=O)NCC2(O)CCC(C)C2)n1 C1(C(=O)NCC2(C#C)CC2)CC(CC)CCN1C(C1CCC(=O)NC1)=O CC1(C(=O)NCC2(CNC(=O)CCc3ccc(O)cc3)CCCC2)CNC(=O)C1 C(CCCC(=O)NCCOCCCCCNC(=O)CC1CCNC(=O)C1)OCC c1(CC(=O)N(CCC2(NC(CCN(C)CCO)=O)CC2)C2CC2)cccnc1Cl c1(SCC(=O)NCC(CC)NC(C23CCC(CF)(CO2)C3)=O)nc(C)cc(C)n1 C(C(N=[N+]=[N-])C(=O)NCC=CCC(=O)NCCC1CCN(C)C1=O)OCC N1(C(C=CC=CC)=O)CC(F)(F)CC1C(N1CCC2(CCC2)C1)=O c1(C(=O)NCc2occ(C(=O)NC(C=C)CO)n2)ccc(CC)nc1 c1(OC)cccc(N2CCCC(CN(C)C(C3CCCC3C)=O)C2)c1[N+](=O)[O-] C#CC(C)CN=C(NC(C#C)CC1CC1)NC1CCCCC1 N1(C(C(C#C)(C)C)=O)CC2CN(C(=O)C=Cc3ccc(C)s3)CC2(C)C1 CC1OCCN(C(C2(CNC(C3CCCOC3)=O)CCCCC2)=O)C1C C1(N(CCNC(c2c(C)nns2)=O)C(c2ccnn2C(C)C)=O)CCCCCC1 C1(CC(=O)NC2(CC)CC(C)(C)C2)C2CCCC2N1C(c1cnncc1OC)=O C(=O)(C1=NN(CC)C(=O)CC1)NCCN(C(=O)Cc1ccc(F)cc1C)CCC C(=O)(C1=NOC2(CCC2)C1)NC1CCC(NC(c2c(C)nc(C#N)cc2)=O)C1 C1(CC)(CO)CCN(C(=O)C(=O)NC(C2CCOC2)COC)C1 c1(C(=O)OC)c(NC(C2C3CC2N(C(c2csnc2C)=O)C3)=O)sc(C)c1C Cc1cc(C(N2CCCC2C(=O)OC(C)(C)C)C(=O)NC2CCOC2)n[nH]1 C1(NC(C(OC)OC)=O)CN(C(c2ccc(OC(F)(F)Cl)cc2)=O)CCC1CO C1(C(=O)NCC2CC(C(=O)NC3C(C#N)CCC3)C2)CCC(C2CC2)C1 c1(CC(N2CC(CC=C)(NC(C3CCCC3(F)F)=O)C2)=O)nsc2ccccc12 Cc1cccnc1C(=O)NCCC(C)(C)CNC(c1oc(C(F)(F)F)nc1C)=O c1(OC)cnnc(C(N2CCC2C(=O)NCCC2CCC(C)(C)O2)=O)c1 CC(CCSc1ccco1)N=c1[nH]c(N2CCC(=NO)CC2)nc2ccccc12 c1(C(N(C2CCCCC2)C(C(C)C)C)=O)ccc2c(c1)CCC2(C)C CCC(CCC(=O)N(CCCC(O)CO)C)NC(c1cn(C)c(=O)cn1)=O C(CC1=CCN(C(C2CCCCO2)=O)CC1)NC(C1CC(F)C(=O)N1)=O N1(C(C=CCOC)=O)CCN(C(=O)C(N2CCC(C)C2)=O)CC1C(C)C c1(C(N(CCN(C(=O)CC2CCCCC2C)CC)CC)=O)nnn(C)c1C C1(OC)COCCN(C(C2CCC(C(C)C)N2C(=O)CCCF)=O)C1 c1(OCC)cc(Cl)ccc1C(=O)NC1(C)CCN(CC(C)CC)C1 N1(C(c2cc(C(CC)CC)no2)=O)CCOCC(NC(=O)C(C)=C2CCC2)C1 CC1(C)CN(C(=O)CC23CCCC2C3)CC(CNC(=O)CCC(N)=O)O1 Cc1cccc(C(=O)NC2CCC2NC(C2COC(C)(C)CO2)=O)c1O C(=O)(C(F)C(C)CNC(=O)C(C)COC)NCCOCCC#C c1(C(=O)NC(C(C)NC(C(CC)F)=O)(C)C)ccc(OC(C)C)c(OC)c1 c1(CC(N2C(CNC(C3CN(CC(C)C)C3)=O)COCC2)=O)cccc(C#N)c1 C(C(O)C(CC)CC)NC(CC1(NC(c2c(CC)cncc2)=O)CCC1)=O C1(C(=O)Nc2ncc(CCO)s2)CN(C(c2cc(Cl)ccc2Cl)=O)CCC1O CC1(C)CC(CNC(c2ccc(F)cc2F)=O)N(C(C2CCCCS2(=O)=O)=O)C1 C1(CNC(C(F)=CCC)=O)N(C(c2ccnn2CCC)=O)CCC1(C)C N1(CC2(C)CCC2)C(=O)CCN(Cc2cccc(-c3ccccc3)c2)C1=O C1(NC(C2CCN(C(=O)C3CC3(Cl)Cl)O2)=O)CCN2CCC1C2 CCCCC(CNC(C1(Br)CC1(C)C)=O)NC(=O)CN1CCOCC1 C1(NC(C2C(OCC)CC2)=O)C2CCCN(C(=O)CCP(C)(C)=O)C2C1(C)C c1(OC)ccc(-c2ccc(O)c(C)c2)cc1NC12CCC(NS(C)(=O)=O)(CC1)C2 C1(C(=O)NCc2scc(C(=O)O)n2)COCCN1Cc1ccc(-c2cccnc2)o1 CN=c1[nH]cc(C(=O)NCC2CCN2C(C2CCN(C)C2)=O)s1 C(C(=O)N(C)CCC1CN(C)C1)(C(C)(C)C)NC(c1c(C)nco1)=O C1(NC(c2c(C)cco2)=O)CN(c2ncc(F)cn2)CCC1O C1(CC)CN(C(c2ccn(CCNC(C3C4CC(=O)CC34)=O)c2)=O)CC1O c1(C(C(=O)NCC2CC(CNC(C(CSC)OC)=O)C2)C)ccc(F)cc1 N1(C(Cc2ccn(C)n2)=O)CCC(C(N2CCCCC(F)(F)C2)=O)C(C)(C)C1 C1(O)(NCc2cccc(COC)c2)CCCN(C(=O)OC)C1 C1(C(C)NC(C2C(=C)C2)=O)CCN(C(=O)C(C)NC(=O)Cc2cccs2)CC1 c1(C(N2CCC(O)(CNC(C3CC(C)(C)C3)=O)C2)=O)c(Cl)ccc(F)c1F Cc1ccc(O)c(CC(=O)NCCC(C)(C)NC(=O)Cc2ccon2)c1 CCCCC(C(=O)NCCCCCCF)NC(=O)CCCCNC(C)=O C(=O)(C(C(C)C)NC(=O)CC1CCCOCC1)NCC1N(CCOC)CC1 Cc1nn(Cc2ccccc2)c(C)c1S(=O)(=O)NC(CO)CCn1cccn1 C1(CC(=O)NC(C=O)C)CCC(C)(C)O1.C#CC(C)(C)N CC(C)C(C)C(=O)NC(CNC(=O)C(C)OC1COC1)C1CC1 c1(OC)cc(NC(C2CC(O)CN2C(C2COCOC2)=O)=O)cc(O)c1 N1(C(COCC)=O)C(CNC(=O)C(C(C)(C)C)SC)CCC2CCCCC12 C1(CNC(c2n(CC)ncc2Cl)=O)CCC(C)CN1C(c1ocnc1C1CC1)=O CC(=O)C(C)CC(C)C(=O)N1CCCCC2(CCC2)C1 c1(OCC)ccc(N)c(C(N2CC(F)(F)CC2CNC(=O)C=C2CCCC2)=O)c1 N1(C(CC(CCC)C)=O)CC(NC(=O)COCC2CC2)CC2(CCOCC2)C1 c1(C(C)Sc2nnnn2C2CC2)ccc2c(c1)CCO2 C(=O)(C(N)CC(F)F)N(C1CCCC(C)C1)C(C)C1CC1 C(=O)(C1c2c[nH]nc2CN1C(c1cc2n(n1)CCO2)=O)NCC(CC)n1cccn1 c1(NCC)nccnc1N1CCCC(Oc2ccccc2Cl)C1 Cc1nn(C)c(C)c1CNC(=O)CC1(NC(=O)CC2CCCC(=O)C2)CCC1 c1(C(=O)NC(CC)CNC(=O)CC2CCCCO2)n[nH]c(C)c1C c1(OCC(=O)NC(C(C)NC(Cc2scc(C)c2)=O)CO)cccc(Cl)c1C Cc1cccn2nc(C(=O)NC3CN(C(=O)C(C)(C)C)CCC3C)cc12 c1(C(N2CC(CC(=O)OC)C(C)C2)C(=O)NC2CCCC2)sc(C)c(C)c1C c1(C(N(CCC(C)NC(C2CCOC2)=O)C)=O)c(F)ccc(Cl)c1F c1(C(=O)NCCCCC(N2CCC(C)(CO)C2)=O)ccc(F)c(O)c1 c1(NC(N(C)CC23OCC(C(=O)OCC)(C2)C3)=O)cncc(C#N)c1 c1(OCC#C)ccc(C(=O)NC2(CNC(C3CCOC(=O)N3)=O)CC2)cc1 C(=O)(C(C)S(=O)(=O)C(C)C)NC1CC(F)(CNC(c2c(OC)ccnc2F)=O)C1 C(=O)(C(C(C)(C)O)NC(=O)CCSCCC)NC(CCC)CO c1(SC)ncc(C(=O)NCC(C)CNC(c2cnc(CC(C)(C)C)s2)=O)n1C Cc1cc(C)c2c(c1)N(C(c1ccc(F)c(Br)c1)C(=O)NC1CC1)CC2 N1(C(c2c(C)cc[nH]2)=O)CCC2CCC(NC(=O)CC3CN4CCC3CC4)C1C2 CC1(C)C(CC(=O)NCCCC2(NC(=O)CSS(C)(=O)=O)CC2)CC1O c1(C(=O)O)cc(Cl)c(O)c(S(=O)(=O)NCC2CN(Cc3ccc(O)c(O)c3)C2)c1 C(=O)(C1=CNC2=NCCC2=C1)N1CCC(CC)C1CNC(c1occc1C)=O CC(C)CC(C(=O)NC1(C(=O)O)CCN(C)C1)N(C(=O)C(CO)OC)C N1(C(=O)CCC2CCC2)CCC(C2CCCN2C(c2nncs2)=O)CC1 C(C1COc2ccccc21)N(C(C(N)Cc1cccc(Br)c1)=O)CCO CC1(C)CC(CC(N2CCC(O)(C(C)CNC(=O)COCCCF)C2)=O)C(=O)O1 CC1=NNC(=O)C1CC(=O)NC1CN(C(=O)Cc2cccc(O)c2)C1 C1(C(=O)NCC2(C)OCCN(C(C3CC(O)(CC)C3)=O)C2)CCc2nnnn2C1 Cc1nc(C(N2CC3CC3(CNC(=O)CCC(=O)c3ccc(Cl)s3)C2)=O)n(C)n1 c1(NC(C)=O)cc(C)c(S(=O)(=O)N2CCCC2(C)C(C)O)c(C)c1 C(=O)(C(C)(C)CCC#N)N1CC(CC(=O)NC2(O)CCOCC2)(OC)C1 C=C1CC2(C1)CC(C(=O)NC(C)CNC(=O)CC1CCNC(=O)C1)C2 c1(OC)ccc(CN2CCCC(C)(C(N3CCN(CCCO)CC3)=O)C2)cc1Br Cc1ccn2cc(C(=O)NC3(CNC(=O)C=Cc4cnc[nH]4)CCC3)nc2c1 c1(NC(C(=O)N(CCN(C)C)C(=O)OC)=O)ccc(OC2CCC(C)(C)C2)cc1 N1(C(C(C2CN(C(c3cc(Cl)ns3)=O)C2)OC)=O)CC(=O)N2CCCC2C1 c1(CC)ccccc1C(=O)N(C1CCC(NC(c2cn(C)cc2C)=O)CC1)C C(C(C)(C)C1CCC1)(c1nnnn1C)NCC1CN(C(CC)=O)C1 C#CCC(C)C(=O)N1CCCCC1CNC(=O)CCNC(=O)CCc1cnco1 C1(NC(C(C)=C(CC)C)=O)CCCCC1NC(=O)C=CC1CCCN1C C(=O)(C(C)SC)NC(CN(C(=O)CC1(CNC=O)CC1)CC)C N1(C(CC2(CC(=O)OC)CC2)=O)CCCC(NC(c2ncn(C(C)(C)C)n2)=O)C1 n1(CC)c(CCNC(c2ccncc2)CC2CCCCC2)nc2ccccc12 c1(-n2ccc(CNC(=O)Nc3c(C)ncnc3)n2)c(F)cccc1F C1(F)(C(=O)NCCC2(O)CN(C(c3c(C(C)=O)cco3)=O)C2)CCS(=O)(=O)C1 c1(OCC(=O)NC(C(C)(C)NC(CSCCOC)=O)C)cc(F)ccc1Br N(C1CN(C(=O)C(F)C(C)C)Cc2ccccc21)C(C12CC(CCC)(C1)C2)=O c1(C(N2CCC(C)(CCNC(C3CCC(=O)O3)=O)C2)=O)c[nH]c2nccc(Cl)c12 C1(NC(c2nnn(C)n2)=O)CC2CC(C1)CN(C(=O)COc1ccc(O)cc1)C2 CP(C)(=O)CN1CC(C(=O)NCCC2(NC(=O)CCC3CC3)CCC2)C1 N1(C(CO[Si](C)(C)C)=O)CCCC12CCCN(C(C1CC1(F)F)=O)C2 N1(C(Cc2c(C)ocn2)=O)CCC(NC(=O)CNC(=O)CC(C)C)C(O)C1 c1(C(=O)NC(C(C(C)C)NC(CCC)=O)C)sc2ncccc2c1Cl N1(C(COC(C)C)=O)CCCC1C(=O)NCC(=O)NC(C)(C)CN(C)C1CC1 C1(NC(C(CCCC)O)=O)CS(=O)(=O)C2CN(C(=O)C3=CCOCC3)CC12 c1(C(C(=O)NCc2cc(CNC(C)=O)on2)O)c(C)cccc1C c1(C(=O)NCC2CCN2C(c2n[nH]c(C3CC3)n2)=O)cc2n(n1)CCCC2O c1(C(N2CC3CC2CN3C(C2SCCCS2)=O)=O)c(F)cccc1Cl c1(-c2ncc(C(N3CCC(CC(C)C)CC3)=O)nc2)cc([N+](=O)[O-])ccc1F Cc1c(F)ccc2[nH]c(C(=O)NC3CCN(C(=O)Cc4ccns4)C34CC4)cc12 CCCCC(O)C(C)C(=O)NC1(CC(=O)NC2CCC3(CC2)N=N3)CCCCC1 N1(c2ncnc(C)c2F)CC(NC(=O)CNC(=O)CC(C)C)CC12CCOCC2 N1(C(CCCSC)=O)CCC(NC(c2cc(Cl)nnc2O)=O)C(C)C1 Cc1ccc(N(CCNC(=O)CCOC2CCC2)C)cc1C(C)(C)C c1(CC(N2C(CNC(CC(C)N(C)C)=O)CCC2)=O)ccc(S(C)=O)cc1 CCCCCCC(C)C(=O)NCc1c[nH]nc1C(=O)NC1CC2C(C1)C2(F)F C(=O)(CC(C)(O)COC)N(C(C)C(=O)NC1(C)CC1)CCC C1(NC(c2c(C)ccs2)=O)CC=C(C(=O)NCC2CCCS2)C1 C1(NC(C(C)(C)OCC)=O)CCN(C(=O)CCNC(=O)C=CCl)CC1C CC1(C)CCN(C(c2cncc(CC#N)c2)=O)CC1CNC(=O)Cn1cncn1 C(c1cc2ccccc2o1)=CC(=O)NC1CCN(C(=O)Cc2nnc(O)s2)C1 C1(C#N)(C(=O)NCC(CN(C)C(C2C3CCCOC23)=O)(C)C)CCOCC1 C1(NC(C2C(C)=C2)=O)CC1C1CCCN(C(c2cncc(N)n2)=O)C1 N1(C(c2cncc(C#C)c2)=O)CCOC2(CCN(C(=O)CCC=CBr)C2)C1 C1(CCC)CN(C(c2ccon2)=O)CCN1C(=O)CC1CC2CCC(C1)C2 C1(C(=O)NCCN(C(C(C)(C)OCC)=O)C)CNC(=O)CC12CCOC2 c1(C(=O)NCC(C)NC(C(C(CC)C)O)=O)ccc2nc[nH]c2n1 N1(C(CC2(C=C)CCC2)=O)CC2CC(C1)N(C(c1ccc(C#N)[nH]1)=O)C2 CC1CC(CNC(=O)CCC2CCOC2)CCN1C(c1cc[nH]c1)=O C(=O)(C1CCc2nnc(C)n21)NCC(C)NC(C1=C(CC)OCCC1)=O C1(NC(C(N2CCOCC2)C)=O)C=CCN(C(c2ccnc(C3CC3)n2)=O)C1 CC1CN2CCN1C(C(N1CC(CCNC(=O)C(O)CC3CCCCC3)C1)=O)C2 CC(C)(CF)C(=O)Nc1cc(CNC(=O)CC2CC(CCNC(C)=O)C2)on1 N(C(=NCC)NCC1(CO)CC2CC2C1)CC(CCC)C N1(C(C(COCC)C)=O)CC2CCC(NC(c3ccn4cccc4c3)=O)(C2)C1 c1(CC)cn2c(n1)CC(C(N1CCC(NC(c3ccc(Br)o3)=O)C(F)C1)=O)CC2 N1(C(=O)OC(C)(C)C)CCCC(F)(CSC2CCCCN2CCc2ccco2)C1 c1(-c2scc(C(=O)NCCC)n2)cc(F)cc2[nH]ccc12 Cn1cc(C(C)(C)C(=O)NCC2CCN2C(c2cc(-c3ccco3)cs2)=O)cn1 N1(C(C(C)n2cnnn2)=O)CCC(C(=O)NC2CCCCC2C#N)=C(F)C1 c1(C(=O)NCCN(C(CNC(=O)OC)=O)C)cnn(C2CCOCC2)c1 C(CN=c1[nH]c(=NCC(C2CC2)C2CC2)[nH]c2c1COC2)N1C(C)CCCC1 CC1(C)CN(C(C2(C)CCCS2)=O)CC1C(=O)Nc1cc(O)cc(F)c1 N1(c2nnc(C3CCC(OCC)C3)n2C)CCNC(=O)C1c1cnn(C)c1 C=CCC(CC=C)C(=O)N1CCC(CNC(=O)C(COC)N(C)C)C1(C)C c1(OC)ccnc(C(=O)N(C2CCN(C(=O)CC3C=CCC3)CC2)C)c1N Cc1[nH]c(=N)nc(O)c1NC(=O)CC1(n2cncn2)CNC1 Cc1nc(NC2CCC(NC(c3cnn(C(F)(F)F)c3)=O)CC2)[nH]c(=N)n1 C1(O)(C(C(=O)N(C(C)CO)C)NC(=O)CP(C)(C)=O)CCCCC1 CC(C)C(C)(C)C(=O)NC12CC1CN(C(C1CC1Sc1ccccc1)=O)C2 C(=O)(CC(C)(C)C(F)(F)F)N1CCC(N(C(=O)CNC(=O)OC(C)(C)C)C)CC1 c1(C(C)=O)ccc(C(=O)NCCCCNC(=O)C(F)(F)C2CCOCC2)nn1 CCCCCC(=O)N(C(CNC(=O)CN(C)C(=O)NC)C1CC1)C c1(C(N(CCN(C(COCCCC)=O)C(C)C)C)=O)cccc(Cl)c1 c1(C(N(C2CN(C(c3ccc(Cl)cc3N)=O)CC2F)C)=O)[nH]cc2c1CCC2 O=[N+]([O-])c1cccc(F)c1CS(=O)(=O)Nc1nccc(N2CCCC2)n1 C=CCCC(N=c1cc(C)[nH]c(=NCC(COC)OC)[nH]1)C1CC1 C1(C(N(CCNC(C2N(C(=O)OC)CCC2)=O)C(C)C)=O)CNC(=O)C(C)(C)C1 c1(OC)ccnc(CNC2C=CCCCC2)c1 C1(CC(=O)NCC(F)(F)CO)CCC(NC(=O)CC2CCCOC2)CC1 CC(C)C(C)(O)C(=O)NCCC(C)CCNC(c1ccc(C2CCCC2)cc1)=O N1(c2cc(C)ncn2)CCCC(C)(CNC(c2conc2C(C)C)=O)C1 CC1(C)CC(NC(=O)CNC(=O)OC(C)(C)C)CN(C(C23COCC2C3)=O)C1 N1(C(C(C)CC2CCCCC2)=O)CC=C(CNC(C2CCCC3CC23)=O)CC1 CC1CCC(CO)N(C(c2coc(Br)n2)=O)C1 N1(C(C2CN(C)C(=O)N2)=O)CCC(F)C(NC(=O)C=Cc2cccc(Cl)c2)C1 c1(C(=O)NC2CCN(C(CN3CCC(C)CC3)=O)C2)cnn(C)c1S(C)(=O)=O N1(C(C(C)N(C)C)=O)CCOC2CN(C(c3cnn(C)c3N)=O)CC12 N1(C(C=CC)=O)CCCC2C1CCCCN2C(c1coc(C(C)(C)C)n1)=O C(C)(C(C(=O)NC(C)(C)CCCOC)C(C)C)NC(CCC(=O)NCC)=O C1(NC(=O)Cc2ccc(Cl)cn2)CCC2CC1CN2C(c1n[nH]c2c1CCC2)=O c1(C(=O)NC2CCCC(NC(C3=C(C)OCCS3)=O)C2)c(F)c(F)cc(F)c1F CCC(CCC(=O)NC1(c2cccs2)CC1)NC(c1cc(C)n(C)c1C)=O C12(CNC(c3c(C)nns3)=O)CCC1CCN2C(=O)CCCc1ncco1 N1(C(C(n2cnc(C#N)n2)C)=O)CCC(C)(NC(=O)C(=O)Nc2ccccc2)C1 c1(C(N2C(C)CN(C(CCC=C)=O)C(C)C2)=O)coc2c(F)c(Cl)ccc12 c1(C(=O)NCC(C)NC(C(c2cnn(C)c2)OC)=O)oncc1C c1(NC(c2n(CC(=C)C)nnn2)CCc2c(Cl)cccc2Cl)cc(O)ccc1C c1(CCC(=O)NC(C2CC(NC(c3nccn3C)=O)C2)C)ccccc1N(C)C c1(C(=O)NC)cc(-c2ccccc2C2(C)OCCO2)cc2[nH]ncc12 C1(C(=O)NCC(CN(C(c2c(C)cc(F)s2)=O)C)O)CC2(C1)CC21CCC1 C(=O)(CCCC(=O)N(C)CC1CCCC1NC(C1CCC(OC)C1)=O)NC Cc1ccc(C(C)NC(C2(C(C)NC(C3CCCN3C)=O)CC2)=O)nc1 C1(CNC(C2(C)ON=C(C)C2)=O)CC2(C1)CN(C(=O)CC1CN3CCC1CC3)C2 N1(C(c2nc(CCCC)sc2)=O)CCC2(CNC(=O)COC3CC3)CCCCC12 C(=O)(C1CCc2cccnc21)N(CCCNC(C(C(=O)OCC)C(C)(C)C)=O)C Cc1cc(=NC2CCCc3c(OC)cccc32)[nH]c(=NCc2ccncc2N)[nH]1 c1(NC(C(COCC)N=[N+]=[N-])=O)cccc2c1OCCO2 CON(C)CCCNC(C1CCN(C(=O)CC2(O)CCC2)C1)=O c1(C(C(=O)NCC2C(C)(C)OCC2)(F)F)cc(C(F)(F)F)cc(F)c1 C(=O)(C1=NN(C)C(=O)CC1)NCC1N(C(c2nc(C)n(C)n2)=O)CC(C)(C)CC1 C1(NC(CCNC(=O)NC)=O)CCN(C(C2CC(OC)C2)=O)C1 S(=O)(=O)(CCC(F)(F)F)NC1C2CN(C(c3ncsc3Br)=O)C(C2)C1 S(=O)(=O)(c1ccc(-c2ccco2)c(OC)c1)Nc1c(C(=O)OC)sc(C2CC2)n1 S(=O)(=O)(c1cnc(NCC2CCCC2O)c(Cl)c1)NCC1(C)CCC1 N1(CC(=O)NCCCN(C(=O)C(F)(F)C2CCOCC2)C)CCC(O)CC1 c1(CN=C(NC(CC)C)NC(CO)CCF)cn2ccccc2n1 C(=O)(C1c2ccccc2C(=O)N1C)NCCCNC(C=C1CCC(C)C1)=O c1(C(=O)Nc2ccc(SC)c(F)c2)cc2n(n1)CCCN(C(=O)C(C)Br)C2 Cc1ccc(F)c(C(=O)NCC(C)(O)CNC(=O)CC2OCCO2)c1Br c1(C(=O)NC2(CC#C)CCC2)c[nH]nc1OCC N1(C(c2cc(Cl)cnc2O)=O)C2CCC1CC(NC(C1(O)CC3CC1C3)=O)C2 c1(C(=O)NC(CCCNC(C(C)NC(=O)C(C)(C)C)=O)C)cccc(F)c1C#N c1(CCNC2(c3n(CCCC)nnn3)CC(C#N)C2)nc2cc(C)ccc2n1C N1(C(C2(NC(=O)Cn3cccn3)CCN(C)C2)=O)CCN2CCOCC2C1 C(=O)(CC(C(=C)C)OCC)N1CCC(NC(CCOCC#C)=O)C1C N1(C(C(=O)NC(C)C)=O)CC(NC(=O)C(C)OCCN(C)C)C(C)C1 Cc1cn(CC(=O)NC2(CN(C)C(C3CC(F)(F)C3)=O)CC2)nc1C(F)(F)F C1(CC(=O)NC2C(CNC(C(C)(C)C)=O)COC2)CCC2(CCCC2)CC1 C1(F)(C(=O)NCCC(C)(C)NC(=O)CC2CC(=O)NC(=O)C2)CCC(F)(F)CC1 N1(C(C2N(C(C(C)=CCC)=O)CCC(CC)C2)=O)CC(C2=NOC(C)C2)C1 C12(NC(c3c(CCC)occ3)=O)CCC(C1)N(C(C1(COC)CCCCO1)=O)C2 c1(C(=O)NC(C(CO)NC(C(CC)SC)=O)C)cnn(CC)c1C1CC1 C1(NC(Cc2c(C)n(C)nc2)=O)CN(C(C2CC2(F)F)=O)CC12CC2 CC(C)C(O)C(C)C(=O)NCCC1(C)CCN(C(=O)C(C)(C)N2CCCC2)C1 c1(OC)cccc(C(N2CCC=C(CNC(C3(C)C=CCCC3)=O)C2)=O)c1O c1(NC(C2CN(C(C3CCC(C(N)=O)C3)=O)C2)=O)ccc2nccn2c1 N(C(=NCCCCc1ccc(Cl)s1)NC1CCOCC1)CC1OCCN(C)C1 C1(C(=O)NCC(C2CC2)NC(C=Cc2n(C)ncc2)=O)CN2CCC1(C)CC2 c1(NC(C2C(NS(C(C)C)(=O)=O)C2)=O)cccc2c(Cl)ccnc12 CC1(C)CC(C(N2CCC(CF)(NC(c3occc3Cl)=O)C2)=O)CCO1 c1(CN2CCC(N(C)C(C3CCCCO3)=O)C2)cccc(F)c1F C1(CNC(c2c(N(C)C)cncc2)=O)CC2CCC1N2C(c1scnc1Cl)=O c1(NC2CCCC(C(=O)OC)CC2)ncnc2ncc(Br)cc12 N1(C(c2ccc([N+](=O)[O-])cc2OC)C(=O)NC)CCOC2(CCC(F)(F)CC2)C1 c1(CC)ccc(N2CCN(C(=O)NCC3CC4(C3)N=N4)CC2)c(F)c1 [N-]=[N+]=NC1CCC(C(=O)NCCC2CC(F)(F)CN2C(C2CCNC2=O)=O)CC1 c1(C(=O)NCC2C3CN(C(COCCC)=O)C2C3)ccc([N+](=O)[O-])[nH]1 n1(CC)nc(C)cc1C(=O)NC(C(=O)NC1CC(C)C1)C1CCC1 CC(O)(CC(=O)N1CCCC2(CC(NC(C3(C(F)F)CC3)=O)C2)C1)C(F)(F)F CC(C)C(CN(C)C)C(=O)NC1CCC(NC(=O)CCc2cncc(O)c2)CC1 c1(C(=O)NC(C(C)C)C(C)NC(c2cnsn2)=O)cc(O)c(F)cc1N Cn1c(C(=O)NC2CCC(CNC(C3CC4CC3C3CC43)=O)C2)cc(Cl)c1Cl C(=O)(CC1OCc2cc(Cl)ccc21)NC(CC=C)CNC(C1CC2(CSC2)C1)=O O=C(C1=CCCOCC1)NC12CCC(CN(C(=O)CCCNC(=O)C3CC3)C1)C2 C1(CC(=O)NC(C=C)CO)CN(C(c2ncoc2CC)=O)CC1C c1(C(=O)NC2CCCN(C(C(C3CC3)OCC)=O)C2)ccc(CO)c(Cl)c1 c1(CC(N2C(C)(CC)CC(NC(=O)Cn3cccc3)C2)=O)csc2ccccc12 CC(C)C(C)(C(=O)N1CCC1CNC(=O)CCNC(N)=O)c1ccccc1 c1(NC(C2C3CCN(C(C(C=CC)O)=O)CC32)=O)ccc2c(c1)COC2 N1(C(CC(CNC(=O)Cc2cscn2)OC)=O)CCCC(O)(C(N)=O)C1 Cc1nc2c(s1)CCCC2C(=O)N1CCC(OCCNC(C2CC=CCC2)=O)C1 CC1(C)CC(NC(C2(n3ccnn3)CC2)=O)CC(C)(C)S1(=O)=O CC1(CNC(c2c[nH]cc2Br)=O)CC(F)(F)CN1C(C1CCc2c[nH]nc2C1)=O N1(C(CC(CC)C(F)F)=O)CCc2nc(CNC(=O)COCCN(C)C)sc2C1 c1(C(N2CCC(C(C)NC(C3COC(=O)N3C)=O)C2)=O)cncn(C)c1=O C1(C(N2CCC(NC(c3cccc(SCC)c3)=O)C2C)=O)CCC(F)(F)CC1 C(=O)(C1CCc2cc(F)ccc21)N1CCC(C)C(CNC(C2CC2F)=O)C1 CCCC(C)CC(=O)NCCC1CN(C(c2cncc(O)c2)=O)CCO1 C1(C(=O)NCC2(CC)CCCC2)(CC)CCN(C(C2CCCC2)=O)C1 C(=O)(C1=CCCCCC1)NCCC(C)N(C)C(C1CCC2(CCC2)C1)=O N1(C(c2c(C)cc(C)o2)=O)CCCC(F)(C(=O)NCCc2ncccn2)C1 C#Cc1cnc(NC(C2CC2NCc2ccc(C(F)(F)F)c(F)c2)=O)cn1 N1(C(c2ccc[n+]([O-])c2)=O)CCCC(N=c2cc[nH]cc2[N+](=O)[O-])CC1 N1(S(c2c(C)nn(CCOC)c2C)(=O)=O)CCC(C)CC1C1CCC(C)O1 c1(C(N2CCC(O)(CC)CC2)=O)cnn2c1CNCC2 C(C1CN(C(=O)C(F)(F)CO)CC1C(=O)NC1CC(C2CC2)C1)=CC CC1CCN(C(c2cc(C(F)F)cs2)=O)C(CNC(c2cnc(N)c(N)c2)=O)C1 c1(CN2C(C(=O)Nc3ccc(Cl)nc3)CC(F)C2)c(F)c(F)cc(F)c1F Cc1cc(=NC2CCCN(C(c3cccc4c3ccn4C)=O)C2)[nH]c(C2CC2)n1 Cc1cc(=O)c(C(=O)NC2CC3CN(C(=O)Cn4nccc4N)CC23)cn1C C(CC(C(C)C)NC(=O)CCCc1csc(=N)[nH]1)NC(C1CC(SC)C1)=O N1(C(c2c(C)nccn2)=O)CCCC(NC(c2csc([N+](=O)[O-])c2)=O)C(F)C1 C(=O)(CCC(=O)NN(C)C)NC(C)CCNC(C1CCSC1)=O N1(C(=O)COC2CC2)CCC2(CCCN2C(C2CCOC3(CCC3)C2)=O)C1 CC1=C(C(=O)N2CCOC(C3CN(C(=O)CC(C)N(C)C)C3)C2)CC1 C(CC(C)C)(CS(=O)(=O)NC1CCN(S(C)(=O)=O)CC1C)OC Cc1cc(NS(C)(=O)=O)c(F)cc1Br.N12CC(C)(C1)CC(=O)N1CCC(C1)C2=O c1(C(N2CCC(N(C)C(C3CS(=O)(=O)C3)=O)C2)=O)cccc(SC2CC2)c1 C(C)(CCC(=O)NCC1CCN(C)C1)NC(c1ccc(CC)[nH]1)=O CC(C)CC(F)C(=O)N1CC=CC1CNC(=O)CCCSC(C)(C)C C(=O)(CC(C)(C)O)N(C1CCN(C(C23CCCC2(C(N)=O)C3)=O)CC1)CC#C c1(CNC(C2CCC(C)C2)=O)nnn(C)c1C(=O)NCCc1ccnc(O)c1 c1(OC)cccc(CC(O)C(=O)NC2(CO)CCN(C(=O)C(=O)NC3CC3)C2)c1 Cc1nc(C)n(CC(=O)NCC2CCC(C(=O)NCCC3CCCCC3)CC2)n1 C[Si](C)(C)CCCC(=O)N(CC(F)(F)F)Cc1cccs1 C(C(CC(=O)NCC(C1CCCCC1)O)OC)NC(c1ccn(CCC)n1)=O C(C(O)CC(=O)NCC1(C(=O)N)CCN(C)C1)N(C)C.C12(CC1)C(=O)NC2.C1CC1 c1(CN(C(=O)NC(c2ccco2)COC)C)cccc(SC(F)(F)F)c1 Cc1nn(C)c(C)c1C(=O)NC1C2CC1N(C(C1SCCS1)=O)C2 CN(CCCCc1ccccc1)N1CCC2(CO)CCC1C2 C1(NC(CC2(COC)CC2)=O)CCN(C(=O)C(O)Cc2[nH]cnc2C)C1C N1(CC)N=C(C(=O)N(C)CCNC(c2nn[nH]c2C(F)(F)F)=O)CCC1=O N1(C(C2C(NC(c3c(C)oc(C#N)c3)=O)CCCC2)=O)CC2(CCC2)CC1C N1(C(CSCC)=O)CCCC2CN(C(c3ccc(C(F)(F)F)o3)=O)CCC12 c1(C(N2CC3(C(C(=O)NC4(C(=O)OC)CCC4)C3)C2)=O)ccc2c(c1)ncn2C C=C1CC2(C1)CC(C(N1CC(F)(c3cn(CC(C)(C)[N+](=O)[O-])nn3)C1)=O)C2 Cc1cnc2ccc(C(=O)NCCC3CN(C(c4cc(Br)n(C)c4)=O)C3)cn12 N1(C(C(CN(C)C)O)=O)CCC(C(=O)NC(c2ncccn2)(C)C)=C(F)C1 N1(C(C2(C(=O)NC)CCC2)=O)CCC(C)(CC(=O)NC2CC(C(C)(C)O)C2)C1 c1(NC(=O)OC(C)(C)C)cc(CNC2C=CCC2)cc(C(F)(F)F)c1 C1(C(N2CCC(O)(C(C)NC(C34CC(F)(C3)C4)=O)C2)=O)CCC2(CCCC2)C1 C(=O)(C1=CCC1)NCCN(C(C1CC(C(C)(C)C)C1)=O)Cc1ccccc1 N1(C(C(CC)(C)CNC(c2cc([N+](=O)[O-])c[nH]2)=O)=O)CC2CC(F)CC2C1 N1(C(C(C(C)C)N(C)C)=O)CCC12CN(C(C1CCCN1c1ncccn1)=O)C2 c1(CC)ccc(F)c(C(=O)NC2C3CCN(C(c4cnnc(O)c4)=O)C23)c1 c1(NCc2cc([N+](=O)[O-])c(O)cc2)cc(-c2cccc(F)c2)nc2ccccc12 C1(CNC(c2nncc(OC)c2)=O)(NC(=O)CC(C)C(C)C)CCCCC1C CC(C)CCN=C(NCC1OCCO1)N1CCC(CCC#N)CC1 C1(CNC(CSCCCC)=O)(NC(=O)Cc2ccc(C(F)F)cc2)CCOCC1 O=C(CC1COCc2ccccc21)NC1CCN(C(=O)Cc2ccns2)CC1O c1(C(=O)NC2C3CN(C(C(CCC)CCC)=O)CC32)cnc2cc(O)nn2c1N C1(CCNC(C2CN3CCN2CC3)=O)CCN(C(c2cnc(Cl)s2)=O)CC1(F)F C1(C(N(C)CC#N)=O)CN(Cc2cc(Br)c(F)cc2O)CC(F)(F)C1 c1(C(N(CCCNC(c2cnn(C(C)C)n2)=O)C)=O)ccc2c(c1)C(C)CO2 c1(N(C)C)c(C(=O)NCCCNC(=O)C(C)(C)C(N)=O)nnc2ccccc12 C(CC(O)C(=O)NC1(C(=O)NCC23CCC(CC2)C3)CC(F)(F)C1)N(C)C n1(CCC)nc(C)cc1C(=O)NC(CNC(=O)C(C)O)CC C1(C(=O)NCCc2nc(C)on2)N(C(C2CC(C)C2)=O)CCCC1(C)C C1(CNC(Cn2cc(C(C)=O)nn2)=O)CCCCN(C(c2cncnc2)=O)C1 CC#CCC(C(=O)NCC12CCCC1CCO2)NC(=O)C=CCN1CCC1 C1(OC)CCC(C(=O)NC(C2CC=CCC2)C(=O)NCCN2CCOC2=O)CC1 C1(O)(C(COC(C(=O)OC)OCC)C)CCN(C(=O)CCc2csnn2)C1 n1(CC)nc(C(N2CCC(Cc3cccc(F)c3)C2)C(=O)NCC(C)C)c(C)n1 C1(CC(=O)NCc2nccs2)CCCN(C(=O)CC2CCCCO2)C1 C1(C(N2CCC(CNC(C(C)OCCCC)=O)C2)=O)(C(=O)OC)CC1(C)C c1(C(=O)NCC(CC)NC(=O)Cc2csc(C)n2)c(C)oc(C)c1C CCC(CNC(=O)Nc1cccc(CN2CCCC2=O)c1)(CC)SC N1(C(C2(COC)CC(=C)C2)=O)CCCC2(CCN(C(C3SCCS3)=O)C2)C1 c1(C(c2cocc2Br)NC(=O)NCC2(C(F)F)CCC2)cccnc1 C(=O)(C(C)(C)S(C)(=O)=O)NC(CC)CNC(C1CCCCC1(F)F)=O Cc1ncc(CCC(=O)NC(C)C(CO)NC(c2cnc(N(C)C)s2)=O)s1 c1(NC(=O)NC2CCCC23OCCO3)nc2cc3c(cc2[nH]1)OCO3 N1(C(c2n(CCC#N)ncc2)=O)CCC(CNC(C2(n3cccn3)CC2)=O)CC1 c1(OCC)c[nH]nc1C(=O)NCCCCCOCCNC(=O)Cc1ccco1 n1(CC)ncc(C(=O)NCC2(C)CCCC2NC(C2COCCOC2)=O)c1C C(c1ccccc1C#N)=CC(=O)NCC1(C)CCCN(C(CC2(C)CCC2)=O)C1 N1(C(c2c(C)cnnc2)=O)C2CCCC1CN(C(c1coc3ccccc13)=O)C2 N1(C(C2(F)CCN(C(CC(C)=C(C)C)=O)C2)=O)CCc2c(C#N)cccc21 C1(N(C(=O)CCn2cc(Cl)cn2)CC)CCCN(C(=O)CC2(O)CCOC2)C1 C(CCCCCC(=O)N(CCNC(C)=O)CC1(C)CC1)n1cc(COC)nn1 C1(NC(C2CCCN(CC)C2)=O)CCN(C(=O)CC2CCCC2)CC1(C)C C1(O)(C(C)NC(c2nocc2C(C)(C)C)=O)CCN(C(C2COCCOC2)=O)C1 Oc1ccc(-c2ccccc2)cc1CNCc1nnnn1C1CC2CCC1C2 C1(C(N(C(CF)CF)C)=O)CCN(C(C2C=CCS2)=O)C1(C)C Cc1cc(=NCc2cccc(Br)c2F)[nH]c(=NC(CCO)C(F)F)[nH]1 C1(NC(C(C=C)O)=O)CN(c2cc(Cl)nc(C)n2)CCC12CCC2 c1(NC(CCN(C(C(CC=CCC)C)=O)C2CC2)=O)ccc(F)c(O)c1 c1(NC(C2CC(O)CN2Cc2c(I)ccnc2Cl)=O)ncc(Br)c(O)n1 c1(SC)cccc(C(=O)NC2CCCCC2NC(=O)Cc2cnnn2C)c1Cl C1(CC)CCC1CN(C(=O)CCNC(=O)CCNC(=O)OC)C1CC1 c1(SCC(=O)NC23CC(CNC(C4CC(F)(F)C4)=O)(C2)C3)ccncc1 c1(C(=O)NCC2C(NC(C(COC)OC)=O)COC2)cccc(CS(C)(=O)=O)c1 c1(C(CC)C)nc(-c2occc2Cl)n(C(C2CCCCC2)C)n1 C1(CCNC(COCCC)=O)CCN(C(c2coc(Br)n2)=O)C(C)C1 C12(C(=O)NC(CC=C)C(=O)OC)CCC(CC1)N(C(=O)C=Cc1cccnc1)C2 c1(C(=O)NCC2(F)CC(CNC(C(c3ccccc3)SC)=O)C2)ccn(C)c1C c1(CNC(CS(CC)=O)=O)nc2c(s1)CCN(C(C1(C)C(C)(C)C1(C)C)=O)C2 c1(CC)nc(C)c(C(=O)NCCCOCCCNC(C2CCOC2C)=O)s1 c1(C(=O)NC2CC(CCNC(C3CCSC3)=O)C2)nc2n(c1Cl)CCCC2 N1(C(c2ccc(OC)cn2)=O)CCN(C(C2(C)CCCCC2)=O)CC1C(F)(F)F C1(C(=O)NC2(C)CCN(C(C(C)=C(CC)C)=O)CC2)CCN(S(=O)(=O)N(C)C)C1 N1(C(C(Cc2c(C)n[nH]c2C)C)=O)CCC(C)(NC(C23CC(CO2)C3)=O)CC1 C1(CNC(C(COC)C)=O)CCCCC1NC(c1ccn(CC2CC2)c1C)=O C12(NC(C(C)SC)=O)CCOCC1CN(C(c1ccc(Br)cc1O)=O)C2 C1(NC(C=CC(C)(C)C)=O)CC2CCC1N(c1cc(-n3ccnc3)ncn1)C2 c1(C(=O)NCCC(C)NC(N2CCCCCC2)=O)cc(Cl)ccc1NC1CCC1 c1(C(=O)NCCCN(C(C2CCCCC2(C)C)=O)CC)nccc2ccccc12 c1(C2N(CC(COc3ccc(OCC)cc3)O)CCC2)ncc(F)cc1F C1(CC(N)=O)CCCN(C(=O)C(Cn2cccn2)NC(C2CCOCC2)=O)C1 c1(C(=O)NC2CCC(NC(=O)CC(O)C3CCCC3)C2)ccc2ncnn2c1 c1(OCC(=O)NCC(CC)NC(C2COC(=O)N2C)=O)ccc(C)cc1C C(=O)(C1=Cc2cc(F)ccc2OC1)NCC1CCN(C(CC(C)O)=O)C12CC2 C1(C(C)C)CN(C(C2C3CCN2CC3)=O)CCN1C(c1cc(C(F)F)[nH]n1)=O C1(CC)COC(C)CN1CCc1ccccc1.c12ccccc1C(=O)N2 N1(CC(N2CCCC(N(C(C3ON=C(CC)C3)=O)C)C2)=O)CCP(C)(=O)CC1 C1(CNC(c2cn(CC)nc2)=O)CCC(C)CN1C(c1cc(C(F)F)ccn1)=O C1(Nc2nccc(N(CCC(=O)N(C)C3CC3)C)n2)CCC2(CCC2)OC1 c1(OC)cccc2cc(C(=O)NCCNC(=O)CC(C)SCC(C)O)c(=O)oc12 C#CCC(CC)NC(=O)C(CSCC)NC(=O)C(C1CCC1)OCC c1(N(C(c2c(C)ccc(C)c2N)=O)C)ccc(S(=O)(=O)C(F)(F)F)cc1 C1(CCCCNC(COCCC=C)=O)CCCN(C(=O)C(F)(F)CO)C1 c1(C(=O)NC2CN(C(Cc3c(C)con3)=O)C(C)C2)ccccc1P(C)(C)=O N1(C(=O)CCSc2ccc(Br)cc2)CC2(CCCC2)C1C(=O)O N1(C(CC2(C=C)CCC2)=O)CC(CNC(c2cn(CC)nn2)=O)C2(CC2)C1 c1(CC)ccc([N+](=O)[O-])cc1NC1(C(=O)O)C2CCCC12 Cc1ccn(C(C)C(=O)NC(CO)C(=O)NCC2(CO)CC=CC2)n1 C(=O)(CC(C)(C)C(F)F)NC(C(C)C)CCN(C)C(C1CC(C)(C)C1)=O c1(C(=O)NC2(CCOC)CCN(C(C3CCC3C)=O)C2)cncn(C)c1=O C1(CC)(CC)CC(NC(c2c(C)nn(C)c2C)=O)CN1C(=O)Cc1nccn1C CCCCC(C(=O)NC1COCC(C)(C)C1)NC(=O)C(CC)CCC c1(OCC)cc(Br)ccc1NC(C1CCC(NC(=O)C=Cc2cnccn2)C1)=O N1(C(C23N(C(C4N(C)CCOC4)=O)CC(C2)C3)=O)CCCN(C=O)CC1 c1(NC(C2N(c3ncc(C(=O)OC)cn3)C3C(C2)C3)=O)ccc(Br)cc1O N1(C(CCNC(=O)Oc2ccco2)=O)CC(F)(F)CC1CNC(C1CCCO1)=O C12(C(=O)NC3CC(N(C)C(c4ncn5c4CCC5)=O)C3)CCC(C)(CC1)CO2 CCS(=O)(=O)c1ccc(Cl)c(C(N2CCC(CNC(=O)CNC=O)(OC)C2)=O)c1 c1(C(N(C(CCC)C)C)=O)cncc(CNC(=O)CCC2CCC(C)O2)c1 CCCS(=O)(=O)C(C)C(=O)NCCN(C(=O)C(C)=C1CCC1)CC1CC1 C1(CCOC)CCN(C(C2CCN(C(c3cccc(F)c3)=O)C2)=O)CC1 c1(CNC(=O)CCC(=O)Nc2ccc([N+](=O)[O-])cc2)c(F)ccc2[nH]cnc12 C(=O)(C(CC(C)CC)NC(=O)C(=O)C(C)(C)C)N1CC(n2cc(CC)nn2)N(C)CC1 CC1CCCC=C1C(=O)NC(C)C(CO)NC(=O)Cc1ccc(F)cc1Br Cc1cc(N)cnc1C(=O)N(C1CCN(C(C2CCC3C2C3(F)F)=O)CC1)C N1(C(C(c2nnc(S)n2C)OC)=O)CC(C)(C)C1C1CCCO1 Cc1cc(C(=O)NCC2(CNC(=O)C(F)C3CCCC3)CC2)c(C)n1C Cc1ccc(C(=O)NCC2C3CCC(C3)N2C(c2n[nH]c(C)c2F)=O)c(C)n1 S(=O)(=O)(c1cnc(NCC2CCCOCC2)c(Cl)c1)N(C)Cc1c(C)nco1 C1(F)(C(=O)NCC(CNC(c2cccc(Cn3cccn3)c2)=O)O)CCCOC1 c1(C(=O)NCC(C)N(C(c2cc(C)c(C)nn2)=O)C)ccc2c(n1)CCC(C)C2 CC(CC(=O)NC1(C)CC1)C(C)(C)NC(=O)C(O)CC(N)=O c1(C(=O)NCCC23CCC2CN(C(C2COC2)=O)C3)cc2c(cn1)OCCO2 N1(C(C=C(C)C)=O)CC(C)OC2(CCN(c3ccc([N+](=O)[O-])cc3C(C)=O)C2)C1 C(CCC(N)=O)(C(=O)OCC1CCNC1=O)N(C)C(=O)OC(C)(C)C C1(C(=O)NC(CC)CN(C(=O)CCNC(N)=O)C)CC2(CCC2)CO1 C(=O)(C1=CCC(C)CC1)N(C1CCCN(C(=O)CN2CCOCC2)C1)CC N1(C(C(=O)NCc2c(CC)cccn2)C)CCc2ccccc21 N1(C(Cc2nc(C)[nH]n2)=O)CC(NC(c2ccc(N)c(O)c2)=O)CC12CCCC2 c1(C(=O)NCC(C)NC(c2ccc3cn(C)nc3c2)=O)cnn2c1CC(C)CC2 c1(CSC)noc(CCC(=O)N2CC(C(C)NC(=O)CC3CCC(O)C3)C2)n1 C1(C(=O)NCC(CNC(=O)C#CC2CC2)C(F)(F)F)(NC(C)=O)CCC(C)CC1 N1(C(C(C)Cc2ccncc2)=O)CCC(NC(=O)CCN2CCCC2)C(C)(C)C1 N1(C(C)C2CC2)CC(C(N2CCOCC2CCNC(c2cscn2)=O)=O)CC1=O C1(C(=O)NC(c2ccccc2)CC)CC2CCC(C1)N2C(C1CC12CC2)=O C1(OCC)COCCC1CC(=O)Nc1cccc(NC(=O)Cc2ccsc2)c1 C1(CNC(C2CC(C#N)C2)=O)CN(C(=O)CSCCC#N)C2(CCC2)C1 CCN=c1ccc(C(=O)NCC2C3CN(C(=O)CCS(C)=O)CC23)c[nH]1 C1(NC(COCCCOC)=O)CCC(NC(=O)CN2CCCC2CO)CC1 Cc1[nH]nc(Cl)c1C(c1nnnn1CCN1CCOCC1)NCC1(C)CC=CCC1 N1(C(Cc2c(C)ccs2)=O)CCCC2(CC(NC(c3cn(C)nn3)=O)CO2)C1 N1(C(c2n(CC)ncn2)=O)CCC(NC(c2ccc(Cl)cc2C)=O)C(F)(F)CC1 O=C(CC(C(F)(F)F)C1CCC1)NC1CN(C(=O)C(F)(F)CN2CCCC2)C1 N1(C(Cc2ccn(C)n2)=O)CCC2(CCCCC2NC(=O)C=Cc2cncs2)C1 c1(CSC)cccnc1C(=O)NC(C)CCN(C)C(c1ncccc1N)=O CC(=O)C(C)CC(C)C(=O)NCC1CC1NC(C12CC(F)(C1)C2)=O CCCCC(CC)C(=O)N(C(c1cccc(Cl)c1)CC)C(c1ccc(C)cc1)=O c1(OCC)ccc(S(=O)(=O)N2CC(C)(CO)C2)cn1.c1(C(=O)N)cncn1C C1(N(C(=O)Cc2cccs2)C)CCCC(NC(=O)CC2CCC(C)(C)O2)C1 c1(N2CC(COC)N(C(C3CCCCCC3)=O)CC2)ncc2ccccc2n1 Cc1cc(-n2cccn2)nc(NC2CCN(C(=O)CCCC3CC3)CC2C)n1 C(=O)(C1=NOC(C)C1)NCC1N(C(c2[nH]cc(C(C(C)C)=O)c2)=O)CCC1 N1(C(C(C)NC(C)=O)=O)CC2CCC1CN2C(c1ncc(C(C)(C)C)o1)C c1(CN(CC(C)(C)C)C(c2ccc(Cl)s2)C(=O)Nc2ccccc2)cccc(F)c1 c1(CC(=O)NC23CC2CN(C(=O)Cn2cnnc2)C3)coc2ccccc12 c1(N(CC(=C)C)C)nc2cccc(F)c2c(=NCC2CCCOC2C(C)C)[nH]1 N1(C(=O)NCC2(CCO)CCCC2)CCOC2CCCCC12 c1(C(=O)NCc2c(C(=O)NC(CCC)C3CC3)scc2)ccccc1OCC N1(C(C(C=C=C)C)=O)C2CCC1C(C(=O)NC(CF)C(F)(F)F)C2 Cc1ccnc(C(N2CCC(N(C)C(c3ncc(F)cc3F)=O)C(C)C2)=O)c1F C1(c2nnnn2CC)(NCCOCC)CN(C)CC1C C1(NC(c2c(CC)c[nH]n2)=O)CC2CCC1CN2C(=O)C(c1ccccc1)C CS(=O)(=O)C1CN(C(=O)Cn2cccc2)CC1NC(C12CCC(CC1)C2)=O c1(CN2CC(NC(c3cc(C)cc(Cl)c3)=O)C2)cc([N+](=O)[O-])cc(Br)c1O Cc1cccc(F)c1C(=O)NC1(C(N2CCCC(CC(N)=O)C2)=O)CC1C C(N1CCC(F)C1)S(CC1C(C)C1)(=O)=O.C1(N)CCCCC1 c1(C(=O)NCC2(C#N)CN(C(c3ccc(C)n3C)=O)C2)cc2ccccc2[nH]1 C(=O)(C(C(C)(C)C)n1ccnn1)N1CC(C(C)NC(c2csc(O)n2)=O)OCC1 Fc1cccc(C2CCCCN2c2cc(Br)ncn2)c1 c1(CNC(CCOC(C)C)=O)cc2cc(F)ccc2[nH]1 C(C(CO)CC(C)C)NC(CN(CC(C)C)C(=O)CC1CCCC(=O)C1)=O N1(C(c2cc(C)oc2)=O)CCC2CCCC12CNC(c1cnn(C)c1N)=O N1(C(N2CC3(C)CC2(OC(C)(C)C)C3)=O)CC(O)CC12CCCC2.C1(=O)CCCO1 c1(C(=O)NCCN(CCC)C(C2CC2CF)=O)cc(S(=O)(=O)NC)c[nH]1 CCC(C)C(O)C(=O)NCC(C1CCC1)NC(c1cnn(C)c1SC)=O c1(OCC(=O)NCCCN(CCCNC(C(F)OC)=O)C)cc(Cl)ccc1Cl Cc1cccc2c(O)nc(CN3CCN(C(=O)Cc4cccc(Cl)c4)CC3)nc12 c1(OCC)c(Br)cc(CN(c2nccs2)CC)cc1Br S(=O)(=O)(c1ccc(C(=O)N(C)C(c2cc(C)ccc2C)C)cc1)NCC N1(C(C)C(N2CCC(N(C(=O)CCCC3CCC3)CCO)C2)=O)CCC(O)CC1 c1(OC)ccc(CC(N2CCN(C(C3CCCN3C(N)=O)=O)CC2C)=O)c(F)c1 N1(C(CCN(C)CC)=O)CCC(Cn2cc(CC3(OC)COC3)nn2)C(F)(F)C1 N1(C(C(=O)OC(C)(C)C)=O)CC(C(=O)NOC2CC(O)C2)C2(CCC2)C1 CC1CN(C(=O)C#CCNC(=O)C(O)C2CCCC2)CCN1C C1(NC(c2cn(CCO)nn2)=O)CCC(CNC(=O)C(O)Cn2cncn2)CC1 c1(CC(=O)NC2CCCC(NC(C(C)OC)=O)C2)cccc([N+](=O)[O-])c1C C1(C(=O)NC(C2(O)CCN(C(c3cnn(C)c3)=O)C2)C)CCCCCCC1 c1(C(=O)NC2(CNC(CNS(CC)(=O)=O)=O)CCCC2)cc2ccc(F)cc2[nH]1 C(=O)(CCCCC(C)(C)C)N1CCC(NC(C(CC=C)C(C)C)=O)C12CC2 O=C1CC2(CCC2)C(C(=O)NCCCCNC(=O)C2=CCCO2)CN1 C1(NC(=O)Cc2ccon2)CC2C1CCN2C(=O)CSc1cccc(Br)c1 CCC(F)(F)C(C)(C)C(=O)NCC1CCC(NC(=O)Cn2cc([N+](=O)[O-])cn2)C1 C1(OC)CC2(CCC(C(=O)NCC3CCC(NC(=O)CCCCC#N)C3)CC2)C1 c1(COCC)ccc(CN(c2ncc(-c3ccccn3)s2)C=O)s1 c1(C(=O)NC2C(NC(C(C)SC)=O)CCC2)ccc2c(c1)N(C)CC2 C1(C(=O)NC2CN(C(CCCN(C)C)=O)CC2O)CC12CCSCC2 c1(CNC2CC(NC(C3C(C)C3)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 CC(O)CCN=c1cccc(S(=O)(=O)NCCc2ccncc2)[nH]1 C1(C(=O)NCC2C(NC(C(CC)CC3CCCCC3)=O)C2)CN(CP(C)(C)=O)C1 Cc1c(C(N2CC3C(CNC(c4cnc(O)o4)=O)C3C2)=O)oc2ccc(F)cc12 C(C(CNC(=O)OC(C)(C)C)S(C)(=O)=O)NC(=O)NC(c1cn[nH]c1)C Cc1c(C(N2CCC(N(C(=O)CSC3CC3)C)C2)=O)[nH]c2c(C)cccc12 C=CC(C)(CC)C(=O)NC(C)CC(C)NC(c1nc(Cl)ccc1Cl)=O CC1Cc2ccc(F)cc2C1NC(=O)CCCOCCCN c1(OC)cc(C(N2CCC(NC(=O)C3=CCC3)C(C(C)C)C2)=O)ccc1Cl c1(OCCC(=O)NC2CCC(NC(CC#N)=O)C2)ccccc1F c1(C(N2CC(CC(C)NC(=O)COc3ccc(Cl)cc3)C2)=O)c[nH]c(=O)cn1 C1(NC(C(C)C)=O)CCCC(NC(c2ccccc2-n2ccnn2)=O)C1 C1(C(=O)NC2C3N(C(c4scc(C)c4Cl)=O)C(CC3)C2)CCC2(CCOCC2)O1 C(=O)(C1=NOC(C2(O)COC2)C1)N1CC2C(N(C(=O)CC3CC4CC4C3)C)C2C1 N1(C(c2c(C)coc2C)=O)CC2=C(C1)CN(C(=O)C(C)Cc1cnc[nH]1)C2 c1(C(=O)NCC2N(C(C(C3CCOCC3)C)=O)CC=C2)cc2n(n1)CCCN2 C1(NC(C2(C#C)CCCC2)=O)CC12CCN(C(c1coc(CO)c1)=O)CC2 CC(CC(=O)NCC1C=CCN1C(C1(C(=O)NC2CC2)CCC1)=O)C(C)(C)C C12(CNC(c3c(CCC)n(C(C)C)nc3)=O)CC(CO1)N(C(=O)C(C)SC)C2 CC(c1cccc(Cl)c1)=CC(N1CC=CC(NC(C23CC2C3)=O)C1)=O n1(CC(=O)N(C(C)CCNC(c2coc(Br)n2)=O)C)cnc([N+](=O)[O-])n1 N1(C(c2cccc(C(=O)NC)c2)=O)CC(C)CN(C(c2ncoc2C)=O)CC1C n1(CCC(N2CCC(c3cnccn3)C2)=O)cc(C2(F)COC2)nn1 CC1=C(C)CC(C(N2CCC(CC3CCCN3C(=O)C3=CCCS3)CC2)=O)CC1 c1(C(=O)Oc2nccc(NC(=O)OCC)c2)ccc2csnc2c1 c1(C(=O)OC)csc(C(=O)NCC2CC(NC(c3ccc(C(F)(F)F)o3)=O)C2)n1 N1(C(C(=O)NCC(=C)C)C2CCC2C(F)(F)F)CCN(Cc2cnc(Cl)s2)CC1 c1(OC)ccccc1C(=O)N(CCCCCCNC(C1CC(C)(C)O1)=O)C N1(C(c2cc(C(C)C)on2)=O)CCCC(O)C1C.C1C(=O)N1CC1CC1 C=CC1CN(C(c2c[nH]c(=NCC)s2)=O)CC1NC(=O)C(C)CC c1(C(N2CC(CNC(C(C)=C(C)C)=O)C(C)CC2)=O)cc(Cl)c2n[nH]cc2c1 N1(C(COc2cn(C)nc2)=O)CC2CCC1C1CN(C(=O)CCC(N)=O)CC21 c1(OC(C)C(=O)NCCNC(C2C=CCN2C(=O)C2CC2)=O)ccccc1F c1(C(=O)NC2CCN(C(=O)CC3=CCCC3)CC2)cc2cccnc2o1 Cc1sc(N)c(C(=O)NC2CC2NC(=O)C(C)Cc2ccc(F)cc2)c1C C(CNC(C1(C)CC(NC(c2cc(CCO)on2)=O)C1)=O)(C(F)(F)F)OC C1(CCNC(CN2C(C)CC2)=O)CSCCN1C(=O)C=C1CCN(C)CC1 C(=O)(CC(C)(C(F)F)N(C)C)NC1(CO)CN(C(c2c(C)c(Cl)ccc2)=O)C1 C(=O)(C(C)(C1CC1)NC(=O)CC1C=CC(NC(=O)CCCOCC2CC2)C1)OC C(CC(C)(C)C)(C(=O)NC1(CN(C)C(c2sc(C)nc2C)=O)CC1)OC c1(CCC)onc(C)c1C(=O)N(C)CCNC(=O)Cc1ccccc1OC(F)F N1(C(c2nc(C)nc(O)c2)=O)CCC2(CCN(C(=O)C=Cc3nc[nH]n3)CC2)C1 c1(C(N)=O)cccc(CN2CCC(C(=O)NCc3ccncc3F)C2)c1 C1(NC(C(CC=C)CC)=O)CN(C(=O)CCc2cccc(O)n2)CCC1(C)C C1(CN(C(C2CN(C(C)C)C2)=O)C)C2CN(C(C3(C)CC3(F)F)=O)CC12 C(=O)(CS(=O)(=O)C1CCCC1)NC(C(C)(C)NC(CC(C)C(F)F)=O)C C1(C)(NC(C(C)OCCC=C)=O)CCN(C(c2sccc2SC(F)F)=O)CC1 c1(-c2c(OC)cc(C)c(C)c2)ccc(N=c2ncc3cc(Br)ccc3[nH]2)nc1 c1(OC)cc(-c2cccnc2C(=O)Nc2cc(OC(F)F)n[nH]2)cnc1F C1(NC(CC2C(CC)C2)=O)(CC)CCN(C(=O)C=Cc2ccc(O)cc2)CC1 c1(C(=O)NC(CN(C(=O)CCCN2C(=O)CCC2=O)CC)C)ccc(Cl)cc1F Cc1cc(NC(=O)CCCCCO)nc2ccccc12.N12CCC(CC1)C2=O C1(CNC(C(CCCC)F)=O)CCC2CN(C(C3(C#N)CCOC3)=O)CC12 N1(C(c2cnc(CC)[nH]2)=O)CC(NC(C2(C#N)CCCOC2)=O)CC12CCCC2 S(=O)(=O)(c1cnn2ccc(N3CCC(C)(N(C)C)C3)nc12)N1C(C)CC(C)CC1C N1(CC)CCCC(ONC(=O)C(O)C2CN(C(=O)NC)C2)C1.C1(=O)C(C)N1 c1(CC)nc2c(C(=O)NCC(C)CN(C(=O)C(C)C(C)COC)C)ccnc2[nH]1 C1(N(C(c2ccc(C(OC)OC)o2)=O)C)CCN(C(=O)CC2(C)OCCO2)CC1 c1(OC)sc(C(=O)NCC(O)CN(C(=O)CC(C)OC)C)cc1Br c1(C(C(=O)NCCNC(c2cnn(C)c2)=O)N(CC)CC)ccc(SC)cc1Cl Cc1ccc2c(c1)C(N)C(C(N1CCC(Oc3ccc(C(=O)O)cc3)C1)=O)C2 N1(C(c2c(Cl)cc(C)nc2)=O)CC(NC(c2oc(C)nc2C)=O)C(S(C)(=O)=O)C1 c1(C(=O)NCC(CO)NC(c2cnn3ccsc23)=O)c(Cl)ccc(F)c1F c1(-c2cn(C)nc2)ncccc1NC(C1CC(O)C1)=O c1(C(N(CC(=O)NC2CN(C)CC2O)C2CCC2)=O)cncn(C)c1=O C(C)(CO)(C(=O)NCCCOCC1CC1)NC(C1ON=C(C)C1)=O N1(C(c2ccc(O)nn2)=O)CCN(C(c2ccc(Cl)c(F)c2F)=O)C2(CC2)C1 N1(C(COCCOCC#C)=O)CC(NC(=O)C(C)n2cnnn2)C2(CCC2)C1 C1(CC(=O)NC(CSCC)C(=O)NCC2(C)CCN(C)C2)CCCN(C)C1 C1(C(NOCC(C(C)C)O)=O)CN(C(C2CN(C)CC(C)O2)=O)CC1(C)C N(C(=NCc1cccnn1)N1CCC2(O)CCOCC2C1)C(CC)C N1(C(COCCC)=O)CCN(C(c2csnn2)=O)C(c2nccn2C)C1 c1(OC)c(C(N2CCOC(O)C2)=O)cc(-c2ccccc2)cc1Cl c1(-c2onc(C3C(C)(CC)C3)n2)ccc(C(F)(F)F)cc1Cl CC1CN(C(c2ccon2)=O)CCC1N(C(=O)Cc1c[nH]ccc1=O)C C1(C)(CCNC(C=C2CCN(C)C2)=O)CCN(C(=O)CCc2ccc(O)cc2)C1 N1(C(C2(C)CC(C)C2)=O)CCC(C(C)C(=O)NCC2CCCOC2)CC1 C1(NC(COC)=O)CN(C(=O)C(C)Cc2ccc(Cl)cc2)CC12CCC2 C1(OCC(=O)NCCCN(C(=O)C(C)(C)F)CC)CCOCC1 Cc1cc(S(=O)(=O)N2CC3(CCC(=O)N3)C2)cc(C(=O)O)c1C c1(C(=O)NCC23C(CN(C(c4nc(C)sc4)=O)C2)C3)c(O)nnc2c1CCC2 Cc1cc(C(=O)NCCC2CC(NC(c3[nH]c(C)nc3C)=O)C2)c(O)nn1 N1(C(C(OC)OC)=O)CCC2(CCCN(CNc3ccc(I)c(OC)c3)C2)C1 C(=O)(CCCc1ccccc1)NCCCCNC(C(c1cscn1)N(C)C)=O C(=O)(C(C(=O)NCCOCCCNC(c1ccoc1C)=O)OC)OCC c1(OCC)ncc(C(=O)NC2CCCC(C(=O)NCCSC)C2)cn1 c1(C2(C(N(CC(C)NC(c3cccc(F)c3)=O)C)=O)CC2)cccc(Br)c1 CC#CC1CCN(C(c2[nH]ccc2CNC(=O)C(C)C2CCCC2)=O)CC1 c1(C(N2CCCC(COC)(CO)C2)=O)cc(C)nc2[nH]nc(C)c12 c1(CC)nc(C(N2CCC(NC(C3CN(CC)CCO3)=O)CC2)=O)c(N)s1 c1(CCC(=O)NC(C(C)C)CNC(=O)C(C)c2ncco2)ccc(C#N)cc1F c1(CC(=O)NCC(=O)OCCC2CC23CC3)cccc(O)c1 CN1CCOCC1C(=O)NCC1CC(C(F)(F)F)CN1C(=O)CCCC#N N1(C(c2cc(C)sc2N)=O)CCC2CCN(C(C3CN(C)CCO3)=O)CC12 C1(C)(C(C)C)CCN1C(c1ccc(CNC(c2ccccc2)=O)s1)=O c1(C(=O)NC2CCCN(C(c3n[nH]c(C)c3Cl)=O)CC2)nnn2c1CCCCC2 c1(NC(=O)COC(c2cccc(CO)c2)=O)ccc(Cl)cc1Cl N1(C(C2(CSC)CC2)=O)CCN(CCNC(=O)CC2(C)CC2F)CC1 C12(CCCC1)C(=O)NC2.C(=O)(CN(C)C(C)=O)NC(C)C N1(C(C(C)CN(C)C)=O)CCN(C(=O)CNC(c2cnc(O)nc2O)=O)CC1C N1(C(c2ccc(CNC(c3c(CC)ocn3)=O)cc2)=O)CCOC(C)C1C CCC(C#N)(CC)C(=O)N1CC(N(C(=O)C=CCF)C)C2(CC2)C1 Cc1ccnc(O)c1C(N1CCC(O)C(N(C(=O)CCOC2CCCC2)C)C1)=O CC(C)(C)CC(C(=O)N1CCCC1CF)NC(c1ccsc1)=O N1(C(C(N2CCC(CN(CCCCl)CC)CC2)=O)=O)CCc2ccccc2C1 N1(C(C(CNC(C(C(C)C)SCC)=O)O)=O)CC2(CC(O)C2)C1 c1(C(N(CCCNC(C2(C)CCCO2)=O)CC)=O)cc(Br)c(Cl)s1 c1(C(=O)NCc2cn(C3CN(C(C4CC=CC4)=O)C3)nn2)cc(CO)ccn1 C(=O)(CC(C)(C)C(C)(F)F)NC(C)CCNC(C1(c2ccccc2)CCOC1)=O CCC(O)C(=O)OC.C1(CCOC(C)(C)C)CN1.C(=O)(C1CC1)O c1(CN(C)C(c2cc(-c3ccccc3)nn2C)=O)ccnc2ccsc12 c1(C(C)OC)nc(C(=O)NC(C)(C)CCNC(=O)C(C)CC2CC2)cs1 c1(C(=O)NC2C(NC(CCCn3ncc(C)c3)=O)CCC2)cnn2ccn(C)c12 c1(OC)nn(C)cc1CNC(=O)C(=O)NCC(c1ccncc1)C C(CC(=O)NCCn1cc(CN(C)C)nn1)NC(COCC)=O.COC C=CCC(CNC(c1cnnn1C)=O)C(=O)N1CCC(N2CC=CC2)C1 C1(NC(c2ccc(C(C)(C)OCC)cc2)=O)C2CC1N(C(=O)C(C)C1CC1)C2C N1(C(COC(C)=O)=O)CCOCC(C)(CNC(=O)CC2CN3CCC2CC3)C1 C1(C(N(CC(=O)NCC)CC)=O)CC2(CCN1C(=O)CSCC(N)=O)CC2 CC(C)C(N=c1[nH]c(Cl)nc(C2OCCO2)c1C(N)=O)C(=O)N(C)C C1(CN(C(=O)C(c2ccccc2)NC(C2CC2(Cl)Cl)=O)C)CCCC1(C)C C(=O)(CCS(N)(=O)=O)NCC1N(C(c2ccc(C(C)=O)o2)=O)CC=C1 C1(C)(C(=O)OC)CCN1C(C1(CNC(=O)C(n2cc(C)cn2)C)CCC1)=O NC1(CC(=O)NCCOCc2ccc(F)cc2F)CCCS(=O)(=O)C1 C=CCCCC(C(=O)N(C)Cc1cncnc1)NC(=O)C(C1(C)CCOCC1)C C(=O)(CCCC(C)(C)C)NCCCC(=O)NCC(CC=C)NC(=O)C(C)C(C)(F)F N1(C(COCC)=O)CC(CC(=O)N(C)Cc2ccncn2)CC1C C=CCN=C(NCC1C(F)(F)C12CCC2)N1CC(C)N(C)C(C)C1 c1(C(C)C)ccc2cc(C(=O)NCCCN(C)C(C3CCS(=O)CC3)=O)[nH]c2c1 C(=O)(CC(F)(F)C(C)C)NCC1CC(NC(C(C)(C2CC2)OC)=O)C1 C1(C(=O)NC(CCC)CC)CCN(C(=O)CC2CC(C)=NO2)C(C)C1 c1(OC(C(=O)NC2C(NC(C3(CCCC)CC3)=O)CC2)CC)ccccc1C C1(N(C(=O)CCc2ccccc2)C)CC2CCC(C1)N2C(c1ncccc1N)=O c1(NC(C(c2cc(Br)c(Cl)s2)N(C(CC)(C)C)C)=O)cccc(OC)c1 c1(CC(=O)NCc2c(CCNC(C)=O)ocn2)cccc2cnccc12 c1(N(CCCNC(C)=O)C)cc(S(=O)(=O)NCC(O)C2CCC2)ccc1C#N C1(CC=C)(C(=O)NC(C2(CSC)CC2)C)CCN(C(=O)C(Cl)Cl)C1 N1(C(c2cc(CNC(C(CC#C)C3CC3)=O)on2)=O)C2CCC1CC(F)C2 C(=O)(C(CC)CCOC)NC(C(=O)NCc1c(CC)nn[nH]1)C N(C1CN(C(C2(C3CCC3)CC2(F)F)=O)Cc2ccccc21)C(C1CCC1)=O c1(CNC2CCC(C(=O)NCc3ccsc3)C2)cc(Cl)nc(Cl)c1 CC(C)(C)C(=O)NCCCC(c1ccccc1)N(C(=O)CC1(C(F)F)CC1)C(C)C c1(N(C2Cc3ccccc3C2)C)[nH]c(=NCC(C)(C)CS(C)(=O)=O)nc2scnc12 N1(C(C(C)SCCCC)=O)CC(F)CC1CNC(c1noc(CC)c1C)=O c1(CCNC(=O)NC2CCCC2C(F)F)cn(CC2CC2)nn1 c1(CC(=O)NC2C(CNC(C3(C)CCCO3)=O)CC2)ccc(Br)nc1 N1(C(C2C3(CC(C)(C)C3)C2)=O)CCCC12CCN(C(c1sccc1Cl)=O)C2 N1(C(C(c2cccc(C)c2)=O)=O)CCC(NC(C2CCCN2C(C)C)=O)C2CC12 C1(C2CCCO2)(C(N2CC(NC(C(C)=CC)=O)CC3(C2)CC3)=O)CCCO1 CC(CCN(C)C)C(=O)NCC1CN(c2ncns2)CCO1 c1(OC)ccc(C(=O)NCC(CNC(C23CCC(CO2)C3)=O)CO)cn1 Cc1cccc2cc(C(N3CCN(C(=O)Cn4ccc(=N)[nH]4)CC3C)=O)oc12 C(=O)(CS(C)(=O)=O)NC(C(=O)NCC(C1CCCC1)C)Cc1cc[nH]n1 N1(C(CC2(OC)CC2)=O)C2CCC1CC(F)(CNC(=O)CCCCC(C)(C)C)C2 N1(CCNC(C2N(CC)CC2)=O)CCCN(C(c2cnnn2C)=O)CC1 C1(CC(=O)NC2(C(=O)NCCc3n(C)cnn3)CC(CO)C2)CCCC2CC12 CN1N=C(C(=O)NC2CC3CC(C2)N(C(=O)CSc2cccs2)C3)CCC1=O N1(CC)CCC(C(=O)NCC2(NC(=O)CC#N)CC2)C1 N1(C(C(C)C(C)(C)C)=O)C2CCC1CC(NC(C1(c3ccncc3)CCC1)=O)C2 C(N=c1ccn(CC(=O)NCC(N)=O)c(O)n1)c1ccc(OC)c(C)c1C N1(C(c2ccccc2S)=O)CCC2(CCN(Cc3cccc(Cl)c3)C2)C1 c1(C(N(C(C(=O)NC(CCCC)CO)C)CC)=O)cc(O)nc(O)n1 c1(C(=O)NCC2(NC(C3(CCC)CC3)=O)CC2)ccc(N(C)CC)nc1.C=O C1(CNC(C2C(C)(C(C)C)C2)=O)CCN(C(c2ccccc2SCC#N)=O)CC1 c1(C(=O)NCC(CN(C(c2c(CC)nns2)=O)C)O)ccc(OC)c([N+](=O)[O-])c1 C(C(C(=O)OC)N(C(=O)C(CNN(C)C)c1ccccc1)C)OCC=C N1(C(C2ON=C(C)C2)=O)CC(NC(C2CC(C(F)(F)F)C2)=O)C(C2CC2)C1 N1(C(C(C)n2cncn2)=O)CCN(C(c2nncn2C2CC2)=O)CC1CO CCC(C(=O)NC1CC(C(C)NC(c2ccc(C(F)(F)F)o2)=O)C1)C1CC1 c1(SC(C)(C)C)ccc(C(=O)NC2(C)CC(NC(C3C4CCC3CC4)=O)C2)cn1 C1(C(=O)Nc2cc(-n3cc(CNC(CC)=O)nn3)ncc2)CCC(F)(F)CC1 Cc1cc(C(=O)NC2CC(C(F)C(=O)NCCC34CC(CCO3)C4)C2)cnc1O c1(C(C)C)ccc2ncnc(N3CCC(N4CC(C(F)F)C4)CC3)c2c1 C1(OC)CC(C(=O)NC(C)Cn2cccn2)N(C(=O)C=CCN2CCC2)C1 CC1CN(C(=O)CC(CC2CC2)NC(=O)CC2CCCN(C)C2)CC(=O)N1 c1(CC(=O)NC2CCCC2NC(C2CC(F)C2)=O)ccc2c(c1)OCCO2 C1(CCNC(c2nc(C)n(C)c2)=O)CCN(C(=O)CS(=O)(=O)C2CC2)CC1(F)F C1(CNC(COC2(C)CCC2)=O)CCC(NC(=O)CC2CCCCO2)CC1 CC1C(C(=O)NC2CN(C(=O)CS(=O)(=O)CCO)CC23CC3)=Cc2ccccc21 CC(C)C(O)CCN=c1[nH]c(=NC(C)CC(C)(C)C2CC2)[nH]c2c1CCCC2 C(=O)(C1=NOC(C)C1)NC1(CCCNC(C2(OC)CCCSC2)=O)CC1 c1(C(N2CCN(C(c3c(SC)scc3)=O)CC(O)C2)=O)cccc2ncn(C)c12 c1(C(=O)NCCN(C(=O)Cc2nc[nH]n2)CCOC)cccc(C(F)(F)F)c1 c1(NC2C(=C)COC2)cc(-n2cccc2)cc(Cl)c1 C1(C(N2CC(C(=O)OC)(CC)C2)=O)CCC(C(C)C)N1C(c1c[nH]c(C#N)c1)=O c1(C(=O)NCCN(C(C2CC2(COC)CC)=O)CC)ccc2c(c1)C1CCC2O1 c1(CN(CCCNC(c2c(C)nns2)=O)C(C)C)ccc(Cl)c([N+](=O)[O-])c1 c1(C(=O)NC2CN(C(c3n(CCC)ncc3)=O)C(C)C2)ccc2c(c1O)CCC2 c1(C2(CNC(CCC)CO)CC2)ccc(-c2cccnc2OC(=O)C2CC2)cc1 C(c1cc(C)ccn1)=CCNC(c1n(CCCSC)nnn1)(C)CC1CC1 N1(C(CCC(=O)OCC)=O)CC2CCCC(C1)N2C(=O)C(CC)SC c1(CC(=O)NCC(CNC(C(c2ccccc2)NC(N)=O)=O)F)ccc(O)cc1 n1(CC)nccc1C=CC(N1CC(NC(c2cc(C)oc2C)=O)C(O)C1)=O CCCCC(O)C(=O)NC1CCC(C(=O)Nc2cnc[nH]2)C1 c1(C(=O)NC2C(C)N(C(C3CC4(C3)CC4F)=O)CC2)cc2ccc(F)cc2o1 N1(C(C2CCN(C(=O)NCC)C2C)=O)CCCC(NC(=O)CN(C)CC2CC2)C1 Cc1cc(=NC(=O)CN(CC(C)NC(=O)CCC2CCC(O)CC2)C)[nH]o1 C1(C(N2CC(CNC(C3CC(C)(F)C3)=O)OCC2)=O)Cc2ccncc2C1 N1(C(CC(C)(C)O)=O)CCCCC(NC(c2ncnn2C2CCOCC2)=O)CC1 c1(SCC=C)ccccc1C(=O)NC1CN(C(=O)CNC(=O)CCC)CC1F c1(C(CNC(=O)C(CC)C2CCC2)NC(c2c(CC)c[nH]n2)=O)cccc(C)c1 c1(NC(C2(CC#C)CC=CCC2)=O)ccc2sc(S)nc2c1 C#CC(C)(C)C(=O)NCC1CCC1NC(=O)C(F)C(C)C N1(C(CCCC=C)=O)CCC2CCN(C(c3cc(CC4CCC4)c[nH]3)=O)CC2C1 CC(F)(F)CCC(=O)N1CC(NC(c2cc(=O)cc[nH]2)=O)CC(O)C1 C1(NC(c2nc(COC)sc2)=O)CCCN(C(c2sc(COC)nc2C)=O)C1 CC1CCc2c(C(N3CC4CC3C4NC(C3CN(CC(C)C)C3)=O)=O)csc2C1 O=C1CCC(C(=O)N2CC3(CNC(C45CCCCC(F)(C4)C5)=O)CC2CO3)=NN1 C=CC1(CC(=O)NC(c2ncnn2C)C)CN(C(c2cnnn2C2CC2)=O)C1 C1(C(N(C)Cc2c(C)cco2)=O)CC(F)(F)CN1C(=O)CCCC(=O)N(C)C c1(CNC(=O)NCCCOCCCN(C)CC)cnoc1CC(C)C C12CN(CC1(C)C)CC(=O)N2C.N1(CC(C)C)CCCC1CN(C)C c1(C(N(C(C)CNC(c2[nH]nnc2C2CC2)=O)C)=O)c(O)ccc(Cl)c1F c1(CN=C(NC(C#C)COC)NC(C)COC)ccc2ncccc2c1 N1(C(C2(CC#C)CCC2)=O)CC2CCC1C(CNC(C1CCC(C(N)=O)O1)=O)C2 CCC(C)CC(C(=O)NCc1ccncc1CO)NC(=O)C(=O)N(C)C C1(C(=O)NC(CNC(c2nc(C(C)C)sc2)=O)C)CC2(COCCO2)C1 N1(C(c2c(CC)ocn2)=O)CCC(CNC(C2CSC2)=O)C(O)C1 c1(C(=O)OC(C)(C)C)cc(F)c(C(=O)NCc2c(C(=O)OC)cccc2)cc1F c1(NC(c2ccnc(C(=O)NC3C(COC)C3)c2)=O)cc(Cl)cc(OC)c1OC C1(CNC(=O)COCCc2ccccc2)CN(C(C2(F)CCOC2)=O)CC1(F)F CN1CC(=O)NC(CC(N2C3CCC2CC(NC(c2cnn[nH]2)=O)C3)=O)C1=O c1(OCC)ncccc1C(=O)NCCC1CC(NC(=O)C(C)(C)NS(C)(=O)=O)C1 Cc1ncc2n1CCN(C(C1CC(C)(NC(c3cccc4ccoc34)=O)C1)=O)C2 N1(C(=O)OC)CC2CC1CN2C(=O)CC=CCNc1ncc(C(=O)OC)nc1 c1(C(=O)NC2CC3CCC(C2)N3C(=O)CC2CCCO2)ccc2cncnc2c1 c1(C(=O)NCC(=O)NC)nn(-c2ccccc2F)c2c1CCC2 N1(C(c2ccc(N)cn2)=O)CC2CC1CN2C(c1csc(O)n1)=O CCCC(CC)CCC(=O)N(CC(=O)NC1CCC(F)CC1)CCC N1(C(C(F)=C(C)C)=O)CC(O)(CCNC(c2cnsn2)=O)C1 c1(C(=O)NC(C2CCCN2C(c2c[nH]c(C(F)(F)F)c2)=O)(C)C)c[nH]ccc1=O CC1(C)OC(=O)CC1C(N1CCN(C(=O)CCc2nc(C3CC3)no2)CC1)=O CC(F)(F)C(F)(F)CC(=O)NCC1(C)CN(C(c2sccc2F)=O)CCO1 Cc1cc(=O)c(C(N2CCCCC2CCNC(=O)C(F)OC(F)(F)F)=O)c[nH]1 c1(CC(N2CC(C(=O)Nc3c(C(=O)NC)cccc3)C2)=O)ccc(Br)cc1I N1(C(C(N2CCOCC2)C)=O)CCC(F)(F)C(C(=O)Nc2cccnc2)C1 c1(OC)cnc(F)c(C(=O)NCC2C3CN(C(C4(C#N)CCSCC4)=O)CC23)c1 N1(C(C=Cc2ccc(CC)cc2)=O)CCCC2(CCN(C(=O)CCSC)C2)C1 C(=O)(C(CC(F)F)C1CCC1)N(C1CC(NC(=O)Cc2nc(=N)[nH][nH]2)C1)C C(=O)(CCCC(=O)N1CC(CNC(c2conc2C2CCC2)=O)C2CC12)NCC CC1(F)CCCCN(C(=O)COCCNC(=O)CCCCC#N)C1 c1(C(N(CCNC(C(C)OCC)=O)CC)=O)ccc(F)c2ccccc12 c1(C(N2CCC(c3ccccc3)(NC(CCC=C)=O)C2)=O)cc(C)nc(C)c1 C1(CNC(c2nc(C(C)OC)sc2)=O)CCCCN(C(c2nc(Cl)cs2)=O)C1 C1(OC)CC(CNC(=O)CCCNS(C)(=O)=O)N(C(=O)CCCc2ncco2)C1 C1(NC(c2c(C)cco2)=O)CC2CC(NC(C3CC3c3nccn3C)=O)C2C1 n1(CC)nc(C(C)C)cc1C(=O)NC(C)C(C)NC(=O)Cn1cccnc1=O CCCC(CCC)C(=O)NCC1(OC)CN(C(=O)Cn2c(C)cc(O)cc2=O)C1 C(CC(C(=O)Nc1ccc(Cl)cc1)NC(=O)CCC1(C#N)CCC1)=CC N1(C(c2cccc(COC)c2)=O)CCN(C(c2cc(C#N)c[nH]2)=O)C(C)C1 c1(C(N2CCC(NC(C(C(C)C)N3CCCCC3)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 C1(C(=O)Nc2c(C)ncnc2)CC2C=CC1N(C(C1(Cl)C3CCC(=O)C13)=O)C2 c1(OCC#C)ncccc1C(=O)NCC(C1CCCC1)NC(C1CCOC1)=O C1(CC)CN(C(C2CC2(C)C)=O)CCC1NC(=O)CN(CCCCCC)C C1(CC)CCN(C(=O)Cc2csc(C)c2)C1C(=O)NCC1CCCOCC1 Cc1cccc(C)c1CC(=O)NC1CCC(NC(C23CC(CO2)C3(C)C)=O)CC1 C1(CC(=O)NC2C=CCN(C(c3cc(CSCC)on3)=O)C2)CN2CCC1CC2 N1(C(C=Cc2cncc(C)c2)=O)CC2(COC(CNC(=O)C(C)C3CCC3)C2)C1 CCCC(C)CC(=O)N(CCCCCCNC(=O)CCn1cccn1)C C(C(C)(CC(C)C)NC(=O)C1=NOC(C(C)(C)C)C1)NC(c1c(C)cc(C)s1)=O N1(C(CCC=C)=O)CCN(C(C2CC(=O)N(C(CC)CC)C2)=O)C2(CC2)C1 C#CCC(C)(C(=O)NCC(C)OCCO)NC(=O)CC1OCCC1C c1(CC)cc(C)c(NCC(C2CCCC(=O)N2)(C)C)cn1 C(=O)(N=c1cc[nH]c(C)c1Br)NCC1CCN(c2ncc(OC)cn2)CC1 c1(C(N2CCC(O)(CNC(C(CCC)=CCC)=O)C2)=O)ccc(F)c2[nH]ccc12 N1(C(Cc2c(C(C)C)con2)=O)CCN(C(c2ccc(=O)oc2)=O)C2CCC12 c1(NC(C(=O)N(C2CCCN(C(COCCC)=O)C2)C)=O)ccc(C#N)c(Cl)c1 N1(C(C(C)Oc2ccccc2)=O)CCOCC1CC(N1CC2CC2C1)=O CCC(C)C(C(=O)Nc1nnc(-c2nn[nH]n2)s1)N1CCCC1 C1(NC(C2CCC(=O)C2)=O)CN(C(=O)C=C2CN3CCC2CC3)C2(CCCC2)C1 C1(NC(CC2CC(=C)C2)=O)CN(C(=O)Cc2ccc(C)cc2)C2(CCCOC2)C1 c1(OC)ccc(Cl)c(C(=O)NCC(C2CCCC2)NC(=O)CO)n1.C1C(=O)O1 Cc1cc([N+](=O)[O-])ncc1C(=O)Nc1ccc2c(c1)COC2 C=CC1CCCN(C(c2ccnc(CNC(c3ccsc3C#N)=O)c2)=O)C1 c1(OC)ccc(NC(N2CCCC(Cc3cccc(F)c3)C2)=O)c(OC)c1Br c1(C(N(CC)Cc2cc(F)ccc2F)=O)cc(C2=CCSCC2)n[nH]1 c1(C(=O)NCCCC(C)(C)NC(=O)CCCC2CC2)cc(S(N)(=O)=O)c(Cl)o1 C1(C2CCCC2)(C(N2CCOC3CN(C(CCCSC)=O)CC32)=O)CCNC1=O N1(C(CCc2cc(C)no2)=O)CCN(C(C2(O)CCOC2)=O)CC(C)C1 C(C1CCN(C(C2(C)COC2)=O)CC1)=CC(=O)NC1CC(C)OC1=O c1(CNC(c2c(C(C)C)nco2)=O)ccccc1CNC(C1CCCC12CC2)=O C1(NC(c2nc(C)c(C)s2)=O)CC2CN(C(=O)C(C)C3CCC3)CC2C1 N1(C(CSCC#C)=O)CCC2(C=C(C(=O)NCC(O)CC3CCCC3)C2)C1 C1(C(N2CC(NC(c3c(OCC)ccs3)=O)C(F)C2)=O)CCC2(CC1)CC2 CC1CCC(Cl)=C(C(=O)N(C2CC23CC3)C)C1 c1(C(N2CCC(CNC(CCCCCC)=O)CC2)=O)cc(=NC)[nH]cc1Br C1(C(=O)NC2CC(NC(C(Cc3cn(C)nc3)O)=O)C2)C2CCCCCC12 C1(NC(COC)=O)CN(C(c2ccc(Cn3cccc3)cc2)=O)CCC1C C1(NC(C2(CC=C)CCC2)=O)CC(C)N(C(=O)COCc2ccccc2C)C1 C1(CCC)CCCN1C(=O)CCC1(NC(=O)COC2CCCC2)CCC1 C1(CNC(CC(C)OC)=O)CC(NC(c2ncsc2C2CC2)=O)C(O)C1 C(=O)(C(C(=O)NCCOCC(=O)NCc1cncc(CN(C)C)n1)OC)OC Cc1cccc2c1C(NC(C1CCCN(CC(C3CCNCC3)O)C1)=O)C(=O)N2 c1(CC(=O)NCC(CC(F)(F)F)NC(C(C(C)C)O)=O)ncn2c1CCCC2 Cc1cccc(F)c1CC(=O)NC1(C)CCN(C(=O)CC(C)C)CC1 N1(C(CCCC)=O)CCCC2(CC(NC(c3sc(Br)cc3F)=O)CO2)C1 c1(CN(C(CC)C)C(C2COCC2Sc2ncccn2)=O)cc(C(C)(C)C)oc1C C1(NC(C)=O)CCN(C(=O)COc2cccc(C(C)C)c2)CC1C S(=O)(=O)(c1cc(C(F)(F)F)ccc1NC1C=CC(CO)C1)N1C(C)C(O)CC1 c1(C(=O)NCC(CCNC(C2C(C)OCC2)=O)O)ccnc(-c2ccco2)c1 CC1C(NC(c2cc(C(F)(F)F)ccn2)=O)CCCN1C(c1cnsc1)=O CN1CCN(C(c2occc2C2CC2)=O)CC1CNC(=O)CCc1cnn(C)n1 c1(C(=O)NCCC(C)NC(c2ncnc(O)c2Cl)=O)cccc2c1NCCC2 c1(C(=O)NC2CC(NC(CSC)=O)C23CCC3)nnn2cc(C)nc(O)c12 Cn1cncc1CCNC(=O)C(Cc1cnc[nH]1)NC(=O)CC1CCCSC1 CC1=NOC(C(=O)NCC2(C3CCCCO3)CC2)C1C CCC(C)C(C(=O)NCc1ccccc1Br)NC(=O)Cc1nccn1C c1(C(N2CCC(O)(CN(C(=O)Cc3ccnn3C)C)C2)=O)ccsc1S(N)(=O)=O c1(C(=O)NC2CC(NC(C3C(C=C)CC3)=O)C2)ccc(-c2ccccc2)nc1O N1(C(C(CCCC)NC(=O)CCc2ccncn2)=O)Cc2c[nH]nc2C(C)C1 C1(NS(CC=C)(=O)=O)C=CC(=O)N=N1.C12CCCN1C(=O)C2 c1(C(N(C(CNC(c2cc(C)ns2)=O)C2CC2)C)=O)cc2cc(Cl)ccc2n1C C1(C(=O)NC(CNC(CC=C)=O)C)CCCN1C1CCCCC1 C(CCC)(CCC)NC(C(CC1CCOCC1)NC(C(C=CC)O)=O)=O c1(OC)ccncc1CNC(C1CC(NC(=O)CCCC2CCCO2)CCO1)=O C1(OC)CC(CNC(C2(C)CS(=O)(=O)C2)=O)N(C(=O)CCCc2csc(C)n2)C1 C1(O)(CCNC(=O)CC(O)C2CC2)CCCN(C(=O)CCCc2cnccn2)C1 c1(C(N2CC3(CCN(C(CC(=C=C)C)=O)C3)C2)=O)cnc2sc(C)cn2c1=O CN1CCc2nc(C(=O)NC3CC4CC3N(C(=O)CCc3cn[nH]c3)C4)sc2C1 C(C)(CN=c1ccnc(NC(CC(F)F)c2ccccc2)[nH]1)OC C1(O)(C(C)NC(c2c(CC)nns2)=O)CCN(C(=O)C(N2CCOC2=O)C)CC1 c1(C(=O)NC2C3CCC(CN(C(C(CC)C)=O)C3)C2)cncc2c(F)cccc12 CC(C)C(O)CC(=O)N1CC2(CO)CC1(C(=O)NCC(c1ccccc1)O)C2 S(=O)(=O)(c1ccc(C(C)(C)C)cc1)NC(C1(C(=O)O)C(C)C1)=O CC1CCN(CCc2cn(CCCC(=O)N3CCC3CC3CCCC3)nn2)C1 c1(NCC2C(C)COCC2)ccc(S(=O)(=O)NCC2(CC3CCC3)CC2)c(Br)c1 c1(C(N2CC(OC)(CNC(=O)CCCF)C2)=O)c(Cl)ccc2cc(CO)cnc12 c1(C(=O)NC23C(NC(c4c(C)con4)=O)CC(CC2)C3)cccc2ccn(C)c12 c1(C(=O)NCC2CCN(C(c3cn(CCC)nn3)=O)C2)cccc(S(C)(=O)=O)c1 c1(NC(C2N(Cc3cccc(OC)c3OC)CCOC2)=O)csc2ccncc12 C(=O)(CCCC(=O)OC)N1CCC(N(CCCCC)C)C1 C1(CNC(Cc2ccc(N)cc2)=O)CN(C(C2(C(N)=O)CC2)=O)CCCO1 CC(C)CC(CNC(=O)C(C)(C)N(C)CC)NC(C1CCCN1c1nccs1)=O c1(CNC(=O)NC(Cc2cscn2)Cc2ccccc2)noc(C(F)(F)F)n1 C1(NC(C(CCCOC)C)=O)CC2CCC1N(c1ccnc(-c3nccs3)n1)C2 c1(C(=O)NCC2C(NC(CC(C)C)=O)CCCC2)cc2c(nn1)OCCS2 CN1CCCC(CC(N2CCC(C(C)(C)C)(CNC(=O)C(C)(C)CF)C2)=O)C1 C1(C(N2CCC(C#N)C2)=O)CCCCCN1C(=O)C=C1CCC1 c1(C(=O)NC(C)(CNC(=O)CCc2cnoc2)CO)ccc(C2CC2)cc1Cl c1(C(N2CCN(C(c3cc(F)cc(Cl)c3)=O)C(CO)C2)=O)cc(Cl)cnc1Br N1(C(CN(C2CCC2)C)=O)CC2CCC1CN2C(=O)CCC1CCCOC1 C=C(C)CC(C(=O)N=CC(=O)OC)NC(=O)C(C)CCCOC Cc1occ(C(F)(F)F)c1CC(=O)NCC(C(C)C)NC(C1(CC(F)F)CC1)=O C(CC(C(=O)NCc1ccc(C)nc1)NC(=O)CC1CCCC1O)SC c1(SCC)cnccc1C(N1CCC(CCOC)(NC(=O)CC(C)C)C1)=O C(=O)(C(C)(C)C(O)C(C)C)N1CC(OC)(CNC(=O)C=Cc2cccc(F)c2)C1 C1(NC(C2CCC(C)O2)=O)CN(C(=O)CC2=CCN(C)CC2)Cc2nccn2C1 C1(C)(CNC(C(COCC)NC(=O)CN(C)CCOC)=O)CCc2ccccc21 N#CCCCCCC(=O)N1CCCC(NC(C2(C(F)F)CC(F)(F)C2)=O)C1 N1(C(Cc2c(C)noc2Cl)=O)CC2CCC(C1CO)N2C(c1ccoc1)=O N1(c2c(F)cnc(C(=O)OC)n2)CCc2sc(-c3ccc(O)c(C)c3)nc2C1 CN1C(=O)OCC1C(=O)NCCN(C)C(C1(NC(c2ccccc2)=O)CC1)=O C1(C(=O)NC2CN(CCOC)C2)(CC)CCN(C(=O)C(C)=C2CCCC2)C1 c1(C(N2CCCC(C(C)(C)C(=O)N3C(CO)CC3CO)C2)=O)ncccc1O c1(-c2nc(-c3cn(C)nc3)nn2CCCC(F)F)n[nH]c2c1CC(C)(C)CC2 CCCC(CCCS(C)(=O)=O)C(=O)NC1CC(CNC(=O)C2=NOC3(CCC3)C2)C1 C(c1cncnc1O)=CC(N1CC(CNC(=O)C(F)(F)CC2CC2)C1)=O c1(-c2n(CCOC)c(N3CCOC(C(C)(C)C)C3)nn2)nccn2cccc12 c1(C(N(C(C)C(=O)NC(CC2CC2)C2CC2)CCC)=O)cn2ccccc2n1 Cc1ccc(CNC(C2CC(C)N2C(=O)C=Cc2cocn2)=O)cn1 C1(CCC(=O)NCC(C(C)O)C)CCCCN1C(C1CCC(N(C)C)C1)=O c1(C(C(=O)NCC(=C)C)N(CC(=O)NC2CC2)CCOC)cc(Cl)ccc1Cl CCCC(C(=O)N1CCCC1CCCNC(c1ncccc1CC)=O)NC(C)=O Cc1cc(C(=O)CSCC(N2CCCC2CSC2CC2)=O)cs1 N1(C(c2snc(C)c2N)=O)CCC2CCN(C(c3coc(O)n3)=O)C2C1 CC12CC(NC(=O)C=CC3CC3)(C1)C1(CN(C(=O)COC3CCCOC3)C1)O2 c1(C(N)=O)ccc(NCC2CCN(C(C3CC4C(C3)C4(C)C)=O)C2)c([N+](=O)[O-])c1 n1(CC(N2CC(NC(C=COCC)=O)C3(C2)CC3)=O)c(C)nc2ccccc12 c1(NC(C2CC(F)CN2C(c2ccccn2)=O)=O)cc(F)c(Cl)cn1 C(CCCC(C)(C)C(=O)NN)NC(c1ccc(N2CCN(C)CC2)c(F)c1)=O CC(C)(CO)C(O)C(=O)NC1CCCOC1 C1(C(N(CC(C)NC(=O)Cc2cncs2)C)=O)CC12C1CC3CC(C1)CC2C3 n1(CC(=O)NCC(N2CCCOCC2)=O)c(C2CCNCC2)nnc1S N1(C(c2n(C)ncc2[N+](=O)[O-])=O)CCCC2(CCN(C(=O)C(N)=O)CC2)C1 C1(C(=O)NC2C(CCOC)CCC2)CCC(C)CN1C(=O)Cn1ccnn1 CC1OC(=O)NC1C(=O)NC1CCCC1CNC(c1ccc(C(C)(C)C)o1)=O c1(C(=O)NC2CN(C(=O)CNC(=O)C3CC3)CC2F)cnc2cc(Cl)ccn12 C(N=c1ccc(Br)c(S(=O)(=O)NCC#Cc2ccccc2Cl)[nH]1)C1(OC)CCC1 c1(CC(=O)NC(c2cc(Cl)sc2Cl)C)c[nH]c2ccncc12 C1(COC)CC(CNC(=O)CCC2(O)CCC2)N(C(=O)CCCn2cccn2)C1 c1(CC(=O)NCC(C)(C)NC(=O)CS(=O)(=O)NC2CC2)cc2ccccc2o1 c1(C(=O)NCCSc2ccc(OCCOC)cc2)cc2c(C)nn(CCCl)c2s1 c1(C(=O)OC)no[nH]c1=NC(=O)CC1CCN(C(=O)CC2CCCC2)C1 c1(NC(=O)Nc2c(C(=O)OC)cc(Br)cc2C)cc(C)c(F)cc1Br N1(C(=O)CCCCC2CC2)CCC2CCN(c3nc(Cl)ncc3C3CC3)CC2C1 C1(C(=O)NC)CN(C(=O)CCCC2CCCO2)CC1c1ccc(C)cc1 CCCC(C(=O)NC(CCN(C)C)C(=O)N1CC(N2CCC2)C1)OCC C1(N(C(c2n(CCC)nc(C)c2)=O)C)CC2CCC(C1)N2C(c1cc(Cl)c[nH]1)=O c1(C(N2C(CCNC(C3C(C#N)C3)=O)CCCC2)=O)cc2ccc(F)cc2[nH]1 N1(C(CC)=O)CCCC2(CCN(C(C3(C)COC(C)CO3)=O)C2)C1 c1(C(=O)NC(C(C)C)CCNC(c2cc(C#N)c[nH]2)=O)cc2c(F)cccc2[nH]1 c1(OC)ccc(Cl)c(S(=O)(=O)NC(C)C(F)F)c1 CC12CCCCC1CN2C(=O)CC(O)CNC(c1cnco1)=O C(=O)(C(CC(C)(C)C)OC)NCC(=O)NCCCN(C(c1cccs1)=O)CC c1(C(=O)NCC(C2CCN(C(C3CCC3)=O)CC2)(C)C)ccc(Br)cc1N Cc1cccc2c(C(=O)NC3CC3CNC(C3(C4CCCCO4)CC3)=O)n[nH]c12 CC1(NC(=O)CN(C(=O)C=Cc2ccco2)CC2CC2)CCOCC1 Cc1cccc2c1OCCC2Nc1nccc(N2CCC(n3cccn3)C2)n1 c1(C(N2CCC(CNC(C3(CCCC)CC3)=O)C2)=O)cnc(Br)c(OC)c1 c1(C(Cc2ccccc2)NC(Cc2n(CC)cnc2)=O)ccccc1Br C1(NC(c2ccc(=N)[nH]n2)=O)CC2(C1)CN(C(C1(O)CC1)=O)C2 N1(C(C2(NC(C3N(CC)CC3)=O)CC(O)C2)=O)CC2CN(C)CC2C1 CC1CN(C)CC1C(N1CCCC1CNC(c1cnn(C)c1)=O)=O C1(C)(C(N2CC(NC(c3c(C)cc(F)cc3)=O)C(C)(C)C2)=O)CCC(C)C1(C)C N1(C(COC)=O)CC(CNC(C2(Br)CC2(F)F)=O)(OC)C1 CCCCC(CC)CC(=O)NCCCC(CO)NC(=O)C(C)c1ccco1 CC(C(C)C(=O)N(CCC(F)(F)F)C)NC(c1cccc(=O)o1)=O C1(F)(CNC(C2CC(O)(C(F)(F)F)C2)=O)CCN(C(=O)CSC2CCOC2=O)C1 c1(C(N2CC(Cn3cc(C(C)O)nn3)OCC2)=O)cc(F)c(C(F)F)c(F)c1 c1(C(N2CC(F)(C(=O)OC)C2)=O)ccc2sccc2c1 n1(CCN(CCC)CC2CCCO2)c(N(c2cccc(COC)c2)C)nnc1C c1(C(=O)NCC2N(C(CCc3ccc(C)s3)=O)CC2)coc2c1CS(=O)(=O)C2 C(=O)(C1=CC2(CCOCC2)C1)NCC1N(C(=O)OC(C)(C)C)CCC(C)(C)C1 N1(C(C(c2c(C)n[nH]c2C)C)=O)CCCC2CN(C(=O)Cc3n[nH]c(=N)s3)CC12 c1(CN(C(c2nccc(OC)c2)=O)C(C)C)cc2ccccc2n1C c1(C(N2CC(N(C(C3CC(SC)C3)=O)C)C(C)(C)C2)=O)ccc(S(C)(=O)=O)o1 c1(NC(CC)CSC)ncnc2cc(Br)c([N+](=O)[O-])cc12 C(CNCCO)(C(C)(C)C)NC(CCOCCOC)=O.C(=O)(C(CC)O)NCC(F)(F)F C(=O)(N=c1ccn(C2CC2)[nH]1)C1CCCC(NC(C(CCC)F)=O)CC1 N1(C(CSCC=CC)=O)CCCC2CN(C(=O)C(C)=CC)CCC12.C(C)(C)(C)NC(=O)O c1(C(=O)NCC(C(=O)NC(CC#C)CO)N(C)C)nn(C)cc1C N1(C(CC(CCC)C)=O)CC2=C(C1)CN(C(=O)CCCCNC(N)=O)C2 CCC(CC(=O)NCc1nnnn1C)NC(c1cc(C2CC2)[nH]n1)=O C(=O)(C(C(F)(F)F)NCc1c(CS(=O)(=O)NC)cccc1)OCC C1(OC)CC(C(N2CC3CC3(NC(c3c(C(F)F)cnn3C)=O)C2)=O)CC1OC C(C(F)(F)C(=O)NCC(C)N(C)C(c1cccc(CC(=O)OC)c1)=O)OC CCCCC(C(=O)NCC1CN(C(=O)C(c2cc(F)cc(F)c2)O)C1)N(C)C C1(C2CCN(C(c3conc3C3CC3)=O)C2)(NC(=O)C=C(Cl)Cl)CC1 C1(C(=O)NC2CN(C(C(C)CSC(F)(F)F)=O)C2)CNC(=O)CC1C C1(N(C(c2cc(C)co2)=O)CC)CCN(C(=O)CC(c2ccccc2)SC)CC1 CN1CC(=O)NCC1C(=O)NCc1csc(-c2ccccc2)n1 c1(NC(c2ccc(NCc3cccc(C)n3)cn2)=O)ccc2ncn(C)c2c1 C1(NC(c2cccnc2)C(C)C)C2CCCC1CC2 CCC(CC(C)CO)NC(=O)CCCNC(C1(O)CCCC1)=O c1(NCC(=O)NCC2(O)CN(C(C(=O)NCCNC(C)=O)=O)C2)ccc(F)cc1 C1(CNC(C2CCN(CC)C2)=O)CN(C(=O)CCc2cncc(O)c2)CCCO1 C(C)(C(C(=O)NC1CCCC1CF)C(C)C)NC(c1n(CC)nnc1)=O c1(C(=O)NCC(C)N(C(c2n[nH]cc2C)=O)CC)oc(-c2ccccc2)nc1C C1(NC(c2c(C)coc2)=O)C2CC3CN(C(c4cnc(Br)s4)=O)C1C3C2 Cc1cccc(F)c1C(N1CCC(N(C(=O)CCc2cc[nH]n2)C)CC1)=O C1(NC(C(CC)CC(F)F)=O)CCC2(CC1)CN(C(c1csnc1C)=O)CCO2 n1(CC(=O)NC(CC)CNC(=O)CC2(NC(C)=O)CC2)nc(C)c(Cl)c1C C1(C(=O)NC(CCC)CO)C2CCC(C2)C1NC(c1nc(C)oc1C)=O C#CCC(C(=O)NC1(CO)CN(C(c2sc(N3CCCC3)nc2Cl)=O)C1)C1CC1 C1(C(=O)NCCC2CCCN2C(=O)Cn2ncnn2)CC(C(F)(F)F)(NC2CC2)C1 C1(CNC(Cc2c(C)n(C)nc2)=O)CC2(CCN(C(c3cc(Cl)ns3)=O)C2)CO1 C1(C(N2C(Cl)(C(=O)OC)CC2)=O)(NC(=O)CCCC(C)O)CCN(C(C)=O)CC1 C1(O)(C(C)NC(=O)C=C2CCCC2)CCN(C(=O)CC(C)(C)O)C1 N1(C(C(COC)COC)=O)C(C)CC2CN(C(=O)COc3ccc(Cl)cc3)CC12 c1(C(CNc2ccccc2)=O)c[nH]c2cccc(F)c12.C12CNCC(C1)C(=O)N2 C1(C)(COC)CCN(C(=O)COC2CC(NC(=O)C(C)(C3(C)CC3)OC)C2)C1 Cc1nc(NC2CC2)sc1C(=O)NC(CNC(C1CN(C)CCO1)=O)C1CC1 N1(C(=O)NCCS(CC)=O)CCS(=O)(=NS(C)(=O)=O)CC1 c1(C(N2C3CC(CC(NC(c4c[nH]c(Br)c4)=O)C3)C2)=O)ccc([N+](=O)[O-])c(O)c1 n1(CC(=O)N(CC(=O)OC(C)(C)C)Cc2nc[nH]n2)nc(C)cc1CC c1(NC(C2C(NC(C=CC(C)C)=O)CCC2)=O)cccc([N+](=O)[O-])c1F CN(C)NC(=O)CCC(=O)N(C(C(N1CCC(N=[N+]=[N-])C1)=O)C1CC1)C c1(OC)cncc(CCC(=O)NCC2CCCCC2NC(C2(OC)CCC2)=O)c1 N1(C(=O)CC2CCN(C(C3C4CCC(F)C34)=O)C2)CCC2CCC(C1)S2 C12(C(=O)NCC3(CNC(C4OC5CCC4C5)=O)CC34CCC4)CCCC(CO1)C2 Cn1cc(C#N)cc1C(=O)NCC(C)(O)CNC(c1csc(C2CC2)n1)=O N1(C(c2c(CC)csc2)=O)CCN(C(c2cc(C)c(Br)o2)=O)C2CC12 CCCC(CCC)C(=O)N1CCCC(NC(c2cnc3[nH]cncc2-3)=O)C1 c1(C(=O)NC(c2ccc(OC)cc2)C)cccc(Sc2c(Cl)ccnc2Br)c1Cl CC1CN(C(=O)CCC2(C)CC2)CC(C)C1NC(=O)Cc1n[nH]c2c1CCCC2 C(CC)(CCCC(=O)NCC=CC)NC(C(C)OCCC#C)=O C1(C(=O)OC)C(F)(F)C12CC(C(=O)NC(C)CCNC(c1cocn1)=O)C2 C1(NC(CC=C=C)=O)CC(CNC(C2CN(c3nnnn3C)C2)=O)C1(C)C C1(CCN(C(Cc2nc(C)oc2)=O)C)CCN(C(c2cc[n+]([O-])cc2)=O)CC1 C(c1ccc(=N)[nH]c1)=CC(=O)N(CC(=O)O)C.N1(C2(CC(=O)N)CC2)CCCC1 C1(O)(CCNC(C(CCC)N(C)C)=O)CCN(C(c2ccsc2Cl)=O)CC1 N1(C(CCC=CC)=O)CCCC(C)(NC(c2cncc(OC)c2C)=O)C1 C1(CC)CCC(C(=O)NC2(C(=O)NCCC3CC(C)(C)C3)CC(F)C2)O1 c1(CNC2CC(C(N(C)CC3(C#N)CC3)=O)C2)sccc1Cl C1(C(=O)NCC(C)=CC(=O)NC(c2cscn2)C)(OC)CCSC1 C1(C2CCCN(C(=O)COC3CC=CC3)C2)(NC(=O)Cc2cnoc2)CC1 Cc1cnc(NC2CN(C(=O)C(C)CC3CCC3)CC(C)(C)C2)nc1S(C)(=O)=O CC1CN(C(C2COCC2NC(C2C3CCC(F)(F)C23)=O)=O)CC(C)(C)C1 C1(NC(C(C(C)C)S)=O)CCOC2(CCN(C(=O)CC3CCC3)CC2)C1 c1(C(=O)N(N2CCCC2C(=O)NC2C(SCC)C2)C)coc2cc(C)c(C)cc12 c1(-c2ccc(C(N3C(C(=O)OC)CC3)=O)o2)ccc(F)cc1 C1(C(=O)Nc2cc(OC)c(F)cc2)CCC2CCC1N2C(C1CC2CC1CC2O)=O c1(OC)cnc(C(=O)NCCOC2CCN(C(=O)C=Cc3nnn(C)n3)C2)cn1 Cc1nn(CC(=O)NC(C)C(C)NC(c2ccc(F)c(O)c2)=O)cc1[N+](=O)[O-] c1(C(c2n(CCCCC)nnn2)N)cc(Cl)sc1C.c12cncn1C2.OC N1(C(=O)C=CCN2CCOCC2)CC2CCN(C(C3CCCCC3O)=O)C2C1 C1(NC(COCCCCOCC#C)=O)(CO)CN(C(C2CCCCC2)=O)C1 C(C(=O)N(C)CC1CCN(C(c2sc(C(C)(C)C)nc2C)=O)CC1)(C(C)C)OC N1(C(C2CCC(NC(CC)=O)C2)=O)CCC(C2CN(C(=O)C=CBr)C2)CC1 C1(C(N(C2CCN(C(=O)CCCCn3ccnn3)CC2)C)=O)CCCCC12CC2 c1(C(=O)NCC23CC2CN(C(c2ncc(Cl)cc2Cl)=O)C3)c[nH]c2ncccc12 N1(C(C2(CC)CC2)=O)CCC2(CCN(C(=O)CC34COC(C(=O)OC)(C3)C4)C2)C1 CC1CN(C(=O)CN2CCC2)CC1CNC(c1cccc(OC(F)(F)F)n1)=O c1(C(=O)NCCCN(C(C)C)C(C2COC(=O)N2)=O)cccnc1O CCCC(C)(CCC)C(=O)NC1CCCC(NC(=O)Cc2cc(C3CC3)no2)C1 c1(C(=O)OC)ccc(C(=O)N(C)CC2CCCN2C(C2(CC(C)C)CC2)=O)o1 N1(C(c2c(OC)cc(OC)c(Br)c2)=O)Cc2c[nH]nc2CC(C)C1 CC(C)C(C)C(CNC(C1(C2CC2)CCC1)=O)NC(=O)Cc1cc(F)ccc1F CC(CC(=O)NC1CCCN(C(c2cnc(C3CC3)s2)=O)C1)C(C)(C)C C(=O)(CCCCc1ccccc1)NC(C1CN(C(C(N2CCC(C)C2)=O)=O)C1)C C1(C(=O)NC(c2csc(C(N3CC(CO)C(O)C3)=O)c2)C)CC2C(C1)C2(C)C C(=O)(C(CC(F)F)N(C(=O)CO)CC1CCCC1)C(=O)CC1CCOCC1.C(CF)N N1(C(CCCC#CC)=O)CC2CC(C(N3CCC(O)C3(C)C)=O)C(C2)C1 N1(C(C(=O)NCCNC(C(C)C)=O)=O)CCCC([Si](C)(C)C)C1 c1(C(=O)OC)cc(Cl)c(CN2CCC(F)(F)C(C(N3CC(C)C3)=O)C2)c(Cl)c1 C(=O)(CC(F)(F)Br)NC(CNC(C(CC)c1ccccc1)=O)(C)CO c1(OC)ccc(C(N2CC(CNC(c3nncn3C)=O)C(C)C2)=O)cc1 C=C1CC(C(F)(F)F)(C(=O)NC2CC(CNC(=O)C(O)Cc3ccccn3)C2)C1 C1(CN2CCC(NC(CCOCCOCC)=O)C2)CCOC1CNC(=O)C1CC1 C(C(C)C(=O)NOCCCOC)N(C(CCOCCCOC)=O)C C1(C)(C(=O)NCC(C)(C)NC(c2cc(COC)no2)=O)CCC(C)=C(C)C1 c1(C(=O)OC(C2CC2)C2CC2)cnn2c1S(=O)(=O)CCC2.c1ccccc1 C#Cc1c[nH]nc1C(N1CCC(NC(=O)CCc2cn(C)cn2)C1)=O N1(C(C(C)Oc2ccccn2)=O)CC2CCN(C(=O)C3=CC(C)(C)C3)CC2C1 C1(C(N2CCN(CCNC(c3ccsc3Cl)=O)CC2)=O)SC2C=CC1CC2 CC(C)(C#N)CS(=O)(=O)NCc1cnc2sccn12 C(C)(CC(C)CC)N(C(C1(CNC(=O)C(C)N(CC)CCSC)CC(=C)C1)=O)C c1(C(=O)NC2C(C)N(C(=O)CC3CCC3)CCC2)nccc2c(Cl)cccc12 N1(C(C)=O)CC(NC(=O)CC2(n3cccc3)CCOCC2)C2(CC2)C1 C1(CC(=O)N(CCCCNC(c2csc(C(F)F)c2)=O)C)CCCCC1F c1(C(C)(C)C)noc(CCCC(=O)NCC2(O)CC(NC(C3(O)COC3)=O)C2)n1 C(C(C)CC(=O)NCc1noc(C2CC2)n1)NC(c1ccn(CCC)n1)=O C(CC(=O)NCCC1CCCOC1)(C(C)(C)C)NC(C(=O)NCC)=O C#Cc1ccc(C(=O)NCC(O)CN(C(=O)C#CC(C)C)C)nc1 C1(C(=O)NCCN(CC(C)O)C(=O)CNc2cccnc2)CCCCNC1=O C1(C(=O)NCC2(CC)CCOC2)C(C2CC2)CCN1C(c1ccnc(C)c1N)=O N1(C(=O)CCc2cnco2)CC2CC1CN2C(c1cccnc1O)=O N1(C(c2c(CNC(C(C)C3CCC3)=O)c[nH]n2)=O)CCCC12CCCOC2 N1(C(Cc2c(C)cccn2)=O)CCC2CCCC12C(=O)NC(C1CCOC1)C C1(C(CNC(=O)CC(=C)Br)(C)C)CCN(NC(C2C(=C)C2)=O)CC1 C(=O)(C(CC(C)C)NC(N)=O)N(CCOCCN(C(CC(=C=C)C)=O)C)C c1(C(N2C(CNC(C(CC=C)C)=O)CC2)=O)sc2nnc(S)n2c1C Cc1c(NC(=O)CC(C)CNC(C2CCCCCCC2)=O)cccc1Cl C1(CNC(C(C)OC)=O)CCC(F)(CNC(=O)C(O)Cc2ccc(F)cc2)CC1 C1(NC(c2c(C)onc2-c2ccccc2)=O)CCN(C(C2(F)CCC2)=O)CC1F CC1(C)CN(C(C(c2csc(C(F)(F)F)n2)=O)CC2(O)CCCCC2)CCC1O N1(C(C2C3(CCN(C(CC(C=C)C)=O)CC3)C2)=O)CCc2ccccc2C1 C1(NC(C2(C)CC2)=O)Cc2ccccc2N(C(=O)CSCc2cccs2)C1 c1(C(=O)NC2C3(CN(C(c4cccc(C)c4F)=O)C3)CC2)ccn2nccc2n1 Cn1ncc2c(NC3CCN(C(=O)C(c4cscn4)N(C)C)CC3)ncnc12 N1(C(=O)C=CBr)CCC2(CCCCN(C(c3cccc([N+](=O)[O-])c3Cl)=O)C2)C1 C12(CNC(CCNC(=O)CO)=O)CC(CNC(C3(CCF)CC3)=O)(CO1)C2 Cc1ncn(O)c1C(=O)NCC1CCC(CN(C(C2C3CC4C(C3)C24)=O)C2CC2)CC1 N1(C(C2(C)CC(=C)C2)=O)CC2(C1)SCCC2NC(c1ccncc1Br)=O C1(NC(c2c(C)n[nH]c2)=O)CC2CC(C1)N(C(c1cc(O)nc(C3CC3)n1)=O)C2 CCC(CC(=O)NCc1ccc(C(=O)NCCSCC(C)C)s1)SC O=S(=O)(c1cn[nH]c1)N1CCCC1CNCc1c(Cl)cccc1I C(=O)(C1CCCn2c(C)cnc21)NC(C)CNC(c1cc2ccoc2cc1F)=O c1(C(N2CCC(N(C(=O)CC3(CO)CC3)C)C2)=O)ccc(F)c(F)c1 C1(CNC(C2N(CC)CC2)=O)CN(C(=O)C(C)c2cccs2)CCN1C c1(C(=O)NC2(CNc3ccc([N+](=O)[O-])cn3)CCCC2)cccc2c1CCOC2 N1(C(CC2CCN(C3CCC(C)O3)C2)=O)CCN(CC2CC2)C(=O)C1 Cc1cc(C(=O)N(C)CC2CCCN2C(c2nnn(C(C)C)c2C)=O)c[nH]c1=N c1(C(=O)NCCN(C(C(C(C)C)C)=O)C2CC2)c[nH]c2cccnc2c1=O N1(C(CCn2ncc(C)c2)=O)CCN(C(=O)CCCN(C)C(C)C)CCC1C C1(c2cccc(NC(C(N3CCN(C)CC3)=O)=O)c2)CNC(C)(C)CO1 C(=O)(CC(C)CC(F)(F)F)N.c12ncnc(OC)c1C(=O)N(C)C1CN2C1.CO C1(NC(C(C)(F)F)=O)CC2CCC1N2C(c1ccc(Oc2ccccn2)cc1)=O Cc1cnc2c(cnn2CC(=O)NC23CCN(C(=O)C=CCO)CCC2C3)c1 C(=O)(CCCCC(N)=O)N1CCC(C)CC1C(=O)N(C)CC1(C)CC1 C(C(C)(C)CC(=O)N1CC(O)(CN(C)C(c2cc(C)cc(Br)c2)=O)C1)OC C1(CNC(CC(C)OC)=O)CCCC2(CN(C(c3nnccc3C)=O)C2)O1 c1(C(N2C3CN(C(C(CCC)(C)C)=O)CC2CC3)=O)cc2c(cc1Br)OCO2 C12(C(=O)OC(C)(C)C)CCC(C1)C(C)(NC(=O)OCCN(CC)CC)C2 C1(C(=O)NC2CN(S(CC=C)(=O)=O)CC2F)CCc2cccc(OC)c2C1 N1(C(C(C(C)C)N(CC)CC)=O)CC2(CC(CNc3ccc(F)c(C)c3)C2)C1 C1(NC(C(CC2CCC2)OC)=O)(CNC(=O)C=Cc2ccncc2)CCCCC1C C(=O)(C(CC)C(C)C)NC(CCC)CNC(C1CCCC1)=O Cc1c(C(=O)NC2CCCC(NC(C3CCC(C)O3)=O)C2)c(C(F)F)nn1C N1(C(CCCOCC)=O)CCC(CNC(c2cc(C3(C)COC3)no2)=O)C(C)C1 C(=O)(C(F)(F)C(F)F)NC(CC(C)NC(=O)CSCc1ccc(F)cc1)C C(CC(CO)NC(C1(C(C)NC(=O)Cc2ccnn2C)CC1)=O)=CC c1(C(=O)NC2CCC(CCNC(=O)CC3CC3)C2)ncc(Cl)cc1O Cc1csc(C=CC(=O)NC(C)CCCCNC(=O)CCc2nc(C)cs2)n1 S(=O)(=O)(c1cccnc1NCc1ccc(=N)[nH]c1)NC(CC)CC(C)O C(=O)(C(C)S(=O)(=O)C(C)C)N(CC(C)N(C(c1ccc(CCC)s1)=O)C)C Cc1csc(=NCC(=O)N2CC(CNC(C3CCCSS3)=O)CC2C)[nH]1 N1(C(c2c(CC)n(CC)nc2)=O)CC2CC(NC(C3CC=CCC3C)=O)C2C1 C=C=CCCC(=O)NCC(N1CCN(C(C2(C)CCC(C)C2)=O)CC1)C C(=O)(C(C)C(CC)CC)N(CCCC(=O)NCCNC(=O)OC)C C(=O)(C1CCc2nccn21)N1C(CNC(c2cccc(F)c2Cl)=O)CCC1 N1(CCC(=O)N(CC(=C)C)Cc2ccco2)CCC2(CC1)CC(O)CO2 C=CCC(C)(C)C(=O)N1CC(N(C)C(C23CCOC(C)(C2)C3)=O)C2(CC2)C1 C(C)(C)(CC(=O)NCC1CC(F)CN1C(=O)Cc1csc(NC=O)n1)SC CC1CCCC1C(=O)NCCCOCCNC(c1ccnn1C(F)F)=O C1(NC(C2C(CC)OCC2)=O)CN(C(=O)Cc2cscc2OC)CC1C(F)F C(=O)(C(F)C(C)CNC(c1cccc(OCC(F)F)n1)=O)N(CC)CC n1(C(C)C)ncc(C(N2CC(O)(C(F)C(=O)NCCOCC3CCCC3)C2)=O)n1 C1(NC(=O)NC(c2ccc(Br)cn2)COC)CCNC(C(F)(F)F)C1 C12(CNC(c3cnc[nH]3)=O)CN(C(c3ccc(Cl)cn3)=O)CC1CCO2 CCC(O)C(C)(C)C(=O)NCC(O)CN(C)C(c1c(C(C)C)n[nH]c1C)=O C(=O)(C1CCCc2ccccc21)NCC#CCNC(=O)CN1CCCC1CO C1(C(N(CCNC(C2CCC(C)S2)=O)CC)=O)CCCCCC1 N1(C(=O)Cn2cc(F)ccc2=O)CC2C3CCC(C2C1)N(C(=O)C(F)F)C3 C1(c2nc(CCC)[nH]n2)CCCN(CN2CC(C(=O)OC(C)(C)C)CC2=O)C1 C12(CNC(C3CCC(C(F)(F)F)O3)=O)CC(CNC(C3CCCO3)=O)(CO1)C2 N1(C(c2cc(C)nn2C)C(=O)NC)CCCC(C)(C)C1C(=O)OC N1(C(=O)Nc2cnn(C3CCC3)c2)CCC12CCCOC2 C1(C2CN(C(=O)Cc3cc(F)ccc3Cl)C2)(NC(C2CCC=CCC2)=O)CC1 c1(C(N2CCCC2c2ccc(C)nc2)C(=O)NCCC)ccc(OC)nc1OC C(=O)(C(C(=O)NC1CCC(NC(=O)C(N)=O)CC1)C1CC1)OC(C)(C)C N1(C(Cc2nc(C(C)C)on2)=O)CC(NCc2cncc(Br)c2)C(F)C1 c1(OC)ccccc1-c1noc(CN(C(C)CNC(c2cnc(C)s2)=O)C)n1 CCC(CC(=O)N1CC(O)(CN(C(=O)CC2(O)COC(C)(C)C2)C)C1)C(F)F c1(OC(c2c(OCCC)cc(C)cc2)=O)cc2c(nn1)CCCC2 n1(C(CC)CC)nc(C(=O)NCCC2(CNC(c3ccoc3Cl)=O)CC2)cc1C C1(CC)(CC)CC(NC(=O)C(C)(C)n2cc(Cl)cn2)CN1C(=O)C(C)SC C1(C(N2CC(CCn3cc(C(O)(C4CC4)C4CC4)nn3)C2)=O)C2CCCCCC12 C(=O)(C1CCCn2cnnc21)N1CC2OCCN(C(c3cnn(CC)n3)=O)C2C1 C1(CNC(CC2C(C)CCC2)=O)CCCN(C(C23CC(C)(CO2)C3)=O)CC1 N1(C(C2CC(C)N(C)C2)=O)CC2CC(NC(c3ccn(C)c(=O)c3)=O)C(C2)C1 c1(NCC)cccc(C(=O)NCC(N2CCN(C(=O)C(C)N(C)C)CC2)C)c1 c1(C(=O)NC23CC(CNC(C4CCC4n4cccn4)=O)(C2)C3)ncccc1CO c1(C(N(C)CC2CCN(C(C3(C)CCOC3)=O)C2)=O)ccnc2ncnn12 C1(NC(C2(C)C(C)CN(C(c3cnn[nH]3)=O)C2)=O)CC2CC1OC(=O)N2 C1(NC(=O)CCN2CCC(O)CC2)CC(O)CN(C(=O)CSC2CCS(=O)(=O)C2)C1 C1(CNC(c2c(C(C)C)occ2)=O)COCCN(C(c2ccc(F)nc2F)=O)C1 CC1CC(NC(=O)C(C)(C)C2CCCCC2)CN1C(=O)Cc1ccccc1O c1(C(=O)OC)ccc(Cl)c(CNC(C23CC2CN(Cc2ccon2)C3)=O)c1.OC CC1CC(=O)NCCN1C(=O)CN(C1CCC1)C(C1CCN1C)=O n1(C(C)C)cc(C(=O)NCC(C)(C)NC(C2CN(C)CC2C)=O)c(Br)n1 Cc1sccc1C(=O)NCCCC(=O)NCc1noc(C(N)=O)n1 N1(C(CN(C)C)=O)CCc2cc(-c3cc(F)ncc3F)ccc2C1 CP(C)(=O)C1CCCCC(Nc2cc(Cl)cc(Br)c2OC(F)F)C1 C1(CNC(CCN(C(C)=O)C)=O)CN(C(C2CC2(Cl)Cl)=O)CC2(CCC2)O1 c1(C(=O)NCC2C(NC(CN(CCC)C)=O)C2)cc2c(nc1O)C(C)(C)CCC2 c1(C(=O)NC2CCN(C(COC)=O)CC2C)ccc(C2=CCOCC2)cc1 c1(COC)nc(C(=O)N(C2CCC(NC(C3(CC(C)C)CCCC3)=O)C2)C)co1 Cc1ccc(CN=C(NCc2c(C)noc2C)NCC2CCCCO2)c(C)c1 c1(-c2cnc(C)s2)ccn2ncc(C(=O)Nc3cc(C)ccc3Br)c2c1 c1(C(N(C(C)CNC(C2COC(C)C2)=O)CC)=O)cnc(OCCOC)cn1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1CC(NC(=O)NCc2ccccc2F)C(O)C1 C(C(=O)N(C1CCCC1)C(C)=O)(C(C)(C)C)OC(CCc1cc(C(=O)OC)[nH]c1)=O c1(C(N2CC(NC(CCC=C=C)=O)C3(C2)CC3)=O)cnn2c1CC(C)CC2 c1(CC)cc(NC(C23CCN(C(c4cccc(C)c4)=O)CC2C3)=O)cnc1C N1(C(C(=O)NCCSC)C2COC2)CCC(c2ccccc2)C(O)C1 c1(C(N2CC(COC)N(C(c3ccc(Cl)[nH]3)=O)CC2)=O)cccc2c1CCO2 C1(CCCNC(C2CC2F)=O)CCN(Cc2nccs2)CC1 c1(-c2n(C(COC)C3CC3)nc(-c3cnn(CCO)c3)n2)ccc2n[nH]cc2c1Cl c1(CC(=O)NC(C2(C(=O)NC(C(COC)C)C)CC2)C)ccc(F)nc1 c1(C(N(C)CCOCCNC(c2ccc(Cl)[nH]2)=O)=O)ccc(N(C)C)cc1F Cc1cc(C(=O)NC2CCN(C(c3ccc(C4CC4)s3)=O)CC2C)c(O)nn1 N1(C(CCc2c(C)noc2)=O)CC(NC(=O)C(n2cc(Cl)cn2)C)C(C)C1 C1(C(N(CC(CN(C(CCC)Cc2ccccc2)C)O)C)=O)CC12CCCC2 c1(CCC(=O)O)ccnc(N2CCC2COC2CCCCC2)n1 C(=O)(C1CNC(=O)c2ccccc21)N1CCC2(CN(C(CSCC#N)=O)C2)CC1 C(CCC(N)=O)(C(=O)NCC1CCC1NC(=O)CCS(=O)(=O)N(C)C)NC(C)=O C1(NC(C2ON=C(C(C)C)C2)=O)CN(C(=O)C(C)(C)O)CC2(CC2)C1 CCCCC(CC(=O)N(C)CCOCC1CC1)NC(=O)C(C)(C)N=[N+]=[N-] C1(O)(CNC(=O)C=Cc2cscn2)CCN(C(C2(c3ccccc3)CC2)=O)CC1 Cc1nc(=N)[nH]cc1C(N1C2CCC1(CNC(c1cnns1)=O)CC2)=O C1(OCCOc2nccc(C(=O)OC)c2)CN(C(c2ccon2)=O)CCC1F c1(CNC(C=CCCC)=O)nc2c(s1)CN(C(c1ccncc1CC)=O)CC2 C1(C(N(C)CC2CCC2)=O)CCN(C(=O)C(O)C2CC2)CCO1 C(=O)(C1=CCC(NC(=O)Cn2ccc(C)n2)C1)N(CC(=O)OCC)C N1(C(C2(CC)CCCC2)=O)CCCOC(CNC(=O)COC2COC2)C1 N1(C(C2(C)CCC(F)(F)CC2)=O)CC2CCN(C(C3COC(=O)C3)=O)CC(C2)C1 N1(c2nnc(C)n2CC2CCOC2)CCn2cccc2C1.n1(CC)ccc(CS)n1 C1(=O)C2CCc3ccc(nc32)O1.c1(OCCCOC)ccc(F)cc1C(=O)OC N1(C(CC)=O)CCCC1C(=O)NCC(CC)NC(=O)CCSC CCC(O)(CNC1CCC(CS(C)(=O)=O)C1)C(F)(F)F CCCCCC(C(=O)N(C)CCN(C(c1cnnc(C)c1)=O)C(C)C)C(C)C Cc1ccc(CNC(C2C=CC(NC(C3C4CCCC34)=O)C2)=O)nn1 C1(NC(Cn2ccc(C)n2)=O)CCC(CNC(=O)C(c2ccc(F)cc2)O)CC1 c1(C(=O)NCC(CCNC(=O)CC2CCSC2)OC)cnc[nH]c1=N C(=O)(C(F)C(C)(F)F)NC1(C(N(CC(F)Cl)C)=O)CC(CO)C1 c1(CC(C)C)c(C(N2CC(CN(C)C(C3CC3(F)F)=O)C2)=O)cnn1C CC1(C)CCOC1C(N1CCCC1(C)CCC(=O)NCCCC(N)=O)=O N1(C(c2scc(CC)c2)C(=O)NCCSC)CCOCC1C#N CCC(O)C(F)(F)C(=O)NCC1(F)CCN(C(C2CCCNS2(=O)=O)=O)CC1 CC(C)CC(C(=O)NC(C)C(C)NC(c1cnco1)=O)N(C)C C(=O)(C(F)(F)C(C)O)NC12C(CN(C(C(C(C)C)NC(COC)=O)=O)C1)C2 C=CCC(CC)C(=O)N(C)CC1CCN(C(C2COCCO2)=O)CC1 c1(C(=O)NCC2(O)CN(C(CC3C(C)(C)C3)=O)C2)sccc1C#N CCCCCS(=O)(=O)CC(=O)NCC1CCCN(C(C2(COC)CCC2)=O)C1 N1(C(CNC(C(C)O)=O)=O)CCC(CCC=O)C1.CCCCCN(CC)CC N1(C(c2c(COC)nn[nH]2)=O)CCC(C)CC1CNC(C1CCC(OC)CC1)=O c1(CC(=O)NC2CC(CC(=O)OC)C2)ccc(F)cc1.C1(C2CCC2)C(=O)O1 C1(NC(CS(=O)(=O)NC)=O)C2CC1N(C(=O)C=CC1CCCC1)C2C C1(NC(=O)Cn2ccc(Br)n2)COCC1NC(C12CCC1C2)=O N1(C(c2c(C#N)cn[nH]2)=O)CCN(C(c2cc3ncc(Br)cc3o2)=O)C2(CCC2)C1 C1(C(=O)NC(C)C(=O)NCC2CC2(C)C)(CC)CCC1 CCCCC(CC)CC(=O)NCC1CCC(C(=O)N(C2CCN(CC)C2)C)CC1 N1(C(C2CCCN(C(Cc3n(C)ccn3)=O)C2)=O)CCC(O)C(C)(O)C1 CC(C)CC(C)(C)C(=O)NCCN(C1CCCCCC1)C(=O)C(C)c1ccco1 c1(NC(C2CC(F)CN(Cc3ccc(CO)o3)C2)=O)cc(F)ccc1[N+](=O)[O-] c1(NC(C2CC(CNC(c3ccn(CCOC)n3)=O)C2)=O)c(Br)cnn1C C1(F)(C(=O)NCCOCCCNC(=O)C=CBr)CC12CCCCC2 c1(C(N(C2CCN(C(C3CC4CC4C3)=O)C2)CC)=O)c(C(F)F)cnn1C C1(NC(C2(CC)CCCO2)=O)CC2CC1CN(C(=O)CC1CCOC1)C2 c1(C(=O)NC2CC(C)(NC(C3ON=C(CC)C3)=O)C2)cc(F)cc(S(N)(=O)=O)c1 c1(C(N)=O)cccc(OCC(=O)NCC(O)CNC(C2CC3CC3C2)=O)c1 N(C(=NCc1ccc(C)o1)NC(C1CCCO1)C)Cc1onc(COC)n1 Cc1cc(C(N2CC(CCNC(C3C4CC4C4CC34)=O)C2)=O)c(C)cn1 c1(C(=O)NC2CC(O)(CNC(C3(C)CC(=C)C3)=O)C2)ccccc1C(C)=O c1(NCc2c(C)scc2)ccc(Cl)c(P(C)(C)=O)c1 CN1CCN(c2ncccc2C(=O)NC2CC(Br)C2)CC1 C1(NC(CCCOCCC)=O)CCN(C(c2ncccc2C(F)(F)F)=O)C(C)C1 c1(-c2cnc(OC)nc2N2CCCC(CN)C2)ccc2c(c1)oc(=O)n2C Cc1c(C(=O)NC2CCC2NC(=O)CS(N)(=O)=O)cncc1F c1(OC)cc(C)cnc1C(=O)NC1(C)CC(NC(C2CCOC(=O)CC2)=O)C1 C(=O)(C1=NNC(=O)C1)NC(C)(CNC(c1coc(C2CC2)n1)=O)Cn1cccn1 C1(C(CNC(c2n(CC#C)ccc2)=O)(C)O)CCN(C(c2cscc2Cl)=O)CC1 N1(C(c2c(C)n(C3CCC3)nc2)=O)CCN(C(=O)C2=CCCCO2)CC(O)C1 C(C(C)C(C)(F)F)NC(C=CCN(C(CC=CCCCCC)=O)C(C)C)=O S(=O)(=O)(c1c(OC(F)(F)F)ccc(Br)c1F)NCC1C(C)OCC1 CC1(C)CCCN(C(=O)CCC2CCC2)C1C(N1CCC(OCCF)C1)=O c1(CN(C(CCN(CC#C)C(c2nocc2Cl)=O)=O)C)ccc(C)cc1 C1(CNC(=O)CCC2CCC2)CCC(CNC(C23CC(CO2)C3)=O)CC1 N1(C(C(=O)NCC(=C)C)C(C)C2CCOCC2)CCCCC2(CCC2)C1 Cc1ccc(NC(=O)CN2C(C(=O)O)COCC2C)cc1Cl c1(CC(N2C(C3(NC(C(C(C)C)SC)=O)CC3)CCC2)=O)cc2ccccc2o1 C12(NC(=O)C3=CCCOC3)CCN(C(=O)COc3cncc(Cl)n3)CCC1C2 C=CC1CN(C(c2csc(C3CCCCC3)c2)=O)CC1NC(=O)C#CC1CC1 C1(CC(N2CC(C(Cn3cc(COC)nn3)F)C2)=O)CC2(CCCC2)CO1 N1(C(c2ccc(O)nc2)=O)CCC2(CCC(N3CCCCCC3)CC2)CC1 N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)C(CO)N(C)C)CC1c1cn[nH]c1 C12(C(N(CCCC)C)=O)CCC(CC1)N(C(C1CC3(CCC3O)C1)=O)C2 c1(OC)cc(N)c(C(=O)NC(C)C(C)NC(c2cc(Cl)sc2Cl)=O)cc1F c1(NC(C2C(NCc3ccc(C(=O)OCC)[nH]3)C2)=O)ncc(Br)nn1 c1(C(C)C)ccc(C(=O)NC(C(N2CC(CCO)(CC3CCCC3)C2)=O)C)s1 c1(N(C2CCCCC2)C(c2nnnn2C2CC2)C)ccccc1OCC(F)F C1(C)(OC)CC2CC1CC2NC(=O)NN1CC(c2ccc(C(F)(F)F)cc2)C1 N1(C(C2C(NC(c3c(CC)nc(C)o3)=O)CC=CC2)=O)CCN2CC(O)CC2C1 C(=O)(C(C(C)(C)C)NC(C)=O)NCC(CC)(CC)NC(C(C)OCCCC)=O c1(C(=O)NC(C(=O)NC2(C#C)CCOC2)(C)CO)ncc2ccccn12 c1(CC(C(=O)N(CCCNC(=O)C(C)O)CC)C)ccc(OC(F)F)cc1 S(=O)(=O)(C1CC1)NCC(=O)NC(C1CCN(C(C2CCC2)=O)C1)(C)C CC(C)CC(C)(CNC(=O)CCc1ccsc1Cl)NC(C1CCOC1)=O N1(C(c2n(COC)ncc2)=O)CCOC(CNC(=O)C(O)C2CCC2)C1 C(=O)(C(C(C)(C)C)N(C)C)NCC(CC(=O)NC(Cn1ncc(C)c1)C)O c1(C(=O)NC(C2CCN(C(CC(=C)C)=O)C2)C)c(Cl)cccc1Cl N1(C(c2c(CC)cccn2)=O)CCC(NC(=O)Cc2cc(C)[nH]n2)C(C)C1 N1(C(c2cc(OC)no2)=O)CCN(C2CN(C(C3CCCC3(F)F)=O)C2)CC1 c1(N(C)CC2(Cn3cncn3)CC2)nc2cc[nH]c2c(=NC2CC(CCF)C2)[nH]1 C1(CC(N)=O)(NC(c2cnn3c2CCC3)=O)CCN(C(C2CC2Cl)=O)CC1 C12(C(N(C3CCN(C(=O)C(=O)NCC(F)(F)F)C3)CC)=O)CC(OC)C1C2 C(=O)(CS(=O)C(F)(F)F)NC(C1CCN(C(C(c2cn(C)nc2)O)=O)C1)(C)C N1(C(C2(CCC)CC2)=O)CC2CCC(C1)C2NC(c1c[nH]c(C(N)=O)c1)=O c1(OC)cc(N)c(C(N2CCC2CNC(=O)C(=O)N(C)C)=O)cc1Br CCC(C)(O)C(=O)NCC(C)(O)CNC(=O)CC(=O)OC(C)(C)C CCCCC(C(=O)NCC1CCCC1NC(c1cc(Cl)no1)=O)NC(N)=O Cc1nn(C)c2ncc(C(N3CCC(OC)C3)C(=O)NCc3ccccc3)cc12 C1(CNC(CCOCC#C)=O)CN(C(=O)CSc2nnnn2C)CC12CCC2 c1(C(N2CCCC(C(C)(C)O)C2)C(=O)Nc2c(C)cccc2)ncc(Br)cc1C c1(CCC)ccc(NC(C2CCCCN2C(C2CC(C(=O)OCC)C2)=O)=O)cc1 N1(C(C2C(CC)CCCC2)=O)CC2(CO)CC1(C(=O)N(C)Cc1ncco1)C2 N=c1[nH]c2cc(C(N3CC(C(N)=O)(CNC(=O)CCC4CC4(F)F)C3)=O)ccc2s1 C1(F)(CC)CCN(Cc2cccnc2O)CC1 C1(COC)(CNC(=O)CN2CCCC2C)CN(C(=O)CCc2cnn(C)c2)C1 C(=O)(C1=C(Cl)CC1)NC(CNC(=O)CCc1ccc(Cl)s1)CO c1(CNC(=O)NC(CN(CCCC)C)C)ccc2ccc(Br)nc2c1 C1(NC2(c3nnnn3C3CCCC3)CC(CC(C)C)C2)CCCCC1CCO CC1(O)COCCN(C(C2CCCCN2CC=CCc2cc(F)cc(F)c2)=O)C1 c1(CNC(C(=O)NC(c2ncc(C)o2)C)=O)cc(C)c(C)cc1O c1(CCC(=O)NCC(CNC(c2cc(C)c(C)s2)=O)(C)O)ccc(Cl)c(F)c1 N1(C(c2cncc(OC)n2)=O)CC2(C1)CN(C(C1OCCO1)=O)CCO2 S(=O)(=O)(c1cccc(CNC(=O)N(C)CC2(OC)CCSC2)c1)NCC C(C(O)CN=c1ncnc2[nH][nH]c(C)c1-2)NC(C(CCC)OCC)=O c1(C(N2CCC(C(CNC(CCCC=C)=O)(C)O)CC2)=O)ncc(Cl)c(N)c1Cl N1(CC(=O)NC2CCC(N(C(C=CCC(=O)OC)=O)C)C2)CCN(C)C(=O)C1 N1(C(=O)CCc2cnc[nH]2)CC2CC1CCN2C(C1COCCOC1)=O c1(C(=O)NC2C(C)CN(C(c3cnsn3)=O)C2)cnn2ccc(Br)cc12 N1(CC)CC(C)N(CCN2CCC(n3cnc(C(=O)OC)c3N)CC2)CC1C CCCCCC(C(=O)NC1CCCNC1=O)N1CCC(CN(C)CC)C1 C1(C(NOCC=C)=O)CCN(C(c2cnncc2O)=O)C1C(C)C CCCC(C(=O)N1CCN(C(=O)Cc2cncnc2)C(CO)C1)C(C)C c1(C(C(=O)N(CC(COC)O)C)NC(=O)C(N)=O)cccnc1 c1(OC)ccccc1C(N1CCC(C(N2CCN(CC(=O)O)CC2)=O)CC1)=O Cc1cc(Cl)cc(C)c1C(=O)NC1CCCN(C(C2CCNC2=O)=O)C1 CC(C)C(C(=O)N(C)CCn1ccnc1)NC(=O)CSc1ccc(Br)o1 C(CC(C)C(=O)NCCCCNC(C1CC(O)CN1C(C)=O)=O)OC c1(C(=O)NCC2CCCN2C(c2ccc(I)cc2)=O)ccc([N+](=O)[O-])o1 c1(OC)nc(C)ccc1C(=O)N(C(C)CNC(c1nccc(C(F)F)n1)=O)C c1(C(=O)NC(C(C)NC(=O)Cn2nnc(=O)[nH]2)CO)ccc2c(c1)OCC2 N1(C(C(CC2CN(C(=O)CN3CCOCC3)C2)F)=O)CC(C2CCCCC2)C1 C1(C(=O)N(C2COCC2(C)C)C)(CC)CCCN1C(C12CCCC1C2)=O c1(C(N(C)CC2CCN(C(C3CC3F)=O)CC2)=O)ccc2nsnc2c1 N1(C(c2cc(CCOC)on2)C(=O)NCCOCC)CCC2(C1)OCCO2 O=S1(=O)CCC(C(c2nnnn2C2CCCC2)Nc2cnc(C3CC3)cn2)CC1 Cc1ccccc1CS(=O)(=O)NC(c1c[nH]nc1C(F)(F)F)=O Cn1cccc(C(N2CCC(O)(CNC(=O)C(c3ccc(Cl)cc3)O)C2)=O)c1=O C1(CNC(CCOCCC)=O)Cc2ccccc2CN1C(=O)C(C)OCCOC c1(C(=O)NCC2CN(C(c3ncc(CC)nc3)=O)C2)ccc2scc(C)c2c1 CN1CCN(C)CC(NC(=O)CCC2(C)CN(C(=O)CC3(O)CCC3)C2)C1 N1(C(c2c(COC)noc2)=O)CC2(CCCC2N=c2ccnc(S(C)(=O)=O)[nH]2)C1 c1(C(=O)OCC)cc(C#N)n(C)n1.C12CCN(CC1)C(=O)CCc1nc(no1)C2 N1(C(C(C)SC)=O)Cc2ccnn2CC(NC(c2cc(C3(C)CC3)n[nH]2)=O)C1 c1(C(=O)NCC(C2CC2)NC(=O)CN2CC=CC2)cc([N+](=O)[O-])c[nH]1 CC(C)C(C)(CNC(c1cc[nH]c1)=O)NC(=O)C(C)n1ccnc1 CCCC(C(O)C(=O)N1CC=CC1CN(C)C)NC(c1snnc1C)=O Cc1ccnnc1C(=O)NCC1(C)CCN(C(c2ccc(F)o2)=O)C1 CCCCC(CCCC)NC(C1(C)C=CCN1C(C1OCCC1C)=O)=O CCCC(CC)CC(=O)NCC(O)CNC(=O)Cc1ccc(OCC#N)cc1 c1(C(=O)NCC(CC=C)NC(C2CSCC(=O)N2)=O)cnc(C)cc1C C1(N(C(C(C=C=C)C)=O)C)CCN(C(=O)Cc2ccc(O)cc2Cl)CC12CC2 O=C1CCC(CNC(=O)N(C2CCCC2)Cc2ccccc2Br)CN1 N1(C(C2(Oc3ccccc3)CCOC2)=O)CCC(CNC(C2(OC)CC2)=O)CC1 Cc1oc(CO)cc1C(=O)NCC(C)(O)CNC(=O)Cn1cccn1 N1(CC(=O)NC(COCC)(C)C)CC(C(F)(F)F)CCC1C(F)(F)F C#Cc1cc(F)c(C(=O)NC2(CC=C)CCN(C(C3CC(C)=NO3)=O)C2)cc1F Cc1cc(N2CCC3NCCC3C2)nc(=NCc2nc(C(F)(F)F)cs2)[nH]1 C1(F)(CNC(C(C)NS(CC)(=O)=O)=O)CCCN(C(c2cc(Cl)c(C)cn2)=O)C1 c1(C(=O)NC(C(CO)NC(C(CC)n2cncn2)=O)C)ccnc2c1cnn2C N1(C(C(CC)OCC)=O)CCC(C)C(NC(C2CC(=O)N(C3CC3)C2)=O)C1C c1(C(N2CC3N(C(c4c(Br)ccc(C)c4)=O)C3C2)=O)c(C)cc(Br)cc1F C#Cc1cnn(C)c1C(=O)NCCCCCCN(C(=O)Cc1ccnn1C)C Cc1ccc2ncccc2c1C(=O)NCCN(C)C(C1CC1(F)F)=O CCCCCC(O)C(=O)NC1C=CCN(C(c2cc(Br)cc(F)c2O)=O)C1 C(=O)(C(C)(F)C(F)(F)F)NCC(C)NC(c1c(C)[nH]c(C)c1C)=O C1(NC(c2c(C)nc(C)o2)=O)CN(C(C2(P(C)(C)=O)CC2)=O)CCC1F C#Cc1ccc(C(=O)NCCC2CC(F)(F)CN2C(c2occc2CC)=O)cc1 C(C(F)(C(=O)NCc1ccc(CO)o1)C(C)C)NC(c1[nH]cc(C)c1C)=O C(CC(C(N)=O)NC(=O)C(C1(O)CCCCC1)NC(=O)CCOC1COC1)OC CC(CCC(=O)NC(C1CCN(C(=O)CCc2nccs2)C1)C)N(C)C C12(NC(=O)NCC3C4CN(C(=O)CC5CCOC5)CC34)CCCC1C2(F)F CN1CCN(CCC(=O)NCC(C2CC2)NC(=O)Cc2nccn2C)CC1 C12(C(=O)NCC3(C)CCCC3O)CCC(NC(=O)CCS(C)(=O)=O)(CC1)C2 Cc1c(C(C)NC(c2ccnc(Br)c2F)c2nnnn2C(C)C)cccc1F C1(NC(C2(C=C)CCC2)=O)CC(NC(=O)COCC2CC2)C(O)C1 Cn1nnc(CNC(c2ccnnc2)=O)c1C(N1CCCC(CF)C1)=O c1(CC(=O)N(CC(C)CNC(c2cn(C)nc2O)=O)C)ccc2c(c1)CCOC2 n1(CC(=O)NC(C2CCN(C(c3cc(C)ns3)=O)C2)C)cccc(N)c1=O c1(C(NOC(C(=O)NC)CC)=O)cc(C#N)c[nH]1.C12CCCN1C2=O N1(C(CN2CC(C)C2)=O)CC(CNC(=O)CCOCC(F)(F)F)C2(CC2)C1 c1(C(N(C2CCCN(C(c3cnc(C)o3)=O)C2)CC)=O)nn(C)nc1Br c1(C(=O)NCC23C(CN(C(C4N(CC)CCC4)=O)C2)C3)c(C)cc(Cl)cc1C N1(C(c2nc(CC)oc2)=O)CC2CN(C(C34CCCC3C4(F)F)=O)CC(C1)O2 CCC(C(=O)OC)N(C(CO)C(C)NC(C12CC(CO1)C2)=O)CCOCCO c1(C(=O)NCCN(C(c2cnc(C(C)(C)CF)o2)=O)CC)cnn(C(C)(C)C)c1 N1(c2cc(NCCOC(CC)CC)nc(COC)n2)CCCC(C2CCC2)C1 C1(C(=O)NCC(=O)OC(C)C)CN(C(C2CCCCC2(C)C)=O)C2(CCC2)C1 N#Cc1c[nH]c(C(=O)N(C2CC2)CC2CCCN2C(c2ccc(C(N)=O)[nH]2)=O)c1 C(=O)(CCCC(CC)NC(c1cnnc(O)c1)=O)NCC(C)OCC=C N1(C(C=CC=CC)=O)CC(CNCC2CCCN2C(=O)C(C)C)C(C(F)(F)F)C1 CC1=NC(C)(CNC(c2cccc(CN3C(=O)CSC3=O)c2)=O)CS1 C12(CNC(C(COC)(C)C)=O)CCC1CCN2C(=O)CCCc1nc(C)no1 C(=O)(CCC(C)CCCC)NCc1ccc(CN(C(C(C=C)(C)CC)=O)C)cc1 C(c1ccc(Br)o1)=C(C)C(N1CCN(C(=O)C=CC(C)(C)C)CC1)=O c1(CCCCC)ccc(C(=O)Nc2ccc(CO)cc2)cc1.N12CC(C)CC1C2=O c1(C(=O)NCCC2(O)CN(C(C3(N=[N+]=[N-])CC3)=O)C2)cccc2c1CCCN2 N1(C(C2CN(C)CC2C(F)(F)F)=O)CCCC2CN(C(=O)C(F)(F)C3CC3)CC12 c1(C(N(CC(C)NC(=O)COCCCOC)CC)=O)cc2ccccc2cn1 C12(CNC(C#CC(C)C)=O)CCCC1N(C(=O)Cc1nc[nH]n1)CCC2 C1(CC)CCCC1C(N1CC(N(C)C(c2cnn(C3CCOCC3)c2)=O)C1)=O CC1=NOC(C(=O)NC(C)CCCNC(=O)C=CCO)C1 N1(C(c2ccn(CCNC(c3n(CC)ccn3)=O)c2)=O)CC(N(C)C)C(C)C1 CS(=O)(=O)c1ccc(C(=O)NCC2CCC2NC(=O)Cc2cccnc2Cl)[nH]1 C1(NC(C2(SC)CCC2)=O)CN(C(c2cn(C3CCC3O)nn2)=O)CC1SCC c1(C(=O)NCC(C2CCCCC2)NC(C2C(C)C2C)=O)cnc2nccn2c1 n1(CC)cc(C(N2CCCC(CN(C)C(C3CC3(F)F)=O)C2)=O)c(C(C)C)n1 CC1CC(NC(c2coc(C3CC3)n2)=O)CCN1C(C12CCC(C1)OC2)=O C(=O)(C#CC(C)(C)CNC(c1oc(CO)cc1C)=O)NCC(C1CCCC1)OC N1(C(C(C(C)C)SCC)=O)CCC(CNC(=O)CCc2cccnc2C)C(O)C1 C(=O)(C1Cc2ccccc21)N1CC(SC)C(NC(c2ccc3nsnc3c2)=O)C1 C(c1cnc[nH]1)=C(C)C(=O)N(C(C)CCNC(=O)Cc1csc(C(C)C)n1)C C1(C(N2CC(O)(CNC(Cn3ccc(C)n3)=O)C2)=O)CCN(C2CC2)C1=O Cc1cccnc1CC(N1CCC(CN(C(=O)CN2CC(C)(C)C2)C)C1)=O CC1(C)CC(CCNC(C23CC2CCN3C(c2n[nH]c(=N)[nH]2)=O)=O)CO1 c1(C(=O)NCC2CN(C(COC(CC)C)=O)C(C)C2)cccc(N=[N+]=[N-])c1 Cc1ccc([N+](=O)[O-])c(C(=O)NC(C)CNC(c2cc(Cl)c(Cl)cc2N)=O)c1 C1(NC(C(C=C)c2ccccc2)=O)CCCCN(C(=O)C(C)C2CC2)C1 c1(C(C(=O)NCc2cccs2)N(C(CSC)C)C)ccc(Cl)o1 C(C1=CCCN(C(C2C3CCC(=O)C23)=O)C1)NC(CC1(C)CC1)=O Cc1cnc(C(=O)OC2CCN(C(=O)OC(C)(C)C)CC2F)cc1C CN=c1[nH]c(C(=O)NCC2CC(O)CN2C(=O)CCC(F)F)cs1 C(=O)(CC(C(F)(F)F)n1ccnc1CC(=O)OC)NC1C(C)CCCCC1 c1(C(=O)NC(CC(C)C)CNC(=O)C(C)(O)C2CC2)ccc(F)c2ccsc12 c1(C(=O)NC(C)CCNC(C2CC(=O)CO2)=O)ccc(Cl)cn1 CN=c1ccc(C(N2CC3(CC3)CC2C(=O)NCCC2CC2C)=O)c[nH]1 c1(-c2cn(CCC(=O)N(C(C)(C)C(=O)O)C)nn2)cccc(OC2CCCC2)c1 C1(CC)C(NC(c2sccc2C)=O)CCCN1C(C1(F)CCOC1)=O N1(c2n(CCOCC=C)c(C3(C)CCOC3=C)nn2)CC2OC(C)(C)OC2C1 C1(NC(C(c2ccc(F)cc2)CC)=O)CN(C(=O)CCCn2cccc2)CC1O C1(c2c(C)ncs2)CCN(C(c2cccc(Br)n2)C(=O)NC2CCC2)CC1 N1(C(C(C)OCCC(C)C)=O)C(C(=O)NCC2CC(CN(C)C)C2)CCC1C C1(NC(CC(CNC(C2C(SCC)CCCC2)=O)C)=O)CCC2(CC1)N=N2 CCC(CC)C(C)C(=O)NC1CN(C(=O)CN(C)C(N)=O)CC1c1ccccc1 CC1CC(NC(=O)CC(c2cccc(F)c2)O)CN1C(c1n[nH]cc1Cl)=O C(C(C)(C)COCC1(O)CCCC1)NC(CN(C)C(=O)NC(C)(C)C)=O C(=O)(C(C(CC)CC)OC)NCC1CC(F)(CNC(c2ccc(C#C)cn2)=O)C1 c1(OC)c(CC(C2CC(NCC(O)CCO)C2)=O)cccc1F N1(CC)CCN(CCC(=O)NC(CNC(=O)C(C(C)C)OC)CO)CC1 N1(C(C(CCF)NC(Cn2c(C)ccn2)=O)=O)CCC2(C=CCO2)CC1 c1(CC(=O)NCCCCNC(=O)CC23CCCC2C3)ccc(OC(F)F)nc1 C1(C(N(C)Cc2n(CC)ccn2)=O)CC(NC(=O)C=CC2CCCC2)C12CCC2 c1(-c2cccc(C(=O)OC(C)(C)C)c2)cccc2[nH]nc(NC(N)=O)c12 c1(C(N2CC3(C(C(N4CCC(C)(C(=O)OC)C4)=O)C3)C2)=O)c(F)cc(Cl)cc1F N1(Cc2cncc(C)n2)CCC2(CC1)CC2(C)C(=O)NCC(O)CO C(=O)(C1=C(Cl)CCCC1)NCc1nccc(C(N2C(CC)CC(O)C2)=O)c1 c1(N2CCC(OCCNC(CC(C=C)c3ccccc3)=O)C2)ncnc(Cl)c1Br C1(OC)CC(C(=O)NC(C)(CNC(=O)CCn2ccccc2=O)CO)CC1OC C1(NC(c2c(C)cn(C)n2)=O)CCC(C)N(C(c2ncc(Cl)cc2O)=O)C1 Cc1[nH]nc(C(N2CCCC(CNC(=O)CCC3CCCO3)C2)=O)c1Br Cn1nc(C(=O)NCc2ncc(C(=O)NCCOC3CCOC3)cn2)cc1Cl Cc1cc(C(=O)N(C)CC2(O)CN(C(=O)C(F)(F)CC3CC3)C2)c(N)c(Cl)n1 c1(C(N2C(CNC(CC3(OC)CC3)=O)CCC2)=O)cccc(O)n1 C1(C(=O)NC(C)CC2CN(C(=O)Cc3cscn3)C2)CCn2nccc2C1 C(=O)(C(CC#CC)NC(=O)C(F)C(C)(F)F)NC1(C)CC(=C)C1 c1(C(N2CC(NC(C(CC)SC)=O)C(O)CC2)=O)ccc2cnccc2n1 Cc1cc(CN2CCOC(CC(=O)NCc3ccc(F)cc3Cl)C2)cc(C)n1 N1(C(C=CC(C)NC(C=CCCC)=O)=O)CC(C)(CO)CC1(C)C CCCCCCCC(C)NC(=O)C#CCNC(=O)CC(C)=C(C)C Cc1ccc(C(N2CCCN(C(c3ncsc3C3CC3)=O)CC2C)=O)c(N)c1C C(C(=O)C1CCCc2ccccc21)OC(N=c1ccc(C#N)c[nH]1)=O c1(C(N2CCN(C(C3C(=C)C3)=O)C(C3CC3)C2)=O)cc(C)c(F)cc1Cl C1(C(=O)O)C(O)CCCN1Cc1ccc(-c2ccc(-n3cnnc3)cc2)cc1F C1(OCC)CCC(C(=O)N(C)CC2(NC(=O)CSc3nccn3C)CC2)CC1 C1(NC(Cn2c(C)cnc2)=O)CCCN(C(=O)CCc2ccc(Cl)nc2)C1C Cc1ccc(OCCC(=O)NCC(C)NC(c2nccnc2N)=O)c(Br)c1 N1(C(C2(C)CCC(=O)NC2)=O)CC2CN(C(C3CC(=O)C3C(C)(C)C)=O)CC2C1 C(C(CNC(=O)CNC(=O)NC)C(F)(F)F)NC(c1c(CCC)n[nH]c1)=O CCCCC(O)CC(=O)N(CC(C)NC(c1cnc(OCCOC)c(Cl)c1)=O)C C1(C(=O)NCC2CCCN(C(CC(C)(C)O)=O)C2)CCC(F)(F)CO1 C#Cc1cncc(C(=O)NC(CC(=C)Cl)C(=O)N2CC(c3ncccn3)C2)c1 c1(OCC)cccnc1C(N1CCC(C2CCCN2C(C2CCCN2C)=O)C1)=O N12CC3(CCC(O3)C1=O)C2.C(=O)(C(Br)C(C)(C)C)OC(C)(C)C CCCCCCCCOCC(=O)N(C1CN(C(c2ncn(CC)n2)=O)CC1F)C CC1CC(OCc2nc(Cl)nc3[nH]ccc23)CC(C)S1(=O)=O c1(CNC(C(C)OCC=C)=O)cncc(C(=O)NC(C)(C)CN(C)C)c1 c1(OC)ncnc(N2C(C(=O)Nc3ncc(F)cc3Br)CC3CC23)c1C N1(C(c2cc(COC)nn2C)C(=O)NCCCCCC)CCC(O)C(F)(F)CC1 N1(C(CC2N(C)CCC2)=O)CCSCC1C(=O)N(CC(c1nn[nH]n1)C)C N1(C(CC=C)=O)CCC2CCN(C(=O)C=C(Cl)Cl)CC2C1 c1(CN2C(C(=O)Nc3ccc(C(=O)OC)nc3)CC(C)C2)cccc(C)c1O C1(CNC(CCc2onc(C(C)OCC)n2)=O)CC(C)CCN1C(=O)C=C(C)C c1(C(N(CCS(C)(=O)=O)C)=O)cccc(CNC(=O)CC2CCC(=O)N2)n1 c1(C(=O)NCCN(C)C(C2CCC2F)=O)ccc2c(c1)CCNC2=O N1(C(C(C)OCC=C)=O)CC(n2cc(-c3ccncc3Cl)nn2)C(C)C1 C1(C(=O)NC(COC)C(C)C)CCN(C(=O)CN2CCNC(=O)C2)CC1(C)C CCCCCC(O)C(=O)NC1CN(C(=O)Cc2sc(C3CC3)nc2C)CC1C Cn1[nH]c(=NC(=O)CONC(c2c(F)ccc(F)c2Br)=O)cc1C(N)=O CC(F)(F)CCC(=O)NCc1cc(C(=O)NCCCC(O)CO)n[nH]1 C1(NC(c2cc(C)sc2C)=O)CCN(C(=O)C=Cc2ccc(Cl)s2)CC1O Cc1cnc(C(N2CCC(NC(c3cn(C4CCC4)nn3)=O)C(O)C2)=O)c(C)c1 c1(CCC(N2CCC(C(C)NC(c3c(C)con3)=O)CC2)=O)nnc(O)nc1O C1(NC(C#C)=O)CC2(C1)CN(Cc1cc(Br)cc(I)c1)C2 CC1CCC(C(N2CCC(CN(C)Cc3ncoc3C3CC3)C2)=O)CC1 N1(C(Cc2c(C)occ2)=O)CC2CCN(C(=O)CC3(C)CCCO3)C2C1 Cc1cc(C(=O)NC(C)CCCNC(=O)C(O)CN(C)C)[nH]c1C C1(NC(CN(S(C)(=O)=O)C)=O)CCN(C(=O)COc2ccc(F)cc2)CC1(C)C C=CCC(C)(CC)C(=O)NCC1CCCN1C(=O)Cn1cccc(C)c1=O Cc1c([N+](=O)[O-])ccc(N2CC(c3cc(F)cc(F)c3)(O)C2)c1I C1(COC)C(OC)C(OC)CN1Cc1sc(C)c(C)c1Br c1(C(C)NC(c2n(CCC)nnn2)C=Cc2ccccc2)ccc(C#N)cc1 c1(OC)cccc(CC(=O)C(=O)NC2CC(CNC(c3cnc(C)[nH]3)=O)C2)c1 N1(CCCNC(c2cnc(OCC)s2)=O)CCN(C(c2nc(Cl)sc2C)=O)CC1 N1(C(CNC(C(CC)C)=O)=O)C(C(=O)NCc2[nH]c(C)nc2C)CCC12CC2 c1(CC)oc(C)cc1C(=O)NCCCN(C)C(C1(OC)CCCCC1)=O c1(C(C(=O)N(CCCOCCNC(c2cnco2)=O)C)(F)F)ccc(F)cc1F c1(NC(C2NCC(C=C)C2)=O)ccc(Cl)cc1Cl C1(C)(C(=O)NC2C(SC)CN(C(c3cc(O)cs3)=O)C2)CCCC1(F)F CC1(C)CC(=O)N(CC(N2CC(NC(=O)Cc3ccnc(O)c3)C2)=O)O1 C1(NC(c2ccc(CO)o2)c2nnnn2CCCF)CCn2nccc2C1 C(CC(=O)NCCCCCO)(C(F)F)NC(C(CC)=CC)=O C(=O)(C#CC1(C)CC1)NCC(CCCC)NC(=O)C(C)Cc1cccnc1 CC(C)C(C)CC(=O)NCC(CC1CC1)C(=O)NC1(c2nc[nH]n2)CC1 Cc1cncc(C(=O)NC(CNC(=O)C(=O)N(C)C)C(C)(C)C)n1 C1(CCn2cc(CCC(C)O)nn2)CCN(C(=O)C(c2ccnn2C)C)CC1 c1(C(N(C=O)Cc2cc(Br)c(F)cc2F)C)ccc2c(c1)OCCO2 Cc1oc(-c2ccccc2)nc1CNC(=O)C(=O)Nc1cncc(N2CCCC2)c1 N1(C(CCSC)=O)CC2(CCC(CNC(C3CC3CC(C)(C)C)=O)O2)C1 C(=O)(CCC1=NNC(=O)CC1)NC1CC(NC(c2cc(OC)no2)=O)C1 C1(N(C(CCN(CCCCC)CCC)=O)C)CCCN(C(C2CC3(CC3)C2)=O)C1 c1(SC)ccc(C(=O)NC2(C)CN(C(=O)CC3CC(C)=NO3)C2)s1 N1(C(c2noc(C)c2C)=O)CCC2(CC1)CC2C(=O)Nc1ccc(O)cc1Br c1(C(=O)NC2C(NC(C3(C#N)CC34CCC4)=O)COC2)cnc2[nH]ncc2c1 C1(c2cn(CCC3CN(C(C4(C=C)CCC4)=O)C3)nn2)CC2CCC1CC2 C1(C)(OC)CCCN(C(c2cc(Cl)c(F)c(Cl)c2)C(=O)NC2CC2)CC1 c1(C(N2CC3C(CNC(C4CCN(C(C)=O)C4)=O)(C3)C2)=O)cccc(=S)n1O C#CC1(C(N2CCN(C(=O)C(F)(F)C3CCCC3)CC2)=O)CCCC1 CC(C)(O)C(C(=O)N1CCC(c2ccco2)C1)NC(=O)CCOC1CC1 CCC(CC1CCCC1)C(=O)N(CCCCNC(C1CCCN1S(C)(=O)=O)=O)C C1(NC(CC=C)=O)CS(=O)(=O)CC1NC(c1nn(C(C)C)cc1Br)=O C=C(C)C1OCCC1CNC(=O)CC(C)(C)N(C)C(c1ccc(Cl)o1)=O Cc1nn(C)c(C)c1CCC(=O)NC1(CC(=O)N(CC2CC2)CC2CC2)CC1 C1(CNC(c2c(COC)ccs2)=O)CN(C)CCN1C(C1CCOC1C)=O c1(C(C)C)nc(Cl)cc(=NC2CC23CC(NC(=O)CC2CCCOC2)C3)[nH]1 N1(C(C)=O)CCC2(COC(CNC(c3cc(C(F)F)[nH]n3)=O)C2)C1 c1(CNC(C(C)O)=O)cn(CCNC2(CO)CC2C(F)(F)F)nn1 c1(C(N2CCCC(CC(=O)OCC)C2)=O)cnc2c(Cl)cccn12 C(C(COC)C(=O)NC(C(N1CCC(COC)C1)=O)c1ccoc1)OC c1(C(N2C(CNC(C3(F)CC=CC3)=O)CC3CC23)=O)cncc2c1CCC2 Cc1nc(CNC(=O)CCC2CC2)oc1C(=O)NCC1CC2(CCC2)C1 C1(C(=O)NCC(C)(C)C(N)=O)(CC)CCN(C(=O)C(C)Cn2cccn2)CC1 c1(N2CC(C(C)C)OCCC2)ccc(S(=O)(=O)N2CCC(C)S(=O)CC2)cc1F O(C1CCCCc2ccccc21)C(Cc1cn(C)nc1Br)=O C(=O)(C(C)(C)C(C)(F)F)NCC1CC(OC)CN1C(C1CCCS1)=O C(=O)(C1=NOC2COCC12)NC(CCCC)CNC(c1occc1C(C)C)=O c1(OC(C(=O)NC(CCN(C(C(C)=C2CCC2)=O)C)C)C)cc(Cl)cc(Cl)c1 c1(C(=O)NC2C=CC(CNC(C(C)O)=O)C2)ccc2c(c1)CC(=O)N2 C1(C(=O)Nc2cccc(O)n2)CN(C(C2CC=CCC2)=O)CC(F)(F)C1 C1(S(C)(=O)=O)(C(N2CC3CC(CNC(c4nc(C)[nH]n4)=O)C3C2)=O)CCOCC1 c1(C(=O)NC(C(C)C)CNC(=O)C(C)Cc2ccco2)cc2cccnc2[nH]1 C1(NC(C(=O)N(CCCn2ccnc2)C)=O)COCC1N1CCOCC1 C1(CNS(=O)(=O)C(Cl)(Cl)Cl)CC2(C1)CN(Cc1c(Cl)ccnc1Br)C2 N1(C(c2c(OC)cnnc2)=O)CC(C(=O)NOCC2CCC2)C(C)(C)C1 C1(CNCC(O)COC2CCCCO2)Cc2cc(F)ccc2NC1=O c1(C(=O)NC2C(NC(C34CC(CCC)(C3)C4)=O)CC2)cnccc1N(C)C C1(CC)CN(C(C2CC3(CC3)C2)=O)CC1C(=O)NCc1cn[nH]c1 c1(C(N2CC(CNC(=O)CC3NC(=O)NC3=O)OCC2)=O)cc(Cl)nnc1O N1(C(=O)NCCc2cc(OC)cc(OC)c2)CC(C)OC(C)(C(F)F)C1 c1(C(N2C(CNC(c3nccc(N(C)C)c3)=O)CCC2)=O)cc(Cl)cc(Br)c1 C(=O)(C(C)CN(C)C)N(CCCNC(CC=C(C)C)=O)CCO c1(CN2CC(NC(Cc3cccc(OC)c3)=O)C(O)C2)ccccc1C#N Cc1n[nH]c(C)c1CNC(=O)CNCCNC(=O)C(C)(C)C CCCC(C(=O)NCc1c(C(=O)NCCn2cnnc2O)c[nH]n1)OC N1(C(C(C)SCC)=O)CC(C(=O)NC2CC=C(C)CC2)C(C)(C)C1 N1(C(C(CC(C)C)NC(c2ncc(C)nc2)=O)=O)CCC2(CCOC2)C1 c1(CCC(=O)O)ccc2c(c1)CCN(C(c1cc3n(n1)CCCNC3=O)=O)C2 c1(NC(=O)CC2CCCN2Cc2cc3ccncc3[nH]2)cccc(S(=O)(=O)O)c1 C1(N(C(=O)C(F)(F)F)C)CN(C(C2C3CC2C(C)N3)=O)CCC1c1ccccc1 C1(C(=O)NC2CCC(CCNC(CNS(CC)(=O)=O)=O)C2)CCCCN1C(C)=O c1(SC)cc(C(N2CC(CNC(c3n[nH]cc3C)=O)C3CC23)=O)oc1C C#CC1(C(=O)NCCCc2cccnc2)CN(C(=O)CC2(C)CCCC2)C1 c1(-c2cn(NC(=O)CN3CCOC3=O)nn2)cc(Cl)ccc1F.C12(CC1)CC2.c1(S)ccccc1 N1(C(C2(CCOC)CCC2)=O)CCC(NC(C2CCS(=O)CC2)=O)C(F)C1 Cc1nn(C)cc1C(=O)NC1(CNC(C23CC2C3)=O)CC1 c1(C(=O)NCCNC(C(C)C)=O)ccc(-c2cc(C(F)(F)F)ccn2)cc1 c1(C(=O)NCC2OCCC(NC(C(C(C)O)N(C)C)=O)C2)cccc2[nH]ncc12 N1(C(c2n(C)cc(C)n2)=O)CC2CC1CC2N1CCC12CCCC2 n1(CC)cnc2c(NC3CCC(SC)C3)[nH]c(=NC3CCCn4ncnc43)nc12 C#Cc1ccc(CC(N2CC(C(N3CC(N(C)C)C3)=O)C(COC)C2)=O)cc1 C1(C(=O)NC2C(NC(=O)Cc3cccnc3Cl)CCCC2)CC2(C1)CC(O)C2 N1(C(c2cccc(O)n2)=O)CCC2CN(C(=O)CC3CCCC3O)C2C1 N1(C(c2c(C)c[nH]n2)=O)CC(CNC(C2CCN(C)C2=O)=O)OC(C)(C)C1 N1(C(C=C(CC)C)=O)CC(C2CCCN(C(=O)C(CN(C)C)N(C)C)C2)C1 Cc1cc(N)cc(C(N2CCCCC2CCNC(=O)C2=CCS(=O)(=O)C2)=O)c1F C(=O)(CCCC(=O)N1CC(N(C)C(c2cc[n+]([O-])cc2)=O)C2(CC2)C1)NCCC CS(=O)(=O)C1CN(C(=O)C(N)Cc2ccco2)C2(CCOCC2)C1 c1(C(C)C)nc(NCC2(CF)CC(F)(F)C2)cc(=NC2CCn3nnnc3C2)[nH]1 c1(C(=O)NC(CN(C(C(C)OCC#C)=O)C)C)noc(-c2ccccc2)c1C C1(SC)CN(C(C2CC(C)CCO2)=O)CC1NC(=O)CN(C1CCS(=O)(=O)C1)C C#CCC(CC(=O)NCCc1cc(C)[nH]n1)NC(=O)C(C)C(C)C N1(C(C2CC(C)(C)C2)=O)CCC2CN(C(c3cc4c(s3)CCCC4)=O)CC2CC1 Cc1ccc(CN(C(c2cc(C#N)ccn2)C(=O)NC2CCCC2)C)cc1Cl C(=O)(C(C)(C)CC1CCCCC1)NC(C(C)NC(CN(C1CC1)CC)=O)CO C1(N(C(c2c(CC)occ2)=O)C)CCN(C(=O)CSc2ccccc2)CC1C c1(C(CNC(C(c2cccnc2)NCCCC)=O)NC)ccccc1 CC(C(=O)NCCC1CCCCN1C(C1CCC(O)C1)=O)C(F)F C1(N(C(C=CC(N)=O)=O)CC2CC2)CCN(C(c2snc(Cl)c2Cl)=O)CC1 c1(NCCCOCCNC(c2cc(CC)nn2C)=O)ncnc2cccc(F)c12 CC(C)CC(C(N)=O)N(C)C(C1CN(C(C2(C)CCCC2O)=O)CC12CC2)=O CC1CCCC1C(=O)NCC(C)(C1CC1)NC(c1nncn1C1CC1)=O CS(=O)(=O)c1ccccc1C(=O)NC1CCC(NC(c2cnns2)=O)CC1 n1(CC)cc(C(=O)NC2CC(CCNC(c3cc(C(C)(C)C)n[nH]3)=O)C2)c(C)n1 C(=O)(C1=CCCOCC1)N1CC(CNC(C2(F)CCOC2)=O)CC(C)C1 C(=O)(CC(C)CC(=O)NCCCNC(c1nc(Cl)c(Cl)s1)=O)OC c1(C(=O)NC(C2CCCCC2)CNC(C2(CSC)CCC2)=O)ccsc1Cl C1(OCC)CCCC1ONC(C1CCC(C2CCC2)O1)=O C1(C(=O)NCCN(C(C)C)CC)CCN(C(=O)C=Cc2ccccc2)CCO1 C1(C)(C(N2CCCC(CC)C2)=O)CCN(OC(C=C2CCOC2C(=C)C)=O)CC1 N1(C(C(CC=C)CC=C)=O)CCCC2(CCC2NC(C2CC3C=CC2CC3)=O)C1 C(C(C)(O)CC(=O)N1CCC(C=CC(=O)NCCCCC(N)=O)CC1)OC CC1(C)CC(C(N2CC(CNC(C3CC(O)C3)=O)C3(CC3)C2)=O)C(C)(C)O1 N1(C(CC(CC)C2CCC2)=O)CCOC(C)C1C(=O)NCC1(C(C)(C)OC)CC1 c1(CN(C(=O)CC2(NC(c3cocn3)=O)CCCCC2)C)cnn(C)c1O c1(OC)ccc(C=CC(=O)NCCC(C)CCNC(=O)CCCC(C)C)cc1O C=CCC(C)C(=O)NC1(CCNC(=O)C(F)(F)C2(OC)CCC2)CC1 Cc1ccc2[nH]c(C(N3CCC4CC4(NC(=O)C(Cl)=CCl)CC3)=O)cc2c1C n1(C(=O)OC)ccc2nc(Cl)nc(N(C)Cc3cccnc3C(F)(F)F)c12 C(=O)(C(O)CCCNC(C12C=CC(CC1)C2)=O)NCCCCCCN(C)C C=C(C)CCC(=O)NCC1(COC)CN(C(=O)C(CC=C)NC(C)=O)C1 N1(C(C(=O)NC)=O)CCC2CN(C(=O)C(C(C)C)N3CCCS3(=O)=O)CC12 C1(NCC(C)(C)CC2CN(C(=O)Cn3cc(CO)nn3)C2)CCCC1C1CC1 c1(C(N2CC3(CN(C(CCC)=O)C3)C2)=O)cnc2[nH]c(C(F)(F)F)nc2c1 c1(C(N2CCCCC(CNC(C3CC3F)=O)C2)=O)cc2ccnn2cn1 N#Cc1ccc(CNC2CCOC(c3cccnc3)C2)c2ccccc12 CC1(C)CC(NC(C2(C)CNC(=O)C2)=O)CN(C(c2cc3c(s2)CCC3)=O)C1 C(=O)(CCS(C)(=O)=O)NC(C(C)(C)NC(Cc1ccc(C(=O)OC)cc1)=O)C c1(C(N2CC(CCNC(c3c(OC)ncc(F)c3)=O)C2)=O)ccc2occc2n1 c1(-c2cncc(C)c2)cnn2cc(C(=O)NC(c3ccc(Br)cn3)C)cnc12 C=C(C)CCC(=O)N1CC(CNC(=O)CC2CCOC(C(C)C)C2)C(C)C1 c1(NCC(C)OCC=C)ccc2c(S(N)(=O)=O)cccc2c1 C=CCC(CC=C)C(=O)N1CC(C2CC2)OC(C)C1 C1(C(N(CCCN(C(=O)CNC=O)C)C)=O)CC2(CC2)CO1 C12(C(N(CCN(C(=O)CC3C=CCC3)C(C)C)C)=O)CCC(C)(C1)OC2 C(c1cn(CCC#N)c2ccccc12)=CC(N1CCCCC1C1(NCCCl)CC1)=O c1(CNC(N2CC3CCC3(C(F)(F)F)C2)=O)cc(F)cc(F)c1 C12(CNC(c3c(C)nn(C)c3F)=O)CCCC1N(C(=O)C1=NOCC1)CCC2 N1(C(Cc2cc(C)on2)=O)CC(CNC(=O)C(C)N(C)C)CC1C C1(C(N2CC(NC(C(=O)NCC)=O)(CO)C2)=O)CCC2(CCC2)CO1 c1(C(=O)NC2CN(C(=O)C(F)CC3CC3)CC23CC3)ccc2nc(O)[nH]c2c1 CCCCCC(C)(C)C(=O)N1CCCC(CCNC(C2CCCCCCC2)=O)C1 c1(C(N(CC(=O)NC(CC)COC)C2CCC2)=O)ccc(C)cc1C N1(C(C2CCCC23CCC3)=O)CCCC2CCNCC12 N1(C(C(=Cc2ccco2)C)=O)CCC2CC2(NC(=O)C=Cc2csc(C)n2)CC1 C1(NC(CC(C)SC)=O)CC12CCC(NC(=O)CNS(=O)(=O)N(C)C)CC2 CCCS(=O)(=O)CC(=O)NCCC1CCC(NC(=O)CSc2ccccc2F)C1 C1(C(=O)NCC(COC)O)CC=CCN1C(=O)CC1(OC)CCC1 N1(CC(N2CCCC(NC(c3cccc(Cl)c3)=O)C2)=O)CCc2ccccc21 C1(NC(C2CCCS2)=O)CC12CCN(C(=O)CCC1CC1(F)F)C2 C1(NC(C(CSC)(C)NC(c2ccsc2C)=O)=O)CCCOC12CCC2 C(=O)(CC(C(F)F)NC(c1cc(O)ccc1F)=O)NCC(C(C)(C)C)O C1(NC(CSCCC)=O)CCCCN(C(C2CCC2C(C)(C)C)=O)C1 c1(-n2c(-c3sccc3F)nc(C(C3CC3)OCC)n2)cc(F)cc(F)c1 c1(CNC(c2cc(O)ccc2Cl)=O)nc(CNC(C2CCCCS2)=O)cc(O)n1 C1(CNC(C=C2CCC(C)C2)=O)CN(C(=O)Cc2cnnn2C)CC2(CCC2)O1 C1(F)(CNC(=O)CCc2cccnc2)CCC(NC(=O)CCc2cnc[nH]2)C1 CC1(F)COCCN(C(c2coc3c2CN(C(=O)CC2CC4CCC2C4)C3)=O)C1 N1(C(c2c(CC)n[nH]c2)=O)CC(C(=O)NC2(C)CCCOC2)C2(CCC2)C1 CCCC(C(=O)NC(CNC(=O)Cc1csc2ccccc12)CCOC)C(C)C CN1CCCC(C(N2CCN(C3CN(C(=O)CSc4cn[nH]c4)C3)CC2)=O)C1 C1(C)(CS(N2C(C(=O)OC)CC2CO)(=O)=O)CCCCC1(F)F CN1CCC2OCCN(Cc3nc(-c4cnn(C)c4)nn3C3CC3)C2C1 C(=O)(C1=CCCC(C)(C)C1)NC1CN(C(c2n(C)nc([N+](=O)[O-])c2)=O)CC1(C)C S(=O)(=O)(c1ccc(F)c(Br)c1)N1C(C)(C(=O)Nc2cc(I)cnc2Cl)CC1 C1(N(C(C(C)NS(C)(=O)=O)=O)C)CCN(C(c2sccc2C(=O)OC(C)(C)C)=O)C1 N1(c2cc(C)nc(C(F)(F)F)n2)CCn2ncc(CNC(=O)C(C)O)c2C1 C1(NC(=O)C2=C(Cl)CCC2)CCCC12CN(C(=O)C=Cc1cnc(O)nc1O)C2 c1(CC)nc(C)c(C(=O)NC2C=CC(CNC(=O)CCP(C)(C)=O)C2)c(C)n1 C=C(C)c1ccccc1NC(=O)C(C1CCCN(C(C2CC=CCC2C)=O)C1)C C1(C(N2CCC(OCC(N)=O)C2)C(=O)NCCC#N)CC2CCC1CC2 N1(C(C2(CC=C)COC2)=O)CC(NC(C2CCCOC2)=O)CC2(CC2)C1 CN1CCC(C(=O)NC2C=CC(CNC(=O)CCCn3ccccc3=O)C2)CC1 c1(OC)cc(C(=O)NC2C(N(C)C)CN(C(C3(OC)CC3)=O)C2)ccn1 c1(N2CCCC(OC)C2)nc2ccc(Cl)cc2c(=NCC2CN(C)CCO2)[nH]1 C1(C(N(C(CC)CC)CCO)=O)CC2(CC(NC(C3CC4CCC3CC4)=O)C2)C1 N1(C(CCC#CC)=O)CCCC(O)(CNC(=O)C=Cc2cnc(C)s2)C1 C1(CNC(c2c(C)cc(C)o2)=O)CCN(C(=O)Cc2nc[nH]n2)C12CCC2 Cc1n[nH]c(C)c1CCN(C)C(C1C2CN(CC(=O)NCc3ccco3)CC12)=O CCC(CC)(CCNC(c1ncccc1N)=O)NC(=O)CC1CCCCC1(F)F C(CN=c1[nH]nc(O)s1)N1CCN(C(C2N(N=O)CCC2)=O)CC1 CCCCCC(C)(C)C(=O)N1CCCC1CN1CCC(=O)NC(C2CC2)C1=O c1(CC(=O)N(C(CNC(C2C(C)(COC)C2)=O)C2CC2)C)cc(C(F)(F)F)n[nH]1 C1(C(=O)OC)CCN(C(c2cncc(OC(C)C)c2)=O)C12CCSCC2 CCCC(C(=O)N1CCC(NC(=O)CNS(C)(=O)=O)C1)NC(N)=O C1(C(=O)NC(CC(C)NC(c2c(CC)nc[nH]2)=O)C)CCc2ncncc2C1 C1(NC(CC(CC)(F)F)=O)CC2CC(C1)N(C(=O)Cc1ncoc1C)C2 C1(NC(=O)COCC2CCOC2)CCN(C(c2cc(CO)on2)=O)CC1F c1(C(=O)NC(C(=O)NCCCc2n(C)ncn2)=O)cccc(-c2ccncc2)c1 Cn1nc(CNC(C2(Cl)CC2(C)C)=O)c2c1CCN(C(=O)C1=NNC(=O)C1)C2 CCCCC(CNC(=O)CCc1ccc(C2CC2)o1)NC(c1ocnc1C1CC1)=O N(C1CCc2cccnc21)C(C1CC(C)(C)N(C(=O)C(=O)C2CCCC2)CC1)=O C(=O)(C(C(C)(C)C)N1CCNC1=O)N1C2C(NC(C(CC#C)C)=O)C(C2)C1 c1(NC(CC(CNC(C(CCC)CC)=O)C2CCC2)=O)ccc2ncnn2c1 C(C(C(=O)NCC(Cl)Cl)NC(C1CC(C)(C)C1)=O)OCC S(=O)(=O)(c1ccc(Cl)c(NC(NC2CCn3ccnc32)=O)c1)NC(C)(C)C c1(NC(N2CCC(C(=O)OCC(N)=O)C2)=O)cc(Br)sc1C(=O)OC c1(C(N2CCC3(NC(c4cc(SC)oc4C)=O)C(C2)C3)=O)nc(C)c(C)[nH]c1=O C1(CC(=O)NC2CC(C(C)O)C2)CCCN1C(=O)CC1CC(F)(F)C1 N1(C(C(C(CC)C)C)=O)CC2(C1)C(NC(c1ccco1)=O)CCS2(=O)=O C=CC1(CC(=O)NCCC(O)CCC)CN(C(c2cnn(C)c2Cl)=O)C1 N1(C(=O)CC2CCC2)CC2OCCN(C(C3CCN(NC(CC)=O)C3=O)=O)C2C1 C(c1ccc(Cl)cc1)=CC(=O)NC(C1(CNC(C(CC)OC)=O)CC1)C Cc1cccc(C(=O)NC2CCCC2NC(=O)CC2COC(C)(C)C2)c1 C1(CC(=O)NCC2(CN(C)C)CC2)N(C(C2CC3CCC2CC3)=O)CCC1(C)C c1(C(N(CCN(C(C2CC2(C)C)=O)CC)CC)=O)cnc(Br)c(O)c1 c1(C(=O)NCC2C(NC(C=CC)=O)C2)cc(=O)c2ccccc2[nH]1 c1(CC(=O)NCCCCc2cn(CCCCCC)nn2)cn(CC)nc1C N1(C(C(CCC)OC)=O)C(C)CC2CN(C(c3cccc4oc(=N)[nH]c34)=O)CC12 CC(CCN(C)C)C(=O)N(c1ccccc1)C(c1cccnn1)=O C1(C(=O)NCC2(C(=O)NC(C#C)C3CCC3)CCC2)CNC(=O)CC1C C12(CNC(c3cc(C)nn3C)=O)CCCCC1CN(C(c1cc(CF)on1)=O)C2 n1(CC(=O)NC2CC(CNC(C)=O)CC2O)cc(C(F)(F)F)cc(Br)c1=O n1(CCC)nc(C)cc1C(=O)NCC1(O)CN(C(=O)C(C)Cc2ccco2)C1 N1(C(c2c(CC)scc2)=O)CC(NC(C2(CF)CC(F)(F)C2)=O)C(C2CC2)C1 Cc1ccc(C(=O)N(CC(C)(C)NC(=O)Cc2ccnn2C)C)c(Cl)c1C c1(N2C3CCC(NC(Cc4cc(C)[nH]n4)=O)C(C3)C2)ncnc2ccc(Cl)cc12 C(=O)(CC(F)(F)Cl)N(CCN(C(C(c1ccc(CC)s1)=O)=O)C)C(C)C c1(CCC)cnnc(C(=O)N(C2CN(C(c3sccc3C(C)C)=O)CC2F)C)c1 C1(C(N2CCC(NC(C3CN(CC(C)C)C3)=O)C2)=O)C(F)(F)C12CCC2 N1(C(c2c(CC)scn2)=O)CCCC(CN(C(=O)C(C)(C)c2ccno2)C)C1 c1(CN2CC3C(C(=O)NCc4cc(C)oc4C)(C3)C2)cc(Cl)nc(Cl)c1 N1(C(C(C(CC)CC)OC)=O)CCCC2(CCCN2C(=O)CC2CC3(CC3)C2)C1 C1(NC(c2c(COC)cco2)=O)CCN(C(=O)CS(=O)(=O)NC2CC2)CCC1CO N1(C(C(n2c(C)cc(C)n2)C)=O)CCC(C)(CNC(C23COCC2C3)=O)CC1 N1(C(=O)OC(C)(C)C)CCC(C2CCC2)(C(=O)N=c2cc(C(=O)NC3CC3)[nH][nH]2)C1 C1(C(=O)NCCC(C)NC(=O)C(F)(F)Sc2cnn(C)c2)CC2(C1)CC2F N1(C(c2ccc(CCC)[nH]2)=O)CCC2CC(C1)CN(C(=O)CC(C)CN(C)C)C2 N1(C(C2C(C=C)CC2)=O)CCCOC(CNC(c2nocc2CC)=O)C1 c1(CC)ccc(Br)cc1C(=O)NCC(CNC(c1cc(C)ns1)=O)OC CCCC(C(=O)N(CC(C)NC(=O)CC(c1ccccc1OC)C)C)N(C)C N(S(=O)(=O)N(C)c1ccc(C)cc1)C1CC(CC)C1 N1(C(CS(CC)(=O)=O)=O)CCOC2CCN(C(C3CCC4CC34)=O)CC12 C=C1CC(C(=O)NCCn2nnc(C(C)C)n2)(CNC(=O)C(OCC)OC)C1 N1(C(C(CCSC)OC)=O)CC2(NC(=O)C(=Cc3ccco3)C)CCCC2(F)C1 c1(C(=O)NC2CC(C(N3CC(C#N)OCC3)=O)C2)c(Br)cc(Br)c(O)c1Br N1(C(CSc2cccc(C)c2)=O)CCN(C(c2ccncc2Cl)=O)C(CC2CC2)C1 N1(C(=O)CC2CCCO2)CCCC2(CCN(C(C34CC5CC3C4C5)=O)C2)C1 S(=O)(=O)(CC(F)(F)F)N1C(C(=O)Nc2c(C)cncn2)CCCC1 C1(NC(CCOC(C)C)=O)CC2CC1N(C(=O)CCc1cscc1Br)C2 C1(NC(C(CC#C)C2CC2)=O)CN(C(c2ccnc(CO)c2)=O)CCC12CCC2 CC(CF)CC(=O)NC1CC(NC(C2(OCc3ccccc3)CC2)=O)C1 c1(OC)cc(C(=O)NCC(C2CC2)N(C)C(c2ccco2)=O)c(C)cc1O CN1CC2(CCN(C(C34CC3CN(C(c3cccc5cncn35)=O)C4)=O)CC2)C1 c1(CC)cc(C(=O)NCCc2ocnc2CNC(=O)Cc2nc(C)cs2)ncn1 C(=O)(CCC(O)C(C)(C)C)N1CC(OC)C(NC(=O)C(C)Cc2cnco2)CC1 CCC(F)(F)CC(=O)NCC1CN(C(c2cccc(CO)c2)=O)CC1(C)C c1(CCC(=O)N(CC(CNC(COCC(=C)C)=O)(C)C)C)c(Cl)cncc1Cl c1(OCC(=O)NCC2(NC(=O)CCc3cnn[nH]3)CCOC2)cc(F)cc(Cl)c1 Cc1cc(C)c(C(=O)NCC2CCCN2C(C23CCN(CC2)CC3)=O)c(C)n1 C=CCC(CNC(C1CCC(=O)N(C)C1)=O)C(=O)Nc1ccc(SC)cc1 N1(C(c2cn(CCO)nn2)=O)CC2COCC2(C(N2CC3CC3C3CC23)=O)C1 c1(NC(C(CCC)OC)=O)cc(Cl)c(NC(N2CCC2C)=O)c(Cl)c1 CC1=C(C(=O)NC2(C)CC(NC(=O)C(c3c(F)cccc3F)(C)N(C)C)C2)CCO1 c1(C(N2CC(N(C(C(C)C3CC3)=O)C)C(O)C2)=O)cc2cccnc2cn1 N1(C(C(C(CC)O)C)=O)CC(C2CCCN(C(=O)CCc3ccsc3)C2)C1 N1(C(C2CN(C)C2)=O)CC(CNC(C2(CC3CC3)CCCO2)=O)C2(CCC2)C1 CCCC(CNC(=O)C(CNC(=O)C=CC1CCC1)CCC)CCO C(=O)(CC(C)C(C)(C)NC(c1nc(C)ccc1F)=O)NCCCCCC#C c1(C(N2CCOCC(NC(C(C)NC(C)=O)=O)C2)=O)cnc(O)n(C)c1=O C(CN=C(NC1CC1)N1CCCC(n2ccnn2)C1)c1cccc(Cl)c1 C1(C(=O)NC(CC(=O)OC)C)CCCCCN1C(=O)C(=O)N(C)C n1(CC(=O)NCC(N(C(CCS(=O)(=O)NC)=O)C)C2CC2)c(C)cc(C)nc1=O C(=O)(C1CCc2ccccc21)NC1CCCCN(C(c2c(C)nncc2)=O)CC1 N1(C(CCSCC(C)C)=O)CC(NC(C2(C)CC2c2ccccc2)=O)C(C)C1 C1(CN(C(C(=O)NCC)=O)C)CCCN(C(C2CC(SC)C2)=O)C1 CC1(CNC(C2(C)CCCN2C(=O)CC2CC=CC2)=O)COCCO1 C(C(C(=O)N1CCC(COC)C1)OC)NC(C(OCC)OC)=O c1(C(N2CCN(C(C(C=C)O)=O)C(C)C2)=O)c(OC)cc(OC)c(Cl)c1N c1(C(=O)NCC2CN(C(C3CC(CF)C3)=O)CCO2)cccc(C#CC2CC2)c1 CC1(C)CN(C(c2ocnc2C(F)F)=O)CC1NC(=O)CC1CCC(=O)NC1=O N1(C(C(Cc2ccccc2Br)NC(CC(C(C)C)O)=O)=O)CC(O)(C2CCC2)C1 N1(C(c2ncc(C)nc2)=O)CCC(NC(c2nccnc2Cl)=O)C(F)C1 C(CNC(c1ccccn1)=O)(C(C)(C)C)NC(C(C)(C)NC(=O)NCC=C)=O C1(CNC(CCc2cn(C)nc2)=O)CC(F)CN1C(=O)CO N1(C(C2C(C)(CC)C2)=O)CCCC(CO)(NC(=O)CC2(O)CCCN(C)C2)C1 c1(CC2CN(C(CCc3c(OC)ccc(F)c3)=O)C2)cc2c(F)cccn2n1 c1(C(=O)NC(CC)CNC(=O)Cc2cocn2)ccc2n[nH]cc2n1 C1(CNC(COCCOC)=O)CN(C(=O)CCC)CC1C c1(OC(C(=O)N(CC(C)NC(C(CCC)C)=O)C)C)ccc(C#N)cc1 C1(NCC(=O)ON)Cc2ccccc2C1NC(N1CC2CC1C(=O)N2)=O N1(C(C(Cc2ccsc2)NC=O)=O)CCOCC(CNc2ncc(Cl)cn2)C1 CC1=NN(C)C(=O)C1CC(=O)NCC1(CNC(c2cccc(O)c2Cl)=O)CCC1 C(C(C)(C)CC(C)O)NC(C1(NC(CCN(CCC)C)=O)CSC1)=O c1(C(=O)OC)nc(N2CC3CC3(CNCC3(c4ccccc4)CC3)C2)ncc1F N(C1CCc2cc(Br)ccc21)C(CSc1n(CCOC)c(-c2cccs2)nn1)=O N1(C(C=Cc2occ(C(=O)OC)c2)=O)CCC2C(CCN2C(=O)CC(C)CF)C1 CC1CCCC1(C(=O)NC1CC(CC2CC2)C1)NC(c1cc(C(F)F)on1)=O c1(OC)ccnc(CC(=O)NC2(CCCNC(c3n[nH]cc3OC)=O)CC2)n1 C1(C(=O)NC2(CO)CCCN(C(CC3(OC)CC3)=O)C2)CCCC12CCOCC2 c1(C(=O)NCC23CC(CNC(CC(C=C)(C)C)=O)(OC2)C3)ccc(F)c(O)c1F C1(C(N2CC(CCNC(C(C)(C3CC3)OC)=O)C2)=O)CNC(=O)CC12CCC2 N1(C(C(CC)N(CC)CC)=O)CCC(C2CC2)(CNC(C2(OC)CC2)=O)C1 C12(C(=O)NC(C3(OCc4ccccc4)CCOCC3)C)OCCCC1C2(F)F N1(C(c2cc(-c3ccccc3Cl)no2)=O)CC2C(CNC(C3(CF)CC3)=O)C2C1 c1(N(CC(COC)(F)F)C)nc(N2CC(=O)N3CCCC3C2)c2sccc2n1 CC(C)C(CN1CC(=O)N(Cc2ccccc2-c2ncc(C=O)s2)C1=O)C(C)C c1(C(=O)OC)cnn(CC(=O)OCc2ccnn2CC(F)F)c1 N1(C(COCC=C)=O)CCC(C)C(N(C)C(c2cc(C(=O)OC)no2)=O)C1 c1(N(CCN=c2cncc[nH]2)C)cc(Br)ccc1S(=O)(=O)NC1C2CCCOC12 c1(C(N2CCC(O)(C(C)NC(c3ccoc3C3CC3)=O)C2)=O)cc(F)cc(F)c1 c1(CC)cc2c(CC(=O)NC3CCC(NC(=O)C(C)C(F)F)C3)csc2s1 N1(S(C)(=O)=O)CCCCC1C(=O)NC1C=CCN(C(C2(O)CCC2)=O)C1 N1(C(C(C(C)C)N(CC)CC)=O)CCCC(NC(=O)CC2CC3(CC3)C2)C1C C1(c2cn(C)nc2)CC1N=c1[nH]c(=NC2CCSCC2)[nH]c2ncn(C)c12 C1(c2n(C(CC)(C)C)nnn2)(NC2CCN(CCF)C2=O)COC2(CCC2)C1 C1(CC(=O)N(C2CCN(C(=O)Cc3cc[nH]c3)C2)CC)C(=O)N(C)N=C1C c1(NC(C2C3CN(C(CC(=O)OCC)=O)C2C3)=O)ccc([N+](=O)[O-])cn1 C1(NC(CCCCCC#C)=O)CCN(C(C2CC23CCOCC3)=O)CC12CCC2 O=C(CCC(F)F)NN1CCCC1C(=O)NC1CCC(O)CC1 C1(C(=O)NCC2CCC(NC(=O)COC3CCOC3)C2)CC12CCS(=O)(=O)CC2 C(C(C)C(F)C(=O)NCCN1CCCNC1=O)NC(c1ccc(C#C)o1)=O C(CCCCC(=O)N1CCC(C(C)(C)NC(c2csc(C#N)c2)=O)C1)=CC C1(C(=O)NC2C(CNC(=O)Cc3cnns3)C2)CCCCO1 C(=O)(C1=CCCCC1C)NC(C(C)C)CCNC(c1nc(C2CC2)cs1)=O CC1=C(C(=O)NCC2(C(C)(C)O)CN(C(=O)CC3CCCN(C)C3)C2)COCC1 n1(C(c2c(C)cccc2)c2nc(-c3cscn3)nn2C)c(=O)oc2ccccc12 C12(C(N(C(C)CNC(=O)CCNS(C)(=O)=O)C)=O)CC(CO)(C1)C2 C12(C(=O)NC3(C)CCCN(C(C4(C)CCCCO4)=O)C3)CC3CC(C(=O)N1)C2C3 C(=O)(C1=NOC(C)C1)NC1(C)CN(C(c2n(CC)ccn2)=O)C1 C1(F)(CNC(CCSC)=O)CCC(CNC(=O)CC2CCCC(O)C2)CC1 Cc1cc([N+](=O)[O-])cc(C(=O)NCCC(O)CNC(=O)Cc2ccoc2C)c1Cl N1(CC(=O)NC(c2cn(CCCC(=O)NCC(F)(F)F)nn2)C)CCOCC1C C(=O)(C(O)C(F)F)Nc1ccc(Cl)cc1.c12ccccc1CN1CC(C1)NC2=O c1(NC(c2cc(C)c(Oc3ccc(F)cc3)cc2)=O)ncc2c(n1)COC2 C(CO)(CCCCNC(=O)C(O)C(F)F)NC(c1c[nH]nc1[N+](=O)[O-])=O CS(=O)(=O)c1cc(NC(=O)Cn2cc(COC3CCOC3)nn2)co1 N1(C(c2occ(C(N)=O)c2)=O)CCC(CO)(NC(=O)CCc2cncs2)C1 c1(C(N2CCCC(C(C)C(=O)O)C2)=O)cc2n(n1)CCNC2=O c1(C(N2C3CN(Cc4ccc(C#N)cc4)CC2C3)=O)cc2cn[nH]c2cn1 c1(CC)nn(C)cc1C(=O)NCCCC1CCCCN1C(C1CC(=O)N(C)C1)=O C12(NC(C=C(CC)CC)=O)CCN(C(c3ccc(OC(F)(F)F)nc3)=O)CC1C2 c1ccc2c(c1)OCC2CNc1cc(N2CCC3(CCCC3)C2)ncn1 N1(C(C(CC)NC(c2ccc(Cl)cn2)=O)=O)CCC(C)(C(C)C)CC1 c1(C(C)C)cc(C(=O)NCC(CO)NC(=O)Cn2ccnn2)ccc1F c1(C(=O)NC2(C)CCN(C(C3(C)CCC3)=O)C2)ccc(Br)c(O)n1 C1(C#CC(=O)NCC2CN(C(=O)CC3CCCCC3)CCC2C)(CC)COC1 C12(NC(c3ccnn3C3CC3)=O)CCN(C(=O)CSCc3ncc[nH]3)CC1C2 Cc1ccc2c(c1)SC(C(N1CCC(NC(c3cccnc3)=O)C1(C)C)=O)C2 C(=O)(CCC(=O)N1CCC(O)CC1)NC(CC(C)NC(C1(F)CCC1)=O)C c1(C(N2C3CC(CNC(C(COC)N(C)C)=O)C(C3)C2)=O)cnn2c1CCCC2 c1(C(=O)NC2(C(N(C(C)CC(N)=O)C)=O)CCC2)ccc(=N)[nH]n1 N1(C(c2cn(C)c(=O)cc2)=O)CCN(C(=O)CCSC(F)(F)F)CC(C)(C)C1 C(N=c1cc(C)[nH]c(=NCC2CCCO2)[nH]1)C1CC(=C)C1 CC1CC(NC(=O)CCSC(F)(F)F)CCN1C(C1CCCSC1)=O C(CCC(=O)NC1CN(C)CC1(C)C)(C(C)C)NC(c1cc(OC)nn1C)=O C1(NC(C(c2ccc(CC)s2)=O)=O)CCN(C(=O)C(O)CC)CC1 N1(C(CC(CC)C)=O)CC(NC(=O)C2=CCCSC2)C2CC2C1 c1(OC)ccc(CN2CC3CN(C(c4cc(F)ccc4Br)=O)CC23)c(Cl)c1OC c1(CN(CCCCCC)CC(N2CCC(CC#N)C2)=O)cccc(Cl)c1 C1(NC(Cc2ccc(OCC)cn2)=O)CN(C(c2csnn2)=O)CC2CC12 C(=O)(CC(C)C(F)(F)F)N(C(C)C(=O)NC(CO)CCO)CC c1(NC(N(CCCOC)Cc2ccccc2O)=O)ccc2c(c1)S(=O)(=O)NC2 C1(C(N2CC(C)C2(C)C)=O)CC(N=[N+]=[N-])CN1C(=O)Cn1ccccc1=O c1(C(C)=O)ccc(C(N2CCC(O)(CNC(=O)C=Cc3cnccn3)C2)=O)nn1 C1(C(=O)NCC2(O)CC(NC(c3cncc(N)c3)=O)C2)CCc2nccn2CC1 N1(C(c2cc(CNC(c3cn(CC)nc3C)=O)[nH]n2)=O)CC2CC(C)C2C1 C#CCCCC(C)C(=O)NCC1CN(C(C2CCCN2C)=O)C1 C(=O)(CC(C)C(F)(F)F)NC(CCSC)C(=O)NCc1cc(F)ccc1O C1(CC)CN(C(c2cccc(C(C)C)c2)=O)CCN1C(=O)C=C1CCN(C)CC1 CC(CO)CCN=c1[nH]c(N2CCC3(CC2)CN(C)CCN3C)nc2c1CCC2 C1(CC(=O)NC(CN(C(C2(C)CC(=C)C2)=O)C)CC)CCC(C)(C)O1 c1(-c2n(-c3ccc(C)cc3C)nc(C3CCC(=O)N3)n2)cc2cc(Br)ccc2s1 C(=O)(CCCCCO)N1CCC(C)C1CNC(=O)Cc1cncn1C c1(OC)ncccc1CNC(c1ccccc1C(C)C)c1nnnn1C1CCC1 c1(C(N2CCN(C(c3cc(C)ncc3C)=O)C(C)C2)=O)cc2ccccn2c1 Cc1sc(C(N2CC(NC(c3ccc(Br)cn3)=O)CC2C)=O)c(C)c1C C1(NC(=O)Nc2ncnc(OC)c2OC)CC2CCCCN2C1 CCC(C)(C)C(=O)C(=O)N1CCC(CC(N2CC(N(C)C)C(O)C2)=O)C1(C)C CN1CCN(C(=O)CCc2cn[nH]c2)CC1C(=O)Nc1cccnc1 CCC(C)(C)C(O)C(=O)N(CCNC(=O)C=CC(C)CC)C1CC1 c1(CN(C(C2N(CC)CCCC2)=O)C)ccc(Cl)cc1O.C12CCCN1C2=O C1(OCC(=O)N(CCCNC(C(C)=CC)=O)CC)CCCCC1C CC(Cl)(CCl)CS(=O)(=O)NC(=O)C(=O)NCC1CCC(c2ccccc2)CC1 c1(CCN2CCN(C(=O)NC3CCNCC3)CC2)ccccc1Cl N1(C(CC2CCN(OCC)CC2)=O)CCC2(CC1)CC(C)N(C(=O)CNC=O)C2 CCC(C)CC(=O)C(=O)NCCn1ccc(C(=O)NCCN(C)C2CC2)c1 c1(C(N(CC(CNC(C(CCOC)C)=O)O)C)=O)cncc2c1CCCC2 CCC(CC(=O)NC1CCCC1CC(=O)N(C)Cc1cccc(O)n1)SC c1(C(=O)NCCC(CNC(c2cscc2Cl)=O)O)noc2cc(F)ccc12 C#CC1(O)CCN(C(=O)CC2CCC(NC(=O)CC(C)CC(=O)OC)C2)CC1 C1(O)(c2cn(Cc3cccc(C)c3)nn2)CCN(C(C2CCC(=O)N2)=O)CC1 C1(CNC(=O)C(O)Cn2cncn2)CC(O)CN1C(c1ccc(Cl)o1)=O C(CN=c1nc(C)cc(C)[nH]1)C1CCN(C(CCC)=O)C1 c1(C(N(CCCN(C)C(C2(C)CCCO2)=O)C)=O)ccc(N)cc1O C1(N=[N+]=[N-])(C(=O)NCC(C(CC)C)CO)CCN(C(=O)CN2CCCC2=O)C1 Cc1ncncc1C(=O)NCC1CCCN1Cc1cccc(-n2ccnc2)c1 CON=CC(=O)NCC(C)(CO)NC(C1CC(=O)C1C)=O c1(C(N(CC(C)NC(C2CC=CC2)=O)C)=O)cc(C(F)(F)F)ccc1N N1(C(C(CC=C)CNC(c2cccc(CO)c2)=O)=O)CCC(C)(C2CC2)C1 C(CCCS(C)=O)OC(=O)C(F)CC1CN(C(=O)OCC)C1 CCCCC(CC(=O)NCc1noc(C(N)=O)n1)NC(C1(C)SCCCS1)=O C1(NCC(N2CC(CCO)(NC(C(C)OCC)=O)C2)=O)CCCCC1N(C)C c1(C(N2CCN(C3CCN(C(C)C)C3=O)CC2C)=O)cnn2ccccc12 c1(CC(=O)NC2CCCC(CNC(CC3(C)CC3)=O)C2)cc(F)cc(F)c1 C1(F)(CNC(C2CCC(C(=O)OC)O2)=O)CCCN(C(c2ccnnc2S)=O)C1 C1(C(N2CCC(CCNC(=O)C=Cc3cnccn3)C2)=O)CC2COCC2C1 n1(CC(=O)NCC(C2CC2)NC(C(N2CCSCC2)C)=O)cnccc1=O N1(C(CCC(=O)NC)=O)CC(C)C(NC(c2cnn(C)n2)=O)C(C)C1 S(=O)(=O)(c1ccc(C(=O)N(C(CC)C)C)cc1)N(Cc1ccc(SC)cc1)CC C1(C(C)(C)C)(CNC(C2CCCCC2c2nc[nH]n2)=O)CCN(C(=O)CO)C1 C1(CNC(C2(NC(=O)CC3CCC3)CSC2)=O)CC(CO)CO1 C1(NC(C23CC(NC(c4ccn(CC)n4)=O)(C2)C3)=O)CCCCC1(F)F C1(C(=O)NC2C(NC(CCSCCC)=O)CCOC2)CCCCCS1(=O)=O C(=O)(C1=CC(C)CC1)NC1CCC(NC(Cn2c(C)c(Cl)cn2)=O)C1 C(=O)(CCCCC(N)=O)NC(C(C(C)C)N(C(CCC)=O)CC)C CN1CCC(NC(=O)C(CC2CCC2)NC(=O)C(C2CCOCC2)=O)C1(C)C C1(CCOC)(OC)CCN(C(=O)CCCN2CCCC2)C1.C(C1C(=O)N1)OCC CC1(CNC(=O)Cn2cccnc2=O)CCCC1NC(c1cscc1F)=O CN1N=C(CC(=O)NC2COCC2NC(c2ncnc3c2CCCC3)=O)CC1=O CC1COCC(C(N2CC(F)CC2CC(=O)NC2CC2C(F)(F)F)=O)O1 N1(C(CCCOCC)=O)CC(C)CN(C(c2ccc(C)c(F)n2)=O)C(C)C1 C1(NC(C(C)n2ccnc2)=O)CC(C(=O)O)C12CCC2 c1(CSC)cccc(C(=O)NC2(C)CCN(C(=O)COc3cn[nH]c3)C2)c1 C1(C)(CC)CCC(C(=O)NCC#CCNC(=O)C(F)(F)C2CC2)O1 c1(C(N2CCC(N(C(c3nn(C)cc3Cl)=O)CC)CC2)=O)c(O)nnc(C)c1C C1(CNC(CCC=C)=O)CN(C(=O)CC(C)C(F)(F)F)CC12CCC2 Cc1nnc2n1CC(C(=O)NCC1CCN(C(c3ccoc3)=O)C13CC3)C2 Cc1ccc(CC(N2CCC(C)(C(=O)Nc3cccc(F)c3C)C2)=O)c(C)c1 CN1CCCC(C(=O)NC2CC2NC(c2ccc(Cn3ccnc3)cc2)=O)C1 N1(C(C2CC(OC)C2)=O)CCC2(CC1)CC2CNC(=O)C1=C(C)CCOC1 C1(CCC(=O)NCCCN(C(C2(CCF)CCC2)=O)CC)CCCN(C)C1 C1(N2CCN(C(c3cc(CC)no3)=O)CC2)CCCCNC1=O c1(C(N(CCCN(C(CC2CCN(C)C2)=O)C)C)=O)ccc(F)c(O)c1 N1(CC(=O)NCc2ccc(F)cc2)CC2(CCCCC2)CC1C(=O)O c1(C(N2C(C(=O)NC3(C(C)C)CC3)CC=CC2)=O)c[nH]c2ncccc12 CC1(C)CN(C(C2(O)CCCC2)=O)CC2(CN(c3nc4cc(F)ccc4o3)C2)O1 c1(OC)cc(Cl)ccc1Cn1c(N2CC(c3ccccc3)OCC2)nnn1 c1(C(=O)NCC2C(NC(C(C)SC)=O)CCC2)cc(O)nc(C2CC2)n1 S(=O)(=O)(c1ccc2c(c1)nnn2C)N1CCN(C)C(C2CC2)C1 C1(C(NOCCCOC)=O)CCC(CNC(=O)C=C(C)C2CC2)O1 Cc1ccc(C(N2CCCCC2C(=O)NCC(C)(F)C(C)(C)F)=O)nc1O CN1CC=C(C(=O)NCCCC2CN(C(C3CC(C)(C)C3)=O)CCO2)C1 c1(COC)cncc(C(=O)NCC2CCN2C(c2ccc[n+]([O-])c2)=O)c1 c1(NC(c2nc(CN(C)C)c(Cl)cc2)=O)sc2nc3n(c(=O)c2c1C)CCC3 C(=O)(N1CCC(C(=O)NC2CCCOCC2)O1)C1(SC)CCC1 C1(C(C)(C)C)CNC(=O)CN1C(=O)C(CNC(c1ccc(O)cn1)=O)CC1CC1 c1(C(=O)NC2CN(C(C3(CCOCC)CCC3)=O)CC2C)cnc2c(c1)CCC2 c1(C(=O)NC(CNC(C(CCSC)OC)=O)C2CC2)coc2c1NC(=O)CCC2 n1(CC(=O)NCC2(F)CN(C(C3CCC3(F)F)=O)C2)cc(Br)ccc1=O N1(Cc2cc(C)no2)CCC2(NC(=O)CCc3ccncn3)CCCC12 c1(NC2CCCC(NC(CC(C)(C)O)=O)C2)ncnc2c1CCO2 N1(C(CCc2ccc(C)o2)=O)CCC(CNC(C2CC(F)C2)=O)C(C)C1 N12CC3(CCCCC3)C1NC2=O.C1(COC)(OCc2ccccc2)CCOC1 c1(NCC2(OCC)CCC2)ccc(S(=O)(=O)N2CCN(C(C)CO)CC2)cc1Br N1(C(=O)Nc2ncc(C(F)(F)F)s2)CCC(c2cccs2)CC1 c1(NC=O)ccc(C(=O)NCC2CCN2C(c2ccc(-c3cnc[nH]3)cc2)=O)cc1 N1(C(c2cccn(C3CCC3)c2=O)=O)CCN(C(C2CC=CCO2)=O)C(C2CC2)C1 c1(CC)ccc(C(=O)N(C)CC2CC(F)CN2C(c2csc(COC)c2)=O)cc1 c1(C(=O)NCC2C=CC(NC(Cc3c(C)ncs3)=O)C2)cn(C)c(=O)cn1 Cc1cc(C#N)ccc1C(N1CC(CC(=O)Nc2ccc(F)cc2F)C(C)C1)=O C=CCCCCCC(=O)NCC1CC2CN(C(c3ccc4cc[nH]c4c3)=O)CC12 C1(CCC)(NC(=O)C(C)C(F)(F)F)CCN(C(c2ccc(C)cc2)=O)CC1 CC(C)(C)CC(=O)NC1CCCCC1NC(=O)CCC(=O)c1cccnc1 c1(OC)ccc(F)cc1C(=O)NC(C)CC(C)NC(=O)COCCF c1(COCC(=O)O)cccc(-c2cn(CCCCC(=O)NCC(F)(F)F)nn2)c1 c1(CNC(CCN(C)C(=O)NC2CCC2C(C)(C)C)=O)nc(CO)cs1 C(CCC(O)CO)N(C)C(C1CC(CNC(=O)Cn2nccn2)C1)=O Cc1cncc(C(N2CCCCC2C2CCN(C(C3(C)COC3)=O)C2)=O)n1 C(C)(CCCC(=O)N1CCOC(C(C)C)C1)NC(C1C(=C)C1)=O C1(N(C(c2c(C)c[nH]n2)=O)C)CN(C(c2ccc(C#N)cn2)=O)CCC1O c1(CCC(=O)NC(CN(C(C(CSC)C)=O)C)(CO)CO)ccc(C)cc1C C12(NC(C3(C(=O)OC)CC3)=O)CC1CN(C(c1occc1Cl)=O)C2 n1(CC(=C)C)c(N2CCN(C3CCN(CC)C3)CC2)nnc1-c1ccc(O)nc1 C(C(CC(=O)NCC1(O)CCCOC1)C1CCC1)NC(C1(C)C(C)(C)C1)=O c1(CN(C)C(C2CCCN2C(c2cc(-c3ccco3)[nH]n2)=O)=O)cnnn1C CC1CCc2nc(C(N3CCCCC(NC(=O)Cc4cncn4C)C3)=O)cn2C1 Cc1nn(C)c(C)c1OCC(=O)NCC(O)CNC(C1(C(C)C)CCC1)=O N1(C(=O)NCCOCCC#C)CC(C)c2ncccc21 C1(O)(C(=O)NCC=C)CCN(C(C2(c3cccs3)CCCCC2)=O)CC1 Cc1ccc(CCC(=O)NC2(CNC(=O)Cn3cc(CN(C)C)nn3)CC2)s1 C1(NC(c2nccc(CC)c2)=O)CN(C(C2CC(=O)NC2(C)C)=O)CC1(C)C c1(C(=O)NCCCN(C(=O)CC(C)(C)C#N)CC)cc(C)ccc1Cl C1(OC(CC(=O)OC(C)C(=O)c2ccco2)=O)CCCC(F)(F)C1 Cc1cccc(C(C)C(N2CC(n3cc(-c4ccns4)nn3)(CO)C2)=O)c1 C1(N(C(CC(CC)O)=O)C)CC2CCC(C1)N2C(c1ccc(F)cc1)=O c1(OC)cc(C(=O)NCCN(C(=O)CC2CCC(C)CC2)C)ccc1C#N C(CCCC(=O)NCCCN(CCCNC(=O)C(C)COC)C)CC.OCC N1(C(CCN(C(=O)CCC2CC2(F)F)C(C)C)=O)CCOCC(C2CC2)C1 C1(CC(=O)NCC(CC(=O)N2CC(SCC)C2)C)CC2(CCO1)CC2 N1(C(C2(C)N(C)CCC2)=O)CCCC2CN(C(=O)C=C3CCCC3)CCC12 C(=O)(CCCCCC(C)O)NC(CCN(C(c1ccc(=NC)[nH]c1)=O)C)C c1(CC(=O)N(CC(C)NC(c2c[nH]nc2OCC(F)F)=O)CC)nnc(S)n1C C(CCCCCN(C)C(c1n[nH]cc1CC)=O)NC(C=CC(=O)OCCCC)=O N1(Cc2nnc(C(C)C)o2)CCCC(CO)(NC(=O)CC2CCC(C(N)=O)O2)C1 c1(C(=O)NC(CNC(C2(CC)COC2)=O)C2CC2)ccncc1C(F)F C1(COC)CN(C(=O)CC(Cl)Cl)CCN1C(=O)CCCOC(C)(C)C c1(OC)ccc(Cl)c(C(=O)COC(C2C=CCN(C(=O)OC)C2)=O)n1 C(=O)(C(C)C(F)(F)C(F)F)NCC(CC=C)CO.c12ccccc1O2 c1(OC)cc(OC)c(C(N2CCC(NC(=O)CCNC(=O)C=CCl)C2)=O)c(F)c1 O=C(N=c1ccn(CNCc2ncnc3sccc23)[nH]1)NCc1ccccc1 c1(C(=O)NC(CCCC)C(=O)N2CCCCC(C)C2)cc2ccccn2n1 N1(C(CN(C(C)C)C)=O)CC(N(C)C(c2cc(Cl)nnc2O)=O)C2(CC2)C1 CC(O)(C(=O)NCCn1cnc(C(N2C3CSCC2C3)=O)c1)C(F)(F)F c1(OC)ncc(C(N2CCC(CO)(CNC(=O)CC3CC4CC4C3)C2)=O)cc1C c1(C(N2CCC(NC(C3(CC#C)CCCC3)=O)C(F)C2)=O)cccc(C#N)c1C n1(CCC(=O)NC2CC(NC(C34CCC(CC3)C4)=O)C2)nc2ccccn2c1=O c1(OC)cc(C)sc1C(=O)NCC(C)NC(=O)C=Cc1nc[nH]n1 C(=O)(CC(C1CC1)NC(C1(O)CCC1)=O)N(CC=C)CC1CC1 C1(CNC(C2(CCC=C)CN(C(c3ncn(C(C)C)n3)=O)C2)=O)CCOCC1C C1(NC(c2cccs2)=O)CC2CC1CN(C(c1cccc(OC(F)(F)F)n1)=O)C2 c1(C(=O)NC2C(C)CN(C(=O)CCC3CCCCC3)C2)ccn2cccc2c1 CC1CC(CNC(c2occc2CNC(=O)C2=CCCSC2)=O)CC(C)C1 C1(N(C(C(C(=O)OC)Oc2cccc(CSC)c2)CC)C)CS(=O)(=O)CC1O C1(C(=O)NCC(C)(C)NC(c2scc(COC)c2)=O)CCn2ncnc2C1 C(C)(CC(=O)N(C(C)C(=O)N(C)C1CC1)C)CC1(NC(C)=O)CC1 CCCCCC(O)C(=O)NCC1CCN1C(=O)C=Cc1cscn1 c1(C(=O)NCCC(C)N(c2ncnc(Cl)c2Br)C)cnc2[nH]c(O)nc2c1 c1(C(N2C(CNC(c3c(C)ccc(C)n3)=O)CC3CC32)=O)cn2c(n1)CCCC2 C1(N(C(CCC)=O)CC2CCCO2)CCN(C(=O)CCC2CCCN2C)CC1 Cc1cn2c(CC(=O)NC3CC(CNC(=O)Cc4ccoc4)C3)csc2n1 C12(NC(c3ncncc3F)=O)CCN(C(c3ccc(O)c(F)c3)=O)CC1C2 Cc1cc(NC(c2cccc(OCCCOC3COC3)c2)=O)cc(O)c1 C(CCC(=O)N(C)Cc1ncc(COC)s1)NC(=O)OCC N1(C(c2c(=O)ccn(C)c2)=O)CCC2CN(C(=O)CSCC3CCCO3)C2C1 c1(C2C(C(N(CC(O)CNC(=O)CCCCNC(N)=O)C)=O)C2)cccc(C#N)c1 N1(C(c2c(OC)c[nH]n2)=O)CCC(NC(c2cc(Cl)cc(Cl)c2)=O)CC1C Cc1ccc(C(=O)N(CCCCN(C)C(C2CC23CC3)=O)C)c(O)c1 c1(CC)cc(C(=O)NCC(C(C)(C)C)NC(C2CC3CCC3C2)=O)cc(N)c1 Cc1cc(C(=O)NCC(F)CNC(=O)Cc2c(C)noc2C)ncc1N c1(C(c2n(C(CC)(C)C)nnn2)NCC2(COC)CCC2)ccc(Br)c(Cl)c1 CC1CS(=O)CCN1C(C1CC2CCC1N2C(c1ncccc1Cl)=O)=O C1(C)(CNC(CC(C)(C)OC)=O)CCN(C(c2ccc(F)s2)=O)CC1 C1(C(=O)NC2(C)CC(NC(=O)Cc3cnc[nH]3)C2)COCCN1C=O N1(C(CS(=O)(=O)N(C)C)=O)CCC(C2(O)CN(C(=O)C(C)(O)C(F)(F)F)C2)CC1 C1(C(N2C3CC(CC(NC(C(C)(C)F)=O)C3)C2)=O)CCCCC12OCCO2 Cn1ncc2cc(C(=O)Nc3cccc(CNC(c4ncnc(O)c4F)=O)c3)sc12 N#Cc1ncccc1-c1cn(CC(c2cccc(N3CCCC3=O)c2)=O)nn1 c1(C2(C)CNC2)cn(CC(=O)NC2CC(n3cnnc3)C2)nn1 N1(CC(N2C(c3[nH]c(C(=O)OC)c(C)n3)CCC2)=O)Cc2ccc(Br)cc2C1=O n1(CC(=O)NC(C)CCCNC(c2cccc(F)c2O)=O)cc(S(C)(=O)=O)cn1 C(=O)(C#CC1CCCCC1)N(C)CC1CCC(C(=O)O)CC1 C1(C(CNC(C(C)SCCCC)=O)O)CCN(C(c2cncn2C)=O)CC1 N1(C(C(CCC=C)(F)F)=O)CC(CNC(=O)CC(C)SC)OC2(CCC2)C1 CCC(O)CCN=c1cc(C)[nH]c(=NCc2ccc(SC(F)F)cc2)[nH]1 N1(C(c2sc(C)c(O)n2)=O)CCC(NC(=O)Cc2cccnc2Cl)C(C)C1 c1(CN2CC(NC(c3sccc3F)=O)C(O)C2)cnc2ccccc2c1 c1(C(=O)NC(C(=O)NCC(C)OCC=C)Cn2cncn2)cc[nH]c(=NC)c1 N1(C(C=Cc2cn(C)nn2)=O)CCC(NC(=O)CCc2ccoc2)C12CCC2 N1(C(C(C)CO)=O)CCC2C(C(N3CCCC3(C)C3CCC3)=O)C2C1 CCC(C)CC(C)N(C)C(c1occc1CNC(C1(CC)COC1)=O)=O c1(C(N(CC(C)N(C(=O)C(F)C(F)(F)F)C)C)=O)cccc(F)c1F C(=O)(C1c2cnn(C)c2CN1C(=O)OCC(C)(C)C)NC(C(F)=CC)=O C1(C(=O)OCC)CCCN(C(=O)Nc2cnn(C(C)(C)C)c2CN2CCCC2)C1 O=S(=O)(c1cc(Br)c(Cl)s1)N1CCC(Nc2cccc(Cl)c2)CC1 n1(CCC)c(N)c(CCc2cc(C)n(-c3cccc(C#N)c3)c2C)c(O)nc1=O c1(C(C(=O)OCC2N(CC(C(C)(C)C)F)C(=O)CC2)=O)ccc2c(c1)OCO2 N1(C(=O)OC(C)(C)C)CC2CC1(C(=O)NOCC1CC13CCC3)C2 N1(C(c2c(C)cc[nH]2)=O)CCC(F)(CNC(=O)CC=CCc2ccccc2)C1 c1(C(N2CCCC(c3nccs3)C2)C(=O)NCC)cccc2cnn(C)c12 c1(OCC(=O)NC2C(NC(C(c3ccc(C)cc3)C)=O)C2)nc2ccccc2s1 C1(CNC(=O)CCCc2cc[nH]n2)COCCN(C(c2cnco2)=O)C1 CCC(C)CC(=O)NCC1(NC(=O)CCc2ccc(SC)cc2)CCOC1 N1(C(C(CCC)(C)C)=O)CC2CCCC(NC(C3CCSC3)=O)(C2)C1 C1(N(C(=O)CCCc2ncco2)CC)CCCN(C(C2(F)CC=CC2)=O)C1 c1(SC)ncc(N)c(C(=O)N(CCC(F)(F)F)C(C)C2CC2)n1 C(CCN=c1[nH]c(=NCCC2CC(O)C2)[nH]c2c1CCCC2)OC(=N)O C(C)(CCCCC#N)(c1nnnn1CSc1ccccc1)NCC(CCC)OC N1(C(C(C=C)CC)=O)CCC2(CC2C(N2CC3CC3C3CC23)=O)C1 c1(C(=O)NC2CCC(N(C)C(c3ccns3)=O)C2)ccc(F)c(Br)c1 c1(C(N(C(CCC2N(C)CCC2)=O)C2C3COCC23)=O)c(F)cccc1[N+](=O)[O-] c1(C(N(CC(C)(C)NC(C)C(=O)NC(C)(C)C)C)=O)cc(C2CC2)ns1 N1(C(C(CC)Oc2ccc(C)cc2C)=O)CCC2(CC1)CNCC2C(=O)O c1(C(=O)NC2CC(OC)CN(C(C3CCOC3)=O)C2)cc2ccccc2n1C c1(SC)cscc1C(=O)NCC(CNC(=O)Cn1nnc(=O)[nH]1)CO C1(CNC(CCN(C(=O)C(C)=CC2CC2)CC)=O)CCCCO1 N1(C(C(C2CCC2)OC)=O)CC(NC(c2nocc2C(C)C)=O)C2CCCC2C1 c1(C(=O)NC(C(C)C)CNC(C2CN(C)C(=O)N2)=O)cccc(C#CC2CC2)c1 CC(CCCNC(=O)CCC1CCOC1)NC(=O)C(C)Sc1ccccc1 c1(C(N2CCC(C)C(NC(=O)Cc3nncs3)C2)=O)ccc(Cl)c(C#N)n1 CC(C)CC(F)(F)C(=O)NC1CCCC(NC(c2ccc(F)c(F)c2)=O)CC1 c1(OC)cc(C(N2CC(C)C(C)C2)=O)c(-c2cnc(=N)[nH]c2)cn1 CC(C)CS(=O)(=O)CC(=O)N1CCN(C(C2CCC(=O)N2C)=O)C(CC2CC2)C1 C1(NC(c2ccn(C)c2)=O)COC2(C1)CN(CC1CCC(F)(F)C1)C2 C1(NC(C(C)OCCC#C)=O)CN(CCOc2ccccc2OC)CCC1C N1(C(c2n(CC)nc(C)c2)=O)CC(C)(C)OCC1CNC(=O)C1=CCCSC1 c1(C(N2CCC(C(N(CCCO)C(C)C)=O)CC2)=O)cc(Cl)c2cn[nH]c2c1 c1(C(N2CCCC2C(=O)N(C)C)C(=O)NC)n[nH]c2ccc(OCC)cc12 C(=O)(CC(C)(CN(C)C)C(F)(F)F)NC1C2CN(C(CCOCC)=O)CC21 N1(C(CN(C(C(C=CC)O)=O)C2CC2)=O)CCCC2(CC(O)C2)C1 C1(C(N2CCC(N(C)C(c3n[nH]cc3Br)=O)CC2)=O)CCn2nnnc2C1 c1(C(=O)NCC(C)(CC)NC(CCCCC)=O)cc2ccccc2c(O)n1 C(=O)(C(C)CC(C)(C)C)NC1C(n2cc(CCCOC)nn2)CCCC1 C1(c2c(COC(C3C(C(C)C)OCC3)=O)cnn2C)CC2(CCO1)CC2 C1(C)(C(N2CC(CNC(c3nc(CC(C)C)sc3)=O)C(C)C2)=O)CCC(O)CC1 C1(C(C)C)CN(C(=O)CN(C)C)CCCN1C(=O)CSCc1nccn1C c1(CN(C(C2CCCN2CC)=O)C2CC2)ccc(CC(=O)NC2C(CC)C2)cc1 CC(C)C(C)C(=O)NCC1CCCC1CN(CCC(=O)OC(C)(C)C)CCCO N12CC(OC)C(C1)C2=O.C(=O)(CS(C)(=O)=O)NC1N(CCC)CCC1 C1(C(N2CC(C)(CNC(c3cc(CF)on3)=O)OCC2)=O)CCCC2CCCN12 C#Cc1cccc(C(c2nnnn2C)NCc2ccnn2C2CCCC2)c1 C12(CNC(C3(CCCC)CCCC3)=O)COCCN1CCN(C(=O)C(C)O)C2 Cc1cc(CN(C(=O)C(C)(Br)C(C)C)C2CC2)c2[nH]c(C)c(C)c2c1 C(=O)(C(C)(C)S(C)(=O)=O)N1CC2C(N(C(CSCc3nc(C)sc3)=O)C)C2C1 C(c1ccco1)=CC(=O)NC(C)C(=O)NCCOCCNC(C1CCSCC1)=O CC(CO)N(C1CCCC1)N(C)CC(=O)OC1CCCC1 N1(C(C2(SC)CC2)=O)CCCN(CCCCNC(C2(C)CC(F)(F)C2)=O)CC1 c1(NC(=O)NCc2nnc(S)n2C2CC2)cnc2ccccn2c1=O CON1CCC(CC(N2CC(N(C)C(c3nc(O)c(C)s3)=O)C(O)C2)=O)CC1 C(=O)(CC(C(F)F)n1ccnc1)NC(C)CCCCNC(c1cc(O)cs1)=O CCCCCCC(F)C(=O)N(C)CC1(CNC(c2ccc(CO)o2)=O)CC1 c1(C(=O)NCC2(CNC(C(CC)O)=O)CCCC2)nnn(C)c1C(F)F c1(CC)ncoc1C(N1CC(CO)(NC(c2cnn(CC3CCOC3)c2)=O)C1)=O N1(C(C(COC)N(C)C)=O)CC(NC(=O)C(=Cc2cccnc2)C)C(C)(C)C1 C(=O)(C1CCCc2cccnc21)NCCCC(C)NC(c1c(CC)oc(C)c1)=O CC1=NOC(CC(=O)NCCOCCC(=O)NCc2ccncc2)C1 N1(C(c2ccc(OC)cc2N)=O)CCCN(C(C2C(C)C2C)=O)CC1C N1(C(c2c(Cl)cccc2Br)=O)CC2CCN(C(c3cnccc3Cl)=O)C2C1 N1(C(CCCN(C)C)=O)CCCC(CNC(c2nnn(C)c2C(F)(F)F)=O)C1 Cc1cc(C)c(C(=O)N(C2(C(N3CC(CO)CC(C)C3)=O)CC2)C)cn1 N1(CC)CCC(C(=O)NC2CC(CNC(C3(F)CC3(Cl)Cl)=O)C2)C1 C(=O)(CCCCC(C)(C)C)N1CC(NC(COC(CC)(C)C)=O)N(C)CC1 C1(NC(C2CC3(C2)CC32CC2)=O)CC2CCC(C1)N2C(C1C2(CC2)C12CC2)=O C1(C(=O)NC2(CC)CCOC2)CN(C(=O)C2=C(C)CCC2)CC(C)(C)C1 CCCC(C)(C)CC(=O)NCc1cccc(NC(C23CC4CC(CC2C4)C3)=O)c1 C(=O)(C(C)C(F)(F)C(F)F)NC1C2(CN(C(c3n(CCC)nc(C)c3)=O)C2)CC1 Cc1ccc(C(C)CC(=O)N(CCC(C(C)C)NC(c2csnc2C)=O)C)cc1 N1(C(c2cnc(CC)[nH]2)=O)CC(NC(c2c(Cl)n[nH]c2C)=O)C(C)C1 C=CCCC(F)(F)C(=O)NCC(O)CCNC(=O)CCc1cc(OC)no1 CC1(C)CC(NC(=O)COCC(F)F)CN1C(c1cnc(C2CCOCC2)s1)=O c1(C(N2CC(NC(C=COCC)=O)(CO)C2)=O)cnc2snc(C)c2c1 N1(C(COCCOC)=O)CCC(OCCC(=O)N(C)C(C)C)C1.C1C(=O)N1 C1(N(C)C)(C(N2CCCC2CNC(=O)CCC2CCC2)=O)CCCSC1 Cc1ccc(O)c(C(N2CC=CC(C(=O)NC3CN(C)CCC3O)C2)=O)c1 C1(C(=O)NC2(CC=C)CC2)(CNC(=O)C(C)C2CCCC2)CCOCC1 N1(C(=O)CC2CC(C3CCCCC3)C2)CC2CCCC(C1)N2C(=O)C=CCO C1(C)(C(N(C2CCN(C)C2)C)=O)CN(C(C2CN3CCN2CC3)=O)C(C)(C)C1 C(=O)(C(CC(C)(C)C)NC(c1cc(C)c(O)nn1)=O)NC(CN(CCC)CC)C C(=O)(CCN(OC)C(=O)C1CC2(CCN1C(=O)CCC1CCCO1)CC2)OC C1(C(C)(C)CNC(=O)C(O)C2CCCC2)CCN(C(c2sccc2CO)=O)CC1 C1(NC(C(C2CC2)OC)=O)(CNC(c2nc(C(F)(F)F)ns2)=O)CCCC1 C1(NC(c2cc(C)c(C)s2)=O)CC2CC(NC(c3ccnc(O)c3)=O)C1C2 S(=O)(=O)(c1cn[nH]c1)N1C(C)CCC1C(=O)Nc1cccc(C(N)=O)c1 C(C(C)NC(=O)CCc1ccsc1)(C(C)C)NC(c1cc(COC)no1)=O C1(NC(C2(C)C(CC)CCC2)=O)COC2(C1)CN(C(C1CC13CCCC3)=O)C2 c1(NCCS(=O)(=O)N2CCCC2)cc(=NC2CCC2)[nH]c(Cl)n1 C(C1c2ccccc2CCN1C(=O)C=CC1CCCC1)NC(c1coc(Cl)n1)=O N1(C(C(CC=CC)C)=O)CCCN(C(=O)Cc2ccc(F)cn2)C(CO)C1 c1(CCC(=O)NCCN(C(=O)Cn2cc(C#N)cn2)C)c(F)cccc1F CCCCC(C(=O)NC(c1nccnc1C)C)NC(c1cc[n+]([O-])cc1)=O c1(C(=O)NCC2CCC(C)CN2C(=O)CCOC2CCC2)c(Cl)ccc(F)c1N c1(C(=O)NC(COC)C(=O)NCCC2CCOC2)ccccc1O C1(CC)(NC(c2nccn2C)=O)CCCN(C(C2CC(=C(F)F)C2)=O)C1 N1(C(C2C(OC)(OC)CC2)=O)CC=CCC1C(=O)NC(C1CSC1)C c1(C(=O)NC2C(F)CCN(C(CC(=O)OC)=O)C2)cccc2cc(Cl)ccc12 c1(C(N2CCC(N(C(C(CC)OC)=O)CCO)C2)=O)ccc2ccn(C)c2c1 C(=O)(CCC(CF)CF)N(CCN(C(=O)CC1COCC1(C)C)C(C)C)C O=S(=O)(c1ccc(Br)cc1Nc1ncccc1F)N1CCC(C2CCOC2)C1 C1(NC(c2cccc(C(=O)NC)c2)=O)CCN(C(c2cnncc2O)=O)CC1C c1(C2(n3cccn3)CN(S(CCNC(=O)C3CC3)(=O)=O)C2)ccc(Br)cc1 c1(C(N2CCC(F)(CNC(c3coc(C4CC4)n3)=O)C2)=O)cnc2[nH]cnc2c1 c1(CNC(C(n2cc(C(CC)(O)CC)nn2)COC)=O)cc(C(N)=O)ccc1C C=CCC(C(=O)N1CCCC1C(=O)NCC1CCCC12CC2)NC(C)=O c1(OC)c(Br)cc(C(N2CC3CN(C(c4csc(C)n4)=O)C3C2)=O)cc1Br N1(c2ccc(C(=O)OC(C)(C)C)cn2)CC2CCCC2(C(N)=O)C1.c1(=O)c(=O)[nH]1 c1(-c2c(C)nc(CCO)s2)cccc2cccc(Cl)c12 c1(NC(C2(SC)CN(C(=O)C(F)CCC(C)C)C2)=O)ccc(C)c(O)c1C c1(CC)ccc(C)nc1NC(C1C=CCN1C(c1nc(C2CC2)cs1)=O)=O C12(CNC(c3cccc(F)c3F)=O)CCCCC1N(CC#N)CC2 Cc1ncc(C#N)cc1NC(=O)C1=CCN(C(c2cc(C)n(C)c2)=O)CC1 N1(C(c2c(C)noc2C(F)F)=O)CC2CCC(NC(=O)CC3CC3(Cl)Cl)CC2C1 N1(C(C2(CC)CCOC2)=O)CC(N(C(=O)CSCCC#N)C)C2(CC2)C1 C1(NC(CC2C3CN(C(C#CC(C)(C)O)=O)CC32)=O)CCCCCCC1O N1(C(CC2C(=O)NC(=O)N2)=O)CCOC2CN(C(C3CCCS3(=O)=O)=O)CC12 C(=O)(CC(C1CC1)NC(=O)C(C)(O)C1CCCCC1)NC c1(NC2C(C)(CC)C2)ccc(S(=O)(=O)NCC2CN(c3ncccn3)C2)c(Br)c1 C1(C(=O)NC2COC3CN(C(C4C(C#C)C4)=O)CC32)C2CC3CC(C2)CC1C3 C(C(=O)Nc1ccc(C2CCCOC2)cc1)(C(C)C)(C(C)C)NC(C)=O N1(C(c2c(C)oc(C#N)c2)=O)CCC2(CC1)CN(C(c1cc(Cl)cc(Cl)c1)=O)C2 C1(C(C)(C)NC(C=CSC)=O)CCN(C(=O)C(F)=C2CCC2)CC1 C1(NC(Cc2cn(CC)nc2)=O)CCCCC1CNC(=O)C(CO)OC C1(C(N2CCC(n3cnnn3)C2)C(=O)NCCOC)CCC(SC)C1 Cc1ccc(C)c(C(=O)N(C2(CC(N3CCOC(C)C3C)=O)CC2)C)c1 C1(CC(=O)NCC2CCN(C(c3ccc(C)[nH]3)=O)C2)CCCCCC1(F)F N1(CC)CCOC(C(=O)N(CCNC(C2(C)CC2(C)C)=O)C(C)C)C1 c1(C(=O)Nc2cc(O)ncn2)ccc(S(=O)(=O)N2CCCCC2)cc1 Cc1oc(=NC2CC(Sc3ccccc3)C2)[nH]c1C1CN(C(=O)OC(C)(C)C)C1 N1(C(C2C(CCC)C2)=O)CC2(CNC(C3(OCC)CCOC3)=O)CC(F)(C1)C2 CC1(C)CCC(CC(N2CCCC2C(C)(C)NC(=O)C2CC2)=O)OC1 C1(CC=C)(NC(=O)Cc2cnnn2C)CCN(C(=O)C(F)C2CCC2)C1 c1(C(N(C2CN(C(C3(C)CCC(C)CC3)=O)C2)C)=O)cc2n(n1)CCNS2(=O)=O N1(C(c2cc(CCC)[nH]n2)=O)CC(O)CC1(C)C(N1CCC(C2CC2)C1)=O Cc1ccc(NC(=O)N(C)C)c(C(=O)NCCC(C)N(C(=O)C(O)C(F)F)C)c1 c1(NC(N2CCCC2C(=O)CCc2ccccc2)=O)ccccc1Br N1(C(CNC(N)=O)=O)CC2CC(NC(c3cnc(C(F)F)nc3)=O)CC1C2 C(C(CC(=O)NC1(CO)CCC(C)C1)NC(=O)CCc1nccn1C)OC C1(NC(COC(C)(C)C)=O)CCCC1C(=O)Nc1ccnn1C1CC1 N=c1[nH]c(CCC(=O)NC2CC2NC(c2sccc2OC(F)F)=O)cs1 N1(C(c2c(C#N)scc2)=O)CC(C2(NC(=O)Cc3cncs3)CC2)C1 CCC(C)(O)C(=O)N1CCCCC1C(=O)NCc1cnsc1 C(=O)(C1CCc2ccccc21)N(CCNC(c1c(CC)n(C)nc1)=O)CCOC N1(C(C2(SCC)CC2)=O)CCC(O)(CNC(=O)C(C(C)C)NC(N)=O)C1 N1(C(C(CC)n2ccnc2)=O)CC2(CC(C(=O)NC(COC)C(=O)OC)CO2)C1 C1(C(N(C2COC(C)(C)C2)C)=O)(CNC(c2csc(C#N)c2)=O)CCCCC1 C#CCC(C(=O)NCCC(C)N1CCC1)NC(=O)C=C(C)C1CC1 C1(c2onc(C(c3ccc(N4CCCS4(=O)=O)cc3)C)n2)CCc2nn[nH]c2C1 c1(C(=O)NC(CCNC(C(CC)(C)F)=O)C)ccc(Cl)cc1F c1(CSCC(=O)Nc2ccc(-c3ccncc3)cc2)ccc(Br)cc1 O(C1CCCc2ccccc21)CC(=O)NC1CCC(NC(C2CCSCC2)=O)C1 N#Cc1cc(C(=O)OC2CCC(C#N)C2)cnc1C(F)(F)F c1(C2C(C(=O)NC(C3CCN(C(c4cnco4)=O)C3)C)C2)cccnc1 c1(C(=O)NC2(CC(=O)N(C)CCn3cccn3)CC2)ccncc1 CCC(C)CCC(=O)NCC(C)CNC(=O)COc1ccccc1C N1(C(CNC(CCC(C)C)=O)=O)CCN(C(=O)C(C)(C)C(N)=O)CC(C)(C)C1 N1(C(C2N(C(CC=O)=O)CCC2)=O)CCCCC(C(=O)NOCC(F)F)C1.NC N1(C(CCCC(C)(F)F)=O)CCCC2CN(C(C3(C)CCOCC3)=O)CCCC12 C#CCC(C)C(=O)N(C(C)CNC(c1ccc(NCc2ccco2)cc1)=O)C C(=O)(C(F)(F)C(O)C(C)C)NC(CCNC(C1(CCOCC)CCC1)=O)(C)C C1(C(CNC(c2cc(OC)ns2)=O)(C)O)CCN(C(C2CCC(=O)O2)=O)CC1 c1(C(N2CC(C(C)NC(C=CC=CC)=O)C2)=O)cc(O)cc(C#N)c1 C(=O)(C(CC(=C)C)OC)N1CC(C(=O)NC(c2ncc[nH]2)C#C)(CC)C1 n1(CCCC)ncc(C(=O)NC2CC(O)(CNC(C3CC=CCC3)=O)C2)c1C C1(CNC(COCCCC)=O)CN(C(=O)C(C)CC(F)F)CCC1(C)C C1(NC(CSCc2cccc(C)c2)=O)CN(C(c2nc(C)no2)=O)CC2(CC2)C1 c1(C(=O)NCCOCCCF)ncccc1Cl C(=O)(C(F)C(C)(C)O)NC(CC=CC)C(=O)N1CC(CO)C1(C)C C(=O)(CCCCC(N)=O)NC(c1cccc(OC)c1)CNC(C1(CC=C)CC1)=O c1(COC)nc(CC(=O)NC(C2CCN(C(C3(n4cncn4)CC3)=O)C2)C)cs1 C(CC(C(=O)N1CCNC(=O)C1)NC(=O)CC1CC(C2CC2)C1)N(C)C c1(CN2CCC(NC(c3c(SCC)cccc3)=O)C2)c(Cl)cccc1I N1(CCC(C)(C)C#N)CC=C(c2cccc(Br)c2)CC1 C12(C(=O)NCC3CC(NC(C4(C)CC(OC)(OC)C4)=O)C3)CC(C1)C(C)(C)O2 c1(CCC(=O)NC2C(NC(c3ccc(C#C)o3)=O)COCC2)cccc(F)c1F CCC(C)(CNC(=O)C(C)Cn1cccn1)C(=O)NCC1CCC(C)(C)O1 c1(CCC(N2CC(COC)(NC(c3cc(Cl)n(C)n3)=O)C2)=O)cnc(C)nc1O C1(NC(C(C)C(C)O)=O)C(C)(C)CN(C(=O)CCC(N)=O)CC1(C)C CC1CCC(C(=O)O)N1c1ccc(C(F)(F)Cl)cn1 C1(C(=O)NCC(C)CC2CC2)COCC1NC(C1CC1Cl)=O CCCC(C#N)C(=O)N1CC(O)CC1CNC(=O)CCc1nnc(O)nc1O CCCCC(C)(F)C(=O)NCC(c1ccc(N(C)C)cc1)NC(C1CC2CC2C1)=O C(=O)(C1=Cc2ccccc2C1)NC1CCN(C(CC2ON=C(C)C2)=O)C(C)C1 N1(C(CC(COC)(C)O)=O)CCN(C(c2cnc(C3CC3)nc2)=O)CC(C)(C)C1 C1(C(=O)OC)CN(C(=O)CCC2CCC(=O)N2)CC2(CCC2)O1 N1(C(C2CCC(C(=O)OCC)C2)=O)CC(C(=O)O)CC12CCOCC2 C1(C(=O)NCc2cn(CC)nc2)CN(C(=O)CC2COCCO2)C(C)(C)C1 c1(C(N2CC3C(CNC(C4CCC(OC)CC4)=O)(C3)C2)=O)cc2ccncc2[nH]1 Cc1c(C(=O)NC2(C)CCN(C(C3C(C)CC3C)=O)CC2)nn(C)c1N c1(CNC(=O)NC2C=CC(C(=O)NC)C2)nccn2ccnc12 Cc1ccc(=N)[nH]c1C(=O)NCC(C1CCCC1)NC(=O)CCN1CCCCC1C C1(C(N(C2CCN(C(Cc3c(CC)con3)=O)C2)CC)=O)CSCC(=O)N1 C=CCCCC(C(=O)N1CCCC(N(C)C)C1)NC(c1ncc(F)cc1F)=O c1(SC)ccc(C(=O)NC2(C(N3CCCC3CNC(N)=O)=O)CC2)o1 N1(C(=O)NCCCl)CCC2C1CCN2C(c1ccc2n[nH]cc2c1)=O C1(NC(=O)CCc2ncccn2)CCN(C(C2CC3CCC2C3)=O)C12CCCC2 C12(C(=O)NCC3CN(C(=O)Cn4ccc(C5CC5)n4)CCO3)CCC(CC1)CC2 C=C1CCC(C(=O)NCCC(O)CNC(c2cccc(C(F)F)c2)=O)CC1 c1(C(N2CCN(CC(CC)CC)CC2)=O)cc2c(C)cccc2o1 C(=O)(CCC(C)(C)C#N)N1CC(CC(C)NC(CC(CC)CN(C)C)=O)C1 CCC(C)CC(C(=O)NCCOCCCF)NC(=O)C(C1CC1)SC c1(OC)ccnc(CN2CCCC2CC(=O)NCCC2CCCN(C)C2)c1 C1(C(=O)NCC(CNC(c2cc(CC)[nH]n2)=O)OC)CCc2c(nnn2CC)C1 N1(C(C=Cc2c(C)nccc2)=O)CCN(C(c2cc(CO)[nH]n2)=O)C(C)C1C c1(C(C(=O)NCC2(CNC(C3CCC(C)C3)=O)CC2)=O)ccc(Cl)cc1 C1(CC(=O)NC2(COC)CCC2)CCN(C(C2C=C(C)CS2)=O)C1 C(=O)(CS(=O)(=O)C1CC1)N1C(COC)(CNC(=O)CC2C(C)C2(F)F)CCC1 c1(C(=O)NC2CCC(C(=O)NCC3C(C)CCC3)C2)ccc(C#N)s1 Cc1nn(CC(N2CC(CNC(c3cnns3)=O)CC2C)=O)cc1Br c1(C(N2CCC(N(C(c3c(C)scc3)=O)C)C2)=O)cc(O)c2nc(C)n(C)c2c1 C=Cn1nncc1C(=O)N(C(C)C(=O)Nc1csc(Cl)c1)C1CC1 C1(N(C(CSCC)=O)C)CCCN(C(=O)CN2CCCCC2)CC1 N1(C(CCNC(=O)CO)=O)CC(COC(=O)C(F)(F)F)C(c2cn[nH]c2)C1 N1(C(CC=CC=C)=O)CCC(C(C)C(=O)NCCS(C)(=O)=O)CC1 C#Cc1cccc(C(=O)NC2CN(C(c3cnns3)=O)CC2O)c1F c1(CC(=O)NCC(CC)(C)NC(c2ccc(C(F)F)cc2)=O)ccc(Cl)nc1 c1(C(N2CC(n3cc(-c4cncc(C)c4)nn3)OCC2)=O)nc(C)ncc1Br CC(C)CCC(F)C(=O)N1CC(CNC(=O)C=Cc2cscn2)OC(C)(C)C1 c1(CCNC(N(CCOCC=C)C)=O)cnn(C)c1 CC1OCCC1CC(=O)NCCn1cc(CNC(C2CC23CCC3)=O)nn1 C(=O)(C(C)C(F)(F)F)NCC(c1cccc(C)c1)NC(=O)CCCCCF C1(C(=O)NC(c2c(C)cccn2)c2ccccc2)(N(C)C)CCCCCC1 C1(NC(C2CSCCN2C(=O)CCCC2CC2)=O)CC12CC(O)C2 C(CN=C(NC1CCOCC1)NC1CCNC(=O)C1)N1CCC(C)CC1 CCC(CC(=O)CNC(=O)CC1CCN1C(=O)OC)NC(=O)C(C)SC(F)(F)F C=CC1OCCC1C(=O)NCCCCCCN(C(=O)C(F)C1CCC1)C CC1C(C(=O)NC2CC(CNC(=O)COCC(C)(C)C)C2)C(O)C(=O)N1C N1(C(CCC(C)(C)F)=O)CCC2(COC(CNC(=O)CCCCCF)C2)C1 N1(C(CC(C(C)C)C)=O)CC(NC(c2ccc(CO)cc2F)=O)CC(C)(C)C1 N1(C(C(CC=C)N(C)C)=O)CCOCC(CNC(c2ccnn2C(F)F)=O)C1 c1(CN(CCCNC(C(C)O)=O)C(c2ccoc2C(F)(F)F)=O)cccnc1 C1(CC=C)(NC(c2cncc(N)n2)=O)CCCN(C(c2ncc(C(F)F)s2)=O)C1 N1(C(C2COCCN(C(C3CCN(CC)CC3)=O)C2)=O)CC2CCN(C)CC2C1 N1(C(CC2(C)CC(F)(F)C2)=O)CCC(NC(=O)CC2CCC2)CC1C1CC1 Cc1cc(C(=O)NC23CC(C2)N(C(=O)Cc2cncnc2)C3)cn(C)c1=O Cc1ccc(C(N2CC3CC3(CNC(c3cccc(O)n3)=O)C2)=O)c(O)n1 c1(C(=O)NCC2(F)CC(NC(CCOCCOC)=O)C2)ccc(Cl)cc1C C(CC(C)CC)(C(=O)N(C1(CCO)CC1)C)NC(C(CC#C)O)=O C1(CNC(CN(CCC#C)C)=O)CCCCN1C(=O)CC(C)N1CCCC1=O C1(CC(=O)NC2CC(F)C2)CC2(CC2)CN1C(=O)Cc1ccco1 C1(CNC(Cc2scc(C)n2)=O)CC(NC(=O)CCS(C)(=O)=O)C1(C)C c1(NCC2(OC)CN(C(c3cnc(Cl)s3)=O)C2)[nH]c(=O)n(C)c(=O)c1C#N c1(C(N(CCN(C(=O)CNC(N2CCCC2)=O)C(C)C)C)=O)cc(C2CC2)sn1 CC1(CNC(=O)OC(=O)C(Cc2cccc(Cl)c2)=NO)CS(=O)(=O)C1 c1(C(=O)NCC(CNC(=O)Cc2cc(C3CC3)nn2C)OC)noc(C)c1SC N1(C(c2cccc(OCC)c2)=O)CC2CC(NC(C3(C(=O)NC)CC3)=O)CC2C1 c1(C(N2CC(C(C)NC(c3c(CC)scc3)=O)C2)=O)ccc(Cl)c(F)c1N c1(C(=O)NC(C2CCN(C(CCS(C)=O)=O)C2)(C)C)cc(S(C)(=O)=O)co1 CN1CCC(C(=O)N(CCCNC(=O)C(C)(C)C2CCC2)C2CC2)C1=O N1(C(C2CCC(CNC(Cc3c(C)ccs3)=O)C2)=O)CCCC(C)C1 C1(C(N2CC(OC)(CNC(=O)CN(C3CCCC3)C)C2)=O)C(Cl)(Cl)C12CC2 C1(O)(CCNC(=O)C2=CCSC2)CCCN(C(=O)C(F)C2CCCC2)C1 C1(C(=O)NCc2n(CC)ccn2)CCN(C(C23CCC(CC2)C3)=O)CCO1 c1(N2C(CCC=C)CCC2)nc(N(C)C[Si](C)(C)C)nc2ccc(OC)cc12 Cc1cc(F)ccc1CNC(=O)C#CCNC(c1cc2n(n1)CCC2)=O N1(C(CC=CC=C)=O)Cc2ccccc2C(NC(=O)CN2CCC(F)(F)C2)C1 C(=O)(C1CCc2c[nH]nc21)NC(C1CN(C(=O)CCOCCN(C)C)CCO1)C N1(C(C2C(C)(C)C2NC(C2CCC(C3CC3)C2)=O)=O)CC2(C)COCC2(C)C1 C1(NC(=O)Nc2cccc(OCCOC)c2)CCCCCCC1OC c1(OC)ccc(CNC(=O)C(C(C)C)NC(c2ccc(C)o2)=O)cc1 c1(CC)nccnc1NC(c1cc(NC(c2cc(C)nn2C)=O)cn1C)=O CCC1=C(C(=O)NCC(C)(CO)NC(c2cc(COC)cn2C)=O)SCCO1 C1(C(=O)NCC2CC(NC(C3(C=C)CC3)=O)C2)CCC2C1C2(F)F N1(C(C2CCC(=O)N2)=O)CC(NC(c2cnc(C(F)(F)F)nc2)=O)CC(F)(F)C1 C1(NC(c2c(OC)nccc2)=O)CC2CCC1CN(C(=O)Cn1[nH]cnc1=N)C2 CC1OC2(C(N3CCC(CN(C)C(C4OCC5CCCC45)=O)C3)=O)CCC1CC2 CC(=O)CCCC(=O)NCC(C)(C)CC(=O)NCC12CCCCC1C2 c1(NC(COCC(=O)N(C)C)=O)cccc(C(=O)NC2CNC(=O)C2)c1 CCC(CC)C(F)C(=O)N1CCCC(N(C(c2[nH]cnc2C)=O)CC2CC2)C1 N1(C(c2cnc(C)nc2)=O)CCCC(CNC(=O)C(C)Cc2cnc[nH]2)CC1 c1(C(=O)NC(C)(CNC(=O)CCCC(F)F)C2CC2)cc(O)nc2ccccc12 Cn1ncc2c(NCCC=CBr)[nH]c(=NCC3CCOCC34CCCC4)nc12 N1(C(=O)C=CC(=O)OC)C(C(=O)NOCC(F)F)CC1C.C1(C)CC(=O)N1 c1(N(C(=O)CCCC2CC2)C2(CNC(C(C)NC(N)=O)=O)CCC2)ccc(F)cc1 C=CC(CCC)CC(=O)NC1(C2CCCN2C(c2oc(CO)cc2C)=O)CC1 C1(C(=O)Nc2cncc(OC)c2)CC12CCN(C(=O)C(C)N1CCCC1)CC2 C1(C)(CNC(CCN(C(C(C)NC(C)=O)=O)CCO)=O)CC2CCC1C2 Cc1cccc(OCC(=O)NCC2CC3(CC3)CN2C(C2CCCSS2)=O)c1C C1(C(=O)NC(CCCNC(c2c(C)c[nH]c2)=O)C)CC12CC(OC(C)(C)C)C2 Cc1nscc1CC(=O)N(CC(O)CNC(c1c[nH]nc1C(F)(F)F)=O)C C(=O)(C1CCc2nccn21)NC1C(CNC(c2ccc(C)c(C#N)c2)=O)C1 c1(Cn2ccnc2-c2ccccc2-c2cnc(SCC)cn2)cc(O)cc(O)c1 C(=O)(CC(CN(C)C)CC)NC1CN(C(C2CC(CCC)C2)=O)C(C)C1 n1(CCC)ccnc1C(c1nnnn1CCC)NCCC(=O)NC(N)=O c1(C(=O)NC2C(F)CCN(C(CC3CCC(C)(C)C3)=O)C2)cc2n(n1)CCCO2 c1(CCC)cc(C(=O)NC2CC(C)N(C(=O)Cc3ccnc(OC)c3)C2)ccn1 C1(NC(CCc2c(C)noc2C)=O)CS(=O)(=O)CC1NC(c1cn(C)cc1C)=O N1(C(CC#C)=O)CC2CN(C(=O)CNS(=O)(=O)CCCC)CC2C1 C1(CNC(c2cnc(C)nc2C2CC2)=O)CCC(C)(C)CN1C(C1CC1(Cl)Cl)=O C1(C(=O)NCCCNC(C)=O)(NC(=O)CC2CN(C)CC2O)CCCCC1 CC(C)CCC(O)C(=O)N1CCOCC1CNC(=O)Cn1ccnc1C(C)C CC1(C(N2CC(F)(CNC(C3CC(n4ccnn4)C3)=O)C2)=O)CC2CC2C1 c1(CC(=O)NC(CCNC(C(C)(C2(C)CC2)OC)=O)C)c(C)noc1C n1(CCOC)c(N2CCCC(C)C2)nnc1Cn1ccnc1C C(CC(C)C)(C(=O)NCC(O)CCOC)N(C(COCCCC)=O)C CC(CC(F)(F)F)C(=O)NC1CC(C(F)F)(NC(=O)CCc2nncs2)C1 c1(C(N2CCCN(C(C(C(C)C)OC)=O)CC2)=O)cc(C)cc(Cl)c1N C1(NC(=O)CC2CCS(=O)(=O)C2)CN(C(C23CSC(C2)C3)=O)CC1C1CC1 c1(NC(Cn2cc(C(CC)(O)CC)nn2)=O)ccc2c(c1)CCO2 c1(C2CC(C(=O)NCC(CNC(Cc3c(C)ccs3)=O)C)C2)cccc(F)c1 c1(C(=O)NC2CCC(CCNC(C(C)(F)F)=O)C2)nncc2ccccc12 c1(C(c2nnnn2-c2ccccc2)NCCNC(COC)=O)csc(C(F)F)c1 CC(C)(O)C#Cc1ccc(C(C(=O)O)NC(C2CC3(CNC3)C2)=O)cc1 C1(COC)CN(C(C2CC(F)C(=O)N2)=O)CCN1C(=O)C(=O)N(C)C c1(C(=O)NCCCCN(C(C(CC2CCC2)OC)=O)C)ccc2nccn2c1 C1(NC(C2(NC(C)C)CC2)=O)CC2CCCC(C1)N2C(C1CC(C)C1)=O c1(OC)nc(C(N2CC(CC(=O)Nc3ccc(I)c(C)c3)C2)=O)ccc1Br c1(C(N2CCC(NC(C(CCC)C)=O)C(F)C2)=O)ccc(F)c(C#N)c1 c1(Sc2nc(SC)[nH]n2)cccc2c1sc1ccccc21 C(CCCC(=O)N(C1CCN(C(c2cncnc2C(C)(C)C)=O)C1)C)SC c1(C(=O)NC(Cn2cc(C(=C)C)nn2)C)cc2cc(Cl)ccc2n1C N1(C(C(CC)OCC)=O)CC=C(CNC(c2c(Br)nnn2C)=O)CC1 N1(Cc2ncc(C)nc2)CCN(c2ncc(C(F)(F)F)cn2)CC1C N(C(=NCCCF)NCC(C)(O)CC)C(C#C)CCC Cc1c(F)ccc(NC(C2CSC(=O)N2)=O)c1F C1(CC(N2CCC(N(CC)NC(=O)CC3(SC)CC3)C2)=O)CCCC12CC2 c1(C(=O)NCC2CC(F)(CNC(C3C(C#N)C3)=O)C2)ccc2snnc2c1 c1(OC)cncc(C(N2CCC(NC(=O)C3=CC(C)(C)C3)C2C(C)C)=O)c1C C1(C(=O)NC(c2cccc(C)c2C)C(=O)OC)CCC2OCCC2N1 C1(C(=O)NC2CC(CCF)C2)CC12CCN(C(=O)C(F)C(F)(F)F)CC2 C(=O)(CCS(C)=O)N(C(C)CNC(=O)CCN1CCC1)CC C(=O)(C(C)(F)C(F)(F)F)NC1C(C)CN(C(=O)CCn2cccnc2=O)C1 N1(C(c2cc(C(=O)OCC)co2)C(=O)NCC(=C)C)CC(=O)NCC1C(=O)OC C(C(O)CN(C)C(C1CCCC1)=O)N(C(=O)CCNC(c1cccs1)=O)C CCC(C)C(C(=O)NCC(=O)Nc1ccc(CCO)nc1)N(C)C C(=O)(CS(C)(=O)=O)N(C(CC)C(=O)NCc1coc(C)n1)C c1(-c2cc(C)no2)ccc(S(=O)(=O)NCc2cnc3occc3c2)s1 C(=O)(C(O)CCC(C)C)N1C(C(=O)NCc2ccc(CC)s2)CN(C)CC1 C(=O)(C1=C(CCl)N(CC2CCCO2)C(=O)NC1c1ccc2cc[nH]c2c1)OCC C1(F)(CNC(Cc2scc(C)c2)=O)CCCN(C(=O)C(N2CCCC(O)C2)C)C1 c1(C(N2C(CNC(c3c(C)cc(=N)[nH]c3)=O)CC2)=O)cc(C)c(Br)c(C)c1 C(C)(CC(C)CC)N(C(C1(NC(COCCCC)=O)CCCC1)=O)C N1(C(c2ccc(CC)cn2)=O)CCN(C(c2ccc(F)c(C)c2)=O)CC1CC c1(CC)cn2c(n1)CCC(C(N1CCN(c3ccc(F)cn3)CC1C)=O)C2 C1(NC(C2N(C(C(c3cncnc3)C)=O)CCC2)=O)CN(C)CC1C C1(N(C(c2c(C)con2)=O)C)CCCN(C(=O)C=Cc2cn[nH]c2)C1 c1(CC)nn(C)c(N2CCN(C(=O)COCC(F)F)CC2CC)c1[N+](=O)[O-] c1(OC)cc(Cl)ccc1C(=O)NC(C)CCN(C(=O)CCCOC(C)(C)C)C c1(C(N2CC(CNC(C(CC=C)CC)=O)C2)=O)cc(Br)c(OC)cc1C c1(C(=O)NC(C2CCN(C(c3ccnn3C3CCC3)=O)C2)C)cc(=O)cc(Cl)[nH]1 N1(C(C(C)(O)C2CC2)=O)CC2=C(C1)CN(C(C1(c3ccc(Cl)c(F)c3)CC1)=O)C2 C(=O)(C(O)C(C)(C)C)NCC(CC(C)C)NC(=O)CC1C(C)(C)C1(C)C C(=O)(CC(C)CC(C)C)N1CC(CCC)C(C(=O)NCC2(C)CC3C=CC2C3)C1 CC1CCC(OCCNC(=O)CC2C=CC(NC(=O)Cc3ccoc3)C2)CC1 N1(C(C=CCCCCC)=O)CCCN(Cc2ccc(Br)c(Cl)c2)CC1C Cc1coc(C=CC(=O)NC2CN(C(=O)CCC(C)N(C)C)C2)n1 c1(C(=O)OCCC2CC2)c(F)ccc(S(=O)(=O)CC2CC2)c1F C1(C(=O)NCC2(NC(=O)CCn3cc(C)cn3)CCCCC2)(OC)CS(=O)(=O)C1 c1(NC(=O)C(F)OC(F)(F)F)c(C)csc1Cl.CCCN1CC1 c1(COc2cccc(C(=O)NC(c3cn(CC)nn3)CC)c2)ccc(F)cc1 CON(CCC(=O)NCC1CCOCC1C)C(=O)CC(C)(F)F CCCCC(O)C(=O)N1CC2CC1C2C(=O)Nc1cncc(Cl)c1 N1(C(Cc2cc(C)ns2)=O)CC(NC(c2cccc3ccnn23)=O)CC(C)(C)C1 N1(C(c2cc(C)c(F)cc2)=O)CCC2(NC(c3cscn3)=O)CCCC12 C1(C(=O)NCC(C2CCCC2)C)CN(C(=O)Cn2c(O)nnc2O)CCN1C C1(C(N(C2(CC(=O)N(CC(C(C)C)C)C)CC2)C)=O)CCOC(=O)CC1 C1(NC(COC)=O)CN(C(=O)C=C2CC2)CC1OC c1(CC(=O)N(C)CC2COCCN2C(=O)COC2COC2)csc2ccccc12 c1(C(=O)NCC(CC(F)(F)F)NC(COCC)=O)nn(C)c2ccccc2c1=O C=CC1(CC(=O)N(C2CN(C(=O)Cc3cnccn3)CC2F)C)CCOCC1 C1(O)(c2onc(CC)n2)CCCN(N2CCN3CC(O)C23)CC1 c1(C(N(C2CCOC2)CCNC(COCC(C)C)=O)=O)ccncc1F N12CCN(CC1)C(=O)Cc1cccc(c1)OC(C)C2.C(=O)(C(C)(C)F)C1CC1 CC1OC2CCC1(NC(C1CC(NC(c3cccs3)=O)C1)=O)C2 CCCCC(CCCC)NC(C1CC2(CC2)C12CCC2)=O CCC(C)(O)C(=O)N1CCCC(NC(c2cn(C)c(C)n2)=O)C1 CC1CCC=C1C(=O)N(C)CC1CCCCN1C(c1cnc(CC(C)(C)C)o1)=O c1(CC(=O)NC2C(NC(C3(C)CCC3)=O)C2)csc2nc(-c3cccs3)cn12 C(=O)(C1c2ccccc2CN1C(c1cccnn1)=O)Nc1cnc(OCC)nc1 Cc1cc(N)c(F)c(C(=O)N(C)CCN(C)C(c2ncsc2C2CC2)=O)c1F N1(C(COCC(=O)NC)=O)CC(C(N)=O)(CNC(C2CC2(C)C(C)C)=O)C1 c1(C(=O)NCC2C(C)(C)C2C(=O)NC2CC2(C)C)ncnc(O)c1F C1(C2CCN(C(C3(Cl)CC3(F)F)=O)CC2)(NC(C2=C(C)S(=O)(=O)CC2)=O)CC1 c1(C(=O)NC2CCCCN(C(CS(C)(=O)=O)=O)C2)ccc2c(c1)CCC2=O CCC(C)C(O)C(C)C(=O)NCC12CCCC(CN(C(=O)CCCN=[N+]=[N-])C1)C2 C1(COC)(CNC(c2ccns2)=O)CCN(C(c2ccc(CCO)cc2)=O)CC1 n1(CC(=O)NCC2CCC(NC(=O)CC3CCOC3)C2)ccc(Br)cc1=O N1(C(=O)OC(C)(C)C)CC(C2CC2)C(F)(c2nc(Cn3cccn3)no2)C1 Cc1ccc2cc(C(=O)N(C(CNC(=O)CN=S(C)(C)=O)C3CC3)C)cn2c1 N1(C(c2ccc(CNC(c3n(C)c(Cl)nc3)=O)nc2)=O)CCC2(CCC2)C1 c1(C(COC(CC)(C)C)=O)cc(F)ccc1OC(C)C(=O)OC C#CCCCCCC(=O)NCC(C(=O)NCCCC(C)(C)CO)OC N1(C(=O)OC(C)(C)C)C(C(=O)NCCC(O)C(F)(F)F)CC2CCCCC12 c1(CNC(C(C)(C)NC(C2C(C)C2C)=O)=O)cncc(F)c1 Cc1cc(Cl)nc(Cl)c1NC(C1CC1C(=O)Nc1ccc2nncn2c1)=O C1(CNC(COCCOCC)=O)CN(C(c2cnc(CC)nc2O)=O)C(C)(C)C1 N1(Cc2c(C)nc[nH]2)CCCC(N(C(=O)Cc2ccccc2F)C)CC1 n1(CCC(=O)NCCN(C(=O)C(C)C(C)(C)C)C(C)C)cnc2sccc2c1=O c1(C(N(CCC)CCNC(c2cn(C)c(O)n2)=O)=O)cc(Cl)c(OC)c(Cl)c1 CON(C)CCCNC(C1(CNC(c2nnsc2C)=O)CC2(CC2)C1)=O C1(C2(C(N3CCC(C)C3)=O)CCC2)CCCCN1C(=O)CN1CCCCCC1 C1(N(C(c2ccn(CCC)n2)=O)C)CN(C(=O)CC2CCN(C)C2)CC12CC2 c1(OC)ccc(C(=O)NC2(C)CCN(C(C3(S(N)(=O)=O)CC3)=O)C2)c(OC)c1 CCCC(C(=O)N(CC)CC1CCCC1)NC(c1cn(C)nn1)=O c1(C(N2C(C)CC(NC(c3cc(C(C)=O)oc3C)=O)C2)=O)cnc2occc2c1 c1(OC)ccc(CC(=O)NCCCCCN(C(=O)CSCC(C)C)C)c(OC)c1 Cc1ccc(C(=O)N(C)CCN2CCN(C(C3CC3(Cl)Cl)=O)CC2)c2c1CCC2 c1(CC)nccn1C(C)CC(=O)N1CCC(NC(=O)COc2ccon2)C1 c1(OC)nccc2cc(NC(=O)Nc3nnc4n(c3=O)CCCC4)ccc12 N1(C(C(C=C)c2ccccc2)=O)C2CCC1C1CC1(NC(=O)CCSCCC)C2 n1(CC)nnc(C(=O)NCC2CCN(C(=O)CC3CC34CC4)C2)c1C C1(NC(C2(NC(C)(C)C)CC2)=O)CN(C(=O)CN(CCCC)CC)CCC1F C1(C(N(C)CC2C(C)OCC2)=O)CN(C)CCN1C(C1CN2CCC1CC2)=O N1(C(c2c(C)noc2)=O)CCCC(O)(CNC(C2CC2C2CC2)=O)CC1 C(CCCCCS(=O)(=O)CCO)n1cc(CC2C(C)N3CCC2CC3)nn1 C(=O)(C1=COCCC1)NCCn1ccc(C(N2CC(C(CC)CC)C2)=O)c1 c1(OC)ccc(C(CNC(C2CC=CCC2)=O)NC(=O)Cc2cnoc2)cc1 N1(C(C2(CC)CCOC2)=O)CCCN(C(=O)CCn2cc(Cl)cn2)C(C)C1 c1(C(N2CCN(CC)CC2)C(=O)NCCOCC)cn(C)nc1Br CCC(C(=O)NC(C)(CNC(c1cccc(C(=O)OC)n1)=O)C1CC1)C(C)O Cc1nc(-c2ccsc2)sc1C(=O)N(C)CCN(C(C1CCCN1C)=O)C(C)C C(C(C)(C(=O)N(C)CC1(CO)CC1)NC(=O)CC1CCOC1(C)C)SC c1(OCC)cccc(CN2CCC(N(C(=O)COC(C3CS(=O)(=O)C3)=O)C)C2)c1 C(=O)(CCCN1CCCCC1)NCCN(CCOC)C(c1coc(Br)n1)=O C12(CNC(CC#N)=O)CCC(NC(c3cc(CCO)on3)=O)(CC1)CO2 N#Cc1ccc(N)c(C(=O)NC2CCCC(NC(c3cccc(F)c3)=O)C2)c1 c1(C(N2CCC(OCCNC(C=C(C)C(F)F)=O)CC2)=O)ccc2c(c1)CCN2 c1(C(=O)NC(C)CCCNC(=O)CC(c2ccccc2F)C)n[nH]c2c1COC2 CN1C(=O)c2ccccc2C1CC(=O)NC1C2CC1CN(C(=O)CS(C)(=O)=O)C2 C(=O)(C1=CC2CCCCCCC12)N(CC(=O)NCC1CCOC1)C1CC1 N1(C(CCC(C)C)=O)CCCC(NC(C2CCN(c3ncccn3)C2)=O)CC1 C1(C(=O)NCC2(O)CCN(C(CC3(COC)CC3)=O)C2)CC(C)(C)OC(C)(C)C1 CC(C)C1=NOC(C(N2CCN(C(C3CC(O)C3)=O)C(c3ccccn3)C2)=O)C1 c1(C(=O)NCC2(COC)CN(C(=O)CCC(=O)C3CC3)C2)cc(Cl)c(F)cc1F C(N=c1ccc([N+](=O)[O-])c(O)[nH]1)c1nc(C)sc1 N1(C(c2cccc(O)n2)=O)CCOCC2(COCCN2C(=O)CCCCCF)C1 C1(CC=C)(C(=O)NCc2cn(CC)nn2)CCCN1C(=O)Cc1cc(C)nn1C C1(C(=O)NOCC(O)CO)N(C(c2cc3n(n2)CCO3)=O)CC12CCCC2 c1(CC(CNC(c2ccns2)=O)N(C)C(C2(C(F)F)CCC2)=O)ccccc1 C(C(C)(C)CNC(=O)C(c1cncnc1)C)NC(C(=O)NCCOCCOC)=O C1(CN(C(Cn2ncc(C)c2)=O)C)CCCCN1C(=O)C(C1CCC(=O)N1)C Cc1nn(C)c(C)c1C(C)C(=O)N(CCN(c1nccnc1F)C)C(C)C c1(NC(C2COCCN(C(C3(Br)CCC3)=O)C2)=O)ccc(Cl)c(C(F)(F)F)c1 C1(NC(CSCCC)=O)CN(C(c2scnc2C(F)F)=O)CC1OC C1(NC(C(C)C2CCC2)=O)CCC12CCN(C(=O)CCc1ccc(O)nn1)CC2 N#Cc1ccccc1NC1(NC2CCC(C3CCN(C4CCC4)C3=O)C2)CC1 CON1CCC(C(=O)NCCOC2CCN(C(c3cnc(C)c(N)c3)=O)C2)CC1 c1(C(=O)NCC2CC(NC(=O)Cn3ncnn3)CC2O)coc2c1COC2 N1(C(C)=O)CCCC(C(N2CC(CCCCNC(=O)C(C)(C)CF)C2)=O)C1 CC1(C)C=C(C(=O)NCC2COCCN(C(C3CCCC3O)=O)C2)C1 C(=O)(C(C)(O)C(F)(F)F)N(CCC(C)NC(c1c(C(C)C)nns1)=O)C CC1CCCN(C(=O)CN(C)C2CC2)C1CCNC(=O)Cc1ccnc(OC)c1 C#CCC(CC(=O)Nc1cncc(C2CC2)c1)NC(c1cnn[nH]1)=O C12(CNC(C3C(NC(=O)COC4CCOCC4)CCOC3)=O)CCC(F)(CC1)C2 Cc1ccccc1C=CC(=O)NC(C)(CNC(=O)CCc1cnccn1)C1CC1 CC(C)(C)C#CC(=O)NCCC1CCCCN1C(c1ncc(Cl)nc1Cl)=O C(C1CCCCC1)=CC(N1CC(C(N2CC(CO)C2)=O)(CC)C1)=O C1(c2cn(CC3C=CCN(CCc4nc(SC)oc4)C3)nn2)CCC(C)=CC1C c1(C(=O)NC2CN(C(C(CC)C)=O)CC2C#N)cc(OC)c(O)c(C(C)(C)C)c1 C(=O)(CC(F)(F)CC(=O)N1CCCC1C1CCN(C(c2ccc(F)o2)=O)C1)OC c1(C(=O)NCCOCCNC(c2cc(C)no2)=O)cc(N)ccc1Cl N1(C(C2C=CCC2)=O)CCC2OCCN(Cc3cc(C(F)(F)F)cc(F)c3)C2C1 C1(N(C(Cn2ccc(C)n2)=O)C)CN(C(=O)CCN2CCC(O)CC2)CC12CC2 N1(C(C=CCC)=O)CCC(NC(c2ncccc2N(C)C)=O)C(CO)C1 Cc1cccc(C2(C(=O)NC(C3CCN(C(c4c(Br)cnn4C)=O)C3)C)CC2)c1 Cc1cccc(N(CCC#N)C(C2CCC2)=O)c1C.c1(N)sc(Br)nc1C C1(NC(C2ON=C(C)C2)=O)CC2(CCCN(C(=O)Cn3cncn3)C2)C1 Cc1ncc(CC(=O)N(CCN(C(=O)CCc2nncn2C)C)C(C)C)[nH]1 C1(N(CC(=O)OCCCN(S(C)(=O)=O)C)C)CCC1F C(=O)(C1=NOC(CNC(C2CN(C3CCC3)C2)=O)C1)N1CC(CSC)C1 C(=O)(C(CNC(=O)C#CC1CCC1)C(C)(C)C)N(CCC#C)CC C1(CC)CCCCC1OCC(=O)N(CCNC(=O)C(C)(C)O)C(C)C C(C)(C)(C(=O)NCCN(C(C1CC(C)C1)=O)CC1CC1)OCCC N1(C(COCCCCCC)=O)CCCC(N(C(=O)C(C(C)C)SC)CCO)C1 C1(CNC(C(=O)NCc2nc(-c3ccc(F)s3)no2)=O)CCS(=O)(=O)C1 Cc1c(C(=O)NC(CO)C(=O)NCc2noc(C(N)=O)n2)cccc1O C1(C(N2CC(C(C)NC(C(CC=C)CC)=O)C2)=O)CN(C)CCN(C)C1 C(=O)(C(O)C1=CCCCC1)NC1CC(OCC(N2CC[Si](C)(C)CC2)=O)C1 C=C(C)CC(C)C(=O)N1CC(NC(=O)C=CSCc2ccco2)C(C)C1 C(C(CC(F)(F)F)NC(=O)Cc1ccns1)NC(CCc1nnc(C)n1C)=O c1(C(N2CC(C(C(=O)NC(c3ccoc3)C)O)C2)=O)cc(CCO)on1 N1(C(C=CC=CC)=O)CCC(NC(c2coc(CSC3CC3)n2)=O)CC1C C12(CC(=O)N(CCCC=C)CC)CCC1CN(C(c1cccnc1S)=O)C2 c1(C(N2CCC3(NC(C(C4CCCCC4)C)=O)C(C2)C3)=O)c(O)cc(F)cc1F C(C)(C(C)C(=O)NC(C)Cc1cn[nH]c1)NC(C1(CCOC)CCC1)=O C(=O)(C(CC1CCCCC1)C(C)C)N(CCNC(C(OC)OC)=O)C Cc1nc(C(=O)NCC(C2CC2)NC(=O)C(C)n2cncn2)c2ccccn12 Cc1cc(C(N2CC(O)(CNC(=O)C(CO)c3ccccc3)C2)=O)nn1CCO N1(C(Cc2cn(C)nn2)=O)CCC(CCNC(C2CC(=C3CC3)C2)=O)CC1 CC(C)(CCNC(=O)C(F)C1CCOC1)C(=O)NCC=C(Cl)Cl c1(N2CCC(N(C(=O)CCn3cccn3)CCC)C2)nc2ccccc2s1 C1(C(N(C(C(C)SC)C)C)=O)(NC(=O)C(C)NC(=O)C2CC2)CCOCC1 C1(C(=O)NC(CCCCNC(CCC2C(C)=NOC2=O)=O)C)COC2COCC12 C(CCOc1ccccc1)(C(=O)O)NC(CN(C1CCC1)C(C)=O)=O.OCN C1(C(=O)NCC2C=CCC2)CC(O)(CNC(C2(CCF)CCC2)=O)C1 C#CC1CN(C(c2cc(C)c(C)nn2)=O)CCN1C(c1ccc2nc[nH]c2n1)=O c1(NC(C2C(O)CCN2C(c2c(Br)cccc2Br)=O)=O)nc(Br)ccc1Br c1(SCC(c2cccs2)=O)cnc2n1CC(CO)CC2.N12CC3(CC3)CC1C2=O c1(CNC(C=CC(CC)C)=O)cn(C2CCN(C(C3COC3)=O)C2)nn1 N1(C(c2cccc(C)c2Cl)=O)CC2CCOC2(CNC(c2c(C)noc2N)=O)C1 C(C(O)CNC(CN(C(=O)C(O)c1ccsc1)CCOC)=O)NS(N)(=O)=O C1(COC)(NC(C2CC2C2CCCO2)=O)CN(C(c2oncc2COC)=O)C1 Cc1c(O)cc(C(N2CCC(NC(C3(c4ccccc4)CC3)=O)C2)=O)cc1O CC(C)CC(CNC(=O)CC=C(Cl)Cl)C(=O)NCC1(n2cccn2)CC1 C1(C(N(CCC(C(C)C)N(C)C)C)=O)CCC(C2CCC2)CC1.C12(CC1)C(=O)N2 N1(CC2N(C3CC=CC3)CC2)CCc2cccc(Cl)c2C1 N1(C(CCCOC(C)=O)=O)CCC(CN(C(=O)CC2CCOC2C)C2CC2)CC1 CC(=O)CCCCC(=O)NC1(C(=O)NC2CCN(C)CC2)CCSC1 Cc1cccc(CNC(C2CC3CC3N2C(=O)C=CC2CCOC2)=O)c1O C(=O)(CCCC1CCC1)NCC(C)CNC(=O)COCC1CCCO1 c1(OC)ccc(CNC2C3CN(C(c4cc(C)cc(Cl)c4)=O)CC23)c(Cl)c1 C1(C(=O)NCc2cccc(C)c2)CN(C(c2cc(C)no2)=O)CC1(C)C Cc1c(C(=O)N(CCC(C)NC(=O)C(O)C2CC2)C)sc(Cl)c1Cl S(=O)(=O)(c1cc(C(=O)NCC(CO)NC(C2(OC)CCC2)=O)c(C)o1)NC C=CCC(CC)C(=O)NC(C1(C(=O)NC(C)C(C)(C)CO)CC1)C c1(C(N2C(C3N(C(C(n4c(C)ncc4)C)=O)CCCC3)C2)=O)ncc(F)cc1N C1(C(=O)NCC2CCCN(C(c3nc(C)oc3)=O)C2)CCC2C(C1)C2(F)F Cc1ccc2ncn(CC(=O)NCC3CCC(C)N(C(=O)CC4CCC4)C3)c2c1 c1(CCC(=O)NCC2CC(NC(=O)CCn3ccnc3)C2)csc(Br)c1 c1(OC)cc(C)c(C(=O)NC2CN(C(c3c(C)noc3N)=O)CCC2C)c(C)c1 c1(C(=O)NCCCN(C(c2c(OC)ccnc2)=O)C2CC2)cnc2[nH]ccc2n1 c1(NC(c2n[nH]c(CNC3CCC3)n2)=O)ccc(N2CCNCC2)c([N+](=O)[O-])c1 C1(COC)(NC(c2nc(C3CC3)cs2)=O)CCN(C(c2cnsn2)=O)CC1 C(=O)(C(C#N)C(C)C)NC(CCOCC)C(=O)NCCCC1(C)CC1 C1(NC(C=CC2CCN(C(Cc3nc(C)oc3)=O)CC2)=O)CCn2cncc2C1 N1(S(c2ccc(OCC)cc2)(=O)=O)Cc2cc(Br)ccc2CC1C c1(OCC)c(CNC(=O)NC(c2cccc(C(F)(F)F)c2)CCO)ncnc1Cl c1(C(N(CC(CC)NC(c2nccn2CC)=O)C)=O)cc(CO)ccn1 C1(CN(C(C(C)=CC)=O)CC)CCCN1C(=O)C(CC)NC(=O)CC C1(CNC(C(CNC(c2n(CC#C)cnn2)=O)CC2CC2)=O)OC(=O)CC1(C)C C1(NC(=O)COC2COC2)CCC(NC(=O)CC2CCCO2)CC1 c1(SC)ncc(Br)c(N2CC3C(C(=O)Nc4ncc(Br)s4)C3C2)n1 Cc1n[nH]c(C)c1CC(C)C(=O)N(CCCN(C)C(c1cnc(Cl)n1C)=O)C C1(C(N(CCC=C)CC)=O)CC2CC1CC2NC(C1CC1(F)F)=O N1(C(c2cc(CN3CCCC3)c(Cl)cc2)=O)CC2CC(COC)C2C1 N1(CC)CC(NC(=O)Nc2cccc(Cn3cc(C)cn3)c2)CC1=O C1(C(C)OC)CCN(C(C23CC2CCN3C(C2CC(SC)C2)=O)=O)CC1 C=CC1OCCCC1C(=O)NC1CC(NC(C2Cc3cscc3C2)=O)C1 C=C(C)C1CN(C(=O)C(C)CN(C)C(C2(c3ccno3)CC2)=O)CCO1 C1(C(=O)NCCN(C(CC)C)C)CC2CC1CC2NC(=O)C#CC(C)(C)C CCC(C(=O)OC)C(=O)N1CC(NC(c2cc3scnc3[nH]2)=O)C(O)C1 c1(OC)nn(C)cc1CNC(=O)CC1CC(C)N(C(=O)CC(Cl)Cl)C1 C(C(O)CC(C)(C)C)N(C(CC1(N(C(=O)Cc2ccnn2C)C)CC1)=O)CCO C(=O)(C#CC1CC(F)(F)C1)N1CCN(C(C=CC=CCCCCC)=O)C(C)C1 c1(CN2CCCC(C(N3CCC(O)(C(F)(F)F)C3)=O)C2)ccc(F)c(Cl)c1 C1(C(=O)NCCCC(C)NC(C=C(C)c2ccco2)=O)CS(=O)(=O)CCO1 C1(CCC(=O)NC2CC(NC(COCCN(C)C)=O)C2)CCN(C)CC1 Cc1cccc(CCC(N2CCC(N(C)C(c3ccoc3)=O)C(C)C2)=O)c1Br CCC(CNC(=O)CCCC#N)(CC)NC(=O)C(=O)NCC1CC1 C1(C)(NC(C2CCC(N(C)C)CC2)=O)CCCN(C(=O)CC2CC2(Cl)Cl)C1 Nc1cccc(F)c1C(=O)NCC1CCCCN1C(=O)Cc1cncnc1O C1(CNC(C)=O)CCC(C(C)NC(C2(N(C)C(C)C)CC2)=O)CC1 N1(C2CCN(C(CCN(CC)CC)=O)C2)CCN(C(C23CCC(CC2)O3)=O)CC1 C(=O)(N=c1[nH][nH]cc1C(F)(F)F)C12C(CN(C(c3cc(Br)ccc3O)=O)C1)C2 O=C(CN=c1cc[nH]cc1)NC1CCN(C(=O)CCCC(F)(F)F)CCC1(F)F c1(OC)ccc(C(N2CC(CNC(c3cncs3)=O)C3CC23)=O)c(F)c1 C12CN(CCS1)C2.N1(C(=O)CN2CCCC2)CCN(Cc2csc(Br)n2)CC1 C12(NC(C3=NNC(=O)C3)=O)CCCC1N(C(C13CCC(C(F)F)(CC1)C3)=O)CC2 n1(CC(=O)NC23CC2CN(C(=O)CCCn2ccnc2)C3)ncc2cccnc12 c1(SC)nc(C)cc(=NCC2(O)CCN(C(=O)CC3CCC(C)C(C)C3)CC2)[nH]1 C1(CC(N2CCOCC(NC(C3(CO)CCCC3)=O)C2)=O)CCC2(CCC2)OC1 C1(O)(CNC(=O)COCC2CCC2)CCCN(C(c2ccc(Cl)o2)=O)CC1 C(=O)(C=C1SCC(=O)N1C)NC1CN(C(C(C)OCCC(C)C)=O)CC12CCC2 C=CCC(COC)N=c1[nH]c(=NCC2(CCO)CN(C)C2)c2ccccc2[nH]1 C#CC(C)(C)C(=O)N1CCOC(C(=O)NCC2(C#N)CC2)C1 CC1CN(C(=O)CC(c2ccc(Cl)cc2)O)CCN1C(c1cc(C2CC2)ns1)=O Cc1c(Br)csc1C(N1CC(O)(CN(C(=O)CNC(=O)C2CC2)C)C1)=O c1(OC)ccsc1C(=O)NCCC1CCN(C(=O)CCSCC(N)=O)C1 C(=O)(C(O)C(C)C)NCC(CCNC(C(CO)OC)=O)OC C12(NC(C3(C(C)C)CN(C(=O)NC45CCC(CC4F)C5)C3)=O)CC1COC2(C)C C(=O)(C(C#N)C(C)(C)C)N1C(CC(=O)NCC2CCC(C)(C)CC2)CCC1 C=CC(C(=O)NCn1ccc(C(=O)N(CC(=O)OC)CC2CC2)c1)OC c1(COC)cc(C(N2CC(CNC(C3(C(F)(F)F)CC3)=O)CC2C)=O)c(C)o1 c1(CC(=O)NCCC(C)N(C)C(c2ncn(C)n2)=O)ccnc(F)c1 C1(C(N(C23CC(C2)C3)CC)=O)COC2(C1)CN(C(c1cccc(C#N)c1)=O)C2 Cc1nn[nH]c1C(=O)N(CCNC(=O)CCC#N)Cc1ccccc1 C(CCC(=O)NCCCOCCC(N1CCCC1CN(C)C)=O)=C(C)C N1(C(c2cc(C)c(Cl)cc2F)=O)CCN(C(=O)Cc2ccco2)C2CCCCC12 c1(C(C(=O)NCCN(CC(C)O)C(C2C(C#C)C2)=O)(F)F)ccc(C)cc1 N1(C(C2CCCN(C(N)=O)C2)=O)CCC2(CC1)CN(C(C1CC3C=CC1C3)=O)C2 C1(C)(CNC(c2ccc(CSC)o2)=O)CN(C(=O)C(C)(CO)NC(C)=O)CC1C C1(OCC(=O)NC(C)CC2CN(C(=O)CSc3nncs3)C2)CCC(F)(F)CC1 N1(CCNC(N2CC(C)SC(C)C2)=O)c2ccccc2N(C)S1(=O)=O Cc1ccnc2sc(C(=O)NCCCN(C)C(C3CC(C)(O)C3)=O)c(C)c12 C(=O)(C1=NOC(C)C1C)NC1CCCC(NC(Cn2c(C)nc(C)n2)=O)C1 c1(NC(C2CC(NCc3cc(Br)cc(I)c3)C2)=O)ccc(I)c(Br)c1 c1(C(N2CCC(N3CCN(CC(=O)N(CC)CC)CC3)C2)=O)cc(=O)n(C)cn1 Cc1cscc1CNC(=O)CC1CCN1C(=O)C(n1nccc1C)C CCC(CCC(=O)N1CCCC1)NC(C1CN2CCN1CC2)=O.C1CC(=O)N1 c1(CC)c(C(=O)NCC(C)N(C)C(C2CC3(CCC3O)C2)=O)sc2ccccc12 c1(CNC(C=CCC)=O)ccc(CNC(C2(C)CCCCO2)=O)c(F)c1 c1(CC(=O)NCC(CC)NC(C2(NC(N)=O)CC2)=O)csc(-c2nc[nH]n2)n1 C1(C(=O)NCCCC(=O)NC(C)(C)CC2CCOC2)CC(O)C(F)C1 n1(CC(=O)NCC(C2CC2)NC(C(C)C#N)=O)ccc2c(=O)n(C)c(=O)n(C)c12 c1(C(N2CC(C)(COC)C2)=O)ccc(NC(c2cccnc2)=O)cc1Cl N1(CCC)CC(N=c2[nH]c(=NC)[nH]c(=NCC3CCCN3C3CCCC3)[nH]2)C1 CC1CCC(C(N2CC(O)(CNC(=O)CCc3ccc(Cl)cc3F)C2)=O)C(=O)N1 c1(CC(C)C)ncc(C(C(=O)NCC2CCOC2)N(C)C(C)C)s1 N1(C(Cc2cn(C)nc2)=O)CCN(C(c2cnccn2)=O)C(c2ccccc2)C1 N1(C(C(C)C2(O)CCC2)=O)CC(C(N2CCC(NC(=O)C3CC3)C2)=O)OC(C)C1 Cc1ccc(C(=O)NCC2CCCN2C(c2occc2C)=O)c(SC2CC2)c1 C1(C)(NC(C2(NC(CCc3cn(C)nc3)=O)CSC2)=O)CS(=O)(=O)C1 C1(C#N)(CCC=C)CCN(C(c2ccccn2)C(=O)NCCCC)CC1 N1(C(C(CN(C)C)O)=O)CCC(O)CC1C(=O)NC1(CO)CC(F)(F)C1 C1(C(=O)NCC2CN(C(c3c(OCC)cc(Cl)cc3)=O)C2)CC1C1CCOCC1 C(=O)(C(C)(C)C(C)C)NC(CC)CNC(C1CCC(C(N)=O)C1)=O N1(C(c2c(CC)csc2)=O)CCC(C(F)F)(CNC(C2CC2C(F)(F)F)=O)C1 N1(C(c2c(CC)ocn2)=O)CC2CC1CN(C(C1CCS(=O)(=O)C1(C)C)=O)C2 c1(CN2C(C(=O)Nc3cnc4sccc4c3)COCC2)c(F)cccc1[N+](=O)[O-] NS(=O)(=O)c1coc(C(N2CC3CCC3(NC(C3CC3F)=O)C2)=O)c1 CCCC(CC)C(=O)NCCCC1CN(C(C23CC4CC2C3C4)=O)CCO1 C1(CNC(Cc2nnc(C)o2)=O)CC2CCC1N2C(=O)CSCC1CCCCO1 C12CN(CCO1)C(=O)CNC2=O.c1(C(C)=O)cnc(CC(C)(C)C)o1 CCC(C)CN=c1nc(N2CCN(CC(=O)N(C)C)CC2)c2c([nH]1)CCC(C)C2 Cn1ccc2c(C(=O)NC(CNC(c3cnn(C4CC4)c3)=O)C3CC3)cccc12 C(=O)(C#CC1(CC)COC1)N1CC(OC)C(NC(c2ccc(O)nc2Cl)=O)C1 c1(C(N(CC(C)O)CCNC(C2CC2F)=O)=O)cc(C(N)=O)cc([N+](=O)[O-])c1 c1(C(N2CCC(N(CCC)C(c3ccc(Cl)s3)=O)C2)=O)ccc2c(c1)NCCC2 C1(NC(C2N(CCC)CCCC2)=O)CC2(CCCCN2C(C2CCC2)=O)C1 C1(CC=C)(C(=O)NC2CCN(C(=O)CN3CC4CC4C3)C2)CCCC1 N1(C(c2cccs2)=O)CCC(C2CCCN2C(c2csc(Cl)n2)=O)C1 Cc1cc(C(=O)NCC(C)(C)CNC(c2nccc(Cl)c2C)=O)nc(C)c1 c1(CC)ccc(C(=O)NC2CCC(C)(NC(=O)CCCC3CCC3)CC2)cc1F C1(C(N(C2CN(C(C3CCCC(OC)C3)=O)C2)C)=O)CC2CCC(C1)N2C CC(CC(F)F)C(=O)NC12CC(CNC(=O)CCC3CCCO3)(C1)C2 c1(C(=O)NCC2CC(OC)C2)cc(C)c(-c2ccc(CO)cc2)cn1 CC1CN2CC(C)C1C2=O.c1(NC(=O)CCc2cncs2)nnnn1C.C1CNC1 N1(C(CC=CC=C)=O)CCCC(N(C)C(c2cc(C(N)=O)ccc2OC)=O)CC1 CC1(C)Cc2ccccc2C(C(=O)N2CC3(C2)OCC(O)C3O)N1 C(=O)(C1=NN(C)C(=O)CC1)N1CCN(C(C(CC)O)=O)C(CC2CC2)C1 c1(C(N(C2CCN(C(C3CNC(=O)C3)=O)C2)CC)=O)csc(C(F)F)c1 CCCC(CNC(C12CSCC1C2)=O)NC(=O)CC1CCCCO1 C=CC1(C(=O)NCCn2cc(C)cn2)CCN(C(=O)C(O)C2CCCC2)CC1 C(=O)(CC1=NNC(=O)C1)N1CCC(NC(Cc2n(C(C)C)ncc2)=O)CC1C c1(C2(C(N3CCC(NC(C=CS(C)=O)=O)C3)=O)CC2)ccc(F)c(Cl)c1 c1(CC(=O)N(C2CN(C(=O)CC3(C)CC3)CC2F)C)cncc(F)c1 CCCC(C(=O)NCCCN(c1ccnc(-c2ccccc2)n1)C(C)C)OCC C1(NC(CNC(C)=O)=O)CCN(C(=O)Cn2ncn(C)c2=O)C(C)C1 CC(CC(=O)NC1CCCCC1C(=O)NCC1(C)CCCC(=O)N1)C(C)(C)C C1(C(N(CCS(C)(=O)=O)C)=O)CCN(C(C2(CCF)CCC2)=O)CCO1 N1(C(C2C(CNC(COC3(C#C)COC3)=O)CCCC2)=O)CCc2c[nH]nc2C1 C1(NC(=O)CC2C=CC(NC(=O)C(O)Cn3cncn3)C2)CNC(=O)OC1 N1(C(CC(C)C)=O)Cc2ccnn2CC(NC(=O)C(F)C(C)(C)O)C1 C1(NC(c2cc(C)ns2)=O)CN(C(c2ncoc2-c2ccon2)=O)CC1C1CC1 C(=O)(CC(C)F)N1CC(C(C(=O)NCCNS(N)(=O)=O)OC)C1 N1(C(c2c(C)con2)=O)CC(C)(C(N2CC3(CCC2CO)CC3)=O)CC1(C)C c1(C(N(C)CC2CCSC2)=O)ccc(CNC(C2OCCC2(C)C)=O)nc1 C(=O)(C1=NOC(C)(C)C1)NCC1N(C(c2cc(C)c(Br)s2)=O)CC2(CC2)C1 N1(C(CCCC)=O)CCN(C(c2nc(C)nn2C)=O)C(c2cccnc2)C1 N1(C(c2ccc(OC)cc2C(F)(F)F)=O)CC(C(=O)O)CC(C)(C)C1 c1(C(=O)NC(CNC(C2C(CCOC)C2)=O)CO)cc(Cl)c(Cl)c(Cl)c1 c1(C(=O)NCC2C(NC(c3n(C)nnc3)=O)C2)csc(Cl)c1Cl CC1(C)C=C(C(=O)N2CC(CNC(=O)CCCC#N)CC2(C)C)C1 N1(C(c2cc(C(C)=O)c(C)o2)=O)CCC(NC(c2n[nH]cc2Cl)=O)C(CO)C1 c1(CNC(C(C)N(C)C)=O)cccc(CNC(C2CCCC(N(C)C)C2)=O)c1 S(=O)(=O)(c1cccc(F)c1)NCC(N1CC(N(C(=O)CC2CC3(COC3)C2)C)C1)=O N1(C(CCOCCC)=O)CCCC2(CCN(C(c3cc(C)n(C(F)F)n3)=O)C2)C1 c1(C(c2n(CC=C)nnn2)NC2CC(Cl)(Cl)C2)ccc(C(N)=O)c([N+](=O)[O-])c1 N1(C(C2(C)CCCOC2)=O)CC2CCC(NC(c3csc(C4CC4)n3)=O)CC2C1 c1(COC)nnc(N(C(C)CNC(=O)CC2CC(F)(F)C2)C)s1 S(=O)(=O)(c1cccnc1NC1CC(=O)N(C2CC2)C1)NCC(CC)O c1(OC)cccc(C(=O)NCC(O)CCNC(C2CC2c2ccn(C)n2)=O)c1C CC(C)C(C)(O)CNC(=O)C(c1cccs1)NC(c1cnnc(O)c1)=O c1(CC)cc(CC(=O)NCC2CC(NC(C3CSCN3C(C)=O)=O)C2)n(C)n1 N1(C(CCC=CC)=O)CCN(C(=O)Cc2c[nH]c3cccnc23)C(C)C1C N1(C(C(C)(C)C2CCCO2)=O)CC2CC2(CNC(c2ccncc2F)=O)C1 CC1(C(=O)NOCC2CCOC2)C=CCN1C(C1CCSCC1)=O C1(NC(C2C(C)(C)CC2)=O)CCC2CC1CN2C(=O)C=Cc1ccc(=N)[nH]c1 C1(N(C)C(c2cnco2)=O)CCCC(NC(c2ccnc(O)c2)=O)C1 c1(C(N2CC(F)CC(NC(C=C(C)c3cccs3)=O)C2)=O)ccc2nncn2c1 c1(C(N2C(CNC(=O)CC3CC=CCC3)CCC2)=O)cc2c(=O)cc[nH]c2s1 C(=O)(C1CCCc2scnc21)NC1C(NC(Cc2c(C)ccs2)=O)CC1 C1(CNC(Cn2cc(-c3onc(C)n3)nc2)=O)COCCN1C(=O)C(C)C CCC(C#N)C(=O)N(CC(C)NC(=O)CCn1cccn1)C n1(CC(=O)NCCCOCCN(C)C(C2CC(CCO)C2)=O)ncnn1 Cc1nc(C(N2CCSCC2CCNC(C2CCC(N(C)C)C2)=O)=O)c(C)n1C Cc1cc(C(C(=O)NC2CCOCC2)N(CCSc2ccccc2)C)cnc1C C(=O)(CC(C)C(C)(C)C)N(CC(C)CNC(C1CC(=C(F)F)C1)=O)C N1(C(c2cc(C)oc2C(F)(F)F)=O)CCN(S(=O)(=O)CC2CCC2)C(CC#N)C1 C#CC(C(C)C)NC(c1conc1C(C)NC(c1cc(CCO)on1)=O)=O c1(C(N(CC(C)NC(CC2CCC(C)CC2)=O)C)=O)cc(Br)ccc1N C12(C(NOCC(N3CC(OC)(CN(C)C)C3)=O)=O)CC(CCO1)C2 N#CC1CN(Cc2ccc(C(F)(F)F)cn2)CCN1C(c1cccc(O)c1F)=O N1(C(Cc2nc(C)sc2)=O)CC2(C1)SCCC2NC(c1cc(C)c(C)s1)=O c1(C(=O)NCC(CNC(CC2CC(OC)C2)=O)(C)O)ccnc2ccnn12 Cc1c(C(=O)NCC2CC2NC(C2CC3(C2)CC(O)C3)=O)[nH]c2c1CCCC2 C1(CNC(C(N)=O)=O)Cc2ccccc2CN1C(=O)C(F)CC1CCC1 N1(C(c2cccc(F)n2)=O)CCC2(C1)CN(C(c1ncoc1C(F)(F)F)=O)C2 Cc1cc(=NCc2cc(C)c(C)s2)[nH]c(=NCCc2c[nH]c3cnc(Cl)cc23)[nH]1 C(C(=O)N=c1ccn(CC)[nH]1)N(C(=O)C(CCC)N(C)C)CC#C c1(NC(N2CC3(OCC(C(=O)OCC)C3)C2)=O)cnc(O)c2c1NCCC2 C1(NC(CN2CC(C)C2)=O)CC2CC1N(C(C1(C)CC=CCC1)=O)C2 c1(CC)cccc(C(=O)NC2C=CCN(C(=O)CCCN3C(=O)CNC3=O)C2)n1 N1(C(c2ccc(CC(C)C)nc2)=O)CC2(C1)CN(C(=O)C(F)=C1CCC1)C2 C(=O)(C(C)CC(=O)N1CCOC(C)(CNC(=O)CSCc2cccs2)C1)OC C1(C(N(C(C(=O)NCCCc2cnn[nH]2)C2CC2)C)=O)CC12CCOCC2 C1(C(=O)NC2C(NC(=O)CCc3nncs3)CC2)CC2(COCCO2)C1 Cc1ccnc(C(=O)NC2CCCCC2CNC(c2snnc2C)=O)c1N c1(CN2C(C(N3CCC(C(N)=O)CC3)=O)C3CCC2C3)cc(O)c(Br)cc1O c1(N(C2CC23CCNCC3)C(c2ccc(OC)cc2OC)=O)ccn2nccc2n1 c1(C(=O)NCC(CCC)NC(C2CCCC2(C)C)=O)ncncc1Cl C(C(C)(C)C(=O)NCC1CC(NC(=O)CCc2ccc[nH]2)C1(C)C)OCC N1(CC)C(=S)NC(c2c(N)cc(Br)cc2Cl)C(C(=O)C(F)(F)F)C1(O)C(F)(F)F c1(CC)ncc(C(N2CCC(N(C(=O)C(F)(F)COC)CC)CC2)=O)c(O)n1 c1(OC)ccn2cc(C(N3CC(C4CN(C(C5CNC(=O)N5)=O)C4)C3)=O)nc2c1 C1(NC(c2c[nH]c(-c3ccncc3)n2)=O)CC2CN(C(C3CSC3)=O)CC2C1 C1(n2cc(C(C)NC)nn2)CCC(NC)CC1.C1(C=O)CCOCC1 C1(C)(CC(=O)NC(CC)CN(C)CC)CCN1C(C1CCCCC1)=O c1(N2CC3(CN(C(C(C(CC)C)O)=O)C3)C2)ccnc2nc(C)nn12 N(C(=NCCC(C)=O)NC1CCN1c1ccc(Cl)cc1)CC(C)OC N(C(=NCC1CC1)NCc1cccc(Br)n1)C(CCC=C(C)C)C Cc1ccc(S(N)(=O)=O)cc1C(C)NCCCc1[nH][nH]c(=N)c1C#N C1(NC(C2CC(C)CC(C)(C)C2)=O)CCC2CN(Cc3ccon3)CC2C1 c1(C(N2CC3CN(C(=O)C4=CCS(=O)(=O)C4)CC3C2)=O)c[nH]c2cc(F)ccc12 c1(CC(=O)N(CCCNC(C2=C(C)CCC2)=O)C2CC2)ccc2c[nH]nc2c1 c1(OC)cc(C2CCCN(C(=O)C(C3CCS(=O)(=O)CC3)NC)C2)ccc1F Cc1cc(C)c(C(=O)NC(C(=O)NOC2CC3CCC2C3)C2(O)CCC2)o1 Cc1nc(C(=O)NC2CC(CC(=O)Nc3[nH]cnc3C#N)C2)ccc1F C1(C(=O)NCCCCCNC(C2(OCC)CCOCC2)=O)CCn2cncc2C1 c1(C(=O)OC)sc(=NC2CC(NC(C3CCc4nncn4C3)=O)C2(C)C)[nH]c1Cl C1(C)(CC)CCN(Cc2coc(-c3ccccc3)n2)C1 CC1C(C(=O)NCC2(O)CN(C(=O)C(C)(F)F)C2)C1(F)F N1(C(CN2CC(CC)C2)=O)CC2C3CCC(C2C1)N(C(c1cncc(N)n1)=O)C3 C1(OC)(CNC(C2CC(=C3CC3)C2)=O)CCN(C(=O)CN2CCCCC2)C1 c1(C(=O)NCC(CNC(C=C(CC)CC)=O)(C)OC)ccn2nncc2c1 C(=O)(C1c2c[nH]nc2CN1C(=O)CCCn1cccn1)NCCC(=C)C Cc1nsc(C(=O)NCC2(C)CCCN2Cc2ccccc2)c1Br c1(CC2(CNC(=O)COc3ccc(Cl)cc3CC)COC2)c(F)ccc(F)c1O C1(C)(C(N2CC(CNC(C)=O)C2)=O)CCN(C)C1=O.N12CCN(CC1)CC2=O C(=O)(C(F)C(F)(F)C(F)(F)F)NC(CNC(c1n(CC)c(O)nc1)=O)CCOC C(=O)(CS(=O)(=O)c1nnc(-c2ccccc2)n1CC1CC1)Nc1c(CC)ocn1 N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CC(F)CC1CNC(=O)CSC(F)(F)F C=CCC(CC)C(=O)NCc1ncoc1CCNC(=O)CC1CCOC1=O C1(C(N2CCC(C)C(CNC(=O)C3=CCCSC3)C2)=O)C(C)(C)CCCC1(C)C c1(CN(C(C(C(C)O)(F)F)=O)C)cnn2c1CN(C(=O)C(F)C(F)(F)F)CC2 CC(=O)CCCCC(=O)N1CCC2(CC2)CC1C(=O)NC1CCCC2(CCC2)C1 N1(Cc2cccc(OC(C)C)c2)CCC2(CC1)CC(NC(c1cc[nH]c1)=O)CO2 N1(C(c2c(CC)non2)=O)CCOC(CNC(=O)CC2C=CCC2)C1 C(CCCN=[N+]=[N-])NC(COC1CCN(C(C(C)CC2CCC2)=O)C1)=O Cc1nc2sccn2c1C(=O)NC1CC1NC(c1cnc2cnccc2c1)=O C1(NC(c2cn(CC)nc2)=O)CC2(C1)CC(NC(=O)C(c1ccc(F)cc1)C)C2 N1(C(CCSCC)=O)C2CCC1CC(N(C)C(C1CCCN(C(=O)CC)C1)=O)C2 c1(C(=O)OC)ccc(C(=O)NCCCN(C(=O)CCC2CCN(C)C2)C)cc1O C1(NC(C(C)=CC(C)(C)C)=O)CCCC(C(=O)NC2CN(C)NC2=O)C1 C1(C)(NC(c2cc(C)c(C)o2)=O)CCCN(C(C2CN(C3CCOC3)C2)=O)C1 N#Cc1cccc(CC(N2CCCOC(CCNC(c3ccsn3)=O)C2)=O)c1 c1(C(CC)NC(=O)C(Cc2ccccc2)CC(C)C)cccc(S(=O)(=O)NC)c1 N1(C(COCC=C)=O)CC(F)(F)CC1CCNC(=O)C(C)CC(F)F c1(C(N2C(CNC(CN(C(C)=O)C)=O)C=CC2)=O)nn(C)c(Cl)c1Br N1(C(C(C)OCC)=O)CCN(C(=O)CCC(=O)c2cnn(C)c2)C(CF)C1 n1(CC=C)cc(C(=O)N(CC(CC)NC(c2csc(CC(C)C)n2)=O)C)cn1 C1(NC(=O)CC2CCSCC2)CCCCC1NC(C1(CF)COC1)=O c1(CNC(=O)NC2CC(C)(Cc3cc(C)c(F)cc3)C2)cc(F)c(N)cc1F Cc1onc(Br)c1C(=O)NC1CC(CNC(=O)C(c2ccc(Cl)cn2)(F)F)C1 C1(CC=C)(NC(=O)C(F)C2CCOC2)CCN(C(c2snnc2C)=O)CC1 N1(C(C2CC(C)SCC2)=O)CC2(CCN(C(c3ccn4ccccc34)=O)CC2)C1 Cc1cc(C(=O)N(C(C)CN(C(=O)Cn2cnc([N+](=O)[O-])c2)C)C)ccc1F N1(c2snc(COC)n2)C2CCC1CC(NC(=O)C1=CS(=O)CCC1)C2 C12(CCSC1)C(=O)N2C.c1(CNC(C2C(C)CC2)=O)cn(C)cn1 C1(NC(CSCCOC)=O)CN(C(c2nc(O)sc2C)=O)C2(CCC2)C1 Cc1ccc2c(c1)C(C(=O)N1CCN(C(=O)C(C)(F)F)CC1)CC2 C=CCC(C(=O)N(C)CCN(C)C(c1ccc(CN=[N+]=[N-])o1)=O)N(C)C C(=O)(C1=NN(CC(C)C)C(=O)CC1)NCCC(C)NC(c1c(CC)nc(C)o1)=O C1(CNC(C=NOC)=O)CCCN(C(c2cnc(Cl)cc2Cl)=O)CC1 O=c1oc2ccccc2n1CC(O)CNC1C=C(c2ccccc2)CC1 N1(C(=O)NC(CCSC)C)CCc2cc(C#N)ccc2C1 c1(OC)ccc(C(=O)NC2(C)CCN(C(c3cc4ccsc4[nH]3)=O)C2)c(N)c1F c1(C(N2CC(CNC(Cc3cnc(C)o3)=O)C(O)C2)=O)c(C)nc(C)n1O N1(C(CC(C)n2ccnc2)=O)C2CCC1CC(CNC(C1(O)CC1(C)C)=O)C2 c1(C(CO)NC(C2(CF)CC2)=O)ccc(C2CCCCC2)cc1 c1(CNCCC(CC)CN(C)C)ccc2c(c1)CCC2 N1(C(C2C(C(=O)OC)C=C2)=O)CC2CC1C2C(=O)Nc1ccnc(C2CC2)c1 C1(C(=O)NCc2cn[nH]c2)(NC(C(C)c2ccco2)=O)CCC(C)(C)C1 C1(C(=O)NC(CNC(C(c2cccc(Cl)c2)CC)=O)(C)CO)CN2CCC1CC2 c1(C(=O)NC23CC(CNC(Cc4nc(C(C)C)sc4)=O)(C2)C3)ccc(O)c(N)n1 C1(NC(C(N(C)C)C2CC2)=O)CCOCC1NC(=O)C=C1CCSCC1 c1(C(=O)NC2CCCC(C(=O)N(c3ncc(Cl)c(O)n3)CC)C2)nccc2nc[nH]c12 C1(NC(CC(n2c(CC)ncc2)C)=O)CC(C)CN(C(=O)CN2CC(C)(C)C2)C1 Cc1cc(C(=O)Nc2cc(Br)nn2C)ccc1OC(c1ccccn1)C Cc1cc(CC(N2CC(O)(CCNC(c3ccc(C)nn3)=O)C2)=O)cc(C)c1 N1(C(=O)C2=CCCSC2)CCCCCC(NC(C2(F)CC=CCC2)=O)C1 C1(CNC(c2c(CC)[nH]cc2)=O)CCC(C)CN1C(c1csc(C2CC2)n1)=O C1(NC(c2cccc(F)c2F)=O)CN(C(=O)CC2CCS(=O)(=O)CC2)CC12CC2 C1(CNC(c2n(C(C)C)ncc2)=O)C2CC1N(C(C1CCSC1)=O)C2 Cc1cc(C(N2CC(O)(C(F)C(N3CCC4(CC4)C3)=O)C2)=O)nc(C)c1 c1(OC)ccc(S(=O)(=O)NCC2CCCN2C(C2(F)CCC2)=O)cc1Br N1(C(c2nn(CCOC)c(=O)cc2)=O)CC2C3CCC(C2C1)N(C(=O)C=CSC)C3 C(=O)(CS(=O)(=O)C12CC(C1)C2)N1C(CNC(c2ccc(C)c(O)n2)=O)CC1 C1(N(c2ccco2)C=O)CCCC12CN(CC1CC1)C2.c1(-n2ccnn2)cc[nH]c1 C(CC(CNC(c1ccc(CC(C)C)s1)=O)NC(=O)C(c1ccccc1)F)OC C(=O)(C(CCF)NC(C1CCCCN1CC)=O)NCC=C C1(O)(CNC(CCOC)=O)CCCN(C(C2CN(C)CCO2)=O)CC1 C#Cc1ccc(CC(=O)N(C2CCCC(NC(=O)CS(=O)(=O)N(C)C)C2)C)cc1 Cc1ccnn1CC(=O)NCCNC(c1csc(COc2ccccc2)n1)=O Nc1c(C(N2CCC3(CC(NC(=O)CC4C=CCC4)C3)C2)=O)cc(F)c(F)c1F CCCCC(=O)NC1COCC1CNC(c1ccnn1C(C)C)=O C1(NCCNC(=O)NC2C(C(=O)OC)CCOC2)CCCCNC1=O N1(C(C2C(C)(C)C2(C)C)=O)CC(NC(c2ccccc2Cl)=O)C(F)(F)C1 Cc1cc(C(=O)NC2(CCNC(=O)CC3NC(=O)NC3=O)CCC2)c(C)c(C)c1 C12(NC(c3ccc(CC)cc3O)=O)CCCC1CN(C(=O)C=Cc1ccoc1)C2 C1(C(=O)NCCC(COC)OC)CC2C=CC1N(C(=O)CCCCC(C)C)C2 c1(C(=O)NC2CC(CNC(c3c(COC)scc3)=O)C2)coc2c1CCCC2 CC(O)CCCCCC(=O)NCC1CCN1C(C1(c2ccccc2)CCOC1)=O CCC(CC(=O)NC1CCC(NC(=O)C(F)(F)Sc2ccc(Cl)cc2)C1)C(F)F c1(SCC(=O)NC(C2CCN(C(=O)CSc3ccncc3)C2)(C)C)ccccn1 C(=O)(CCCCC(=O)N1CC2CC(NC(=O)C=Cc3ccc(C)cc3)C1C2)OC c1(C(=O)NCC2CC(NC(CC(C)(F)F)=O)C(O)C2)cccc2c1NC(=O)CC2 C=CC1CCCCC1.c1(C(=O)NCCOCC=C)cccnc1C(F)F c1(C(N2C3CC(NC(C(CCC)(C)C)=O)C(C3)C2)=O)ccc2cnccc2c1 C1(C(=O)NCC(C)CNC(c2coc(N(C)C)n2)=O)CCc2cc(F)ccc2O1 c1(NC(C)=O)sc(Cl)cc1C(=O)NCCC(C)NC(C1CC1(C(C)C)COC)=O N1(C(c2nc(C(=O)OCC)oc2)=O)CC(CNC(=O)CCCNC(C)=O)C(O)C1 C1(C)(C(N2CC(O)(C(=O)OC)C2)=O)CC(O)CN1C(C1C=CC=CC=C1)=O S(=O)(=O)(c1cc(Br)ccc1OCC(=O)NC)N(CCCC)Cc1ccc(Cl)cc1F C(=O)(C1=CCCCCC1)NC1CCCN(C(CCc2cc(C)no2)=O)C1 C1(CNC(=O)C=CC2CCC2)CCN(C(C2CCCN2C2CC2)=O)CC1(F)F C1(NC(c2n(C)nnc2)=O)CCN(C(c2ccc(C3CC3)o2)=O)CC1F Cc1cccc(CC(=O)NCC2CCCCN2C(C2CCCC(C(N)=O)C2)=O)c1 N1(C(CNC(C)=O)=O)CCC(C2CCCN2c2cc(O)ncn2)CC1.C(C(=O)N)N N1(C(c2nccc(C)n2)=O)CC2CCCCC2(CNC(C2CN(C(N)=O)C2)=O)C1 N1(C(C2C(C=C)C2)=O)CC(NC(=O)CCNS(=O)(=O)CC)CC2(CC2)C1 C1(C)(NC(c2c(CCC)n[nH]c2)=O)CCCCC1C(=O)NCCCC1(O)CCC1 C1(C)(CNC(C(C2CC2)OCC)=O)CCN(C(=O)CCCCc2cnn[nH]2)CC1 N1(C(C(C)OCCOC)=O)CCOC(C)(CNC(C2(C)CCC3CC3C2)=O)C1 N(C1CN(C(=O)C2CCc3nccn32)Cc2ccccc21)C(C=COCC)=O CC1(C)CC(CNC(=O)CS(N)(=O)=O)CN(C(c2cnc(O)c(Cl)c2)=O)C1 CCC(C(=O)NCC=CCNC(c1ccc(C2CCCO2)nn1)=O)C(F)(F)F C1(CCCNC=O)CCCCN1C(=O)CC1CCCC12CC2.C1(CO)(CO)CCC1 C1(NC(c2c(C)con2)=O)(CO)CCN(CCOC)CC1.C1CCC1 N1(C(C(C)c2cccs2)=O)CCC2(CNC(C3(CO)CCC3)=O)CCCC12 N1(C(c2c(C)ccnc2O)=O)CCCN(C(=O)CCOC2CCCCC2)CCC1 N1(Cc2cc(C)cc(Br)c2O)CCCc2c(CO)cccc21 c1(OC)ncccc1NC(=O)C(C1CCCN(C(C2(C)CC=CC2)=O)C1)C C1(NC(C(C)(C)CF)=O)CC1C1CCN(C(C2CCCNC2=O)=O)CC1 CC(C)C#CC(=O)N(C(C)CNC(c1ccc(-c2ncon2)cc1)=O)C CCCC(C)(CCC)C(=O)NC(C)CCC(N1CC2CCC(C1)N2CC)=O c1(CN(C2CN(C(c3ccc(O)cc3)=O)C2)C)cc(OC(F)(F)F)ccc1O c1(C(=O)NC2C(C(=O)NC(C(=O)OC)CO)C2(C)C)cccc(F)c1 CC(C)C(C)(C)C(=O)N1CCOCC(C(=O)NC(c2nccc(O)n2)C)C1 C(c1c2c(nn1C)CCCC2)=CC(=O)NC(C(=O)OC)(C)Cc1cccnc1 c1(COC)nc(OC)cc(NC(C)CNC(=O)CCC2CCCC2)n1 c1(C(=O)NCC2CCN2C(=O)CCc2ncc[nH]2)cc2c(Br)coc2cn1 N(C1COc2cc(Br)ccc21)C(c1n(C(C)C)nnn1)(C)CCI C(=O)(C1c2c[nH]nc2CN1C(=O)CC1=CCCCC1)N(CC(C)C)CCO c1(CCNCC2C(Cl)(Cl)C2)ccc2c(c1)OC(F)(F)O2 C1(NC(C(CC)SC)=O)CN(C(=O)Cc2nc[nH]n2)CCC12CCOCC2 C1(C(=O)NCC#CC(=O)NCCC(=O)OC(C)=O)(OC)CCC(C)C1 c1(C(=O)NCC2(CNC(C=CC(=O)OC(C)(C)C)=O)CCC2)cncc(F)c1Cl c1(C(N2CCC(C(=O)NC3COCC3N(C)C)(CC)C2)=O)ccnc(C)c1C C1(OC(c2csc(-c3cccnc3)n2)=O)CCCC2CCOC12 C1(NC(c2c(C)ccnc2)=O)CCN(c2ccc(C(F)(F)F)cn2)CC1F C=C1CCN(C(c2cocc2C)=O)C(C(=O)NCC=CC)C1 N1(C(CCC#CC)=O)CC2(CCC2NC(c2nc(C)ncc2Cl)=O)C1 CCCCC(C(=O)NCCCCCNC(C1CC2CC2(CC)C1)=O)C(C)C Cc1ccc(C(=O)NC23CC2CN(C(=O)COCc2ccccc2C)C3)c(O)n1 C(=O)(C1=CCCN(C(c2cc(C)c(N)cn2)=O)C1)NC(C1CCCCC1)CC c1(C(N2C(CNC(Cc3cn(C)nn3)=O)CC2)=O)c[nH]c2ncccc12 CCC(C(=O)N1CC(O)(C(C)(C)CNC(=O)CSC2CCOC2=O)C1)C(F)(F)F c1(C(N2CC(N(C(C3CCC(CC)C3)=O)C)C2)=O)cn(C)nc1-c1ccoc1 C1(NC(C2(F)C(C)C2)=O)CN(C(c2onc3c2CCCC3)=O)C2(CCC2)C1 C=CC1(C(N2CCC(C(N3CCC(C)C3CN(C)C)=O)C2)=O)CCOCC1 c1(OC)nc(Cl)c(C(=O)NCC(C)(C)CNC(=O)Cc2nncn2C)s1 c1(C(N2CCC(NC(C(CC)SC)=O)C(F)C2)=O)csc2c(OC)cccc12 N1(C(C(C)C)=O)CCN(C(=O)CC(F)(F)Br)C(C2CC2)C1 c1(CC)ccc(C(c2nnnn2Cc2ccc(OC)cc2)NC(C)C2CC2)cc1 c1(C(N2C(C)(CNC(=O)CC=C(Cl)Cl)CCC2)=O)cnc(O)c2ccccc12 c1(C(=O)NCC2(O)CN(C(=O)C(F)=C3CCCC3)C2)ccc(F)c2ccccc12 C(C(O)CC(=O)N1CCCC1CNC(=O)CC1CC12CC2)N(C)C C(=O)CC(C)(C)OC.C(C(CCO)NC(=O)CCCNCCOC)OC CC(CC(N)=O)C(=O)NC1COCC1CNC(c1cc(CO)[nH]n1)=O c1(C(C)C)ccc(C(=O)N(C2C3CN(C(c4ccc(=N)[nH]c4)=O)CC23)C)cc1Cl N1(C(C23CC(NC(c4[nH]cc(C)c4C)=O)C(OC2)C3)=O)CCC2CCCC2CC1 C(C(COC)CC(=O)N1CC(CNC(=O)CC2CCCC(C3CC3)O2)C1)OC C(=O)C1=CC2(CN(N(CC(c3nn[nH]n3)C)C)C2)OC1.C1(C=O)OC2CCC1C2 C1(NC(CC(C)c2ccccc2)=O)CC2CC(NC(C3CCC3)=O)C2C1 Cc1ccc(Oc2ccc(C(=O)NCC(C)N(C)C(c3cnns3)=O)nc2)cc1 N1(Cc2ncc(C)s2)CCN(C(=O)Nc2cccc(C(C)(C)C)c2)CC1CC#N C(C(C(=O)NCC(O)CNC(=O)CCC(=O)NC1CCCC1)C(C)(C)C)OCC=C c1(C(=O)NC2C(NC(c3c(CC)c[nH]c3)=O)CCC2)cccc2c1C(C#N)C2 C(CCCCCNC(C1(F)C2CCCC12)=O)NC(C1(CC(C)C)CCCC1)=O c1(CC)nc(C)c(C(=O)NC(C)C(C)NC(=O)C(c2cccc(F)c2)(C)C)o1 c1(N2CC(C(=O)NC(C(n3ncc(C)c3)C)=O)C2)nc2ccccc2s1 CCC(C)(C)CC(=O)NC1COCCN(C(c2nc(Br)cnc2N)=O)C1 C1(CNC(C(c2cccnc2)OC)=O)CCOC1C(=O)NCC1CC(F)(CO)C1 CCCC(C(=O)NCCCN(C)C1CC1)NC(c1snc(O)c1Cl)=O c1(C(N2CC(CNC(c3c(OC)nsc3)=O)C(C)C2)=O)ccc(F)cc1C CC1CN(C(C2(C)CCCN2C)=O)CC1NC(c1coc(C(F)F)n1)=O c1(CC(=O)NCC(C)N(C(=O)C=Cc2ccco2)CC)ccc(C)cn1 C=CCCN=C(NCC)NCC(C)(O)C.N1(N2CCC(O)CC2)CCOCC1CC N1(C(C2C(C)(CC)C2)=O)CCC(O)(c2cn(-c3c(F)cccc3F)nn2)CC1 c1(N2CCC(CC)CC2)nc(=NCC=CCOC)[nH]c2c1ncn2CC C1(C(N(CCC)CCNC(=O)C(O)C(F)(F)F)=O)CC(c2ccccn2)=NO1 c1(C(N2C(C(N(C)Cc3ncc[nH]3)=O)CSC2)=O)cccc(F)c1 N1(C(C2C(C)(C)NC(=O)C2)=O)CCC(C2(NC(c3cc(=O)cc(Cl)[nH]3)=O)CC2)C1 CC1CCn2c(C(=O)NCC3(O)CN(C(=O)C(C#N)C(C)(C)C)C3)cnc2C1 C1(C(=O)NCCCNC(C2C(C(N)=O)C2)=O)Cc2ccc(F)cc2O1 N1(C(C2(CN)CC(=C)C2)=O)CCS(=N)(=O)CC1.C1(C(=O)N)CCCC(O)C1 c1(OCC#C)ncccc1C(=O)NC(c1cscn1)C c1(C(N(C)CC2CCCCN2C(C2CC2F)=O)=O)c(F)cncc1Cl C=CC(C)(O)CC(=O)N(CCCCC(=O)NC(C)C(=O)OC)C N1(S(=O)(=O)c2ccccn2)CCc2ccc(F)c(F)c2C1 N1(C(c2cnc(C(C)C)o2)=O)CCC2CC12C(=O)NCCC1CCCCO1 C1(NC(=O)CCNC2CN(C(N3CCCCC3)=O)C2)CC2CC3C(C2)C13 CCC(C)(CO)C(=O)NCC1CC(O)CN1C(=O)CCC(=O)c1ccc(Cl)cn1 n1(C(CC)C)ccc(=NC(=O)C2c3c[nH]nc3CN2C(=O)CC2(C)CC2)[nH]1 C1(N(C2CCN(C(=O)COCC(F)F)C2)C)CCCN(C(=O)C(=O)N(C)C)C1 C(=O)(C(C(C)C)n1cnnc1)N(C1CCN(c2snc(CC)n2)C1)CCOC c1(C(=O)NC(C)CNC(=O)COCc2ccccc2)cnc2c(ccn2C)c1 c1(CCC(=O)NCC2(C)CCN(C(c3cnc(S)[nH]3)=O)C2)csc2ccccc12 C1(OC)(CNC(C2CC3(CC3)CO2)=O)CCN(C(=O)C(C(C)C)SC)CC1 C(CC)(C(=O)NCC1CC1CNC(c1cnsc1C)=O)=CCCC C(=O)(C1CCCn2ccnc21)NC(C)CN(C)C(C1CC(=O)N(C)C1)=O Cc1ccc(C(=O)N(C2CCCN(C(=O)C(C)OC3CCCC3)C2)C)nc1 C(=O)(C(C)(C)CCNC(=O)Cc1cccs1)NC(CCC)C(=O)NC N1(C(CCC2C(C)C2)=O)CC2CCC(C1)C(NC(C1CC1C1CCC1)=O)C2 C1(CCC)CCN(C(C2(CCNC(c3ncnn3CC)=O)CCC2)=O)C1 N1(C(c2nc(CC)sc2)=O)CCCC2(NC(c3nc[nH]c3C(F)(F)F)=O)CC2C1 C1(C(C)C)COCCN(C(=O)C(C)(C2CCC2)NC(=O)C=C2CCOCC2)C1 Cc1cccc(CNC(C2CC(O)CN2C(c2cccc(Cl)c2C)=O)=O)c1C c1(C(N(CCNC(=O)C=Cc2nccs2)CC)=O)ccc(C)c(C)c1N c1(C(=O)NC(C)CNC(C2(Cl)CC2(F)F)=O)c(C(F)(F)F)nn2ccccc12 C1(NC(C2CN3CCC2CC3)=O)CN(C(C2CC(F)C(=O)N2)=O)CCC1CO N1(C(c2cnc(CC)nc2)=O)CC2(CC(C(=O)NC(C)C(=O)NC(N)=O)CO2)C1 C1(C(=O)NCC(C#C)CC2CC2)C(O)CCN1C(=O)CC1CCOC1C N1(C(C(C)(C)OC(C)C)=O)CCOCC(C)(CNC(=O)CC(C)O)C1 CC1CN(C)CCC1N=c1nc2sccc2c(NCCC2(C)CC2)[nH]1 Cc1nn2ccccc2c1C(N1CCCC(NC(=O)CC2CC(F)C2)C1)=O C1(NC(CCc2onc(N(C)C)n2)=O)CC2CC1N(C(C1(N(C)C)CC1)=O)C2 N1(c2ccnc(SC)n2)CCCC(C2CC2NC(=O)CCNC(=O)C(C)(C)C)C1 c1(-c2nc(CC)nn2CC(F)F)ccc(CC(C)C)cc1C N(C1CN(C(=O)C(C)CCCOC)Cc2ccccc21)C(C=CC)=O C=C=C(C)CC(=O)NCC1(C)CCCN1C(c1cnn(CC(F)F)n1)=O N1(CCC(=O)NC(C(C)NC(COCCCCC)=O)CO)CCCCC1=O c1(C(=O)NCC2N(C(c3c(C)cccc3)=O)CCC2C)cccc(C)c1N C1(C)(C(N(C)CC2N(C(C(C)OCCC#C)=O)CCC2)=O)CCC(=O)N1 C(c1cc(OC)ccc1OC)=CC(=O)N(CC(CC)Nc1cc(Cl)ncn1)CC N1(C(C(C(=C)C)(C)C)=O)CCC2CCN(C(c3ccc4cnoc4c3)=O)CC2C1 CC1(C)C(NC(C2CCCC2(F)F)=O)CCN1C(=O)Cc1cccc(C(F)F)c1 c1(CC)ncc(C(N2CCC2C(=O)NC(CO)C2(C)CC2)=O)o1 N1(C(c2n(C)ccc2)=O)CCC2CCN(C(c3ccn4c3CSCC4)=O)CC2C1 c1(C(=O)NC2C(NC(C(c3c(C)nn(C)c3)C)=O)CCC2)cncc2c1CCC2 C1(C(=O)NC2CCCCN(C(c3ccc(CC)nc3)=O)C2)CCCCCS1(=O)=O Cc1cc(C(N2CCCC2C(C)NC(c2snnc2C)=O)=O)cc(Cl)c1 c1(C(N(CCNC(=O)CC2(c3ccon3)CC2)CC)=O)ncnc2c1CCCC2 CC(C)(C)CCC(F)C(=O)NCC1CN(C(=O)Cc2ccc(F)cc2F)CCO1 c1(C(=O)CN2CCCCC2C(c2ccc(Cl)cc2)C)ccc(C(F)(F)F)cc1-c1cnccn1 C1(NC(C(n2cccn2)C)=O)(CO)CCCN(C(=O)OC(C)(C)C)C1 N1(C(C(CCC2CCC2)NC(=O)C=Cc2ccco2)=O)CCCCC(CO)C1 c1(C(N(C)CC2N(C(C=CC=CC)=O)CCOC2)=O)cn(CC)c2ccccc12 C(C)(C(=O)N1CCN(C(C2(C)CCCOC2)=O)C(C)C1)(C(C)C)NC(C)=O C1(CC(C)NC(C2CC2C#N)=O)CCN(C(c2cn(C)c(C(F)F)n2)=O)CC1 C12(CCNC(C=CCOC)=O)CCC(C1)N(C(=O)C(=CC1CCCCC1)F)C2 C(=O)(C1=CC2C=CC1C2)NCC1N(C(C(C=C)C)=O)CC(O)C1 CC1(CO)CN(C(C2COCCN2Cc2ccc(Cl)nn2)=O)CCC1O c1(C(=O)NC2(COC)CCN(C(c3nncs3)=O)C2)cc2cccc(C)c2o1 c1(C(=O)OCC)nn(C)cc1-c1cn(CC2CCN(Cc3cnns3)C2)nn1 N1(C(C(CCOC)OC)=O)CC2CCC1C1CN(C(c3nccnc3N)=O)CC21 C1(C2(C(N(CC=C)CCC)=O)CC2)CCCN1C(=O)CC1(C)CCCO1 c1(C(=O)NCCCNC(C2(COC)C=CCC2)=O)cc(C)cc(Cl)c1 C1(C(=O)NCCNC(CCCC(=C)C)=O)C2Cc3cc(Cl)ccc3C12 CC(CN(C)C)CCC(=O)NCC(C)(C1CC1)NC(c1cnc(C(C)(C)C)o1)=O CCCC(CC)CC(=O)N(CC(O)CNC(c1cc(C(C)=O)cn1C)=O)C CC(F)(F)CCC(=O)NCC=CCNC(c1scc(F)c1Br)=O C1(NC(C(C)NC=O)=O)CCCC(C(=O)NC2CCCC(O)C2)CC1 C(=O)(C(CCOC)OC)NC(CCC(N1CCC(COC)CC1)=O)C CC1C(=O)NCCN1C(c1ccc(N(C)C)cn1)=O.c12ccnc(c1)NC2=O c1(C(=O)NC(C(C)OC)C(N2CC3(CCCN3C)C2)=O)cc2ncccc2[nH]1 C1(CNC(CCCOCCC)=O)CC(F)(F)CN1C(=O)CCN1CCC(F)C1 Cc1ccc2c(C(=O)NC(CNC(c3cc(F)c[nH]3)=O)CC(F)(F)F)c[nH]c2c1 C1(C(=O)NCC2(F)CCCN(C(C3CC4(CC4)C3)=O)C2)CCCCC12CCC2 c1(OC)cncnc1C(=O)NC1CC(C(=O)NCCC(F)=C(F)F)C1(C)C C#CCCCC(C)C(=O)NC(C)(C)C(=O)NC1CC1C(=O)NCC C(C(=O)N(C(C)(C)C)C1COC1)(C(C)C1CCC1)N(CCN(C)C)Cc1ccsc1 N1(C(c2c[nH]c(=NC)s2)=O)CC(O)CC1(C)C(=O)NC1(C)CSC1 C(=O)(C1=NOCC1)NC(c1ccccc1)CN(C(=O)CSCc1cscn1)C C1(C(N(CC(C)O)CCNC(c2cc(C)sc2)=O)=O)CCOC1(C)C c1(CC)ncsc1C(=O)NCCC1(NC(=O)CCC2CC2)CC1 C(=O)(NNC(=O)c1cccc(Cn2cc(C(C)O)nn2)c1)OC(C)C c1(C(N(c2cccnc2)CCCC)=O)cc2c(s1)C(C)(C)CCC2 C1(C(=O)NCC2CCSCC2)CN(C(c2ccc(F)c(F)c2Br)=O)CCC1(F)F C12(C(=O)OC)CCC(CNC(C34CC(C(F)F)(C3)C4(C)OC)=O)(CC1)OC2 c1(NCC2(CN(C)C)CC2)nc(NCCCCS(N)(=O)=O)nc2c1ncn2C C1(NC(c2cnc(C)o2)=O)CC(C)N(C(=O)CN(C)Cc2ccccc2Cl)C1 N1(C(C23C(C)OC(C)(C2)C3)=O)CCCN(C)c2cc(F)ccc21 Cc1cc(CNC(C2CN(C(=O)CCc3ccc(=N)[nH]c3)C3CC23)=O)cc(Cl)c1 C(=O)(CC1=CCN(C)CC1)N1CCC(C(F)F)(CNC(Cc2nc(C)oc2)=O)C1 C1(C(=O)OC)CC2C(CC1C(=O)NCc1ccc(O)c(Br)c1)C2(F)F C(C(C(=O)NC1CCCN(CC(=O)OC)C1=O)C(C)(C)C)OCC=C N1(C(C(CCC)NC(C2CCC=CCC2)=O)=O)CCC(=C(F)F)CC1 CCCC(CC(C)C)C(=O)NCC(CC(=O)NC1CCC(C)(C)CC1)OC C1(C(=O)NC(CC)C(F)(F)F)COC2(C1)CN(C(=O)C(C)(C)CNC(C)=O)C2 N1(C(C=C(C)CNC(=O)COC(C)(C)C)=O)CCC(CCCO)C1 N1(C(C(CCC)O)=O)CCCC12CCCN(C(=O)CCN1CCN(C)CC1)C2 c12cnc3ccnn3c1CNC2=O.c1(C(=O)OCC)cc(C(F)(F)F)n(C)n1 c1(CC)cc(C)c(C(N2CCCC2C2CCCOC2)=O)o1 c1(-c2nc(NC(=O)NC3CC3)sc2)cccc(Nc2ccccc2)c1 C1(NC(CC(COC)NC(C2CCSCC2)=O)=O)CCN(C)C(=O)C1 C1(SC)CC(NC(=O)COC2CC(NC(=O)CCOC3COC3)C2)C1 C(=O)(C1CCc2snnc21)NC1(CNC(C2(C)N(C)CCC2)=O)CCCCC1 C(C(=O)NOCC(O)CO)(C1C(C)(C)C1)NC(C1(F)CCOCC1)=O C1(C)(CNC(COCC)=O)CN(C(c2cnc(C(F)(F)F)cn2)=O)CC1C Cc1[nH]c(C#N)cc1C(N1CC(C)(C)CC1CNC(C1(C)CCCN1C)=O)=O c1(-c2c(CN(C)Cc3ccc(OC)nn3)n(C)nc2)ccc(OC)c(C)c1 S(=O)(=O)(c1cccc(N2C3CCC2CC(=O)NC3)n1)NC(CC)CN1CCCC1 CC1=CC(C(N2CCC2CC(=O)NCC=CBr)=O)SC1 Cc1cc(N2CCCC(c3ccncn3)C2)nc(=NC(C)CCc2cn[nH]c2)[nH]1 c1(C(=O)NCC(CNC(=O)C(C)c2ccsc2)OC)cn(C)nc1C(F)(F)F N1(C(C(Cc2ccco2)NC(=O)Cc2ccsn2)=O)CCC(F)(F)C(O)C1 CC1CN(C(C2CCCCO2)=O)CCN1C(c1nn(CC(F)(F)F)cc1Cl)=O n1(CC(N2C(CNC(=O)CC3(O)CC3)COCC2)=O)ccc([N+](=O)[O-])n1 c1(C(=O)NCC2(F)CCN(C(C(CC)CC(F)F)=O)C2)nsc2ccc(C)cc12 Cc1nnc2n1CCC(C(=O)NCC1(C)CCCN1C(C1CC3(CC3)CO1)=O)C2 c1(C(=O)NC(C(C)(C)NC(CC(COC)(C)C)=O)C)cc2c(o1)CCCNC2=O C(C)(N=c1ccnc(N2CCCOC(C)C2)[nH]1)c1c(CC)nccn1 c1(C(=O)NCCCC(C)(C)NC(c2cccnn2)=O)cnc2sccn12 C1(N(C(CCN(C(C2C(C)SCCC2)=O)C)=O)C)CCOC(C)(C)C1 c1(C(=O)NCC2N(C(CSC(C)C)=O)CC2)cncnc1C(C)C C1(NC(c2n(CCC)nc(C)c2)=O)C(C)CCN(c2cc(C)nc(C)n2)C1C CCC(C)CCCC(=O)N1CCCC1(C(N1CCC([N+](=O)[O-])CC1)=O)C(C)C CC1(CNC(=O)C(C)(C)c2ccccn2)CC(NC(=O)CN2CCSCC2)C1 N1(CC(=O)NCC2(F)CC(NC(Cc3cc(C(N)=O)sc3)=O)C2)CCS(=O)CC1 S(=O)(=O)(c1cnccc1N1CCC(OC(C)(C)C)C1)NCC(C)O C1(C(=O)NC(c2cccc(Cl)c2)C)CC12CCN(C(c1cc(Cl)ccc1O)=O)C2 c1(C(=O)NCCCN(C(=O)C(C)CC(F)F)C(C)C)cnc(O)c2cccnc12 N1(C(CC2CCC(=O)C2)=O)CC(=O)NCC1C(N1CC2(CCCO2)C1)=O C12(CC(=O)NC(C3CCCN3C(=O)C(C)C(C)C)C)COC(CF)(C1)C2 C1(C(C)C)CN(C(=O)CCOCC(F)(F)F)CCN1C(c1ccc(F)c(Cl)c1)=O c1(CN2CC(NC(C(C)(C)C)=O)C(F)C2)c(Br)ccc(Cl)c1Cl C12(C(=O)NCC3CC[Si](C)(C)C3)CC(CCO1)N(C(=O)CC1CCC(=O)NC1)C2 Cc1nc2ccccn2c1NC(C1(O)CCN(c2ncnc3c2ccn3C)C1)=O CCCCC(C(=O)NC1CC2(C(=O)NCC(C)CO)COC1C2)N(C)C N1(CC(=O)NC2CCC(CC(=O)NC3CCCCC3CCO)C2)C(=O)CNC1=O CC(C)(C)CCCC(=O)N1CCC(Cn2cc(-c3cnccn3)nn2)C1 CC1(NC(c2cnc(-c3ccccc3)nc2)=O)CCCN(C(c2cocn2)=O)C1 c1(NC(=O)OC)cc(C)c(NC(=O)C(=O)NCc2csc(C#N)c2)cc1C c1(COC)nc(NCCc2cnc(C)[nH]2)cc(=NCC2(CCO)CCC2)[nH]1 C1(C(=O)NCC2CCC2(F)F)CC2CCC(C1)N2C(=O)C#CC1CCCC1 Nc1cc(C(=O)NC2CC(NC(C3CN4CCC3CC4)=O)C23CCC3)cc(F)c1 c1(CN(C(c2sccc2C)C(=O)NCC=C)CC)ccc2cc[nH]c2c1 Cc1cc2cc(NC(C34COCC3C4(F)F)=O)ccc2o1 S(=O)(=O)(c1ccc(NC2(c3ccc(F)cn3)CC2)c(F)c1)NC1C(C)CCCC1 c1(OC)cc(Br)ccc1C(=O)C(=O)NCC1CN(C(=O)CCC2CCC2)C1 Cc1cc(C(=O)NCc2nc(CNC(C3C4CC5C(C4)C35)=O)cs2)sc1C c1(CC(=O)NC2(CC=C)CN(C(C3CSCCS3)=O)C2)c[nH]c2cc(F)ccc12 C1(C(=O)NCCC(C)CCNC(C2CCCN2C2CC2)=O)CC(C(C)(C)C)=NO1 CCCC(C)(CC)C(=O)NCCCCN(C(=O)CC(C)N1CCCC1=O)C N1(C(C(C)NC(CC)=O)=O)CCOCC(F)(CNC(c2nn(C)cc2SC)=O)C1 N1(C(C(CC=C)CC=C)=O)CCC2CN(C(=O)COCC3CCCO3)CCC12 c1(C(N(C(C)CNC(=O)CCCCSC)CC)=O)cccn2nccc12 N1(C(CCn2c(C)ncc2)=O)CCC2CCC(C1)N2C(C1CC=CCC1)=O c1(C(=O)NC2C(C)N(C(=O)Cc3cncc(C#N)c3)CC2)cc(O)cc(O)n1 CC1CCN(c2cc(NCc3ncoc3C(F)(F)F)ncn2)CCS1 c1(CC(C(=O)O)NC(c2ccc(C(=O)OC)cn2)C)ccc(Br)c(F)c1 C1(C(=O)O)CC12CCCCC2.C1(CN(CC)CC)CCCN1C(=O)C1CC1 C1(NC(CC(CC)(F)F)=O)CCC(O)CN(C(=O)Cc2c(F)cccc2F)C1 N1(C(C(C)(C)OC)=O)CC2(C(=O)NCCC34CC(CCO3)C4)CCC1CC2 c1(C(=O)NC(CC)C(=O)NCC2(F)CCN(C)C2)c(C)ccn1C N1(C2CCC(=O)NCC2)CCC2CC(C(=O)NC3CCC3O)C2C1 Cc1ccc(CC(N2CC(OCCNC(=O)C(C)(C)C3CCCO3)C2)=O)o1 C1(c2n(CCOCC)nnn2)(NCc2ncccc2Cl)CCC(CC)C1 S(=O)(=O)(c1cccc2cnccc12)NCC(C(CC)CC)O N1(C(=O)COCc2nccs2)CC2(CC(NC(=O)C3=CCCCCC3)CO2)C1 C1(C)(C(=O)NCC2(CN(C)C(C3CC(=C4CCC4)C3)=O)CC2)CCCC1O Cc1cc(F)sc1C(=O)NCC(C1CCOC1)NC(c1ccncc1N)=O c1(-c2n(CCOCC)nc(-c3ccsc3)n2)cccc2ccncc12 C1(CNC(c2cn(C)nc2O)=O)CCC2(CN(C(=O)C=CC3CCOC3)C2)O1 N1(C(C(CSC)C)=O)CCC2CCN(C(C3CCC(C)CC3)=O)CC2C1 C=CC1(C(=O)NC2CCCC(CNC(c3cnns3)=O)C2)CCCCC1 N1(C(CC(C)N(C(CCCSC)=O)C)=O)CC2(C1)CC1(CCC1)C2 Cc1c(C=CC(=O)N(C2CCN(C(=O)C(C)S(N)(=O)=O)C2)C)cnn1C CN1CCC(C(=O)NCCc2ocnc2CNC(C2CNC(=O)C2)=O)C1 CCC(CC(=O)N(C)CC1CCCCN1C(=O)CS(C)(=O)=O)C(C)(C)C CN=c1[nH]cc(C(N2CCCC2(C)CCC(=O)NCC(O)C(N)=O)=O)s1 C1(N(C(=O)CCc2ccon2)CC)CCCN(C(=O)CCn2nc(C)cc2C)C1 C1(C(N2CC(NC(c3sccc3Cl)=O)C(CC3CC3)C2)=O)CCCC12CCC2 C1(OC)CCCCC1C(=O)OCC(=O)NC1CN(C(=O)C(F)OC(F)(F)F)C1 N1(C(CC(C(C)OC)NC(COCCCOC)=O)=O)CC(CO)CC12CCC2 c1(C(=O)NCC23C(CN(C(C4(COC)CCCO4)=O)C2)C3)occ2c1CCOC2 c1(COC)cc[nH]c1C(=O)NC(C)(C)C(=O)Nc1cccnc1 c1(C(N2CC(C(N(CCCC)CCCC)=O)NCC2)=O)ccc2c(Br)nn(C)c2c1 C(=O)(C1=NN2CCCN=C2N1)NCCCC(C)(C)NC(c1n[nH]cc1Br)=O CC#CC1CN(C(=O)CN(C(=O)Cc2ccc(C)o2)C(C)C)C1 Cc1cc2[nH]c(C(=O)NC(C)CN(C)C(C3CCCC(O)C3)=O)cc2o1 c1(NC(C2C(C(=O)NCC3CCN(C)CC3)C2)=O)cc(Cl)c([N+](=O)[O-])cc1O C1(C(=O)NC(c2ccc(C)cc2)C)CC2CN(C(=O)CCC3(C)N=N3)CC2C1 Cn1cnc2c(C(N3CC(Nc4cc(O)ncn4)C4(CCC4)C3)=O)cccc12 c1(C(N2C(C(C(=O)N(CC(=O)NC(C)(C)C)C)(C)C)CCC2)=O)cncc(F)c1 c1(C(N(C2CCN(C(=O)CCCOC)C2)CC)=O)cc2ncn(C)c2cn1 CC1CC2(CCN(C(C3(C)CCN(C)C3=O)=O)CC2)CN1C(c1cc(Cl)no1)=O Cc1nn(C)c(C(N2CCCC2c2cccs2)C(=O)NCCC2CC2)c1Cl c1(OCC)cc(Cl)ccc1C(N1CC2C(NC(=O)C(COC)NC(C)=O)C2C1)=O C(=O)(CCC1=NNC(=O)CC1)NC1CC(CNC(C2(C)C(C)C2)=O)C1 C(=O)(CC(C(F)(F)F)NC(c1ncc(F)cc1N)=O)NC(c1nc(CC)on1)C C1(=CC(N2CCC(NC(C3C(C)OC(C)C3)=O)C2C2CC2)=O)CN2CCC1CC2 N1(C(C2CCC(=O)N2)=O)CCCC(NC(c2ncsc2Br)=O)C1 C=CCCC(C(=O)N(C)CCO)NC(C1CCCC1)=O.C1CCC1 CCCCC(CC)C(=O)NCc1ccc(C(=O)NCCC(C)N2CCCC2)cn1 C1(O)(C(=O)NCC(C)NC(c2cccc(C(N)=O)n2)=O)CCOC1(C)C N1(C(c2cnc(C)nc2O)=O)CCCC2(NC(c3cccs3)=O)CCCC12 C(=O)(C(C)C(C)NC(c1sncc1C)=O)NCC=CCCOC N1(C(C(C2CC2)OC)=O)CCCC(C)(NC(c2c(C(F)(F)F)cccc2Cl)=O)C1 c1(C(N(C2C3CN(C(=O)CCNS(C)(=O)=O)CC23)C)=O)nccnc1Cl c1(CC)cccc(C(=O)NC2CC(C(C)NC(C(CN(CC)CC)F)=O)C2)c1N C1(C(=O)NCC2(O)CCN(C(C3(COC)CCC3)=O)C2)CC2CCC(C1)O2 n1(CC(N2C(C)CC(CNC(C3(CO)CC3)=O)C2)=O)ncc2cccnc12 Cc1cc(CCC(=O)NCC(C)NC(c2[nH]c(O)nc2C)=O)c(C)s1 c1(OC)ccc(NC(=O)CC2CCCN(S(=O)(=O)CC#N)C2)cc1Br C1(C)(C(N(C2CN(CC(=O)NCc3ccccc3)C2)C)=O)CC1(F)F c1(CCC)ccc(C(=O)NCC2CCCC2NC(C2(COCC)CC2)=O)cc1 C1(CNC(CSC)=O)CCC2(CN(C(=O)CCOc3ccccc3C)C2)O1 Nc1cc(Cl)nc(C(=O)NC2CCN(C(c3nncn3C3CC3)=O)CC2)c1Cl C(N=c1[nH]c(N2CC(c3cc(C)[nH]n3)C(C)(C)C2)nc(=N)[nH]1)C1(OCC)CCC1 N1(C(C2N(C)C(=O)CC2)=O)CCCC2(C1)CN(C(c1cncn1C(F)(F)F)=O)C2 Cc1ccc(C(C)N(CC(F)(F)F)C(=O)C=CCOC(C)=O)o1.C(C)(C)(C)O CCCCCCCC1CCN1C(C1CC(n2cc(CC3(O)CCSC3)nn2)C1)=O C12(C(=O)NCC3CCC(C)C3)CC(CN(C(=O)C(F)F)C1)C2 C(CCC)(C(=O)NCC1CCCN1C(c1[nH]nc(C(F)(F)F)c1C)=O)=CCC c1(CCNC(C23OC(C)C(C2)C3)=O)c(F)ccc(F)c1Br c1(C(C)(C)C)ncc(C(=O)NC(C2CCOC2)CNC(=O)Cc2cn[nH]c2)o1 C1(C(=O)NCC2(C)CC(C)(C)C2)(CC)CCCN(C(=O)C(F)=C(C)C)C1 Cc1cc(NC(C2(NC(=O)C(C)C(F)F)CCC(C)(C)C2)=O)cc(O)c1 C=CC(C)(C)C(=O)NC(CN(C)C(c1cc(-c2ccns2)on1)=O)CC N1(C(c2ccc(NC)cn2)=O)CCCC(NC(c2cn(C(C)C)cn2)=O)CC1 CC(C)C(CNC(c1n[nH]c(=N)[nH]1)=O)C(=O)NC1(CO)CC2CCCC12 N1(C(c2cnc(OC)s2)=O)CCCC2C1CCN2C(=O)Cn1nc(C)oc1=O C12(C(=O)NCC#C)C(NC(C3CN(C(C)C)C3)=O)C3CC1C2C3 c1(C(=O)NOCC2CC2)ncoc1CNC(c1ccc(C(F)F)o1)=O O=C(Cn1cc(C2C3COCC23)nn1)NNC(=O)NC1OCCO1 c1(C(CC(C)C)NC(=O)C(=O)Nc2ccc(Br)cc2)ccc(F)cc1 C(CC(=O)N1Cc2ccccc2CO1)(c1ncccn1)C(=O)OC(C)(C)C CC1CN(C(=O)CCCc2cccc(Cl)c2)CC(C)N(C(=O)COCCF)C1 N1(C(c2ccc(OC)o2)=O)CCCC2(CCCCC2NC(c2oncc2C)=O)C1 c1(COCC(N2CC(NC(C3CCC(C)O3)=O)(CO)C2)=O)ccccc1Cl C1(NC(C2(CC)CCOCC2)=O)CCC2CC1CN2C(C1CCC(CC)CC1)=O C(=O)(C(F)(F)CCC(N1C(CNC(C2CC(C)(F)C2)=O)CC1)=O)OC(C)(C)C C(=O)(C(O)CC(C)(C)C)NCC(CNC(c1cnc(C(C)O)s1)=O)(C)F N1(C(C(c2ccc(C)cc2)=O)C)CCC2C(C1)NC(=O)N2C c1(CC(=O)NC2CC23CC(NC(C2(O)CC2)=O)C3)c[nH]ccc1=O c1(C(C(=O)NCCCSC)N(C)CC2CCOC2(C)C)sc(Br)cc1C C12(CC(=O)NC)COC(CCOCCOC3CCN(C(C(C)C4CC4)=O)C3)(C1)C2 CC(C)(CC1CC1)C(=O)NCC1C2CC1N(C(c1ocnc1C(F)F)=O)C2 C1(C(=O)NC2(C)CC(NC(C3CN(C(C)C)C(=O)C3)=O)C2)OCCN(C)C1=O C1(NC(c2c(C)coc2C)=O)CCN(C(C2CC3(CCO2)CC3)=O)CC1F N12C3CCCC1CN(C3)C(=O)COCCOCC2=O.c1(COCC)nnc(C)s1 N1(C(=O)C(O)Cn2cncn2)CC2CC1CN2C(C1(c2cccc(F)c2)CC1)=O C(CCCCCC(=O)N1CCC(O)(CN(C(=O)CN2CCC(C)(C)C2)C)C1)SC N1(C(C(CCOC)(C)C)=O)CCN(C(C23CCC(CC2)C3(C)C)=O)CC(O)C1 c1(C(C)C(=O)NCc2nc(-c3cccs3)n[nH]2)ccc(F)cc1F Cc1cc(C(=O)NCC2(C(=O)NC3CCN(C(C)(C)C)C3)CC2)cc(O)n1 C(N=c1ccnc(N2CCOCC(F)(F)C2)[nH]1)c1cc(O)nc(O)n1 C1(N(C(C(N2CC(C)C2)C)=O)C)CCCN(C(c2nn[nH]c2Cl)=O)CC1 Cc1cc(C(=O)NCC2(C)CCCN2C(C2CC(F)(F)CS2)=O)cn(C)c1=O C(=O)(C1=C(Cl)CCCC1)NC(C(C)OC)C(=O)N1CC(N2CCOCC2)C1 C1(NC(C2C(C(=O)NCC#C)C2)=O)CCN(C(=O)CC2=CCCC2)CC12CCC2 C1(CCCNC(C2(C)CCCC2)=O)CCN(C(=O)CCC2(O)CCOCC2)CC1 CC1(C)CN(C(C2CCOCC23CCC3)=O)CC(CNC(=O)CN2CC=CC2)O1 c1(C(NOCC(=O)N(CCCO)CC)=O)cc(C)c(C)nn1 S1(=O)(=O)c2ccc(C)c(c2)C(=O)OCCN1C.c1(OCC)cccc(Br)c1 C1(N(C(C(C)Cn2ccnc2)=O)CCNC(C2(C(F)F)CC2)=O)CCCCCC1 N1(C(c2ncccc2CO)=O)CCCC(N=c2nn[nH]n2Cc2ccccc2)C1 C12(CN(C(=O)CN3CCC(c4cc(F)ccc4F)C3)CC)CCCCC1OCC2 C(C(C(=O)NCC1CC1(C)C)N(C)C)NC(C(C1CCC1)OC)=O C1(NC(CC(C)n2ccnc2)=O)CN(C(=O)CSCC(F)(F)F)C(C)(C)C1 C(=O)(N=c1[nH][nH]c2c1CN(C(c1ccc(Cl)c(I)c1)=O)C2)c1ccc(C)c(F)c1 C(=O)(CCCC(F)(F)F)NCCC(C)(C)C(=O)Nc1cccc(OCF)c1 O=S(=O)(c1cccnc1NCCC1CC1C1CC1)NCCN1CCSCC1 N1(c2ncnc(C)c2F)CCC2(CCN(C(=O)Cc3c(F)cncc3Cl)C2)C1 C(CCCCC(=O)NC1CCN(C(c2cccc(C#N)n2)=O)CC1F)N(C)C N=c1[nH]c(C2CC2)ncc1C(N1CC=CC1CNC(=O)CCC1CCOC1)=O N1(C(CCC=CCC=C)=O)CCCCC(CNC(=O)Cc2cc(Cl)sc2Cl)C1 CC1CC(C(N2CCC(OCCNC(c3c[nH]c(Br)c3)=O)C2)=O)CCS1(=O)=O N1(C(C2(F)CN(C(c3c(N)non3)=O)C2)=O)CC2(CCC1CO)CC2 N1(C(C2Cc3ccccc3C2)=O)CC2CCC(C1)C2NC(C12CSCC1C2)=O C=C(C)CC(C(=O)Nc1ccc(C(F)(F)F)cc1CO)NC(C1CCCC1)=O C12(CNC(CC)=O)CN(C(c3cn(-c4cnn(C)c4)cn3)=O)CC1CCO2 CC1C(NC(C2(C3CCCO3)CCC2)=O)CCN1C(=O)CC1CCCC(=O)N1 c1(N(C(C2C(NC(C(C)NC(CC)=O)=O)CCCC2)=O)C)cc(C)ccc1C CC(C)CC(C(=O)N1CCOCC(C(=O)N(C)C)C1)NC(=O)C(=O)NC(C)(C)C C(=O)(CC(C)(C)C(=O)NCC1CC(OC)CN1C(=O)CC1CC(N(C)C)C1)OC C1(C(N(C)CC2CC2C(F)(F)F)=O)CNC(=O)CN1CCN(C)C Cn1ccc(NC(=O)CC2CC2CNC(=O)OC(C)(C)C)n1 CCC(CCCC(=O)N(C(C)CC)C)NC(=O)C(C)CCN(C)C O=C1CC(=O)CC(C(=O)N(CCC(=O)NC2CCN3CCCC23)CC2CC2)C1 c1(NC(C)=O)ccc(F)c(C(=O)NC2CCCCC2CNC(=O)CC(C)(C)F)c1 CCCCCC(O)C(=O)NC1CCCC(C(N2CC(C3CC3)(COC)C2)=O)C1 CC1CC(=O)CCC1C(=O)NCC1CN(C(C23CC4CC2C3C4O)=O)C1 Fc1ccccc1CNC(=NCC1CC1(Cl)Cl)NC1CCOCC1 c1(C(N2CCN(C(C3N(C)CCCC3)=O)C3C2C3)=O)c[nH]c2cc(C#N)ccc12 N1(C(C(COC)NC(C)=O)=O)CC(N(C)C(c2cccc(OC)n2)=O)C2(CC2)C1 O(NC(=O)C(c1ccco1)NC(c1cccn1C(C)C)=O)CCCC(=O)OC C(N=c1[nH]c(N2CCOC(C(N)=O)C2)nc(=N)[nH]1)c1ccc(NCC(C)C)cc1 N1(C(C#CC(CNC(CC=C(C)C)=O)(C)C)=O)CCC2(CC1)CN(C)C2 C1(CNC(C2CCCN(CC)C2)=O)CN(C)CCN1C(C1OCCO1)=O C1(C(=O)NC2CCN(C(=O)C=C(Cl)Cl)CC2CO)Cc2ccccc2CO1 N1(C(CCSCCC)=O)CC2CC(NC(=O)CCC=CC(C)C)CC2C1 c1(C(N2C3(CNC(C4(NC(C)C)CC4)=O)CCC3CC2)=O)coc2ccccc12 Cc1cnc(C)c(NC(C2CC3CC3N2C(c2cc(F)ccc2O)=O)=O)n1 CC1(C(N2CCOC(C(=O)NOCc3ccccc3)C2)=O)CC2CC2C1 C1(OCC)CC2(C1)CC2CCNC(CCC(=O)N(CCN1CCC2CC12)C)=O C(=O)(CN=S(C)(C)=O)NCC1CC(OC)CN1C(C1CCCN(C(C)C)C1)=O N1(C(C=CC(CC)C)=O)CCC(CN(C(=O)CN2CCCNC2=O)C)CC1 N1(C(C(C(C)C)F)=O)CCCN(C(=O)CC2CC2)CC1C C(C(C)(C)C(=O)N(C)CC1CCN(C(c2ccc(C3CCOC3)cc2)=O)C1)OC C1(NC(COCCOCC#C)=O)CCCCCN(C(=O)C2=CCCC2C)C1 Cc1[nH]ccc1C(=O)NCC(Cc1ccccc1)NC(=O)CC1C=CCC1 C1(C(=O)Nc2c(C)csc2)CN(C(=O)CCc2cn[nH]c2)CC1C CCCCC(O)C(=O)NC(C)(C)CNC(c1cc(C(F)F)cs1)=O CC1(C)CCC(NC(=O)C(c2ccco2)NC(=O)Cc2ccc(O)cc2)C1 c1(CNC(C(C)C2CC2)=O)cn2c(n1)CC(C(=O)O)CC2 C1(OC)CCC2(C(N3CC(C(C)NC(=O)CS(=O)(=O)NC4CC4)C3)=O)CC12 c1(C(=O)NCCCN(C(C(CCC)C)=O)C2CC2)c(C)oc(C)c1C C1(C(=O)NC(COCCCNC(C(C2CC2)SC)=O)(C)C)CC2CC1CC2(F)F C(=O)(CC(C)CC(F)(F)F)NCCOCCNC(C(C1CCCC1)OCC)=O N1(C(C2C(C)C3CCC2C3)=O)Cc2occ(C(N3CCC(C)C3CO)=O)c2C1 c1(CNC2C(C)CN(C(=O)OC(C)(C)C)C2)oc2ccccc2c1C(F)F C(c1cccc(OC)c1)=CC(=O)NC(CNC(c1ccc(CC)cn1)=O)CO Cc1ccc(C(N2CC3CCC3(NC(=O)CN=S(C)(C)=O)C2)=O)c(C2CC2)c1 N(C(=NCC(C)N(C)C)NC(c1cccc(Cl)c1)C)C(C=C)C C(=O)(CC(F)(F)C(F)F)N1C(CNC(c2ccc(Cl)s2)=O)CC(OC)C1 Cc1nn(C)c(C)c1CC(N1CCC(NC(c2cccc(=O)o2)=O)C(O)C1)=O C1(C(N2CCC(O)(C(C)NC(c3ccc(O)nc3)=O)C2)=O)COC2(CCC2)C1 Cc1ncc(CCC(=O)NC(CNC(=O)C(O)c2cnc[nH]2)C2CC2)s1 C12(CNC(c3cnc(S)[nH]3)=O)CCCC1CCN2C(c1coc(C(F)(F)F)c1)=O N1(C(c2sc(CC)c(C)c2)=O)CC(CNC(C2CCC(=O)N(C)C2)=O)C(C)(C)C1 c1(CC)ccc(NNC(=O)N=c2[nH]nc(CCC(=O)OC)s2)cc1F CC1(C)CN(C(=O)CN(C2CCC2)C(C2CC2[N+](=O)[O-])=O)CC1CO c1(C(N(C2CCN(C(C3CC(F)C3)=O)CC2)CCC)=O)ccc2nc(O)[nH]c2c1 c1(C(N(C2CCN(C(=O)C=C3CCOCC3)C2)CCC)=O)ccn2c1CSCC2 c1(C(=O)NC(CCNC(CCCNC(C)=O)=O)C)ncn2c1CCC2 C1(N(C(CNC(CCC)=O)=O)C)CCCCN(C(=O)C(C)=C(C)C)C1 N(C(=NCCCC1CC1C)NCC1CC1)CC(c1c(C)nn(C)c1C)O CC(CC(=O)NCC1CC(C)CCN1C(C1CC(N(C)C)C1)=O)C(C)(C)C N1(C(C(CC)n2cccn2)=O)CCC(C(CO)NC(=O)CN(C)CC)CC1 C1(CC=C)(NC(=O)C(C)CC)CCCN(C(=O)CC(=O)OCC)C1 N1(C(C(C2CN(C(=O)CC3CC=CCC3)C2)OC)=O)CCCOCC1C c1(NCc2cn(C)nc2)cc(-c2ccnn2C2COC2)ccn1 c1(C(=O)NC23CC(CNC(CCC=C)=O)(OC2)C3)ccc2ncn(C)c2n1 CC(C)(CNC(c1cnc(=N)[nH]c1)=O)CC(=O)NC(CCO)C(F)F Cc1cccc(CC(=O)NC(c2cccnc2)C(=O)N(C2CCCN(C)C2)C)c1 C(C(C)(C)CC(C)C)NC(C=CC1N(C(CC(=O)OCC)=O)CCC1)=O C12(CC1(C)C)C(=O)N2.CC(C)(C)NC(=O)CCOCCNC1CC1.C1(=O)CN1 CCC(CC(F)F)C(=O)N(CCCCN(C)C(C1C=C1C)=O)C c1(C(c2n(CC=C)nnn2)NC2CCS(=O)(=O)C2)nc(C)c(C)n1C C(=O)(C(=O)N=c1cc(C)o[nH]1)N1C(C)CC2CN(C(C(C)OCC)=O)CC21 CN1CC2CCN(C(C34CCC(NC(=O)CCCC#N)(CC3)C4)=O)C2C1 Cc1ccncc1CC(N1CCC(CNC(=O)C(O)C2CC2)C1)=O C1(NC(c2cnc(C3CCC3)s2)=O)C=CCN(C(C2(CCF)CCOCC2)=O)C1 CCCC(CCC)=CC(=O)NCCCN(C1CCCC1)C(=O)CC1CC(F)(F)C1 c1(SC)cc(C(=O)NC(C)(CNC(=O)C(C)(O)C2CC2)C(C)C)c(C)o1 C(=O)(C(CCCC)NC(N)=O)NCC(CCCC)NC(=O)CCNC(N)=O CCC(CCC(=O)N(C)CCc1cnc[nH]1)NC(=O)CSC1CC1 C1(NC(c2cc(OC)c(C)cc2)=O)COC2C(NC(=O)CCCC#N)COC12 c1(N(c2n(CC(CSC)OC)nnn2)C)ccnc(OC)c1Br C1(CC)CN(C(c2ccc(CO)o2)C(=O)Nc2ccccc2C)CC(=O)N1 N1(C(Cn2c(C)cc(O)cc2=O)=O)CC2(C)CN(C(=O)C=CCF)CC2(C)C1 C1(CCNC(c2ccc(CCC)cc2)=O)CC(F)(F)CN1C(=O)CCCN(C)C C(=O)(C(C)C(O)C(C)C)NC(CC)CC(=O)NCC1C(C)C1C c1(C(N2CC(CO)C(C)C2)C(=O)NCCC)ccc(OCC(F)F)cc1 N1(C(CC(C)OC)=O)CCOc2ccccc2C1CO Cc1ccc2n[nH]cc2c1C(=O)NCC1CCN(C(=O)C(C)O)CC1(F)F C=CC1(C(N2CC3CC(F)CC3C2)=O)CCN(C(c2cccnc2C)=O)CC1 C(CC(=O)NCc1ccccn1)(C(C)C)NC(c1c(C)n[nH]c1)=O c1(OC)ccc(C)cc1CN(C)CC1CCCN1C(c1cnc(C(F)F)cn1)=O c1(COC)nc(C(=O)NCCOCCN(C2(n3ccnn3)CC2)C)cs1 C1(C(=O)NCC(N2CCCCC2)=O)CC2CC1CC2NC(c1cn(C)ccc1=O)=O C1(C2CN(C(c3ccnc(-c4ccco4)c3)=O)C2)(NC(c2c(C)[nH]cc2)=O)CC1 C(=O)(CC(C)OC)N(CC=CC(=O)N(CC(=O)NCC)CC)C CCC(N=c1[nH]c(=NCCCN(CC)CC)[nH]c2c1CCC2)C1CCOCC1 N1(C(c2ccc(C)cc2)=O)CCC(NC(c2cncc(N)c2C)=O)C2(CCC2)C1 C1(C(N2CC3CC3C2C(F)(F)F)=O)CCC2(CCCCC2)C1 C(C(C)C)(C(O)C(=O)N(C1CC(NC(=O)C(C)Oc2cccnc2)C1)C)OC Cc1cnc(C(N2CCC(C3CCC(C(=O)N(C)C)O3)CC2)=O)cn1 CCCC(C)(C)CC(=O)NCCN(C)C(c1cc(N)c(OC)cc1F)=O N1(C(CC=C)=O)CC(CNC(c2c[nH]ccc2=N)=O)C(C(F)(F)F)C1 N1(C(C=CC(=O)OC(C)(C)C)=O)CCC(NC(c2ccc(CO)cc2)=O)C12CC2 Cc1ccc(C)c(S(=O)(=O)NC2CCN(C(=O)CCC3CC3)CC2O)c1 C(=O)(CC(C)C(C)(C)C)N1CC(CC=C)(NC(C23COCC2C3)=O)C1 c1(CC(C)OC(c2cc(O)ncn2)=O)cccc(Cl)c1 Cc1cccc(Cl)c1C(c1nnnn1C1CC1)NCCNC1CCSC1 N1(C(C2(CC(C)C)CCNC2=O)=O)CC2(CCC2NC(=O)CCF)C1 C1(C)(NC(CCC(C)C)=O)CCN(C(c2c[nH]cc2Cc2ccccc2)=O)CC1 c1(NC(C)=O)cccc(C(=O)NCC2CCCN2C(c2csnn2)=O)n1 Cc1nc(CO)sc1C(=O)NCC(C1CCN(C(C2(C)COC(=O)N2)=O)CC1)O c1(C(=O)NC(CNC(CNC(CC)=O)=O)CO)nc2ccccc2nc1C C1(NC(C(n2ccc(C)n2)C)=O)CN(C(=O)C(F)(F)C2CC2)CC(F)(F)C1 O=C(Cc1cccs1)C(=O)NCC1CN(C(=O)CCn2ccnc2)C1 c1(C(=O)NCCCCNC(C2(F)C(C)C2)=O)sc(Br)cc1Cl c1(C(=O)NC(CN(C(C2CC2(Cl)Cl)=O)CC)C)ncc(C(F)(F)F)cc1Cl c1(NC(=O)NC2N(C)c3ccccc3C2)ccc2cc(S(N)(=O)=O)ccc2c1 C1(C(=O)NCC(C)NC(c2c(Cl)ccc(C)c2)=O)Cc2ccc(Cl)cc2C(=O)O1 c1(C(N2CCC3(NC(=O)Cn4ncnn4)C(C2)C3)=O)cc(Cl)cc2cccnc12 C1(C(=O)NC(C2(O)CN(C(C(CCCC)O)=O)C2)C)CN2CCN1C(C)C2 CCCCCNC(C1(CNC(C2CC(F)C2)=O)CCC1)=O c12ccc(=O)n(c1)CC1CCCN1C2=O.Cn1cc(COc2ccc(F)cc2)c(Br)n1 C1(NC(CC=C)=O)CN(C(c2cc(CC)n(CCO)n2)=O)C(C)(CC)C1 N1(C(C=Cc2cccc(N)c2)=O)CC2CCC(NC(C3(CCF)CC3)=O)CC2C1 C(C(C)(C)C(=O)NCCC1CN(C(=O)Cc2nc(C)sc2C)C1)SC C(=O)(CCS(C)(=O)=O)NCCCCCCN(C(C12CC(OC)C1C2)=O)C n1(CC)nc(C(=O)NC2COCC2NC(=O)C(C)(CC)OC)cc1O Cc1ccc(CN2CCC(N(C(=O)C=Cc3cccc(O)c3)C)C2)cc1C#N c1(C(N(C2CCC(n3cc(C(N)=O)nn3)CC2)C)=O)ccc(-c2nccs2)cc1 c1(C(=O)NCC(C)CNC(c2cccc3sncc23)=O)cnc2nccn2c1 c1(C(N2CC(N(C(=O)CC3CC34CC4)C)C3(C2)CC3)=O)ccc(Cl)c(F)c1N CC(C(=O)NCC(c1cc(F)cc(Cl)c1)NC(C1(CC#N)COC1)=O)S(C)(=O)=O c1(CCCC)noc(C(C)NC2C=CCSC2)n1 CC(CCCCNC(=O)C(C)(O)C1CCC1)NC(=O)C(C)(C)CO N1(CC(=O)NCc2cccc(OCCC)c2)CCC2CC3(CCC3)C2C1 C(CCCC(=O)N1CCCC1C1CCN(C(c2cnsn2)=O)CC1)OC c1(OC)ccc(C(N2CCC(NC(=O)CC3CCCN3)CC2)=O)cc1N n1(CC)c(C)cc(C(=O)NC2CCN(C(c3ccc(NC(C)C)cc3)=O)C2)c1C C1(CNC(CCCSC)=O)CC2CCCC2N1C(=O)CN1CCCC1C CN1C(=O)CCC1C(=O)NC1COCC1CNC(=O)COC1CCCCCC1 Cc1c(C2(C(N3CC(F)(CNC(=O)CC=C(Cl)Cl)C3)=O)CC2)cccc1F CC(C)(CNC(C1CCN1C(C1CN(C2COC2)C1)=O)=O)CCCO N1(C(c2c(OC)nc(C)cn2)=O)CC2CCC1CN2C(=O)CC1OCCC1(C)C C(CC(CC)C(=O)NCC12CC(CO1)N(C(C1(SC)CCC1)=O)C2)=CC c1(CC)[nH]ccc1C(=O)NC12CC(C(=O)NC3CC(C)C3)(C1)C2 c1(C(=O)OC)coc2cc(C(N3CC(CNC(=O)C(C)C(C)(F)F)C3)=O)[nH]c12 c1(CNC(c2cccc(OC(C)C)c2)C)c(OC)cccc1O c1(OCC(=O)NC(C2CCCN(C(C(C(C)C)O)=O)C2)(C)C)ccc(Cl)c(Cl)c1 Cc1nsc(C(N2CC(CCCCNC(C3(C)CCNC3=O)=O)C2)=O)c1N c1(C(=O)NCC#CCNC(Cn2[nH]c(=N)c(Br)c2)=O)n[nH]c2ccccc12 c1(CC(C(=O)NCC2(NC(c3ncc[nH]c3=O)=O)CCOC2)O)ccccc1Cl c1(OC)cc(C(=O)NCCCN(C(=O)CCC(C)OC)CCO)cc(F)c1C#N N1(C(C2(OC(C)=O)CC2)=O)CCN(CC2CCN(C(=O)C(C)CO)C2)CC1 c1(C(=O)NC2C(CNC(c3nc(COC)[nH]n3)=O)CCC2)cc(C)cnc1C N1(C(CC2CCN(C)C2)=O)CC2CC1C1OCCOC21 c1(CC)sc(C(=O)NC2CN(C(=O)C(C)OC3CCCC3)CC2O)cc1C C1(CC(=O)NC2COCC2CNC(c2cc(Cl)cc(Cl)c2)=O)CCC(F)(F)CO1 CC1CC(F)CN1C(C12CC1CCN2C(=O)C(CO)N(C)C)=O N1(C(CC(=C)C)=O)CC2CCC(C1)C2NC(=O)CCCCOCC N1(CC(=O)N(C2CCN(C(C3C(c4ccccc4)C3C)=O)C2)CC)CSCC1=O C(=O)(CC(C)(C)C(C)=O)N1CCCC(N(C(c2n(CC)ncc2Cl)=O)C)CC1 N1(C(Cc2c(C)non2)=O)CCOCC1CNC(c1ccc(Cl)[nH]1)=O C(CC(=O)NCC1(F)CCN(C)C1)(C(F)F)NC(c1c(CC)occ1C)=O C#CCC(C)(C)C(=O)N1CCC2C(C(=O)N(C)OCC(F)(F)F)C2C1 c1(OC(C)C)cnc(N2CCCC(CNC(=O)C=Cc3nccs3)C2)nc1 N1(C(C2(COC)CCC2)=O)CCC(NC(c2cn3c(n2)CCC3)=O)C(CO)C1 N1(C(CCN(C)C(C2CCCOCC2)=O)=O)CC(O)CC1C(N)=O C1(CCC(=O)NCC2C(NC(=O)OC(C)(C)C)C2)CCCC(=O)N1 c1(C(=O)NCCC2CCN(C(=O)C3=CCOC3)CC2)noc2ccccc12 c1(C(N2CC(C)C(NC(=O)C(C)n3cccn3)C2)=O)cc(Br)ncc1Br Cc1ccc(C(=O)NC(C)C(CO)NC(=O)C(C)n2cnnn2)nc1O C1(NC(C=NOC)=O)C=CCN(C(=O)CC2CC23CC3)C1 c1(C(=O)NCC(C)(O)CNC(C2(C(F)(F)F)CC2)=O)nccc2c1CNC2=O N#Cc1nc(=NCCCCCCNC(=O)CCc2cncc(F)c2)cc[nH]1 S(=O)(=O)(c1ccc(O)cn1)NC(CCc1cccc(OC)c1)C N1(C(C(C)SC)=O)CCC2C(NC(=O)CCN3CCOCC3)C12 c1(C(N(CC(CC)NC(CCSCCCC)=O)CC)=O)c[nH]c2c(C)cccc12 N1(C(CC(C=C)C)=O)CCC2CN(C(c3ccc(OCCCC)cc3)=O)CC2C1 N1(C(c2n(CC)nnc2)=O)CCC(NC(=O)C(C)NS(C)(=O)=O)C12CC2 c1(C(C)C)cc(C(C)(C)NC(C2CC2c2ccccc2)C)n[nH]1 c1(C(N2CCC(N(C)C(C3CCCN3C=O)=O)C2)=O)cc2n(n1)CC(C)(C)CO2 Cc1ccc(O)c(C(=O)NCCC(C)NC(=O)C(C)Cc2ccnn2C)c1 c1(N2CC(CCOC)OCC2)nc(NCC(C(C)C)OCC)c2c(ncn2C)n1 c1(CCC(=O)NC23C(CN(C(C4CC(C)C4)=O)C2)C3)c[nH]c2ccccc12 c1(C(=O)NC2CCC(CC(=O)NCCc3nc(CC)[nH]n3)C2)ccc(C#N)o1 N1(C(C2C(OC(C)=O)C2)=O)CCC(F)(C(=O)NC2(CO)CC2)CC1 Cc1c(C(=O)NC(CNC(C23CCC(CC2)C3)=O)C2CCC2)c(C(F)F)nn1C N1(C(C=CC(CC)=CC)=O)CCC2C1CCCN2C(=O)Cn1cnnn1 C(=O)(C1=CCCCCC1)N1CCN(C(C(C)CC2CC2)=O)CC1CC1CC1 C(=O)(C1=CCC(C)CC1)N1CCN(C(C2N(CC)CCOC2)=O)CC1.C1CO1 C1(CCNC(C=C(C)C(C)C)=O)CCN(C(C2(c3ncco3)CCC2)=O)CC1 N1(C(C2=CC(C)(CC)C2)=O)CCC(CCNC(=O)CNC(=O)OC)C(F)(F)CC1 C1(N(C(=O)COC(n2ccc(SCC)n2)=O)C)C2CC3C(C2)C13NC(COC)=O c1(C(=O)NC(CCCC)CNC(=O)C(C)OCCOCC)ccc2nnnn2c1 CC(CCNC(C1(C)CCN(C(c2cccc(C3CC3)c2)=O)C1)=O)C(F)F N1(C(CCC(=O)NCC)=O)CCCC(O)(CNC(C2CC2C(C)(F)F)=O)CC1 C1(NC(c2cc(C)no2)=O)CN(C(c2cc(CF)on2)=O)CC1C c1(C(N(CCC(C)NC(=O)C2CC2)C)=O)cccc(O)n1 C(=O)(C(C)(C)CC1CCOCC1)N(CCCNC(=O)C(F)n1ccnc1)CC N1(C(C2CC(C)(C)O2)=O)CCC2(CCCN(C(=O)COC(F)(F)C(F)(F)F)C2)C1 C12CN(CC13CCOCC3)S(=O)(=O)C2.CC(C)CC(C)CC=O.CC[Si](C)(C)C C1(C(=O)NC2CCC(NC(C3(C)CC3(F)Cl)=O)CC2)CC2C=CC1C21CC1 N1(C(c2cc(F)cs2)=O)CCC2CN(C(=O)C(F)(F)C(F)F)CC2C1 c1(NC(c2cnn3c2OCC3)c2n(CC=C)nnn2)cc(C)cnc1C CC1(CC(=O)NC2CCN(C(C3(n4ccnc4)CCCC3)=O)C2)CCC(=O)N1 C=CCCC(C)N=c1[nH]c(=NCc2cc3c(s2)CCCC3)[nH]c2ccc(Cl)cc12 N1(C(C2(CC=C)COC2)=O)CCC(NC(c2cccc(OC)c2)=O)C(F)C1 c1(C(N2CC(CNC(C(C(C)C)NC(=O)OC)=O)C2)=O)cnc2nccnc2c1 c1(C(=O)NC2CCC(NC(c3c(C)cc[nH]c3=N)=O)C2)coc2c(F)cccc12 CCC(C)C(O)C(C)C(=O)NC1(C2CCCN2C(=O)CCCC2CCC2)CC1 C1(C(N(CCC(C)O)C)=O)CCCN(C(c2ccncc2)=O)C1 C1(C(=O)OC)CC(C(F)(F)F)CN(C(=O)COc2cc(C)cc(C)c2)C1 c1(OC)nn(C)cc1CNC(=O)C(CCSC)NC(C1SCC=C1C)=O CC(C(C)(C)O)N(C(=O)CN(C(=O)CC1CCCN1C)C1CCC1)C C1(C(N(CC(CC)NC(=O)CNC(c2ccncc2)=O)C)=O)(OC)CCSC1 N1(C(=O)NCC2(C(C)(C)C)CCCCC2)CCC(C(F)(F)F)C(CN)C1 c1(C(=O)NCC2C(C(=O)NCC3(C)CNC(=O)O3)OCC2)cccc(C#N)c1 C(C)(CC(=O)NC(C1(CNC(=O)CCOCC2CCC2)CC1)C)SC CC1CN(C(=O)CCNC(=O)CO)CCC1C(=O)NCCC1CCCN(C)C1 c1(C(N(CCCN(C(C2CC(C)NC(=O)C2)=O)C)C)=O)cnn2c1CC(C)CC2 C1(CNC(c2cc(C)ncn2)=O)CCC12CCN(C(=O)Cc1c[nH]nc1O)CC2 C(=O)(CCC(C)CN(C)C)NC(C(=O)NC(CC(C)C)CO)C1CCC1 N12CCc3onc(c3C1)C2=O.N1(CC=CC(=O)OCC)CCC(N2CCCC2)C1 c1(C(=O)NC(CCN(C(CCCCSC)=O)C)C)cc(C)c(C)cc1Cl C(CC(=O)NCC(C)CN(C)C(c1cc(OC)cc(C)n1)=O)(C(C)C)OCC c1(OC)ccc(C(F)F)cc1C(=O)NCC(C1CC1)NC(c1n[nH]c(C)c1Cl)=O C(C)(N=c1nc[nH]cc1C#N)C1CCCN(C(c2ncc(C)nc2)=O)C1 C1(C(=O)NCCC2CC(NC(CCOC(C)=O)=O)C2)CCc2nc(C)ncc2C1 c1(NC(C(CNC(C(CC=C)CC)=O)C)=O)cnc2[nH]cnc2c1 C(=O)(CCS(N)(=O)=O)NC1C=CC(CC(=O)NCc2cc(COC)no2)C1 N1(C(C(C2CCCO2)NC(c2ccncc2)=O)=O)CCOC(C2CCC2)C1 C1(NC(CS(CC)=O)=O)CN(C(=O)CCNC(c2ncccc2O)=O)CC12CC2 N1(C(c2c(C)nc(C(C)C)s2)=O)CCN(C(=O)CNC(=O)NC2CC2)C(CF)C1 CC(CSc1ccccc1)C(=O)NCC(CNC(c1cc(C(F)F)[nH]n1)=O)CO c1(CC)ncc(C(=O)NC2CC(C(C)NC(=O)CC3CSCCO3)C2)[nH]1 c1(C(C(=O)NCC(CNC(CCC(=C)Cl)=O)F)C)ccc(Cl)c(Cl)c1 C1(NC(c2c[nH]c(Br)c2)=O)CN(C(c2cccnc2C(F)(F)F)=O)CC12CC2 Cc1cccc2c(C(=O)N(C)Cc3cn(-c4ccccc4Cl)nn3)cnn12 c1(C(=O)NC2CCC(CNC(CNC=O)=O)CC2)cc(F)c(F)cc1I c1(COC)nc(Cl)cc(=NC2CCN(C(C3CCCC3C)=O)CC2CC)[nH]1 c1(OC)ccnc(CC(=O)NCC#CC2CC2)c1OC c1(CC(=O)NCC(C)(C2CC2)NC(c2cc(Br)co2)=O)ncccc1O Cc1cc(C(=O)NC2COCC2NC(=O)Cc2ccc(C)s2)c(F)cc1N C1(COC)(NC(C2(OC)CCOC2)=O)CCN(C(c2cncc(C(C)=O)c2)=O)C1 N1(C(CN(C)C(c2cccs2)=O)=O)CC2(CCN(C(C3CCCC(=O)O3)=O)C2)C1 C1(OCCC(=O)NCCN(C2CCCC2)C(=O)CC2CC=CCC2)CCCOC1 N1(C(CC2CC(OC)C2)=O)CCC(O)C(N(C(=O)CC2CCCC(F)(F)C2)C)C1 C1(NC(Cn2c(CCC)ncc2)=O)CN(C(=O)CS(=O)(=O)CC)CC1N=[N+]=[N-] N1(C(CCNC(C)=O)=O)C2CCC1CC(F)(CNC(C1(C(F)F)CCC1)=O)C2 N1(C(C=CCC)=O)CCC2C(CCN2C(=O)C=CCN2CCCCC2)C1 CCS(=O)(=O)c1ccc(CC(=O)N=C2CCN(C)CCN2)cc1 C1(CC(=O)NCCCCN(C(C(N2CCOC2=O)C)=O)C)CSCCS1 C1(C)(CC)CC(NC(=O)C2=CC(C)(C)C2)CN1C(=O)Cc1sc(O)nc1O O(NC(=O)C(CC(C)C)ONC(C1(C)CCCN1C)=O)CC=C(C)C CCCC(C(=O)NC(CNC(c1ncncc1Br)=O)CC)OC C1(CC(=O)N(C)CC2CCN(C(=O)CCc3cn(C)cn3)C2)CCCS(=O)(=O)C1 C12(C(=O)NC3CCC(NC(Cc4c(C)n[nH]c4)=O)CC3)CCCC1CS(=O)(=O)C2 C1(c2nc(OC)c(C)s2)CCCN1N1CCC(C(N2CCCCCC2)=O)CC1 C1(C(N2C(C)CCC2C)=O)CC2(CC(NC(=O)Cc3cnn(C)c3)C2)C1 C(=O)(C(CO)NC(c1cc[nH]n1)=O)NCC(CC)N1CCCC1 C=CC(CCC)CC(=O)N(C1CCN(C(=O)Cc2ccc(OCC)nc2)C1)CC C1(NC(c2c(C)nc(C(C)(C)C)s2)=O)CCCN(C(=O)Cc2ccsc2C)C1C c1(N(C(=O)CNC(c2ccsc2)=O)C)c(C(=O)O)cccc1C(=O)O c1(C(=O)NCC(CC(C)C)NC(=O)Cn2ncnn2)ccn2c1CSCC2 c1(C(=O)NC(C)CCCNC(C2(C)CCC(C)C2)=O)ccncc1N=[N+]=[N-] O(NC(=O)CC=CCNC(C1CCC(C(N)=O)O1)=O)CCCC=C Cc1ccc(C(N2CCCCC2Cn2cccn2)C(=O)NC2CC2)cc1F c1(C(N2CC(NC(COCC=C)=O)C(C(F)F)C2)=O)n[nH]c2c(OC)cccc12 C12(C(C)NC(=O)C(O)C3CN(C(c4cn(C)nn4)=O)C3)CCC(CO1)C2 O=C(CC1CCOc2ccccc21)NCC1(NC(C2CCS2(=O)=O)=O)CCCC1 N1(C(C=C(C)c2ccco2)=O)CCN(C(C23CCC2C3)=O)CC1C(C)(C)C c1(CCC(N2CC(NC(C(C)(C3CCOCC3)OC)=O)C2)=O)cc(C)nc(C)c1 N#CC1(F)CCN(C(=O)C(C2CC2)NC(=O)CC2CCCC(=O)N2)C1 C1(NC(=O)C=Cc2ccco2)C2CCC1N(C(=O)CNC(c1ccco1)=O)C2 Cc1ncc(CCC(=O)NCC2CCN(C(=O)Cc3cnn(C)n3)C2)s1 C(=O)(CC(C(F)(F)F)c1cccc(F)c1)NC(CNC(c1c(C)scn1)=O)CO CCCCCC(CC)C(=O)N(CCC(=O)N(C)CCOC(C)=O)CCCO C(c1ccc(OC)cc1C)=CC(=O)NCCNC(C1(SCC)CC1)=O c1(C(N2CCN(C)C(CNC(C3(C(F)(F)F)CC3)=O)C2)=O)cnn2ccccc12 c1(CC(=O)NCCNC(c2c(C(C)=O)cn(C)n2)=O)ccc(S(C)=O)cc1 CCC(C#N)C(=O)NCc1ccc(C(N2CC(NC(=O)NC)C2)=O)cc1 N1(C(C(C)NC(=O)OCC)=O)CC2CC2(CNC(=O)C(C)(C)O)C1 N1(C(C(Cn2cccn2)NC(c2ccn(C)n2)=O)=O)CCCC(CO)CC1 CC(C)C(F)(CNC(C1(C)CNC(=O)C1)=O)C(=O)N1CC2CCC2C1 C(C(=O)N=c1cc[nH]c(C)c1F)C1CCC(NC(C(CC(C)C)NC(C)=O)=O)C1 c1(N2CCCC3(N(C)CCC3)C2)cc2ccc(Br)cc2c(Cl)n1 c1(NC(C(CNC(=O)CSc2cn[nH]c2)O)=O)cccc2[nH]ccc12 C(C(C(=O)N1CCC(c2nc[nH]n2)C1)NC(=O)CCc1cnco1)N(C)C C1(NC(CN(C)C(N)=O)=O)C2CCCN(C(C3OCCN(C)C3=O)=O)C2C1(C)C CC1(C(=O)NCC(C)(C2CC2)NC(C2CCS(=O)(=O)CC2)=O)CC2CCC1C2 c1(N(CC(CN(C(=O)CC2CC(=O)NC(=O)C2)C)O)C)ncc2ccccc2n1 Nc1cc(C(=O)NC2CCN(C(C3CCCOC3)=O)C2)ncc1Cl c1(NC(=O)NC(C#CCC)(C)C)nc2ccc(N)cc2s1 c1(OC2CN(C(=O)NC3C(C)(C(C)C)C3)C2)ccc(Br)cc1 c1(NC(CCCNC)C)nc(C(C)C)ncc1Br.CS C(=O)(N=c1nc(-c2ccccc2Cl)[nH]s1)NC1C(SCC)CCC1 C1(NC(c2c(OC)csc2)=O)CN(C(c2cccc(F)c2N)=O)CC1(C)C N1(CC)CCCCC1C(=O)N(CCCc1scnc1C)C CC1(CNC(=O)C=CCn2cncn2)CCCN(C(C2OCC3CCCC23)=O)C1 C1(C(=O)NCC2(C(=O)NC3(C(=O)OC)CC3)CC2)CC1(F)F C(C(C)(C)C(=O)N1CCCC(CN(C(=O)CC2(OC)CC2)C)C1)OC N1(C(CC(CC)OC)=O)CCC2(CCC(C(=O)NCCC3CCCC34CC4)O2)CC1 c1(C(C)C)nc(C(=O)N(CC(O)CNC(c2ncoc2Br)=O)C)co1 c1(OC)ccc(CO)cc1C(=O)NC1CC(NC(=O)CC2CCCC2(F)F)C1 C(=O)(CCCCN(C)C(C)C)NCC1(O)CC(NC(C2CN(CC(C)C)C2)=O)C1 c1(C(=O)NCC2C=CCN2C(c2cc3c(s2)CCC3)=O)ccc2cnccc2n1 CCC(CNC(=O)C(C)CN(C)C(C1CNC(=O)N1)=O)(CC)CO c1(C(N(C(CNC(Cn2c(C)ccn2)=O)C2CC2)C)=O)coc2c1C(O)CCC2 N1(CCCCCC)C(=O)CCN(C2CC(C)(C)Oc3cc(F)cc(F)c32)C1=O C1(C(N2CCN(CC(N3CC(C)OC(C)C3)=O)CC2)=O)(CN)CC2CCC1CC2 CCC(C#N)C(=O)NCC(C)N(C(=O)CCCc1cnn[nH]1)C Cc1cc(C(N2CCCC(C(C)NC(c3ccc(Cl)s3)=O)C2)=O)cc(C)c1C#N N1(C(C2N(C(C)=O)CC(O)C2)=O)CCC(NC(c2ccnnc2)=O)C12CCC2 C(=O)(C(C)(C)C(F)F)N1CCCC(CNC(C(C(C)C)N(CC)CC)=O)C1 c1(C(N(CC(CNC(C2(COC)CC=CCC2)=O)(C)C)C)=O)cc(C)cc(C)c1 C(=O)(CC(O)C(C)CC)N1CCN(C2CN(N3OCC(O)C3=O)C2)CC1.CC C(=O)(CC(CCCC(C)C)NC(=O)C(c1ccccc1CC)O)OCC C(CCCCC1CC1)(C(=O)NCCOCC1CC1)N1C(C(=O)NC)CCC1 c1(C(=O)NCC23CC(CNC(C4CC(C#C)(O)C4)=O)(OC2)C3)cc(Cl)cc(Cl)c1 CCCC(CNC(C1CN(C)CCN1C(C1CC(=O)C12CCC2)=O)=O)CCO CC(C)(C)CCCC(=O)NC(CC(=O)N1CCC(n2cnnn2)C1)C(F)(F)F C1(NC(c2c(C)n[nH]c2)=O)CCC2CN(C(C3CC4(C3)CC4(F)F)=O)CCC2C1 C(=O)(C(C#N)C(C)(C)C)NCCCC(C)(C)NC(=O)C1=CCCC1 CC(C)C(CCc1ccccc1)C(=O)NC(CNC(=O)CNS(N)(=O)=O)C1CC1 C(=O)(C1COc2ccc(Cl)cc21)N1C(C)CC(NC(c2cnoc2)=O)CC1 N1(C(CNC(CC)=O)=O)CCOCC1CN(C(=O)C(C)NC(=O)CC(C)(C)C)C CCC(CC(=O)N1CC(F)(F)CC1OCC(=O)Oc1cnn(C)c1)C(F)F N1(C(COCCOC)=O)CC=CC(CNC(=O)Cc2ccncc2Cl)C1 c1(C(=O)NC2CCC(CCNC(CCCSCC)=O)C2)ccccc1F CC(C(=O)N(C1CCCN(C(c2ccc(CS(C)(=O)=O)cc2)=O)C1)C)S(N)(=O)=O C(c1ccc(C)cc1)=CC(=O)NC1CCCC(NC(C2(CC#C)CC2)=O)C1 N1(C(c2n(CC)ccc2)=O)CC2(CCC(CNC(C3(C4CC4)CCCO3)=O)O2)C1 c12ccc(c(F)c1)C(=O)N1CCCC(O)(C1)CNC2=O.S(=O)(=O)(C1CC1)N.CCN N1(C(c2nc(C)sc2)=O)CC2CC1CCC2NC(c1cccc(O)n1)=O N1(C(CCOC)=O)CC(C(=O)NCCc2c(C)noc2C)C(C2CC2)C1 C(=O)(C1=Cc2cc(Br)ccc2OC1)NCC1N(C(CN(C)CC)=O)CCC1 n1(CC(=O)NCCCN(C)C(c2cnc(S)n2C)=O)nc2n(c(=O)c1=O)CCC2 c1(COc2cccc(C(=O)OC3(C(=O)OC)CCCC3)c2)ccc(F)c(C#N)c1 Cc1cnc(C(N2CCC(C(=O)NCC3(O)CCCCCC3)C23CC3)=O)c[n+]1[O-] CC(C)CCC=CC(N1CCC(NC(C2(Cl)CC2(F)F)=O)C1)=O N1(C(c2ccc(C)nc2C)=O)CC(NC(C2CC(C)(O)C2)=O)C(S(C)(=O)=O)C1 C1(CNC(C2(F)CC2)=O)COC2(COCCN(C(C3(F)CCCC=C3F)=O)C2)C1 C1(C(=O)NCC2N(C(CSCC)=O)CCC2CC)CC2CC1CC2O C(=O)(CCCC(C)(c1nnnn1C1COC1)NC(c1ccc(Br)cc1)C)OC CCCCC(C)C(=O)NC1C=CCN(C(=O)CSc2nnnn2CC(F)(F)F)C1 C(CC(C)(C)C)N(C(c1ccn(C(C)(C)C)c1)C(=O)NC1CC(F)(F)C1)CC [N-]=[N+]=NCCCC(=O)N1CC2CC(C1)N2C(=O)C(F)C1CCOC1 c1(C(=O)NCC(C(=O)NC(C)C(C)(C)O)C)ccn(C)c(=O)c1 N1(C(c2cccc(CC)c2)=O)CCC2(CCC2)C(NC(C2CC2COC)=O)C1 c1(C(C2(OC)CCN(C(C(=O)OCC=C)=O)C2)N(C)C)ccc(C(F)F)c(Cl)c1 Cc1ccnc(CN(C)C(c2coc(C(C)NC(=O)C(C)CC3CC3)n2)=O)c1 c1(OC)ccc(C=CC(=O)NCC2CCN2C(c2nc(Cl)sc2Cl)=O)cc1OC C(CC(=O)NC1(CNC(c2oc(C)cc2C)=O)CC1)(C1=CCCC1)OCC N1(C(C(CO)N(C)C)=O)CC(CNC(C2(C)SCCCS2)=O)C2(CC2)C1 C1(C(N(C)Cc2cccc(OC)c2)=O)CCCN(Cc2ccc(F)c(I)c2)CC1 C1(C(N2C(C(=O)Nc3cnn(CCF)c3)C=CC2)=O)CCC2(CC1)CC2 C1(CC)CCN(C(=O)CC(CNC(c2cccc(=O)o2)=O)C2CCC2)C1C c1(Cn2c(CCC(C)N(CCC)C)nc(-c3ccc(C)o3)n2)cc(Cl)ccc1Cl N1(C(CC2(CC)CCC2)=O)CCC(O)(CN(C)C(c2ccccc2OC)=O)C1 N#CC1(C(N2CCC(C3CCCN3c3ncccn3)C2)=O)CC2CCC1CC2 Cc1ccc(C(N2C3CN(C(=O)C(C)(C)c4ccccc4)CC23)=O)cc1Cl Cc1cc2cccc(C(=O)NC3CC(C(N4CCN5CCCCC5C4)=O)C3)c2[nH]1 C(C(C)(C)C1=CCCC1)N1CC(CCCC(=O)NC23CCC(C(=O)OC)(CC2)C3)C1 N1(C(C(C)Oc2cccc(C)c2)=O)CCC(NC(=O)C(F)C2CCC2)C12CC2 N(C(=NCCF)NCc1ccccc1)CC1C(C(C2(O)CCCOC2)O)CC1 c1(C(=O)OC)ccc(NCC2CC2)cc1OC(F)(F)C(F)(F)F N1(C(CSCC)=O)CCC(NC(c2cc(Br)co2)=O)C(CC)C1 N1(C(c2ccc(C3CC3)s2)=O)CC(C2CN(C(c3ncc4[nH]ncc4n3)=O)C2)C1 C12(CCNC(C(C)(C)n3cccn3)=O)CCC1CN(C(C1(CO)CC1)=O)C2 C1(C)(NC(CC(C)N(C(=O)CC2NC(=O)NC2=O)C)=O)CCC(C)C1 C(=O)(C(CC1CC1)NC(=O)CN1CC2CC2C1)NC(c1ccnn1C)CC c1(CC)cccc(C(=O)NC2CC(NC(C3CCC34CCC4)=O)C(O)C2)c1O n1(CCC(N2CC(CC=C)(NC(=O)CC3C=CCC3)C2)=O)cnc([N+](=O)[O-])c1 c1(C(=O)NC2CN(C(COCCC#C)=O)CC2C(F)F)cc2cc(F)ccc2o1 CCCC(C(=O)NC1(COC)CN(C(=O)CC2CCC2)C1)n1ccc(C2CC2)n1 N1(C(C2(C#N)CCOC2)=O)CC2(COC(CNC(=O)C(=O)NCC(F)F)C2)C1 CN1CCOC(CNC(C2CC(O)CN2C(=O)CCc2cccn2C)=O)C1 C12(NC(C3CCCCC(C)(C)C3)=O)CCCC1(F)CN(C(=O)C=CCO)C2 c1(OC)cc(C(=O)NCC(c2ccccc2)N(C)C(C2CC2C)=O)cc(Cl)c1 CC#CCC(C(=O)N(C)CC1CC1C)NC(=O)CCC(C)CC Cc1c(-c2nc(Cc3ccc(Br)cc3)nn2CC(N)=O)cnc2ccnn12 CCCC(C(=O)NC1(CCNC(c2cc(CCO)on2)=O)CCC1)NC(C)=O C1(C(=O)OC(C(=O)Nc2ccc(C(C)=O)cc2)C)CCc2cnn(C(C)C)c2C1 N1(C(C(CC#C)C2CC2)=O)CCOCCC1C(=O)NC(C)Cc1cccs1 CC(CF)CC(=O)N(C)CCN(C)C(c1nc(C(C)(F)F)cs1)=O Cc1nc(O)nc(C)c1CC(=O)NCC(CNC(C1(Cl)CCC1)=O)CO c1(N2C(C(=O)Nc3ncc(Cl)cc3O)CC3(CC3)C2)ncnc2cc(F)ccc12 C1(C(N(C)CC2(NC(c3cnn(C(C)C)c3N)=O)CC2)=O)CCCC1S(C)(=O)=O N1(C(CCOC)=O)CCCC(CCNC(c2cc(SC)oc2C)=O)CC1 C(C(=O)N(C)OC1CCCC1)(C1CCCCO1)NC(C1C(C(C)C)C1)=O N1(C(C(CC(=C)Cl)NC(=O)C(C(C)C)NC(C)=O)=O)CC2(CCC(=O)O2)C1 CN1CCC(C(=O)NCCC2(C)CCN(C(c3ccc[n+]([O-])c3)=O)C2)CC1=O CCCC(C)(C)C(=O)NCC1CN(C(=O)C(CCOC)OC)CCCO1 N1(C(CC(CC2CC2)NC(c2cc(C)nn2C)=O)=O)CC(=O)N(C)CC1C C(C(N=[N+]=[N-])C(=O)NC1CCC(C(N2CC(CC(F)F)C2)=O)C1)OCC C1(NC(=O)NC2CCC(CC#N)C2)CC2CC1CC2F C1(CC)CN(C(C23CC(OC)C2C3)=O)CCN1C(=O)COC1CCCC1 C(C)(C)(C(C)CC(=O)NCCc1c[nH]nc1O)NC(c1ccn(COC)n1)=O c1(C(N2C(CNC(c3cncc(N)n3)=O)CC(F)C2)=O)cc(F)c(F)cc1F C(C)(C(CC(=O)NC12CC(F)(C1)C2)NC(c1cc(N)cc(F)c1)=O)OC C(CCCCCNC(C1CC2CC1C2)=O)N(C)C(C1CC1F)=O C(=O)(CCCCC#Cc1ccccc1)N(C1CCN(C(C(CC)C)=O)CC1)C c1(CCCNC(=O)C(N2CCN(c3cccc(Cl)n3)CC2)=O)ccc(O)cc1 C1(CNC(c2c(C(=O)OC)scc2)=O)C2CN(C(C3CC4(CCC4)C3)=O)CC12 c1(C(C)=O)cccc(C(=O)N(CC(C)CNC(C2(C)CSC2)=O)C)c1 c1(CCC(=O)NC(C2CN(C(CCC#C)=O)C2)C)ccc(F)c(F)c1 C1(NC(C(C)SCC)=O)CCN(C(C23CCC2CC3)=O)C(C)C1 c1(C(N2CC(NC(C3CC(C)(C)C3)=O)C3C2C3)=O)cnn2cc(Br)cnc12 S(=O)(=O)(c1ccc([N+](=O)[O-])c(Cl)c1)NC1C(C(=O)Nc2cncs2)C1 CS(C)(=O)=NC(=O)c1cc(C2OCCO2)on1 N1(C(C(n2cc(Br)cn2)C)=O)CCCCC(CNC(c2cncnc2)=O)CC1 C1(NC(C2CCC(C)C2)=O)CC1C1CCCN(C(c2ccc3scnc3c2)=O)C1 N1(C(c2c(CC)cco2)=O)CCSCC1C(=O)NCCc1cnnn1C N(C(=NCCC1CCC(=O)N1)NCc1c(Br)nnn1C)C(C)C1CC1 N1(C(C=CC(C)(C)SC)=O)CCC(N=[N+]=[N-])(C(N2CC(C(C)N(C)C)C2)=O)C1 c1(CC(=O)NCC(C)(C)NC(c2cc(F)cc(N)c2F)=O)ccn2cncc2c1 c1(NC(C)=O)ccc(C(=O)NC(C)Cc2cccc(C(C)(C)C)c2)nc1 N1(C(CN(C)CC)=O)CCN(C(C23CCCC2C3(F)F)=O)CC1CCOC c1(C(c2n(CCC)nnn2)Nc2ccc(C)nc2)ccc(C(C)CC)cc1 Cc1ncn2ccc(C(=O)NCC3(CCNC(=O)C=Cc4cccs4)CC3)cc12 Cc1cc(C(=O)N(CCCOCCNC(c2ccn(C)c2)=O)C)c2nccn2c1 N1(C(c2[nH]c(=NC)sc2)=O)C2CCC1C(C)C(NC(=O)C(C)S(C)(=O)=O)C2 C1(O)(CCNC(C(C)(C)C2CCCC2)=O)CCN(C(C2C=CCCC2)=O)C1 C(c1ccccc1)=C(CC)C(=O)OC(C)C(=O)C1CCC1 c1(NC(C2C(C(=O)Nc3c(C#N)cno3)C2)=O)ccc(F)c(F)c1O c1(C(=O)NCCOCCNC(=O)CCc2ccc(F)nc2)cccc(F)c1CO C1(C)(CNC(C(CC)(C)CC)=O)CC(F)(F)CN1C(=O)Cc1ccc(C)c(F)c1 c1(C(=O)NCCC(C)(C)NC(CSCC#C)=O)cc(C)cc(Br)c1F c1(N2CCC(C)(CN(C)C)C2)ccc(S(=O)(=O)NCc2c[nH]ccc2=N)c(Cl)c1 CN1C(=O)NC(C2CCN(CC(=O)Nc3ccc(=N)[nH]c3)CC2)C1=O C1(C(=O)NC2CC2C(=O)NC2CN(Cc3ccco3)C2)CC2CCC1C2 CC1CCCc2nc(C(N3CCOC(CCNC(=O)C(C)(C)C#N)C3)=O)cn21 c1(C2C(CN(CCCCC)CC(=O)NCCCNC(=O)OC)C2)cnc(C)[nH]1 CC1CCN(C(C2CC(=O)N2)=O)CC1CNC(=O)C(c1ccc(F)cc1)F C(C(C)(CC)N(C(CC)CC)C1CCCC1)NCC(=O)NCC(=O)NC(=O)NC c1(OC)nc(N2CCC(C)(NC(C3CCC(C)CC3)=O)CC2)nc(C)c1F C(=O)(CCC(C)(C)F)N1CC(C)C(CCNC(c2ncccc2C(C)(C)C)=O)C1 c1(NCC)ccc(S(=O)(=O)NC(C2CCN(S(C)(=O)=O)CC2)C)c(Br)c1 C(c1nc2ccccc2o1)=CC(=O)NCC1CCN(C(=O)CCF)C12CC2 c1(C(=O)NC2(CO)CCN(C(=O)CSc3n[nH]c(O)n3)C2)cnn2cccnc12 CC1(CNC(C2(C)CC2(F)F)=O)CN(C(=O)COc2ccc(F)cc2Cl)CCO1 Cc1ccc2c(c1)CC(NC(CN1C(SCC3CCS(=O)(=O)C3)CCCC1)=O)O2 C#CC(CNC(=O)C(C)N(C(c1scnc1C)=O)C1CC1)CC(C)(C)C c1(NC(C(CNC(c2ccc(CC)[nH]2)=O)O)=O)ccnc(OC)c1 N1(C(c2c(CC)nccc2)=O)CCC2CC2(C(=O)NC2CCNC(=O)C2)CC1 C12(NC(c3[nH]cc(CC)c3)=O)CCCCC1CN(C(c1nocc1Cl)=O)C2 N1(Cc2nc(C)cc(C)n2)CC=C(CCNC(c2cc(C3CC3)n(C)n2)=O)CC1 c1(C(=O)NC(C)CCNC(=O)CC(F)(F)Cl)cc2cn[nH]c2cn1 c1(C(=O)NCCCC2(NC(CC3(C)CC3)=O)CC2)cc2n(n1)CCCO2 C1(CNC(C=CC(C)(C)C)=O)CCCCN1C(c1ccc(-n2ccnn2)cc1)=O c1(-n2c(CC3CCC(OC)CC3)nc(CC(CC)C)n2)cccc2nc[nH]c12 C12(NC(C(C)NC(CC)=O)=O)CCCC1N(C(C1CCCC3CC13)=O)CCC2 c1(C(=O)OCC)nc(=NCC(C)CNC(C2CCC3CC3CC2)=O)cc[nH]1 c1(C(=O)NC2(CO)CCCN(C(C3CC(N=[N+]=[N-])C3)=O)C2)nc2c(s1)COCC2 C(C(=O)NCc1ccc(C)nc1)(C(C)CC)NC(c1ccc(NC)cc1)=O c1(N2CCC(CCCC)C2)nc(N2CCC(CC(F)(F)F)C2)cc(C)n1 C=CC(C)(CC)C(=O)NCC(C)(CO)NC(=O)CCOC1CC1 CC1CCCC1N=c1nc(N2CCC(C)(N3CCC3)CC2)c2ccccc2[nH]1 c1(C(=O)NC(c2cccc(C)c2)CNC(C(CC)F)=O)ccc(C2CC2)nc1O c1(OC)ccc(C(C)Nc2ccc(NC(C3COC(=O)N3)=O)cn2)cc1 C1(F)(CNC(C(C)OCC2CC2)=O)CCN(C(=O)CCc2ccccc2Cl)C1 CCCC(O)CC(=O)NC1CCCC1NC(c1cn(CCC2CC2)nn1)=O C1(SC)COCC1NC(=O)CCCN(C(=O)C(C)OCC1CC1)C C1(NC(C=CCC)=O)CC2CN(C(c3cc[nH]c3C(C)C)=O)CC12 CC1CC(N=c2[nH]c(=NCc3cocn3)c3cc(F)cc(F)c3[nH]2)CS1 C#CC1(C(=O)Nc2cccc(OC)c2C)CCN(C(=O)CC2CC(CC)=NO2)C1 CCCC(CC)C(=O)N(CCN(C(c1cnc(CC(C)(C)C)s1)=O)CC)CC N1(C(C(c2ccc(Br)cc2O)=O)=O)CCC2(CC1)OCCC2O N1(C(c2c(OC)cc(Cl)cc2)=O)CC2CS(=O)(=O)CC2(NC(=O)C=C(C)C)C1 c12c(sc(C)c1C)N(N(CC)CC)C2=O.C1(C=O)CC(n2ccnn2)C1.C1(C)CC1 C1(COC)(NC(c2cc(CO)[nH]n2)=O)CN(C(=O)CCc2ccc(Cl)s2)C1 Cc1cc(C(F)F)oc1C(=O)NCC(CO)NC(=O)Cc1cnccn1 c1(CNC(C2(C(N)=O)CC2)=O)ccc2c(c1)CCN(C(C1CC3CCC3C1)=O)C2 c1(OC)ncc(CN2CCC(NC(=O)Cc3ccc(Cl)cn3)C(F)C2)cc1C N1(CCC(N2CC(CC)C(N)CC2)=O)C(=O)Cc2ccccc2C1=O N1(C(C(C(C)C)CNC(=O)CC(C)n2ccnc2)=O)CC2(C)CCC2(C)C1 N1(C(CC(CC)C)=O)CCC2(CCOC2)C(CNC(=O)C2=CCC(C)CC2)C1 C1(O)(CNC(CC(C)N(C)C)=O)CCN(C(=O)Cc2cc[nH]c2)C1 O=C(NOCCO)C1c2c[nH]nc2CN1C(=O)C1=CC2C=CC1C2 CC(C)C(C#N)C(=O)N(C(C)CCNC(c1cccc(F)c1Br)=O)C C1(O)(CN(C(=O)Cn2cc(Cl)cn2)C)CCN(C(=O)Cn2cnnc2)C1 CC(C)CC(CNC(C12CCC(C)(C1)OC2)=O)C(=O)NC1CC12CC(O)C2 CC1COC(CO)CN1C(c1c[nH]nc1CNC(c1ncncc1Cl)=O)=O C1(CNC(=O)NC(c2cccc(OC(F)(F)F)c2)CO)CC2CCCC2O1 n1(CC(=O)N(CC(CN(C(CCCc2ccc(C)s2)=O)C)O)C)cc(Cl)c(C)n1 c1(C(C(=O)NC(CC)(C)C)N(C2CCCC2C#N)C)ccncc1CC c1(C2CCN(C(=O)NCC3(CSC)CC3)C2)nc2ccccc2o1 C(=O)(CC1=CCCCC1)NC12CCC(NC(=O)Nc3c(C)c(F)ccc3)(CC1)C2 c1(C(=O)NCC2C(NC(C(CSC)C)=O)CC2)nc(C2CC2)ncc1Cl CC1(C)C2CCC1(C(=O)NC13CCCN(C(c4cccnc4N)=O)CC1C3)CC2 C(C(C(=O)N(C)CCNC(C1CCCN1CCC(C)C)=O)OC)OC c1(CN(C(=O)CC2C(C)(C)C2(C)C)C)nnc2n1CCCC2C(F)(F)F c1(OC)nccc(C(=O)N(C2(CC(=O)NCCN3CCNC3=O)CC2)C)n1 c1(C(=O)NC2CCC(CNC(C(CC)F)=O)C2)ccnc2[nH]c(CC3CC3)nc12 N1(C(CC2C(CC)C2)=O)CCN(C(C2(c3ccccc3)CC2(C)C)=O)CC1C c1(C(=O)NC2CC(CNC(C(CC=CC)C)=O)C2)c(O)nnc2c1COCC2 n1(CC)cc(Cl)cc1C(=O)N(CCNC(c1sc(OC)nc1Cl)=O)C1CC1 C1(C(N(CC(C)(C)NC(=O)CN2CCCCC2)C)=O)CC12CCC1(CC1)CC2 C1(CCSC(F)(F)F)CC2CN(CC(=O)OC(CCCCC)=O)CCN2C1=O C(=O)(C(C)(C)C(F)(F)F)N1C(CNC(c2c(O)ccc(CC)c2)=O)CC1 C1(C(C)(C)NC(C(N2CCOC2=O)C)=O)CCCN1C(=O)CCn1cnnn1 N1(C(CCC2CCC(=O)N2)=O)CC2CCC1CN2C(c1nccc(Cl)c1O)=O N(C1CCCNc2ccccc21)c1cccc(CC)c1.OC c1(C(=O)NCC2C(NC(C(CSC)C)=O)CCCC2)ncnc2ccsc12 CCC(CNC(C1(CCOC)CCC1)=O)(CC)NC(=O)C(c1ccc(C)cc1)C Cn1c(C(=O)NCC2CC2NC(c2cc(Cl)no2)=O)cc2ccccc12 N1(C(c2ccc3c(n2)OCCO3)=O)CCC2(CCN(C(C3CC(O)C3)=O)CC2)C1 N(C)(S(=O)(=O)NCc1cccc(Cl)c1)C(C1CCCC1)C c1(NC)ccccc1C(=O)NC1CCC1C(=O)NC1CCC(C(N)=O)C1 c1(C(N2C(CC)CN(C(C34CCCCC3OCC4)=O)CC2)=O)cc(C)c(C#N)cn1 c1(C(=O)NC(C(=O)OCC)C2CC2)ccoc1CNC(c1cncn1C)=O c1(NCC2(C#C)CNC2)cc(SC2CCCC2)ccn1 c1(C(N2CCC(S(C)(=N)=O)CC2)C(=O)NCC=C)cc2ccnc(Cl)c2s1 c1(C(N(CCC(=O)O)CC)=O)ccc(Br)c2c1OCCC2 N1(C(c2nnc(C)s2)C)CCC2(CC1)CC2(C)C(=O)N(C)C Cc1cc(C(C)(C)C(=O)NCCN(C(=O)CC(O)c2cc(C)cs2)C)cs1 CC1Cc2ccc(F)cc2C1NC(=O)Cc1c[nH]c2ccccc12 c1(C(N2C(CCNC(=O)CC34CCCC3C4)CCC2)=O)cc2n(n1)CCNC2=O c1(CNC(C(CC)O)=O)ccc(C(C)NC(=O)CNC(=O)C2CC2)cc1 c1(C(=O)NCCC(CC)(CC)NC(=O)C(O)CC(C)C)cn2c(C)cccc2n1 C12(C(N3C(C)CCC(CNC(C(C)OCC=C)=O)C3)=O)C3C4C1C1C2C3C41C c1(NC(CCCC)c2nnnn2CC2CCOC2)ccc(SC(F)F)cc1 C(=O)(C1=CCCOC1)N1CCC(N(C(Cc2c(COC)cccc2)=O)C)C1 C1(CCNC(CSCCC)=O)C(C)CCCN1C(c1scnc1C)=O Cc1nccc(Cl)c1C(N1CC2C(NC(c3ccc[nH]3)=O)C2C1)=O C1(C(=O)Nc2ccc(COC)cc2)CCC2(CC2)N1C(=O)C=Cc1cc[nH]c1 C1(C(N(CCCCO)CC)=O)CC(=O)CN1C(=O)C=C(C)C C1(NC(c2cc(CC)[nH]n2)=O)CC2CC(NC(c3cscc3C(F)(F)F)=O)C1C2 c1(N(C)C)ccc(S(=O)(=O)NCC(N2CCC3NCCC23)=O)cc1[N+](=O)[O-] C(=O)(CCC(F)(F)F)NC(C(=O)NCC(CO)N(C)C)CCF Cc1cccc(Br)c1C(C(=O)N(C)CCC1CCCO1)NC(C1CC1Cl)=O c1(C(N2CCC(C=C)(C(=O)NOCCN(C)C)C2)=O)cccc2cc[nH]c12 C#CC1(NC(=O)CC2(CNC(C3(COC)CNC(=O)C3)=O)CC2)CCCOC1 N1(C(C2C(=C)CC2)=O)C2CCC1C(C)C(NC(c1nc(C(C)(C)C)no1)=O)C2 CCC(CC)(CC)C(=O)NCC(c1ccccc1)NC(c1cnn(C)c1N)=O C1(CN(C(=O)C=CC2(C)COC2)C)CCCN(C(=O)C(C)(F)c2ccon2)C1 Cc1cc(C)cc(S(=O)(=O)N2CCCC(C)(C(N3CCN(C)C(C)C3)=O)C2)c1 C1(C2CCN(C(=O)Cc3cccc(O)c3)C2)(NC(CC2C(C)=NOC2=O)=O)CC1 C(CCN=c1[nH]c2ccc(O)cc2s1)N(C(c1n(C)ncc1C(F)(F)F)=O)CCO c1(CN2C(C(=O)OC)CC(NC(c3ccnc(C)c3)=O)C2)ccc(NC)cc1Cl c1(CC(=O)NCC(C)CN(C(=O)C(F)CC)C)nc([N+](=O)[O-])n[nH]1 Cc1cc(C(=O)NC(CNC(=O)C=Cc2nccs2)C2CC2)cc(C)n1 C1(CSCC)CCC(C(N2CCN(C(C3C4CC5C(C4)C35)=O)CC2)=O)CC1 C1(F)(C(N(CC(CC)NC(c2cnc(O)cc2OC)=O)C)=O)CCCN(C)C1 N1(C(C2N(C(c3ccnnc3)=O)CC(=O)NC2)=O)CC2CCC1C(O)C2O C=C(CNC(=O)C(OC)OC)CCNC(c1[nH]nnc1C(F)F)=O Cn1nc2c(c1C(N1CCCC(F)C1)=O)CN(C(=O)C1CC1)CC2 N1(C(CN(C(=O)OCC)C)=O)CCCC(O)CC1C(=O)N(C)CCc1cccs1 C1(C(N(CCCC(=O)NCc2ccc(C#N)s2)C)=O)CC(F)(F)CO1 c1(C(N2C(C(=O)Nc3ccccn3)CC3CC32)=O)c(F)cncc1Br c1(NC2(CNC(C(CC)N(C)C)=O)CC2)cc(COC)nc(C(C)(C)C)n1 c1(C(=O)NC(CNC(c2ncccc2F)=O)C2CC2)ccc2c(c1)CC2 C1(NC(COC2(C)CCCC2)=O)CN(C(C2CCCOC2)=O)Cc2ccnn2C1 c1(OC)ncnc(OC)c1C(=O)NCC(C)NC(c1sccc1C#N)=O C(C(CC(F)(F)F)NC(C1CC1C1CCC1)=O)NC(=O)Cn1ccc(C2CC2)n1 c1(C(N2CCC(NC(c3c(C)noc3N)=O)C(F)C2)=O)cccc2occc12 CC(C)CC(C(=O)NCC(C)(C)CNC(C1CC2CCC1C2)=O)n1ccnc1 N1(C(CC=C(C)C)=O)CC(CNC(c2cnn(CC(F)F)c2)=O)C(F)(F)C1 Cc1cnc(C(N2CCN(C)CC2C(N2CCOC(C)(C(C)C)C2)=O)=O)cc1C Cn1ccc(CC(N2CCC2C(=O)N(CC(N2CCOCC2)=O)CCO)=O)n1 Cc1cc(F)cc(C)c1C(N1CC(NS(=O)(=O)CC#N)C(C#N)C1)=O C=C(C)CCCC(=O)NC1CC2(C1)CC(C(=O)NC1CC13CC(O)C3)C2 C1(C(N(CC(C)OC)CC)=O)C=CCN(C(=O)CN2CCCNC2=O)C1 CCC(C)(COC)C(=O)NC1CN(C(=O)CCNC(c2cccs2)=O)CC12CC2 c1(C(=O)NCC(C)CN(C)C(c2cc(O)cc(O)n2)=O)ccnc2c1CC(=O)N2 c1(C(N2CCC(N(C)C(C34COCC3C4)=O)C2)=O)cc(C2CC2)ccn1 N1(C(C(COC)NC(C)=O)=O)CCC2CCCC(C1)N2C(=O)Cc1cncn1C C1(NC(C2CCCCCC2)C(=O)O)CN2CCC1c1ccccc12 CCCC(C(=O)NCC1(O)CN(C(=O)CSC(F)(F)F)C1)OC C#CCC(C)(C(=O)N(C(C(N)=O)C1CC1)C)NC(C1CCC(=O)NC1)=O c1(CN=C(NC2C(C)NC(=O)CC2)NCc2ccco2)cnn2ccccc12 C1(NC(c2c(C)cnc(F)c2)=O)CCN(Cc2cccc3[nH]ncc23)CC1(C)C C1(CC(N)=O)CCNCC1.c1(CNC(=O)NCC(F)F)cnc(C(F)F)cn1 C1(CC=C)(NC(c2cnncc2NC)=O)CCN(C(=O)C(F)C(C)C)C1 N1(C(C(C)(N(C)C(c2cc[nH]c2)=O)C2CC2)=O)CCC(C(N)=O)C1 N1(CCN(C)C(C2CC3CCC2O3)=O)CCN(C(C2CCN(C)C2)=O)CC1 C1(CC(=O)NCC(C(C)C)NC(c2ncsc2C2CC2)=O)CCC(C)(C)CO1 CCCC(O)C(=O)NC1CCN(Cc2nccn2CC)C1 c1(C(=O)NC2CC(NC(C3(CC#C)CCCO3)=O)C2)onc(C)c1C CS(=O)(=O)c1ccc(C(=O)NC(CNC(=O)C2=CCS(=O)(=O)C2)C2CCC2)nc1 c1(C(=O)NC(C(C)NC(c2cc(CC)c(C)s2)=O)C)n[nH]c(C(C)C)c1[N+](=O)[O-] N1(CCNC(C(CCCC)=O)=O)CCN(C(=O)C(C)(CC)CC)CC12CCC2 C1(CNc2nc(C)nc(O)c2)CC2CCC1N(C(C1(CO)CCOCC1)=O)C2 c1(CC(=O)NCCCCC2CN(C(C3CC(C)OC3)=O)C2)ccccc1[N+](=O)[O-] c1(C(=O)NCC2C(NC(C(C)C3CC3)=O)CC2)ccc2c(cnn2C(F)F)c1 C1(NC(C(CCC)C)=O)CN(C(=O)Cn2ncc(Br)c2C)CC12CCC2 c1(C(N2CCC(F)(CNC(CCC=C=C)=O)C2)=O)c(OC)ccnc1OC C(=O)(C1=CC2(CCOC2)C1)N1CC(CCNC(C(c2cn(C)nc2)(F)F)=O)C1 C1(CNC(c2nn(C)c(O)c2)=O)CCCC2(CCN(C(C3CC3C#N)=O)CC2)O1 C12CCCN1NC(=O)CONC2=O.Cc1ccc(CC(=O)NC(C)C)cc1 N1(C(CN(C)CC)=O)CCCC2CN(C(C3(C4=CCCCCC4)CC3)=O)CC12 C(C(CO)(CO)NC(=O)C=CCO)N(C(=O)CC1(C)CC1F)C C1(CN(C)C(C2(F)CC2)=O)CCCN1C(=O)CCC1CC1(C)C C(CC(N)=O)(C(=O)NCC(=O)N(C)O)NC(C(C)OCCN(C)C)=O c1(C(=O)NC2CC(CNC(C(CC)=CC)=O)C2)ccnc(OC(F)(F)F)c1 c1(OC)cc(C)c(C(=O)NC(CNC(C2CCCO2)=O)C2CCC2)c(F)c1 N1(C(C(CC#CC)NC(c2cc(CC)no2)=O)=O)CCCCN(C)CC1 N1(C(C2(C)CC2(F)F)=O)CCC2(CC1)C(NC(c1cc(CO)on1)=O)CS2(=O)=O c1(C(=O)NCC(CC)NC(C2CC(=O)N(O)C2)=O)ccc2c(C)cc(O)nc2c1 C1(NC(C(C)(C)SC)=O)CC(C)N(C(=O)C(C)OC2CCCCC2)C1 c1(C(=O)NCC2CN(C(Cn3ncc(C#C)c3)=O)CC2C)cc(F)cc(C)c1O C1(NC(CC(CC)C2CC2)=O)C2CC3C(C2)C13C(N1CC(N=[N+]=[N-])C1)=O CC(=O)CCCC(=O)NCC1(O)CCCN(C(=O)CCC(=O)c2ccc[nH]2)C1 CN1CC(NC(c2ccc(CNC(=O)CCNC(N)=O)o2)=O)C2(CC2)C1 C1(CC)C(NC(=O)CCOCC2CCC2)CCN1C(C1OCCCO1)=O N1(C(c2c(CC)nns2)=O)CCN(C(c2coc(CS(C)(=O)=O)n2)=O)C(CO)C1 C#CCCC(O)C(=O)NC1(C(=O)NCc2cnn(-c3ccccc3)c2)CCCC1 CC1Cc2cc(N)ccc2CN1C(=O)C(N1CCC2(CCCC2)CC1)=O C1(C(N2C(C(N(C3(C4CC4)CC3)C)=O)C=CC2)=O)CC2(CCO1)CC2 c1(C(N2C(C)CC(CC(=O)NCC3CC(C)C3)C2)=O)ncnc2cc[nH]c12 CC1(CNC(c2ccc(NC3COC3)cc2)=O)CCCN1C(=O)CC(F)(F)F c1(NCCc2ncc(CC)s2)nc(N2CC=CCC2)nc2scnc12 C(=O)(C(CO)C(F)(F)F)NCC(CCC)C(=O)NCc1nc(CC)no1 N1(C(CN(C(C)C)C)=O)CC(=O)CC1C(=O)NC1CC(CF)C1 Cc1[nH]nc(C(N2CCN(CC(=O)N(CCCF)C)CC2)=O)c1Cl c1(OC(C(=O)NCC2CCN(C(c3c(C#C)c[nH]n3)=O)C2)C)cccc(C)c1C C=CCCC(F)(F)C(=O)NCC(C1CCC1)NC(C1(C)CCCNS1(=O)=O)=O c1(C(N2CC(C(N)=O)(CNC(C3CC(C)SCC3)=O)C2)=O)cc([N+](=O)[O-])n[nH]1 N1(C(CCc2cc(C)no2)=O)CCC(C)C(CNC(=O)CNC(=O)NC2CC2)C1 c1(N2CCN(CC)CC2C)cc(-c2cnccc2N)c2cccc(F)c2n1 O=C1CCC(CC(=O)NCC2CCN(C(C3(F)CC=CCC3)=O)CC2)CN1 c1(C(N(C(C)CNC(C2(c3cccnc3)CC2)=O)C)=O)cc2n(n1)CC(F)C2 N1(C(=O)Nc2ccc(OC)cc2)CCC2(C1)CN(CC(O)CC(F)(F)F)C2 c1(C(C)C)ncncc1C(=O)NCC(C)N(C)C(C1CCOC1(C)C)=O c1(C(N2CCC(F)(CNC(COCCC)=O)C2)=O)cnc2c(C)cccc2c1 C1(NC(C(C)(C2CC2)NC(C)=O)=O)CCCCN(C(C2CC(F)C2)=O)C1 C(c1nc2ccccc2[nH]1)=CC(N1CC(CC)N(C(c2cnc[nH]2)=O)CC1)=O Cc1ccc(Cc2nc(C3(C(=O)NC4CCCC4)CC3)nn2-c2ccccc2)cc1 CCCC(C)(O)C(=O)N1CCC(C(=O)N(CC(C)SC)C)O1 O=C1CCCC(C(=O)NC2C=CC(CC(=O)NCc3cnn(CCF)c3)C2)N1 C1(CC(N2C(C#C)CCC2)=O)CN(C(c2cnn(C(F)F)c2)=O)CC12CC2 C1(NC(C2CCCN(S(=O)(=O)C3CC3)C2)=O)CC(=O)N(C2CCCCC2)C1 CCC(C)(C)CCCC(=O)NCCN(C(C1OCCC1C)=O)Cc1ccccc1 Cc1oc(Br)cc1C(N1CC(F)CC1CNC(c1cnn(C)c1C)=O)=O CCC(=O)CCC(=O)NCC(O)CNC(=O)CC1COCC1(C)C c1(C(=O)NCC2CN(C(C(COC)OC)=O)C3(C2)CCC3)ccc(C#N)c(C)c1 N1(C(C(c2ccco2)NC(c2c(C)cc(N)cn2)=O)=O)CC(C2=NOC(C)C2)C1 CC(C)C(F)(CNC(=O)CCC(=O)C1CC1)C(=O)NCC1CC12CC2 c1(CNC(=NC)NCc2ncccc2N(C)C)nc2cc(F)c(F)cc2[nH]1 N1(C(C2C(C)CCOC2)=O)CCN(C(c2ncc(F)cn2)=O)C(c2ncc[nH]2)C1 c1(C(=O)NC2CCCN(Cc3cc(OC)ncc3)C2)ccc([N+](=O)[O-])o1 c1(OC)cc(C(=O)NCC2C(C)CCN2C(=O)CCCC#N)sc1Br C(=O)(C1=CCC(NC(C2CC2(F)Cl)=O)C1)N1C(CC)(CC)CC1 C12(NC(=O)C(N3CCOCC3)C3CC3)CCN(C(=O)CC3CCOC3=O)CC1C2 C1(NC(=O)NCC(c2ccc(F)cc2)Oc2ccc(Cl)cc2)CCCC12CCNC2 c1(C(N2C(C)CCC(CNC(C3(C(=O)OC)CC3)=O)C2)=O)ccc2cnsc2c1 C1(NC(=O)CC(O)CC2CC2)CC12CCN(C(C1COCCO1)=O)CC2 Cc1cc(O)ncc1C(=O)NC(CO)CCCCNC(=O)CN(C1CCC1)C c1(CNC(N(C2CC2c2ccccc2OC(F)F)C)=O)cc(C(F)(F)F)ccc1F c1(NC(c2n(C(C(=O)OC)C)nnn2)CC(C)C)ccccc1-c1ncco1 C1(OC)CC(CNC(c2cnc(C(C)C)o2)=O)N(C(c2cccc[n+]2[O-])=O)C1 C1(F)(C(=O)NC2CC(C(C(=O)NCC3C(C)OCC3)F)C2)C(C)(C)C1(C)C c1(C(N2C(CNC(CS(=O)(=O)N(C)C)=O)CCCCC2)=O)cccn2nnnc12 c1(OC)cc(C)ccc1C(=O)NCCCCCN(C(=O)CC(C)NC(N)=O)C C(CCN=c1[nH]c2c(c(=NC(C)c3nc(=N)[nH][nH]3)[nH]1)CCC2)SCC Cc1nc(C(C)C)oc1C(=O)NC(C)C(C)(C)NC(c1cnc(=N)[nH]c1)=O c1(C(C)C)ccc(C(CNC(=O)CN2CCCC2)NCc2cc(C#N)no2)cc1 c1(C(=O)NCCC(CC)(CC)NC(CSCCC)=O)ccc(F)c2c1CCC2 c1(CNC(=O)Nc2ncc(CC)s2)cc(C)n(-c2cc(C)on2)c1C C1(C(=O)NC(c2cscn2)CO)CCN(C(=O)C=CC2CCOC2)C1 Cc1cc(CC(N2CCOC(CNC(c3ncnc(C)c3C)=O)C2)=O)cc(C)c1 N1(C(C2C(CCC)C2)=O)CC2(C1)CN(C(c1cnco1)=O)CCO2 c1(C(=O)NC2CN(C(CN(C)C(=O)C3CC3)=O)CC(O)C2)ccn2ccnc2c1 Cc1cc(C(N2CCC(C)(CNC(C34CC(O)C3C4)=O)CC2)=O)c(N)cc1F c1(C(N(C)CC2(O)CCN(C(C(C)OCCC=C)=O)C2)=O)cc(F)cc(Cl)c1 C1(C(=O)NC2(C)CCCN(C(c3ccnc(S)c3)=O)C2)CC2(CO1)CC(F)(F)C2 CCS(=O)(=O)c1cccc(C(=O)NC23CCN(C(=O)COCCOC)CC2C3)c1 c1(NC(C(C2CC2)OC)=O)cccc(OCCN2CCOCC2)c1 c1(SC)cnn(C)c1C(=O)NCc1nc(CNC(=O)CC(C)NC(N)=O)cs1 C(=O)(CN=c1cc[nH]cc1)NC1CC(NC(C=Cc2ncn(C)c2)=O)C1 C(CCC(=O)NC(CN(C)C)C(=O)NCC1COCC1O)OC(C)=O c1(CC(=O)NCCC2CCCC(C(F)(F)F)O2)cccc2cnccc12 N1(C(=O)C=CC2CCCCC2)CCOCC(NC(C2(F)CCCCC2)=O)C1 Cc1cc(=NCC2(C)CCCCO2)[nH]c(N2CC3CCC2CN3c2ccccc2)n1 c12cnc(c(C)c1)N(S(C)(=O)=O)C1CCN(CC1)C2=O.CCOC N1(C(C(C2CCN(C(C(C3CCC3)OCC)=O)C2)F)=O)CCC=CC1CC N1(C(CSCCOC)=O)CCC(N(CC=Cc2ccncn2)CC2CC2)CC1 C12(NC(C3OCCN(C(C(C=C)O)=O)CC3)=O)CC3CC(CC1C3)C2 c1(C(N2CC(CC(=O)NCCCC(C)(C)O)OCC2)=O)cc(F)ccc1O CN1CCC(C(=O)NCc2n[nH]cc2C(N2CCC(N3CC(O)C3)C2)=O)CC1 C(CNC(c1c(C)nn(CC(F)F)c1C)=O)(C(C)C(C)C)NC(CCOC)=O CCC(C)(C)CC(=O)N1CCCC(N(C(=O)CC2COCC(C)(C)O2)C)C1 C(C(=O)NOCCO)(C1CCCO1)NC(C(CN(C)C)O)=O C(CCCCOC(C)(C)C)(c1nnnn1CCNC(C)=O)NC(COC)(C)C C(=O)(C1CCCc2cncn21)N1CC(C)C(CNC(c2cc(N)ccc2F)=O)C1 c1(CC(=O)NC(CC(C)C)CNC(=O)CC2CCOC2)nc(F)ccc1Cl C(N=c1[nH]c(=NCCC2CN(C)C2)c2ncccc2[nH]1)C1(OCC)CCC1 N1(C(CNC(=O)NC)=O)CCC2(CC1)CCN(C(c1ccnc(C)c1C)=O)C2 c1(C(=O)NC2C(NC(c3c(SCC#N)cccc3)=O)C2)nnn2c1C(=O)NCC2 c1(CC)cccnc1N1CCC(CCC(=O)NCC(c2cccc(F)c2)C)CC1 Cc1ocnc1C(=O)NC1(CCNC(C23CC(F)C2C3)=O)CC1 C1(C(=O)NCC2(O)CC(CO)C2)(NC(C(C)=C(CC)C)=O)CC(O)C1 C=CC(O)C(=O)NCC1(CNC(C2CC=CCC2)=O)CC1 c1(C(=O)NCC(CCCC)NC(c2cc(C)nc(O)c2)=O)cc(Cl)nc(Cl)c1 c1(N2C(C)CC(CNC(C3N(C(C)=O)CCC3)=O)C2)ccc([N+](=O)[O-])c(O)n1 c1(C(N2CC(NC(C(CC)C)=O)C(C)C2)=O)c[nH]c2ccc(Br)cc2c1=O c1(C(C(=O)NC(C)CNC(C2(C#N)CC23CCC3)=O)C)ccc(S(N)(=O)=O)cc1 N1(C(c2c(C)ccc(OC)n2)=O)CCC2CN(C(=O)CSC3CC3)CCC2C1 C1(NC(CCCC#C)=O)(CNC(c2cnc(Cl)cc2N)=O)CCCCC1C c1(C(N2C3CN(C(C=CCOC(C)(C)C)=O)C(C3)C2)=O)nc(F)c(F)cc1F c1(-c2cn(C3CCN(C(C(CC)(C)O)=O)C3)nn2)cc(NCOC)ccc1OC N#Cc1ccc(CNC(c2ccc(=NCc3ccnc(O)c3)[nH]c2)=O)cc1F C1(C2CCC2)(CNC(C(CC)=CC)=O)CCN(C(=O)CCOC2CCOC2)CC1 Cc1ccnc(O)c1C(N1CCC2(NC(c3ccc(N(C)C)cn3)=O)CC2C1)=O N1(C(Cc2c(C)ccnc2)=O)CCC(C(=O)NOCCCO)C(C)(C)C1 C1(NC(CC(=O)N(C)C)=O)C2CC(O)C1N(C(=O)C=Cc1ccoc1)C2 c1(C(N2CCCC(NC(c3c(C)scc3)=O)CC2)=O)ncnc2c1cnn2C C(=O)(C(F)(F)C(F)F)NCC(CNC(C12C(C(=O)OCC)(CCC1)C2)=O)O Cc1nccnc1C(=O)N(C)CC=CC(=O)NCC1(F)CCN(C)C1 C12(COC)CC(NC(C3CCCN(C(C)C)C3)=O)(CN1C(C1(C)CC1(F)F)=O)C2 C(=O)(C(C)CN(C(=O)CCc1cn(C)nn1)C)NCC(C)OCC#C C1(CN(C(c2nc(O)c(C)s2)=O)CC)CCCCN1C(=O)C(C)OCC(C)C c1(C(=O)NC2CCCC(C#C)C2)cc(OCCC)c(O)c(OC)c1 c1(CCCC)ccc(C(=O)N(C(C)C2CC2)Cc2nnc(CC)n2C)cc1 CCC(C(=O)NC1(CO)CN(C(C2(C#N)CC3CC3C2)=O)C1)C(F)(F)F c1(C(=O)NC2C=CCN(C(Cc3ccc(C)o3)=O)C2)ccc([N+](=O)[O-])cc1F C1(NC(C2CN(C)CC(C)O2)=O)CCCC12CN(C(=O)CC(C)(C)O)C2 C1(O)(CN(C(CC2CC(OC)C2)=O)C)CCN(C(c2cc(C)c[nH]2)=O)CC1 C(CCC(=C)C)(C(=O)N(C1CCN(Cc2ccccc2)C1)C)N(CC=C)CCC CCC(C)C(O)C(C)C(=O)NCc1cn(CC(=O)Nc2cc(C)cc(C)c2O)nn1 CC(C)C(C)(C)C(=O)NCC1CN(C(c2cnc(-c3ccncn3)nc2O)=O)C1 N1(C(Cn2nnc(C)n2)=O)CCN(C(=O)CN2CC=CC2)C(CO)C1 Cc1ccc(=N)[nH]c1C(=O)NC1(CNC(C2CC2C(F)F)=O)CCOC1 N1(C(C2CC(C)C2)=O)CCN(C)C(C(N2C3CSCC2C3)=O)C1 c1(C(N(C2CC(NC(Cn3c(C)ccn3)=O)C2)C)=O)ccc(S(N)(=O)=O)nc1 C(=O)(CC(O)CC1CC1)NCC(C1CCCCC1)NC(C(C)(C)OC(C)C)=O C1(CCC)(NC(c2csc(C(F)(F)F)c2)=O)CCCN(C(C2(N(C)C)CC2)=O)C1 c1(C(=O)OC(c2ccccc2)CCC)csc(C(=O)NCCNN2CCC2C)n1 c1(C(=O)NC(C2CCN(C(c3nccc(C)n3)=O)C2)(C)C)n[nH]c2ccccc12 C1(CNC(C(C)(O)C2CC2)=O)CC2CCC(C1)N2C(c1cnnn1C1CCC1)=O C(C(C)CC(=O)NCc1occc1C(N1CCC1C1CCCC1)=O)OC c1(C(C)C)cc(=NC(C)CC(C)NC(=O)CC2(C)CCCO2)[nH]c(C(C)C)n1 C(=O)(C1=CCS(=O)(=O)C1)NCCCCC(C)NC(=O)Cn1nccn1 C1(SC)CCN(C(c2sccc2CNC(C2CCC2C#N)=O)=O)CC1 c1(CC)nc(C)c(C(=O)NC2CCCCC2CNC(C2SCCS2)=O)o1 c1(C(N(CCCNC(c2n(CC)ncc2)=O)C2CC2)=O)cc(C)c(O)c(C)c1 CC1CN(C(c2cn(-c3ccc(Cl)cc3)nn2)=O)CC1NC(=O)CCC1CCC1 C1(CNC(=O)CC2CCC2)CCCC2(CN(C(C34CCCN(CCC3)C4)=O)C2)O1 N1(C(c2ccc(NC(C)=O)s2)=O)CCC(C)C(CNC(=O)C(C)c2ccco2)C1 N1(C(c2ncc(CC)cn2)=O)CCCOC(CN(C(=O)C(C)C(C)(F)F)CC)C1 CC1=CCC(N=c2ccnc(N3CCN(CCC(F)(F)F)CC3)[nH]2)CC1 c1(-n2c(C)cnn2)ccc(C(=O)NCCNC(C2COCCO2)=O)cc1 C(CC(C(=O)NC1CC1CC)NC(c1ccc(C)s1)=O)OCC N1(c2nnc(C)o2)CCCC(C(C)NC(c2ocnc2C2CC2)=O)C1 C1(C(=O)NCCN(C(C)C)CC)(NC(C23CSCC2C3)=O)CC(O)C1 N1(C(C(C)C2CC2)C(=O)NCc2ccccc2Br)CCOCC2(CC2)C1 CCC(C(C)C)C(C(=O)NCCOC)N(C1CCS(=O)(=O)C1)CC C(=O)(C1=NOC(C)(C)C1)NCC1CCN(C(C2C(C)(CC)C2)=O)CC1O N1(C(c2cnc(C)[nH]2)=O)CCn2cc(NC(=O)Cc3ccc(O)cc3)nc2C1 O=C1OC(NC(C2Cc3nncn3C2)=O)Cc2ccccc21 S(=O)(=O)(c1ccnc(NNC(=O)C2CCS(=O)(=O)C2)c1)NC1CC1CC(C)(C)C c1(CN(C2CC(=O)N(C3CCC(=O)C3C)C2)C(C)=O)cc2ccccc2nc1Cl c1(C(N2CC(CCO)(NC(CCc3scc(C)n3)=O)C2)=O)cc(C)n(C(F)F)n1 c1(C(=O)NC2(C)CN(C(C3CCCO3)=O)C2)nc(Br)c2ccccn12 C1(C(C(=O)N(CC(F)F)CC)C)CCN(C(C2CCN(C)C2C)=O)CC1 N#Cc1ccc(C(=O)NCC(O)CC(=O)NCCCn2nccn2)cc1 C(C)(C(C(C)C)NC(c1cnc(C)n1C(F)F)=O)NC(C1(CC#C)CCCC1)=O C(CC(C)(C)C)(C(=O)NCC1(O)CCCN(C(C2CCC=CCC2)=O)CC1)OC C#Cc1ccc(C(=O)NCC(C2CCOC2)NC(=O)Cc2nnc(S)n2C)cc1 N1(C(CSCC)=O)CCCC(C)(CNC(c2ncc(C)cc2OC)=O)C1 CCCCCC(CC)C(=O)NC1CC(C)(C(=O)N(CC(C)(C)COC)C)C1 Nc1c(F)cc(F)c(F)c1C(N1CC(NC(=O)CCc2cn[nH]c2)CC(O)C1)=O C1(C(N(CCC(=O)OCC)CC=C)=O)CCN(C(=O)Cc2cc[nH]c2)CC1O c1(C(N(C(C)CNC(=O)COc2cncc(Cl)n2)C)=O)c(F)cccc1F c1(NC(=O)NCC2CS(=O)(=O)C2)cc(Br)cc2c1OCO2 C12(C(=O)NCC3N(c4ncc(C(=O)OC)cc4Cl)CCC3)CCC(C)(CC1)OC2 C(=O)(C1OC(=O)c2ccccc21)NCCCOCCNC(CS(C)(=O)=O)=O N1(C(C(CC(F)F)NC(c2c(C#C)c[nH]n2)=O)=O)CCc2sccc2C1 c1(C(=O)NC(C)C(C)(C)NC(C2CC(C)(F)C2)=O)cnnc(-c2ccccc2)c1 c1(N(CC(CC)C)CC)cc(=NCC(=O)NC2CCCC2)[nH]c(C(F)(F)F)n1 C#CCC(C)(C(=O)NC1CCN(C(C)=O)C1)NC(c1c[nH]c(=NC)s1)=O c1(C2N(C(=O)C(C3CCOCC3)F)CCC2)cc(Br)ccc1Cl C1(C)(C(=O)NC2C(NC(C=C(C)C(C)(C)C)=O)CC2)CC(=O)N(C)C1 N1(C(C=C(CC)C)=O)CCC(NC(c2cc(COC)cn2C)=O)C(CC)C1 c1(C(N2CCC(c3cnn[nH]3)C2)C(=O)NCC)ccn(C(F)F)n1 N1(C(C(c2ccccc2)SC)=O)CC2(CC(NC(=O)CCn3ccnn3)CO2)C1 C(C(=O)Nn1cccn1)C1(NC(c2[nH]cc(C(C)=O)c2)=O)CC1 N1(Cc2c(C)cc(C)[nH]2)CC2CCCC(C1)C2C(=O)NC1CCCC(O)C1 C1(N(C)C(C2CC(O)CN2)=O)CCCN(C(c2c[nH]c(=N)s2)=O)C1 C12(C(N3CCC(NC(c4c(C)n[nH]c4)=O)(CF)C3)=O)CCC(N=[N+]=[N-])C1C2 c1(OC)ccc(C(=O)NCC2(CNC(=O)CC3(CO)CC3)CCOCC2)cc1 C1(CNC(c2nc(C(C)C)sc2)=O)CCN(C(=O)CC2CCCN2C)C1(C)C c1(C(=O)NC2CCC(C)N(C(c3cc[nH]n3)=O)C2)ncc(C#N)cc1Cl c1(NC2(CNC(c3ccc(N(C)C)cc3)=O)CC2)nc2cccc(F)c2s1 C1(C)(CNC(COC(C)C)=O)CCCN1C(=O)C=Cc1cscn1 C1(OCC)CN(C(=O)Cc2ccccc2)CC1CNC(=O)CCc1ccon1 c1(N2CCCC(O)(CNC(c3c(C)csc3)=O)C2)nccc(S(C)(=O)=O)n1 C(=O)(C1CCc2nccn21)N1CC(NC(C=NOC)=O)C2C1CCC2 CCCC(C(=O)OC)C(=O)NC(CNC(c1ccc(CO)o1)=O)C1CC1 C1(NC(C2C(NC(=O)Cc3cc(F)ccc3F)C2)=O)CC2(C1)CS(=O)(=O)C2 C12(NCc3ccc(C(=O)OC)cc3)CC(CN3CC4(CCCC4)C3)(CCO1)C2 N1(CC(N2CCC(NC(c3cccn3C(F)F)=O)CC2)=O)CCCCC(O)C1=O c1(C(=O)NCC=CCNC(C(C)CC2CC2)=O)cccc(-n2cccn2)c1 N1(C(C2CC(=C)C2)=O)CC(CNC(C2CCCCS2(=O)=O)=O)CC12CCC2 c1(C(N2CCC(O)(CN(C(CCCCSC)=O)C)C2)=O)cc(C)c2[nH]cnc2c1 C1(NC(C(C)(C)Oc2ccccc2Cl)=O)CC2CC1N(C(C1(C)CCOC1)=O)C2 c1(OC)ccc(C(=O)NCC2CCCC(NC(=O)C=C3CCC3)C2)cc1OC CCC(C)(C(=O)NC1CCC(CCNC(C23CC(CO2)C3)=O)C1)OC C(CN=c1cc(C)nc(CC2CC2)[nH]1)(N(C(C=C(C)c1cccs1)=O)C)C1CC1 CC1=CCN(C(C2CC3CC3N2C(=O)C(C)N=[N+]=[N-])=O)CC1 CC(C)C(F)(CNC(=O)C=Cc1cncs1)C(=O)N=c1ccn(CC2CC2)[nH]1 C1(NC(c2n(CC=C)nnn2)c2ccn(CCC)n2)CCCC(C2CC2)C1 c1(C(N2C(C(=O)Nc3cc(O)cc(O)c3)CC(O)CC2)=O)ccc2ncnn2c1 CCC(C)(C(=O)NC(c1ccc(CNC(=O)C=Cc2cn(C)cn2)cc1)C)OC C1(CC)CCCC1(C)NC(=O)COC(C)(C)CNC(=O)CN1CCCCC1C N1(C(C(C(C)C)O)=O)CCCC(O)(CNC(c2[nH]ccc2-c2cccs2)=O)CC1 N1(C(c2ncc(CC)s2)=O)CCN(C(c2cc(Cl)nn2C)=O)CC1CCO N1(C(Cc2c(C)occ2)=O)CCN(C(=O)CC2CCCNC(=O)C2)C(CCO)C1 Cc1cc(F)c(C(=O)NC2CCCCN(C(C3CCCCN3N=O)=O)C2)cc1F c1(C(C(=O)NCCC(=O)OCC)N(C)CCC2CC2)ccc(S(N)(=O)=O)cc1F CN1CCC2CN(C(c3ccc(NC(=O)NC(=O)C(Cl)(Cl)Cl)cc3)=O)CCC12 C(N=c1[nH]c(=N)[nH]c(=NC2CCOC3(CCSCC3)C2)[nH]1)C1(CCOC)CCC1 CCCCCCC(F)C(=O)NC(C)(C)CN(C)C(C1(C)CCN(C)C1=O)=O C(=O)(C1=C(SC)CCCC1)NC(CN(C(=O)Cc1scnc1C)CC)C c1(CC2(N(C(N3CC(n4cnnc4)C3)=O)CC3CC3)CCC2)ccccc1 C1(C(=O)NCC(C)(C)NC(c2cn(CCCC#N)nn2)=O)CCCC(F)C1 C1(CNC(CSCC)=O)CCCN1C(C1(C)CC1)=O.C(C)(=O)O CCCCS(=O)(=O)CC(=O)NCC(C)NC(C1CCCN1Cc1nnn(C)n1)=O c1(C(N2C(C)CC(NC(CCN(CC)CC)=O)C2)=O)ccn2ccccc12 c1(NCCCCCC)[nH]c(=NCC(C)CC(C)C)nc2c1ncn2C c1(OC)ccncc1C(=O)NCC1CN(C(=O)C(C2(O)CCCC2)F)CC1C C1(C(N2CC3(CNC(C4(Cl)CC4)=O)CC2CO3)=O)CCc2nc[nH]c2C1 c1(C(N2C(CNC(C(c3n(C)ncc3)O)=O)COCC2)=O)cn2c(n1)CCC2 Cc1cc(C(=O)NCCOCCNC(=O)C(c2ccccc2Cl)(C)C)n(C)n1 Cc1c(C(=O)NCC2(CN(C)C(c3c[nH]nc3-c3ccsc3)=O)CC2)ccn1C c1(C(CC)C)nccc(=NCCNC(c2ncoc2-c2ccccc2)=O)[nH]1 N1(C(COCCCCOCC#C)=O)CC(OC)CC(NC(c2coc(Cl)n2)=O)C1 c1(C(N2CCC(C(C)(C)NC(CCC=CC)=O)C2)=O)cccc(OC(C)(C)C)c1 N1(C(C2OC3CCC2C3)=O)CCC(N2CCNCC2)CC1 C(CCC(C)C(=O)N1CCC(O)(CNC(c2ccc(OC)cc2OC)=O)C1)OC Cc1nn(C2CCCCO2)c(C)c1C(=O)NCC1CCN1C(=O)C(F)=CCCF CCC(C)CC(=O)N1CCCC1C(C)(C)CNC(=O)C=CCCc1ccccc1 c1(C(=O)NCC(C)N(C)C(C2COC(C)(C)CO2)=O)cccc(F)c1C#N C=C(C)CCCC(=O)NC1(COC)CN(C(c2nccn2CC)=O)C1 C#Cc1cncc(C(=O)NCC2CC(C)(C)CN2C(=O)C#CC2CC2)c1 C1(NC(c2csc(-c3ccco3)n2)=O)CC2CN(C(=O)C(F)C3CCC3)CC2C1 C(C(O)CCNC(C1CS(=O)(=O)C1)=O)NC(COCC=C)=O C(C(=O)N1CCC(C(N2CCC(C(F)(F)F)C2)=O)O1)C1CC(=O)NC1 c1(CNC(NC(CC=CC)C)=NC)cccc(OCCOC)c1 c1(C(=O)NC(c2cn(C)nn2)C(=O)Nc2cn(CCOC)nc2)ncc(F)cn1 c1(C(N2C3CC(CNC(Cc4nnc(C)o4)=O)C2CC3)=O)cc2cccn2cn1 N1(C(CCc2nc(C)c(C)[nH]2)=O)CCC2CN(C(=O)C(C#N)C(C)C)CCC2C1 C1(C(=O)NCCCN(C(c2c(Cl)nn(C)c2Cl)=O)CC)CC(S(C)(=O)=O)C1 C1(NC(c2ccc(C(=O)OC)s2)=O)CCC(NC(=O)CC2CC3COCC23)CC1 N1(C(CC2CC(OC)C2)=O)CC(NC(=O)C=CC2CCCO2)CC1(C)C c1(C(N2CC3CN(C(c4c(C)ccn4C)=O)C3C2)=O)n[nH]c2c1CCC2C C1(CC)CCCN(C(c2c[nH]c(=O)cn2)=O)C1C(N1CC2C(C(=O)OC)C2C1)=O C1(CC(=O)NCC2(O)CN(C(C(C=C=C)C)=O)C2)Cc2ccc(Cl)cc2C1=O C(N=c1[nH]c(=NC2CC3(CCCCN3)C2)[nH]c2c1COC2)c1n(C)c(Br)nn1 CC(CCC(=O)N(C)CC1(C#N)CCC1)NC(C1CCCSC1)=O C1(C)(C(=O)NCc2nccc(C(=O)Nc3ccc(C)s3)c2)CC2CCC2C1 CC(C)(C)CCC(=O)N1CCOCC1CC(=O)NCC(CO)C1CCC1 c1(C(=O)OC)ccc(Cl)c(NC(C2CCCN2C(=O)Nc2cccc(Cl)c2)=O)c1 C(C)(C(=O)NCC1CCC(NC(C2CCCO2)=O)C1)(c1ccccc1)OC N1(C(CNS(N)(=O)=O)=O)CCOC2CN(C(c3cc(Cl)c(F)cc3F)=O)CC12 C1(NC(c2c(C)cc[nH]2)=O)CC2CC1CC2C(N1CC(=O)NC(C(C)C)C1)=O c1(OCC=C)cccc(-c2cnc(C(N3CCC(N4CCOCC4)C3)=O)nc2)c1 N1(C(c2c(CC)scn2)=O)CCCC(NC(=O)C=Cc2ccnn2CC)C1C CCC(C)CCC(=O)N1CCOCC1C(=O)Nc1cc(O)ccc1C C(=O)(C(C(C)(C)C)C1CCC1)NC1(C)CC(NC(Cc2c(OC)nccc2)=O)C1 C=Cc1cc(C(N2CC(C)CCC2CNC(C2(C=C)CCC2)=O)=O)cc(F)c1 C1(CC(N2CCC(N(CCC)C(c3n[nH]cc3Br)=O)C2)=O)C(C)(C)C1(C)C c12cc(ccc1O)C2=O.c1(C(=O)NC(C)C(C)(C)NS(C)(=O)=O)cc(Cl)cn1C C(CCCC(CO)NC(c1ccc(C)cc1)=O)NC(c1c(CC)ncs1)=O N1(C(c2cn(C)nc2C(C)(F)F)=O)CC2(C1)CN(C(C1CC1C(F)F)=O)C2 CC1CC2(CC(NC(C3CN(C(=O)CC4CCC(=O)C4)CCN3C)=O)C2)C1 C1(NC(COC)=O)CC12CCN(C(=O)CC(c1ccc(F)cc1)NC(C)=O)C2 c1(CCOC)c(C)csc1C(=O)N(C1CC(NC(=O)CC2(CSC)CC2)C1)C CN1CCC2CN(C(C3CC3NCc3c(Br)cc(Br)cc3Br)=O)CC2C1 C1(C(C)NC(c2c(C)[nH]cc2)=O)CCCN(C(=O)CCCN2C(=O)CNC2=O)C1 C(=O)(C(C(C)(C)C)NC(=O)COC(C)=O)NCCOCC(C)C Cc1cn2c(CCC(N3CC(O)C(O)C3CNC(=O)C=CCO)=O)csc2n1 c1(C(N2CCC(CNC(C3(C4CC4)CC3)=O)C2)=O)ccc2cccnc2c1F N1(C(C(C(C)CC)N(C(c2c(CC)c[nH]c2)=O)C)=O)CCOCC(F)(F)C1 C1(Cc2cccc(OC)c2)CC2(CO1)CN(C(C1Cn3c(C)nnc3CN1)=O)C2 CC(Cc1ccccn1)C(=O)NC1C(C(=O)Nc2cc(C(=O)C(F)(F)F)c[nH]2)C1 Cc1ccoc1CNC(=O)C(c1cnn(C)c1)NC(C1CC1C(C)C)=O CCCC(CC)C(=O)N1CCN(C(=O)C=Cc2ccsc2)C(c2ccnn2C)C1 C1(CC(=O)NC2CC(CC(=O)NCC(C)N(C)CCOC)C2)CCCCCC1 CCCC(CCC)C(=O)NCC(O)CC(=O)N(CCOC)CCOC(C)=O c1(C(=O)NCC(CN(C(=O)COCc2nc[nH]n2)C)(C)C)cc(C#N)ccc1O C(C)(C)(CC(=O)N1CCC(F)(CO)C1)NC(C(n1c(C)ncc1)C)=O N1(C(CCn2c(=O)sc(C)c2C)=O)CC(CO)C2(C1)CN(C(c1ccco1)=O)C2 CC(CNC(c1cc(CO)on1)=O)CC(=O)N(C1CCN(C)C1=O)C c1(C(N2C(CNC(c3ccc(Cl)o3)=O)COCC2)=O)cn2ccsc2n1 C1(CNC(C=CCOC)=O)CC(C(=O)NCC2C=CCCC2)CO1 CN1CCC(C(=O)N(C2CCN(C(=O)C(C)N3CCC3)CC2)CC2CC2)CC1=O N1(C(C(C)CCO)=O)CCCC2(CNC(c3cnn4ncccc34)=O)CCCC12 c1(CCC(=O)NC(C2(CNC(COC(CC)C)=O)CC2)C)cc(Cl)no1 N1(C(COCC)=O)CCC2(CCC(CNC(C3CC3C3CCC3)=O)OC2)CC1 c1(CC)cc(C(=O)NC2COCC2NC(c2ncnn2CC)=O)nn1CCO c1(C(N2C(CC)CN(C(=O)C(C)O)CC2)=O)cc(Br)c2c(c1)OCCO2 C1(c2ncc(C)s2)CCCCN1S(=O)(=O)Cc1ccc(C(C)(F)F)cc1 CCCCC(C)CCC(=O)NC(C)(CNC(c1ncc(C#N)cc1Cl)=O)C(C)C c1(CNCC(CO)F)cccc(F)c1I c1(CC(N2C3CCC(C3)C2CNC(=O)C(F)(F)CO)=O)cccc2nsnc12 N1(C(C2(c3ccc(C)cc3C)CC2)=O)CCN(C(=O)CC(=O)N(C)C)CC12CCC2 CCC(C(=O)N1CC(NC(C2(CO)CC2(F)F)=O)C1)OC c1(NC(=O)NC2CC2)ccc(OCc2ccncc2)cc1C.CCC1CN1 N1(C(CCC(C)SC)=O)CCCC(C)(CNC(C23CC2COC3(C)C)=O)C1 Cc1ccc(C(=O)NC2CCCC(NC(C3(C)CC4CC4C3)=O)C2)cc1Cl C1(CCNC(=O)C(=O)NCc2cccc(N3CCC3=O)c2)CCS(=O)(=O)CC1 N1(C(C2CCCCS2)=O)CC2CC(C1)N(C(c1ccnn3ccnc13)=O)C2 CC1CCC(C(N2CC(C3CCCCO3)C2)=O)N1C(=O)CCc1cnc(O)[nH]1 C1(C(=O)NC2CN(C(C(=Cc3ccncc3)C)=O)CC2C)CCc2nccn2C1 C1(C(=O)N(C)Cc2cn(C(c3ccccc3Cl)C)nn2)(CC)CCCC1O C1(C(=O)NC2CC(CO)C2)CN(C(=O)CSc2ccoc2)CC12CC2 N1(C(COC(CC)C)=O)CC(C)(NC(=O)Cc2cn(C)cn2)C1 C=CC(CCC)CC(=O)N(CCCCCNC(=O)Cc1c(C)nc(O)nc1C)C CC1CC(=O)NCCN1CCCCCC(=O)N(C)C C(=O)(CCCS(N)(=O)=O)NC(C1CN(C(c2n[nH]cc2[N+](=O)[O-])=O)CCO1)C N1(C(CSCC)=O)CCN(C(c2ccc(N)c(SC)c2)=O)CC1CF CC(C)C(CCN(C)C(C1(CCF)CC1)=O)NC(c1nncn1C)=O Cc1cncc(NC(=O)C(Cn2cncn2)NC(=O)Cn2nccc2C)c1 N1(C(CCCC=C)=O)CC(C(=O)NCC(=O)NCC(C)C)CC(C)C1 C=CC1(C(=O)Nc2cccnc2)CCN(C(=O)C(=Cc2ccccc2)C)C1 c1(C(=O)NC2(CO)CN(C(CNC(C(CC)CC)=O)=O)C2)cnn2c1OCCC2 C1(CCNC(CCN(S(C)(=O)=O)C)=O)CCCN(C(C2(C)CC=CC2)=O)C1 c1(C(N2CC(CC(=O)Nc3cc(Br)nc(Br)c3)C2)=O)cc(O)ccc1[N+](=O)[O-] CCCC(CCC)CC(=O)N1CC2CC1C2C(=O)NCC1CN(C)CCO1 c1(C(=O)NCc2c[nH]nc2C(N2CC(N3CCCC3)C2)=O)c[nH]c2cnccc12 CC1(C)C(CNC(C2CCS(=O)(=O)N2)=O)CCN1C(c1nccc(Cl)c1O)=O c1(CC(=O)NCCCC2N(C(CC3(OCC)CC3)=O)CCC2)cccnc1Cl c1(C(N(CC(CN(C(C(CC=C)CC)=O)C)O)C)=O)nn(C)c2c1CCC2 c1(C(C)CC(=O)N(C(C)CCNC(c2cncs2)=O)C)ccccc1F c1(C(=O)NC2CC(CC(=O)Nc3ccc(O)c(F)c3)C2)cc2cnccc2[nH]1 Cc1oc(C(C)(C)C)cc1C(=O)N(CCCN(C(=O)Cc1cc(Cl)sc1Cl)C)C CN1CCCC(NC(=O)NC2COCC2NC(=O)COCC2CCCO2)C1 N1(C(=O)NC2C(CCN(C3CCCC3)C(=O)OC(C)(C)C)C2)CC2CC2C1C#N CC(CC(F)F)C(=O)N(CCC(N1CCC(F)(CO)C1)=O)CC1CC1 C(=O)(C(C)(C)NC(C)=O)NCC(c1ccccc1)CNC(C(F)=CC)=O CC1C(NC(=O)Cn2cncn2)CCCN1C(=O)CCC(=O)c1ccc[nH]1 CCC(F)(C(=O)OC)C(=O)N1CC(CCNC(c2cc(C(F)(F)F)nn2C)=O)C1 C(CCN=C(NCCC(=O)NCc1ccco1)NCC(C)SC)NS(CC)(=O)=O CN1CCCC(N=c2[nH]c(=N)[nH]c(=NCCc3ccsc3Cl)[nH]2)CC1 N1(C(Cc2c(C)n[nH]c2C)=O)C2CCC1CN(C(C1(CC#N)CCCC1O)=O)C2 c1(CC(=O)NCC(CN(C(CC2C(C(=O)OC)CCC2)=O)C)C)nn(C)cc1Cl N1(C(C2(O)CCCN(C(=O)OC)C2)=O)CCCC12CCCN(C(=O)CNC=O)C2 c1(C(N(C2CCN(C(C3CC(C)C3)=O)C2)CCO)=O)cc(C#N)ccc1O CC1(C)COc2cc(C(=O)NOCc3cn(CC4CCCCC4)nn3)ccc21 O=C(C1=CC2(CCN(C(=O)C(O)Cn3cncn3)C2)C1)NCc1ccc(O)cc1 N1(C(c2c(C)cc(CC)o2)=O)CC(C(N2CCC(C(N)=O)CC2)=O)CCC1(C)C N1(C(CC(C)OC)=O)C2COCC1CC(NC(=O)CN(C)Cc1ccccc1)C2 C(=O)(CC(C)c1cnn(C)c1)NC(CC)CNC(=O)CC1(n2cccn2)CC1 c1(C(=O)NCC2N(C(CC=CC=C)=O)CC(O)C2)sc(Cl)c(Cl)c1OC C1(CC(=O)NC(CCN(C(=O)CSc2nc[nH]n2)C)(C)C)CCC(=O)NC1 c1(OC)ccnc(C(=O)NC(CO)C(C)NC(C2CC2(F)F)=O)c1OC c1(C2CC2)cnc2[nH]ccnc1-2.CC1(C)COCC1CC(N1CCC(NCC)C1)=O CCC(C)(CCC(C)C)C(=O)NCC12CCCC1N(C(=O)Cn1cnnn1)CC2 c1(C(=O)NCC2CN(C(CCC=C)=O)C3C2C3)cnc(O)c2ccccc12 Cc1oc(C2CC2)nc1C(=O)NC1C=CC(CNC(C2CC3CCC2O3)=O)C1 C1(C(N2CCC(CCNC(CCc3c(C)noc3Cl)=O)C2)=O)CCC(C)(C)CO1 c1(C(=O)NCC2CCC(C)N(C(c3cc(C)n(C)n3)=O)C2)cc(F)c(F)cc1O c1(NC(C2CC(NC(C(c3ccccc3)C)=O)C2)=O)cnc(Cl)nc1 c1(C(=O)OC)ccc(C2CCCN2C(=O)C(n2ccc(C3CC3)n2)C)cc1 C1(CC(N2CC(O)(COC)C2)=O)CN(C(c2cc(OC)cs2)=O)CCC1C C1(C(=O)NCCCC2(NC(CN(C3CC3)CC)=O)CC2)Cc2c(C)cccc2O1 CC(C)(F)CCC(=O)NCC1(C)CN(C(c2cnc(C(F)(F)F)s2)=O)CCO1 c1(C(N2CCC(NC(C(C(C)C)C)=O)C23CCC3)=O)ccc2ncncc2c1 N1(C(C(CC)(C)C)=O)CCN(C)C(C(N2C(CO)CC2C)=O)C1 c1(SC)cc(C(N2CC(CCNC(c3ccc(O)cn3)=O)C2)=O)ccc1F C1(OC)CCC(c2cn(C(C)CNC(=O)C(C)Oc3ccc(C)cc3)nn2)CC1 C(CCN=c1c(C#N)c[nH]c2cc(F)cc(F)c12)N(C)C(C1(C)C=CCCC1)=O CC1(C)C(CNC(=O)C(=O)Nc2ncc[nH]2)CCN1C(=O)CC1CCCCC1 N1(C(C=COCC)=O)CC2CCN(C(C3CN4CCCC4CO3)=O)C2C1 C1(NC(C(C=C)(F)F)=O)CCCCCC1C(=O)NCC1CC1C(=O)OC C1(C)(C(=O)NCC(C)(C2CCC2)NC(=O)C(C)(C)n2cccn2)C=CCC1 c1(CNC(c2nc(C)c(C)n2C)c2n(C(CC)C)nnn2)cn(C)c(=O)nc1O CC(C)CC(C(=O)NCCc1cccc(O)c1)NC(c1ccc(C2CC2)cc1)=O C1(NC(CC=C=C)=O)CN(C(c2csc([N+](=O)[O-])c2)=O)C2(CCOC2)C1 C1(C(=O)NCC=CCCC)CC(CC)CCN1C(=O)CCS(N)(=O)=O c1(OC)cc(C(N2CCC2CNC(=O)CC2CCCC2)=O)cc(F)n1 C12CCN(CC1)C2=O.c1(SCC(=O)N(CCCN(C)C)C)c[nH]nc1C(C)(C)C c1(OC)ccc(NC(=O)C(C)NC(C2COC(=O)N2C)=O)cc1C C=C(C)CCC(=O)Nc1cccc(CNC(C2(C)CCC(=O)N2)=O)c1 S(=O)(=O)(c1ccc(N(C)CCc2nccs2)c(C#N)c1)NCCCC(C)CO N1(C(C2C(C)(C)C2(F)F)=O)CCOC(C)(CNC(=O)CN(C2CCCC2)C)C1 C12(C(N(CC(CNC(C(CC)(F)F)=O)O)C)=O)CCC(CC1)C2(C)C N1(C(CC(C(=C)C)OCC)=O)CCC2(C1)CN(C(c1c[nH]cc1C)=O)CCO2 c1(CC)cccc(F)c1NC(=O)CC1CCCCN1C(=O)CSCC(F)F CC(CC(=O)N1CC(CNC(c2cn(C)[nH]c2=N)=O)C(C)(C)C1)C(F)(F)F C1(NC(C(C(C)NC(c2ccsc2)=O)C)=O)CC2C(O)C(O)CC12 C(=O)(C1CCCc2cccnc21)NC(CNC(=O)CC1(O)CCCCC1)CO C1(CNC(C2C(CC)C2)=O)CCCN(C(=O)CCC2CC2)CC1 c1(C(=O)NCC2CCC(C(=O)Nc3cc(Cl)cnc3O)C2)cc(F)cnc1O N1(C(C2CCC(CC)O2)=O)CCC(NC(=O)CCn2ccc(C)n2)CC1C C1(CCCNC(C(C)N(C)C)=O)CCCN1C(=O)C=Cc1cn[nH]c1 Cc1ccc(F)c(C(=O)NC(C)C(=O)NC(c2cccnc2)CO)n1 CCC(C)(C#N)C(=O)NCC(O)CNC(c1ccnc(C)c1)=O N1(C(c2cc(C)ns2)=O)CCCN(C(=O)COCC2CCCOC2)C(C(C)C)C1 C(=O)(CCCC(=O)C(C)(C)C)N1CC(C(C)C)N(C(c2nn(C)cc2Cl)=O)CC1 N1(C(C(CC#C)(C)NC(c2ccc(F)s2)=O)=O)CCC2(CCC2)C(O)C1 c1(C(=O)NCCC2(CNC(CC3C(C)(C)C3)=O)CC2)cnc(-c2ccccc2)o1 C(=O)(C(CNC(C1CCCO1)=O)CC(C)C)Nc1c(CC)onc1C C1(CC(=O)NCCC(C)NC(c2cc(C(N)=O)no2)=O)CC2(CCC2)CCO1 N1(C(c2c(CC)ocn2)=O)CC2CC2(NC(c2cn(C)nc2-c2ccoc2)=O)C1 C12(CC(=O)NCC(C)(F)F)CCC1CN(C(=O)CC1(O)CCOC1)C2 C1(CC)COC(C)(C)CN1C(C1CN(C(=O)CCc2ccc[nH]2)CCN1C)=O N1(C(c2cc(OC)ns2)=O)CCCCC1CNC(c1ccc(C(F)F)o1)=O NC(=O)CCCCC(=O)NCCCC1CCCN1C(=O)CCS(N)(=O)=O CC(C)CCC(=O)NC1CCCC1N1CCN(C(c2ccccc2NF)=O)CC1 N1(C(C(CC)C)=O)CC2CCC(CNC(c3ncc(F)c(OC)n3)=O)(C2)C1 N1(C(COC(C)=O)=O)CCC2CCN(C(c3cc4c(C)n[nH]c4nc3O)=O)C2C1 c1(C(N2CC(C)(C(=O)NC(c3ccsc3)C)C2)=O)ccc2occc2c1 c1(OC)ccc(C(N2CC3C(N(C)C(C4CCCCN4N=O)=O)C3C2)=O)c(F)c1 N(C(=NCCCSc1ccccc1)NC1CC12CCC2)C1CC(CC(C)(C)C)C1 C(C(F)(F)CCC(=O)NC(c1cc(Br)no1)C)n1cc(CCCC)nn1 CC1CC(C)N(C(c2cnc(CC3CC3)s2)=O)CCN1C(=O)CSCCC#N c1(C(CNC(=S)NCC23CC(CCO2)C3)C(F)(F)F)c[nH]c2ccccc12 N1(C(=O)NC(c2ncc(-c3ccccc3)[nH]2)C(C)C)CC(F)C(F)C1 C(CC(C(C)C)NC(=O)Cc1csc(NC=O)n1)N(C(CC(=C)C)=O)C S(=O)(=O)(c1ccc(CC(=O)O)c(F)c1)NC(c1cnc(OC)c(C)c1)=O C1(NC(C=C(C)C)=O)CN(C(c2cnc(C)nc2C)=O)C2(CCCC2)C1 N1(C(C2(C)CNC(=O)C2)=O)CC2CC(C1)N2C(C1(F)CCCCC1)=O c1(CCCC(=O)NC2(CC=C)CN(C(c3c[nH]cc3C)=O)C2)ccccc1Br C(C(=O)N=c1cco[nH]1)N1CC(CN(C)C(c2ccnc(F)c2F)=O)C1 C1(C(C)C)CCC(C)CCN1C(c1cc(Cl)ncc1Cl)C(=O)NC(C)(C)C C1(C)(C(=O)NCCN(C(C(COC)C)=O)CC(C)O)CCCN(C)C1 c1(C(=O)NC2C3(CN(C(C4CC(SC)C4)=O)C3)CC2)cc(C)c(C)nc1C Cc1cc(C(N2CCC(C)(C)C2CNC(=O)CC2CCN(C)C2)=O)cc(C)c1 C1(CC(N2CCN(C(CNC(=O)C(F)F)=O)CC2)=O)Cc2ccccc2O1 C(=O)(C(CC(C)(C)C)OC)N(C(C)C(=O)NCCCN1CCOCC1)CC C1(NC(C2C(C)(C(C)C)C2)=O)CCC2CN(C(=O)Cc3cnn(C)n3)CC2C1 C=CCCCCC(=O)NCC1(NC(c2ccc(O)nc2)=O)CCCCC1C Cc1sc(O)nc1C(=O)NCC1(F)CCN(C(=O)C(F)C2CCC2)C1 C1(C(=O)NC(CNC(c2ccnc3cc[nH]c23)=O)CO)Cc2cc(Cl)ccc2O1 C1(CC(N2CC(CCC=C)(C(=O)NC(C)Cc3nncn3C)C2)=O)CCN(C)C1=O Cc1ccc2scc(C(=O)NC3CCN(C(=O)CCc4cc[nH]n4)C(C)C3)c2c1 N1(C(C(N2CC(C)OC(C3CC3)C2)=O)=O)CC2CCCN2CC1CO c1(C(N2CC(N(C(C3C(CC)C3)=O)C)C3(C2)CC3)=O)cc2ccccc2o1 c1(CN(CC(C)C)C(=O)NCC2(C)CSC2)nocn1 c1(C(N2CC(COC)(CNC(=O)CCN3CCC3)C2)=O)nc(OC)cc(OC)n1 C1(OCC)CN(C(=O)CCn2nnnc2C(c2sccc2Br)NC)CC1(C)C C1(C(N(C(C(=O)OCC)C)C)=O)CCN(C(=O)C(C2CCCCC2)F)C1 C1(C(=O)NCC(CN(C)C(C2(CO)CC2(F)F)=O)(C)C)C2CCCCC12 C(=O)(CC(C)CCC(=O)NCCCCCCNC(=O)CC(=O)NC1CC1)OC c1(C(=O)NCCC(=C)CNC(=O)C(C)CF)cnc(C)c2c1COC(C)(C)O2 c1(C(N2CCN(C(C3CC(CC)C3)=O)CC(O)C2)=O)ncnc2c1ccn2C c1(NC(C2CCCO2)C)ccc(S(=O)(=O)NCc2cnc3n2CCCC3)cc1Cl c1(C(N(CCC)CCNC(c2oncc2C)=O)=O)ccc(OC2CC2)cc1F N(C(=NCCN1CCCCCC1)NCC1(C)CCOC1C1CC1)CC(=C)C C1(NC(C(COC)NC(C)=O)=O)CN(C(=O)C(F)OC(F)(F)F)CC1O.C(C)(=O)O C(=O)(C(C)(C)CC(=O)NCC1OCCC1C(=O)NC(CO)C(C)CC)OC N1(C(C(=O)NCC)=O)CCCC(C)(C)C1CNC(=O)C=C(C)c1ccccc1F CCC(CC(=O)Nc1nccc(C)n1)N(C)C(=O)NC(c1nncn1C)CO C(=O)(C(CCC(N)=O)n1cnnn1)NCC1CCN(C(CC(C)(F)F)=O)C1 N1(C(Cc2scc(C)c2)=O)CCC2(CCN(C(c3cccc(C)c3C)=O)CC2)C1 C=CCC(C)(C)CC(=O)N1CC2(CC2)CC1CNC(=O)C(C)n1cccn1 N1(C(CC(=C=C)C)=O)CC2(CC(C(N3CC4CC5CC4C3C5)=O)CO2)C1 C1(CNC(C=C(C)C(C)C)=O)(NC(=O)C(F)CC2CCC2)CCCC1 CC(C(C)(C)NC(=O)C=Cc1cscn1)NC(c1cc(Cl)no1)=O N1(C(c2n[nH]c(C)c2C)=O)C2CCC1C(CNC(c1ccc(Br)cc1)=O)C2 N1(C(CCCCC)=O)CCOC2(CCN(C(=O)CCc3cccnc3C)CC2)C1 CCC(CC(=O)N1CC(CC(C)NC(c2cccc(C(C)C)c2)=O)C1)C(C)(C)C C(=O)(C(C)(O)C(C)c1ccccc1)NC1C(NC(CCSC)=O)C1 c1(OC)ccc(C2CC(COC(=O)CCCC3CC3C)C2)c(F)c1 c1(SCC)cc(C(=O)NCC2CCCN2C(=O)C(C)C2CCC2)ccn1 Cc1ccc(CN2CC(NC(C3CCCN(C(=O)C4CC4)C3)=O)C2)c(F)c1F C1(C(N(C2CCOCC2)CCC)=O)CCCC(NC(=O)C(C)CC#N)C1 C1(NC(C2C(C(=O)OC)C2)=O)CC(N(C(=O)CCn2cncn2)C)C1 C1(C(N2CC(CNC(C(C)(C)N(C)C)=O)CC2(C)C)=O)CCc2ccnn2C1 c1(C(=O)NC2CN(C(C3=CCCCC3C)=O)C2)c[nH]c2cccc(C#N)c12 C1(OC)CC(CNC(=O)Cc2nnc(C)o2)N(C(C2(c3cc[nH]n3)CC2)=O)C1 Cn1ncc(C(=O)NC2CCCCC2CNC(C2(CF)CCOCC2)=O)c1F C1(CNC(C2=CCSC2)c2n(-c3c(Cl)cccc3)nnn2)C2(CCC2)C12CCC2 N#Cc1c(N2CCCC(CCNC(c3cc(CO)[nH]n3)=O)C2)ncc2c1CCC2 C1(NC(c2[nH]c(CC)c(Cl)n2)=O)CC(OC)CN(C(C2CCCSC2)=O)C1 Cc1ccc(C(=O)NCC(O)CN(C)C(C2CC3CCC2C3)=O)nn1 c1(C(=O)NCCC2CC(NC(Cn3ncc(C#C)c3)=O)C2)cccc2nncn12 CCC(C)(C(=O)N1CC(C2CN(C(c3coc(-c4ccccc4)c3)=O)C2)C1)C(N)=O C(=O)(C1=NOC(C(=O)NCCC2CN(C(C3(C(F)(F)F)CCCC3)=O)C2)C1)OC C(=O)(C(O)C(F)(F)F)NCC(C(=O)N(CC(CCC)C)C)N(C)C c1(C(=O)NC2CC(NC(C3N(C(C)=O)CCC3)=O)C2)c(C)ccc2nonc12 C(C)(C(CC(=O)NCC1(OC)CCSC1)NC(=O)Cc1cnn(C)c1)OC C(C(C)C(=O)NCC(=C1CN(C(=O)CNC(C2CCCC2)=O)C1)F)OC C(=O)(CC1=NNC(=O)C1)N1CC(O)(CCNC(c2cccc(C)c2F)=O)C1 C(c1cc(C)c(C)cc1C)=CC(N1C(C(=O)OC)CCC(C(=O)O)C1)=O c1(NC(C2C=CC(NC(C(COC)OC)=O)C2)=O)ccccc1C(C)C CCCC(CCC)C(=O)NC(C(=O)N1CC(C(C)OC)C1)C(C)(C)C c1(C(=O)OC)cc2ccc(N(C)C(c3cccc(-n4ccc(C)n4)c3)=O)cc2o1 Cc1ccc2sc(C(=O)NC3CCN(C(c4cn(C)nn4)=O)CC3(C)C)cc2c1 c1(OC)ccc(C(=O)NC2(c3nn[nH]n3)CCC2)cc1[N+](=O)[O-] c1(-c2cc(C(=O)NC(c3ccc(C)o3)C)n[nH]2)ccc(F)cc1F c1(C(=O)NCC2C(NC(C3(C)CCCO3)=O)C2)ccnc(-c2ccccc2)n1 C1(NC(c2n(C)cnn2)=O)CN(C(C2CC2(Cl)Cl)=O)C2CCCCC12 CC(C)(CC(F)F)C(=O)N1CCCC(O)(CNC(=O)CCC2=CCCC2)C1 CC(C)CC(C)C(=O)N1CC(N(C)C)C(CNC(=O)COC2CCCC(C)C2)C1 c1(C(N(C)CC2N(C(c3n(CCC)ncc3)=O)CCC2)=O)c(OC)cccc1F c1(N2CCC(CC)OCC2)nc(N2CCSC(C)(C)C2)c2[nH]ccc2n1 C1(CC)CCCC1(C)C(=O)NCc1cc(C(=O)NCc2ncccc2O)ccn1 C1(C(N(C2CC(C#N)C2)CC(=O)NC(C)(C)CC2CCOC2)=O)CCC(=O)NC1 CC1CCC(NC(=O)C=CCN2CCC2)CN1C(C1CC2(CSC2)C1)=O N1(C(c2cc(OC)c(Cl)s2)=O)CC(C2CCCCN(C(C3CC3F)=O)C2)C1 N1(C(c2cn(CCC)nc2)=O)CC(NC(=O)C(C)=CC2CC2)C(SC)C1 C1(NC(C(C(=O)OCC)OC)=O)CN(C(=O)CCS(=O)(=O)NC)C2(CCC2)C1 Cc1cnncc1C(=O)NC1(C(=O)NOCC(N)=O)CC1(C)C c1(CC(N2CCN(CCN(C(CCC#C)=O)C)CC2)=O)c[nH]c2cc(F)ccc12 C1(N(CCCNC(C2CC2F)=O)C(c2cnsn2)=O)COC(Cn2cccn2)C1 Cc1cc(O)nnc1C(=O)NC(C)(C)CCNC(c1cc(C2(C)COC2)no1)=O C1(C(=O)NCC(C(C)C)NC(C2CC(=C3CCC3)C2)=O)CCCCC1O Cc1nc(C(N2CC(C3CN(C(=O)Cn4cnnn4)CCO3)C2)=O)sc1C n1(CCC)cc(C(=O)NC(C2(O)CN(C(=O)CSCC)C2)C)cn1 C(=O)(CC(C(F)(F)F)NC(C1CC(=O)CC(=O)N1)=O)NC(c1n(CC)ncn1)C C1(CC(=O)NCCN(C(c2cnn(C)n2)=O)CC)Cc2ccccc2NC1=O c1(C(N2CC(O)(CNc3ncc(I)cn3)C2)=O)cc2ncccc2[nH]1 C1(C(=O)NCC2CCCN(C(C(CC)C)=O)CC2)CC2(C1)CC1(CC1)C2 N1(C(CC(CC)(C)C)=O)CCN(C(c2ccoc2CC(N)=O)=O)CCC1C C1(CNC(C2(CC=C)CN(C(c3cnsc3C)=O)C2)=O)CCCCC1C c1(C(=O)NC2C(CNC(CC3(COC)CCOCC3)=O)C2)cc2cccnc2[nH]1 C1(C)(C(=O)NC(CN(C(CSCCC)=O)C)C)CC(C(C)C)=NO1 C1(C(=O)Nc2cn(C)nc2)=CN2C(=NNC2C)C=C1.N12CCCN(CC1)C(=O)C2 CCCC(CCC)C(=O)NCC1CCCC1C(N1CCC(F)(C(=O)OC)C1)=O C(=O)(C1=CC2C=CC(C1)C2)N(CC(C)CNC(=O)Cc1ccc(C(F)F)cc1)C C=C(Cl)CC(C(=O)N(C1CCOCC1)CCC)NC(c1ccc(=N)[nH]n1)=O c1(N2CC(C(C)(C)C)C2)ccc(NC(=O)CCn2cc(Br)cn2)cc1F c1(CCC)cccc(C(N2CCC(OCCNC(=O)C=C3CCCC3)C2)=O)c1 C1(C(N2CCC(CCCO)C2)=O)CCCC(c2nn[nH]n2)C1 c1(CC(=O)NCCCC(C)NC(C2(OC)CCOC2)=O)cccc(F)c1O N1(S(C)(=O)=O)CCCc2cc(-c3nc(-c4ccncn4)no3)ccc21 N1(c2ccnc(C(CC)C)n2)CC2CCC(NC(=O)CS(N)(=O)=O)CC2C1 C(=O)(C(=O)N(O)C(C)C)NC(CC)CNC(c1nccnc1-n1ccnc1)=O N1(C(C2CCCC(C)C2)=O)CCCOC(CCNC(c2ccnc(F)c2O)=O)C1 CC1(C)CC(C(=O)NCC2(C(C)(C)C)CCN(c3ncccn3)C2)CC(C)(C)C1 c1(SCC(=O)N(CC(C)NC(Cc2nc(OC)oc2)=O)C)ccc([N+](=O)[O-])cc1 N1(C(CCOCCOCC)=O)CC(C)CN(C(=O)Cc2ccsc2Cl)C(C)C1 c1(C(N2CCCN(C(c3onc(C)c3C)=O)C(C)C2)=O)c(F)ccc2ccoc12 N1(C(c2c(OC)cnnc2)=O)CCN(C(c2cnc(C(C)C)s2)=O)C(CCO)C1 Cc1cc(C(N2CCC(C(C)NC(c3cnc(=N)[nH]c3)=O)CC2)=O)cc(C)n1 C=CCCN=C(NCC1CCS(=O)(=O)N1)NC1CCN(CC(F)F)C1 C1(O)(CNC(CCC=CC)=O)CCN(C(=O)CCn2ccnn2)CC1 C1(NC(C2C(C)C2)=O)(CO)CN(C(c2cn(C)cn2)=O)C1 C12(C(=O)NCc3cccc(CC)c3)CCC(CN(C(=O)C=Cc3nccs3)C1)C2 CCCC(C)C(=O)NC(c1ccccc1)CNC(=O)C(N)=O N1(C(CN(C2CC2)CC)=O)CCCCCCC1C(=O)NCc1ccnc(F)c1 O=C(C1=CCOC1)NC1CN(C(C23CC(O)C2C3)=O)CC1O c1(C(=O)NCC2CCCN2C(C2(n3cccn3)CC2)=O)cnnc(O)c1 c1(C(C)(C)C)nnc(Cn2cc(CNCCCO)nn2)s1 c1(N2CCC(F)(CNC(c3ncc(N(C)C)nc3)=O)CC2)nc(C#N)ncc1Cl c1(C(=O)NC2CCCN(C(C(F)=CC)=O)C2C)cc(OC)c(OC)cc1O C1(C(=O)OCC2CC(COC)C2)CC12CCOc1ccccc12 CCC(C(C)CN(C)C)(c1nnnn1C(C)(C)C)NCCc1ccncc1C C1(NC(C(C)(C)c2ccno2)=O)CCN(C(c2ccc(CO)o2)=O)C12CCC2 C(=O)(C(CC(C)C)n1ccnc1)N1CCC(C(CNC(CNC(C)=O)=O)C)CC1 Cc1nccc2c1CCN(C(c1ccc(F)c(Br)n1)C(=O)NCC(F)F)C2 c1(C(=O)NC(CC(C)NC(c2coc(C(F)F)n2)=O)C)ccc2cccnc2n1 C(=O)(CCC(C)(C)F)N1CCC(CC(C)NC(Cc2c(C)noc2)=O)CC1 C1(N(C(C(C)Cc2cccnc2)=O)C)CN(C(=O)C=Cc2ncco2)CC12CC2 C1(C)(N(C)C)CCN(C(c2cc(CNC(C3CN(C4COC4)C3)=O)on2)=O)C1 N1(C(=O)NCC2CCNC(=O)C2)CCC(C(=O)N)C2CCC12.CC(C)(C)O Cc1cnccc1C(=O)NCCCCN(C(=O)C(C)SCC1CCCO1)C c1(N(C)Cc2ccc(C)c(F)c2)nc(=NC2CCC(F)CC2)[nH]c2ccccc12 C(=O)(CCCCC(F)(F)F)NCC(C1CCC1)NC(C1N(C=O)CCC1)=O c1(C(N(CC(C)NC(=O)Cn2cnc(=N)[nH]2)CC)=O)noc2c1CC(C)CC2 C1(CO)COCCN(c2nnnn2Cc2nc(C3CCOCC3)n[nH]2)C1 c1(C(=O)NC2CC(C)(C(C)C)OCC2)cc(C(F)(F)F)cc(Cl)n1 C(=O)(C1=NN(CC)C(=O)CC1)N(C1CCN(C(C2C(=C)CC2)=O)C1)CC Cc1nccn1CCC(=O)NC1CC(C)(NC(=O)CC2CCOC2C)C1 c1(OCC(=O)NCC(=C2CN(C(C(C(C)C)OCC)=O)C2)F)c(C)cccc1C C1(NC(C(C)OCCOC)=O)CCN(C(C2CCC(OC)CC2)=O)C12CC2 C(=O)(C(C)(C)CF)NC(C)C.C(=O)(C(=O)NC)N(CCNCC)CC N1(C(CC(CCCCC)O)=O)CC23CCCC2(C1)CN(C(=O)CN1CC=CC1)C3 CCCC(C)(C)CC(=O)N(C)CC1(NC(=O)CCC2CC2(C)C)CC1 c1(C(N2C(C3(NC(CCSCC)=O)CC3)CCCC2)=O)ccn(CCO)c(=O)c1 C(C)(C(=O)N(CCC(=O)N1CCC1CO)CCCO)NC(CCCC)=O c1(C(=O)NC(C(=O)NC(C(=O)OC)CC#N)C)ccc(F)c(Cl)c1 CCCCCC(O)CC(=O)NC(C(=O)NCc1nnnn1CC)C(C)CC c1(C(N2C3CN(C(CCS(=O)(=O)NC)=O)C(CC3)C2)=O)c(C)nc2sc(C)nn12 c1(C(=O)NCC(C)NC(=O)C(C)CC2CCCCC2)cc(Br)ncc1N(C)C c1(C(N(C(C)CNC(=O)Cc2cc(F)ccc2Cl)C)=O)cc(Cl)c(F)cc1F C1(NC(C(C)SC)=O)CCCCCN(C(c2c(F)ccc(F)c2Br)=O)C1 C1(C(=O)NCC2N(C(c3nc(CCOCC)oc3)=O)CCC2)CCCS(=O)(=O)C1 c1(OC)cc(C(=O)O)nc(C(=O)NC2CCCCC2O)c1 C1(NC(C=CCCC)=O)CCCCC12CCN(C(=O)C=Cc1cnc(C)s1)CC2 c1(C(=O)NC2CC(CNC(c3nn(C)c(O)c3)=O)C2)ccc(S(=O)CC#N)cc1 Cc1ccc(=O)n(CC(N2CCC(NC(c3c(C)cncc3C)=O)C(F)C2)=O)n1 C1(C(NOCC(C)(C)O)=O)CC(O)CN1C(c1nc(=N)cc[nH]1)=O C(C)(C)(C(=O)N1CC(O)CCO1)C1CCN(C(C(C)OCCC(C)C)=O)C1 c1(C(N2CCC(NC(C(CC(C)=O)C)=O)C(F)C2)=O)cc(F)cc([N+](=O)[O-])c1Br Cc1cc(C(=O)NCCCCN(C)C(c2c[nH]nc2I)=O)n[nH]1 N1(C(c2cc(CC)on2)=O)CCCC2(NC(c3ccccc3OC)=O)CC12 c1(C(N2CC(N(C(Cc3nnc(C)s3)=O)C)C2)=O)cc(CN(C)C)ccn1 C1(C(CNC(C(n2cc(C(CC)O)nn2)C)=O)(C)O)CCC(F)(F)CC1 CCCC(C)(O)CC(=O)NCC1(NC(c2ncc(Br)cc2C)=O)CCC1 c1(N2CCC(CC(C)NC(CN(CC)CC)=O)CC2)ncc(Br)c(O)n1 N1(C(=O)Cn2nccn2)CC2CC1CN2C(c1cc(C2CC2)ns1)=O C1(S(=O)(=O)N2CCC2)(CC)CC1.N12CC(C1)NC(=O)C1CC1C2=O C(=O)(CC(C(F)(F)F)N(C)C1CC1)NCC1=CCN(C(C(C=C=C)C)=O)CC1 c1(CCC(=O)N2CCC2Cn2ccc(C(=O)O)n2)nc(-c2cccs2)no1 c1(CC)nn(C)c(C(=O)N(C)CCNC(c2ocnc2C2CC2)=O)c1Cl N1(C(c2ccn(CC)c2C)=O)CCN(C(=O)CNc2ncccn2)C(C)CC1C C(CCCCCCC(F)(F)F)N1C(CC(C)C)CC(O)C1 N1(C(CCC2CC(C)C2)=O)CCCC1C(C)NC(c1nccn1C)=O C1(C(=O)NC(CC)CCCO)CCCN(C(=O)CC2CSCCO2)CC1 N1(C(CNC(C)=O)=O)CCC2CN(C(c3c[nH]cc(Br)c3=O)=O)CC2C1 CC1(NC(=O)NCc2ncco2)COC(C)(C)OC1 c1(C(N2C(CNC(C(CCC)=CCC)=O)CCC2)=O)nc(O)c(C#N)cc1C CCCCCCCCOCC(N1CCC(NC(c2snnc2C2CC2)=O)C1C)=O S(=O)(=O)(c1cc(C)cnc1N1CCC(c2ccncn2)CC1)N(CCSC)CC N1(CC=C)CCC(NC(=O)C(CCF)NC(=O)CC2CCC(=O)C2C)CC1 c1(OCC(=O)NC(C)C(C)NC(=O)Cn2cccnc2=O)cncc(Br)c1 CS(=O)(=O)c1ccc(CC(CC(=O)NCCBr)NS(=O)(=O)c2cccc(Cl)n2)cc1 C12(NC(=O)CCc3cnoc3)CC(CNC(C3CC=CC3)=O)(C1)C2 Cc1nnc2cc(N3CC(NC(C4CCCC(C)(C)C4)=O)CC(C)(C)C3)ncn12 C1(CCNC(C=CC)=O)(NC(c2ccoc2)=O)CCN(C(=O)COC)C1 CCC(CC)C(=O)N(C)CC1CCCN1C(c1ccc(-c2ncc[nH]2)nc1)=O N1(C(C(C)n2cccn2)=O)CCCCC12CN(C(C1CC(CC(F)F)C1)=O)C2 c1(C(C)NC(C2CC(N(C)C)C2)=O)nc(C(=O)NCC(O)CS(C)(=O)=O)co1 c1(C(=O)NC2CN(C(C(CSC)OC)=O)CC2C)ccc(F)c(C)c1Cl c1(N2CC3C(C)C3C2)ccc2cc(S(=O)(=O)NCCc3cnoc3)ccc2n1 c1(CC(=O)NC(C)Cn2cc(CNC(=O)CC#N)nn2)ccc2c[nH]nc2c1 Cn1nc2c(c1C(N1CC(C3(NC(c4ccc(F)c(Cl)c4)=O)CC3)C1)=O)CCC2 c1(C(=O)NC2CC2C(=O)NCCn2cc(Br)cn2)cc(Cl)c(Br)c(Cl)c1 C12CC(C)(C1)NC(=O)CC1CC(C1)O2.CC(C)(C)OC(C1(O)CC1)=O N1(C(C2CC(=C)C2)=O)CC(C2CCCCN(C(=O)CCC3C(=O)ON=C3C)C2)C1 C1(C(=O)NCc2ccc(OC)nc2)CN(Cc2ccc(C)cc2Cl)CCC1O c1(CC(N2CC(CCCCNC(CNS(CC)(=O)=O)=O)C2)=O)c(C)nn(C)c1Cl Cc1c(C(=O)NC(C2(O)CN(C(C3CC(F)C3)=O)C2)C)ncn1C CCCCC(CN(C(=O)CC(C(F)F)NC(=O)CN1CCNC1=O)C)CC N1(C(C2(C#N)CC=CC2)=O)CCC2CCN(C(c3ccc(C4CC4)o3)=O)C2C1 Cc1cnc(C(=O)NCC2(O)CCCN(C(=O)Cc3nc[nH]n3)C2)cc1Cl C1(c2cn(CC(=O)OC)nn2)CN(C(=O)CNC2(C)CCCC2C)CCO1 c1(C(=O)NC(C)CCCNC(c2cccnc2)=O)n[nH]c2c1CS(=O)(=O)CC2 CCN=c1[nH]c(C)c(C(=O)NC2(CNC(=O)Cn3cc(C(C)O)nn3)CCC2)s1 C1(N(C(C2N(C(C)=O)CCC2)=O)C)CC2CC1N(C(C1CC(C)(O)C1)=O)C2 N1(CCNC(=NCCSC)NC2CC3(CCCCC3)C2)CCC2(C)C(C1)C2(Cl)Cl c1(C(=O)NC(CNC(CCC)=O)CC)cc(C)ncc1C N1(C(c2c(Cl)cn(CC)n2)=O)CC(CNC(c2cnc(COC)s2)=O)CC1(C)C C1(OC)CCC2(C(N3CCC(CCNC(=O)C(c4ccccc4)F)CC3)=O)CC12 Cc1nc2cc(C(N3CCCC(CNC(=O)CC4C(C)C4(F)F)C3)=O)cnc2[nH]1 N1(C(=O)NC)CCC(NC(C2(C)C=CCN2C(=O)CCC(=O)N(C)C)=O)CC1 C#CCC(O)C(=O)NCCC(C)NC(c1c(C)ncn1O)=O C1(CC(=O)N(CC(=O)OCC)CC#C)CN(C(C)=O)CC1C(F)(F)F C(=O)(C1=CCCSC1)N1CCC(C(C)NC(c2nocc2Cl)=O)C1 C1(CC(=O)NCC(N(C(=O)CS(=O)(=O)N(C)C)C)C2CC2)CCCCC1(F)F c1(C(=O)NC2C(C)(CNC(CC=CC)=O)CCC2)cc(NCC)ccc1[N+](=O)[O-] C1(NC(C2CCN(C(C3(C)COC3)=O)C2)=O)CC2OC(=O)CC12 Cc1ccc(F)c2c1CN(C(c1cc(F)c(F)c(F)c1)C(=O)NC1CCC1)CC2 N#CC1=C(C(=O)NC2CC(O)CN(C(=O)CCc3c(F)cccc3F)C2)CCC1 C1(C(N2CC(N(C)C(c3cc(Cl)c[nH]3)=O)C2)=O)CCCCC1O N1(C(c2c(C)nc(O)cc2)=O)CCCC(C2CC2NC(c2ccnnc2C)=O)C1 C1(CNC(c2c(C)noc2C)=O)CCC(C)CN1C(C1CN(C2CCC2)C1)=O c1(C(N(CCCNC(c2ncc(F)cn2)=O)CC)=O)ccc(=O)n2c1CCC2 c1(NC)c(C(=O)NC2CCC(CNC(=O)CC(C)C(C)C)CC2)cccc1F c1(CS(N2CC(O)(C(C)(C)C)C2)(=O)=O)ccc2c(c1)OCCO2 n1(CC(=O)NC2C(C)CN(C(=O)C(C)(C)CF)C2)nc2n(c(=O)c1=O)CCOC2 N1(C(c2c[nH]c(=N)[nH]2)=O)CCC(NC(=O)C2=CCSC2)C(c2ccccc2)CC1 CC(CNC(=O)CNC(C1CC1(Cl)Cl)=O)CN(C)C C(=O)(CC(c1ccccc1)NC(=O)COC(C)(C)C)NCC(CN(C)C(N)=O)O C(=O)(C(C)(O)C(C)(C)C)NC(CC)CNC(c1csc(C)c1Br)=O c1(OC)ncc(Br)cc1CN1CC2CC2(C(=O)Nc2ccc(O)cc2C)C1 c1(C(CNC(c2cscc2C(F)(F)F)=O)NC(c2cnc[nH]2)=O)ccccc1F C1(C(=O)NCC2CC(NC(c3nn(C)c(O)c3)=O)C2)CCC(C2CCCO2)O1 C1(N(C(c2cn(CC)nc2C(C)C)=O)C)CCCN(C(=O)CSC(F)(F)F)CC1 C(=O)(C(F)C(C)CNC(c1ccn(C)n1)=O)N1C(CC)C(O)CC1 c1(C(=O)NC(C)CNC(C2(CO)CC2)=O)ccnn1C(C)(C)C O=C(C1=CCCOCC1)NC12CCCN(c3cc(C(F)(F)F)ncn3)CC1C2 c1(C(C2(CNC(=O)Nc3cscn3)CCC2)C2C(SC)C2)ccccc1 C(C(CC(=O)N(C1COC(C)(C)C1)C)NC(C1(c2cc[nH]n2)CC1)=O)OC c1(CC)nc(C)c(C(=O)NCC2(F)CCC(NC(c3cc(Cl)cn3CC)=O)C2)s1 c1(C2C(CC(=O)NC(C)C=CC(=O)NC3CCC3)C2)ccccc1 c1(C(=O)NCCCCCNC(C2(n3cncn3)CC2)=O)sc(Cl)cc1Cl Cc1ccn(CC(=O)N(C(C)CNC(=O)CCc2cc(C)[nH]n2)C)c(=O)c1 C(=O)(C1=NN2CCC(C)N=C2N1)N1CC(O)(C(C)NC(C(F)=C(C)C)=O)C1 c1(C(N2CCC(NC(C(COC)OC)=O)C(F)C2)=O)ccc2cc(O)ccc2c1 C#CC1CCN(C(=O)CC2CN(C(=O)C3=CCSC3)CC2C)C1 c1(CCOCC(N)C(=O)NC2(CN3CCOCC3)CC2)ccc(Cl)cc1 C(=O)(C(CCC(N)=O)N(C)C)NC(C(C)C)C(=O)NC1CCNC(C)CC1 C=CC1(CC(=O)N(CCNC(=O)CN(c2ccncc2)C)C2CC2)CCCCC1 CN1CCC(OCCC(=O)NCC2CCCC(NC(C3CC3(F)F)=O)C2)CC1 C1(NC(=O)C=Cc2cccc(F)c2)CN(C(C2CCC2(F)F)=O)C2(CCC2)C1 C1(C(=O)NC2(CC#C)CC2)CC2CC1CN(C(=O)C(c1cncnc1)C)C2 CCC(CC(=O)NC1COCC1CNC(=O)CS(=O)(=O)CCOC)C(F)F C1(CNC(c2nc(C(C)C)oc2)=O)C(C)CCN1C(c1cc(Br)n[nH]1)=O C(=O)(CC(O)CC(C)C)NC(CNC(CCN)=O)C1CC1.C(=O)(C(=O)CSC)OC CCC(CC)CCC(=O)N(C(C)C(N1CCC(CC(F)F)C1)=O)CC c1(C(N2C(CCNC(c3ccc(CCC)s3)=O)CCC2)=O)ccc(C)c(C)c1N CC(C)C(C(C)NC(c1ncccc1C1CC1)=O)NC(=O)CCc1ccccc1 CC1(C(=O)N2CCC(C3(NC(=O)CC4=CCCC4)CC3)C2)CCCc2ccccc21 C(CCC(C)(C)C(=O)NC1C=CCN(C(=O)CC2(C)CC2)C1)OC CC(C)C(F)C(=O)N1CCSCC1CCNC(C1CCCC(C)C1)=O N1(C(C2C(CC)CCC2)=O)CC(O)(C2CCN(C(c3ncn(CC)n3)=O)CC2)C1 N1(C(C)=O)CC(O)CC1C(N1CCCC(N(C(=O)C(C)(C)NC(C)C)CCO)C1)=O C1(NC(=O)CC2COCC2O)CC12CC(NC(c1ccccn1)=O)C2 C1(NC(=O)CSc2n[nH]c(O)n2)CC2CCC(C1)N2C(C1CC12CCSCC2)=O CC(F)(F)CC(C(=O)N1CC(C)(C#N)C1)NC(=O)OC(C)(C)C C1(NC(C(C)CN(C)C)=O)CC2(CCC(NC(=O)C(F)CC3CCCC3)CC2)C1 Cc1ncncc1C(=O)NC(C)C(C)(C)NC(C1CC(c2ccccc2)C1)=O N1(C(C2(CCC)CC2)=O)CCN(C(c2cc3n(n2)CCC3)=O)CC(C)(F)C1 N1(C(C)=O)CS(=O)(=O)CC1C(=O)N(CC(O)CN(C(=O)C#CC(C)C)C)C c1(CNC(C(C)OC(C)=O)=O)ccc(C(N2CCOCC2CN(C)C)=O)nc1 N1(C(CC2N(CC)C(=O)CC2)=O)CC(CNC(=O)CCC(N)=O)CC(C)C1 CN1CCCC(c2cn(C(c3nc(C(F)(F)F)cs3)C3CC3)nn2)C1 C12(CNC(c3c(C)ncs3)=O)CCCC1CCN2C(=O)Cn1cccn1 N1(C(c2cccc(C(C)C)c2)=O)CC2(C1)CN(C(=O)CC(C)C1CC1)C2 N1(C(C(CC)OCC)=O)CCC(O)(Cn2cc(-c3cn(C)cn3)nn2)CC1 C1(CNC(c2c(C)cc(OC)nc2)=O)C(C2CC2)CCN1C(C1CC=CCC1)=O CC1(CNC(C2C=CCCN2C(=O)CC2CCCC3CC23)=O)CCC(O)CC1 N1(C(c2ccn(C3CC3)n2)=O)CCC2CC2(C(=O)Nc2ccsc2)CC1 C1(C)(CNC(C(F)OC)=O)CCCN(C(c2nccc(C)n2)=O)C1 C(=O)(C(F)(F)C1=CCOCC1)N1CC(CNC(C(C(C)C)O)=O)C2(C1)CC2 NS(=O)(=O)CCCNC1(c2cn(CCc3ccc(O)cc3)nn2)CCC1 Cn1nc(C(=O)NC(CO)CCCNC(C2CCCSC2)=O)cc1F C1(C(=O)NCC2CCC(CN(C)C(C3CC34CC4)=O)CC2)CCC2(CCC2)O1 C1(N(C(COCC(C)C)=O)C)CCN(C(c2n[nH]c3c2CCC3)=O)CC12CC2 C(C(C)(O)C(C)C)NC(C1C(CNC(COC)=O)CCC1)=O N1(C(=O)C(C2CC(F)(F)C2)O)CCCC12CCS(=O)(=O)CC2 C12(NC(c3cnccn3)=O)CC3CCC(C1C2)N3C(C12CCCCN1CCC2)=O C1(NC(=O)CCc2cc(Br)cs2)CN(C(c2cnsc2)=O)CC1O N1(C(C(COCC)C)=O)CCCC(O)(CN(C(=O)COC2CCCCCC2)C)C1 C(=O)(CCCCCCc1c[nH]c2ccccc12)NCC1(OC)COC1 CC1(NC(C2CC2(Cl)Cl)=O)CCN(C(C2(Cc3cccs3)CC2)=O)C1 c1(C(=O)NCc2scc(CNC(C(CSC)O)=O)n2)ccnc(C)c1 NC(=O)CCCCC(=O)N1CC(C(=O)NC2CCC3(CC2)CC3)C(F)C1 CC1(C)C(CNC(C2CC(C3CC3)=NO2)=O)CCN1C(C12CCC(C1)C2)=O C(C)(C(CC(=O)NCCC1CCC(C)(C)C1)NC(C1CCOC1C(C)C)=O)OC N1(C(C(=O)NC(C)C)=O)CCCC12CCN(C(C1CCC1C(N)=O)=O)CC2 C1(C(NOCCN(C)C)=O)CCC(C2CC2)N1C(=O)C=Cc1ccncn1 Cc1ccc(C)c(CC(N2CC(C(=O)Nc3cc(Cl)nnc3Cl)CC(F)C2)=O)c1 C(=O)(C1=C(C#N)CCC1)NC(C1CCCCC1)C(=O)NCC(C(C)(C)O)F C1(N(C)C)CN(C(C2(C3CCCO3)CC2)=O)CC1CO.c12cnccc1NC2=O C(CC(O)C(=O)NCCC(=O)NC(c1csc(C)n1)C)SC C(=O)(CC(C)(C)CNC(=O)C=Cc1ccnn1C)N1C(CC)CCCC1 C1(C(=O)NCC(C)CCl)CCCC12CCN(C(c1cc(F)c[nH]1)=O)C2 c1(C(=O)NC(C2CCN(C(c3ccc(Cl)cn3)=O)C2)C)ncncc1C#N N1(C(c2cc(C(C)=O)on2)=O)CC2(NC(C3CC(F)(F)C3)=O)CC1C2 c1(-n2cc(C(N(C(c3n(CC)nc(C)c3)=O)C)C)nn2)cc(F)cc(Br)c1 c1(C(=O)NCC2CN(C(C(c3ccccc3)SC)=O)C2)nc(C)ccc1Br C1(CCC)(NC(c2c[nH]nc2OC)=O)CCCN(C(c2cncc(SC)c2)=O)C1 N1(C(Cn2ccc(C)n2)=O)CCC(NC(c2cc(C(F)F)ccc2F)=O)C(F)C1 C(=O)(N=c1[nH]nc(Cl)c(C)c1C)NC(c1cccnc1)CC c1(OC)ccc2nccc(CNC(=O)NCC(C)(O)C3CC3)c2c1 C=C(C)CC(C(=O)N(C1CC(C#N)C1)CC(=O)NCCC(C(C)C)OC)OC Cc1c(C(C)NC(C2CC(C)CN2C(=O)Cc2cncs2)=O)cnn1C CC(C)CCC(F)C(=O)N(CCC(=O)NCC1COCC(=O)N1C)C1CC1 C(=O)(C1NCc2nc(C)ncc21)OC(C)(C)C.C1(C(=O)OCC)COC2CN1C2 C(=O)(C1=CCCCO1)N1C(CN(C(C(CCC)N(C)C)=O)C2CC2)CCC1 C1(c2nc(CNC(C(C3CC3)SC)=O)[nH]n2)CCN(C(C23CC(C)C2C3)=O)CC1 c1(C(=O)NCC(C(C)(C)C)NC(C2N(CCC)C(=O)CC2)=O)cc(F)ccc1C C(C(C)(CO)NC(c1cn(C(F)(F)CO)nn1)=O)NC(C(C)NC(=O)NC)=O N1(C(C(C2CN(C(C=CC(C)C)=O)C2)O)=O)CCC2(CC=CCO2)C1 C1(NC(C(C(C)C)O)=O)CN(C(c2cnc(C(F)(F)F)s2)=O)C2(CCOCC2)C1 C(=O)(CS(=O)(=O)C1CC1)N1CC(CCC)N(C(=O)C=C(C)C(C)C)CC1 C12(NC(c3cnc(C)o3)=O)CCCC1CN(C(=O)Cn1cc(C3CCC3)nn1)C2 c1(NC(C)=O)cc(C(=O)N(C23C(CN(C(=O)N(C)C)C2)C3)C2CC2)ccn1 n1(CC(=O)NC2CC(CNC(c3n(CC)ccc3)=O)C2(C)C)nc(O)ccc1=O N1(C(c2c(C)nn(C)c2F)=O)CCC2(CC1)CCN(C(=O)C(C)C1CC1)CC2C Cc1cc(N)cnc1C(=O)NC1CC(CNC(=O)CC2CCC(F)(F)CO2)C1 Cc1nc(CC2CCC2)oc1C(=O)N(CC(C)CNC(c1cc(CO)[nH]n1)=O)C c1(C(N2CC(CN(C)C(c3cnc(Br)o3)=O)C2)=O)csc(C(F)(F)F)n1 Cn1ncnc1CCNC(=O)CCCC1(NC(=O)C(O)C2CC2)CCC1 C(C(CN=C(NC(C)CN(C)CC)NC1CCC2(C1)OCCO2)C(C)C)OCC N1(C(C=C(C)CNC(c2scc(C)c2C)=O)=O)CCN(C)CC(C)C1 c1(C(=O)NCC2CCC(C)CN2C(=O)COCC2(F)CC2)coc(S(N)(=O)=O)c1 c1(NC(C(CCOC)NC(c2ccnnc2)=O)=O)cnc(C)c(C#N)c1 N1(C(CC2CCC(C)(C)C2)=O)CCCCC(C(=O)NCC2CC3(C2)CC(O)C3)C1 C1(CNC(=O)C(CO)C(F)(F)F)C(C2CC2)CCN1C(=O)CCn1ccnn1 CC(O)(CNC(c1sccc1C1CC1)=O)CNC(C1CC1c1ccco1)=O Cc1ccc2c(c1)CC(C(=O)NC(C)(C)CNC(=O)CC1CCC3(CC1)CC3)S2 C(=O)(CC(C)P(C)(C)=O)N(CCN(C(C(C)=C1CCCC1)=O)C)C(C)C N1(C(c2c(C)ccnc2)=O)CCC(C2(NC(C3CCC(CCO)CC3)=O)CC2)C1 CCCCC(O)C(=O)NC1CCN(C(c2cn(CCN(C)C)nn2)=O)C1(C)C CN1CCC(C(=O)N(C)CCNC(=O)CCc2cncn2C)CC1 N1(CCNC(=O)OC(C)(C)C)CCCC(C)(NS(=O)(=O)CC2CS(=O)(=O)C2)C1 CC1(C)CC(C(N2CC(F)(CO)C2)=O)N(C(c2cnc3n2CCC3)=O)C1 C(C(COC)CC(=O)N1CC(C(=O)N(CC(C)OC)C)C(C)C1)OC N1(C(C(C)OCCC=C)=O)CCN(C(=O)C=Cc2ccc(Cl)cc2)C2(CC2)C1 C(CC)(C(=O)NCC#CC(=O)N1CCCC1C1CCOC1)OCC CCCCC(CNC(=O)C=C(Cl)Cl)NC(=O)C(O)COCc1ccccc1 c1(C(N(C(C(=O)NCC(C)C(F)F)C2CC2)C)=O)ccc(O)nc1 c1(OC)cncc(C=CC(=O)NCC2CC2NC(=O)CCCN2CCOC2=O)c1 N1(C(c2cc(Cl)n[nH]2)=O)CCCc2cc(-c3ccccc3F)ccc21 CCC(CC(C)C)C(=O)NCC1(CNC(=O)C(C)CC2CCCC2)CCC1 c1(C(N(C(CN(C(c2c(C)ccnc2)=O)C)C)C)=O)[nH]ccc(=O)c1C Cn1nnc(C(=O)NC2COCC2CNC(=O)CCc2cccc(F)c2)c1N CC(C)(C)C(=O)C(=O)N1CC=CC(C(=O)NOCCC2CC2)C1 C=C(Cl)C(C)(C)C(=O)N1CCC(O)(CN(C)C(C2(CC)CC2(F)F)=O)C1 C1(COC)(NC(c2c(Cl)ccnc2C)=O)CCCN(C(c2cccc(N)c2)=O)C1 C1(C(N2CC3CC2CC3O)=O)CCOCCN1C(=O)Cn1ccnn1 C1(CNC(=O)CC2CC2)CC(NC(=O)C(O)c2ccco2)C1 N1(C(c2sc(Br)cc2Cl)=O)CCCC2CNCCCC12 c1(C(=O)NCC2CN(C(c3cnn(CC)n3)=O)C2)c(Br)nc2n1CCC2 C1(CC)CN(C(=O)C(C(C)C)N2CCCC2=O)CCC1N=c1[nH]nc(C#N)s1 C(=O)(C(C)(C)C(=O)NC(CNC(c1ccccc1OC1CC1)=O)C1CCC1)NC C1(NC(c2cccnc2)=O)CCC(C(N2CC(NC(=O)C3CC3)C2)=O)C1 CCC(CC(=O)N1CCC(C)(CNC(=O)CCCCN(C)C(C)=O)C1)C1CC1 Cc1cccc(F)c1N(C(=O)CONC(=O)CN1C(C)CCC1C)C1CC1 n1(CC(=O)NCC(C2CCC2)NC(c2ncn(C)c2)=O)ncccc1=O c1(OC)ccc(C)c(C(=O)N(C)CC2CCN(C(=O)C(C)S(C)(=O)=O)C2)c1N C1(CN(C(C(N2CCSCC2)C)=O)C)CN(C(=O)Cc2ccsc2)CC12CC2 c1(CC)cc(C(N2CCSCC2C(=O)NC2(CCO)CCC2)=O)c(C)o1 C1(C(=O)NC2(C3CN(C(C4N(C(N)=O)CCC4)=O)C3)CC2)CCn2cncc2C1 C1(C(=O)NC23CC(F)(C2)C3)(CC)CCN(C(=O)C2=CCCC2)CC1 C1(C(=O)NCCOCCNC(C(CC=CC)C)=O)CCC(F)(F)CC1 c1(C(=O)OC)cc(Cl)c(N2CCC(CCNC(c3[nH]c(C)nc3C)=O)C2)nc1C C#CCCCCC(=O)N1CC2(C)CC1(C(=O)NCCOC1CCOC1)C2 c1(N2CCN(CC#CC)CC2)ncnc(C)c1C#N C1(CC(=O)NCC2CC(NC(c3ccc([N+](=O)[O-])o3)=O)C2)CC(=O)NC(=O)C1 Cc1cccc2cc(C(N3CCCC(CCN=c4[nH]nc(O)s4)C3)=O)nn12 c1(C(=O)NCCSCC(=O)NC(C(CCC)O)CO)ccc(C#N)cc1C C1(NC(C2(C#C)CCC2)=O)CN(C(c2c(C)nn(C)c2Cl)=O)CCC1C N1(C(C2N(C(C(C)Cc3ccccc3)=O)C3CCC2C3)=O)CCCC(C)(O)CC1 c1(NC(=O)NCC2(OC)CCS(=O)(=O)C2)ccc(C#N)c(CSC)n1 N1(C(CC(CC)C)=O)CCCCC(CCC(=O)NCCc2ccc(F)cc2)C1 c1(OC)cccc(C(=O)NCC(CO)NC(=O)CCc2ncccc2C)c1 N1(C(C(=O)NCC(F)(F)F)=O)CCCC2(CNC(=O)CSc3ccccc3)CC12 c1(C(=O)NC(CNC(C2(CCC=C)CC2)=O)CCC)onc2c1CCCC2 C1(CNC(=O)Cn2cc(Cl)cn2)C2CN(C(c3cnncc3O)=O)CC12 C#CCCCC(=O)NCC(c1ccc(C)cc1)NC(C1(C)COC(=O)N1)=O c1(C2C(C(N(CC(CC)NC(=O)C=Cc3cnc[nH]3)C)=O)C2)cccc(Cl)c1 Cc1cc(O)c(Cl)cc1C(=O)NC1(CCCNC(C2C=CCCC2)=O)CC1 C(c1cccnc1)=CC(=O)N(C)CC1N(C(C(CC)F)=O)CCC1 CC1(CCNC(C2(C)COCCO2)=O)CCN(C(c2ccccc2C2CC2)=O)C1 C1(NC(c2ccc[n+]([O-])c2)=O)CC(O)CN(C(=O)CCC=CBr)C1 c1(C(N(CC(CC)NC(C2CCC(=O)N2)=O)CC)=O)cccnc1OC(F)(F)F c1(C(N(C)CCNC(c2ccc[nH]2)=O)=O)ccc2c(c1)C(=O)OC2 Cc1cccc(N(C(=O)NCc2nc(C(C)(C)O)n[nH]2)CC2CC(Cl)=NO2)c1 N1(C(C2CC23CCC3)=O)CC2(CCN2C(C2CCCC2F)=O)C1 C1(C)(CC)CC(C(=O)NCC(C2CCNCC2)C)CCO1 C1(C(N(CCCN(C)C)CC)=O)CC2CC1CC2NC(=O)CN1CCC(O)CC1 N1(C(c2c(OCC)cccc2)=O)CCCCC(NC(=O)C=C2CCSCC2)CC1 N1(C(c2n(CCCC)ncc2)=O)CC(C)C(C)(CNC(=O)CCOCC(C)C)C1 C1(CC=C)(C(=O)NCCC2CCCN2C)CCCN1C(=O)Cc1cccs1 N1(C(CCSCCN(C)C)=O)CC2(CC(NC(c3cnc(C(F)(F)F)s3)=O)C2)C1 C1(NC(C(CC)C)=O)CCN(C(C23CC4CC2C3C4)=O)CCC1CO Cc1cc(N)cnc1C(=O)NC(C(=O)N(C1CC2CC2C1)C)c1ccoc1 N1(C(C=Cc2cc(C)no2)=O)CCN(C(C2CCCN2C(C)C)=O)CC1CCO C1(NC(C2(CCC=C)CCCC2)=O)CCCCC1CNC(=O)C1=CSCS1 N1(C(CCCNC(=O)OCC)=O)CCCN(C(=O)CC2(CO)CCCC2)CC1C C1(C(N(C2CCCN(C(c3ccc(CO)s3)=O)C2)CC)=O)C(C)(C)C1(C)C c1(CC(=O)NCC23CC(NC(C(C)OC(C)(C)C)=O)(C2)C3)cnn2ccccc12 Cc1cc2[nH]c(C(=O)N(C)CC3CCN(C(=O)CC(C)(F)F)C3)cc2o1 N1(C(c2cnc(C(=O)OCC)s2)C(=O)NCC)CCC(O)(C(Cl)(Cl)Cl)C1 C1(C(N(CCCNC(=O)C(C)Cc2ccco2)C(C)C)=O)CCc2ncnn2C1 c1(C(N(CC(CN(C(c2c(C)c[nH]n2)=O)C)O)C)=O)coc2c(C)cccc12 O=C(CCN=C(NCc1cccs1)N1CCC(NCC2CC2)C1)N1CC1 N1(C(C=C2CCN(C)C2)=O)CCC(NC(c2cc(C(F)F)no2)=O)C(C)(C)C1 CC1CN(C(=O)CC2CC(=O)NC2=O)CC(C)CN1C(=O)C=CBr c1(N(C2CCN(C(C3CCC(CC)CC3)=O)C2)C)nc2cccnc2s1 N1(C(CC2CN(C)C2)=O)CCCC1CCNC(=O)Cn1cnnn1 c1(OCCC(=O)NC(CNC(C2(n3ccnn3)CC2)=O)CO)cccc(Cl)c1Cl C1(OC)(CNC(=O)CC(=O)NCC(F)(F)F)CCN(C(=O)CC2(C)CC2)C1 c1(C(N(CCCCN(C)C(C2CCC(O)C2)=O)C)=O)[nH]nnc1-c1ccccc1 C1(C(=O)NCCSC)CC(C)N1C(=O)Cn1cnc(=N)[nH]1 N1(C(C(C(C)C)O)=O)CCC(NC(=O)C=CCF)C(O)C1 c1(C(=O)NC2CCC(NC(C(N(C)C)C3CC3)=O)CC2)c[nH]c2ccc(F)cc12 c1(CN(CCOC)C(c2ccccc2)C)ccc(Cl)cc1 CC(C)(CNC(=O)CNC(N)=O)CCNC(c1cccc(-c2ccoc2)c1)=O C(=O)(CN=c1cc[nH]cc1)N(CCN(C(=O)C(CO)C(C)(C)C)C(C)C)C c1(C2(C(=O)NCC(C)NC(=O)C(CN(C)C)N(C)C)CC2)ccc(F)cc1F CC1OCCN(C(c2ccncc2)=O)C1C(=O)NC1CC(CCO)C1 CCC(CN=c1nc(N(C)CCc2ccccc2F)c2sccc2[nH]1)C(C)(F)F c1(CC)n[nH]c(=NC(=O)N(C)C(c2cccc(O)c2)C)s1 c1(NC(C(CCSC)O)=O)ccc(NC(C2CN(C(C)=O)C2)=O)c(C)c1 C1(NC(C(C)NC(=O)NC)=O)CCSC12CN(C(c1scnc1C(C)(C)C)=O)C2 N1(C(CSCC#C)=O)CCC(N=c2[nH]nc(C(=O)OC)o2)C(CC)C1 c1(CC=C)cc2cc(OC)c1o2.c12csc(n1)CNC2.c1(C)ccccc1.OCC c1(CCC(=O)NCC(C)NC(C2CC2c2ccsc2)=O)cccc2c1OCO2 CCCCCCC(C)C(=O)N1CCC(CCC(=O)NCC(C)C#N)CC1 C1(C(=O)OC)CCC(C(=O)NCCS(C)(=O)=O)(NC(CCO)CC(C)C)CC1 CCC(C)CC(C(=O)N(C)Cc1ccc(C)cc1)NC(c1cc(C#N)c[nH]1)=O c1(C(CNC(c2c(CC)nco2)=O)NC(=O)CCSC)ccccc1OC C1(C(=O)OC)Cc2c(C)cccc2CN1C(=O)C(=O)Nc1cccnc1 C1(NC(CCOCC(C)C)=O)CN(C(=O)C(C)c2cc[nH]n2)C2(CCOCC2)C1 C1(C(C)O)COC(c2ccccc2)CN1CC(=O)C1CC1 N1(C(C2C(CC)N(C)CC2)=O)CCC2CN(C(c3ncc(Br)cc3C)=O)C2C1 c1(C(=O)NC2C(C)CCN(CCO)C2)cc2ccccc2s1 N1(C(C(=Cc2ccco2)C)=O)CC2CC(C1)CN(C(=O)CC(=O)NC1CC1)C2 CC1CN(C(=O)CC(C)n2cccn2)CC1CCNC(C1CC(O)C1)=O C1(CNC(=O)C=CCn2cncn2)CC(F)(F)CN1C(c1cccc(CF)c1)=O N1(C(C2CN(C(Cc3c(C)noc3C)=O)CC(F)C2)=O)CCc2ccccc2C1 CC1OC2(C)CC1(C(N1CC3CC3(NC(C3CCCCC3O)=O)C1)=O)C2 CCC(CC)(CC)C(=O)N1CCCC(NC(C2CCCN(C(C)C)C2)=O)CC1 C(=O)(N1CC(C)(O)CO1)C1CCN(C(c2cc(CC)[nH]n2)=O)C1CC C1(C(=O)Nc2cc(Br)cc(Cl)n2)CN(C(c2ccc(O)cn2)=O)CC(F)(F)C1 S(=O)(=O)(C1CCOCC1)NCC1N(C(C(C(C)C)O)=O)CCCC1 c1(C(=O)NC(CC=C)CNC(=O)Cc2csc(S)n2)cnc2c(cnn2C)c1N N1(Cc2nc(CCCC)sc2)CCC2(CN(C(C3CCC4CCCCN34)=O)C2)C1 C1(C(=O)NCC#CC(=O)NCC(C)C2CC2)C2CC3C(C2=O)C13 c1(CC(=O)N(C)CC2CCN(C(C3(C)CCCN3C)=O)C2)nc2ncccn2n1 N1(C(CC(CC)SC)=O)CC2CC(C1)C2NC(=O)C(N1C(=O)CCC1=O)C N1(C(C(=O)NCC2CCOCC2)=O)CCOC(CC(c2ccc(O)cc2)=O)C1 N(C(=N)N1CCCC(Cc2nnn(-c3ccc(F)cc3)n2)C1)CC(C)C N1(C(C2C(CCC)C2)=O)CC2CCC1CN2C(C1(OC)CCSC1)=O C1(C(=O)NC2CN(C(c3n(CC)ncc3)=O)CC23CC3)CCc2c(nnn2C)C1 C#CCC(O)C(=O)N1CC(CCC=C)(C(=O)NCC(C)C(=O)OC)C1 c1(CCNC(CN(C)C(N)=O)=O)ocnc1CNC(=O)CCc1cnn[nH]1 c1(C(N2CC(NC(C(C)P(C)(C)=O)=O)C(O)CC2)=O)ccc2n[nH]cc2c1 C#CCC(C)(C)C(=O)NCCCNC(=O)C(C)Cc1ccc(Cl)c(Cl)c1 C(CCCC(C)(C)NC(=O)Cc1ncn2c1CCC2)NC(C1C(CC)CCC1)=O C(=O)(C(C)(C)CC(=O)N1CCC(O)(CNC(C2OCCO2)=O)C1)OC N1(C(c2cc(OC)c(C)nc2)=O)CCCC12CCN(C(=O)CC13CCCC1C3)C2 Cc1cc(C(=O)NCCC(C)NC(=O)Cc2cncs2)ncc1C#N C1(CC(=O)NCC(CN(C(C2COC(=O)C2)=O)CC)(C)C)CCN(C(C)=O)CC1 C1(CNC(c2ccc(CO)s2)=O)CCCN(C(=O)C(F)(F)CO)C1 N1(C(=O)OC(C)(C)C)CCCC2(CNc3nc[nH]c4ncnc3-4)CCCC12 c1(COCC(=O)NC2CN(C(C(C(C)C)O)=O)CC(F)C2)ccc([N+](=O)[O-])cc1 CC1C(NC(c2cc(-c3ccco3)on2)=O)CCCN1C(C1CS(=O)(=O)C1)=O C1(CNC(c2onc(CC)c2C)=O)CN(C(C2CC3CCC2O3)=O)CCCO1 c1(CN=C(NC2CCN(C(CCC=C)=O)C2)NC(C)C)cc(C)nc(O)c1 CC1=C(C(=O)NCC2(F)CCN(C(c3c[nH]c(=N)s3)=O)C2)CC1 CCC(C)C(=O)C(=O)NCCC1(C(N2CCC(COC)CC2)=O)CC(=O)C1 c12ccc(cc1)-c1cccc(n1)-c1nccn1C2.c1(CCOC)noc(CO)n1 N1(C(C(c2c(C)cccc2)(F)F)=O)CC2CC1CC2CNC(=O)C(C)NC(N)=O C1(NC(c2cc(C)on2)=O)CCCC12CCN(C(c1cccc(N(C)C)n1)=O)C2 C1(CC)Oc2cc(Br)ccc2C1NC(=O)C(=O)NCC#CCc1ccccc1 c1(NC(CC(=O)OCC)C)nc2cccc(C#N)c2n1C N1(C(C=NOC)=O)CC2CCN(C(c3cc4scnc4[nH]3)=O)CC12 CC(CC(N)=O)C(=O)NCC1CCN1C(c1cc(-c2ccc(O)cc2)on1)=O C1(C(=O)OC)CCC(F)CN1C(C1CC(C)CN(Cc2ccccc2)C1)=O C1(CCNC(c2c(C)nc(CO)s2)=O)CN(C(=O)CNC=O)CCS1(=O)=O N1(C(CC(=O)OCC)=O)CCOCC1CC(N1CCC(C)(COC)C1)=O c1(CC(=O)N(CC(C)NC(C2C(OCC)C2)=O)CC)cnc2ncccn12 C(=O)(CS(=O)(=O)CCO)N1CC(OCCNC(c2ccc(N)cc2F)=O)C1 C12CC3CN(CC13)C2=O.C1(COCC)CCCN(c2cc(OC)ncn2)C1 c1(C(=O)NC2CCN(C(C=NOC)=O)CC2CO)n[nH]c2c1CCOC2 Cc1nc(C)c(C(N2CCC(NC(=O)CC3CCCC(C)C3)C2)=O)c(C)n1 c1(C(N2C(CCNC(CC3CC(C)(C)C3)=O)COCC2)=O)ccc2cc[nH]c2c1 Cc1cc(C(=O)NC(C2(O)CCN(C(C3(N(C)C)CCC3)=O)C2)C)cnc1O c1(CC)occ(C)c1C(=O)NCCCN(CCCNC(=O)CN1CCSCC1)C C12(C(=O)NC3CCC(F)(CNC(c4ccc(C)s4)=O)C3)CCC(CO)(CC1)C2 N1(C(=O)NC)CC(C(=O)N(CC(C)NC(=O)Cc2ccsn2)CC)C1 c1(C(N2C(CC)C(NC(C3(C)CCC3)=O)CC2)=O)ccc(S2(=O)=NCCC2)cc1 Cc1cc(C(N2CCC(NC(=O)C(C)(Cl)Cl)C(CO)C2)=O)cc(N)c1Cl C1(C(=O)NCC(=O)Nc2ccccc2)CCCN1CC(F)F O=C1CC(C(=O)NCCC2CCN(C(c3ccn(CCF)n3)=O)C2)(CF)C1 c1(OC)cccc2c1OCCCC2NC(=O)NCCCCC(F)(F)F c1(OCC(OC)OC)ccc(C)cc1NC(C1CC(F)CN(C(C)=O)C1)=O c1(C(N(C2CC23CC3)C)=O)nc(Br)cnc1N.CCC(CN)NC=O c1(CC)cc(C#N)c(NC(C2CC(O)CN2C(C2CCC(C)(C)CC2)=O)=O)s1 c1(C(=O)NCCC2(NC(=O)CC3(O)CC3)CC2)csc(C(F)(F)F)c1 N1(CC(Cc2cn(C(COCC)C(=O)OC)nn2)O)Cc2ccccc2C1 C1(CC(N2CC(C(N)=O)C2)=O)C2CCCC2N1C(C1(O)CCCCC1)=O c1(C(=O)NCCC2(O)CN(C(C3C(C)CCS3)=O)C2)cccc2c1OCCN2 c1(C(N2C(C(=O)NC(C)(C)CO)CC3(CC3)C2)=O)cc2cc(Br)ccn2n1 N1(C(C2(C(C)=O)CC2)=O)CC2(C1)CN(C(=O)CNc1nccc(OC)n1)C2 C1(NC(C2CCCN(CC)C2)=O)CCN(C(C2CCS(=O)(=O)C2)=O)CCC1CO c1(C(=O)NC2C(C)N(C(c3cnnc(O)c3)=O)CC2)ccc2c(c1)CCOC2 N1(C(c2ccc(OC)cc2)=O)CCC(F)(C(N2CCCC(N(C)C)C2)=O)CC1 C1(CNC(C=CC=CCC)=O)CCCN(C(=O)C(C)CCC)C1 C12CCC(CC1)CNC(=O)C2.C1(NC(C2(OCC)CCC2)=O)COC(C(F)F)C1 CN1N=C(C(=O)NC2(CNC(=O)CC3CC(F)(F)C3)CCCC2)CCC1=O c1(C(=O)NC(C2CCN(C(C3C=CCC3)=O)C2)(C)C)cc2[nH]ccc2s1 c1(OC)csc(C(=O)NC(CNC(C2COCC2(C)C)=O)C(C)C)c1OC C1(C(=O)NC(CCCC)CNC(=O)CCC(=O)NC2CCCC2)CCCS(=O)(=O)C1 C1(C(N2CC(NC(=O)C(=C3CCCCC3)F)CC(C)C2)=O)CC(C)(C)OC1(C)C Cc1cnc(C(=O)NC2CCC(N(C(=O)C(C)n3cccn3)C)CC2)c(F)c1 c1(C(N(C(=O)C(=O)NC2(F)CC(C(=O)OC)C2)CC)C)cccc([N+](=O)[O-])c1 Cc1cc(C#N)ccc1C(=O)NC(C)C(C)C(=O)NCC1CN(C)CCN1C C1(CNC(=O)Cc2csnn2)CC2CCC1N2C(C1CCC2CC2C1)=O c1(C(=O)NCC2C(NC(C3(C#C)CCOCC3)=O)CCC2)c[nH]c2cccnc12 N1(C(C2C(C=C)CC2)=O)CC(NC(c2snnc2C(C)C)=O)CC(C)(C)C1 CCCC(C)(O)C(=O)N1CCC(CC(N2CC3CCC3(OC)C2)=O)CC1 C(=O)(C#CC1CCCCO1)NC1C(CO)CCN(C(CN(C)C2CC2)=O)C1 c1(C(N2CC(C=C)C(NC(=O)Cc3csc(Cl)n3)C2)=O)ccc2nc[nH]c2c1 c1(N(CCOCC)CC)ccc(S(=O)(=O)N2CC(C)CC(C)C2)c2ccncc12 N1(C(C(CC=C)(C)C)=O)CCC(C2CC2)(CNC(C2(OC)CCOCC2)=O)C1 C1(O)(CCNC(c2nc(C)sc2)=O)CCN(C(=O)Cc2ccc(O)cn2)C1 c1(OC)c(O)cc(C(=O)NC(c2ccc(O)nc2)C)cc1C#N C(N=c1[nH]cnc(NCC(C)Cn2nc(C)cc2C)c1C)c1occ(C)c1 Cc1cc(F)cc(C(N2CCN(C(c3c(F)cc(O)cc3F)=O)C3CC23)=O)c1O C(=O)(C#CC1CCCO1)NCC1CC(NC(C(C(C)C)O)=O)C1 c1(C(C(=O)NCC2(F)CC(CNC(C3CC(=C)C3)=O)C2)O)ccccc1Cl N1(C(CC2(CSC)CC2)=O)CCC2CN(C(c3cccc(NC(N)=O)c3)=O)C2C1 c1(C(N2CCC(OCCCC(=O)OC)CC2)=O)cc(Br)c(C)cc1Br C1(CCC(=O)NC(C2(O)CCC2)C)CCCN(C(c2cc(=O)cc[nH]2)=O)C1 Cc1cccc(C(=O)NC2CC2CNC(c2ccc(NC(N)=O)cc2)=O)c1C CC(C)CCCCCC(=O)N1CCN(C(=O)C(C)(C)CC2CC2)CC1CO c1(C(=O)NCC2(C)CCC(NC(c3ncn(C)c3)=O)C2)nc2cnccc2s1 N1(C(COCC#C)=O)CC(CNC(=O)Cc2c(C)nc(O)nc2C)C2(CCC2)C1 C=C(F)C1(CC(N2CCCC2C2(C(=O)NC3CC(=O)N(O)C3)CC2)=O)CCC1 CC(C)(C)CCn1cc(-c2nc(-c3ccc(C)o3)sc2)nn1.CO c1(CC(N2C(C(C)NC(C3CC3OCF)=O)CCC2)=O)ccc(OC(F)F)cc1 N1(C(c2c(CC)cncc2)=O)CC2C=CC1C(C(=O)NCC(C)(COC)CC)C2 c1(C(=O)NC(C)CC(=O)NCCC(O)C2CCC2)nccnc1N N1(C(C(C)(CO)OC)=O)CCN(C(c2cc3ccccc3cn2)=O)CC12CCC2 c1(C(=O)NC2C(CNC(CCCC(N)=O)=O)C2)cc2cc(Br)cnc2s1 CC(CNC(c1ccccc1)=O)(CO)N.C(=O)(CC=CCC1CCCC1)C(=O)CS c1(CCNC(=O)Nc2nc(C(=O)OCC)c(CC)s2)ccc(F)c(F)c1 C(CN=c1nc2c(cnn2C)c(NCCc2n[nH]c(O)n2)[nH]1)OCCOC CC1(C(N2CCCCC2CNC(C2CCCC2CF)=O)=O)CCOCC1 c1(C(N2CC3C(C(=O)Nc4cnc(OC)nc4)(C3)C2)=O)ccc(C)nc1Br Cc1cc(C(=O)N(CC(O)CNC(c2cc(CO)n(C)n2)=O)C)[nH]c1C C1(C#C)(NC(C2(CC#C)CN(C(c3coc(C)c3)=O)C2)=O)CC2CCCC12 N1(C(CCN(C(=O)C(C)n2cccn2)CC=C)=O)CCCC2CCCCC12 Cc1nc(NC2(CNC(c3cc(Cl)cn3C)=O)CCC2)c(Cl)cc1C#N C(C(C)N=c1[nH]c2ncnc-2c(C(=O)NC)[nH]1)NC(CCc1ccnc(C)n1)=O N1(C(c2c(CC)cc[nH]2)=O)CC(NC(c2ccc(C(C)=O)[nH]2)=O)C(SC)C1 Cc1cccc(C2CC2C(=O)NC2CC2(F)F)c1.C12(O)CN(C1)C(=O)CCCOC2 c1(C(N(CCCNC(C2COCC2C(N)=O)=O)CC)=O)cc(C)cc(Cl)c1 N1(C(c2c(C)cn(C)c2)=O)CCC(F)CC1C(=O)N(C)CCC1CCCN1C C12(C(N(CCNC(CN3C(C)CCC3)=O)C)=O)CCC(CC1)C2(C)C N1(C(c2ccn(C)n2)=O)C(CNC(c2[nH]nnc2C2CC2)=O)CC2CC12 C1(F)(CNC(CCNC(COC)=O)=O)CN(C(=O)CC2CCC(C)O2)C1 c1(C(N(CCCOCCN(C(c2c(C)cc[nH]2)=O)C)C)=O)c(C)noc1C(C)C N1(C(c2ccc(CNC(C(CC(C)C)OC)=O)o2)=O)CCC2CCCC2C1 C1(NC(Cc2cc(C)sc2)=O)COCCN(C(C23CCCC2CCC3)=O)C1 N1(C(C2(F)CCN(C(C(C)NC(=O)OC)=O)C2)=O)C2CCC(C(N)=O)C1CC2 C1(CNC(C(C)(C)C2CC2)=O)CC12CCN(C(C13CCCN(CCC1)C3)=O)CC2 C(=O)(C(C)C(O)C(C)C)N1CCC(C(=O)N(C2CCN(OC)CC2)C)(OC)C1 C(=O)(C#CC(C)(C)C)Nc1cn(-c2ccn(C(C(C)C)C(=O)N3CCCC3)n2)nn1 c1(CC)cc(C(=O)N(CCCNC(c2cncc(O)c2)=O)C)cc(Cl)n1 C1(NC(CN2CC(CC)C2)=O)CCN(C(=O)C(c2ccccc2Cl)C)CC1C Cc1nc(CCNC(=N)NCCCOC(C)(C)C)n[nH]1 N1(C(C(C2(O)CN(C(C3CC3(F)Cl)=O)C2)F)=O)CCCC12CCOC2=O c1(C(=O)NCCN(C(C2(CC=C)CC2)=O)C)cnn(C)c1CC C(=O)(CCCCCC(C)(C)C)Nc1cccc(NC(C2CC(C)=C(C)CC2)=O)c1 C1(NC(C(C)SC)=O)CC2CCC(C1C)N2C(=O)CCCCCF c1(C(=O)NC(C)CCCNC(C2(C#N)CC=CC2)=O)cnc2c(c1)CCCC2 N1(C(CC#N)=O)CCCC(CCCCNC(C2CC(=O)NC2=O)=O)C1 c1(C(=O)NC(CCCNC(CC2C(CC)C2)=O)C)nccnc1C C1(CNC(c2cc(CC)ncn2)=O)CN(C(c2nccn2C(C)C)=O)CCN1C C1(C(=O)NC(C)CSC(F)F)CCC2(CC2)N1C(=O)C(C)Cn1cccn1 c1(C(=O)NCC(CCCC)NC(=O)CC2CN(C)C2)nc2ncccn2n1 Cc1c(C(=O)NCC2C(C)CCCN2C(=O)CC(C2CC2)C2CC2)c(Cl)nn1C C(C(=O)N=c1cc(C(F)F)[nH][nH]1)c1ccc(OC)nc1 C(CNC(c1n[nH]cc1Br)=O)(CC(C)C)NC(CCN(C(C)=O)C)=O c1(C(=O)NC(C)CCCNC(c2ncncc2F)=O)cccc(=O)n1C N1(C(C2(CCC=C)CC2)=O)CC(C(=O)NC2(C)CC3CCC2C3)C2(CCC2)C1 CC1CCC=C1C(=O)N1C2CCC1C(CNC(=O)CN1CC(=O)NC1=O)C2 N1(C(CC2(CC)CCC2)=O)C2CCCC1CN(C(c1ccoc1)=O)C2 C1(C2CCSCC2)(NC(C(=O)NCC(C)S(N)(=O)=O)=O)CC1 Cc1sc(NC(=O)CN2CCSC(C(C)C)C2)c(C)c1C C1(CNC(C2CC3CCCCN3C2)=O)CC2(CC2)CN1C(C1CCCCS1)=O Cc1sc(Br)nc1C(N1CCCCC1C)C(=O)NCC1CCCO1 N1(C(c2ccc(C)o2)=O)CC2(CCN(C(=O)CN3CCc4ccsc4C3)CC2)C1 CC1(C)CCN(C(c2sc(Br)c(Cl)c2Cl)=O)CCS1=O N1(C(C2C3CN(C)CC32)=O)CCN(C)C(C(=O)NC2CC(C(C)(C)O)C2)C1 C12(C(=O)NC3C(OC)C(O)C3)COC(C1)C(NC(c1cc(C(N)=O)co1)=O)C2 C12(C(=O)NCC(C)=CC(N3CCCC3Cn3cccn3)=O)CCOC(C)(C1)C2 c1(C(C)OC(C(C(C)C)F)=O)cnc2ccsc2c1 c1(NC(=O)CCCN(C)C)cc(Br)ccc1I.CC1CC2CN1C2 C1(CC(C)C)Oc2cc(Br)ccc2C1NC(N1CC(C)C(C)C1C)=O C(=O)(CC(O)CN(C)C)NC(C1C(C(=O)Nc2c(CC)csc2)C1)C CC(CCC(=O)NC(C)C(CO)NC(=O)CSCC(F)F)N(C)C C(=O)(N=c1cccn[nH]1)C12C(C)(C)C1CN(c1ncnc3occc13)C2 C1(NC(c2c(CC)onc2)=O)CCSC12CN(C(=O)C=Cc1ccc(=N)[nH]c1)C2 c1(C(=O)NC2C(NC(Cc3nc(C)c(C)o3)=O)CC2)cncc2c1CCC2 c1(CNc2cc(N3CC(COCC)OCC3)nc(C)n2)ccc(S(N)(=O)=O)s1 C1(C(=O)NCC(CNC(Cc2n(C)nnc2)=O)O)CCn2cncc2C1 c1(C(N2C3C(C(=O)NCCCC4CC(C)C4)C(C3)C2)=O)ccnc(O)c1F C1(C2CC2)(NC(C)CCCO)CCCCC1 CC(=O)CCCC(=O)N1CC(NC(C2CC2C2CC2)=O)CC(C)C1 c1(CNC(C(CC)O)=O)nc2c(s1)CN(C(=O)CCCC(C)=O)CC2 c1(C(N2CCC(NC(C(C#C)(C)C)=O)C2)=O)ccc(N)c(F)c1Br C(=O)(C(C(C1CC1)OC)N1CCC(CCc2ccccc2)CC1)NCC(=C)C c1(C(c2nnnn2CC2CCOCC2)NCNS(N)(=O)=O)cn(CC2CC2)nn1 C(=O)(CNC(C1(CC(N)=O)CC1)=O)NC(C1(SCCO)CC1)C c1(C(N2C(CNC(=O)CO)CCCC2)=O)ccc([N+](=O)[O-])cc1C(F)(F)F c1(C(C(=O)N(C)CCNC(c2ccnn2C(F)F)=O)O)ccccc1Cl c1(C(=O)NCCC2CCC(NC(C(Cn3ccc(C)n3)C)=O)C2)cn(C)nc1O C12(C(=O)NCCC(CCNC(CCC(C)C)=O)C)CCC(CC1)CC2 CN1C(=O)NCC1C(N1CCCC1CNC(=O)Cc1cnn(C)c1C(F)(F)F)=O C1(NC(C2CC(CN)OC2)=O)CN2CCC1C2 C1(C)(CNC(c2n(COC)ncc2)=O)CCCN1C(=O)COc1cccc(O)c1 c1(C(N2CCC(O)(CNC(c3ccc(C#C)cc3)=O)C2)=O)ccc(C#C)c(F)c1 N1(C(CCCC2CCN(C(c3c(CC)[nH]cc3)=O)CC2)=O)CC(C2CC2)C1C1CC1 C(C(CC(C)C)C(=O)NOCC(N1CC(OC)C1C1CC1)=O)OC c1(OC)c(C(=O)NCCCC(C)NC(C2CCCCC2)=O)oc2ccccc12 C(=O)(C(C)(C)CCCO)N1C(C)CN(C(c2cc(O)cc(O)c2)=O)CC1 N1(C(CC2(C)CC2)=O)CCN(C(=O)CN2CCCC2CO)CC1 N1(C(c2ccnc(Br)c2)=O)CC2(CCC(NCc3cnc(O)nc3O)C2)C1 N1(C(Cc2c(C)occ2)=O)CC(NC(C2(n3cccn3)CC2)=O)C(O)C1 C=CCC(C)C(=O)NC1CC(C(N2CC(C)(C#N)C2)=O)CC1O C#Cc1cccc(OCC(=O)NC2CN(C(=O)CCC(=C)C)C3CC23)c1 CC(CCc1ccccc1)CC(=O)NCC(O)C(=O)OC(C)(C)C CCCC(C(=O)N1CCCC1C1(NC(c2csc(CC)n2)=O)CC1)S(N)(=O)=O C(=O)(C(C)(C)C(C)(C)O)NCc1cn(CC(=O)NCC(C)(C)C)nn1 Cc1ncc(C(N2CCN(C(=O)CCCNC(c3ccco3)=O)CC2)=O)c(=N)[nH]1 C1(NC(C(C)(F)Cc2ccccc2)=O)COC2(CCN(C(=O)CNC=O)CC2)C1 N1(C(C2(OC)CCCC2)=O)CC(C)OC2(CCN(c3cncc(C#N)n3)C2)C1 C1(CC)CCCCC1(c1nnnn1C1(C)CC1)NCCCSC(F)(F)F C1(NC(C2(COCC)CC2)=O)CC2C1CCN2C(c1cccc(C(F)F)n1)=O C=CCC(C(=O)N(C(C)C(=O)NCC1CCCN1C)C)C(C)C C1(C(N(C)CCc2ccccc2)=O)CCC2(CC2)N1C(C1CC(C)(C)C1)=O c1(C(N(CCCN(C)C(c2ncn(C)n2)=O)C)=O)cc(Br)ccc1N c1(C(C(=O)NC(CCN(C(C=CCCC(C)C)=O)C)C)(F)F)cc(F)cc(F)c1 c1(C(N2CC(C(C(=O)N(CC(C)C(F)(F)F)C)OC)C2)=O)ccnc(C)c1N CN1CC(=O)NCC1C(=O)NNC(=O)c1ncon1 Cc1cc(C(N2CCCC(O)(CNC(C3CC(O)C3)=O)C2)=O)c2cnn(C)c2n1 c1(C(C)C)noc2ncc(C(N3CCC(C)C3CNC(=O)C3=CCCC3)=O)cc12 C(CCC(C)C(=O)NCCCC(C)(C)NC(C1CCCCC1(C)C)=O)OC Cc1nn(-c2ccc(F)cc2)cc1C(N1CC(CNC(=O)CO)C(C)C1)=O c1(C(=O)NC23CCN(C(Cc4c(C)scc4)=O)CC2C3)cnc2c(c1)CCC2 C(=O)(C(C)(F)F)N(C1CCN(C(C2CC(CF)C2)=O)C1)CCC CC1CC(N(C)C(c2cc(CNC(=O)Cc3ccn(C)c3)cs2)=O)CCO1 c1(C(=O)NC(C(C)NC(C2C(C)CCO2)=O)(C)C)ccc(S(C)(=O)=O)o1 N1(C(CSC)=O)CCCC(O)(CCNC(=O)CCC2(C)CC2)C1 N1(C(C=C(C)C(F)F)=O)CC2OCCN(C(=O)C(C)N3CC(C)C3)C2C1 C(=O)(C(C(C)(C)C)NC(c1ccc(C2CC2)o1)=O)N(CCCC#C)C N1(C(C(C)CF)=O)CCC2(CCC2CNC(c2ncccc2N)=O)CC1 C12(NC(CC)=O)CCN(C(c3cccc(OCc4nc[nH]n4)c3)=O)CCC1C2 N1(C(c2cc(OC)ncc2)=O)C2CCC(C2)C1C(=O)Nc1ccc(I)cc1 c1(NC(N2CCN(C(C)C(F)(F)F)CC2)=O)ccc(Cl)nc1P(C)(C)=O C1(C(=O)NC(CC=C)CC=C)CCC(C)(C)N(C(=O)C=CC)C1 c1(OCC(=O)NC2(CC(=O)NC3CC3)CCC2)ccccc1C(F)(F)F CC1(C)CN(C(C2COCCO2)=O)CC(CNC(c2ccc(C(F)F)cn2)=O)O1 N1(Cc2cnc(C)s2)CCC(NC(=O)Cc2cccc(C(F)(F)F)c2)CC1C C1(CNC(C2(C(F)F)CC(=C)C2)=O)CCCCN1C(=O)CCOCC(F)F N1(C(CC(C(C)C)NC(=O)CC2CCCN(C)C2)=O)CC2(CCC(C)OC2)C1 C1(CNC(c2cc(C(F)(F)F)cc(O)n2)=O)CC2(CCOC2)C1 c1(C(N(C2CCCC2)CCNC(C2CCS(=O)(=O)C2)=O)=O)cc(Cl)c(Cl)s1 c1(OC)ccc(C)cc1NC(=O)C(CC1CC1)NC(=O)CC=C(Cl)Cl c1(C(=O)NCCCCNC(C2C(OCC)C2)=O)cc(Cl)c(F)cc1OC N1(c2nc(N3CC(CCC)OCC3)nc(C)c2)CCOc2ccc(F)cc2C1 CCC(CC(C)C)C(=O)N(CCN(C)C(c1nnsc1C(=O)O)=O)CC.C(C)=O c1(C(=O)NC2(CO)CCN(C(C3CCCCS3)=O)CC2)cccc2nonc12 c1(C(=O)NC(CN(C(CCC(=O)OCC)=O)CC)CC)nn(CC)cc1[N+](=O)[O-] C#CCC(CC(F)F)C(=O)NC1CN(C(=O)CCCOC(C)C)C(C)(CC)C1 C1(NC(C(c2c(C)cccn2)(F)F)=O)C2CC(O)C1N(C(=O)CN(C)C(C)C)C2 C1(OC2(C(N(C)C)=O)CC2)CCOCC1.C12CC(C1)CNC(=O)CN(C)C2=O c1(C(=O)NCC(CC2CN(C(CCOCC)=O)C2)(C)C)cc2ccc(F)cc2s1 C1(c2n(CC(=C)C)nnn2)(NCCOCCCO)CCC(P(C)(C)=O)C1 c1(C(=O)NCC(CNC(c2n(CC)ncc2)=O)C)c(C)cccc1[N+](=O)[O-] N1(C(C(C)(C)OC(C)C)=O)CC2ON=C(CNC(c3ccc(F)c(F)c3)=O)C2C1 N1(C(c2snc(CC)n2)=O)CCC(C)C(C(F)(F)F)C1 c1(C(=O)NC(CC(C)NC(CC2(COC)CC2)=O)C)c(C)cc(Cl)cc1C CC(C)CC(C)(C)C(=O)NC(C)CCN(C)C(c1conc1C1CC1)=O Cc1ccc(CC(=O)NC2CN(C(=O)Cc3cc(F)ccc3Cl)CC2O)c(C)c1 c1(C(=O)NC(C)CNC(=O)CC2CSC2)c(O)nc(=O)n2c1CCC2 C1(CNC(c2c(CC=C)cccc2)=O)CC2(CC2)CN1C(=O)CNS(=O)(=O)CC CC(C)CC(C)CC(=O)NC(C)(C)CN(C)C(c1cnc(C(C)(C)C)[nH]1)=O C(=O)(CC(CC)C(C)C)NC(C(C)(C)NC(c1c(CC=C)cccc1)=O)C N1(C(CCSCC)=O)CCOCC1CCNC(C1CCCN1C(C)=O)=O c1(C(=O)NC(c2nc(C(C)C)sc2)C)cc(C(F)(F)F)c(F)cc1N C1(N(CC#C)C(C2CC2=C)=O)CCN(C(C2CCC(=O)C2)=O)CC1 c1(OC)cc(F)c(NC(C2CCCN(C(c3cccs3)=O)C2)=O)cn1 C1(S(N)(=O)=O)(C(N(CCOCCNC(C(C(C)C)OCC)=O)C)=O)CCCC1 C1(NC(c2cnc(C)o2)=O)CN(C(=O)C(c2c(C)n[nH]c2C)C)C2(CCCC2)C1 CC(C)(F)CCC(=O)NCC1CC1CNC(c1cccnc1S)=O c1(C(=O)NC(CC)CNC(=O)CCN2CCCC2)cc2cc([N+](=O)[O-])ccc2[nH]1 N1(C(=O)CC2CCOC2)CC2CC(C1)N2C(=O)CC1CC(C2CC2)C1 c1(C(=O)NC)[nH]c(C)c(C(=O)NC(C)C(C)C(=O)Oc2ccccc2)c1C Cc1nn(C)c(C)c1NC(=O)NCc1ccc(-n2ncnc2C)cc1 C1(F)(CNC(=O)C(O)C2CC2)CCC(CNC(C2(O)CC2)=O)CC1 C1(C(=O)N)CC(=O)OC1(C)C.C(=O)(C(C1(O)CCC1)CC(C)(C)C1CC1)NCC c1(C(N2CC3(C(NC(C(F)OC)=O)CCS3)C2)=O)cc(F)cc2cnccc12 C1(CNC(C=C2CCC(C)CC2)=O)CC(C)CN(C(=O)CCc2cscn2)C1 C12(NC(COCC(=O)NC)=O)CCN(C(c3cc(COC)[nH]n3)=O)CC1C2 c1(C(c2nnnn2CC2CC2)NCC(CCC=C)(C)C)cn2cc(Br)ccc2n1 C1(C(=O)NCCN(OC)C)CCN(C(C2CC2C2CCC2)=O)CCO1 C1(NC(C2OCC(C)C2)=O)CC(=O)N(C2CN(C(=O)CCNS(C)(=O)=O)C2)C1 c1(SCC(=O)NCCN(C(c2coc(Br)c2)=O)CC)ccc(F)c(F)c1 C(=O)(CCCCC(=O)NC1CCCCC1C(N1CCC(C(C)(C)C)CC1)=O)OC Cc1ccc(C(=O)C(=O)NC2(CO)CN(C(=O)C(C)(C)c3ccc(Cl)s3)C2)cc1 Cc1c(NC(=O)Cc2ccccc2NC(c2n[nH]cc2I)=O)ccc(C#N)c1Cl N1(C(c2c(CC)c[nH]c2)=O)CCC(CNC(c2ccnc(S)c2)=O)(OC)CC1 NS(=O)(=O)C(C(=O)N1CCC(F)(CNC(=O)C=C2CCC2)C1)c1ccccc1 n1(CCC(=O)NCC2(NC(C=CCC)=O)CC(OC)C2)cc(Br)c(C)n1 CC1(C)COC(C(=O)NCC2(NC(=O)CC3CCCCCO3)CCCC2)C1 c1(CC)nc(=N)[nH]cc1C(N1CC(NC(C2(C)CC(F)(F)C2)=O)C2CC12)=O c1(COC)nn(C)cc1C(=O)NC(C1CCN(C(=O)CC2CCOC2)CC1)C S(=O)(=O)(c1ccc(=NCCC2(CO)CC2)[nH]c1)N1C(c2n(C)ncc2)CCC1 C1(NC(C)=O)CCN(C(=NC2CCS(=O)(=O)C2)NC2C(C)C2C)C1 C1(C(=O)NCCN2CCOCC2=O)CCC2(CC2)N1C(C1CC1c1ccco1)=O c1(CN2C(=O)C2)c(F)cccc1Cl.C1(CC(=O)OCC)CCCC(F)(F)C1 c1(-c2ncc(C(=O)NC3C(NC(CC(CC)C)=O)C3)s2)c(F)cccc1F C1(F)(C(=O)NC(CNC(C(C(C)C)N(CC)CC)=O)CC)C(C)(C)C1(C)C Cc1cccc2c(C(N3CCN(C(c4c[nH]c(C#N)c4)=O)C(C)C3)=O)coc12 c1(C(=O)NC2CCCN(C(C(CC)n3nccc3C)=O)C2)cc(C#N)ccc1F C1(CNC(Cc2ncc(CC)[nH]2)=O)CCN(C(C2(C)CCCC2C)=O)C1(C)C CN(C(=NCCF)NCC12CCC(CC1)C2(C)C)CC1CNC(=O)O1 C1(CNC(=O)N(C2CCC2)CC2N(C(C)=O)CC2)CCC(C(=O)O)N(C)C1 c1(C(=O)NC(CC)C)ccc(NC(=O)NCC2ON=C(C)C2C)cc1Cl c1(CCC)[nH]nc(C(=O)NCC(C(C)(C)C)NC(C2CC2(C)C)=O)c1[N+](=O)[O-] c1(OC)cc2c(cc1C(N1CC3CCC1C(O)C3)C(=O)NC(C)C)OC(C)C2 CC1CCC(C)(C(N2CCC(NC(=O)C#CC(=O)N(C)C)C(F)C2)=O)C1(C)C N1(C(c2c(C)onc2)=O)CC(NC(=O)C(O)C2CCCC2)C2CCCC12 N1(C(C=CC(C)(C)SC)=O)CCCCC1CC(C)O.C12(CC1)CC(=O)NC2 C(CCNC(=O)CNC(C1CCCC1)=O)(C(C)C)NC(C1(C(F)F)CC(=C)C1)=O N1(C(C2CC(C)(C)OCC2)=O)CCC(C2CC2)C1CNC(=O)CCn1cnnn1 N1(C(C(CC)C(C)C)=O)CCc2nc(CNC(=O)C(C)CC(C)O)sc2C1 C(C(C)(C)C(=O)NC1CN(C(C2CCS2(=O)=O)=O)C1)OC C=C(Cl)CCC(=O)N1CCOCC1CNC(=O)CCC1CC1(F)F N1(c2cc(C)ncn2)CCC(NC(c2csc(C3CCCO3)n2)=O)C(O)C1 CCC(CC(=O)NC1(C(=O)NCC2CC(F)(F)C2)CC(O)C1)C(C)C CC(C(=O)N1CCNC(=O)C1)(C(F)(F)F)N(C)C(c1cc2ccc(Br)cc2[nH]1)=O C1(C)(CC(=O)NC2C(CCOC)CCC2)CCN(C(=O)CNC(=O)C2CC2)CC1 c1(C(=O)NCCOC2CN(C(C(C)(C)CF)=O)C2)ccc2c(c1)OCC2 Cc1cc(C2CC2)ccc1C(=O)NCC(C)NC(=O)C(C)Cc1c(C)noc1C C(=O)(N=c1[nH]nc(Cl)c2c1CCC2)Oc1c(C=CC=CC#N)ccc(OC)c1 C1(NC(c2cn(C(C)C)nn2)=O)C=CCN(C(=O)C(c2ncccc2F)(F)F)C1 C(N=c1nc2sccc2c(N2CCOCC(C)(F)C2)[nH]1)c1nn(C)nc1Br N1(C(C2CC(C)(O)C2)=O)CCN(C(c2ccc(O)nc2Cl)=O)C(CC2CC2)C1 N1(C(=O)Nc2ccc3ncccc3c2Cl)CCCCC12CCS(=O)(=O)CC2 c1(CN2C(C(=O)OCC)CC(F)C2)cnc2n1CCCCC2 C(=O)(C1=CCCN(C(=O)CC2COC3(CCC3)CO2)C1)OC C(=O)(C1CCc2nccn21)N1C(CN(C(c2c(CC)nc(C)nc2)=O)C)CCC1 C(CC(C)C(=O)NCC1(C(=O)NC(Cc2ccco2)CO)CCCC1)=CCC N1(C(C(C2CCCOC2)OC)=O)CCC12CN(C(c1cc3c(s1)CCC3)=O)C2 C12(C(N3CC(N(C)C(c4ccc(Cl)s4)=O)C3)=O)CCCC(CCC1)C2O C(=O)(C(C)CCCC(C)C)NC1CCN(C(c2cc(C)sn2)=O)CC1 Cc1ncc(Cl)c(C(=O)NC2CCCCC2NC(=O)C(C#N)C2CC2)n1 N1(C(C(CCCC)O)=O)CC2CCCN(C(=O)Cc3nocc3C)C2C1 c1(C(=O)NCC2(O)CN(C(C(C)c3ccco3)=O)C2)cncn(C)c1=O C=CC1CN(C(=O)C(C)(C2CC2)N(C(=O)CNC(C2CC2C)=O)C)C1 N1(C(C2(C=C)CCCC2)=O)CCOC2(C1)CN(C(c1c[nH]c(=N)c(C)c1)=O)C2 c1(C(N2C(C)C(C(=O)NCc3nn[nH]n3)CCC2)=O)cccc2[nH]ncc12 N1(C(C(C(C)O)C)=O)CCN(C(c2ccccc2C(F)F)=O)CC12CCC2 CC(C)C(=O)C(=O)NCC1CC1C(=O)NC(CO)CCF N1(C(c2cn(C)nc2)=O)CCC2(CC1)CC2C(=O)NCC(c1ccccc1)F c1(NC(C(c2occ(C)c2)N(C)Cc2n[nH]c(C)n2)=O)cccc([N+](=O)[O-])c1 CC1(C)CC=C(C(=O)N2CC3CC(C2)CN(C(=O)CC(O)C2CCCC2)C3)CC1 c1(C(=O)NC2C(CNC(C3N(CC)CC3)=O)C2)ccc(C)c(Br)c1C C1(NC(C2C(NC(C3C(C)(C)OC(=O)C3)=O)CC=CC2)=O)Cc2ccccc2C1 c1(NC(C2N(Cc3c(OC)c(Cl)ccc3)CC2)=O)ccc2cn(C)nc2c1 C(=O)(C(C)(C)CCCNC(=O)CSc1nc[nH]n1)NCC1CCN(C(C)=O)C1 c1(C(=O)NCC2CCC2C(N(C2CCS(=O)(=O)C2)C)=O)ccc(N)cn1 NCCCC(O)C(=O)N1CCC(n2cc(-c3cn[nH]c3)nn2)CC1 c1(OCOC)cccc(C(=O)NC(CNC(=O)C(C)N(C)C)C(C)C)c1 N1(C(c2ccc(C(=O)OC)[nH]2)=O)CC(CNC(C2(Cl)CC2(C)C)=O)C(O)C1 C1(CC#C)(C(=O)NCC(F)CNC(c2cnn(C)c2OC)=O)CCOCC1 C1(C(=O)NC(CN(C(c2nc(CC)sc2)=O)CC)C)CCCOC1CC(C)C c1(C(=O)OCC(C(CC)(C)C)=O)cc(Br)cc(S(C)(=O)=O)c1F C1(CNC(C(C)C2CC2)=O)CCCN(C(c2ccn(-c3ccncc3)n2)=O)C1 c1(OCC)cncc(C(=O)NC2CCN(C(=O)CC3(OC)CCCC3)C2)c1 c1(OC)cc(OC(C)C)ccc1N(C1CC2CCC(C1)N2)C(c1cc(C)[nH]n1)=O Cc1ccnc(CNC(=O)CC2CCN(Cc3ccc(C(F)F)cn3)C2)c1 C1(CNC(C2(C(C)C)CCN(C(CC(=C=C)C)=O)C2)=O)NC(=O)CC1(C)C c1(C(N2C(CNC(CC3C(C)C3)=O)CCCC2)=O)cc2cc(N)ccc2[nH]1 c1(NC(CC(C)NC(C2CC23CCOCC3)=O)=O)c(O)cccc1F Cc1nn(C(C)C)cc1C(=O)N(C1CN(C(=O)Cc2cncnc2)CC1F)C c1(C(=O)NC(C(C)NC(c2c(C)nc[nH]2)=O)C)cccc(Cn2cncn2)c1 CCCC(CCC)C(=O)NCC1CC(C)(C)CN1C(C1CCC1c1nc[nH]n1)=O c1(OC)cc(C)ccc1C(N1CCC(O)C(NC(C2(CN(C)C)CC2)=O)C1)=O c1(C(=O)NC2CN(C(c3cc(C)nn3C)=O)CC2O)ccc(C(F)(F)F)cc1C C1(CC(=O)N(CCCNC(=O)Cc2ccn(CC(F)(F)F)n2)C)CCC2(CC1)CC2 C1(NCCNC(N(C)CCN2CCCCC2)=O)CCN(C2CCCCC2)CC1 c1(OC(C)C(=O)NCCNC(c2[nH]nnc2C2CC2)=O)ccccc1C(F)(F)F Cn1ccc(C(=O)NCC2CN(C(=O)COCCF)C(C)(C)C2)cc1=O C(=O)(C(CCCC)C(C)C)N(CCC(=O)N(C)CC1OCCC1(C)C)CC=C CC(C)(C)CC(O)CC(=O)NCC1CCCN1C(=O)CSCC1CCCCO1 N1(C(N)=O)CCC(C(=O)NCC=CCNC(c2ccc(CO)o2)=O)CC1 C1(CNC(C(CC)N(C)C)=O)CN(C(=O)COCP(C)(C)=O)C(C)(C)C1 C1(NC(c2cc(C)[nH]n2)=O)CC2CC1N(C(c1cnc(C(F)F)s1)=O)C2 c1(-c2cn(C3C(N4CCC(OC)C4)CCC3)nn2)cc2occc2s1 CC(C)CCCC(=O)N(C1CCCN(C(c2cocn2)=O)C1)CCF c1(C(N2CC(C)CC(NC(CC(C)F)=O)C2)=O)cc(F)c(Cl)cc1Cl c1(OC)ccc(C(=O)NCC2CC(C(=O)N)OC2)s1.C1CO1.C1CO1.C1CO1.OC c1(OCC(=O)NCC2C(CNC(=O)CCCCCF)C2)ccc(Cl)c([N+](=O)[O-])c1 C1(CNC(c2cscn2)=O)COCCN(c2nc(Cl)ncc2Br)C1 C(=O)(C(F)C(C)(C)O)NC(c1ccccc1)C(N1CC(N(C)C)(C(N)=O)C1)=O C1(N(C)C)CCCN(CCC(=O)NCC(C)(C)CNC(=O)CC2(C(F)F)CC2)C1 N1(C(=O)COCC2CCCC2)CCC(O)(Cn2cc(-c3ccccc3Cl)nn2)C1 N1(C(CSCC=C)=O)CCOC(CNC(c2ccoc2CCC)=O)C1 Cc1cncc(CC(=O)NCCNC(=O)CCOc2ccccc2)c1 C1(C(N2CCC(CC3CC3)CC2)=O)CC2(CCN(C(C3CC(CF)C3)=O)C2)C1 c1(-n2cc(CCC#N)nn2)ccc(C(=O)NCC2CCOC2)cc1 N1(C(=O)Cc2ccccc2)CCN(C(C2CS(=O)C2)=O)CC1c1cn[nH]c1 C12(CNc3ncccc3C3CC3)CC1CN(OCC)C2 c1(C(=O)NC2CN(C(c3c(C)snc3)=O)CC2F)cnc2ccccc2c1 Cc1ocnc1C(c1nnnn1CC1CCCO1)NCc1csc(Br)c1 N1(c2cc(OCC)ncn2)CCC(NC(C2CCCN(C(N)=O)C2)=O)C(O)C1 C1(C(=O)NCC(CN(C)C(c2nnn(-c3ccccc3)n2)=O)O)COCC1(C)C CCCCC(C)C(=O)N1CC(OC2CCN(C(c3n[nH]cc3Cl)=O)CC2)C1 c1(CC)ccc2cc(C(N3CCC4(CCC4NC(=O)CC(F)F)CC3)=O)[nH]c2c1 c1(CNC(C2CCC(C)O2)=O)ccc(C(C)NC(=O)C(Cl)=CCl)cc1 Cn1c(C(N2CC(OCC(=O)NC(C(N)=O)C3CC3)C2)=O)cccc1=O N1(C(CN(S(C)(=O)=O)C)=O)CC2(CC(NC(C3CCC(CC4CC4)O3)=O)CO2)C1 c1(OC)ccc(C(C(=O)O)NC(C2CCO2)=O)cc1 Cc1ccc(OCCC(=O)NC(C)C(CO)NC(c2cccs2)=O)c(C)c1 C1(C(=O)NCC2(CC)CC2)(CO)CCN(C(c2cn(CC)cn2)=O)C1 CCCC(C(=O)N(C)CC1CN(C(=O)CC(O)CC)CCO1)C(C)C CCC(C(=O)NCCC1(CNC(=O)C(O)CC)CC1)n1ccnc1CNC(C)C c1(OC(C(=O)NC2C(NC(CC=CC)=O)CCC2)C)ccc(OC(C)=O)cc1 C(CCC(C)CC(=O)N1CCC(N(C)C(c2n[nH]c(C)c2Cl)=O)CC1)=C(C)C CCC(C(=O)NC1(C(N2CC3(C)COCC3(C)C2)=O)CSC1)C(C)(C)CC N1(C(c2cc(C)n(C)c2C)=O)CC2(CCC2)CC1C(=O)NCCC(O)C(F)F c1(C(N2C(CCCNC(CN(C)CC)=O)CCC2)=O)ccc2c(c1)NC(=O)C2=O C1(NC(CCN(C(=O)COCc2nc[nH]n2)CC=C)=O)CCCN(CC)C1 N1(C(C)=O)CCCC2(NC(=O)Cc3cccc4c(C)csc34)CCCC12 c1(C(N(CCN(C)C(c2csc(Cl)c2)=O)C)=O)cc(O)c2sccc2c1 CC1(C)CC(CC(N2CCOC3CC23)=O)N(C(=O)C(CO)NC(N)=O)C1 C1(c2n(CC=C)nnn2)(NC(C)Cc2cccs2)CC2(CCC(C)(C)CC2)C1 Cc1cc(C#N)cnc1C(N1CCC2CC12C(N1CC(O)(c2cnn[nH]2)C1)=O)=O c1(C(=O)NCC2(F)CCCN(C(C3C(C#N)C3)=O)C2)ncn2c1CCCC2 N1(C(CC(C(C)C)O)=O)CC(CNC(=O)Cc2nncn2C)OC(C)(C)C1 c1(CN2CCC(O)(CO)CC2)cc(Cl)c(F)cc1F.N#CC1CC(N2CC2=O)C1 c1(OC)cc(C)c(S(=O)(=O)NC2(C(=O)O)CCOC2)c(C)c1 c1(C(=O)NCC(CC)NC(c2nn[nH]c2C(F)(F)F)=O)c[nH]c(=NC)s1 n1(CCCOC)c(N(C2CC(C(F)(F)F)C2)C)nnc1C1CCCS1 C(C)(C(=O)NC1CC(NC(C2(C(=O)N(C)C)CC2)=O)C1)(C(C)C)OC c1(CNC(CCCCC#N)=O)cc(Cl)cc2c1OCC2.C12C3CCC(C3)N1C2=O Cc1cccc(F)c1CC(=O)N(CCCCCCNC(C1CC(C)OC1=O)=O)C C1(NC(C=Cc2cnc(C)s2)=O)CC2CC(NC(c3cc(C(C)C)[nH]n3)=O)C1C2 CC1(C)CCC(CNC(C2CC2CNC(C2CSC2)=O)=O)OC1 C1(NC(COc2ccc(C)cc2Br)=O)CN(C(=O)CNC=O)CCC12CCC2 n1(CC(=O)NCC2CCCN(C(C(CC)C#N)=O)C2)cc2ccccc2n1 c1(C(=O)Oc2ccc(CON)cc2)c(F)ccnc1Cl c1(C(C)C)cc(C(=O)NCCOCCCN(C(=O)Cc2cncn2C)C)n(C)n1 CC1(C)C(C(=O)NCC(C2CCC2)NC(c2ccnc(OC3CC3)c2)=O)C1(C)C C1(C(N(CCC)Cc2n[nH]c(CC)n2)=O)CCN(C(=O)C(C)CC)CC1 C#Cc1cncc(C(=O)N(C2(C(N3CCN(C)C(CC)C3)=O)CCC2)C2CC2)c1 c1(C(=O)NCC(C)N(C(=O)C(F)C2CC2)C)cc(F)cc2ccoc12 N1(C(CC(CC)C2CCC2)=O)CC(C)C(C)(C(=O)NCC2CC23CCOCC3)C1 C=CC(F)(F)C(=O)N1CC(O)(CCNC(c2ncccc2C2CC2)=O)C1 C=CCC(CC(C)C)C(=O)NCCC1(C(=O)NCC2(CSC)CCCCC2)CC1 CC(C)(C)C(CNC(c1ccsc1C#N)=O)C(=O)NCC1C=CCOC1 C#CCC(C(=O)NC(CO)C(C)CC)NC(=O)CSC(C)(C)C C1(F)(C(=O)NCC2N(C(=O)CCn3ccnn3)CCC2)CC2(CCC2)C1 C(N=C(NC1CCCCC1)N1CCN(C(C)(C)COC)CC1)c1n(CC)ncn1 C#CCC(C(=O)N1CCC(CC)(CC)C1)NC(c1cc(C(C)C)[nH]n1)=O c1(C(=O)NCC2CN(C(C3C(C(C)(F)F)C3)=O)CC2(C)C)coc2cc(O)ccc12 C1(C(CNC(C(C)C2CCC2)=O)(C)C)CCN(C(=O)Cn2nnc(=O)[nH]2)CC1 N1(C(CC2(CSC)CC2)=O)CCC(CO)C(NC(c2oncc2C)=O)C1 c1(CCCC)cn(C2CC3(C(N4CC(COC)C4)=O)CC23)nn1 C=CCC(CC(C)C)C(=O)N1CCC(N(C(=O)CCC2CCCC2)CCO)C1 c1(NC(C)=O)cnc(C)c(C(N2CC(CNC(c3ccn(C)n3)=O)C2)=O)c1 C1(NC(C2CCC(CC)CC2)=O)CN(C(c2cc(N)cc(N)c2)=O)CC1(C)C C1(NC(CC(C)NC(N)=O)=O)CC(=O)N(C2CN(C(=O)Cn3ncnn3)C2)C1 C1(NC(=O)Cc2cnccn2)CCC(O)CN(C(=O)CC2CCCCCCC2)C1 C(=O)(C(C)(C)CCCNC(c1c[nH]c(=N)o1)=O)Nc1cn(CC)nc1 CC(C)C(F)(CNC(C1CC(F)(CF)C1)=O)C(=O)NC12CCN(CC1)C2 c1(CSc2n(CCC)c(Cc3cc(O)nc(S)n3)nn2)ccc(C)c(Br)c1O CCCC(CCCNC(=O)CCCc1nncn1C)NC(C1(CO)CC1)=O N1(C(c2nn(C)c(Br)c2)=O)CC(C2CN(C(=O)Cc3cccs3)C2)C1 C(=O)(CCCC(N)=O)N1C(OCCn2cc(C(C)=O)nn2)C=CC1 C(=O)(N1CCCc2ccnn21)C1C(NC(c2ncn3ccccc23)=O)C1 CCCC(CC)C(=O)NC(CNC(c1c(F)cccc1Cl)=O)C1CC1 c1(C(N2CC3CCN(C(CCCN(C)C)=O)C3C2)=O)ccc2c(=N)[nH][nH]c2c1 c1(C(N2CCC(CNC(c3c(C(C)(C)C)ocn3)=O)C2)=O)cnn2ccncc12 C(=O)(C(C)CS(C)(=O)=O)NCC(CCCC)NC(=O)C(CC)CC C1(CCN(C(=O)CSc2ccncc2)C)CCCCN1C(C1CCCNC1=O)=O N1(C(C2CCC(NC(Cc3ccn(C)n3)=O)C2)=O)CCN(CC(F)(F)F)CC1 c1(N(C(C)(C)C2CC2)C)ccc(S(=O)(=O)N2CCS(=O)(=O)C(C)(C)C2)cn1 N1(C(C2(C#C)CCC2)=O)CC=CC(NC(C2CC(=O)N(Cc3ccco3)C2)=O)C1 C1(C(=O)NCCc2cccc(COC)c2)CCC(=O)N(CC(F)(F)F)C1 Cc1ccc(C(=O)NC(CCF)C(=O)NC23CCN(CC2)CC3)nc1C O=C(C#CC1CCC1)NC(C1CCOC1)CNC(=O)C(c1ccc(Cl)cc1)(F)F C1(C(N2CC(NC(=O)COCc3ccnc(O)c3)C(O)C2)=O)(CC)CCCCC1 N1(CC(=O)Nc2cccc(C(C)=O)c2)CCC2C(F)(F)C2(c2ccccc2)C1 Cc1ccc(C(N)=O)cc1C(=O)NC1CCC(NC(=O)C(=Cc2c[nH]cn2)F)C1 N1(C(C(c2cccc(O)c2)C)=O)CCCCC(NC(C2CC3CCC2O3)=O)C1 C1(C(=O)NC(C(C)OC)C(N2CCCC(C#N)C2)=O)CN(C)CCN1C c1(C(C2CCN(C(C)(C)C)C2)C)cccc(C#N)c1.c12cn(nn1)C1CN(C1)C2 c1(NCCN2C(CC)COCC2)[nH]c(=NC2CCCCC2F)nc2sccc12 C1(C(=O)NCCCC(=O)NCCSCC)CCOC(C)C1 C1(CN(C(=O)CN2CCCCC2)C)CCCN(C(C2CCC(=O)NC2)=O)C1 C1(C(C)C)(C(=O)NC(C)C(C)F)CCCN1C(C1CC1C1CC1)=O c1(C(c2cn(CC(C)NC(c3ccc(CC)s3)=O)nn2)(C)O)ccc(F)cc1 C1(NC(CC(=C=C)C)=O)CN(C(=O)CN2CCOCC2)C(C)(CC)C1 N1(C(C2(C=C)CCOCC2)=O)CC(CNC(=O)CC(C)(C)C#N)C2(CCC2)C1 c1(C(=O)NCC(C)N(C(c2ccc(OC)o2)=O)C)cnc(O)n1C N1(C(C(C#C)(C)C)=O)CCC(C)C(NC(=O)CC2OCCCC2(C)C)C1 N1(C(C(=O)NC2C3(CN(C(C)=O)C3)CCC2)=O)CCC2(CC1)CNC(=O)O2 C1(CCCC)CCC(C(=O)N(CCCN(C(=O)C(C2CCC2)OC)C)C)CC1 C1(NC(CCc2nnc(C)n2C)=O)CCCC(NC(C2CC(C)(C)C2)=O)CC1 c1(C(=O)NCCN(C(=O)CCCCO)CCOC)nc(Cl)ccc1F N1(C(COCCC)=O)CC2(CCC(NC(c3c(Cl)cc(Cl)cc3Cl)=O)CC2)C1 C1(NC(=O)CN2CCCCCC2)CC1C1CCN(C(=O)C(F)OC(F)(F)F)CC1 c1(CC(=O)NCC2C(NC(CNC(C(CC)CC)=O)=O)C2)c(O)ncnc1O C=C(C)CCC(C)NC(c1cc(CNC(=O)C(C)n2cccc2)[nH]n1)=O c1(CC(=O)NCc2cn(CCCC)nc2C)ccc(Cl)c2cccnc12 C1(CNC(c2c(CC)scn2)=O)CC(C)N(C(=O)C(O)C2CCCC2)C1 Cc1cc(Sc2cnn(C)c2C(F)(F)F)c(C(F)(F)F)cc1[N+](=O)[O-] N1(C(C23CC(C)C2C3)=O)CC2(CCCN(C(c3n[nH]c4cccnc34)=O)C2)C1 C1(CNC(=O)CC2CCOCC2)CC2(CCCC2)CO1.C12CCN(CC1F)C2=O C1(C(=O)NCCOCC(C)(C)O)CCCCC1(C)NC(C1CCOC1C1CC1)=O N1(C2CN(C(=O)NCC3=CCCC3)C2)CCCS1(=O)=O C1(C(=O)OCC)CCC2(CCCN2C(c2ccc(CNC(=O)OCC)o2)=O)CC1 C1(CN(C)C(c2ccoc2Br)=O)CCCC(NC(c2cncnc2)=O)C1 CC1(F)CCCCN(C(C2CC(F)(F)CN2Cc2ncc[nH]2)=O)C1 Cc1noc(C)c1C=CC(=O)N(C)CCOCCCN(C(=O)CC1CC12CC2)C c1(CC)ccc(C(=O)NCC2CC2CNC(C2(CC)CC2(F)F)=O)o1 C=C=CC(C)C(=O)NCCCCN(C)C(c1nccc(-c2sc(C)nc2C)n1)=O C1(CC(=O)NC2(CNC(C3CC4CC4C3)=O)CCCC2)CCCCO1 c1(CNC(COC)CC2CCOCC2)nc(C)cn1C N1(C(c2c(C)c(F)cnc2)=O)CCC2CN(C(=O)CCc3cnoc3)C2C1 c1(OCC)cnc(C(N2CCC(C(C)NC(c3ncc(Cl)n3C)=O)CC2)=O)cn1 C#CCC(O)C(=O)NCC1CCCN1C(c1c(C2CCOCC2)noc1CC)=O N1(C(C2CCC(n3cc(CCCC(C)O)nn3)C2)=O)CCC(C#N)CC1 c1(NCC2(COC)CCC2)[nH]c(=NCC2(S(C)(=O)=O)CCCC2)nc2scnc12 c1(OC)nccc(C(=O)NC2CC(NCc3c(F)cccc3F)C2)c1F C1(n2cc(CN(C)C(=O)OC(C)(C)C)nn2)CN(C(=O)Cn2ncc(Br)n2)CC1O C(CC(CC)C(=O)N1CCC(CC(=O)NCCCC(C)CO)C1)=CC N1(C(CC)CC)CC(C(N2CC(C(C)NC(=O)COCCCOC)C2)=O)CC1=O CC(C)CCCC(=O)N1CC(CNC(=O)C(C)C2CCCO2)CC1C CCCCCCC(CC)NC(C1CC(C)CN(C(=O)Cc2cc(C)cs2)C1)=O c1(C(N2CCCN(C(C(c3ccn(C)n3)(C)C)=O)CC2)=O)ccn2c1CCCC2 n1(CCCOC)c(N2CCCC(c3nc(C)no3)C2)nnc1C1CCCCN1C N1(C(c2cccc(C)c2F)=O)C2CCC1CC(N(C)C(C1CC3CC1C3)=O)C2 CCC(CCC(=O)NC1CCN(C(=O)CCSc2nnnn2C)CC1O)OC C(C(C)(C)CNC(=O)C(C1CCN(C(c2cnn(C(C)C)c2)=O)C1)C)OC C(C)(CSC)(C(=O)N=c1cc(C)n(C)[nH]1)NC(C(C(CC)O)C)=O C1(C(C)C)CCC(C(N2CC(c3nncn3C)C2)=O)N1C(=O)COc1ccsn1 Cc1cnnc(C(=O)NC2(CF)CCN(C(=O)CCOCC3CC3)C2)c1 Cn1nc(CC(N2CC(NC(=O)C(C)(O)C3CCOC3)C2)=O)cc1C(F)(F)F N1(C(CC(C)(F)F)=O)CCC2(C)CN(C(=O)CC3CC3(Cl)Cl)CC12 N1(CCCCCNC(COCCCCCC)=O)CCCC(C(N)=O)C1 n1(CC)c(C)nn(CC(=O)N(CC(C)NC(C2(C)COC2)=O)C)c1=O C(CCN(CC(C)C)N1CCC2(CCCN2C)C1C)OC c1(COC)cccnc1C(N1CCC(N(C)C(c2ccnc(O)c2)=O)CC1)=O N1(C(C2CN(C)C(=O)N2)=O)CC2CCCC(NC(=O)CCC3CC3(Cl)Cl)C2C1 C1(NC(=O)C2=COCCC2)CC2(CCN(C(=O)Cc3ccc(Br)cc3Cl)C2)C1 N#Cc1ccc(CNCC23CC2CN(C(=O)C=Cc2ccc(O)cc2)C3)nc1 Cc1cc(-n2cc(-c3cnn(C)c3CNC(c3ccc(F)s3)=O)nn2)cc(F)c1 c1(C(=O)NC(CCCCNC(CC2(OC)CCCC2)=O)C)ccc(F)cc1Cl N1(C(CCC(=C)Cl)=O)CCCCC2(CCN(C(=O)C(C)COC(C)=O)C2)C1 S(=O)(=O)(c1ccc(SCCOc2ccc(NCC)cc2)c(Cl)c1)N(CC#N)CSC c1(C(=O)NC2CCCN(c3nc(C#N)cc(C)n3)C2)cccc2ccncc12 c1(C(N2CCCC2C(=O)NC(C(C)(C)CO)c2nccn2C)C)cccnc1F CC(N=c1ccnc(NCc2cccc(N3CCCC3=O)c2)[nH]1)C1CCCCO1 c1(OC)ccc(C(N2CC3C(NC(c4ccn(C)n4)=O)C3C2)=O)nc1 C1(NC(c2cc(CC)ncc2)=O)C2CCN(C(=O)Cn3ccnc3C)CC12 C1(C(=O)NCCC(=O)N2CCCC2)CCCC1(C)NC(C(C)C)=O Cc1cc(C(N2CCN(C(c3n[nH]c4c3COC4)=O)C3CC23)=O)n2ncnc2n1 C1(N(C(=O)CCSC2CCC2)C(C)C)CCCCCC1 Cc1[nH]nc(C(=O)NC2(C)CCN(C(=O)CCC3CCCN3C)C2)c1Cl Cn1ncc(C(=O)NCCCCC2CN(C(c3cnc(C(F)F)s3)=O)C2)n1 N1(c2ccnc(NC3C(COC)OCC3)n2)CCOCC(OC2CC2)C1 CC1CN(C(C2(F)CCCOC2)=O)CC1NC(c1nccn1C)=O N1(C(C=C(CC)C)=O)CCC(NC(c2cc3nnn(C)c3s2)=O)C(CO)CC1 C1(C(N2C(C(=O)OC)C=CCC2)=O)CN(C(c2nn(C)cc2C)=O)CC1(F)F C(C(F)(F)C(=O)NCC(C)(C1CC1)NC(C1CC(C)CCO1)=O)OC Nc1cccc(CCC(N2CCCC2CNC(C2CC3CC2C3)=O)=O)c1 C1(NC(C(CC)N(C)C)=O)CCN(c2nc(C(=O)OC)cc(C)n2)CCC1CO N1(C(C2CCC(C)(C)C2)=O)CC(NC(c2ccc(CC3CC3)s2)=O)C2(CC2)C1 C(C(C)(C)C(=O)NCC1CC(C)N(C(=O)CCc2ncc(F)cn2)C1)OC c1(C(=O)NC(c2ccnn2C)C(=O)NC(C)C(C)(C)CO)cccn2cncc12 C1(NC(C(CC)C)=O)(CC)CCN(C(C2CC(NS(C)(=O)=O)C2)=O)CC1 N1(C(CC2N(C)CCCC2)=O)CCc2c(c(CNC(=O)CC3CSC3)nn2C)C1 C(=O)(CC(C(F)F)NC(=O)CN1CCN(C)CC1)N(C1C(C)CC1)C C1(C(C)(C)C)C(NC(C2CCC(=O)NC2)=O)CCN1C(=O)CNc1nccs1 C(=O)(CCCCCNC(C)=O)NCCC1CN(C(C=COC)=O)CC1C N1(C(CCC=C)=O)CC(C2(Nc3nc(C(F)(F)F)ns3)CC2)C1 c1cnc(Br)o1.C1(C(=O)NC)CCCO1.C12CC(C1)CCOCC(=O)N2 Cc1ncccc1C=CC(N1CCC1CNC(=O)CC(O)C1CC1)=O C(=O)(CC(C)(O)CCC)NCc1c(CNC(CN(CCC#C)C)=O)cccn1 CN=S(C)(=O)c1ccc(C(=O)N(C(C)CN(C(=O)CCn2ccnc2)C)C)cc1 Cc1ccc([N+](=O)[O-])cc1C(N1CC(NC(=O)C=CC(C)(C)C)CC1C)=O N1(C(c2ccc(C(F)F)o2)C(=O)NC(CC)C)CCOCC(O)C1 c1(C(N2CC3C(CNC(CCCSC)=O)C3C2)=O)cc2c(s1)CCOC2 c1(CNC(=NCC)NCc2cnc(C3CC3)o2)ccc(C)c(C#N)c1 C1(NC(C=C(CC)C)=O)CC2(C1)CN(C(C1(c3ccc(Br)s3)CC1)=O)C2 CC1=C(C(=O)NCC(F)CNC(C2CCCCN2C)=O)C(C)(C)CCC1 c1(C(=O)NC2CCC(CNC(c3csnc3Cl)=O)C2)ccc(=O)n(C2CC2)c1 C12(C(=O)NC(CC(C)C)CNC(c3ccc(C4CC4)o3)=O)CC3CC(CC1C3)C2 c1(C(=O)NCCC(CCC)NC(=O)CC(CC)C(C)C)cnc2cc[nH]c2c1 C1(CCNC(CCCC=C)c2nnnn2Cc2ccco2)CCC(C)(C)CC1 C1(CC(N2CCC(O)(CN(C(=O)C(C)(C)CF)C)C2)=O)CCC(C)(O)CC1 c1(C(C)(C)NC(=O)OCc2cnc(C3CCC3)s2)ccc(C(F)(F)F)cc1 N1(C(C2C(C)C2)=O)CCCC(NC(=O)CCc2ccc(Br)cn2)C1C c1(C(=O)NC2CC(n3cc(C(CC)(O)CC)nn3)C2)cnc2c(c1)COC2 c1(C(=O)NC2C(CNC(c3c(C#C)c[nH]n3)=O)CCC2)ccc2ccoc2c1 N1(C(C2(C(=O)OC)CC2)=O)CCCCC(CNC(C2(C)CC3CCC2O3)=O)C1 c1(C(N2CC(F)(CNC(C(C=C)(C)O)=O)C2)=O)ccc([N+](=O)[O-])c(N)n1 C1(CNC(C2CC3(CCC3)CO2)=O)CCC2CN(C(=O)Cc3ccsc3Cl)CC12 C(=O)(C(C)CC(C)(C)C)NC1C(F)CCN(C(COCCSC)=O)C1 c1(C(=O)NC2(CO)CCCN(C(COCC(C)C)=O)C2)ccc2c(c1)CNC2=O Cc1nc[nH]c1CNC(C1(C(=O)NCc2ccn(C)n2)CC1)=O Cc1scc(C(=O)NC(C)CNC(=O)CCc2nncn2C)c1C Cc1cc(Cl)ccc1C(=O)NCC1CCCC1NC(=O)CC1COC(C)(C)C1 CC1(C)CC(CNC2CC3C=CC2C3)CCO1 c1(C(=O)OC)cnc(C(=O)NCC(C2CC2)N(C(=O)C(O)C2CCCC2)C)cn1 C1(C(=O)NCC2(COC)CCCN2C(C2CC(C)(F)C2)=O)Cc2ccccc2O1 C(=O)(CS(F)(F)(F)(F)F)N(C1CCCN(C(=O)C2=NOC(C)(C)C2)C1)C c1(C2C(C(N3CCC(CCNC(=O)CCc4ncco4)C3)=O)C2)ccccc1Cl c1(C(N(CCNC(c2ccc(F)s2)=O)CCOCCO)=O)cccnc1O Cc1cn2cc(C(=O)NCCC(C)NC(C3CCC3(F)F)=O)cc(F)c2n1 C12(CNC(C(=O)N(CC(C)(C)C)Cc3ccc(Br)cc3)=O)COCCN1CCOC2 c1(C(=O)NCCCN(C(=O)C(C)NC(C(C)(C)C)=O)CC)n[nH]cc1C(F)(F)F C(=O)(C#CC1(C)COC1)N1CCC(CCC(=O)NC(CCC)C(C)(C)C)CC1 c1(CC)cc(C(=O)NC2CC(C)(CNC(=O)C(C)CSC)C2)oc1CC N1(C(COC(CC)(C)C)=O)CC2CC(O)C1C2NC(=O)CCn1cc(C)cn1 CCN=C(NCc1ccc(Br)cc1)NCc1cn(CC(F)(F)F)nn1 c1(OC)cc(CNC(=O)CCOC2CN(C(=O)C(C)=C3CCC3)C2)cc(Cl)c1 C1(C(=O)NCC(CSC)(C)C)COC2(C1)CN(C(c1c(C)ccn1C)=O)C2 c1(CC)ccc(C(C(=O)NC(CN)C(C)(C)OC)C(C)C)cc1 c1(CC)nc(C)oc1C(=O)N(C)CCOCCCNC(C1CCCSC1C)=O CC(=O)CCCC(=O)NC1CCC(NC(C2C(C)C2(F)F)=O)CC1 C1(C(=O)NCCC23CC(C)(OC2)C3)CCc2ncc(Br)n2C1 C(=O)(C(C)(C)CCSC)N1C(CC)C(NC(c2csnc2C)=O)CC1 Cc1nnc2cnc(C(N3CC(CNC(C4C(C)C4C)=O)OC(C)(C)C3)=O)cn12 c1(NC(c2nc(-c3ccc(OCCC)cc3)sc2)=O)ccc(OC)c(Cl)n1 C1(C(N(CCN(C(=O)CC2CCCNC(=O)C2)CC)CC)=O)CCCC1C1CC1 C1(CCC)(NC(=O)C(CO)NC(=O)COC)CCN(C(C2CC2(Cl)Cl)=O)CC1 N1(C(N2CC(OC)C(F)C2)=O)CC(C)Oc2ccncc21 C[Si](C)(C)C1(CNC(C2CCC(NC(c3nsnc3O)=O)CC2)=O)CC1 C(=O)(CC(C)CC(C)(C)C)N1CC2CCN(C(c3cc(C)[nH]c3C)=O)C2C1 c1(C(=O)NCC2(F)CC(NC(c3cc(C)oc3)=O)C2)nc(C(C)C)oc1C CCC(CC(F)(F)F)C(=O)N1CCCC(C2CCCCN2C(C2SCCS2)=O)C1 N1(C(CNC(=O)OCC)=O)CCC(C(=O)NC2CCN(C)C2(C)C)C(O)C1 N1(C(CC2(CSC)CC2)=O)CCC2CCCC12C(N1CCC(n2cnnn2)C1)=O c1(N2C(C3CCN(C(C(COC)(C)O)=O)CC3)C(C)(C)C2)ncnc2ccsc12 c1(C(=O)OC)cc(C(N2CCC(c3ccc(C)cc3)CC2)=O)c2ccccn12 C12CCCN(C1)CC(=O)NC(C)CC(=O)N2C.C(C)(C(C)C)=CC N1(C(CC(CC)OC)=O)CCN(C(=O)C(C)CC(=O)OC)CC1c1ncc[nH]1 Cc1cnc(C(N2CCCC2CNC(=O)Cc2cc(F)ccc2F)=O)cc1C c1(OC)ccc(Br)c(CC(=O)NCC2CN(C(C3CC(C)CO3)=O)C2)c1 S(=O)(=O)(c1ccc(N(C)CCN(C)C)c(Br)c1)N1C(C)CCC1CNCO C1(N(C(C(C)SCC)=O)CCOC)CCN(C(=O)CC2CC=CCN2C)CC1 Cc1nc(O)ccc1C(=O)NC1CN(C(c2c(C)noc2C(F)F)=O)CCC1C c1(C(N2C(CCC(=O)NCc3ccsc3)CCC2)=O)ccc2ncsc2c1 C1(NC(c2cn(CCC)nc2)=O)(CC)CCN(C(=O)C(C(C)C)N(C)C)CC1 Cc1cc(NCCCCO)ncc1S(=O)(=O)N1CC(c2ccccc2)OCC1C CCCCC(C)(F)C(=O)NCC1CN(C(c2cn3nc(C)sc3n2)=O)CC1(C)C C#Cc1cnc(C(N2CCOC(CCCNC(c3c[nH]nc3Cl)=O)C2)=O)c(C)c1 Cc1ccc(C(=O)N(C)CCC2CCCCN2C(=O)COCCCF)n1C Cc1nnc(CC(=O)NC(C)(CNC(=O)CC(O)C2CCCC2)C2CC2)o1 Cc1cc2sc(C(=O)NC(C)(CNC(=O)CC#N)C3CC3)c(C)c2cc1C CC1CCCCC1(CNC(=O)CNc1ccc(O)cc1)NC(c1cccnc1)=O c1(N(CC(CC)O)C)ccc(S(=O)(=O)NCc2c(C)nn(C)c2C)c(Br)c1 c1(C(C(=O)NC(C)CNC(C2CC2(F)F)=O)O)ccc(Cl)cc1F CC(N=c1ccnc(N2CCC(F)(c3ccccc3)C2)[nH]1)c1ncc(F)cc1F C1(CNC(CN2CC(C)C2)=O)N(C(c2ccc3scnc3c2)=O)CCCC1(C)C Cc1cc(C(N2CCC(OCCNC(=O)C(C)N(C)C)C2)=O)c(C)s1 CCC(C)(O)C(=O)N1CCC(C(C)NC(c2cccc(OC(C)C)c2)=O)CC1 N1(C(c2c(CC)cncc2)=O)CC(C)C(NC(C2(NC(C)=O)CCC2)=O)C(C)C1 c1(OC)ccccc1C1(C)CC1C(N1CC2CC1C2NC(=O)COCCCF)=O c1(CC(=O)NCC2N(C(c3c(C)ccnc3)=O)CC(F)C2)ccc2nonc2c1 c1(OC(C)C)ccc(NC(C2CC3(C2)CN(Cc2ccccc2I)C3)=O)cc1Br c1(C(=O)NC(C2CN(C(=O)C3=NNC(=O)CC3)CCO2)C)ccc(Cl)c(F)c1O Cc1ncc(C(=O)Nc2cccc(NC(=O)CC3CCC(=O)N3)c2)cc1N c1(OC)cncc(C(N2CC(C(C(=O)NC3CCC(C)(C)C3)OC)C2)=O)c1 C(C(O)CNC(=O)C(C)OCOC)OC(N(CCOC)C)=O.C(C)(C)(C)O C1(NC(C(=Cc2ccccn2)C)=O)(CO)CCN(C(=O)C(C(C)C)N(C)C)CC1 Cc1cc(F)c2c(c1)CCN(C(c1ccc3c(c1)OCC3)=O)C2 C1(C(=O)NC(CCC)CCC)CC2(CCN1C(=O)C(C)SC)CC2 CCC(C)(C(=O)NCC(CNC(c1csc(-c2cccc(Cl)c2)n1)=O)OC)OC c1(C(N2CC(C(N)=O)(CNC(C3C(C)COCC3)=O)C2)=O)c(F)ccc(F)c1Cl N1(C(C(C(C)(C)C)O)=O)CCC2CCCC12CNC(=O)Cc1ccc(O)nc1 CC(CC(F)F)C(=O)NCCN(CCOCCO)C(c1c[nH]nc1C1CCCO1)=O CCC(C)(CNC(C1(F)CCCN(C(c2cc(OC)ns2)=O)C1)=O)C(N)=O c1(OC)cnccc1C1(C(=O)NCC(C)CO)CC(N)C1 C(=O)(C(F)(CNC(C1CC1C1CCC1)=O)C(C)C)NCC1(C#C)CCOCC1 c1(NCC2(CCC)CCC2)nc(N2CCS(=O)CC2)nc2c1ncn2C C12(NC(c3n(CC)ccn3)=O)CCN(C(=O)Cn3ncnn3)CCC1C2 C1(CC)CN(C(c2cnc(Cl)s2)=O)CCC1NC(c1cn(CCOC)nn1)=O C(=O)(CCC(C)(C)[N+](=O)[O-])NCC12CC(NC(CCc3c(C)ncs3)=O)(C1)C2 C1(NC(CC=C)=O)CN(C(c2ccc(Cl)c(OC(F)(F)F)c2)=O)CCC1(F)F c1(C(N(C(CC)CC(=O)NC2COC(C(F)F)C2)C)=O)cccc(C)c1N c1(C(=O)NC2C(NC(CN(C(COC)=O)C)=O)CCC2)ccc(F)cc1C1CC1 C(=O)(C(O)CN(C(=O)C=CCOC)C)NCC(CC)OC C(=O)(CCC1CCc2ccccc21)NCC(CNC(C#CC1(C)CC1)=O)(C)O c1(C(=O)NCC2CN(C(C(C(C)C)O)=O)CC2C)cccc2c1CCCC2 CC(C)(C)CCC(=O)C(=O)N1CCC(CF)(NC(c2cc3ncccn3n2)=O)C1 c1(CC(=C)C(=O)NC(C)CCC=C(C)C)ccc(F)cc1F N1(C(c2cc(C)ncc2C)=O)CC2(C1)SCCC2NC(=O)C(O)C1=CCCCC1 c1(-c2n(CCCO)nc(-c3cncc(Br)c3)n2)ccc(Cl)cc1Cl N=c1sccn1CC(N1CC(O)(CNC(C2CC(=O)N2)=O)C1)=O Cc1ccc(CC(=O)NC(C)(C)CCNC(=O)Cc2ccoc2)cc1O CCC(C)(C)C(=O)NC12CC1CN(C(C1(c3cncnc3)CCCC1)=O)C2 c1(NC(CN(c2nnc(CC(C)C)s2)CC)=O)cccc(C)c1 c1(C(N(C2CCCC(NC(C=CCCC)=O)C2)C)=O)cc(C)c2[nH]nnc2c1 C1(NC(CN(C)C)=O)CCCC1NC(=O)C(CO)NC(=O)Cc1ccccc1 c1(C(N(CCCNC(=O)C(O)COC)CC)=O)cn2cnnc2cn1 c1(OC)cc(C(=O)NC2CC(CNC(=O)C(C)O)C(O)C2)c(F)cc1Br c1(C(N2CCC(NC(CCCn3c(C)nc(C)n3)=O)C2)=O)ccn2c1CCCC2 CCCCCCC(=O)N1CCCCC1C1CCN(C(c2nn(C)cc2Cl)=O)CC1 C1(NC(c2c(C)nn[nH]2)=O)CC(F)(F)CC1NC(c1cnns1)=O Nc1nccnc1C(N1CCCCC1CCNC(=O)CN1CC2CC2C1)=O Cc1nc2ccc(F)cc2c(NC2(C)CCc3ccccc3C2)c1C C(=O)(C(C)(F)C(C)(C)F)NCC(CC(C)C)NC(C1CCCC2CCCN12)=O N1(C(CCC(C)OCC)=O)CCC(NC(=O)CCC(C)N(C)C)C2(CCC2)C1 CS(=O)(=O)c1ccc(C(N2C3CCC2CN(C(=O)CCN2CCC(F)C2)C3)=O)o1 C1(CNC(CCOCC)=O)COCCN(C(C2CCCCNC2=O)=O)C1 C(=O)(CC(CN(C)C)C(F)F)NCCCN(C(=O)CN(C)S(N)(=O)=O)CC N1(C(C(CCC)OC)=O)CCC(C2CC2NC(c2nsnc2O)=O)CC1 C1(C(N(CC(=C)C)C)=O)C=CCN(C(C2CCCC2CCC)=O)C1 C1(C(N2CC(CCC#C)C2)=O)CC2CCC1N2C(=O)CC1CCC(C(C)C)CC1 N1(C(CC(C)n2ccnc2)=O)CC2(COC(CNC(=O)Cc3ccsc3)C2)C1 N1(C(CCN(C)CC)=O)CC(C(=O)NC(C)CCC(=O)OC)CCC1(C)C N1(C(C(n2cc(-c3ccc(CCC)cc3)nn2)C)=O)CCC2CCC(C1)S2 C#Cc1ccc(Br)c(C(=O)NCC(CNC(=O)C=CC(C)C)C(F)(F)F)c1 c1(CC(=O)N(CC(CNC(COC)=O)O)C)cccc(Cl)c1F c1(NCC=CCNC(c2c(CCC)occ2)=O)cc(C)nc(COC(C)C)n1 N1(C(c2cnc(C(=O)OC)s2)=O)CCCCC(NC(C2(C)CCCC2C)=O)C1 C(=O)(CCCCCCN=[N+]=[N-])N1CC2N(C(c3c(C)cc(F)cc3)=O)C(C2)C1 c1(OCC(=O)NCC(C2CC2)NC(C2CCCOC2)=O)cncc(Br)c1 C1(CNC(=O)CNC(=O)NC2CCCO2)CCCN(C(c2cc(Cl)no2)=O)C1 c1(CNC(C2(CC=C)CCC2)=O)ccc(C(=O)N(C(CCO)C(F)F)C)cc1 c1(C(=O)OCC)ccc(NC(=O)NCC2CN(C)CCN2C)cc1C C(=O)(CCCCC(=O)NC)N1CC(CNC(C(CCCC)O)=O)C1 c1(C(=O)NC2CCC(CN(C)C)CC2)ccc(N)c(-c2nccs2)c1 C1(C(=O)NCC2C(NC(=O)Cc3cnc[nH]3)C2)CC2(CCC2)CO1 CCCCCC(CC)C(=O)NCCC1CCCN1C(c1ccc(CC)nc1C)=O Cc1ncc(C(N2CC(C(N3CCC3CN=[N+]=[N-])=O)CC2(C)C)=O)c(=N)[nH]1 C12CC3CCC1N(C3)C2=O.C1(C2CC2)(CNC(=O)OC(C)(C)C)CCNC1 c1(C(=O)NCC2CCC(NC(C(CC)(CC)OC)=O)C2)cnc2ccc(C)cn12 C1(NC(C(c2cccs2)NC(C(CN(C)C)O)=O)=O)CC2CC1C(O)C2O C#CCC(C(=O)NCCCOCCN(C(=O)C(C1CCCCCC1)C)C)C1CC1 c1(C(F)F)nc(OC)cc(=NC2CCOC(C3CCCCN3C(=O)C=CCO)C2)[nH]1 C1(C(=O)NC2CC(NC(CSCCC(C)C)=O)CC2O)CCC([N+](=O)[O-])CC1 N1(C(C2N(C(c3c(C)nccn3)=O)CC(O)C2)=O)C2CCC1CC(C)C2 C=CC(C)(CCOC)C(=O)N1CCCN(C(=O)C(C)OCC(C)C)CC1 N1(C(CNC(C)=O)=O)CCC2(NC(C3C4CCC3(C)C4(C)C)=O)CCCCCC12 C(=O)(C(C)(C)CCC(=O)NC(c1nccn1C)CO)OC.C12CN(C1)C(=O)O2 C(=O)(C1CCc2nccn21)N1CC(C#C)N(C(c2cncc(NC)c2)=O)CC1 C1(C(C)NC(=O)C(C2CC2)C2CC2)CN(C(=O)CC=C(Cl)Cl)CCO1 c1(C(C)SCCN2CCOC2=O)c(F)cccc1F Cc1ncc(CC(N2CC(CNC(C3CCC(=O)N3)=O)C(O)C2)=O)c(O)n1 c1(C(N2CC(NC(c3ccncc3)=O)CC23CCC3)=O)cc2c(Cl)cccn2n1 c1(C(N2CCC(NC(C3C(C)OCCC3)=O)(CF)C2)=O)ccc([N+](=O)[O-])c(O)c1 CC1CN(C(c2ccc(C#N)cc2)=O)CCC1NC(=O)C(C1CC1)C1CC1 c1(SC)nc(N2CC(C)(C)CC2CNC(c2ccncc2Cl)=O)cc(C(F)F)n1 C1(NC(c2cc(OCC)no2)=O)CC2CCC(C1C)N2C(C1CC2CCCC12)=O c1(C(=O)NCCC(=O)NCCCCCC=C)c(C)ncnc1C C(=O)(C1(C)CCc2ccccc21)NC1CC(NC(c2cn(C)nn2)=O)C(O)C1 N1(C(CC2CC(=C)C2)=O)CC(NC(c2ccc(OC(C)C)cc2)=O)C(C2CC2)C1 C1(NC(=O)Cc2nc(C(F)(F)F)cs2)CCOCC1NCCN1CCC(O)CC1 N1(C(CCN(C)CC)=O)CCOC(CCNC(c2cn(CC)nc2C)=O)C1 N1(C(c2c(C)ccnn2)=O)CCN(C(c2ccns2)=O)C2CCCCC12 c12ccc(OC)c(F)c1CNC2=O.c1(CCC)cn(C(C)(C)C)nn1 CCC(C(=O)N1CCC(C(=O)NOC(c2cnn(C)c2)C)(OC)C1)C(C)(C)CC C=CC1(C(N2CCCC2CC=CC)=O)CCCCC1.N12CCCC(F)(C1)C2=O N1(C(CCC2CC(OC)C2)=O)CCCCCC1C(N1CC2CC2(CO)C1)=O CN1C(=O)NCC1C(=O)NCC1CC1CNC(c1ccccn1)=O C1(CCCC)CN(C(=O)CC2CC(=O)NC2=O)CCN1C(c1cn(CC)cn1)=O C1(CNC(C=COCC)=O)CC(C)(C)CN1C(c1cnn(C)c1N)=O Cc1c(Br)cc(Cl)c(NC(C2CCN(C(c3ccc[n+]([O-])c3)=O)CC2O)=O)c1Cl C1(NC(c2nn(C)c(F)c2)=O)CC2CCC1CN2C(=O)C=Cc1ccco1 C1(NC(c2cn(C)nn2)=O)CCCCN(C(C2(N(C)C)CCCCC2)=O)CC1 c1(C(N2CC(OC)C(NC(c3cc(C(C)C)no3)=O)C2)=O)cc(C)ccc1F C1(CNC(C(C)OC)=O)CC(F)(F)CN1c1nc(C(=O)OC)ns1 C1(C2CCN(C(c3cscc3Cl)=O)C2)(NC(c2cc(C)c(C(F)F)nc2)=O)CC1 C1(CC(=O)OCC)CCN(C(c2cc(C(C)(F)F)on2)=O)C1(C)C c1(C(CC)C(=O)Cc2csc(N3CCOCC3)n2)cc(F)cc(Br)c1.N1CCC1 c1(C(=O)NCC2N(C(C(C=C=C)C)=O)CCCC2)cc(O)nc2[nH]c(=N)ccc12 C(=O)(C(F)(F)C1=CCOCC1)NC1CC2CN(C(=O)COC3CCOC3)C1C2 c1(C(=O)NC2CC(OC)CN(C(=O)CC3CC4CC4C3)C2)cc(C)c(F)cc1Cl c1(C(=O)NC2C(CNC(c3c(C)cc(CO)o3)=O)CCC2)cccc(F)c1N c1(OCCCN(C)C)ccc(C(=O)Nc2cnn(C3CC3(F)F)c2)cc1 c1(C(=O)NCC(CNC(c2c(C)n(C)nn2)=O)(C)C)n[nH]c2c1CCOC2 C(=O)(C1CCCn2nccc21)NCC1CCN(C(C(C=C)(C)O)=O)CC1CC O=C(C#CC1CCC1)NCC1CCCC1NC(c1cnn(-c2ccncc2)c1)=O C1(NC(=O)CCc2ccsc2Br)CCCCC1NC(C1C2CCCC12)=O N1(C(c2cccc(Cl)c2)C(=O)NC(c2ccc(CN)cn2)C)CCC(O)C(F)C1 C1(NC(=O)Nc2ccc(-c3cn(C)nc3)cn2)CCC2CCCC2C1 c1(C(N2CCN(C)C(CNC(=O)C=CS(C)=O)C2)=O)ccc2cnccc2c1 C1(NC(C2CCC(CCCC)CC2)=O)CN(c2ncnc(C)c2OC)CCC1C C1(CNC(CC(=O)NC)=O)COCCN(C(=O)C#CC2CC2)C1 c1(C(N2CC3N(C(C(C)Oc4ccccn4)=O)C3C2)=O)cc2cc[nH]c2cc1Cl c1(NC(C)=O)cccc(NC(=NCC2CC2(Cl)Cl)NCC2CCCO2)c1 c1(C(N(C)CC2CCN(C(c3ccoc3Br)=O)C2)=O)cc(N)cc(O)c1 C1(NC(=O)CSc2ccncc2)CC12CCN(C(c1ccc(Br)c(F)c1)=O)CC2 C(C)(CCC(=O)NCC(CC1CCCC1)C(=O)N(C1CCCCC1O)C)OCC CC(C)(C)C1=NOC(C(N2CC(CNC(C3CC4C=CC3C4)=O)C2)=O)C1 N1(C(COCC(=O)OC)=O)CC2C3CCC(C2C1)N(C(=O)C(C)OCC(C)C)C3 C1(CNC(C(C)=C2CCCC2)=O)CC2CCC(C1)N2C(=O)CNC(=O)CCC1CC1 Cc1ccc(CCC(=O)NCC2(NC(c3ccc(O)cc3)=O)CCCC2)cc1 c1(C(N2CCC(NC(C3C(CC)C3)=O)C2C2CC2)=O)ccc(=O)n(C)n1 c1(N2C(=O)C2)ccccc1C.c1(SC)nnc(-c2ccc(O)cc2)n1CC(N)=O C(=O)(CS(=O)(=O)CCOC)NC1CCN(C(C(C=C)(C)O)=O)CC1F Cc1oc(CCN)nc1C(N1CC(n2cc(Cc3ccccc3)nn2)C(C)C1)=O c1(C(C(=O)NC(CC)CN(C(=O)CCc2cn[nH]c2)C)O)ccc(C)cc1 C(=O)(C(Cc1ccco1)NC(=O)C(C)n1cccc1)N(CC(COC)C)C c1(C(=O)NCC2(NC(c3cc(C(=O)OC)no3)=O)CCOC2)c(F)cccc1F c1(OCC)ccc(CC(=O)NC(C)CCCNC(C2(OC)CCC2)=O)cc1 CC(C)C(O)C(=O)N1CCC(OCCNC(C2(c3cccs3)CC2C)=O)CC1 C(CCCC(=O)N=c1ccn(C2CC2)[nH]1)NC(C1N(C)C(=O)CCC1)=O C1(NC(C(C2CCOCC2)OC)=O)CCCC1CNC(C1(F)CCC1)=O C1(C(=O)N(C)C)CCCN2CCCCC12.c1(OC)cc2c(C(F)(F)F)cc1[nH]2 c1(CC(=O)NCC2CC2NC(c2nc(Cl)sc2Cl)=O)c(F)cccc1Cl C1(CNC(C2CC(O)(CNC(c3ccc([N+](=O)[O-])[nH]3)=O)C2)=O)CCC2(CC2)CO1 C(=O)(C(C)(F)C(F)(F)F)NCCOC1CCN(C(c2cc(CC)oc2C)=O)C1 c1(C(C)=O)cc(C(=O)NC(C(=O)NCC2(CC(C)C)CC2)C2CC2)n[nH]1 C(=O)(CS(=O)(=O)CCCC)NC1CN(C(C(F)=CCC)=O)C(C)CC1 C1(C(=O)NCCOCCCNC(CC2N(C)CC=CC2)=O)CCC=CCCC1 N1(C(c2c(N)ccc(Cl)n2)=O)CCc2nc(CNC(=O)CCC3CCC3)sc2C1 C=CCC(C)(O)C(=O)N1CC2CC1(C(=O)NCc1ncc(CO)o1)C2 c1(N2CC(CCOC)(NC(C3CCN(CC#C)CC3)=O)C2)nc(C)nc(O)c1C C12(C(N3CCC(C#N)C3)=O)CCCC1CCN2C(C1CC2CC2C1)=O C1(CNC(C2(COC)CCC2)=O)CCC(NC(c2scnc2C)=O)C1 CC1CCCn2c(C(=O)NC(C)CCNC(=O)CNC(c3ccncc3)=O)cnc21 CCC(CC)C(C(=O)NCCN(C(C1CCCC1)=O)Cc1ccccc1)OC C1(CC)(NC(C2CC(Cl)(Cl)C2)=O)CCN(C(=O)Cc2ncncc2Cl)CC1 c1(C(=O)NC2CCC(CNC(c3ccc(Br)o3)=O)C2)ccnc(S)c1 C12(C(=O)NCCC(=O)NCC(COC)O)C=CC(CC1)C2 C1(NC(=O)OC(C)(C)C)CC2(CC(NCC3C4OC(=O)OC34)CCS2(=O)=O)C1 C(C)(C(CC(=O)NC1CC(C(C)C)C1)NC(C1CCOC1(C)C)=O)OC C(=O)(CC(CC(C)C)NCC1CCC(c2nc[nH]n2)O1)OCC CC(C)C(C)C(CNC(=O)CCCCCF)NC(=O)Cn1ccc(C2CC2)n1 C(CC(=O)Nc1c(C)nn(C)c1C)(C(F)F)NC(c1cccc(C)n1)=O c1(OCC)ccc(NC(C2CN(C(=O)C(=O)NCC3(C#N)CCCC3)C2)=O)cc1 CC1CCC(CC(=O)NC2CCCC2NC(=O)Cc2cc(Br)cs2)C1 S(=O)(=O)(c1ccc(F)cc1)ONC(C1C(C)CCN1C(=O)C1=CCCSC1)=O C12(NC(C34CC(C)C3C4)=O)CCCC(CN(C(c3cocn3)=O)C1)C2 C1(C(=O)Oc2c(COC)ccc(CS(C)(=O)=O)c2)CCN(C(=O)OC)C2(CC2)C1 C(CCCCC(=O)N(C)Cc1cnco1)NC(c1c(CC)n(C)nc1)=O c1(OCC)cc(N2CCN(C)CC2CNC(=O)C(C)N(C)C)ccc1[N+](=O)[O-] C1(C(N(C)Cc2nc(C)sc2)=O)CCC(C(C)C)N1C(c1cnn(C)c1)=O C12(NC(Cc3ccc(CC)cc3)=O)CCCC1N(C(C1(C)C=CCCC1)=O)CC2 c1(C(=O)NCC2(C)N(C(c3ncc(OC)cn3)=O)CCC2)ccc(C)c(Cl)c1F C1(NC(c2cn(CC=C)nn2)=O)CCCCC12CCCN(C(C1(C)CC1)=O)C2 C1(CC(=O)NC2CC(C(C)NC(CCCN(C(C)=O)C)=O)C2)CCC(C)(C)O1 C1(NC(CCc2ccn(C)c2)=O)CCCC(NC(=O)CN2CCCNC2=O)C1 C12(COC)COC(C(N3CC(O)(C(C)NC(=O)C(C)c4cccs4)C3)=O)(C1)C2 N1(C(C2CC(OCC)C2)=O)CC(C)CN(C(c2ccc(CC)c(C)c2)=O)C(C)C1 c1(CC=C)cccc(CC(C(=O)NC(CC2CC2)CO)NC(=O)C(OC)OC)c1 Cc1nscc1CC(=O)NCCN(C(=O)C=CBr)CC1CC1 C(=O)(CCCCN(C)C)NC1CC(C)(NC(C(C2CCCC2)NC(C)=O)=O)C1 C1(OCC(=O)NCCCCNC(c2n[nH]cc2Br)=O)CCC(F)(F)CC1 c1(CCC)noc2nc(C)cc(C(=O)NCC3(NC(=O)OC(C)(C)C)CCC3)c12 c1(SCC(N2CCC(COCC)C2)=O)ccc(Br)cc1.C1CC(=O)N1 c1(C(N2CC3C(CNC(C4(CCF)CCC4)=O)C3C2)=O)ccc(F)c(Cl)c1 C1(C)(CNC(C(C2CN(C(C3C(CCC)CCC3)=O)C2)OC)=O)CSC(C)=N1 C(=O)(C(CCOCC)NC(=O)CC1COC(=O)C1)NCCC=CC=C c1(C(=O)NCC2(NC(C3CC(CCC)C3)=O)CC2)ccc(CC)cc1O N1(C(CC2CC(OC)C2)=O)CCC(CN(C(=O)CCc2ccc(C)o2)C)C1 c1(N(C)CC2CCN(C(=O)C=Cc3ccccn3)CC2)nc(Cl)nc2[nH]ccc12 c1(OCC)ccc2cc(CN3CCN(C(C)CO)C(C)C3)ccc2c1 Cc1cc(C(=O)NC(C(=O)NCCCS(C)(=O)=O)C2CCOC2)cc(C#N)c1 C1(NC(c2n[nH]c(CC)c2Br)=O)CCCN(C(=O)CC=C(C)C)CC1F CC(C(=O)NC(C)(CNC(=O)C=CC1CCC1)C1CC1)NC(N)=O C1(NC(C(CC)OCC)=O)COCCN(C(c2cocn2)=O)C1 CCN=c1cc(C(=O)NCC2CC(NC(=O)C(n3nc(C)cc3C)C)C2)cc[nH]1 N1(C(CSCCC(C)C)=O)CCC(NC(C2CCC(C)(C)CO2)=O)C(CO)CC1 c1(C(=O)NC23CC(CNC(C4CCCOC4)=O)(C2)C3)occ2c1CCCC2 C(=O)(C(O)CC(C)C)NCC1N(C(C(c2cc(C)ncn2)(F)F)=O)CCCC1 c1(C(N2CC(CNC(C(n3c(C)cc(C)n3)C)=O)C(C)C2)=O)cc2n(n1)CCO2 c1(C(=O)NC2CCC2CNC(c2ocnc2C(F)F)=O)ccc(F)c(Cl)c1F c1(C(=O)NCC2CN(C(c3ccsc3Cl)=O)CCO2)c[nH]c2nc(F)ccc12 N1(C(c2cncc(C)c2)=O)CCC(CNC(=O)C(C)OCCC(C)C)C(F)(F)C1 c1(C(=O)NCC2(OCC)CN(C(C(C(=C)C)(C)C)=O)C2)cccc([N+](=O)[O-])c1 N1(C(C=CC)=O)CCN(C(c2cc(Cl)ccn2)=O)C(C)C1C c1(C(=O)NC2CC3CC(NC(C4C(C)C4C)=O)C3C2)cc(Cl)cc([N+](=O)[O-])c1O Cc1cccc(C)c1OCC(=O)NCC(C)NC(c1ccc(C(F)F)cc1Cl)=O N1(C(c2cccc(Cl)c2)=O)CCC2(C1)CN(C(C1CC=CCC1)=O)CCO2 C(CN=c1[nH]c(N(C)Cc2ccccc2)nc(=N)[nH]1)(c1ccccc1Cl)N(C)C C1(CNC(CC2(OC)CN(C(c3nc(O)sc3C)=O)C2)=O)CCCC12CCC2 c1(-c2c(CNc3cc(CCC(C)C)nn3C)n(C)cn2)ccc(C#N)cc1N n1(CC)nc(C(N2CCC(CCC(=O)N=c3cco[nH]3)C2)=O)c2ccccc12 C(=O)(C(C)C(C)NC(=O)C(CCC1CCC1)NC(=O)CC1CCCCN1C)OC N1(C(C(C)N(C)Cc2ccccc2)=O)CCc2cc([N+](=O)[O-])cc(Br)c21 N1(C(CCN(C(=O)C(O)C(F)(F)F)C(C)C)=O)CCC12CCC(C)CC2 O=C(CCCCCCCC1CC1)NC1CC2(C1)CC2NC(c1ccc(O)cn1)=O N1(C(C2(C)CC(C)C2)=O)CCCC2(C1)CN(C(=O)C1=NOCC1)C2 N1(C(C(=O)NC2CC2)=O)C(CC(=O)O)CCC1C1CC1.C1(=O)C(=O)NN1CC(F)F c1(OC)cc(N2CC(OCCNC(C3CCC(C)(CC)O3)=O)C2)ccc1[N+](=O)[O-] c1(C(=O)NC2C=CC(CNC(Cc3cc(CC)no3)=O)C2)cc2scc(Cl)c2[nH]1 CCCCC(C)C(=O)N1CCCC1(C(=O)NCc1cccc(CO)c1)CC CC1CN(C(C)=O)CCC12CCN(CCc1cccc(Cl)c1)CC2 CC1CC(NC(C2CCCNC2=O)=O)CN(C(c2cccc(O)c2Br)=O)C1 c1(C(=O)NC23C(C)OC(CNC(=O)C(C)(C)F)(C2)C3)cc(Cl)c(N)c(Cl)c1 c1(C(=O)NCC2CCN(C(C3C(OCC)CC3)=O)C2)ccc(OC(C)(C)C)cn1 C(C(C)C(F)(F)F)N(C(C(Cc1ccco1)NC(C1N(CC)CC1)=O)=O)C c1(OC)cccc(CN(C(=O)NCc2ccc(F)cc2O)C)c1Br C1(C(=O)NC2CN(C(C3(O)CCCC3)=O)CC2F)CC2(C1)CC(O)C2 c1(C(N(CC(C)(C)CNC(=O)C=CC(F)(F)F)C)=O)ccc2c(c1)CC(C)(C)O2 C(=O)(CCCN=[N+]=[N-])N(C1CCN(C(CCOCCCOC)=O)C1)C c1(CC)ccc(OCCC(=O)N(CCCNC(=O)C=Cc2sccc2C)C)cc1 c1(CCC(=O)NC2C(NC(C3N(C)C(=O)CC3)=O)C2)ccc([N+](=O)[O-])cc1Cl c1(C(C(=O)NCCCF)N(CCCC)C2CC2)ccc(OC)c(Br)c1 c1(C(=O)NC(C)CCCCNC(=O)CCCSC(C)(C)C)c[nH]c2nc(Cl)ccc12 Cc1ccc(C)c(C(N2CC(O)(CNC(c3ccnc(C(F)F)c3)=O)C2)=O)n1 N1(C(C2CC(SC)C2)=O)CCOC(CNC(c2c(CO)n[nH]c2C)=O)C1 c1(CC)nn(C)cc1C(=O)NC1CC12CC(NC(c1ccc(C(C)C)nc1)=O)C2 C12(C(=O)NCC(CC#C)(C)CO)CCC(CN(C(=O)COCCSC)C1)C2 c1(C(=O)NC2CCCN(C(C)C(=O)NCc3cocn3)CC2)ncc(Cl)cc1Cl C1(NC(C2CCN(CC)C2)=O)CCCCCC1C(=O)NCCCCCSC c1(C(=O)NC2CC(NC(c3c(O)ccc(CC)c3)=O)C2)cccc2ncc(C)n12 C(=O)(CCCCCS(N)(=O)=O)N(CC(CN(C(C(CCCC=C)(C)C)=O)C)O)C Cc1cc(F)c(C(C)C)cc1Nc1cn(C(C)(C)C)nn1 N1(C(CC2(C)CC(F)(F)C2)=O)CC(NC(c2ccn(C3CC3)n2)=O)CC2(CC2)C1 N1(C(Cc2ccc(OC)cc2)=O)CC(C)(C)C(NC(=O)C2=CCC2)C(C)(C)C1 c1(CCCN(CCCO)C(C)C)cnc(-c2ccccc2)[nH]1 c1(C(=O)NCCN(CCC)C(c2cc(F)ccc2C)=O)c(OC)ccnc1F c1(OC)ccc(C(N2CCCC(CCNC(=O)C(F)C(C)C)C2)=O)c(C)c1 CC(C(CO)NC(=O)Cn1nccn1)NC(=O)C(F)(F)C1CCOCC1 N1(C(c2c(CNC(C(C)SCC)=O)cco2)=O)CC2CCC(O)C(O)C12 N1(C(C2(OCC)CCCC2)=O)CCCCCC(NC(c2cccc(N)c2C)=O)C1 C1(CNC(C2CCS(=O)(=O)C2)=O)CC(F)CN1C(c1ccc(C(F)F)cc1)=O Cn1cc(C=CC(N2CCCCC2CCCNC(=O)CC2CCCOC2)=O)cn1 C1(C)(CCC=NC(c2c(C)oc(Cl)n2)=O)CCCN(C(C23CC4CC2C3C4)=O)C1 C1(NC(c2ncn(CC)n2)=O)CC(C(=O)NCC2(C(C)(F)F)CC2)C1(C)C Cc1cncc(C(=O)NC2CCCC2C(N2CCOCC2CCO)=O)n1 N1(C(C(C2CCN(C(=O)C#CC3CC3)CC2)C)=O)CC(CO)OCC1C c1(-c2ccc(Cl)cc2)n[nH]c(=NCC2OCCc3sccc32)o1 C=C(C)CCCC(=O)NC1CCCCCC1C(=O)N(C1CCN(CC)C1)C n1(CC)nc(C(=O)NC(CCOCCO)C(=O)N2CC(COC)C2(C)C)cc1O c1(C(C)OCC)nc(CC(=O)N(C)CC2CCN(C(=O)CSS(C)(=O)=O)C2)cs1 c1(NC(=O)NC23CC(C(C)(C)C)(C2)C3)ccc2scnc2c1 c1(OCC)c(C)cc(C(=O)NC2(C)CCN(C(C3(CO)CCCO3)=O)C2)cc1C C1(N(C(=O)N)C(n2cccc2)C)(CC23CC(CC(F)F)(C2)C3)CCOC1.CC(C)O C(C(F)(F)C(F)F)OCC(N1CC(NC(CCSCC(C)C)=O)C1)=O.C1CN1CO C1(c2cnccc2)CCN(CCOc2cc(C)ccc2Br)CC1c1nn[nH]n1 c1(OCC)ccccc1C(=O)NC(C(=O)NC1CCCCC1)C1CCOC1 C1(C2CC2)(NC(c2c(SC)n(C)nc2)=O)CCN(C(=O)C=Cc2nccs2)C1 N1(C(COCC)=O)CCOCC12CCN(C(=O)C1CC1)C2 C1(C(=O)NCCS(CC)=O)CN(C(=O)CSC)CC12CCC2 c1(C2N(C(N=c3cnn(COC)[nH]3)=O)CCC2)c[nH]c2ccccc12 CCCCCCCCCCC(c1nnnn1C1CC1)NCC(C)Cn1cccn1 C1(C(N2CC(C)C2)=O)CC12CCN(c1ncc(Br)c(C(F)(F)F)n1)C2 C1(CNC(C2C(C)C2)=O)CN(C(=O)Cc2ccc(F)nc2)CCC12CCC2 N1(C(=O)NC(c2n(CC)ncc2)C)CCC2(CCO2)C1 C(=O)(C(CCCCc1ccccc1)N(C1CCCC(C)C1)C)NCCSC C1(CCC)C(=O)N(C(c2n[nH]cc2-c2cccc(F)c2)=O)CC1C(=O)OCC c1(OC)ccc(C(C)OC(c2ccc(-n3ccnc3SC)cc2)=O)nn1 N(C1CCc2ccc(Br)cc21)C(C1CN(C(c2ccncn2)=O)CCS1)=O N1(C(c2cc(C(C)=O)on2)=O)CCC(C)C(CNC(c2ccncn2)=O)C1 c1(C(=O)NC(C(C)C)CCN(C)C(C2CC2C(C)O)=O)cnc2sccc2c1 c1(OCCOC)cc2cc(CN3CCC3Cc3ccccc3)[nH]c2cc1OC O=C(C1Cc2ccc(F)cc21)NCCCOCCNC(c1ncoc1C1CC1)=O N1(CC)CC2CN(C(C34CC3CCN4C(=O)C(N3CCOC3=O)C)=O)CC2C1 N1(C(CC(=C)Br)=O)CCC2CCN(C(c3ccc(S(N)(=O)=O)o3)=O)CC12 Nc1c(F)ccc(F)c1C(N1CC2CCN(C(C3CCS(=O)(=O)N3)=O)C2C1)=O c1(C(=O)NC2C(NC(c3cc(CC)ncc3)=O)COC2)c(C)ncn(C)c1=O Cc1nc2cccc(C(=O)NC3CCCCC3NC(=O)C(C)OCC3CC3)c2s1 c1(CCNC(C2C(CNC(c3scc(C)c3)=O)OCC2)=O)cccc(O)c1 N1(C(Cc2cnc(C)[nH]2)=O)CCN(C(=O)C#CC2CCC2)C(C)C1C c1(C(c2nnnn2Cc2cccs2)NCC(=C)Br)c(C2CC2)cnn1C N1(C(c2cc(C)ccn2)C(=O)NC(CC)(C)C)CC2(CCC2)C1c1ccccc1 C(=O)(C(O)P(C)(C)=O)NCCCC(C)NC(CCn1ncc(C)c1)=O C(CC(C)CC)(C(=O)N(C)Cc1ccnn1C)NC(C(C)=CCC)=O C1(C(=O)NCC(CC(C)C)(C)NC(=O)Cc2csnn2)CCC2(CCOCC2)C1 c1(C(N2CC(C)C(CNC(=O)CC3CC3)CC2)=O)ccc2cnnn2c1 C1(C(N2CC(C)(CC=C)C2)=O)C(CC)CCN1C(=O)C1=CCSC1 Cn1nccc1CCNC(=O)C(Cc1cnc[nH]1)NC(=O)CCC1CCC(=O)C1 Nc1c(C(=O)OCC2C(c3ccccc3)C2(F)F)cc(Cl)c(Br)c1F C1(CCNC(Cc2n(C)cnc2)=O)CCN(C(c2ccsc2)=O)CCC1(F)F N1(C(c2c(C)cccn2)=O)CC2CC1CN(C(=O)CC=CC(C)(C)C)C2 c1(C(=O)NCCNC(C2(C3CC3)CCC2)=O)cc(F)ccc1Cl c1(C(=O)NC2CC(NC(=O)CO)C2)c(Br)nc2n1CCC2 C(C(O)C(=O)NCCCCC1(NC(=O)CN2CC(C)(C)C2)CC1)=CCCC CCC(CC(=O)N(C)Cc1ccnc(C)n1)NC(=O)CCCN(C)C(C)=O c1(CN2CCC(CNC(=O)Nc3nn[nH]c3Br)C2)ccc(O)cc1 C(=O)(CCC(=O)NN(C)C)N1C(C(=O)NCC23CCC(OC)C2C3)(CC)C=CC1 C(=O)(C1CCCc2nccn21)NC1(C)CN(C(c2ccnn2CCF)=O)C1 Cc1nc2cccc(C(N3C(C)C4CC3C4NC(C3(C)CCNC3=O)=O)=O)c2[nH]1 c1(OC)ccc(C(C)NCC(C)C(C)(F)F)c(Cl)c1 c1(OCCNC(=O)Nc2sccc2Cl)ccccc1O CN1CCC2CN(c3nc(NCc4ncoc4C(F)F)c4ccsc4n3)CCC12 C(C1c2ccccc2CCN1C(=O)CC1CCNC1=O)NC(c1n(C)cnc1)=O c1(C(=O)NCC(CC=C)NC(=O)Cn2nnc(=O)[nH]2)cnc2[nH]cncc1-2 c1(-n2c(-c3ncn(-c4cc(C)sc4)c3)nc(Cn3cccn3)n2)ccc(F)c(C)c1 c1(OC)cc(C)cnc1C(=O)N(C)CC1(CNC(C2CCC(=O)O2)=O)CC1 c1(NC(C(C)NC(C)CCc2ccco2)=O)nc2c(s1)CCC2 C1(C(CNC(CCOC)=O)(C)O)CCCN(C(c2ccoc2CC(N)=O)=O)C1 c1(N(C(=O)C(C2CCN(C(=O)CSC(C)(C)C)C2)F)C)ccc2occc2c1 c1(C(=O)NCC2(NC(C3CC3c3ccco3)=O)CCC2)n[nH]c(C2CC2)c1Br C=CCCCCCC(=O)NC1CN(C(C2CCCCN2CCC)=O)CC1C N1(C(c2c(OC)cccc2)=O)CC2(CC(NC(=O)C(O)CC3CCCCC3)C2)C1 C1(C(=O)OC)CC(=O)N(C)C1C(=O)NC(C)CNC(c1cn(C)nc1C)=O Cc1nc(CC(=O)NC2CCC(CNC(c3sccc3C)=O)C2)cs1 CC1(C)COCC(C(=O)NC2COCCC2NC(=O)CCc2csc(=N)[nH]2)O1 C1(C(N(CCCCN(C)C(=O)OC(C)(C)C)C)=O)CC2CCC1CC2NO c1(OC)ccc(NC(=O)C(C)=CC2CC2)cc1S(=O)(=O)N(C)C Cc1ncnc(C(=O)N(CCNC(=O)CCS(C)(=O)=O)Cc2ccccc2)c1C N1(C(c2cnn(CC)c2C)=O)CCCC(NC(c2ccnn2C(F)F)=O)C1C C(CCNC(C1CC2CCC2C1)=O)(C(C)C)NC(COCC)=O C1(CC)CCN(C(=O)CCOCC2CCC2)C1C(=O)NCc1c(C)coc1C N(C1CCc2cc(F)c(F)c(F)c21)CCN1C(C)CCCC1C c1(C(=O)NC2CN(C(C(Cn3ccc(C)n3)C)=O)CC2C)c(C)cc(O)nc1C C1(C(N2CC(C)SCC2)=O)CC(C)(C)CCN1C(=O)CC1COC(=O)C1 C1(C(=O)NCC2CCCC2N(C)C)(CC)CN(C(c2cc(C(N)=O)[nH]n2)=O)C1 C#Cc1cc(C(N2CCC3(CC2)CC3NC(=O)C=C(CC)CC)=O)ccc1Cl C(=O)(C1=CC2(CCN(C(=O)Cc3n[nH]c(C)n3)C2)C1)NCC(C(=O)OC)(C)C c1(NC(C2C(Nc3ncc(C)cn3)C2)=O)cc(Br)ccc1I CC1CC(NC(=O)C(c2cccnc2)O)CN(C(=O)C=C(C2CC2)C2CC2)C1 N1(C(c2cc(COC)no2)=O)CC2CCCC2(CNC(C2(F)CC2(Cl)Cl)=O)C1 Cc1oc(C)c(S(=O)(=O)NCC(C)Oc2ccccc2Cl)c1C(=O)O N(C1CCCc2ccccc21)C(c1n(CCOCC)nnn1)c1occc1Br O=C1CC(C(=O)N2CCC3CC23C(=O)OCC)=NN1.c12ccccc1C2 c1(NC(c2ncn(C)c2)=O)cccnc1CN1CCCCC1C(N)=O c1(OCC)ccc(F)cc1NCc1ccc(F)c(OC)c1 C(=O)(C(O)CNC(C12CC(n3cc(CNS(N)(=O)=O)nn3)C1C2)=O)OC N1(C(C(C2(OC)CCOCC2)(F)F)=O)CC2(CCN2C(C2CC23CC3)=O)C1 c1(OC)ncc(CNC(=O)COC2CC(C)N(C(=O)OC(C)(C)C)C2)cc1Cl N1(C(C(CC=C)C)=O)CCCN(C(=O)C2=CC(C)(C)C2)C(C)C1 n1(CC(=O)NC2CCC(C)(CNC(=O)C=C3CCSCC3)C2)ccc([N+](=O)[O-])n1 C(c1c(Cl)cccc1Cl)=C(C(=O)NCCC(=C)CNC(=O)C(C)CC(F)F)C C1(NC(=O)CC2C=CCC2)C2CC1CN(C(=O)CCNC(c1cccs1)=O)C2 c1(NCc2onc(C(C)C)n2)cc(C2CCOCC2)ncn1 C1(CN(C)C(C2(C3CCCO3)CCC2)=O)CCCN1C(C1CC2CC2C1)=O CCCCC(O)CCC(=O)NCC1(CCNC(=O)C=Cc2ccncc2C)CC1 CCC(CC)(C(=O)NC(C1CCCC1)CNC(=O)Cc1nc[nH]n1)OC Cc1cc[nH]c(=N)c1C(N1CCCC(NC(C2CC2C(F)(F)F)=O)C1)=O N1(C(C2(C)C(C)(C)C2)=O)CCC2CN(C(=O)CCC3CCCO3)C2C1 C1(C)(CNC(C2C(C)(C)CO2)=O)CCN(C(C2(c3ccc(F)cn3)CC2)=O)C1 C1(F)(CNC(C(CC)NC(C)=O)=O)CCCN(C(=O)C(C)(C)c2ccno2)CC1 CCC(CC(=O)N(C1CCC(NC(C2(CO)CC(F)(F)C2)=O)CC1)C)SC C1(C(N(CCCCNC(c2coc(C3CC3)n2)=O)C)=O)CC2(CCOC2)C1 N1(C(C(C#C)(C)C)=O)CC2(CCC2NC(c2nc(Cl)ccc2OCC)=O)C1 C1(C(CNC(CCC2N(C)CCC2)=O)O)CCN(C(=O)Cc2cnnn2C)CC1 CCCCC(C(=O)NCC12CC(CN1C(C1COC(=O)N1C)=O)C2)C(C)C C1(OC)CC2(C1)CN(C(=O)C(CC1CC1)NC(=O)CC(C)(C)C)C2 C1(NC(C2(N(C)C)CCCC2)=O)COCCN(C(c2cc(O)ncc2F)=O)C1 N1(C(C(C)C2CC2)C(=O)NC2CCCCC2)CC2COCC2(C)C1 c1(C(N2CCCC(F)(CNC(=O)Cc3ccsn3)C2)=O)oc2ccccc2c1Cl c1(C(N(CCC(C)NC(c2cn(CC)nc2)=O)C)=O)nn(C)c(=O)cc1C N1(C(C)=O)CC2(C1)CN(C(C1CC3(CC3)CN1C(=O)Cc1nonc1C)=O)C2 C1(C(=O)NCC(C(=O)NC(C(C)n2cccn2)C)O)(CO)CCCCO1 c1(CC(=O)NC(CC)CNC(=O)Cn2cc(CO)nn2)noc(C)c1C#N Cc1nc2ccccc2cc1NC(=O)NC12CC(F)C1C2 C12(NC(=O)Cc3cccnc3)CCC(C1)N(C(=O)C(c1ccc(Cl)cc1)O)C2 c1(C(C(=O)NC2(C)CC2)N(C)CC2(OC)CCCC2)ccc2c(c1)CCC2 C1(C(=O)NC2(CNC(C(n3ncc(C)c3)C)=O)CCC2)CC1C1CCC1 C(=O)(C1CCc2cccc(O)c21)N(CC(CN(C(CCNC(=O)NC)=O)C)O)C C1(C(N2C3CC(CN(C(C4(CC)CC4)=O)C3)C2)=O)CC2CC1C1OC(C)(C)OC21 CC(C)CC(CN=c1cc[nH]cc1C#N)NC(C1CCCN1C(=O)C(C)(C)C)=O C1(C(=O)NC2CC(CNC(=O)C3=CCCOC3)C2)CCC2CCCCN12 N1(Cc2cccc(NC(N)=O)c2)CCCCC(NC(c2ccc(CF)cc2)=O)C1 C1(C(=O)NCC(C)CCO)CCCN(C(=O)CCN(C)CCO)CC1 C=C(C)C(C)(O)C(=O)NCCC1(O)CCN(C(=O)CCNc2ccccn2)CC1 c1(C(=O)OC(C(=O)OC)C2CCC2)c(I)cnn1C(C)C c1(C(N2CC(CNC(=O)CN3CCCC3)CC(C)C2)=O)ccc([N+](=O)[O-])nc1 C1(C(C(=O)NCCOC)N(CCS(C)(=O)=O)C)CCCC1C C=CC(C)(CC)C(=O)N1CC(O)(CNC(c2cc(-c3csc(CO)n3)c[nH]2)=O)C1 N1(C(C2CCCCO2)=O)CC2CCC1C1CN(CC3CCSCC3)CC21 CCCC(CCCNC(C1(c2ccccc2)CCOC1)=O)N=c1cc(C)nc(Cl)[nH]1 N1(C(CCn2ncc(C)c2)=O)CCN(C)CC1C(N1CC(CO)(CO)C1)=O c1(NC(C(CC#C)ONC(c2cc(O)cc(=O)o2)=O)=O)ccc2c(c1)OCO2 C1(N(C)C(c2nocc2Cl)=O)CCCCN(C(c2ccn(CC(F)(F)F)n2)=O)C1 c1(OC)ncc(F)cc1C(N1CCC(C)C(NC(=O)CC2(O)CCOCC2)C1)=O N1(CC(=O)NC(C2CCN(C(c3cc(CO)[nH]n3)=O)C2)C)CCCNC1=O c1(C(=O)NCC(C)(C)NC(C(C)OCC)=O)cc(S(N)(=O)=O)c(C)cc1C N1(C(=O)CCN2CCC2)CCC2CCN(C(=O)CC3CC(F)C3)C2C1 CCCC(CC)C(=O)N(CC(CC)NC(c1cc(NC(C)=O)ccc1C)=O)CC C(=O)(C(C)(F)C(=O)N(CCCNC(=O)CN1CCSCC1)CC1CCCC1)OC c1(CN(C2CCCC(NC(=O)OC(C)(C)C)C2)C)ccc([N+](=O)[O-])cc1 C1(O)(CN(C(c2cc(CCC)c(C)s2)=O)C)CCN(C(=O)C=CC(C)C)CC1 N1(CC)N=C(C(=O)N2CC(NC(=O)CCOc3ccc(F)c(Cl)c3)C2)CCC1=O CN1CC(O)CC1(C)C(N1CC2(CNC(C3CCC4CC34)=O)CC1CO2)=O C(c1ccc(Cl)cc1F)=CC(N1CC(CNC(c2ccc(Cl)c(O)c2)=O)C1)=O C(=O)(C(C(C)OC)NC(c1[nH]ccc1C)=O)N1C(C)(C(=O)NC)CC1 C=C(F)C1(CC(=O)NC2(C3CCCN3C(C3(S(N)(=O)=O)CC3)=O)CC2)CCC1 c1(CC(CC)C)nc(-c2cc(OC)nn2C)n(-c2ccccc2OC)n1 N1(C(CC(C)(C)OC)=O)CCN(C(=O)CC2CCC3CC23)C(CCO)C1 CC1=C(C(=O)N2CC(F)(CNC(c3cccc(C4CCCOC4)c3)=O)C2)CCC1 Cc1cc(C(=O)NC2CCN(CCCCCSc3ccccc3)C2)co1 Cc1cncc(C(=O)NC2CCN(C(c3ccnc(O)c3)=O)C2)c1 N1(C(C(C)N(C(CCc2cc(C)no2)=O)C)=O)CC2(COC(=O)C2)C1 N1(C(C2CC(OC)C2)=O)CCOC(C)(CNC(C2(Cl)CC2(C)C)=O)C1 CCCCCCC(=O)NCCC(C)NC(=O)C=Cc1cccn1C c1(OC)ccc(C(C)C(=O)NC(C)CCNC(c2ccsn2)=O)cc1OC N(C)(C(=NCC1CC1)NCC(=O)N(C)CC1CC1)CCOC.c1(O)ccccc1C c1(C(=O)NC2(C(=O)NCC3(OC)CCC3)CSC2)cn(C)cc1C C(N=c1cc[nH]cc1[N+](=O)[O-])C1COCCN(C(=O)CSc2ccccn2)C1 C1(NC(CC(=O)NCC)=O)C2CCC(C2)C1C(=O)N(CC(C)(O)C1CC1)C CC1CCN(C(=O)C(c2ccn(C)c2)C)C1C(=O)NCC1CNC(=O)CO1 C12(NC(C(CC)C)=O)CCC(NC(c3sccc3I)=O)(CC1)C2 N1(C(COCC(=C)C)=O)C2CCC1CN(C(C1(OC(C)=O)CC1)=O)C2 CC(C)(O)CCC(=O)NCC1=CCN(C(C2CSCC(=O)N2)=O)CC1 N1(CC(C)C)CCCN(C(c2cocc2Br)C(=O)NC(C)C)CC1 N1(C(c2c(C)nsc2)=O)CCN(C(c2cncc(F)c2C)=O)CC1CC(F)F CC1CN(C(C2CCCC(O)C2)=O)CC1CNC(C1(CCN(C)C)CC1)=O C1(c2ccccc2)(NC(=O)C(O)C2CCC2)CN(C(c2nc(C3CC3)cs2)=O)C1 c1(C(N2CC(C)C(CNC(=O)C(c3cscn3)N(C)C)C2)=O)cn2ccccc2n1 Cc1cccc(C(=O)NCc2cccc(C(=O)NC(c3ncnn3C)C)n2)c1O N1(C(CS(CC)=O)=O)CCC(C)C(CNC(=O)C(C)(C)c2nccs2)C1 c1(CC(=O)NC(C2CC2(F)F)CC)ccc(S(C)(=O)=O)c(C)c1 C12(CC)CCC(C(N3CCCC(CNC(c4cnccc4C)=O)C3)=O)(CC1)CO2 c1(NCC2C(C)(C)C2CO)cc(=NC2CCc3c(Cl)cccc32)[nH]c(C(F)(F)F)n1 c1(C(N2C(CNC(=O)CC3CN4CCN3CC4)C=CC2)=O)ccnc2ccsc12 C1(C(N2C(CC)C2)=O)CCC(C)CC1.c1(C(=O)N)nocc1C(C)C.C1(C)CCCC1 N1(C(C(C)NC(=O)NC)=O)CC2CCCC(CNC(=O)C(C)(C)CC(C)C)C2C1 c1(CC(=O)NCC(F)CNC(C2CC3CCC2CC3)=O)cccc2cnccc12 c1(CC(=O)NCC(C)NC(C2CC2(F)F)=O)nc2ccccc2s1 N1(C(CC(=C)Br)=O)CCN(C(c2ccc(N)c(O)c2)=O)CCC1C CCC(F)(F)C(C)(C)C(=O)N1CCC(CN(c2cc(C(=O)NC)ncn2)C)C1 c1(C(=O)NCC=CCNC(C=CCCC)=O)cccc(OC)c1 c1(OC(C)C)cccnc1CNC(C1CCC1c1ccccc1Cl)=O N1(C(c2nc(C#C)sc2)=O)CC2(C1)CN(C(=O)C(O)CC(N)=O)CC2CO C(=O)(CC(C(F)F)C(C)(C)C)NC(C(C)C)CNC(c1nsnc1O)=O C1(C(=O)NCC2N(C(CNC(CC)=O)=O)CC2)CCCN(c2cc(C)ncn2)C1 C(=O)(CC(C)(C)C(C)(F)F)NCC1C(C)CCN1C(c1cnccc1Cl)=O C(=O)(C(C)C(O)C(C)CC)NCC1(C(N2CCC(NC(=O)CC)C2)=O)CC(=C)C1 C1(CC)C(NC(c2cnc(C(F)(F)F)cn2)=O)CCN1C(C1CC1C(C)C)=O c1(SC)nc(O)c(C(=O)OC(c2ccc(F)cc2Cl)C)cc1C#N CC1=C(C)CC(C(=O)N(C2C3CN(C(c4ccc(O)nc4C)=O)CC23)C)CC1 c1(C(=O)NC(C(=O)NCC2C(OCC)CC2)C2CC2)cnc(Cl)s1 Cc1cc(C)n2ncc(C(N3CCC4(CC(NC(=O)C5=CCC5)CO4)C3)=O)c2n1 c1(C(=O)NC2C(C)CN(C(=O)C(O)C3CC3)C2)oc2ccccc2c1Br C(=O)(C1=NOC2(CCOC2)C1)N1CCC(NC(=O)CCOc2ccc(F)cc2)C1 c1(NC(C)Cc2ccco2)ccc(S(=O)(=O)NCCC2CCCN(C)C2)cc1Br Cc1ccc(C(N2CCCC(C3(C(F)(F)F)N=N3)C2)=O)cc1I c1(C(N(CCC(C)NC(=O)CNC(c2ccccc2)=O)C)=O)ccnc(Cl)c1O Cc1cc(COCC(=O)NCC2(F)CN(C(C34CCCC3C4)=O)C2)no1 c1(-n2cc(-c3c(C)con3)nn2)cccc(CCNC(C2CCS(=O)(=O)N2)=O)c1 S(=O)(=O)(CC(=O)N1CCCC1CCNC(C1CC(n2cnnc2)C1)=O)NC C(C(C(=O)NC(C)(C)C)N1CCC(CC2CCOCC2)C1)(C1CC1)OC c1(CC)nn(C)cc1C(=O)NCC1CC(NC(=O)Cn2nc(C)cc2C)C1 C1(CC)CN(Cc2csc(-c3sccc3Br)n2)CCC1CC(N)=O N1(C(C(CC)N(C(=O)CCc2ccsc2)C)=O)CC(C)C(O)C(C)C1 c1(C(c2nnnn2CC2CCCO2)NCC=C)cccc2ccncc12 C1(CNC(c2nc(CC)oc2)=O)CC2CCC1N2C(=O)CN1CCC1 O=C(C1=COCCC1)NC1CCN(C(c2ccc(Br)c(F)c2)=O)C1C1CC1 c1(C(N2CC(CC(C)NC(=O)CSCCOC)C2)=O)ccccc1SC(F)(F)F C1(C(N2CCCC(CN(C)C)C2)=O)CCCN(C(=O)C(C)(C)CNC(N)=O)CC1 C(=O)(CC(C(C)CC)NC(=O)C(C)(O)CCN(C)C)NCC1N(CCC)CCC1 C(=O)(CCCCCNC(C1CC2C=CC1C2)=O)NC(c1nnc(O)n1C)C N1(C(c2c(CC)ccs2)=O)CC(NC(=O)C2=CCCSC2)CC1(C)C C1(COC)(CNC(=O)CC2CC(SC)C2)CCN(C(C2(O)COC2)=O)CC1 C1(CNC(=O)NCC(=O)N(C)Cc2ccco2)COC2(CCC(C)CC2)O1 O=Cc1cccc(CN2CCOC(C(=O)NCCc3cccc(F)c3)C2)c1Br C1(NC(c2n(CC)ccn2)=O)CN(C(=O)CCn2nc(C)nc2C)CC2(CC2)C1 N1(C(c2cc(CSC)c(C)s2)=O)CC2CCN(C(=O)C(C)c3cncs3)CC2C1 c1(C(=O)NCC(CNC(C2(Cl)CC2(C)C)=O)OC)ccn2nccc2n1 c1(OC)ncccc1C(N1CCOC(CCCNC(c2coc(OC)n2)=O)C1)=O c1(OCC(=O)N(CCC(C)NC(CCC#C)=O)C)cc(C)ccc1Br N1(c2cc(C)nc(NC3CC4(C3)CC(C)C4)n2)CC2CCCC(C1)N2C C1(NC(C(C)OCCOC)=O)CN(C(c2c(C)cncc2F)=O)CCC1O C(=O)(C(C)(C)C1CCOC1)N(CCCC(=O)NC1CC(C(C)O)C1)C O=[N+]([O-])c1nn(-c2ccc(F)cc2)nc1CCc1cnc(O)nc1 C12(CNC(CC3N(C)C(=O)CC3)=O)CN(C(=O)COC(F)F)CC(F)(C1)C2 n1(CCC(=O)N(C(C)CNC(=O)C=Cc2cccs2)CC)ccnc1C C(=O)(C(C(C)(C)C)n1cc(CO)nn1)NC1CCCN(Cc2c(C)cncc2)C1 C1(C(C)=O)CCCN(C(=O)NC(C2CC=CCC2)c2noc(-c3cccs3)n2)C1 C1(CC(N2CC(C(=O)OC)(COC)C2)=O)CCCN(C(=O)CSS(C)(=O)=O)C1 c1(C(=O)NC2C(CNC(Cc3n(C)nnc3)=O)C2)nc(Br)sc1Cl c1(C(=O)NCC2CC(NC(C3N(CCC)CCC3)=O)C2)cnc(O)c(Br)c1 c1(CC(=O)N(CC(C)NC(=O)CNS(C)(=O)=O)CC)occc1C C(CN=c1[nH]c(=NCC(C)N2CCC(C)CC2)c2ccc(OC)cc2[nH]1)OC N1(C(C(C)(CO)OC)=O)CCOC2(CCC(NC(C3CCCCO3)=O)CC2)C1 C(CN=c1nc2sccc2c(NCC2CCCC2(F)F)[nH]1)(C1CCC1)OCC Cc1nc(C(N2CC3CC(N(C(=O)C(C)P(C)(C)=O)C)C2C3)=O)c(=O)[nH]c1C CC1(C)COC(C(=O)NC2(NC(c3ccc(F)cc3)CCO)CC2)C1 Cc1ccccc1-n1nnnc1C(C)C(=O)N(CCCN(c1ccc(Cl)cn1)C)C c1(CC)csc(C(c2nnnn2C(C)C(=O)OC)NCCCNC(N)=O)n1 c1(C(N(CCNC(C2CCC(=O)N2)=O)CC)=O)ncc(F)cc1C C1(O)(CC(=O)NCC2C(NC(C3(CC#N)COC3)=O)CCCC2)CCCCCC1 N1(C(C(F)=CCC)=O)C2CCC1CN(C(=O)C(=O)Nc1cnn(CC)c1)C2 C1(C(C)(C)NC(C2C(C)C2)=O)CCCN1C(c1ccoc1C(F)(F)F)=O C(=O)(C(C)(F)C(F)(F)F)NCC1CC(OC)CN1C(=O)C=Cc1ccncc1 Cc1ccc(C)c(N(C)C(C2CCN(C(c3cnc(C)nc3C)=O)C2)=O)c1 C1(NC(Cc2cnc(C)s2)=O)CCN(C(=O)C(O)CC(N)=O)C(C)C1 N1(C(C(CCCC)C)=O)CC2CCC1C1CN(c3ncnc4cc(C)[nH]c34)CC21 C(CC(C(=O)N1CC(NC(C)=O)C1)NC(c1cc(Cl)n[nH]1)=O)SC c1(NC(C2CN(C(C3CCN(C)CC3)=O)CC(F)C2)=O)cc(F)c(Cl)nc1Cl C1(NC(COCCCOC)=O)CC(CC(N2CC=C(C)CC2)=O)C1(C)C c1(SCCC)ccc(C(=O)NCC(C2CC2)NC(c2cn(C)nc2CC)=O)cc1 c1(SC)cccc(CC(=O)NC2CC(CCNC(=O)CSc3ccncc3)C2)c1 c1(C(=O)NC(C(=O)NC2(CCC)CC2)c2cccs2)c[nH]c(=N)o1 C1(n2cc(CNC(CC)=O)nn2)CCCN(C(=O)C(C)CN(C)C(C)=O)CC1 N1(C(CC2(C)CNC(=O)O2)=O)CCC2(CC1)CC2CNC(=O)CC1CC1 C1(COC)(NC(=O)Cc2cccc(NC(C)=O)c2)CCCN(C(=O)C(C)(C)C)C1 CCC(CCC(=O)NCCc1cc(CC)no1)NC(=O)C(C)C(C)(C)C C(CN=[N+]=[N-])(C(=O)N1CCC(C(N)=O)CC1)NC(C(C)N(C)C)=O CCC(CC(C)C)C(=O)NC1CN(C(=O)Cc2cccn2C)C1 C1(C(=O)NC(C)C)CCN(c2nnc(CC3CCCC3)n2CCCS(C)(=O)=O)CC1 Cc1cc(C(F)(F)F)ncc1C(N1CC(CC(C)NC(c2cccn2C)=O)C1)=O c1(NC(C(=O)N(n2cncn2)CCC)CC)cccc(Cl)c1Cl C1(NC(=O)CONC(c2n[nH]c(O)n2)=O)C(=O)OC2CCCC12 Cc1ncnc(C(N2CC(O)CC2CC(=O)N(C(C)CO)C)=O)c1C C(=O)(CC(O)C(C)CC)N1CC(CC=C)(C(=O)NCC(C)N=[N+]=[N-])C1 c1(CNC(C=CC2(C)COC2)=O)nnc2n1CCN(C(c1ccc(CO)o1)=O)C2 c1(C(=O)OC)sc(C(N2CC(O)CC2CNC(=O)C(F)n2ccnc2)=O)cc1C C(=O)(C#CC1CCCCO1)N1CC2C(NC(C(CC)C(C)C)=O)C2C1 Cc1ccc(C(=O)NC2CCCC2C(=O)NCCc2ccc(F)cc2)c(C)n1 CCCCCC(C)CC(=O)N1CCN(C(C2CCCOC2)=O)C(C2CCCC2)C1 N1(C(C=CCC)=O)CCCC(COC)(NC(C2(NC(N)=O)CCCCC2)=O)C1 C1(C(=O)NC2(CNC(C(C)c3ccco3)=O)CC2)COC(C)(C)CO1 c1(CCC(=O)NCC(C)NC(C(C)Cn2ccnc2)=O)ccccc1F C1(NC(CSCCOC)=O)CCC2(CCN(C(C3Cc4cccnc4C3)=O)C2)C1 c1(CNC(c2ccc(OCc3ccccc3)cc2)C(=O)NC)nnc2n1CCOC2 Cc1cc(N2CC(C)C(C)C2)ncc1S(=O)(=O)N1CCC(CN(C)C)CC1 c1(C(C)C)nccc(C(=O)NCCC2CSCCN2C(C2CCCC2O)=O)n1 C(=O)(C(C(C)(C)C)C1CCCO1)N1CCC(OC)(CNC(C2CC(O)C2)=O)C1 N1(C(C2(C(=O)OC)COC2)=O)CCN(C(=O)CN2CCS(=O)CC2)C(CF)C1 N#Cc1nc(=NC2CCN(c3ccccc3)C2=O)cc[nH]1 C(=O)(CC(C)(C)CC(=O)NC1CCN(C(=O)Cn2c(C)cc(C)nc2=O)C1)OC c1(C(N2CC(Cn3cc(C4(C)CCCC4)nn3)OCC2)=O)nccn2ccnc12 Cc1onc(CO)c1C(N1CC(NC(=O)CCCC#N)C(c2ccnn2C)C1)=O Cc1ccc(C(=O)NCC2CCCN2C(C2CC(=C(F)F)C2)=O)cc1O c1(C(N2C(C(C)NC(CCOCC(C)C)=O)CCCC2)=O)c[nH]c2ccncc12 Cc1cc(C(=O)NCc2cc(C(=O)N(C)CC3CCCCO3)n(C)n2)ncc1N C(=O)(C1=CNC2=NCCCC2=C1)NC1CC(NC(C2C3(CC(C)(C)C3)C2)=O)C1 CCC(C)(C(=O)NCC1CC(F)CN1C(c1cc(CN(C)C)c[nH]1)=O)C(F)F C#CCCCC(=O)N1CCOCC1CCNC(c1sc(NC2CC2)nc1C)=O Cc1nn(C)cc1S(=O)(=O)N1CC2CC2(CNC(c2ccc(F)nc2C)=O)C1 c1(C(=O)NC2(C)CC(NC(C3CN(CC(C)C)C(=O)C3)=O)C2)ccn2ccsc12 N1(C(c2c(C)nsc2)=O)CC2CCC1CC2NC(C1CC2CC2C1)=O Cc1c(C(F)(F)F)n[nH]c1C(=O)NC(Cc1cncnc1)C(=O)N(C)C CC1CC(C(=O)NCC(O)CCC2CC2)N1C(=O)COC1(C)CCC1 C1(CNC(=O)C=C(Cl)Cl)CN(C(=O)COc2cccc(F)c2)CCC1(F)F C(=O)(C(O)CC(N)=O)NC(C(C)C)CCNC(=O)Cc1cnc(C2CC2)[nH]1 N1(C(CC2CC(=O)NC2=O)=O)CC2CC1CN2C(c1ccccc1)=O c1(COC)nc(=NCC(C)N(C(=O)C(CC)NC(N)=O)C)s[nH]1 CCCC(C)CC(=O)NCCCC(C)NC(=O)Cc1c(C)nn(CC)c1C C1(CCNC(=O)C2=CCOC2)CN(C(c2cc(C3CCC3)on2)=O)CCS1(=O)=O c1(C(=O)NCC(CO)NC(C(c2n(C)cnc2)O)=O)scc2c1CCCC2 C1(CC(=O)NC(c2ccccc2Cl)COC)CCC2(CCC2)CO1 C=C(C)CCCC(=O)NC1(C)CCN(C(=O)C(C)N=[N+]=[N-])C1 c1(CC)nn(C)cc1C(=O)NCCCCN(C(=O)CCc1nc(O)n[nH]1)C C(=O)(CS(=O)(=O)CCOC)NC1CN(C(C2(C)CCN(C(C)=O)C2)=O)CC(C)C1 N1(C(C(=Cc2cccs2)C)=O)CC(NC(c2cnc[nH]c2=N)=O)CC1C c1(CN(C(C)C)Cc2ccc(OCCO)cc2)cncc(C(C)(C)C)c1 C(=O)(CCC(=O)c1cccnc1)NC(C)(CNC(=O)C=Cc1ncc[nH]1)CO c1(CC(C)C)ccccc1COC(=O)CSc1nnnn1C Cc1cnc(NC2CN(C3CCOCC3)C2)c(S(=O)(=O)N2C(C)CCC2C)c1 Cc1cnc(C(=O)Nc2cccc(NC(c3ccn(C)c3)=O)c2)nc1 N1(C(C(CC)=CC)=O)CC(NC(=O)CC2CCCC(C)C2)C2(CCOCC2)C1 c1(C(=O)NCCN2C(c3cccc(C)c3)C(=O)NCC2)cnn2c1OCC(O)C2 C1(C)(CNC(CN2CCN(C)CC2)=O)CCCN(C(c2cc(C#N)no2)=O)C1 c1(CC#N)cccc(NC(c2cccc(CCCc3ccccc3Cl)c2)=O)c1 c1(C(=O)NCC(C(C)(C)C)NC(C(CC)SC)=O)cc(N)ccc1C c1(CCC(=O)NC2C(NC(c3c(C)cno3)=O)CCOC2)cnc2n1CCOC2 C12(C(=O)NCCCCC=C)CC(CO1)N(C(=O)CC1CCOC1=O)C2 C1(C(N(CC(C)N(C(C)=O)C)C)=O)(NC(=O)CC2CCSC2)CCN(C)C1 N1(C(C(C)C2CC2)=O)CCC(C)(C)C1C(=O)NCC1CCCCC1(C)C CCC(C)C(C)C(=O)NCCCN(c1nc(Cl)ncc1C(N)=O)C C(CC(CO)N=c1cc(F)nc(C(C)(C)C)[nH]1)N(C)C c1(C(=O)NC2CC(CNC(=O)C=Cc3cc[nH]c3)C2)ccc(F)nc1F C123CC(CN1C2)C3.C1(CNC(N(C)Cc2ccccc2)=O)CCCC(N)C1 C(=O)(C(CC(C)C)N(C)C(C1CN(C(C)C)C1)=O)N1CCC(C(CC)C)CC1 c1(C(=O)NCCC(C)NC(c2cc(-c3ccoc3)[nH]n2)=O)cnc(N)c(N)c1 C1(CCNC(=O)CC(O)C2CCCC2)CCCN(C(=O)C(=O)NCC(F)F)CC1 C=CC(CC)CC(=O)NCC1COCC1NC(=O)CCN1CCC(N(C)C)CC1 c1(C(=O)NC(C2CC(F)(F)C2)C)n[nH]c2c1CN(C(c1c[nH]nc1C(F)F)=O)C2 N1(C(C(C)C(N)=O)C)CC(C(F)(F)F)C(F)(CO)C1 C1(C(C(=O)O)OC)CCN(C(c2cn(-c3ccc(C)cc3)nn2)=O)CC1 CC(CCC(C)(C)C)C(=O)NCCOCCCNC(c1cncc(C(F)F)c1)=O C(C1=NOC2CCCCC12)n1cc(C2N(C(C3(CC)CCCO3)=O)CCC2)nn1 c1(C(N(CCC(C)NC(c2ccc(C3CCCO3)[nH]2)=O)C)=O)csc(=N)[nH]1 c1(C(N2C(CNC(CN(CC)CC)=O)COCC2)=O)csc2nccn12 CCC(C)(C)C(=O)N(C(CNC(=O)CC1CCCC12CC2)C1CC1)C C(CCCC(CO)NC(=O)CC(C)CF)NC(c1c(C)c[nH]c1)=O N1(C(C(CC)C#N)=O)CCCC2(NC(C3CC4CC4C3)=O)CCCC12 c1(COCCC)ccc(C(N2CCC(C(C)C(=O)NC(C)CCC=C)C2)=O)cc1 C12(C(=O)NC3C(NC(CC4CN(C)C4)=O)COC3)CCC(=O)N1CCS2 C1(C(=O)NCCN(CCC)CC)(CNC(=O)Cc2cc(C)cs2)CCCO1 C(=O)(C1=CCS(=O)(=O)C1)N1CC(NC(=O)CSCc2ccc(Cl)cc2)C1 C#CCC(CC(=O)N1CC=CC(OC)C1)NC(c1cnn(C)c(=O)c1)=O c1(CSCCNC(C(C)(C)N2CCOCC2)=O)ccc(Cl)cc1 Cc1ncsc1COCC(=O)N(CCCCCNC(c1n[nH]cc1C(C)C)=O)C C1(C)(CC(=O)NCCOCCC=C)CCN(C(=O)CC2CCOC2)C1 CC1=CCC(C(=O)N(C2CCCC2)CCNC(c2cc(Br)n[nH]2)=O)CC1 C(=O)(C1COc2ccc(Cl)cc21)NC1C2OCC(NC(=O)CCC(F)F)C2OC1 Cc1cc(C(=O)NCC(O)CNC(=O)Cc2ccc(C(N)=O)nc2)oc1Br c1(OC)cc(C)c(C(N2CCC(CF)(NC(=O)CN=S(C)(C)=O)C2)=O)cn1 CC(C)CC(CCO)NC(=O)CN(C(=O)CCc1cnoc1)C N1(C(c2nc(OCC)sn2)=O)CCC(C2CN(C(c3ccoc3)=O)C2)CC1 C(=O)(C1=CCCCCC1)N1C(CC(=O)NCc2n(CC)ncc2)CCC1 C1(NC(C(C)(N(C(C(CC)OCC)=O)C)C2CC2)=O)CC(CO)C2CC12 CC(c1cccnc1)=CC(=O)NC(C)CNC(=O)C(c1ccc(N(C)C)cc1)C N1(C(C(C)(C)O)=O)CC2CCCC(CNC(C3CC34CCOCC4)=O)C2C1 C(=O)(CCCCN=[N+]=[N-])N1CCC(C(=O)NC2(C(=O)OC)CC2C)CC1 C(=O)(C(F)CC(C)(C)C)N1CCSCC(C)C1.C1(=O)C(CC(F)F)N1C C12(C(C)C)COC(C(=O)NCC3CCCCC3CNC(=O)Cc3cc[nH]n3)(C1)C2 c1(C(=O)NCC2CN(C(c3nn[nH]c3C(F)(F)F)=O)CCO2)cc(Cl)c(Cl)nc1Cl C=CC(C)(O)CCCC(C)C(=O)N1CCC(CCNC(=O)C(F)=CC2CC2)CC1 C1(F)(CNC(=O)CC=C(Cl)Cl)CCN(C(=O)Cc2cccnc2)CC1 c1(C(=O)NCC2C3CN(C(C4(C)CC4(F)F)=O)CC32)[nH]nc2ncnc(O)c12 C(CNC(=O)Cc1nocc1C)(CC(=O)N(C)Cc1csc(C)n1)OC CC1C(C=CC(=O)NCCCOCCNC(C2(C)CCCOC2)=O)C1(Cl)Cl N1(C(C=Cc2ncn(C)c2)=O)CC2(CCN(Cc3ccc(Cl)cc3F)CC2)C1 N1(C(C=C(C)Cl)=O)CC2CCN(C(=O)CCOc3ccccc3)C2C1 Cc1sc(=NC2CCOC3(CCC3)C2)[nH]c1-c1ccc(Cl)cc1 N1(C(C(CC#C)C2CC2)=O)CCN(C(c2cc3occc3[nH]2)=O)CC1C1CCC1 c1(C(N(CCNC(C(CC=C)CC)=O)CC)=O)ncnc2c1cnn2C Cc1cn2c(n1)C(C)CC(C(N1CC(NC(=O)C(C)(C)F)C1)=O)C2 c1(CCNC(CC)(C(=O)N(C)C)c2ccccc2)ccc(SC(C)C)nc1C C1(OC)CC(CNC(c2occc2C)=O)N(C(=O)CC2(C)CCOCC2)C1 Cc1cc(C(=O)NCC2(O)CCN(C(=O)C=Cc3cn(C)cn3)C2)c(C)s1 c1(C(=O)NC2CCN(C(CCCOCC=C)=O)CC2F)nnc2n1CCCC2 C1(C(=O)NCC2(OC)CN(C(Cc3ccc(OC)s3)=O)C2)COCC(C)(C)O1 c1(C(=O)NC2C(NC(CC=CC=C)=O)C2)cc(N2CCNC2=O)ccc1F Cc1ccc(=O)n(CC(N2CCCC(N(C)C(c3ccncc3O)=O)C2)=O)c1 c1(C(C)(C)C)cccc(N(C(C2CC2c2ccccc2)=O)Cc2cccs2)c1 C(=O)(CS(=O)(=O)CC(F)(F)F)N1CCC(OC)(CNC(C2CCC2CF)=O)CC1 Cc1nc2[nH]ccc2c(=NCC(C)(C)NC(C2CCCCN2CC(F)F)=O)[nH]1 N1(C(C2C(C)(C)C2)=O)CC(CNC(=O)CNc2ccccc2C(F)F)CC1(C)C CCCC(C(=O)N1CCN(C(c2c[nH]c(C#N)c2C)=O)CC1CC(F)F)C(C)C Cc1sc(C(=O)NC(C2CCN(C(=O)COC(C)C)C2)C)cc1Br C(=O)(C(=O)C(C)C)N1CC(CC(=O)N(CC(F)F)CCO)(OC)C1 CC1CN(C(C2CC2C)=O)CC1NC(C1(c2ccc(Cl)nc2)CCC1)=O N12CC3(CCC3)CC1C2=O.c1(CC)c[nH]cc1C(N1CCC(C(C)(C)OC)C1)=O N1(C(CCCCC=C)=O)CCC2(CCCN(C(=O)CC3CCCN3C(C)=O)C2)C1 C1(CC)CCCN(CC(=O)NCC2(CN(C)C(C3C(Cl)(Cl)C34CC4)=O)CC2)C1 N1(C(C(CC(C)C)O)=O)CCCN(C(C2CCCN2C(=O)C(F)(F)F)=O)CC1C S(=O)(=O)(c1ccc(N2CCC=C(C)C2)c(F)c1)NC(c1ncc(C)s1)CC CCC1=C(C(=O)NCC2=CCN(C(c3cccc4cc[nH]c34)=O)CC2)CCCO1 c1(C(N(CC(CN(C(C(C)SCC)=O)C)O)C)=O)ccc(Cl)cc1Br C1(NC(CC2CC(C)C2)=O)CCCN(C(c2ccsc2)=O)C1C C1(F)(C(=O)NCC(C2CCN(C(c3ncsc3C3CC3)=O)CC2)F)CCCCCC1 c1(C(N2CCN(C(CCNC(=O)NC)=O)CC2CF)=O)nn(C)c2ccccc12 N1(CC(=O)NC2CN(C(Cc3scc(C(=O)OC)c3)=O)C2)C(=O)CN(C)C1=O Cc1oncc1S(=O)(=O)NC12CC(C(C)(C)O)(C1)C2.N12CCC(CC1)C2=O C12(C(=O)N)C3C4C1C1C2C3C41C(F)F.c1(SC)ccc(-c2cccc(CO)c2)cc1 c1(OC)cc(O)c(C(=O)NCC2(O)CCN(C(=O)C3CC3)C2)cc1Br c1(CNC(C2(C(F)F)CCNC2)=O)cnn2ccccc12 c1(C(N(CCOC)CCNC(=O)Cc2csc(C)c2)=O)ccc(Br)cn1 c1(C(N2CCC(N(C=O)Cc3ccc(OCC)cc3C)C2)=O)ccc2cc[nH]c2n1 c1(C(=O)NC(C(=O)NCC2(CO)C(C)(C)C2)C2CCCC2)ccc(=N)[nH]c1 CCCC(CCCNC(c1cnc(O)cc1C)=O)NC(c1c[nH]nc1F)=O c1(CCC)n[nH]cc1C(=O)NC1CC1NC(c1coc(C2CCCCC2)n1)=O CCC(CC(=O)NC(CNC(c1nnn(C)c1C(F)(F)F)=O)CO)C(F)F N1(C(Cc2cnc(C)s2)=O)CCC(F)(C(=O)NCC2(O)CCCOC2)C1 C(=O)(CC(O)C(C)C)NCCN(C1CCCCC1)C(c1c(C#C)c[nH]n1)=O c1(C(NNC(COc2cccc(C(N)=O)c2)=O)=O)ccc2c(c1)OCO2 Cc1ccc2sc(N3CC4(CCC4)CC3CNC(=O)C3=CCCCC3)nc2c1C c1(C(N2CCN(C(C3CCCCCC3)=O)C3CC23)=O)cc2cccc(Cl)c2[nH]1 C1(N(C(=O)COCCN(C)C)C)CCC(NC(c2cn(C(C)(C)C)cn2)=O)CC1 C(C)(CC(F)(F)F)NC(CCCNC(C1(OC)CCSC1)=O)=O C1(C)(NC(c2n(CC)ccn2)=O)CCCN(C(c2ccc(OC)c(N)n2)=O)C1 C1(CNC(C(C)OCC)=O)CC2CC2N1C(c1ccnn1Cc1ccccc1)=O C=C(C)CC(C)C(=O)N1CCC(C(C)NC(c2cscc2SC)=O)C1 Cc1nc([N+](=O)[O-])cn1CC(N1CC2C(N(C)C(C3CC(F)CN3C)=O)C2C1)=O C1(CNC(C(C)S(C)(=O)=O)=O)CC12CCN(C(=O)C=Cc1ccccc1)CC2 C1(N(C(=O)CCCc2cccs2)C)CCC(NC(C2CCC2(F)F)=O)CC1 C(=O)(CCCCN(C)C)NCCN(C(c1ccc(C(=O)OC)o1)=O)CC C1(COC(c2ccc(NC3COC3)nc2)=O)OCC2CC(=O)C1C2 c1(NC(C2(COC)N(C(CCCC)=O)CC=C2)=O)ccc(C2CC2)nc1C c1(C(=O)NC(CC(=O)OC)C)cccnc1-c1cscc1C CCC(N=c1ccnc(NCc2ccccc2-c2cccnc2)[nH]1)C1CCCO1 c1(NC(C)=O)cc(Br)ccc1C(=O)Nc1cccnc1C(=O)N(CC(F)F)C C(C(C)(C)C#CC(=O)NC(CCO)c1ccco1)NC(C1CCN(C)C1=O)=O c1(C(N(C)CC2COCCN2C(C2COCCO2)=O)=O)cc2cn[nH]c2cn1 C1(C(=O)NCC2(CO)CCCO2)CCCCC1NC(C1CCCC1O)=O c1(C(N2CC(C)(NC(c3c(CC)ncs3)=O)C2)=O)cc(F)cc2nc[nH]c12 c1(C(=O)NCCC(=O)Nc2cccc(C3CC3)c2)cn2c(n1)CCC2 N(C1CCc2ccc(Cl)cc21)C(C1CN(S(CCC(=O)OC)(=O)=O)CC(F)C1)=O N1(C(c2cc(C)n(C(F)F)n2)=O)CC(NC(c2cccc(Cl)c2N)=O)CC(O)C1 c1(CC)onc(C)c1NC(c1ccn(CCNC(=O)CCN(C)C)c1)=O C12(CNC(c3c(Cl)cccc3Cl)=O)CCC(CC1)CN2C(=O)Cc1cnccn1 CC1=NOC2(C1)CC(C(=O)NC1(CNC(c3cc(F)c(Cl)c(N)c3Cl)=O)CC1)C2 C(=O)(C(O)CC(F)F)N(C)C(c1ccc(Cl)cc1)c1ncc[nH]1 C1(O)(CNC(C2(CC)CCC2)=O)CCCN(C(C2CN(C)C(=O)CCO2)=O)CC1 c1(C(N(C2CC3(C2)CN(CC)C3)C2(F)CCCN(C)C2)=O)cc(F)c(F)cc1Cl C1(C(N(C2C(C)CCC2)C)=O)CC(O)CN1C(C1CC(F)C1)=O N1(C(C2CCC(C)CC2)=O)CCCC12CCN(C(=O)C1=COCC1)C2 C1(C(N2CC(N(C(=O)C(=O)NCC(F)F)C)C2)=O)CN2CCC1(C)C2 c1(C(=O)NCc2cc(C(N3C(COC)CCCC3)=O)ncc2)cnccc1C#N C1(C(=O)NC23CC(CNC(C(C)OCCOC)=O)(OC2)C3)CCOCC12CCC2 N1(C(c2cc(C)ns2)=O)CCCC12CCN(C(=O)Cc1ccc(F)cn1)CC2 C=CC(CCC)CC(=O)NC1(C(N2CC(O)(CCC)C2)=O)CC1(C)C C1(C)(C)CCCO1.C(C(=O)N(CC(=O)NC)C)OC.C12(CC1)C(=O)N2 C1(C(C)O)CCN(C(=O)CCC2(C)CN(C(=O)C(C)(C)n3cccn3)C2)C1 c1(CSCC(=O)NCc2ncoc2C(F)(F)F)ccc(Cl)s1 N1(C(c2c(C)csc2)=O)CCCN(C(C2CCCC(C(N)=O)C2)=O)CCC1 C12(CNC(CCC#CC)=O)CC(NC(=O)C(O)C=CC)(CCO1)C2 C(=O)(C(=O)C(C)(C)C)NC1(C(=O)NC(c2cnccn2)C)CC(F)C1 c1(OC)cccc2cc(CNCC(C)(C)C3CCCO3)oc12 N1(C(C2N(CC)CCC2)=O)CC(F)(F)CC1CNC(C1CCCN1)=O C(=O)(C1=CCCOC1)N(CCNC(C12CC(CF)(CO1)C2)=O)CC1CC1 c1(-c2ccn(CC(C)C)n2)cccc(C(=O)NC2(C)CCCC2C)c1 C(C)(CC(=O)NCCCCN(C)C1CC1)NC(C(N1CCNC1=O)C)=O c1(NC(C2CC3CC3N2C(c2ccc(O)nc2)=O)=O)cccc([N+](=O)[O-])c1Br C1(CC(=O)NC(CC=C)CNC(c2ccc(Cl)cc2N)=O)COCC(C)(C)O1 c1(C(=O)NC2CCC(CNC(CC3CC(CC)C3)=O)C2)cccn2c(C)cnc12 c1(C(=O)NC2C(CNC(CCCOC(C)C)=O)CC2)cn2c(n1)SCC2 Cc1ccc(O)cc1C(N1CCC(C(C)CNC(=O)CO)CC1)=O c1(C(=O)NC(C2CCN(C(CC3C(C)OCC3)=O)C2)C)cnn(C)c1C(F)F Cn1nc(C(F)F)cc1CSC1CCC(C(=O)NCc2ncccn2)CC1 c1(C(=O)NC(C2CCN(C3CCN(C)C3=O)CC2)C)cc(F)cc(F)c1 C1(NC(CC(C=C)C)=O)CCC2(CCN(C(C3CC(C)CCO3)=O)C2)C1 C1(C(=O)NC(C2CN(C(Cc3c(C)n(C)nc3)=O)C2)C)CC12CCSCC2 N1(C(C(c2ccc(Cl)cc2)C)=O)CCC2(CC1)OCCC2NC(=O)CC(F)(F)F c1(NCC(C)NC(=O)OC(C)(C)C)cc(N(C)CC2CCCCN2C)ncn1 C1(NC(C2C(C(=O)N(c3cc(O)n[nH]3)C)C2)=O)Cc2ccc(Br)cc2C1.C=O.CCO N1(C(c2c(C)ccs2)=O)CCN(C(=O)Cc2ccc3c(c2)OCO3)CC(CO)C1 c1(-c2nc(NC(C3(OC)CCC3)=O)sc2C)ccc([N+](=O)[O-])cc1F Cc1c(C(N2CCN(C(C3(C(=O)C4CC4)CC3)=O)CC2CCO)=O)cncc1Cl C12(NC(COC)=O)CC1CN(C(=O)C(C)Cn1cccn1)C2 C1(C(C)NC(C=COCC)=O)CCCN(C(c2cc(C(C)(C)C)[nH]c2C)=O)C1 C(CN=c1[nH]c(C2CC2)nc(=N)[nH]1)OCCNC(C1CC2(CC(C#C)C2)C1)=O N1(C(C2C3(CC(NC(CC(C)SC)=O)C3)C2)=O)CC(F)(F)CC1C CCCCCCC(C)C(=O)NCC(C(C)C)NC(=O)CC(C)CC(=O)OC c1(C(=O)NCC(=C)CCNC(=O)C(CCC)OCC)ccc2ncccc2c1F Cc1cccnc1CC(N)C(=O)NC1CCCN(c2ccccc2)C1 C1(C(=O)NC(CN(C(=O)C=C2CCC2)C)(C)C)CS(=O)(=O)CCO1 CCC(CC)CCC(=O)NCC(CC1CCCC1)C(=O)NCCC1CCN(C)C1 C1(CNC(C2CC=C(C)CC2)=O)CCN(Cc2ccc3nonc3c2)CC1(F)F c1(SC)nc2ncnc(N3CCCC(C(C)NC(=O)C(C)C)C3)c2s1 C1(C(=O)NC2CC(C)(NC(C(C(C)C)OC)=O)C2)CCOCC12CCCCC2 C(=O)(CC(C)(C(F)(F)F)N(C)C)N1CCC(NC(C(C(C)C)CN(C)C)=O)CC1 C1(CNC(c2ccc(CC)cc2)=O)CCN(C(=O)CCCc2ncco2)CC1C c1(CN2CCC(CNC(Cc3ccc(C)cc3)=O)C2)ccc(N(C)C)c(Br)c1 c1(OC)cccc(CN(C)C(C2(O)CCN(C(C)(C)C)C2)=O)c1OC c1(CC(C)C(=O)NCCc2ccn(C)n2)cccc(O)c1 C1(C2CCNCC2)(C(=O)NCCC(CCCC(C)C)C)CCOCC1 C12(C(=O)NC(C(C)SC)C)CCC(CC1NC(=O)CC1(C)CC1)C2 N1(C(c2cnc(OCC)s2)=O)CC2CC3CC2C1C3NC(C1CC(F)(F)C1)=O c1(OC)ccc2c(c1)CCCC2C(=O)N1C2CCC1C(CNC(=O)C(C)(C)C)C2 c1(C(N2CCCC(N(C(C3C(C=C)C3)=O)CC)C2)=O)cc(O)nc(O)c1 c1(C(F)F)nc(C2Cc3ccccc32)n(-c2ccc(Cl)cc2Cl)n1 N1(C(C2(CC=C)CC2)=O)CCN(C2CCCN(C(=O)C(C)COCC)C2)C(=O)C1 N1(C(c2ccccc2N2CCC(O)CC2)=O)CCNCC1c1ccccn1 CN(C(=O)C1CCOC1c1ccccc1)N1CCS(=O)(=O)CC1 C1(C(N2CCC(N(C(c3c(C)cc(C)s3)=O)C)C2)=O)CCCCS1(=O)=O CC1CCN(C(=O)C(=Cc2cnn(C)c2)Cl)CCN1C(C1CCN(C)C(=O)C1)=O N1(C(c2c(CC)n(CC)nc2)=O)CCC(C)C(N(C(=O)CN2CC(F)(F)C2)C)C1 CCC(CC(=O)NCCN(C(=O)CC(C)COC)CCc1ccccc1)C(C)C CCC(CC)C(C)C(=O)NCC1CC2CCC1N2C(=O)C(C)(C)CO c1(C(=O)NC(C)CCNC(=O)C(C)NC(c2ccco2)=O)ccn2c1CCC2 CCCCC(F)(F)C(=O)N1CCC(NC(c2ccnn2COC)=O)C(CC)C1 N1(C(c2cc(C(C)(C)C)n[nH]2)C(=O)NCCOC)CCC2CC12C Cc1cc(C(=O)NC(C)C(C)NC(=O)CCc2cccnc2C)c(C)cc1Cl C1(C(=O)NCC(CCC)(C)C)CNC(=O)CN1C(=O)C(COC)N(C)C c1(C(N(CC(C)N(C(=O)C=CI)C)C)=O)ccsc1C(F)F CC(C)C(C(c1ccccc1)NC(=O)CSC1CC1)NC(=O)C=Cc1ccsc1 C(=O)(C(C)(C)CC(C)C)NC(CNC(c1c(C)ccnc1C)=O)CC(C)C C1(CC(=O)NCCCCC(C)NC(c2n[nH]c3c2CCC3)=O)CCC2(CC1)CC2 c1(CNC(C(C2CCC2)NC(CCOCCOC)=O)=O)ccc(Cl)cn1 C1(NC(CCCCC)=O)CC2CC1CN2C(c1cn(C)nc1C(F)(F)F)=O c1(C(=O)NCC=CCNC(C2CC(CC)C2)=O)ccc2nc(C)cn2c1 C1(C(=O)NC(CC(=O)NC(C)C)C)CC2CCC(C1)N2C(=O)C(F)C(C)(C)O C1(NC(N(C)C(C2C(C(=O)OC(C)(C)C)C2(C)C)C)=O)CCC(=O)N1 C#CCCC(C(=O)N1CCCC(C)(N(C)C)C1)NC(=O)CCc1ccnn1C O=C(CC(Cc1cccs1)Nc1ccncn1)N1CC2CCC1C2 c1(C(=O)NCC(CC(C)C)NC(=O)CC2CCCN2C)[nH]nc2ncccc12 c1(C(N2CCCC(CN(C)C(c3cc(CO)on3)=O)C2)=O)ccc(N)cc1Cl C(C(CC(C)C)NC(C1CC=CCC1C)=O)NC(C(CC1CC1)OC)=O C1(C(N2CCC3(CCN(C(COCC)=O)C3)C2)=O)Cc2ccc(Cl)cc2C(=O)O1 c1(C(=O)NC(CC)CN(C(C2(CC)CNC(=O)C2)=O)CC)ncc(N)nc1C c1(CN2CCC(CC(N3CC4=CC(=O)SC4CC3)=O)C2)ccc2ccccc2n1 N1(C(CN(C2CCC2)C)=O)CCC(NC(=O)CC2CCC(O)C2)C1C C1(NC(C2=NOC(C)(C)C2)=O)CCOC2(CCN(C(=O)C=CC3CCC3)CC2)C1 c1(C(N2C3C(CNC(C4CCC(C)C4)=O)C(C3)C2)=O)ccc2c(n1)NCC(=O)N2 CC1CCC(CC(=O)NCC2CN(C(=O)COC3CCOCC3)C2)C1 CC(C(C)(C)C)=CC(=O)NCC1OCCC1C(=O)NCCCCN1CCC1 C(=O)(C(F)C(F)(F)C(F)(F)F)NC1C(CNC(=O)CSCc2cscn2)C1 C(=O)(C(C)(F)C(=O)NCC1(C(=O)N)CC1)NC(CCOC)C.C1(C(=O)NC)CCC1 C#Cc1cnc(C(=O)NCCCCC(N2CCSC3CCCC23)=O)c(C)c1 c1(OC)cc(CC(=O)NC2CC2NC(c2cc(N)ccn2)=O)ccc1Br n1(CC(C(=O)NCC(C)(C)NC(CC(COC)C)=O)(C)O)ccc(C)cc1=O c1(C(N2CC(CNC(C(C)(F)F)=O)OCCC2)=O)nc2cccnc2s1 C1(NC(c2c(C)con2)=O)CCN(C(c2ccc(-c3ccccn3)o2)=O)CC1O N1(C(COc2cn(C)nc2)=O)CC2CC1CN2CC(=O)Nc1nc(C(F)F)no1 N1(C(C(CC)CCOC)=O)CCC2CN(C(c3cccc4c[nH]nc34)=O)CC12 c1(OCC(=O)NC(c2ccc(I)cc2)C)cccc(C#N)c1.C(CN(C)C)N C12(C(=O)NC(CC(C)NC(CCc3cc(C)n(C)n3)=O)C)CCCCC1C2(F)F CN1CCC(C(=O)NC2C3CCCC23)(NC(C2CCC2(F)F)=O)C1 Cc1noc(C(C)NC(=O)C(C)NC(C)(C)C)n1 c1(CC)cccc(C(=O)NC(C)CN(C)C(C2CC(=O)N(C(C)C)C2)=O)n1 CS(=O)(=O)CCCC(=O)NC1CCN(C(C2C3CC4C(C3=O)C24)=O)C12CCC2 c1(CC(=O)N(C(C)CNC(=O)CS(=O)CC)CC)ccc(C)cc1Cl C=CC1(C(=O)NC(CC(C)C)C(=O)OC)CCN(C(C2CN(C(C)C)C2)=O)C1 c1(C(N(C(C)CN(C(=O)CC(C)c2ccncc2)C)C)=O)cc(O)nn1C c1(C(N2CCOC(C3CCOCC3)C2)=O)cccc2ccsc12 N1(C(=O)Cc2cc[nH]n2)CCC2(CCCN2C(=O)CCCC2CCC2)C1 C1(CO)C(C)N=C2N=c3ncn(C)c3=C(N2)N1.C(CCOC(=N)O)SC c1(C(N(CC)Cc2cn(-c3ccc(C)c(Cl)c3)nn2)=O)cncc2ccccc12 C(=O)(C(F)CCC(C)(C)C)N1CC(F)CC(NC(C2CCCC(C)CC2)=O)C1 N1(CCCC(=O)Nc2c[nH]c3ccccc23)CCC2(O)CCCCC2(O)C1 C1(C(=O)NC(C2CCC2)C2CC2)CCN(C(c2cc(Br)ccc2F)=O)CC1O N1(C(C=CC=CC)=O)CCC(C(=O)N(C2CC2C)C)C1C C=CC(C)(C)CC(=O)NC(C(C)NC(=O)C=Cc1cscn1)C(C)C C(=O)(C1=CC2CC(C1)CC2O)NCC1(OC)CCC1.c12nc(cs1)CC(=O)NC2 N1(C(C2(C(=O)NC)CCC2)=O)CC2(CCN(C(C3CC4CC4C3)=O)C2)C1 Cc1nn(-c2ccccc2)c(Cl)c1NC(C1CCCN1C(c1cccs1)=O)=O c1(C(=O)NC(C2N(C(CCNC(COC)=O)=O)CCC2)C)ccc2cc[nH]c2n1 Cc1c(C(=O)NC23CCN(C(=O)C(C)N4CCCC4)CC2C3)sc2ccccc12 C1(SC)CCN(CC2CC3COCC23)CC1 C1(N(CC)CC)CCN(C(C2CC2)=O)C1.C1C(=O)NCCSC1 C(=O)(CC1=NN(C)C(=O)C1)NCCNC(c1c(Br)ccc(C)c1)=O N1(C(CCC2C(C)(C)C2)=O)CC(F)CC1CNC(C1CCC(C)CC1)=O c1(C(=O)NCCN(C(c2cn(C3CCOC3)nc2C)=O)CC)cccc(O)c1 c1(C(=O)NCCN(C(C23CCC(C2)C3)=O)CC)cccc(CS(C)=O)c1 Cc1c(NC(c2c(Br)cnn2C)C)ncnc1NC(c1ncc(F)cc1F)C C1(N(C(Cc2cc(CC)nn2C)=O)C)CCCN(C(C2CCC(C)(C)C2)=O)CC1 C=C(C)CCCC(=O)N1CC(C2CN(C(=O)C(C3CCOCC3)C)CCO2)C1 N1(C(CCC2CCCN(C)C2)=O)CCC2(NC(C3CC4CCCC34)=O)CCCC12 C12(NC(CSCC)=O)CCCC(NC(c3cc(C)c(C)cn3)=O)(C1)C2 Cc1cscc1C(N1CCC(CN=[N+]=[N-])C1)C(=O)NCc1cccs1 N1(C(C(Cn2cncn2)NC(COCC=C)=O)=O)CC(C2(C)CC2)C1 c1(CCC)nc(C(=O)NCC2(CNC(=O)COc3ccccc3)CCC2)co1 N1(C(Cc2cccc(C)c2C)=O)CCC(NC(C2(CCO)CC2)=O)C(CO)CC1 Cc1occc1CC(=O)N(C)CC1CCCN1C(C1(c2cc[nH]n2)CCC1)=O C(C(CC(F)(F)F)NC(C1(C)CC(C(F)(F)F)C1)=O)NC(C(CC)SC)=O N1(C(c2cc(C)sn2)=O)CCC(C(=O)NCC2C=CCOC2)CC1 c1(OCCOC)ccc(NC(C2CC2C(=O)OC(C)=O)=O)cc1Cl.C(C)(C)C N1(C(C2CC(SC)C2)=O)C2CCC1CC(CCNC(=O)C=CC1CCOC1)C2 c1(C(C(=O)NC(CO)C(C)NC(c2ccc(C(C)C)o2)=O)OC)ccccc1Cl N#Cc1ccc(S(=O)(=O)NCC2CC(F)(F)CO2)cc1NCc1ncoc1C1CC1 C1(NC(CCSC)=O)CC(O)CN(C(=O)COc2c(F)cccc2F)C1 C1(CNC(C(CCC)=CCC)=O)CCCC2CN(C(C3(C)C=CCCC3)=O)CC12 N12CCC(CC1)NC(=O)C2C.c1(C(N2CCCCC2)=O)cc(C(N)=O)c[nH]1 c1(C(N(CCN(C(=O)CC2CCOC2)C)C)=O)cc(-c2ccn(C)n2)on1 C12(C(N3CC(CC=C)(C(=O)NC4CC(=O)NC(=O)C4)C3)=O)CCC(N=[N+]=[N-])C1C2 C(=O)(CCCC1CCOCC1)N(CC(CNC(CCOCC)=O)O)C c1(C(=O)NCC2CCN(C(=O)C3=C(Cl)CCOC3)C2)ccc2nc(O)[nH]c2c1F N1(C(CC(=C)C)=O)CCC(C2CCN(C(c3cc(C(=O)OC)no3)=O)CC2)C1 C(C(=O)NC(C1CCN(C(C2CC(OC)C2)=O)C1)C)(C(C)C)NC(C(C)C)=O C1(C(=O)NCCN2CCOC2=O)CC2COC(CCO)CN2C1 C1(NC(C2(C(C)C)C(C(=O)OC)C2)=O)CCCN(C(=O)CC2CCOCC2)CC1 N1(C(CCCC=C)=O)CCC2CN(C(C3CCCC(=O)N3)=O)CC12 c1(C(=O)NC2C(OC)CN(C(c3ccc(Cl)cc3F)=O)C2)ccc2n[nH]cc2n1 c1(-c2cc(C(=O)NCCCN(C(=O)CO)C3CC3)sc2)ccc(F)cc1 c1(C(=O)NCC(C)N(C(CC(CC)(F)F)=O)C)c(Cl)c2ccccc2n1C C1(CCC)CN(C(=O)C(C)c2ccco2)CCN1C(c1scc(C)c1Cl)=O N1(C(c2cncc(C)c2)C(=O)NC2CCC2)CC(C)N(S(C)(=O)=O)C(C)C1 c1(C(N2CCCC(NC(=O)CCn3ccccc3=O)C2)=O)n[nH]c2c1CCC2 c1(OC(C(=O)N(CCNC(CCC)=O)CCOC)C)ccc(Cl)c(C)c1 c1(NC(=O)NCCN2CC(C)(O)C2)nnc2n1CCCCC2 Cn1cc(C(=O)CN2CC(CC(c3ccn(C4CCC4)n3)OCC3CC3)C2)cn1 N1(CCC2=CC(C)(c3c(OCC)cccc3)C2)CCCC(C)(C(=O)O)C1 C1(NC(c2ncc(C)s2)=O)CCCN(C(c2n[nH]c(C3CC3)c2C)=O)C1 N1(C(CCC2CCC(=O)N2)=O)CCC(C2CN(C(C3(F)CCOCC3)=O)C2)CC1 CC1CC(N=c2ccn3c(Br)cnc3[nH]2)CCN1C(=O)CN1CCCCS1(=O)=O c1(C(=O)NC2CCN(C(C3(C)CCCCO3)=O)C2)cc(N)ccc1Cl Cc1ccc(NC(=O)CC2CN(Cc3ncc(Cl)s3)C2)c(C)c1C c1(C(N2CC(CCC=C)(C(N3CC(C(=O)N(C)C)C3)=O)C2)=O)cncnc1C c1(-c2nc(NS(Cc3cn(C(C)(C)C)nc3)(=O)=O)on2)ccccc1C(F)(F)F CC(C)C(O)C(C)C(=O)N(CC(=O)N(C)C)C1CCC1.c12nc(co1)C(=O)N2 c1(C(=O)NC2C(C(=O)Nc3c(OC)nc(Cl)cn3)C2)cc(F)c(F)cc1C c1(CO)cc2cccc(NCC3CC4CCC3C4)c2s1 c1(OC)c(C)cc(C(N2CCCCC2c2cn(C3CCCC(C)C3)nn2)=O)cc1C N1(C(C(C2CC2)SC)=O)CCOC(C)(CNC(c2nnc(O)nc2O)=O)C1 C1(F)(C(=O)NC(C)(C)C(=O)NO)CCCN(C(C2CCOC(C)(C)C2)=O)C1 c1(C(=O)NC(CC)CNC(=O)C(C)CCOC)cc(C#N)ccc1Cl CC(C)CC(CN=c1cc(Cl)nc[nH]1)NC(=O)C(F)(F)C1(O)CCCC1 C1(CC)CC(C(=O)NC2(CNC(=O)COCCCCCC)CCOC2)CCO1 N1(C(COCCC(C)C)=O)CC2(NC(=O)CC3CCN(C)C3=O)CCC1C2 C1(C(N2CC(CNC(CCc3ncc(C)[nH]3)=O)C(C)C2)=O)CCc2n[nH]cc2C1 C1(NC(c2c(C)n(-c3cccc(F)c3C)nn2)=O)CCCc2ccccc2C1 CCCC(C(=O)Nc1sccc1C(=O)OC)NC(C1CC(N(C)C)C1)=O c1(C2C(C(=O)NC(CCCOC)c3cccnc3)C2)ccncc1F c1(C(N2CC3CC(NC(C4(C)CCCCO4)=O)C3C2)=O)cc(F)cc(F)c1O N1(C(CC=C)=O)CCC2(CCC(CNC(c3cc[nH]c3C3CCCC3)=O)O2)CC1 CC1=C(C(=O)O)CCN(C(C2CCCCN2C(=O)OCC(C)C)=O)C1 CCC(C)C(O)C(C)C(=O)N1CCN(C(=O)CC(C)(C)C)CC1C Cc1ccnn1C(C)C(=O)N(CCNC(C1(CCCCl)CCC1)=O)CC1CC1 C1(C=C)(C(N(CCC=C)CC)=O)CCN(C(c2ccc(C)[nH]2)=O)C1 O=C1CCOC(C(N2CCCCC2CC(=O)NCC2OCCC2C(Cl)Cl)=O)C1 C1(NC(c2c(CC)c[nH]n2)=O)CN(C(c2nccn3cnnc23)=O)CC12CCC2 C1(NC(CC2(CN(C)C)CCC2)=O)CCOCC1C(=O)NCCCn1cnnn1 N1(C(CN(C(C(C)C)=O)C)=O)CCC(C(=O)NC2CC(F)C2)C1C(C)C C1(O)(C(C)NC(=O)C(C)C(C)O)CCN(C(C2(C3CC3)CC2)=O)CC1 C1(C(=O)NCc2scc(CNC(C3CCC3(F)F)=O)n2)CCc2ccccc2O1 C1(C(=O)NC(c2nccs2)CC)CC2CNCC2C1 C#CC1CN(C(=O)C(CCOCC)NC(c2ccnnc2)=O)CCO1 S(=O)(=O)(c1ccc(C)cc1)N1C(C(=O)NCCNC(CCOC)=O)CCC1 c1(CC(C)NC(=O)C(N)=O)cccc(CNC(=O)Cc2coc(C(F)F)n2)c1 C(=O)(CC(C)CC(=O)N(C1CCCN(C(=O)C=Cc2ccsc2)C1)CCO)OC c1(C(C)=O)ccc(C(=O)NCCN(C)C(c2c[nH]nc2C2CCCCC2)=O)nc1 Cc1cnccc1C=CC(=O)NCCC(O)CNC(c1ccc(Br)cn1)=O C(=O)(C(CO)C(C)(C)C)N1CC(CNC(CCc2cc(OC)c(F)cc2)=O)C1 C(=O)(CCN(C(=O)CCC1OCCO1)CCO)NC(COCC)C C12(NC(c3cc(C)sn3)=O)CN(C(c3ccc(C(N)=O)o3)=O)CC1CS(=O)(=O)C2 c1(C(=O)OC)cc2oc(C(=O)NC(C(C)NC(C)=O)C(C)C)cc2[nH]1 C1(NC(C2(CCC=C)CC2)=O)CCCC(C(N2CC(O)(c3nn[nH]n3)C2)=O)C1 Cc1ncc(C(=O)NC2CCCC2NC(c2c(Br)n[nH]c2C)=O)cc1C#N c1(C(=O)NCC(CNC(C(C)OC(C)(C)C)=O)F)cnc(C(F)(F)F)c(Cl)c1 N1(C(c2n(CC)nc(C3CC3)c2)=O)CCC2CN(C(c3cnsc3)=O)CC2CC1 N1(C(C23CN(C(=O)CC4(O)CCCC4)C(CC2)CC3)=O)CCC2(CCCOC2)C1 C1(CCN)(OC)CCCCC1CC(c1n(CCCCCC)nnn1)(C1CCCC1)C C12(NC(CN(CCC)C)=O)CCCCCC1N(c1cc(O)nc(COC)n1)CC2 c1(OC)ccc(-c2nc(CC(C3CCCO3)C)n(Cc3ccccc3)n2)cn1 CC(C(=O)NC1CC2(C1)CC2NC(=O)Cc1cc(F)ccc1O)C(F)(F)F C#CC1CN(C(=O)C(C(C)OC)N(C)C)CCN1C(c1ccc(Cl)cc1C)=O C1(NC(C2C(C)C2C)=O)CN(C)CC1S(C)(=O)=O.c1(C(=O)N)cnn(CCO)c1 CC(C(=O)NC(CC1CC1)C(=O)NCCC1=CCCCC1)C(F)(F)F CC1(C)CC(C(=O)NCC2CCCC2)CCN1C(C1CCC(C2CC2)C1)=O Cc1ccc(C(=O)NCC(C)(C)OCC(=O)NCCc2nc(=N)[nH][nH]2)n1C CCC(C(=O)OC)C(=O)NCCCCCCNC(C1CCCO1)=O C1(O)(c2c(C(=O)NC(CN(C(C(C)=CC)=O)CC)CC)cco2)CCOCC1 Cc1c(C(=O)NCC(CO)NC(c2cc(O)nn2C)=O)nnn1-c1cnn(C)c1 C=CCCCCC(=O)N(C1CCCN(C(=O)CC2CC(CC)C2)C1)CCO C#Cc1cc(C(=O)NC2CCN(C(=O)C(F)(F)c3cnccn3)C2)cc(Br)c1 C#CCCC(C(=O)NC1CCS(=O)(=O)C1)NC(c1cc(F)cnc1O)=O c1(C(=O)NC2CC3(CC(NC(C4CCC(OC)C4)=O)C3)C2)cc(C)c(C)cc1C N1(C(c2cc(C(F)F)on2)C(=O)NC2CCCC2)CCCC(C2OCCO2)C1 C(=O)(C1CCCc2ccnn21)NCC12CCC(NC(C=CC(C)C)=O)(CC1)CO2 C1(CC)CN(C(C2(c3ccsc3)CC2)=O)CCC1NC(=O)C1=CCCCO1 c1(N(C2(CCO)CN(C(=O)CO)C2)C(CN2C(C)CCC2C)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NCCN(c2cc(C(C)C)ncn2)CCC)ccc(C=NOC)cc1 c1(OC(C)C(=O)NCC2(F)CN(C(c3cc(C(F)F)no3)=O)C2)ccccc1Cl Cn1ccnc1C(C(=O)NCC(=O)NC1CCC1)N(C)CCOC.C(C)(C)(C)OCC#N c1(N(C(C)C)Cc2c(C)cccc2C)ncnc2c1ncn2C(C)C(O)C(C)C N1(C(c2cn3cc(C)ccc3n2)C(=O)NCCOC)CCCCC(S(C)(=O)=O)C1 N1(C(c2c(N)nccc2)=O)CCCC(NC(=O)CC(C2CC2)C2CC2)CC1 n1(-c2ccc(C)cc2)ncc2c1CCCC2NC(=O)NC1CCc2ccccc2C1 C1(NC(c2c(C(C)C)ocn2)=O)CCN(C(c2cc(C#N)c[nH]2)=O)CC1O N1(C(c2nn(C)c(O)c2)=O)CCC2(C)CN(C(C3CC4CCC3C4)=O)CC12 c1(C(=O)NCCC(CCNC(C(C)(C)OC)=O)C)ccn2nccc2n1 C1(CC(=O)NCC2CC(NC(c3ccnn3CCF)=O)CC2O)CCCC1(F)F C(=O)(C1=CC2(CCN(C(C3COCOC3)=O)C2)C1)N1CCC(C(CC)C)CC1 N1(C(C(c2ccc(Cl)s2)C)=O)CC=CC1CNC(=O)CCN1CCCC1=O c1(C(=O)NC2CCN(C(c3nc(C)sc3)=O)C23CCC3)ccc2cn(C)nc2c1 C(=O)(N=c1ccn(CCC)[nH]1)C1(CC=C)CCN(C(=O)C(C(C)C)NC=O)C1 C1(CNC(C2(SC)CC2)=O)(CNC(=O)CCCc2cnn[nH]2)CC12CCC2 n1(CC(=O)NCC2C3CN(C(=O)C(F)C4CCCC4)CC23)cnc([N+](=O)[O-])n1 c1(C(=O)NC2C(C#N)CN(C(=O)Nc3ccccc3)C2)cc(F)c2cn[nH]c2c1 c1(NC(=O)NC2CC(NC(C(C)(C)Br)=O)C2)ccc(Cl)cc1 N1(CC(=O)N(CC(C)NC(=O)Cn2cc(C3CCC3)nn2)CC)CCC(C)(O)C1 C1(NC(c2c(C(C)C)occ2)=O)CN(C(=O)CCCS(C)(=O)=O)CC1C1CC1 CC1OC2(CO)CC1(C(=O)NCC1CCCN(C(c3ncc(F)cc3F)=O)C1)C2 C=C1CC2(C1)CN(C(=O)C=CCNC(c1coc(COC)n1)=O)C2 N1(C(=O)CC2CCCC2)CC2CCN(C(C3C4CCCCCC34)=O)C2C1 c1(C(=O)NCC(C2CCNC2)O)ccc(-c2nn[nH]n2)cc1Cl c1(OC)cc(C)c(C(N2CCC(NC(C3CC(OC)C3)=O)C2)=O)cn1 CCC(CC(F)F)C(=O)N(C1CCN(C(=O)C(C)=CC2CC2)CC1)CC CC1CNCCC1CNCc1ccccc1SC(F)(F)F c1(Cn2cc(C3(C)CN(C(=O)CCCC4CCCC(O)C4)C3)nn2)cccc(Br)c1 C(CCCCCNC(C1(C)CCNC1=O)=O)NC(C=CC)=O C1(C)(OC)CCCN(C(c2ccnc(CNC(=O)C(C)(O)C3CCC3)c2)=O)CC1 C1(N(C(=O)Cc2scnc2C)CC)CCCN(C(=O)CN2CCS(=O)CC2)C1 N1(C(CCCNC(C)=O)=O)CCCCC1C1CCCN(C(c2csnc2C)=O)C1 C1(C2(O)CCCN(C(c3cn4c(n3)C(C)CCC4)=O)C2)(C(=O)OC)CCC1 c1(C(=O)NC(C(=O)NC(c2cccnc2)CC)C2CCCC2)cc(C)c(O)nn1 C12(C(N3C(CNC(=O)C=Cc4cn[nH]c4)CCCC3)=O)CC3CC(CC(C3)O1)C2 C1(C(=O)NC2C(CCOC)C2)CN(C(=O)CC2CC(F)C2)CC1C(C)C c1(C(N2CC(CNC(CSCC(=O)OC)=O)C3C2C3)=O)nc(C)c(C)[nH]c1=O CCCC(C)(O)C(=O)NCC1CCC(CNC(c2ncc(N)cn2)=O)CC1 N1(C(c2c(C)nns2)=O)CC2C(NC(=O)CNc3ncccn3)C2C1 C1(C(=O)NCCN(C(C)C)C(C2CC(F)(F)C2)=O)CC2COCC(C1)C2(F)F C12(NC(c3ccc(C(=O)OC)[nH]3)=O)CC(C1)N(C(=O)C=C1CCSCC1)C2 N1(C(CC(=O)NCC)=O)CCN(C(=O)CN(C)S(N)(=O)=O)C(CC)C1 C(=O)(C1CCc2cccnc21)NC(CNC(c1ccc(C(C)C)o1)=O)(C)C Cc1nc(C2CCC2)sc1CC(=O)NC1(C)CC(NC(C2CC(C)(C)C2)=O)C1 C12(CNC(NC3CCS(=O)(=O)C3)=NCC3CCCO3)CCC(CC1)OC2 C1(CNC(=O)COC2CC=CC2)CN(C(=O)C2=NNC(C(F)(F)F)C2)CCCO1 N1(C(C2CC(=C)C2)=O)CC(C)(C)CC1C(=O)NCCc1ncn(C)n1 c1(C(C)(C)C)ocnc1C(=O)NCCOCCNC(C1CCC(CN(C)C)O1)=O CC(CC#N)C(=O)N(C1(C(=O)NC2CCCSCC2)CC1)C C12(C(=O)NC)CCC(C(=O)N=c3[nH][nH]cc3C(=O)OC)(CC1)CC2 c1(CN2CCC(CC(=O)Nc3nc(C(=O)OCC)c(C)s3)C2)ccc(Cl)c(O)c1 N1(C(c2[nH]cc(C#N)c2)=O)CC2CCOCC2(NC(=O)C2=CCCCCC2)C1 c1(C(N2CC(C(C)NC(=O)C(C)(F)F)C2)=O)cncc(F)n1 C1(C(C2CC2)NC(=O)NCC2CCCCS2(=O)=O)COc2cscc2O1 c1(COC)cnc(N2CCCC(NC(c3coc(Br)c3)=O)C2)nc1 C1(N(C(Cn2c(C(C)C)nnn2)=O)C)CCN(C(=O)CC2CC3(CC3)C2)CC1 CN1CCC(C)(CNC(=O)CC2CC2CNC(c2nc(Cl)cs2)=O)C1 c1(CC(=O)NCC2(NC(C3CCC4CC34)=O)CC2)cccc(Cl)c1F C1(CCC(=O)NCC2CCCCN2C(=O)CCc2cncs2)(OC)CCOCC1 n1(CC(=O)NCC(C2CCC2)NC(=O)COC2CCC2)cncn1 CC1(NC(=O)Cn2cncn2)CCN(C(c2coc(O)n2)=O)CC1 C12(Cc3c(N)cccc3)CCCCN1CCC2.c12cn(nn1)C1(CC1)C(=O)NC2 C1(CNC(CCN(CCC)C)=O)CN(C(=O)C(F)(F)c2csc(=N)[nH]2)CCC1C C1(O)(C(C)NC(C2CCCC2C(F)(F)F)=O)CN(C(C2COC(=O)N2)=O)C1 C1(NC(C(CC)F)=O)CC2(NC(c3cccc(NS(=O)(=O)CC)c3)=O)COC1C2 C1(NC(CCN(C(CC)CC)C)=O)COCCC1CNC(=O)C(C(C)C)NC=O C(=O)(CCS(N)(=O)=O)NCCC1N(C(c2[nH]ccc(=N)n2)=O)CCOC1 c1(N2CCCC3(NC(c4cc(C)n(C)n4)=O)C(C2)C3)nc(Cl)nc2c1COCC2 Cc1cc(C(=O)N(C)CCOCCN(C)C(c2ncsc2C2CC2)=O)cc(C)c1 c1(OC)cc(C(N2CC(NC(c3c[nH]c(C)c3)=O)CC2(C)C)=O)ccc1C c1(-n2c(C(C3CC3)NCC(C)(C)O)nnn2)ccccc1Cl.c1(OCC)ccccc1 N1(C(C2CC(CC)(CC)C2)=O)CCCC1(C)CNC(=O)C(C)Oc1ccccn1 Cc1cnc(S(C)(=O)=O)nc1N1CC(C(=O)NCC(C)(C)F)CC(F)C1 Cc1[nH]nc2ccc(C(=O)NC34CC(CNC(C5CC5C)=O)(C3)OC4C)cc12 Cc1sc(C2CCCN2Cc2scc(C(c3ccccc3)SC)n2)nc1C1CC1 C#Cc1ccc(C(=O)NC2(C(=O)NC3CCOCC3F)CCC2)nc1 O=C(N=c1[nH]n(-c2ccccc2)cc1Cl)Nc1cccn(CC(F)(F)F)c1=O N1(C(CC2(C)CC2(F)Cl)=O)C2CCC1CN(C(=O)COC1CCCC1)C2 c1(C(N2CCC(N(C(=O)CC3CCCCC3)C)C2)=O)ccc2c(c1)C(=O)CCC2 c1(CC(=O)NCc2c(C(N(C(CC)COC)C)=O)cco2)cccc(F)c1 C1(C(N2CCC(NC(CC(=O)NCC(F)(F)F)=O)C2)=O)CCC2(CCOCC2)O1 c1(NC)ccc(N=c2ccn(CC(=O)OC)[nH]2)cc1C(F)(F)F c1(C(=O)NC2CC(N(C(CCOCCOCC)=O)C)C2)oncc1C C(=O)(C(C(C)(C)C)SC)NC1C(CNC(c2nc(CCC)oc2)=O)COC1 C#CCC(CC#C)C(=O)N1CCOCC1CNC(=O)CC1(C)CCCO1 c1(C(=O)NC2CC2NC(C2CC2[N+](=O)[O-])=O)[nH]c2ccccc2c1Br N1(C(C(C)SCc2ccccc2)=O)CCC(C)C(NC(=O)CCNC(N)=O)C1C C1(NC(c2cn(C)nc2)=O)COC2(CCN(S(=O)(=O)c3cccnc3Cl)CC2)C1 C1(C(=O)NCC2(CCC=C)CC2)(NC(=O)Cc2cc[nH]n2)CC(F)C1 c1(C(=O)NC2CN(C(CC(CC)OC)=O)C2)ccc2ccccc2n1 C(=O)(CCCOC(C)(C)C)NCCN(CCC(C)O)C(C)=O C(c1ccncc1C)=CC(=O)N(C(CN(C(C1N(C(=O)OC)CCC1)=O)C)C)C c1(CC(C)(C2CC2)N(C(c2nnn(CC)c2C)=O)C(C)C)ncnc2c1c(Br)nn2C N1(S(C)(=O)=O)CCC(C(=O)NC(C2(O)CCCCC2)CNCC2C=CCC2)CC1 C1(CNC(CCNC(c2ccncc2)=O)=O)CN(C(C2(Cl)CC2)=O)CCC1(F)F CC1CCCN(C(=O)C(O)C2CN(C(c3ncccn3)=O)C2)CC1 C12(CNC(C(CC(C)C)OC)=O)CN(C(=O)C=Cc3ccccc3)CC(F)(C1)C2 c1(C(C)NCCC(C)F)nccc(C(F)(F)F)n1 Cc1cccc2cc(C(=O)N(CC(C)(C)NC(=O)C=C3CCN(C)CC3)C)oc12 C(CC(C)C(=O)N(CCC(C(C)C)NC(c1csc(CO)n1)=O)C)=CCC C(=O)(NN=c1ccc2nccn2[nH]1)C(N1CCC(C)CC1)=O C(C)(CCCCO)N(C1CCC1)C(C1CC(=C2CC2)C1)=O.C12(CCC1)N(C)C2=O N1(C(C=CC(C)NC(=O)C(C)(O)C2CCC2)=O)CC(=O)NC2(CC2)C1 C12(CNC(C(SC)SC)=O)CC(CCO1)N(C(C1C3CCC(C3)C1C)=O)C2 CCCCCCn1nnnc1C(c1csc(C(=O)OC)c1)NCC1CCC(=O)N1 c1(CC(=O)N(CC(C)N(C(CCc2onc(CCC)n2)=O)C)C)cn(C)nc1C CS(=O)c1ccc(C(N2CCC(O)C(NC(=O)C(C)(C)C(N)=O)C2)=O)cc1 C1(C(=O)OC)CCCC(C(N(C2CCC(NC(c3c[nH]nc3Cl)=O)CC2)C)=O)C1 c1(C(N2C(CNC(C3CCC(C)CC3)=O)COCC2)=O)cnc2ccnn2c1N c1(C(c2cccs2)NC(CC(C)NC(=O)OC(C)(C)C)=O)cc(F)ccc1O c1(CNC(C(n2cc(CNc3ccccc3)nn2)C)=O)ncc(Br)s1 C1(NC(=O)Cn2ccnn2)CN(C(=O)COCC2CCCO2)CC1n1cccn1 C(=O)(CCN=C(NCc1ncccc1OC)NCC(=C1CCCC1)F)NC CC1(C)CC(C(=O)N2CCC3CCC23CNC(=O)CC2CCSCC2)=NO1 CC1CCCN(C(C2CCCN2C)=O)C1CNC(=O)C=CCCc1ccccc1 C1(C(=O)NCCCN(C(C2(C)CN(C)C(=O)C2)=O)CCO)CC2(C1)CC1(CC1)C2 Cn1[nH]c(C(=O)NC2CCCCC2NC(C2CC2(C)C(F)(F)F)=O)nc1=O CN(OCC(F)(F)F)C(=O)C(c1cn(C)nn1)NC(C1(C)CCOCC1)=O c1(C(=O)NCc2c(CN(C(CC=CCC)=O)C)cccc2)cc2scnc2[nH]1 N1(C(c2nccc(COC)c2)=O)CC(NC(C2C3CC4C(C3)C24)=O)C2(COC2)C1 c1(C(N2CC(OC)(CNC(=O)C#CC3(C)CC3)C2)=O)ccc2c(c1)CCC(=O)N2 c1(CC(=O)N(C2CCCC2)CCNC(=O)C=C2CC2)c[nH]nc1O c1(C(C)C)ccc2[nH]nc(C(=O)NS(=O)(=O)CC(C)(C)C)c2c1 C1(NC(=O)C2=COCCC2)CC12CCN(C(c1cc(F)ccc1N)=O)CC2 C(=O)(C(C)(C)C(=O)NCCC1CCC(NC(=O)C(C)c2cncs2)C1)OC O=Cc1sc(CN2CC3CC(NC(=O)CCc4cnc[nH]4)CC3C2)c(Br)c1Br C(CCCCCC(=O)NCCCc1cncnc1)n1cc(C(C)(C)O)nn1 CCC(F)(F)C(=O)N(CCCCCCNC(=O)C=CCO)C Cn1[nH]cnc1=NC(=O)c1nccc(NC(c2cc(C(N)=O)ccn2)=O)n1 CC(C)CC(C)C(C(=O)NCC1CCCO1)N1CC(=O)NC(C(C)C)C1 c1(NC(C2CN(C(CC)C)C(=O)C2)=O)ccc(OC(F)(F)F)cc1C C1(CNC(Cc2c(CC)con2)=O)CC(C)CN(C(=O)CCC(=O)NC)C1 N1(C(C(CSC)C)=O)CC(C(=O)NCCCn2ccnn2)C(C)C1 C1(NS(CCC)(=O)=O)CC2CCC(C1)N2Cc1cncc(Br)c1C C1(NC(C(C)OCCOC)=O)CC2CC(C1)N(C(C1CC3CCC(C1)C3)=O)C2 c1(CNC(C2(C#N)C(C)C2)=O)ccc2c(c1)CCN(C(=O)C(C)(Cl)Cl)CC2 c1(N2CCCN(C)CC2)nc(=NCCCc2cncc(F)c2)[nH]c2c1CCCC2 C1(C(=O)OC2(C)CCC(C)CC2)C2CNC(=O)C2CCN1C(C(C)(C)C)=O N1(C(C(C(C)C)N(C)C)=O)C2CCC1CN(C(=O)C=Cc1cn(C)nn1)CC2 c1(C(=O)OC)ccc(C)c(C(C)NC(=O)C(=O)NC(c2ccc(CO)cc2)C)c1 CC(C)C(CC(=O)N1CC2(CC(NC(C3OCCN(C)C3=O)=O)C2)C1)C(C)C C#CCC(CC(=O)N=c1ccn(CC)[nH]1)NC(=O)CC1CCC(=O)N1C S(=O)(=O)(c1ccc(NCC(C)Cn2cccn2)c(Cl)c1)NC(CC)CO c1(C(=O)NCC(CN(C)C(c2csc(C(N)=O)n2)=O)(C)C)cc2[nH]ccc2s1 c1(C(=O)NC(CN(C(C2C(COC)(COC)C2)=O)C)(C)C)cc([N+](=O)[O-])oc1C C1(O)(CNC(C(CC)CC)=O)CCCN(C(C2(C#N)CC3CC3C2)=O)CC1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1CC(C)N(c2nc(Cl)cn3ccnc23)C(C)C1 C=CC1CCCCN1C(C12CC1CCN2C(=O)C1=CCCCC1)=O Cc1ccccc1NC(C12CC(Br)C1C2)=O C1(Cc2ccc(N3CCOCC3)s2)CN(NCc2nc(C)sc2)CC1C Cn1cc(C(C(=O)NCCC(=O)NC(N)=O)NC(=O)Cc2ccc(Cl)o2)nn1 c1(C(N(CCOCCNC(C2CCC(C)(CC)O2)=O)C)=O)c(C)nc(O)nc1C C1(C2CCC2)(C(=O)NCC2CN(C(c3cc(C)cc(Cl)c3)=O)C3C2C3)CC1(F)F N1(C(c2occ(C(=O)OC)c2)=O)CCC(CO)(CNC(c2c[nH]cc2C)=O)CC1 C(=O)(C#CC1CCCO1)NCC1(CCCNC(C(CC)n2cncn2)=O)CCCC1 C(=O)(C1=COCCO1)N1CC(SC)C(NC(=O)C(C)c2ncco2)C1 c1(CC)cc(C)c(C(N2CC(C(C(=O)NC(c3ccc(C)cc3)C)OC)C2)=O)o1 C(=O)(C#CC1CCCO1)NC1(CNC(=O)COC2CCCCC2)CC1 C1(F)(C(N2C3(C(N4CC(OC)C(OC)C4)=O)CC3CC2)=O)C(C)(C)C1(C)C C1(N(C(C2CC(CC(=O)NCC3(CC)CCC3)C2)=O)C)CN(CC(=O)OC)C1 C(=O)(C(CCCCC(=O)OC)N(C1CCN(CC(F)(F)F)C1=O)CC(C)C)NC C1(C(=O)NCCCCCNC(CC#N)=O)CCCC2(CC2)C1 C(CCC(=O)NC1CCC(CCNC(=O)COC(C)C)C1)OCCOCC c1(SCCCC(=O)N2CC(CCNC(=O)CC3C=CCCC3)C2)ccc(F)cc1 N1(C(C(C)CC2CCCC2)=O)CCc2c(CNC(=O)CN3CCC3)cccc2C1 Cc1cc(C(N2CCC(C)(NC(C3CC(F)C(=O)N3)=O)CC2)=O)cc(F)c1C c1(NC(Cc2ncc(-c3c(C)cc(O)cc3)cn2)=O)c(Cl)ncc2ccccc12 c1(C(N(C)CC2(NC(C(CSC)O)=O)CC2)=O)cccc2c1NC(=O)CO2 C(=O)(CN=S(C)(C)=O)OC.C(=O)(C#CC1(C)CC1)NC1c2c(cccc2)C1 c1(NC(c2nccc(-c3cc(C)ncc3)c2)=O)cccc2c1OCCC2 C12CC(N(C(C3CCC3)=O)C1)C(=O)N2C(=O)Cc1ccc(Br)cc1.C(CO)SC c1(OC(C(=O)NCC2(CCNC(c3cc(C)oc3)=O)CC2)C)cccc(C#N)c1 Cc1cnn(C)c1CNC(=O)CN(C)C(c1csc(F)c1)=O N1(C(C=C(CCC)C)=O)C2CCC1CC(O)(CNC(=O)C(C)(CC)C(N)=O)C2 N1(C(c2cc(C)c(F)cn2)=O)CCCN(C(=O)Cc2cccc(F)c2F)C(C)C1 C1(C(=O)OC)CN(N(CC2CCCCO2)Cc2ccccc2)C1 N1(C(c2n(CC)nc(C)c2)=O)CCCCC(NC)C1 n1(CC)cc(Cl)c(C(N2CC=CC2CNC(c2ccnc(C(F)(F)F)n2)=O)=O)n1 c1(C(N(CCN(C(=O)C(n2cc(Br)cn2)C)CC)CC)=O)cccn1C c1(NCC2OCCCN(c3ccccc3)C2)c[nH]c2c(F)cccc12 Cc1c(CC(N2CCOC(CCC(=O)N(C3CC4CC4C3)C)C2)=O)cnn1C N1(C(Cc2c(C)non2)=O)CC2CS(=O)(=O)CC2(NC(=O)C=CC2CCCC2)C1 C(C)(CCCCNC(c1ncoc1C1CCC1)=O)NC(c1cc(CC)no1)=O S(=O)(=O)(c1cccnc1)N1C(C(=O)NCc2c(F)ccc(OC)c2)CCC1 C(C)(CN=C(NCc1nnc2cccnn12)NC1CC1)(C1CCOCC1)OC N1(C(C2CCCN(C3CCC(=O)NC3)C2)=O)CC(C(=O)O)OC2(CCC2)C1 N1(C(CNS(N(C)C)(=O)=O)=O)CC(OC)CC(NC(=O)Cc2c[nH]nc2O)C1 CC1COCC1N=c1nc2sccc2c(NCC(=O)N=S(C)(C)=O)[nH]1 CCS(=O)CC(=O)N1CC(NC(=O)C(=O)Cc2ccccc2)CC1C N1(C(Cc2nc(C)oc2)=O)CCCC2(NC(c3coc(S(N)(=O)=O)c3)=O)CC2C1 N1(C(C2OCCN(CC)C2)=O)CCN(C(=O)C(CC)N(CC)CC)CC(C)C1 N1(CCC(=O)NC2CCS(=O)C2)Cc2ccccc2C1=O c1(C(N2CC(CC=C)(OCCC(=O)NC)C2)=O)ccc2c(c1)C(C)C(C)O2.OC N1(C(=O)CSc2n[nH]c(O)n2)CCC(NC(=O)Cn2cc(-c3cscn3)nn2)CC1 Cc1cccc(CC(N2C3CCC(C3)C2CNC(c2c(C)n[nH]c2C)=O)=O)c1C N1(C(C(N2C(Cc3cn(C)nn3)CCC2)=O)=O)CCC(Cn2cnnc2)CC1 CCCC(CC(C)C)C(=O)NC1(C(=O)NC2CCC3(CC3)C2)CC1(C)C N1(C(C(COC)OC)=O)CCN(C(C2(C3CCCO3)CCCC2)=O)C(C)C1 C1(NC(c2cc(C(N3CCC(NC(=O)NC)C3)=O)n(C)n2)=O)CC(C2CC2)=NO1 c1(N(CCC=C)C)ccc(C(N2CC(CNC(c3ccc(OC)s3)=O)C2)=O)cc1 c1(C(=O)NCC(CC=C)NC(=O)CCc2ncc(F)cn2)ccc(CC#N)cc1 CSC1=C(C(=O)NCCC2CCN(C(=O)CCCNC(N)=O)C(C)C2)CCCC1 c1(C(=O)NC2CCC2NC(C2CSC2)=O)cc2c(Cl)ccc(Cl)c2[nH]1 c1(OCCOC(c2ccc(-c3cc[nH]n3)cc2)=O)ccc(F)c(F)c1 C(CCC(=O)NO)NC(c1n(C(C)(C)C)nnn1)c1sccc1C1CC1 Cn1cnc2cc(CC(=O)NC(CNC(c3cc(O)cc(=O)o3)=O)CO)ccc12 Cc1c(C(N2CCCC2CNC(=O)CCCCCN(C)C)=O)cccc1C1CC1 C1(CCC(=O)NC2CCCC(SC)C2)CCc2ccccc2C1=O CCC(CC)(CO)C(=O)NCCC1CC(NC(C2CCC(=O)N2C2CC2)=O)C1 CCC(CCC(=O)N(C1CCCC1C#N)C)NC(=O)C(C)n1ccnn1 c1(CC)cc(C(N2CCS(=O)C(C)C2)C(=O)NC)ccc1OCC c1(C(=O)NCCC(C)N(C(CCc2cnc(C)o2)=O)C)ccc2c(c1)CCC=C2 N1(C(C=CC2N(C(C=Cc3n(C)ncc3)=O)CCC2)=O)CC(C)(C(=O)O)CC1(C)C c1(NC(C2CCN(C(C3CC3)=O)CC2)=O)ccc(Br)cc1O c1(C(=O)OC)ccccc1NC(C1CCCC1NCc1sccc1C)=O C(=O)(C(CC1CC1)NC(=O)CONC(=O)Cc1cn(C)cn1)OC N1(C(C2CN(C(C(C)SC(C)C)=O)CC2C)=O)CC(CO)CC(C)C1 C1(C(=O)OCC)(C(=O)NCC(C2CCCC2)NC(=O)C(C)C)CC=CC1 C1(CC(=O)N(CC(CC)OC)C)CN(C(=O)CN(CC(C)(C)C)C)CCO1 C12(CC)CN(C(C3(C)CC=CCC3)=O)C(CNC(=O)CN(C(=O)C(C)C)C)(C1)C2 c1(C(N(C2CCC(CNC(CN(C3CCC3)C)=O)CC2)C)=O)cc(=N)[nH]c(Cl)n1 c1(CC(=O)N(CCNC(C(c2cccc(Cl)c2)C)=O)C2CC2)ccccc1Cl CC1CC(C)(C(=O)NC2CC(NC(c3cncc(OC(F)F)n3)=O)C2)CC(C)O1 Cc1nc(C(=O)C(=O)NC(C)(CNC(=O)CN(C)C)Cn2cccn2)cs1 c1(C(N(C2CCCN(C(=O)Cc3ccn(C)n3)C2)C)=O)ccc([N+](=O)[O-])cc1 C(C(Cl)C(C)(F)F)NC(CN(C(=O)C=Cc1cnn(C)c1)CC#C)=O C1(OC)CCN(C(=O)CC2(N(C(=O)Cc3ccc(F)c(F)c3)C)CC2)C(C)C1 C1(NC(C(=O)N(C(C=C)C2CC2)C)=O)CC2CCC(C1)N2Cc1ccccc1 Cc1ccc(C(N2CCC(NC(C3CC3c3ccccc3)=O)C(F)C2)=O)cc1Cl C1(C(N(C2CCN(C(c3cnn(CC)c3)=O)CC2)CCC)=O)CCCC(=O)O1 N1(C(C=C(C)C(F)F)=O)C2CC1CN(C(C1(C(F)F)CCCC1)=O)C2 CC(C)C(CCN(C(=O)C(C)C(=O)OC(C)(C)C)CC)NC(C1CC=CC(O)C1)=O CC1(C)COCCN1Cc1ccc(C(=O)NCc2cccnc2OCCO)cc1 c1(C(N(C2CCCC(NC(c3cncc(OC)c3)=O)C2)C)=O)cc(N)c(F)cn1 C(=O)(CCC(F)(F)C(F)(F)F)N1C(C(C)NC(C2CCC(C)(C)CC2)=O)CCC1 C1(CC)(CNC(C2(COC)CC3(CC3)C2)=O)CCCN(C(=O)CSC(C)C)C1 C=CC1(CC(=O)N(C)CC2CCN(C(c3cn(C)c(O)n3)=O)CC2)CCOCC1 Cc1c[nH]c(C(=O)NCC(CC(C)C)NC(=O)COc2cccnc2)c1C c1(OCC)cnc(NC(C(C)NC(c2n[nH]c(C)n2)=O)C(C)C)nc1 Cc1cc(CC(=O)NC(C2CCCN2C(=O)C(=O)NC(C)C)C)ccc1CO Cc1ccc(CC(=O)N(C)CC2CCN(C(=O)C(C)OC(C)(C)C)C2)c(F)c1 CC(C)C(CC(=O)N1CCOCC1CN(C)C(c1cnsn1)=O)C(C)C C1(C(N2CC(NC(c3cc(C)c(Cl)s3)=O)C(C)C2)=O)CCc2nnc(O)n2C1 C1(CC(=O)NCC(C)CN(C(=O)C(O)Cc2cnn(C)c2)C)(CC=C)CCCC1 N1(CC(N2C(CCNC(C(C)NC(N)=O)=O)CCCC2)=O)CCCNS1(=O)=O Cc1ncc(C(N2CCCC2(C)CNC(C2CC2F)=O)=O)c(Br)c1Cl C=CCC(CC=C)C(=O)NCC1CCN(C(C2CNC(=O)C(C)(C)C2)=O)C1 c1(CNC(C2CN(C(=O)OC(C)(C)C)CC(C)O2)=O)cncc2ccc(F)cc12 C1(C(N2CC(CC(C)NC(=O)CCn3ccnn3)C2)=O)CCCCCCC1 N=c1[nH]c(NC(=O)NCc2cn(CC(=O)NCc3ccccc3)nn2)cs1 C1(NC(C(c2ccc(Cl)cc2)C)=O)CN(C(C23CC(CO2)C3)=O)CC2CCCC12 C(=O)(C(C(C)(C)O)NC(=O)CSCCC#N)N1CCC(C)(C)C1 C1(NC(c2ccc(CC)o2)=O)CCCN(C(c2cc(=O)n(C)cn2)=O)C1CC C=C(Cl)CC(C(=O)NC(c1nnc(C)s1)C)NC(=O)C(C)OCCOCC CC(CCCCNC(=O)C(C1CCCO1)C1CC1)NC(=O)CC1CC(=O)NC1=O S(=O)(=O)(c1c[nH]ccc1=NCCC(=O)Nc1ccccc1)N(C(=O)CC1CC1)C c1(C(N2CCC23CCCSC3)C(=O)NC2(C)CC2)ccc2nccnc2c1 C(C(C(C)(C)C)NC(=O)CCCN1CCCCC1)NC(CCCOC)=O CC(=O)CCCC(=O)NCCC(C(C)(C)C)NC(=O)Cc1cn(C)nc1C(F)F C(=O)(C(C)S(=O)(=O)C(C)C)NCCCC1CCN(C(C(CC(=C)C)C)=O)CC1 Cc1cccc(Cl)c1C(N1C2CCC1C(C(=O)NC(c1cccc(F)c1)C)C2)=O C=CC1CN(C(=O)CCN(C(=O)C(C2CC2)OCC)C)CCO1 N1(C(C2(CCC)CCNC2=O)=O)C2CCC1CC(NC(c1cc[nH]c1)=O)C2 N1(C(C(C(C)C)F)=O)CC2(CCC(NC(c3cc(C(N)=O)co3)=O)CC2)C1 N1(C(C(CC)C(C)C)=O)CC2(CNC(c3ccco3)=O)CCC1CC2 CCC(Cc1ccccc1)CC(=O)N(C(C)CCNC(=O)CC(O)CN(C)C)C C1(CCCCCC)CCCC1(c1nnnn1C(C)(C)CC)NCC=C(Cl)Cl C(=O)(C(C(C)(C)C(N)=O)NC(N)=O)N(C)CCNC(=O)CNC(=O)OC(C)(C)C CC(C)C=CC(=O)NC(C)CN(C(=O)COC(=O)CO)C CN1CCN(C(C2CCCN(C(c3cccc(I)c3)=O)C2)=O)CC1(C)C C1(CNC(=NCC)NCCc2ccccc2Br)COC2(CCCC2)O1 CC1CCC(C)(C(=O)NCC(Cc2ccccc2F)NC(C2CCCC2O)=O)C1 N1(C(CCN(C(CC)CC)C)=O)CCC(NC(=O)C=Cc2cncs2)C(O)C1 c1(C(N2CC3(CC(NC(c4cnc(SC)nc4)=O)C3)C2)=O)cc(C)c(Cl)c(C)c1 c1(C(N2CCCC(NC(=O)CC3CSCCS3)C2)=O)cc(F)cc([N+](=O)[O-])c1 C=C(C)C1OCCC1C(=O)NCC1CCC1NC(c1ccc(C(C)(C)C)nc1)=O CC1=NC(C(=O)N(CC(C)CNC(C2(N(C)C)CCCC2)=O)C)CS1 C(=O)(C(C(C)C)(C(C)C)C1OCCO1)NCc1cn(C2CCC(OC)CC2)nn1 C1(NC(c2cc(C)ncc2C)=O)C2CCCN(C(C3CCCCS3)=O)C2C1(C)C C=CCC(C)(O)C(=O)N1CCC(CCC(N2CCOC(CC)C2)=O)C1 C(=O)(C1=CC2CCCC12)NCC1CN(C(c2n(CC)nnc2)=O)C(C)C1 C(=O)(CCCC(C)(C)NC(C1CCCC(=O)CC1)=O)N1CC(CCC#C)C1 S(=O)(=O)(c1ccccc1)C(=O)N(CCCN(C(CC(C)F)=O)CC)CC1CCCC1 c1(C(C)C)ncc(C(c2nnnn2C2CCOC2)NCC(C)(C)OCCO)[nH]1 CS(=O)(=O)c1cccc(CC(=O)NC2(c3ccccc3)CCCN(C(C)(C)C)C2)c1 C(=O)(C#CC1CCCCC1)NCC(=O)NCC(N1C(CC)CCCC1)=O C1(NC(C2(CC=C)CCC2)=O)CN(C(=O)Cn2cncn2)CC1O C(C(=O)NCC12CC(CNC(=O)CCC(C)SC)(CO1)C2)(C(C)C)OCC c1(C(=O)NC(C2CN(C(=O)CC3CCOCC3(C)C)C2)C)ccn2cccc2c1 N1(CCc2ccc(OC(F)(F)F)cc2)CC(C2CCNC2)C1 C1(NC(C2C(CCC)C2)=O)CC2CCC(C1F)N2C(c1cnc(O)c(C)c1)=O c1(C(N2CCC(C)C(CNC(c3ccno3)=O)C2)=O)cccc2nsnc12 C(CN=c1[nH]c(N2CCC(N3CCCC3)C2)nc2c1CCC2)N(C(CC)C)C C1(CNC(Cc2cc(C)[nH]n2)=O)CN(C(c2csc(C)c2N)=O)CCC1(C)C c1(CC)cccc(C(=O)NCC2CCN(C(=O)CCSCC(C)C)CC2C)c1C Cc1nn(C)c(N)c1C(=O)NCC(C)(C1CC1)NC(=O)CN1CCOCC1=O c1(C(N(CC(C)NC(c2ccc(N3CCOCC3)cc2)=O)C)=O)nc(=O)n(C)[nH]1 N1(C(c2c(C)ccc(C)n2)=O)CC2CCCC(C1)N2C(=O)CCCCN(C)C C#Cc1cnn(CC(=O)N(C)CC2C3CN(C(C4(OC)CC4)=O)CC23)c1 N1(C(C2CC(C#N)C2)=O)CCN(C(C2CC3C=CC2O3)=O)C(C2CCCC2)C1 c1(C(=O)NCC2C(NC(CSCCC#N)=O)C2)coc2c1C(=O)NCCC2 N1(C(c2cn(CCC)nc2)=O)CC(NC(=O)C(N2CCOC2=O)C)C(C2CC2)C1 C1(O)(C(C)C)CCN(C(N(c2ccoc2Cl)CC(C)CN2CCCC2)=O)C1 N1(C(C2(CC)CC2(F)F)=O)CCC2CN(C(=O)C(C)(C)C3CCCO3)CC2CC1 C1(SCC(N2CCC(CC(C)CO)CC2)=O)CCc2ccccc2C1 C(c1ccccc1F)=CC(=O)NC12CN(C(c3cn(CC=C)nn3)=O)C(C1)C2 Cc1cc(C(=O)NC(C2CCOC2)CNC(=O)CCCc2nccs2)sc1C c1(C(=O)NC2CCN(C(C(CC)CC(C)C)=O)C2(C)C)ccc2cnccc2n1 O(NC(=O)C(C(C)O)NC(=O)Cn1cnc(C#N)n1)CCCC(=O)OC CC1=CCC(C(=O)N(C2CCC(NC(c3nnn(C)n3)=O)CC2)C)CC1 N1(CC(=O)NC(C2CC3(CCC3)C2)C)CCN(C(c2cc(C(N)=O)[nH]n2)=O)CC1 c1(-c2cc(C(=O)NC3(CNC(=O)COC(F)F)CCCC3)n[nH]2)cc(F)cc(F)c1 C1(C#N)(OC)CC(C(N2CCC2CNC(C2CC(=O)N(C)C2)=O)=O)C1 c1(C(=O)NC2(CCNC(=O)CSCC(F)(F)F)CC2)nnc(O)nc1O c1(C(N2C(Cn3cc(CS(C)(=O)=O)nn3)CC2)=O)cc(SC2CCCC2)ccn1 N1(CCC#C)CCC(C(C)CNC(=O)Cc2ncc(CC)[nH]2)CC1 N1(CC(=O)NC(c2ccccn2)=O)CCCCC1c1ccc(C(F)(F)F)cc1 N(C1CN(C(c2onc(C)c2C)=O)CCc2ccccc21)C(CC=C)=O c1(CN2CC(O)(CNC(=O)CC3CCOCC3)C2)c[nH]c2cccnc12 C(=O)(CS(=O)(=O)CC(F)(F)F)N1CCC(NC(c2n(CC)nnc2)=O)CC1C N1(C(C(C)(C)C2CCCC2)=O)CC2(CCCCN2C(c2cc(F)cnc2O)=O)C1 CC(C)CCC(O)C(=O)NC1CC2CC(NC(c3nocc3C(C)C)=O)C2C1 Cc1c(C(N2CC3C(NC(c4ccncc4Br)=O)C3C2)=O)oc2ccccc12 C(Cc1cnc[nH]1)(C(=O)NC(C)Cc1ccncc1)NC(CNC(CCC)=O)=O c1(SC)c(C(=O)N(C)CCOCCCN(C)C(C2CC3CCC3C2)=O)cnn1C CCCCCCC(CC)C(=O)N(C)CC1COCCN1C(c1ccc(C)cc1)=O C12(CNC(C(C)N(C)C)=O)CCC(C1)N(C(c1ccc(Cl)nc1O)=O)C2 C1(C=C)(C(=O)NC(c2ccccc2)C#C)CCN(C(C2CC2(F)Cl)=O)CC1 c1(C(=O)NCC2(C)CCN(C(=O)Cn3cccn3)C2)ccnc2c(F)cccc12 c12ccc(C(F)(F)F)cc1C(c1n(CCC)nnn1)N2.n1(CC)nc(C)cc1C CCCCCCC(C)C(=O)NCCC1CCCN1C(c1ccc(=NCC)[nH]c1)=O C1(N(C)C(c2cn3c(n2)CCC3)=O)CCCCN(C(=O)C(C)(C)c2ncco2)C1 N1(CCCNC(C2(CCC)CC2)=O)CCN(C(=O)CC(C)CC)CC1 C(=O)(C1=CC(C)CC1)NCc1ccc(CNC(C=CC)=O)cc1 c1(C(N(CCNC(C(CC)c2cccnc2)=O)C)=O)cc[nH]c(=N)c1[N+](=O)[O-] c1(CC)cc(C(=O)NCc2ccc(C(N3CC(N4CCC4)C3)=O)o2)n(C)n1 C1(C(N(C(C)C(=O)N(C2CCC2)CC2CC2)C2CC2)=O)CC12CCCCC2 c1(C(=O)NC2C3CC(NC(C(C)n4ccnn4)=O)CC32)cccc2oncc12 C1(C(=O)NCCN(C(C(=O)N(C)C)=O)C2CC2)CCN(c2nccs2)CC1 N1(C(c2ccc(NC(N)=O)cc2)=O)CCCCCC1CNC(c1cc(Cl)cs1)=O CC1(CNC(C2(CO)CC(F)(F)C2)=O)CN(C(=O)CCn2ccnn2)CCO1 c1(C2(C(N3CCC(NC(C(CC)OCC)=O)CC3)=O)CC2)ccc(Cl)cc1Cl C1(C#N)(C(N2CC(C(C(=O)N(CC(C)C(F)(F)F)C)N(C)C)C2)=O)CCCOC1 C1(NC(C2N(CC)CC2)=O)CC2(CCC(CNC(=O)CCNC(=O)CO)OC2)C1 C1(CNC(CCCC=C)=O)CC(C(C)C)CCN1C(c1cc(=O)cc(Cl)[nH]1)=O c1(CC)nn(C)cc1C(N1CCN(CC(=O)N(CC(O)C(F)(F)F)C)CC1)=O c1(C(=O)NC2(c3ccc(-n4ccnn4)cc3)CC2)cc(C(F)(F)F)ccn1 C(=O)(CC(O)C(C)(C)C)NC(CCN(C(c1c(C)cncc1)=O)C)C(C)C C(=O)(C(C)CC(=O)OC)NC1CC(CC(=O)NC(CC#CC)CO)C1 C(=O)(C1CSc2ccccc21)N(C1CN(C(CCCC#CC)=O)CC12CC2)C N1(Cc2c(C)noc2C)CCCC(C)(C(N2CCC23CN(C)C3)=O)C1 c1(OC)cc(F)ccc1C(N1CCCC(C)C1CNC(=O)Cc1conc1C)=O C1(CC)CN(C(C2CCC(C(C)C)N2C(c2nnc(S)n2C)=O)=O)CCO1 c1(SCCC(=O)NCCNC(Cc2c(C)occ2)=O)cc(F)ccc1F C1(CCOCC)(C(=O)N(C)CCN(C)C(C2(CC)CCC2)=O)CCCC1 CC(C)(C)CC(O)C(=O)NC1COCC1CNC(c1cc2n(c1)CCSC2)=O c1(CC)ncc(C(=O)NCC(C(C)C)NC(C2CCC2Cc2ccccc2)=O)[nH]1 c1(C(N(C(C)CNC(=O)CC2SC(=N)NC2=O)CC)=O)cc(C)cc(OC)c1C c1(C(N(C(CCNC(C2(CC)CCC2)=O)C)C)=O)cc(OC)c(Br)s1 Cc1ccc(-c2ccc(C(N3CCCC3c3ccncc3C)=O)o2)cc1 C(CCC(C(=O)N(C)CC1CCCCCC1)NC(c1cc(C)no1)=O)OC N1(C(CSCCCC)=O)CCN(C(=O)C=CCCc2ccccc2)CC1C(F)F c1(NC(C2CCC(Nc3c(F)cnc(C)n3)C2)=O)cc(F)c(Cl)cc1F N1(C(=O)NCc2ccc(CC3CCC3)cc2)CC2CC(C1)c1cccc(=O)n1C2 N1(C(COCCOC)=O)CCCC(C2CN(C(=O)C(F)(F)c3ccccn3)C2)C1 C1(CNC(C(C)(C)n2cnnn2)=O)CC2(CO1)CN(C(C1(O)CCOC1)=O)C2 c1(N(C)CCOC2CC2)nc(N2CC3OCCOC3C2)nc2scnc12 C1(C(=O)NC2CCC(NC(c3cc(C(CC)CC)no3)=O)C2)CC2(CCCC2)C1 c1(C(N2CC(NC(CC(CC)SC)=O)C(C)(C)CC2)=O)cccc2[nH]cc(Cl)c12 c1(OC)cc(C)ccc1Cc1nccc(CC(=O)NC2CS(=O)(=O)CC2CO)n1 C=CCCCC(C(=O)N1CCCC(F)CC1)NC(=O)C(CC=C)NC(C)=O N1(C(CCCOC)=O)CCN(C(c2ccnn2C(F)F)=O)C2CCCCC2C1 C(CCC(O)CO)NC(CN(C(CNC(=O)NC)=O)CC1CC1)=O C(c1ccccc1Br)=CC(N1CC(NC(C(COC)(C)OC)=O)C(C)C1)=O C1(CC)(NC(C(CCNC(C2CCNC(=O)C2)=O)OC)=O)CCCCC1 CC(CO)C(=O)NCC(O)CN(C(=O)CC(c1cccs1)n1cccc1)C C(=O)(CC(C(F)F)C(C)(C)C)N1CC(C)N(C(c2ccc(N)cc2F)=O)CCC1 N1(C(c2c(N)csn2)=O)CC(NC(c2ccc3ccoc3c2)=O)C2CCCCC12 N1(C(C2CCC(CNC(c3ccc(C)c(O)c3)=O)O2)=O)CCCC2(CCCC2)C1 C1(CNC(C=C(C)C)=O)CC2(CO1)CN(C(=O)Cc1ccc(CO)cc1)C2 C1(NC(C(C(C)C)CO)=O)CN(C(c2ncccc2F)=O)CCC12CCOCC2 c1(CC)ocnc1C(=O)NC(CC1CCC1)C(=O)NCCSCCO N1(C(c2cnc(C)s2)=O)CC(NC(C23C=CC(CC2)C3)=O)C(O)C1 O=C1NCc2ccc(C(=O)NCCS(=O)(=O)Cc3cn(CC4CC4)nn3)cc2N1 c1(CC(=O)NCCNC(CN(C2CC2)CC)=O)ccc(Br)cc1C#N C12=NC(=NCCC3(OC)CN(C3)C1=O)NC=C2.c1(OC)ccc(CO)cc1 CCC(CC(=O)N1CCCC(C)(C(=O)NCCC(=O)NCC)C1)C(C)(C)C C(CN=C(NCc1ncc(C)cc1C)NCC1COC(C)(C)O1)SC c1(OC)c(C)nc[nH]c1=NCC1CC(C)N(C(c2cnn(C)n2)=O)C1 N(C1COc2ccc(F)cc21)C(c1cncc(N)n1)=O c1(C(N2CC(C)C(NC(=O)CCNC(N)=O)CC2)=O)c[nH]c2cc(F)c(F)cc12 CC(C)(C(=O)NCC(O)CC(=O)N1CC2(CSC2)C1)C(F)(F)F C1(C2(C(N(C3CN(C(C4CCN4C4CCCC4)=O)C3)C)=O)CC2)CCCC1 C1(C(=O)NCCSC(C)C)CC(O)C(O)CC1CNC(C1CCN(C)C1=O)=O CC(C)(CCO)NC(c1conc1CNC(=O)C=CCF)=O C1(NC(CC2C(C)C2)=O)CN(C(=O)CSCC2CCCCO2)CC2(CC2)C1 c1(NC(CC2N(C(C3CCN(C)C3)=O)CCCC2)=O)ccc(Br)c(F)c1F C1(C(N(C2CC(C(NOCC(=O)OC)=O)C2)C)=O)C2CCC(C2)C1C c1(C(N(CCCCCCNC(C2CC=CCC2)=O)C)=O)ccn2cccc2c1 S(=O)(=O)(c1cc(Br)nn1C)NCCCCOC(C)C C12(NC(CC3C(C)(C)C3)=O)CCC(CNC(c3ccc(C(N)=O)o3)=O)(C1)OC2 c1(CC(=O)NC2CCCN(C(c3occc3Cl)=O)C2)cccc2nsnc12 Cc1snc2sc(C(=O)NC3CCN(C(=O)CN4CCCC4)CC3F)cc12 S(=O)(=O)(c1cnc(Cl)nc1)NC1CCN(C(c2cc3ccccc3o2)=O)CC1F c1(CNC(CC2(NC(C(OC)OC)=O)CCC2)=O)ccc(Cl)c([N+](=O)[O-])c1 O=C(C#CCNC(C1(CO)CCCC1)=O)NCCCC1CCCCC1 C1(OC)CC(CNC(=O)CSCC2CCCO2)N(C(=O)Cc2ccncc2C)C1 C(N=c1[nH]c(N2CCCSC2)nc2cc(C(F)(F)F)ccc12)c1n(CC)cnc1 N1(C(CCCC(=O)OCC)=O)CCCC2(NC(=O)CCc3ccccc3)CC2C1 CC(C)CC(C(=O)NCCCOC(F)(F)F)ONC(=O)C(C)C1CCOCC1 N1(C(c2c(OC)csc2)=O)CCc2sccc2C1CNC(C1(O)CC1)=O N1(C(CCC(=C)Br)=O)CCC2(CCN(C(=O)CCCC(C)CC)C2)C1 C(=O)(C(F)C(C)CNC(c1cn(CC)nc1C)=O)NC(CCC=C)C N1(C(c2ccc(CC)[nH]2)=O)CC(NC(c2cc(C)cnn2)=O)CC(C)(C)C1 N1(C(CNC(=O)NC)=O)CCCC1C1CCN(C(C2CN(C(C)=O)C2)=O)C1 N(C(=NCC(C)COC)N1CCC(c2ccccc2)C1)CC(=O)N(CC)CC c1(OC)ccc(C(=O)NCc2csc(CNC(=O)CCSCC(N)=O)n2)c(C)c1 C(N=c1nc(N2CCC(O)C(CO)C2)c2c([nH]1)COC2)c1c(C)coc1C CCCCCCC(C(=O)N1C2CCC1(CNC(=O)C1=CCOC1)CC2)NC(C)=O C1(CC=C)(NC(=O)C(C)SCCCC)CN(C(C2CCOC2)=O)C1 CCCC(CNC(=O)COC(C)(C)C)C(=O)N1CC(CO)CC(C)C1 CCCC(C#N)C(=O)N(C(C)CCNC(C1CC(O)(CCC(C)(C)C)C1)=O)C N(C1CC2(CN(C(c3cc(C)c(O)c(N)c3)=O)C2)n2ccnc21)C(C(C)OC)=O c1(C(N2CC3C(NC(C4CCCCC(=O)N4)=O)C(C3)C2)=O)ccc2ccsc2c1 CC1c2ncc(C(N3CCC4COCC4C3)=O)n2CCN1C(c1cnoc1)=O CC1=C(C(=O)NCC2CCCN2C(c2nc(Cl)sc2Cl)=O)Cn2ncnc2N1C c1(N(C)Cc2c(OC)c(Br)ccc2)c(Br)c(C(=O)O)nc2ccccc12 C(c1ccc(OC(F)F)cc1)=CC(=O)NCCC1N(C(C(C)C2CC2)=O)CCC1 C1(NC(COCCOCC)=O)C(C)CCN(C(C2CC(=O)N2)=O)C1C C1(N(C(c2c(C)cc(Br)o2)=O)C)CN(C(=O)C2=NNC(=O)C2)CCC1C N1(CC(=O)N(C)CC2N(C(CCC(CC)O)=O)CCC2)C(=O)CC(C)(C)C1=O c1(C(N2CC(C(C)NC(C(C)=CC)=O)OCC2)=O)n[nH]c2cc(Cl)ccc12 C1(CC(C)O)CCN(C(C2CC(CCNC(=O)CNC(=O)C(C)(C)C)C2)=O)CC1 Cc1cnc2n1CC(C(N1CC=C(CNC(=O)C(F)(F)C(F)(F)F)CC1)=O)CC2 C1(OC)CC(CNC(=O)CCC2CCCC(=O)N2)N(C(c2ncc(F)cn2)=O)C1 N1(C(c2csc3ccccc23)=O)CC2CCCC(C1)N2C(=O)CC1CCOCC1 c1(C(=O)NCC2(CN(C(C3CCC(OC)C3)=O)C)CC2)cnn(C)c1C(C)(F)F CCCCC(CNC(C1(C)CCCO1)=O)NC(c1coc(OCC(F)(F)F)n1)=O N1(C(=O)NC2(CC(=O)OC)CCC2)CCC(C(C)O)CC1.c12nc(n[nH]1)S2 C1(N(C)C(c2ccc(F)cc2)=O)CCCN(C(=O)C=CCN2CCCC2)CC1 N1(C(C=Cc2cncc(C)c2)=O)CCN(C(=O)CC2(C)OCCO2)CC2(CC2)C1 c1(NC)cnccc1C(N1CCCC(N(C(=O)CC2CCCC(=O)N2)C)C1)=O Cc1nc(C(=O)NC2CCCN(C(C3CN(C4CCOC4)C3)=O)C2)c(=O)[nH]c1C C1(NC(c2n(C)ccn2)=O)CN(C(=O)CCC2CNC(=O)N2)CC1C(F)(F)F C(=O)(C1Cc2ccccc21)NCC1CN(C(CCCN(C(=O)OC)C)=O)CC1O c1(C(N(CC(C)O)CCNC(CCCC(OC)OC)=O)=O)cn(C)c(=O)nc1O c1(N(CCCNS(C)(=O)=O)C)nc(=NCCC2CCCC2)[nH]c2c1CCCC2 N1(c2nc(C)c(C#N)cc2Cl)CCCC(C2CC2NC(=O)Cc2cc[nH]n2)C1 c1(C(C)C)cc(C(=O)NC(C2CCCC(c3ccccc3)O2)C2CC2)n(C)n1 O=C1CC(C(=O)NC2CN(C(=O)Cc3ccsc3)CC2C(F)(F)F)=NN1 N1(C(CCC(C)=O)=O)CC(C(N2CCC23CCCC3)=O)CC(F)C1 C(CC(N)=O)(C(=O)NC1CC(CO)N(C(=O)CCC2CC2)C1)NC(CC(C)C)=O N1(C(c2nc(C#C)sc2)=O)CCC(CO)C(NC(c2ccn(C3CC3)c2C)=O)C1 C1(O)(Cn2cc(C(C)N(C)C)nn2)CCN(C(=O)C(F)CC2CCCCC2)CC1 CCCC(C(=O)NCC(O)C1(Cl)CC1)NC(C1CCOC1C(C)C)=O c1(CC)noc(CC)c1CC(=O)NCCCCNC(=O)CCCCN1CCCC1 Cc1nc(C)c(C(C(=O)NCCC2CC2)N(C)CC23CC(C2)C(C(F)(F)F)N3)s1 c1(CC)ccc(C(=O)N(C(C)C(=O)NC2CC2(C)CC)C)[nH]1 c1(C(=O)NC2(C3N(C(CCCC)=O)CCCC3)CC2)cc(C2CC2)nc(O)c1 C(=O)(C1COc2ccccc21)N1CCC(N(C(=O)C2=CCC2)CC)C1 N(C1CCc2cccc3cccc1c23)C(c1cc(C)c(-c2cccc(Cl)c2)s1)=O c1(N2CCCC(OCCC)CC2)nc(=NCCOC)[nH]c2c1SCC2 CCC(C)(C#N)C(=O)NC1CC(CNC(c2nocc2C2CC2)=O)CC1O c1(-c2cn(CC(C)(C)CNC(C3C(CO)CCCC3)=O)nn2)cnccc1C#N Cc1nn(C)cc1-c1cn(CCNC(=O)NC2(c3cccc(Cl)n3)CC2)nn1 N1(C(c2c(CC)n[nH]c2)=O)CCN(C(=O)CCc2cnn[nH]2)C(C)C1C N1(C(c2c(Cl)cccc2Cl)C(=O)NCCCOCC2CC2)CCC2CCC(C2)C1 c1(CC(N2C(C)(CNC(C(C)OC)=O)CCC2)=O)cccc(F)c1Cl C1(NC(C2(C)CCCS2)=O)CC1C1CCN(C(c2c[nH]c3nccc-3c2)=O)CC1 C1(NC(c2c(CCC)occ2)=O)CCC(CNC(C2CC3CC2C3)=O)CC1 C(=O)(C(C)(F)C(C)(C)F)NCC(=CC(=O)N(C(C(=O)OCC)C)C)C c1(C(c2nnnn2C(C)C)(CC)NCc2ccc(Br)s2)ccccc1OC Cc1cc(CC(=O)NC2CC3CC2CN3C(C2CC(=C3CC3)C2)=O)ccc1O C1(CC)(NC(=O)CCCn2ccnc2C)CCN(C(=O)C(C)OCCN(C)C)C1 O=C1CC2(CCN(C(C3CCN(C(=O)c4csc(Cl)c4)O3)=O)C2)CN1 C1(C(N(C)CC2CCCN2C(c2csnn2)=O)=O)CCn2c(O)nnc2C1 c1(C(N2CCN(C(C3CCCC3)=O)C(CO)C2)=O)nc2cccnc2s1 N1(C(C(C)C2CC2)=O)CCC(O)(CCNC(=O)CCN2CCC(F)C2)CC1 n1(CC(=O)NC2CC(NC(C(C3CC3)OC)=O)C2)cc(C(F)(F)F)nn1 N1(C(c2ncn(CC)n2)=O)CC(NC(=O)CCc2cc(C)nc(C)c2)CC(C)C1 c1(C(N2CCC(O)(CNC(C(C)S(N)(=O)=O)=O)C2)=O)cc(S(N)(=O)=O)oc1Cl Cc1cc(Br)ccc1S(=O)(=O)N1CC2CC1CN2C(=O)CCC1(CN)CCC1.N c1(C(C(=O)OC)NC(=O)C(c2cccnc2)NC2C3COCC23)ccc(F)c(Cl)c1 C1(CNC(C(C)OCC#C)=O)CC(CNC(c2csc(C(C)C)n2)=O)CO1 c1(C(=O)NC(CCNC(C(C)OCC#C)=O)C)cc(C(C)(C)C)nn1C C1(C(=O)NCCOCC(=C)C)COCCC1NC(=O)C(C)(C)CF c1(C(N(C2CC3CC2CN3)C(=O)C(F)Cl)=O)cc2cccc(F)c2s1 c1(CC(C)NC(c2c(CSC)cco2)c2nnnn2C)ccccc1Cl N1(C(C=C(C)Cl)=O)CCN(C)CC1CNC(C1CCC2(CC1)CC2)=O C1(C(=O)NC(CC)CSC)(OC)CCN(C(c2coc(Cl)n2)=O)CC1 c1(CCOC(C)C(=O)NCCNC(=O)CC(O)c2ccccc2)ccccc1 C(=O)(C(CC#CC)NC(c1ccc(F)c(F)c1)=O)N1C(CCC#C)CCC1 CC1(C)CCCCC1(C)NC(C12CC1CCN2C(=O)CCn1cnc(=N)[nH]1)=O C1(NC(COCC(=C)C)=O)COC2(CCN(C(c3ccc(C(C)(C)C)[nH]3)=O)C2)C1 c1(-c2ccc(CN(CC(C)C)C)s2)cccc2c1nnn2C1CCCCC1 c1(OC)ccc(CC(=O)NC2(CN(C(=O)Cn3cc(C)cn3)C)CC2)c(Cl)c1 c1(C(=O)NCCOCCN(C)C(C2CCC(=O)O2)=O)cc2ccsc2n1C c1(CC(N2CCN(C(c3n(CC)ncn3)=O)CC2C)=O)c(F)cccc1C#N CC(O)CC(=O)N(C(C)(C(=O)NCC1(C#N)CC1)C1CC1)C c1(OC)ccnc(C(N2CCC(F)C(NC(c3ccco3)=O)C2)=O)c1OC Cc1ncnc(C(=O)NCC(C2CCC2)NC(c2cccc(N(C)C)c2)=O)c1C c1(CC)onc(C(=O)NC(Cc2cc[nH]n2)C(=O)NC2CC2c2ccsc2)c1C C(=O)(CC(F)(F)C(C)C)N1CCCC(N(C(c2[nH]cc(CC)c2)=O)CC)C1 c1(N(C2CCCOC2)CC)nnc(-c2nc(C)ns2)n1CC1CC1 c1(CC)ncc(C(=O)N(C2CCC(NC(C3(Br)CC3)=O)CC2)C)c(C)n1 C(CCN=c1[nH]c(Cl)ncc1C)OCCNC(c1cc(C)oc1C(F)(F)F)=O c1(C(=O)NCC2CN(C(C3CCCCC3)=O)CCO2)cc2c(O)ncnc2cn1 N1(C(c2c(C)cn(C)n2)=O)CCN(C(c2cc(N(C)C)ccn2)=O)C2CCC12 C1(C#N)(Cc2cn(CC(=O)N(C)Cc3ncc(Cl)n3C)nn2)CCCCC1 c1(C(N2CCC(OC)(CNC(=O)CCS(C)=O)C2)=O)cncc(F)c1Cl N1(C(c2c(OC)ccs2)=O)CCCCC(NC(=O)CC2CC(OC)C2)C1 C1(CC(=O)OC)CC2(CCN(C(=O)Cc3sc(S)nc3C)CC2)CO1 c12ccc(cc1)C(=O)N(C)C2.C(=O)(CCC(C)C)NCC1CN(C(=O)NCC)C1 C#CCC(C)(CNC(=O)CCC1(NC(=O)CCCSC)CCCC1)CO c1(SC)ccc(C(C)NC(C2CSCCN2C(=O)CC2CCCCO2)=O)cc1 C(=O)(C#CC1(C)CCCO1)NCC1CCCCN(C(C2(CC)CC(C)(C)C2)=O)C1 C1(N(C(=O)CSc2ccccc2)C)CC2CCC(C1)N2C(=O)CC1(CSC)CC1 c1(C(=O)NCC(C)CNC(=O)Cc2ccco2)cc(S(N)(=O)=O)ccn1 c1(CN2CC(F)(C(N3CCC(C(F)(F)F)C3)=O)C2)nc(Br)ccc1F Cc1c(C(=O)NC2CN(C(C3CCN(C)C3=O)=O)C2)cccc1Br N1(C(CNc2c(C)cccc2)=O)CCC2(CC1)CC2C(N1CC2CC1CN2C)=O C=CC(CC)C(=O)N(CCNC(=O)C(CO)N(C)C)CCOCCO C(=O)(C(O)CC(F)F)N1CCCC(C(N(CCOC)C)=O)C1 c1(OC)cc(OC)c(C(N2CC(NC(C3CC(C)(C)CO3)=O)C(O)C2)=O)cc1N CN1C(=O)CCC1C(=O)NC(C)(C)C(=O)NCCN1CCNC1=O C12(C(=O)OCC)COC(NC(=O)C(=O)NCC(C3CCCCC3)NC(C)C)(C1)C2 C1(NC(=O)CC2CCCN2CCF)CC2CC(NC(c3cc(O)nc(Cl)c3)=O)C2C1 Cc1ncn(CCNC(=O)CCN(C(=O)C2=CCSC2)CC2CC2)c1C Cc1onc(C(=O)NCC(C)CN(C(=O)CC2OCCO2)C)c1Br C#Cc1cnn(CC(=O)NCC(c2ccc(F)cc2)NC(=O)C(COC)SC)c1 N1(C(CCC=CC)=O)C(C(=O)NCc2nn[nH]c2C2CC2)CC2CC12 N1(CCC(C2CN(C(=O)Cc3cncc(O)c3)C2)C)CC2CCC1C2 CC(CN=c1[nH]c(=N)[nH]c(=NCC2COC(=O)N2)[nH]1)NC(=O)OC(C)(C)C c1(C(=O)NC(C(C)C)(C)CNC(c2cc(Cl)ns2)=O)ccc2nncn2c1 C(=O)(CCCCN=[N+]=[N-])NCCCCC(=O)NC(CCOC)C c1(NC(=O)OC(C(=O)NCCCCNC(C=CC)=O)C)ccccc1 c1(C(=O)NCC2C(NC(c3c(OCC)cccn3)=O)C2)ccc(C#N)c(F)c1 C(C)(CCCC(=O)NCC[Si](C)(C)C)NC(C(CC)n1cncn1)=O C1(CNC(N(C(c2ccccc2OC)C)CC)=O)CCCCNC1=O c1(C(N(C(C)CNC(c2cn(C3CCC3O)nn2)=O)C)=O)nc(Cl)sc1Cl C1(CSc2ccccc2)CCN(C(c2ccccc2)C(=O)N(S(C)(=O)=O)C2CC2)CC1 N1(C(C2C(C)(Br)C2)=O)CCCCC12CC(NC(c1ccc[n+]([O-])c1)=O)C2 C12(NC(C3N(C)CC3)=O)CCCC1N(C(c1nn(C)cc1Cl)=O)CCC2 O=C(C1=C(Cl)CCOC1)NCC12CCC(CC1)N(C(=O)C#CC1CCOC1)C2 c1(C(=O)NCC2CC(OC)CN2C(=O)C=C(C)Cl)cc2c(=O)cc[nH]c2s1 C12(C(=O)NCc3n(CC)ncc3)C(NC(C3CCC(=O)N3C)=O)C3CC1C2C3 C1(C(=O)NC(c2cncnc2)C)CCN(C(=O)CCC2CCC2)CC1O C12(C(N3CC(O)(CNC(c4nccc(C)c4N)=O)C3)=O)CC3CC(C(=O)N1)C2C3 C1(N(C(=O)NC(C2CCOC2)C)C)CCN(c2ccccc2)CC1 NS(=O)(=O)c1cccc(NC(=O)NC2CC(F)CN2C(=O)C2=COCCC2)c1 C(C)(CC(C)N=c1ccnc(CO)[nH]1)NC(c1ccc(N(CCC)CC)cc1)=O c1(OC)c(F)cc(C(=O)NC2C3CC(O)C2N(C(C2CC(F)C2)=O)C3)cc1Cl N1(C(c2ccc(C)cc2Cl)=O)CCN(C(=O)CN2CC(C)C2)C2CCCCC12 c1(C(=O)NCC(C)N(C)C(c2ccc[nH]2)=O)ccc(C2CCCO2)[nH]1 c1(C(N2CC(NC(C3(C)CC3)=O)C(C3CC3)C2)=O)cc2ccccc2cc1Cl N1(C(c2ccc(C(C)C)nc2)=O)CC2(CCCC2N(CC#N)C(=O)OC(C)(C)C)C1 CCCCC(C)CCC(=O)NCCCNC(c1ncnc(OC)c1F)=O c1(C(N2C(C)(C(=O)NCc3c(C)ccs3)CC2)=O)cc(Br)cc([N+](=O)[O-])c1Cl N1(C(c2cc(C)cc([N+](=O)[O-])c2)=O)CCCCC(N=c2ccc(C#N)n[nH]2)C1 C(=O)(CC(C)(C)CC(F)F)NC1CN(C(C2(C)CN(C)C(=O)C2)=O)CC1N=[N+]=[N-] c1(CC(N2C(CNC(C3CC(=O)N3)=O)CCC2)=O)c(Br)ccc(F)c1F N1(CC=C)CCN(C(=O)CC2COCCN2C(C2CCCN2C=O)=O)CC1=O C1(CC(=O)NCC2(O)CC(CNC(C3(SC)CC3)=O)C2)CC(O)C1(C)C C(C(=O)NCC1CC(F)CN1C(=O)C(O)C(F)F)(C(C)C)NC(C)=O CC1CC(NC(C2(CF)CCC2)=O)CN(C(c2c[nH]nc2Br)=O)C1 c1(C(=O)NCC2CCCN2C(=O)CSc2nncs2)ccn2nncc2c1 c1(N(CC(C)O)Cc2cccc(OCC)c2)ccnc(F)c1I N1(C(C(CC)NC(=O)CN(C)C)=O)CC2CCN(C(=O)CCSC)CC12 CC1CC(N=c2[nH]c3c(c(=NCc4ncn(C)n4)[nH]2)CCCCC3)C1 N1(C(CSCCCC)=O)CC2CC1CN2C(c1ccc(C2CCC2)nc1)=O CC1CCCCC1(CNc1ncccn1)NC(C1CS(=O)(=O)C1)=O C1(C(=O)NCC2N(C(CSc3n(C)nnn3)=O)CC=C2)CCC2(CCC2)O1 N1(C(C2C(F)(F)CCN(Cc3c(C)c(Br)cnc3)C2)=O)CCC2(CC1)CN(C)C2 c1(C(N2CC(NC(c3cnc(Br)o3)=O)C(F)C2)=O)cccc2cc[nH]c12 c1(OC)ccc(CC(=O)O)cc1S(=O)(=O)N(Cc1ccccc1)C.C(=O)(C(N)=O)O c1(C(N2CC(C)(NC(Cn3ncc(CC)c3)=O)C2)=O)ccc(N)cc1Cl C1(COC)CCC(=O)N(C(=O)CC2CCC2)C1.c12ncccc1OC2=O C1(CNC(C2CCN(C(C)=O)C2)=O)(CO)CCN(C(=O)Cn2cccn2)C1 C1(CC(=O)NCC(C2CC2)NC(=O)Cc2cccc(Cl)c2)CC2(CCC2)C1 N1(C(c2cc(OC)c(C)cc2)=O)C2CCC1CN(C(C1C(C)(C)C1(F)F)=O)C2 C#CCC(CC(=O)NC)NC(C1(C)COC(=O)N1)=O CC1(C2CCCN(C(c3ccc(-c4ccccc4)nn3)=O)C2)COC(=O)N1 c1(C(C(=O)N(C2CCCC2)CCNC(CSCCC)=O)F)ccc(F)cc1 C(CC(C)CCNC(=O)C=Cc1csc(C)n1)NC(C(C)(C)SC)=O C1(NC(CC(CCC)O)=O)CN(C(c2ccc(C)s2)=O)C2(CCCCC2)C1 CCC1=C(C(=O)NCC2(n3cccn3)CCN(C(C3CC3=C)=O)CC2)SCCO1 N1(C(c2cnnc(O)c2)=O)CC2CCC1C1CN(c3ncncc3Cl)CC21 c1(NC(C2CN(C(C(=Cc3cn[nH]c3)C)=O)C2)=O)ccc(F)c(F)c1 Cc1ccc(C(F)(F)F)cc1C(N1CCC(CC(=O)NCc2occc2C)C1)=O c1(NC(C(C)N(C(C(CCCC)C)=O)C2CCC2)=O)cnc2ncnn2c1 N1(C(CC)=O)CCOC(CS(=O)(=O)Oc2ccccc2)C1 CC1(C)Nc2ccccc2C1NC(c1ccccc1C(O)C(F)(F)F)=O Cc1cn2c(C(=O)NCC(C)N(C(=O)CCC3CC3C)C)cnc2s1 C1(C)(CC)CC(C(=O)NC(C)CN(C)C(C2(C)CCCN2C)=O)CCO1 Cc1[nH]nc(O)c1CN(C(C1CCN1C(=O)CCC1CCCC1)=O)C(C)C CS(=O)(=NC(=O)c1ccc2c(Br)cccc2c1)C1CC(C(=O)O)C1 CCCC(CCCNC(c1cnc(S)[nH]1)=O)NC(c1nccn1C(C)C)=O c1(C(=O)NCC(C2CCCC2)NC(C23CCC2C3)=O)cc2ccnc(Cl)c2[nH]1 c1(CC(=O)NC(C(=O)OCC)Cc2ccc(C#N)cc2)c[nH]c2cnccc12 C1(NC(C)=O)CCCC12CCC2.C1(=O)C(OC)CC(C(=O)OCC)N1C C1(C(=O)NC(C2CCN(C(C3SC4C=CC3CC4)=O)CC2)C)CC2C(C1)C2(C)C O=C1CN(C(c2coc(CO)c2)=O)C(C(N2CC(CCO)C2)=O)CN1 c1(OC)cc(C(N)C(=O)NC(C)C(Cc2ccccc2)OC)cc(OC)c1OC C(=O)(C(C(=O)NC(CC1CC1)CC(=O)NCCc1cccc(O)n1)OC)OC C(=O)(C1=CCN(C(=O)C(O)(C2CC2)C2CC2)CC1)N1CCC(C)(OCC)CC1 c1(C(N2CC(C)(CCC(=O)NCC(C)O)C2)=O)ccc(C#N)cn1 C1(NC(=O)CC2COCCO2)COC2(C1)CN(C(c1ccc(O)c(F)c1)=O)C2 C(C)(C(C)S(C)(=O)=O)NC(CC(=O)NC(C)=O)c1ccccc1 c1(C(N(CCCC)C)=O)ccccc1C(=O)NC(c1ccccc1C)CO CCC(CN=C(NC(C)C)N1CCC2(C1)Oc1ccccc1O2)CC(F)(F)F C1(NC(C2(C(=O)OCC)CCC2)=O)CS(=O)(=O)CC1NC(c1cc(C)[nH]n1)=O C1(C(=O)NCC(CNC(c2ccc(NC(N)=O)cc2)=O)OC)CS(=O)(=O)CCO1 Cc1nnc(C(C)(C)NC(C2CC2C(C)NC(c2c[nH]nc2C(C)(C)C)=O)=O)s1 C1(CNC(COc2cn(C)nc2)=O)CN(C(C2(F)CCCCC2)=O)CC1C(F)(F)F N1(C(CN(C)C(N)=O)=O)CCC2(CC(NC(=O)CC3CCCC34CC4)C2)C1 c1(C(=O)NC2(CNC(C3N(C)CCC3)=O)CCCC2)cnc(Br)c(N)c1 N#Cc1cncc(C(N2CCCN(C(=O)Cc3ccc(Br)s3)CC2)=O)c1 C=CC(O)C(=O)NC(CO)C(=O)NC1(CN(C)C)CCCC1 c1(OCC)cccc(CC(=O)NC2CN(C(=O)CSCCC#N)C3CC23)c1 C1(NC(c2cn(CCC=C)nn2)=O)CCCCC1CNC(C1(C)CC2CC2C1)=O N1(C(c2c(CC)nns2)=O)CCCCC1CCNC(C1SCCCS1)=O C1(C(N2CCC(C)(CNC(c3ccc(O)nc3)=O)C2)=O)CCc2ncccc2C1 c1(C(CC2CC2)NC(C2C(CNC(C3C(C)(C)C3)=O)CC2)=O)ccccc1 C(=O)(C(CNC(c1cnc(S)nc1)=O)C(C)(C)C)N(CCN(C)C)CC C(=O)(CC(C)NC(c1c[nH]c(=N)o1)=O)NCC(n1ccnn1)C CC1CCOC(C(N2CC(CC(C)NC(=O)C(C)(C)C3CCCO3)C2)=O)C1 C1(NC(c2cc(C)oc2C)=O)CC1C1CCN(C(=O)C(C2CC2)N(C)C)CC1 c1(C(=O)NC2CN(C(C3N(CC)C(=O)CC3)=O)C(C)C2)ccc2cccnc2c1 c1(C(=O)NCC2CN(C(c3cc(Cl)no3)=O)CC23CC3)ccc2ncsc2c1 C(N=c1[nH]c(=NCCC2=CCCCCC2)[nH]c2c(F)cccc12)C1(CC)CCC1 N1(C(c2c(OC)nccc2)=O)CC23CCCC2(C1)CN(C(c1nncs1)=O)C3 N1(C(CN(C)CC)=O)CCCC(C2CCN(C(C3(CF)CC4(CCC4)C3)=O)C2)C1 C1(C)(NC(=O)NCC(C(C)C)c2cccnc2)COc2ccccc21 C1(n2cc(NC(c3cccc(C)c3)=O)nn2)CC2CCC1CC2(C)O c1(C(=O)NC2CC(N(C(=O)COc3ccon3)C)C2)cc[nH]c1-c1ccccc1 CP(C)(=O)C1CCCCC(c2nnnn2-c2ccccc2)(NCC2COC2)C1 N1(C(c2cncc(C#C)c2)C(=O)NC(C)C(=O)OC)CC(N(C)C)CC(C)(C)C1 Cc1nc(Cl)cc(Cl)c1C(N1C2CC1CN(Cc1cnc[nH]1)C2)=O N1(C(c2ccc(OC)cn2)=O)CC2CCC(C1)N2C(C1(CC(F)F)CCC1)=O N1(C(C(CN(C)C)NC(C(C(C)O)N(C)C)=O)=O)CCC12CC(O)C2 c1(C(=O)NC(CC(=C)Cl)C(=O)N2CCC(C(F)F)C2)nccc2[nH]ccc12 Cc1cc(C(N2CCCC2CNC(C23CCOC(C)(C2)C3)=O)=O)c2c(c1)CCO2 c1(C(N2CC(CNC(C3CCCC3)=O)OCCC2)=O)cc(F)c(O)c(Cl)c1 C1(C(=O)NCC(CN(C(=O)CCc2ccc(CO)o2)C)(C)C)CCCC(C#N)C1 c1(C(=O)NCCn2cc(CC(=O)OCC)nn2)ccc(-c2ccsc2)nc1 CCC(CCCC(=O)N1CCCCC1C(F)F)NC(C1CCN(CC)C1)=O c1(-c2cn(CCC(=O)NC3C(F)(F)C34CC4)nn2)cccc(Cl)c1Cl CCC(CC)CC(F)C(=O)NC(C1CC(NC(=O)C(C)CC2CCC2)C1)C CC(O)(CC(=O)NCC1(C(N)=O)CN(C(c2cnn(C3CCC3)c2)=O)C1)C1CC1 Nc1cc2c(cc1C(N1CCOC(CCNC(=O)Cc3nc[nH]n3)C1)=O)OCO2 C1(C(N2C(C)CC(NC(c3cscc3Cl)=O)CC2)=O)CCC2CC1C2(C)C CN1CC(C(=O)NCCCOC2CCN(C(c3ccc(N)cn3)=O)CC2)CC1=O C1(CC)CCN(C(C2CCC2CNC(=O)COC2CC2)=O)CC1 c1(C(=O)NC2CC(NC(C3(C)CCC3)=O)C2)cc(=O)cc[nH]1 c1(OC)c(C(=O)OC(C)C(=O)NO)cc(Cl)cc1C c1(C(=O)NCCCN(C(=O)CN2CC(C)(C)C2)C)cnc2c(c1)NC(=O)CN2 C1(CC)CN(C(=O)Cc2ccc(F)cc2)CCC1NC(c1cc(C)nc(C)n1)=O C1(NC(Cc2nc(C(C)(C)C)sc2)=O)CN(C(C2(CF)CC2(F)F)=O)CC12CC2 C(C)(C(CC(=O)N(CCO)CC1CC1)NC(=O)CC1CCOC1C)OC Cc1cc2c(C(N3CCN(C(c4cc(O)c(Br)c(O)c4)=O)CC3)=O)nccn2n1 Cc1ncc(Cl)c(C(=O)NCC(C)NC(=O)Cc2ccccc2)n1 C1(C(N(C(CNC(COCCCC)=O)CC)C)=O)CCCCN1C c1(Oc2ccc(NC(=O)Nc3csnn3)cc2)ccc(Cl)cc1Cl c1(CN=C(NCc2ccc(N(C)C)cn2)NCC(F)F)cccc(OCCCC)c1 C1(C(N(CC(COCC)O)C)=O)CCCC1NC(=O)C=C1CCCCC1 n1(CC(N2CC(NC(COCCOC)=O)C(C)CC2)=O)cnc2sccc2c1=O C12COCCC1NC2=O.c1(C(N2CCC(C(=O)NC)C2)=O)cc(OC)nn1C CCC(CNC(=O)C(c1cn(C)nn1)NC(C1CCCN1C1CC1)=O)(CC)CC N1(C(CNC(CC)=O)=O)CCOC(CC(N2CCC(F)(CF)C2)=O)C1 N1(C(C2CC(C)C2)=O)CC(Nc2cc(O)ncn2)CC2(CCC2)C1 c1(C(=O)NCC(=O)NC(CNC(c2c(CC)non2)=O)CO)cccc(OC)c1 C1(CCNC(C2(C)CC(F)C2)=O)CN(C(=O)Cc2ccccc2O)CCS1(=O)=O c1(C(=O)NC2CN(C(C(C3CC3)SC)=O)CC2C)ccnc2c1ncn2C C12(C(N3CCC(NC(CC(CC)C)=O)C(O)C3)=O)CCC(CC1)C(C)(C)O2 CC1CCC(NC(c2csc(C(N)=O)n2)=O)CN1C(=O)COc1cccnc1 N1(C(CCCC2C(C)C2)=O)C(C(=O)N(C2CC3CCC2CC3)C)CCC12CC2 Cc1nc(=NC(CNC(c2cccc(C#N)c2C)=O)CO)s[nH]1 N1(S(C(CC)C)(=O)=O)C2CCC1CC(NC(c1ccc(OC(F)F)cc1F)=O)C2 CC1CCN(C(=O)CCC2CCOCC2)C1C(=O)NC1CN(C)CC1C N1(C(C(C2CC(C)(C)C2)OC)=O)CC2C(CNC(C3CCC4(CCC4)C3)=O)C2C1 c1(N(C)C)cncc(C(=O)NC2CCCC(NC(c3sccc3C(F)F)=O)C2)n1 N12CCN(CC1)C(=O)CSCC2.Cc1cc(C(=O)NNC(=O)CN)on1 CON=CC(=O)NCC1CCC(NC(=O)C(C)n2cccc2)C1 C1(NCCOCc2c(C)cncc2)CP(C)(=O)CC1O n1(CC(=O)NC2C(CNC(c3c(CC)con3)=O)CCC2)cc(C#N)cn1 CC(C)C(C)(O)C(=O)NC1CC=CCC1C(N1CCC(O)(C(N)=O)CC1)=O C1(COC)(CNC(=O)CCc2cn[nH]c2)CN(C(=O)COC2CC(F)(F)C2)C1 C(=O)(CC(F)(F)CS(C)(=O)=O)N1CC(C)C(CNC(=O)CC23CCCC2C3)C1 Cc1ccc(C(N2CCCC(N(C(=O)CCC3CCOC3)C)CC2)=O)cc1C N1(C(c2cnc(Cl)c(F)c2)C(=O)NC)CCC2(CCCCN2C)C1 C1(OC)C(NC(c2ccc([N+](=O)[O-])s2)=O)CN(C(=O)C(C)OCCOC)C1CO N1(C(CN(C)CC)=O)CCCC(C)C1CNC(c1ccnc(F)c1N)=O CC1=CCN(C(c2cnn(CC)c2)C(=O)N(C2CCC2)Cc2ccccc2)CC1 C1(C(N2CCCC(O)(CCNC(C=CC(C)(C)C)=O)C2)=O)CN(CP(C)(C)=O)C1 c1(-c2ccncc2)cnccc1SCCC1CCC1 C1(NC(C)=O)CC2CCC(C1)O2.C12CCCN(C1)CCn1cc2nn1 c1(C(=O)NCC(C)NC(c2cc(SC)c(F)cc2)=O)ccc2c(=N)[nH]cnc2c1 c1(NC)ccc(F)cc1C(=O)NC1(CCCNC(c2cc([N+](=O)[O-])c[nH]2)=O)CC1 c1(C(=O)NCC2(CNC(c3cc(C)n(C)c3)=O)CC2(F)F)ncc(N)cc1Cl C#Cc1cnn(C)c1C(=O)NCC1(CNC(C2(CC(C)C)CCNC2=O)=O)CC1 C12(NC(C3CCN(CC(C)C)C3)=O)COC(C1)C(NC(c1ccn(C)c1)=O)C2 c1(C(=O)NC)ccc(NC(C2CC23CN(Cc2c(Br)cnn2C)C3)=O)cc1 c1(CC)nc(C)oc1C(=O)N(C1CN(C(C2(C)CC2(F)F)=O)C1)C c1(C(=O)OC)cnc(C(=O)Nc2cccc(CO)n2)cn1 CC(C)C(C)(CNC(=O)C(C)C1(O)CCC1)NC(c1cn(CCO)nn1)=O N1(C(C2CCC(CC)CC2)=O)C2CCC1CN(C(C1C3CCC4C(C3)CC14)=O)C2 NS(=O)(=O)C1(C(=O)NCC2(NC(c3ccc(O)nc3)=O)CCOC2)CC1 C1(NC(c2c(=N)[nH]cnc2)=O)C2CCC1N(C(c1cccc(C3(C)CC3)c1)=O)C2 C(=O)(C1CCCc2ccnn21)NCC1CN(C(C2CC(=C)C2)=O)CC12CC2 N1(CC(=O)N(CC(CNC(C2C(CCOC)C2)=O)C)C)CCc2sccc2C1 c1(C(C(=O)NCCNC(N(C)C)=O)NC(=O)C(F)F)cccnc1 c1(C(N2CC(NC(CN(C)CC)=O)CC2(C)C)=O)cccc2c1OCC2 Cc1ccc(CC(=O)NCCCOCCNC(=O)CC2(C)CC2(F)F)cc1O C1(C(CO)NC(c2cocn2)=O)CCN(CCN2CCC2=O)CC1 CC1CN(C(C2CN(CC(F)(F)F)C2)=O)CCN1C(=O)C(F)C(C)(C)O N1(C(COCC(=O)OC)=O)CCC(C(=O)NCCc2cn(C)nn2)C1C c1(C(c2nnnn2CCCOCC2CC2)NC(C)CCO)c(Br)ncn1C N#CC1CN(C(=O)CC2CCC2)CC1NC(=O)C=Cc1cccs1 N1(CCC(=O)NCC(C)(C2CC2)NC(C(C)NS(C)(=O)=O)=O)CCCCC1=O c1(C(N(C)CC2(CNC(=O)CSc3nc[nH]n3)CC2)=O)cnn2c1CCC2 c1(N2CCCC(CN(C(C3C(C)(CC)C3)=O)C)C2)nc(Cl)ncc1OC c1(C(=O)NC2(CC=C)CN(C(=O)C=Cc3cccnc3)C2)ccc(CSC)cn1 c1(CC)oc2ccccc2c1CC(=O)NCC(O)CNC(C1CC12CCCC2)=O C1(NC(c2ccc(C)cc2)=O)CC2CC1CN2C(=O)COc1cccc(F)c1 N1(C(C2C(C(C)C)C2)=O)CC(NC(=O)CNC(=O)COc2ccccc2)C(O)C1 CCCC(C(=O)N1CCC1)N(C)C.C12CCN(CC1)C(=O)C(=O)NCCO2 C1(NC(c2scc(C)c2Cl)=O)CCN(C(c2cc(Cl)cc(Cl)n2)=O)C(C)C1 N1(C(Cc2c(C)nsc2)=O)CCOC(C(C)NC(=O)COc2ccsn2)C1 C1(C(N2CCCC(N(C(CC=CCC)=O)CC)CC2)=O)CN2CCCCC2CO1 N1(C(=O)COCC(F)F)CC2CCCC(C1)N2C(C1Cc2cccnc2C1)=O c1(OC)cc(CN2CCC(C)C2C)cc(C(=O)Nc2ccccc2)c1OC C12(C(=O)NCCN(C(CN(C3CCOC3)C)=O)C3CC3)C3C4C5C3C1C5C24 C1(N(C(C(CC=CC)NC(=O)CSc2cn[nH]c2)=O)C)CCCC(C)(C)C1 c1(CC(CC)C)nc(C(O)C2CC2)n(-c2ccc(C(C)C)cc2)n1 N1(C(CC2CCN(OC)CC2)=O)CCCC2CN(C(c3ccc(Cl)o3)=O)CCC12 N1(C(c2cc(C)n(C)n2)=O)CCN(C(c2ccc([N+](=O)[O-])n2C)=O)CC(CO)C1 C12(NC(COCC(=O)NC)=O)CCC(NC(C3COCCN3C)=O)(CC1)C2 C#Cc1cnc(C(N2C3CCC2C(NC(=O)C(C)CSC)C3)=O)c(C)c1 Nc1ccc(C(N2CC3C(C(=O)NOCCCO)C3C2)=O)nc1 CCCC(C(=O)NC(C1(O)CCN(C(c2ccnc(CO)c2)=O)C1)C)S(N)(=O)=O c1(C(=O)NCC(CNC(C2CCO2)=O)OC)[nH]c2ccccc2c1Br Cc1ncccc1C=CC(=O)NCCNC(C1(OC(C)C)CCCCC1)=O C1(NC(CCC=C=C)=O)CCC(C)(C)CC1CNC(c1cccc2c[nH]nc12)=O C1(N(C)C(C23COC(CF)(C2)C3)=O)CCCC(N(C)C(c2ncccc2F)=O)C1 c1(C(=O)NCC(C)(C)NC(C2CN3CCN2CC3)=O)ccc(Cl)c(N)c1 N1(C(Cc2c(C)ocn2)=O)CC2(CNC(c3c(O)cccc3F)=O)CCC1CC2 CC1CC(C(=O)NCCC2CCCC23CC3)N(C(c2cn(CCO)nn2)=O)C1 CC(C)CCC(O)C(=O)NCC(CC1CC1)C(=O)NC1(C2CCCO2)CC1 O=C(C(O)CCNC(C1(CO)CCCC1O)=O)NC12CC(F)(C1)C2 c1(C(C(=O)NC2COC2)N(CC)CC2CC2)cn(CC2CC2)nn1 Cc1cc(C)c2nc(N3CCC(C)C3CNC(c3ncccc3CO)=O)sc2c1 C1(C)(CNC(C2(CC)CCC2)=O)CCC(NC(=O)Cc2ccccc2F)C1 Cc1cc(C(=O)N(C)CCN(C(=O)C(CO)NC(=O)C(C)C)C(C)C)cn1C N1(C(C(CC2CCC2)OC)=O)CC(C(=O)NCC(C)F)C2(CC2)C1 N1(C(c2nn(CC)c(O)c2)=O)CCC(C2CN(C(C3CCC(F)CC3)=O)C2)CC1 c1(C(=O)NC(C2N(C(C=CC(CC)=CC)=O)CCC2)C)cc(C2CC2)cc(F)c1 c1(OC)cc(CCCNC(=O)NCC(C(=O)O)C2CCOCC2)ccc1Cl N1(C(C(C(C(C)C)O)C)=O)CC2CCN(C(c3nn(C)cc3[N+](=O)[O-])=O)CC2C1 c1(C(N2CCC(OC)(CO)C2)=O)cc2n(c1)CCNC2 c1(CCC=C)ccc(C(=O)N(C2CN(C(=O)CC3CC3)CC2O)C)cc1 CC(C)(C(=O)NCCC1COCCN1C(C1OC2CCC1C2)=O)C(F)(F)F C(CC(=O)NCC1CC2(CCC2)CO1)(C(C)CC)NC(CCC=CCC=C)=O c1(N2CCC(C)(SC)C2)nc(=NCCC(C)c2cn[nH]c2)[nH]c2ccsc12 C1(OC)C(OC)CN(C(=O)C(=O)C(F)(F)F)C1CNC(C1COCCN1C)=O C1(NC(CCC(=O)N(CCC)CC)=O)CN(C(=O)C2=CCOCC2)CCC1CO c12ccc(cc1)[nH]2.C1(C(=O)NC(CNS(C)(=O)=O)=O)CN(CCF)CC1F N1(C(CCSC)=O)CCCC2C1CCN2C(c1cc(-c2ccccc2)co1)=O C1(OC(c2cnc(S)[nH]2)=O)CN(C(=O)N(C2CCCOC2)C(C)(C)C)CC12CC2 c1(C(=O)NC2CC3(CCN(C(CC4CC(=O)C4)=O)C3)C2)ccc2nc(O)[nH]c2c1 CC(C)C(N=c1[nH]nc(C#N)s1)C(C)NC(=O)Cn1cc(C2CCC2)nn1 C1(c2n(CC(=C)C)nnn2)(NCc2cc(Br)no2)CC2CCCC12 CC(O)(Cn1ccccc1=O)C(=O)NC(CNC(c1csc(C(F)F)n1)=O)CO N1(C(C(CCC)NC(C)=O)=O)CCOC2(CCC(NC(c3cc[nH]c3)=O)CC2)C1 C1(NC(=O)CC2(CO)CC2)CCN(C(C2CN3CCCN2CC3)=O)CCC1CO c1(N2CCN(CC#CC)CC2)ncnc(N2CCC(CSC)C2)c1C N1(C(C=Cc2c(C)ccs2)=O)CCC(CNC(C23CCCC2CCC3)=O)C1(C)C c1(NC(C(C)NC(=O)NC2CCN(c3nccn3C)C2)=O)ccc(C#N)cc1 c1(C(=O)NC2CC(CC(=O)NC(c3ccccn3)CO)C2)cc(Cl)sc1Cl C(=O)(C#CC1CCCO1)N1CC(N(C(c2ccc(CC)c(F)c2)=O)C)C(O)C1 c1(OC)nc(Cl)ccc1C(=O)NC1CCCC(CN(C(=O)CNC=O)C)C1 c1(C(=O)NCC2C=CC(NC(CCS(N)(=O)=O)=O)C2)csc2ccc(F)cc12 c1(C(=O)NC2(CNC(COCCCC#C)=O)CC2)cnc2occc2c1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(C(C)NC(c2ccc(C(N)=O)cn2)=O)CC1 C1(C(=O)OC)CCCC1C(C)C.C(=O)(C(C)=C)OCC N1(C(C2N(CCC)CCC2)=O)CCC(F)(CNC(c2nocc2C(C)C)=O)C1 N1(C(c2ncn(-c3cn(C)nc3)c2)=O)CCN(C(c2cnns2)=O)C(CF)C1 N1(C(C2(Cc3cccnc3)CC2)=O)CCC2(CC1)OCCO2 C1(NC(CC2CCC(=O)N2)=O)CN(C(=O)CC2CC=CCC2)CC2(CC2)C1 N1(C(C=CC2(C)COC2)=O)CCC(F)(C(N2CCC(CC3CCC3)C2)=O)C1 C#Cc1cccc(C(c2nnnn2CCOC)NC(COC)CCO)c1F C1(O)(C(=O)NCC(=CC(=O)NC(C2(CO)CC2)C)C)CC(CF)C1 c1(C(N(CC(CN(C(C(C)CCN(C)C)=O)C)O)C)=O)cccc2ccsc12 CC(C)CCCC(C)NC(c1ccncc1NCc1cnc(N(C)C)nc1)=O c1(C(N2CC(NC(C(CC)F)=O)C(c3ccccc3F)C2)=O)cc(Cl)ccc1F c1(CNC(c2n[nH]cc2Cl)=O)ccc2c(c1)CCN(C(C1C3CCC(=O)C13)=O)C2 c1(C(N(CC(C)NC(C(C(CC)(C)C)O)=O)C)=O)ccc2c(C)cc(Cl)nc2c1 C(CCC(=O)NCC1CCC1NC(=O)Cc1ccn(C)c1)N(C(C)=O)C(C)C C1(CCNC(c2c(C)n(C3CCC3)nc2)=O)CC2CCC(C1)N2C(C1CCC1)=O C(N=c1[nH]c(=NCC(C)(C)CCO)c2ncccc2[nH]1)c1cc(C)oc1C c1(C(N(C2CN(C(=O)CC3CSC3)CC2O)C)=O)cnn2ccncc12 Cc1cccc(CCNC(C2(NC(=O)C=CCCC(C)C)CC(F)(F)C2)=O)n1 C1(C(=O)OC)CCC(C(N2CCC(CNC(=O)CC3CCCCC3)C2)=O)CC1 C(=O)(C1=NOC2(CCC2)C1)N(C1CCC(NC(=O)C(C)(C)C#N)C1)C CCCC(C)(CC)C(=O)NCC1C2CC1N(C(=O)C=Cc1cn(C)cn1)C2 c12cc(OC)c(Br)cc1OC2=O.C(=O)(CCSCc1ccco1)NCC(=O)OC Cc1cc(-c2noc(C(C3CCC(C)(C)CC3)(C)C)n2)ccc1I C(=O)(CCC[N+](=O)[O-])NC(CCCC)CNC(C1CCCN(C)C1)=O C1(C(N(CCOC)CCNC(C2CCCN2S(C)(=O)=O)=O)=O)CC1C1CCCCC1 N1(C(=O)C2=CCCCO2)CC2CN(C(=O)CCc3ccsc3)CC2C1 CC12CC1CCN2C(c1cc(CC2CCCCN2)on1)=O c1(N(C(CS(CC)(=O)=O)=O)C2CNCC2F)nc(C)nc2ccccc12 c1(CN2C(C(C)C)CN(C(c3cscn3)=O)CC2)c(F)c(F)c(F)c(F)c1F CC1CN(C(C2C3(CCC3)C23CCC3)C(=O)NCCCF)c2ccccc21 c1(C(=O)NCC(CC=C)NC(c2conc2C(C)(C)C)=O)c(OC)cccc1C Cc1cc(C(N2CCN(C(=O)C(C)N3CC(C)C3)C(CO)C2)=O)c(Cl)cn1 C1(C(=O)NC(C(=O)NC(CN(CC)CC)C)C)C2CCC(C2)C1C FC1(F)C(CNC(=NCC2SCCS2)NCc2cccs2)C12CCOCC2 C(=O)(CCCS(C)(=O)=O)N(C1CN(C(c2ccco2)=O)CCC1O)C C(=O)(C(F)C(F)(F)F)N(C)C(C1CC(N2CCCC2)C1)=O.C1(CC)CCCN1 N1(C(C(C=C)C)=O)CCC2(CC(NC(C3C4CCCC34)=O)C2)C1 C(CC(C(C)(C)C)NC(=O)Cc1cccs1)N(C(C(CC)C#N)=O)C c1(SCC)cncc(C(N2CCC(CNC(c3ccc(F)cn3)=O)(OC)C2)=O)n1 CCC(C)(C#N)C(=O)N1CCC(CC(=O)Nc2cnn(C3CC3)c2)CC1 Cc1cccc(Br)c1CN(C1CCC1)CC(C1CCCC1C)=O N1(C(c2cc(C)on2)=O)CC(C)OC2(CCN(C(c3cn(CCO)nn3)=O)C2)C1 C1(CNC(c2cncc(OCC)c2)=O)CN(C)CCN1C(c1ccc(Cl)[nH]1)=O CCCCCCCc1cn(CCCNC(c2ccccc2)Cc2nc[nH]n2)nn1 N1(C(CCC(=C)C)=O)CC2(CNC(C3CC(O)(c4ccco4)C3)=O)CCC1CC2 N1(C(C(CC)N(C)C)=O)CCCC2(CCC2NC(C2CC(CCO)C2)=O)C1 c1(CC(=O)NCCC(C)NC(C2(C)CC2(Cl)Cl)=O)c[nH]c2cccnc12 C(CC(O)C(=O)NCC1CN(C(=O)CCSc2nnnn2C)CC1C)SC N(C(=NCCCCl)NC1CCC(N(C)C)C1)CCCSCc1cc(C)on1 c1(C(N2CCCN(c3c(C#N)cccc3)CC2)=O)cc(F)c2c(c1)OCCO2 N1(CCCNC(=NC)NC2CN(C)CC2O)C(=O)c2ccccc2C1=O n1(CC(=O)N(CCCNC(=O)CC2CCCOC2)CC)nc(C)cc1C c1(C(=O)NCC2N(C(CC(C)n3cccc3)=O)CCC2)ccc(S(C)(=O)=O)[nH]1 c1(C(=O)NCC(CC)N(C(=O)CCc2ccc(F)cc2)C)cc(C)n(CCO)n1 C1(C(=O)NC(C2CCN(C(C3CC34CCC4)=O)CC2)C)CC(C)(C)CN1C c1(C(=O)NCC(C)(O)CNC(=O)C=CC(F)(F)F)cc(Cl)c(Cl)cc1N c1(CC)ccc(N)c(C(=O)NC2CCC2CNC(=O)C=CC2(C)CCOCC2)c1 N1(C(c2cc(COC)[nH]n2)=O)CCN(C)C(CNC(=O)CC2CCCO2)C1 C=CC1(NC(c2conc2CNC(=O)COC(C)(C)CC)=O)CCCCC1 c1(C(=O)NCCCCN(C(CN(C)C(N)=O)=O)C)ccc(F)c2occc12 Cc1cc(Br)c(I)cc1NC(C1CC1c1ccccc1C)=O C1(NC(c2n(C)nc(O)c2)=O)CN(c2cnc(C#N)cn2)CC2(CCC2)C1 C(=O)(CCCCCOC)N1CCC(N(CC#C)C(C2(COC)CCCC2)=O)CC1 C1(OC)CCCCC1C(=O)NCCC(C)N(C)C(c1cccc(CC(C)C)c1)=O CN=c1[nH]cc(C(N2CC(C(C(N3CCOC(C4CCC4)C3)=O)OC)C2)=O)o1 N1(C(c2nc(OCC)oc2)=O)CC(C)CN(C(=O)CC#N)C(C)C1 c1(C(=O)NC2CCN(C(C(CC=C)CC=C)=O)C2)cc2ccc(COC)cc2[nH]1 [N-]=[N+]=NC1(C(=O)NCc2ccc(O)cc2F)CCN(C(=O)CCCC2CC2)C1 c1(C(C(=O)NCC2CN(C(C3(C)COC3)=O)C2)OC)cccc(Cl)c1 C1(C(N(C2CSC2)C)=O)C2CC3C(C2NC(=O)C2=C(Cl)CC2)C13 C=CCC(C(=O)N(C(C)CN(C(=O)CCCc1ccc(O)c(F)c1)C)C)C(C)C c1(C(=O)NC(CC)CC)cccc(-n2cc(CCC3CCOC3)nn2)c1 C1(NC(C(CC=C)NC(=O)CC2CCOC2C)=O)CCCOC12CCC2 N(C(=NCCc1cnn(CC)c1)NC(C)C)CC.C12(CCC1)C(=O)N2 c1(C(C(=O)NC2CN(C(c3cnc(C)s3)=O)C2)O)cccc(F)c1 c1(OC)cc(C)ccc1C(=O)NC(C)CCNC(c1ccc(F)cc1O)=O C(=O)(CCC(=O)OC(C)(C)C)NCC(CC)NC(=O)Cc1nonc1C c1(C(=O)Nc2cc(C)cc(C)n2)cc2c(-c3cncc(O)c3)cccc2s1 CCCCC(F)C(=O)NCC1CN(C(=O)CCOC2COC2)CC12CC2 C1(NC(CN(C2CCCC2)C)=O)CCCC(NC(c2cc(Br)nn2C)=O)C1 N1(C(C2OCCC(NC(C=CC(C)(C)C)=O)C2)=O)CCc2ncsc2C1 Cc1ccc2nonc2c1C(=O)NCc1ccccc1CNC(=O)CCCCCO CC1CN(C(C2CCCC2CNC(c2cncnc2)=O)=O)C(C)C(C)(C)O1 N1(C(c2cc(C)sc2)=O)CC(NC(=O)C(C)Cn2cccn2)CC(F)C1 c1(C(=O)NCCOC2CCN(C(CC3CC(SC)C3)=O)C2)cc2c(s1)CCC2 C1C(C)(C)CC(=O)N1.Cc1cc(CCCCCN2CCOCC2)n[nH]1 C1(C(=O)NC2CN(C(CC)=O)C2)CC=CC(NC(C2CCN2C)=O)C1 c1(OC)c(C(N2CCN(C3CC3)C(C)C2)C(=O)NC2CCOC2)cccc1O c1(C(=O)NCC(C)CN(C(=O)CC2CCCCC2O)C)cn2cc[nH]c(=O)c2n1 c1(OC)cncnc1Nc1cccc(NC(C)=O)c1.c12nc(C)c(s1)c(=O)[nH]2 CC(C)C(CCN(C(=O)C(C)(C)C1CCCO1)C)NC(=O)C(O)CC1CCCC1 c1(C(=O)NC2C(C)CN(C(CCC#C)=O)CC2C)ccc(S(=O)(=O)CC)cc1 CC(C)CC(C)(C)C(=O)NC1CC(NC(c2ccc(Cl)c(F)c2F)=O)C12CCC2 C(CCC(C)C(=O)NCC(C(=O)NCc1ccns1)N(C)C)OC C1(C(=O)NCCN(C(COCC=C)=O)CCOC)CCc2ccccc2C1 C1(C(N(C)Cc2n(CCC)cnn2)=O)CCCN(C(C)CCOC)C1 N1(C(=O)C=C(Cl)Cl)CC2CC(NC(C3(C4CCCCO4)CCOCC3)=O)C1C2 c12nc(sc1Cl)N2.c1(C(=O)OCC)conc1SC.C12CCCC1OC2=O c1(C(=O)NCC(C)NC(c2cc(NC(C)=O)ncc2)=O)coc2c1CSC2 c1(C(N(CCn2cc(-c3cc[nH]n3)nn2)CC)=O)cc2c(OC)cccc2s1 c1(CC(=O)NC2(CNC(COCC)=O)CCOC2)n[nH]c2ccccc12 N1(CC(CCOCC)O)CC23CCCCC2(COC3)C1 c1(CC)noc(C(C)NC(=O)COC2CCOC2)n1 N(C(=NCCN(S(C)(=O)=O)C)NC1CCC1)C(CC)C.C12=CC=C(C=C1)C2=O C(=O)(C(CC)CCCCC)N1C(CNC(C(CC)=CC)=O)CN(C)CC1 c1(OCC(=O)NC2CCCCC2CNC(c2nsnc2O)=O)ccc(Cl)nc1 N#Cc1nccnc1N1CCC(CNC(c2ccc(-n3cncn3)nc2)=O)CC1 C(=O)(C1=CCC2CCC1N2C(c1cnn(C2CC2)c1)=O)N(C(C)CO)C C(=O)(C1COc2ccc(F)cc21)N1CCN(C(=O)CCc2cc[nH]n2)CC1CO CCCC(CC)CCC(=O)N1CCC(CNC(=O)C2=C(C)OCCS2)(OC)C1 c1(CC)oc(C(N2CCC2CNC(C2C(C)(C)C2(F)F)=O)=O)cc1C S(=O)(=O)(c1ccccc1C(F)(F)F)N1CCC(C(=O)Nc2cnn(CCO)c2)C1 C1(NC(C2(C=C)CCC2)=O)CC(OC)CN(C(c2nccn2CC)=O)C1 c1(C(CCO)NC(c2cscc2I)=O)ccccc1Br N1(C(C(C)(C)NS(C)(=O)=O)=O)CCC(C2CCN(C(C3(O)CCSC3)=O)C2)CC1 C(C(C)C(F)C(=O)NC1(c2cnc[nH]2)CC1)NC(C(C)OCC)=O c1(C(=O)NC(CCC(=O)NC(CC)COCC2CC2)C)cc(C)c(C)cn1 c1(OCCOC)ccc(C(N2CC(C(C)NC(C3CCCC3C)=O)C2)=O)cc1 C1(C2CC2)(CNC(Cc2c(C)ccs2)=O)CCN(C(=O)C(O)CN(C)C)C1 c1(OCCN(C)C)cccc(C(N2CCCC2(C)CNC(c2cnsn2)=O)=O)c1 C1(C(N2CCCC(OCCC)C2)=O)CC2CCC(C1)N2C(c1cc[n+]([O-])cc1)=O CON1CCC(CC(=O)NC(C)CCCNC(=O)CC23CC(C2)C3)CC1 n1(CCCC(=O)NC2CCC(CNC(CC3(C)CC3(F)Cl)=O)C2)ccccc1=O n1(CC(=O)N(C2CCN(C(=O)COC3CC3)C2)CC)ccc(Br)n1 c1(C(N(CCOC)CCNC(C2CCC3(CC3)C2)=O)=O)cc(F)c(C)cc1F c1(CC)cc(C(=O)NCC(COC)NC(=O)CCc2ccco2)n[nH]1 C1(C(=O)NCCc2c(C)n[nH]c2C)CN(C(c2cccc(=O)o2)=O)CC1(F)F C1(NC(CCC)=O)CC(F)(CNC(=O)COCC(N2CCCC2)C)C1 C12(C(N3CC(C(=O)OC)C3)=O)CCN(C(=O)C3=CCCC3)CC1C2 c1(C(=O)NC2CCCN(C(c3cc(COC)[nH]n3)=O)C2)ccc(S(=O)(=O)NC)o1 c1(N2CCC(SC)CC2)nccc(=NC(CCO)c2cccc(F)c2)[nH]1 c1(COC)cc(C(=O)NC2(CO)CN(C(=O)C(C3CCCOC3)OC)C2)cs1 C(=O)(C1=CCN(C(c2ccn(COC)n2)=O)CC1)NC(C#C)CC1CCC1 C1(C(C)C)CCC(C(=O)NC(C)C(C)(C)NC(c2cn(C)nc2C2CC2)=O)CC1 C#CCCC(O)C(=O)NC1C2CC1N(C(=O)C=Cc1cccs1)C2C N(C1CN(C(c2scnc2C(F)F)=O)CCc2ccccc21)C(=O)CSC1CC1 c1(C(N2CCOC3CN(S(=O)(=O)CCl)CC23)=O)c[nH]c2c(Cl)cc(Br)cc2c1=O Cc1nn(CC(F)(F)F)cc1NC(=O)C(N1CCC(CC(=O)N(C)C)C1)=O C=CC1CCCN(C(C2(C=C)CCN(C(c3cnncc3OC)=O)C2)=O)C1 c1(C(N(CCCNC(c2ccns2)=O)C(C)C)=O)cn(C)cn1 c1(C(N2CC(c3cccc(C(=O)O)c3)C2)=O)c(Br)nc2n1CCCC2 C1(OC)(CNC(=O)CC2COCCOC2)CCN(C(C2(O)CC2)=O)C1 c1(C(N(CC(C)NC(c2cc3scnc3[nH]2)=O)CC)=O)ccc2cncn2c1C C1(CNC(=O)CC2CCC2)CCCN(C2CC2)C1 C#CCCC(O)C(=O)NC1CN(C(=O)CCc2cc(Br)cs2)C1 C#CCCCCCCC(=O)N1CCC(N(C(=O)Cc2cnccn2)CC)C1 N1(C(c2c(C)c[nH]c2)=O)CC2CCC1CN2C(=O)Cc1c(C)ncnc1C c1(CCC(=O)NC(C)(CNC(c2coc(Cl)c2)=O)C2CCC2)cc(F)cc(F)c1 c1(CCC(C)NC(C)CC(C)N)ccccc1F c1(C(=O)NCCC(C)N(C(C(C)c2cncs2)=O)C)cc2cccc(F)c2o1 C(=O)(CC1CNc2ccccc21)NC1CCN(C(C=CC)=O)CC1 C1(C)(NC(CN2CCC(C)(C)C2)=O)CCC(NC(C2COCCO2)=O)CC1 C1(CC(=O)NC(C#C)(C)C2CCC2)CN(C(c2csnn2)=O)CCC1C C(C(C)(C)CC=C)NC(c1n(CC(=C)C)nnn1)C1CCSCC1 C#CC1CCCCN1C(C1(C)C=CCN1C(C1CCC1C(C)(C)C)=O)=O c1(CC)c(C(N2CC(CNC(=O)CSc3nncn3C)C(C)C2)=O)nnn1CC CC1CC(N=c2nc(C3CCOC3)[nH]s2)CCC1(F)F c1(NC(C2C(O)CCN(Cc3cc(C)c(Cl)nc3)C2)=O)nc2cc(F)ccn2n1 c1(C(N2CCCC(O)(CNC(C(CC)(C)C#N)=O)C2)=O)cc2cc[nH]c(=O)c2s1 C1(NC(c2c(CC)cno2)=O)CCCCC1NC(c1cnn(CC(C)C)c1C)=O CCCCC(C)CCC(=O)NCC1CC12CCN(C(=O)C=CC(C)(C)C)CC2 c1(C(N2C(CNC(C(C3CCC3)OC)=O)CCC2)=O)ccc(OC)cc1C(F)F C(=O)(C(O)CSC)N1CC(CC(=O)N(C2(C(=O)OC)CC2)C)C1 n1(CC(=O)NCCC2CN(C(C(CC)C(C)O)=O)C2)[nH]cc2c(=O)ncnc1-2 O=C(CS(=O)C(F)(F)F)NCCNC(=O)CC1CSCCO1 c1(OC)ccc(C(N2CCC(C)C(NC(=O)CCCSC(C)C)C2)=O)c(OC)n1 C1(C(N2CCC(N(C(=O)CC=CC(C)(C)C)C)C2)=O)C2CNC(=O)C12 C(CC(CC)C(=O)NC(C)(CSC)C(=O)NCCC1(C)CCOC1)=CC c1(C(=O)NCCN(C)C(C2CCNC(=O)C2)=O)ccnc(OC2CC2)c1 Cc1nn(CC(=O)NCC(C)(CO)NC(=O)Cc2cnc[nH]2)cc1Cl c1(C(C(=O)NC)N(C)CCc2ncc(C)s2)ccc(C)cc1 CC(=O)CCC(=O)N1CC2CC2C1C(=O)NCCC(=O)NO C(=O)(C1=CCCC1)N1C(C)(CC(N2CCC(OCC)C2)=O)CC1 CC1(CNC(c2cccnn2)=O)CCC(NC(c2cc(C(F)(F)F)ns2)=O)CC1 c1(OC)cc(C(=O)NC2CCCC(CNC(c3cccc(F)c3)=O)C2)cc(C)n1 Cc1cc(C(=O)NCCN(C(=O)C(F)(F)CO)C(C)C)cnn1 Cc1ncc(CNC2C=CC(C(=O)NCC3CC3)C2)[nH]1 CCC(C)(C)CC(=O)NC(C)(CNC(=O)CCCc1cc(O)ccc1C)C1CC1 C(=O)(CCCCCC(C)(C)C)N(C1CN(C(C2CCC(C)O2)=O)C1)C c1(C(N2CCC(C)(NC(c3ccn(C)n3)=O)C2)=O)ccc2c(c1)CCC=C2 C1(NC(c2c(CC)cncc2)=O)CC2(NC(C3CC=CCC3)=O)COC1C2 O=C(C1=CCOCC1)NCCC1(C(N2CC(O)(C(F)(F)F)C2)=O)CC1 C#CC1CCCN(C(=O)CCC2CC(NC(C3CCCOC3)=O)C2)CC1 c1(CC)nn(C)c(C(=O)NCC2CC(NC(c3cc(OC)ns3)=O)C2)c1Cl CCCC(C)(C)C(=O)NC1CN(c2nnn(C)n2)C1 N1(C(C(CNC(C2C(C)C3CCC2C3)=O)CC2CC2)=O)CC(C2CCCCC2)C1 O(NC(=O)CCOC1CC(NC(C2CCCO2)=O)C1)CC CC(C)C(C(=O)N1CCCCC(CNC(=O)C(F)(F)C(F)F)CC1)C(C)C C1(c2cn(CCN(CC)CC)nn2)CCN(C(=O)CC2(C)CCCC2)C(C)C1 CC(C)(CCS(C)(=O)=O)NC(c1cc(C(N)=O)cs1)=O C12(C(CNC(CC3N(C)CCC3)=O)NC(=O)CC3CC3(Cl)Cl)CCC(CC1)C2 CCCCC(O)C(C)C(=O)N1CCC(NC(=O)C=CC2CCCN2C)C(C)(C)C1 c1(C(=O)NC(CCC)CC(=O)NCCn2nc(C)nc2C)ccc2cncn2c1 CC(O)C(F)(F)C(=O)NC1CC(NC(C2(c3ccccc3F)CC2)=O)C1 c1(C(N2CC(NC(c3ccc(Cl)cn3)=O)C(F)C2)=O)cccc2c(Cl)ccnc12 c1(C(N2CCC(CNC(C3CC3C(F)(F)F)=O)C2)=O)ccncc1Br c1(C(N2CCC(O)(C(C)NC(CCCOCC)=O)C2)=O)cc(Cl)ncc1F C(=O)(C(F)(F)C(C)(C)O)NC(C)C(CCc1ccccc1)NC(=O)CCCF CC(C)(CCNC(=O)C1=CCCC1)C(=O)NC1CCC(C(N)=O)CC1 CC(C)CCCC(C)NC(=O)N(C1CCN(Cc2cnc(C3CC3)o2)C1)C C1(NC(C2(C3N(C(CCC=C)=O)CCC3)CC2)=O)CCC(C)CC1 CC1(C)CN(C(c2cnn(C3COC3)c2)=O)CC1NC(=O)CCn1cc(Cl)cn1 C1(C(=O)NC2CCCC2CNC(c2nc(Cl)oc2C)=O)(OC)CCSCC1 C1(NC(Cc2c(C)ncs2)=O)CCN(C(=O)Cc2cncn2C)CC1F CC(CNC(C1CCC1c1ccccc1)=O)C(=O)N(C)C C(C(COC)CC(=O)N(C(C)CCNC(c1cccc(=S)n1O)=O)C)OC C1(CNC(CCOCCC)=O)CCC(C)N(C(=O)CSc2cn[nH]c2)C1 CCC(C(=O)N1CCC2CC12C(=O)NCCCN(C)C)C(F)(F)F C1(CC=C)(NC(c2ncccc2F)=O)CCN(C(=O)CSCC2CCCC2)CC1 c1(OC)cc(CC(=O)NC(C2CN(C(C3CCCCC3(C)C)=O)C2)C)ccc1Cl N1(C(c2c(CC)c[nH]c2)=O)CCC(C)C(CC(=O)N(C)CCN2CCCCC2)C1 Cc1cn2cc(C(N3CC(NC(c4cc[nH]c4C)=O)CC(F)C3)=O)sc2n1 N1(C(C2CC(=O)NCC2)=O)CC2(C(=O)NCCC(F)(F)F)CCC1CC2 CC(C(=O)N1CCN(C(c2cnn[nH]2)=O)CC1C1CC1)S(=O)(=O)C1CCOCC1 C1(c2n(CC=C)nnn2)(Nc2cnc(OC)c(Cl)c2)CCCCC1CN(C)C C(=O)(CCC(C)(C)C)NCC(CCCC)NC(c1ccc(OC2CC2)cc1)=O C1(C(=O)NC2CC(CNC(c3c(CCC)nsc3N)=O)C2)CCOCC1(C)C N1(C(=O)CC2CC2)CCC(C(F)(F)F)C(Nc2nccc(C(F)F)n2)C1 C1(NC(c2nc(NC(C)=O)sc2)=O)CC(O)CN(C(c2nnc(S)n2C)=O)C1 C1(C(N2CC(NC(c3c(C)cno3)=O)C(O)C2)=O)CCCCN1N=O c1(CC(=O)NCC2N(C(C(CC)N(CC)CCCCC=O)=O)CC2)ccc(C#N)nc1 c1(SC)nc(N2CC3(CC(CC(=O)Nc4ccc(CO)cc4)C3)C2)ncc1Br C(=O)(C(C(C)C)N(C)C)NC(C(C)C)CNC(=O)CCc1cncn1C CC1(C)CC(NC(C2CCOC2=O)=O)CN(C(c2ccsc2Cl)=O)C1 O=NN1CCCCC1C(=O)NCC1CCCCN(C(c2cn(C(F)F)cn2)=O)C1 N1(C(c2cn3nc(C)sc3n2)=O)CC(C(=O)NC2CCCCC2)CC2OCCC12 C1(CNC(C(N2CCC(C)(CC#N)C2)=O)=O)CC2(C1)CC1(CCC1)C2 c1(C(N2CCCC(CCNC(C3CCC(O)C3)=O)C2)=O)ccc(F)c(Br)c1 CCC(C)CCC(=O)N1CCCC1CN(c1cc(C)cnc1C)C.C(=O)(C1CC1)N N1(c2cc(NCC(CC)(C)C(N)=O)nc(COC)n2)CCn2ncc([N+](=O)[O-])c2C1 C1(CCC(=O)N(C(C)(C)C2(C(=O)O)CC2)C(C)C)CCCCO1 N1(C(C2(COC)CN(C(C3CCC(=O)NC3)=O)C2)=O)CC(C)(C)C2CCCC12 CC(C)CC(C)(CN=c1ccnc[nH]1)NC(c1cnc(C(C)(C)C)o1)=O CC1Oc2cc(-c3nnc(-c4ccon4)o3)ccc2NC1=O n1(C(C)C(N2CCC(C)C(NC(C3CCC(C)C3)=O)C2)=O)cnc2ccccc12 N1(C(CC2CN(C(C3(C=C)CCC3)=O)CC23CC3)=O)CCCN(C)CCC1 c1(C(=O)NCC(C(C)C)NC(CCC(C)=O)=O)ccc2cnc(C)cc2c1 c1(C(CNC(CSCC)=O)NC(C2CC=CCO2)=O)ccc(F)cc1F N1(C(C2(CC)C=CCC2)=O)CC2(C1)CN(C(=O)CSc1n[nH]c(C)n1)C2 CCC(F)(F)C(C)(C)C(=O)NC1CCCC(CN=c2cc(Cl)nc[nH]2)C1 C(CC(C)(C)C(=O)NCC(C)C(=O)NCC1(O)CCCCC1)SC c1(C(=O)NCCCCCNC(C2CCC2)=O)cn(CC(F)(F)F)cn1 c1(C(N(C2CC(NC(C(C)c3cc[nH]n3)=O)C2)C)=O)cnc(-c2cccnc2)s1 C1(C(NOCC(=C)Cl)=O)(CC)CCN(C(c2cncc(OC)n2)=O)C1 Cc1ccccc1CC(N1CC=CC1CNC(=O)CCN1CCC(F)C1)=O C=C(C)C(C)(C)C(=O)N1CCCC(F)(C(=O)NCC(C)CC(F)(F)F)C1 N1(C(c2c(C)sc(O)n2)=O)CCCCC(NC(C2(CC(C)=O)CCCC2)=O)C1 N1(C(c2c(C#C)cn(C)n2)=O)CC2(CC(C(=O)N(CC(O)CO)CC)CO2)C1 N1(C(COCCSC)=O)CCCCCC(Nc2ccnc(-c3ncc[nH]3)c2)C1 N1(C(c2c(C)noc2)=O)CC=CC(C(=O)NC(C)C(F)(F)F)C1 CC(CCO)N=c1[nH]c(N2CCCCC(CO)C2)nc2c1COC2 C1(CC(=O)N(CC(CN(C(=O)CC2CC3(CC3)CO2)C)O)C)CC(C)(C)CO1 C1(C(C)C(=O)NCC2=CCCC2)CCN(C(=O)C(C)c2ccco2)CC1 C(CNC(C1(O)CCSC1)=O)(CC(=O)NC(C(O)CO)C1CC1)OC N1(C(C2N(C)C(=O)OC2)=O)CC2(C1)CN(C(C1CC3CCCCC13)=O)CCO2 C#CC1CN(CC(=O)Nc2ccc(C)cc2Br)CC1O Cc1cccnc1C=CC(N1CCC(NC(c2ccnnc2S)=O)CC1C)=O C(=O)(C1=NN(C)C(=O)CC1)N(CC(=O)N(CCCCC)Cc1cncnc1)C C=CCCC(CC(C)C)C(=O)N(CCNC(=O)Cc1csc(C(C)(C)C)n1)CC c1(COCC)cccc(CNC(=O)CC(O)Cn2cc(-c3ccccc3)nn2)c1 C#CCCCCCCCC(=O)N1CC(O)(C(C)NC(C)=O)C1 Cc1cccnc1CC(=O)N(C1CN(C(c2c(CO)noc2C)=O)CC1F)C S(=O)(=O)(c1c(C)cccc1Cl)N1CC(NC(C2N(C(C)=O)CCC2)=O)C(C#N)C1 n1(CC)cc(C(=O)NC(C2CC(NC(=O)C(COC)NC(C)(C)C)C2)C)c(C)n1 c1(C(=O)NC(CC)CN(C(=O)C(C)n2cncn2)C)cccc(C(F)(F)F)n1 n1(CC)c(C)nn(CC(=O)NCCN(C)C(c2ncc(Br)cn2)=O)c1=O CC(C)(CC(F)F)C(=O)NCCCCN1CCCN(C(C2CC(O)C2)=O)CC1 C(=O)(C1=CCCSC1)N1CC(CCCCNC(CC2(C=C)CCC2)=O)C1 C12(C(N(CC(C)(C)NC(c3ccnn3C3CC3)=O)C)=O)CCC(C(F)F)(CC1)C2 C12(CC(=O)N(C(CCNC(c3n(CC)ncn3)=O)C)C)CCC(CC1)CC2 Cc1ncnc(O)c1C(=O)NC1CC2CC(NC(C3(C(F)(F)F)CC3)=O)C2C1 Cc1cccc(F)c1CC(=O)NC1CCN(C(=O)Cc2cnn(C)c2)CC1CO N1(C(c2c[nH]c(=N)o2)=O)CC(=O)N2CCOCC2(CNC(=O)COC(F)(F)F)C1 CC(CN(C)C)CCC(=O)N1CC(CC(=O)NC2(CO)CCC2)C2(CC2)C1 C1(NC(C(C)OCC)=O)CCC(NC(=O)CC2CC(F)C2)CC1 N1(C(=O)C(F)Cc2ccccc2)CCN(C(c2cnc(Cl)s2)=O)C(CCO)C1 c1(C(N(CCN(C(=O)CC2(N(C)C)CCC2)C)C)=O)ccc(=O)n(C)c1 CC(C)CC(O)CC(=O)N1CSCC1C(=O)N(C(C)C(C)C)C1CC1 C(C)(C)(CCCCC(=O)N1CCN(C(=O)CC2=CCCC2)C(C)C1C)OC C1(NC(CCC(C)(C)NC(=O)C2=CCCCC2)=O)CCCCCCC1O C1(C(N(CCC(C)NC(CCOCC)=O)C)=O)Cc2cc(C)ccc2S1 c1(C(N2CC(O)(CNC(c3cccc(C)c3F)=O)C2)=O)cnc2c(F)cccn12 CCCCCCCC(F)C(=O)N1CC(CNC(=O)Cc2cc(C)no2)C(C)(C)C1 C1(CC(=O)NCC(C)(C)CCNC(=O)C=Cc2ccccc2)CC(=O)NC(=O)C1 N1(C(C2N(C(CC)=O)CCCC2)=O)CCN(C(=O)C#CC(C)(C)C)C(CCO)C1 C1(NC(C2CCCS2)=O)CC2CCC1CN(C(c1nccc3c1NCCC3)=O)C2 N1(C(C2(CC(C)C)CCC2)=O)CC2CC(NC(=O)CCc3cn(C)nc3C)C2C1 c1(C(=O)NC(C)CNC(c2occc2-c2ccccc2)=O)ccnc2[nH]nnc12 Cc1cc(CC(=O)NC2(CCNC(=O)CCSCC3CC3C)CC2)sn1 c1(C(c2n(CCCC)nnn2)NCCS(=O)(=O)N(C)C)ccc(C)nc1 N1(C(C(C2CCCC2)OC)=O)CCC(CNC(C2CN(C)C2)=O)C(O)C1 N1(C(c2c(C)c(=O)cc[nH]2)=O)CC2(CCN(C(c3c[nH]c(=N)s3)=O)CC2)C1 C(C)(C)(CC(=O)NCC(C1CCN(C(=O)C(F)=C2CCCC2)CC1)C)OC N1(C(C2CC2(F)F)=O)CC(NC(C23CC2Cc2c[nH]nc23)=O)C2CCCC12 N1(C(c2sc(C)c([N+](=O)[O-])c2)=O)CC2CN(C(=O)CC3CC(=O)C3)CC2(C)C1 c1(NC(C2N(C(c3nccc(CC)c3)=O)CCC2C)=O)ccc2cnccc2c1 c1(C(N2CC(NC(C(C)c3ccsc3)=O)C(C)C2)=O)ccc(N)c(Cl)c1 c1(C(=O)NC2C(NC(C3CN(C(C)C)C(=O)C3)=O)CCC2)ccc2cc[nH]c2n1 c1(C(=O)NCCN(C(=O)CN2CCC(O)CC2)CC)nc(=N)cc[nH]1 C(C)(CN=c1[nH]c(N2CCC(CS(N)(=O)=O)C2)nc(=N)[nH]1)(C1CCOCC1)OC CCCCCCC(C)NC(=NCCc1ccc(Cl)cc1Cl)NCc1[nH]nnc1C C#CCC(CC(=O)NCCCCC1CC1)NC(=O)CCCC(=C)C C1(NC(CSCC(=O)OC)=O)CCN(C(C2(C(C)(C)C)CCC2)=O)CC1 C(=O)(C1Cc2ccccc21)NC(CN(C(C(C=CC)O)=O)C)(C)C Cn1cc(C(=O)NC(C)(C)CNC(=O)CC2CSC2)c(OCCCS)n1.CC#N N1(C(C2N(C(CC3(C(=C)F)CCC3)=O)CC=CC2)=O)CC2(C1)CC(C)(C)C2 c1(C(N2CC(CNC(C3CC(C)(C)C3)=O)C3C2C3)=O)ccc2nc(S)[nH]c2c1 n1(C(C)C)cnc(CNC(c2coc(CNC(=O)C(C3CCCCC3)C)c2)=O)n1 NS(=O)(=O)CCCCNC(c1ccc(C(F)(F)C(F)(F)F)cc1)=O c1(OC)ccc(C=CC(=O)NCCC(C)NC(c2ccc(F)c(F)c2)=O)cc1 c1(CC)c(C(=O)NCCOC2CCN(C(=O)C(O)C3CC3)CC2)nnn1CC C(=O)(C(O)CC(F)(F)F)N1C(C(=O)NC2CN(C)C(=O)C2)CCCCC1 N1(C(C(=CC2CCCC2)C)=O)CC2CC1C2NC(=O)CC1CNC(=O)O1 C(=O)(C1=Cc2ccccc2OC1)NCCC1N(C(C(CC)C)=O)CCCC1C N1(C(c2ccn(CC(F)F)n2)=O)CCOC2(CCN(C(C3CC=CCC3)=O)C2)C1 Cc1ccc(F)c(C(=O)NC(CC(=O)N(C2CC3CCC2O3)C)C2CC2)c1 c1(C(=O)OCC)ccc(C(=O)NN2CCC2CF)cc1 C12(C(=O)NCc3c(CCNC(C4(CC(C)=O)CC4)=O)ocn3)CCCC1C2(F)F c1(NCC(=O)NC2C(CNC(=O)CCOC3CC3)C2)ccc2ncsc2c1 C#CCC(C(=O)NCCCc1ccco1)NC(=O)C=Cc1ccccc1 CC1CC=C(C(=O)NC2(CO)CCN(C(=O)C=CCN3CCCCC3)C2)CC1 c1(-c2n(CC)ccn2)cc2ccccc2nc1C(=O)NCC1CCC(CO)CC1 C(CC(F)F)(C(=O)N1CC(CO)C(O)C1)N(C(C=CCC)=O)C c1(C(=O)NC(CNC(CNc2cc(C)oc2C)=O)C)cc(Cl)ccc1C(C)C c1(C(N(CC(C)(C)CNC(=O)C(=O)NCC)CC)=O)cc(OC)c(C)c(OC)c1 N1(C(c2cc(C)ncc2C)=O)CCCCCC(NC(=O)C(C)CC(N)=O)C1 C(c1ccc2[nH]ccc2c1)=CC(=O)NCC(C)NC(C1(C#C)CC1)=O c1(CNC(CCN(C(C=CCC)=O)CCO)=O)ncnn1C1CC1 c1(CNC2C=CC(C(=O)Nc3ccc(C)cn3)C2)cc(F)cnc1Cl N1(C(C(c2cn(C)nc2)(C)C)=O)CCN(C(C2CC2F)=O)C(CO)C1 O=C(C1=CC2C=CC1C2)NCc1ocnc1C(=O)NC1CCCC1(F)F n1(CC(=O)NCC2(NC(CC(C)(C)O)=O)CCOC2)cnc2c1CCCC2 c1(COC)cncc(C(=O)N(C2CC(NC(c3cc(Cl)cnn3)=O)C2)C)c1 C12(C(=O)NCC3C(NC(=O)Cc4cscn4)CCC3)CCC(C(F)F)(CC1)CC2 N1(C(CCCCNC(C2=NOC(C)C2)=O)=O)CCC2(CCOC2=O)C1 Cc1cc(C)c(CC(=O)N(CC(C)CNC(=O)Cc2nc(C)sc2C)C)c(C)c1 Cn1ncc(C(=O)NC2(CCNC(c3cn(C(F)(F)CO)nn3)=O)CC2)c1C#N C1(CC=C)(NC(=O)CCNC(c2ccsc2)=O)CCN(C(=O)C=C(C)C)C1 c1(C(=O)O)cc(Br)ccc1NCc1cccc(C(F)(F)F)c1 Cc1ccc(C=CC(=O)NC2COCC2NC(=O)Cc2cnns2)c(C)c1 N1(C(=O)Cc2cnns2)CC2CCC(C(N3CCOCC34CC4)=O)(C2)C1 c1(C(=O)NCCN(C(=O)Cc2cnnn2C)CC)ccc2nc(O)[nH]c2c1 C1(CNC(c2c(OC(C)C)cccc2)=O)CC2(C1)CN(C(C1CS(=O)(=O)C1)=O)C2 c1(CS(C)=O)c(C(=O)OCC(C2CCC(F)(F)CC2)=O)oc2ccccc12 N1(C(C(C(CC)O)C)=O)CC2CCCN(C(=O)CSc3cccc(F)c3)C2C1 CC12CC(C(=O)NC3CC3CNC(c3nc(C4CC4)cs3)=O)(CCO1)C2 c1(C(=O)Nc2cc(I)ncn2)cc2c(-c3ccc(CO)o3)cccc2s1 c1(CNC(CCC2N(C(C3CCN(C)CC3)=O)CCC2)=O)ccc2ocnc2c1 O=C(N=c1[nH]oc2cccnc12)C1CN(Cc2ccc(F)c(Br)c2F)CCO1 c1(C(N(C(C)CNC(=O)Cc2nc(C)sc2Cl)CC)=O)csc(=NC)[nH]1 N1(C(CCCC(N)=O)=O)CCCCC2(CCN(C(=O)CCN3CCCC3=O)C2)C1 c1(C(N2CC(N(C)C(C34CCC3C4)=O)C(O)C2)=O)ccc(Br)cc1F c1(SC)ccc(Cl)c(NCC2(C)CC2)c1.C12(F)CC(C1)NC2=O.C12(CC1)C(=O)N2 c1(C(=O)NC2(CNC(c3c(-c4n(C)ncc4)nn[nH]3)=O)CC2)cc(N)ccn1 c1(CC)oc2ccccc2c1CNC(=O)N(C)CC(c1cc(OC)ccc1F)C c1(C(N2CC(NC(C(CC=C)(F)F)=O)C(OC)C2)=O)cc(S(=O)(=O)NC)cn1C C1(C)(C(c2n(CC)nnn2)Nc2ccc(SC)cc2)CCCCCC1 c1(OCC)ccc(C=CC(=O)NCC2CCN(C)C2C)cc1C C(C(C)(C)CC(=O)NC(C)(CO)C(C)(C)O)NC(CCc1n(C)cnn1)=O N1(C(CN(CC)CC)=O)CC2(CCN(C(C3CC4C=CC3C43CC3)=O)C2)C1 N1(CC)N=C(C(=O)N2CC(N(C(=O)CCCC3CCCC(=O)N3)C)C2)CCC1=O N1(C(=O)NCC(c2ccc(F)cc2)(F)F)CC2C(C(F)(F)F)CC2(C(=O)O)C1 N1(C(CNC(CCC(C)C)=O)=O)CC2CCCC2(NC(C23CC(C)(C2)OC3C)=O)C1 CC1(C)CC(NC(=O)COCC2CCOCC2)CN(C(c2cncc(N)n2)=O)C1 CCCC(CNC(=O)CC1CCN(C(C2(C3CC3)CCCO2)=O)C1)CCC c1(OC)nccc(CNC(C2CCC2CNC(=O)CC2(O)CCOC2)=O)n1 N1(c2n(CCC3CC(C)(C)OCC3)nnn2)C(CO)CC2CCCCC12 C1(NC(C2N(C(=O)NC3C(OC(C)C)C3)CCC2)=O)CCCC12OCCO2 CC1(C)CCCC(CC(=O)NC23CC(C2)N(C(c2cccc(Cl)c2Cl)=O)C3)C1 C(CCCCCNC(c1cn(CC(N)=O)nn1)=O)N(C(CN(CCC)C)=O)CC C(C(CC1CC1)C(=O)N(C(C)COC(C)C)CCOC)NC(CSC)=O c1(C(=O)NCC2CN(C(C3C(=C)C3)=O)CC2c2cncn2C)cccc(Cl)c1C C1(CNC(C(C(C)C)C)=O)CN(C(=O)CCN(C)C(=O)OC(C)(C)C)C(C)(C)C1 C1(=O)C(C)(C)C(C)N1.C(=O)(CCCNC(C)=O)N(C(C(C)SC)C)C c1(C(c2nnnn2CC)NCc2n(CC)cnc2)cccc(S(C)(=O)=O)c1 c1(C(N2C3CC(NC(C4CCCCC4)=O)(C3)C2)=O)ccc2ccoc2c1 C1(NC(c2cc(C(F)F)[nH]n2)=O)CC2(C1)CN(C(c1coc(Br)n1)=O)C2 C1(C(N(C)CC2(NC(c3cn(CCC(C)C)nn3)=O)CC2)=O)CC2CC1CO2 C12(NC(CN(CCC)C)=O)CCCN(C(c3ccc(Cl)nc3O)=O)CC1C2 CCCC(CC)C(=O)NC1CN(C(c2sccc2F)=O)C(C)(C)C1 N1(C(CC=CC=CCC)=O)CC(C(=O)Nn2ccnn2)C(C)(C)C1 C#CCC(C(=O)NOC(CC)CC)NC(=O)CCCCCC c1(C(=O)NCCC(C)NC(=O)CN(c2ccncc2)C)c(N)cc(Cl)cc1F Cc1sc(N)c(C(N2CC3CCC3(CCNC(=O)C3=C(Cl)CC3)C2)=O)c1C N1(C(C(CC)C#N)=O)CCC(N=[N+]=[N-])(C(=O)Nc2cccc(C)c2C)C1 C1(C)(C(N(CC(C)NC(C2(C)CCC(=O)C2)=O)C)=O)CCS(=O)(=O)CC1 N1(C(C(C(C)(C)O)F)=O)C(C(=O)NC2COC(C(F)F)C2)C2CC(O)C1C2 c1(COC)nn(C)c(CN)c1CC(N1CCCC1)=O.C12(CCOCC1)C(=O)N2 CCCCC(C)(F)C(=O)N1CCC(C2CC2)(NC(=O)CCC2CC(F)(F)C2)C1 CC1CCC(NC(=O)CSC2CC2)CN1C(=O)CCc1ccccc1C(F)(F)F c1(C(=O)NCc2cccc(Cl)c2)n[nH]c2ccc(-c3ccnn3C3COC3)cc12 c1(C(C(=O)NCC2N(C(CCOC(C)C)=O)CCCC2)O)ccc(Cl)c(Cl)c1 c1(NS(C)(=O)=O)cccc(NCC2C=CCCC2C(F)(F)F)c1 Cc1nc(C)n(CC(=O)N(C(C)CN(C)C(C2(Nc3ccccc3)CC2)=O)C)n1 c1(CC)ccc(S(=O)(=O)CCOC(=O)CCN(CCCO)C(C)C)cc1 C1(C(=O)NCCCCN(C)C(C2(F)CC=CCC2)=O)CN2CCC1CC2 c1(CNCCNC(c2cccc(F)c2F)=O)cc(F)ccc1Br c1(C(=O)NCC(CC)NC(C2(C)COCC2(F)F)=O)cc2n(n1)CCCC2 Cn1nc(CC(=O)NC2CC(CNC(=O)CC3CCCO3)C2)cc1C(F)(F)F C1(NC(C(CC=C)CC)=O)CC1C1CCN(C(c2cnc[nH]c2=N)=O)CC1 C1(CCOC)(NC(=O)CCCn2cccn2)CCN(C(c2cc(C)on2)=O)C1 C(=O)(C1=C(C)CCCC1)NC1(CCOC)CCN(C(=O)CC2CCNC(=O)C2)C1 C(=O)(CCCCN(C(=O)COc1ccn(C)n1)C)N1C(C)CCC1 C1(C(C)(C)C)(CNC(c2occc2C2CC2)=O)CCN(C(C2CCSCC2)=O)C1 CC(CC(F)F)C(=O)N(CCNC(=O)COCc1ccnc(O)c1)C1CC1 c1(C(C)NC(c2c(CC)cnn2C)c2n(CC(=C)C)nnn2)cc(C)cc(C)c1 N1(C(C2(CCCNC(c3ccsn3)=O)CCCC2)=O)CC2CC2C1.C(C)OCC C1(CNC(c2c(C)cco2)=O)CC12CCN(C(=O)CC1(C)CCS(=O)(=O)N1)CC2 c1(C(=O)NC2C(C)N(C(C)C(N3CCCCC3)=O)CCC2)cnc2n1CCOC2 N1(Cc2ccc(C(C)C)cc2)CC(NC(=O)CCc2ccc(O)cc2)C(C#N)C1 c1(C(=O)NC(CSCCNC(C=CC)=O)(C)C)ccc(NC=O)cc1 N1(C(C2C(CNC)CCC2)=O)CCC(c2nccn2C)CC1 c1(NC2CN(C(COCCOCC)=O)C(C)C2)cc(C(C)(C)C)nc(Cl)n1 c1(C(N2CCC(NC(=O)Cn3cccn3)(CO)C2)=O)ccc(Cl)c(F)c1F N1(C(C(C)=C2CCCC2)=O)CCCC2(CC(NC(=O)C3Cc4ccccc43)C2)C1 c1(C(=O)NC(CC(C)NC(c2n(C(C)C)ncc2)=O)C)cccn2nnnc12 CC1=C(CNC(=O)C(C2CCN(C(=O)C(=O)C3CCCC3)C2)F)CCC1 C1(CNC(CC(C)SC)=O)CC(F)CN1C(=O)C(C)NC(c1cccs1)=O N1(C(C(COC)C)=O)CC(CNC(=O)COCC(=O)OC(C)(C)C)C(O)C1 O(NC(=O)C(CNC(C1CCCC(C#N)C1)=O)CC1CC1)CCCOCC C1(CNC(c2c(C)nco2)=O)CCCC12CCN(C(c1ccsc1C#N)=O)CC2 C(C)(CO)(CN=c1ccnc(N2CCCC(CO)C2)[nH]1)OC Cc1cc(Cl)ccc1NNC(=O)C=Cc1ccc(F)cc1F C1(C(C)O)CCC(NC(=O)CCC2CCCN2C(c2cnco2)=O)CC1 Cc1ccc(NC(=O)C(C2CC2)N(C)C(C2CCCOCC2)=O)cc1F C1(CNC(c2ccc(F)cc2)=O)CCCN(C(c2sccc2CO)=O)CC1 C(=O)(C1CCCc2c1ncn2C)NCC(C)NC(c1cc(C#C)cc(F)c1)=O C(c1ccncc1)=C(C)C(=O)NCC(C)CNC(=O)COCC1CCOC1 c1(C(N2CCC(NC(Cc3ccn(CC)n3)=O)CC2)=O)ccc(Cl)cc1C c1(C(=O)NC2CCCC(NC(CCC(CC)C)=O)C2)ccc(=O)n2c1COCC2 C1(OCCC(CC2(CO)CCOCC2)O)CCC(F)(F)CC1 c1(C(N2C(CN(C)C(C3(CO)CCCO3)=O)CC(F)C2)=O)cncc(Cl)c1Cl CC(=O)C(C)CC(C)C(=O)NCc1ccc(C(=O)NCC2(C(C)(F)F)CC2)o1 CCCC(C)(O)CC(=O)N1C2CCC(C2)C1CC(=O)NCC1CCCCN1C C1(C2CCCCC2)(NC(C2N(C(C(CC)Cl)=O)CC(O)C2)=O)CC1 C=C(F)C1(CC(=O)NC(C)CN(C)C(c2n[nH]c(CC)n2)=O)CCC1 C#CCC(CC(=O)NC(CC)C(C)(C)C)NC(=O)C(OC)OC c1(C(C)C)ccc(C(=O)NCCC(O)CNC(C2CCCC2F)=O)cn1 c1(CC(=O)NC(CCOC)CNC(=O)Cc2ccco2)ccc(F)c(F)c1 CCC(CC)CCCC(=O)N1CC(NC(c2csc(COCC)n2)=O)C2CC12 C1(NC(=O)NC(CO)C(=O)O)CCC(O)CC1 c1(C(=O)NC2(CCCC(=O)NC3CC(C#N)C3)CCC2)ccc2c[nH]nc2c1 N1(C(c2c(CNC(Cc3ccc(C)nc3)=O)ccs2)=O)CCC2C(O)C(C)(C)C12 c1(CC)ncc(C(=O)NCC(C)(CNC(c2ccccc2OC)=O)OC)cn1 N1(C(CC(CC=C)(C)C)=O)C2CCC1C(F)C(NC(=O)C(F)C(C)(F)F)C2 C1(CC(N2C(C(=O)NC(C(=O)OCC)C3CC3)CCC2)=O)CCC(=O)NC1 c1(C(=O)NC2C(NC(c3csc(Cl)c3)=O)C2)ccccc1Oc1ccccc1 N1(C(C(CCC)O)=O)CCC(NC(=O)Nc2ccc(OC(F)(F)F)cc2)C(C)C1 N1(C(C2CCC(CC)O2)=O)CCC(C(C(C)C)NC(c2cccc(=O)o2)=O)CC1 C1(C)(C(=O)NCC2(NC(C3CCC(CC)O3)=O)CCC2)CC(C#N)C1 C(c1cnc2ccccc2n1)=CC(=O)NC(C)CCNC(C1(Cl)CC1)=O Cc1cc(C(N)=O)cc(C(=O)NC2CC2NC(C2(C#N)CC3CC3C2)=O)c1 c1(NC(c2onc(-c3ccc(C)cc3)n2)=O)c(-c2ccccc2)nc2ncccn12 n1(CC)c(=O)sc2c(NC(c3cnn(-c4ccccc4)c3)=O)cccc12 C(=O)(CC(C)C(=O)N1CC2CC1(CNC(C1CCC(F)CC1)=O)C2)OCC c1(C(=O)OC(C(C)OCC=C)C)cnn2c(C(F)F)cc(C)nc12 c1(C(N2C(CNC(CCC(=O)NCCC)=O)CC2)=O)cc2cc(F)ccc2cn1 N1(C(C(C(C)C)SC)=O)CCCC(C(N2CCC(N(C3CC3)C)C2)=O)C1CO C1(C(=O)NCC2N(C(=O)CCC(N)=O)CCN(C)C2)COc2ccccc2C1 c1(C(=O)NCCC2CN(C(C3(OC)CCSC3)=O)C2)sc2ncccc2c1Cl N(C1COc2cc(Br)ccc21)C(C(=O)Nc1cccc(SC)n1)=O C1(OC)CC(NC(=O)CC2(C)CCCC2)CN(C(C2OCCN(C)C2=O)=O)C1 N1(C(CCNC(N)=O)=O)CC2CCC1CN(C(c1ccncc1NCCO)=O)C2 C=CCCCC(=O)NC1CC1NC(c1cn(CC(N)=O)nn1)=O c1(NC(c2cc[nH]n2)=O)noc2c1CN(CC(=O)NC1CCCCC1)CC2 C1(C(N2CCC(C(=O)NC3CC(C(C)C)C3)(CO)C2)=O)CC(=O)NC(C)C1 C#CC1(C(=O)NCc2cncc(C(=O)NCC3(CN=[N+]=[N-])CC3)c2)CC(=O)C1 C(CCCC(CO)NC(C1CC1c1cccs1)=O)NC(c1c(C(C)C)cco1)=O Cc1ccc(S(C)(=O)=O)cc1C(=O)NCC1=NOC2CN(C(=O)C(C)(F)F)CC12 CCC(CC)C(C)C(=O)NCC12CCC(CC1)N2C(=O)C=CCOC(C)(C)C C(=O)(C(C#N)C(C)(C)C)NCc1cc(C(N2C(C(CC)O)CCCC2)=O)ncc1 CCCCS(=O)(=O)NC(C1(C)CCN1C(=O)NC(=O)C(Cl)(Cl)Cl)=O C1(N(C(C2CCC(C)(CC)O2)=O)C)CC2CCC(C1)N2C(C1CCC2(C1)N=N2)=O Cc1cc(Cl)nc(Cl)c1CNC1CC(CC(=O)Nc2cnccc2C(N)=O)C1 C=CCCC(C)(C)C(=O)NC1CCC1NC(=O)Cc1ccn(C(C)C)n1 c1(NC(CC)CNC(=O)CNC(=O)Nc2ccccc2)ccnc2ncnn12 C1(NC(COC)=O)CC(CNC(c2ccccc2C(F)(F)F)=O)C1(C)C S(=O)(=O)(c1ccccc1)NCC(=O)NC1CCOC(CNC2CC(F)(F)C2)C1 c1(C(N2CCC(CN(C)C(C3COC(=O)N3)=O)C2)=O)ccc(F)c(CO)c1 C1(C(C)(C)OC)CCC(C(=O)OC(c2ccc(C(F)(F)F)nc2)C)CC1 N1(C(c2cncc(C)c2)=O)CCC(C)C(NC(C2CC2(C)C(C)C)=O)C1 C12CC(CN1N1C(C(=O)OC)CC1)C2.c1(C=O)ccc(C(=O)N(C)C)nc1 C1(NC(C(Br)=C(C)C)=O)CN(C(c2ccc(F)cc2F)=O)C2CCCCC12 c1(C(N(C(CC2(C=C)CCC2)=O)C)=O)ccc(CN(CCCOC)C)cc1 N1(C(c2cnc(C(C)C)[nH]2)=O)CC(NC(c2cnc(Cl)c(N)c2)=O)CCC1C c12cccc(c1)CNC(=O)NC2CN(C)C.c1(COC)ncc(C(F)(F)F)s1 CCCCC(O)C(C)C(=O)NCc1cnn(C)c1C(=O)NOCc1ccccc1F C1(NC(CCCCN(C(C2OCCN(C)C2)=O)C)=O)CCCC(F)(F)C1 c1(CC(N2C3C(NC(CCCC(C)C)=O)CC(C3)C2)=O)ccccc1S(C)(=O)=O C1(C2CCOCC2)(C(=O)NC(C(C)NC(c2cnc(O)n2C)=O)(C)C)CC1 C(CCC(C)C(=O)NCc1cc(C(=O)NC2CC3(CC3)C2)ccn1)OC C(c1cn[nH]c1)=C(C)C(=O)N(CCC(C)NC(=O)C=CCO)C N1(C(C2(CC)CCNC2=O)=O)CC2CCC(C1)N2C(C1(C)CC=C(C)CC1)=O Cc1nccc(C(N2CCC(OCC(N3CCC4CC34C)=O)C2)=O)c1N c1(CC(=O)NCC2CCC(NC(C(COC)(C)O)=O)C2)c(C)nn(C(C)C)c1C N1(Cc2nc(N(c3cc(O)ccc3Br)C(C)=O)sc2)CC2CC=CCC2C1 c1(CC(=O)N(C)CC2CCN(C(c3cocc3C(N)=O)=O)C2)n[nH]c2c1CCCC2 C(C(=O)NCC(c1ccccc1)NC(=O)Cc1ccc(C)nc1)(C(C)C)NC(C)=O C1(C(N2CCCCC(C(c3nn[nH]n3)O)C2)=O)CCNC12CCS(=O)(=O)CC2 CC1(F)CC(C(=O)N(CCCNC(=O)CC2CCCO2)CC2CCCCC2)C1 c1(C(N2CC(C)C(NC(C3CN4CCC3CC4)=O)C2)=O)cccc2[nH]ncc12 C1(CNC(c2ccn(CCF)n2)=O)CCC(=O)N1.C12(CC1)C(C)NC2=O c1(C(N2CCCC(c3cn(CCCCC)nn3)C2)=O)cc([N+](=O)[O-])cnc1O C1(C2(CC(C)=O)CCC2)(CNC(c2ncccc2NS(C)(=O)=O)=O)CCCCC1 N1(C(C2=CC(C)C2)=O)CC(CO)C2(C1)CN(C(C1(C(=O)NC3CC3)CC1)=O)C2 c1(C(N2CCC(C)(NC(=O)CC3CCOCC3)C2)=O)cnc2c(c1)CNC(=O)N2 C=CCC(F)(F)C(=O)N1CCC(NC(C2(NC(=O)OC(C)(C)C)CC2)=O)C(C)C1 C1(CC)C(NC(c2cnco2)=O)CCN1C(=O)CCOCC(C)C C1(NC(c2cc(CNC(c3c(CC)ncnc3)=O)no2)=O)CCc2nncn2C1 C(=O)(C1=CC2CC(C1)CC2O)NCC(CCCC)NC(c1[nH]cc(C)c1C)=O c1(N2CCC(NC(C3CCC4(CCC4)CO3)C)C(C)C2)ncnc2c1CCC2 CCCCCC(CC)C(=O)NCCN1CCN(C(=O)C=CC(=O)NC2CC2)CC1 c1(C(=O)NCC2OCCC(NC(CCOC)=O)C2)cnn2cc[nH]c(=O)c12 N1(C(c2cn(CC=C)nc2)=O)CCCCC1CN(C(=O)CC(C)c1ccco1)C N1(C(c2c(OC)cc(C)s2)=O)CCC2CCCC(C1)N2C(=O)COCC1CCC1 CC(CCC(=O)NC1CCN(C(c2cc(C3CC3)nn2C)=O)C1C1CC1)N(C)C C1(S(C)=O)(CNCCCN(C2CCCCC2)CC)CCC1 C(N=c1nc2ncccc2c[nH]1)C1CN(C(CS(C)(=O)=O)=O)CC1C(F)(F)F c1(C(C)O)ccccc1Nc1cnc(-n2cccn2)cn1.C12CCN(C1)C2=O C1(C(=O)NC2CCC(CNC(C(CCC)NC(N)=O)=O)C2)CC2CC2CC1C c1(NC23CCC(C(=O)Nc4ccc(C)c(CO)c4)(CC2)C3)ccnc2ccnn12 N1(C(C=CCNC(C2(CC)CC(C)(C)C2)=O)=O)CCSC2CCCC12 N1(C(c2cc(C)cc(Br)c2)=O)CC2CN(C(=O)C=Cc3ccc(O)cc3)CC2C1 c1(C(N2C(C)CC(NC(=O)C=CC3CCCCC3)C2)=O)cc(F)cc2nn[nH]c12 n1(CCOCCOC)nnnc1C(C(C)(c1ccccc1)OC)NC(C)(C)C N1(C(CCCOCC=C)=O)CC2C(CNC(=O)CCN3CCC3)C2C1 CC1=C(C(=O)N(C2CN(C(c3nonc3N)=O)C2)C)C=C2CCCN=C2N1 N1(C(C(C=C)(C)C)=O)CC2CC(CNC(C3CC3c3ccncc3)=O)C2C1 C1(NC(N(CCCC(=O)OC)CC=C)=O)CCN2CCCC2C1 CC(CC(=O)NCCNC(c1ccc(C(C)(C)C)s1)=O)C1CCCCC1 C=CC1(CC(N2CCC(C)C(NC(C34CC3COC4(C)C)=O)C2)=O)CCCCC1 C(=O)(C=C1SCC(=O)N1C)NC1(COC)CCN(C(c2cnc(CCC)s2)=O)C1 CC(C)(C(=O)N1CCC(CSC2CC2)C1)ONC(c1coc(C(N)=O)c1)=O C(CCS(C)=O)(C(=O)NCC(C1CC1)NC(=O)CCCc1cccs1)N(C)C C1(NC(C=C(COC)C)=O)CCC1C(=O)NC(c1cscn1)CO C(CCO)(C(C)(C)C)NC(C(COC)NC(C1COCCN1C)=O)=O C=CCC(C(=O)NC1(C(=O)NC(CC)C(C)(C)O)CCCCC1)OC N1(C(C2(OC)CN(C(c3ccc(SC)o3)=O)C2)=O)CCC(C(F)F)CC1 c1(OCC)ccc(C(=O)NC2(CCNC(C3CN(S(C)(=O)=O)C3)=O)CC2)cn1 c1(SC)nc(C)c(CCC(=O)NC2(CCCNC(C3(C)CC3F)=O)CC2)c(O)n1 c1(OCC)ccc(C(C(=O)NC2CCCO2)N(CC)CC)nn1.C(C)(C)(C)O N1(C(=O)CSCc2ncc[nH]2)CCN(C(c2cc(C3CC3)on2)=O)CC1CCO S(=O)(=O)(c1cc(F)ccc1F)N1CC2CN(C(c3ccccc3O)=O)C2C1 N1(C(CN(C(COC)=O)C)=O)CC(C)CN(C(C2(C)CC3(CCC3)C2)=O)C(C)C1 N#CC1(CC(N2CCC(NC(C3(CCS(N)(=O)=O)CCC3)=O)CC2)=O)CCOC1 Cc1oc(C(N2CCC2CNC(c2ccc(CO)cc2)=O)=O)cc1S(C)(=O)=O c1(C(=O)NCCC(C(C)C)NC(C2CCCCC2)=O)ccc2ccnn2c1 N1(C(C(C)(C)c2cnc[nH]2)=O)CCCC(CNC(c2ccc(CF)cc2)=O)C1 c1(OC)ncc(C(N2CCC(Nc3nccc(N4CCOCC4)n3)C2)=O)cn1 c1(C(=O)NCC(C)NC(c2c(C)c[nH]c2)=O)ccc(C(C)C)nc1O C1(C(=O)NC(c2ccncn2)C)(NC(CC2C(CC)C2)=O)CCN(C)C1 C=CCCCCCCCC(=O)Oc1cccc(C(=O)NC(C)C)c1C C1(C(=O)NCCCN(C(C2COC3CC2C3)=O)CC)CNC(=O)CC1C(F)(F)F C(C(C(=O)N(C)CCc1cnn(C)c1)NC(=O)CCn1ccnc1C)OCC C1(OCC)CN(C(=O)C=CSCc2ccco2)CC1NC(c1ccc(=O)oc1)=O c1(C(N2C3CN(C(C(CC=C)(C)C)=O)C(C3)C2)=O)c(Cl)sc2nnsc12 C1(NC(c2n(C)cnc2)=O)CCC2CN(CCOCc3ccccc3)CC2C1 C1(CCC)CCCN(C(C2CCN(C(c3cncc(C)n3)=O)C2)=O)C1 C1(CNC(C2C(C3C(C)C3)C2)=O)CC2(CO1)CN(C(C1(C)CCCOC1)=O)C2 c1(C(N2CC(N(C(=O)CSC(C)(C)C)C)C(F)C2)=O)csc2ccccc12 c1(C(=O)NCC(CCCC)NC(=O)Cn2nnc(=O)[nH]2)cc[nH]c2nccc1-2 CC1=CC=CNC(=O)C(=O)NCC1CCN1CC(OCCCO)C1=O C1(CNC(c2c(CC)c[nH]n2)=O)CCC2COCCC2C1 CCC(C)(C)CCN=c1[nH]c(=NC)[nH]c(=NCC2(OC)CCCSC2)[nH]1 N1(C(CCSC)=O)CC(NC(=O)C(c2ccc(F)cc2)CC)CC(F)C1 c1(CCC(=O)NCCC(C)NC(C2CCCC2)=O)csc(Br)c1 N1(C(CC(CCC)CC)=O)CCN(C(c2cccc(CCO)c2)=O)CC12CCC2 N1(C(N2CCN(CCc3ccccc3)CC2)=O)CCCC(CF)C1 C1(C(=O)NCc2occ(C(N(C)Cc3ccncc3F)=O)n2)CC2C=CC1CC2 N1(C(c2c(C)nc(CC)o2)=O)CCC2CC2(NC(=O)Cc2ccc(F)cn2)CC1 c1(N2CCC(NC(=O)NC34CCC(F)(CC3)CC4)C(F)C2)ccc([N+](=O)[O-])cn1 C(C1CCOc2ccccc21)NC(N1CC(C(=O)OC)C(c2cn(C)cn2)C1)=O C1(OC)CC(CF)N(C(=O)CN(C(C2CC(O)C(F)C2)=O)CC2CC2)C1 c1(C(N(C)CC2N(C(CCC3CC(C)C3)=O)CCOC2)=O)c2c(nn1C)CCC2 N1(C(C2C(C)C2)=O)CCC(CNC(c2cc3sccc3n2C)=O)C(F)(F)CC1 c1(C(=O)Nc2cccc(C3CCCCC3)c2)cc2cc(Cl)c(Cl)cc2[nH]1 C1(CC(N2CC(CNC(C3N(CC)CC3)=O)(OC)C2)=O)CCC(F)CC1 c1(C(N2CC(O)(CCNC(CC3CCC(C)C3)=O)C2)=O)c[nH]c2ccncc12 Cc1ccc2ncc(C(=O)N(C)CCN(C(=O)CC(C)N3CCCC3=O)C)n2c1 c1(OC)cc(F)c(F)cc1C(N1CC2CC2(NC(=O)C2=CCS(=O)(=O)C2)C1)=O N1(C(CN2CCCC(NC(C3(OC)CCSC3)=O)C2)=O)CC2CC2(OC)C1 C(C(O)CN=c1ccnc[nH]1)NC(c1ccc2nc(O)[nH]c2n1)=O c1(C(N2CC3(CNC(=O)C(F)F)CCC2CC3)=O)ccccc1S(=O)C(F)(F)F C1(C(=O)NCCSCC=C)CN(C(=O)C(C2CCCCC2)O)CC1C N1(C(c2cc(O)cs2)=O)CC2C(C(=O)NOCCC(F)F)C2C1 CC1CCc2ncc(C(N3CC4CC(NC(=O)COCCCF)C3C4)=O)n2C1 NS(=O)(=O)CCCCCCC(=O)NC1CCC(NC(=O)COC2CCCCC2)C1 Cc1oc(C)c(C(N2CCCCC(NC(=O)C(CCO)N(C)C)C2)=O)c1C C1(C(=O)NCC(=O)OC(C)C)CCCN(C(=O)CC2CCCOCC2)CC1 S(=O)(=O)(c1ccc(=NCc2c(C)nn(C)c2C)[nH]c1)N(C(C(CC)CC)C)CC CCCCC(O)CC(=O)N(C(C)(C)CC(=O)NCc1ccnc(C)c1)C c1(CCC(N)=O)ccc(C(=O)NC2CCCN(Cc3ccncc3Cl)C2)cc1 C1(CC(=O)NCC(C2CCOC2)NC(c2ccncc2)=O)CCC2(CC2)CO1 N1(C(CN(C2CCCC2(F)F)C)=O)CCOCC1CNC(c1ccccc1)=O CC(C)(C)C(CC(=O)NC1CCC2CC1CN2C(=O)C#CC1CC1)C(F)F CC1CCC=C1C(=O)NCC(O)CC1(C)CCCO1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1(NC(CCCC)=O)CC1 C1(c2n(CCSC)nnn2)(Nc2sc(Cl)nc2Cl)CCCN(C(C)(C)C)C1 C1(C)(C(N(C)CC2(O)CN(C(COc3cc(C)on3)=O)C2)=O)CCC(=O)NC1 c1(C(=O)NCC2N(C(C(C)CO)=O)CC(O)C2)csc2ccc(F)cc12 c1(C(=O)NC(c2occ(C(N(C3CCC(C)C3)C)=O)n2)C)ccccc1O c1(C(N2C3CN(C(CCCC(=O)OC)=O)C(CC3)C2)=O)cnc2ccccc2c1 C(C1c2ccccc2CCN1C(=O)COC(C)(C)C)NC(C(C)CNC(N)=O)=O C12(C(=O)NC3CC4CC(OC)C4C3)CCCC1CN(C(c1cc(C)c(C)[nH]1)=O)C2 c1(N)ccsc1.CC(C)COCC(=O)NC1CC1NC(C1(C(=O)N)CC1)=O c1(C(C(=O)NC2CN(C(c3c(C)cno3)=O)CC2O)O)ccc(F)cc1F CC1CCC(NC(=O)CC2CCN(C)C2=O)CN1C(C1CSCN1C)=O C(=O)(C1=CC2(CCN(C(c3cnnn3C)=O)C2)C1)NC1CCN(CCC)C1 C(=O)(CCCC(=O)NCC1(NC(=O)COC2CCOC2)CCOC1)OCC C(=O)(C(C)CS(C)(=O)=O)NCC1(NC(c2cc(C)c(C)o2)=O)CC1 C(C#Cc1cccnc1)NC(C(C(COC)C)C)=O N(C1CCCOc2c1ccc1ccccc21)Cc1cc(Br)c(I)cc1 c1(C(=O)NCCCN(C(=O)CCS(C)=O)CC)nccc2cccnc12 c1(C(=O)NC(CN(C(CN(C2CC2)CC)=O)C)C)n[nH]cc1F C1(C(=O)NCc2n(C)ncc2)CC12CCN(C(=O)COCC1CC1)C2 C1(NC(c2cccc(OC)n2)=O)CC12CCN(C(=O)CC(C)C(C)C)C2 CC1(C)CCC(C(N2CC(NC(c3ccc(CC#N)cc3)=O)C2)=O)O1 Cc1cc2cc(CNC(c3cc(-c4ccc([N+](=O)[O-])cc4F)on3)=O)ccc2s1 N1(C(c2cnn(C(C)C)c2I)C(=O)NCc2cccs2)CCC(C)(C)C1C N1(C(C=CCCC)=O)CC(NC(=O)C=Cc2nnn(C)n2)CC1(C)COC Cc1cc2ncc(C(=O)NCC34CC(CO3)N(C(C3CCC(C)O3)=O)C4)cc2[nH]1 C1(C(N2C(CN(C(=O)Cc3cnsc3)C)COCC2)=O)CC2CC1C1C2C1(F)F CCC(CC)(CO)C(=O)N1CC=CC(NC(=O)C=Cc2cscn2)C1 c1(SC)nccc(N(CC(C)NC(=O)C(n2nc(C)cc2C)C)C)n1 C(=O)(C=CS(C)(=O)=O)NCC1N(C(C=CC=CC)=O)CC=C1 c1(CC)ncc(C(N2CCOC(C)(CNC(=O)C(O)C(F)(F)F)C2)=O)c(O)n1 C(CN=c1nc2sccc2c(N2CC34CCC3(COC4)C2)[nH]1)Oc1ccc(Cl)s1 C(=O)(C1=CSCCO1)N1C(CCNC(c2ccn(CC)c2C)=O)CCCC1 C1(CC)CN(C(C2(COC)CN(C(=O)C3=COCCC3)C2)=O)CC12CC2 Cc1ccc(Cl)cc1NC(=O)C(C1CCN(C(=O)C(C)n2ccnn2)CC1)C Cc1cc(F)c(C(=O)N(CC(C)CNC(C2CC3CCC2O3)=O)C)c(Br)c1 c1(C(=O)NC2(C(COC)O)CC2)ccc(CNC(C2CC(C)C2)=O)s1 Cc1cc(C(N2CC(NC(c3cc(C)n(C(F)F)n3)=O)C(O)C2)=O)c(N)cc1F c12cc3c(s1)CCN(C3)C(=O)Nc1nc-2cs1.C(CNC=O)OCC.C(CCl)O C1(NC(C(C2CCOCC2)C)=O)CCN(C(C2C(C)(C)C2(C)C)=O)C1C c1(C(N2CC(S(CC)(=O)=O)C2)=O)ccc2c(c1)SCC(=O)N2 C(=O)(C(C)(C)Cc1cccc(Cl)c1)NC(C)CN(C(=O)CC1C=CCCC1)C c1(SC)ncc(C(=O)NC(CO)C(C)NC(C2C(C)(C)C2(F)F)=O)c(O)n1 C(c1cnccn1)=CC(=O)NCC(CNC(c1ncnn1C(C)C)=O)OC c1(C(N2CC(CC=C)(NC(C3C(C)CC3C)=O)C2)=O)ccc(Cl)cc1Br N(C1CCc2cc(CNC(c3ncsc3C(F)(F)F)=O)ccc21)C(C1C(C)C1)=O Cc1c(F)ccc(C(N2CCC(NC(c3cnsn3)=O)C2C)=O)c1Cl N1(C(c2c(CNC(c3cncc(CC)c3)=O)occ2)=O)CCC(O)C(C)C1 c1(C(C)NC(=O)C(N2CCCC2c2nnc3n2CCCC3)=O)cc2ccccc2s1 N1(C(c2c(C)con2)=O)CCCCC(CNC(=O)C=C2CCOCC2)C1 c1(C2CCN(S(CCN(CCC)C(=O)N(C)C)(=O)=O)C2)c(OC)cc(Br)cc1F C(N=c1nc(O)c2ccccc2[nH]1)C1CCCN(C(C2(C)CCCCO2)=O)C1 C12(CNC(C3CC(CN(C)C)C3)=O)CC1CN(C(=O)COc1ccn(C)n1)C2 N1(C(CC2CCC(NC(C3CC34CCCCC4)=O)CC2)=O)CC2(CCC2O)C1 N12CC(NC(CSCC)=O)CC1C2.C(=O)(CS(=O)(=O)NCCOC)NC(C)(C)C CC1(C)OCCNC1C(=O)Nc1ncc(Cl)c(C(F)(F)F)n1 Oc1c(F)cc(CNC2(CN3CCCCC3)CCCCC2)cc1F c1(NC2(CNC(c3c(C)oc(C(C)(C)C)c3)=O)CCC2)ncnc2[nH]cc(I)c12 C1(NC(c2c(C(C)NC(C3(CC)CCOC3)=O)noc2)=O)CCN(C)C(=O)C1 c1(OC)ccc(CN2CCC2C(=O)Nc2cnn(C3CCCC3)c2C)cc1Br C1(CC)CC(C(=O)N(C)CC2CC(O)C2)CCN1C(c1cc(C)cs1)=O C1(NC(C(CO)NC(C(C)C)=O)=O)(NC(=O)CN2CC3CCC2C3)CCCCC1 Cn1nc(C(N2CCCC(CO)(NC(=O)C(C3CCOCC3)F)C2)=O)cc1C#N N1(C(c2c(CC)non2)=O)CC(C)(C)CC1C(=O)NCCNS(=O)(=O)CC c1(C(=O)OC)c(CCC(=O)NC2(c3cnn(C)n3)CCC2)c(C(F)(F)F)nn1C CCC(F)(F)C(C)(C)C(=O)NCC1(C)CN(C(=O)COC2CCOC2)C(C)(C)C1 C(=O)(C1=CC2CCC(C1)C2)N1CC(CC(C)NC(=O)CN2CC3CC3C2)C1 C(=O)(CC1CCc2ccccc21)C(CNC(=O)OC)=O.C1(NC)CCN(CC)C1 Cc1nc(C(=O)NC2CCCC(NC(C3(CO)COC3)=O)C2)ccc1Br C(C1CC(=O)Nc2ccccc21)NC(C(C)NC(c1ccc(Cl)c(Cl)c1)=O)=O c1(OC)ncc(C)cc1NC(C1CC(NC(=O)Cc2ncccc2F)C1(C)C)=O c1(C(=O)NC2CCC2CNC(c2coc(O)n2)=O)cc2c(Cl)cccc2[nH]1 c1(C(N2CCN(C(C(C)SCCCC)=O)CC2)=O)cc2c(OC)cc(Cl)cc2[nH]1 CC(C)CC(C(=O)N(C)CCNC(=O)C(C)C(F)(F)C(F)F)C(N)=O CC12COCC1(C)CN(C(=O)NCCc1ccc(-n3cccn3)cc1)C2 C1(COC)(NC(=O)CN2CC(F)(F)C2)CCN(C(=O)C(F)C2CCCC2)CC1 C1(C(=O)NC(CC=C)C2CC2)CC(O)C(O)CC1CNC(=O)CC(C)C(=O)OC N1(C(C2C(C=CC)CN(C(=O)CCCCCOC)C2)=O)CC2CCC1C(O)C2O CC(C)(CNC(C1C2CCCC12)=O)CCNC(=O)COc1ccccc1Cl c1(N2CC(C)(NC(CCCCC(C)C)=O)C2)nc(Cl)nc2cccc([N+](=O)[O-])c12 C1(CN(C(=O)CCc2cc(Cl)cs2)C)C2CN(C(c3cc[nH]c(=N)c3)=O)CC12 C1(OC)CC(CN(C(=O)CC2CCC(=O)C2)CC)N(C(=O)CN(C(=O)C(C)C)C)C1 N1(C(C(C(CC)C)O)=O)CCC2(CC1)CC2NC(c1ccsc1)=O C(=O)(C(CNC(c1cc(O)ccc1C)=O)C(C)(C)C)N(CCCOCC)C c1(C(N2C(CNC(CCCC(=C)C)=O)C(O)C(O)C2)=O)cc(S(N)(=O)=O)oc1C N1(C(C2(CC=C)CCCC2)=O)CC2ON=C(CNC(=O)Cc3cc[nH]n3)C2C1 N1(C(CC(CC)(F)F)=O)CCOC2CN(C(C3CCC34CCC4)=O)CC12 n1(CC)nc(C(=O)N(C)CC2COCCN2C(=O)C=CSC)cc1C1CC1 C1(CC)CN(C(C2(OC)CCOCC2)=O)CCN1C(c1csc(Cl)n1)=O C(C(=O)NCc1ccc(OC)cc1)(C1=NOC2CC12)N(C1CN(C)S(=O)(=O)C1)C N1(CC(=O)NC2CCC2NC(c2ccc(=O)oc2)=O)C(=O)CCCC1=O C1(CNC(CSCC#C)=O)(OC)CCN(C(=O)CC2CCOC2(C)C)CC1 N1(C(C2(SC)CC2)=O)CC(CNC(=O)C(C)Oc2ccc(C#N)cc2)C2(CC2)C1 CCCCC(C)C(=O)N1CC(NC(c2cc(N)cnc2C)=O)C(C)C1 n1(CCCC(=O)NC2C(CNC(C3CC(SC)C3)=O)CC2)nc(C)cc1C N1(C(CCOCC)=O)CC=C(CCNC(C2OCCC2c2cnn(C)c2)=O)CC1 c1(C(=O)NCC(C(C)C)NC(C)=O)cnn(-c2ccncc2)c1C CCS(=O)(=O)C=CC(=O)NC1CCC(CNC(c2cc(CO)[nH]n2)=O)C1 c1(C(N(C2C(C)CCN(C(CC(C)C)=O)C2)C)=O)nc(=N)[nH]c2ccccc12 C(c1ccc2c(c1)COCC2)=Cc1onc(CC)n1 Cc1cc(C)c(C(=O)NCC(C)CC(=O)NCCCCCCF)s1 c1(C(C(=O)NCC2CCN2C(=O)C(C)C2CC2)OCC)ccccc1 N1(C(C(CCC)C)C(=O)NCCC2CC2)CCc2cc(C)cc(C)c2C1 C1(CNC(c2nc(CC)sc2)=O)C(C2CC2)CCN1C(=O)CSC(F)(F)F N1(C(c2n(CC)ccn2)=O)CC(C2(NC(C3CCCSC3C)=O)CC2)C1 N1(C(C(CC)F)=O)CC2CCC1CN2C(c1c(C)nn(C)c1-n1ccnc1C)=O C1(C(=O)NC(C(C)C)CN(C)C)CCCN1NC(=O)CCC(N)=O C(=O)(CCN=C(NCc1nccs1)NC1CC1(c1ccccc1OC)C)NC N1(C(CCc2cc(C)on2)=O)CCC(F)(CNC(C2C3COCC23)=O)CC1 C1(NC(=O)Cc2ccc(C(F)(F)F)cc2F)CC2CN(C(=O)CSC(F)F)CC2C1 C1(CC(C)C)(C(=O)NCC2CC(C)N(C(c3csc(O)n3)=O)C2)CCNC1=O Nc1cc(C(=O)NCC2CN(C(c3ncc(Cl)s3)=O)C2)nc(O)c1 C1(NC(c2c(CC)nco2)=O)CC2CC(C1)N(C(=O)CC1CC(C)(C)C1)C2 C1(NC(C(=Cc2cnc[nH]2)C)=O)CC2CCC(C1C)N2C(c1cccn1C)=O N1(C(C=CC)=O)CCn2nc(C)c(CNC(=O)COc3cccnc3)c2C1 CC1(C)NC(=O)CC1C(=O)NCCC1(NC(c2cc(C(N)=O)[nH]n2)=O)CCCC1 c1(OC(C)C)cccc(NC(C2COCCC2NC(c2cc[nH]c2)=O)=O)c1 c1(Sn2nccc2-c2cccc(CCC(N)=O)c2)cc([N+](=O)[O-])cnc1O N1(C(C2C(C)CC2)=O)CCC(C2(O)CN(C(C3(NC(N)=O)CC3)=O)C2)CC1 N1(C(c2cc(CC)oc2C)=O)CC2CCC(NC(C3CCCCS3)=O)CC2C1 CC1C(NC(C2CC(F)(CO)C2)=O)CCCN1C(c1cncc(OC(F)F)c1)=O C1(F)(C(=O)NCC(C)F)CN(C(c2cc(C3CC3)[nH]n2)=O)C1 N12CCCC(O)(CC1)SC(F)(F)C2=O.C1(C(C)=O)CCC(O)CC1 c1(C(N2C3C(NC(C(C=C)(C)C)=O)CC(C3)C2)=O)cc(C)cc2ccncc12 C12(CCCC1)c1cn(nn1)C(C)C(=O)N2.C1(C(=O)NCCOC)CCCCC1 CCCCC(CNC(C1CCCCN1C)=O)NC(=O)CC1CCCC1C N1(C(C(CCC)C)=O)CC(NC(c2ccccc2OC2CC2)=O)CC2(CCC2)C1 Cc1cc(C(N2CCC3CC2CN(C(C2(C)CCCO2)=O)C3)=O)cc2nc[nH]c12 CC(C)CC(C(=O)N1CC(CO)C(F)C1)ONC(c1cccc(F)c1F)=O C1(NC(CC2(CC)CCOCC2)=O)CN(C(c2cccnc2O)=O)CCC1C Cc1cc(C(=O)NCC(CC(C)C)NC(C2CC3(C2)CC3F)=O)oc1C C(=O)(C(C)(C)C(c1ccccc1)NCC(c1cccc(OC)c1)C)OC CC1CCN(C(=O)CNC(N)=O)C(CNC(C23CCCC(CO2)C3)=O)C1 c1(SC)cc(C(=O)NC2(CO)CN(C(c3coc(C)n3)=O)C2)ccc1NC(C)=O N1(c2c(C)cncn2)CCc2ccc(C(=O)NCCc3ccccc3)cc2C1 c1(C(=O)NC2C3N(C(c4c(C)c[nH]n4)=O)C(CC3)C2)cc(C)nc2onc(C)c12 N1(C(CC(C)(C)C#N)=O)CC(F)(F)CC1(C)CNC(=O)CC1CC2(CCC2)CO1 N1(C(CCCC=C)=O)CCC(C)C(CC(=O)N(C)CCSC)C1 C1(NC(C2C(C)(C)C2)=O)CCC(F)(CNC(=O)CC2(N3CCCC3)COC2)C1 C1(CN(C(=O)Nc2cnc(OC)s2)CC)CCN(c2nccc(Cl)n2)CC1 C1(C(=O)NCCN(C(C2C(CC)C2C)=O)CC2CC2)CC(=O)N(C(CC)CC)C1 C1(F)(CNC(c2cc(CCO)on2)=O)CC(CNC(C2(F)CC2)=O)C1 CN=c1[nH]c(C(=O)NC2(CCNC(c3cncc(OC)n3)=O)CC2)cs1 c1(CCOCC)nc(C(N2CCC(CN(C)C(C3CC3CSC)=O)C2)=O)co1 Cc1csc2cc(C(N3CCC(C(C)NC(=O)CC(C)P(C)(C)=O)CC3)=O)[nH]c12 CC1CCN(C(=O)C(C)(C)C#N)CC1CC(=O)NCCC1CCCC1 c1(C(N(C(CNC(C2(C)CC(=C)C2)=O)C)C)=O)ncc(C)cc1F C1(CC(=O)NC2(CC(=O)OC)CC2)C2CCCC2N1C(c1cccc(C#N)c1)=O c1(NCC)scnc1C(=O)NC(C)C(=O)NCC12CCCC1C2 C1(C(=O)NCCC(C)NC(COCC)=O)CCCC(=O)CC1 N1(C(CCc2c(C)noc2)=O)CCC(C)C(N(C(=O)CCc2ccncc2)C)C1 Cc1ccc(Cl)cc1OCC(=O)NC1CCC(C)N(C(=O)CC2CC(F)C2)C1 n1(CC(=O)N(CCC(=O)NCCCc2cnc[nH]2)CCO)ncccc1=O Cc1nn(CC(=O)NCC(CNC(C2(CC(C)C)CCC2)=O)CO)cc1Cl CCCCCC(=O)NCC1COCCN1C(c1cccc(OCC(=O)NC)c1)=O N1(C(c2c(C)oc(C3CC3)n2)=O)CC(CNC(C2(C3CC3)CC2)=O)C(F)(F)C1 C=CC1CN(C(c2c[nH]nc2CNC(C2CCCC(OC)C2)=O)=O)CC1O C1(NC(=O)CC2C=CCCC2)C2CCC1N(C(=O)Cc1ccsc1Cl)C2 C(=O)(CC(CC)c1ccccc1)NCC(CNC(c1c(CC)cco1)=O)OC S(=O)(=O)(c1ccccc1F)Nc1cccc(C(=O)NC(CC)CO)c1 Cc1c(C(=O)NC2CCCC2NC(=O)CCCC2CCC2)[nH]c2c1C(=O)CCC2 N(C(=NCCC(C)C)N1CCC(c2ccccc2F)C1)CCC(C)=O N(C1CCc2cc(Cl)ccc21)C(=O)Cc1c(Cl)cccc1[N+](=O)[O-].C1C(=O)N1 N1(C(CC2(CNC(C(C)NC=O)=O)CC2)=O)CC2CC=CCC2C1 c1(CC(=O)N(CC(C)O)CCNC(=O)CCC2CCCC2)ccc2oc(O)nc2c1 C(=O)(C1=CCC(NC(=O)Cn2cnnc2O)C1)NC1(C)C(C)(C)C1 C1(NC(c2ccc(Br)cc2)=O)CN(C(C2(CF)CC2)=O)CC1n1cccn1 c1(C(=O)OCC)cc(C)nnc1N1CCC(COC)(NC(=O)C(C)C(C)CC)C1 N1(C(C2C(C=C)C2)=O)CCC2(CCCC2CNC(=O)CS(N)(=O)=O)CC1 S(=O)(=O)(c1ccc(N2CCc3sc(C)cc3C2)cc1Br)NC(CC=C)C C1(C(N(C)C)=O)CCN(C(=O)NCC2C=CCCC2)C1 N1(C(CC(=C)C)=O)CCCC12CCN(C(C1CC(=O)N(c3cn[nH]c3)C1)=O)C2 N1(C(C(F)=C(C)C)=O)CCN(CC2(NC(C3COC(=O)N3)=O)CC2)CC1 c1(C(=O)OCC)ccc(S(=O)(=O)NC(C(=O)OCC)C(=O)NC2CCCC2)o1 c1(C(=O)NCC(COC)OC2(CO)CC3CCC2C3)c(C)ncnc1C N1(CC)C(=O)COC(NC2CC2C(C)(C)C)C1c1ccnn1C CC1CN(C(=O)CCn2cccn2)CCN1C(=O)CC1CC=CCN1C C1(N(C(C2OCCC2C)=O)CC)CCN(C(c2ncsc2Br)=O)C1 c1(C(N2CCCN(C(c3c(C)cc(C)[nH]3)=O)CC2C)=O)cnn2c1CC(F)(F)C2 C(=O)(C1=CC2CCC(C1)C2)NCC(C(C)C)NC(CNC(=O)OCC)=O S1(=O)(=O)c2ccc(c(F)c2)NCc2cccc(c2)CN1.C1(CCC)(CSC)CC1 Cc1cc(C(=O)NCC2CC3CN(C(c4cnc(C)o4)=O)CC23)c(O)nc1C c1(CCCC(=O)NC2(CNC(=O)CSc3nncs3)CC2)ccc(F)c(F)c1 NC(=O)CC(O)C(=O)NCc1csc(C(N2CCCC(N=O)C2)=O)c1 c1(NC(=O)Nc2cccc(C3OCCO3)c2)ccc(C2CC2)nc1 C12(C(=O)NC3(C)CC3)CC(CO)(C1)OC2(C)C.N12CCC(C1)N(CCO)CC2=O c1(C(N(C(C)CNC(=O)Cc2nnc(S)n2C)CC)=O)cc(OC)n(C)n1 Cc1sc2ncnc(NC(C)CC(C)NC(c3cnc(C4CC4)[nH]3)=O)c2c1C N1(C(Cc2ccc(CC)s2)=O)CC2OCCCC2(C(=O)NC(C)CO)C1 N1(C(c2c(C)cc(CC)o2)=O)CC2CCCC1CN(C(c1cc(Cl)nn1C)=O)C2 C(CNC(=O)COOCO)(CC(F)(F)F)NC(C1(OC)CCSC1)=O.c1ccccc1 C(=O)(CC(CC)C(C)C)NC1CC(C(C)NC(C(C=C=C)C)=O)C1 c1(C(=O)NC2CN(C(C3CCCS3)=O)CC2F)ccc2nccnc2c1 N1(C(c2c(C)oc(Br)c2)=O)CCN(C(=O)CC2C(C)(C)C2(C)C)C(C)C1C CC(C(=O)NC1CC(CCNC(=O)Cn2cc(C3CC3)nn2)C1)C(C)(C)C c1(CN(C(c2csc(-c3cccs3)n2)=O)Cc2nn[nH]n2)nc2ccccc2[nH]1 c1(C(N2CC=CCC(C)(C)C2)=O)cc2ncncc2s1 C(=O)(C1CCCc2cncn21)NCc1c(CN(C(C2(OC)CC2)=O)C)cccc1 c1(C(=O)NCC2(F)CN(C(c3cc(C)c(F)cn3)=O)C2)nn(C)c(=O)cc1C C12CCc3nnc(n3C1)NC2=O.c1(CC#N)ccc(N2CCCCC2)nc1 C1(CCOC)(NC(=O)C=CCO)CCN(C(=O)C(O)CC2CCCCC2)C1 N1(C(Cc2c(C)nc[nH]2)=O)CC2(CCC2)CC1CNC(c1cc(Br)n[nH]1)=O C#CCC(C(=O)N1CCCC1(C)CCCO)NC(C1CS(=O)C1)=O C1(C(=O)NCCC2CC(NC(C3CC4CC4C3)=O)C2)CC2COCC(C1)C2(F)F c1(CN2C(CNC3CC(CC)(CC)C3)CC2)ccc(Br)cc1 c1(CNC(C=C(CC)CC)=O)ccnc(OC)c1.C12(CSC1)C(=O)N2 Cn1cc(Br)c2c(C(N3CC(C)(C)CC3CNC(=O)CCF)=O)ncnc12 N1(C(=O)NCCC(C)C)CC2CN(C(=O)CCCc3ccc(Cl)cc3)C2C1 C(C(C)(CC(C)C)NC(C1CC(OC2CC2)C1)=O)NC(C1(C(F)F)CC(=C)C1)=O N1(C(c2cccc(SC)c2)=O)CCC(NC(c2ncsc2C2CC2)=O)C(F)C1 N1(C(c2cc(O)ccc2O)=O)CCC(F)(F)C(Nc2ncccn2)C1 C(=O)(CC(C(F)(F)F)n1ccnc1)NCC1(O)CN(C(=O)OC)C1 CC1=C(C(=O)NC2CCCCCC2NC(=O)Cc2cn[nH]c2)C(=O)OC1(C)C CCCCC(C(=O)N=c1cc2ccccn2[nH]1)NC(=O)C(O)CSC N1(C(c2c(CC)onc2)=O)CC(NC(C2(O)CC2)=O)CC1(CC)CC c1(CCC(=O)NC(C2CCCN(C(=O)C(C)(C)C#N)C2)C)c[nH]c2ccccc12 N1(CCC)CCCC(CNC(=O)CC(C)(C)C)C1.N12CCCCC1C2=O c1(NCC2CN(C(C3CCC(CN(C)C)O3)=O)CC2C)ncnc2c1CCC2 CCS(=O)CC(=O)NC(Cc1ccccc1)CCNC(c1cnc(CF)s1)=O c1(C(N2CC(NC(C(c3ccccc3)C)=O)C(O)C2)=O)cc(Cl)c(F)cc1F C(=O)(CCN(CC(C)C)C(c1ccon1)=O)NCCC=CCCC c1(CN2CC(C)N(C(C34CCC(CC3)CC4)=O)CC2)ccc2c(c1)OCO2 c1(C(=O)NCCC(CCNC(C(=Cc2cnc[nH]2)C)=O)C)cc(CO)ccc1Cl c1(C(=O)NC(C(=O)OCC)C2COC2)c(F)c(F)c(Br)c(F)c1F C1(C(C)(O)CNC(=O)C=Cc2cnc[nH]2)CCCN(C(C2CCCCC2)=O)C1 c1(C(N2CC(CCNC(c3c(C)snn3)=O)OC(C)C2)=O)ncnc2c1CCC2 C1(N(C(C(C2CN(C(C)=O)C2)O)=O)C2CC2)CCNC1=O C1(F)(CNC(C(C)N(C)C)=O)CCC(CNC(c2cc(C(F)F)nn2C)=O)CC1 C1(CC(=O)OC)CC(n2cc(C3(OC)CN(C(=O)C(C)(C)CC)C3)nn2)CCO1 C=Cn1nccc1C(=O)NCC(C)(C)OCC(=O)NCC1COC(CO)C1 C1(c2n(CC)nnn2)(NCCOCc2ccccc2OC)CCC(C)SC1 C(=O)(CCC(C)(F)F)N1CCCC(CCNC(COCCC)=O)C1 C(=O)(C(C)(C)CC(F)F)N(CCC1CCN(C(C2(C)CCC(C)C2)=O)CC1)C C1(C(=O)NCC(C)NC(C2C(C)(CC)C2)=O)CSCCS1 C1(C(C)C)CN(C(c2scnc2Cl)=O)CCN1C(C1CCCN1C)=O c1(C(=O)NCC2C(CC)CCN2C(=O)Cc2cnn(C)c2C)nnc(O)nc1O c1(C(N2C(CNC(COCCOCC#C)=O)CCC2)=O)cnc2c(ccn2C)c1 c1(C(=O)NC2CN(c3ncncc3Br)CCC2(F)F)cccc2nc(Cl)sc12 C(C(C(=O)N(C1CCCCC1)CCOC)C(C)C)NC(c1cc(CC)no1)=O C12(NC(c3cc(C)on3)=O)CCCN(C(=O)CNC(=O)Cc3ccccc3)C1C2 C1(C(N2C(C(=O)NCc3ccc(C(C)C)cc3)C(O)CC2)=O)C2CC3C(C2=O)C13 c1(N(C(=O)Nc2ccc(C(CC)=O)cc2)C)cccc(C(=O)OC)c1C CC1COCC2(CCC2)N(C(=O)C(N2CCC(C)CC2)=O)C1 N1(C(c2ccc(C)o2)=O)CCCC2(CCCN(C(c3cc(Br)ccc3Cl)=O)C2)C1 C(=O)(C#CC1CCCCC1)N1CCC(N(C(c2cc(CC)ncc2)=O)C)C1 c1(C(=O)NC2CCC(NC(CC3C(C)(C)CCO3)=O)CC2)cccc2ncsc12 CCC(C)C(C(=O)NCCCOCCNC(c1cocc1C)=O)c1ccccc1 CC(CC(=O)NCCn1cc(C(=O)NCC2CN(C(N)=O)C2)nn1)C(F)(F)F N1(C(c2c(CCC)cccc2)=O)CCC(NC(=O)C(C)OC(C)=O)C12CCC2 C12(C(=O)NCC(C)CN(C)C(c3csc4nccn34)=O)CCCCN1CCC2 CC(CCC(C)(C)C)C(=O)NN(C)C.c1(C)ccccc1-n1cc(CC2CC2)nn1 C(=O)(C(C(=O)NCCCC(C)NC(=O)CN(C)C(c1ccsc1)=O)OC)OC c1(C(=O)NCc2ccnc(-c3nn[nH]n3)c2)ccc(Cl)c(C2CC2)c1 c1(OC)ccc(Cl)c(C(=O)N(C2CN(C(C3CCCCC3C)=O)C2)C)c1 N1(C(C2CCC(C)(C)C2)C(=O)NC(c2ccccc2)C)CCC12CCSCC2 c1(CC)cn2c(C(=O)NCC#CCNC(=O)CC3(O)CCCCC3)cccc2n1 O=C(N=c1[nH]nc(Cl)cc1O)c1occc1OC(F)F C1(NC(c2ccc(OC)o2)=O)C=CCN(C(=O)CC2CC2c2ccccc2)C1 C1(C(=O)OC)CC(S(C)(=O)=O)CN1C(=O)CC=CCNC(=O)CC1CCOCC1 N1(C(C)=O)CCCCC1C(N1CCCCC1CCNC(=O)CCn1ccnc1)=O CC(CNC(=O)CCCF)(CO)NC(=O)CCCc1ccsc1 CC1Cc2cccc(C(N3CC4(C3)CN(C(=O)COC3CCOCC3)C4)=O)c2O1 Cc1ccc(OCCC(=O)NC(C)(CNC(=O)CC2CCCCO2)C(C)C)cc1 Cc1cc(C)c(C(=O)NCC2(C)CCN(C(C3CCCOC3C)=O)CC2)c(O)c1 C1(CC)(NC(c2conc2C)=O)CCN(C(c2ccc(C)nc2C2CC2)=O)CC1 C(=O)(C(C#N)C(C)(C)C)NCCC(C)N(C(C(=O)NC(C)C)=O)C c1(OCC)cccc(NNC(=O)NC2CCN(CC(=O)N=c3cc(C)o[nH]3)C2)c1 c1(C(Cn2c(N3CCCC(NC(=O)OCC)C3)nnn2)(C)O)cc(Cl)ccc1Cl Cc1cccc(C=CC(=O)NC(CNC(=O)CN2CCSCC2)C(C)C)c1 C1(N(C(C)(C)C)C(=O)COC2CCOC2)CCN(C(C2(C)CCCS2)=O)CC1 N1(Cc2cccs2)CC(C(=O)OCC(C)OCC)CC1=O N1(C(C2CC(C)OC2)=O)CCCC2CN(c3ncc(O)cn3)CC12 N1(C(c2c(CC)ncs2)=O)C(C(=O)NCC(O)CCC2CC2)CC2CCCC12 C1(C(C)OC)CCN(C(C2CCC=CC2NC(C2CCCN(C)C2)=O)=O)CC1 O=C(O)C(F)(F)C(c1ccccc1)NC(=O)CC1CCCCO1 c1(CC(N2CCN(C(c3noc(CC)c3C)=O)CC2)=O)ccc2ncsc2c1 N1(C(c2c(CC)cnn2C)C(=O)NCCOCC)CCC23CCC(CC12)C3(C)C c1(C(=O)NC2CC2CNC(C(CC)C(C)O)=O)ccc2oc(C)nc2c1 C=CC1(C(N2CCN(C(C3CCC3)=O)C(CC3CC3)C2)=O)CCCCC1 C(CC(=O)NCC1CC2C(C1)C2(F)F)(C(C)(C)C)NC(C(C(C)(C)C)=O)=O c1(OC)ccnc(OC)c1C(=O)NCC(O)CNC(c1cc(F)cs1)=O C1(NC(c2cnc(C(C)(C)C)o2)=O)CCN(C(=O)CCC2CC2(Cl)Cl)C12CC2 c1(C(=O)NC(c2cn(CCCOC)nn2)C)cccc(OC)c1Cl C1(C(=O)NC(C2CCCN2c2cc(Cl)ncn2)(C)C)CCc2nnc(O)cc2C1 C1(C(N2CC(C)(NC(c3cccc(CC)c3C)=O)C2)=O)CCc2cnnn2C1 c1(C(N2CCN(C(c3csc(C)c3N)=O)C3C2C3)=O)ccc(S(N)(=O)=O)o1 C1(C(=O)NC2CN(CCC)C(=O)C2)CCN(C(=O)Cc2ccccc2C)C12CC2 Cc1cc(C)c2nc(NC(=O)NC3(C4CCC4)CCC3)sc2c1 N(C(=NCc1ccccc1)N1CCCC(O)CC1)C(C1(Cl)CCOCC1)C C1(CC(=O)NC(C)C(CO)NC(=O)CNC(C2CCOCC2)=O)CCCOCC1 c1(NC(C(N2CCC(CO)C(O)C2)c2n(C)nnc2)=O)cccc([N+](=O)[O-])c1 Cc1nc(C(=O)NCC2C3CN(C(=O)CC(C)NC(N)=O)CC23)nn1C CCC(CN(C)C)C(=O)NC1CCC1NC(c1cccc(O)n1)=O C1(NC(C(=O)NCC)=O)CC2CC1CN2C(C1CCCN1C(C)C)=O c1(OC)nc(C)ccc1C(=O)N(C(C)CCNC(C1CC(C)N(C)C1)=O)C N1(C(C2(F)CCN(C(c3c(CC)occ3)=O)C2)=O)CCOC(C)(C)C1C CC(CCC(C)(C)C)C(=O)NC(C)(CO)C(=O)Nc1cccc(C#N)c1 C(C)(C)(C#Cc1cn(C2COCC2O)nn1)NC(C(C)c1ccco1)=O C1(C)(CNC(C2(OC(C)C)CCC2)=O)CCN(C(C2(C)CC2(F)F)=O)C1 CCC(C)(CNC(=O)C(C1CCOCC1)O)NC(=O)Cc1cnn(C(C)C)c1 Nc1ncc(Br)cc1C(=O)NCC(F)CNC(=O)C1=CCCOC1 c1(C(N2C3C(NC(c4cn(C)nc4Cl)=O)CC(C3)C2)=O)cccc2c1ccn2C N1(C(c2ccccc2F)=O)CCOC(CNC(C2(CO)CCC2)=O)C1 CC1CN(C(=O)C=CBr)CCC1CNC(c1coc(C#N)c1)=O c1(C(N2CCC(O)(CNC(C=Cc3scc(C)n3)=O)C2)=O)cccc2oncc12 CC1CN(C(c2cc(=N)[nH]c(Cl)n2)=O)CCC1CNC(c1nocc1Cl)=O CCCCCC(CC)C(=O)NC1(C(=O)N(CC(O)COC)C)CC(F)(F)C1 C1(C2C(NC(=O)C(F)C3CC3)CCO2)CCN(C(=O)C=CC2CCC2)CC1 CCCCCC(F)C(=O)NCCC1CN(C(=O)C(C(C)CC)NC(N)=O)C1 Cc1cc(CC(=O)N(CCCNC(c2cn(C(C)C)nn2)=O)CCO)cc(C)c1 N1(C(COC(C)=O)=O)CCCC12CCN(C(c1sc(C(F)(F)F)cc1C)=O)C2 c1(C(=O)NC2CCCN(C(C(c3ccc(O)cc3)=O)=O)C2)ccc2n[nH]cc2n1 CCC(CNC(c1cc(C)n(C)n1)=O)(CC)C(=O)NCc1nccc(O)n1 C1(N(C)Cc2nc(-c3cccs3)no2)CN(CCN2C(=O)CCC2=O)CC1(C)C C1(C(N2CC(C)(NC(c3cocc3C)=O)C2)=O)(NC(C)=O)CCCC1 C1(CC(=O)NCC=CCNC(C(N2C(CC)CCC2)=O)=O)CS(=O)(=O)CCO1 C(=O)(CCCC(=O)c1ccccc1)NC(C(C)C)C(C)NC(C1(CSC)CC1)=O c1(NC(=O)CCc2cncnc2)c(Cl)cccc1[N+](=O)[O-].C12(CC1)CCN(C1CC1)C2 C1(CC(=O)NCC(O)CCO)CN(C(=O)CC2CCCC3CC23)CCO1 C1(C(=O)NCC2(COC)CCCC2)CCN(C(=O)C2(C#N)CCCOC2)O1 N1(C(CC2(NC(C(C)CC3CC3)=O)CC2)=O)CCC(C)C(F)(F)C1 Cc1ccc(-c2nc(C(=O)NC(C)CN(C(=O)Cc3ccsc3C)C)cs2)cn1 C1(NC(C2C(C)(C)C2)=O)CN(C(=O)CC2CCN(CC(F)F)CC2)CC1O c1(C(C)(F)C(=O)NCCCNC(=O)Cc2coc(C(F)F)n2)ccc(F)cc1 C(=O)(C1=CCCOCC1)NCCC1CN(C(C(C)Oc2c(Cl)ccc(C)c2)=O)C1 c1(C(=O)NCC2(CN(C(C(C(C)OC)O)=O)C)CC2)c[nH]c2cc(F)ccc12 CC1CC2CN(C(C3CC=CCO3)=O)CC2N1C(c1cnc2cccnc2c1)=O CCC(C(=O)NC(C1(NCC2CC2Cl)CC1)=O)C(C)C c1(C(N(CC(O)CNC(c2cnncc2O)=O)C)=O)cc2cccc(Cl)c2[nH]1 c1(OC)c(C(N2CC3CC2C3CNC(=O)C(C)C2CCOC2)=O)ccnc1Cl Cc1cccc2cc(NC(C3CN(c4nccc(C(N)=O)c4[N+](=O)[O-])C3)=O)[nH]c12 N1(C(c2cnc(Cl)s2)=O)CCC(CN2CCN(C(C3CC3C(F)F)=O)CC2)CC1 c1(SC(C)C(=O)NC2CC(NC(=O)C=CC3CC3)C2)ccc(F)cc1 c1(C(=O)NCc2ccc(C)s2)cc(CNC(=O)CC2(C#N)CC2)ccn1 CC1CCN(C(C2C3CC(=O)CC23)=O)C1CNC(=O)C(C)(Cl)Cl C#Cc1ccc(C(=O)NCCCC(CC)CC)cn1 C(=O)(C(C)(C)C(=O)N1CC(NC(C2CCC=CCC2)=O)CC(C)C1)OC c1(CNC(NCC(=C)Br)=NCCc2ccccn2)ccc2cnn(C)c2c1 N1(C(c2csc(C(=O)OC)n2)=O)CC(OCC)CC(F)(F)C1 c1(C(=O)NC(C(C)(C)C)CNC(c2cnc(O)o2)=O)cn2ccc(CO)cc2n1 C1(NC(C(COc2c(OC)cc(C)cc2)(C)C)=O)CCN(C)C2(CC2)C1 C(=O)(CCC(C)(C)C)N1CC(CNC(c2cnn(C)c2Cl)=O)C(C(F)(F)F)C1 C(=O)(C1=CCC(NC(=O)CC2C=CCCC2)C1)NC1(C(=O)OC)CCCC1 C(CC(=O)NCC1(C)CC2CC2C1)(C(F)F)NC(c1c(CC)c[nH]c1)=O CC(O)C(C)CN=c1cc[nH]cc1S(=O)(=O)NCC1(N2CCCC2)CCOCC1 c1(OC)ccccc1C1(C(=O)NC(C)(C)CCNC(c2ccsc2)=O)CC1 S(=O)(=O)(c1ccnc(F)c1)N1CCC(CN(C(C)C)C)CC1 c1(CC)cc(F)ccc1C(=O)NC(C1CCCN1C(=O)CCc1ccn(C)c1)C C1(NC(CC2(N(C(c3c(C)cccn3)=O)C)CC2)=O)CCN2CCCCC12 CN1CCC(C(=O)NCC(c2ccccc2)CNC(=O)CC(F)F)CC1 C1(NC(=O)C=Cc2ccoc2)CC2CC1CN2C(c1cnsc1)=O CC1COC(C(N2CC(N(C)C(c3cc(C4CC4)on3)=O)C2)=O)C1 C1(F)(C(N2CCC(NC(c3nnc(C(C)(C)C)s3)=O)C2)=O)C2CCCC12 C=C1CC(CNC(=O)NOCC(=O)N(C)C)(CC2(F)CCC2)C1 c1(CC(=O)NC2C(NC(C(CC)SC)=O)COCC2)cc2ccccc2nc1O C12(NC(CCOCC#C)=O)CCC(CN(C(=O)CC(C)CC(=O)OC)C1)C2 c1(CCC(=O)NC(CC)CN(C(=O)C(C)Cc2ccncc2)C)nc(C)c(C)o1 C1(N(C(=O)Cc2ccoc2)CC)CCN(C(C2CCCCN2S(C)(=O)=O)=O)CC1 N1(C(CSCCOC)=O)CC(NC(c2c(Cl)nn(C)c2Cl)=O)CC(F)C1 C1(C(=O)NC2CCC(CS(C)(=O)=O)CC2)Cc2ccc(Cl)cc2S1 N1(C(COC2(C)CCOCC2)=O)CCC(C2CC2)C1CNC(c1ccc(Cl)[nH]1)=O C(=O)(C(CC)NC(c1ccc(CNC(=O)C(c2ccn(C)n2)C)s1)=O)NCC c1(Nc2ncnc(N(C)C)c2Br)ccc([N+](=O)[O-])cc1S(C)(=O)=O O=C(NOC(c1cn(C2CC2)nn1)C1CC1)C(F)c1ccccc1 C(=O)(CC(COC)NC(C1CN(C)C(=O)N1)=O)Nc1c(CC)nsc1 N1(C(C2OCCN(C(C(=O)NCC)=O)CC2)=O)CC(O)CC(C)(C)C1 OC1CCN(c2nccc(-c3cccc(Br)c3)n2)CC1O c1(C(=O)NC(C)(C)CCO)coc2c1CN(C(C1CCC(C#N)CC1)=O)C2 N1(C(C(C(C)(C)O)F)=O)CCCC2(CCC2NC(=O)COC2CCC2)C1 Cc1cn2cc(C(=O)NC(C)CNC(c3cnc(S)nc3)=O)cc(C)c2n1 CC(C)CC(O)C(=O)NCC1(C)CCN(C(c2cn(C)nc2-c2cccs2)=O)C1 C1(N(C(C(CC)OC)=O)C)CCCN(C(c2ccc(-c3ccccc3)cn2)=O)C1 N1(C(CC2CC(CC)C2)=O)CCC2CCN(C(c3n[nH]cc3Br)=O)C2C1 c1(C(N2CC3N(C(C(C4CC4)SC)=O)C(CC3)C2)=O)ccc2[nH]c(=O)cnc2c1 CCCCCCC(C)(C)C(=O)NCCCC1CCCN1C(=O)CCC1CC1(C)C C1(C(=O)NC2CCC(NC(C3(CO)CCOCC3)=O)CC2)CN2CCC1CC2 CN1CCC(O)(CC(=O)NC2CC3CC(NC(=O)CNC(=O)C4CC4)CC23)CC1 c1(C(N(C2CCCN(C(=O)C(F)(F)C(O)C3CC3)C2)C)=O)cnc2occc2c1 CCC(CC(=O)NCC(C1CC1)NC(c1cc(Cl)c(Cl)[nH]c1=N)=O)C(F)F c1(OC)ccc2nccc(NCC3(C(=O)C(CC(C)C)N)CC3)c2c1.C1(CO)CC1 c1(NC(C(CCNC(C2(CCN=[N+]=[N-])CC2)=O)OC)=O)cnc2[nH]cnc2c1 Cc1nc(C(=O)NCCC(=O)NC2CC23CC(O)C3)sc1C c1(CC)ccc(C(=O)NCC2(NC(=O)C(C)n3cncn3)CCOCC2)c(C)n1 CC1(C)C(=O)NCCN1C(c1cc(-c2ccc3c(c2)CCC3)on1)=O C1(CNC(CN2CCC(C)C2)=O)CN(C(=O)CC2=CCCC2)CC(C)(C)C1 CC1CC2(CCC2)CN1C(c1cc(CNC(C2CN(C)C2)=O)[nH]n1)=O C(=O)(N(CCCO)OC)C1CN(C(C(CC)(C)OC)=O)CC12CC2 C1(NC(Cc2cc(C)no2)=O)CCN(C(=O)Cc2sc(O)nc2O)CC1C N(C1CCc2sc(Cl)cc21)C(N1CC=CC(CO)C1)=O C1(O)(CNC(C2C(CC)C2)=O)CCCN(C(=O)C(=CC2CCC(C)CC2)C)C1 Cc1cc(NC(c2ccnc(Cl)c2O)=O)ccc1NC(c1ccn(C(C)C)n1)=O N1(C(CC(C)(C)C(F)F)=O)CCC2C(CCCN2C(c2cc(O)cc(=O)o2)=O)C1 C(=O)(C(C(C)C)n1cnnn1)NCC(c1ccccc1)N(C(CCC=CC)=O)C n1(C(C)C)ncc(C(N2CCC(CNC(C3CN(C)CCO3)=O)C2)=O)c1F N1(C(CC(C(C)C)C)=O)CCCC2(C1)CN(C(C1(C(F)F)CCCO1)=O)C2 Cc1cc(C(=O)N(CC(C)NC(=O)C(CO)c2ccccc2)C)n[nH]1 C(=O)(C1CCCc2nnn(C)c21)NC(CNC(C(CSC)(C)C)=O)CO c1(NC(C2CCCCN2C(c2cc(Cl)c(F)c(Cl)c2)=O)=O)c(Cl)ccc(O)c1Cl N1(C(C(C)NC(CC)(C)C)=O)CCC(NC(=O)C2=C(Cl)CC2)C12CCCC2 Cc1cc(C(=O)NCC2(C)CCN(C(C34COCC3C4)=O)C2)nc(C)n1 C1(NC(C2C(C)(C)C2NC(=O)Cn2cnnc2O)=O)CC2CCC(C1)C2O C1(NC(C(COC)OC)=O)CCN(C(c2cnc(S)nc2)=O)C1(C)C c1(N2CCC(NC(c3c(C)nc(O)cc3)=O)C2C)nc(Cl)nc(C)c1F CC(O)(CNC(=O)C(Cc1ccco1)NC(C1CC12CCC2)=O)CO C1(NC(c2c(OC)nn(C)c2)=O)CCC12CCCN(C(c1cnc[nH]1)=O)C2 N1(C(C2OCCN(CC)C2)=O)CCOCC(NC(=O)CCCN=[N+]=[N-])C1 Cc1ccc(C)c(C(=O)NCC23CC2CN(C(c2cnn(C(C)C)c2)=O)C3)c1N c1(NC)cncc(C(=O)NC2CCN(C(=O)C(c3cccnc3)OC)C2)c1 c1(C(C2CCCCC2)N(C)Cc2c(C(=O)OC)ncs2)cccc(OC)c1 N1(c2cc(NC3CCN(C)C(=O)C3)ncn2)CCCOCC12CCCC2 C=CC(CCC)CC(=O)N1CC2CCC(NC(=O)Cc3c[nH]ccc3=O)(C2)C1 C12(CC(=O)Nc3ccc(CC)o3)CCC1CN(C(C1CCC(OC)CC1)=O)C2 CCC(CNC(C1CCCCN1C(C)C)=O)(CC)NC(=O)CCCF CCCCC(CCCC)C(=O)N(CC(O)CNC(=O)C(CO)C(F)(F)F)C Cc1cc(C)n(CC(=O)NCCN(C(=O)C(C)(C)C(N)=O)C2CC2)c(=O)n1 CCCCCC(CC)C(=O)NC(C1CCCN1c1ncc(Cl)c(O)n1)(C)C C1(C(N(CCCNC(c2c(C(C)C)n[nH]c2)=O)C(C)C)=O)CCCOC1C C1(C(=O)NC(CNC(C=CSC)=O)(C)C)C(F)(F)C12CC2 c1(CN(CCC)CCN(C)C)cc(-c2ccc(C)o2)ccc1OC c1(C(N2CC(OCC(N3CCC(C)(C)C3)=O)C2)=O)cc(O)cc(=O)o1 N1(C(=O)OC)CCCC(C(=O)NCC2CCC(CNC(=O)C(F)(F)CF)CC2)C1 C(=O)(CC(C)CC(=O)NC(c1nocc1C(=O)NC1CC2CCCC2C1)C)OC CC1CC(O)CN(C(c2cccc(C(C)(C)C)n2)C(=O)NC2CC2)C1 c1(OC)cc(C(N2CCC(C(C)NC(c3c(F)ccnc3Cl)=O)C2)=O)ccc1C C12(CNC(=O)Cn3nnc(=O)[nH]3)CN(C(c3cnc4n3CCS4)=O)CC1CCO2 N1(C(C(CC=C)(C)C)=O)CC2CC(O)C1C2NC(c1ccc(F)cc1OC)=O C1(N(C(=O)CC2CSCCO2)C)CCCCC1N(C)C(C1CC12CCCC2)=O c1(OC)cccc(C(=O)NC2CN(C(c3cc(C)ncn3)=O)CC2F)c1 c1(C(=O)NCCn2cc(COC(=N)O)nn2)sc2cc(Br)ccc2c1Cl CC1CN(C(=O)CCCC(C)(C)C)CC(C)C1NC(=O)Cc1cc[nH]c1 N1(C(CCN(c2nn(C)cc2C)C2(OC)CN(C)C2)=O)CC2CCC(CC2)C1 N1(C(C(CC#C)C)=O)CCC2C1CCCN2C(c1cc(=O)n(C)o1)=O c1(C(=O)NOCC2CCCO2)ccc2cccc(F)c2n1 N1(C(c2c(CC)noc2)=O)CC2CC1C2CNC(c1c(C)noc1C(F)(F)F)=O c1(C(N2C(CNC(C3CCc4c[nH]nc4C3)=O)C=CC2)=O)cc2cccnc2[nH]1 C1(C(N2CCC(Cn3cc(C(C(=O)OC)(F)F)nn3)CC2)=O)CCCCC(=O)N1 c1(CC(=O)NCC23CC2CN(C(c2ns[nH]c2=O)=O)C3)ccc(C(F)(F)F)cc1 c1(-c2cc(C)c(C#N)cc2)ccc2cc(NC(C3CCCO3)=O)ncc2c1 C1(NC(C(CC)OC)=O)CCN(C(c2cnn3cc[nH]c(=O)c23)=O)CC12CCC2 CCCC(C)(CC)C(=O)NC1CCN(CCCNC(=O)CC2CCSC2)C1 C1(CCNC(=O)CCF)CC(F)(F)CN1C(=O)CC(O)C1CCCC1 CN1CC(NC(=O)C2=CCC(NC(=O)CCC3CCC(=O)C3)C2)C2(CC2)C1=O c1(C(N2CCN(CCOCCOC)CC2)=O)ccc2ncnn2c1 c1(C(N2CCC(C)C2CNC(c2cc3cscc3s2)=O)=O)cc2occc2n1C N1(C(C(c2ccccn2)C)=O)CC(NC(=O)C(C)CC2CCC2)C2CCCCC12 C1(C2CC2)(C(=O)NCC(C)(CO)CO)CN(C(=O)CN2CCOC2=O)C1 c1(CN(C(c2ccc(Cl)nc2)C(=O)NC)C)cc(Cl)c(O)c(Br)c1 N1(C(C(C(C=C)C)C)=O)CCn2nc(C(=O)Nc3c(C)cccc3C)cc2C1 c1(CC(=O)NC(CC)CNC(C2CC(F)(CO)C2)=O)ncncc1Cl C1(NC(C(CC)OCC)=O)CN(C(c2cc(C)ccc2N)=O)CCC1(C)C c1(OC)ccc(OCC(=O)NCCCCN(C(=O)C(C)(C2CC2)OC)C)cc1 CC1(C2CCN(C(c3cn(CCNC(c4ccc[nH]4)=O)nn3)=O)C2)CC1 C1(N(C(c2nc(C)oc2)=O)C)CN(C(C2(CNS(N)(=O)=O)CC2)=O)CC1O C1(CNC(c2c(C)cccn2)=O)N(C(=O)Cc2cc[nH]c2)CCCC1(C)C N1(C(c2c(C)nccc2)=O)CCC(C)(C)C1CC(=O)N(C)Cc1cc(=O)cc[nH]1 C1(CC)(CC)Oc2ccc(NCC3CCCN(C(=O)OC(C)(C)C)CC3)cc2O1 Cc1ncc([N+](=O)[O-])n1CC(=O)NCC(C)(C)CNC(=O)CC1CCCC1C CCCCC(CNC(C1CC1OC)=O)NC(c1ccc(OCC(F)(F)F)o1)=O N1(C(C(CCC=C)NC(c2csc(=N)[nH]2)=O)=O)CCN(C)C(=O)C1C C1(CC(=O)NC2CC(CNC(CCNC(=O)CO)=O)OCC2)CC(O)C12CCC2 N1(CC(C)NC(=O)C(CNC(C2CNC(=O)O2)=O)N(C)C)CCCC1=O Cc1ncccc1C(=O)NCCC(C)(C)CNC(=O)CCCc1nncn1C N1(C(C(CCC)C)=O)C(C)CC2CN(C(=O)CCCOCCOC)CC12 N1(C(C(C)n2cccn2)=O)CCN(C(=O)CN2C(=O)CNC2=O)CC1C1CCC1 Cn1cnc2cncc(C(=O)NCCNC(=O)CCCn3ccnc3)c12 N1(C(c2c(C)nn(CO)c2)=O)CCCC(NC(=O)COC(C)(C)C(F)(F)F)C1C C1(O)(CNC(C=Cc2n(C)cnc2)=O)CCCN(C(=O)CC(C)(C)O)CC1 C1(NC(=O)Cc2nnc(O)s2)CN(C(c2cccc(-c3cc[nH]n3)c2)=O)CC1O CC1=C(C(=O)NCC2(NC(c3ccc(C(F)F)cc3)=O)CC2)C(=O)OC1(C)C O=C(CC1=CCCC1)NCC1(CNC(=O)C(F)C2CCCC2)CC1(F)F N1(C(C2CC(C)N2C(=O)CCc2cccs2)=O)CCN(C)C(C)C1 C#CCC(C(=O)N1CCC(NC(c2ccc(COC)cc2)=O)C1CC)C1CC1 C(N=c1[nH]cnc(NCC(C)(C)S(C)(=O)=O)c1C)c1cncc(SCC)c1 c1(C(N2C(CN(C(=O)CN3CC4CC4C3)C)COCC2)=O)n[nH]c2c1COCC2 Cc1ccc(F)c(C(N2CCC(CNC(=O)C(C)(O)Cc3ccccc3)C2)=O)c1 N1(C(C2C(C)C2)=O)CCC(N(C(=O)CSCCN(C)C)C)CC1.C12CCC(C1)N2 N1(c2c(OC)cncn2)CC(NC(=O)CCNC(c2ccccc2)=O)CC(C)C1 c1(CC)ccc(C(=O)NC2CC23CC(NC(=O)C(C)(C)CSC)C3)cc1 C1(C(N(C(C=C)C2CC2)C)=O)(NC(C2CCCN2C(=O)C2CC2)=O)CC(F)C1 c1(OC)ccc(C)nc1C(N1CC(CNC(c2cccnc2C)=O)C1)=O c1(C(N2C(CN(C(CSCC=C)=O)CC)CCC2)=O)cc(N)ccc1C N1(C(C(C)N2CCCC2)=O)CC2CCCC2C1C(N1CCCC(O)C1C)=O c12ccc(cc1)C(=O)NC2.C1(CCNC(C)=O)CCCCN1C(=O)COC(C)C CC1CN2CCN1CC2C(=O)NC1(CCNC(=O)CC2CCCSC2)CC1 C1(CNC(c2cc(C(C)C)[nH]n2)=O)(NC(=O)C(O)C(C)C)CCC(F)(F)CC1 c1(C(N(CCC(=O)NCC2CCC(CO)CC2)CC)=O)cccc(C)c1C#N C1(NC(CC2CCC(OC)CC2)=O)CN(C(C2(F)CCOC2)=O)CC12CC2 N1(C(CC=CCC)=O)CCOCC1CC(=O)NC(CO)C(C)(C)C N1(C(CNC(CCc2n(C)cnn2)=O)=O)CCCCC(CO)C1 N1(C(C2(NC(C(C)CC(F)F)=O)CCCCC2)=O)C2CCC1CC(F)C2 CCCC(C)C(=O)NC(C)CCN(C)C(C1CC1c1cnn(C(C)C)c1)=O n1(CC(=O)N(CCC)CCNC(=O)C(O)Cn2cncn2)cnc2c1CCCC2 N1(C(C(C)SC)=O)CC(NC(c2cscc2SC)=O)CC1(C)C C1(CC(=O)NCC(CC)NC(=O)C(C)(C)CSC)SC2=NCCN2C1=O N1(C(=O)NC(c2ccccc2O)C)CCOCC(NC(C2(C)COC2)=O)C1 N1(CCC(=O)N(CCOCCN(C(CS(CC)=O)=O)C)C)C(=O)NC(C)(C)C1=O N1(C(C2C(C(=O)OC)C2)=O)CC(C2CCCN(C(=O)CCCC3CCCC3)C2)C1 C(CCCC(CO)NC(=O)C(C)C1CCCC1)NC(c1c(CC=C)cccc1)=O N1(C(C(CC)C)=O)CCC2CN(C(c3cc4cc(Cl)ccn4n3)=O)CCC12 CC(C)CC(C)(CNC(=O)C(c1ccc(F)cc1)CO)NC(=O)CNC(N)=O N1(C(c2ccnc(OC)n2)=O)C(C(=O)N(CC(C)CO)C)CCC12CC2 C1(C(=O)NCC2(F)CC(NC(=O)CC3CCCO3)C2)CCCOC1c1cc[nH]n1 CC(C)CC(F)(F)C(=O)NCC(C1CC1)N(C(=O)C(C)Cc1ccc(F)cc1)C N1(CCC(=O)NCC(C2CC2)NC(c2c(CC)nns2)=O)C(=O)NC(C)(C)C1=O C(CC(C(=O)NOC1CCCC1)NC(=O)C(C1CCCC1)OC)OC C=CC1COCC1NC(C12CC(CO1)C2)=O N1(c2c(C)cc(-c3nn[nH]n3)cn2)CCc2nc(C(=O)N(C)C)ccc2C1 N1(C(c2c(CC)ccs2)=O)C2CCCC1CN(C(c1cc(C(C)C)n(C)n1)=O)C2 c1(C(=O)NC2CCC(CC(=O)N(CCN=[N+]=[N-])C)C2)cc2ccccc2o1 C(=O)(CCCCC(=O)NCC1CC(C)N(C(=O)CCc2nc(C)cs2)C1)OC C1(C)(C(N(CC)Cc2ccoc2)=O)CN(C(c2cccc(O)c2F)=O)C(C)(C)C1 CC(CC(=O)N(C)CC1(O)CCN(C(=O)CN2CCCC2)C1)CC(C)(C)C Cc1nc(C)n(CC(=O)NCc2ocnc2C(=O)NC23CC(C2)C3)n1 C(C)(C(=O)N1CC(CC(N2CC(N(C)CCO)C2)=O)C1)N(C(C)=O)C c1(OC)cc(O)c(C(=O)N=c2ccn(-c3ncccc3Cl)[nH]2)cc1Br N1(C(C2C(=C)C2)=O)CCC(CF)(NC(=O)COCc2ccccn2)C1 C1(C)(C(c2cnn(C)c2)C)CN(C(=O)Cn2cc(C3CCC3)nn2)C1 C1(NC(Cn2c(C)c(Cl)cn2)=O)CC(NC(c2cc(C)n(C)c2C)=O)C12CCC2 C1(N(C(=O)C(F)OC(F)(F)F)C)CN(C(=O)Cc2csc(=N)[nH]2)CC1F C(=O)(C(C)(O)C(C)C)N1CC(CC=C)(NC(=O)C(N2CCSCC2)C)C1 C1(C)(NC(CC2C(CNC(c3c(CC)cccc3)=O)C2)=O)C(C)(C)C1(C)C c1(C(N(CCC)CC2CCCO2)=O)cn2c(n1)CCN(CC1CC=CCC1)CC2 C12(C(=O)NCC3C(C(=O)NC(c4ccsc4)C)CC3)COCC1C2 CC1(C)C(NC(=O)C(F)C2CCOC2)CCN1C(C1CCN(CCO)C(=O)C1)=O c1(-c2cn(C3CCC(NC(CCc4cnn(C)n4)=O)C3)nn2)cncc(N)c1 c1(C(N2CC(NC(=O)CC3CCCCC3O)C3(C2)CC3)=O)ccc2nncn2c1 c1(C(=O)NC2C(CNC(=O)Cn3nnc(C(F)(F)F)n3)C2)ccnnc1S C1(C(N2CCN(C)C(=O)C2)=O)CN(C(C2CCS2(=O)=O)=O)CCC1(C)C c1(OC)ccc(C(O)CNC(C2CCN(C(c3c(C)n[nH]c3C)=O)C2)=O)cc1 C1(NC(C2ON=C(C)C2)=O)C2CC1CN(C(c1ccccc1C(F)(F)F)=O)C2 C1(N(C(c2c(C)nns2)=O)C)CCN(C(C)C(=O)NCc2ccccn2)CC1C C1(CNC(CCN(C(CC2C(CC)C2)=O)C)=O)CCCC1(C)C CCC(C)C(C)C(=O)NCc1ccccc1CN(C)C(c1ncnc(C)c1C)=O C1(F)(CC)CCN(C(=O)CC2CC(NC(=O)C=Cc3cc[nH]c3)C2)C1 c1(N(C)C)cncc(NC(C2C=CCN(C(C3CC(F)(CF)C3)=O)C2)=O)c1 C1(C(=O)NCC2(F)CCOC2)(NC(Cc2c(C)n(C)nc2)=O)CCC(C)(C)C1 C=CC1(C(=O)NCC2(OC)CN(C(=O)CC(C)c3cnn(C)c3)C2)CCOCC1 c1(C(=O)NC2CCCN(Cc3cc(F)c(Cl)cc3O)C2)cccc([N+](=O)[O-])c1F N1(C(C(=O)NCC)C(C)C2CCCC2)CCN2CC(O)CC2C1 C(=O)(CC(C)(C)C(=O)NCCC1CN(C(=O)C(C)OCC(C)C)CCCO1)OC N1(C(C(c2cc(C)sc2)(F)F)=O)CCC2(NC(=O)Cc3ccnn3C)CCCC12 N1(C(C2N(CCC)CCC2)=O)CCCC1(Cn1ccc(CC(=O)NCC)n1)CC c1(NC(c2nnnn2CC2CC2)(C2CCCOC2)COC)cc(Br)ccc1C CCC(CCCC(=O)NC(C)C1CC1)NC(=O)C=C(C)C(C)C C1(=O)C(NC(=O)OC(C)(C)C)CCNCCN1C.c1(COC)cscn1 C12(NC(Cc3nc(C)sc3C)=O)CCCC1CN(C(=O)C=CC1CCOC1)C2 C=CCC(C)(C)CC(=O)OCC1NC(=O)NC1=O.c1(C(=O)NCC)cscc1 c1(C(C)(C)C)cn2c(n1)C(C(=O)N1CC3CC1C3NC(c1cn[nH]c1)=O)CCC2 N1(C(Cc2n(C)nc(CC)c2Cl)=O)CC(C)OC2(CCN(C(=O)C(C)(C)C)C2)C1 C1(c2cc(C)on2)CCCN1N1CCC(C(C)(C)O)C1 CC(C)CCC(F)C(=O)NC(C(=O)NC1CCCC(C2CC2)C1)C1(C)CC1 CN1C2CCCC1CN(C(C1C3CCC(C3)C1NC(c1ccc[nH]1)=O)=O)C2 N1(C(Cc2c(C)ocn2)=O)CC(NC(=O)CN(S(C)(=O)=O)C)CC1CO C(=O)(CC(C)CC(C)(C)C)NCC1(F)CCC(NC(C2(COC)CC2)=O)C1 N1(C(CSCC#C)=O)CCC2(CCCN2C(=O)COCC2CCCO2)C1 c1(C(N2C(C)CC(CCNC(C3(O)CCCC3)=O)CC2)=O)coc2c1CCCC2 c1(C(=O)NC)ccc(-c2cncnc2N2CC3CC(O)C2C3)cc1F c1(C(N2CC(NC(=O)Cn3ccnn3)C(O)C2)=O)ccnc2ccc(F)cc12 c1(OCC)ccccc1NC(=O)NC1CCCC1NC(=O)CC1(C#N)CCC1 C1(C(N(CC(c2nn[nH]n2)C)C)=O)CC2CCCC2N1C(C1C=CCCC1)=O C#Cc1cc(C(=O)NC2CCN(C(c3ccc(N)c(N)n3)=O)C(C)C2)ccc1Cl S(=O)(=O)(CCC(F)(F)F)NC1CCN(C2CCN(c3ccc(C)cc3)CC2)CC1 N1(C(C(c2ccn(C)n2)C)=O)CC(CNC(=O)C(C)(C)N(C)C)C(C)C1 C1(CCC)CN(C(C2(C#N)CCCOC2)=O)CCN1C(=O)Cc1ccccc1Cl C(CC1=CCN(C(C2CCC3CC3CC2)=O)CC1)NC(=O)CC1CNC(=O)N1 c1(C(=O)NC(C2CN(C(=O)CC3C=CS(=O)(=O)C3)C2)C)cnc(C2CC2)nc1 c1(C2(C(=O)NC3C(NC(C4CCC(=O)N4)=O)C3)CC2(Cl)Cl)ccc(F)cc1 c1(CC)cc(CCC(=O)NC(C)Cc2ccnc(N(C)C)c2)ccc1O Cc1ccc(O)cc1C(=O)NOCC(N1CC(C2CCCO2)C1)=O c1(C(N2CC(O)(C(C)NC(C3CCC(C)(CC)O3)=O)C2)=O)cc2n(c1)CCCC2 Cc1cc(C(=O)NC2CC2NC(c2cncc(Cl)c2)=O)ncc1S(N)(=O)=O Cc1cc(Cl)c(C(C)NC2CCN(CCCO)CC2)cn1 N1(C(C(CC=CCC)C)=O)CCC(C)(C)C(NC(C2(N(C)C)CCCCC2)=O)C1 c1(C(=O)NC(C(=O)NCCC(C)SC)C2(O)CCC2)ccc(CF)cc1 Cc1cc(C(N2CC(C(=O)NCc3nc(C)c(C)[nH]3)CCC2C)=O)c(C)nn1 N1(C(C(=O)N(C)C)=O)CCC2(CC1)CC2(C)C(=O)NCCS(=O)(=O)NC1CCCC1 C1(NC(Cc2cccc(OCC)n2)=O)CC2CC(NC(=O)CNC(N)=O)C2C1 C1(C(N2C3C(NC(C4N(C)CCC4)=O)CC(CC3)C2)=O)CCCC12CCOCC2 c1(C(N2C(CNC(=O)CSc3cccs3)CC(O)C2)=O)noc2c1CCCC2 N1(C(CCCOCCOC)=O)CCC2CC1CN(C(=O)CN(S(C)(=O)=O)C)C2 CCC(C(=O)N1CCC(N(C(=O)CCCOCC)CC2CC2)CC1)C(C)O CCCC(C)(CC)C(=O)NCC1(C)CCN(CC2CCC(C)CC2)CC1 O=C(CC1=CCCCC1)NC1CC(CNC(C2(c3ccno3)CCOCC2)=O)C1 Cn1cc(NC(=O)CCC2CCN(C(=O)CCn3ccnn3)C2)c(C#N)n1 N1(C(c2n(C)c(S)nn2)=O)CC2(CCN(C(C3CN4CCCN3CC4)=O)CC2)C1 N1(C(Cc2cn3cc(C)sc3n2)=O)CC2C(C1)C2N=c1[nH]c(Cl)ncc1Br c1(C(N2CC(COC)(CNC(c3cc(CO)ncn3)=O)C2)=O)nccc(Cl)c1C C1(C2CCC2)(C(=O)NC(C)(CNC(C2CCCC(=O)O2)=O)C2CC2)CCCCC1 c1(N(C)Cc2ccc(C)c(C)c2)nc(N2CCCN(C)CC2)c2c(n1)COC2 c1(C(N(C2CCN(C(c3nc(=O)n(C)[nH]3)=O)CC2)C)=O)cnc2ccncc2c1 C1(NC(c2c(C(C)(C)C)ncs2)=O)CCC2CCN(C(=O)Cc3cccs3)C12 c1(C2N(C(=O)NC3CCN(c4ccccc4)C3)CCC2)ccc(F)cn1 C1(NC(C(C)(C)C)=O)CCCCC1CNC(c1ccc(-c2cc(O)ns2)cc1)=O N1(C(CCC2(C)CN(C(C=CCN(CC)CC)=O)C2)=O)CCCC(OC(C)=O)C1 N1(C(C=CCC)=O)CCC(NC(c2nc(OC)c(C)s2)=O)CC1C CCC(CC(=O)NC(C1(O)CCN(C(=O)CCn2cnnn2)C1)C)C1CCC1 c1(C(=O)NC23C(CN(C(C=C(C)Cl)=O)C2)C3)sccc1S(C)(=O)=O c1(CNC(C2(C(C)(F)F)CC2)=O)ncccc1CNC(=O)CNc1ccsn1 N1(C(c2cc(C(NC(=O)C(c3cccnc3)O)C3CC3)no2)=O)Cc2ncsc2C1 C(C(=O)N=c1cc(-c2cccs2)[nH][nH]1)(c1cccc(OC)c1)SC c1(C(C(=O)NCC(CNC(COC)=O)C)O)ccc(C(C)C)cc1 C#Cc1cncc(C(=O)NCC2COCCN2C(c2ccc(CO)cc2F)=O)c1 Cn1ccc2c(C(=O)NC3CC34CCN(C(=O)COC(F)(F)F)CC4)ncnc12 C1(NC(C(C)OCC)=O)COC2(CNC(=O)CCCCc3cnc[nH]3)CC1C2 C1(CC(=O)O)C2CCC(C2)N1C(N(CCCC=C)C(C)(C)C)=O.C1CC1 C(C(CC(F)(F)F)NC(c1ccsc1OC)=O)NC(C(CC)SC)=O c1(CNCC2CCN(C(c3cncn3C(F)(F)F)=O)C2)cc(Cl)sc1Cl Cc1ccc2c(c1)N(C(C1CCC(NC(C3CC3[N+](=O)[O-])=O)CC1)=O)CC2 CCC(CC)CCCN(C)C(C1CCCN1C(=O)COCCOC)=O c1(NC2C(SCC)CCC2)[nH]c(=NCCN2CCCCC2=O)nc2scnc12 c1(C(N2CC(NS(CCOC)(=O)=O)C3(C2)CC3)=O)ccc(O)c(F)c1F.C1(O)CCCC1 Cc1ccc(F)cc1-c1nc(C(=O)Nc2cscn2)ccc1F Cc1c(C(C)NC(c2cncc(N(C)C)c2)=O)oc2ccccc12 Nc1c(Cl)ccc(F)c1C(N1C2CCC1C(NC(c1cnc(C3CC3)o1)=O)C2)=O c1(CN(CC(C(C)C)C)Cc2ccccc2)ccc(Br)c(C#N)c1 N1(Cc2scc(C)n2)CCN(C(c2csc(CCP(C)(C)=O)n2)=O)CC1 N1(C(C(C(=O)OC)C)=O)C2CCC1C1CC1(NC(=O)C=C(C)c1cccs1)C2 C1(C(=O)NC(CNC(Cc2cccc(OC)c2)=O)C(C)C)CCC(C)(C)CC1 C=CCN=C(NCCC(C)(C)COC)NCC1(CF)COCCC1=O Cc1csc2c(CC(=O)NC3CC4CN(C(c5cnn[nH]5)=O)CC4C3)cccc12 c1(C(N2CCN(C(C(C3CCCCC3)C)=O)CC2CO)=O)nccn2nccc12 N1(C(C(CC(CC)C)C)=O)C2CCCC1CN(C(=O)CN(c1ccccc1)C)C2 Cc1ccc(C(CNC(C2CC2(Cl)Cl)=O)NC(c2ccn(C(C)C)c2C)=O)cc1 c1(C(N2C(CC(=O)OC)CC3(CC3)C2)=O)csc(S(C)(=O)=O)c1 C=CC(F)(F)C(=O)NCC1(F)CN(C(c2cnn(CC3CCCC3)c2)=O)C1 C=CCN(Cc1ccccc1)N1CCC(CC(=O)N(C)C)C(F)(F)C1 C(=O)(C(C)(C)C(O)C(C)C)N1C(C(=O)OC)CC(Oc2cccc(OCC)c2)C1 c1(CC)nc(C(N2CCCC2C2CCN(C(c3cnsc3)=O)C2)=O)c(N)s1 C1(CNC(COCC(=C)C)=O)CC2CC1CN2C(C1C=CCC1)=O N1(C(c2sncc2C)C(=O)NC(CC)(C)C)CCCCC1CCC(F)(F)F c1(C(=O)OC)ccc(CO)cc1NC(C1(C(C)C)CCC1)=O c1(CCC(N2CC(NC(c3cc(C)sc3)=O)C3C2C3)=O)c(O)nc(=N)[nH]c1C c1(C(N2CCN(CC(C)(C)NC(=O)CC3CC(F)C3)CC2)=O)ccc(C#N)cc1 C1(CCN(CC[Si](C)(C)C)C)CCC2(CCC2)O1.c1(CC)cscc1Br c1(C(N2CCC(N(C(c3cccnc3C)=O)CC)C2)=O)cccn2c(O)nnc12 C1(C(=O)NCCC2(O)CN(C(C(C=C)O)=O)C2)(C(=O)OC(C)(C)C)CCSCC1 Cc1ccc2c(c1)OC2.c1(C(=O)NCc2cccnc2)c[nH]nc1Cl C1(CC(=O)NC(c2cnccc2C)=O)COCCN1CC.c12cnoc1NC2=O c1(-n2c(-c3coc(C4CCC4)n3)nc(CC(C)OC)n2)cc(Cl)nc(Cl)c1 c1(OC)ccc(CN(C2CCCSC2)C(=O)NCC2C3CC4C(C3)C24)cc1 c1(C(C)NC(C(COC)NC(=O)C(O)Cn2cncn2)=O)c(C)n[nH]c1C C1(CNC(C(COC)(C)C)=O)CC2CCC1N2C(c1cncc(C(C)C)c1)=O O=S(=O)(c1ccc(-c2csc3ccccc23)cc1)NCCc1cccc(F)c1Cl C1(C(c2n(CCOC)nnn2)NCCSC)(COC)CCCCO1 N1(C(c2cc(C)n(C)c2)=O)CC2CC(NC(c3nn[nH]c3C(F)(F)F)=O)C2C1 CC1=C(C(=O)N2CCC3CN(C(=O)CC4CC(=O)NC4=O)CC23)C(C)(C)CCC1 N1(C(C=COC)=O)CCOC(C(C)NC(c2cnccc2N(C)C)=O)C1 S(=O)(=O)(c1ccc(NCC(C)OC)nc1)N(C(CCCC)(C)C)CC C1(C(=O)NCC2(CO)CCN(C(=O)C#CC3CC3)CC2)CCN2CCCC2C1 CC(C(=O)N1CC(F)(CNC(C23CCC(F)C2CC3)=O)C1)S(C)(=O)=O CS(=O)CCC(=O)N1CC2CC2C1CNC(=O)CCCC1CCOCC1 C1(NC(=O)NCc2cc(C)nn2C)CCCC(OC(C)(C)C)CC1 C1(NC(CC=CC=C)=O)CCN(C(=O)C(C)(C)C(C)C)CC1(C)C Cc1cccc(F)c1CC(N1CC2CC1C2NC(=O)Cn1nnc(=O)[nH]1)=O N(C(=NCCc1ccc(O)c(OC)c1)NC(C)C)Cc1cn(CC)nc1 N1(C(c2cnc3ccnn3c2)C(=O)NC(CC)(C)C)CCCN2CCCC2C1 C1(CC(=O)OC(C(CCC)N(C)C)=O)CN(CC(C)(C)C)CC1(C)C n1(CC)nc(C)c(C(=O)N(C)CC2(O)CCN(C(C3(SC)CC3)=O)CC2)c1Cl c1(CC(=O)NCCN(C)Cc2cn(-c3ccncc3)nn2)ccc(S(N)(=O)=O)s1 N1(C(C=C(COC)C)=O)CCCC(CCC(=O)NC(CCO)C2CC2)C1 c1(C(N2CC(NC(c3c(Cl)cnc(SC)n3)=O)C(F)C2)=O)cc(Br)cc(Br)c1O n1(CC)nnnc1C(C)(C1CC1)NC1(c2cccs2)CC1 C(=O)(C1Cc2ccc(Cl)cc21)NC1C(CNC(c2c(COC)cccc2)=O)CC1 c1(C(=O)NCC=CCNC(c2ccn(CCC)n2)=O)cc(Cl)ccc1OC Cc1c(C(=O)N(CCCNC(C2CCCOC2C(C)C)=O)C)ccc2cncn12 NS(=O)(=O)CCCC(=O)NCC1CC(NC(C2CC3CCC2CC3)=O)C1 CC(CC1CCOCC1)C(C(=O)NC1CCOC1)N(C1CCN(C)CC1)C N1(C(c2cc(-c3ccc(OC)c(Br)c3)no2)=O)CCC2(CC1)CCS(=N)(=O)C2 C#CCC(CC(=O)NCC(C1CCCCC1)C)NC(c1ccc(C)s1)=O C(c1cccnc1)=C(C)C(N1CCC(C)(NC(=O)C=CC(F)(F)F)C1)=O Cc1ccc(C(=O)NC2(CO)CCN(C(C3(C)C=CCC3)=O)C2)c2ncccc12 N1(C(Cn2c(C)c(Cl)cn2)=O)CCC(CCNC(c2cn(C)c(O)n2)=O)CC1C C(CS(=O)(=O)CCN=c1[nH]c(=NCC(C)OC)[nH]c2c(F)cccc12)OC C1(CC(=O)NC2C3CN(C(C4C(CC)C4)=O)C2C(O)C3)CC2(CCOCC2)CO1 Cn1cc(C(N2CC(C(=O)N(N3CCOCC3)CS(=O)(=O)CC3(C)CC3)C2)=O)cn1 C=CCC(CNC(c1ncccc1Cl)=O)C(=O)NC(CC(=O)NC)C1CC1 C(=O)(CC(C)C1CCC1)NCC(N(C(C=CCOC)=O)C)C1CC1 Cc1ccc(C)c(C(N2CCC(C)N(C(C3(F)CCCC3)=O)CC2)=O)c1N C1(C(=O)NCC(=C)Br)CN(C(=O)Cc2nc(=N)[nH][nH]2)CCC1(C)C N1(C(CC(CNC(C(=O)NCC)=O)OC)=O)Cc2ccccc2C1 C1(NC(CC(C=C)C)=O)CN(C(c2nc(C(F)(F)F)cc(C)n2)=O)CCC1C Cn1cc(C(=O)NCCNC(=O)C(C)(C)NS(C)(=O)=O)cn1 N1(C(Cc2cccc(C)c2)=O)CCN(C(c2cc(O)nc(Cl)c2)=O)CC1C Cc1ncc(Br)c(N2CCC(NC(c3ncn(C)n3)=O)C(O)C2)n1 N1(C(Cn2nnc(C)n2)=O)CC2(CCN(CCCC(C)(C)C)CC2)CC1C CCCCCC(CC)C(=O)NCC1CC(F)CN1C(c1ccn2c1CCCC2)=O C1(C)(C(=O)NC2CCC(CCC(=O)NCC(C)(O)C3(C)CC3)C2)CC2CC2C1 C1(=O)C(CC(C)C)ONC(=O)CC(C)N1.c1(CC)cc(CCO)on1 N1(C(C=C(CC)C)=O)CCC2(CC1)CC2CNC(C1CC2CCC1C2)=O C(=O)(C(F)C(F)(F)F)NCC(CNC(c1c(OC)noc1C1CC1)=O)C c1(C(N(C2CCCC2)CCCNC(C2OCC(C)C2)=O)=O)cnc2occc2c1 N1(C(C2CCCS2)=O)CCC2(CCCN2c2nc3cccnc3s2)C1 Cc1c(C(=O)N(C)CC2CCCN2C(=O)CCCC2CCCC(=O)N2)ccn1C c1(N(C(=O)NC(c2cccc(OCC)c2)CCC#C)CCC)cc(N)ccn1 C1(C(C(=O)NCC2CCOC2)N(CC(F)F)C(C)C)CCCC(C)C1 C(=O)(C1=CCCC1P(C)(C)=O)N1CC(C(C)NC(CCCCCOC)=O)C1 C1(C(N2CCC(C)(C)C2)=O)CC2(CCN1)CCOCC2 c1(NC(=O)NCC2(C(F)F)COC2)ccc(F)c(F)c1.C1CC(=O)N1C(C)=O c1(CN(C(c2c(C)cno2)=O)C)ccccc1CNC(=O)CC1CC(C(F)F)C1 c1(C(C(=O)N2CC(OCCNC(C(CC)=CC)=O)C2)C)nc(F)ccc1Cl N(C(=NCc1cccc2c1OCCO2)N1CC(C)N(C)C(C)C1)C(CC)C C1(C(=O)NCC2(CCNC(C(C(C)C)O)=O)CC2)CCc2ncnn2C1 n1(CC(=O)NCC(CNC(C2CCSC2)=O)OC)ncc2ncccc12 N1(C(CCC(CC)C)=O)CCC(C2CC2)(CNC(c2ccon2)=O)C1 c1(OC)cc(F)ccc1C(=O)NCC1CN(C(=O)Cc2ccc(Cl)s2)CCCO1 N1(C(C(C2CCCCC2)OC)=O)CC2CC(NC(C3(C)CC3)=O)CC(C2)C1 c1(C(=O)NC(C(=O)N2C(C)(CC)CC2)CCOCCO)ccc(C)c(O)n1 C(=O)(C1=C(C#N)CCC1)NCC(C1CCN(C(C(CC(C)C)C)=O)CC1)(C)C C1(CNC(C(C)NC=O)=O)CN(C(=O)CCc2cccnc2F)CC(C)(C)O1 c1(OCC(=O)N(CC(CNC(C(COC)(F)F)=O)C)C)c(F)c(F)cc(F)c1F c1(C(=O)NC2CN(C(c3c[nH]nc3Br)=O)CCC2O)cc2cncn2c(O)n1 c1(CCNC(C2(CCCOC)CCCC2)=O)cc(Cl)sc1Cl C1(NC(C2N(C(C)=O)CCC2)=O)C2CC(NC(c3csc(Cl)c3)=O)CC12 C12(NC(C3CCC(CC)O3)=O)COC(CNC(c3cc(C4CC4)on3)=O)(C1)C2 C(C(C(=O)N1CCc2nn[nH]c2C1)C(C)(C)C)NC(C(COC)N(C)C)=O c1(C2(C)C(c3cn(C)nc3)C2)nc(CC2CCCC2)nn1-c1ccnc(O)c1 C1(C(N2C3C(NC(C(CCCC)(C)F)=O)C(C3)C2)=O)CCn2c(cnc2C)C1 c1(CC(N2CCC(O)(CNC(C3CCC(C)CC3)=O)C2)=O)cc2ccccc2[nH]1 C1(C(=O)NCC(CC)NC(c2cnc[nH]c2=N)=O)CC(c2ccccc2)=NO1 c1(OCC(=O)NCCNC(c2cc(Cl)no2)=O)ccc(Cl)cc1 NS(=O)(=O)c1cc(C(=O)N(CCCNC(C2(C(F)F)CCCC2)=O)CCO)cs1 CC(c1ccccc1)=CC(=O)NCc1cc(C)c(C(N2CC(S(N)(=O)=O)C2)=O)o1 CN=c1[nH]nc(CC(=O)NCCC2CCCN(C(C3(C(F)F)CCC3)=O)C2)s1 C1(CNC(C=CCN(CC)CC)=O)CCCN(C(c2cnn(C)c2SC)=O)CC1 C=CCC(CC)C(=O)NCc1cc(C(=O)NC(C)CN(CC)CC)no1 N1(C(c2noc(CC)c2C)=O)CCC(C2CC2)C1C(=O)NC1(C)C(C)(C)C1(C)C C1(C(Cn2cc(COC)nn2)F)CCN(C(c2c(Cl)nsc2Cl)=O)CC1 C1(CCNC(=O)CCNC(c2cccs2)=O)CCCN1C(c1ccsc1)=O C1(C(N2C(C(N)=O)CC2)=O)COC2(C1)CN(C(=O)C=Cc1ccc[nH]1)C2 N1(C(c2nc(C)c(C)s2)=O)CCC2(CCN(C(C3CCC(C)NC3=O)=O)CC2)C1 c1(C(N2CC(NC(C(CC)(C#N)CC)=O)C(C)C2)=O)cncc2ccc(F)cc12 c1(C(=O)NCCN2CCN(C(C3C(C)C3)=O)CC2)ccc2c(c1)OCCCO2 Cc1ccccc1CCNC(=O)C=CC1CCCN1C(=O)C(C)O n1(CC(=O)NC2CC(CNC(=O)C(F)(F)C3CC3)C2)ncc2ccccc12 N1(C(C(C)C2CC2)=O)CCC(F)C(NC(c2cnc(N3CCOCC3)nc2)=O)C1 c1(OCC)c(C(N2CCC(CN(C(=O)CC3CC(C)=NO3)C)C2)=O)cccc1F c1(C(=O)NCC2(C=C)CCC2)cccnc1CC.C1(=O)C(CC)N1.C(=O)(C1CC1)N C(C1(CC(=O)OC)CCOc2ccccc21)Nc1ncc(OC)cc1F CC1CC(NC(=O)C=CC(=O)NC2CC2)CN(C(=O)C#CC(=O)N(C)C)C1 C(C(=O)NC1CCOCC1)(C(C1CCCC1)OC)N(C(C)COC)CC=C CCC(CC)(C(=O)NC1CC1NC(=O)CSc1ccc(F)cc1)OC C(=O)(C(C(C)C)NC(=O)C(N1CCOCC1)C)NCc1c(C)nns1 c1(C(N(CC(CN(CCSC)C)O)C)=O)ccc2cc(C)ccc2n1 CCC(C)C(C(C(=O)NC(C)C(=O)OC)N1CC(C)OC(C)(C)C1)OC Cc1cc2c(cc1C)N(C(C1(C)CC3(CCC3)C1)=O)CC2 S(=O)(=O)(c1ccc(-c2cccc(O)c2)cc1)N1C(C)(CC)CC1 c1(C(=O)NC2CN(C(CC3(C)CCCCC3)=O)C2)cc2nc(F)ccc2o1 CN1C(=O)CCC1C(=O)NCCN(C(C1CCOC1)=O)Cc1cccc(Cl)c1 c1(NC(C(=O)N(CC)CC2CC3(CC3)C2)=O)cccc(NC(=O)OC(C)(C)C)c1 Cc1nc(C)n(CCCC(=O)NC2CCN(C(c3coc(C(F)(F)F)n3)=O)C2)n1 c1(C(N2CCC(N(C(C=C(COC)C)=O)C)C2)=O)cc(=O)n(C)c2ccccc12 C1(CNC(C=C(CCC)C)=O)CCCCN1C(=O)COc1cc(C(F)(F)F)ccn1 N1(C(C(C)=CC)=O)CC(C)CN(C(=O)Cc2c(F)cccc2Br)CC1C c1(NC2CC(CC(C)(C)C)C2)ccccc1CCP(C)(C)=O C(=O)(CCC(C)S(C)(=O)=O)N1C(CN(C(C(CC=C)(F)F)=O)C)CCCC1 CC1CC(C)(C(=O)NC2CCN(C(=O)COCCN(C)C)CC2CO)CCO1 c1(C(N2CCN(C(c3nccc(CC)c3)=O)C(C)C2)=O)c(C)cc(C)cc1O N1(C(CCOCC#C)=O)CCN(C(=O)C(O)C2CCCC2)CC(C)C1 N1(C(C2N(C(CCC)=O)CCC2)=O)CC(NC(C2CCCN2C)=O)CC(F)(F)C1 C12(C(N3C(C)CC(F)C3)=O)CCC(NC(=O)NC3CCC(N=[N+]=[N-])C3)(CC1)CC2 C1(OC)CCCC1NC(C1(CO)CCC1)=O.C12CCCN1C2=O Cc1ccccc1OCC(=O)NC1(CNC(C2(c3ccncc3)CC2)=O)CCC1 C12(CNC(C3CC(C(C)C)C3)=O)CCC1CN(C(=O)CCc1cccc(O)c1)C2 Cc1conc1CNC(C1CCCC1CNC(C1CCC1C(C)(C)C)=O)=O c1(NC)ncc(C(=O)NCC2CN(C(c3ccnn3C(C)C)=O)CCO2)cc1Cl N=c1cc[nH]cc1C(=O)NC1CCN(CCNC(=O)Cc2ccccc2)CC1 CC1(NC(c2cncc(N)c2)=O)CCN(C(=O)CC23CNC(=O)C(C2)C3)CC1 C(C(CC(F)(F)F)NC(=O)CC12CCCC1C2)NC(c1cncc(C(C)C)c1)=O C(=O)(CC(=O)NC(C)CC(C)NC(=O)C(C1CCCC1)NC(C)=O)OCC CCC(Cc1ccccc1)CC(=O)NC1C2(NC(C3(CO)CC3)=O)CCC(C1)C2 c1(C(CNC(=O)NCc2ccn(C)n2)OC)ccccc1C c1(C(N(CCCNC(=O)CC2CC2C2CC2)C)=O)cc(O)nn1C C(=O)(CCC(CF)CF)N1C(C(C(=O)NCC2(O)CCC(C)C2)(C)C)CCC1 c1(C(=O)NCCOCCNC(CC=C)=O)c[nH]cc1CC C1(CNC(Cc2cccc(SC)c2)=O)CN(C(=O)CC2CCC2)C2CCCC2O1 c1(C(N2C(CNC(c3cccc(F)c3O)=O)CCCC2)=O)cc(Cl)cc(Cl)c1O N1(C(C2OCC(C)C2)=O)CC2CCCN(C(c3ccc(-c4ccco4)o3)=O)C2C1 CC1(CNC(=O)CC2(C#N)CC2)CCC(NC(c2csc(CO)n2)=O)C1 c1(OC)cc(OC)c(F)c(CN2CCC2C(=O)NC2CC(CO)C(O)C2O)c1F CC12CCCC(C(N3CCC(CNC(=O)C=Cc4ccc(F)cc4)C3)=O)(CO1)C2 c1(COC(c2csc(-c3ccccc3)c2)=O)ccc(O)nn1 c1(C(=O)NCC2CN(C(C(c3ccccc3Cl)(C)N(C)C)=O)C2)nnccc1C C(=O)(C1=CC2CCCC12)OC1CC(=O)OC1 C(=O)(C(CC(C)C)C(C)C)N1CCN(C(c2c(C)ncs2)=O)CC1C CCCCCCC(CC)NC(=O)CC1C=CC(NC(C2CCC(F)CC2)=O)C1 C1(COC)CCN(C(C2(CNC(=O)C=CC3CC3)CC(C)(C)C2)=O)CC1 C1(C)(C(N2CC(CN(C(C(F)=C(C)C)=O)C)OCC2)=O)CCCCCC1 c1(C(N2CCCC(CC=C)(NC(C3CCC(F)C3)=O)C2)=O)c(C)cc(=O)oc1C CCC(C)C(O)C(=O)NCC1CC(NC(c2ccc(CO)nc2)=O)C1 C1(CCNC(c2c[nH]c(Br)c2)=O)CCCCN1C(c1ccc(CO)nc1)=O C(=O)(C1=COCCO1)NCC1CC(NC(C(C)(C)c2ccccc2)=O)C1 C#Cc1cc(F)ccc1CN1CC(C(N2CC(OC)C2)=O)CC(F)C1 C1(CC(C)NC(CC=C)=O)CC2CCC(C1)N2C(=O)Cc1ccc(C)cc1 c1(C(N(C2CN(C(CC(CC)CC)=O)CC2(C)C)C)=O)cnn2ncccc12 C(=O)(C(C)(C)C(=O)NCC1CC(O)CN1C(C1(N2CCCC2)CCCC1)=O)NC C1(C(N2CCC(SC)C2)=O)CC12CCN(C(=O)C1=COCC1)CC2 C(=O)(CC(C)(C)CC(F)F)N1CC2(OCC(NC(Cc3c(C)occ3)=O)C2)C1 CC1CC(C#N)(C(N2CCOC(CC(=O)NC(c3nncs3)C)C2)=O)C1 CC1(O)CCN(C(c2cc3c(s2)CCC3)C(=O)Nc2ccccc2)CC1(C)O C1(C(=O)NCC(=O)NCC(=O)NCC(CCC)C)CSCC(=O)N1 Cc1ccc(C(C)NS(=O)(=O)C2CC2c2cccc(Br)c2)c(C)c1 Cc1nccc(Cl)c1C(=O)NCC1C(C)CCCN1C(=O)C1=NOCC1 C1(CNC(c2cn(CC=C)nn2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)CC1 c1(CNC(C)=O)ccc(C(=O)N(C2CC(NC(C3CC=CC3)=O)C2)C)cc1 Cn1cc(Cl)cc1C(=O)NC1C2CN(C(=O)CC3CNC(=O)O3)CC12 C1(OC)(CNC(=O)CC2CCN(C)C2)CCN(C(c2c[nH]ccc2=O)=O)C1 C(=O)(C1=CCN(C(=O)C2=NOC(C)(C)C2)CC1)NC1C(CC)CCCC1 C1(C)(C(=O)NC(CCC)CNC(c2ccnc(O)c2)=O)CCC2CC2C1 c1(C(=O)NCCN(CCC)C(C2CC(C)CO2)=O)ccncc1-c1ccccc1 N1(C(c2cnn(C)n2)=O)CC(C(=O)NC2CC(=O)NC2=O)CCC1(C)C CC(C)CC(F)C(=O)NCC1C=CC(NC(=O)CCc2cn[nH]c2)C1 CC(C)(O)C(F)(F)C(=O)N1CCC(C(N2Cc3cccnc3C2)=O)CC1 N12CCc3[nH]nc(c3C1)C2.c1(C(=O)O)ccc(C(F)F)nc1 c1(NC2CCC(N)(CC(=O)OC)CC2)cccc(N=S(C)(C)=O)c1 C(=O)(CC(C)CC(C)(C)C)NCC#CC(N1CCCC(C)(CCC)C1)=O c1(C(=O)NCCCNS(CC)(=O)=O)ccc(C(F)(F)C(F)(F)F)cc1C c1(N2Cc3c(O)nccc3CC2)nc(=NCC2CC2(F)F)[nH]c2c1CSC2 C1(CC(=O)NC2CN(C(c3cc(-c4ccccn4)c[nH]3)=O)C2)CN2CCC1CC2 C1(NC(C=C)=O)CCOCC1C(=O)Nc1cccc(OC(C)C)c1 CC1CC(CCNC(=O)C=C2CCC2)CCN1C(=O)CC(=O)NC1CC1 N1(C(c2c(C)ccc(O)c2)=O)CCCC(O)(CNC(=O)CSCC(F)F)CC1 C(CC(F)F)(C(=O)NCc1ccns1)NC(C1CCN(C)CC1)=O c1(C(N2CCN(C(COC(C)=O)=O)C3C2CC3)=O)cccc(C#CCO)c1 C(=O)(C1SCCc2ccccc21)N1CC(C)C(NC(C2(C)CCOCC2)=O)CC1 CC(C(=O)NCCOCCNC(=O)CN1CCC(F)(F)C1)C(F)(F)C(F)F N1(C(Cc2ccc(C)o2)=O)CCC=CC1C(N1CCC(N(C)C)CC1)=O C#Cc1cc(C(=O)N(C)CC2(O)CN(C(C3CCC3C)=O)C2)cc(Br)c1 N1(c2cc(C)ncn2)CC2CCN(Cc3cc4cc(Br)ccc4[nH]3)CC2C1 C1(CNC(CCN(CCCCC)C(C)C)=O)CC(F)CN1C(c1ccns1)=O C1(C(=O)NCCC(C)NC(c2cnc(C3CC3)nc2)=O)CCC(=O)N1C CCC(CCCC(=O)NCC1CCC(=O)O1)NC(C1(CF)CC(=O)C1)=O CCC(C)CC(=O)C(=O)N1CCC=CC1C(=O)NC1(c2cc[nH]n2)CC1 CC1Cc2c(Cl)c(Br)cc(F)c2CN1N1CCCC1c1ncccn1 N1(C(CC2C(C)=NN(C)C2=O)=O)CCC(NC(=O)Cc2cc(C)on2)C12CCC2 N1(C(C2CCN(C(C(CC=C)C)=O)C2C(C)C)=O)CCC12CCC(C)CC2 C1(C(=O)Nc2c(CC)ccnc2)CC2(CCC2)CN1C(C1CCCC1C(C)C)=O CC1=C(C)CC(C(=O)NCC2C(C(=O)NC34CC3CN(C)C4)C2(C)C)CC1 N1(C(c2ncc(C)cc2C)=O)CCC(NC(=O)C(F)(F)C(C)(C)O)C(C)(C)C1 CC(C)C(N=c1nc2[nH][nH]cc-2c(O)n1)C(C)NC(=O)C(O)CCc1ccccc1 N1(C(c2cc(OC)no2)=O)CCC2CN(C(C3CCC=CCCC3)=O)CC2CC1 C1(F)(CN(c2ncccn2)C(c2ccc(C3(O)COC3)cc2)=O)CCCNC1 C1(OC)(CNC(C2CC(Cl)(Cl)C2)=O)CCN(C(=O)CCC2C(=O)NN=C2C)CC1 C(=O)(C1=CCC(NC(c2ccccc2F)=O)C1)NC(C1(O)CCC1)C C(CC(C)(C)C(=O)NCCC1CCCO1)NC(c1c(C)ccnc1)=O c1(NC(c2ccc(OC)c(Br)c2OC)=O)cc(C#N)c(F)cc1C CC(C)CCCC(C)C(=O)NCC1COCCN1C(c1ccnn1C)=O C1(C(=O)NC(CN(C(C2(CC#C)CC2)=O)C)C)CN(C)CCO1 C1(C(N(CCCNC(Cc2cccs2)=O)CC)=O)CN(C(=O)NC)CCO1 C1(C)(C(=O)NC(CN(C(=O)Cc2sccc2C)CC)C)CCC2CC2C1 CCC(C(=O)N(CC(C)(C)CNC(c1ncccc1C(F)(F)F)=O)CC)C(C)O N1(C(CCC)C(=O)NCCCC2CC2)CCc2c(O)cccc2C1 C(=O)(CC(C)C(C)(C)C)N(C(C(CC)C)C(=O)N(CC(O)CO)CCO)C C1(CNC(CN(C)C)=O)CCC2(CC1)CCN(C(C1CCC3(CC1)CC3)=O)CC2 C=CCC(C(=O)NC(CNC(=O)C=Cc1ccccc1)(CC)CC)OC Cc1ccc(C(=O)NC2(C3CN(C(C4(C#N)CC4)=O)C3)CC2)c(F)c1Cl N1(C(C(CCC=C)NC(=O)Cc2cccs2)=O)CC2C(=O)NC(=O)C2C1 c1(C(=O)NCCC(C)NC(CC=C=C)=O)cccnc1C(F)F c1(C(c2cccs2)NC(=O)NCCC(C)(C)O)ccc(F)cc1 C(=O)(CCCCCF)NC1C(OC)CN(C(=O)CCCC2CCOCC2)C1 N1(C(C(c2ccc(Cl)cc2)CC)=O)CCC(F)CC1(C)C CCC(C(=O)NCCN(C(=O)C(C)COC)C1CC1)C(F)(F)F c1(C(=O)NC(C)CCNC(=O)CSc2nccn2C)sc(F)cc1Cl c1(CC)nc(C)[nH]c1C(=O)NC12CC(CNC(C3(O)CCOCC3)=O)(C1)C2 C1(N(C(CN(CC)CC)=O)CC)CCN(C(c2cc(C(F)(F)F)n[nH]2)=O)C1C CCC(C)C(C)C(=O)NCc1cc(C(=O)NCCC2(C)CC2)ccn1 C12(C(=O)NCC3CC(C(=O)OC)C3)CCC(CN(C(C3(C)C=CCC3)=O)C1)C2 c1(C(=O)NC(CCOC)CNC(C2COCCOC2)=O)ccc(F)c(C)c1Cl C(=O)(C(CN(C)C)C(C)C)N(C(C)C(N1CCC(CC(C)C)CC1)=O)CC C1(CNC(C(C)CF)=O)CCCN(C(C2(C)CC(F)C2)=O)C1 C(=O)(CS(=O)(=O)C(C)(C)C)NCC(c1ccccc1)N(C(C1C(=C)C1)=O)C N1(C(c2cn[nH]c2)=O)CCC(F)(F)C(CNC(C2(F)CCCCCC2)=O)C1 N1(C(C2(C#N)CC(C)C2)=O)CC2(COC(CNC(=O)COC3(C)CCC3)C2)C1 N1(C(C2CCC(C)(C)CC2)C(=O)NCCOCC)CCCCC(S(C)(=O)=O)C1 N1(C(C2CCS(=O)CC2)=O)CC2CCC(C1)C2N1CCCCC1 C1(C(=O)OC)C2CC1N(C(C1(CNC(=O)OC(C)(C)C)CC(C)(C)C1)=O)C2 C#Cc1ccc(CC(N2CCC(C(=O)Nc3cccc(F)c3)C2C)=O)cc1 CC(CCN1CCCC1)N=c1[nH]c(=NCC2(CC3CC3)CC2(C)C)[nH]c2c1CSC2 C1(C(=O)NCCn2c(CC)nnc2)CN(C(=O)C(C2(O)CCCC2)F)CC1C C1(C(=O)NCCN(C(C(CN(C)C)(F)F)=O)C)OCCOC12CCC2 CN1CCN(C(c2ccn(C)c(=O)c2)C(=O)NCCCC2CC2)CC1=O N1(C(C2C(C#C)C2)=O)CC2CN(C(C3(c4ccc(C(N)=O)cc4)CC3)=O)CC2C1 c1(C(=O)NCCC(C)N(C)C(C2CC2(Cl)Cl)=O)cn(C)nc1-c1ccncc1 C(=O)(C(CCC1CCC1)NC(c1cc(CO)on1)=O)NCC(CC)n1cccn1 Cc1ncc(C)c(NC(N2CCN(c3cccs3)C(=O)C2)=O)n1 C1(C(N(CC)Cc2ccc(O)cc2)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CC1O N12CC3CCCC(C3C1)C(=O)NOCC2.O=C1CC1NC(=O)C(F)(F)F N1(C(C2CCC(OC)C2)=O)CC2=C(C1)CN(C(c1c(Br)cnn1C)=O)C2 C(=O)(C(CNC(=O)C(F)CC1CCOC1)N(C)C)N(CC(=O)OC)CC1CC1 C(=O)(C(C)(C)C1CCN(C(=O)C(O)CN(C)C)C1)NCC(c1ccncc1)C c1(C(=O)NC2C(C)N(C(c3csc(O)n3)=O)CCC2)ccc2c(c1)CCCC2 c1(OC)cc(NC(=O)C(CCNC(=O)C(F)=CC2CC2)OC)cc(F)c1 C1(C(=O)NC2CN(C(CC(CC)(F)F)=O)CC2C)COc2ccc(F)cc2C1 N#Cc1nc(Br)cnc1NC(C1CCCN(C(c2cnc3snnc3c2)=O)C1)=O Cc1ccc(CN=C(NCC(F)F)NC2COC3CC2C3)c(SC(F)(F)F)c1 CC1CN(C(c2c(C(F)(F)F)ncn2O)=O)CCC1NC(C1CN(C(N)=O)C1)=O C1(N(C(C(CC)C)C(=O)OC)C(=O)C(C)=O)CCC2(CCNCC2)CC1 C(=O)(C(CC(C)C)NC(=O)OC)N(CC(CNC(c1noc(CC)c1C)=O)C)C Cn1c(C(N2CC(S)CC2Cn2cc(CCS(N)(=O)=O)nn2)=O)cc2sccc12 c1(C(N2CCC(CNC(=O)CC3COCCO3)CC2)=O)cc2cc(Cl)ccc2s1 N1(C(C2C(C)C2)=O)CCC(C2CCCN(C(C3CCc4nn[nH]c4C3)=O)C2)C1 c1(NC(C)=O)cccc(F)c1C(=O)NC1CN(C(=O)C2CC2)CC1F C1(C(=O)NOCC2CCC2)C(C2CC2)CCN1C(c1occ2c1CCC2)=O CC#CCCC(=O)N1CCCC(NC(C2CCC(N(C)C)CC2)=O)C1 C1(NC(C(C)S(N)(=O)=O)=O)COC2(C1)CN(C(=O)C#CC1(C)COC1)C2 N1(c2c(C#N)cncc2)C2CCC1CN(C(c1cc(CN)no1)=O)C2 C1(CNC(c2cn[nH]c2)=O)CN(C(c2cn(CC(F)(F)F)cn2)=O)CCCO1 c1(CC)csc(C(F)(F)C(=O)OCC=Cc2cnco2)n1 Cc1cccc(OC(C)C(=O)NC(C)CC2CCN(C(C3CCC3)=O)CC2)c1 c1(C(=O)NC(C(=O)NCC)C)n[nH]cc1CNC(c1cc(COC)on1)=O c1(OC)nccc(Br)c1C(N1CC(N(C2CCC2)C(C2C=CCCC2)=O)C1)=O N1(C(C2(C)CCC(N(C)C)C2(C)C)=O)CCC2C(C1)C2(F)F c1(CCC(=O)NCC(=C)CCNC(c2csc(O)n2)=O)ccncc1Br c1(C(N(C2CCC(NC(=O)Cc3ccon3)C2)C)=O)cc(C2CC2)ncn1 C12(CNC(C(C)=CC3CC3)=O)CCCC1N(C(=O)CC(O)C1CC1)CCC2 c1(CC(=O)NC2C(CNC(CN(C)CC)=O)CC2)c[nH]c2cc(Cl)ccc12 C1(C(C)C)CN(C(=O)CC2CCSCC2)CCN1C(C1CCOC1)=O CC1=C(C(=O)N2CCC(C)(NC(=O)CCC3CCCCN3C)C2)C(C)(C)CCC1 c1(C(=O)NC2CC(CNC(CC(COC)(C)C)=O)C2)ccc2c(c1)NC(=O)CC2 c1(CNC2C(C(=O)Nc3c(C#C)nccn3)C2)cnc2ccc(C)cn12 c1(C(=O)OCC2(CC(=O)OC)CCOCC2)cc(Cl)c(Br)cn1 CN(C(=NCC12CC(CO1)C2)NCC1CCCCO1)Cc1cc(F)cc(F)c1 C=CCCCC(=O)NCC(C)NC(c1ncoc1-c1ccccc1F)=O c1(OC)cc(C(N2CCN(Cc3cnc(Cl)cn3)C3CC23)=O)cc(O)c1O C(N=c1nc2c(cnn2C)c(NCC2CC3CCC2CC3)[nH]1)c1ccc(SC)s1 C12(C(N(CCC)CCNC(=O)CC(C)C)=O)CC(COCC)(CO1)C2 C1(N(C)C(c2ccc(C#N)s2)=O)CCCN(C(=O)CCNc2cncnc2)CC1 N1(C(CCSCCC)=O)CCN(C(=O)CC2CCN(C)C2)CC(O)C1 C1(NC(C2N(C(C)C)CCC2)=O)CC12CC(NC(=O)C1CC1)C2 N1(C(c2cc(CC)nc(O)c2)=O)CC2(COC(CNC(C3(F)CC3)=O)C2)C1 Cn1c(CCC(N2CCCC2(C)C(C)(C)C)=O)nnc1S O=C1OC2CCC1CN(C(C1CCC(n3cc(CCCCO)nn3)C1)=O)C2 N1(C(C(CCC)OCC)=O)CCC2(CC1)OCCC2NC(c1cnccc1Cl)=O c1(OC)cc(C)c(C(=O)NCC2C=CCN2C(=O)CNS(=O)(=O)NC)c(C)c1 C1(C(C)C(N2CCC(n3ccnc3)C2)=O)CCN(C(C2CC2(F)Cl)=O)CC1 N1(C(c2c(C)nsc2)=O)CCC2(C1)CN(C(=O)CCC1CC1)C2 c1(C(N2C(CNC(c3cnc(C)[nH]3)=O)CC2)=O)cncc(Cl)n1 N1(C(CC)=O)CCCC(O)(CNC(c2cccn(C3CCSC3)c2=O)=O)CC1 N1(C(c2cc(OC)nc(Cl)c2)=O)CCN(C(=O)CC(C)N(C)C)C2CCC12 C1(CC(=O)NCC(C)N(C(CCc2onc(CC)n2)=O)C)CCCC1(F)F C(=O)(C1CCCc2cncn21)N1CCC(COC)(NC(c2cc(CO)[nH]n2)=O)C1 N(S(=O)(=O)N1CCCC1C)C(CCC)Cc1ccc(C(F)(F)F)cc1F N1(C(c2ccc3c(c2)COC3)=O)CCC2C(CCCN2C(=O)Cc2ccon2)C1 N1(CC(=O)NCCc2ccn(-c3ccccc3)n2)CCCCC1Cn1cncn1 Cc1cccc(C)c1CN1CCCC(NC(=O)C(C)Cc2c(C)n[nH]c2C)C1 C1(C(=O)NCC2C(NC(C(C(=O)OC)(C)F)=O)CC2)CC2(C1)CC(F)(F)C2 C(=O)(CCCC(=O)NC(C1CCN(C(=O)C(C)OCCOC)CC1)(C)C)NC C1(CNC(c2nc(COC)sc2)=O)CC2(CC2)CN1C(=O)C(C)n1ccnn1 CC1SCCCC1C(=O)NC1(C)CC(C(=O)NCCOC2CC2(F)F)C1 C(C1CCCCCC1)=CC(=O)NC(CC(C)C)CNC(=O)CC1CCC(C)(C)C1 CCS(=O)CC(=O)NC1COCC1CNC(c1[nH]c(-c2ccccc2)nc1C)=O C1(NC(CNC(CC)=O)=O)COC2(CCN(C(c3ccc(Cl)c(O)c3)=O)CC2)C1 N1(C(C2(CC=C)CC2)=O)CCCC1CNC(=O)C(O)CC1CC1 CC(C)(O)C(F)C(=O)NC1CN(C(=O)Cc2nc(=N)[nH][nH]2)CC1F c1(OC)cnccc1C(=O)NC(C)C(C)NC(=O)C(F)(F)c1csc(=N)[nH]1 C(C(C)(C)CC(=O)Nc1cncnc1C)NC(c1oc(CC)c(C)c1)=O C1(C2CN(C(Cc3c(NC(C)=O)cno3)=O)C2)CN(C(=O)CC(C)(C)O)CCO1 c1(C(=O)NC2CCC(NC(C3C(F)(F)C34CCC4)=O)CC2)c(F)ccc(F)c1F N1(C(=O)CCC2CCC(=O)N2)CC2CCC(NC(=O)CSCc3cccs3)(C2)C1 S(=O)(=O)(c1ccc2oc(O)nc2c1)N1CCC(F)(C(N2C(C#N)CCC2)=O)CC1 c1(C(=O)NCC)nccnc1Sc1ccc(Cl)cc1.c12ccccc1[nH]c(=O)[nH]2 c1(C(=O)NCC(CN(C(c2cccc(C3CC3)n2)=O)CC)(C)C)cc[nH]c(=N)c1 CCCCC(O)C(=O)NCC1CC2(CC2)CN1C(C1CCCN(CC)C1)=O N1(C(C2(c3ccnc4ccccc34)CC2)=O)CCOC2(CCc3ccccc32)C1 c1(C(=O)NC2CN(C(C3ON=C(C(C)C)C3)=O)CC3C2C3)ccc2c(cnn2C)c1 C(C(C)C(F)C(=O)NC(CCO)C(F)(F)F)NC(C1CN(C(C)=O)C1)=O c1(COC)nc(N2CCC(NC(c3c(Cl)cncc3Cl)=O)C(O)C2)cc(O)n1 CCS(=O)(=O)CC(=O)NCc1ccccc1CN(C(=O)Cc1conc1C)C c1(CC(=O)NCC2(OC)CN(C(c3cncc(C)c3)=O)C2)ccccc1SC C(=O)(C1CCc2snnc21)NC1CCCC(NC(C(C)(C)n2ccnn2)=O)C1 N1(C(C(=O)NCC(c2cnn(C)n2)C)=O)CCC(C(F)(F)F)C(F)(F)C1 C1(NC(C=C(C)CNC(=O)CC2CCCC2O)=O)CC=C(C)CC1 Cc1ccc(C(=O)NCC2(C)CCCN2C(C2COC(C)C2)=O)cc1N C(=O)(C#CC1CCCO1)N1CC(CNC(CC(c2ccc(CC)cc2)C)=O)C1 N1(Cc2nc(-c3ccc(OC)cc3)oc2)CCC2(CC1)CNC2C(C)C c1(CC(=O)NC2C(C(N3CCCN(C)CC3)=O)CCC2)c(F)cc(F)cc1F c1(C(N2C(C)CC(CNC(c3cc(C(C)=O)oc3)=O)C2)=O)ncnc2sccc12 C1(CNC(=O)C(O)c2ccsc2)CCN(C(=O)CC2CCCCO2)CC1 C1(C(=O)NCCN(CCC)C(c2cc(CC)nnc2C)=O)CCn2ccnc2C1 c1(C(=O)NCC2(C(N)=O)CN(C(CN(CCC)C)=O)C2)ccn(CC2CC2)c1C C(=O)(C(O)CC(N)=O)N(CC(=O)N(CCCO)C)C(C)C C(=O)(C(C)CC(F)F)N1C(C(=O)NC2CC(C)OC2=O)CC(OC)C1 S(=O)(=O)(c1cc(C(=O)OC)ccn1)NCC(=O)NC(c1ccncc1)CC C(C(CO)(CO)NC(c1cc(C2CC2)nn1C)=O)N(C(=O)CC1CCCC1)C c1(C(N2CCC(CNC(c3ccccc3C(F)F)=O)C2)=O)c[nH]c(=O)cn1 C1(CNC(CC2(C)CCCCC2)=O)CC2(CC2)CN1C(C1CCCC(F)(F)C1)=O C1(C)(C(=O)OC)CC(C(N2CCC(NC(=O)C(C)COc3ccccc3)C2)=O)C1 N(C1CCc2sc(Br)cc21)C(CC)C(c1ccc(Cl)cc1)=O C(=O)(C(CC)C(C)(C)CC)NCC(CC)NC(c1ccnc2c1ncn2C)=O C1(CN(C(CCc2onc(CC)n2)=O)C)CN(C(=O)Cc2ccns2)CCO1 c1(C(=O)NC2CN(C(C3(Cl)CC3)=O)CC2C2CC2)cc(=O)n2ccsc2n1 Cc1nc(C(=O)NCCC(O)CNC(=O)C=CC2CCC2)cc(O)n1 N1(CC(=O)NC2CC(NC(c3sccc3F)=O)C2)CSCC1=O c1(C(N2C(CCC(=O)NCCn3ncnn3)CCC2)=O)cc(=O)cc[nH]1 C(=O)(C1CSc2ccccc21)NC1CCCN(C(c2cc(CC)nn2C)=O)C1C N1(C(COC(CC)(C)C)=O)CC(C)CN(C(=O)CCCc2ncco2)CC1C C12(NC(C(C)NC(C)=O)=O)CCCN(C(C3CC(=O)N(C)C(=O)C3)=O)CC1C2 N1(C(CC(C=C)C)=O)CCN(C(=O)C(CC)(CC)CO)CC2(CC2)C1 C1(NC(c2ccccc2Cl)=O)(CO)CCN(C(=O)CCC(F)(F)F)CC1 N1(c2snc(COC)n2)CC2CC1CCC2NC(C1CCc2nncn2C1)=O N1(C(Cc2c(C)sc(Br)n2)=O)CC(C)c2ccccc21 Cc1cc(CC(=O)N(CCC(C)NC(=O)Cc2ccco2)C)on1 C12(CNC(=O)Cc3csnn3)CCC1CCN2C(c1cccnn1)=O N1(C(c2cc(C)on2)=O)C2CCC1CC(F)(CNC(=O)C=CC=C(Cl)Cl)C2 CCCC(CC(C)C)C(=O)NCCC(C)(C)NC(C1COC2(CCC2)C1)=O CC(C)(C)CC(O)C(=O)N1CC(C2CC2)(C(N2CCS(=N)(=O)CC2)=O)C1 CC1CN(C(=O)CC2CC3(C2)CN(C(=O)CCCCN=[N+]=[N-])C3)Cc2c[nH]nc21 c1(CC(=O)NC2C(C)N(C(C3CCOCC3)=O)CC2)cc2ccccc2cc1O c1(C(N2C3CC(NC(C(C(C)C)OC)=O)C3CC2)=O)ccc(Cl)c(Cl)c1O N1(C(c2cc(C)c(=O)n(C)c2)=O)CCC2(CC1)CN(C(C1CC1C)=O)CC(C)O2 Cc1n[nH]c(C)c1CCNC(C1CSCN1C(=O)C(C)(C)n1cccn1)=O CCS(=O)(=O)CCNC(=O)C=CC(C)(C)NC(=O)CNC(=O)CC(C)(C)C N1(C(=O)CSc2n[nH]c(O)n2)CCCN(C(c2cccc(F)c2F)=O)CC1 N1(C(C2N(C)CCOC2)=O)CC2CC(Nc3ccncn3)CC1C2 N1(C(CCSCCC)=O)CCC(C)(CNC(=O)C(C2CCC2)OCC)C1 C1(CNC(C(CC#C)C2CC2)=O)CC(C(=O)NOCCC(=C)C)=NO1 N1(C(C(CC)=CC)=O)CC(C)CN(C(=O)C(C)(C)N(C)C)CC1C N1(C(C(=CC2CCCC2)C)=O)CCN(C(C2CCS(=O)(=O)N2)=O)C(C(C)C)C1 C1(NC(Cn2c(C)cc(C(F)F)n2)=O)CC2CC1N(C(C1C(C)C1C)=O)C2 C1(C(N2CCN(C(c3n(C)cc(Cl)c3)=O)C3(C2)CC3)=O)COc2ccccc2O1 C1(C(=O)NC2CC(COC)C2)(COC)CCCN1C(=O)CN(CC(C)(C)C)C N1(C(C(C)(O)C2CC2)=O)Cc2ccc(CNC(c3ccnn3C(F)F)=O)cc2C1 C(=O)(C(CO)NC(N)=O)N1CC(C(C)NC(=O)Cc2ccon2)C1 c1(CC(N2CC(C)(NC(C(C)NC(C)(C)C)=O)C2)=O)cncc2ccccc12 CC12CCCC1NC(=O)CN(c1ncnc3c1ncn3CCC(O)C1CCC1)C2 O=S(=O)(c1cncc(Br)c1Cl)N1CC(c2ncc(C(F)(F)F)cc2F)C1 CCCC(C(=O)N1CC(NC(=O)C(OC)OC)C(CC)C1)NC(=O)OC Cc1ccc2cc(C(=O)NC3(CNC(C4(C#N)CC4C(F)(F)F)=O)CC3)ccc2c1 C(=O)(C1=CCCC1(C)C)NCCN(CCCN(C)C)C(c1cnc(C(F)(F)F)s1)=O C(=O)(CCCC(=O)NCc1ncoc1C1CCN1C(=O)NC1CCCCC1)OC O=C1CSc2ccc(C(N3CCN(C(=O)C=CC4CC4)C4CCC34)=O)cc2N1 C(CC(C(C)(C)C)NC(=O)Cc1cncs1)N(C(=O)COC1(C)CCC1)C c1(CC)ccc(N)c(C(N2CCC(CNC(=O)C(F)(F)CO)C2)=O)c1 c1(C(N2CCN(C(c3cc(C)ncn3)=O)C(CO)C2)=O)c([N+](=O)[O-])c(C)nn1C Cc1cc(C(=O)NC2(CO)CCCN(C(c3snnc3C)=O)C2)cc(Cl)c1 c1(C(=O)NC2CCN(C(C3(N(C)C)CC3)=O)C2)cc(O)ncc1Br c1(C(=O)NCC2(Nc3cc(CC4CC4)nc(Cl)n3)CCC2)cccc2cnsc12 CC(C(O)C(F)F)NC(c1cnn(CCNC(=O)CCc2cnn[nH]2)c1)=O N1(C(c2c(CC)nc[nH]2)=O)CCCN(C(=O)CCC(C)(C)C)C(C)C1 Cc1ncc(Cl)c(C(N2CC(NC(c3cc[nH]c3)=O)CCC2C)=O)n1 C=CC(CC)CC(=O)NC(C(=O)Nc1cnc(CO)nc1C)C1CC1 c1(OCC)ccc(C(C)NC(=O)NCCNS(N)(=O)=O)cc1.C1CCC1 C(CC(O)C(=O)N1CC(N(C)C(C2(C(F)(F)F)CCCCC2)=O)C1)OCC c1(C(N2CCC(C)(NC(c3ncn(C)c3)=O)C2)=O)cc2ccc(C(N)=O)cc2[nH]1 n1(CC)ncc2cc(C(=O)NCCC(C)CCNC(=O)Cc3ccco3)cnc12 Cn1ncc(CNC(c2nc(Cl)cs2)=O)c1C(=O)NC1CC(CC(C)(C)C)C1 c1(C(=O)NCC2CC(NC(=O)COc3ccc(F)cc3)C2)ccccc1[N+](=O)[O-] c1(C(N2CC(C(N)=O)C(NC(=O)C(F)C3CCC3)CC2)=O)ccn2c1CSCC2 C1(N(CCOC)C(C)=O)CCN(C(=O)C(N)=O)CC1.C(C)(C)(C)ON c1(C(N2CCCC(CNC(C(F)OC)=O)C2)=O)ccc(O)c(N)c1 N1(C(CCNC(c2c(Cl)cn(C)n2)=O)=O)CCC(CO)C(C)(C)C1 S(=O)(=O)(CC(COC)OC)CNC(NC1CCCC(CC)C1)=NC N1(C(C(C)C)=O)CCC(c2nc(C3CN(C)CCO3)nn2C2CCSC2)CC1 n1(CC(=O)NC(CCNC(C=C(CC)C)=O)C)sc2ccccc2c1=O C1(C(=O)NC(CN(C)C)C(N2CCC(O)(CN(C)C)C2)=O)Cc2nccn2C1 Cn1ccn2ncc(C(N3CC4(CC(NC(c5ncc(Cl)s5)=O)CO4)C3)=O)c12 C1(NC(c2cccc(OC)n2)=O)CN(C(=O)C(C(C)C)C(C)C)CC2CCCC12 C1(NC(=O)OC(C)(C)C)CC2CC1CC2(C(F)(F)F)NC1CCCC(C(N)=O)C1 c1(COC)cc(C(C(=O)NC2CCCOC2)N(CC(N2CCOCC2)C)C)on1 N1(C(=O)Cc2ccccc2C(F)(F)F)CC2CC1CN2Cc1ccncc1Br C1(C)(NC(C(CCSC)NC(c2nc(Cl)cs2)=O)=O)CC(C)(C)OC1=O C12(C(N3CCCC3Cc3cn(Cc4ncon4)nn3)=O)CCC(CC1)C2 C(=O)(CC1=CCCCC1)NC(C(CO)NC(c1c(C)nn(C)c1Cl)=O)C c1(CNC(C2C(C(=O)Nc3cccc(CCC)n3)C2)=O)cccc(C)c1F c1(OCC(c2n(C)ncc2)(c2nnnn2C)NC2CCCCO2)cccc(Cl)c1 C(C(C(F)(F)F)n1cncn1)NC(c1n(CC(=C)C)nnn1)c1cc(C)ns1 Cc1cc(C(=O)NCC2(O)CC(NC(=O)C(F)CC3CCCC3)C2)no1 c1(C(=O)NC2CC(C)(NC(C(CC)CCOC)=O)C2)[nH]nc2ncccc12 c1(C(=O)NC(C)CNC(C2(C(F)(F)F)CC=CCO2)=O)cnc2ccccc2c1 c1(C(=O)NC2C(C)CN(C(=O)Cn3cnnn3)CC2C)nccc2ncncc12 C(=O)(C1CC(=O)Nc2ncccc21)NC1CC(CNC(C(CC(C)C)F)=O)C1 n1(CCC(N2CCC3C(NC(CC(C)C)=O)C32)=O)c(=O)oc2cc(Cl)ccc12 C(=O)(CCCC(F)(F)F)N1C(C)CC(CNC(c2ccnnc2)=O)C1 C(=O)(CCCN=[N+]=[N-])N1CC(CC(=O)NCC(C)SC)OCC1 C(=O)(CS(=O)(=O)CC)NC(CCCC)CNC(C1C2CCC1CC2)=O O=C1NC2CN(C(C3CC(O)CN3C(C3CCCOCC3)=O)=O)CC2O1 C12(CNC(c3cnc(OC)nc3)=O)CCC(CC1)N2C(C1COC(=O)N1)=O N1(C(c2c(C)c[nH]c2)=O)CCC2(C=C(C(=O)NCC(C)(O)CC(C)C)C2)C1 Cc1cccc2c1CC(C(=O)NC1CCC(NC(C3CC3C)=O)CC1)O2 O=S1(=O)CC2CN(Cc3ccc(I)c(F)c3)CC2C1 c1(C(=O)NCC=C(C(=O)N(C(CC)C2CC2)C)C)nccnc1N CC(CC1=CCCCC1)NC(c1cn2c(n1)CCCC2)C c12ccc(cc1)NC2.c1(OC)ccsc1OC.c12nnnn1CC2COC N1(CCN(C(CC2(NC(C3C(C)(CC)C3)=O)CC2)=O)C)CCOCC1 c1(C(=O)NCC(CC)NC(=O)CC2(c3ccccc3)CC2)cnccc1N(C)C N1(C(C2C(C)CC(C)O2)=O)CC=C(CNC(=O)C(N)=O)CC1 c1(C(=O)NC2C3CCN(C(C4CC5(CC5)CO4)=O)C23)cc(Cl)c(Cl)c(Cl)c1 CCC(C(=O)NCC(=O)N(C)CC1CCN(Cc2ccccc2)CC1)C(C)O C(CCCC(=O)NC1(C2CCCN2C(=O)CCC2CCCO2)CC1)N(C)C N1(C(C=CCCC)=O)CC2(C1)CN(C(c1ccccc1C(C)=O)=O)C2 CC1(C(N2CCCC2C(=O)NCC2=CCCOC2)=O)CCNC1=O N1(C(C)=O)CCCC(C(N2CCC(N(C)C(C3CC4(C3)CC4F)=O)CC2)=O)C1 c1(C(N2CC(CC)(CNC(C3CN(CC)CCO3)=O)C2)=O)cc2n(n1)CCC2 c1(NC(c2c(C(=O)OCC)ccs2)=O)ccc2c(c1)CCN(C(C)C(=O)OC)C2 c12cccc(c1)NC(C(=O)OC)N(C)C2=O.C1(C2CC2)(CC(=O)NC2CC2)CC1 N1(C(CCCSC)=O)CC2C3CCC(C2C1)N(C(c1cc(C)n(C)c1)=O)C3 c1(C(=O)NCC2CC(NC(CC3C(C)CCC3)=O)C2)cc(Br)c(C(F)F)s1 c1(N2CCC=C(C(=O)CC)C2)cc(C(=O)OC)nc2ncnn12 c1(C(=O)NCC2N(C(Cc3c(C)ocn3)=O)CC=C2)ccnc(-n2cccn2)c1 O=C1CN(C(c2nccs2)=O)C(C(N2CCn3nccc32)=O)CN1 c1(OCC(=O)NCCN(C(=O)CCNCC2CCC2)C)c(F)c(F)cc(F)c1F c1(C(N2CCC(NC(=O)C#CC3CCOC3)C(F)C2)=O)cc2ccc(F)cc2[nH]1 N1(C(c2ccn(C)n2)=O)CCCC(C(C)(C)C(=O)NCc2ccncc2F)CC1 N1(C(C2C(C)(C)C2CNC(=O)C=Cc2nccs2)=O)CCCC(F)CC1 C=C(C)C1OCCCC1C(=O)NCC1=CCCN(C(=O)Cc2cncs2)C1 CC(C)C(F)C(=O)NCC#CCNC(=O)CN(C)Cc1ccc(Cl)s1 c1(C(N(CCNC(C2(CC)CN(C(C)=O)C2)=O)CC)=O)nn(C(C)(C)C)cc1Cl C=CCC(CC(F)F)NC(=O)CCC1CCCN(C(=O)Cn2cc(CO)nn2)C1 CC1CN(C(=O)CC2OCCO2)CCC1CNC(C1CC(O)C1)=O C1(NC(CSC)=O)CC(C)CN(C(C23CC(F)(C2)C3)=O)C1 c1(C2(C(=O)NCC(C)(C3CC3)NC(CC=C)=O)CCC2)cc(F)cc(C#N)c1 c1(C(=O)NC2CCCCN(Cc3ncc(C)c(Br)c3)C2)cc2ncccn2n1 N1(C(=O)NC(c2cnn(C)c2)C)CC(NC(=O)OC(C)(C)C)C2(CCC2)C1 C1(C(=O)Nc2ccc(C)nc2I)CC12CCN(C(c1c(Cl)cncc1Cl)=O)CC2 C(=O)(C(C)CC(F)(F)F)N1C2CC(NC(c3c(C)nc(Br)s3)=O)C2CC1 c1(CC(N2C(CC(=O)N(c3ccccc3)CC)CCC2)=O)ccc(F)c(Cl)c1F N1(C(C2(SCC)CC2)=O)CCC(C)C(NC(=O)C(C)=O)C1 c1(CN2C(CNC(CC(C)C)=O)CCC2)cccc2c1oc1ccccc21 c1(C(=O)NCC(CO)NC(=O)C2=CCOCC2)nnc(O)c2ccccc12 C(=O)(CC(C)N(C)C(c1c[nH]nc1CNC(c1cc(C)no1)=O)=O)OC c1(C(C(=O)NC2CC(NC(C=C(CC)CC)=O)C2)=O)ccc(O)cc1 CCC(CC)C(F)C(=O)N(CC(O)CNC(=O)CC(CC)C1CCC1)C c1(C(=O)N(CCOC)C)ccc2nccn2n1.O=C1CCN1CC1CC1.C1CC1 C1(COC)(NC(=O)Cn2cc(C)cn2)CN(C(C2CCN(C(C)=O)C2)=O)C1 N1(C(c2c(C)nc(C)s2)=O)CCC(C2CC2)(NC(c2cc(Cl)ccc2F)=O)C1 c1(C(=O)NC(C)(C)C(O)C(F)(F)F)cccc(S(=N)(=O)C(F)F)c1 c1(OC)cccc(N2CCC(C(=O)N(C(C)C(=O)O)Cc3ccccc3)C2)c1 c1(-c2ccc(C)cc2O)cnc2ncc(C(N3CCOC4CC34)=O)n2c1 Cc1c(O)ccc(C(=O)NC(CNC(=O)C(CC2CC2)CC2CC2)CO)c1C Nc1c(Cl)cc(NC(C23CC2CN(C(c2cc(C(F)(F)F)n[nH]2)=O)C3)=O)cc1Cl CON(C(=O)C=CCNC(c1cc2ccccc2o1)=O)C(C)C c1(C(=O)NC2(C)CCN(C(C3CCC3C(F)(F)F)=O)C2)cccc2c[nH]nc12 N1(c2c(C)cncn2)CCC(O)(CC(=O)N(C)CCN(C)C)CC1 N1(C(C(C)OCCC(C)C)=O)CC=CC1C(=O)NCC(O)C1(Cl)CC1 C1(C)(N2C(=O)NC(C)(CC(C)C)C2=O)CCN(S(N)(=O)=O)CC1 c1(C(=O)NCCCCC2(NC(c3n(CC)ccc3)=O)CC2)cnc(N(C)C)cn1 C1(NC(c2cc(C)oc2)=O)C(C)CCN(C(C2CCCSS2)=O)C1C CC1(C(=O)NC2CCN(CCNC(C3CCCCNC3=O)=O)CC2)CCC2CC2C1 C(CC1=CCN(C(=O)CSCc2cscn2)CC1)NC(Cc1c(C)cco1)=O c1(CNC(C(CC)C(C)O)=O)ccc2c(c1)CCCC2NC(c1cc(C)[nH]n1)=O N1(C(CC=CCC)=O)CCCN(C(=O)C(=O)Nc2ccccc2)C(CO)C1 C(C(=O)NC(CNC(=O)C(C(C)C)C1CCC1)C(C)C)(C(C)C)SCC c1(C(=O)NCC(CCCC)NC(=O)CCOC(C)C)[nH]cc2c1CCC2 N1(C(C(=O)Nc2c(C)cc(Br)nc2)=O)CC2CC1CS(=O)(=O)C2.C1(C)(C)C(=O)O1 CCC(C(=O)N1CCC1CNC(c1cc(S(C)(=O)=O)oc1C)=O)C(C)(C)CC c1(NC(C(C)(F)F)=O)cccc(NC(=O)CCc2cncnc2O)c1 C(C(CC(C)C)C(=O)NC1(CO)CC(OC)C1)NC(C(C=C)C)=O Cc1ccn(C)c1C(N1CC=CC1CNC(C1(c2ccc(F)cc2)CCC1)=O)=O C=CCC(CC(F)F)C(=O)NC1C=CCN(C(C2OCCOC2C)=O)C1 CC(CNC(=O)C=Cc1ccoc1)CC(=O)NCC(C)(C)F C(=O)(C(CN=[N+]=[N-])NC(=O)Cn1cncn1)N(CC(N1CCCC1)C)C C(=O)(CC(F)(F)C(F)F)N1C(CCC)CN(C(c2cn(C(C)C)cn2)=O)CC1 S(=O)(=O)(c1cccc(=NCCCCCCF)[nH]1)NC(C)C(C)S(C)(=O)=O C#CC1CN(c2nc(-c3ccccc3)nc(C)c2I)CCN1C C(=O)(C1OCCn2ccnc21)NC12CN(C(C3CCCC(=O)N3)=O)C(CC1)CC2 c1(C(=O)NC(CCN(C(COCCCCC)=O)C)C)ccc(OC(F)F)cn1 CC1(C)CC(CC(=O)NOCc2ccccn2)N(C(=O)CC2CC(=O)C2)C1 c1(OCC(=O)NC2CC(CNC(C3(C)CC3(Cl)Cl)=O)C2)cc(Cl)cc(Cl)c1 c1(OC(COC)C(=O)N2CCC(c3ccc(Cl)cc3)C2)cc(F)cc(F)c1 N1(C(c2c(C(=O)O)c(Br)ccc2)=O)CCC2(CC1)CC(c1ccc(Cl)cc1)C2 c1(C(=O)NCC(CC=C)NC(=O)C=CC=CC)c(C)cc(C)cc1N C1(OC)(CNC(=O)COC2CC2)CCN(C(c2cccc(C(C)(C)C)c2)=O)CC1 Cc1cnc(C(=O)NC(CC2CCC2)C(=O)NC(c2ccccc2O)C)cn1 N1(C(c2c(Cl)ccc(C#N)c2)=O)CCC2CN(C(=O)CSC(F)(F)F)CC2C1 c1(C(n2cc(CONC(C3CCNCC3)=O)nn2)CC)ccc(F)cc1 Cc1ccc(O)nc1CNC(=O)CCCC(C)NC(=O)C(O)C1CCCC1 C(=O)(C(CC(F)F)NC(c1ccc(C2CC2)[nH]1)=O)N(C(C)CN(C)C)C C(=O)(CC(C)(C)CC(C)OC(C1(c2nc(C)cc(C)n2)CC1)=O)OC Cc1nn(C)c(C)c1CCC(=O)NC1CC1CNC(=O)CC(C)(C)CN(C)C N1(C(C(C)=CC2CC2)=O)CCCC(O)(CNC(=O)Cn2cnc(C(N)=O)n2)C1 C(CCCCCNC(=O)Cn1c(C)csc1=O)NC(CSc1nc(C)[nH]n1)=O c1(CC(=O)NC2C(C)N(C(c3cnn[nH]3)=O)CC2)ccc(Br)c(F)c1 c1(C(=O)NCCCN(C(=O)C(F)C2CCOC2)C2CCCC2)cc(C2CC2)on1 c1(C(=O)NC(CC(=O)NC2CCC=CCC2)C(F)F)ccc2occc2c1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CCCCC(CNC(=O)CN(C)C(=O)C2CC2)C1 C1(NC(Cc2c(CC)n[nH]c2CC)=O)CCN(C(=O)CSCCC#N)C12CCC2 N1(C(C2CCN(CCC)CC2)=O)CCCC2CN(C(=O)CCC(C)C)CC12 C(C(C)C(=O)N(CCO)OC)N(C(C(CC)(CC)CO)=O)C C(=O)(CC(F)(F)CC(=O)NC1CN(C(C2CCCOCC2)=O)CC1C)OC CC1=C(C(=O)NC2CCC(CNC(c3cc(O)ccc3O)=O)C2)SCCO1 N1(C(C(C)OC)=O)C2CCCC1CN(C(C1CCN(c3cnccn3)CC1)=O)C2 C(=O)(CC(C)C(C)C(C)C)N1CC(C2(NC(c3onc(C)c3C)=O)CC2)C1 C1(C(N(C(CNC(Cc2cccc(SC)c2)=O)C)C)=O)CCOC2(CCCC2)C1 CCCC(C)CC(=O)NC1(CC(=O)Nc2cc(CO)cc(F)c2)CC1 N1(C(c2cnc(OC)c(C)c2)=O)CCCCCC(NC(c2scc(C)c2C)=O)C1 c1(OC)ccc2[nH]c(C)c(C(=O)NC(CNC(=O)C=C(C)C(C)C)CO)c2c1 C1(C(CNC(CN(C(C)C)C)=O)F)CCN(C(=O)CC(F)(F)F)CC1 c1(N(c2ccc(F)cc2)C(c2cccc(Cl)c2C(F)(F)F)=O)cncc([N+](=O)[O-])c1 c12ccc(nc1)S(=O)(=O)NCC(OC)CNC2=O.C1(COC)(CO)CCCC1 N1(C(c2ncc(NC)nc2)=O)CCC2(CC(NC(=O)C(C3CCOC3)OC)C2)C1 C1(C(N(C(C)C(=O)NCCc2noc(CC)n2)CCC)=O)CC2(CCCO2)C1 C1(CC=C)(NC(c2cc(C)c(Br)s2)=O)CCN(C(=O)C=CC)C1 C1(CCNC)CN(C(=O)OC2(C(=O)NC(C)(C)C)CCC2)CC1C C(CCC(C)C)(C(=O)N1CCCN(C)CC1C)NC(CC1(CC)CCC1)=O C(=O)(C(C)CC(F)(F)F)N1C(C(=O)NC2CN(C(C)C)C2)CC(=O)C1 N1(C(C2(OCC)CCCC2)=O)CCC(O)(C(C)CNC(=O)Nc2scnc2C)C1 Cc1sc(Br)nc1C(=O)NC1CCCC1CNC(=O)C(C)CC1CC1 c1(C(C(=O)NC(CC#C)COC)C)ccc(C(F)F)cc1 C(CCCC(=O)N(C(C)CCNC(=O)CC1(CO)CCOCC1)C)OCC Cc1ccc2c(C(=O)NCC3C(C)CCN3C(=O)C#CC3CC3)cnn2c1C N1(C(CCC(=O)OC)=O)CC2CC(NC(c3c[nH]cc(C)c3=O)=O)CC1C2 CC(C)(C)C(CO)C(=O)NCC1(C)CCN(C(C2CC(OC(F)F)C2)=O)C1 C1(NC(C)=O)C2CC(NC(=O)C(C3(O)CCCC3)F)CC12 C(=O)(C(F)(F)F)NCCNC(N1CCC(Cc2ncccn2)C1)=O C(CC(C)CC)(C(=O)NC1CN(C)CC1C)NC(C(CC=C)CC)=O N1(C(Cc2c(C)cccn2)=O)CC(CNC(=O)C(F)(F)C2CCCC2)C(C)(C)C1 c1(C(N2C3C(NC(=O)CC4CC=CCC4)CC(C3)C2)=O)c[nH]c2ccc(Cl)cc12 c1(C(=O)NC2CC(NC(C=C(C)c3cnn(C)c3)=O)C2)cnn2c1NCC(C)C2 CC12CCC1CN(C(C1CNCC13CCC3)=O)C2 N=c1[nH]c(Cl)c(Cl)c(=NC2CCCC(CO)C2)[nH]1 c1(C(=O)NCCCN(C(C2C(C)(CC)C2)=O)C)cc(C2CCCCC2)on1 CON=C(C(=O)N1CC(=C(F)CNC(=O)CCCN=[N+]=[N-])C1)c1ccco1 N1(C(C=CSC)=O)CC2CC(NC(=O)Cc3ccc(F)cc3)C1C2 c1(C(=O)NCC(CNC(CCC(=C)C)=O)C)cccc(Cl)c1C N1(C(=O)CC2(O)CCCOC2)CCCC2(CCN(c3cc(Cl)ncn3)CC2)C1 N(C(=NCC1CCN1C)N1CC(C)C(C)C1)Cc1cc(C)on1 c1(C(c2n(CC)nnn2)NC2CCC(=O)NC2)cccc(-c2ccccn2)n1 CCCCCCCCc1ccsc1C(=O)NCC(CC)NC(c1cc(Cl)c[nH]1)=O CC1=NS(=O)(=O)N(C)C=C1C(=O)N(CC(C)NC(=O)C(C)Cn1cccn1)C N1(C(C(C)C(C)(C)C)=O)CC(NC(c2cnn(C)n2)=O)CC12CCC2 CC1(C)CN(C(C23CCCC2C3(F)F)=O)CC(C)(C)C1NC(=O)Cc1ccco1 c1(CCCC)ccc(-c2cccnc2C(=O)N(C)C(C2CCC(=O)N2C)=O)cc1 N1(C(c2c(C)con2)=O)CC=CC(NC(=O)C(N2CCN(C)CC2)C)C1 c1(C(N2CCC(NC(C(C#C)(C)C)=O)C(F)C2)=O)ccc2n[nH]cc2c1F c1(C(=O)NCC2CN(C(=O)CC3C=CS(=O)(=O)C3)CC2O)ncc(Cl)cc1F C12(NC(CC(C=C)(C)C)=O)CCCC1N(C(C1CCCCN(C)C1=O)=O)CCC2 CCC(C)CC(=O)C(=O)N1CC2(C(=O)NCC(O)C(F)F)CCC1CC2 N1(C(=O)Nc2c(C)onc2OC(F)F)CCNC(C)C1C C1(C)C(=O)NC12CC2.c1(CN(C(C2(COCC)CC2)=O)C)cocn1 c1(CC)c(C(N2CCC2C(=O)NCc2ccccc2OCCO)=O)cnn1CC C1(O)(C(C)NC(C2C(CC)C2)=O)CCN(C(C2CCCOC2)=O)CC1 N1(C(C(CC)CC)=O)CCCC(O)(CN(C)C(c2cc(O)ncn2)=O)C1 N1(C(C2CCN(C)O2)=O)CCC(COC(=O)Nc2ccnnc2O)CC1 C#Cc1cc(C(=O)NC2COCC2NC(=O)CCc2cnc(C)s2)ccc1Cl N1(CCN(CCC)CCNC(c2cnsc2)=O)C(=O)NC(CCSC)(CC)C1=O C1(F)(CNC(c2cnc(C(C)OCC)s2)=O)COCCN(C(=O)CSCC)C1 CC1(C)OC2CN(C(c3cccc(Cl)c3)C(=O)NCC3CCCO3)CC2O1 c1(OC)ccnc(NC(C2CCCC2NC(c2cccc(F)n2)=O)=O)c1I CCC(CNC(C1CN(C)CCO1)=O)(CC)C(=O)N(C)Cc1ccccc1C C1(C(=O)O)CN(Cc2nc(C3CC3)cs2)CC1C1CCOCC1 C(=O)(C#CC1CCC(=O)CC1)NC(C(C)C)C c1(C(N2CC(C(C(=O)NC3(N(C)C)CCC3)OC)C2)=O)ccc(COC)c(F)c1 c1(C(=O)NC2CC(C)(COC)N(C(=O)C=CCO)C2)cc(C)c(C)nc1C C(=O)(C(C)N(C(=O)CC1CC(NC(=O)CCC2CC2(F)F)C1)C)OCC S(=O)(=O)(c1cc(C)cnc1NCCC(C)CC(C)(C)C)NCc1cc(SC)on1 N1(C(CCCC#C)=O)CCCC(CC=C)(C(N2CCOCC2CCC)=O)C1 C1(NC(Cc2c(CC)cccc2)=O)CCc2nc(NC(=O)C(O)C(C)C)sc2C1 C(=O)(C(C)(C)CC#N)NCC1CC(NC(c2c(COC)cc[nH]2)=O)C(O)C1 c1(C(=O)NC(CC)CN(C(=O)C(COC)OC)CC)[nH]nc([N+](=O)[O-])c1Cl C1(N(C(c2cc(SC)oc2C)=O)C)CCCN(C(=O)CC2(O)CCCOC2)CC1 c1(C(=O)NCCNC(c2ccc(C3C(C)C3)o2)=O)ccc(NC(=O)C2CC2)cc1 CCC(CC(F)F)C(=O)N1CCCCC1CCNC(C1CC2CCC(C1)N2C)=O C(CC(=O)NCCCN(C)C(c1cc(Br)cnc1S)=O)(C(C)C)OCC C(=O)(C1CCCn2cnnc21)N1CCCN(C(=O)CC2CS(=O)(=O)C2)CC1CO C(CCCC(CO)NC(C1(CO)CCCO1)=O)NC(c1n(C)ncc1)=O c1(NC(C2CC2F)=O)cccc2c(-c3ccc(NCCO)cc3)cccc12 n1(CC)nc(C(=O)N(C(CNC(=O)CCF)C2CC2)C)c(=O)c2ccccc12 C=C(C)CC(C)C(=O)NCCOC1CN(C(=O)C(c2ccc(C)s2)C)C1 c1(C(N2CC(CC(C)NC(CCCCCC#C)=O)C2)=O)cc2cc(C)ccc2[nH]1 c1(SC)ccc(C(N2CC(NC(=O)CC3(CO)CC3)C3(CC3)C2)=O)c(Cl)c1 c1(C(=O)NC2C(CNC(=O)CN3CCC3c3cccnc3)CC2)ccc(F)cn1 CCC(CCC(=O)NC(C)C1=CCCC1)NC(=O)CC(C)(C)COC c1(C(C(=O)OCCSC(c2ccccc2)C(=O)OC(C)(C)C)F)cccc(Br)c1F N1(CCCOC(C2CC2C(=O)Nc2ccccc2)=O)CCOCC1 CC1CCCC(CCNCC(c2ccc(O)cc2)O)C1 N1(C(C(C)C2CCC2)=O)CCC(N(CCO)C(c2cc(Br)n(C)n2)=O)CC1 c1(C(=O)NC2CCC(CCNC(C(N)=O)=O)C2)cccc(CCO)c1 N1(C(c2c(NC)scn2)=O)CCC(NC(C2CCC(C)(C)CC2)=O)C12CC2 c1(C(N2CC(C)C(NC(C3(C)CCCCO3)=O)CC2)=O)cccc2c1OCC2 C1(NC(=O)CN2CCCCC2)CCC2CN(c3cc(C(F)F)ncn3)CC2C1 Cc1nc(C2CC2)oc1C(=O)NC1CN(C(C23CCC(C(=O)O)(C2)C3)=O)CC1O CN=c1[nH]c(=NCC2CC(F)(F)C2)[nH]c(=NCCc2cn[nH]c2)[nH]1 n1(CCN(C(C23CSC(C2)C3)=O)C2CC2)cc(C2CC23CC3)nn1 C(CCCO)(CCSC)NC(=O)NCCC(OC)OC CC#CCC(C(=O)NOC(C)C(=O)OC)NC(=O)C(CC)CCCCC N1(c2cc(N(CCOC)Cc3ccco3)ncn2)CC(C)SC(C)C1 c1(CC)nc(C)ncc1C(=O)NCC1C(C)CCCN1C(C1CCCCN1C)=O C1(C(N2C(CNC(c3nc(-c4cn(C)nc4)sc3)=O)CCC2)=O)CCCC1(C)C C(CCC(O)C(=O)N(CC(N)=O)C)NC(c1c(CC)cns1)=O C=CC(C)(CC)C(=O)N(CC(C)O)CCNC(c1cc(N)ccc1O)=O N#Cc1cc(CNC(C2COCCN(C(C3CC34CCNC4)=O)C2)=O)cc(Br)c1 Cc1cc(F)ccc1C(N1CCC(O)(CNC(c2ncoc2C)=O)C1)=O N1(C(C(C(C)C)NC(N)=O)=O)CCC(NC(=O)C=Cc2ccsc2)C2(CCC2)C1 C1(CC(=O)NC(c2ccncn2)C)CCN(C(C2CC(F)C2)=O)C1 c1(OCC)cc(NC(C2CCCCN2C(C2CC(=O)NC(=O)C2)=O)=O)ccc1F N1(C(c2cc(C#N)sc2)=O)C2CCC1CC(NC(C1CC=CCC1)=O)C2 c1(C(C)C(N2CC(O)(CNC(C3CC3c3ccco3)=O)C2)=O)cc(F)cc(F)c1 C1(CC=C)(C(N2CCC(C)(CNC(c3ccc(CO)nc3)=O)C2)=O)CCOCC1 CC(C)C(N=[N+]=[N-])C(=O)N(CC(N1CCC(N2CCCC2)C1)=O)C N1(C(C2C(OCC)C2)=O)CCOCC(CNC(C2CCS(=O)CC2)=O)C1 c1(CC)n[nH]c(CC)c1CC(=O)NCC1CC1NC(=O)C=Cc1ccc(Cl)s1 c1(C(=O)NC2CC(CNC(CCSCCC)=O)C23CCC3)ccn2ccnc2c1 CCC(F)(F)C(=O)NC(C)C(C)NC(=O)CCc1ncccn1 C1(NC(c2cc(N)cc(O)c2)=O)CC(NC(=O)Cc2cnsc2)C12CCOCC2 c1(NC)ccc(F)cc1NC(=O)CC1(OC)CCC1.C12CC1C(=O)N2 N1(C(C2(F)C(C)C2)=O)CCC(N(C(=O)CNC(c2ccccn2)=O)C)C1 C1(C(=O)OC)CC(C)(NC(=O)CC2(NC(C34COCC3C4)=O)CC2)C1 N1(C(CCSCC)=O)CCC(CN(C)C(C2(C(=O)NCC)CCC2)=O)C1 CC(N=c1[nH]nc(O)s1)C1CCN(C(c2cc(C3CC3)nn2C)=O)CC1 C(C)(CCCCN=c1[nH]cnc2cc(C(=O)OC)ccc12)NC(CN(CC)CC)=O N1(C(c2cnn(C)c2N)=O)CC(C)(C)CCC1CNC(C1CC2CCCCC12)=O CC1(C)COC1C(=O)NCC(CNC(c1c[nH]nc1C(F)(F)F)=O)CO c1(C(=O)NCC(C)(C2CCC2)NC(C(F)=CCC)=O)nsnc1O C(=O)(C(O)COCOC)N1CC(C(C(=O)NCC(C)(O)c2ccco2)O)C1 C(=O)(C(C)CCCC)N(CC(=O)NCCNC(=O)NC)CC#C C1(Nc2c(C)ccc(Cl)c2)CC2CN(C(=O)OC(C)(C)C)CC2C1 Cc1nonc1CC(=O)NC(CN(C(=O)C(O)CN(C)C)C)Cc1ccccc1 C12(C(=O)NC3C(OC)CC3O)CC(CN(C(c3cn(C4CC4)nn3)=O)C1)C2 n1(C(CC)C)ccc(=NC(=O)C2CC(N(C(=O)CC(O)C3CCCC3)CC)C2)[nH]1 C(=O)(C(C)(C)C(C)(F)F)NCC1C(C(N(C2CCOC2=O)C)=O)OCC1 c1(-c2c(C)ccc(C#N)c2)ccc2c(c1)C1(CCN(C(=O)C(C)S)C1)C(=O)N2 c1(C(=O)NC(CC2CN(C(C(CC)F)=O)C2)C)cncc(NS(C)(=O)=O)c1 CC1CC(NC(C2(c3ccc(F)cc3)CC2)=O)CCN1C(=O)C(C)CC1CCC1 c1(C(N2CC3C(NC(c4c[nH]c(=NC)s4)=O)(C3)C2)=O)n[nH]c2c1CC(C)CC2 N1(C(C2N(C(C(CC)n3ccnc3)=O)CCC2)=O)CCC(C(=O)OC)CC1 c1(CC)ccc(Cl)cc1C(=O)NC1(C(=O)NC(C(=O)OC)C(C)O)CSC1 N1(C(=O)NCc2ccc(CC)c(F)c2)Cc2ccccc2CCC1C Cc1cccc(C)c1NC(=O)C(N1CCCC(C(C)(F)F)C1)c1cncs1 c1(C(=O)NC2C3CC2CN(C(C2C4CCCC24)=O)C3)ccc2cc(Cl)ccc2c1 C12(CCNCC1)C(=O)N1CCCCC1C2.C1(C)CCC1.CCCO N1(C(C2CC3C=CC2C3)=O)CCC2(CC1)CCN(C(C1CC3(CCO1)CC3)=O)C2 C1(C2CN(C(c3ccc(Br)cc3)=O)C2)(NC(CCn2ncc(C)c2)=O)CC1 CCCC(CCC)CC(=O)N1CC(O)CC1CNC(=O)CC1(CC)CCOCC1 c1(CC(=O)NC2(C(N3CCCC3C)=O)C(C)C2)cc(Br)ccc1O C1(C(C)C)CN(C(c2cn(CCCF)nn2)=O)CCN1C(=O)COC1CC1 C1(C(=O)OC)C=CCCN1C(=O)C(C)CN(C)C(c1cnn(C(C)C)c1)=O C1(NC(C=CCCC)=O)CC(C(=O)NC(c2cscn2)C)C12CCC2 c1(NC(=O)NC(c2cccc(Cl)c2)CC)nc2cc(C#N)ccc2o1 Cc1ccc(NC(=O)COCCN(C)C)c(OCC2CCOC2)c1 C=C1CCN(C(=O)C=C(C)CCC)C(C(=O)NC2COC3(CCC3)C2)C1 Cc1c(Cl)c(C(=O)NCC(=C2CN(C(=O)CC3OCCC3(C)C)C2)F)nn1C C1(C(=O)NCc2c(C)nn[nH]2)CN(C(C2(O)CCCC2)=O)CCN1C CCCCC(CN=c1cc(C)nc(C)[nH]1)NC(=O)C1CNC(=O)c2ccccc21 C1(CC(=O)NCC2(C(C)NC(CSC(C)C)=O)CC2)CCCSC1 c1(OCC)ccc(C)cc1CNC1COCCN1C(=O)Cc1ccc(Br)[nH]1 c1(CNCCN(C(c2c(CC)nn(C)c2)=O)C)c(F)cccc1Cl C1(C(N2CC(COC)(NC(c3sccc3F)=O)C2)=O)CC(C2CC2)=NO1 N1(CC(c2ccc(C)cc2)=O)CCC(O)(C(=O)NC2(C)CCCC2)CC1 n1(CC)cc(Cl)cc1C(=O)NCC1CCN(C(c2n[nH]c(C)c2Br)=O)CC1 c1(C(=O)NC(C2CCCCC2)C(=O)NC(CCCCC)C)c[nH]c(C#N)c1C CCC(C(=O)NCC(C)CN(C)C(c1ccc(C(F)(F)F)o1)=O)C(C)(F)F c1(C(=O)NCC2N(C(CCOCC)=O)CCC(C)C2)cc2c(nc1O)CCSC2 c1(CCC)cc(C(=O)NC2(C)CCN(C(c3coc(N(C)C)n3)=O)C2)n(C)n1 CCCCC(O)CC(=O)NCC1(CCNC(=O)C(CC)c2cccnc2)CC1 c1(OC)cccc([N+](=O)[O-])c1CN1CCNCC1C(=O)Nc1ccnc(C#N)c1 C=CC1(C2(C(=O)NCC3CC3CNC(=O)CCCC(CC)CC)CCC2)CCC1 c1(C(=O)NCC2N(C(C=CCCC)=O)CC(OC)C2)ccc2c(c1)CCCCN2 Cn1ncc2c1CN(C(=O)C(CC1CC1)NC(C1C=CCCC1)=O)C2 C1(NC(C=CC=CC)=O)C(C)CCN(CC(=O)NC2CCCC2)C1C N1(C(c2ccc(C=C)cc2)C(=O)Nc2ccccc2)CC(N(C)C)CC12CCC2 c1(C(=O)NCC(CCNC(c2cnc(C3CC3)o2)=O)O)occ2c1CCOC2 C(=O)(C(C(C)(C)C)NS(C)(=O)=O)NCC1N(C(CC(C)(C)C)=O)CC(F)C1 C1(C(C)C(=O)NC2(C)CC(NC(c3ccc(Br)o3)=O)C2)CCC(C)(C)CC1 N1(C(C2CC2CF)=O)CCOC(CNC(=O)C(F)(F)CC(C)(C)C)C1 C1(NC(c2c(C)sc(O)n2)=O)CCN(c2snc(Cl)c2C#N)CC1C Cc1ccc(C(N2CCC(C)(C(=O)NCCc3nccnc3C)C2)=O)c(F)c1 C1(CC#C)(C(N2CC(CC(C)NC(c3cc(C)c(C)s3)=O)C2)=O)CCCCO1 C12(C(N(C)CC3(C)CCCC3NC(C3COCCO3)=O)=O)CCCN1CCC2 C1(C2(O)CN(C(C3CC34CC4)=O)C2)(CNC(C2CC(C)N(C)CC2)=O)CC1 C1(NC(C=CSC)=O)CN(C(C2CC3CCC(C2)O3)=O)CCC1CO C1(C)(CC)CCCC(NC(=O)CCc2ccc(OC)cc2)C1 c1(C(N2C(C)CC(NC(c3cc(C(CC)C)no3)=O)C2)=O)ccc(C)c(CO)c1 c1(N2CCN(C(C(C(C)C)N(C)C)=O)CC(O)C2)ccc([N+](=O)[O-])c(C(N)=O)c1 c1(C(=O)OCC)c(CC(C)C)csc1NC(C1OCCOC1C)C N1(C(C(C)OCC(C)C)=O)CCOC(C(=O)NC(C)Cc2cn[nH]c2)C1 C1(=O)CC(COC)CN1.c1(CC)nccn1CCN(C(=O)C(CC)OC)CC c1(COC(c2ncc(OC)s2)=O)nc(Cl)ccc1Br N1(C(=O)Nc2sc(CC)c(C)n2)CCc2c(ccnc2Cl)C1 Cc1noc2ncc(C(=O)NCC(CO)NC(=O)CC3(O)CCCOC3)cc12 C(=O)(C(F)CCC(C)(C)C)NC(N(CC(c1cccnc1)N1CCCC1)C)=O N1(C(CC(C)(C)SC)=O)CCC(C2CCOCC2)(CNC(=O)C(C)CC2CC2)C1 C1(NC(C2(COC)CCCCC2)=O)CC(O)CN(C(=O)CCN2CCC(F)C2)C1 C(=O)(C(C1=CCCCC1)N1CC2CCN(C)C2C1)NCCC CC(CC(N)=O)C(=O)NCCOCCN(C(=O)Cc1ccco1)C Cc1ccc(C(=O)NCC(=O)N(C2CC2)Cc2cccnc2F)cc1[N+](=O)[O-] c1(OC)ccc(C(N2CCCC(C(=O)NCCN3CCCC(C)C3)C2)=O)cc1I C1(NC(C2CCCCC(C)(C)C2)=O)CN(c2nc(Cl)ncc2Cl)C2CCCCC12 C1(C)(NC(C2C(OC)C2)=O)CCN(C(c2nn(-c3ccccc3)cc2C)=O)C1 c1(C(=O)NCCCNC(C(C)(C)C2CCOC2)=O)ccc(C2=CCCC2)cc1 N1(C(C(CC)SC)=O)CC2(CC(NC(C3CC3C(F)F)=O)CO2)C1 C1(C(=O)NC(CCSC)C)C(C)OCCN1C(=O)C(CN(C)C)N(C)C Cc1cncc(CCNC(=O)C=CCC(C)(C)NC(c2sccc2C)=O)n1 C1(CC(=O)NCC(COCC)NC(=O)CN2CCS(=O)CC2)CCCC(OC)C1 c1(C(=O)NCC(CNC(c2nc(C(C)OC)sc2)=O)CO)ccnc(CO)c1 C1(NC(=O)CNC(=O)CCF)(CO)CCN(CCOCc2ccco2)CC1 c1(C(=O)Nc2c(C)nc(Cl)cc2)cc2c(-c3ccc4oncc4c3)cncc2s1 N1(C(C2OCC(C)C2)=O)CCCC2(NC(=O)C=Cc3cccc(F)c3)CCCC12 N#CC1CC(C(=O)NCC(C2CCCCC2)NC(C2CCOCC2)=O)C1 C1(CCC(=O)N(C2CCCC2)CCNC(C(C)n2cncn2)=O)CCN(C)CC1 Cc1ccc(C(=O)NCC23CCC(C2)N(C(c2sccc2C(C)C)=O)C3)nc1O Cc1ccc(C=CC(=O)N(C)CC2CCCN2C(c2cc(C(F)F)cs2)=O)s1 c12cc(c(F)cc1[N+](=O)[O-])NCC1CCN2C1.C(=O)(C=CCN(C)C)NC.CO CC(CN(C)C)CCC(=O)NCC1(C(=O)N(C)CCF)CC1 Cc1oc([N+](=O)[O-])cc1C(N1CCCC(CNC(c2coc(C#N)c2)=O)C1)=O CC1(C)CN(C(=O)C(C)(F)c2ccon2)CC1NC(C1CCCS1(=O)=O)=O Cc1cc(C(=O)NCC2CCC(NC(C3CC(C)C3)=O)C2)c2nc(C)n(C)c2n1 N1(C(=O)C2=NOC3(CCC3)C2)CC2C3CCC(C2C1)N(C(c1sccc1F)=O)C3 S(=O)(=O)(c1ccc2[nH]c(=NC(C)C(C)CO)sc2c1)NCc1ncc(C)nc1 C1(C2CCCN(C(c3ccc(N4CCCC4)c(C#N)c3)=O)C2)(C(=O)OC)CC1 C(=O)(C(C)CC(C)CC)NCCNC(=O)CC1(CO)CC1.O(C(F)F)C(C)O N1(N(C(C)(C)C)C)CCCC(NC(=S)Nc2c(-c3ccccc3)ncn2C)C1 N1(C(C(COCC(=O)N(C2CCC2)C)O)=O)CC(C(=O)N(C)C)CC12CCC2 c1(C(N(C2CCC(NC(=O)COCC(C)(C)C)CC2)C)=O)cnc(S)nc1 c1(CC(=O)NC2CC(CNC(CC(=O)NCC)=O)C2(C)C)c(C)nn(C)c1Cl N1(C(C)=O)CCCCC1C(=O)NC(CNC(c1cc[nH]c(=N)n1)=O)C1CC1 Cc1oncc1C(=O)NC(C)C(N1CC(F)(CNC(c2csc(Cl)n2)=O)C1)=O Cc1ccc2snc(C(=O)NCC(O)CNC(=O)CC3CC3(C)C)c2c1 c1(C2C(C(=O)NCCCOCCNC(C3(C)CCC3)=O)C2)cc(F)ccc1F c1(C(=O)NCC(C2(O)CN(C(c3ncccc3F)=O)C2)(C)C)cc(F)ccc1F C1(OC)CCC2(C(=O)NC3CC(NC(=O)Cn4c(C)csc4=O)CC3O)CC12 Clc1cc2c(N3CCC4CC(c5ccccc5)CCC4C3)ccnc2cc1Cl C(=O)(CCC(O)C(C)(C)C)N1CC(CNC(CCC2C(C)C2)=O)C(C)(C)CC1 N1(C(CCc2nc(C)sc2)=O)CCC2(NC(=O)CSCCC#N)CC2C1 C1(CCC(=O)NC2CC(O)C2)(NC(CNC(N)=O)=O)CCCC1 c1(C(C)NC(c2cnn3ccncc23)=O)ccc2c(c1)CC(C)O2 c1(C(C(=O)NCC)N(C2CC2)Cc2ccccc2Br)cc(C(=O)OC)ccn1 c1(CC(N2CCCN(C(C(C)OC)=O)C(C)C2)=O)ccc([N+](=O)[O-])cc1F C1(NCC2C(=O)NC(C(F)(F)F)CC2)CCN(Cc2ccccc2)C2(CCC2)C1 N1(C(CC2C(NC(C3(C(C)C)CC3)=O)CCC2)=O)CC2CCCCC2C1C c1(N(C)C)ccc(CNC(=O)CC(C)(C)N(C(=O)CCCc2cnn[nH]2)C)cc1 N1(C(C2(CC)CCOC2)=O)CCC(OCCNC(=O)Cc2cn[nH]c2)CC1 CC(O)(C(=O)NCC1CCCN1c1ccncn1)C(F)(F)F c1(NCc2snc(C)n2)cc(N2CCN(C3CCS(=O)(=O)C3)CC2)ncn1 C12(NC(=O)CCC3CCCC(=O)N3)CCC(CC1)N(C(=O)Cc1cncnc1)C2 c1(CC)nc(C)[nH]c1C(N1CCCC1C(C)NC(=O)CC1(O)CCOCC1)=O C1(NC(c2cnc(OCC)nc2)=O)CCN(C(C2CCCN2C)=O)C12CC2 C1(NC(C2CCCN2C2CCCC2)=O)C2CC1CN(C(c1ccccc1F)=O)C2 CC1CC(NC(C2(CCF)CCOCC2)=O)CN1C(C1(c2ccno2)CCC1)=O Cc1nc(C(=O)NCC2C=CC(NC(=O)C(C)CC(C)(F)F)C2)c2ccccn12 c1(NCC2CC(NC(c3n(CC#N)ncc3)=O)C2)ncnc2scc(Br)c12 C(CC(C(C)C)NC(=O)Cc1ccnn1C)NC(C(C)NC(CC)=O)=O N1(C(C(N2CC(C)C2)C)=O)C2CCC1CC(CNC(=O)Cc1ccncc1Cl)C2 C1(NC(=O)COCC2CCCC2)COCC1NC(=O)COCC1CC1 C1(C(N2CCN(CCNC(C(CN(C)C)O)=O)C(=O)C2)=O)CC2OC(=O)OC2C1 c1(C(=O)NCC2CC(NC(C=Cc3cn(C)nn3)=O)C2)ccc(N)cc1O C1(CC)CCCN(CC(=O)NCC(C)(O)CNC(C2(C3(C)OCCO3)CC2)=O)C1 [N-]=[N+]=NCCCCC(=O)N1CC(CCCCNC(=O)CCCCN2CCCC2)C1 CCCC(F)(F)C(=O)NCC1OCCC1C(=O)Nc1conc1CC C(=O)(C(CC)CC(F)(F)F)N(CCC)CCNC(c1c(C)coc1CC)=O Cc1cc(C#N)cc(Cl)c1NC(=O)CC1CCCN(C(=O)CCC(F)(F)F)C1 CC1CN(C(=O)CC2CCCSC2)CC(C(=O)NCCC2NC(=O)NC2=O)O1 c1(C(=O)NC2CC(CNC(Cc3n(C)ccc3)=O)C2)cc(F)c(CO)c(F)c1 C(CS(=O)(=O)c1ccccn1)NCc1cnc(C(C)O)s1 c1(-c2nc(NCc3cccc(OCC)c3O)sc2)ccn2cnnc2c1 N1(C(c2c(N)ccc(CC)c2)=O)CC(C)CN(C(c2nc(C)n(C)n2)=O)CC1C c1(CNC(NC2C(C)CCCC2C)=NCC2CCC2)ccc2c(n1)CCCC2 N1(C(C2(NC(C3CN4CCC3C4)=O)CC(O)C2)=O)CCC2(CC1)CC2 C(c1ccc(C)c(Cl)c1)=CC(=O)NC1C2CCN(C(CCC=C)=O)C21 O(NC(=O)C(O)CC1CCCC1)CC(=O)N(CCN(CC=C)C)CC c1(NC(C=CC(CC)C)=O)cccc(NC(c2cc(N(C)C)ccn2)=O)c1 CCCC(O)CC(=O)N1CC(NC(c2cccc(NC(N)=O)c2)=O)C2(CC2)C1 C=C=CCCC(=O)N(CCCN(C)C)CCNC(c1ccc(N(C)C)cn1)=O N1(CC)CCC(N(C(=O)C(CCNC(=O)CC(C)(C)O)OC)C)CC1 Cc1noc(C)c1C(c1nnnn1-c1ccccc1)NC(C)C(C)(C)CO Cc1n[nH]c(C)c1CNC(c1cnc(CNC(=O)C=CCCC(C)C)nc1)=O N1(C(C2CN(C)C2)=O)CC2(CCCN(C(C3CCCC(O)C3)=O)C2)C1 N1(C(c2cccc(C(=O)OCC)c2)=O)CC(NC(C23CC(CO2)C3)=O)CC(O)C1 N1(C(c2cc(C)no2)=O)CC2(CC(CC(=O)NCCc3scnc3C)C2)C1 c1(C(N(CCC(N2CCC(N(C)CC)C2)=O)CC)=O)cccc(OC)c1 N1(C(C2(C)C(C)OCC2)=O)CCC2(CC1)CC2C(=O)NCc1nn[nH]n1 Cc1cc(F)ccc1C(F)(F)C(=O)NCC(C)N(C)C(c1ccnn(C)c1=O)=O N1(C(CC(CC)C2CC2)=O)CCC(C)(C)C(C(=O)NCCCC(O)CO)C1 CC1CN(C(C2CSCCN2C(c2ccnc(Cl)c2F)=O)=O)CC(C)N1C Cc1ccc2[nH]nc(C(=O)NCC3CC(F)(F)CN3C(c3coc(C)n3)=O)c2c1 C1(C(=O)NC(CCCNC(c2c(OC)nccc2)=O)C)Cc2ccccc2N1C C1(C(=O)NCC(CC)CO)CCCCCN1C(=O)C(C)N=[N+]=[N-] c1(CC(=O)N(C2CCCCC2N)CC)cccc(Cl)c1Cl C(=O)(C1=Cc2ccccc2C1)N1CCN(CCNC(CCCOC(C)C)=O)CC1 N1(C(C(C)O)=O)CCC2CCCC(C1)N2C(=O)CCc1cccc(Br)c1F C(CS(=O)(=O)CC(=O)N1CC2CCC2(CC(=O)NCc2cnsc2)C1)OC C1(C(N2CC(O)(CNC(C=C(C)c3ccco3)=O)C2)=O)OC2CCC1CC2 N1(C(C)C)CCCCC1C(=O)NC1(CCNC(=O)CC2CCC(=O)N2)CC1 C1(C(N2CCC(C3CCCO3)C2)=O)CN(C(=O)CC=C(Cl)Cl)CC12CCC2 CC1=C(C(=O)NCC2CN(C(C3CC(C)(C)CO3)=O)C2)CC1 N1(C(CC(C)C2CC2)=O)CCC2C(NC(=O)Cc3csc(Br)n3)CC12 C1(NC(c2cc(C)nc(O)c2)=O)CN(C(c2c(C)ccn2C)=O)CC(C)(C)C1 Cc1ccn(CC(=O)NC(C)(C)C(=O)N(C)CC2(O)CCCC2)c1 Cc1c(C(N2CCN(C)CC2CNC(=O)CC2CCOC2)=O)cccc1Br C(=O)(C(C)CC(C)C)Nc1cccc(NC(C(CC)(C)F)=O)c1 N1(C(CC2CCC(C)(C)O2)=O)CC2(CCCC2)C1C(N1CC2CC2C1)=O C(=O)(C1Cc2ccc(F)cc21)NC1CC(C)(NC(C(C(CC)CC)F)=O)C1 C1(NC(C(n2c(C)ncc2)C)=O)CN(C(C2CC(C#N)C2)=O)CC12CC2 N1(C(C=Cc2n(CC)ncc2)=O)CCN(C(=O)C(N2CCCC2)C2CC2)CC(O)C1 C1(C(N2CC(F)(F)C2C2CC2)=O)CC2CCC1N2C(C1(CO)CCOC1)=O Cc1cccc(CNC(=O)C(C2CC2(C)Br)N(CC(=O)N(C(C)C)C(C)C)C)c1 CC1CN(C)CCCN1C(c1cnc(C2OCCO2)s1)C(=O)Nc1ccccc1 C1(C(N2CC3CC(C(N4CCC4CC4CC4)=O)CC3C2)=O)CCC(C2CC2)CC1 C(CCN(C(=O)Cc1c(Cl)cnn1C)C)(C(C)C)NC(C(CC)OC)=O CC(C)C(F)(CNC(C1CC2CC1CC2=O)=O)C(=O)NC(C)C(O)C(F)F C#CCC(CC(=O)OC)NC(C1C=CC(NC(C2CCC(C(N)=O)C2)=O)C1)=O C1(O)(C(=O)NCCNC(C2N(CCC)CCC2)=O)CCc2ccccc2C1 Cc1ccc(F)c(Br)c1C(=O)NCCC1(CNC(C2CNC(=O)N2)=O)CC1 C1(C(=O)NCC(CNC(c2n(CC(C)C)ncc2)=O)(C)F)CCS(=O)(=O)N1 Cc1cc(C(=O)O)cc(C)c1OC(c1ccc(C(C)C)c(F)c1)N(C)C C1(C(N2CCC(F)CC2)=O)CSCCN1C(=O)Cn1c(O)nnc1O c1(C(=O)NCC(C2CCCCC2)NC(C(C)(C)C)=O)sc(F)cc1Br C(CCCCCNC(C1CC(CF)C1)=O)NC(=O)CC1CCOC1 N1(C(C(CC)(F)F)=O)Cc2occ(C(=O)NCC(C)(C)CO)c2C1 CS(=O)(=O)c1cnc(NCC2CCCC2NC(c2ccccn2)=O)c(Cl)c1 N#Cc1ccc(CN2CCC3CC(C(N4CC(O)C(F)C4)=O)C3C2)c(F)c1 C=CCC(F)(F)C(=O)N1CC(O)(C(C)NC(=O)COc2cncc(Br)c2)C1 C12(C(=O)NCC(CC=C)NC(=O)CC3CC(C)(C)CO3)CCC(C#N)(CC1)CC2 c1(SC)nc(O)c(C(=O)N(C(C)CNC(c2ccc(Cl)s2)=O)C)cc1C#N CCCC(C)C(CO)NC(C1(CCNC(=O)CC2CCSCC2)CCC1)=O N1(C(CCC)=O)CC(NC(c2ccc(C(C)(C)C)cn2)=O)CC1(C)COC C1(CCC)(NC(c2ccnc(OC)c2F)=O)CCN(C(=O)CSC(C)C)CC1 c12ccc(c(OC)c1)S(=O)(=O)NC(=O)CN2.C1(C(CC)OC)CCCCC1 C(N=c1ccc2cc(S(=O)(=O)O)ccc2[nH]1)C1CC(N)C(O)C1 C#Cc1cc(C(=O)NCC(C)(CO)NC(=O)C(CC)C2CCOCC2)cc(F)c1 C1(CNC(C(=O)NCC(F)F)=O)CN(C(c2n[nH]c(C3CC3)n2)=O)CCC1(F)F C1(NC(C(CCC)(C)C)=O)CC2CN(c3nc(C(F)(F)F)cc(C)n3)CC2C1 CN1CCCC2(CCN(Cc3cn(Cc4nccs4)nn3)C2)C1=O N1(C(COCc2cc(OC)ncc2)=O)CCN(C(=O)CCCC(F)F)CC(O)C1 N=c1[nH]nc2ccc(N3CCN(C(=O)CCc4cc(Cl)cs4)CC3)nn12 C1(CNC(CC(=O)NCC#C)=O)CN(Cc2nnc(C3CC3)o2)CCCO1 C(=O)(N=c1ccn(CC2CC2)[nH]1)C1CC(NC(C(CCN(C)C)(C)C)=O)C1 Nc1ccc(-c2cn(CC(=O)Nc3ccccc3C(F)(F)F)nn2)cc1 c1(CC)cccc(C(N2CC(Nc3ncncc3Br)C(C)(C)C2)=O)c1F C1(S(=O)(=O)c2ccccc2)(C(=O)NC(C)CNC(C2CC=CC2)=O)CCC1 C12(C(N3CCC(NC(C(N4CCOC4=O)C)=O)C3)=O)CCC(CF)(C1)OC2 N1(C(C=NOC)=O)CCC(C(F)(F)F)C(NC(c2oc(C)cc2C)=O)C1 c1(C(=O)OC)cc(C(=O)NCC=CCNC(C2(C(C)C)CCC2)=O)ccc1C C#CCC(CC(=O)NCC1CN(C(C2(CCC)CC2)=O)CCO1)c1ccccc1 C(=O)(CC(O)C(C)(C)C)NCC1(NC(C2N(C)C(=O)CC2)=O)CCCCC1 c1(C(=O)NC2(C(N3C(CNC(C)=O)C=CC3)=O)CC2(C)C)ncn(C)c1C C(=O)(CC(C)CC(C)C)NCC1CCN(C(C=C(C)C)=O)C(C)C1 C(=O)(CCC(=O)C(C)(C)C)N1CCC(C)(C(N(C)Cc2cnccn2)=O)C1 C1(NC(=O)C(C2(O)CN(C(=O)C=CCN3CCC3)C2)F)CC12CCCC2 C1(NC(c2c(OC)n[nH]c2)=O)CN(C(=O)CC2C=CCCC2)C2(CCCCC2)C1 c1(C(=O)NC(CNC(C=CC(=O)OCC)=O)C)ccc(OC)c(C)c1C CCC(C)(C#N)C(=O)N1CC(CNC(C2CC(O)(C(F)(F)F)C2)=O)C1 C1(C)(NC(C(c2n(C)ncc2)NC(c2ccc(Cl)s2)=O)=O)CCC2(CC1)CC2 C1(CCNC(=O)C(c2ccc(Cl)cc2)CO)CCCN(C(=O)C(F)(F)C2CC2)C1 C1(CC)C(NC(=O)Cn2ccc(C)c2)CCCN1C(=O)CCCn1cccn1 c1(C(=O)NCC2CCCN(C(CC(C)F)=O)C2)cc(N)c(F)cn1 C1(C(=O)N(C(C)(C)C)Cc2cnc[nH]2)C=CC(NC(N)=O)C1 N1(Cc2n(CC)cnn2)CC2C(NC(=O)Cc3nnc(C)s3)C2C1 n1(C(C)C)c(CCC(CC(N)=O)c2ccccc2)nnc1Br N1(C(=O)C2CC2)CC2OCCN(C(=O)Cc3cnns3)C2C1 C1(NC(CC2(C)CCN2C(C2CCSCC2)=O)=O)CC(=O)N(O)C1 CN1CC(N(CC(c2ccccc2)C2CC2)CC(=O)NC2CC2)C(O)C1 N1(C(c2ccc(C)nn2)=O)CCC(CO)C(NC(c2coc3c2CSC3)=O)C1 c1(C(CO)NC(c2scc(C(=O)OC)c2)=O)ccc(OC)c(OC)c1 N1(C(CCC=CC)=O)CC(C)CCC1CNC(=O)C(N1CCC(C)CC1)=O C(=O)(C1CCCc2cncn21)N1CC2C(CNC(CCC#N)=O)(CCC2)C1 CC(CCC(=O)NCCN(C)C(C1CCS(=O)(=O)N1C)=O)S(C)(=O)=O C1(CC)(NC(C2CCC(n3cc(CNC(=O)NC)nn3)C2)=O)CCOC1 c1(OC)ncc(C=CC(=O)NC2CC3(C2)CN(C(=O)CC2CC2(Cl)Cl)C3)cn1 c1(C(=O)NCCC2N(C(C(COC)O)=O)CCC2)ccc(C(C)C)cc1 C=CCCC(F)(F)C(=O)N(CCCCNC(c1cc(OC)cc(C)n1)=O)C C(C(=O)N(C(C)CC(=O)NCc1ccc(Cl)cc1)C)(C(C)C)SC c1(NC(N)=O)cccc(F)c1C(=O)NCC1CC(NC(c2cnco2)=O)CCO1 N1(C(C23CCC(C)(CC2)OC3)=O)CCC(C2CC2NC(C2CCCO2)=O)CC1 C1(C(C)C)CCC(C(=O)NC(Cn2cncn2)CC)N1C(=O)CC1OCCO1 C1(NC(C(C)OCc2ccccc2)=O)CN(C(=O)C(F)C(F)(F)F)CCC1C C12(CNC(C3(CC=C)CCC3)=O)CC1CN(C(C1(C(C)(C)O)CCC1)=O)C2 C1(C(N2CCC(OCCNC(c3c(C)cccn3)=O)C2)=O)COC(C)(C)CO1 c1(C(N2CC(CNC(c3cc(C)cc(O)c3)=O)OCC2)=O)cnc2ccoc2c1 c1(C(N2C(C(=O)Nc3c(C(N)=O)cccn3)CCC2)=O)cccc2c1NCCC2 N1(C(C)(C)C)CC(C(=O)NC2CCC(NC(=O)C3CC3)CC2)CC1=O N1(C(c2ncc(OC)nc2)=O)CCCN(C(c2ncccn2)=O)C(C(C)C)C1 C(CC(C)C)(C(=O)NC1CC1NC(C1(C#N)CCSCC1)=O)NC(C)=O C1(C(=O)NC(CC)(CC)CCNC(C2CCC(C)(C)C2)=O)CCc2c[nH]nc2C1 C1(C(=O)NCCC2C(C)CN(C(=O)Cc3ccccc3)C2)CC(S(C)(=O)=O)C1 N1(C(c2cc(C)no2)=O)CCN(C(c2cnn(C)n2)=O)C(c2cccc(Cl)c2)C1 N1(c2n(CCOC)c(CCCCC#N)nn2)CCOc2c(C)cccc2C1 N1(c2c(OC)cncn2)CCC(NC(=O)CC(C)(C)C)CC(C)(C)C1 C1(CNC(=O)NCCCC(CC)O)CCCCC1(C)C c1(OC)ccc(N)c(C(=O)NC(C)CC(C)NC(c2ccncc2OC)=O)c1 c1(C(N2CC(CCCNC(COCCC)=O)OCC2)=O)ccc(O)c(F)c1 c1(C(=O)NC2C(NC(C3CCC(C)(C)CO3)=O)CC2)cccc2c1CNC2=O C(CCCC(C)NC(C1CC(CN(C)C)C1)=O)NC(C=CC(=O)OCC)=O C1(NC(c2c(C)n(C)nn2)=O)CC(NC(=O)C=C2CCOCC2)C12CCOCC2 C12(CC3N(C(=O)N(CC(O)CO)CCO)CC(F)(F)C3)CC3CC(CC(C3)C1)C2 c1(C(=O)NCCC(C)(C)NC(C2OCCC2(C)C)=O)cccc(CCO)c1 Cn1ncc(=NC(=O)CC2CN(Cc3cc(Cl)ccc3O)C2)[nH]1 Cc1cc(C)cc(C=CC(N2CCOCC2CCC#N)=O)c1 Cc1c(C(N2CC(CC(C)NC(=O)C(C)CO)C2)=O)c(O)nc2ccccc12 c1(CCOCCN(CCNC(c2cnoc2)=O)C(C2CCO2)=O)ccccc1 C1(c2nnnn2C2(C)CC2)(NCCSC(C)C)CCC2CC12 N1(C(c2ccc(C(C)=O)o2)=O)CC(C)(C)C(NC(=O)C=CCO)C(C)(C)C1 C1(O)(C(=O)NCC(CC)(C)OC)CCCCC1O C1(CCNC(C2CC=CCC2)=O)CCCCN1C(=O)Cc1ccsc1Cl C1(C(N(C2CN(C(C(CCC)=CCC)=O)C2)C)=O)CN2CCC1CC2 C12CCCCN(C1)C(C)c1cnc([nH]1)CC(=O)N2.c1(CC)ncc(C(C)C)o1 C(C#Cc1cnn(C)c1)NC(CC(C(C)C)NC(C(COC)(C)C)=O)=O C1(CNC(C2=C(C)CCC2)=O)CCN(C(c2ccc3occc3c2)=O)CC1(F)F c1(OC)cc(C(C)=O)ccc1OCC(=O)NCC(O)C(C)(C)O C(c1cccc(O)c1)=CC(=O)NCC1CN(C(c2n(CC)ccn2)=O)C(C)C1 C(=O)(CCCCC(=O)N1CC(O)(CNC(C2CC(F)(CO)C2)=O)C1)NC N1(C(c2n(CC)cc(Cl)c2)=O)CC(NC(C2CC3C=CC2O3)=O)CC2(CC2)C1 c1(C(N2C(C)CC(NC(c3c(C)n(C)cn3)=O)C2)=O)cccc2cccnc12 C=CCC(C)(C)CC(=O)NC1CCC(N(C(=O)CCCCN(C)C(C)C)C)C1 C1(C(N(C)Cc2cc(OC)cc(F)c2)=O)CCn2cnnc2C1 N1(C(c2ccc(Cl)c(C)c2Cl)=O)CCOC2(CCN(S(=O)(=O)CCCl)CC2)C1 c1(CC(=O)NC(C)CCNC(C2CCCC2C)=O)ccc2c(c1)ncn2C Cc1cnc2c(C(N3CC(NC(c4nc(Cl)sc4Cl)=O)C4CC34)=O)cccn12 C1(N(C(CC(C)OC)=O)C)CCN(C(=O)CS(=O)(=O)NCC2CCCO2)CC1 C=Cc1ccc(C(=O)NC(CNC(=O)CCc2cccnc2)C(C)C)cc1 CC1CCN(C(c2cnn(CC(F)(F)F)n2)=O)CC1NCN(C)C1CC1 N1(C(C2CCN(CC)C2)=O)CCC2(CC1)CC2(C)C(=O)N(c1ccccn1)CC C1(C)(C(N2CC(CNC(C3(C)CC3)=O)C(O)C2)=O)CCCS1(=O)=O c1(CC(=O)NCCN(C(C2N(C(CC)=O)CSC2)=O)C2CC2)cccc(Cl)c1 c1(C(N(C(C)C(=O)NC(CN(CC(C)C)C)CC)CCC)=O)sc(CC)nc1C C12(C(=O)NC(C3CCN(C(=O)CC4C=CCC4)CC3)C)C3C4C1C1C2C3C41C#N c1(C(C(=O)NCC23OCC(C(=O)Nc4n(C)ncc4)(C2)C3)O)cc(Cl)cc(Cl)c1 c1(OC)nccc(NC(C2CC2NC(=O)C=Cc2ccc(O)cc2)=O)c1Br C1(CN(C)C(c2cnc(S)[nH]2)=O)CCCC(NC(C2(c3ccsc3)CC2)=O)C1 CC(C)C(C(=O)NCC1CCCC1N(C)C)C(C)NC(=O)CC1(C)CC1 C1(C(=O)NCCC(C)N(C(c2nc(OC)nc(O)c2)=O)C)CCC2(CCC2)CO1 c1(C(N2CCCC(NC(CCC(=C)Cl)=O)C2)=O)oc2ccc(C)cc2c1C C1(NC(C(CC)C)=O)CCCCC12CCN(C(c1ccn(C3CCCC3)n1)=O)C2 CC1(CO)C=CCN1C(C1OCCC1CNC(C1CS(=O)(=O)C1)=O)=O C1(NC(=O)COC2CCCCC2)CCCCCN(C(C2(C3CCCO3)CCC2)=O)C1 N1(C(C(CCC)(C)CC)=O)CCC2(C1)CN(C(C1(C)CCCCO1)=O)CCO2 N1(C(c2c(OC)scc2)C(=O)NC2CC2)CCCC(n2nc(C)cc2C)C1 N1(C(C(C)OCCC#C)=O)CCN(C)C(CNC(C2(n3cccn3)CCC2)=O)C1 c1(N2CCC(OCCNC(C=C(C)Cl)=O)C2)cc(Cl)ncn1 c1(C(N2CC(CN(C)Cc3ccsc3Br)C2)=O)c(I)ccnc1F C1(OCC(=O)NC(C(=O)NC(CC)CN(C(C)=O)CC)C)CCCCCC1 C(=O)(CC(C)(O)C(F)(F)F)NC1CC2CN(C(CCC(C)(C)C)=O)CC1C2 Cn1ncc2c1CN(C(C1CC(F)(F)CN1Cc1cccc3nonc13)=O)CC2 CCCC(CNC(c1ncccc1C)=O)C(=O)N(CC(C)C)CC(C)C C1(NC(CCCC(=C)C)=O)CN(C(C2(C)COC(C)(C)OC2)=O)CC2(CCC2)C1 CC1=C(C(=O)N(C)CCNC(=O)CCOc2cccc(Cl)c2)CCC1 N1(C(CCC2C(C)=NOC2=O)=O)CCCC(C)C1CNC(=O)C=C1CCN(C)C1 C1(C(N2CC(O)(CCNC(c3cncc(O)c3)=O)C2)=O)COCCC1(F)F Cc1cccc(NC(C(=O)NCc2ccnnc2)C(C)C)c1C c1(C(=O)NCCC(C)N(C(C2CCC(CC)O2)=O)C)cc(C(F)F)ccc1Cl C1(CNC(C(C)O)=O)CC2CCC(C1)N2c1ccc(C(F)(F)F)cn1 N1(C(c2ccc(-n3cc(C4CCCC(O)C4)nn3)o2)=O)CCCC(O)(CO)CC1 C1(CC=C)(NC(c2ncccc2C)=O)CCCN(C(=O)C(C)NS(=O)(=O)CC)C1 n1(C(C)C)cc(C(=O)NC2CC2NC(=O)COC2CC=CC2)cn1 C1(CNC(C2N(CCC)CCC2)=O)(COC)CCCN1C(=O)Cc1cccn1C N1(C(C2(C)COCCO2)=O)CCC2C(C(=O)NCC(F)C3CCC3)C2C1 CCCC(C)(CC)C(=O)NCCCNC(c1ccc(C#N)c(C)c1)=O N1(C(=O)C2=CCCOC2)CC2CCC1CN2C(c1cn(C2CC2)cn1)=O c1(C(=O)NCCC(=C)CNC(=O)C(C)CO)cn2c(n1)CCC(C)C2 C1(C(=O)Nc2cc(C(=O)OCC)[nH]c2)CCCCN1c1ccnc(SC)n1 N1(C(COC(C)C)=O)CCC(C2CCN(C(=O)C3=CNC4=NCCCN34)C2)CC1 C1(C(=O)N(C(C23CC4CC2C3C4(F)F)=O)CC2CC2)CCC2(CCNCC2)CC1 Cc1nc2cc(C(N3CC(CNC(=O)CC4CS(=O)(=O)C4)C3)=O)ccc2o1 C1(CC(=O)NCCCN(C(=O)CCc2nncs2)CC2CCCC2)CCNC1=O C1(C(=O)NCC(C2CCC2)NC(=O)Cc2cc(C3CC3)on2)CCCC2(CC2)C1 S(=O)(=O)(c1cnc(NCC2(S(C)=O)CC2)c(Cl)c1)N(C)Cc1cccc(F)c1F C(=O)(CC(C)(C)C(F)(F)F)N(CC(C)NC(Cn1c(C(C)C)nnn1)=O)C C=CCCC(C(=O)NCc1cc(O)cc(F)c1)NC(=O)CCc1ccco1 c1(OC)ncc(C(=O)NC2C=CC(CNC(=O)C3CC3)C2)cn1 N1(C(C2C3CCOCC23)C(=O)NCC)CC=C(c2ccc(C)cc2)CC1 C1(NC(C2(C=C)CC2)=O)CC12CCN(C(=O)C(C)(C)N1CCCCC1)CC2 C1(OC(c2ccc(Cl)o2)=O)C2CC3C(=O)OC1C3O2 N1(C(C(C)=C2CC2)=O)CCN(C(=O)C(C)C(F)F)C(c2cn[nH]c2)C1 c1(C(=O)NC2CC(CNC(c3cn4c(n3)SCC4)=O)C2)ccc2sccc2c1 c1(C(=O)NC(CNC(C(C)NC(CC)=O)=O)(C)CC(C)C)ccnc2[nH]ncc12 C(C(C(C)C(C)C)NC(c1c(Br)c(C)nn1C)=O)NC(CCC)=O C(=O)(C1Cc2ccccc21)NC1(COC)CN(C(=O)CCc2ccsc2)C1 c1(C(=O)NCC(C)CNC(c2ccc3cncn3c2)=O)cccc2c1COCC2 C1(CC)CN(C(C23CC(CO)(C2)C3)=O)CCN1C(c1c(C)coc1C1CC1)=O c1(C(=O)OC)ccc(NC2(F)CN(C(=O)C(C)Oc3ccccc3)C2)c(I)n1 N1(C(CC(=O)NCC)=O)CCCC1(C)CNC(c1cn(C2CCOC2)nc1C)=O C1(CNC(C(n2cc(-c3ccnn3C3CC3(F)F)nn2)C)=O)CCC2(CC2)C1 c1(NC(=O)CCc2ncc[nH]2)cccc(NC(=O)C(O)CC2CCOCC2)c1 Cc1cc(=NCCOCC2CC2)[nH]c(NCC2CCCCC2c2ccccc2)n1 c1(C(N2CCC(NC(=O)COC(F)(F)F)CC2)=O)cc2c(O)cccc2[nH]1 C(N=c1[nH]c(=NC2CCC(C)C2)[nH]c2c1COC2)c1c(C)sc(Br)n1 N1(C(c2cc(C)c(CO)cn2)=O)CC(C)CN(C(=O)C=Cc2cocn2)CC1C S(=O)(=O)(c1c[nH]c(C(=O)N(CC(C)NC(=O)C(C)(C)C(N)=O)C)c1)NCCOC N1(C(C23CCCC2C3)=O)CCC2(C1)CN(C(C1(Cl)CC1(F)F)=O)C2 Cn1ncc2cc(C(N3CC(NC(c4cccs4)=O)CCC(O)C3)=O)sc12 C(=O)(C(C)n1cncn1)NCC1(C(C)NC(CC)=O)CC1 C1(NC(C(CO)OC)=O)CN(C(C2(C)CCOC2)=O)CC1CO CC(C)S(=O)(=O)C(C)C(=O)N1CCCC(NC(c2ccn3ccnc3c2)=O)C1C C=CCC(C)C(=O)NCc1cn(C2CCN(C(=O)C(C)n3ccnn3)CC2)nn1 C(C(C(=O)NCC1CCN(C(C)C)C1)NC(=O)C(C)=CC1CC1)OC c1(C(=O)NCc2c(C(=O)NCCC3C(C)CCO3)con2)occ2c1CCC2 c1(C(N(C(C)CN(C(=O)Cc2nc(=N)[nH][nH]2)C)C)=O)ncc(F)cn1 c1(C(N2CCCC(CO)(NC(C3(F)CCCCC3)=O)C2)=O)ncn2c1CCC2 N1(C(C(C=CC)O)=O)CCC(CNC(c2cn(C(C)(C)C)nc2C)=O)C12CC2 C1(NC(C=CCC)=O)CC2(CCN(C(=O)CN3CCN(S(C)(=O)=O)CC3)C2)C1 C=C(C)CC(C(=O)N1CC(O)CC1C(=O)NC1CCC(C)CC1)OC C1(C(N(CCN(C(=O)CCc2cscn2)C)C)=O)CC1(F)F C1(OC)CC(C)CN(C(=O)CC(CC2CC2)NC(=O)C(n2nccc2C)C)C1 c1(C(=O)NC2C(C(=O)NCC3(O)CCC3)C2)ccc(Br)c(C(F)(F)F)c1 C(=O)(CC(C)C(C)(C)NC(=O)CC(C1CC1)C1CC1)Nc1ccc(OC)nc1 c1(C(=O)OC)cc(CCC(=O)NC(C)CCNC(C2CN(C)C2)=O)c[nH]1 C1(C(=O)NC(C(=O)NC)CC2CC2)CNCCS(=O)(=O)C1 c1(OC)cc(C)cc(C(=O)NCC2(F)CCC(NC(=O)C(F)(F)C(C)O)C2)c1C c1(CNC(NCC(CC)OC)=NCCOC)nc2cc(C)ccc2n1C Cc1c(F)cc(C(N2CCC(F)(C(=O)NCc3ccccc3)CC2)=O)cc1Br C=CCC(C(=O)NC1CC(C(=O)NCC(F)C(C)(C)O)C1(C)C)C(C)C C1(C(N(CCN(C(C=NOC)=O)C)C)=O)CC(O)CN1C(c1cnc(N)cn1)=O C1(CCC(=O)NCCCN(c2nncs2)C)NC(=O)NC1=O CC1CCCC1(C)C(=O)NC1CCN(C(C2(Br)CC2)=O)CC1 N1(C(C2CC(N(C(C(C)n3cccc3)=O)C)C2)=O)CC2C(=O)NC(=O)C2C1 c1(C(=O)NCCOCCN(C)C(C2CC(C)(O)C2)=O)cc(C(F)(F)F)c(Cl)cn1 c1(CC(C)C)ccc(-c2nc(CC(C)C)nn2-c2cnnn2C)cc1 N1(C(C(CC)OCC)=O)CCCC(C)(C)C1CNC(c1ccc2c(c1)COC2)=O C(=O)(C1CCc2nnc(C)n21)N1CC(NC(CC=CC)=O)C(OC)C1 Cc1ccc(NC(N2CCC(N(C)C(c3cnoc3C3CCC3)=O)C2)=O)cc1C c1(C(=O)NC2C(NC(CCNC(N)=O)=O)C2)cnc(O)cc1C(F)(F)F C(CC1OCCc2ccccc21)C(NNC(C(N1C(C)(C)CC(c2nn[nH]n2)C1)=O)=O)=O O=C(CC(C1CC1)C1CC1)NCCCC1CCN(CCN2CCCCC2)C1 CCC(C)(C)C(O)C(=O)N1CC(CC(=O)Nc2cnc(C)c(C)c2C)CC1(C)C c1(CCn2cc(CC(O)C3CCC3)nn2)cn2ccccc2n1 Cc1nc(O)c(Br)cc1C(=O)NCC1CN(C(c2cnsn2)=O)CC1C N1(C(c2cn3ccccc3n2)=O)CCOC2(CCN(C(C3CC4CC4C3)=O)C2)C1 N1(C(=O)C=Cc2ccco2)CCC(N2CCN(C(=O)CN3CCC3)CC2)CC1 C1(O)(C(C)NC(c2cc(C)nnc2)=O)CCN(C(=O)C(C)(C)CF)CC1 CCC(CC)C(F)C(=O)NCC(CNC(C1CN(C2CCN(C)CC2)C1)=O)CO N1(C(Cc2cc(C)nn2C)=O)CC2CCC1C1CN(C(=O)C=CC3CC3)CC21 n1(CC(=O)NC(CCNC(C=C(C)Cl)=O)C)ncn2cccc2c1=O c1(OC)c(C(C)NCC(=O)N(C)CC2(OC)CCC2)cccc1Cl c1(C(N(C2C3N(C)C(CCC3)C2)C(C)(C)C)=O)cnc2cc(Br)ccc2c1 c1(C2(NC(=O)NC3CCCN(c4cccnc4)C3)CC2)ncc2c(n1)CCC2 Cc1c(C(=O)Nc2nc3ncc(Cl)cc3s2)c(C)n2ccncc12 c1(N2CCC(C(C)(C)CNC(=O)C=C3CCC3)CC2)cc(Cl)nc(S(C)(=O)=O)n1 Cc1ccc(COC(C)C(=O)NCC=CCNC(C2CCOC2(C)C)=O)cc1 CC1(C)CC(NC(=O)CC2CC3(CC3)CO2)CN1C(c1ccoc1Cl)=O c12cccc(c1)C2.c1(CC(=O)OC)cn(CC(=O)N(CC(C)O)C(C)C)nn1 c1(C(=O)NCC2(CN(C(CCCC)=O)C)CC2)cc(C)c2c(O)nc(O)nc2n1 Cc1c(Cl)cnc(NCC(C(C)(C)C)NC(c2cc3ccccn3n2)=O)c1C#N N1(C(C(CCC)OCC)=O)CC(CNC(C2(F)CC2)=O)C(C)(C)C1 Cc1cc(Cl)nc(N)c1C(=O)NCCCCCNC(c1ccc(C(N)=O)o1)=O Cc1cc(C)cc(S(=O)(=O)N2CCC=C(C(=O)NCCCS(C)(=O)=O)C2)c1 C(=O)(C1CCCn2nccc21)NC1CC(C)(NC(C(CCC)NC(C)=O)=O)C1 C1(C(=O)NCC(CSC)(C)O)CC(C)CCN1C(=O)CC(=O)NC1CC1 N1(CC)C(C)CN(C(=O)C(C)(CO)NC(c2cncs2)=O)CC1C Cn1ccnc1C(F)(F)C(=O)NCCCNC(C1CCOC1C(F)(F)F)=O C1(NC(=O)C(N2CCOC(c3ccccc3)C2)=O)CCN(CCF)C1=O C#CCCCCC(=O)N1CCCC1CNC(=O)CNC(=O)Cc1ccc(N)cc1 N1(C(CC=CC=C)=O)CC2CC(NC(C3CC34CCSCC4)=O)C(C2)C1 C1(C(=O)NCC2(CNC(c3ncn(C)n3)=O)CC23CCC3)CC(=O)OC1(C)C Cc1nc(Br)c(CNC2(c3nnnn3Cc3ccccc3)CC(C)N(C)C2)n1C C1(CC(=O)OCC)(NCC2NCC23CCC3)CCOCC1 N1(C(CCC)=O)CCN(C(c2cn(C)nc2-c2ccoc2)=O)CC1C C1(NC(C(CCC)C)=O)CN(C(C2C(F)(F)C23CCC3)=O)CCC1C C1(C(=O)NCC(C)NC(c2ncc3ccccn23)=O)CCCCC12OCCO2 N1(C(CCCNC(=O)OC)=O)CC(C(=O)NC(c2nn(C)cc2O)C)CC(C)C1 CCCC(C(O)C(=O)NCCC1CC=CCC1)NC(=O)COCCF c1(C(=O)NC2C=CC(CC(=O)Nc3cncnc3O)C2)cccc2ncccc12 c1(C(=O)NCC2OCCCN(C(C(=O)NCCOC)=O)C2)ccc(C#N)cc1F c1(C(=O)NC2CCCN(C(CCN(CCC)C)=O)C2)cc(NC(C)=O)ccc1C C(=O)(CS(=O)CCC(F)(F)F)N1CCC(O)(CN(C(=O)Cc2ccccc2)C)C1 N1(C(C2(CC(=O)OC)CC2)=O)CCC2(CC1)CC2C(=O)NCC(O)C(C)C C(=O)(C1=NOC(CNC(C2C3(CC3)C23CC3)=O)C1)NC(C)C(=O)NC1CC1 CC(F)(F)C(=O)NNC(=O)c1cccc(Cc2ccc3occc3c2)c1 c1(-c2cn(C(CNC(C3CC(=C)C3)=O)C)nn2)cc(C)cc(F)c1 C(=O)(CC1OCCc2sccc21)N1CC(F)CC(NC(CNC=O)=O)C1 CN1CC2CCC(C1)N2C(C1C2CCC(C2)C1NC(C1(C)CCCOC1)=O)=O c1(C(C)=O)ccc(NC(=O)C(C)SCc2nc[nH]n2)cc1 N1(C(Cc2cccc(CC)c2)=O)CC(NC(=O)C=CC2CCCC2)C(C#N)C1 CC1(C)OCCC1CC(=O)NCCNC(C1C(C)(C)C1(F)F)=O CC1(C)COC(C)(CNC(=O)C(=O)Nc2c(Cl)ccc(Cl)c2Cl)CO1 Cc1coc(C(N2CCC(NC(c3ccc(-n4ccnc4C)nc3)=O)C2)=O)c1C c1(NC(c2n(CCC)ccn2)c2nnnn2CCCF)cc(CC)c(F)cc1C C1(C(=O)NCC2C(C)=NOC2=O)CC2CC(O)CC(C1)C2.C12CCN1C(=O)N2 c1(NC(c2n(CCCC)nnn2)C2(COC)CC2)cnc(C)c(Br)c1 c1(CC)c(C(=O)NC(C)CN(C)C(c2cnc(C(N)=O)cn2)=O)cnn1C C1(C(=O)NC(CC(C)C)CNC(=O)C=Cc2ccccc2)CCCS(=O)(=O)C1 C1(CCNC(CSCC(C)=O)=O)CCN(C(c2ccnnc2)=O)CC1 c1(OC)ncc(C(N2CC(NC(c3cc(C)ncc3C)=O)C(C)C2)=O)cc1C C1(C(N(CCCOC)CCO)=O)CCCCN1C(=O)CCc1nc(C)no1 NC1CC(C(=O)NCC2(c3ccc(F)cc3F)CCCC2)CCC1CO C1(CNC(C(C)NS(C)(=O)=O)=O)CCC(F)(CNC(=O)CC2CCC2)CC1 C1(CCC(=O)NC(C(=O)NC2C(CC)C2)c2cccs2)(OC(C)=O)CCCC1 CC1CCC(=CC(=O)N(CC(=O)NC2(C(F)F)CCCC2)CCN(C)C)CC1 C1(c2cn(C)nc2)C(C(=O)NC(C2CC2)C2CC2)CC(=O)N1CCON C=C=CCC(=O)NC(C)CN(C)C(c1cn(Cc2ccccc2)cn1)=O N1(C(C(C)NC=O)=O)CCCCC(CNC(=O)CCOCC2CC2)C1 C1(CC(=O)NCC2(C(=O)OC)CCC2)CN(C(c2coc(C)c2)=O)CCC1C C1(NC(C2N(C(C(C)OCC#C)=O)CC(C)C2)=O)CC2C(O)C(O)CC12 C1(NC(c2ccnnc2S)=O)CC2CCCC(C1)N2C(=O)C(F)C1CCC1 N1(C(CN(C(C)C)C)=O)CC=C(CNC(C2CCC3CC3CC2)=O)CC1 O=S(=O)(c1nc(C(F)(F)F)cs1)N1CCn2nccc2C1 C(=O)(C1=CCCC(C)(C)C1)NC1CC(c2n(C)ncc2)OCC1 CC1CN(C(C2CCOC2)=O)CCCN1C(c1cc(C(F)(F)F)ccc1O)=O c1(NC(c2csc(-c3cnccn3)n2)=O)nccc2c(F)cccc12 C12(CC(F)(F)C1)N(CCc1ccccc1)C2=O.N1(CC)CCC(N(C)C)CC1 CC1(C(=O)NC2COCCC2NC(=O)C=C2CN3CCC2CC3)CCCS1(=O)=O N1(C(C(C)O)=O)CCCCC(NC(=O)CSc2ccccc2Cl)CC1 c1(OC)ccc(C(N)=O)cc1C(=O)NCC1CC=CCC1 c1(C(N2CC(C)C(NC(C3(CO)CCOCC3)=O)C2)=O)cc(O)nc(N(C)C)n1 c1(SC)cc(C(N2CC3CC2(CNC(=O)C2=CCSC2)C3)=O)ccc1[N+](=O)[O-] C1(NC(C2N(CC)CC2)=O)CCN(C(c2nscc2Br)=O)CC1 c1(C(N(C)CC2N(C(C(c3cn(CC)nc3)=O)=O)CCC2)=O)cccn(C)c1=O N1(C(c2c(CNC(CCc3n(C)cnc3)=O)occ2)=O)CCCC2CC12 N1(C(=O)C2=CCCOC2)CC(NC(C2(c3ccccc3)CC(F)C2)=O)CC2(CC2)C1 C(N=c1ccnc(NCC(c2ccsc2)C)[nH]1)c1c(CC)snn1 C1(N(C(c2ccc(N(C)C)cc2)=O)C)CCOC(C)(C)C1.N12CCC(C(O)C1)C2 n1(CC(N2CCC(NC(=O)Cn3ncccc3=O)C2)=O)ncc2ncccc12 c1(C(=O)NC2CC3CN(C(COCCC#C)=O)C2C3)ccc2c(O)ncnc2c1 N1(C(C(C)Oc2ccccn2)=O)CC2CCC1C1CN(C(=O)C(C)(C)CF)CC21 c1(C(N2CCN(C(CC)=O)CC2C(C)C)=O)nsc2ccccc12 Cn1nc2c(c1C(=O)NCC1CC(NC(=O)CCC(C)(C)C)C(O)C1)CSCC2 C1(C(N2C(C)CN(C(C3CC4(C3)CC(O)C4)=O)CC2)=O)C2Cc3ccccc3C12 c1(C(=O)NC2C=CC(CNC(c3cc(C)oc3)=O)C2)ccncc1C(F)F CC1=NOC(C(=O)NCC2(CNC(c3cc(C)oc3C)=O)CCCC2)C1C C1(C(NOC)=O)CN(C(=O)CC2CC=CCN2C)CC1C(C)C Cc1nc(CC(F)(F)F)sc1C(=O)NCC1(C)CCN(C(=O)C2=CCOC2)C1 c1(OC)cc(C(=O)NCC(F)CNC(c2csc(Cl)c2)=O)ccc1Cl CCCCCC(O)C(=O)NCc1cccc(C(=O)NCC2CC=CCC2)n1 C1(N(c2cc(Cl)c(Br)cc2Br)C(c2ccc(Br)cn2)=O)COC2(CCNCC2)C1 C1(NC(C2C(=C)C2)=O)CC(OC)CN(C(=O)CSc2cccnc2)C1 Cc1ccc(C)c(C(N2CC3(CO)CC2(C(=O)NCc2cccc(C)c2F)C3)=O)n1 c12ccc(cc1)CNC2=O.N1(CC2(CC(C)C)N=N2)CC(c2cccs2)CC1C.O C1(N(C(c2cc(C)n(C(C)C)n2)=O)C)CN(C(=O)Cn2nccc2C)CCC1C C#CCCCCCC(=O)NCCOC1CCN(C(C2SCCS2)=O)C1 Cc1cccn(CC(=O)NCC2CN(C)CCN2C(=O)Cn2cc(Cl)cn2)c1=O C1(CC(=O)N(CCCNC(c2ccns2)=O)C(C)C)CCC(=O)NC1=O n1(CC)nc(C(=O)NCC2COC(CNC(C3CCCN3C=O)=O)C2)cc1O C(CCC(=O)NC(c1nc[nH]n1)CC)NC(C1(CC#C)CC1)=O C1(CNC(c2ccco2)=O)Cc2ccccc2CN1C(=O)Cc1ccccc1F c1(CNc2cncc(C(C)(C)O)c2)ccccc1S(=O)(=O)c1ccccc1 N1(C(c2c(CC)n(C)cc2)=O)CCCC(C)(C(N2CCCCC2)=O)C1 N1(C(C(c2c(C)noc2C)(C)C)=O)CC2CN(C(=O)C(C)C(C)(F)F)CC2(C)C1 C1(n2cc(CCN(C(=O)CC3CCC(=O)O3)C)nn2)C2CC3C(C2)C13 c1(C(=O)NC(C(C)NC(c2ncc(C)cn2)=O)CO)cnn2c1NCC(C)C2 C(=O)(C(C)CC(F)(F)F)N1C(CNC(c2c(Cl)nc(OC)s2)=O)CC1 N1(C(C(C(CC)CC)C)=O)CCC(=O)NC2CN(C(c3ccnn3C)=O)CCC12 c1(NC(N2CCC(CC)CC2)=O)ccc2cnn(C)c2c1 C1(CNC(C=CCOC)=O)CC2CCC1N(C(=O)C1=CCCOC1)C2 CCC(O)C(F)(F)C(=O)N1CC2(COC(CNC(=O)CCCn3ccnc3)C2)C1 c1(CC(=O)NCC2CN(C(c3cnc(C(F)F)s3)=O)CC2O)ccc(F)cc1F C1(NC(C(CCSC)O)=O)CC2(CCN(C(C34CC(C(C)C)(CO3)C4)=O)C2)C1 C12(C(=O)OC)CCCC1(C(=O)N(CCCNC(c1cccc(C3CC3)c1)=O)C)C2 c1(C(N2CC3CC(NC(C4ON=C(C)C4)=O)C3C2)=O)cccc2c1NCCC2 c1(OCCCC)ccccc1C(=O)NCC12CC1CN(C(c1conc1C)=O)C2 CC(C)C(O)C(F)(F)C(=O)NC1CN(C(=O)Cc2ccon2)C2CCCC12 c1(C(C)(C)C)cc(NC(=O)NCC2(C)CCOC2C2CC2)nc(Cl)n1 Cc1ncc(NC(=O)C(CC(F)F)N(C(=O)C(C)NC=O)C)cc1Cl C1(C(=O)NC(c2scc(C)n2)C)(NC(c2c[nH][nH]c2=N)=O)CCC(C)(C)C1 c1(-c2c(CNCC(=O)NCCc3ccccc3)cccc2)cc(F)c(O)c(F)c1 C1(C(N(CCOCC=C)C)=O)N(C(=O)CCC(C)(C)C)CCC1(C)C N1(C(=O)Cc2ccc(F)cc2F)CC2CCN(C(C34CCC(CC3)O4)=O)CC2C1 CCC(C)(O)C(=O)NCCN(C(C12CCN(CC1)C2)=O)Cc1ccccc1 Nc1cccc(C(=O)NCC(O)CNC(C2(C(O)C(F)(F)F)CCC2)=O)c1 C1(C(=O)NC(CC2CN(C(C3CC(OCC)C3)=O)C2)C)CC(=O)N(CC)C1 C#CC1(CNC(=O)C(C)(CO)NC(=O)C(CC)N(C)C)CCOCC1 C1(CNC(c2cc(F)n[nH]2)=O)CN(C(=O)CNC(C2CCCC2)=O)C2(CCC2)C1 Cc1cc(C(=O)NC2(CC)CN(Cc3cccnc3)C2)cc(Cl)n1 CC1CN(C(c2cc(Cl)c(Cl)n2C)=O)CCC1CNC(C1CCCSC1)=O C12(NC(COC3C(C)CCCC3)=O)CCC(CN(C(=O)C3=COCC3)C1)C2 C(C(CNC(=O)CN(C)C1CC1)S(C)(=O)=O)NC(c1cnc(CC)nc1)=O N1(C(CCn2nc(C)c(Cl)c2C)=O)CCCC12CCCSC2 N1(C(=O)CCc2ccc(Br)c(F)c2)CCOc2ccc(Cl)cc2C1 C1(N(C(CC2(CNC(=O)CCn3ccnn3)CC2)=O)C)CCC(C(=O)OC)C1 N1(C(C2(CCOCC)CCC2)=O)CC2CC(NC(=O)C(=Cc3c[nH]cn3)F)C2C1 C(CC(CC)C(=O)NCCC1CCCN1C(=O)CSCC(F)(F)F)=CC N1(C(C(C(C)=O)(C)C)=O)CCC2(CC1)COC(C(=O)Nc1nccnc1Cl)C2 C(N=c1[nH]c(=NCc2cccc(Cl)c2Br)[nH]c2cc[nH]c12)c1c(F)cccc1F N12CC3CCCC3(C1)C(=O)NOC(CC(C)C)C2=O.Cc1nncc(C(N)=O)c1C c1(C(=O)NCC2CCN2C(=O)C=CC(F)(F)F)cnc2[nH]ncc2c1 c1(NCc2cc(C)ncn2)nc2ccccc2n1-c1ccccc1 C(c1ccc(F)cc1)=CC(N1CC(NC(CCCc2ncc(C)o2)=O)C(C)C1)=O CC#CCCCC(=O)N(CC(C)NC(C1CCCC(=O)O1)=O)C c1(-c2cnc(NC)s2)cc(C)c(S(=O)(=O)NC(C)C(=O)N(C)C)cc1C c1(C(=O)NC(CC=C)CNC(=O)CN2CC3CC3C2)cccc2[nH]ncc12 N1(Cc2c(C)cccc2)C(=O)CN(Cc2ccc(OC(F)F)nc2)C1=O C[Si](C)(C)CCCNC(=O)C(C1CCN(C(=O)CC(=O)NCC(F)F)C1)F N1(C(CCN(C(=O)CCC(F)(F)F)CC)=O)CCCC(F)(F)CC1 C(=O)(C(C)Cc1cccnc1)NCCC(C)NC(C1(C#N)CCC1)=O C(C)(C)(C(=O)N(C)CC1(C(=O)NC2COC(Cn3cccn3)C2)CC1)OC c1(C(N2C(Cn3cc(CN(C)S(N)(=O)=O)nn3)CCC2)=O)ccc(Br)cc1[N+](=O)[O-] N1(C(CC(C)CN(C)C)=O)CCCC(C)(CNC(c2cccc(Cl)c2)=O)C1 c1(C(C)N(C)Cc2ccc(C(=O)O)s2)ccc(Cl)c(Cl)c1 c1(CC(=O)NCC(CC)(C)NC(c2cnn(CCF)c2)=O)cccnc1O C1(CC(=O)Nc2n[nH]cc2C2CC2)C2CCC(C2)N1C(=O)Cn1cnnc1 CC1CN(C(=O)CONC(C2CCCN2C(C)(C)C)=O)CC(C)(C)CO1 CCC(F)(F)CC(=O)N1CCC(CC(N2CCCC2CC2CC2)=O)CC1 c1(C(N(CCC(C)NC(c2cnn(C(C)C)c2F)=O)C)=O)ccccc1[N+](=O)[O-] C1(NC(C(C)OCC#C)=O)CCC(C)N(C(=O)COCCCC(C)C)C1 N1(C(Cc2cccc(OCC)n2)=O)CCCC(CC)(NC(=O)CCOC2CC2)C1 N(C(=NCC1CCOC1)NCC(C)(C)OCC1CC1)Cc1ccc(CC(C)C)s1 c1(C(=O)NCCC(CNC(C2C(=C)C2)=O)O)nc(O)nc(O)c1OC C1(c2nnnn2C)(NC(CCc2ccc(OC(C)C)cc2)C)CC12CCOCC2 c1(C(N(C2CCN(C(C3CCC(C)O3)=O)C2)CC)=O)c(C)nc2sccn12 n1(CCOC)nc(C(=O)N(C)CCN(C)C(c2ccc(Cl)cc2Cl)=O)ccc1=O c1(N)ncc(Cl)nc1Cl.c1(C(=O)Nc2cccc(N)c2)ccc(Cl)cc1OCCO N1(C(C(C)C)=O)CC2CCCC2(CNC(=O)C(C)Cc2cccnc2)C1 C(=O)(C1CCc2c[nH]nc21)NCC(C1CC1)NC(=O)CCCN1CCCCC1 Cc1cc(C(=O)NC(CNC(=O)CC2CC23CC3)C2CCC2)c2n[nH]cc2c1 C(CCCC(C)(F)F)NC(CN(C(=O)Cc1ccon1)CCOC)=O C1(NC(c2cc(C(N)=O)oc2)=O)CC(NC(=O)C(O)Cc2ccccn2)CC1O C1(C)(CNC(C(COC)OC)=O)CCCN1C(c1cc(C(F)(F)F)cs1)=O N1(C(COC)C)CCN(N2CCN(C3CCS(=O)(=O)C3)CC2)CC1 c1(C(=O)NCCCCC(C)NC(c2ccc(=O)n(CCF)n2)=O)cc(C#N)ccn1 n1(CC)cnc2c1=NC1=NCC(=O)NC=2N1.C1(SCC2CC2)CN2CCC1CC2 C1(C2CCN(C)CC2)(C(=O)NC2CC3(CN(C(c4cc(C)sc4)=O)C3)OC2)CC1 c1(C(N2CCC(NC(=O)C=CCO)CC2C2CC2)=O)cc2ccccc2cc1F CN1N=C(CC(=O)N2CC(NC(c3ccc(O)nn3)=O)CC23CCCC3)CC1=O c1(C(C(=O)NC(c2ccccc2)C)N(CC(C)OC)C)ccc(Br)cn1 CC1(NC(=O)CCOC2CC2)CCN(C(c2ccccc2-c2cc[nH]n2)=O)CC1 C=CC1(C(=O)NC2CN(C(c3cc(CC)no3)=O)CC2C(F)(F)F)CCOCC1 C#CC1(C(N(C)C[Si](C)(C)C)=O)CCN(C(=O)C(F)n2ccnc2)C1 c1(SC)ccc(Cl)c(C(=O)NC2CN(C(=O)Cn3nnc(=N)[nH]3)CC2C)c1 Cn1nc(Br)cc1C(N1CC(CNC(c2cn(CCF)nn2)=O)C(O)C1)=O CCCCCCCCCC(=O)NC1CCN(C(c2csc(C(C)=O)n2)=O)CC1O C=CC(CC)CC(=O)NCC1C2CN(c3nc(C(C)C)ncc3Br)CC12 c1(CSC)cccc(C(=O)NCC(C)CNC(c2cc(Cl)c(Cl)s2)=O)c1 CCC(C)(CCC(C)C)C(=O)N1CC(F)(CNC(=O)CN2CC(C)(C)C2)C1 CC1CCC(O)CN1C(C1CCCOCC1)C(=O)NC1COC1 CC1CN(C(c2ncn(C)n2)=O)CC1NC(=O)C(F)C1CCC1 CC1(C)CCN(C(c2ccc(F)o2)=O)CC1CNC(=O)C(F)(F)c1ccccc1 C1(C)(CNC(C(C)C#N)=O)CC(F)(F)CN1C(=O)CCc1ccc(Cl)nc1 CC(C)(CCCNC(c1ncccc1C1CC1)=O)NC(=O)CSCC(N)=O c1(SC)cccc(C(=O)NC2CCCN(C(=O)Cc3cc(C)nn3C)C2)c1Cl c1(C(=O)NCC(CCOC)NC(C2(O)COC2)=O)cncc(Cl)c1 C1(CC)CN(C(C2CCCNC2=O)=O)CCN1C(=O)CCN(C)CC c1(C(=O)NC(C)CCNC(c2cc3n(c2)CCOC3)=O)cnn2c(N)ccnc12 N1(C(c2c(CC)cns2)=O)CCN(C(=O)CC2CCCC(C)O2)CC1 N1(C(C(C)O)=O)CCc2c(CNC(=O)Cn3cc(Br)ccc3=O)cccc2C1 Cc1ncc(C(=O)NC(C)CN(C(=O)CCc2csc(=N)[nH]2)C)c(C(C)C)n1 N1(C(C(C(C)C)NC(c2ccccc2)=O)=O)CC2CC(C(F)(F)F)C2C1 C=C1CCC(C(N2CCC(C(=O)NC3CCN(C(C)C)C3=O)(C(C)C)C2)=O)CC1 c1(C(C(=O)NC(CNC(C2(COC)CC2)=O)C)C)c(C)noc1C C(=O)(CC(C)(O)COC)NC1C(NC(C2(CC)COC2)=O)CCC1 C(=O)(CCS(C)=O)N(C1CC(C(=O)NCC2(n3nccn3)CC2)C1)C c1(C(=O)NCCCC#C)ccc2c(c1)CN(C(c1ccoc1)=O)CC2 C1(CNC(C2(CC=C)CCOC2)=O)CC(C)(C)CN1C(=O)C1=C(C)CCC1 N1(C(C2C(=C)C2C(=O)OC)=O)CCN(C(c2cc(C)ccc2O)=O)CC1C C1(CCC)CN(C(c2nnn(C(C)(C)C)n2)=O)CCN1C(c1cnc(C)nc1)=O N1(C(C(C2CC2)OCC)=O)CCC2(C=C(C(=O)NC(C)(C)CC3CCCC3)C2)C1 C(C(F)(F)C(F)F)CCn1cc(C(N(C(CCc2onc(C)n2)=O)C)C)nn1 C=C(Cl)CCC(=O)NC1CN(C(C2(COC)CCOCC2)=O)CC1C c1(C(=O)NCC(CNC(=O)CCOCC(F)F)OC)cnn(C)c1Cl c1(C(=O)NC2(CN(C(C3CC(C)OCC3)=O)C)CC2)cnn(C)c1C#N N1(C(CC=CCC)=O)CC2CCCC(NC(c3cnc4ccnn4c3C)=O)(C2)C1 c1(C(=O)NCC2(CCNC(C(C(C)O)N(C)C)=O)CC2)sc(C#N)cc1Cl c1(C(=O)NC2CN(C(CCCOCC)=O)C(C)C2)cc(C(F)F)ccc1Cl Cn1c2c(ccc1=O)C(NC1CCNCC1(F)F)CCC2 O([Si](C)(C)C(C)(C)C)C(CC)CNc1ccc(Cl)cc1Cl C1(CNC(CS(=O)(=O)NCC)=O)CC2(CCC2)CN1C(c1c(Cl)cnn1C)=O N1(C(CCCNC(=O)OC)=O)CCC2CN(C(C3(C)CCC3)=O)CCC2C1 Cc1ccn2ncc(C(=O)NC3CC4CCC3N(C(C3(O)CCSC3)=O)C4)c2n1 N1(C(c2c(C)sc(Cl)n2)=O)CC2CCCC(NC(=O)C=CC3CCCCC3)C2C1 N1(C(c2c(CCC)occ2)=O)CCC(C)C(CNC(C2(CSC)CCC2)=O)C1 C(=O)(CC(C)(C)C(F)(F)F)N1C(C)(CNC(c2ccc3c(c2)NCC3)=O)CCC1 c1(SCC(N2CCC(NC(c3ccn(C(C)C)n3)=O)CC2)=O)ccc(F)c(F)c1 N1(C(C(COCC=C)C(C)(C)C)=O)CCC(C2CC2NC(=O)CCC(N)=O)CC1 Cc1ccc(S(=O)(=O)NC2CCC(NS(=O)(=O)c3cccc(Cl)c3F)C2)c(F)c1 N1(C(CCCNC(=O)OCC)=O)CCCC(C)(NC(=O)CC(COC)CC)C1 C1(NC(Cc2scc(C(C)=O)n2)=O)CN(C(C2C3COCC23)=O)C2(CCCC2)C1 N1(C(CN(C)Cc2ccccc2)=O)CC(NC(c2csc(CO)n2)=O)CC(O)C1 c1(C(=O)NC2(CCCNC(Cc3c(C)ocn3)=O)CC2)ccc2sccc2c1 C12CN(CCC1CO)C(=O)C=CC(=O)O2.C(CCC=CC(=O)NCO)=C(C)C.C(C)(C)=C Cc1nc(C2CC2)[nH]c1C(=O)NC(C)CCCCNC(=O)CC1CCCC12CC2 C1(NC(CCN(CCC)C)=O)(CO)CCCN(C(C2(C#N)CC2(C)C)=O)C1 C1(N(C(CC)Cc2ccc(C)cc2)CC)CC(CC(=O)OC)CN1 c1(-n2ccc(C(=O)NC3CCN(C(C4C(C)C4C)=O)C3C)n2)ccc(Cl)cc1F Cc1cc(F)ccc1C(N1CCCC(C(C)NC(=O)C2=COCCC2)C1)=O C1(CC=C)(NC(c2cccc(CNC(=O)CN3CSCC3=O)n2)=O)CCCCC1 C1(C(=O)NC(CNC(CCNC(=O)NC)=O)C)CCCN1C1CCCCC1 CCCCC(C)C(=O)N1CCC(C)C(CNC(c2cnc(O)cc2C)=O)C1 Cn1nc(C(=O)NC(C)(C(=O)NC2CC(O)C(O)C2)C2CCC2)cc1O C(=O)(CCCC(=O)NC(C)CCC(N1CCOCC(C)C1)=O)OC Cc1onc(C(=O)NC2CN(Cc3ccnc(F)c3)CC2F)c1C c1(C(=O)NC2(C3CCN(c4cc(C)ncn4)CC3)CC2)ccc2cnn(C)c2c1 c1(CC(=O)NC)cccc(NC(=O)NCC(N2CC=CC2)C)c1 C(CN=c1[nH]cc2ncnc-2[nH]1)c1c(C)non1 N1(C(C(C(C)C)O)=O)CCC2CC(NC(c3cnn4ccncc34)=O)CCC2C1 c1(C(=O)NC2CC(CNC(C3C(C#C)C3)=O)C2)cc(C)c(Br)cc1C C1(CNC(c2cc(CCC)n(C)n2)=O)CC2CN(C(=O)C=Cc3cscn3)CC12 C(=O)(CCN=[N+]=[N-])N(C1CCCC1)CC(=O)NC(c1cccs1)CC CCC(CC)(CC(=O)OC)C(=O)N1CC2CC(CNC(c3ccsn3)=O)CC1C2 C1(C)(CNC(C(C(C)C)O)=O)CN(C(=O)CCc2cc(Cl)cs2)CCO1 C1(CCC(=O)OCC)CCC(NC(C2CCN2C(=O)Cc2cnoc2)=O)C1 N1(C(c2c(Cl)cnc(C)n2)=O)CC(NC(=O)Cc2cn(C)cn2)C2(CCCC2)C1 C1(c2nnnn2C(C)C(=O)OC)(NCCCCCC)CC2CCC(C1)S2 C1(C(N2CCC(COC)(NC(=O)CC(O)CN(C)C)C2)=O)Cc2ccccc2C1 c1(C(=O)NCC2CN(C(CNC(=O)OCC)=O)C(C)C2)c(N)ccc(F)c1C N1(C(CCCCC(C)=O)=O)CCC2C(CCCN2C(c2coc(CO)c2)=O)C1 c1(C(N2CC(CNC(CNC(C)=O)=O)OCC2)CC)ccc(F)cc1F C1(C(N2C(CN(C(=O)CCC3CC3)C)CCC2)=O)CC2CCC1CC21OCCO1 C(=O)(CC1OCc2ncccc21)NCCCNC(C=C1CCC(C)CC1)=O c1(C(C(c2ccc3c(c2)CCC3)C#N)=O)ccc2cc(Cl)ccc2c1 C(=O)(C(F)(F)C(F)F)N(CCNC(c1c(C)nn(C2CC2)c1)=O)C1CC1 O=C1NCC2(CO1)CN(C(=O)C(O)Cn1cncn1)C2.[nH]1ccccc1=O N1(C(c2c(CC)onc2C)=O)CCC2C(CCCN2C2CC2)C1 C(=O)(C(CCCC(C)C)N1CCCC1Cc1cnn(C)c1)NC(CC)C C1(CC(=O)N(CC(C)NC(=O)C(C)(C)N(C)C)C)CC1C1CC1 N1(C(C(=O)NC)=O)CCOCC(C(=O)O)C1.C1CC(C(F)F)c2ccc(cc2)O1 C(=O)(C(CCC)C(=O)OC)N(CC(C)NC(c1cnc(CCC)s1)=O)C c1(NC(C)=O)cnc(O)c(C(=O)NC2CCN(C(c3cc(F)cs3)=O)C(C)C2)c1 N#Cc1cccc(NC(C2CCCCC2NC(c2ccccc2CO)=O)=O)c1Cl c1(NC2CCC(NC(c3c(C)ncs3)=O)C2)nc(C(C)(C)C)nc(=N)[nH]1 n1(C(C=C)C)nc(-c2ccnc(Cl)c2)nc1C1CCN(C)C1=O CC1CN(C(=O)Nc2ccc(CN3CCN(C)CC3)cc2)C(C)(C)C1 C1(CNC(c2cc(C)n(C(F)F)n2)=O)CN(C(=O)CC2CC=CC2)CCCO1 C1(NC(CCc2ccn(C)n2)=O)CCCCC1CNC(=O)CC1CCCCC1O C(=O)(C(C(C)O)N(C)C)NCc1c(C(N(CC(C)C)CC(N)=O)=O)n[nH]c1 Cc1nc(C)n(CC(=O)NCC2CCN(C(c3ccc(CC(C)C)nc3)=O)C2)n1 C(CCCC(=O)NC1CC1NC(=O)CC1CC2(CC2)CO1)OCC CC(CN=C(NCC1CCC1)NC(C)C1CC1)Oc1ccccc1 C(=O)(C1CCCn2nccc21)NC1(C)CC(NC(c2ccc(F)c(O)c2F)=O)C1 C1(NC(c2cnn(CCC)c2C)=O)(CNC(=O)C2=CCCC2)CC2CCC1CC2 c1(OC)ccc(C(N2CCCC2CN(C)C(c2ccsc2OC)=O)=O)cc1F N1(C(c2n[nH]c3c2CN(C(CNC(=N)N)=O)CC3)=O)CC2CC3CC(C2)CC1C3 C1(C(N(CC(C)CNC(C2CCCC23CCC3)=O)C)=O)CNC2=C1CCCC2 C1(C(N(CCCNC(=O)CC2CC(F)C2)C(C)C)=O)CCC(=C2CCC2)CC1 N1(C(Cc2n(C)nnc2)=O)CCCC2C(NC(C3CC4(CSC4)C3)=O)C(C)(C)C12 C1(NC(=O)C2=COCCO2)CC2(CCN(C(c3n[nH]cc3F)=O)C2)C1 c1(C(=O)NC(CC)CNC(=O)CC2CC2(C)C)coc(C2CC2)n1 C(=O)(CCC1CCc2ccccc21)NCC1(C)CCCN1C(=O)CNS(N)(=O)=O Cc1cc(F)c(NC(C2CCCN2C(c2ccccc2CO)=O)=O)cc1[N+](=O)[O-] N1(C(C2CC(=O)NC2)=O)CC(C2CN(C(=O)CC3CCNC(=O)C3)C2)C1 Cc1ncc(Cl)cc1NC(C1(NC(c2cnccc2C)=O)CCN(C)C1)=O CC1CN(C(C2(CO)CC2)=O)CC(CCNC(c2n[nH]cc2Cl)=O)O1 Cc1c(C(=O)NCC(C)NC(=O)CSc2nnc(-c3cccs3)n2C)cncc1Cl c1(C2(C(c3nnnn3C)NCCc3n(CC)cnn3)CC2)ccc(F)c(F)c1F C(=O)(CCCC(F)(F)C(F)(F)F)N1CC2(N(C(CC(CC)SC)=O)CC2)C1 c1(C(=O)NCC(CN(C(C(CC(C)C)OC)=O)C)C)ccc(C)c(Br)c1C C(=O)(C(C(C)C)C1CCC1)NCC1(NC(C(C)NC(=O)OC)=O)CCOC1 c1(NC(C2CCC2C(c2ccccc2)c2ccccc2)=O)cnnc(I)c1 CCC(CC)CCC(=O)NC(CC)CC(=O)N(CCCN1CCCC1)C c1(C(=O)NCC(CC=C)NC(=O)C(C)OC)ncc(C(=O)OC)cc1Cl C(C(CNC(c1ccnn1CCCC)=O)C(F)(F)F)NC(C(C=C)O)=O c1(C(N2CC(N(C)C(c3cc(Cl)cn3C)=O)C(F)C2)=O)cc2n(c1)CCC2 c1(C(=O)NC(C2CCN(C(c3c(C)nc(CC)o3)=O)C2)C)cc([N+](=O)[O-])oc1C c1(C(C)(C)C)cccc(C(=O)NC2(C)CC(NC(C3CCC(O)C3)=O)C2)n1 C1(CNC(=O)Cn2cccc2)C(C2CC2)CCN1C(=O)Cc1cnns1 C1(C(C)CCO)CCCCN1C(=O)Cn1cc(CCN(C(C)(C)C)C)nn1 N1(C(c2csc(C)c2C)=O)CC2(CCN(C(=O)C(C)(C)c3cnco3)C2)C1 C1(N(C(CC(C)N(C)C)=O)CC2CC2)CCN(C(=O)C2=CCSC2)CC1 c1(OCC(=O)NC(CC)CNC(=O)CNC(=O)OC)ccccc1C C=CCCCCC(=O)N(C1CCCN(C(c2csc(C(F)F)c2)=O)C1)CCO C(=O)(CCCC(C)(C)C#N)N1CC(OC)(CNC(C2CN(C(C)=O)CCO2)=O)C1 c1(CN2C(C(N3C4CCC3CC4)=O)C=CC2)cccc(Br)c1Br c1(C(N2CCOCC2CCC#N)C(=O)NCCC#N)cccc2c1nnn2C c1(NCc2c(F)ccc(C(C)(F)F)c2)cc([N+](=O)[O-])ccc1C#N C(=O)(C(CCOCC)NC(=O)C(C)NC=O)NCC1N(CC)CCC1 CC(C)CC(CC(=O)NC1COCCC1O)NC(=O)C(C)c1ccco1 Cc1sc(O)nc1C(=O)NC1CC(C(=O)NC(C)CCC(C)C)C1 C(CCC(C)C(=O)N1CC(C(C)NC(C2C=C2C)=O)C1)OC C1(C(=O)NCC(CO)NC(C2CC(=C3CCC3)C2)=O)(OC)CCC1 c1(OC)ccc(F)c(C(=O)NC(CNC(c2cc(Cl)cc(Cl)c2)=O)CO)c1N C(CCC(O)C(=O)NCC1(CN=[N+]=[N-])CC1)NC(c1cnn(C)c1Cl)=O C12(O)CCN(C1)C(=O)CC1(CCC1)OC2C.C(C(=O)NCO)N(CCOC)C C12(C(=O)NCCN(CCCN(C)C)C(c3ccc(F)cc3F)=O)CC1COC2(C)C N1(C(c2c(OC)ccnc2)=O)CC(C)(C)CC1CNC(=O)C(C)C(C)O CC1CN(C(c2cccc(O)n2)=O)CCC1CNC(=O)CC(C)(C)C1CC1 C1(C(=O)NCC(C=C)(C)C)C(CC)CCN1C(=O)C(C1CC1)OCC C1(c2ccccc2)(SCC=C(C)C)CCCC(=O)N1.S1(=O)(=O)CCCN1 C(=O)(CC1=CCN(C)CC1)NC1CN(C(C=C(COC)C)=O)C(C)CC1 N1(C(C2(C)CCN(C)C2)=O)CCCC(NC(=O)CSC(F)F)CC1 c1(OC)cc(C(=O)NC2(C)CCCN(C(c3ccc(C)nc3)=O)C2)cc(Br)c1 NS(=O)(=O)CC(=O)NCC1CN(C(c2csc(-c3ccoc3)n2)=O)CCO1 n1(CC)cc(C(=O)NC(C)(C)CNC(c2coc(OC)c2)=O)c(C(C)(C)C)n1 c1(C(N2CC(c3cn(C4CCOC4)nn3)(NC=O)C2)=O)c(F)cc(Br)cc1F c1(-c2n(C)c(-c3ccc(Br)cn3)nn2)ccc(S(=O)(=O)N2CCNC(=O)C2)cc1 C1(NC(CC2(C)CCS(=O)(=O)N2)=O)CC2CCC(C1)N2CC(F)(F)C(F)F c1(C(=O)NCCC2CCC(NC(C3CCC=CCC3)=O)C2)ccnn2ccnc12 C1(CC)CN(C(C2CC2c2ccoc2)=O)CCN1C(c1ccc(SC)s1)=O c1(CC(=O)NC(C2(CNC(c3[nH]cc(CC)c3)=O)CC2)C)ccnc(F)c1F CCCC(F)(F)C(=O)N(CCCCCC(=O)Nc1cnc(SC)nc1)C N1(C(C(C=C=C)C)=O)CCC2(CC1)C(NC(c1csc(Cl)c1)=O)CS2(=O)=O CC(C)CCCCC(=O)N1CC2(CO)CC1(C(=O)NCC1(O)CC=CC1)C2 c1(CC(C(=O)N(C2CCN(C(c3cnc(OC)s3)=O)C2)CC)O)ccc(F)cc1 c1(N2CC(O)(CCNC(c3c(C(C)(C)C)ocn3)=O)C2)ncnc2c1CCO2 C1(C(=O)NCC2CN(C)C(=O)C2)CN(C(=O)C#CC2CCC2)CC12CC2 c1(CC2CCN(C(C(C(C)C)NC(C3CCCCC3)=O)=O)C2)cccc(C#CCO)c1 C1(SC)CN(C(=O)CC2CC2)CC1n1cc(CCN2CCOCC2)nn1 c1(C(N(CCC(C)NC(C2CCCCS2)=O)C)=O)cccc2ccsc12 c1(C(=O)NCC(CC)NC(c2cnc(NC)cn2)=O)csc([N+](=O)[O-])c1 C1(C)(NC(c2c(C(C)NC(=O)CCN3CCC3)noc2)=O)CN2CCC1CC2 C=CCCCCC(=O)NCCC1C(C)CCCN1C(c1cc([N+](=O)[O-])n[nH]1)=O C1(C(=O)NCC2C(NC(c3cnc(O)c(Cl)c3)=O)C2)CC(C2CC2)=NO1 C1(CNC(C2(NC(c3c(C)scc3)=O)CCC2)=O)CC(C)OC(C)C1 C1(C)(NC(C)C(C(=O)OC(C)(C)C)N(C)C)CCC(C)(C)CC1 Cc1cc(N)c(C(=O)N(CCCCNC(=O)C(O)CCC(C)C)C)c(F)c1 C=CC(C)(O)CC(=O)NCC(C)(CNC(c1sc(C2CC2)nc1C)=O)OC c1(C(N(C2CN(C(=O)COC3CCC3)C2)C)=O)c(F)cc(Br)c(F)c1F C(=O)(C(C)N(OC)C(=O)C1(CCNC(=O)Cc2cncn2C)CC1)OC CC(C)(O)C(F)(F)C(=O)NC1COC2C(NC(c3n[nH]cc3[N+](=O)[O-])=O)COC12 N1(C(c2c(C)nsc2C)=O)CC(C(N2CCC(C)(C)C2C)=O)C(F)(F)C1 C1(C(N2CCC(C(C)Nc3ncc(Br)cn3)C2)=O)CN(C)CC(C)O1 CN=c1[nH]cc(C(N2CC(NC(=O)C(c3ccccc3)C)C(O)C2)=O)o1 C1(CC(=O)NCC(F)F)CCCC(NC(=O)CC2CCOCC2)C1 C1(CNC(=O)CCc2ccc[nH]2)OCC2CCN(C(=O)C(Cl)Cl)CC12 c1(CC)ccc(CC(=O)NC(C)CCNC(c2ccc(F)o2)=O)cc1F N1(CCN(C(C2CC(CC)C2)=O)C)CCN(C(=O)C(C)NC2CC2)CC1 C1(NC(C2CC2C(F)F)=O)CCC2(CC1)CN(C(C1CC13CCCC3)=O)CCO2 C(=O)(C1=C(CC)OCCC1)N1C(CC)CN(C(C2CN(CC(F)(F)F)C2)=O)CC1 CC(C)C(C(=O)N(C)CC1(NC(C2C(F)(F)C23CC3)=O)CC1)n1cc(Br)cn1 C1(CNC(C2(C)C=CCCC2)=O)CCCCCN1C(c1ccc[nH]1)=O c1(CC)cc([N+](=O)[O-])ccc1NC1CN(C(C2CC23CCOC3)=O)C1 c1(OC)cnc(F)c(C(=O)NCCCC(C)NC(=O)C(C)(C(C)C)OC)c1 C1(C(=O)OCC)CN(C(c2ccnn2COC)C)CC1(C)C(F)F c1(C(=O)NC2CC3CN(C(C(C)(O)C4CCC4)=O)C2C3)ccn2ncnc2c1 c1(C(N(CC(CN(C(=O)C(F)C2CCOC2)C)O)C)=O)nc[nH]c1C(F)(F)F N1(C(c2c(CCC)n[nH]c2)=O)CCCC(C(N2CCC(F)(CF)C2)=O)C1C N1(C(CNC(CNC(C)=O)=O)=O)CC(N(C)C(c2ccc(C)nn2)=O)C(F)C1 c1(C(C(=O)NCC(=C)C)N(CCC(C)C)CCC#N)cc2ccnc(Cl)c2s1 C1(NC(C(c2ccnn2C)C)=O)CN(C(c2nc(Cl)ccc2N)=O)CC1C1CC1 C1(C(N(C(CCNC(c2cn(CCC)nc2)=O)C)C)=O)CC2CCC(C1)C2O C1(O)(CNC(CCOCC(C)C)=O)CCN(C(C2CCCC23CCC3)=O)CC1 C(CCC(F)(F)F)(C(=O)NC1CC1)NC(=O)CCOC1CNC1 C12(C(=O)NC3C4CN(C(C(C(C)(C)C)O)=O)CC43)CCC(C(F)(F)F)(CC1)CC2 c1(C(=O)NC(CCNC(CN(C2CC2)CC)=O)C)cc(Cl)cc(Cl)c1[N+](=O)[O-] N1(C(CCOCC#C)=O)CCN(C(c2ccc(N)cc2OC)=O)C(C)C1C C1(C(=O)NCC2(C)CCN(C(=O)Cc3nn(C)cc3Cl)C2)(OCC)CCSCC1 C(CCCCC(=O)N1CCC(C(C)NC(=O)CCc2csc(=N)[nH]2)C1)OC C1(OC)CCNCC1C(=O)NCC(O)CCc1ccccc1 c1(CN2C(C)(C(=O)Nc3cccc(NC(=O)OC)c3)CC2)cc(F)c(F)c(F)c1 c1(OC)ncc(C(N2CCCc3c(CN)cccc32)=O)c2ccccc12 C(CC1CC1)(C(=O)NCC(O)CCNC(c1csc(CC(C)C)n1)=O)OC Cc1cc(Cl)cc(Br)c1NC(C1CC(F)(F)CN1Cc1cc(Br)cc(Cl)c1F)=O C1(NC(C2CCCN(CC)C2)=O)CC2(CCN(C(c3cc(=O)n(C)o3)=O)C2)C1 C(C)(C)(CC(F)C(=O)NCCOC(=O)C1CC1)NC(C1C(C)CC(=O)CC1)=O N1(C(C(COC)N(C)C)=O)CCN(C(c2cc(OC)ncn2)=O)CC(O)C1 Cc1ccc(N)c(C(=O)NC2CC(CNC(C3(CO)CC3)=O)C2)c1F C1(CCC(=O)OC)CC(CO)N(C(=O)NCCC(C(=O)O)c2ccc(F)cc2)C1 N1(C(CSCCC)=O)C(CNC(c2cnn(C)c2COC)=O)CC2COCC12 N1(C(C(C)C)=O)CCN(C2CCN(C(c3csc(CC(F)F)n3)=O)CC2)CC1 c1(OCC)ccc(Cl)cc1CCN1CCC(OC(c2[nH]c(C)cc2C)=O)C1 CCC(CC(=O)NC(C1CCN(C(=O)Cc2sc(S)nc2C)C1)(C)C)SC N1(C(c2n(C)nnc2)=O)CCC(C2CN(C(c3ccc(C4CC4)cn3)=O)C2)C1 c1(CC(C(=O)Nc2n(CC)nc(CN)c2)N)nccc2ccccc12 c1(C(N2CC(O)(C(C(=O)NCC3CS(=O)(=O)C3)F)C2)=O)c[nH]nc1[N+](=O)[O-] CC1=C(C(=O)NCC2CCN2C(c2cnc3n2CCCC3C)=O)S(=O)(=O)CCO1 c1(OC)cccc(C(N2CC(C(O)C(=O)NC3CC4C=CC3C4)C2)=O)c1 Cc1ccc(C(c2cnccc2Cl)NC2CC(NC(=O)OC(C)(C)C)C2)cc1F C1(CC(=O)N(C2CCN(C(c3cc(C)n(C(C)C)n3)=O)C2)CC)CC2CCC1C2 CCC(CCC(=O)NCc1cn(CCNC(c2ccc(Cl)cc2NC)=O)nn1)OC CCCC(C(=O)N(CC(C)C(=O)NCCOC(C)=O)C)OC C1(C(=O)NC(c2ccncn2)(C)C)CCCN(C(=O)C=C2CCCCC2)C1 CCC(CNC(C1CCCN(C(C2CC=CCC2)=O)C1)=O)C(C)(F)F N1(C(Cc2c(C)noc2Cl)=O)CC2(CCCC2NC(=O)Cn2nnc(=N)[nH]2)C1 CN=c1cc(C(=O)NC(C(=O)NCCc2ccsc2)C(C)(C)C)cc[nH]1 CC(CC(=O)NC1(C2CCCN2C(=O)CN2CCCC2=O)CC1)c1cnn(C)c1 C1(OC)CC(NC(=O)CCc2ccoc2)CN(C(c2coc(C(F)(F)F)c2)=O)C1 c1(C(=O)NCC2(NC(C(CC(C)C)O)=O)CCC2)cc2c(s1)CCC2=O C(CC(C)N=c1[nH]c(N2CCCCCCCC2)nc2ncn(C)c12)SC C=CCC(C(=O)NCCCCCNC(c1ccnc(OC)c1)=O)C(C)C Cc1cocc1C(=O)NCC12CC(NC(=O)C(C)NC(N)=O)(C1)C2 C123CCC(CC1n1cc(nn1)-c1ccc(cc1)N2)C3.C(=O)C1CC1.CCS c1(C(N2CCC(C(=O)Nc3nnco3)C(O)C2)=O)c(O)c(Cl)cc(Cl)c1Cl S(=O)(=O)(c1cccs1)NC1CCN(Cc2cc(OC(CC)C)ncc2)CC1 C#CC1CCCCN1C(C1(C)CN(C(=O)CC2CCC(C)(C)O2)CC1C)=O C(C(C)(C)C1=CCC(C)(C)CC1)NC(C(c1cn(C)nc1)(C)C)=O N1(C(C2CN(C(C)=O)C2)=O)CCC2C(C1)NC(=O)CN2C(C1CCC12CCC2)=O CN=c1[nH]c(=NCc2nncs2)[nH]c(=NCc2ccc(F)cc2Cl)[nH]1 c1(C(N2CC3CC(CNC(C45CC(CO4)C5)=O)C3C2)=O)c(F)ccc(F)c1F N1(C(C(n2c(C)ncc2)C)=O)CC(C(N2CC3CC3(CO)C2)=O)C(C)C1 C12CN(C(=NCCCCl)NCC1N(C)C)CCS2.c1(CC)cc(Cl)ccc1Cl c1(C(=O)NC2(C)CC2)cc(C2CC2)nc(O)c1.N12CCN(CC1)C(=O)CN1CC2C1 CP(C)(=O)c1cnn(CC(=O)NCC(C)(C2CC2)NC(c2sccc2Cl)=O)c1 c1(C(=O)NCC2CN(C(CCc3cnc(C)o3)=O)C(C)C2)cccc2ccoc12 c1(CC(=O)NC(CC)COC)ccnc(O)c1 C(CC(C(C)(C)C)NC(c1cc2n(n1)CCC2)=O)N(C)C(C1CCC2(CC2)C1)=O C(=O)(C(C)(O)CC=C)NC1C(C(N(C(CC#C)C)C)=O)CCCC1 C1(CNC(C=CC)=O)CCC12CCN(C(C1CC1CC(=O)OC(C)(C)C)=O)CC2 N1(CC=CCC2CCN(C(=O)C(O)CCn3cncn3)CC2)CC(F)(F)C(F)(F)C1 C(=O)(C1=NOC2(CCOC2)C1)OCc1ncn(C)n1 N1(C(C(C)c2cc[nH]n2)=O)CC2CC(C1)N2C(=O)CC1CCCSC1 c1(C(=O)NCC2C3CN(C(c4c(C)ccs4)=O)C2C3)cccc(Cl)c1[N+](=O)[O-] C1(CCF)C(=O)N1.C(C(=O)NC1(C(=O)N(C)C)CC1)=CCOC Cc1cc(=NCC2CCOC2C)[nH]c(=NCc2cnc(Br)cc2C)[nH]1 C#CC1(NC(C2(CCNC(C3CCCCC3C)=O)CCCC2)=O)CCCCCC1 c1(C(=O)NCC2(C)CN(Cc3ccccc3)CCO2)ccc2ncoc2c1 C1(CNC(C2(CNC(CC(C)OC)=O)CC(C)(C)C2)=O)OCCCC1(C)C N1(C(C(CCC)C(C)C)=O)CCC2(CCCN2C(c2cn(C)nc2OC)=O)CC1 N1(C(c2nc(CCOC)oc2C)=O)CC2CN(C(=O)CCCC(C)C)CC2C1 CCC(C)C(C(=O)NCC(CCNC(C1(CCOC)CC1)=O)OC)OC C#CCCCCC(=O)N(C)Cc1ccccc1CNC(=O)C(CC)C(=O)OC C1(C(c2nnnn2C(C)C)(CC)NCc2nc(Br)sc2C)CCC2CC1C2(C)C N1(CC(=O)NCC2CC(O)CN2C(=O)C(O)CC(F)(F)F)Cc2ccccc2C1 c1(C(=O)NC2CCN(C(c3cncc(O)c3Cl)=O)CC2)noc2c1CCCCC2 N1(C(CCCC#C)=O)CC(NC(=O)C(CC)CCc2ccccc2)CC2(CC2)C1 CCC1=NOC(C(=O)NCC(CC2CC2)C(=O)NC23CCC(CC2)C3)C1 N1(C(C(C)O)=O)CCn2ncc(S(C)(=O)=NC(=O)C(C)CS(C)(=O)=O)c2C1 C1(C(N2C(C)(C(=O)NC)CCC2)=O)CCN(C(=O)CC2(N(C)C)CC2)C(C)(C)C1 CC1(C(N2CC(O)(CNC(=O)C3=C(Cl)CCC3)C2)=O)CC(C2CC2)=NO1 c1(C(=O)NC2C(C(C)C)N(C(C3(F)CCOC3)=O)CC2)ccc2nccnc2n1 c1(CNC(=O)OC(C)(C)C)cc(F)cc2nc(S)[nH]c12.C1CCNCCC1 CC(C(=O)NOCC(N1CCCC(C(N)=O)C1)=O)N(C)C CCCC(C)(CCC)C(=O)N1CCCOC(CNC(C2OCCC2C)=O)C1 C(CC(C(=O)N(C)C)N1CCC(C(=O)NCc2cccs2)CC1)SC c1(CC(=O)N(C2C3CC(OC)C(C3)C2)C)ccc2c(c1)CCC2 N1(C(C2CC(C)OCC2)=O)CC2(C1)CN(C(c1cnn(C(C)(C)C)c1)=O)C2 O=C1CC(CC(=O)NCCCNC(C2C3CC(F)(F)CC23)=O)CCCN1 C(=O)(C(C)(F)C(C)(C)F)N(CCNC(c1cc(C)sn1)=O)C C#Cc1cn(C)nc1C(=O)NC(C(=O)NOCC1CC2C=CC1C2)c1ccco1 c1(C(N2C(C)(CNC(=O)C(O)C(F)(F)F)CCC2)=O)cnn2c1OCCC2 C(CN=c1cc(C(F)F)nc[nH]1)C1CCC(NC(c2ccn(C(F)F)n2)=O)C1 c1(C(=O)NC(C)(C)CNC(c2ccc(Cl)o2)=O)ccc2c(C#N)c[nH]c2c1 c1(CC)cc2c(NC(c3ncsc3-c3ccccc3)=O)ncnc2s1 c1(OC)c[nH]c(C(=O)NCC2CN(C(=O)C(C)N(C)C(C)=O)CC2C)cc1=O C=C1CC2(C1)CC(C(=O)N(CC(C)CNC(=O)CC1SC(=N)NC1=O)C)C2 Cc1cc(N)c(C(=O)NCC2CCCCN2C(=O)CC(F)(F)C(C)C)nc1C c1(OCC)cc(N(C)CC2CCN(C(=O)C(C)NC(N)=O)CC2)nc(C)n1 c1(N(C(=O)NCC(C)OC)C)sc2nnc(S)n2c1C.N1(C=O)CCCC1 c1(CC(=O)NC2CC(CNC(C3CC3(F)Cl)=O)C2)ccc(O)cc1 c1(OC)ncc(-c2cnoc2)cc1-c1ccoc1 C1(SC)CCCCC1N=c1[nH]c2c(c(=NCCc3cc(C)ccc3Br)[nH]1)COC2 N1(C(C(C)OCCN(C)C)=O)CCCC2(CNC(=O)CC3CC3)CCCC12 C#Cc1ccc(C(=O)NCC(C(=O)NCCCC(=O)NC)C(C)C)cn1 CC1C(C(=O)NOC2CCCC2)CCN1C(c1nc(=N)cc[nH]1)=O c1(CC(N2CCC(NC(CCS(C)=O)=O)CC2)=O)ccc(F)cc1F CC(C)(C)CCC(=O)N1CC(F)(F)CC1C(N1CC(n2ccnc2)C1)=O C1(NC(C(CC)OC)=O)CCC2(CC1)CC(NC(=O)CCn1cnnn1)C2 n1(CCNC(C(=O)N(C)C)=O)cc(C(C)(C)NC2CC(F)C2)nn1 C12(NC(Cc3c(Cl)cn(C)n3)=O)CCN(C(=O)CC3(C)CCC3)CC1C2 c1(CCNC(=O)NCC2CC3(C2)OCCO3)nnc2n1CCNC2=O C1(C)(C(C)C)CCN1C(=O)CCCC1(NC(C2(C)CCCC2)=O)CCC1 N(C1COc2ccccc21)C(=O)Nc1nc(C(F)(F)F)c(I)s1 c1(C(C(=O)NCCCN(CCCNC(C2(C(F)F)CC2)=O)C)C)ccc(F)cc1 C(=O)(CC(C)C(F)(F)F)NC(CCCNC(CCN1CCN(C(C)C)CC1)=O)C C=CCCC(C(=O)NCC1(C(N)=O)CC1)NC(c1cnn[nH]1)=O N1(C(=O)Cc2cccs2)CC2(CCN(CC(O)COc3ncc(Cl)cc3Cl)C2)C1 c1(C(=O)NC2(CCCC(=O)NCC3ON=C(C)C3)CCC2)ccc(C#N)c(C)c1 C(C)(C1CCCCC1)=CC(=O)NC1C(CNC(CNS(CC)(=O)=O)=O)C1 c1(C(=O)NC(CN(C(=O)C(F)Cc2ccccc2)C)(C)C)cc(N)c(O)c(F)c1 c1(NC(CCSCC)C)ncc(S(=O)(=O)NCCC(C)(C)CO)cc1Cl CC1CCC(CC(=O)NC(CC2CCC2)C(=O)NC2CC(n3cncn3)C2)CC1 N1(C(c2c(C)coc2C2CC2)=O)CCCC(NC(c2c[nH]nc2C(F)F)=O)CC1 C(C(C)C(F)C(=O)N(C)Cc1nccn1CC)NC(CC)=O CC(CN(C)C(c1ccc(C#N)o1)=O)C(=O)Nn1ccnn1 c1(C(=O)OC)ccc(NCc2cn(CCCNC(C3CC(O)C3)=O)nn2)cc1 C(CCCC(=O)NC(C1CN(C(=O)C=CC(C)C)CCO1)C)NC(C)=O C1(C(=O)NCC(C)NC(C(C)SC(C)C)=O)CCCSC1 c1(OC)ccc([N+](=O)[O-])c(NCCNC(=O)NC2(C)CCCO2)c1F c1(C(N(CC(=O)NC2CC2CNC(=O)OC(C)(C)C)C)=O)ccc(Cl)nc1 c1(CN2CCC(NC(CCC3CC(OC)(OC)C3)=O)C2)cccc([N+](=O)[O-])c1 C1(N(C(C(F)=CCC)=O)C)CCCC2CN(C(c3ccc(Cl)cc3)=O)CC12 c1(C(C(=O)N(CCCOCCN(C(C(F)OC)=O)C)C)N(C)C)ccc(Cl)cc1 n1(CC)nc(C)c(C(N2CCC3C(NC(=O)C4=COCCO4)C23)=O)c1C C(=O)(C(CNC(C1CCC1OC(C)=O)=O)C(C)(C)C)NC(C1(OC)CCC1)C c1(C(N(CC#N)CC#N)=O)[nH]nc2ncc(-c3ccc([N+](=O)[O-])cc3)cc12 C(=O)(C(O)C(C)(C)CO)OCC1CCN(C)CC1 C1(F)(CNC(C(C2CC2)SC)=O)COCCN(C(=O)Cn2ccc(C)n2)C1 CC(C)CCC(=O)C(=O)NC(C)CCCC(=O)NC1C=CCCC1 N1(C(CN2C(C)CC2)=O)CCCC1CCNC(c1csc(-c2nc[nH]n2)n1)=O Cc1nc(C(C)C)sc1C(=O)NCc1ccccc1CNC(C1CCC(=O)O1)=O Cc1c(Cl)ccc(C(N2CCCC2CN(C)C(c2ncnn2C)=O)=O)c1N Cc1ccc(CSCC(=O)NC2CCOCC2NC(c2coc(CO)c2)=O)cc1 Cc1cccc(-c2ccc(C(N3CC(CO)(NC(C4CC4(F)Cl)=O)C3)=O)n2C)c1 c1(C(=O)NC2C(CC)CN(C(=O)CCCSC)CC2)cnn(C)c1S(N)(=O)=O C(=O)(CC(C)(C)N(C(=O)CC1C=CCC1)C)N(CC(=O)OC)CC c1(C(=O)NCC2OCC(CNC(c3ccsc3)=O)C2)oc2ccccc2c1Cl c1(C(=O)NC2CCCC(CC(=O)NCCN(C)CC)C2)ccc2n[nH]cc2c1 N1(C(CC2CCN(C(CNC(N)=O)=O)CC2)=O)CCC(O)(c2ccccn2)CC1 CCCCC(CC)C(=O)NCC1(C(=O)OCC(C(=O)NCC2CC2)OCC)CC1 C(CCNC(=O)Cc1ccsc1Cl)(C(C)C)NC(c1c(OC)scc1)=O n1(CC(N2CC(CNC(C3CC(O)(CC#C)C3)=O)C(C)C2)=O)ncc(C#N)c1N N1(C(c2cncc(OC)n2)=O)CC(O)CCC1C(=O)NC1(C)CCCC1C C1(NC(=O)OC(C)(C)C)CCS(=O)(=O)C1.C12CCC(C1)COC2=O N1(C(CC(CCC)CC)=O)CCC2(CCC2)C(NC(=O)CC2C(C)(C)C2(C)C)C1 n1(CC(=O)N=c2cc[nH]cc2)ccc(=NC(=O)N2CCOCC2)nc1O C1(CNC(CS(CC)=O)=O)CC2CCC1N2C(=O)CCc1cnc(C)s1 CC1CC(NC(=O)Cn2nnn(-c3cccs3)c2=O)CN1C(c1coc(Cl)c1)=O CC(C(C)C(=O)NCCOCCOCCNC(C1CC(C(F)F)C1)=O)S(C)(=O)=O C(=O)(C#CC(C)(C)O)N(CCC(N1C(CCC=C)CCC1)=O)C(C)C N(C(=NCCOc1cccnc1)NCC1CCC(C(N)=O)O1)Cc1ccc(C)o1 C1(C(=O)NC2(C)CC(NC(Cn3ncc(C)c3)=O)C2)OC2CCC1C2 c1(C(=O)OC)ccc(I)cc1-n1cnnn1.c12ccccc1COCO2 c1(C(=O)NCCCC(C)NC(COCCOC)=O)cc(Br)c(C)s1 C1(C(=O)NCC(CNC(CNC(=O)OCC)=O)(C)O)(CC)CCCC1 c1(C(C(=O)NCCC2N(C(c3cncs3)=O)CCC2)(F)F)ccccc1F c1(C(=O)NC2CC(OCC(=O)NCC(CC)(C)O)C2)cnnc(C)c1 CC(CC(=O)NCC=CCNC(=O)C(C)Oc1ccc(Cl)c(Cl)c1)CC(C)(C)C N1(C(C2(c3ccc(Br)cn3)CCC2)=O)CC2CC(CO)(CO2)C1 c1(C(N2C(CN(C(=O)CN(C)C(N)=O)CC)CCC2)=O)cccc2c1nnn2C N1(C(CC(CC)C(C)C)=O)CCC2CCC(C1)N2C(=O)CN1CC2C=CC1C2 c1(C(=O)NC2COCCN(C(=O)C=C3CCOCC3)C2)ccc2c(c1)NCCC2 C(C(C(=O)NCC(C1CCCC1)O)C(C)(C)C)NC(CCN(CCC)C)=O c1(OCC(=O)NCCN(C(=O)C=C2CCCC2)CCOC)cnn(C)c1 C1(OCC)CC2(C1)CC2NC(C1CC1CNC(C1(O)CC1)=O)=O C(=O)(C(O)C1=CCCCC1)N1CCN(C(=O)C2CC2)CC(CO)C1 Cc1c[nH]nc1CNC(=O)CCOCCNC(=O)CSC1CC1 C1(C(=O)NC(c2ccccc2)CNC(C2(CO)CC2)=O)CCOC2(CCCC2)C1 c1(C(N2C(C)CC(CC(F)(F)F)C2C)=O)cc(F)c2ccccc2c1 c1(C(N(C(CNC(C(C)=NOCC#N)=O)C)C)=O)ccc2cnn(C)c2c1 C1(CC(=O)N(C)CCOCCN(C(=O)COCC(F)F)C)CC12CC2 C1(NC(c2c(F)cccc2Cl)=O)CN(c2nnc(O)s2)C2CCCCC12 Cn1ncc(C2CC2)c1C(N1CC(CNC(C2COCCO2)=O)C(O)C1)=O CCC(C(C)C)NC(=O)C(n1cc(CN(C(C)C)C(C)C)nn1)C C(O)(CC(=O)N1CCOCC1C1CC1(F)F)(C(F)(F)F)c1ncc(C)o1 N1(C(Cc2n(C)nnc2)=O)CCN(C(=O)C=Cc2nccs2)C(CC(F)F)C1 C1(NC(=O)C(c2ccccc2)F)CC2(C1)CC2C(N1CC(CF)C1)=O c1(C(=O)NCC(C)CNC(=O)C(C)n2ccnn2)cccc(C(C)(C)C)c1 Cc1ccc(Cl)cc1C(=O)NC(c1cn(-c2cncc(Cl)c2)nn1)C C(=O)(C(C)(C)c1csc(-c2cccs2)n1)NCC(C)NC(C1CC(O)C1)=O CCC(CC(=O)NC1CC(CO)N(C(C2CC(CF)C2)=O)C1)C1CC1 C1(NC(=O)CNC(=O)C2CC2)CC2CC1CN2C(c1cccnc1O)=O N1(C(Cn2ccc(C)n2)=O)CCCC(NC(C2CC3(F)CC2C3)=O)C1 CC1CN(C(=O)C(C)(C)COCC(F)F)CC1NC(=O)Cc1ccco1 C(=O)(CCCC(C)(C)C)NCCC(CC)(C)NC(=O)CC=CC(C)(C)C CC(C(C)C(=O)NCC1C=CCOC1)NC(=O)CN(C1CCC1)C c1(OC(C)C)ccc(Cl)cc1S(=O)(=O)N1CC(F)(F)CC1CCO N1(C(c2cc(OC)ncc2Cl)=O)CC2CC3CC2C1C3NC(=O)CNC(=O)OC C1(CNC(C2C(CCC)C2)=O)(NC(=O)C(F)=CCCF)CCOCC1 C1(NC(=O)C2=CCCO2)CC1C1CCCN(c2ncnc3[nH]ccc23)C1 c1(C(=O)NC(CCNC(C(c2ccccc2)OCC)=O)C)cc(C)sc1Br C(N=c1[nH]c(=NCC2CCCO2)[nH]c2c1CCC2)c1sc2ccccc2n1 C(CCC(O)C(=O)NCc1ccccc1F)NC(c1c(C)noc1)=O Cc1c(C(=O)NC2CCN(C(=O)CNC(N)=O)CC(C)(C)C2)nn2c1CCCC2 S(=O)(=O)(c1ccc(Cl)cc1C(=O)O)N(C1CCOC(C)(C)C1)CC C1(C(=O)NCC(CCC)OC)CN(C(=O)C(C)N=[N+]=[N-])CCC1(C)C N1(C(C2CCCC(NC(C(CC)(C#N)CC)=O)CC2)=O)CC2(C1)CC1(CCC1)C2 c1(C(N(CCCN(C(=O)CSc2ccc(O)cc2)C)C)=O)cnc2sccn12 N1(C(C(F)OC)=O)CC23CCCC2(C1)CN(C(c1cnc(F)c(C)c1)=O)C3 C(=O)(CCC1=CCCCC1)NC1C(NC(C(C2CCCCCC2)C)=O)COCC1 N1(C(c2c(C)nn(C(C)(C)C)c2)=O)CCCC(CO)(NC(=O)CC(C)N(C)C)C1 c1(N2CCC(CCC)(CO)C2)cc(N2CCOC(CC)CC2)nc(CC)n1 C12(CNC(c3c(SC)cccc3F)=O)CN(C(c3cc(F)n[nH]3)=O)CC1CCO2 Cn1cc(C(N2CCC(CNC(C3CCCN3N=O)=O)C2)=O)n(C)c1=O C(C)(C)(CC(=O)NCC1(F)CCC(NC(c2cnc(C)nc2)=O)C1)OC Cc1ccc(Cl)c2[nH]c(C(=O)N(C(C)CNC(c3cc(N)ccn3)=O)C)cc12 C(=O)(C(C(C)CC)N(C)C(c1cnn(CC)c1C)=O)NCC(=O)OCC#C C1(CC)(CNC(=O)C(C(C)C)NC(c2cccc(C)c2)=O)CC(C)(C)C1 N1(C(C(CC)SC)=O)CC(NC(C2C3CCC2(c2ccn(C)n2)C3)=O)CC1C Cc1csc(CC(=O)NCC2CC2CC(=O)NC2(n3ccnn3)CC2)c1 c1(C(=O)NC2(CNC(CNC(N)=O)=O)CCC2)cc(O)c2ccccc2c1 CCC(O)(CN(C)C(c1cn(CCNC(c2ncnn2C)=O)nn1)=O)CC C#Cc1cccc(NC(c2cc(Br)c(C)s2)c2nnnn2CC(=C)C)c1 C(=O)(C(C)(F)C(=O)NC1CC(NC(=O)C(C2CCCC2)OC)C1)OCC c1(C(=O)NC23CC(NC(CC(=O)OCC)=O)C(OC2)C3)cc2n(n1)CCCC2O c1(OCC)cnc(C2CN(C(=O)CC3CC(O)C34CCC4)C2)cc1C N1(CC(=O)NCC2(O)CCCN(C(C3(C)COC3)=O)C2)CCCC2(CC2)S1(=O)=O CCC(C(=O)OC)C(=O)N1CCCC1(C)C(N1CCC(C(C)OC)CC1)=O N1(C(C(C)NC(C)=O)=O)CCC(NC(c2ccc(F)cc2)=O)C(CO)CC1 C=CCC(CC(F)F)NC(=O)NCCc1cc(C)ccc1Br C(=O)(CC1CCCc2ccccc21)N1CC(CNC(C2(C=C)CC2)=O)N(C)CC1 C1(OC)CCn2cc(C(=O)Nc3cc(-c4nn[nH]n4)ccc3Cl)nc2C1 C1(NC(=O)CCN2CCC(F)C2)CCN(C(=O)CCC2CC2)C12CC2 CC(C(=O)N(C1(C(=O)NCC2(N(C)C)CC2)CC1)C1CC1)=C1CCCC1 C1(C(N(CC(CNC(C2C(C)C2)=O)(C)C)C)=O)Cc2cc(F)ccc2O1 c1(C(N2CC3CCN(C(CCC(CC)OC)=O)C3C2)=O)ccc2c(c1)C=CCC2 N1(C(c2cccc(=S)n2O)=O)CCC(NC(C2(F)CCOC2)=O)C2(CCC2)C1 c1(C(=O)NCC2(F)CC(NC(C3CC(OC)C3)=O)C2)cccc2cc(Cl)ccc12 c1(CCC)cc(C(=O)NC2(CCNC(=O)COC)CC2)c(C)o1 N1(C(C(C)NC(=O)NC)=O)CCC2(CC1)CC(NC(=O)C(=O)N(C)C)CO2 C(=O)(C1=NOC2(CCOC2)C1)NCC1(C)CCCN1C(C12CC(F)(C1)C2)=O CC(C1CCCCC1)=CC(=O)NCC(C)(C(C)C)NC(=O)CC1(CO)CC1 CC(CCC1CCCCC1)(c1nnnn1C1COC1)NCc1cnco1 C1(C(NC(=NCC2CCOC2)NCC2=CCCCC2)C)CCC(F)(F)CC1 c1(SC)cccnc1C(=O)NCC1CCCC(CNC(=O)C(C)SC(C)C)C1 Cc1cnc(CCNC(=O)CCC2CC(NC(C3(C)CCNC3=O)=O)C2)nc1 c1(OC)cc(C)c(C(=O)N(CCCNC(c2c(C)nn(C)c2Cl)=O)C)cc1Cl CCCC(C)(CC)C(=O)NC(C)C(=O)NCCc1ncn(C)n1 N1(CC)CC(C(=O)N2CC(NC(=O)C(C)(F)F)C(C)(C)C2)c2ccccc21 CC(CC(N)=O)C(=O)N(C1CC(NC(c2c(O)cccc2Cl)=O)C1)C Nc1cccc(CC(N)C(=O)NC2CC(n3ccnc3)C2)c1 C1(SC)CN(C(c2cc(Cl)cnn2)=O)CC1NC(=O)C(C)(C)n1cnnn1 C12CCOCC1Sc1cccc(c1)CC2.C(=O)(C(C(C)C)OC(C)=O)NCCC O=C1CSc2ccc(C(=O)NC34CCN(C(=O)C5=CCCCC5)CC3C4)cc2N1 c1(C(=O)NC(CCNC(Cn2nnc(C)n2)=O)C)cccc2ccnn12 CC#CCCCC(=O)NC(C)C(CO)NC(=O)CCNC(C1CCCO1)=O CCC(C(=O)NC1C2CN(C(C3(c4cccc(F)c4)CC3)=O)CC12)C(C)(C)CC n1(CC(=O)NCC2(CNC(C(CO)OC)=O)CC2)c(C)ccc1C CCC1(c2ccccc2)C(=O)N2CC(CO2)n2cc1nn2.C1(C(N)=O)CC1 c1(C(=O)NCC2CC(NC(c3n(C=C)nnc3)=O)C2)cc(C)cc(C)c1N C1(CC(=O)NCC(CC2CCCC2)C(=O)N2CC3(CC3)C2)CC2(CCC2)C1 Cc1cc(NC(C2CC3CCC2N3C(=O)CC2CCCC23CC3)=O)cc(C)c1C Cc1ncc(C(=O)N(C2CCN(C(=O)C#CC(=O)O)CC2)CCO)cn1 c1(OC)cccc(C(=O)N(C2CN(C(=O)CCSC(F)(F)F)CC2F)C)n1 c1(OCC(N2CC(N(C)C)C3(C2)CC3)=O)cnc2ccccc2c1 CC1OC2(CNC(=O)C(O)C3CC3)CC1(NC(c1ccc(C3CC3)cc1F)=O)C2 N1(C(c2cn(C)c(=O)cc2)=O)CC(NC(=O)C(CO)NC(N)=O)CC2(CC2)C1 C1(CCC)(NC(c2sccc2C)=O)CCN(C(=O)C(CC)SC)CC1 c1(C2CC(C(=O)NCCNC(C3(C(=O)NC)CC3)=O)C2)ccc(F)cc1 c1(SC)cc(=NC(=O)C2CC(NC(C3(C4(C)CC4)CC3)=O)CCO2)[nH]n1C c1(C(=O)NC2CCCCN(C(C3C(OC)CC3)=O)CC2)cccc(Cl)c1[N+](=O)[O-] C(=O)(C(=O)C(C)CC)N1C(CC(=O)NC(CCCC)COC)COCC1 CC(C)C(O)CC(=O)N1CC(C(C(=O)N2CCC2CN=[N+]=[N-])N(C)C)C1 C1(CNC(C2CCCS2)=O)CCN(C(C2CC2F)=O)C1 N1(C(CC(C)F)=O)CCN(CCNC(C2(C(=O)OC(C)(C)C)CC2)=O)C2(CCC2)C1 S(=O)(=O)(c1c[nH]c(C(N2CCN(C(C3CNC(=O)C(C)(C)C3)=O)CC2)=O)c1)NC Cc1nnc2n1CC(C(N1CC(NC(=O)C=Cc3cscn3)CCC1C)=O)C2 N1(C(c2n(CC#C)ccc2)=O)CCC(C)C(NC(c2cccc(Cl)c2F)=O)C1 CC1(F)CN(C(c2cc(Br)co2)=O)CCN(C(c2cc(Cl)c(Cl)s2)=O)C1 CCCC(C(=O)N1CCOC(C)(CNC(=O)C=C2CCC2)C1)S(N)(=O)=O c1(C(=O)NC(CNC(CCC(=C)Cl)=O)CC)cc2cccc(C)c2s1 c1(C(N2CC(CN(C(=O)CCN3CCCC3)C)OCC2)=O)ccn2ccnc2n1 Cc1ccc(C)c(C(=O)OC2CCC(NC(=O)NC3CCC3)CC2)c1C Cc1cc(C(=O)N(C(C)CNC(C2(C)CCNC(=O)C2)=O)C)cc(C)n1 c1(NC(COCC)COC)[nH]c(=NCCNS(=O)(=O)C2CC2)nc2scnc12 Cc1oc(C(=O)NC(C)CC2CN(C(=O)CCn3cc(Cl)cn3)C2)cc1CO C1(O)(CCNC(=O)C2=C(Cl)CC2)CCCN(C(c2cc[nH]c2C2CCC2)=O)C1 C1(C(=O)N(CC(C)C(=O)N(CC(O)CF)C)C)(CC)CC(C)(C)C1 CC1Cn2nccc2CN1C(=O)CCN(CCO)C(c1cccc(F)c1O)=O c1(C(=O)NCC2CCC2NC(C2C3(CC3)C23CC3)=O)cc(F)c(F)cc1F C1(O)(CCNC(CCOC(C)C)=O)CCN(C(=O)C(C2CCCCC2)C)C1 S(=O)(=O)(c1ccc(NCCn2ncc(C(C)SCC)c2)c(F)c1)N1CC(CO)C1 N1(C(C)=O)CCCCC(C2CN(C(c3cn4cc(C)ccc4n3)=O)C2)C1 CCC(O)CC(=O)NC1CCCN(C(=O)C(c2ccc(OC)cc2)C)C1 C(CCCCCC(=O)N1CCC(N(C)C(c2csc(C(C)=O)n2)=O)C(C)C1)SC C#CCC(C)(C)C(=O)NCC12CC1CN(C(c1c(C)nn(C)c1Br)=O)C2 C1(CNC(C(=O)NCC)=O)CN(C(c2ccc(N)c(F)c2)=O)CC12CCC2 c1(C(N2C(CCNC(CCN(C)CC)=O)CSCC2)=O)ccn2cccc2c1 C(C(CO)N=c1[nH]nc(C(C)C)o1)NC(c1cc(CC)n(-c2ccccc2)n1)=O C1(NC(C2C3CC3CN2C(C2CC2C(F)F)=O)=O)CCC12CCCC2 N1(S(C)(=O)=O)CCC(COC(=O)CCC(=O)N2CCCC(N(C)C)C2)CC1 Cc1cc(CNC(=O)N(C)CC2CCS(=O)(=O)N2C)nc(Cl)c1Br c1(CN(C2CN(C(c3cc(C)nn3C(F)F)=O)C2)C)cc(F)cc(Br)c1 C#CC1CN(C(C2C=CCC2)=O)CCN1C(c1cc(O)ccc1C)=O C1(OC)CCn2cc(C(=O)N(C)CCNC(c3c[nH]nc3C(C)(C)C)=O)nc2C1 c1(CC)cc(Br)c(C)cn1.C12CN(CCS1)C(=O)N2.CC=O C(=O)(C(COC)C(F)(F)F)N1CC(F)CC(NC(C2CC(CCC)C2)=O)C1 c1(C(=O)NCC(CC)NC(CC(=C=C)C)=O)ccc(-c2ccccc2)cc1C c1(-c2ccc(COC)cc2F)nc(C2Cc3ccccc32)nn1CC1CCCC1 N1(C(c2cnc(SC)nc2O)=O)CCC2C(C1)CN2C(=O)C1=CC(C)(C)C1 N1(C(C(CC)CC)=O)CCCN(C(c2ccc(N)cc2SC)=O)C(C)C1 N#Cc1ccnnc1NC1CC(CCNC(C2CCCO2)=O)C1 Cc1c(F)cc(C(=O)NCC(CNC(c2cc[nH]n2)=O)CO)c(F)c1N C12(NC(CCc3c(C)noc3Cl)=O)CCCN(C(=O)C(C)(C)O)CC1C2 Cc1nc(C2CC2)oc1C(N1CC(NC(c2c[nH]nc2C(C)C)=O)C1)=O N1(C(c2c(C)cc(F)cn2)=O)CCCN(C(=O)CSCc2cccnc2)CCC1 C12(C(=O)NC3C(CCC)CN(C(C4COCCC4C)=O)C3)CCC(C1)OC2C N1(C(C(CC(C)C)ONC(c2cc(=NC)[nH]cc2)=O)=O)CCOC2CCCC12 N1(C(c2c(C(=O)OC)c(C)on2)=O)CCC(NC(c2cc(C)nn2C)=O)C(C)C1 N1(C(c2cccc(CC)c2)=O)CC(N=[N+]=[N-])CC1C(=O)NCC(O)CC(C)(C)C N1(C(C=CCC)=O)CCOC(C(C)NC(=O)CCCn2c(O)nnc2O)C1 C1(C)(NC(Cc2cccc(CC)c2)=O)CCN(C(C2CC(=O)CO2)=O)CC1 c1(CC)[nH]nc(C(=O)NCC=CCNC(c2nnn(CC)c2C)=O)c1Br C1(C#N)(C(=O)NCCCC(N2CC=C(C)CC2)=O)CC2CC2C1 C(C(CC(C)C)C(=O)N1CCC(CNC(=O)C(C)=CCO)C1)OC c1(C(=O)NCC2(C)CCN(CCC=CCC)CC2)coc2c1C(=O)NCC2 N1(C(c2cccc(OC)c2)=O)CCCC2(NC(c3cc(O)nc(Cl)c3)=O)CC2C1 c1(C(=O)NC2CC(NC(COCCCN(C)C)=O)C2)ncnn1C N1(C(C2CCC(C)CN2C(C2CCNC2=O)=O)=O)CC(C#N)C2(CCC2)C1 c1(CC)ccccc1CC(=O)NCC12CC1CN(C(c1ocnc1C)=O)C2 N1(C(c2cccc(C)c2N)=O)CC2CC(C)N(C(=O)CC3CCC(C)(C)C3)C2C1 N1(C(c2ccnnc2)=O)CCC2CC2(C(=O)N(C2CC2)CC2CC2)CC1 C(=O)(C#CC(C)(C)O)NCC12C(CN(C(C(C)OC3CCOC3)=O)C1)C2 CC1CN(c2ccccc2CNC(c2[nH]nnc2Cc2nn[nH]n2)=O)CC(C)O1 c1(C(N2CCC(CC=C)(NC(c3ccc(C)o3)=O)C2)=O)cc2ccc(Cl)cc2o1 O=C1CCC(C(N2CCC(NC(=O)C(C3(O)CCCC3)F)CC2)=O)CN1 C(=O)(C(CO)C(F)(F)F)N1CCC(OC)(CNC(C2CC(C3CC3)=NO2)=O)C1 C1(C(N2CC(CNC(CNC(CCC)=O)=O)C(O)C2)=O)CC(=O)NC(=O)N1 C(CCN(C)C(C1CCCCS1)=O)(C(C)C)NC(C1(OCC)CCOC1)=O Cc1cccc2[nH]c(C(N3CC4CC3CN(C(c3cc(C#N)no3)=O)C4)=O)cc12 Cc1ccccc1C=CC(N1CC2(NC(c3cc(C)c(C)[nH]3)=O)CCC1C2)=O N1(C(CSCC)=O)CCC2(CNC(=O)C=Cc3ccccc3)CCCCC12 O=C(C#Cc1ccccc1)N1CC2CCCN(C(c3ccnc(Br)c3)=O)C2C1 CC(CC(=O)N1CC(F)(F)CC1(C)CNC(=O)Cc1cnsc1)C(F)(F)F c1(CC(=O)NCC(C)NC(C2CCCCS2)=O)ccc(O)nc1 N1(C(CC2(OCC)CCC2)=O)CC2CN(C(C3COCCC3(F)F)=O)CCC12 N1(C(Cn2ccc(=N)[nH]2)=O)CCC(NC(c2cc(C3(C)CC3)n[nH]2)=O)C(CO)C1 c1(OC)ncc(C(=O)Nc2ncc(-c3ncc(C(F)(F)F)cc3Cl)s2)cc1F N1(C(=O)Cc2cnccn2)CC2CCC1CN2C(=O)C=C1CCCCCC1(F)F CC1CC(NC(c2ccc(C3CC3)s2)=O)CN(C(c2cnc(Cl)c(N)c2)=O)C1 c1(C(=O)NC2C(OC)CN(C(CC3(C=C)CCC3)=O)C2)coc2c1C(=O)NCC2 CC1CCc2onc(C(=O)NC3(C)CN(C(c4ccnc(Cl)c4N)=O)C3)c2C1 N(C1CCOc2c(C(=O)OC)cc(C)cc21)CC(C1CCOCC1)CC C(=O)(CC(C)(C)C)N1C(C(N(C(C)CNC(C2COC(=O)N2)=O)C)=O)CCC1 c12ncc(cn1)C(=O)NC2.C1(CCCOC)(CNC(=O)CC(C)C)CCCC1 C(C1=CCN(C(=O)C=Cc2ccc[nH]2)CC1)NC(Cn1c(C)csc1=O)=O N1(C(CC(C)(C)C)=O)CCC2CN(C(C34CC3CNC4=O)=O)CC12 C(C1=NOC2CN(C(c3cn(C4CC4)nn3)=O)CC12)NC(c1cc(C)c(C)[nH]1)=O C1(C(N(CC(O)CNC(=O)CCc2cnn(C)n2)C)=O)CCCC(N(C)C)C1 C1(N(C(CCCC)=O)C)CCN(C(C23CCOC(C)(C2)C3)=O)CC1C S(=O)(=O)(c1ccc(I)cc1[N+](=O)[O-])NCc1cc(CC)on1 C1(OC)CN(C(=O)C(Cn2ccnn2)NC(=O)C(CO)OC)CC12CC2 C=CCCC(C(=O)NCC1CCOC1C)NC(c1nnsc1C)=O c1(C(=O)NC2CC3(CN(C(Cn4c(C)nnn4)=O)C3)C2)c[nH]c(=O)c2ccnn12 Cc1nn(C)c(C(=O)NC2CCC2CNC(=O)C(F)(F)C2CCCC2)c1[N+](=O)[O-] C1(O)(C(C)NC(=O)COC(F)F)CCN(C(c2cnn(C3CC3)c2)=O)C1 CC(CC(F)F)C(=O)N1CCN(C(C)CNC(=O)CSc2ccncc2)CC1 CC1(C)CC(CNC(=O)N(CCO)CC2CCCN(C3CCC3)C2)c2ccccc2O1 C(c1cccc(F)c1)=CC(=O)NC1CC(C(N2CCCC(N(C)C)C2)=O)C1 N1(Cc2c(C)nc(C)s2)CCC(C)C(NC(=O)CCC2NC(=O)NC2=O)C1 n1(CC(=O)NC(CCCCNC(C)=O)C)nc2n(c(=O)c1=O)CCC2 Cc1cncc(C)c1C(N1CCOCC(CNC(=O)COc2cnn(C)c2)C1)=O c1(CC)n[nH]cc1C(c1nnnn1CC1CCCO1)NCCC1(SC)CCC1 CC(C(=O)NN1CC2CC=CCC2C1)(C(F)(F)F)c1ccccc1 CC(O)C(C)C(=O)N(CCCOCCCNC(=O)Cc1ccccc1F)CCO CC(C)(C)C(O)C(=O)N1CC(NC(C2CCCC(=O)C2)=O)C(C)(C)C1 c1(C(=O)NCC2(F)CCC(NC(CCOCC#C)=O)C2)cc(C)c(F)cc1N c1(C(=O)NCCCNC(c2cnc(OC)s2)=O)ccc2c(c1)CC(C)O2 CCCCS(=O)(=O)CC(=O)NCC1(OC)CN(C(c2cnc(CC(C)C)[nH]2)=O)C1 C(=O)(C(C)CC(C)CC(C)C)NCCN(CCC)C(C1OCCC1CC)=O N1(C(c2cnc(SC)s2)=O)CCN(C(c2ccon2)=O)C(CF)C1 N1(CC(=O)N(C2CC2)CC2N(C(C=C(C)Cl)=O)CCC2)CCC(F)(F)C1 N1(C(C(C)O)=O)CCC(NC(c2cc(Cl)ns2)=O)C1C1CC1 C1(NC(c2cc(COC)on2)=O)CC(O)CN(C(=O)CCc2cccc(Cl)c2)C1 C1(C(=O)NCC(C)NC(=O)C(C)(C)c2cncnc2)CC(C)(C)CO1 CC(C(=O)NCCC1(CNC(=O)C(C2CCCO2)C2CC2)CC1)N(C)C c1(C(N(CC(C)C(=O)NC(C)Cc2ccco2)C)=O)c[nH]c2ncccc12 Cc1ccc(C(C)C(N2CCCC2C2CCCOC2)=O)o1 CCC(C)C(C(=O)NCC(CO)OC)N(C)C(c1cccc(C)c1N)=O C#Cc1cnn(C)c1C(=O)NC1CCCN(CC(F)(F)F)C1=O NC(Cc1ccccc1)C(=O)NCCC1CCC1 C=CC1(O)CCN(C(=O)C(N)CC2CCOCC2)C1 CC(C)(C)C(C(=O)N(c1cccs1)Cc1cn2c(n1)SCC2)N1CCCCCC1 C(CCS(C)(=O)=O)N(C(C(c1cnn(C)c1)NC(COCC(=C)C)=O)=O)C(C)C C(=O)(CS(=O)(=O)C12CC(C1)C2)N1C2CC(NC(C3CC(=C)C3)=O)CC1CC2 N1(c2ccc(NC(=O)NC3(c4cccc(C)c4)CC3(F)F)cc2)CCS(=O)(=O)CC1 C1(N(C(=O)NC(C2CCCC2)CC)C)CCOCC1 n1(CC(=C)C)nnnc1C1(NCC2(CC(=O)OC)CC2)CCC1CC(C)C CN1C(=O)OCC12CN(C(=O)CC(F)(F)c1ccncc1Br)C2 c1(CN(C)C(=O)OC(C)(C)C)ncc(C(=O)NCC23COC(C2)C3)cn1 S(=O)(=O)(c1cnc(NCC2(Cl)CC2(F)F)c(Cl)c1)NCC(C)N(C)C C1(CCC(=O)NC2(CC=C)CCCC2)CCCCN1C(=O)CC1CCCC(C)C1 c1(C(=O)NC(CCOC)CNC(=O)C=Cc2cnccn2)cc(F)cc(N)c1F c1(COC(C2N(C(C)=O)CSC2)=O)c(Br)cnn1C Nc1cc(C(N2CCN(C(c3csc(Cl)c3)=O)C(c3cn[nH]c3)C2)=O)cc(F)c1 C(C)(C(=O)NCC(C)(C)Cn1cc(C(C)O)nn1)(C(C)C)NC(C)=O C12(NC(c3c(C)ccnc3Cl)=O)CCCC1CN(C(=O)NC(=O)C(Cl)(Cl)Cl)C2 N1(C(C(C)CC2CCCC2)=O)CCCC(NC(C2(C)CC(F)C2)=O)C1 C(CC(C)C)(C(=O)NCC(=O)N(C)O)N(C(COCCCC)=O)C Cc1ccc(C(=O)NCC2C3CN(C(c4n[nH]cc4Cl)=O)CC23)c(=O)n1C Cc1cc(O)c(Cl)cc1C(=O)NC(C)CNC(=O)C1=NOC(c2ccccc2)C1 C=CCCN=C(NCCc1c[nH]c2ccccc12)NCC(C)(O)c1cccs1 c1(OC)cccc2c(C(N3CCC(C)C3CNC(=O)CCC(C)(F)F)=O)coc12 C1(CNC(C2(CC)CCCC2)=O)CN(C(c2c(C)cnn2C)=O)CC2(CCC2)O1 N#CC1CC2(CC(NC(C3CC(NC(=O)C(O)CC(N)=O)C34CCC4)=O)C2)C1 c1(C(=O)NC2CN(C(CSC(C)C)=O)C3C2C3)cnc2cnn(C)c2c1 C#CCCC(C(=O)NCC1C=CCCC1)NC(=O)CCn1cc(C)cn1 CCC(CC)C(C(=O)NCCCC1CCCN1C(c1ccco1)=O)OC N1(C(COCc2cc(C)no2)=O)CCC(NC(=O)C2=CCCS2)C(CO)C1 c1(C2N(C(c3csc(C(F)(F)F)n3)=O)CCC2)cncc(Cl)c1 Cc1cccc2c1N(C(=O)CCCCC(=O)c1ccc(F)cc1)CCO2 N1(C(c2c(OC)cncc2)=O)CC2CCC1CN2C(C1CC2(C1)CC(C)C2)=O c1(C(C)NC(C2(C(C)NC(=O)C(F)C3CCC3)CC2)=O)ccccn1 C(=O)(CCCC(C)(C)C#N)NCC#CC(=O)NCc1cc(C)oc1 c1(C(=O)NCC(CC(F)(F)F)NC(c2cc(F)c[nH]2)=O)cccn2nccc12 N1(C(C=C(C)C(F)F)=O)CC(F)(F)CC1CCNC(=O)COC(F)F c1(C(N2CCN(C(C(COC)C)=O)C(C)CC2)=O)cc(OC)cc2c1OCC2 C1(NC(c2cnn3c2CCC3)=O)CCCC(NC(c2snc(Cl)c2Cl)=O)CC1 CCC(CC(=O)NCC=CCNC(=O)C(CC)OC)c1ccc(OC)cc1 c1(C(N2CCC(C(C)NC(C(CC)F)=O)C2)=O)cc(N)ccc1O CC(CC(=O)NCC1COC(CNC(=O)Cn2nc(O)ccc2=O)C1)P(C)(C)=O CC1(C)CCCOC1C(=O)NCCC1CCCN1C(c1cc(C(F)(F)F)c[nH]1)=O c1(C(N(C2CCN(C(CNC(C)=O)=O)C2)CCO)=O)cccc(CS(N)(=O)=O)c1 c1(N2CCN(C(c3ccccc3Cl)C(=O)OC)CC2)ccnc(C#N)c1 N1(C(C2(C)CCN(C(CC(CC)(C)C)=O)C2)=O)CC2CC=CCC2C1 N1(CCOCC)CCC2CCC(C1)N2C(C1CCc2nnn(C)c2C1)=O CCC(C)C(O)C(=O)N1CCOC(CNC(=O)CSCc2csc(=N)[nH]2)C1 Cc1ccc(OCC(N2CCCC2(C)CNC(=O)CN2CSCC2=O)=O)c(C)c1 C1(C(=O)NCC(c2ccccc2)CNC(C2(CF)CC2)=O)CC2(C1)CC2F C(=O)(C(CN)C(C)C)NC(C1CC(O)C(F)C1)=O.C(C)(C)(C1CC1)OC C1(C(=O)NCC(CNC(c2cnc(CCCC)s2)=O)CO)CC12CCOCC2 Cc1nc2sccn2c1C(N1CCC(C)(NC(C2CC3CCC(C2)C3O)=O)C1)=O c1(C(=O)OC)ccc2c(n1)CCCN2C(c1cc2ccccc2nc1Cl)=O N1(C(C(N2CCOCC2)C)=O)CCC2(CCCC2NC(C2C(C)(C)C2(C)C)=O)CC1 N1(C(C(C)NC)=O)CCC2(CCCC2C(=O)N(c2ccc(-n3cccn3)nc2)C)C1 N1(S(CCCC)(=O)=O)CCC2(CC(C(=O)Nc3cc(C(F)F)c(Cl)cc3F)=NO2)C1 C1(N(C2CCCCC2)C(c2ccc(O)nc2)=O)CCc2ccccc2C1 c1(OC)nc(C)ccc1C(N1CC2(CCN2C(c2cc(Cl)cnc2F)=O)C1)=O O(NC(=O)C(C1(O)CCC1)NC(=O)CC(C)(C)SC)CC#C Cc1cc(=NCCC2CCC2(F)F)[nH]cc1S(=O)(=O)NCCN(CC(F)(F)F)C N1(C(CSC)=O)CCN(C)CC1C(N1CC(O)C(O)C1)=O CC1CCCC1NC(=O)NCCN(C)CC1CCOCC1 C1(C)(C(N(CCCC(=O)NC)C)=O)CCN(C(c2nnn(C)c2CC)=O)C1 C1(O)(CCNC(Cc2c(C)ccnc2)=O)CCCN(C(C2CC2C(F)F)=O)C1 C1(NC(c2ccc(CC)cc2)=O)CN(C(=O)C(O)c2ccsc2)CC2(CCC2)C1 c1(C(=O)NCC2N(C(CCN(CC)CC)=O)CC2)ccc(OC)c2ccnn12 c1(C(C)(CC2CCOC2)NCCCn2ccnn2)nnnn1CCCNC1CC1 c1(CN(CC)Cc2scc(OC)c2OC)cc(Cl)cnc1C CCC(CC(=O)NC(c1ccoc1)C)NC(c1ccccc1NC)=O C1(C(C)C)CN(C(c2nnn(Cc3ccccc3)c2Cl)=O)CC1N(C)C c1(C(N2CCN(C(Cc3cccc(CC)c3)=O)CC2C)=O)cnc2c(c1)NCC2 N1(C(C2C(C)(C)C2)=O)CCC2CCN(C(C3(C)CC(F)C3)=O)CC2C1 C(CCC(N)=O)(C(=O)N1CCCC1CNC(c1cc2c(s1)CCOC2)=O)NC(C)=O CCCCC(C(=O)N1CCC2(CC=CCO2)C1)C(C)C c1(C(=O)NCC2(NC(CCCSC)=O)CCCCCC2)c(C)cc(O)nc1C C(C(O)(CNC(C1(C)CN(C(c2ccn(C(F)F)n2)=O)C1)=O)CO)OC c1(OC)cccc(C(=O)N(C)CC2(O)CCCN(C(c3conc3C)=O)C2)c1F C(=O)(C1CCCc2sccc21)NC1CN(C(c2c(C)cc(C)s2)=O)CC1C C1(CNC(=O)CCCCC(F)F)CCCC2(CN(C(C3CCS(=O)(=O)C3)=O)C2)O1 C1(C(=O)NCC2(F)CN(C(=O)COCCN(C)C)C2)SC2C=CC1CC2 N1(CC(N2CC(SC)C(NC(c3ccc(C(C)C)s3)=O)C2)=O)C(=O)CN(C)C1=O N1(C(CCOC)=O)CCC(NC(=O)Cc2ccccc2S(C)=O)CC(C)(C)C1 Cc1ccc(C(=O)NC2CC(C)N(C(c3n[nH]cc3C(F)(F)F)=O)C2)cc1 c1(C(N2CC3C(NC(c4cccc(O)n4)=O)(C3)C2)=O)cc(F)cc2nc(S)[nH]c12 C1(CNC(COCC(C)(C)C)=O)(NC(c2ccc(O)c(Cl)n2)=O)CCCCCC1 C1(O)(CNC(C2CCN(S(CC)(=O)=O)CC2)=O)CCCN(C(=O)C(F)F)C1 c1(C(=O)NCCOCCN(C)C(C2CCC(O)C2)=O)cccc(C(F)(F)F)c1 CC(C)C(C)CC(=O)NCCCCN(C(=O)COCCCN=[N+]=[N-])C c1(C(N2CCC(NC(CN(C(C)C)C)=O)C2C)=O)noc2c1CC(C)CC2 c1(NC(c2c(-c3ccn(C)n3)n[nH]c2)=O)cc(F)cc(F)c1CO C(=O)(C(C(C)(C)C)OC)NCCC1(C(=O)NC(C=C)CO)CCOCC1 N1(C(CCN(C)CCO)=O)CCC2(CC1)CC2(CO)CNC(=O)C1=CCCC1 C(=O)(C(C(C)(C)C)OC(C)(C)C)NCC(CCOC)NC(c1csnc1C)=O C1(CC(C(=O)NCC=C)N(C)Cc2nc[nH]n2)CCC(F)(F)CC1 Cc1sc2ncc(C(N3CC4CCC3CN4C(c3cc(Cl)ccn3)=O)=O)n2c1C c1(C(=O)NCCCC2CCCN2C(C2CCCS2(=O)=O)=O)ncn2c1CCCC2 CC(C)CC(C)C(=O)NCC1CCCC1NC(=O)CC(C)(C)Cc1ccccc1 C(=O)(CCP(C)(C)=O)N1CCC(O)(C(C)NC(CSCC#C)=O)C1 C1(C(=O)NCC2(C(C)NC(c3cccc(F)c3)=O)CC2)CCn2cncc2C1 c1(C(CNC(c2n(CC)nnc2)=O)NC(c2ccnnc2)=O)ccc(C)cc1 C1(NC(N2C(C(C)(C)O)CCC2)=O)CCCCC(F)(F)C1 C(C(CC)(CC)CO)NC(c1c(CNC(CCC)=O)n[nH]c1)=O Cc1cc(C2CC2NC(C2CC(c3ccc(F)c(F)c3)(C(=O)O)C2)=O)ccc1Br c1(C(=O)NCC2(CNC(c3cc(CC)ncn3)=O)CCC2)ccnc2cc[nH]c12 c1(C(N2CCN(C(CC=C)=O)CC(CO)C2)=O)ccc2oc(O)nc2c1 C1(N(C(COCc2ncc(C)o2)=O)C)CC2CCC(C1)N2C(C1CCC2CC12)=O N1(C(c2c(C(C)C)[nH]cc2)=O)CCC(CF)(NC(c2ncccc2F)=O)C1 c1(CC)nc(C)c(C(=O)N(C)CC2(NC(C3CC3c3cnn(C)c3C)=O)CC2)s1 c1(C(=O)NCCOCCCN(C(CCC=C=C)=O)C)ccc(C(C)=O)c(C)c1 c1(C(N(CCCCN(C(C2N(CC)CC2)=O)C)C)=O)nn(C)cc1Cl N1(C(CS(=O)(=O)NC)=O)CCC2(CCCCC2NC(c2cccs2)=O)C1 C1(CC(=O)NC2CC(CCO)C2)CCCN(C(C2CNC(=O)N2)=O)CC1 C1(NC(C(C=C)(C)CC)=O)CCN(CCCC2CCCCO2)CC1(C)C C1(c2ccccc2)(C(N2CC(C)(NC(C3CCC(C)S3)=O)C2)=O)CC2(CC2)C1 C1(C(=O)NC(CC)CNC(=O)C(F)CC2CCOCC2)(CC2CC2)CCOCC1 N1(C(c2cc(CCC)on2)=O)CCC(CC)(NC(c2ccoc2Br)=O)CC1 c1(NCCC(=O)Sc2n(CC)c(-c3ccccc3C)nn2)cc(F)cc(F)c1 N1(C(C2C(CNC(Cc3cc(C)n(C)n3)=O)CCCC2)=O)CC(O)CC12CCCC2 C(=O)(C=C1SCC(=O)N1C)N1C(CNC(C(C)C2CCOC2)=O)CCCC1 N1(C(CCC=C)=O)CC2CCC2(NC(c2ccc(-c3csc(=N)[nH]3)cc2)=O)C1 N1(C(C(C)CC2CCC2)C(=O)NCC2CC2)CCc2c(O)cccc2C1 C(=O)(C1SCCc2ccccc21)NCCC1(O)CN(C(C(C(C)C)CO)=O)C1 c1(CC)nccnc1C(=O)OC.C1(CN2C3CC3C2=O)OCCO1 N1(c2cc(C)c(C3CC3)c(C)n2)CCC2(CC1)CC=CC(=O)N2C c1(C(=O)NC2C(NC(c3csc(CO)n3)=O)COC2)csc(Cl)c1Cl n1(CC)nnnc1C(c1cc(C2CCC2)no1)NCC(C)Oc1ccccc1 Cc1cccc(C(N2CCCC(N(C)C(c3cc(C)n(C)n3)=O)CC2)=O)c1F N1(CC)CCc2cc(OC(C)C)c(OC)cc2CC1.N12CCCC(C1)NC(=O)C2 c1(CC)c(C(=O)NC2CC2NC(c2cc(OC)c(Br)s2)=O)cnn1CC C1(CCOC)CN(C(=O)C(F)(F)C2CCCC2)CCN1C(c1csc(Cl)n1)=O c1(NC)snc(C)c1C(=O)NCCCCCCNC(C1CCCC1(C)C)=O O=C(O)CC(C1CC(F)(F)C1)NC(=O)NCC1CCC(c2ccccc2)C1 C(CC(C(=O)NCCC(O)C1CCC1)NC(c1nc(O)sc1C)=O)SC C1(NC(C2N(C(C)=O)CCCC2)=O)CC2(CCN(C(c3cc(CO)no3)=O)C2)C1 N1(C(C(c2ccccc2)NC(C)=O)=O)C2CCC1CN(C(c1ccccn1)=O)CC2 C1(C)(C(N2CC(CCNC(C3C(C)C3(F)F)=O)C2)=O)CC(C(C)(C)C)=NO1 Cc1ccc(F)c(C(=O)NC(C2CCCN2C(=O)CN2CCC(C)C2)C)c1 CC1(C)CC(C)(CNC(C2CCCCS2)=O)CN1C(c1cc(C(F)F)cs1)=O C1(NC(C2CCC(=C)CC2)=O)C2CCC(C2)C1C(=O)NOCC(C)C O(C=C(C#N)C(=O)N1CCC(NC(c2oc(C)cc2C)=O)C1(C)C)CC N1(C(C(C(C)C)N2CCCCC2)=O)CCC2CCN(C(=O)CC3CC3)C2C1 c1(C(=O)NC)cc(C)c(C)nn1.Cc1cccc(C2CCCN2CC2(CO)CC2)c1 C=Cn1ncc(C(=O)NCC2CC2C(=O)NC2CC(O)CC2O)c1N Cc1ccccc1C=CC(N1CC2(C(=O)NCc3cnc(C)n3C)CC1CO2)=O Cc1ncc(C(=O)NCC(C)CNC(=O)C(C)N(C)Cc2ccccc2)c(C)n1 c1(SCc2nc(CCC)on2)cc(C)[nH]c(=NC)n1 N1(C(C(c2cccs2)NC(COCC)=O)=O)CCC1(C)CC C(CCC(C)C)(C(=O)N(C)Cc1cc(C)cs1)NC(C1(NC(C)=O)CC1)=O C1(C(=O)NC2(CF)CN(C(CC3CCC(C)(C)O3)=O)C2)CC2C=CC1C21CC1 C(=O)(C(COC)CC(C)C)N1CC2(N(C(C(C)SCCCC)=O)CC2)C1 CC(C)CC(F)(F)C(=O)NC(C1CCN(C(=O)COCc2ccccc2)C1)C C1(C(=O)NC(CC)(C)CCNC(c2ccnnc2)=O)CCc2cnnn2C1 C(=O)(C1=CNC2=NCCC2=C1)N1CCCC(CN(C(CC2(C=C)CC2)=O)C)C1 c1(C(=O)NCC(C2CCOC2)NC(C2(OCC)CCC2)=O)cc(C#N)ccc1O C1(NC(c2cccc(C)c2I)=O)CN(C(C2CC3CCC2O3)=O)CC(F)(F)C1 C1(NC(C2N(C(COC3(C)CCCC3)=O)CCC2)=O)CCOC12CCCC2 N1(C(CC(C)OC)=O)CCCC(C)(NC(c2cccc(-n3cnnn3)c2)=O)C1 c1(C(c2n(CCC)nnn2)NCC(C)(C)CCO)cc2cc(Cl)cnc2o1 C12(C(N3C(COC)CC3)=O)CCCC1CCN2C(C1(O)CCCC1)=O N1(C(=O)CCC2CCOC2)CCN(C(c2noc3c2CCCC3)=O)CC(O)C1 C(=O)(CCC(F)(F)CN=[N+]=[N-])NCC1N(C(c2c(C)cc(=O)n(C)n2)=O)CC=C1 Cc1ccc(N(C)C(C2CCN(c3nccc(Br)n3)CC2)=O)c(C)c1 c1(C(=O)NC(CNC(c2c(C)coc2C)=O)(C)C2CCC2)ccc2c(c1)OCC2 c1(C(=O)NCC2C=CC(NC(C(C)NC(COC)=O)=O)C2)n[nH]c(C)c1Cl C1(CC(N2CC(CC(C)NC(C3(C(=O)NC)CCC3)=O)C2)=O)CCCC(C)C1 c1(NC(C)=O)cc(C(=O)NC2CC3(C2)CC32CCC2)ccc1[N+](=O)[O-] C1(CNC(=O)Cn2ccccc2=O)C2CCC1CN(C(=O)CSc1nc[nH]n1)C2 C(CC(C(=O)NC(c1cnc(C)s1)C)NC(=O)Cc1cn(C)nc1C)OC c1(C(=O)NC2CCN(C(c3c(C)cc(F)cn3)=O)CC2O)coc2ccccc12 c1(C(N2CC(NC(C(C)CC3CCC3)=O)C(C)(C)C2)=O)c(F)cc(N)cc1F N1(C(CC(=O)NCC)=O)CCCC(C2CCCN(C(=O)Cc3cnc[nH]3)C2)C1 N1(C(c2ccc3nccn3c2)=O)CCC2CCN(C(=O)Cn3cc(Cl)cn3)C2C1 Cc1c(C(=O)NCCNC(c2cnc[nH]c2=N)=O)c(-c2ccccc2)cn1C c1(C(=O)Nc2c(C(=O)NC3CCNC3=O)n[nH]c2)c(F)cc(F)cc1F N12CCCC(C)(C1)CC2.n1(C(C)C)ccc(C(=O)NC2CCOC2)n1 N1(C(C23CC(C#N)(C2)C3)=O)CCCCCCCCC1.C1(CCC)CN2CC1C2=O C1(NC(C(C)=C2CC2)=O)CCC(F)(CNC(=O)C(C)NC(c2ccoc2)=O)C1 c1(C(=O)NCC2C(NC(C3(O)CCC(CC)CC3)=O)C2)cc2ccc(C)cc2[nH]1 C1(C(N(CC(C)NC(=O)COCC(F)F)C)=O)COc2ccc(Cl)cc2C1 N1(C(CCCOCC)=O)CCN(C(=O)C(C)Oc2ccc(Cl)cc2)CC1C c1(N2CCC(C)C2)nc(N2CCN(c3ccncn3)CC2)nc2scnc12 c1(CCNC(C2CN(C(=O)CC3CC3)CC2(F)F)=O)c(F)cccc1Cl c1(C(=O)NCCC2N(C(C3(COC)CC3)=O)CCCC2C)cc(C)c(C#N)cn1 C1(NC(c2c(C)nns2)=O)CCN(C(C2CCC3CC3CC2)=O)CC1(C)C C1(C(=O)NCC2(CCNC(C3(C)CCC4CC4C3)=O)CC2)CN=C2N=CNN2C1 C1(C(=O)Nc2ccc(NS(C)(=O)=O)nc2)COC2(CCC2)C1 C12(NC(C3CN(CC(C)C)C3)=O)CCC(C1)N(C(=O)C(O)C(C)(C)C)C2 CC(c1ccc(F)cc1)=CC(=O)NCC1CN(C(=O)Cc2n[nH]c(C)n2)CC1C C1(CNC(C(C)SCCCC)=O)CN(C)CCN1C(c1cc2[nH]ccc2s1)=O c1(C(N(c2ncccc2N)C)=O)cccc(CNC(C2CC2[N+](=O)[O-])=O)c1 C(=O)(C(C)Cc1ccc(CC)o1)NC1CN(C(CCOCC#C)=O)C1 N1(C(C2CC(SC)C2)=O)C2CCCC1CC(NC(=O)C(C(C)C)C(C)C)C2 c1(C(=O)NCCC2CC(NC(=O)CC=C(Cl)Cl)C2)cccc(C#CCO)c1 C1(C(=O)NCC2CCN(C(C3(COC)CC3)=O)C2)CC12C1CC3CC(C1)CC2C3 c1(CNC(=O)OC2COC(C(F)F)C2)cnn(Cc2ccccc2)c1 N1(C(C(COC)OC)=O)CC2CC(NC(C3(C)CC=CC3)=O)CC2C1 Cc1cc2c(cc1C)OC(C(=O)NC1CCN(C(c3ccccc3Cl)C)C1)C2 c1(N(C)C)nc2ccc(C(=O)NCC3CC(N)CCO3)cc2o1 N12CCC3(CC3C(=O)Nc3nocc3C1=O)C2.CC(C)(C)SCC(N)=O CC1=C(C(=O)N2CC(CO)(NC(c3snnc3C(C)C)=O)C2)C(=O)OC1(C)C c1(N(C2CN(C(c3cccc(S(C)=O)c3)=O)C2)C)ncnc2[nH]cc(I)c12 CC1=CCC(C(N2CC3CC3C2CNC(=O)Cc2cnc[nH]2)=O)CC1 Cn1ncc2ncnc(N3CC4C(CNC(=O)CC5CC(=O)NC(=O)C5)C4C3)c12 c1(C(=O)NC2C=CCN(C(CCSCCCC)=O)C2)cnc2cc(C)nn2c1C c1(CNC2(SC(c3nnnn3C)C)CC2)csc(S)n1.C(C)(C)(C)OC(=O)O N1(C(C(F)=CCC)=O)CC2CCN(C(c3cc(Br)sc3C)=O)CC12 c1(C(C)NC(C2N(C(C=C(C)C(C)C)=O)CCC2)=O)c(C)noc1C Cc1cc(C(=O)N(C)CC2CCCCN2C(=O)CCCNC(N)=O)nn1C C12(C(=O)NCC3CCN(C(C(C(C)OC)O)=O)C3)CC(C)(C1)OC21CCC1 CC1(C)C(CC(N2CC3CC2(C(N2CC(C)(O)C2)=O)C3)=O)CC1O C12(CNC(C(C)OCCOC)=O)CC(NC(c3cnsc3)=O)(C1)C2 C(c1ccc(C)cc1)=CC(N1CCC(CN(C(=O)C=CCF)CC)CC1)=O C1(CN(C)C(C2CC2F)=O)CCCCN1C(C1CCC(N2CCOCC2)CC1)=O N1(C(C(=O)Nc2cccc(-c3nc(C)[nH]n3)c2)=O)CCC(C2(O)CC2)CC1 C(CC(CC)C(=O)NCCCOCCNC(=O)CC1(C)CCOCC1)=CC Cc1cc(Br)c(NC(c2cnc(C(F)F)cn2)=O)cc1Cl C1(C(N(C2CN(C(c3cc(C)sc3)=O)CC2F)C)=O)CC(C)CCC1C(C)C C1(C(=O)NC(CC(C)C)CNC(=O)CCSCC(N)=O)CC2(C1)CS(=O)(=O)C2 N1(C(CCC2CCC(NC(C3(OC)CC3)=O)C2)=O)CCC12CC(C(N)=O)C2 c1(C(=O)NCC(C2CCCC2)NC(C(COC)(F)F)=O)cc2cc(Cl)sc2[nH]1 C1(C(N2CC(C(=O)OC3CCOCC3)C2)=O)OCC1(C)C.CC1CCC(=O)N1C c1(C(=O)NCC(CNC(c2c(C)cc(=N)[nH]c2)=O)O)ccnc2ccc(F)nc12 Cc1ccc(Cl)cc1C(=O)NCCCCC1CN(C(=O)C2=NOC(C)C2)C1 c1(N2CCCC(CCC=C)C2)cc[nH]c(=NCCC(C)P(C)(C)=O)n1 c1(CC)cc(F)ccc1CC(=O)NCC1CCC1NC(=O)C=C(C)c1ccsc1 c1(C(=O)NCC23C(CN(C(CNC(=O)NC)=O)C2)C3)cc(C)nc2ccnn12 c1(C(N2CCCC(NC(c3c(=N)cc[nH]c3)=O)C2)=O)cnn2c1OCC(F)C2 C1(c2ccc(OC)cc2)CC(C(=O)NCC2(O)CC(NC(=O)C=CSC)C2)=NO1 C(=O)(C1=CCCSC1)NC1(CCNC(C2(C)CS(=O)(=O)C2)=O)CC1 c1(-c2cn(-c3c(C)n(-c4ccccc4Cl)nc3)nn2)cccc2cccnc12 CCC(CN(C)C)C(=O)N1CCC(CC(=O)N(C(C)COCC)C(C)C)CC1 CC1CC(=O)NCC1C(N1CC(C)(C(=O)NCCSC(C)(C)C)C1)=O N1(C(C(C)(C)C)=O)CCN(C(=O)CN2CCN(C(C3CCOCC3)=O)CC2)CC1 c1(C(N2CC(NC(c3n(CC=C)ccc3)=O)C(O)C2)=O)ncc(N)cc1C c1(-c2ccc(C)cc2C)nc(-c2nc[nH]n2)nn1C1CCc2ccccc21 Cc1cc(C#N)cnc1C(=O)NC12CCN(C(c3ccc(CO)o3)=O)CC1C2 C(=O)(C(CC(C)C)NC(=O)CCC1(NC(=O)CC2CCCO2)CCC1)OCC c1(C(=O)NC(C)CCC(=O)O)c[nH]c2cc(C(=O)O)ccc12 C(CC(=O)N1CCC(NC(c2noc(C)c2[N+](=O)[O-])=O)C1C)(C(F)(F)F)OC N1(C(CCC)=O)CC(CNC(C2(c3ccccc3)CCOC2)=O)C(C)C1 C(=O)(CC(C)(C)C(=O)NCCC1CC(NC(c2c(C)nn(C)c2C)=O)C1)OCC c1(OC)cc(F)c(C(=O)NCCC(C)NC(c2ccnc(CO)c2)=O)c(F)c1F N1(C(CN(C(=O)OC(C)(C)C)C2CC2)=O)CCN(C(c2cccc(N)c2)=O)C2CC12 N1(C(c2c(CC)nn(C)c2Cl)=O)CCCC2(CCC(NC(=O)C=C(C)Cl)C2)C1 CC1c2ccccc2CC1C(=O)NC1(C)CN(C(=O)C2=CCCOCC2)C1 C1(C(N2C(C)CC(NC(c3cccc(C)c3N)=O)C2)=O)CCn2c(C)cnc2C1 c1(C(N2CCCC2C2CC2)C(=O)NC2(C)CC2)cnc(-c2cccs2)o1 C(N=c1[nH]c2c(c(=NC3CSc4ccccc43)[nH]1)COC2)C1C(Cl)C1 c1(C(=O)NC2C(NC(c3cc(C)on3)=O)CCC2)cc(C(C)(F)F)ccc1C C(=O)(C1=CC2C=CC1C2)NC1CCC(CCNC(c2c(C)nncc2)=O)C1 C=C(C)CCCC(=O)NCC1CCCCCN1C(=O)C(O)CCn1cncn1 C1(NC(C(C=C)(C)C)=O)CN(C(=O)CCNS(=O)(=O)CC)CC12CC2 N1(C(=O)CCc2nc[nH]n2)CCC2(CCCN2C(c2cc(=O)cc(Cl)[nH]2)=O)C1 C(CC(CC)C(=O)NCC1CCN1C(=O)COCc1cc(C)no1)=CC N1(C(C(C)=C2CC2)=O)CCOCC(NC(c2ccnn2CC2CC2)=O)C1 CC1(NC(C2CN(C3(C)CC3)C(=O)C2)=O)CCCN(C(C2CCC(F)CC2)=O)C1 C1(NC(C=CCC(C)(C)NC(=O)C=Cc2ccncc2)=O)CCC2CC1CO2 N12CC(C(O)C1)N2C.c1(COCCC=O)ccccc1.C1(C=O)CC=CC1 C1(CC(=O)NCCCNC(C(C)C)=O)C2CCCC2N1C(C1CCOC1C)=O N1(C(CC(CC)OC)=O)C2CCC1CC(C(=O)NC(CO)CCO)C2 C12(NC(CS(=O)(=O)N(C)C)=O)CCOCC1CN(C(c1ccc(C#N)cn1)=O)C2 Cc1cc(C(=O)NC2CCN(C(=O)C#CC3CCC3)CC2CO)n2nccc2n1 n1(CC)cnnc1CCNC(=O)C(F)CC1CN(C(C2(CN(C)C)CC2)=O)C1 c1(C(=O)NCC2CN(C(c3cn(CC=C)nc3)=O)C2)cccc(OCC(C)C)c1 c1(C(C)C)cc(C(=O)N(C(C)C(=O)NC2CC(n3cccn3)C2)CCO)n[nH]1 C1(CNC(=O)C=Cc2ccncc2)CC2COCC2N1C(C1CS(=O)(=O)C1)=O C(=O)(C(C#N)C(C)(C)C)NCCC1(C)CCN(C(=O)CC(C)(C)C(F)F)C1 C1(CC(=O)NC(C)CCC2CC2)CCOCC1.C1(=O)C(F)CC2CN1C2 C=C(C)C1OCCCC1C(=O)NCC12CCC(CC1)N2C(C1CC1C(N)=O)=O c1(C(N2C(CNC(CC(CC)OC)=O)CCCC2)=O)c(N)sc(C)c1C CC(C)C(C(C)NC(C1CN(C)C1)=O)NC(=O)CCn1cccnc1=O c1(C(=O)NCC(CCNC(C(C)CF)=O)O)cc2c(s1)-c1ccccc1OC2 CCC(CN(C)C)CC(=O)NCC1(F)CCN(C(c2ocnc2C(F)F)=O)CC1 C(C1CN2CC1C2=O)=CC.C1(NCCO)CCCC1.C(=O)COCCF c1(-c2nnc(N(C)NCC)n2CCOC)ccc(OC)c(OC)c1 CN(C)NC(=O)CCC(=O)NCCC1CC(C(N2CCCC3(CC2)CC3)=O)C1 c1(C(C)C)ccc(O)c(C(N2CC3CC3(NC(c3cccn(C)c3=O)=O)C2)=O)c1 c1(C(=O)NCC2CN(C(=O)Cn3cnc(Br)c3)C2)ccc(OCCF)cn1 N1(C(C(CNC(c2c(C)cccc2F)=O)C(C)C)=O)CCN2CCC1CC2 CC(N=c1nc2c(cnn2C)c(NCC2(CC#N)CC2)[nH]1)c1ccc(Cl)cc1F C#CCC(C(=O)N1CC(c2cc(O)no2)C1)NC(c1sccc1Cl)=O S(=O)(=O)(c1cc(C#N)ccc1C)NC1CCC(C(=O)NCc2c(C)nsc2)CC1 c1(C(N2CC(C)(NC(c3cc(C(C)=O)on3)=O)C2)=O)ccc(CC2CCC2)cc1 CC1(C)CC(NC(c2cnsn2)=O)CN1C(C1CCC(C(N)=O)CC1)=O CCCCC(O)CC(=O)NCCCN(C(=O)CC1COCCN1CC)CC c1(CNC(Cc2onc(C)n2)=O)ccc(Br)cc1.N12CCC1(C)C2=O C(=O)(CCC(CC)NC(=O)CCSC)NC(C=C)C CC(C(=O)NCC1(CNC(=O)CCCc2ccccc2)CC1)C(F)F C1(CNC(C(c2cccc(Cl)c2)C)=O)CCCCC1NC(=O)Cn1nnc(=O)[nH]1 C(=O)(CC1=CCOCC1)NCC(C(C)C)NC(c1ncoc1-c1ccco1)=O N1(C(C(CC)OC)=O)CCC(O)(C(C)NC(c2snc(O)c2Cl)=O)CC1 c1(C(N2CC(CNC(c3ccncn3)=O)CC(C)C2)=O)cnc2[nH]nnc2c1 C(=O)(CCCCCC#N)N(CC(C)C(=O)NCC=CCl)C N1(c2cc(N(C)C)ncn2)CCN(Cc2cc(I)ccc2O)C2CC12 c1(C(=O)NC(C)CNC(c2cscc2C(F)(F)F)=O)ccnc2[nH]ncc12 C=CCCCCCC(=O)NC1CC(C)(NC(=O)Cc2csc(C(F)(F)F)n2)C1 N1(C(C(CCC)N(C)C)=O)CC2CC(C1)N(C(=O)C(CC)c1ccccc1)C2 N1(C(c2csnn2)=O)CCCC1Cc1cn(C2CC2)nn1 C(CN=c1[nH]cnc(Cl)c1C#N)(C1CCCC1)NC(c1c(C)oc(CO)c1)=O C(=O)(NNC(=O)C(C)(C)c1ccccc1)c1c(CN(CC)CC)cccc1 C1(NC(c2cc(OC)ns2)=O)CCCN(C(=O)Cc2ccoc2)CC1 c1(C(N(C)CCNC(C2CCC23CCC3)=O)=O)cc2c([nH]1)CCCC2 c1(C(C)NC(C(CC)SC)=O)ccc(CNC(=O)CCc2ncc(C)[nH]2)cc1 S(=O)(=O)(c1cccs1)NC(C(=O)NCC(CO)NC(CC(C)CF)=O)C C(=O)(C(F)CCC(C)(C)C)N1CC2(C(NC(C(CCC)F)=O)CCC2)C1 C(=O)(C(C)(C)CCCNC(c1ccc(C(N)=O)[nH]1)=O)NCc1cnc(C)[nH]1 C1(C(N2OCC(n3cc(CNC(N)=O)nn3)C2)=O)CC12CCS(=O)(=O)CC2 N1(C(CN2CC(CC)OCC2)=O)CCS(=O)CC1c1ccc(C)o1 Cc1cc(-c2cn(C3CC(NC(C45CCC(CC4)CO5)=O)C3)nn2)ccc1N C1(C(=O)NC23CC(CNC(C4N(C)CC4)=O)(C2)C3)CCCC1C1CC1 Cc1c(NC(N2CCCC(C)(C(F)(F)F)C2)=O)cc([N+](=O)[O-])cc1C(F)(F)F N1(C(C(C2CCCC2)OC)=O)CCC(C(=O)NCC(O)C(C)C)(CF)C1 N#Cc1cc(CN2CCC(C(F)(F)F)CC2)cc(C(F)(F)F)c1 CCCC(C)(O)CC(=O)NC1(CCCNC(C2(O)CCC(C)(C)CC2)=O)CC1 C(=O)(CCCCCCCC1CC1)N1CCC(NC(c2c(OCC)scc2)=O)C(C)C1 c1(C(N2C(C)CCC(NC(c3cnc(CC)s3)=O)C2)=O)cnc2[nH]c(O)nc2c1 C1(OC)CC2(C1)CN(C(=O)C(CC(N)=O)NC(c1csc(F)c1)=O)C2 C1(NC(CC=CC=C)=O)CCN(C(c2cnc(C(F)F)c(C)c2)=O)CC1C CCCC(CCC)C(C)(c1nnnn1CCC1CC1)NC1CC2CC2C1 c1(C2N(C(c3ccccn3)C(=O)NCC)CC2)ccc(OC)c(OC)c1OC c1(C(=O)NC2CCC(SC)C2)c2c(nn1C)CN(C(=O)OC(C)(C)C)C2 C12(NC(c3c[nH]cc(F)c3=O)=O)CN(C(c3cc[nH]n3)=O)CC1CS(=O)(=O)C2 C(C1=CCN(C)CC1)NC(C1CCCN(C(C(C)SCC)=O)C1)=O C(CC(F)(F)C(F)F)(C(=O)N=c1nc(-c2ccccc2Cl)o[nH]1)OC c1(C(=O)NC2C(NC(C(c3cscn3)N(C)C)=O)C2)cccc2c1OCC2 C=C(C)CCCC(=O)N1CCN(C(c2cc(C(F)(F)F)cc(F)c2)=O)CC1C CC1CCc2n[nH]cc2C1C(=O)NC1CC(CCNC(c2ccc[n+]([O-])c2)=O)C1 c1(C(=O)NCCNC(C2CN(C(C3C(C)CC(=O)N3)=O)C2)=O)ccc2cc[nH]c2c1 C1(CNC(CC(C)(C)SC)c2nnnn2C2CCCCC2)CCn2ccnc2C1 N1(C(CNC(CC)=O)=O)CC(C)CN(C(=O)CC2CCCC2(F)F)CC1C c1(NC(C(c2cc(C)cc(Br)c2)N2CCC(O)C2C)=O)ccc2c(c1)OCO2 C1(F)(CNC(CC2CN(C)C2)=O)CCC(NC(=O)CCSCc2ccccn2)C1 Cc1ccc(C(=O)NC(C)(CNC(=O)C(O)Cc2ccc(Cl)cc2)CO)cc1C N1(C(c2c(OC)nc(C)cc2)=O)CCC2CCN(C(C3CN(C)C3)=O)C2C1 Cc1ccc(C(C)C(=O)NCCC2(NC(=O)CCc3cnc(O)[nH]3)CCC2)cc1 C(C(=O)NCC(CCNC(=O)CNC(c1ccccc1)=O)OC)(C(C)C)SC N#Cc1c[nH]c2ccc(C(N3CCC(F)(C(=O)Nc4ccc(Cl)cn4)C3)=O)cc12 CCC(F)(C(=O)OC)C(=O)NCC(C)CNC(C1(Sc2ccccc2)CC1)=O c1(CNC(C2C(SCC)C2)=O)ncccc1CNC(=O)C(COC)OC C1(CNC(CC(=C)C)=O)CC2CCC1N(C(C1CC=C(C)CC1)=O)C2 N1(C(C(CC)C(F)(F)F)=O)CCOC2CN(C(c3cc(C4CC4)no3)=O)CC12 c1(SC(C(N2CC(NC(C(CCCC)O)=O)(CO)C2)=O)C)nc2ccccc2s1 S(=O)(=O)(c1nc(N2CC3CCC(C2)C3O)ccc1Br)N(C)C c1(C(=O)NC2COCCN(C(C(CC)OCC)=O)C2)cnc2c(c1)CCC2 C(=O)(CS(=O)(=O)CCO)N(CC(C)NC(=O)CC1CC(C)=NO1)CC C12(NC(CCCC#C)=O)CN(C(=O)CCN3CCCCC3=O)CC1CS(=O)(=O)C2 c1(CN(C(=O)CC2CCC2)CCNC(C2CC23CCC3)=O)ccccc1 N1(C(c2cccc(N3CCOCC3)c2)=O)CC2CN(c3ccncn3)C2C1 C(C(C)(O)CC(=O)N1CC(n2cc(-c3ccc(N)cc3)nn2)C(C)C1)OC c1(CC(N2CC3C(NC(c4n(CC)ncn4)=O)(C3)C2)=O)ccc2occc2c1 C1(Cc2scc(C(=O)NCCN(C)C(C3CSCCS3)=O)n2)CCCCCC1 c1(OC)cc(C(N2CC(OC)C(NC(C3CC(OC)C3)=O)C2)=O)cc(N)c1O C(CC(C)CCNC(=O)Cc1ncc(C)s1)NC(c1c(CC)noc1)=O c1(COc2nccc(NC(C(=O)NC(C3CCCO3)C)=O)c2)nnc2n1CCC2 c1(C(=O)NCC2N(Cc3c(C)scn3)CCC2)nc2ccc(F)cn2n1 c1(OC)nc(N2CC3CC(NC(C4CCCCC4(C)C)=O)CC2C3)nc(C)c1F c1(C(N(C(CNC(C(C(CC)C)C)=O)C2CC2)C)=O)cccc2c1CCCC2 N1(C(C(C)(C)C(F)(F)F)=O)CCOC2(CCN(C(=O)C=C3CC3)C2)C1 C1(CC(=O)N(CCN(C(=O)C(=O)N(C)C)C(C)C)C)CCC(=O)N1C c1(C(N2CC(NC(CNC(N)=O)=O)CC3(C2)CC3)=O)nnc2ccccc2n1 C(=O)(C(C)CS(C)=O)NCC#CCNC(c1cc(CC)no1)=O c1(CNC2CC(NC(c3ccn(C(C)C)n3)=O)C2)ccc(Br)c([N+](=O)[O-])c1 Cc1nn(C)cc1CCC(=O)N(C)CC1C2CN(C(=O)CNC(=O)C3CC3)CC12 C1(C(=O)NCC2N(C(c3c(C)cco3)=O)CCC2)CC12CC(C)(C)C2 C(CC(C(=O)NCC(C)CC1CCC1)NC(=O)CC1CC(OC)C1)=CC c1(CNc2nccc(=NCC3(OCC)CCC34CCC4)[nH]2)cnn2ccncc12 N1(C2CCN(c3cn(C)nc3)C2=O)CCC(NC(c2cnoc2)=O)CC(C)(C)C1 N1(C(=O)NC2(c3cn(C)s3)CC(O)C23CCC3)CC2(CCCCC2)C1C(C)C N1(C(Cn2c(C)ccn2)=O)CCC(C(=O)NC(C)Cc2nncn2C)C1C CC(C)C(F)C(=O)NCC(c1ccc(F)cc1)NC(C12COCC1C2)=O Cc1cccc(C(=O)NC(C2(O)CN(C(=O)C(O)CN3CCOCC3)C2)C)c1F c1(C(N(CC(C)(C)NC(=O)Cn2nc(O)ccc2=O)C)=O)cc2n(c1)CCOC2 c1(C(N2C(CN(c3n[nH]c4c3CCC4)CC)CCC2)=O)cc(OC)cc(Cl)c1 N1(C(c2cc(C)nc(Cl)c2)=O)CCOC2(CCN(C(=O)C(F)(F)C(F)F)CC2)C1 CCC(CC(C)C)C(=O)NC1(C2CN(C(c3cncc(C)c3)=O)C2)CC1 N1(C(CCC2OCC(C)(C)C2)=O)CC2CCCC2(NC(c2c[nH]c(=N)s2)=O)C1 c1(NC(C2CCN(C(=O)CSc3nc[nH]n3)CC2O)=O)ccc2nc(Br)sc2c1 C#Cc1cc(C(N2CC(CCO)(NC(=O)CC)C2)=O)ccc1C c1(NC(C2CC2(C)C)CC)cc(NCCCN(CC(N)=O)C)nc(C)n1 C(=O)(CC1=CCOCC1)NC(C(C)NC(CCc1cccc(C(=O)NC)c1)=O)C CC(C)(F)CCC(=O)N1CC(C(=O)NC2CCC3(CC2)CC3)CC12CCC2 c1(OCC)cnc(C(N2CCC(CF)(NC(=O)CC(C)C3CC3)C2)=O)cn1 c1(C2(NC(C(=O)OC)CNC(=O)CCN3CCCCC3)CC2)ccccc1Cl c1(SC)cccc(C(=O)NCCCOC2CCN(C(c3cc(Cl)ns3)=O)CC2)c1 CCC(CCOC)C(=O)NC1CCCCCC1C(=O)NC(CN1CCCC1)CO c1(C(=O)NCCCCCNC(Cn2c(CCC)ncc2)=O)ncc(Cl)cc1Cl C(=O)(CCCC(F)(F)CO)NC(C)C(CO)NC(C1CCS(=O)(=O)CC1)=O C(=O)(CC1=CCOCC1)c1cn(C2C(C)(O)CCC2)nn1.C12CCCCC1NC2 c1(N(C(=O)CC2CCCN2C(=O)CCCNC(N)=O)C)ccccc1Cl C1(C(N(C2CCNC2)CCC#N)=O)CC2CNCC(C1)C2=O C(CC(=O)NC(CNC(c1cc(C(C)C)no1)=O)C(C)C)(OCC)OCC C(=O)(C1=CCC(NC(C2C=CCCC2)=O)C1)NCc1n(CCC)cnc1 c1(C(=O)NC2CCC2CNC(C2(c3cc[nH]n3)CCC2)=O)cc2occc2s1 CCC(CC(=O)NCC(O)CNC(=O)CC1CCN(C)C1=O)c1ccccc1 C1(C(=O)NC(C(=O)OCC)C2CC2)CCC2(CC2)N1C(c1cc(CC)nn1C)=O CCCN=C(NCCOc1cccc(C(C)(C)C)c1)NCC(C)C c1(CC(=O)NC(C)C(c2ccccc2)NC(C2CC(C)(C)C2)=O)cncn1C c1(C(=O)NC2C(C)CCN(C(=O)C(C)(C)N(C)C)C2)cc(F)c(F)c(F)c1 CC1CC(C(=O)NC(C2(O)CCN(C(=O)CNC(=O)NC3CC3)C2)C)CCO1 C1(NC(=O)C2=CCSC2)CC2CCC1N(C(=O)Cn1ccc3ccccc13)C2 c1(C(=O)NC(CCC(=O)OCC)C)sc2ccccc2c1Cc1nn[nH]n1 C1(C(=O)NC(C2CCCN(c3ccnc(C(C)C)n3)C2)C)CC(=O)CC12CCC2 n1(CC(=O)NC(CCN(C(C(CC)CN(C)C)=O)C)C(C)C)nc(O)ccc1=O N1(C(c2c(CC)cccn2)=O)CC(CNC(=O)CCC(=O)NC)C2(CC2)C1 C12(NC(CCC(=O)NC)=O)CCC1CN(C(=O)C(C)CO)C2 c1(CC(=O)NC2(COC)CN(C(CC3(OC)CC3)=O)C2)cccc2ccccc12 c1(CN2CC3C(NC(c4ncc(C)nc4)=O)C3C2)cc(Cl)c(O)c(Br)c1 C1(C)(c2cn(CCC(=O)OC)nn2)CN(C(C2COCCC2(F)F)=O)CCO1 C1(C(=O)NC2CCN(C(c3onc(CC)c3C)=O)CC2)CC2(CCCCC2)CO1 C(=O)(C(=O)CC(C)C)N(CCCNC(CCC(=O)NCCC)=O)CC C(=O)(CC(CC)C(F)F)N1CC(C(=O)NCC=CC)C(CCC)C1 Cc1cncc(-c2cn(CCc3ccc(N(C(=O)C(C)C)C(C)C)cc3)nn2)c1 C12(NC(c3c(C)coc3C)=O)CC3CCC(C1C2)N3C(c1cc(CF)on1)=O N1(C(c2c(N)sc(C)c2C)=O)CCCCC(NC(=O)CN2CCC(C)(O)C2)CC1 O=C(CN1CCCOC2CCCC12)N1NC2CC1C(O)C2O C(CN=c1[nH]c(C2CCCCC2)nc(=N)[nH]1)NC(COC1CCCC(C)C1)=O C1(C(=O)NCCCSCC)C2CCC(C2)N1C(c1c[nH]c(=N)c(C)c1)=O C1(NC(C(COC)NC(C(CC)N(CC)CC)=O)=O)CCCC1N=[N+]=[N-] N1(C(C2C(C)(C)C2(C)C)=O)CC2CCC(CNC(=O)CC(F)(F)Cl)C2C1 N1(C(C(CC(C)C)NC(C)=O)=O)CCC2(C1)CN(C(=O)CCC(=O)OC(C)(C)C)C2 C(=O)(CCC(O)C(C)(C)C)N1C2CC(N(C(C3N(C)CCCC3)=O)C)CC1CC2 N1(C(c2nc(C)c(C)[nH]2)=O)CCCC(CCNC(c2ccncc2F)=O)CC1 C12(NC(=O)NCc3ncc(-c4ccc(OC)cc4)o3)CCC(C(N)=O)(CC1)C2 N1(C(C(C2CC(F)(F)C2)OC)=O)CCC(CN(C(=O)CC2CC=CC2)C)C1 c1(C(C(N2CC=CC2Cn2cc(C3(CO)CC3)nn2)=O)O)ccc(F)c(Br)c1 c1(C(N(Cc2cn(Cc3cccc(C(C)C)n3)nn2)O)=O)cncc(Cl)c1Cl Cc1cc(C(N2CCC(C)C(NC(=O)COc3ccon3)C2)=O)c(C)nc1C Cc1ccc(CNC(C2CC23CC(NC(=O)Cc2csc(C)n2)C3)=O)cc1 C12(C(=O)NC3CCC(CNC(COCP(C)(C)=O)=O)C3)CCC(CC1)O2 C1(CNC(C(C=C)(C)O)=O)N(C(=O)Cc2ncc(CC)[nH]2)CCCC1(C)C N1(C(C2(CS(N)(=O)=O)COC2)C)CC2CN(c3nccc(C(F)(F)F)n3)CC2C1 N1(Oc2cn(-c3onc(CC)n3)nc2)CCN(C(C2CCC(Cl)CC2)=O)CC1 C1(C(N2CC(CCCCNC(Cc3ccc(C)s3)=O)C2)=O)CCOC(=O)CC1 c1(C(N(CCN(C(C)C)C(C2SCCC2C)=O)C)=O)cc(F)c(F)cc1Cl c1(COC)ccc(C(=O)NC(c2nc(C(=O)NC(COC)CO)co2)C)cc1 N(C(=NCCCCN(C)C)NCC1(NC(=O)OC(C)(C)C)CCCC1)C(C=C)C c1(-c2nnc(CNC(=O)NC(C3(N(C)C)CC3)C)o2)cccc(O)c1 N1(C(c2nc(C)[nH]n2)=O)CCC2(CNC(c3ccnc(O)c3)=O)CCCC12 C(=O)(C(CNC(c1ccc(F)c(C)c1)=O)C(C)(C)C)NCC1(COC)CC1 n1(CC)nc(C)c(C(=O)NC2CN(C(c3cncnc3C)=O)C3CC23)c1C C1(NC(COC(C)C)=O)CN(C(=O)CN2CC=CC2)CC1C c1(OC)ccc(CC(C)CNC(c2ccccc2-c2cncnc2)=O)cc1 c1(CC)cc(C(N2CC(CNC(=O)C(C)SC(C)C)(OC)C2)=O)c(C)nn1 c1(CNC(=O)COC(C23CCCC(C2)OC3)=O)cc2ccccc2o1 Cc1cc2ccc(C(N3CCC(O)(C(C)CNC(=O)CCC(N)=O)C3)=O)cn2c1 C1(C)(NC(C(N2CC(C)C2)C)=O)CCCC1NC(c1ccc(CCO)cc1)=O CC(CN(C)C)CC(=O)NCCC1(O)CCN(C(=O)Cc2ccn(C)n2)C1 c1(C(=O)NCCC2CCN(C(C3COCCO3)=O)C2)cccc2c1CCCCC2 N1(C(CC2CC(C)C2)=O)CC(NC(=O)COc2ccccc2)CC(C)(C)C1 Cc1scnc1C(=O)NC(C)C(C)NC(=O)C=CCN1CCCC1 C(C1C(C(N2CCCC2C(C)(C)NC(=O)CC2CCCC2)=O)C1(C)C)=C(C)C N1(C(CCC#C)=O)CCCC12CCCN(C(C1(CCO)CC1)=O)C2 C1(NC(C(C)NC(=O)C(F)(F)C2CC2)=O)CCN2CCCC12 C(=O)(CC(CC)C1CCC1)N1C(C(=O)NCC2CCN(CC)C2)CSC1 c1(C(=O)NCC(C)CNC(C2CCCC2C(F)F)=O)ccc2c(c1)NC(=O)CC2 c1(NCC(C)(C)C(F)(F)F)nc2ccccc2nc1NCc1ccc(F)cc1Br Cc1ccc2c(c1)CCC(C(N1CCN(C)CC1CNC(=O)C(C)CF)=O)O2 C(=O)(CN=c1[nH]c(N2CCC(CN(C)C)C2)nc(=NC)[nH]1)NCCC C1(NC(=O)CC(C2CCC2)C2CCC2)CN(C(=O)CC2OCCCO2)CCC1O c1(CC=C)ccccc1C(N1CC(OCCNC(=O)CC2(CC#N)CC2)C1)=O CC1CCN(CC(=O)NCC(C)(C2CCC2)NC(=O)Cc2ncc(Cl)s2)C1 c1(C(N2C(C(=O)OC)CCC2C(C)C)C(=O)NCCSC)ccc(C#N)nc1 N1(C(C)C)CCCC(C)(C(=O)NCCC2CCCC(C)N2)C1 N1(C(C(CC(C)C)O)=O)CC2(CCCCN2C(C2CCCC2C)=O)C1 c1(OCC(N2CC(C(C)NC(C3CC34CC(C)(C)C4)=O)C2)=O)cccc(F)c1F C(CC(C)C)(C(=O)NCC1(NC(c2ccc(C)s2)=O)CCCCC1C)OC C#Cc1ccc(C(N2CCCC2C(C)(C)C(=O)NCC2CCC2C)=O)cc1 Cc1nn[nH]c1C(=O)NC(C)(C)CN(C)C(C1CCCC1O)=O c1(C(N2C3C(CNC(CCC(C)SC)=O)C(C3)C2)=O)coc2ccc(Cl)cc12 C1(SCc2nc(C)on2)CN(N2CCC(c3cccc(Cl)c3)C2)C1 O(NC(=O)C(CNC(c1cccc(CN(C)C)c1)=O)C(C)(C)C)C(C)C C1(C(N2CCCCC2)Cn2cc(C3N(C)CCC3)nn2)OC(=O)CC12CCC2 C(C1CC1)(C1CC1)=CC(=O)NC(C(N1C(CCN(C)C)CCC1)=O)C1(O)CCC1 C(CC(=O)NC(c1snnc1C)C)(C(F)(F)F)NC(c1ccn(CCC)n1)=O c1(N(CC(C)CNC(C2CCOC(C)C2)=O)C)ncc(C#N)cc1F C1(O)(CNC(c2cc(F)cs2)=O)CCCN(C(=O)C=Cc2cnc[nH]2)CC1 N1(C(C(C)OC(C)=O)=O)CCC(C(N2CCOCC2C(F)F)=O)CC1(C)C N1(c2nnc(-c3c(C)cccc3)s2)CCC(F)C(NC(=O)OC(C)(C)C)C1 Cc1nc(-n2nc(COc3cccc(Cl)c3)nc2C2CCC2C)n(C)n1 CON1CCC(C(=O)NCCCN(C)C(C2CCC(C3CC3)C2)=O)CC1 C1(C(=O)NC(CO)CCC2CC2)CC(O)CN1CCN1CCCCCC1 N1(C(C2C(NC(c3cc(I)c(O)c(I)c3)=O)C2)=O)CCC2(CCCOC2)C1 C1(CNC(C2(COCC)CC2)=O)CC2CC(C1)N(C(=O)C#CC(C)(C)C)C2 c1(CC)ccc(C(N2CCC(O)C(N(C)C(C3CCCNC3=O)=O)C2)=O)cc1N C1(C(N2CCC(C(C)NC(C3CCCNS3(=O)=O)=O)C2)=O)CC2(COC(=O)N2)C1 C1(C(=O)NC2C3CCN(C(c4ccc(C)c(C)n4)=O)C32)CCCC(F)(F)CC1 c1(C(N2C3CCC2CN(C(C2CC2C2CC2)=O)C3)=O)ccc(F)c(F)c1Br C1(C(N2CCCC(C(=O)NCCc3cn[nH]c3)C2)=O)OCC2CCCC12 C(=O)(CC(CC)C(C)(C)C)NCCN(CCC)C(C1CC(C)(CC)C1)=O CN1CCN(C(C2CCC3(CC2)CC3)=O)CC1CNC(=O)C1=C(Cl)CCC1 c1(CC)cccc(C(N2CCCC2CN=[N+]=[N-])C(=O)NCCC#N)n1 N1(C(c2c(-c3ccc(C=O)cc3)cccn2)=O)CCC2(CCCO2)CC1 N1(C(C(C)C2CCCC2)=O)CC(N(C(=O)Cn2ncnn2)C)C2(CC2)C1 C1(C(=O)NC2(CNC(C3(O)CC(C)(C)C3)=O)CCC2)CC2(C1)CC21CCC1 CC(C)CC(O)CC(=O)NCCC(F)Cn1cc(-c2cc(Cl)cc(Cl)c2)nn1 c1(N2CC(CO)OCC2)nc(=NCC2CC3C(C2)C3(F)F)[nH]c2c1COCC2 N1(C(C2(C)CC(C)C2)=O)CCC(OCCCNC(C2CC(C(C)C)C2)=O)CC1 C1(C)(CC)CN(C(c2cc(-c3cccc(F)c3)on2)C(=O)NC(C)(C)C)CCO1 c1(SCC2(C(=O)NC3CCN(C(CC=CC)=O)C3)CCCO2)ccc(F)cc1 c1(C(=O)NCC2(CNC(C3(C)CS(=O)(=O)C3)=O)CC2)cccc2[nH]c(=N)oc12 c1(OC)ccc(C(=O)NC2(C)CCCN(C(=O)C(C3CC3)OC)C2)c(F)c1F c1(CCCC(N2CCC(CCNC(C(F)OC)=O)CC2)=O)nc2ccccc2o1 c1(C(N2C(CN(C(=O)Cc3nccs3)C)COCC2)=O)nn(C)c(Cl)c1Cl n1(CC(=O)NCC(CO)NC(c2occ(C)c2)=O)nnc2ccccc2c1=O C1(C(C(=O)N(CCCCC)C(C)C)C)CCCN(C(c2ccn(CC)n2)=O)C1 C1(NC(C(CO)OC)=O)CCOC(C(=O)NC(CO)C(F)(F)F)C1 C(CC(=O)NC(c1cn(C)cn1)C)(C1CC1)NC(CC=C)=O c1(C(C(CO)NC(C(c2ccc(F)cc2)C)=O)O)ccc(Br)cc1 N1(C(c2c(C)ncs2)=O)CC2CCC(NC(c3cc(CC4CC4)on3)=O)CC2C1 N1(C(c2c(CC)csc2)=O)CCN(CC(C)(C)NC(=O)C(C)CC2CCC2)CC1 CC1(C)CC(NC(C2(C)CC2(Cl)Cl)=O)CCN(C(c2nc(Cl)cs2)=O)C1 Nc1cccc(C(=O)NCC2CN(C(C3(C4CCC4)CC3)=O)CCO2)c1Br C1(C(=O)NCC(CC)(C)NC(=O)Cn2nccc2C)CCN(C(C)C)CC1 C12(NC(COC(CC)(C)C)=O)CCN(C(=O)CCOC3CCCC3)CCC1C2 c1(C(=O)NC(CC)CNC(C2(CC(C)C)CCC2)=O)oc(SC)cc1C Cc1nn(C)c(C)c1C(=O)NCC1CCN(C(c2ccc(F)c(Cl)c2)=O)CC1C N1(C(C2(CC(C)C)CC2)=O)CCC2(CC1)C(NC(c1nccn1C)=O)CS2(=O)=O N1(C(C2(OC)CC2)=O)CCCC(NC(c2c(C)nsc2N)=O)C1 CCCCC(C(=O)N(C1CCCCC1)CCNC(=O)CCN(C)C)C(C)C C1(C(N2CCC(CNC(C3CCCCC3F)=O)CC2)=O)CCC(F)(F)CC1 CCC(CC)CC(=O)N1CC2(CNC(=O)C3=NOCC3)CC1(COC)C2 c1(C(CN2CCC(C#N)(C(=O)OCC)C2)=O)n[nH]c2c1CCCC2 C(CC(O)CC(=O)N1CCN(C(c2ncc(C(N)=O)cc2Cl)=O)C(C)C1)SC C#Cc1ccc(NC(C2CCN2C(=O)CCCOc2ccccc2F)=O)cc1 c1(C(N2C(CNC(C(CSC)C)=O)CC(O)C2)=O)ccc(F)c(Cl)c1 CC1(O)CCN(C(=O)CC2(C)CCCN2C(=O)C(F)=CC2CC2)CC1 c1(C(c2nnnn2C2CC(F)(F)C2)NC(c2nccs2)CC)cnc(O)s1 C1(CC=CC)(NC(=O)C=CCCC(C)C)CCN(C(C2(C)CCC(C)C2)=O)CC1 c1(-c2nc(C(C)OCC)nn2-c2cc(C)ccn2)ccc(C)cc1CC C1(C(N2CC(NC(C(CC)OC3CCCCC3)=O)C2)=O)CCC2(CC1)CC(=O)C2 CCC(C)(CCNC(=O)CCOCc1ccccc1)NC(=O)C(C)C1CCC1 c1(OC(C)C)ccccc1C(=O)NCC(C)(O)CNC(=O)CC1COCCOC1 CC(C)C(CCN(C(=O)CCCn1cncn1)C)NC(C1CCN(C)C1C)=O C(CCC(O)C(=O)N1CCC1C1CCCCC1)NC(C1(C#C)CC(=O)C1)=O c1(C(N2CC3CN(C(c4c(C)cco4)=O)CC32)=O)c[nH]c2cc(Cl)ccc12 O=C(C1=CCCN(C(C2CCCCC(=O)N2)=O)C1)NC1CCn2ncnc2C1 c1(OC)ccc(C)cc1CC(N1CCN(C(=O)CC2CCSCC2)C2CC12)=O CC1CN(C(c2cnc3n2CCC3)=O)CC(C)N(C(c2cccc[n+]2[O-])=O)C1 N1(C(CCSC)=O)CCN(C(=O)C(C(C)(C)C)c2ccccc2)CCC1C C(=O)(C1=NOC(C)C1)N(CC(CNC(C(C(C)O)NC(=O)C1CC1)=O)(C)C)C C1(c2ccccc2)(NC(C2C(C(=O)NCc3scc(C)n3)C2)=O)CC2(CC2)C1 Cc1ccc(-c2cn(CCC3CC(NC(C4CC(CCO)C4)=O)C3)nn2)cn1 C1(C(=O)NC2CN(C(=O)CN3CSCCSC3)C2)CCC2(CCOCC2)C1 C1(CNC(c2cc(C)oc2)=O)CN(C(=O)CC2CCC(F)(F)CO2)CCC1(F)F C(CCN(C(=O)CCN1CCOC1=O)C)(C(C)C)NC(C(C)SC)=O N1(CCC(=O)NC(CN2CCC(C)C2)=O)CCN(C)CC1.C12(CC1)CC2 C1(C(=O)NCCNC(C2(CC#C)CCOCC2)=O)CCC(C(C)C)NC1=O CN1CCC(=CC(N2CCC(C(F)CNC(=O)C3CC3)CC2)=O)CC1 N(C1CCc2cc(CN)ccc21)C(CCC(=O)NCC)=O CC(C)(C(=O)NNC(=O)C1(S(C)(=O)=O)CC1)Oc1cccc(C#N)c1 CC1CC2CN(C(C)=O)CC12.C(CC(F)(F)F)N(CCC(=O)OC(C)(C)C)CC N1(C(C2(C(=O)OCC)CCO2)=O)CCC2(CC1)CC2NC(c1cc(F)n[nH]1)=O c1(C(N2CC(NC(C3C(C(=O)OC)CCCC3)=O)C2)=O)cc2c(s1)CC(C)(C)C2 N1(C(CC(CC)CC)=O)CCc2cc(CNC(=O)CNS(=O)(=O)CC)ccc2C1 CCCCS(=O)(=O)N1CCC(C(=O)NCC2CCO2)C1 c1(C(=O)NCc2ccc(C(=O)NCC3CC(OC)C3(C)C)o2)cncn(C)c1=O N1(C(COC2(C#C)COC2)=O)C(CC(=O)NCc2ccc(O)nc2)C2CCCC12 C1(C(=O)NC(c2ccnc(O)c2)C)CCN(C(=O)C2(CC(N)=O)CC2)O1 C1(C(=O)NCC2(CC)CCC2)(CC)CN(C(=O)Cc2cn(C)nn2)C1 c1(SC(C)C(=O)N(CC(C)O)CCNC(C2(C(C)(F)F)CC2)=O)ccccn1 C1(COC)(NC(=O)Cn2nnc(C)n2)CCCN(C(C2(O)CCC2)=O)C1 CCC(C)CC(C)C(=O)Nc1ccc(CCn2cc(C3CCCN3C)nn2)cc1 C1(C(N2CC(CCNC(CC3CC(OCC)C3)=O)C(C)C2)=O)(OC)CCCCCC1 C1(C(=O)NC2(CC(C)C)CC2)(NC(C2COCCO2)=O)CCC(C)(C)C1 Cc1cccc(C)c1C(=O)N(CC(C)CNC(=O)C(C)(C)c1ccccn1)C CN1CCN(C(C2COCC2C(=O)NC2CC(C)(C)CCO2)=O)C(CCO)C1 C1(CC)(NC(=O)CCC2CC(NC(=O)C(C)NC(=O)C3CC3)C2(C)C)CC(C)(C)C1 N#Cc1csc(CNC(C2(NC(=O)CC3CC4CCC3C4)CC(F)(F)C2)=O)c1 C(=O)(CC(O)CC(C)C)NCC1(C(=O)NC(C2CCOCC2)C#C)CC(C)(C)C1 c1(CC(N2CCC(NC(C(CC)(C)OC)=O)C2)=O)ccc(OC(C)=O)c(OC)c1 c1(C(=O)NCCN(C(C2CC(F)(F)CS2)=O)CC)ccccc1-n1ccnn1 C1(N(C(C(=O)NCc2nc(Cl)cs2)C2CC2(C)Br)C)CCCCC1 CCCCC(C)C(=O)N1CCC(CO)(CNC(C2(N(C)C)CCC2)=O)C1 C1(C(=O)NCc2ccc(F)cc2)CCCCCC1NC(C1CC2CC2C1)=O CN1Cc2cccc(NCC3CCC3NC(=O)OC(C)(C)C)c2C1=O C(=O)(C(CC(C)C)N(C)C)N(C(C)CNC(c1cnc(O)n1C)=O)CC N(C1CN(C(c2ccc[nH]2)=O)Cc2ccccc21)C(CC(C)C(C)(C)C)=O CCCCC(C)(F)C(=O)NC1CCCC1CNC(=O)C=C1CCC(C)CC1 C1(C)(COC)CC(NC(=O)COC(C)C)CN1C(c1ccn(CCN(C)C)n1)=O CC(C)S(=O)(=O)CC(=O)NC1CCCCC1CNC(C1CCCC12OCCO2)=O CCCCC(C)C(=O)NCC(C)=CC(=O)NC1CCCCC1(F)F CCCCC(=O)C(=O)N(C1C2CN(C(c3cscc3Br)=O)CC12)C Cc1oc2ccc(NCc3cc(C(=O)O)ccn3)cc2c1C N1(C(CC(C)N(C)C)=O)CCCC2CN(C(=O)CC(C)NC(N)=O)CC12 CCC(C)(C)CN=c1nc2c(ncn2C)c(NCC2CC(F)(F)C(=O)N2)[nH]1 S(=O)(=O)(c1cccc(C)c1C)NCC1CCCN(C(C(CC)C)=O)C1 c1(CN2C(C(=O)Nc3cc(Cl)ccn3)CC3CC32)cn2ccccc2n1 C(=O)(CCCCCCN=[N+]=[N-])N1CC(N(C)C(c2cc(=O)n3nccc3[nH]2)=O)C1 n1(CC)nc(C(=O)N(C)CC2CCN(C(C3CC4CC3C4)=O)C2)cc1C N1(C(C2(OC)CC2)=O)CC(CO)C2(C1)CN(C(c1nn[nH]c1C(F)(F)F)=O)C2 C1(C(N2CC(CS(C)=O)C2)=O)CCC2CCC1N2C(=O)CS(C)(=O)=O c1(C(N2CCC(CCNC(CS(C)(=O)=O)=O)C2)=O)ccc(Br)cc1N(C)C C1(C(C)(C)O)(CNC(CCNS(C)(=O)=O)=O)CN(C(=O)CCCF)C1 N1(C(C=Cc2cn(C)nn2)=O)CC2CC(NC(c3cc[n+]([O-])cc3)=O)C1C2 Cc1[nH]c(C)c(C(=O)NC(C)CN(C(=O)C(c2ccc(Cl)nc2)(C)C)C)c1C CCC(CNC(=O)C(CC(C)C)C(N)=O)N=c1nc(-c2ccc(OC)cc2)[nH]s1 C1(NC(C2C(OC)(OC)CC2)=O)CCC(NC(=O)CSc2nccn2C)CC1 C1(CC(N2CCOCC(NC(c3cocn3)=O)C2)=O)CCc2sccc2C1=O C(C(C)(C)C(C)(C)C)NC(CNC(CNC(C(C)C1CCCC1)=O)=O)=O N1(C(c2cnc(OC)nc2)=O)CCC(CNC(c2cnco2)=O)C(C)C1 C12(C(=O)NCC(CC)NC(=O)C=C3CC3)CCOC1CN(C(=O)NC(C)(C)C)C2 Cc1ccc(O)cc1C(=O)NCCOC(C)(C)CNC(C1CC2CCCC2C1)=O N(C(=NCC(c1cn(C)cn1)N(C)C)NCC1(C(F)(F)F)CC1)C(C)C C(CC(CNC(=O)C(C)Oc1ccccn1)NC(=O)C(C)(C)C)OC C(=O)(C1=NN(CCO)C(=O)CC1)NCC1(C(C)NC(=O)Cc2ccsc2)CC1 C1(CC)(NC(=O)Cc2cnc[nH]2)CCN(C(c2coc(C(C)C)n2)=O)CC1 c1(SCC2CCC(C(=O)NCC(O)CO)C2)cc(Cl)nc(Cl)c1 N1(C(C(C)NS(CC)(=O)=O)=O)CC(CNC(C2(C)CC(C)C2)=O)(OC)C1 C(CC(C)C)(C(=O)N1CCN(C(=O)COCC2CCCO2)C(C)C1)NC(C)=O Cc1cc(C=CC(N2CCC(CN(C(=O)CCc3cnc[nH]3)C)C2)=O)c[nH]c1=N C(=O)(C1=CCCCC1)NC1C(C)N(C(C2CCCO2)=O)CC1 C(N=c1cc(C)[nH]c(=NCC2CCCC2C)[nH]1)c1ncc(CC)o1 Cc1ccc(C(c2nnnn2C2CCCC2)NCc2ccc(Cl)o2)cc1[N+](=O)[O-] N1(C(C=CC)=O)CCN(C(c2ccc(C3CCCCC3)cc2)=O)C2CCCC12 N1(C(C(CC=C)NC(=O)OC(C)(C)C)=O)Cc2nncn2CC1C(=O)OC c1(OC(C(N2C(CCCNC(CCC=C)=O)CCC2)=O)C)cccc(C#N)c1 N1(C(C(C)NC(C)=O)=O)CC(NC(=O)C(C)(C)n2cncn2)CC12CCCCC2 C1(CC(=O)NC2CC(N(C)C(C34CCN(CC3)C4)=O)C2)CC2CC1C1CC21 c1(-c2ccc(C(N3CC4CCCC3CC4)=O)c(F)c2)cc(F)c(C(=O)NC2CCCC2)c(F)c1 Cc1ccccc1C(=O)NCC(=O)NCC12CC1CN(C(C1(O)CCSC1)=O)C2 C1(C(=O)NC23CC(NC(=O)Cc4cccs4)(C2)C3)CCC2(CC1)CNC(=O)C2 c1(NS(C)(=O)=O)cccc(C(N2CC3CC3(CNC(C3(O)CC3(C)C)=O)C2)=O)c1 N1(C(C(C(C)O)N(C)C)=O)CCC(C2CC2)(NC(c2ccc([N+](=O)[O-])[nH]2)=O)C1 N1(C(CCC2C(C)C2)=O)CC(C(N2CC(c3ccccc3)C2)=O)C2(CC2)C1 C12(CNC(C3C(CCC)C3)=O)CN(C(C3CC(=O)NC(C)C3)=O)CC(F)(C1)C2 c1(CC)ccc(C(=O)NC2CC(NC(C3(C)CCC3)=O)C2)cc1[N+](=O)[O-] c1(CC)cncc(C(=O)NCC(O)C(=O)NCC(F)(F)C(F)F)c1 c1(OC)cccc(Cl)c1C(=O)NC1CC1CNC(c1ccc(CSC)o1)=O C1(C)CS(=O)(=O)N1.C1(CC(=O)OC)(CC(=O)OCC)CCCC1 C(=O)(CCS(N)(=O)=O)NCC(CCCC)NC(C1CCC1c1nc[nH]n1)=O N(C1CCc2c(Br)cccc21)C(=O)CN1C(=O)C2CCCCC2C1=O C1(CC)CCN(C(=O)Cn2ncccc2=O)C1CNC(C1CC(F)(F)C1)=O c1(-c2ccc(C(=O)NCCC(C)(C)OC)o2)ccc(C(=O)NC2(CF)CC2)cc1 CCCCC(O)CC(=O)NCC1(CNC(=O)CCNC(=O)NC)CC1(F)F c1(CN(C(C2CCCN(C(CNC(C)=O)=O)C2)=O)CCO)cccc(Br)c1F C(=O)(CCN1CCCC1)NC.C1CCNC(=O)C2(CC2)CNC(=O)N1CC C1(OC)CC2CCC(C1)N2C(=O)CC1CCCC(NC(=O)CCC(=O)N(C)C)C1 C(CC(C)C)(C(=O)NCCCN(CCCNC(c1ccsc1Br)=O)C)OC CN1CC(O)CC1C(=O)NCC1CN(C(c2csc(-c3ncccn3)n2)=O)C1 CC1=NNC(=O)C1CCC(=O)NCC(O)CCNC(C1CCS(=O)CC1)=O c1(C(N(CCOCCNC(CC(C=C)C)=O)C)=O)cn2nc(C)cc2[nH]c1=O c1(C(N(C)CC2CCCN2C(=O)CC2CC2)=O)cc(OC(F)F)ccc1[N+](=O)[O-] C(=O)(C(F)(F)CO)N(C1CN(C(=O)CC2C(C)(C)C2(C)C)CC1O)C CC(C)(C)C(O)C(=O)NCC1CN(C(c2cccc(C(F)(F)F)c2F)=O)CCO1 c1(Cn2cc(C3(C)CN(C(CCCN(C(C)=O)C)=O)C3)nn2)cnnc(O)c1 c1(OC)cc(C)c(C(N2CC(CNC(c3cnsn3)=O)C(C)C2)=O)cc1OC Cc1cc2c(cc(C(=O)OCC(=O)CC3CCCS3)n2CC(F)(F)F)s1 c1(C(N2CC(NC(C(CC)n3cncn3)=O)C(C)C2)=O)cc([N+](=O)[O-])n[nH]1 CC(C)CC(O)C(=O)NC(C)(C(=O)NCC1(O)CC1)C1CCC1 c1(CCNCC(c2cccc(C#N)c2)O)c(F)c(F)c(F)c(F)c1F N1(C(C(CCC)C)=O)CCC(CO)C(NC(=O)Cc2ccc(Cl)cn2)C1 C#CCC(CC(=O)NCC1(C#C)CCCC1)NC(=O)COc1ccsn1 C1(C(N2C3(C=O)CC3CC2)=O)CCOCC12CCCCC2.c1(CC(C)C)c[nH]c2nccc-2c1 C1(CNC(c2cc(C)sc2)=O)CC(NC(C2CCN(CC(C)C)CC2)=O)C(O)C1 c1(CC)ccc(C)cc1NC(=O)C(C(C)C)NC(C1(C#N)CCCOC1)=O C12(C(=O)NCC3C(NC(c4cc(C)c(C)o4)=O)CCC3)CCC(CC1F)C2 N1(C(COCC(=C)C)=O)CC2(CCN(C(=O)C(C)c3ccsn3)C2)C1 C(C)(C)(C(C)CC(=O)N(C)C(c1ncccn1)C)NC(C(C)=C1CC1)=O c1(C(=O)NC(C(=O)NC(CC=C)C)C)cc2occc2[nH]1 C1(C(=O)NCCC)CCCN(C(c2ccn(C)c2CC(=O)O)=O)C1 N1(C(C2CCN(CC)CC2)=O)CC2CC(C(=O)NC3CCCCCC3F)(C2)C1 N1(C(c2ccc(COCC)cc2)C(=O)NCCCOC)CCOC(C(F)F)CC1 N1(CC(C)N(C)C)CCC(C)(C(N2CCN(c3ccccc3)CC2)=O)CC1 CC(C(=O)NCCOCC(=O)NCC1(Cl)CC1(F)F)C(C)(C)C c1(C(=O)NCCCN(C(c2cnc(SC)s2)=O)C)cc2cncn2c(O)n1 C1(NC(c2cn(C)nn2)=O)CCN(C(C2CCC(C(C)(C)O)CC2)=O)CC1O CCC(C)(C#N)C(=O)N1CCC(CCNC(C2(C(N3CCOCC3)=O)CC2)=O)C1 C(=O)(C1=CCCN(C(c2ccc3occc3c2)=O)C1)NC(c1ccc(C)nc1)C N1(C(CCC(=O)N(C)C)=O)CCC2(NC(=O)C=CCn3cncn3)CCCC12 O=C(C#CC1CCOCC1)NCC1CC(F)(F)CN1C(c1ccoc1Cl)=O N1(C(c2ccc(C(=O)O)cc2Cl)=O)CC2OCCN(C(C3CCCS3)=O)C2C1 c1(C(c2n(CC)nnn2)NCC2(C)CCOC2)cn(C)nc1-c1ccccc1 c1(NC2CCN(C(c3c(C)cc(C4CC4)nc3)=O)C2)ncnc2sccc12 CC1CCCCN1C(=O)CN1CCCC(CCNC(=O)CC(C)(C)C2CC2)C1 C1(C(=O)OC)CC2(CCNCC2)CN1C(=O)CN(C)C(N)=O C1(COC)(CNC(C2(C)CCOCC2)=O)CCCN1C(=O)C(c1cccnc1)F C1(C(=O)NC(C(=O)NCC(C#C)OC)CC2CCC2)CN2CCC1C2 Cc1cc(C(N2CCC(NC(=O)COCC(F)F)C(CO)CC2)=O)cc(=O)n1C N1(c2nnc(COC)s2)C(CNC(=O)CC=C(C)C)CC2COCC12 c1(C(=O)NCCCC(C)NC(c2nnn(CC)c2C)=O)cc(C)c(C(F)F)cn1 C(=O)(C1CCCc2cc(C#N)ccc21)NCCCN(C(=O)COCCOC)CC Cc1cccc(N(CCCC(=O)Nc2ccc(Br)cc2)C(N2CCSCC2)=O)c1F C1(C(=O)NC(C)CCNC(c2csc(S)n2)=O)CCCCN1C(N)=O CC(CC(N)=O)C(=O)N1CC(C(C)NC(c2cc3c([nH]2)CCC3)=O)C1 C1(CC)(NC(c2nnnn2CCC2(C)CC2)c2cncs2)CCCCC1 CC1CN(C(c2cccc(F)c2C2CC2)=O)CCCN1C(c1ccc(O)cn1)=O C1(CC(=O)NCC=CCC(N2CCN(c3cccc(Cl)c3)CC2)=O)NC(=O)NC1=O C1(O)(C(=O)NC(CCNC(CC(CC)C)=O)C)CCCC(C)(C)C1 c1(C(N(C(CCNC(c2ccc(C)[nH]2)=O)C)C)=O)csc2cncn12 C=CC1CN(C(=O)CCCCCOCC)CC1NC(c1cc(F)n(C)n1)=O N1(CC(=O)N(C(C)CNC(C2CC(C3CC3)C2)=O)C)C(=O)NC(C)(C)C1=O O=C(CCCCC(F)F)NCCC1CC(F)(F)CN1C(c1cnc(S)[nH]1)=O Cc1cnn2c1CN(C(C1COCCN(c3nccnc3N(C)C)C1)=O)CC2 c1(SC)ncc(N)c(C(=O)NC(CNC(c2csc3cncn23)=O)C(C)C)n1 C1(C(=O)NCC(CC)NC(c2cccc(Cn3ccnn3)c2)=O)CC(F)CN1C C(C)(CCCN=c1[nH]cc2ncnc-2[nH]1)NC(CCCc1ccc(OC)cc1)=O CCCCC(F)C(=O)NCC1(CO)CCN(C(=O)C(C)N(C)C)C1 c1(C(=O)NC2CCN(C(C=CCOC)=O)CC2C)ccc2c[nH]nc2c1 C1(NC(CC(C)OC)=O)C2CC1N(C(=O)CN1CCC(C)(O)C1)C2 N1(C(CC2CCC(OC)CC2)=O)CCCC2(C1)CN(C(C13CC(F)C1C3)=O)C2 C#CCCCC(C)C(=O)NCC(C1CC1)NC(c1cc(F)c(F)c(F)c1)=O N1(c2cc(CC)nc(CC)n2)CCC(C2(NC(=O)C3=CS(=O)CCC3)CC2)CC1 CC(CC1CC1)C(=O)NCCCOCCNC(=O)C(C)(C)c1nncn1C c1(C(=O)OCc2nnc(C3CCCOC3)o2)ncn2c1CCCCC2 c1(C(=O)NCCN(CC(F)(F)F)C)nc(Br)n2c1CCC2 N1(C(c2c(C)scn2)=O)CCOCC1CNC(=O)CN1CCC(F)CC1 Cc1ccc(S(=O)(=O)C2CCN(C(=O)NCCN(CC(F)(F)F)C)CC2)cc1 N1(C(CSCC)=O)CC2(C(N3CCC4(C3)CN(C(C)=O)C4)=O)CC1CCO2 CC1(O)CCCC1n1cc(CCC(=O)NC2CCOCC2O)nn1 N1(C(C(CN(C)C)NC(C(CC)=CCCC)=O)=O)CCCC1(C)COC c1(NC(C)=O)ccc(Cl)c(C(N2CCC(CNC(C34CC(O)(C3)C4)=O)CC2)=O)c1 CC1CCCC(C)N1CCC(N1CCN(C)C(CNC(=O)C(C)CN(C)C)C1)=O C1(C(C)NC(=O)C=CC(C)NC(=O)CCC(C)N(C)C)C(C)(C)C1(C)C C(CCC(CCC)NC(c1sccc1CC#N)=O)NC(CCSCCC)=O CCC(CC(=O)NCCOC1CN(C(=O)Cc2cc(=O)n(CC(C)C)[nH]2)C1)SC c1(CCC)[nH]nc2ccc(C(=O)NCCOCCCNC(C3CC3(F)Cl)=O)cc12 C(CN=c1[nH]c(N(CCCO)C)nc2c1CCCC2)c1cccc(OCC)n1 C12(NC(C3N(C(CC)=O)CSC3)=O)COCCC1CN(C(c1cc(C)co1)=O)C2 c1(CC(=O)NCC(C2CC2)NC(=O)C(c2ccccc2F)O)cnccc1Cl N1(CC)CCCC2C1CCCN2C(=O)CC(c1ccc(F)cc1)C C12(CNC(C(C)c3ccsc3)=O)CN(C(C3C(C)(C)C3(C)C)=O)CC(F)(C1)C2 C1(C(N2CCC(NC(C(C)(C)SC)=O)C2C(C)C)=O)CCC2(CCC2)O1 C1(C(=O)C(F)(F)F)CCN(C(c2nccn2-c2ccc(F)cc2)=O)CC1 CCCCC(C(=O)N1CC=CC(NC(c2cc(C(C)C)nc(O)c2)=O)C1)N(C)C c1(C(N2CCC(NC(C3CC=C(C)CC3)=O)C2)=O)ccccc1S(=O)(=O)C(C)C C1(C(=O)NCCN(CC(C)O)C(c2c(C)csc2)=O)CC2(C1)CC(F)C2 C=CC1CCCN1C(C1CC=CCC1C)C(=O)NCCOCC Cc1ccc(CNCCCNC(C2(F)CCN(Cc3ccco3)C2)=O)c(O)c1 c1(CNC(C2OCCC(NC(C(CC)C)=O)C2)=O)cccc(F)c1C C(CCC)(C(O)C(=O)N(CC)Cc1cn(C)nn1)NC(C(C=C)(F)F)=O C(=O)(C1=CC2C=CC(C1)C2)N1CC(CNC(c2c(N(C)C)cccn2)=O)C(O)C1 CCCCCC(C)(C)C(=O)NCC(CC1CC1)C(=O)N1CCCC(N(C)C)C1 C(=O)(C(CC)OC1CCCC1)NC1(CCC(=O)N(C2CCOC2)C)CCC1 c1(C(=O)NC(CC)CNC(=O)C=Cc2nccs2)ccc2c(c1)nc(O)n2C N1(CC(=C)Cl)C2CCC1CN(C(C1CCC(=O)N(CC)C1)=O)CC2 c1(C(=O)NCC(CC)NC(C(COCC)C)=O)cc(SC)nn1C N1(C(CN2CC(C)C2)=O)CCC(CNC(=O)CN2CCNC(=O)C2)C(C)C1 N1(C(C(C)SCC)=O)CCCC2(CCN(C(=O)C=Cc3ccc(Cl)cc3)C2)C1 n1(C(C)C)cnc2c(N(CC(C)O)C)nc(N(C)Cc3cnc(C4CC4)s3)nc12 c1(C(=O)NCC#CCNC(C(CC=CC)C)=O)c(C)[nH]c2ncccc12 c1(C(=O)NC(C23CCC(CC2)C3)CNC(C(COC)C)=O)ccnnc1O N1(C(COCCC#C)=O)CC2CCN(C(c3cc4nc(C)sc4[nH]3)=O)C2C1 c1(CN(C(=O)Cc2cn[nH]c2)C)ccc(CNC(c2ccc(Cl)s2)=O)cc1 N1(C(C(C)O)=O)CC(NC(C2(O)COC2)=O)CC12CCCCCC2 N1(C(C(C)SC)=O)CCC(C)(CCNC(c2cc(F)c[nH]2)=O)C1 C1(CNC(c2ccnc3[nH]ncc23)=O)CN(C(C23CC(C2)C3)=O)CCC1(F)F C1(NC(c2cc(CC)no2)=O)CN(C(=O)C(C)CN(C)C)CC2CCCC12 N1(C(C(SC)NC(c2cc(C(C)=O)[nH]n2)=O)=O)CCC2C(C(N)=O)C2C1 CCC1=NOC(C(=O)N(C2(C(=O)NCC(F)Br)CC2)C)C1 C(=O)(CC(O)CC(C)C)N1C(CNC(=O)CC2(CO)CC2)CC(OC)C1 CCCCC(CNC(=O)C=CS(C)=O)NC(=O)C(c1cccc(F)c1)(C)C c1(CC)cc(N2CCC(NC(c3cn(C(C)C)nc3C)=O)C(C)C2)nc(C)n1 CC(C)C(C)CC(=O)NCC1CCC1NC(c1c[nH]nc1-c1ccccn1)=O Cc1cc(C(=O)NC2CC(F)(F)CC2NC(c2cnns2)=O)c2ccccc2n1 c1(NC(c2cc(C)cc(Cl)c2)=O)nc2c(s1)CC(NC(=O)CCC#N)CC2 C1(O)(CNC(=O)C(CO)c2ccccc2)CCCN(C(C23CCC(CC2)O3)=O)C1 C1(COCC)(OC(C(=O)NCC)C2CCC2)CN(C(=O)CCNC(=O)C=CCl)C1 c1(C(N(CCCN(C)C)CCNC(C2CC2(C)C)=O)=O)cn2cccc(F)c2n1 CCCCC(O)C(C)C(=O)N1CCC(NC(c2cc(O)cs2)=O)C1 S(=O)(=O)(c1ccc(NCCC(C(C)C)NC)c(C#N)c1)NCCN(C(CC)C)C c1(C(=O)OC)cc(C(=O)NC23CC(CNC(=O)CN4CCNC4=O)(C2)C3)cn1C c1(C(=O)NC(C)CCCNC(=O)C(C)Cn2ccnc2)ncc(F)cc1N CC(C(C(=O)NC1CCC1)N1CCCC1C(N1CCCC1)=O)C1CC1 Fc1cc(Br)cc(CNC23CCCCC2C3)c1F C1(CNC(C(C)OCC)=O)CCN(C(=O)CN2CCC(=O)NC2=O)CC1(F)F Cc1ccc(C(=O)NC2CCCC2(C)CNC(c2nsnc2O)=O)cc1C C1(NC(C(C)(O)C2CCC2)=O)CC(F)CN(C(c2sccc2SC(F)F)=O)C1 C(=O)(CCCC(F)(F)F)NC(CCN(C)C)C(N1CCC(=C(F)F)CC1)=O C1(CC=C)(C(=O)N(CC(C2CCN(c3ncccn3)CC2)=O)CC)CCOCC1 C(CCS(=O)(=O)C(C)(C)C)NC(c1n(CCCSCC)nnn1)C(C)(C)C1CC1 N1(C(c2c[nH]nc2Br)=O)C2CCC1CC(n1cc(C3OCCO3)nn1)C2 Cn1cc2cccc(C(=O)NC3CC3CNC(c3cccc(N)n3)=O)c2n1 CC1CCC=C1C(=O)N1CCN(C(=O)CCCCN(C)C)C(c2ncc[nH]2)C1 c1(OCC)ccc(C)cc1NC(=O)C(N1CCOC(Cn2nc(C)cc2C)C1)=O C(N=c1nc2c(cnn2C)c(NC2CCOCC2C)[nH]1)c1c(CC)nns1 C(=O)(CCCS(C)(=O)=O)N1CC(CNC(c2onc(CC)n2)=O)OCCC1 CS(=O)(=O)c1ccccc1CC(N1CC(O)(CNC(C2(F)CCCOC2)=O)C1)=O C1(NC(C(C)OCC=C)=O)CCCN(C(=O)Cn2cc(CC)cn2)C1 c1(-n2c(C)ncc2)ccc(C(=O)NCC(O)CNC(C2(F)CC2C)=O)cn1 C1(CC(=O)OC)CN(CC(C)CC2CCC2)CC(C)(C)O1 c1(CC(=O)OCC)cnc(NC(c2nn(CC)nc2C)=O)nc1O CC1=C(C(=O)NC2CCN(C(C3CC4CCC3O4)=O)CC2(C)C)C(C)(C)CCC1 C=C(C)C1OCCCC1C(=O)NCC#CCNC(C1CCCCC1C(C)(C)C)=O C1(CC(=O)NC2C(NC(C3(C=C)CCC3)=O)CCCC2)CN2CCN1CC2 C(=O)(C1CCSc2ccccc21)N(CC(C)NC(C1CCN(C(C)C)CC1)=O)C N1(C(c2c(C)nn(CC(F)(F)F)c2Cl)=O)CCC(O)c2cc(Br)ccc2C1 C#CCC(C)C(=O)N1CCC(N(C2CC2)CC)C1.C12COCCN1NC2=O N1(C(C(CCN(C)C)NC(=O)CCN2CCCC2=O)=O)CC(S(C)(=N)=O)C1 c1(C(N(C2CCN(C(CC(C)F)=O)C2)CC2CC2)=O)cccc(Cl)c1 N1(C(CC2(OC)CCCC2)=O)CCCC(CCNC(=O)C(O)C(C)C)C1 C1(CC)CCC(NC(=O)CC(CNC(C2CC2c2cc[nH]n2)=O)C2CCC2)CC1 N1(C(=O)NCC2C(C(=O)OC)C2)CCCC2(CCCO2)CC1 CN1CC2CC1CN2C(C1COCCN1C(C1CCC2(CCC2)O1)=O)=O C1(C)(CNC(CCC=CC)=O)CCCN1C(C1CC1c1ccncc1)=O N#Cc1c(N2CCC3(CC2)CC3C(=O)NC2CCCC2C2CC2)cccc1F c1(NC(c2n(CC)nnn2)c2ccc(COC)s2)cccc(CCC(N)=O)c1 C(=O)(C(CCOC)OC)NC(C(=O)NC(C=C)(C)C)C1CC1 C1(NC(C2C(C)CCN2C(=O)Cn2cc(C#N)cn2)=O)CCC(C2CC2)C1 C=C=CC(C)C(=O)NCC1(OC)CCN(C(c2cc(C(C)C)no2)=O)C1 c1(CC)[nH]ccc1C(=O)NCCCC1CCCN1C(C1CSCCS1)=O CCC(C#N)C(=O)N1CCC(N2CCN(C(=O)Cc3csc(S)n3)CC2)C1 N1(CCC)CCC(OCCN(C(Cc2ccc(OC)cc2)=O)C)CC1 c1(C(=O)NCC(C)NC(=O)C(O)C2CC2)c[nH]c(C(F)(F)F)c1 Fc1ccc(N2CCN(Cc3nnc(C(F)F)s3)CC2)cc1 c1(C(N2CCC(N(C(C3CC(SC)C3)=O)C)CC2)=O)c(F)ccc2c1OCC2 C1(NC(CC2C(C)=NNC2=O)=O)CC2(CC(NC(=O)OC(C)(C)C)C2)C1 C12(C(=O)NC(C(=O)NC3CC=C(C)CC3)CC3CC3)CCN(CC1)CC2 C1(CNC(C=CC)=O)CN(C(C2CCC2(OC)OC)=O)CC12CC2 C=CCC(C)(C)CC(=O)NC1CC(CNC(c2cc(CC)no2)=O)C(O)C1 C1(NC(c2c(CC)noc2C)=O)CN(C(=O)C=Cc2cncn2C)CCC1C C(=O)(C(F)(F)C(F)(F)Cl)OC.C1(n2cc(C(C)(C)O)nn2)CCCN(C(=O)CO)C1 C(CCC(C(=O)Nc1cccc(CCO)c1)NC(C1CCOC(=O)CC1)=O)OC N1(C(C(C)=CC2CC2)=O)CC(N(C(=O)CCC2CCCCO2)C)C(C)(C)C1 C1(C)(C(=O)NCCN(C(C(C2CC(F)(F)C2)OCC)=O)C2CCCC2)CCCC1 n1(C(C2(C)CC2)C)nc(-c2ccccc2)nc1C1C2CCC12 c1(C(=O)NC2CN(C(=O)CCC3CCCC3)C2)c(Cl)cccc1Br CC(C)C(C)(CNC(=O)CCOC1CC1)NC(c1ccc(C(N)=O)cn1)=O CC(C)(C)CC(O)C(=O)NC(C)(C)CC(F)C(=O)N1CCCC(C)(CO)C1 C1(CC(=O)NCCN(C(=O)CCc2ccc(C)s2)CC)COCCN1CC C1(C(=O)NC2CN(C(=O)OC)C2)CCCN(C(=O)Cn2ccnn2)C1C C1(NC(c2scc(C)c2)=O)CCN(C(c2ccc(C(O)CF)cc2)=O)C1(C)C N1(C(CNC(CC)=O)=O)C2CCC1C(NC(=O)C(F)n1ccnc1)C2 N1(C(C2CCN(C(=O)CCc3cncnc3)C2)=O)CC2CCC(CC2)C1 C1(OC(C)C)CCCN(C(=O)CCCNC(=O)CC2C=NN(C)C2=O)C1 N1(C(CCSCCC)=O)CC(C)(C)CC1C(=O)NC1CN(C)CC1(C)C C1(CNC(=O)CCc2cnoc2)CCCC(NC(=O)C(C2CCOCC2)O)C1 c1(C(=O)NCC(C2CCN(C(C)=O)CC2)F)cc2c(Br)cc(Cl)cc2[nH]1 N1(C(c2c(C)csc2)=O)CCC2CCCC12CNC(=O)CCCCN1CCCC1 CCC1(CC)CN(CC2CC(CC(=O)OC)C2)c2ccccc21 Cc1ccc(SCC(=O)NC2CN(C(=O)CC3CC=CCC3)C(C)(C)C2)cc1C CC1CN(C(c2ccn(C3CCC3)n2)=O)CCC1NC(=O)Cc1nnc(O)s1 c1(C(=O)NCc2c(C)cc(-c3nn[nH]n3)cc2)nnc2cc(C#N)ccn12 C12(C(=O)NC(CC)CNC(c3cc(=O)cc[nH]3)=O)CCC(CC1(F)F)C2 c1(C(=O)NC(CCCNC(C(N2CCNC2=O)C)=O)(C)C)cnn2c1N(C)CC2 c1(N(C)C)ccc(-c2csc(C(N3CC(N4CCC(O)CC4)C3)=O)n2)cc1 N1(C(c2c(CC)nccn2)=O)CCC(CNC(C2CCCSC2)=O)C12CCC2 C(=O)(C(C(C)(C)C)OC)NCCCCNC(C(CC)CC1CCCCC1)=O c1(CC(=O)NC2CC(F)(CNC(C(CC)=CC)=O)C2)sc(-c2ccsc2)nc1C c1(C(N2C(C3(NC(C(C)=[SH]C)=O)CC3)CCC2)=O)oc(SC)cc1C c1(C(=O)NCCCN(C)C(C2CCCOC2)=O)cc(N2CCCC2)ccn1 CC(CCN=c1ccnc(NCc2ccc(N(C)C)cc2)[nH]1)C(F)F CCC(C)(CNC(=O)C(O)C1CC1)NC(c1cc(Cc2ccccc2)c[nH]1)=O N(C1CCCn2nccc21)C(=O)Nc1ncnc(OC)c1C C(=O)(CS(=O)(=O)CC1CCCO1)NCc1n(C)c(Sc2ccc(Cl)cc2)nn1 C#CC1CC2(CC(C(=O)NCCN(C(=O)CCN3CCCC3)CC(C)O)C2)C1 N1(C(CC2(C=C)CCC2)=O)CCC(NC(C2CCCN(CCC)C2)=O)C(O)C1 C#CCCCCC(=O)N1CC(NC(C2CCCC2C(F)(F)F)=O)C1 CC1C(C(=O)NCCc2c[nH]nc2O)CCN1C(=O)C(C1CCCCC1)=O c1(CCC)sc(C(=O)N(CCCNC(=O)CC(C)F)C2CC2)cc1Br C1(C(N(C(C)(C)CC(N2CCC(C)(CO)C2)=O)C)=O)CCCC2(CC2)C1 c1(OC)ccc(NC(c2cc(C3CC3)n(-c3ccccn3)n2)=O)cc1C CC1(C)CN(C(=O)C2=NOC(C)(C)C2)C(CNC(c2ccc(Cl)cn2)=O)CO1 CC(C)(C#N)CC(=O)N1CC(CO)(NC(=O)COc2cc(F)cc(Cl)c2)C1 C(=O)(C1=CC2(CCN(C(C3CC4(CC4)C3)=O)C2)C1)NCCCCC#C Cc1ncc(N)cc1C(N1CCC(NC(=O)C#CC(C)(C)C)C1C1CC1)=O C1(C(=O)NCCN(C(CC2CCN(C)C2)=O)CC2CC2)CCCNS1(=O)=O S(=O)(=O)(c1ccc(NCC2CSCCS2)c(C#N)c1)N1CCc2c(nc(C)s2)C1 CCCC(C(=O)NCC1CC(NC(C2CC(F)(F)CC2C(=O)OC)=O)C1)C(C)C C(=O)(C(O)CC(F)F)N1CC(C(C)NC(C2CC2[N+](=O)[O-])=O)C1 N1(C(C23CC(NC(C(COC)OC)=O)(C2)C3)=O)CCC(CO)C(O)C1 N1(C(C(C)Oc2ccc(COC)cc2)=O)CC2(CCN2C(C2CC2(F)F)=O)C1 N1(CC2(OCC)CCCOC2)CCC2(CCCC2)CC1 Cc1ccnc(C)c1C(=O)NCCC(O)CNC(c1cn(C)c(=O)cn1)=O C1(NC(CSCC#C)=O)CC(CC(=O)N(CCCC)CCO)C1 c1(C(=O)NC2CN(C(CCCC)=O)CC2c2ccc(F)cc2)cc(Cl)cnc1O N12CCCN(CC1)C(=O)C2.C12(NC(N3CC(CCCCOC)C3)=O)CCCC1C2(F)F C#CC1(NC(c2ccnc(CNC(C3CC3C)=O)c2)=O)CCC(C)(C)C1 C1(NC(c2cc(OC)no2)=O)C2CCC(C2)C1C(N1CCCCC1C(C)(C)C)=O C=CC(C)CC(=O)N1CCC1C(=O)NC(C)C(C)SC Cc1ccc(CCNC(c2ccc(-c3cn[nH]c3)cn2)=O)cc1 c1(Oc2ccc(C(=O)NCC3C(C)CCC3)cc2)cccc(F)c1F Cc1cnccc1CN(C(C1CCCCC1)C(=O)NCCC#N)C C1(CNC(CNC(c2c(C)occ2)=O)=O)CCC(C)N(C(=O)CC2CC=CC2)C1 c1(COC)nc(=NC2(CNC(c3c(C)ccnc3Cl)=O)CCCCCC2)s[nH]1 CC(C)CC(C(=O)N1CC(CCNC(=O)C(C)N(C)C)C1)c1ccccc1 C1(C(N(C)CC2CN(C(C3CCC(C)CC3)=O)CCO2)=O)CS(=O)(=O)CC12CC2 c1(C(=O)NC(CN(C(CC2(OC)CCCCC2)=O)C)C)ccnc2c1ncn2C c1(CSC)cc(N2CCN(Cc3cn(C(C)C(=O)N(C)C)nn3)CC2)ccc1F CC(CS(=O)(=O)N1CCC(NCc2ccc(Cl)cc2F)CC1)C(=O)O N1(C(C2CC(OC)C2)=O)CC(NC(=O)COc2cc(C)ccc2F)CC1(C)C Nc1c(C(=O)NCc2ncccc2CNC(C2CCNC2=O)=O)ccc(Cl)c1F c1(C(c2nnnn2CC)Nc2[nH]nc(OCC)c2C#N)ncc(Br)cc1OC n1(CC(=O)NC2CCCC(NC(c3c(CC)scc3)=O)C2)cc([N+](=O)[O-])c(C)n1 c1(NC(C2(c3c(-c4cccc(C)c4)cccc3)CC2)=O)cc(F)c(Cl)cc1Cl N1(C(c2ccc(C)cc2Br)=O)CCCC2CN(C(=O)C(C)(C)CO)CCC12 N1(C(CN(C(C2C(C)SCCC2)=O)C)=O)CCC2(C1)CN(C)C2 CCC(CC)CCCC(=O)N1CCN(C(=O)CCCNC(C)=O)C(C2CCC2)C1 C1(CCNC(=O)CC2CC3(CC3)CO2)CN(C(=O)CCOC2CC2)CCS1(=O)=O c1(CN)cncc(-c2csc(OC3CC3)c2)c1 CCCC(C)(C)C(=O)NCC(CCOC)NC(=O)CNC(c1ccc(C)cc1)=O c1(CC)ccc(F)c(C(N2CCC(NC(C3(F)CCOC3)=O)C(O)C2)=O)c1 N1(C(CCC)=O)CCCC(C(=O)NCC(C)CNC(c2ccc(C)cc2)=O)C1 C(C(=O)NOCC1CCC1)(NC(C(COC)OC)=O)SC N1(C(C(C=C)(C)O)=O)C2CCC1(CNC(c1scnc1COC)=O)CC2 C1(NC(CS(=O)(=O)NC)=O)COCCN(C(c2cnc(C(F)(F)F)s2)=O)C1 CCC(CCCC(=O)N(C1CCCCC1)CC1CC1)NC(=O)C(C)N(C)CC CC(CC(=O)NC1(CCNC(C2OCCC2(C)C)=O)CCC1)C(F)(F)F c1(C(C)NC(C(F)=CC)=O)ccc(CNC(c2cnn(C3CCC3)c2C)=O)cc1 C1(CNC(=O)NC(c2cnc(C)s2)C)CCc2nn(C)cc2C1 c1(CN2CC(NC(c3cc(F)ccc3C(F)(F)F)=O)C2)cc(Br)cc2[nH]ccc12 c1(C(N(CCCCCO)C)=O)ccc2c(c1)CN(C(=O)CN(C)C(C)C)CC2 CC1(C)CN(C(=O)C(C)(C2CCC2)NC(C2CC3CCC(C2)C3)=O)CCC1O n1(CC(=O)NC2C(NC(c3c(C)n(CCO)cc3)=O)CC2)c([N+](=O)[O-])cnc1C c1(C(=O)NCC23OCCC(NC(C4(C)CC4)=O)(C2)C3)cncc2c1CCNC2=O C(=O)(C1CCCc2cncn21)N1C(C)CCN(C(c2ccsc2C(F)F)=O)CC1 N1(C(CCOCCN(C)C)=O)CCC(NC(c2cc(C3CCC3)no2)=O)C(O)C1 C1(CNC(C(C)NC(COC)=O)=O)CCCCN1C(C1(c2cc[nH]n2)CC1)=O c1(NC(C(CCSCC)NC(=O)CC2COCCOC2)=O)cc(CC)cc(O)c1 C(CCC(O)C(=O)NCC(C)C(C)(C)C)NC(c1c(CCC)n[nH]c1)=O c1(C(=O)NCC2CCN(C(c3ccc(OC)cc3Cl)=O)C2)cc2sc(C)cc2s1 C=CC1OCCC1C(=O)N(CCNC(=O)C(c1cccnc1)OC)C1CC1 Cc1ncnc(NCC2(NC(=O)CC(C)C3CCCO3)CCCCC2C)c1C#N c1(OC)ccc(-c2cc(CN=C(NC3CCCCC3)NC3CCC3F)no2)cc1 n1(CC(C)C)cc(NC(C2(NC(C3CCCO3)=O)CCCC2)=O)cn1 c1(C(N2CC(O)(CCNC(CC3CCC(C)CO3)=O)C2)=O)cc2ccccc2[nH]1 C1(OC)CCCCC1S(=O)(=O)NCc1noc(-c2cccc(Br)c2)n1 c1(C(C)(C)C)ccc(C(=O)Nc2ccc(OC(F)F)nn2)cn1 C1(C)(CNC(C(C)NC(=O)CC2C=CCC2)=O)CC(F)(F)CN1C(=O)C=CCF c1(C(C)C)ccc(C(=O)NCC2(F)CC(CNC(C3CCN3C)=O)C2)cc1 c1(OCC#C)ncccc1C(N1CCC(C(C)NC(c2coc(CC)n2)=O)C1)=O C(=O)(C1CCCn2nccc21)N(C)CC1(NC(C(C(F)(F)F)OC(C)=O)=O)CC1 C1(NC(CCCC)=O)CCN(c2cc(OC(C)C)ncn2)CC(C)(C)C1 N1(C(=O)CC2(c3nn[nH]n3)CCC2)CCCC(Cn2ccnn2)C1 C(CCCCCCC(=O)N1CCC(NC(c2cc(C)ncn2)=O)C12CCC2)SC N1(Cc2scc(C(=O)OC)n2)CCC(C(C)C(=O)Nc2csc(C(F)F)c2)CC1 N1(C(C2CCC2NC(=O)C(c2cncnc2)C)C)CCC(F)(F)CC1 c1(C(C(=O)Nc2c(C)cccc2)N(C2CCC2)C2CC2)c2c(nn1C)CCCC2 C(=O)(C1CCCc2nncn21)N(CCN(C(=O)CNS(N)(=O)=O)C(C)C)C c1(C(=O)NC(C)CC2CN(C(c3ccnn3C3CC3)=O)C2)cc(Br)n(C)c1 CC1C(NC(C2CCS(=O)(=O)N2)=O)CCN1C(c1ccc(NC=O)cc1)=O C1(C(=O)NCCC2CC(C(N(C3CCSC3)C)=O)C2)CC2CCC1C2 c1(C(N2CCCCC2c2ccc(C)cc2)C(=O)NC)nc(O)sc1C C1(OC)CCC(C(=O)NCc2cc(C(=O)NCc3nnn(C)n3)n[nH]2)CC1 N1(CC(=O)NCc2onc(C(C)OC)n2)CCCCC1CCN N1(C(CCSCCCC)=O)CCCC(C)C1CNC(=O)Cc1ncoc1C c1(CC)nocc1C(=O)OCCNC(=O)CCN(C)CCO.N12CC(C1)O2 Cc1nc(=N)[nH]cc1C(=O)NC1CCCN(C(C2(C3CCCO3)CC2)=O)C1 C1(C(N2C(C(=O)NCC(C#C)OC)C=CC2)=O)C2CC(=O)CC12 O=C(C#CC1CCOCC1)NCC(CC1CCCC1)C(=O)NCC1CCSC1 S(=O)(=O)(c1ccc(Cl)c([N+](=O)[O-])c1)N(C(C1(C#C)CCCCC1)=O)CC=C c1(C(=O)OC)cc(CCNC(=O)CNC(=O)NCc2cc(C)on2)on1 c1(C(N2CCOCC(NC(C(CC)OC)=O)C2)=O)c(C)oc2nc(Cl)ccc12 N1(C(C(CCCC)NC(c2nnsc2N)=O)=O)C2C=CCC1CCC2 c1(C(N2CCC(O)(CCNC(C3ON=C(C)C3)=O)C2)=O)cncc(Br)c1C Cc1ccc(C(N2CCOCC(NC(C3C=CCCC3)=O)C2)=O)c(O)c1C c1(C(N2C(CN(C(C(CC)(C)C)=O)C3CC3)CCC2)=O)[nH]c2ccccc2c1Cl N1(C(C=CSC)=O)CCC2(CCCCC2NC(=O)CCNC(C2CCCO2)=O)C1 C(CC(C(=O)N(C(C)C(N)=O)C)NC(C1CC(C(C)C)C1)=O)SC C1(S(N)(=O)=O)(C(=O)NCC(CNC(C2(C)N(C)CCC2)=O)O)CCCC1 C1(CCNC(CCC(=O)OCC)=O)CCN(C(=O)Cc2cnc(C)[nH]2)C(C)C1 C1(C(=O)NCC2CCN(CCN(C)C)CC2)C(N)C2CCCC12 C1(CC=C)(C(=O)NCC(CC)NC(=O)COC2CC=CC2)CCOCC1 C1(CNC(C2(CNC(C=CC(C)(C)C)=O)CCC2)=O)CC2CCCC2C1 C(=O)(CCCCCCSC)NCC1(C(=O)NCCOC)CC1 Cc1c(CN2CCC3(CC3C(=O)NC(c3ccccc3F)C)C2)ccc(F)c1F CC(C)C(C)C(=O)N(C(CNC(c1csc(-c2cccc(Cl)c2)n1)=O)C1CC1)C C1(O)(CC(N2CC(CN(C(C(C)n3cnnn3)=O)C)OCC2)=O)CCCN(C)C1 c1(-c2occ(C(N(CC(C)NC(CN(C(C)C)C)=O)C)=O)n2)ccccc1Cl C1(C)(C(=O)NCC2CCC(NC(C=Cc3n(C)ncc3)=O)C2)CC(C2CC2)=NO1 C(=O)(CC1=CCCC1)NCC(CNC(C1(CC=C)CCOCC1)=O)C C1(C(CNC(c2cc(OC)no2)=O)C)CCN(C(c2cnn(C(C)C)n2)=O)CC1 C(=O)(C(C(C)C)c1cccnc1)NC1(CO)CN(C(CC(C)C)=O)C1 CCCCC(O)CC(=O)N1CC(N(C(=O)CN(C)C(N)=O)C)C(C)(C)C1 c1(C(N(CCn2cc(CNC3CCCNC3)nn2)CC)=O)cccc2c1OCC2C C12(C(=O)NC(CCC=C(C)C)C)C(NC(C34CCC(C3)C4)=O)C3CC1C2C3 CCCC(CC)CCC(=O)N1CC2CC(C(N3CCC(O)CC3CC)=O)CC2C1 C1(CCCNC(c2c(CC)csc2)=O)CCCCN1C(=O)Cc1c(C)cnn1C N1(C(CC(C)C(C)(C)C)=O)CCC(C2CC2NC(c2ccc(CO)nc2)=O)CC1 c1(CC)cn2c(C(=O)NC3CC(C)(NC(c4cnco4)=O)C3)cccc2n1 Cc1cc(NNC(=O)C2CC(OC3CCOCC3)C2)ccc1F CC#CCCCC(=O)NCC1C=CC(C(=O)NCCN2CCC(OC)C2)C1 C(=O)(C(C)(C)S(C)(=O)=O)NCC12C(CN(C(C3(C(C)C)CNC(=O)C3)=O)C1)CC2 Cc1[nH]c(C#N)cc1C(=O)NC1(C)CCCCC1C(N1CC2CC=CC1C2)=O C1(C)(OC)CCCN(c2nc(N3CCCC(C(F)(F)C(F)(F)F)C3)cc(C)n2)C1 N1(C(c2nn(CC)c(C)c2)=O)CCC2(CC1)CC2NC(=O)CN1CCCC1CO C(C)(C(=O)NCC1(CCNC(=O)C(C)OC2CCCC2)CC1)NC(C)=O S(=O)(=O)(c1ccccc1Cl)N1CCCC(CC(=O)NC2CCC(O)CC2)C1 N(C1COc2ccccc21)C(C1N(C(C=Cc2ccc(C)o2)=O)CCSC1)=O N1(C(C(N2CCC(O)CC2)C)=O)CCC2(CC1)CN(C(=O)Cn1nccn1)C2 c1(COC(N2CC(NC(C(COC)(C)OC)=O)C2)=O)cc(C)c2c(O)n[nH]c2n1 C1(CC)CCN(C(=O)C(C)Cc2ccoc2)C1C(=O)NCC1CC2(CC2)C1 c1(C(N(C2CCC(NC(c3ccc(F)s3)=O)C2)C)=O)ccc2nc[nH]c2c1 C(CCC(C)(C)NC(C1CC1C(F)F)=O)NC(CC1C(CC)C1)=O c1(C(=O)NC2CC(CNC(C(CSC)O)=O)C2)ccnc2ccc(Cl)cc12 CCCCCC(O)CC(=O)NC1CCN(C(=O)Cn2cnc([N+](=O)[O-])n2)C1C C1(CC(=O)N(C(C)C)C)CCCCC1NC(=O)C=Cc1nccs1 C(C(CC(C)C)C(=O)NCCCC(CO)NC(=O)C(C1CCCCC1)C)OC C1(Cl)(C(N2CC(OCCNC(CC3C(C)C3)=O)C2)=O)C2CCC(=O)C12 C1(CCCC)CN(C(c2cc(C)c(C)[nH]2)=O)CCN1C(C1C2COCC12)=O c1(C(N(C(CCNC(CCC(=C)Cl)=O)C)C)=O)cc(C#N)c2n1CCCC2 N1(C(C(CC)OC)=O)CC2(CC2)CC1CNC(=O)CCOCCOC(C)(C)C C1(C(N(CCN(C(C(COC)(C)O)=O)C)C(C)C)=O)CCCCS1(=O)=O c1(C(=O)OC)cn(CC(=O)NCC2CCC(NC(=O)CNC=O)C2)cn1 N1(C(C2C=CCCN2C(=O)Cc2ccns2)=O)CCCN2CCCC2C1 c1(C(=O)NC2C(NC(CCCCC=C)=O)C2)ccc(Cl)c(C)c1O O=C(CCCCC(F)F)NCC(C1CC1)NC(c1csc2nnsc12)=O CCC(C)C(CC(=O)NC(C)CCN(C)C)NC(=O)CC1C=NN(C)C1=O CC1C(C(=O)N(C)CC2CCCN2S(C)(=O)=O)CCN1C(=O)OC(C)(C)C c1(C(C(=O)NCC2(F)CC(NC(C(CC)F)=O)C2)=O)c[nH]c2ccc(F)cc12 c1(C(N2CC3C(C(N4CC(C)NC(=O)C4)=O)(C3)C2)=O)cc(F)ccc1C#N CCC(CCCC(=O)NC1CCN(C2CC2)C1=O)NC(c1csc(Cl)n1)=O c1(C(N(CCC(C(C)C)NC(C2(O)CCSCC2)=O)C)=O)c(Cl)ccnc1F C(=O)(CCCCCn1cnnn1)NCC(C(C)(C)C)NC(=O)COCC(F)(F)F c1(OC)ccc([N+](=O)[O-])cc1C(=O)NCC1CC1NC(=O)COC1CCCC1 c1(C(=O)NCCOCCCNC(=O)CC2CC=CCO2)ccc2ccncc2c1 N1(CC(=O)N(C(C2CC23CC3)=O)Cc2ccccc2Cl)CCN(c2ncccn2)CC1 N1(C(CCc2c(C)cccc2)=O)CC(NC(=O)C(O)c2cnc[nH]2)CC(F)C1 CC(CC1CCCO1)C(=O)NCCC1CC(NC(=O)CCC2(C)CC2)C1 N1(C(C(C)(C)OC)=O)CC2CCOCC2(NC(c2cc(C(C)=O)cn2C)=O)C1 N1(C(C(C)CCN(C)C)=O)CC2(CCOCC2)C1c1cn(CCCCF)nn1 N1(C(C(=O)NC(C)C)CC2CCOC2)CCOC2CS(=O)(=O)CC12 C1(NC(CNC(=O)NC)=O)C2CC3C1C3C2C(=O)NCC(CSC)OC C#CCN(OC)C(=O)C1C2CCN(C(c3cc[nH]c3CC)=O)CC12 C12(NC(CCN(CC)CC)=O)CCCCC1N(C(=O)C(c1ccccc1)=O)CC2 C(=O)(CC(CSC)NC(=O)C(O)CSC)NCC(CC)(C)O Cc1n[nH]c(C)c1S(=O)(=O)N1CCC(O)C(Nc2ncnc3ccccc23)C1 N1(C(c2cc(CC)on2)=O)CC2CC2(CNC(=O)C2=C(Cl)CC2)C1 CCCC(C)C(=O)NC1CN(C(=O)Cc2ccnc(OC)c2)CC1C C(=O)(CCP(C)(C)=O)NC1C(C)CN(C(c2cc(-c3ccc(Cl)cc3)no2)=O)C1 C12(CNC(c3cc(C#N)[nH]c3)=O)CN(C(=O)CC3CCOC3)CC1CS(=O)(=O)C2 c1(NC(C2CC(O)CN2C(=O)Cc2ccc(O)cc2)=O)c(F)ccc(Cl)c1F C1(NC(CN(C(C)=O)C)=O)CCN(C(C2CCCN2C(=O)C(C)C)=O)CC1O c1(OC)cnccc1C(=O)NC(C)CC1CN(C(=O)CC(C)n2cccn2)C1 C1(CC(N2C(COC)CC2)=O)C=CC(NC(=O)C(CO)OC)C1 C1(N(CCc2c(C)ccnc2)C)CCc2cc(Br)ccc2C1 c1(C(=O)NCC2C(C)(C)N(C(C3CC34CC4)=O)CC2)cccc(S(N)(=O)=O)c1 C(C(CC(C)C)C(=O)NC1CC12CC(NC(c1cccc3[nH]ncc13)=O)C2)OC c1(C(N2CCCC(O)(C3CC3)C2)C(=O)NCC(C)C)ccc2ccccc2n1 c1(CN(CCN(CCC(c2ccccc2)C)C)C)c[nH]c2cccnc12 N1(C(c2c(C)ncnc2C)=O)CCC2(CCCCC2NC(=O)CNS(N)(=O)=O)C1 C1(CC)(NC(c2nc(Cl)oc2C)=O)CCN(C(c2cccn2CC2CC2)=O)CC1 C(=O)(C1=CCCCO1)N(C(CCNC(C(CC)NC(c1ccccc1)=O)=O)C)C Cc1cc(C(N2CC(NC(=O)CCCCBr)C(F)C2)=O)nn1C C1(CNC(=O)CC2COCCO2)CC(O)CN1C(c1cc(CCO)on1)=O CC(C)C(F)C(=O)NC(C)(C)CNC(C1OCCO1)=O c1(C(=O)NC2CCC(N(C(=O)CN3CC(C)(C)C3)C)C2)nn(C)c2c1CCC2 C1(C(N(C2CCS(=O)(=O)C2)CC(CC)OC)=O)CCCCC1C(C)(C)C N1(C(c2cnn(C)c2C#N)=O)CC=C(CC(=O)NC2CCOC2(C)C)CC1 c1(CNC2CC(NC(CCC3CCC(C)O3)=O)C2)ncccc1Cl C1(C)(C(N(CC(O)CNC(C2(CC3CC3)CCC2)=O)C)=O)CCCN1C N1(C(CC2(COC)CCOCC2)=O)CC(C)(C)CC1CNC(c1n[nH]cc1F)=O c1(OC)ccc(C(N2CC(OC)C(NC(C3CCN3C3CCCC3)=O)C2)=O)cc1 C=CCC(CC)C(=O)NCCOCCNC(=O)Cc1c(C)ncnc1C C(=O)(C(C)CC(C)C(C)=O)NCC(CC(=O)NC(CC)CCO)O C=CCC(C(=O)NC(C)C(C)NC(C1CCC(CCC)CC1)=O)C(C)C C(C)(CCCCN=c1[nH]cncc1I)NC(C1CC2CC(OC)CC21)=O N1(C(c2n[nH]c(CC)c2Cl)=O)CCC(C)(C)C(NC(c2cnc(O)cc2C)=O)C1 C1(NC(CCS(C)=O)=O)CC2CC(NC(c3ccc([N+](=O)[O-])[nH]3)=O)CC12 C1(C(=O)NC2CCC(NC(C3C(C(=O)OC)C3)=O)CC2)CCC2(CCCC2)CC1 Cc1ccc(OCCCC(=O)NCC(C2CC2)NC(=O)C(C)CO)cc1C c1(C(N(CC(CNC(c2n(C(C)C)cnc2)=O)C)C)=O)ccc(C(C)(F)F)nc1 c1(C(=O)NC2CC(N(C(=O)C(O)CC3CC3)C)C2)c(F)cccc1[N+](=O)[O-] O(N1CCC(CC(N2CCCC(N(C(=O)C(C#N)CC)C)C2)=O)CC1)CC C1(O)(CC)CC(C(=O)OCc2ccc(CC(=O)OC)s2)C1 C1(CN(C(=O)CC2CNC(=O)C2)C)CC(F)CN1C(=O)CCc1c[nH]c(=N)[nH]1 N1(C(CCc2nnc(C)o2)=O)CCC(NC(c2ccc(F)c(Cl)n2)=O)C(F)C1 C1(NC(CCC(=O)N(C(C)C)C)=O)CC(F)(F)CC1NC(C1CC2(CC2)CO1)=O N(C)(C(=NCC(F)F)NCC1CC2C=CC1CC2)Cc1c(C)c(Br)ccc1 c1(Cn2c(N3CC(CC)OCC3C)nnc2-c2cc[nH]n2)cc2ncccc2[nH]1 n1(CC)cnc2nc(N3CCC(CN(C)C)CC3)nc(NCCCCO)c12 C(=O)(CC(C)(O)C(F)(F)F)N1CC(C)(C)C(NC(=O)Cc2ccco2)CC1 C(c1ccc(C)o1)=CC(=O)NC(C(=O)NC(C(=O)NCCC)C)c1ccoc1 c1(C(=O)NC2C(CNC(c3ccc(C(F)(F)F)c(F)c3)=O)C2)ncnc(O)c1Cl Cc1[nH]nc(C(=O)NCC2CC(NC(c3ccc(CN(C)C)o3)=O)C2(C)C)c1F N1(C(C2(COC)C=CCC2)=O)CCOC(CN(C)C(C2CC=CC(O)C2)=O)C1 C1(C(N2C(CO)CC(C)(C)C2)=O)CC12CCN(CC(O)CO)CC2 c1(C(N)=O)cc(C(=O)NCc2nocc2C(=O)NCCCC2CCCC2)n[nH]1 n1(CC(N2CCOCC(NC(c3nc(CC)[nH]n3)=O)C2)=O)c(C)cc(O)cc1=O C1(NC(C2CCC(=O)NC2)=O)CCCCCC1C(=O)NCCN1CCCC(O)C1 C1(C(=O)NC(c2cnn(C)c2)C)CCN(C(=O)Cn2c(C)ccc2C)C1(C)C C(=O)(CC1=CCN(C(=O)C(C)(CC)CO)CC1)N(CCCC=C)CC c1(-c2nnc(NC(C(F)=C(C)C)=O)s2)ccc(F)cc1 c1(C(N(C)CCOCCNC(=O)CC2CCOC2)=O)cc(Cl)ns1 CCC(CC(=O)N1CCC(C(=O)N2CC(O)CO2)C(C)(C)C1)C(C)(C)C S(=O)(=O)(c1cccc(=NCCC(C)CCCC(C)C)[nH]1)NC1(C=C)CCC1 c1(C(CC)C)nccc(=NCC2CCCN(C(=O)CCN3CCC(O)CC3)C2)[nH]1 c1(C(=O)NCC=CCNC(c2c(C(=O)OC)coc2)=O)cc(Cl)cnc1O C1(N(C(COCCCC(C)C)=O)C)CC2CC1N(C(c1cc(Cl)ns1)=O)C2 C1(CNC(c2cc(C)c(C)nc2)=O)CC2(CO1)CC(F)(F)C2 N1(C(CCCC)=O)CCN(CCCNC(=O)CC2CCN(CCNC)CC2)CC1 C12(CNC(Cn3ccc(C)n3)=O)CC(CNC(=O)CC3CC=CC3)(CO1)C2 C1(CNC(C(C=CC)O)=O)CCN(C(c2nc(C)c(C)s2)=O)C1(C)C C12(NC(C(=O)NCC)=O)CCN(C(=O)C(C)(Cl)Cl)CC1C2 c1(OC)cc(F)c(F)cc1CN1CCC(O)(C(=O)Nc2ccc(C)c(F)c2)C1 n1(CC)nnc(C(=O)NC2CC(O)C2CC(=O)NCC(CC)n2cccn2)c1C Cc1cc(N)ccc1C(N1CC=CC1Cn1cc(CCOC(C)C)nn1)=O C1(C(=O)NCC(F)Cl)CCCCCCN1C(=O)Cc1cnsc1 C=CC(O)C(C)(C)C(=O)N1CC2OCC(C(=O)N(C)CCOC)C2C1 C1(NC(c2cnc(C)s2)=O)CCC(C)N(C(c2ccc(C(F)(F)F)cn2)=O)C1 C1(CNC(c2c(OCC)cncc2)=O)CCN(C(=O)CCCCCSC)C(C)C1 c1(C(=O)NCC=C2CCN(C(COCCC)=O)CC2)ccc(C2=CCCC2)cc1 C1(COC)CC(OC)CN1C(C1C(c2cn(CCCC(=O)OC)nn2)C1)=O N1(C(C2N(CCC)CCCC2)=O)CCCC(CC)(NC(c2sccc2Cl)=O)C1 N1(C(C=Cc2nc(C)c(C)[nH]2)=O)CCC2(CCCC2NC(=O)C=CBr)C1 c1(CC(N2C(C)CC(CNC(C3(CC#C)CCCC3)=O)C2)=O)c(C)nn(C)c1C C(=O)(CS(=O)(=O)CCO)NC1CCC(N(C(CSCCC)=O)C)CC1 C1(NC(CC2CC(OC)C2)=O)CCCC(CNC(C2(NC(C)C)CCC2)=O)C1 S(=O)(=O)(c1cccc(=NC2CC(CC(N)=O)C2)[nH]1)NCC1COCC(C)(C)O1 n1(CC)nc(C(=O)NC2CCN(C(=O)C(CCOC)OC)CC2O)ccc1=O C=C(F)C1(CC(N2CC(C(=O)NOCC3CCCCC3)C(F)C2)=O)CCC1 N1(C(=O)Cn2cc(Cl)cn2)CCC2C(CCN2C(c2cn3cccnc3n2)=O)C1 c1(C(N2CC3C(NC(=O)Cc4cncs4)(C3)C2)=O)cccc2ncccc12 N1(C(c2c(C)nc(COCC)s2)=O)CCN(C(=O)CO)C(C)CC1C CC(C)CC(CNC=O)CC(=O)NC(C1CN(C(=O)CC2CCC3CC23)C1)C c1(OC)ccc(C(=O)NC2COCC2CNC(=O)CCN2CCCC2)cc1N C1(NC(c2cc(C)on2)=O)(CNC(c2cnc(N)c(Cl)c2)=O)CCCCC1C N1(C(c2c(CC)ncs2)=O)CCCCC(NC(C2(c3ccc(Cl)cn3)CC2)=O)C1 C1(F)(C(N(C)C)=O)CCC(CNC(=O)C(=O)NCC2(C(N)=O)CC2)C1 CC1CCc2[nH]c(=NCc3cn[nH]c3)nc(N3CC4C5CCC(CC5)C4C3)c2C1 N1(C(c2cc(C(=O)OC)no2)=O)CCC(O)(CNC(C2CCSCC2)=O)C1 N1(C(CC(C)OCc2ccccc2)=O)CCN(C)C(CNC(=O)CCC(N)=O)C1 CCC(C)C(C(=O)N(CCCNC(=O)CCCc1ccccc1)C)NC(N)=O c1(OC)ccc(C(=O)NCCN(C(=O)C(Cl)=CCl)Cc2ccc(Cl)nc2)cc1O Cc1cc(C(N2CCCC2CC(N2C3CCC2CC3)=O)=O)cc(C)c1C N1(C(CCSCCCC)=O)CCC2C(CCCN2C(=O)CCN2CCCC2)C1 c1(OC)ncc(C)cc1C(=O)NCCCC(C)NC(c1[nH]cc2c1CCC2)=O C(=O)(CC(CNC(=O)C(C(C)C)SC)C1CCC1)NC(CC#C)(C)C C(=O)(CCCNC(=O)CC1CC1(C)C)NC(CC)COC c1(CNC(=O)Nc2cc(-c3cccc(OC)c3)on2)cc(OC)nc(Cl)c1 CCC(C)C(C(C(=O)NC1CCCCC1)N1CCCC(N2CC(O)C2)C1)OC C1(C)(OC)CCCN(C(=O)C(CNC(c2ncccc2O)=O)CC(C)C)CC1 CS(=O)c1cccc(C(N2CCSCC2CCNC(C2CCCCS2)=O)=O)c1 C(CCN(C)C(c1cc(C)cs1)=O)(C(C)(C)C)NC(C(CCSC)O)=O N1(C(Cc2cn(CC)nc2)=O)CCC2(CC1)CC2NC(c1sncc1C)=O c1(C(=O)NCC(CC)N(C(=O)CCCCOC)C)cncc(Cl)c1 c1(OC)ccccc1-c1cnc(C2CCCN2Cc2ccc(C)s2)[nH]1 c1(C(N2CC(NC(CCC#C)=O)C3C2C3)=O)cnc2[nH]ccnc1-2 C=C1CC(C(=O)NCCC(=O)NC(C)(C)C)N(Cc2sc(C)nc2C)C1 c1(C(=O)NC2CCCN(C(c3n[nH]cc3Cl)=O)CC2)ccc(Cl)c(Cl)c1O N1(C(c2nn[nH]n2)CC)CCC(COC(F)F)CC1 N1(C(C(COCC)C)=O)CCC(O)CC1C(=O)NOCc1ccc(O)cc1 S(=O)(=O)(c1ccc2c(c1)CCCNC2)N1CC(C2CC(=O)NC2)OCC1 N1(C(c2ccc(C(C)C)cc2)=O)CCC2(C(=O)N3CC(O)CO3)CC2C1 S(=O)(=O)(c1ccc(CCC(=O)N(C2CCCC2)CC(C)O)cc1)NC C1(OCC(=O)N(C2CN(C(C(C)=C(CC)C)=O)C2)C)CCCC(C)C1 C1(C(C)NC(=O)CCOC2CC2)CCCCN1C(c1[nH]ccc1-c1cccs1)=O c1(C(C(=O)OCC)NCC)ccc2c(c1)OC(F)(F)O2.c12cccc(c1)C(=O)N2 N1(CC(=O)NC2CN(C(C(c3cccc(F)c3)C)=O)C3C2C3)CCCCCC1=O N1(C(CCOc2c(C)cccc2)=O)CC(CO)C2(C1)CN(C(=O)CSC(F)F)C2 c1(CC)cnc2ccccc2c1C(N1CCC(NC(=O)CC2CC2(C)C)CC1)=O CC(C)CC(CNC(=O)C(C)(C)C1CCOC1)NC(=O)CCc1cncc(F)c1 N1(C(C2(CC)COC2)=O)CC2CCC1C(CNC(C1CC(F)(F)C1)=O)C2 C1(CNC(CCc2cn(C)nn2)=O)CC12CCN(C(c1sccc1Cl)=O)CC2 CC1CCC(C)(C(=O)NC2C=CCN(C(=O)CCCF)C2)CC1 C(=O)(C1CCCc2ncccc21)N1C(CN(C(=O)CCC(C)(C)C#N)C)CCC1 CCC(F)(F)C(=O)NCCC1(NC(c2cccc(=O)o2)=O)CCC1 C12(CNC(c3c(F)ccc(C)c3)=O)CN(C(=O)Cc3ccnn3C)CC1CCO2 c1(C(=O)NCC(CNC(=O)C=C(Cl)Cl)C(F)(F)F)cc2ccccn2n1 Cc1sc(C(=O)NCCNC(=O)COc2ccc(F)cc2)cc1Br n1(CCCC)nccc1C(=O)NC1CCCC1NC(=O)CSC1CCCCO1 CCC(CC(=O)NCc1ncoc1CCNC(c1cn(C)c(SC)n1)=O)C1CC1 C1(C(=O)OC)CCCCCCN1C(=O)C(CC(C)C)ONC(=O)C(C)SC1CC1 C1(CC(=O)N(CCN(C(=O)COCC2CCCO2)CC)CC)C=CS(=O)(=O)C1 c1(C(C)C)ccc(F)c(C(=O)NCCC(C)N(C(=O)CCC2CC2(Cl)Cl)C)c1 c1(C(N(CC(=O)NCC(C)(CO)CO)CC2CC2)=O)ccc2nccn2c1 c1(SCCC(=O)NC2C(NC(CN3CCC(C)CC3)=O)CC2)ccc(F)c(F)c1 Cn1cc(C(=O)N(C2CCN(C(=O)CC3CCC(O)C3)CC2)CCO)ccc1=O C12(C(N3CCCC(C(=O)NC(CC=C)CC)C3)=O)CC(C)(CCO1)C2 c1(OC)nn(C)cc1CNC(=O)C(Cn1cccn1)NC(=O)CCSC C1(NC(C(C)Cn2cccn2)=O)CC12CCN(C(C1CC(F)C1)=O)CC2 C1(CC#C)(C(=O)NC2COCC2SC)CCN(C(c2cncs2)=O)C1 C1(CC(=O)NCC(C)(CO)NC(C(N2CCOCC2=O)C)=O)CC(=O)NC1=O c1(C(N(C2CN(C(=O)CC3CCC3)CC2O)C)=O)cccc2cn(C)nc12 c1(N2C(=O)CC(C(=O)NC(C(=O)OCC)CC)C2)cc(C)ccc1OC N12CC3C(C3C1)CC(=O)OOCCNC2=O.Cn1cc(OC2CCOC2)cn1 Cc1ccnn1C(C)C(=O)NCC1(C(=O)NC2(CF)CCC2)CCCO1 C1(C(=O)NCCC(=C)CNC(=O)C(F)CC(C)C)CC2(CCCCC2)S1(=O)=O CCCCC(CNC(=O)CCc1ccon1)NC(=O)CCC1CC1(Cl)Cl NC(=O)CC(C(=O)N1CCC1C1CCCC1)NC(C1CCC2(CCC2)C1)=O CN1CCC2(CCN(C(C3CCC(CNC(C4(C)CC5CC5C4)=O)C3)=O)C2)C1 N1(C2CC(C(=O)NCC(C)N(C)C(c3cnc(Cl)[nH]3)=O)C2)CCCS1(=O)=O CC#CCCCC(=O)NC1CCC(NC(c2cn(C3CCOCC3)cn2)=O)CC1 c1(SCC(=O)NCC(C2CC2)NC(C(F)=CC)=O)nnc(S)s1 C1(CN(C)Cc2ccc(N3CCCC3)o2)CCc2cc(I)ccc2O1 CCC(C(=O)N1CCC1CNC(=O)C(=O)N(C)C)N1CCCC1=O CC(C)(CO)C(c1ccccc1)NC(=O)C=CCNC(C1(F)CC=CCC1)=O C1(OC)(OC)CC(C(=O)N(C)CCOCCNC(c2ccsc2Br)=O)C1 Cc1cc(C(=O)NC2CCCN(C(C3(C)CC4(CC4)C3)=O)C2)ccc1O Cc1cccc(CC(=O)NCCNC(c2n[nH]c3c2COC3)=O)c1F Cn1nc(C(=O)NCC2CCN(C(=O)CN3C(=O)CCC3=O)CC2)cc1C(F)F c1(COOC)ccc(C(=O)C(C2CN(C(CC(CC)O)=O)CC2C)=O)cc1[N+](=O)[O-] C(=O)(C#CC1CCCC1)N1CC(NC(Cc2c(C)nn(C)c2Cl)=O)C(C(F)F)C1 CCC(C)C(CC(=O)NCCC(C)C(C)(C)C)NC(C1(CC)CCC1)=O c1(OC)c(CN=c2[nH]cc(CNC(C3CCN(C(C)C)CC3)=O)s2)cccc1C c1(C(N2CC3C(C(=O)Nc4cc(C)no4)C3C2)=O)nc(C)ncc1Br Cc1ccc(Br)cc1S(=O)(=O)N1CC2CN(C(=O)CN3CCOCC3)C2C1 c1(C(=O)NCCCN(C(=O)COCCF)C(C)C)sccc1-c1ccccc1 N1(C(CC(C=C)C)=O)CC(C)(C)OCC1CNC(c1nn(C)cc1SC)=O c1(C(CNC(CC)=O)NC(c2cc(C(=O)OC)nn2C)=O)cccc(C)c1 C1(NC(c2cc(C)no2)=O)CCC(C)N(C(=O)CCOc2ccc(F)cc2Cl)C1 CC1(C(=O)NCCOCCNC(c2ccn(C(F)(F)F)n2)=O)C=CCC1 C(C(=O)NC12CC(C)(C1)C2)(C(C)(C)C)NC(CC1(C)CC1)=O c1(CNC(=O)Cc2ccc(Br)c(O)c2)ccc2occc2n1 c1(C(=O)NCCN(C(C(C)SCC)=O)CC)oc2ccc(Cl)cc2c1C C1(NC(c2cccc(CC)n2)=O)CCCN(C(=O)CC(CC)C2CC2)C1C C(=O)(CCS(C)=O)N(C1CCN(C(=O)C=Cc2cn(C)nn2)C1)CCC C(=O)(C1=CCS(=O)(=O)C1)NC(C)C(CO)NC(=O)Cc1cc(F)cc(F)c1 c1(CCC(=O)NCCNC(C2(C)C(C)(C)C2)=O)ccc2c(c1)OCO2 N1(C(C(C)OCCOC)=O)CC(O)(CCNC(=O)C(C(=O)OC)NC(C)=O)C1 C1(C(N2C(CN(C(c3n(C=C)ncc3)=O)C)CC(F)C2)=O)CN2CCN1CC2C C(=O)(NNc1ccc(F)nn1)c1c(C)nn(C)c1C N1(c2n(CC)c(C#N)nn2)CC2CCC(C(=O)NOC=CC(C)(C)[N+](=O)[O-])(C2)C1 c1(CN2CCC(CCCCCNS(CC)(=O)=O)CC2)ccc(O)cc1F.C(C)(C)O c1(C(=O)NC2(C)CN(C(C(C)CF)=O)C2)ccc(N2CCC(C)C2)cc1 CC(c1cccs1)=CC(=O)NCCC1CSCCN1C(C1CCC(F)CC1)=O Cc1ccc(C(=O)N(CC(C)CNC(=O)C(C)(C)NS(C)(=O)=O)C)c(C)c1 N1(C(=O)CN2CCOC2=O)CCC(CO)(NC(=O)COC2CC2)CC1 c1(C2(C)CC2)cc(C(=O)N(C2CCCC2N(C(=O)Cc2cc[nH]n2)CCO)C)no1 N1(C(CCn2c(C)ncc2)=O)CCN(C(c2csc(C)c2C)=O)C(CC(F)F)C1 c1(C(=O)NC2C(C(C)(C)C)N(C(C3CC3(Cl)Cl)=O)CC2)cnc2ncccn12 C#CCCC(O)CCNC(C1C(O)CCN1C(=O)C(c1cccn1C)=O)=O C1(C(N2CCC(N(C(=O)C(Cn3cccn3)NC)CC)C2)=O)CCCCN1N=O N(C1c2ccccc2CC1NC(c1csc(S)n1)=O)C(C1C(C(C)O)C1)=O c1(NC(C2CC(F)CN2C(c2cc[nH]c2)=O)=O)cc(Br)cc2cc[nH]c12 C=CC1(CC(=O)NC2CN(C(=O)C(C3CCC3)C3CCC3)CC2C)CCCCC1 N1(CCCC)CCN(CC(C(=O)CC2CC3CCC2C3)=O)C(=O)C1.OC C#CC1(NC(C2CCOC2CNC(=O)C(C)(CO)OC)=O)CC(F)(F)C1 CC1CN(C(C2CC2(F)F)=O)CCN1C(=O)C(c1ccccc1)C c1(C(=O)NC(C)CNC(=O)C(C)NS(C)(=O)=O)occc1Cl Cc1cccc(CN(C(=O)C(C)C)Cc2cccs2)c1 Cc1ccc(N(C(=O)C(C)CN(C(=O)C(C)n2cncn2)C)C)cc1C C1(C(=O)NCCN(C)C(c2cnn(C(F)F)c2)=O)CCCCC1P(C)(C)=O [N-]=[N+]=NC(CCC(N)=O)C(=O)NCC1CCCN1C(C1CCc2nncn2C1)=O C1(NC(C2CCCN(C(CC(C)C)=O)C2)=O)CCCCCC1C N1(C(c2ccn(C(F)F)n2)=O)CCCC2C1CCN2Cc1cc(I)ccc1Br c1(-n2c(C)nnc2)ccc(C(=O)NC(C)CCNC(=O)C(C)n2cncn2)cc1 Cc1cnc(Cl)cc1NC(=O)NC1CCC1C N1(S(CC)(=O)=O)CC(O)CC1Cn1cc(Cn2nc(C)cc2C)nn1 n1(CCNC(c2n(CC)nnn2)c2cnc(C(F)F)s2)nc2ccccn2c1=O Cc1ncc2n1CCC(C(N1CCC(N3CCC(NC(=O)CCF)CC3)C1)=O)C2 Cc1cc(I)c(F)cc1NC(C1CCCC(NCc2cccc(CO)n2)C1)=O c1(NC(=O)C(O)CNC(=O)COCC2CC2)ccc(O)c(F)c1 C=CC(CC)CC(=O)NCC1CCCCN(C(=O)CN2CCN(C)CC2)C1 C1(NC(CSC)=O)CCC(C)(CNC(c2sc(C3CCCO3)nc2C)=O)CC1 N1(c2[nH]c(=N)c3c(n2)CCC3)CCC23CCCCC2(C1)C3(F)F c1(-c2c(C(N(C)CCNC(C3CC3F)=O)=O)cccc2)cccc(C#N)c1 C1(C(=O)NCc2ccnc(F)c2)C2CC(O)C(C2)N1C(C1CCCSC1)=O C1(C(N2CC(O)(C(C)NC(c3cc(C4CC4)[nH]n3)=O)C2)=O)CN(CP(C)(C)=O)C1 C(=O)(CC(C(C)C)C(C)C)N1CC(NC(c2c(C)nc(COCC)s2)=O)C1 c1(C(=O)OC)cnc(N2CCC(C)C2CNC(=O)C(c2c(C)n[nH]c2C)C)nc1 C=CCC(CCCCC)C(=O)NC1(COC)CCN(C(=O)CCC(=C)C)C1 c1(CC(N2CCC(N(C(=O)CCN3CCOC3=O)C)C2)=O)ccc(F)nc1 N1(C(CC(C=C)CC)=O)CCC2CN(C(=O)CCc3cnn[nH]3)CC2C1 CC1CN(C(C2(CC(F)F)CC2)=O)CC(CCNC(=O)CC2CCCC3CC23)O1 N1(C(C(=CC2CCCC2)C)=O)C2CC1CN(C(=O)C(C)n1cccn1)C2 C1(C(N2CC(CNC(C3CC4C(C3)C4(F)F)=O)C2)=O)Cc2ccncc2C1 c1(CC(N2CCCC(Cc3c(C)cccc3)C2)=O)c(Cl)ccc(O)c1Cl c1(CC(C(=O)NCCC(=C)CNC(c2cnc(C)[nH]2)=O)C)c(C)nn(C)c1C C12(CNC(CC3(C)N(C(CNC(C4C(C)C4)=O)=O)CC3)=O)CCC(CC1O)C2 N1(Cc2cn(C)c(=O)cc2)Cc2n[nH]cc2CC1C(=O)OC C1(C(N(C(c2ccccc2)CC)CCC)=O)C=CCNCC1 c1(C(N(C(C)CNC(=O)CCP(C)(C)=O)C)=O)sc2cc(F)ccc2c1Cl N1(C(c2ccc(F)c3c2CNC3)=O)CCS(=O)(=O)CC12CNC2 CC1=NN(C)C(=O)C1CC(=O)NCCCCNC(c1sc(C(C)(C)C)nc1C)=O c1(C(=O)NC(C(C)NC(=O)Cc2cc(O)nc(O)n2)C)cn2c(n1)CCCN2 C(=O)(C1=C(C#N)CCC1)NC(C1CCOC1)CNC(CCCc1c(C)ccs1)=O c1(OCCCC(=O)NCC=CCNC(C2CCCCS2)=O)ccc(F)cc1F CCC(CC)C(F)C(=O)N1CC=CCC1C(=O)NOCC(C)C CN1CCC(CC(=O)NCCOCCCN(C(=O)CO)C)C1=O C12(C(N3CC(OC)(CNC(=O)CCNC(C)=O)C3)=O)CCC(CF)(C1)OC2 c1(NCC2CCN(C(c3cc(OC)c(O)c(Cl)c3)=O)C2)ncnc2cnccc12 c1(CC)ncncc1C(=O)NCCCCCCN(C(=O)Cc1cc(C)on1)C CCCC(CNC(=O)C(C)=CC(C)(C)C)C(=O)N1CCC(CNC(N)=O)C1 c1(C(c2onc(C(C(CC)CC)C)n2)(C)C)cc(F)ccc1F CCCC(CC)CC(=O)NCCC(C)NC(c1nccc(OC)c1O)=O C1(C(N2CC3C(CNC(=O)CCN4C(=O)CCC4=O)C3C2)=O)CC2(CCC2)CO1 C1(C(=O)NC(c2cccc(C)n2)C)CC2(CC2)CN1C(c1csc(C)c1)=O C#CCC(O)C(=O)NCCn1cc(CNC(=O)C(C#N)CC)nn1 c1(C(N(CCCNC(C2CC(C)OCC2)=O)C)=O)cccc(Cl)c1[N+](=O)[O-] CC1CN(C(=O)CCn2ccnn2)CC(C)N1C(C1CC2(CCC2O)C1)=O CC1CN(C(=O)COc2cccnc2)CCC1N(C)C(c1coc2c1COC2)=O c1(C(N(CC)CC2CCCN2C(=O)Cc2cc[nH]n2)=O)csc2ccc(F)cc12 C1(NC(C=Cc2c(C)n[nH]c2)=O)CN(C(C2CC(=O)N(C)C2)=O)CC12CC2 c1(C(=O)NC2CC(N(C(COCCSC)=O)C)C2)ccc(C(C)(C)C)nc1 n1(CC)cnc2c(NC(c3cc(Br)no3)C)[nH]c(=NCCc3nncn3C)nc12 C(=O)(N=c1cc2n([nH]1)CCCC2)C1CCN(C(C2(CN(C)C)CC2)=O)CC1(C)C N1(C(C(=O)NC(c2cc(F)cc(F)c2)C)=O)CC2CCC1C(CO)C2 N1(CCN(CC(N)=O)C)CCCC(NC(=O)CCC2CC2)C1 c1(C(=O)NC(C(=O)NCCC(C(=O)OC)C)C2CCC2)nc(C)ccc1F N1(C(CCCCOC)=O)CCC2(CCC2)C(CNC(=O)C(O)CC2CCCC2)C1 C(C1=NOC2CN(C(c3cccc(N)c3F)=O)CC12)NC(c1ccc(SC)s1)=O C1(C(=O)NC(C)C(=O)NO)CC2(CCC2)CN1C(=O)CCCCC1CC1 c1(NC2(CNS(CC)(=O)=O)CCOC2)[nH]nc(OC(C2CC(C)(C)C2)=O)c1Cl c1(C(=O)NCCCCCN(C)C(C2CC(N(C)C)C2)=O)ccnc2c1nnn2C S(=O)(=O)(c1cccc(=NC(CO)C2CCOC2)[nH]1)NC(C)(C)CS(C)(=O)=O c1(OC)cnncc1C(N1CCCC(C(C)C(=O)NCCc2scnc2C)C1)=O C(=O)(CC(C)CC(F)(F)F)NC1CN(C(C2(CC(=O)OC)CC2)=O)CC1N=[N+]=[N-] CON=CC(=O)NC(C)(C)CN(C(=O)Cc1cncn1C)C CCC1=C(C(=O)N2CCC(C(=O)NCCN=[N+]=[N-])C2C(C)C)CCCO1 N1(CC(=O)NCC(CN(C(=O)CCN2CCC(F)C2)C)O)CCCCCCC1=O CC1=CCC(C)(C(N2CCCC(CO)(NC(C3CCCS3)=O)C2)=O)CC1 c1(C(=O)NCCC(=O)N(CCOCC=C)C)ncc(N)cc1C N1(C(C(C)c2ccsn2)=O)CCCN(C(=O)CCn2cccn2)CC1C C1(CC(N)=O)CCCN(C(=O)C(CCF)NC(=O)C2=NOCC2)C1 C(=O)(C(CC(C)C)ONC(c1cnncc1N(C)C)=O)NCc1c(C)nccn1 c1(C(=O)NCCN(C(CC(CC)C2CCC2)=O)C(C)C)coc2c1CCCC2 c1(C(N2CC(NC(c3c(CC)con3)=O)C3C(C2)C3)=O)cc2cccc(Cl)c2o1 c1(C(N(CCCNC(CCCOCCOCC)=O)C)=O)cc(CC)ccc1Cl C1(C(=O)NCCCCCN(C(CN(C(C)=O)C)=O)C)C2CCC1(c1ccco1)C2 C1(C(=O)NC(C#C)(CO)CO)CN(C(c2ccccc2O)=O)CC1C1CC1 n1(CCCSC)nnnc1C(C1CCCO1)(C)NCc1ccn(C2CC2)n1 C1(CCNC(c2cc(C(C)C)nn2C)=O)CC(F)(F)CN1C(C1CC1(Cl)Cl)=O N1(C(C2(SC)CC2)=O)C2CCC1CN(C(c1cc(C3CC3)nn1CC(F)F)=O)C2 CCCCCCCC(C(=O)NCCC#N)N(C(Cc1ccc(O)cc1)C(=O)OC)C C(=O)(C(F)CC(CC)CC)N(C1CCC(NC(CNC(CC)=O)=O)CC1)C c1(C(=O)NCCC2(NC(c3cnc(C)[nH]3)=O)CCC2)[nH]nc([N+](=O)[O-])c1Cl C12(NC(C(C)NC(=O)C(C)(C)C)=O)CCCC1N(C(=O)CC(O)C1CC1)CC2 C1(NC(=O)Cn2cccn2)Cc2ccccc2N(C(=O)C(F)C2=CCCCC2)C1 c1(CC(=O)NC2C(CC)CN(C(=O)CCC3CC3)CC2)cccc(S(C)(=O)=O)c1 CC1CN(C)CC1NC(=O)CNC(=O)C(c1ccccc1F)F C1(C(N(C2CCCCC2)CCNC(C=CC=CCC)=O)=O)CCn2nccc2C1 c1(C(N2CC(O)CC(NC(CCC#CC)=O)C2)=O)cc(C)c2nc(C)nn2c1 N1(C(C(CCC(C)C)NC(C2CCCC(=O)N2C)=O)=O)CCc2nc(O)[nH]c2C1 n1(CCN(CC(C)C)C(c2cn(CC(CC)O)nn2)=O)ncc2ccccc12 c1(CC)cc(C(N2CCCC2CN(C(C2CCCCS2)=O)CC)=O)c(C)nn1 c1(C(=O)NCC2CCC(NC(c3c(C)coc3)=O)C2)ncnc(O)c1F c1(C(=O)NCCCN(C(c2cc(C(C)C)no2)=O)CCO)ccn2c1CCCC2 c1(C(N2CC(OC)C(NC(=O)CN3CCC3C)C2)=O)cnn2c1CCC2 C(C(C)(C)COC)(c1n(C(C(=O)OC)C)nnn1)NC1CCS(=O)(=O)C1 NS(=O)(=O)c1cccc(S(=O)(=O)NCCCc2cnccn2)c1 C1(CNC(c2scc(OC)c2)=O)(CNC(c2cc(Cl)ns2)=O)CCOCC1 N1(C(C2(CCOC)CCC2)=O)CCC(C2CCN(C(=O)CC3CCCC3)CC2)C1 c1(C(=O)NC(CC(C)NC(C(CC#C)CC#C)=O)C)csc2ccc(OC)cc12 N1(C(c2c(C)nc(CC)o2)=O)CC2CC1CCN2C(=O)C(C)CC c1(C(=O)NCC(C(C)C)(C)NC(c2cnco2)=O)n[nH]c2c1CCC(C)(C)C2 c1(CNC2CC(C(=O)OC)C2)cccc2cccnc12 CN=c1[nH]c(=NCC(=O)Nc2cccc(F)c2)[nH]c(=NC(C)c2nncs2)[nH]1 C1(CN(C(c2ccn(CC(F)(F)F)n2)C(=O)NC(CC)C)C)CCCS(=O)(=O)C1 C(=O)(C(C)(C)C(F)(F)F)NC(CN1CCN(C(C=CC)=O)CC1)C C1(C)(C(N(CCNC(c2cn(C)[nH]c2=N)=O)C2CC2)=O)C2Cc3ccccc3C12 C1(CNC(c2nc(CC)sc2)=O)C(OC)C(OC)CN1C(=O)CCn1cccn1 C(CC(N)C(C)(C)C)N(C)Cc1c(N(C)C)ccnc1 Cc1cc(C(F)(F)F)n2ncc(C(=O)OCC(=O)N3CCC3)c2n1 n1(CCCOCC)c(N2CC(OCC)C(F)C2)nnc1-c1ccc(Cl)s1 C1(C(N2CCCC(NC(=O)C=Cc3cc[nH]n3)CC2)=O)CCc2cncn2C1 c1(C(N2CCCC(N(C(=O)C(O)Cc3ccccn3)C)C2)=O)nccc(N)c1Cl C(CN=C(NCCc1ccco1)NCCN1CCCC1)c1ccc(C)nc1 CC1CC(C(=O)NCC2(C)CCN(C(=O)C(F)(F)C3(O)CCC3)C2)=NO1 Cc1ccc2[nH]c(C(N3CC(CNC(=O)COCCF)C(F)(F)C3)=O)c(Cl)c2c1 Cc1cn2c(n1)CN(C(c1coc(CNC(c3n[nH]c(CO)c3C)=O)c1)=O)CC2 Cc1cc(C(N2CCCC(C(=O)N(C)Cc3nncn3C)CC2)=O)c[nH]c1=N C#CCCCCC(=O)N1C(C(=O)NCC2(C)CC3CC3C2)CC1C C1(CNC(CCCC=C)=O)CN(C(=O)Cc2ccc(Cl)cn2)CC1(F)CO Cc1ncc(C(N2CCCCC2C2CCCN(C(c3ccno3)=O)C2)=O)n1C C1(C(N(CC)Cc2cccnc2)=O)CC(C)CN(C(c2ccc(NCC)s2)=O)C1 C1(O)(C(C)NC(c2cn(C)nn2)=O)CCN(c2nnc(C#N)s2)CC1 Cc1ncc(C(=O)NC(c2cc(Cl)ccc2Cl)c2nn[nH]n2)cc1C#N c1(NC(c2n(CC)ncn2)C)nc(=NCC2C3COCC23)[nH]c2c(C)nn(C)c12 N1(C(c2c(C)n(C(C)C)nc2)=O)CCC(C2CC2)(CNC(=O)C(C)C2CCC2)C1 C1(NC(C2N=C(C)SC2)=O)CCN(C(c2cc(C)ccc2O)=O)C1(C)C N1(C(C2N(Cc3c(F)ccc(OC)c3)CC(O)C2)=O)Cc2cc(Br)cnc2C1 C=CC1(C(=O)NC2C=CCN(C(=O)Cc3cccc(NC(C)=O)c3)C2)CCCC1 C1(C(=O)NCCNC(=O)Cc2csc(C(F)(F)F)n2)CC2(CC2)CO1.c1cnco1 C(=O)(CC(C)(C)CC(F)(F)F)N1CCCC(C)(CNC(C(C)OCCC=C)=O)C1 n1(CC(=O)NCC2CCN(C(CCC(=C)C)=O)C(C)C2)ccc(=O)c([N+](=O)[O-])c1 c1(OC)ccc(NC(c2ccc(SC)cc2)c2nnnn2C(C)C(=O)OC)cn1 c1(CC(=O)NCC(CNC(C2CC2C(F)F)=O)F)cc(Cl)ccc1Cl C1(NC(c2ccc(COC)o2)=O)CC12CCN(C(=O)C(C)N(CC(F)(F)F)C)C2 C1(C(=O)NC2CN(C(COCCOC)=O)C2)CC(C(=O)O)C12CCC2 C12(NC(C3(NC(c4nccc(N)c4Cl)=O)CCCC3)=O)CC3CC(CC1C3)C2 CCC(C#N)C(=O)N(C(C(=O)N(C)CCOC(C)C)C1CC1)C C1(CNC(C2C(C)(C)NC(=O)C2)=O)N(c2ncc3c(n2)COC3)CCCC1(C)C C12(NC(c3coc(Br)c3)=O)CC3CCC(C1C2)N3C(c1cc(CF)on1)=O N1(C(CCC=CCC=C)=O)CC2CCC2(CCNC(c2cccn(C)c2=O)=O)C1 C1(C(=O)NCCCCCCC)CNC(=O)CN1C(=O)C(CO)NC(N)=O C1(CNC(c2n[nH]cc2[N+](=O)[O-])=O)CC2CCC1N(C(c1ccc(CO)o1)=O)C2 c1(NC(C2CN(C(c3cc[nH]c3)=O)CCS2)=O)c(F)cc([N+](=O)[O-])cc1Br C1(OC)CN(C(=O)CN(C)C2CC2)CC1C(=O)NOCC(F)F Cc1ccc2c(c1)SC(C(=O)NCC1CC1NC(=O)CS(=O)(=O)CC(C)C)C2 N1(C(C2CC(C)(CC)C2)=O)CCC(C)C(CNC(C2(OC)CC2)=O)C1 c1(N(C)Cc2ccc(OC)cc2)ncnc2c1ncn2CCc1nc(Br)sc1C c1(C(=O)OC)nnc2ccccc2c1N1CC(CNC(=O)CC(C)CC(C)C)C1 CC(C(=O)NCC1(C(C)NC(c2cccc[n+]2[O-])=O)CC1)C(F)F S(=O)(=O)(c1ccc(CCNC(N2CC3CCC(N(C)C)C3C2)=O)cc1)NC c1(OC)nc(C(N2CC3CC3C2)C(=O)NCC2CCCO2)sc1C C(=O)(CS(=O)CC)N(CCC(=O)NC(C#C)CCC)CCCO C(C(O)CCCCC)NC(c1c(CCNC(CC=CCCCCC)=O)n[nH]c1)=O C1(CNC(c2c(C)n(C)cn2)=O)CC2(CC2)CN1C(C1CN(C)CCO1)=O c1(CC)nscc1C(=O)NC1(C2CCCN2C(=O)Cc2cc(C(C)C)no2)CC1 C(=O)(C1CCCc2sccc21)N1C(CN(c2ccnc(C(F)(F)F)n2)C)CCC1 Cn1nc(C(=O)NCc2cc(C(=O)NOC3CC4CCC3C4)on2)cc1CO N1(C(C(C)OC)=O)CC2CCN(C(c3cc(I)ccc3C)=O)C2C1 CC(C)(C)CCC(=O)N1CC(CNC(=O)Cc2cncc(Br)c2)CC(O)C1 C1(CNC(C(N2CCC=C(C)C2)=O)=O)CCC(C)C(C)C1 C12(C(=O)NC(CC(CC)C)C)CC(CN(C(c3nccnc3N)=O)C1)C2 C(CCC1CCC1)(C(=O)N(c1ccncc1)CC)NC(CCC)=O c1(C(=O)NCC2OCC(CNC(=O)Cn3nnc(=O)[nH]3)C2)cc(F)cc(Cl)c1 S(=O)(=O)(CCCS(=O)(=O)C(F)(F)F)NC(c1cccc(CCC)c1)=O N1(C(C(C=C)C)=O)CCCC(C(=O)OC)C1CC.C1C(F)C(=O)N2CC1C2 c1(C(N2C(CNC(=O)C=Cc3cc[nH]n3)COCC2)=O)ccc(F)c2occc12 Cc1cc(C)n2ncc(C(N3CCC(CF)(NC(C4CCC4)=O)C3)=O)c2n1 CS(=O)(=O)CC(C(=O)NNC(=O)C(F)(F)c1ccccc1)C1CCC1 Cc1scnc1C(=O)NCC(C)(C)CN(C(=O)C(C)OCCC(C)C)C N12CCCC(C1)OCC1CC1C2=O.c1(-c2cn(C3CC(OC)C3)nn2)ccc(Cl)cc1 c1(C(N2CCC(NC(c3cc(C)c(Cl)s3)=O)C2C(C)C)=O)cc2c(ccn2C)[nH]1 N1(C(CCC(C)C)=O)CC23CCCC2(C1)CN(C(c1ccc(Cl)c(O)c1N)=O)C3 C(=O)(C(O)C(F)(F)F)NC(c1ccnn1C)C(=O)N(CC(=O)NCC)C C1(C(=O)OC)CCOC12CCN(C(c1cc(Cl)cc([N+](=O)[O-])c1N)=O)CC2 C(CCC)(C(=O)N1CCCC1CN(C(=O)CC1CCCO1)C)=CCC C(C(O)C(=O)NC(C)CNC(c1ncoc1C1CCCO1)=O)=CCCC C(C(O)C(=O)NCC(O)CCNC(=O)C=C1CCC1)=CC(C)C c1(CNCc2c(C)nn(C)c2N2CCOCC2)cn2cccc(C)c2n1 S(=O)(=O)(c1ccsc1C(N1CCC(NC(C2(O)CC(F)(F)C2)=O)C1)=O)NC C#CCCCCCC(=O)N(CCC(=O)NC(CC)C(C)(C)C)C C1(C(=O)NC(C#C)C(C)C)(CNC(=O)CC=C(Cl)Cl)CC2(CC2)C1 C1(N(C)C(c2csc(CC(F)(F)F)n2)=O)CCN(C(c2cncnc2)=O)CC1 c1(C(N2CCN(C(C3CN(C(C)=O)C3)=O)C3C2C3)=O)ccc2cn(C)nc2c1 c1(-n2ccc(C(=O)NCCC(=O)NCc3ccc(F)cn3)n2)ccccc1F N1(C(C(C)=C2CCCC2)=O)CCC(NC(=O)CCc2cn[nH]c2)C(CO)C1 N1(CC(=O)NC(c2cccs2)C)CC(NC(=O)CC(C)C(F)F)C(C)(C)C1 C1(C(N(CCC(=O)NC2CN(C(=O)OC)C2)C)=O)CCCC1C C1(NC(C2(C)C=CCC2)=O)CC=C(C(=O)NCCc2nnc(O)o2)C1 c1(C(N(CCN(C(C(CCSC)NC=O)=O)C)C)=O)n[nH]c2c1CN(C)CC2 CC(CCC(=O)NCC=CC1CC1)NC(C1CC2(CCC2)C1)=O Cc1ccc(CNC(C2CC2C(C)NC(=O)C2=CCCC2C)=O)cc1O c1(OCC)ccc(-c2noc(CS(C)(=N)=O)n2)cc1 CC1(C(=O)NCC(O)CNC(C2(CF)CC2(F)F)=O)CCCO1 N#Cc1cc(F)c(C(=O)NC2COCC2NC(=O)CC2CC2(Cl)Cl)c(F)c1 c1(C(=O)NCCC2CN(C(C=CC(=O)OCC)=O)C2)cc(C2CCC2)no1 Cc1cccc(C)c1C(=O)NCC1CC(CNC(=O)Cc2cnsc2)CO1 N1(C(=O)Nc2n(C)nc(-c3ccncc3)n2)CCC(O)(C2CCC2)CC1 c1(NC(=O)COC(c2cccc([N+](=O)[O-])c2)=O)c(O)c(Cl)cc(Cl)c1Cl N1(C(C(C)(C)SC)=O)CCC(CN(C)C(c2snnc2C)=O)CC1 C(=O)(CC(C)(C)C#N)N1C(C)CC(NC(COCCCC(C)C)=O)C1 c1(C(=O)NC2CCN(C(c3c(Cl)cc(C)c(C)c3)=O)C2)ccc2c(c1O)CCC2 N1(C(C2(SC)CC2)=O)CC(O)(CN(C)C(C2CCN2S(C)(=O)=O)=O)C1 C(=O)(CCCCN(C)C)NCC(COC)NC(=O)C(COC)OC C(=O)(N=c1[nH]nc(C(=O)OC)s1)Oc1ccccc1CN(C)CC N1(C(c2c(O)ccc(N)c2)=O)CC(NC(=O)C(F)n2cccn2)C2CCCCC12 c1(C(=O)NC(CN(C(C=CC=CCC)=O)CC)C)cnc(O)c2cccnc12 c1(C(=O)NCC2C3CN(C(CN(c4ccncc4)C)=O)CC32)cc2n(n1)CCCO2 N(C1CCc2ccccc21)C(C12CN(C(C3(C#C)CC(=O)C3)=O)C(C1)CO2)=O C12(CNC(CN(C(C)=O)C)=O)CC1CN(C(=O)C(C(C)C)n1ccnc1)C2 CC1CCCCC1(C)NC(=O)C=CC1CCN(C(=O)CC2(C)OCCO2)CC1 S(=O)(=O)(c1cc(Br)c(Br)c(Br)c1)Nc1ccc(C(=O)NCC)cn1 n1(CCOC)cc(C(=O)NC2(CNC(C3CCCS3(=O)=O)=O)CCC2)ccc1=O C=CC(C)(C)CC(=O)N1CCC(C)(NC(c2cnc(SC)s2)=O)C1 N1(C(c2nnn(C)n2)=O)CCN(C(c2sccc2F)=O)CC1CS(C)(=O)=O C(=O)(CCCCC#N)NC(CC)(C)CNC(=O)CNc1ccc(C(N)=O)cc1 c12cnc(cn1)C(=O)OCC(O)CO2.Cc1nocc1C(=O)OC(C)(C)C C(C)(C(=O)NC1CCCC1C(=O)N(C)Cc1ccoc1)(C(C)C)OC C(=O)(C1CC(=O)c2ccccc21)NCC1(NC(C(C)C(F)F)=O)CCC1 CS(=O)(=O)C1CCCN(C(C23CC(C(=O)NCc4cncnc4)(C2)C3)=O)C1 n1(CC#C)cccc1C(=O)N(CCC(=O)NCC1CCC(=O)O1)CC1CC1 c1(C(=O)NCC(C)N(C(CCC(C)O)=O)C)ccc(O)c(Cl)n1 c1(C(=O)NCC(C)N(C(=O)Cn2cccc2)C)cnc2ccsc2c1 C1(CC(=O)NCCSCC(=O)Nc2cc(F)ccc2O)CCCCC12CC2 c1(C(=O)NC(C2CCN(C(C3CCC(F)C3)=O)C2)C)cc(C(F)F)[nH]n1 C1(O)(CNC(C(COC)(C)C)=O)CCCN(C(=O)Cc2csc(C)n2)CC1 C1(CCCC)CN(C(=O)C(F)(F)C(C)O)CCN1C(c1cocn1)=O c1(C(=O)NC(c2ccc(C)cc2)CNC(=O)C2=CCC2)c(N)ccc(F)c1F C(N=c1[nH]c2c(c(=NCCCN3CCOCC3)[nH]1)SCC2)c1nc(C)cc(C)n1 C1(C)(C(=O)NCC2(OC)CCN(C(=O)C=CC3CCOC3)C2)CC2(CCC2)C1 c1(C(=O)OC)cc(Br)sc1NC(C1CSCN1C(=O)CC1CN(C(C)=O)C1)=O N1(C(c2cc(OC)cc(Cl)c2)=O)CCN(C(C2CCCN2N=O)=O)CC(CO)C1 C1(SCc2nnc(-c3c(C)oc(Cc4ccccc4)c3)o2)CCS(=O)(=O)C(C)C1 Cc1cc(CC(=O)NCCC2COCCN2C(=O)CCN(C)C)n(C)n1 c1(C(N2CC(OCCNC(c3ccncn3)=O)C2)=O)cc2cccnc2s1 c1(C(N2C(C(C(=O)NCCCN(OC)C)(C)C)CCC2)=O)cnc(C)nc1C CC1(C)CC(C(=O)N2CCCC2CNC(=O)CCOc2cccc(Cl)c2Cl)=NO1 C1(C(C)(C)NC(C(CC)OCC)=O)CCCCN1C(c1csc(CC)n1)=O C1(C(=O)Nc2cccc(Cl)c2)(CC)CCCN(C(c2ccnnc2)=O)C1 C1(C(=O)NC(CC2CN(C(C3(OC)CCCCC3)=O)C2)C)CCCC(F)(F)C1 c1(C(=O)NC(CCCC)CNC(c2cscc2OC)=O)ccc2oc(O)nc2c1 c1(C(=O)NC2C(NC(CC(C)SC)=O)CCC2)coc2c1COC2 c1(C(=O)NCC2(NC(C34CCN(CC3)C4)=O)CCOCC2)ccc2n[nH]cc2c1 N1(C(CC(C)c2cnn(C)c2)=O)CCC(CNC(C2(CCO)CC2)=O)C12CCC2 C(=O)(C#CC1(C)COC1)N(CCCNC(c1c(C2CC2)ccc(C)c1)=O)C(C)C C1(NC(C2C(C=C)OCC2)=O)CCN(C(c2oncc2C)=O)C12CCC2 c1(C2C(C(=O)NCCCCNC(c3ccnnc3O)=O)CC2)ccc(F)cc1F c1(OC2CCN(C(C(C)(C)Nc3ccccc3Cl)=O)C2)ccc(S(C)(=O)=O)cc1 N1(C(CP(C)(C)=O)=O)CC(CNC(C2CCC3(CCC3)C2)=O)CC1(C)C C1(CNC(C(CSC)O)=O)CC2(CCN(C(c3cc(C)cc(Cl)c3N)=O)CC2)C1 C12(C(N3CC4CC(NC(C(C)(C)CF)=O)C4C3)=O)C3C(=O)C4C5CC(C14)C2C35 c1(OCCSCc2nnc(C(C)C)s2)cc(Br)cc(F)c1F Cc1nscc1CC(=O)NCCNC(=O)CCc1cncs1 CCCCCCCC(=O)N1CCN(Cc2ccc(Br)s2)CC1CC#N C1(C)(C(=O)NCCN(C(C)C)C(c2cncc(F)c2)=O)CC2CCC(C1)S2(=O)=O C(=O)(C(C)(C)Cc1ccccc1)NCC1N(C(C2C(=C)CC2)=O)CC1 c1(SC)cc(C)ccc1C(=O)NC1(CF)CN(C(C2C3CCC(F)(F)C23)=O)C1 c1(C(N2CCC(C#N)(NC(C3CC=CCC3)=O)C2)=O)cc(F)c(Cl)cc1Cl Cc1cncnc1C(N1CCCC(CCNC(=O)CCc2csc(=N)[nH]2)C1)=O N1(C(C2C(C)(C)CCCC2)=O)CCN(C(c2ccc3cnsc3c2)=O)CC(O)C1 c1(C(C)(C)C)ccc(C(=O)NCC2CN(C(=O)Cc3csnn3)C2)cc1Cl c1(OCC)ccc(C(=O)NCCN(C(=O)CC2CCSCC2)CC)nc1 C1(OC)CCn2cc(C(=O)NCC3CC3NC(=O)C(F)=CCCF)nc2C1 N12CCC(CC1)C2.N1(C2CN(C(=O)NCCOCCCC)C2)CCCCC1=O C1(NC(c2cn(CC)nc2C2CC2)=O)CC2CN(C(c3ccsc3C)=O)CC12 c1(CC(N2CCOCC(C)(CO)C2)=O)noc2ccc(Br)cc12 C(=O)(C1=C(C)OCC1)NC(CN(C(C1COCC(=O)N1C(C)C)=O)CC)C N1(C(c2c(C)cncc2)=O)CCCN(C(c2ccccc2S(C)=O)=O)CC1C N1(CC(C)C)CCC(C(=O)NC2(CNC(C3CCN(CC(C)C)C3)=O)CC2)C1 C1(CC(=O)NC2(C)CC(NC(=O)CNC(C3CCCC3)=O)C2)CCS(=O)(=O)C1 N1(C(c2c(CC)cno2)=O)CC2CC(C1)N2C(=O)C(=Cc1cccnc1)F Cc1ncnc(C(=O)NC(C)(CNC(=O)C(C)(C)C2CCCO2)C(C)C)c1C c1(C(=O)NCC(=C)CCNC(C2(COC)C=CCC2)=O)c(F)ccc2ccoc12 c1(C(=O)NCCCC(C)NC(CCC=C(C)C)=O)cc(C)c(C)cc1N N1(C(Cc2cnc(C)[nH]2)=O)CC2CCN(C(c3c(C)cccc3F)=O)CC(C2)C1 C1(C#N)(C(=O)NC(C)CN(C(=O)Cc2cnccn2)C)CC1(C)C C1(CN(C(C=C(CC)CC)=O)C)CN(C(c2oc(C(C)C)nc2C)=O)CC12CC2 c1(-c2ccc(C)o2)cnc[nH]c1=NCCCCCCNC(=O)C1=C(Cl)CC1 N1(C(CCOCC)=O)CC2CCC1C(CNC(c1cccc(CN(C)C)c1)=O)C2 c1(C(N2CCC(NC(CCOCC(C)C)=O)C(F)C2)=O)cn(C)c(=O)n(C)c1=O c1(NC(C2C(NC(c3cc(OC)cc(Br)c3)=O)C2)=O)cc(Cl)c(Br)cc1[N+](=O)[O-] c1(CC(=O)NCC2(CCNC(CC(C)F)=O)CC2)cc(Br)ccc1Br C(C(=O)NCC1CCC(C(=O)N(CC(C)O)CCN(C)C)O1)(C(C)C)SC Cc1ccc2c(c1)ncn2CC(=O)NCCC(C)NC(c1cc(O)ccc1F)=O c1(NC(C(C)=C2CCC2)=O)cccc(NC(c2sc(C)nc2CC(C)C)=O)c1 Cc1cccc(C)c1OCC(=O)NC1CCOCC1NC(C1(C)CCOCC1)=O c1(C(=O)NCC(CO)NC(CC(C=C)CC)=O)cc2cccnc2nc1C1CC1 N1(C(c2n(CC)cnn2)C(=O)NCCCC2CC2)CCC(O)(C#CBr)CC1 Clc1ccc(C2(CNC(C3CCCOCC3)c3nnnn3C3COC3)CC2)cc1 C(CCCCC(=O)NC1CC2CCC1(NC(c1cc(CCCO)on1)=O)C2)SC c1(C(=O)NC(CC)CN(C)C(C2CC=CCC2)=O)nccc(OC)c1F N1(C(c2nc(C)oc2)=O)CC(NC(c2cc(Cl)c(Cl)s2)=O)C(O)C1 O=C1CN(c2cccc(OC(F)(F)C(F)(F)F)c2)C(=O)C2CCCN12 N1(C(c2cc(NC(C)=O)ncc2)=O)CC2CCCC2(NC(c2cnsc2)=O)C1 N1(C(=O)CC(C(F)F)c2ccc(F)cc2)CCOc2c(Br)cc(Cl)cc21 CCCCC(CNC(=O)C(C)C1CCCO1)NC(=O)CCOc1cccc(Cl)c1 c1(CCC(=O)NCC(N2CCC(C)CC2)C(C)C)c[nH]c2ncccc12 c1(-n2ccc(C)n2)ccc(NC(C2CCC(Cn3ccnc3)O2)=O)cc1 N12CCOC(C1)C1(CC1)N(C(CC(C)C)=O)CC2=O.c1(CO)ccnn1C C(=O)(N1CC=CCO1)NC(C)CCOc1ccccc1 c1(C(N(CCNC(C2NC(=O)CC2C)=O)CC)=O)ccc(C#CC2CC2)cc1 c1(C(N(CCCNC(C2CC(=C)C2)=O)C2CC2)=O)ccc(SC)c([N+](=O)[O-])c1 N1(C(c2c(C(C)C)n[nH]c2)=O)CC(NC(=O)C(O)C2CCC2)CC2(CCC2)C1 C(=O)(CCCC(F)(F)F)N1C(CN(C(C(CC=CCC)C)=O)C)CCC1 Cc1cc(CNC(C2(CF)CCN(C(=O)CNC(=O)CN(C)C)C2)=O)ccc1F c1(OC)cccc(CCNC(C2CCN2C(c2ccnc(Cl)c2)=O)=O)c1Cl c1(C(N2CCC(NC(c3c(NC)cnnc3)=O)C(C)C2)=O)cc(F)c(C)cc1F CCC(CC)CC(=O)NC(C)CN1CCN(C(=O)CCc2cnccn2)CC1 C1(CNC(C(C)NC=O)=O)CCC(C(=O)NCc2noc(N(C)C)n2)O1 N=c1nc(N2CCSC3(CCCCC3)C2)[nH]c(=NC2CN(c3cnccn3)C2)[nH]1 c1(C(=O)NC(CC)CNC(=O)C(C)N2CCC2)cc2ccccc2nc1O NC(=O)C1=NOC(CNC(C2CCN(C(=O)C=Cc3ccsc3)CC2)=O)C1 c1(C(=O)NC(CC)CN(C)C(C2(OC)CCOC2)=O)c(C)cnn1C c1(C(=O)NCCN(C(=O)C(F)(F)c2cccnc2)C)ccnc2ncccc12 CC1(C(=O)NC(c2ccc(Cl)cc2O)=O)CCN(Cc2c[nH]cc2Br)CC1 Cc1nn2cc(C(=O)NC(CNC(=O)Cn3cnc(C#N)n3)C(C)(C)C)nc2s1 C1(CNC(c2ncc(OC)nc2)=O)CN(C(=O)COCCN(C)C)CC1(C)C CC1CN(C(=O)C2CC2)CC(C)N(C(=O)C=CSc2nc[nH]n2)C1 N1(C(CC(C(=O)OC)C)=O)CCC(C)(C)C(NC(c2cccnc2O)=O)C1 c1(C(N2CC(NC(c3ccc(C)c(C)c3)=O)C(O)C2)=O)cc([N+](=O)[O-])ccc1C c1(C(N2CCCCC(CO)C2)C(=O)NCCCOC)cc(Cl)c(C)cc1Br C(=O)(C1CSc2ccccc21)NCCC1(CNC(C2(C)CCCNC2=O)=O)CC1 Cc1noc(COCC(=O)N(CCN(C)C(c2ncsc2C(C)C)=O)C(C)C)n1 C(=O)(C(C)C(F)(F)F)N(CCOCCC(=O)NCCN(CCC)CC)C C(c1ccc(F)cc1)=CC(=O)N(CC(C)CNC(c1coc(C2CC2)n1)=O)C C1(CC(=O)NCC2(CCNC(CN(CC(C)(C)C)C)=O)CC2)CCCO1 c1(OC)ncccc1C(=O)NC(C1(O)CCN(C(=O)C(C)OCCN(C)C)C1)C C1(C(CNC(=O)Cc2cnoc2)NC(CSCCOC)=O)CCCCC1 c1(C(=O)NC(C)(CNC(c2cc(C3CC3)no2)=O)CO)c[nH]c2cccc(F)c12 c1(C(c2n(CCOCC)nnn2)NC(C)Cc2ccsc2)ncc(Cl)cc1Cl CCC(COC)N=c1cc(C)[nH]c(=NCc2ccc(Cl)c(C)c2)[nH]1 C=CCC(C)(C)CC(=O)NC12CC(NC(=O)CCn3ccc4cccnc34)(C1)C2 c1(C(=O)NC2CC3(CC(NC(=O)CCCC4CC4)C3)C2)ccn2ncccc12 N1(C(C2(CC#C)CCC2)=O)CCC(CCCCNC(C2CCC(=O)N2)=O)CC1 C1(N(CC(C)C)C(c2cnco2)=O)CCN(C(C2CCC(O)CC2)=O)CC1 C(=O)(C(CC(C)C)CC(C)C)NC1C(OC)CN(C(=O)C(CCF)NC(C)=O)C1 c1(OCOC)ccc(CN2CCC2C(=O)Nc2cccc(OC)c2O)c(OC)c1 C1(N(C(c2c(C)onc2)=O)CCC2CCCCC2)C2CCC1CNC2 N1(C(c2onc(C)n2)=O)CCC2(CCCN(C(=O)CCC(C)N(C)C)C2)C1 c1(CN(c2n(CC(=C)C)c(C3CCCC3C3CC3)nn2)CC)nc(C)ccc1C C1(CNC(=O)Cn2cnc(Br)c2)CC(F)CN1C(c1cccc(F)c1)=O C1(NC(C2(NC(c3c(CC)c[nH]n3)=O)CC2(C)C)=O)CCCC(C(N)=O)C1 C(=O)(CCC1=CCCCC1)N1CCC(NC(c2c(=O)ccn(C)c2)=O)C12CC2 C1(CCNC(c2ccoc2)=O)COCCN1C(=O)C1=CCSC1 N1(C(CNC(CCC)=O)=O)CCC(C2(NC(C3(N4CCOCC4)CC3)=O)CC2)C1 c1(C(=O)NC(CC)CN(C)C(C2CC23CCC3)=O)cc(C)n(C(C)(C)C)n1 N1(CC=C)CCCN(C(C(=O)NCC2CCCO2)C(C2CCC2)SC)CC1 C12(NC(C=CCOC)=O)CC(C)(C1)OC21CN(C(c2nn(C)cc2SC)=O)C1 C1(C(N2C(C)(CNC(c3cn(C)nc3C(F)F)=O)CCC2)=O)Cc2nccn2C1 c1(CN(C)CC2(c3cnn(C)c3)CCCO2)cccc(C(N)=O)c1 C(=O)(C(=O)CCCC)N1C(CCNC(C(C=C)C)=O)COCC1 N1(CCn2cc(CCNC(C)=O)nn2)CCCN(C(=O)C(C)c2ccsc2)CC1 C(C(C)(O)C(=O)N1CC2CC2(NC(C2CC(N(C)C)C2)=O)C1)OC Cc1ccc(-c2nc(CCC3CCCCO3)n(CC3CC3)n2)cc1Br C1(NC(C=C(C)C)=O)CCC(C)N(C(c2cn(-c3ncccn3)cn2)=O)C1 Cc1sc(C(=O)NCCCCC(C)NC(=O)C=CBr)cc1Br Nc1cc(C(=O)NCC2CN(C(c3cnn(C4CC4(F)F)c3)=O)C2)ccc1Br c1(CNC(=O)Nc2c(OCC)nccc2)cccc(C)c1F Cc1nccn1C(C)C(=O)NC1CCC1C(N1CCCC1CCCn1ccnc1)=O C1(COC)(NC(=O)C(F)(F)C2CCOCC2)CCN(C(=O)CC(C)O)C1 CC1CC(NC(c2nc(Cl)c(Cl)s2)=O)CN1C(=O)Cc1cccnc1 CC(C)CC(O)C(=O)NCC(F)CNC(C1(O)CN(C(=O)OC(C)(C)C)C1)=O CC1(C)C(C(=O)NCC2(CN(C(=O)CCc3csnn3)C3CC3)CC2)C1C(F)F Cc1ccc(NC(c2sccc2NCc2ccc(O)c(Cl)c2)=O)c(C#N)c1 CC1(C)COCCC1CNCC1CCCN(C2CCCCC2)C1 C(=O)(C(C)(C)C(=O)NS(=O)(=O)CC(C1CCCCC1)OC)OCC CC(C)CC(C)(CNC(C1(C)C(C)(C)C1(C)C)=O)NC(C1CCCOCC1)=O C1(C(=O)NC2CC3(CN(C(c4c(SC)nn(C)c4)=O)C3)C2)CC(=O)N(C)C(=O)N1 N1(C(C2(C)C=CCCC2)=O)CCCC(CCNC(=O)Cc2cnoc2)CC1 CP(C)(=O)CN1CC(C(=O)NC2CCCC2CNC(c2cncc(O)c2)=O)C1 CP(C)(=O)C(O)C(=O)NCC1(O)CCN(C(=O)CCOc2ccc(Cl)cc2)CC1 C(=O)(CC1OCc2ccccc21)N(C(C)CNC(c1ncn2ccccc12)=O)C Cc1cccc(C(=O)N(C)CCN(C(c2ncc[nH]2)=O)C(C)C)c1[N+](=O)[O-] C=CCCC(CC(C)C)C(=O)NC1CC2CC(C1)N(C(C1CC(F)(F)C1)=O)C2 N1(CC(=O)N(CCO)CC2CC2)CCCC1Cc1ccccc1 CCCC(CC)CCC(=O)N1CC(CC(N(C)CP(C)(C)=O)=O)CC1C CN1CC(F)CC1C(=O)NCCNC(=O)C(=O)Nc1ncc[nH]1 CC#CCCCC(=O)N1CCC(NC(=O)C2CC2)C1C N1(C(CSCCC)=O)CCC(CN(C(=O)CCCc2nncn2C)CC)CC1 C1(NC(C2CC(=C)C2)=O)CC(CNC(=O)Cc2sccc2C)C1(C)C C(=O)(CC(C)(O)C(F)(F)F)NCC(C)NC(c1cccc2nc(C(F)F)[nH]c12)=O c1(C(=O)NCC2CCCC(NC(c3ccccn3)=O)C2)cc(O)ccc1Cl n1(CC)nncc1C(C(=O)NCCCSC)N(C)Cc1scnc1C Cc1cncc(C(=O)NC(C2CC(NC(c3cnn(C)c3)=O)C2)C)n1 N1(C(c2cnc(C)[nH]2)=O)CCN(CC(C)(C)NC(=O)C2=CCCC2)CC1 N1(C(c2c(CC)ncs2)=O)CCC(O)C(NC(C2CN(C(C)C)CCO2)=O)C1 c1(C(N2C(CC)C(C(=O)N(CC(F)(F)CO)C)CC2)=O)cccc2[nH]ncc12 C(c1cc2ccccc2o1)=CC(N1CC(OC)C(NC(=O)CCN2CCCC2)C1)=O C(CCC)(C(O)C(=O)N1CCC(CO)C(C)(C)C1)NC(C(C)OCCCC)=O N1(COCC)N=C(C(=O)N2CC3CC3(CO)C2)CCC1=O.c1(C(=O)N)nnccc1C N1(C(c2cc(C)[nH]c2)=O)CCCC(C2CC2NC(c2cc3ncccc3s2)=O)C1 C(CCCC(=O)NCCCCCCNC(C1CC1(C)C(C)C)=O)NC(C)=O C1(C(N(CCCNC(=O)CNc2nccs2)C)=O)CCNC1=O.c12nnnn1C2 N1(C(c2[nH]cc(CC)c2)=O)CCCC12CCN(C(C1CC3CC(O)C(C1)C3)=O)C2 C1(CCC)CN(C(=O)C=C2CCC2)CCN1C(c1sc(Br)c(C)c1C)=O c1(C(N2C(CC)C(C(=O)NC(c3c[nH]ccc3=O)C)CC2)=O)cc(O)ccc1F c1(C(=O)NCC2CCC(C3CC3)O2)cnc2c(Cl)cccn12 C1(C(=O)NC2CN(C(C(C)CCc3cccc(F)c3)=O)C2)CCc2c[nH]nc2C1 c12cc(c(Cl)cn1)N2C(n1cc(C(O)CC(C)C)nn1)=O.C1(Cc2cnn[nH]2)CCCO1 C1(C(C)(C)NC(C(C)=CC2CC2)=O)CCN(C(C23CCCC2CC3)=O)CC1 c1(NC(=O)NC(CSC)CO)cnc2ccnn2c1 C(=O)(C(O)C(C(C)C)OC)N(CC)CC1CCCN(C(=O)C(F)C(F)(F)F)C1 C1(CCC)CN(C(=O)C(O)C2CCCC2)CCN1C(C1CCC2(CC1)CC2)=O C1(C(N(CC(C)NC(=O)Cc2ccccc2F)C)=O)CCn2cncc2C1 N1(C(CCc2nnc(-c3cccc(C)c3)o2)=O)CCc2c(cnn2C)C1 c1(C(=O)NC(C(C)C)C(C)NC(c2coc(Cl)c2)=O)cccc(C(F)(F)F)c1F C(C(C)(CC)C(N)=O)NC(C(CC#C)NC(=O)CSCCC)=O CC(O)C(F)(F)C(=O)NC1CCC(CNC(=O)CSc2ccc(F)c(F)c2)C1 C(=O)(C(C(C)(C)C)OC)NCCN(C(C1CN(CC(F)(F)F)C1)=O)CC C1(CCNC(C(C)OCC(C)C)=O)CCCN(C(=O)CC2CC(F)(F)C2)C1 c1(C(N2CC(CN(C(C(CCC)(C)C)=O)C)C2)=O)ccc2nnc(O)n2c1 C#CCC(O)C(=O)NCCC1CCCCN1C(c1c(Cl)n[nH]c1C)=O C1(OC)CCCCCC1NC(c1nnnn1C1CC1)(C)CNC(C)=O N1(C(CC(C)c2ccco2)=O)C(CNC(=O)CC2CCCC2)CC2COCC12 c1(C(=O)NC2(CC=C)CCCN(C(=O)CSc3nncs3)C2)ccc(C#N)cn1 C1(C(=O)NCC(C)N(C(CCc2c(C)n(C)nc2)=O)C)CCC2CCC1O2 C(=O)(C1=CCN(Cc2ccccc2)C1)NC(CN(C(c1c(CC)nco1)=O)C)C C1(NC(C=NOC)=O)(CO)CCCN(Cc2ccc(C3CCCC3)cc2)C1 c1(C(=O)NC2CC2C(=O)Nc2ccon2)ccc(Oc2cccnc2)cc1 C1(COC)CN(C(=O)CSc2nncn2C)CCN1C(c1ccn(CC#N)n1)=O c1(C(N(C)CC2(O)CCN(C(CC=C)=O)C2)=O)cc(Cl)ccc1OC C1(C(N2CCC(C)(N(C)CC)C2)=O)CN(C(c2ccccn2)=O)CCC1(C)C c1(NC(CC)C(=O)N(C(C2CCC2)C)CCN(C)C)cccnc1Cl c1(N(C2CCC(C)(C)CC2)C)nc2ccccc2nc1NC1CCN(C)CC1 Cc1c(F)ccc(NC(=O)C=Cc2ccc(F)c(F)c2)c1F Cc1cc(CNC(=O)CCCC2(NC(=O)C(F)OC(F)(F)F)CCC2)cnc1Cl N1(CC(=O)NCC23CCCCC2C3)CCN(C(=O)Cc2ccc(O)nc2)CC1 C1(C)(CNC(CC2CCN(C(C(c3cncnc3)C)=O)C2)=O)CCN(C)C1 C1(NC(c2c[nH]nc2-c2cccs2)=O)CCSC12CN(C(=O)C=CC1CC1)C2 C1(F)(CNC(C(C)Cc2cnco2)=O)CCN(C(c2ccc(CO)o2)=O)C1 N1(C(c2ccc(CC)s2)=O)CCC(C(=O)NCC(C)Cc2cn[nH]c2)C1(C)C c1(C(=O)NCC2C(CNC(=O)COCC(c3ccccc3)=O)C2)ccncc1Cl c1(C(=O)NCC2(C)CCN(C(c3cnn(C)c3N)=O)C2)cccc([N+](=O)[O-])c1 C1(C(=O)NCc2cn(CC(=O)N(CC(=O)N(CC)CC)C)nn2)CC(=O)N(C)C1 N1(C(c2c(C)sc(O)n2)=O)CC2CC1CN2C(=O)CC1CCCNC(=O)C1 c1(C(=O)NC2C3CN(C(=O)CCC4CC4(F)F)CC23)ccc([N+](=O)[O-])o1 c1(C(=O)NC2(CC)CCN(C(=O)CCOC)CC2)ccn2ncccc12 Cc1cccc(CC(N2CC(OCCNC(=O)Cc3ccccc3O)C2)=O)c1Cl C12(NC(C=CC)=O)CC(C(N3CCC(CN(C4CC4)CC)C3)=O)(C1)C2 C1(NC(=O)C2CC2)CN(C(c2cc(Cl)n[nH]2)=O)CC1C1CC1 CS(=O)(=O)C1(C(=O)NCC=CCNC(c2cnn(C3CCCC3)c2)=O)CCCC1 c1(C(=O)NC2CCCCN(C(C(C)=C3CCC3)=O)C2)c(C)nc(C2CC2)nc1O C(CN=c1[nH]c(NC2CC2c2cncs2)nc2ccccc12)c1cc(O)nc(=O)o1 C(CO)(CO)(C(=O)O)NC(C1CCN(Cc2ccccc2)C1=O)=O C1(NC(=O)CC(O)C2CCCC2)CCOCC1NC(c1nccnc1C(N)=O)=O C#CC1(C(=O)NCc2ccccc2CN(C(=O)C(CSC)OC)C)CCCC1 c1(N2C(C3CCN(C(C(c4n(C)ncc4)(F)F)=O)C3)CCC2)ccn2ccnc2n1 Cc1ccc(C(=O)NCC(O)C(N2CCCCC2C)=O)cn1 CC(O)C(F)(F)C(=O)NC1COCC1CNC(=O)Cn1cnc(=N)[nH]1 c1(C(N2CCC(C)(CCNC(C3CC3C3CC3)=O)C2)=O)ncc(N)cc1Cl n1(CC(=O)N(C2CN(C(CCc3cnc(C)o3)=O)CC2O)C)ccc([N+](=O)[O-])n1 c1(COC(COC2(C)CCC2)=O)ccccc1SCC1CCCC(=O)O1 N1(C(c2n[nH]c(C)c2Cl)=O)CC(CNC(C2CC2F)=O)OC2CCCC12 CCC(CC)C(C(=O)N1CC(C23C(CO)(CCN(C(C)=O)C2)C3)CCC1(C)C)OC C(=O)(C1=CCC(NC(C2(c3ccccc3)CC2)=O)C1)NC(C)(C)CCF C(C(C)(C)C#CC(=O)NC(CO)CCO)NC(CCCCN(C)C)=O C1(c2ccccc2)(CC(=O)N(C2CN(C(=O)C(C)c3ccco3)C2)C)CCCO1 Cc1ccc(SC(C)C(=O)N(C)CC2CN(C(=O)C(C)(C)C#N)CCO2)cc1 c1(COC)n[nH]c(=NC2CC(CCNC(=O)C(C)(O)C3CC3)C2)s1 N1(C(C(CN=[N+]=[N-])NC(C2C(C)(C)C2)=O)=O)CCOCC2(CCC2)C1 CCCC(CCC)C(=O)NC1CCCCC1NC(=O)CC1CCOC1=O C1(NC(C(CNC(CCc2cc(C)[nH]n2)=O)O)=O)CN(C)C(C)(C)C1 c1(OC)c([N+](=O)[O-])cnc2c(C3COc4ccccc4O3)ccc(C)c12 Cc1cc(C)n(CC(C)C)n1.C12(c3nnnn3C3CC3)COC(C1)CN2 c1(OC)ncc(-c2cn(C(C)C(=O)N3CCC3C3CCOCC3)nn2)c(OC)n1 CN=c1[nH]c(C(=O)NC(CNC(=O)C(c2cccc(Cl)c2)C)C(C)(C)C)cs1 C1(C(=O)OC(c2ccccc2Cl)C)CCc2ccccc2C1O C1(N(C(C2CC(OC)C2)=O)C)CN(C(=O)Cc2cccnc2F)CC1(C)C c1(C(N2CCCC(CNC(C3C4CCCC34)=O)CC2)=O)cnc2ncccn12 N1(C(C(SC)SC)=O)CCCC(O)(CN(C)C(C2CC(SC)C2)=O)C1 Cc1cccc(F)c1-c1cn(CC2C(CNC(C3(C(N)=O)CC3)=O)C2(F)F)nn1 N1(C(C2C(OC)C2)=O)CCC(C)(CNC(c2ccccc2OCC(N)=O)=O)CC1 C(CCCC(=O)N1CCCC1C(C)NC(C1CC1C1CC1)=O)SC C(C(C)(C(=O)NCC(C1CCN(C(=O)COC2CCOC2)CC1)O)OC)OC Cc1csc(=O)n1CCC(=O)N(CC(C)N(C(=O)COc1cnn(C)c1)C)C C12(NC(C3C(=C)C3)=O)CCC(CNC(c3cn(C)c(=O)cc3OC)=O)(CC1)OC2 CCCC(O)C(=O)N1CC(NC(c2cc(-n3cccc3)ccn2)=O)C(CC)C1 N1(C(c2occ(C)c2)=O)CC2CC(C1)CN(C(C1CC1c1cccs1)=O)C2 c1(C(=O)NC2CC2NC(C2CC2(Cl)Cl)=O)cc(F)cc(Br)c1 c1(C(N2CCC(NC(C3(C)SCCCS3)=O)CC2)=O)cc2occc2[nH]1 CC1(C)OCCC(NC(=O)NC=Cc2cccc(CO)c2)CO1.C(C)(C)(C)O c1(CN2CCCC(NC(C3CCN(C)C3)=O)C2)ccc([N+](=O)[O-])cc1O N1(CC(C)C)CCC(C(=O)NCC(C)NC(C2OC3CCC2C3)=O)CC1 C1(C(N2CCN(C(CNC(C(F)=CCC)=O)C)CC2)=O)Cc2nc(C)cn2C1 N1(C(C2C(C(=O)OCC)COC2)=O)CCOCC1C(=O)Nc1ncc(F)cn1 Cc1ncc2c(n1)CCC(NC(=O)CSc1ccccc1O)C2 c1(C(N2CC(C)C(NC(=O)CCn3ccnc3)CC2)=O)cnn2c1CCCC2 CC(C)(C)C(CNC(c1csc(Cl)c1)=O)C(=O)N1CCC(c2cnco2)C1 N1(C(COCCC=C)=O)CCC(NC(=O)C=C(C)I)CC(O)C1 c1(OCCC)nc(C)ccc1C(=O)NC1CC(NC(=O)C(C)=C(C)C)C1 N1(C(C(CCSC)O)=O)CCC(C)(C)CC1C(=O)NCC(N1CC=CC1)=O N1(C(c2cc(OC)ncn2)=O)CCC2CC2(NC(=O)C=Cc2ccoc2)CC1 N1(C(=O)OC(C)(C)C)C(C(N2CC(NC(C3CCCSC3)=O)C2)=O)CC1C C1(NC(c2c(SC)scc2)=O)CC2CC(NC(=O)C=Cc3sccc3C)CC12 N1(C(C2(N(C)C)CCC2)=O)CCC2(C=C(C(=O)N3CC(O)CC3CO)C2)C1 C1(NC(=O)CC2CCCC2(F)F)CC1C1CCCN(C(=O)C=CCO)C1 Cc1cc(Cl)c(C(N2CC3CC(NC(C4CN(C5CCC5)C4)=O)C2C3)=O)cc1N Cc1cnc(N(C)CC2CCN(C(=O)C(C3CCOCC3)C)CC2)nc1C N1(C(=O)NCC(CC=C)c2ccccc2)CCCC(O)(c2cnn[nH]2)C1 C=C(Br)CC(C)(C)C(=O)N1CCC2(CC1)CC2C(=O)NCCSC Cc1[nH]nc(C(N2CC3CC(NC(C4CCOCC4)=O)CC3C2)=O)c1[N+](=O)[O-] C1(N(C(CCC)c2cccs2)C(=O)Cc2ccncc2)CCNCCC1C c1(OC)cc(OC)c(N)c(C(=O)OCCn2cnc(C)c2C)c1 c1(CC)nn(C)c(Cl)c1C(N1CCC(CCN(C(=O)C(C)(O)C2CC2)C)CC1)=O C1(COC)CCCCN1C(c1ccccc1C)=O Cc1ncc(CCC(N2CC(CNC(c3nc(Cl)cs3)=O)CC(C)C2)=O)c(O)n1 C12(CCCC1)C(OC)CCCCN2CC(c1ccncc1)O.N1(CC=O)CCOCC1.CO Cc1c(C(F)(F)F)n[nH]c1C(=O)NCC(C)CN(C(=O)CN1CCC(O)CC1)C C1(C(=O)NCC23CCC(CC2)N3C(C2CC23CCC3)=O)CC1C1CCCCC1 C1(C(N(CCC(C)NC(C2(C)CCOCC2)=O)C)=O)CCOC1(C)C c12ccc(cc1)OC2OC.c1(N(C(=O)COC)C2CC2)cccc(C)c1 c1(C(N2CC(CNC(c3occ(C)c3)=O)C2)=O)cnn2cc(C(N)=O)cnc12 c1(-c2ccc(C(=O)NC3(CNC(COC(CC)C)=O)CC3)o2)ncccc1Cl N1(C(CC2CN(C)C2)=O)CCC2CN(C(C3CC(=C4CCC4)C3)=O)CC2CC1 C1(NC(C(CC)=CCCC)=O)C2CC1N(C(=O)CN(CC(C)(C)C)C)C2 NC1CC2(CCC(CS(=O)(=O)Nc3cnc4ccc(F)cn34)CC2)C1 C(CCCCCCO)SCC(=O)NC(C1CCC(NC(=O)C(C)(C)C)C1)C CC(C(=O)N1CCC(C)(CNC(=O)C2=CC3CCC(C2)C3)CC1)C(C)S(C)(=O)=O C(CCC(CO)NC(=O)C(C)=C1CC1)NC(C(C)N(CC)CC)=O c1(C(=O)NCC(CN(C(=O)CCNC(N)=O)C)O)cnc2sccn12 C(C(C)(CO)NC(=O)CN(C)C1CC1)NC(CC=CC=C)=O c1(C(C)=O)ccc(CC(=O)NCC(Cc2ccccc2)N(C(=O)C(N)=O)C)cc1 c1(CC)cc(N)ccc1C(N1CCC1CN(C(C1(C)CC=CC1)=O)C1CC1)=O O=C(CCC(F)(F)F)Nc1nc(C2CC(F)CN2Cc2ccc([N+](=O)[O-])[nH]2)no1 C1(C(=O)NC2CC3CC(NC(=O)OC(C)(C)C)C3C2)CC2(CNC(=O)O2)C1 C1(NC(c2cc(F)cc(I)c2)c2n(CCCC)nnn2)CCn2ccnc2C1 C1(CC)(NC(C2OCCC2C)=O)CN(C(=O)CNC=O)C1 C1(CNC(C2CC(=O)NC2)=O)CCC(F)(CNC(=O)Cc2cnc(C3CC3)[nH]2)C1 c1(C(=O)NC2C3CCC2N(C(=O)CC2CC2(Cl)Cl)C3)cc(F)c(F)cc1F c1(C(N2CCC(C(N(CC=C)CCO)=O)C2CC)=O)cc(C#N)[nH]c1C N1(CCc2nc(C(=O)OC(C)(C)C)sc2)CCOC(Cc2ccccc2)C1 c1(CC(C(=O)NC2(c3nn[nH]n3)CCC(F)(F)CC2)NC)c[nH]c2ccccc12 N1(C(CC2C(CC)C2)=O)CCC(CF)(NC(=O)CSc2nnnn2C)C1 Cc1cccc2nc(C(=O)N(C3CCCCC3)C(C)=O)cn12.N1(CC)CCCC1 c1(C(N2CC(N(C)C(c3scnc3Cl)=O)C2)=O)ccc2c(c1)C(=O)CCO2 C1(NC(C(C2CC(F)(F)C2)OC)=O)CC(Nc2cncc(Cl)n2)C1(C)C C12(C(=O)NC3(CC=C)CCC3)CCCC1CCN2C(=O)Cn1cc(CO)nn1 c1(C(N2C3C(CNC(CC#N)=O)CC(CC3)C2)=O)cnc2c(c1)OCCN2 C=C(C)CC(C(=O)N(CC1CCC(NC(=O)CC)C1)CC)NC(C)=O c1(C(N2C(C)C(NC(=O)CCc3ccc(F)cc3)CC2)=O)ccc2nn[nH]c2c1 c1(C(=O)OC)cc(NCC2CCSC(C)C2)nn2c(Br)cnc12 c1(C(N2C(CC)CN(C(c3ncnn3C)=O)CC2)=O)cnc2cccc(Cl)c2c1 C(CCC(C)(C)NC(=O)CC1CCN(C(=O)CN2CCCC2C)CC1)OC c1(CCC)occc1C(=O)NCc1cn(CC(C)NC(=O)C(N)=O)nn1 CC1(C)C(C)(C)C1(F)C(=O)N(CCC(=O)Nc1ccc(F)c(C2CC2)c1)C1CC1 CC(=O)C(C)CC(C)C(=O)NCC(C)(C(C)C)NC(=O)C1=CC(C)(C)C1 CC1(CC(=O)NCC(C2CCCCC2)NC(=O)CCOCCN(C)C)CC1(F)F N1(C(=O)CC2CCCCO2)CCCCC(N=c2ccn3nccc3[nH]2)C1 N1(C(=O)COC(F)(F)F)CCC2C(C1)CN2C(=O)CC1CCSCC1 CC1=C(C(=O)NCC2CCCCN(C(=O)Cc3nc(=N)[nH][nH]3)C2)C(C)(C)CCC1 N1(C(C2C(NC(C3CN(C)C3)=O)C3CCC2C3)=O)CCC(O)C(F)CC1 n1(CC)nc(C(N2CC(NC(=O)CCc3nc[nH]n3)CC(O)C2)=O)ccc1=O C1(NC(C(CC)=CC)=O)(CO)CCN(C(c2cc(Br)cn2C)=O)C1 N1(C(CCCCC)=O)CCCC(C)C1CNC(C1(N2CCOCC2)CC1)=O S(=O)(=O)(c1ccc(Br)cc1NC1COc2ccccc21)N1CCCCC(CC)C1 C1(CC(=O)NCc2cc(C(N(C(C)C)CC3CCCO3)=O)sc2)CC2CCC1C2 C1(NC(CC2ON=C(CC)C2)=O)CC2(C(=O)NCCOCC(F)(F)F)COC1C2 Cc1c(C(=O)NCC2(O)CN(C(=O)C=Cc3ccn(C)c3)C2)cnn1CC(C)C C1(C(=O)OC)CC2(C1)CC(c1nnnn1C1CCOCC1)(NC1CCS(=O)C1)C2 c1(C(=O)NC2CCN(C(c3nccc(C)c3)=O)CC2)c(F)cc(C)cc1Cl C(=O)(CCS(=O)(=O)C(F)(F)F)N1C2C(CNC(=O)COC3CC3)(CCC2)CCC1 C1(OC)CN(C(=O)CCCNC(=O)C2CC2)CC1NC(c1cc(C(C)=O)on1)=O c1(C(=O)NC2CCC(NC(=O)CCC3CCOC3)C2)ccn2c1CCCC2 c1(C(C(N2CC(NC(=O)Cn3nccn3)C2)=O)O)cccc(F)c1 Cc1nc(O)[nH]c1C(=O)NCC1(CO)CCN(C(C2(C)CC=CCC2)=O)C1 C1(C(N2CCCC(F)C2)=O)(CC)CCN(C(=O)CCOCCCOC)CC1 C12(COC)CC(NC(c3cc(C)ncc3C)=O)(CN1C(=O)Cc1ccco1)C2 c1(C(=O)NC2CN(C(C=CC=CC)=O)CC2O)cc2cncc(Br)c2s1 CC1(CCNC(c2scnc2C(F)F)=O)CCN(C(=O)Cc2ccno2)C1 C1(C(=O)NCCCn2c(C)ncc2)CN(C(=O)CCCN2CCCC2)CC1(C)C c1(CC)cccc(CC)c1C(N1CC2CC1C2NC(=O)CC(C)O)=O C(=O)(C(C)S(C)(=O)=O)NC1(CNC(CC(C)CF)=O)CCOCC1 N1(C(C2(C(N)=O)CC2)=O)CCN(C(C2C=CCCC2)=O)C(c2ccccn2)C1 c1(C(=O)NCCN(C(C(C)OC)=O)CC(C)O)cc(O)c2ccoc2c1 Cc1n[nH]cc1C(=O)NC(C)C(=O)NCC(C)Cn1cccn1 C1(C(N2CCC(CN(C)C)C2)=O)CN(C(=O)CC2CCC(C)(C)O2)CCN1C c1(C(=O)NC2CCN(C(=O)C(C3CCOCC3)F)CC2F)cccn2nnnc12 Cc1ccc([N+](=O)[O-])c(C(N2CCC(NC(=O)Cc3conc3C)C(C)C2)=O)c1 CCC(C)(CNC(=O)C(c1ccco1)NC(=O)Cn1ccc(C)n1)C(N)=O c1(CC)[nH]nc(C(=O)NCCOC2CCN(C(c3cc(F)c[nH]3)=O)C2)c1Cl c1(CCC(=O)NC(C(C)NC(C(C)OCC2CC2)=O)CO)c(F)cccc1Cl C1(C)(CO)CCN(C(C)=O)CC1.C1(C(=O)OC)CC(C)N1C(C1CN(C(N)=O)C1)=O CCCCC(CC)C(=O)NC(CC)CCCC(=O)NCCCCOCC Cc1ncc(C=CC(=O)NC2CN(C(=O)CC(C)(O)C3CC3)CC2C)s1 Cc1cc([N+](=O)[O-])ccc1N1CCC(C)C(NC(C2CC(CC3CCCC3)C2)=O)C1 C1(CCC)CN(C(c2ccnn2CCC)=O)CCN1C(C1CC=C(C)CC1)=O C1(N(C(CSC)=O)C)CN(C(=O)CNC(=O)CC2CCCC2)CC1O C(CN=c1[nH]cnc(C)c1C#N)C1CC(NC(C(CC)CC2CCCC2)=O)C1 C1(NC(CC2(C#N)CC2)=O)CN(C(=O)CC2CCS(=O)(=O)C2)CC1CC(C)(C)C CCN=c1ccc(C(=O)N(C)CC2CCCN2C(c2cccnc2S)=O)c[nH]1 N1(C(Cc2nc(C)sc2)=O)CCC2CN(C(=O)COCC3(F)CC3)CCC12 C1(CNC(c2n(C)ccn2)=O)CN(C(=O)C=C2CCOCC2)CCCO1 c1(CN(c2ccc(F)cc2)C)ccc(NC(c2ccccc2)CN)c([N+](=O)[O-])c1 C1(C)(CN(C)C)CCN(C(=O)C(CNC(c2cscc2Cl)=O)N(C)C)C1 C(=O)(C1=NOC(c2ccc(F)cc2)C1)N1CCCC(CN(CC(=O)N(C)C)C)C1 C1(C(N2CC(C)(NC(C3(CC(=O)OC)CC3)=O)C2)=O)CC12CCCCC2 CCC(CC(=O)NC1CCOCC1C(N1CCC1(C)CCO)=O)CC(C)C C1(CNC(=O)C(O)C2CCC2)CCN(C(C2CCS(=O)(=O)C2)=O)C12CC2 CC1CCc2sc(C(=O)NC3(CF)CCN(C(C4CSCN4C)=O)C3)cc2C1 Cc1ccc(Cl)cc1C(=O)N(CC(C)CNC(C1CC1[N+](=O)[O-])=O)C C=C(C)CC(C)C(=O)NCCC1CCN(C(=O)CCc2cnn(C)c2C)C1 C1(NC(c2n(C)nnc2)=O)CCN(C(=O)CCC23CCC(CC2)C3)CC1(C)C S(=O)(=O)(c1cnn(C)c1)N1CCN(C(=O)NCc2ccc(NCC)cc2)CC1C C1(CC)CN(C(C2CCN(C)CC2)=O)CCN1C(=O)CC(O)C(C)C C(=O)(CC1=CCCCC1)N1CCCC(CN(C)C(C2COCCOC2)=O)C1 N1(C(c2cc(C)ncc2)=O)CC(NC(c2csc(Br)c2)=O)CC(C)C1 C1(C)(C(=O)NC2CN(C(CNC(C(CC)C)=O)=O)CC2O)C(C)(C)C1(C)C CN1CCOC2CN(C(=O)C=CCN(C)C(c3cccn3C3CC3)=O)CC12 c1(CN(C(N(C2CCN(C)CC2)CCO)=O)C2CC2)c(S(N)(=O)=O)cnn1C c1(COC)nc(C)c(C(N2CC3CC2(CNC(C2CCCCS2)=O)C3)=O)s1 N1(C(CC(C=C)C)=O)CCC(C)(C(C)(C)N)CC1.c1(-c2cn(CCC)nn2)cc(C)n(CC(F)(F)F)n1 C1(C(=O)OC(CCc2ccccc2)C(F)(F)F)COC2CCCCC12 c1(CN(C)CCN(C)CCN(C(=O)C(F)=C2CCCC2)C)nc(C(N)=O)cs1 C(C(C)(C)CC(=O)NCCNC(=O)Cc1cccc(C#N)c1)N(C)C Cc1oc(Cl)nc1C(=O)NC(C(=O)NC12COC(CSC)(C1)C2)C1CCCC1 c1(C(N2CC3C(C(N4CCN(CCOC)CC4)=O)(C3)C2)=O)cc2ccccc2[nH]1 N1(C(CCC=CC)=O)CCN(C(=O)C(C(C)C)C2CCC2)C(C)C1 c1(CCC(=O)N(CCN(C(=O)C(C)OC2CCOC2)CC)CC)nnc(C2CC2)o1 C1(C)(CCC)CCN1C(=O)C(C)CNC(=O)Cc1ccsc1C c1(C(N2CCC(CNC(C(C)Cc3cnc[nH]3)=O)C2)=O)noc2c1CCCCC2 N1(C(c2cn(C)nc2)=O)CC2CS(=O)(=O)CC2(CNC(C2(CCO)CC2)=O)C1 C1(NC(C(C)OCCN(C)C)=O)CC2CCC1CN2C(c1n[nH]cc1Cl)=O c1(-c2cccc(NC(c3csc(C)c3N)=O)c2)nnc2n1CCCC2 c1(C(=O)NCCC(C)(C)NC(C2CCCO2)=O)ccc2oc(=N)[nH]c2c1 c1(CCC)cccc(C(=O)NCC2CCN(C(=O)C(C)NC(=O)NC)C2)c1 C1(C(N2CC(C)(NC(C(C)=C3CC3)=O)CC2(C)C)=O)C2C3CC4C1C1C2CC3C41 C1(N(C(C(CC)OC)=O)CC)CCCN(C(=O)Cc2scnc2-c2cccs2)C1 C1(c2nnnn2C(C)C)(NC2C(OC)OCCC2)CCC(C(C)C)CC1.C1CS1 Cc1cnc2cc(C(=O)NC3CCC3NC(c3cc(C(F)F)ccn3)=O)ccn12 C(=O)(C1=CCCCCC1)NC1CCN(C(c2cn(C(C)(C)C)nn2)=O)CC1CO C1(NC(CC2N(CC)CCC2)=O)CS(=O)(=O)N(C)C12CCN(C(=O)C1CC1)CC2 C1(C(N2CCC3(C2)CN(C(C2CC4CCC(C2)C4)=O)C3)=O)CN2CCCN1CC2 C(=O)(C(=O)N=S(C)(C)=O)NCCOC(C1CN(C(c2c(OC)cncc2)=O)C1)=O Cc1ccn(C)c1C(N1CC(CNC(c2cc(CN(C)C)no2)=O)C1)=O CC1=C(C)CC(C)(C(=O)NCC23CCC(CC2)N3C(C2C(C)(C)C2(C)C)=O)CC1 C1(OC(C)(C)C)CN(C(=O)COCCF)CCN1C(=O)C(F)C1CC1 c1(C(N2CC(CNC(CC(=C=C)C)=O)C3C2C3)=O)ccc(OC)c(F)c1F N1(C(c2cc(C)nn2C(C)(C)C)=O)CCC2CCN(C(c3ccsc3)=O)CC2C1 C1(C(=O)NCCC(C)NC(c2nc(C)oc2)=O)CCCC(CF)C1 C1(CN(C(c2c(C(C)C)nns2)=O)C)COCCN1C(C1CCCCC1)=O c1(C(CC(=O)O)NC(CN)CCO)ccc(I)cc1 C12(NC(C(C)CN(C)C(C3CCOC3)=O)=O)CC3CC(CC1C3)C2 C#Cc1ccc(Cl)c(C(N2CC(NC(C3(C)CCCC3)=O)CC(O)C2)=O)c1 C1(NC(c2cc(OCC)n[nH]2)=O)CCN(C(C2CCC(C(N)=O)N2C)=O)C1C N1(C(c2cc(OC)n[nH]2)=O)CCCC(O)(CNC(C2CC3CCC2O3)=O)C1 C1(C(=O)NCc2cccc(NC(C(n3ncc(C)c3)C)=O)c2)CCN(C)C(=O)C1 c1(NC(=O)OCC)scnc1C(=O)NCC1CN(C(C)=O)C1.C12CC(CO1)CN2 CC(O)CCCCCC(=O)NC1CC(CCNC(=O)C=C2CCN(C)C2)C1 C1(C(N2CCC(N(C(=O)CCCNC(c3ccco3)=O)C)C2)=O)C(Cl)(Cl)C12CC2 c1(N2CCCC(C(C)NC(C3CCCN3C=O)=O)C2)cc(C(F)(F)F)nc(Cl)n1 C1(CC(=O)NC2CC(CCNC(CN(S(C)(=O)=O)C)=O)C2)NC(=O)CN(C)C1=O CC1(C)CC(CNC(C2(CNC(C3(C)CC4CC4C3)=O)CC2)=O)CO1 c1(NCC(CC)CC(F)(F)F)ccc(S(=O)(=O)NC2CCCCC2N(C)C)cn1 CC1(C)CC(CC(=O)NC2CCC(=O)NC2=O)N(C(=O)CC2CC=CC2)C1 c1(C(=O)OC)c[nH]c(=NCC(C)CNC(c2snnc2C)=O)c2ccsc12 CC(F)CC(=O)N(C1CC(NC(c2cc(CO)[nH]n2)=O)C1)C C1(CNC(C(C)(C)C)=O)CC2CN(c3nc(C4CCCCC4)ns3)CC2C1 c1(C(=O)NCCC(=C)CNC(c2ccc(C)nc2)=O)ccccc1SC(F)F c1(OC)cncc(C(=O)NCCN(C)C(c2ncccn2)C2CC2)c1 C1(N(C(C(CC)c2ccccc2)=O)C)CN(C(c2cnc(=N)[nH]c2)=O)CC1(C)C CC(C)CC(C)C(=O)N1CCCC(NC(=O)CCNC(=O)Nc2ccccc2)C1 C12(NC(C(CCC)OC)=O)CCC(CC1)N(C(C1CC3C=CC1CCC3)=O)C2 c1(C(=O)NC2C(C)N(C(=O)Cn3cnccc3=O)CC2)cc(F)cc2ccoc12 c1(OC)cccc(C(=O)N(C)CC2CN(C(=O)C(N3CCCCC3)C)C2)n1 N1(C(c2c(OC)ccs2)=O)CCC(CNC(c2ncc(N)cc2Cl)=O)C(F)(F)C1 N1(C(Cc2c(C)scc2)=O)CC(NC(=O)C(C)CSCc2cccnc2)C(O)C1 N1(C(C2(COC)CC(F)(F)C2)=O)CC2(CCCC2NC(=O)CC(C)P(C)(C)=O)C1 N1(C(CC2CCCN(C)C2)=O)CCC(C(=O)NC2COC(=O)C2)C12CCC2 c1(C(=O)NCC2C(C(=O)NC3(CCC)CCC3)CC2)cnn(C)c(=O)c1 C(=O)(C(=O)N=c1cc(C)o[nH]1)NC1(CC)CCCN(C(c2c(C#C)c[nH]n2)=O)C1 c1(OC)ccc(C(N2CCCCC2CCNC(C2(OC(C)C)CCOC2)=O)=O)nc1 CC(=O)CCCCC(=O)N1CCCCC(C(=O)NCC(C)N(C)C)C1 N1(C(C(COC)OC)=O)CCC(F)(C(=O)NCc2ncc(C)s2)C1 Cc1cnn(CC(=O)NCC2CC2CC(N2CC(CN(C)C)C2)=O)c1 C(=O)(C1CCc2c[nH]nc21)N1CCC(O)(CNC(C2(C)CCC(=O)N2)=O)C1 n1(CC(=O)NC2CN(C(=O)CCC3CC3)CC3(CC3)C2)ncc2ncccc12 C1(CCNC(C(OC)OC)=O)CC(F)(F)CN1C(=O)Cc1csc(C(C)OC)n1 N1(C(C(=O)NCC)C2CC2(Br)Br)CCN(CC(c2ccccc2)=O)CC1 C=CCC(CNC(=O)CCCc1cccs1)NC(C1CCN(C(C)=O)C1)=O C1(CNC(C(COC)C)=O)CN(C(=O)CC(C)(F)F)CC2(CCC2)O1 c1(-n2cc(Cn3ncc(C)c3)nn2)cccc2[nH]ncc12.N1S(=O)CC1 C1(NC(=O)C=CC2CCCC2)CS(=O)(=O)C12CCN(C(c1cocn1)=O)CC2 C1(CNC(c2cnc(C)s2)=O)CC2(CC(NC(=O)C(C)c3ccsn3)C2)C1 c1(OC)ccc(C(N2CCC(CC(=O)NCCOC3CCCCC3)C2)=O)cc1C c1(C(C(=O)NC2CCOC2)N(C(c2cccc(F)c2)C)C)cc(Br)cc(F)c1F C#Cc1cc(C(=O)NC(CNC(=O)C=C(C)CCC)CC(F)(F)F)ccc1Cl Cc1sc2nc(C(C)NC(=O)Nc3cnn(CC(C)C)c3C)nc(O)c2c1C Cc1cccc(CC(N2CCC(CNC(=O)CN(C)S(N)(=O)=O)C(O)C2)=O)c1F N1(C(C2C(C)CCC2)=O)CCC(N2CCC(NC(c3cc(O)cs3)=O)C2)CC1 C=CCC(C(=O)N1CCC(C)N(C(=O)CCS(C)(=O)=O)CC1)C(C)(C)C C(=O)(C(CC(C)C)C(C)N(CCC(C(C)(C)C)NC(=O)OC(C)(C)C)C)OCC N1(n2cc(CNC3(C(=O)NCc4c(C)noc4)COC3)nn2)CCCC(C)C1 c1(CCCNC(=O)NC(C(C)C)C2CCC2)nc(-c2ncccn2)no1 c1(C(N2C(c3cnc(C)nc3)CCC2)=O)cc(Cl)c(C(F)F)cc1F C12(N)CCC(C(=O)NC34CC(NC(c5ccc(F)c(CO)c5)=O)(C3)C4)(CC1)C2 C(=O)(CC1=Cc2ccccc2C1)NCC1CC(OC)CN1C(C1CCC(O)C1)=O N1(C(C(=O)OCC)=O)CC(CC(=O)O)OC2(CCC2)C1.c12cnc(C)c(c1)OC2 N1(C(C(C)C(C)(F)F)=O)CCCC2(C1)CN(C(=O)CCCc1cnn[nH]1)CCO2 c1(N(C2CCCCC23CCC3)C)nc(=N)[nH]c(=NCc2cnn(CCF)c2)[nH]1 Cc1cc2cc(C(N3CCN(C(C4CCC(CO)CC4)=O)C4CC34)=O)ccc2[nH]1 c1(CC(=O)NCCC2CCN(C(c3cc(C)c(C)o3)=O)CC2)cn2ccsc2n1 CC(C)C(C)(CNC(c1cnn(C)n1)=O)NC(=O)C=Cc1cn(C)cn1 C(=O)(CC(CC)C(F)F)N1CCC(N(C(CCOCC#C)=O)CC#C)CC1 CC(C)(C(=O)NCc1nocc1C(=O)NCC1CC1Cl)c1ccno1 c1(CC(=O)NC(CNC(C2(COC)C=CCC2)=O)(C)C2CCC2)cccnc1C N1(C(c2n(CC)cnn2)=O)CC2(CCN(C(=O)CC3CCCNC3=O)C2)C1 C(=O)(CC(C)(C)C(=O)NC(CNC(=O)Cc1nc2ncccn2n1)CC)OCC C(CC(C)C(=O)NCC1CN(C(=O)CN(C)C(=O)OC(C)(C)C)C2CC12)=CCC Cn1ncc(C(N2CCC(CCNC(=O)CCc3c[nH]c(=N)[nH]3)C2)=O)n1 Cc1ncsc1C=CC(=O)NCC1CCN(C(c2cc(Br)n(C)n2)=O)C1 C(CCN(C(=O)COCC(C)(C)C)C)(C(C)(C)C)NC(C1(CC#C)CCOC1)=O C1(CNC(C(CCSC)N(C)C)=O)CCCCN(C(=O)C(C)(C)c2cncs2)C1 C1(C(N2CC(NC(c3c(Cl)cn(C)n3)=O)C(F)CC2)=O)COc2ccccc2C1 C(c1ccccc1)=CC=C(C(=O)N(CC(=O)OCC)CC=C)C.C1CO1 N1(C(C(c2ccc(Cl)cc2)C)=O)CCC2(CCCN2c2ccnc3ncnn23)C1 N1(C(C=CC(N)=O)=O)C2CCC1C(NC(=O)CCCn1cncn1)C2 c1(C(=O)NC(CC)CNC(=O)COCC(F)F)cnn(-c2ccccc2F)c1N N1(C(CCN(C)CC)=O)CC2CCC(N(C)C(c3cc(C)cc(Cl)c3)=O)C2C1 c1(C(=O)NC23CN(C(C(C)NC(C)=O)=O)C(C2)C3)cc(F)cc(C)c1N c12cccc(n1)NC(=O)C2.CCC(C(=O)NC12CC(NC(C)=O)(C1)C2)N(C)C c1(CC)ncccc1C(=O)NC(C)(C)CCNC(=O)C(C)C(C)C C(=O)(C1=NOC(NC(=O)C(C2CC2)OC)C1)N(CCCN(CC)CC)C C1(CC(=O)NC(C(N2C(C)(C(=O)OC)CC2)=O)C)CC2CCC1O2 Cc1ncc(NC(C2CCCN(Cc3cc(Cc4cccs4)on3)C2)=O)nc1C c1(C(N2CCC(N(S(C)(=O)=O)C)C2)C(=O)NCC2CCOC2)sc(Br)nc1Cl c1(NC2(CO)CCN(Cc3cc(Br)cnc3Cl)CC2)ncnc2cc[nH]c12 c1(NC(c2n(CC)nnn2)c2cncn2C(C)C)cccc(OCC(C)(C)O)c1 C1(CNC(CCCOCC)=O)CCN(C(c2c(C)noc2C(F)F)=O)CC1(F)F C(c1cccnc1)=CC(=O)NCC1(CC(=O)NC(CC)C(C)O)CC1 C1(CNC(CC(C)(F)F)=O)C(C2CC2)CCN1C(=O)Cc1nc(C2CC2)cs1 n1(CC)nc(C2CC2)cc1C(=O)NCC1CN(c2nnc(C(F)(F)F)s2)CC1C CC1(C(N2CCC(C)(C(F)(F)F)CC2)=O)CCCN(C(c2ccccc2I)=O)C1 C=C=CCCC(=O)N(C1CCCC1)CCCNC(=O)CNC1(c2ccccc2)CC1 C1(C(N(C(C)CNC(=O)C=CCOCC(F)(F)F)CC)=O)CCN(C)CC1 c1(N(CCC)C)ccc(C(N2CCCCC2CN(C(=O)C2=CCSC2)C)=O)cc1 N1(C(c2n(C)ccn2)=O)CCN(C(C2CC2c2ccccn2)=O)CC1 CCC(CC)C(C)N=c1cc[nH]cc1S(=O)(=O)NCC1CCOCC1(C)C N1(C(C(=Cc2ccccc2)OC)=O)CCN(C(c2cnc(C(C)C)[nH]2)=O)CC1C CC12CC(C(=O)OC(C)(C)C)(C1)C1(CCN(C(=O)CSCc3cccs3)CC1)O2 FC1(F)CCCC(NC2(c3nnnn3C3CCCC3)COC(C3CC3)C2)CC1 C1(NC(COC2(C)CCCC2)=O)CCN(C(C2CC23CC(O)C3)=O)C12CCCC2 C(=O)(C#CC1(C)COC1)N(C)CC1CCN(C(C23CCC(C2)C3(C)C)=O)C1 Cc1cc(C(=O)O)cc(CNC(c2cc(Cl)c(Br)[nH]2)=O)c1 C#CC1(CN(C(CNC2CNC(=O)C2)CO)CC=CCCCCC)CCCC1 C1(C(=O)NCC(COCC)(C)C)CC(NC(=O)CC2CC3C=CC2C3)CCO1 N1(C(C(CC)CO)=O)CC2CCN(C(C3CC=CCC3)=O)CCC2C1 O=c1n(CCN2CCC=C(c3ccco3)C2)nc2ccccn12 c1(C(=O)NC2CC3(CC(NC(=O)CCn4cccc4)C3)C2)cc2sccc2cn1 N1(C(c2ccc(OC)cn2)=O)CC2CS(=O)(=O)CC2(NC(c2cscc2F)=O)C1 c1(NC(C2N(C(Cc3cc(C)no3)=O)CC(C)C2)=O)ccc2c(c1)CNC2=O C1(C(=O)NC2CC2C(=O)NCC2CN(C(C)=O)C2)CCCCC1n1cccc1 C12(C(N3CCC(C(C)(C)NC(CC(CC)OC)=O)C3)=O)CCC(C#N)(CC1)CC2 C#Cc1ccnc(C(=O)NCC(C)CNC(c2cccc(CC=C)c2)=O)c1 CCC(CC(C)O)NC(C1(SC)CN(C(c2csc(C)n2)=O)C1)=O C(=O)(C1=C(F)CN(C(=O)CCCC(C)=O)CC1)NC(CCC)CC N1(C(CC=CCC)=O)CC(NC(=O)CCc2nc(-c3cccs3)no2)CC1(C)C c1(C(N2C(C(=O)NCCCCC3CCNCC3)CCC2)=O)cccc(O)c1 N#Cc1c(Cl)nsc1NCC1CCCCC1NC(C1CC12CCCC2)=O C1(C)(C(N2CC(CC=C)(NC(=O)Cn3ncnn3)C2)=O)Cc2ccccc2NC1=O C=CC(C)(O)CC(=O)N1CCC(N(C)C(c2ccc(CO)cc2)=O)C1 c1(C(=O)NCC(CC(C)C)NC(c2c(CC)ncnc2)=O)cncc(F)c1Cl Cc1ccc(N)cc1C(N1CCC(NC(=O)CCF)C(O)C1)=O N1(C(C2CC(C)N2C(c2cc(Cl)cs2)=O)=O)CCc2cnccc2C1 N1(C(C2N(C)CCC2)=O)CCC2CN(C(C3CC(C)(F)C3)=O)C2C1 c1(C(=O)NC2C(OC)CN(C(C(CC#C)O)=O)C2)ccc(OC)nc1F N1(C(C(C=C=C)C)=O)CCN(C(C2(CC)CC(C)(C)C2)=O)CC1C C1(CNC(C(c2ccccc2)OC)=O)C=CC(NC(=O)CCc2ccncc2)C1 N1(C(C(CC)=CC)=O)CCN(C(c2cc(C)c(N)cn2)=O)C2CCCCC12 c1(OC)ccc([N+](=O)[O-])cc1NC(C1COCCN1Cc1cnc(Cl)c(Cl)c1)=O C1(NC2(c3n(C(C)C)nnn3)CC3COCC3C2)CC2C(=O)NCC(=O)N2C1 Cc1cc(C)n(-c2cccc(CNCC(c3nc(C)c(C(F)(F)F)s3)C)c2)n1 C(=O)(C(C1=CCSC1(C)C)N1CCC(CCO)CC1)NCC c1(-c2ccc(OC)c(C)c2C)cccc2[nH]c(C(=O)NC3CCCC(O)C3)cc12 C(=O)(C(CNC(c1cc(C)on1)=O)C(C)(C)C)N(CC#C)C N1(C(CCn2cc(CNC(=O)OC)nn2)=O)CCc2nc(C)ccc2C1 C1(C(N2CC(CCNC(COCCCC)=O)OCC2)=O)CC2(C1)CC2(F)F n1(CC)cc(CC(=O)N(CCCNC(C2CC3CCC2C3)=O)C(C)C)c(C)n1 N1(C(c2cc(C)sc2C)=O)CC(=O)NC2CN(C(=O)C=Cc3cncs3)CCC12 c1(C(N2CCC(N(C(=O)C(C3CC3)SC)CC)C2)=O)cc2nc(C)cc(C)n2n1 Cc1noc(C)c1C(C)C(=O)N1CC(n2cc(CNC(C3(CO)CC3)=O)nn2)C1 C1(CC(=O)NCC(CC)NC(=O)Cc2csc(C(=O)OC)c2)COC2CC1C2 CC(O)C(C(=O)NCCCNC(=O)CC1(C)CC(F)(F)C1)NC(=O)OC(C)(C)C N1(C(CC(C)(C)C)=O)CC(NC(C2CCNC2=O)=O)CC2(CCOCC2)C1 N1(C(CC(C)CCc2ccc(I)cc2)=O)Cc2[nH]cnc2CC1C N1(C(C=CC)=O)CCCC1CC(N1CC(C2CC2)C1)=O.C12CC(C1)N2C N1(C(CCCc2onc(C)n2)=O)CCC(NC(c2nc(Cl)cs2)=O)C(F)C1 C1(C2CCCN(C(=O)C=Cc3ccccc3)C2)(NC(COCC=C)=O)CC1 Cc1nc2cc(Cl)c(NC(C3(F)CN(C(c4cnc(F)cc4C)=O)C3)=O)cc2o1 CC1(C)CC2=C(C(=O)N1)C(c1cccc([N+](=O)[O-])c1F)NC(=S)N2CC1CC1 C12(C(=O)NCCN(C(CC3CC(=C)C3)=O)C3CC3)CCCCC1OCC2 c1(SC)cccc(C(N2CC3CC2CN3C(c2cc(O)n(C)n2)=O)=O)c1Cl N1(C(c2c(CC)noc2)=O)CC(O)CC1(C)C(=O)NCc1ccn(C(C)C)n1 C1(C(=O)NC2CN(C(C(CC#C)(C)C)=O)CC2(C)C)CCn2cc(C)nc2C1 C1(NC(c2ccc(N)cn2)=O)CC2CCCC(C1)N2C(C1CC12CC2)=O N1(CC(=O)NCC23N(C(C(C(CC)C)C)=O)C(CC2)CC3)CCCCCCC1=O N1(CC(=O)NCCCN(C(=O)CSc2cccc(F)c2)C)CCCCC(O)C1=O C12(C(=O)NCC3CC(NC(CC(C)c4cnn(C)c4)=O)C3)CCC(CC1O)C2 C(=O)(CS(=O)(=O)CCOC)NCCC(=C)CNC(c1ccc[n+]([O-])c1)=O N1(C(CN(C)C)=O)CCC(NC(c2ccccc2OC2CC2)=O)C(CO)C1 c1(C(=O)NCC2CC(C)N(C(=O)CCCC(F)F)C2)cccc2nsnc12 C1(CNC(CC2(OC)CCC2)=O)CCC(C)N(C(=O)CCCC2CCC2)C1 C1(NC(CC(C)C2CC2)=O)CC2(CCN(C(c3cncn3C3CC3)=O)CC2)C1 N1(C(C(=O)NC(CC)CNC(=O)CSc2ccccc2F)CC)C(=O)CCC1=O N1(C(CCCOCC)=O)CC(NC(c2cc(C(C)(C)C)oc2C)=O)C2CC12 c1(C(=O)NC(CC)COc2ccc(C(C)(C)C)cc2)cnc2cccc(Br)n12 c1(OCC(N2CCC(NC(c3nnc(C)o3)=O)C2)=O)cccc(F)n1 C1(C(=O)NCCCOCCNC(C(n2ccc(C)n2)(C)C)=O)CCC2C1C2(F)F c1(C(=O)NC2C(CNC(c3ccn(CCOC)n3)=O)CCC2)cccc(F)c1C c1(C(=O)NC2C(N(C(C(C)C#N)=O)C)CCCC2)ccc([N+](=O)[O-])c(N(C)C)c1 C(C(C(C)C)C(C)C)NC(CC(OC)OC)(C)c1nnnn1C1CCCC1OC N1(C(C(C=C)(C)CC)=O)C(CNC(=O)CN2CC3CC3C2)CC2COCC12 N1(c2c(C)cncn2)CC2CC1CN2C(c1ccn(-c2cccc(F)c2)n1)=O c1(CC(N2C(CNC(C3C(C(=O)OCC)CC3)=O)CC2)=O)csc(S)n1 N1(C(c2cc(SC)oc2)=O)CCCC2CN(C(c3cc(=O)cc(Cl)[nH]3)=O)CCC12 C(=O)(CCCC(F)F)NCCCC.S(C(F)(F)F)CC(=O)OCC(F)F C1(CC(=O)NCCN(C(=O)Cc2sccc2C)CCC)CC(C)=NO1 C1(NC(C2CN(C(C)=O)C2)=O)CCN(C(c2cn(C3CC3)nc2C)=O)C1C1CC1 c1(C(=O)NCCC2(CNC(C34CCCC3C4(F)F)=O)CC2)ncnc2ccsc12 CC(CC1CCC1)N=c1[nH]c(=NCc2cc(Cl)nc(Cl)c2)[nH]c2cccc(F)c12 C1(CNC(C2C(C)CC=CC2)=O)CCN(C(=O)Cc2cccnc2Cl)C1(C)C C1(N(C(=O)COC(F)F)C)CCCC(NC(C2(C#N)CCC2)=O)C1 N1(C(CCNC(C)=O)=O)CCC2(NC(=O)Cc3nnc(C)o3)CCCCCC12 C1(C)(NC(COCCCC#C)=O)CCN(C(C2(OCC)CCCCC2)=O)C1 C1(OC)C2CC3CC1CC(C(=O)NCCC(C)NC(=O)C(C)CN(C)C)(C3)C2 c1(OC)ccc(CO)cc1C(=O)NC(C1CCCCN1C(C1CC(F)C1)=O)C Cn1cncc1-c1cn(C2CCN(C(=O)C(C)(O)c3ccsc3)C2)nn1 c1(OC)cnccc1C(N1CCC(C)C1CNC(=O)CCc1cccnc1C)=O C(=O)(CCCN=[N+]=[N-])N(C1CC(C#N)C1)CC(=O)N(CCCC(C)(F)F)C Cc1ccc(C(C)CC(=O)NCCCCn2cc(C(C(C)C)N(C)C)nn2)cc1 C1(CC)CCCC1(C)C(=O)NCCCN(C(=O)CCC1CCCC(=O)N1)C N(C(=NCCc1cccs1)NCc1ccnn1C)Cc1ncc(C)cn1 N1(C(C(C)=C2CC2)=O)CCCC(C2(NC(C3(C)CCOCC3)=O)CC2)C1 C1(OCCNC(C(C)C2CCC2)=O)(CNC(C2CCCC(=O)O2)=O)CCOCC1 C1(NC(C(F)=CCC)=O)CCC2CCN(C(c3cc(C)n(CC)c3C)=O)C1C2 CC1(CCO)CCN(C(=O)CSC2CC2)C1.C12(CC1)C(=O)N2 CCC(C)C(O)C(=O)NCCCCCCN(C)C(c1ccn(C)n1)=O C(C)(CCNC(C1CC1CF)=O)NC(COCCC)=O c1(C(N(CC(C)NC(c2scnc2C(C)(C)C)=O)C)=O)ccc(F)cn1 Cc1cc(C(N2CCOC(CCCNC(=O)CC3C(C)C3(F)F)C2)=O)nc(O)c1 c1(C(N2CC(C)C(CNC(=O)C(C)NS(C)(=O)=O)CC2)=O)ccn2c1CCCC2 C=C(C)CC(C(=O)N(C)CCNC(c1n[nH]c(CC)c1Br)=O)NC(C)=O c1(SCCNC(c2n(C(C(=O)OC)C)nnn2)=O)cccnc1Cl C12CCN(C1)C2=O.n1(CC(=O)NC2CCC2C(F)(F)F)cnnn1 N1(C(C(CC)Sc2ccccc2)=O)CCCN(C(C2(CCN(C)C)CC2)=O)CC1 C1(C(=O)NCCn2ccnc2)CN(C(=O)C=Cc2cocn2)C2(CCC2)C1 c1(N2CCC(CN(C)CC)CC2)cc(NC(c2ccncc2F)C)nc(C)n1 C1(C(C)NC(=O)CCC2CC2(Cl)Cl)CCN(C(c2c[nH]cc2Br)=O)C1 C1(CNC(C(C)OC2CCOC2)=O)CCCC1NC(=O)CSc1ccccc1 CCS(=O)CC(=O)NC(CCN(C(=O)C=Cc1cn[nH]c1)C)C(C)C C#Cc1ccc(F)c(NC(C)CCN(C)C(=O)OC(C)(C)C)c1 c1(CNC(CC2C(CNC(c3c(CC)ncnc3)=O)C2)=O)ccc(F)c(O)c1 N1(C(C2(CCNC(C(CC)=CCCC)=O)CCC2)=O)CC(CO)C(C)(C)C1 c1(CC(=O)NCC(CC)NC(=O)CCc2cc(C)on2)ccc(S(N)(=O)=O)s1 N1(C(C(N2CCC(NC(C3OCC(C)C3)=O)C2)=O)C)CCC(O)CC1 c1(NC)ccc(C(N2CC3C(CNC(=O)C(C(C)C)NC(N)=O)C3C2)=O)cc1 Cc1cc(C(N2CCN(C(=O)CSc3n[nH]c(O)n3)CC2C2CC2)=O)cc(C)c1 N1(C(C2COCCN2C(=O)CCc2cnc[nH]2)=O)CCC2(CCCNC2=O)CC1 N1(C(Cc2c(C)con2)=O)CC(NC(=O)CCS(C)(=O)=O)CC12CCCOC2 c1(NC23CC(NC(=O)CNC(C4(C(F)(F)F)CC4)=O)(C2)C3)ccc([N+](=O)[O-])cn1 c1(C(N2CC(COC)N(C(=O)Cc3cncs3)CC2)=O)cc(Cl)cc(C)c1N C1(OC)CC(OC(c2[nH]c(-c3cccc(C)c3)nc2C)=O)CC(OC)C1 C(=O)(CN=c1cc[nH]cc1)N1C2C(NC(=O)C(=Cc3c[nH]cn3)F)C(C2)C1 C1(OC2(CC(=O)NC3(n4cccc4)CC3)CC2)CN(C(=O)COCCCF)C1 c1(CCN(CC(O)C(=O)N(CCC(=O)N(C)C)CCO)C)ccccc1N C1(NC(Cc2ccc(C)s2)=O)CC2CN(C(=O)CC(C)C)CCN2C1=O CC1=C(C(=O)N2CCC(C)(C(=O)NC3CC3C(C)(C)C)CC2)CCO1 N1(C(C2(CC#C)CCC2)=O)CC(NC(C2CCCC2C2CC2)=O)C(SC)C1 N1(C(C)=O)CCN(C(=O)C(F)NC(C2(SC)CCC2)=O)C(CC2CC2)C1 Cc1cn(C)nc1C(=O)N(C)CC1(NC(=O)CCc2ncccn2)CC1 N1(C(c2cc(C)n(C(C)C)n2)=O)CCC2OCCN(C(C3CCC(C)O3)=O)C2C1 N1(C(C2CC3CC3N2C(c2ccc(Cl)c(Cl)c2)=O)=O)CCc2sc(Br)cc2C1 C(=O)(C1CCCc2cccnc21)NCC(C)NC(=O)C1=CCCCCC1 C1(NC(c2cn3c(n2)COCC3)=O)CC2(CCN(C(C34CCN(CC3)C4)=O)C2)C1 C1(CC(=O)NC(CCNC(C(C)(C)CC#N)=O)(C)C)Oc2ccccc2NC1=O Cc1nc[nH]c1CC(=O)NC1CC(C)(NC(=O)C(C)OCCC(C)C)C1 c1(C(=O)NC2C3(CN(C(CC(=O)OC)=O)C3)SCC2)ccc2c(c1)N(C)C(=O)C2 C(C(O)CN=c1cc(F)nc[nH]1)NC(C(CC)SC)=O CC1CCCCN(C(c2cn(C(C)C)cn2)C(=O)NCCC2CC2)C1 Cc1cn2cc(CC(N3CCOC(c4ccc(F)cc4F)C3)=O)nc2s1 C=CCCC(CC(C)C)C(=O)N1CCCC(C(=O)NCc2ccnc(F)c2N)C1 C1(C2CCCO2)(C(=O)NC2CC(CNC(C3CCS3(=O)=O)=O)C2)CCCC1 Cc1ccn(CC(=O)NCC(C)CN(C(=O)CCCc2cnn[nH]2)C)c(=O)c1 c1(C(=O)NC2CCN(C(C3C(C=C)C3)=O)C2C2CC2)sc2cc(Cl)ccc2c1Cl C12(C(=O)OCC)CC(C(=O)N(c3ccccc3)CCOC(C)C)(C1)OC2C C(=O)(CC(C)(C)CC(F)(F)F)N(CCNC(c1c(C)c(Br)sc1)=O)C Cc1nc2n(n1)CCN(C(=O)Cc1cc(C(N3CC4(COC4)C3)=O)cs1)C2 n1(CC(=O)NCCc2ccc(OC)cc2F)c(C)nc2ccccc2c1=O CCCCCC(C)CC(=O)NCC1CC(C(=O)NCc2c(C)coc2C)=NO1 C(C(C)(C)C(=O)OCC)N(CC(O)Cn1cccn1)CCC C1(C(=O)NC2C(NC(c3c(C)con3)=O)C2)CCc2c[nH]nc2C1 C12(C(=O)O)C3C4C1C1C2C3C41C(=O)NCC(O)(C(F)(F)F)c1ccccc1 C1(N(C)C(c2cnc[nH]2)=O)CC2CCC(C1)N2C(c1cnnc(O)c1)=O N1(C(C(=O)NCc2c(CCNC(C(C)N(C)C)=O)ocn2)C)CCC(O)CC1 N1(C(C(=Cc2cn[nH]c2)C)=O)CCC(C(N2Cc3cncnc3C2)=O)CC1(C)C N1(C(c2cc(OC)no2)=O)CCC2CN(C(=O)C=Cc3ccncc3)CC12 c1(NC(CC)=O)cncc(C(N2CC(N(C(=O)CC(F)F)C)C2)=O)c1 C1(NC(C(C)CF)=O)CN(C(C2(C#N)CCCCC2)=O)CC2(CC2)C1 CCCCC(O)CNC(C1(C(C)NC(c2ccn(CC)n2)=O)CC1)=O C1(C(C(=O)NC(CC)C)N(C)Cc2cccnc2)CCC2(CC2)C1 c1(OCC)cc(C(=O)NCCNC(=O)CCN(C)C(c2ccoc2)=O)oc(=O)c1 c1(CC(C(=O)NCCN(C(=O)Cc2ccn(C)n2)C)OC)ccc(F)cc1 C1(C(N(C2CCN(C(C3(SC4CC4)CCC3)=O)C2)CC)=O)CC1C1CC1 C(C(=O)N1CC(O)C(O)CO1)C1CCN(C(Cn2c(C)ccc2C)=O)C1 C1(O)(CNC(c2cn(CCCF)nn2)=O)CCCN(C(c2ccns2)=O)CC1 Cc1cc(C(=O)NC2COCC2NC(=O)CCc2nccn2C)cnc1C(F)F N1(C(C)CNC(c2ccnnc2)=O)CCN(C(C2(F)CCCC2)=O)CC1 c1(NC(CC2C(C)(C)C(NC(=O)CSC3CC3)C2)=O)cccc2c1CCC2 N1(C(C(C)(C)OC(C)C)=O)CC2CCC(C1)N(C(c1ccc(F)c(F)c1)=O)C2 N1(C(C2COCCN(C(c3c(CC)nc(C)o3)=O)C2)=O)CC2CCCCC12C N1(C(C2CCN(C(CC)=O)C2)=O)CCCC(NC(c2cscc2OC)=O)C1 C=C(Cl)CCC(=O)NC(CCOCCO)C(=O)Nc1cccc(N(C)C)c1 C1(NC(c2cc(F)ccc2F)=O)CCN(C(c2csc(Cl)c2)=O)CC1F CC(=Cn1ccnn1)C(=O)NCCCC(C)NC(C1SCCS1)=O C1(CC)(NC(=O)C(C)OCOC)CCN(C(=O)C=CCF)CC1 C1(C(N2CCC(CCNC(C34CCCN3CCC4)=O)C2)=O)C(F)(F)C12CCC2 C=CC(F)(F)C(=O)NC1CC(NC(c2csc(O)n2)=O)C1 n1(CC(N2CCC(NC(C3C(C)C3)=O)C2(C)C)=O)nnc2c1CCCC2 C1(NC(c2n(OC)cnc2C)=O)CC2(CCN(C(=O)C=C3CCN(C)CC3)C2)C1 c1(CC)ccnc(C(=O)NC2(CC)CC2(C)C)c1.C1(C)C=CC(=O)N1 c1(CC)ccc(OCC(=O)NC2CCC(C(=O)Nc3ccc(C)cc3)CC2)cc1 CCC(CC)C(C(=O)N(CC(=O)NC1CCC(C(N)=O)C1)C1CC1)OC C#Cc1ccc(C(=O)NC2CC3(C2)CC3NC(c2cnc(C)[nH]2)=O)c(OC)c1 N#Cc1cc(C(N2CCC(NC(c3cnn[nH]3)=O)CC2C2CC2)=O)c(O)cc1N C1(CC(=O)NC(C2(O)CCCCC2)C(=O)NCc2c(C)ncs2)CC2C=CC1C2 CP(C)(=O)CCC(=O)C1C(C(=O)N(c2c(O)cccc2F)C)C(NC)C1 CCC(C)CCCCC(=O)N1CC(C)(C)CC1CC(=O)Nc1cnc(Cl)c(C)c1 C1(C)(NC(C2(C)N(C(c3cc(C)n(C)c3C)=O)CC(O)C2)=O)CN2CCC1CC2 C1(CC(=O)NC)CC(CN(CCn2cc(CCCO)nn2)C(C)=O)C1(C)C Cc1ccc(O)c(C(N2CC(NC(c3cccn(C)c3=O)=O)CC2C)=O)c1 c1(C(CN(C(=O)CN(CC(C)(C)C)C)C)NC(COC(C)=O)=O)ccccc1 CCCC(C(=O)N=c1ccn(C(F)F)[nH]1)NC(=O)CN1CCCC1C Cc1ccc(CC(=O)NC2CN(C(=O)C(N3CCSCC3)C)CC2(C)C)c(F)c1 S(=O)(=O)(c1c[nH]c2cnc(Cl)cc12)NC(c1ccc(N2CCOCC2=O)cc1)=O c1(C(N2CC=C(CNC(C3C(C)CN(C)C3)=O)CC2)=O)c(O)ncc2c1CCC2 C1(CN(C(=O)C(F)n2cccn2)CC)CCC(NC(CC2C(CC)C2)=O)CC1 CC(c1ccco1)=CC(=O)NCCCC1CCCN1c1ccnc(C2CC2)n1 c1(C(=O)NC(C)(C)CC=CC(=O)NC2CCOCC2F)cc(F)ccc1O c1(C(=O)NCCC(O)C(=O)NC(c2ccccc2)CF)ccc2cc[nH]c2c1 N1(C(c2n(CCC)ncc2)=O)CC2CC(NC(C3CC4CCC3CC4)=O)CC2C1 C1(C(=O)NC2(C3N(C(c4cncc(NC)c4)=O)CCC3)CC2)CCCC12CCC2 C1(C(N2CC(CNC(c3ccc(F)o3)=O)C2)=O)CCCC12CC2 CCC(C)C(O)CC(=O)NC(CC)CCCC(=O)NC(c1cnn(C)c1)C C1(NC(Cn2c(C(C)C)nnn2)=O)CCC(C)(CNC(C2CC(F)(F)C2)=O)C1 Cc1cc(C)nc(N2CCN(C(c3cccc(O)c3)=O)CC2CO)n1 c1(C(=O)NCCCC(C)NC(C2COC(C)(C)CO2)=O)cc(S(N)(=O)=O)c[nH]1 c1(C(C)NCc2c(NC)nccc2)ccc(F)c(Br)c1 C12(OC)CCC(C(=O)NCC(CNC(C3CC=C(C)CC3)=O)CO)(CC1)C(=O)C2 N1(C(=O)Cc2nc(C3CCCC3)no2)CC2CC(C1)N(C(c1coc(Cl)n1)=O)C2 Cc1nn(C)c2c(NCc3nc(-c4cccc(C(F)(F)F)c4)no3)ncnc12 N1(C(CCCC=C)=O)CC2CCCCC2(NC(=O)CSc2nc[nH]n2)C1 C=CCC(C(=O)N(C1CCN(C(=O)C(CCCC)ON=C(C)C)CC1)C)C(C)C n1(C(CC)C)nnnc1C(CCC1CC1)NCc1cocn1 C1(NC(c2ccn(CCF)n2)=O)C2CN(C(C3(F)CCCOC3)=O)CC12 c1(C(N2CCC(O)(C(=O)OC)C2)C(=O)NC(CC)C)cc(S(C)(=O)=O)c(C)o1 c1(C(=O)NC(CNC(CCCCOCC)=O)CCOC)c(N)ccc(F)c1F c1(C(N2CC(CC=C)(C(=O)NC(CC3CC3)CO)C2)=O)cc2ccccc2[nH]1 N1(C(c2c(COC)cc[nH]2)=O)C2CCC1CN(C(=O)CN1CC3CC3C1)C2 c1(SC)nc(=NC2CCCN(C(=O)CC34CCCN3CCC4)C2)c(C#N)c[nH]1 Cn1nc(Cl)c(C(=O)N(CCCN(C)C)CCNC(C2C3CCCC23)=O)c1Cl c1(OC)c(Cl)ccc(Cl)c1C(=O)NC1CC(CNC(C2NC(=O)CC2C)=O)C1 CN1Cc2ccccc2C(NC2CCCC2CN)C1 CCC(CC(=O)Nc1cn(C)nc1C(C)C)NC(c1ccsc1C)=O C=C(C)CC(C)C(=O)N1CCN(C(=O)C(C)(C)OC)CC1c1cn[nH]c1 CCCCCCC(CC)C(=O)NCC1CCN(C(c2cnc3ccccn23)=O)C1 C1(CC=C)(C(=O)NCCC2(O)CN(C(c3cc(C(C)C)on3)=O)C2)CCOCC1 N1(C(CN(CC)CC)=O)CCC(n2cc(Cn3cc(C)cn3)nn2)C1 Cc1ccc(C(=O)NC23CC(C(=O)NN4CCCCCC4C(N)=O)(C2)C3)c(C)c1 C1(CNC(=O)OC(C)(C)C)OCCC1(C)C.C12C(C1(C)C)NC2=O C(=O)(C(CCC(C)C)N1CCC(O)(c2cnnn2C)CC1)NC(CC)(C)C C(C(F)(C(=O)NC1COCCC1CO)C(C)C)NC(c1c(C)scc1)=O Cn1cc(C(=O)CN2C(C)(N(C(=O)CC3(CS(C)(=O)=O)CC3)C3CC3)CC2)cn1 C1(C)(CNC(C2CCC3CC23)=O)CN(C(C2(OC)CC(C)C2)=O)CC1C C(C)(C(C(=O)NCC1OCCC1(C)C)C(C)C)NC(c1c(NC)nccc1)=O C(C)(C)(CN=c1[nH]cnc(NCc2cccnc2C(F)(F)F)c1C)OC c1(C(=O)NCc2scc(C(=O)NCC(CC)CC)c2)ccc(C)c(C)n1 c1(CC)ncoc1C(=O)NCCOCC(=O)NCC=C1CCSCC1.C1CC1 Cc1ccc(C(=O)N(CC(N2CCC(OC(C)=O)C2)=O)C2CCC2)c(O)c1 c1(OC)cnc(Nc2ccsc2C(N2CCSCC2C(=O)OC(C)C)=O)nc1C C#CC1(O)CC(C(=O)NCC(CC(=O)N(CC(=O)NCCC)C)C2CCC2)C1 C(=O)(C(F)C(C)CNC(C1CC(F)CN1C)=O)NC(C(C(=O)OC)C)C CC1CCCC(CCO)N1C(c1cnn(C)c1-c1ccccc1)=O c1(C(=O)Nc2c(C(=O)NCC)cccc2)nccc(C#N)c1Cl C1(C)(N(C(=O)CCOC2CN(C(=O)CC3C=CCC3)C2)C)CCOCC1 CCCCC(O)C(=O)N1CCC(C)(C)C1CNC(=O)CCc1ccc(CC)cc1 c1(C(=O)NCC(C)N(C(c2ccc(C(N)=O)s2)=O)CC)ccc(C2CC2)cc1 Cc1c(CC(N2CC(CNC(C3CC(=C4CCC4)C3)=O)CC2C)=O)cnn1C C1(NC(CC2(OC)CCCC2)=O)CN(C(=O)C(C)N=[N+]=[N-])CC1O C1(NC(CCC(=C)Cl)=O)CC2CC(C1)N(C(c1cccc(N)c1F)=O)C2 Cc1cn(C)cc1C(=O)NCCN(C(c1ccc(N2CCCC2)nn1)=O)C(C)C C(CNC(=O)C(C)CSC)(C(=O)NCC1(OC)CN(C)C1)OC C1(N(C(c2nc(C#C)sc2)=O)C)CCCN(C(C2CC2(Cl)Cl)=O)CC1 c1(C(=O)NC2C(NC(C3(CC)CCCC3)=O)CCC2)ccc2c(n1)CCC(C)C2 c1(OC)ccc(C(N2CCOC(C(C)NC(=O)CCc3cscn3)C2)=O)c(Cl)c1 c1(C(=O)NCCCNC(c2c(COC)scc2)=O)ccc(F)c(F)c1F N1(C(c2c[nH]c(=NC)o2)=O)CCC2(CC1)C(OC)CC2NC(c1ccc(C)o1)=O c1(C(N2C(CNC(CCOC(C)=O)=O)CCC2)=O)cc(C(C)C)nn1C c1(CNC(C2C(C)(C(C)C)C2)=O)ccc(C(=O)NCC=CCl)cn1 C1(CCOC)CN(C(=O)Cc2sccc2C)CCN1C(=O)C(=Cc1c[nH]cn1)F Cc1sc(C(=O)NC(C)CN(C)C(C2(O)CC(CF)C2)=O)cc1[N+](=O)[O-] O=C(C1Cc2ccc(F)cc21)NC1CCN(CCCN2CCOCC2)C1 C(=O)(C(C(C)C)NC(=O)Cc1ccc[nH]1)NCC(C(=O)OC)OC C1(NC(=O)NC(C2CCCCO2)CC)CCC(OCC2CC2)CC1 C(CNC(=O)CN1CCSCC1)(C(C)(C)C)NC(C(CC)Oc1ccccc1)=O c1(NC)cc(Cl)ccc1C(=O)NCCC(C(C)C)NC(c1cc[nH]n1)=O C1(NC(C=C2CCN(C)CC2)=O)CC2CC1CN(C(C1CCC(O)CN1C)=O)C2 C(=O)(CC(C)CN(C)C)NC1(C)CC(NC(CC2CC(OCC)C2)=O)C1 c1(CCN=C(NC2CCC(C#N)C2)NC2CCC2)ccc2c(c1)OCCO2 CCCC(CC)C(=O)NC1CCC(F)(CNC(=O)Cn2ccc(C3CC3)n2)C1 C(=O)(C(C)C(O)C(C)C)NC(C(C)C)C(=O)OCC(=O)NCCC1CCCC1 Cc1ccc(C2CC2C(=O)NCC2(NC(=O)COC(C)C)COC2)cc1Br C1(NC(c2cccnn2)=O)CCN(C(C2(O)CCSC2)=O)CC1CO N1(C(=O)Cc2cnccn2)CCC12CCCN(C(C1CC(O)C1)=O)C2 C1(C(=O)NCC2CN(Cc3cc(C4CCC4)no3)C2)CCc2c[nH]nc2C1 c1(C(=O)NCC=CCNC(CCc2cc(C(C)=O)c(C)o2)=O)cc(F)cc(Cl)c1 C(=O)(C1=NOC(CNC(C2CCCSC2)=O)C1)N1CC(CCC#C)C1 C1(C(N(C)Cc2cnn(-c3ccccc3)n2)=O)CCCCC1NC(N)=O C1(NC(c2c(CC)onc2)=O)CC2CC(NC(=O)CCCc3csc(C)n3)CC12 c1(C(N2C(CN(C(C(C)NC(CC)=O)=O)C)COCC2)=O)cc(F)c(F)cc1Cl C(c1ccn(C)c1)=CC(=O)N(CCN(C(c1c(SC)ccs1)=O)C)C C1(N(C)Cc2cc(Br)c[nH]c2=N)CCN2CCCC2C1 N1(C(c2n(C)ncn2)=O)CCC2(CC(NC(c3cnn(C(F)F)c3)=O)C2)C1 CCCCC(C(=O)N1CCCC1(C)CNC(=O)C(C#N)C1CC1)NC(N)=O C=Cc1ccc(C(N2CCOC(C(=O)NCCOCC3CCC3)C2)=O)cc1 S(=O)(=O)(c1cnccc1N1CCCC2(CCOC2)C1)N1CCCC(C#N)C1 N1(C(C2C(CC)C2)=O)CC2CCCC(C1)N2c1ncc2c(n1)COC2 C1(NC(=O)CN2CCN(CCc3ccsc3)CC2)CCc2c[nH]nc2C1 c1(C(=O)NC(CN(C(C2CCC(=O)N(C)C2)=O)CC)C)cnc2c(C)nsc2c1 CC1CCN(c2nccnc2F)CC1NC(=O)C(Cc1ccsc1)NC=O c1(C(=O)NCCc2ccn(CC)n2)cc(F)c(F)cc1Cl Cc1coc2c(C(=O)NC3CC(C)CN(C(=O)C(O)C(F)(F)F)C3)cccc12 Cc1ccc(C(N2CCC3CC23C(=O)NCC2CCC3(CC2)CC3)=O)c(O)n1 c1(C(=O)NC(C)C(C)NC(c2cnc(-c3cnn(C)c3)s2)=O)ccccc1Cl N1(C(=O)CN2CCOCC2=O)CC2CCN(C(c3ccc4nsnc4c3)=O)C2C1 C1(CCC(=O)Nc2cn(CC)nc2)CCCN(C(=O)CCCCOC)C1 c1(C(N2CC(O)(C(C)NC(C(CCCC)O)=O)C2)=O)cc(OC)c(Cl)cc1Cl n1(CC)nc(C(N2CCC(C(=O)N=c3[nH]nc(C)n3C)(C)C2)=O)c2ccccc12 C(C(C)(O)COC)CNC(C(=O)NCCC(C)OCCC)=O c1(NC(C2CC(NC(c3ccnc(F)c3Cl)=O)C2)=O)c(Cl)cnnc1Cl CS(=O)(=O)c1cc(C(N2CC(NC(c3cscn3)=O)C3CC23)=O)cc(N)c1 N1(C(C=C(C)C)=O)CC2COCC2(C(=O)NCc2c(C)cccc2C)C1 C(=O)(C(O)CC(C)(C)C)NCC(CC)NC(C(C)SCCCC)=O N1(C(c2scc(C#N)c2)=O)CCOC2(CCN(C(c3ncncc3Cl)=O)CC2)C1 c1(C(=O)NC2CN(C(c3cc(F)cc(Cl)c3)=O)CC2F)csc2c1CCCC2 C1(C(N(C2CCCOC2)CC)=O)CN(C(=O)C=C=C(C)C)CC1C C12(CNC(=O)C=Cc3ccoc3)CC1CN(C(=O)CCOc1ccccc1F)C2 c1(C(=O)NC(C(C)NC(c2cnc(SC)s2)=O)C)cc2ncccc2o1 c1(OC)cc(C(=O)NC2(C)CCN(C(=O)C(F)C3CC3)CC2)c2ccccc2n1 CC1CN(CC(=O)NCC2CCCO2)CCN1c1cc(N(C)C)ncn1 N1(C(=O)Cc2ccsc2)CCCC2(CCN(C(C3CCCN4CCCC34)=O)C2)C1 C12CCN(C1)C(=O)OC2.S(=O)(=O)(CCOC(C)(C)C)NC(=O)OC(C)(C)C N1(C(C)=O)CCCCC(CCC(=O)NCc2cn(C3CC3)cn2)C1 c1(OC)cc(C(=O)N(C2CN(C(c3cccc(F)c3Cl)=O)CC2O)C)cnc1O c1(C(N2CC(F)CC(NC(=O)CCC3OCCO3)C2)=O)cccc2cnccc12 c1(NC(C2CCC(NC(C3(COC)CC3)=O)C2)=O)cnc(C)c(Br)c1C S(=O)(=O)(c1cccc(F)c1F)NC(CNCCC(N)=O)=O C1(C(=O)NC(c2ccc(C)nc2)C)CCOCCN1C(c1nnccc1C)=O c1(C(=O)NCC(C2CC2)NC(CCCOC(C)=O)=O)nc2cccnc2s1 c1(OC)ccc(S(=O)(=O)N2CC3CN(C(c4cc(C#N)cc(C)c4)=O)C3C2)cn1 C1(C(=O)NC(C2CC2(F)F)(C)C)CCCN(C(=O)CC2CCOC2=O)CC1 S(=O)(=O)(c1ccc(NCc2cnsc2)c(C#N)c1)N(CC(C)C)C1CCC1 N1(C(C2(CCNC(C=CC(CC)C)=O)CC2)=O)CCC2(CCCO2)C1 Cc1cc(CNC(=O)CC(C)(C)C)c2c(c1)CCC2.C1CCCCCOC(=O)C1 c1(CC)ccc(C)c(C(N2CCN(C(=O)Cc3c(C)noc3Cl)C3CC23)=O)c1 CCC(C)CC(=O)NC1C2CC1N(C(=O)C(c1cscn1)N(C)C)C2 C1(NC(C=C(C)CCc2ccccc2)=O)CCCC1NC(c1sccc1CO)=O c1(CC(N2CCC(CCNC(CCC=C)=O)CC2)=O)ccc2c(c1)CCN2C c1(C(N(C2CCN(Cc3sccc3Cl)C2)CCC)=O)ccc(N2CCCC2)nn1 C1(CC(=O)NC2(CN(C(c3cc(C)sc3)=O)C)CC2)CC2(C1)CC1(CCC1)C2 CC1=C(C(=O)NC2CC(N(C(=O)CCC(F)(F)C(F)F)C)C2)S(=O)(=O)CCO1 C12(CC(=O)N(C3CC(NC(c4cc(O)nc(Cl)c4)=O)C3)C)CCC(CC1)OC2 CC(C)C(CNC(=O)Cc1nccn1C)NC(c1ccoc1C(F)(F)F)=O N1(C(C(CN(C)C)O)=O)CC(F)(F)CC1CNC(c1csc(-c2nc[nH]n2)n1)=O c1(-c2nc(CCC(N3CCC(F)(F)C(CO)C3)=O)on2)coc2cc(O)ccc12 c1(C(N2CCC(NC(Cc3c(C)noc3)=O)(CO)C2)=O)cc(=O)n2ccsc2n1 c1(C(=O)NC2CC3CC(NC(C4CN(C)C(=O)C4)=O)C3C2)cn2ncccc2n1 C1(NC(C(=O)NCC)=O)CCC(NC(=O)C(F)CC2CCOCC2)CC1 N1(C(C2(c3ccc(Cl)c(F)c3)CC2)=O)CCC2(CC1)OCc1ccccc12 Cc1cc(F)c(C(N2CCOC3(CCC3)C2)C(=O)NC2CCOC2)nc1Br c1(C(=O)NCC(C)N(C(C(C(=O)OC)C)=O)C)c(C)nn(-c2ccccc2)c1C N1(C(CC)C)CC(C(N2CCN(CCN(C)Cc3ccccc3)CC2)=O)CC1=O CCC(C)CC(C(=O)NCC(C)COC)NC(=O)CCN1CCCCC1 C(C)(C)(C(=O)N1CCC1CNC(C1(Cc2cccnc2)CCC1)=O)OC(C)C C1(C(N2CC(NC(C(N)=O)=O)C3(C2)CCC3)=O)Cc2ccc(F)cc2C(=O)O1 N1(C(C(C)N(C)C)=O)CCC(C(=O)C(C)(C)C)CC1 CC1(C)C(C(N2C3C=CC(C3)C2CO)=O)CCS1(=O)=O CC1CCC(C)(C(N2CC(C)(NC(=O)CC(C)(F)F)C2)=O)C1 C1(CC=C)(NC(=O)CCCCCC)CC2CCC(C1)N2C(c1n[nH]c(=N)[nH]1)=O c1(C(N2CCN(C(=O)NCCCCc3cc(C)no3)CC2)=O)cccc(F)c1F C(C(CC(=O)N1CC(O)(n2cnnn2)C1)OC)NC(C(CC)n1ccnc1)=O N#CC1(C(=O)NC2CCCCC2CNC(=O)CC(F)(F)F)CC2CCC1CC2 CC1(C(=O)NC2CC(C(=O)Nc3nnco3)C2)CCOCC1 C1(NC(c2cc3c([nH]2)CCCC3)=O)C2CC3CN(C(=O)C4=COCC4)C1C3C2 C1(CNC(C(C)NC(CC)=O)=O)CC2COCC2N1C(c1ccc(N)cc1Cl)=O CCC(C)(CNC(=O)COC)NC(c1cnn(CCC(F)(F)F)c1)=O C1(CCC#C)CCCN(c2cc(NC3CCOC3)ncn2)C1 C1(NC(=O)Nn2ccc(C(CC)CC)n2)CCCN(CCCO)C1 c1(CC(N2C(CN(C(c3oc(C)cc3C)=O)CC)CCC2)=O)ccc(F)cc1 Cn1cc(CC(C(=O)O)NC2CCN(C3CCSC3)CC2)c2ccccc12 Cc1cc(C(=O)N(CC(C)(C)NC(c2csc([N+](=O)[O-])c2)=O)C)c2nccn2c1 c1(CCC)c(C(=O)NCCCN(CCC)C(C2CC3(CCC3)C2)=O)nnn1C C1(C)(C(N(C(CNC(c2c(CC)ccs2)=O)C)C)=O)CCCCNC1=O N1(C(C(CCCC)O)=O)CC2CCC(C1)N2C(C1(C)CC2CCC(C1)S2)=O N1(C(C(=O)NCC(F)(F)F)=O)CCC(NC(c2ccc(C3CC3)s2)=O)C(C)(C)C1 C1(CC(=O)NCC(c2ccc(C(F)(F)F)cc2)OC)CCC2(CCC2)OC1 Cc1ccc(I)c(C)c1NC(C1CCC2(CN(C(=O)Cn3cccn3)C2)O1)=O CN1CCN(C(=O)C(C2CCCCCCC2)O)CC(O)C1 C(=O)(C(C)CCC(C)(C)C)NCC(CC)N(C)C(c1ncn(CC)n1)=O CC1CN(C(=O)CSc2cccc[n+]2[O-])CC1CNC(=O)C=CC1CCOCC1 c1(CCC)[nH]nc(C(=O)NC(C2CCN(C(=O)C3=CCCC3)CC2)C)c1[N+](=O)[O-] CC1(C)C(NC(=O)C=Cc2ccncc2)CCN1c1ncc(C(F)F)cn1 N1(C(=O)C2=NOCC2)C2CCC1(c1nn[nH]n1)CC2 C1(C(=O)NCc2ccccc2)CC(F)CN(C(c2cc(Cl)ccc2F)=O)C1 c1(C(=O)NCC)ncc([N+](=O)[O-])n1C.C12CC(C1)C(=O)NCCN(CC)C2=O c1(CC(=O)N(C2CN(C(CC3ON=C(CC)C3)=O)C2)C)cc(OC)ccc1OC c1(C(N2CCCC(NC(CC(C)C)=O)C2C)=O)coc(C#Cc2ccccc2)c1 C(=O)(C1CCCn2nccc21)NC12CCCN(C(CC3(C)CCCO3)=O)CC1C2 N1(c2cc(C)c(CC3CC(C)CC(C)(C)C3)cn2)CC(C)(C)c2ccccc21 N1(C(CCc2cnc(C)o2)=O)CC=CC(C(=O)N(CC(C)C(C)C)C)C1 C(=O)(C#CC(C)(C)CNC(C1(COC)C=CCC1)=O)N(CC(CC)(C)OC)C c1(C(N2CCCC2CC2CC2)=O)cc(-c2ccccc2)nc2c(Cl)cnn12 C12(OC)CCC(C(=O)NC(C)CC3CCN(C(=O)C4CC4)CC3)(CC1)C2 c1(SC(C(=O)NCCC(CNC(CNC(CC)=O)=O)O)C)ccc(C)c(C)c1 C1(C(N2CCC(O)(CN(C(CC(C)C3CC3)=O)C)CC2)=O)OC(C)(C)OC1(C)C Cc1noc(C(CO)NC(=O)CCCNC(=O)Nc2cccnc2)n1 CC1=C(C(=O)NC2C3CCN(C(C4C=CCCC4)=O)C23)SCCO1 C1(C)(C(=O)NCC2N(C(CN(CC(=O)NC(C)C)C)=O)CCC2)CCN(C)CC1 C1(C(=O)NCC=CCCC)(COC)CC2CC2C1 c1(C(NNC(=O)C=Cc2ccccc2F)=O)ccc2c(c1)OCCNC2=O CCC(C)C(O)CC(=O)NC1CCOC1C(=O)NC(C)C(=O)N(C)OC c1(C(N(CCCN(C(=O)Cn2[nH]cnc2=N)C)C)=O)nn(C)cc1Cl C12(CNC(C3C=CC=CC=C3)=O)CC1CN(C(=O)Cc1ccc(Cl)cc1)C2 C(C1c2ccsc2CCN1C(=O)CSc1cn[nH]c1)NC(=O)Cn1nccn1 N1(C=O)CCN(C(c2ccc(COC)o2)=O)CC1.C(=O)(CC(C1CC1)SC)NCC N1(C(Cc2ccc(C)o2)=O)CCC(O)(CNC(=O)CCOCC2CC2)CC1 c1(NC(CN2CC(C)(Nc3ncccc3C(N)=O)C2)=O)cc(CO)cc(F)c1 C1(C(=O)NCC2CC(C(=O)NCCOCC(=O)OC)C2)CC2C=CC1O2 c1(SCCC(=O)NC2(CCNC(C3C(C)(CC)C3)=O)CCC2)nnnn1C c1(C(C)(C)C)ncc(C(=O)NCC(C2CCCC2)NC(c2csc(F)c2)=O)o1 c1(CC)ccc(C(=O)NCC2CCCC2NC(=O)CC(C)(F)F)c(F)c1 C(=O)(C(F)(CC)C(=O)OC)NCC1CC(F)(CNC(CC2ON=C(CC)C2)=O)C1 N1(C(=O)NCc2ccn(-c3ccc(F)cc3)n2)CCC12CCC(CO)CC2 C=CC1(c2nc(-c3cccc(CC(C)C)c3)no2)CCCCC1 C1(CNC(C2C(C)CCC2)=O)COC(C)(C)CN1C(c1cnn2cnnc2c1)=O CC1CC(C(=O)NCC(C)(C2CC2)NC(=O)CNC(N2CCCC2)=O)=NO1 N1(C(CCCC(CC)C)=O)CC2CCCCC2(NC(=O)C=C2CCC2)C1 N1(C(c2c(C)ccc(C)c2)=O)CC(C)CN(C(c2ncc(Cl)cc2Cl)=O)CC1C C(CO)(C(C)N=c1ncnc(N(C)C)[nH]1)c1c(OC)cccc1 N1(C(c2cn(C)nc2CC(C)(C)C)=O)CC2(CCCC2N)C1 c1(NS(CC)(=O)=O)cccc(C(=O)NC2C3CC2N(C(c2nccn2C)=O)C3)c1 C(=O)(C#CC1CCCCC1)N1CCC(N(C(=O)CN(CC)CC)CCC)CC1 N1(C(c2ccc(C)s2)=O)CCN(C(C2CC(=O)N(c3cn[nH]c3)C2)=O)CCC1C N1(C(c2n(CCC)ccc2)=O)CCCCCC1C(N1CC(CO)C(C)(C)C1)=O C1(C(N(CC(C)SC)C)=O)CC(N=[N+]=[N-])CN1C(=O)Cc1csnc1C c1(OC)cc(C(=O)NCCN(CC(C)O)C(C2CC2C)=O)cc2c1OCCO2 c1(C(=O)NCC(CO)NC(C(c2scc(C)n2)(F)F)=O)cnc2cccnc2c1 C(=O)(C1CCCc2nnn(C)c21)N1CCC(N(C)C(C2CC(F)C(=O)N2)=O)CC1 c1(OC)ccc([N+](=O)[O-])cc1S(=O)(=O)NNC(=O)C(N)COC.c12cccc(c1)O2 N1(C(C2C(C(C)C)OCC2)=O)CC2CC1C2C(=O)NCC1CCCCN1C CC1Oc2ccc(C(N3CC(NC(=O)Cc4c(F)cccc4Cl)C3)=O)cc2C1C C1(CN(C(C(C)CN(C)C)=O)C)CCN(C(C2(C#N)CC2(C)C)=O)CC1 c1(C(N2CC(C)(CNC(C3N(C)CCC3)=O)C2)=O)ccc2ocnc2c1 CCC(C)C(C(=O)NCC1CC(NC(c2cn(CCN(C)C)nn2)=O)C1)OC Cc1ccc2c(c1)CCC2NC(=O)NNc1ccccc1F C=CCC(C(=O)NCC(C1CC1)NC(=O)CCN(C)CC)C(C)C c1(N(C2CN(C(C34CC(C)(CO3)C4)=O)C2)C)cc(C(N)=O)ccc1[N+](=O)[O-] c1(C(=O)NC(c2nc(C)cs2)CC)ccc(Sc2cncc(F)c2)cc1 CC1(C(=O)NCC(C)(O)C(F)(F)F)CCN(C(C2CC2(C)C)=O)CC1 C1(C(N2CCC(N(C(C3C(CC)OCCC3)=O)C)CC2)=O)CN2CCC1CC2 C12(C(N3C(CNC(c4ccc5c(c4)CC5)=O)CCCC3)=O)COC(CCO1)C2 C1(NC(=O)Cc2cnsc2)CC2CCC(C1)N2C(c1cc(C2CC2)cnc1Cl)=O C1(NC(=O)CCc2ccc(F)cc2)CC(O)CN(C(c2[nH]cc3c2CCC3)=O)C1 C1(NC(c2c(CC)nco2)=O)CN(C(c2ccnc(OC)n2)=O)C2(CCOC2)C1 c1(C(N(CCNC(C2(S(C)(=O)=O)CC2)=O)CC)=O)ccnc2ncc(C)cc12 c1(CC)cc([N+](=O)[O-])ccc1N1CCN(CCNC(=O)CC2CCC(C)C2)CC1 Cc1[nH]nc2ncc(C(=O)NC3CCC(C)N(C(=O)CCC4CC4(F)F)C3)cc12 c1(CCNC(C(C)N(C(CSCCC)=O)CCC)=O)c(C)cc(C)cc1Cl c1(C(=O)NCCC2(NC(C3CC3Cl)=O)CCOCC2)c[nH]cc(Cl)c1=O c1(C(=O)NC2CCN(C(c3ccc4c(c3)CCN4)=O)C2)ccc2c(c1)CCCS2 C(=O)(C(C(C)(C)C)OCC)N1CC2C(NC(c3cn(CC=C)nc3)=O)(C2)C1 C1(N(C(c2[nH]cc(CC(C)C)c2)=O)C)CCCCN(C(C2CC(=O)C2)=O)C1 C(CN=c1[nH]c(=NC2CCS(=O)(=O)C2C)[nH]c2c1SCC2)(c1ccccc1)OC C1(NC(CONC(C)C)=O)CCC(C)N(C(c2cn(CC(=O)CCC)nn2)=O)C1 N1(CC)CC(C(=O)NC2CCCC(NC(=O)CCc3cnc[nH]3)C2)CCC1=O N1(C(C(C)(C)SC)=O)Cc2[nH]nc(C(=O)NCc3cc(C)co3)c2C1 Cc1csc2ncnc(N(CCC3CCCNC3)Cc3c(Cl)ccc(Cl)c3F)c12 Cc1ccn2cc(C(=O)NC3CN(C(c4ccc(F)cc4Cl)=O)CC3C)nc2c1 CC(C)(CCC(=O)NCC1CC(=C2CC2)C1)NC(=O)Cc1ncccc1F N1(C(c2c(C)ncc(Cl)c2)=O)CCN(C(=O)Cc2ccns2)C(C)C1C C1(CCN(C)C(c2cscc2C(N)=O)=O)CCN(C(=O)C2=NOCC2)CC1 C1(NC(c2cc(Cl)c(F)c(Cl)c2)=O)CN(C(=O)CC2CCOCC2)CCC1(F)F N1(C(C(CCC)OC)=O)CCN(C(c2ccn(C)n2)=O)CC1C C=C=C(C)CC(=O)NC(C)(C)CNC(C1(NC(=O)OC(C)(C)C)CC(O)C1)=O C1(NC(CC)=O)C=CCC(C(N2CCC(C(C)CO)CC2)=O)C1 N1(C(c2cccc(C)c2N)=O)CCC2(C1)CN(C(C1(C)CC1(Cl)Cl)=O)CCO2 C(=O)(C(C)(F)C(=O)NCCC1CCN(C(c2csc(-c3cn[nH]c3)n2)=O)C1)OC CC(C(=O)Nc1cccnc1CNC(=O)C(C)NS(C)(=O)=O)S(C)(=O)=O c1(C(=O)NC2CCC(CNC(CC3CC(CC)C3)=O)C2)ccc(C)cn1 C1(N(C(c2c(CC)onc2)=O)C)CN(C(=O)Cn2cc(C)cn2)CCC1C c1(C(=O)NC2CC3CN(C(Cc4ncc(CC)[nH]4)=O)CC32)c[nH]c2nccc-2c1 C(CCCCCN(C)C(c1ccco1)=O)NC(C1C=C(C)CS1)=O C(C)(N=c1[nH]c(=N)[nH]c(=NC(C)CCC2CCCC2)[nH]1)c1cccc(SC)c1 C12(C(=O)NCCC3N(C(c4n(C)ccn4)=O)CCCC3)CCOC1CC(=O)NC2 N1(C(C2C(OCC)C2)=O)CC(N=c2[nH]c(Cl)ncc2[N+](=O)[O-])CC1C N1(C(C2(OC)CCCOC2)=O)CC(C(=O)NCC2CC2C(C)C)CC(C)C1 N1(Cc2c(OC)nc(Cl)cc2)CCC2(CCC(F)(F)CC2)C1 N1(C(C(CCCC)C)=O)CC2CCN(C(=O)CNS(=O)(=O)CC)CC2C1 N1(C(C(CN(C)C)N(C)C)=O)CC2(C)CC1(C(=O)NCCC1COCCO1)C2 C=CC1(C(N2CC3C(N(C)C(c4cccc(C)c4Cl)=O)C3C2)=O)CCCCC1 n12c(nc3ccccc13)-c1ccc(cc1)C(=O)N2.S(=O)(=O)(c1cccs1)NCC C(C(C(=O)NCc1cccnc1C)C(C)C)NC(C(C=C)(C)O)=O c1(C(C(=O)NC2C(CNC(c3cn(CCOC)nc3)=O)C2)F)ccc(F)cc1 CC(C(C)C)=CC(=O)NC(C)(C)CN(C(=O)CCC1CC1(C)C)C c1(C(=O)NCC2(C)N(C(C3N(CC)CCOC3)=O)CCC2)nc(C)ccc1OC c1(C(=O)NC(C(=O)N(C)CC2(O)CCC2)Cc2cn[nH]c2)ccc2c[nH]nc2c1 Cc1cnc(Nc2ccc(C)c(C(N3CC(N(C)C)C3)=O)c2)nc1C n1(C(=O)NCC(c2ccccc2F)NC(=O)CN2CCSCC2)cccnc1=O N1(C(c2cccc(C)c2)C(=O)Nc2ccccc2)CCS(=N)(=O)CCCC1 Cc1ncc(Cl)c(C(N2CCN(C(=O)CN(C(=O)C(C)CC(F)F)C)CC2)=O)n1 Cc1sc(N)c(C(N2CC(NC(=O)C(C)CC3CC3)CC(C)C2)=O)c1C c1(CC(=O)NC2(CCNC(=O)CCc3cnc[nH]3)CCC2)ccc([N+](=O)[O-])cc1 CC1(C)COC(=O)C1NC(=O)CCCn1cc(CC2CCCOC2)nn1 c1(C(=O)NC(C(C)NC(CSCc2nc(C)sc2)=O)CO)cncc(C#N)c1 c1(OCCCCCC)ccccc1C(N1CC(OCC)C(NC(=O)COC)C1)=O C=C(C)CCC(C)NC(C1CCC(NC(=O)CC2CC(=O)C2)C1)=O Cc1ccc(C)c(C(=O)NC2COCCN(C(=O)C(c3ccc(O)cc3)=O)C2)n1 N1(Cc2ccc(N(C)C)o2)CC(C(=O)NCc2c(F)cccc2I)CC(F)(F)C1 Cc1cccc(C(=O)NC2CC(CCNC(c3cn(C(C)C)nc3C)=O)C2)c1C c1(N2CCCC(NC(C3C(C)OC(C)C3C)=O)C2C)cc(C#N)ccc1[N+](=O)[O-] N1(C(c2c(C)nc(CC)o2)=O)C2CC=C(C(=O)NCC3(SCC)CC3)C1CC2 N1(C(C2CCCC(F)C2)=O)Cc2ccccc2C(CNC(C2CC(O)C2)=O)C1 Cc1cccc(CC(=O)NC2CCCC(NC(c3cc(C)oc3C)=O)C2)c1 c1(NC(C(C)(C)C)=O)ccc(N2CCN(C(c3ccnc(F)c3)=O)CC2)nc1 N1(C(COCC(=O)NC)=O)CC2CCC2(CCNC(c2cnc(C)cc2Cl)=O)C1 c1(CN=C(NC(COC)C)NCC(C)(C)C(C)(F)F)noc2c1CCCC2 CCCC(CNC(C1CC1[N+](=O)[O-])=O)C(=O)NCC(=O)NOCC Cc1ccnc(C(=O)NCC2CCN(C(C3CC4C=CC3CC4)=O)CC2)c1O C(=O)(C1=C(C)S(=O)(=O)CC1)NC1(C2N(C(c3nc(COC)[nH]n3)=O)CCC2)CC1 N1(C(c2cc(Cl)cc(Cl)c2)C(=O)NCCCCCC)CC2(C)CCC2(C)C1 N1(C(c2ccc(CC)cn2)=O)C2CCC1C(NC(=O)CC1(CC)CCC1)C2 C#CCCCCC(=O)NC1CCCC1(C)NC(=O)C(c1ccccc1)F Cc1c(C(N2CCN(C(c3ncn(C)n3)=O)CC2C)=O)ccc2c1CCC2 N1(C(c2[nH]cc(CC)c2)=O)CCCC(CNC(c2ccn(C3CC3)c2C)=O)CC1 c1(OC)ccc(C=CC(=O)NCCC(C)NC(C2(C(C)C)CNC(=O)C2)=O)nc1 N1(C(CCC(C(C)C)NC(=O)CCC2CC2C)=O)CCCC12CCOCC2 c1(SC)ccsc1SC.CCS(=O)(=O)NCCC(=O)NCC1CCN1C(C1CC1)=O c1(C(=O)NCCN(CCOC)Cc2cc(C)[nH]n2)ccc(C(N)=O)o1 C1(CNC)CCCCC1CNc1nnc(CSc2ccccc2-c2cccs2)o1 C1(CNC(C(CC)NC(N)=O)=O)CCN(C(=O)CC2CCC(=O)N2)C1(C)C C1(NC(C=CC=CCC)=O)C=CCN(C(=O)C=CC(=O)Oc2ccc(OC)cc2)C1 C1(C(N2CCC(C)N(C(C3CC4CCC3O4)=O)CC2)=O)CCc2ccccc2C1 C(=O)(N=c1[nH]c(Cl)ncc1O)C1CCCN(C(c2c(C)nc(Cl)cc2Cl)=O)CC1 N1(C(=O)COCC2CCOC2)CCC2(CCN(C(c3cc4sccc4[nH]3)=O)C2)C1 C1(C(N2CC(OC)C(NC(=O)CN(C)C(C)=O)C2)=O)CNC(=O)CC12CCC2 c1(CCNCc2c(OC)cccc2)c(Br)cncc1Br C1(OC)CN2CCCC2(C(N2CCOC(C(C)NC(C3CC3(C)C)=O)C2)=O)C1 C1(C(=O)NC2CC3(CC(NC(C(CC)(C)O)=O)C3)C2)CC(C)(C)SC(C)(C)C1 Cc1noc(N)c1C(=O)NCCCOCCNC(c1ccc(C(C)C)o1)=O c1(C(N2C(C(C)(C)NC(c3cnns3)=O)CCC2)=O)cc2cc(Cl)ccn2n1 C1(C(=O)NCC(CC(C)C)NC(CNC(CCC)=O)=O)CCc2nc(O)[nH]c2C1 N1(C(C2(CC=C)CCC2)=O)CC2CCC2(CCNC(C2(C)CSC2)=O)C1 C1(CNC(C2CC3CCC2O3)=O)CN(C(c2ncc(C(F)(F)F)s2)=O)CCO1 C1(NC(C(C=C)CC)=O)CCN(C(=O)CC2CCCC(=O)C2)CC(C)(C)C1 CC(CNC(C1CN(C(N)=O)C1)=O)C(=O)N(C)CC1CCC1 CC1CCN(CCC(=O)NC2(C)CCN(C(=O)C(C(C)C)NC=O)C2)CC1 c1(C(=O)NC(C2CN(C(=O)C=Cc3ncc[nH]3)C2)C)ccc(-c2ccsc2)cc1 CC1(C)CCOC1CC(=O)NCC1CCCN1C(c1cnnn1C1CC1)=O C(=O)(CC1=NN(C)C(=O)C1)NC1C(C(=O)NC2C(CCOC)C2)CCC1 c1(-c2ccc(N3CCN(C(=O)NC45COCC(C4)C5)CC3)s2)cc(F)ccc1F c1(CNC(c2n(C)nc(C3CCCOC3)c2)=O)cc(Br)ccc1F c1(CC)cc(C(=O)NCc2ccc(CN(C(C)=O)CC3CCC3)cc2)n(C)n1 c1(C(=O)OC)nc(N2CCC(OCc3nc(C)cs3)C2)ccc1C c1(N(C)Cc2ccncc2)nnc(-c2ccc(Cl)nc2)n1CCC1CC1 N1(C(C(N2CCOCC2=O)C)=O)CC2CC(C1)CN(C(C1CCC(=O)N1)=O)C2 CC(C(=O)NCC(c1ccccc1)CNC(=O)CCC(=O)c1ccc[nH]1)C(F)F N1(C(CCSCC)=O)CC(NC(=O)Cn2cnc(C(N)=O)n2)C(C)(C)C1 C1(C(=O)OCCCCCSC)COCC(C)N1C(=O)OC(C)(C)C N1(C(CC2CCC(C)CO2)=O)CC(C)(C)CC1CNC(=O)CCC1CCCOC1 N1(C(C(CC)C(C)O)=O)CCCC(C2CCN(C(C3CCC(F)CC3)=O)C2)C1 c1(C(=O)Nc2ccc(NC(c3ccc(F)cc3F)=O)cn2)c(Cl)cccc1Br N1(C(c2c(SC)scc2)=O)CC(NC(=O)Cc2ccon2)C(O)C1 Nc1ccc(Cl)cc1C(=O)NC1(c2cn(Cc3nccs3)nn2)CCC1 c1(C(=O)NCC2C(NC(COCCOCC)=O)C2)cc(OC)c2occc2c1 CC1CCOCC1C(N1CCCC1(C)C(=O)N(C)Cc1cscn1)=O c1(COC)ccc(C(=O)NC2CCCC2CNC(c2cnn(SC)c2)=O)cc1F N1(C(C2C(C)(COC)C2)=O)CC2CC1CCC2NC(C1CN2CCN1CC2)=O c1(C(N2CC(NC(=O)Cc3csc(Cl)n3)C2)=O)cccc2c3c([nH]c12)CCCC3 C1(CC(=O)NC(C2CN(C(c3cc(C#N)on3)=O)CCO2)C)CCC(=O)NC1 c1(SC)nc2ncnc(NCCOCCNC(C3CC4C=CC3C4)=O)c2s1 Cn1nncc1CC(=O)NCC1COCC1NC(c1scnc1Cl)=O c1(CC(N2CCCC(CC(=O)Nc3cncnc3Cl)C2)=O)ccc(O)c(O)c1 c1(C(=O)NC(C2CCN(C(=O)CS(=O)(=O)N(C)C)C2)C)csc2ncnc(O)c12 N1(C(=O)CCc2cccc(O)n2)CC2=C(C1)CN(C(C13CSCC1C3)=O)C2 C=CCC(F)(F)C(=O)NCC1CCCC1NC(c1sccc1-n1cnnn1)=O c1(N(CCNC(C2CCN(C)C(=O)C2)=O)CC)nnc2c(c1C(=O)OC)CCC2 C(C1=CCN(C(=O)CC2CCS(=O)(=O)CC2)CC1)NC(C1CCCS1)=O c1(C(=O)NCC(C(C)C)NC(CN2CCCC(CC)C2)=O)ccc2cnoc2c1 c1(C(=O)NCCCOCCNC(C(C2CCCOC2)OC)=O)nc(O)c(C)s1 CCC(C)CCC(=O)N(C1CN(C(c2cc(Br)oc2C)=O)CC1(C)C)C c1(C2C(C(N3CCC(NC(C4CC(O)C4)=O)CC3)=O)C2)ccc2c(c1)OCO2 N1(C(C2CCCC(=O)N2)=O)CCC2CN(C(c3ccccc3)=O)CC12 Cc1cnn(C)c1C(=O)N(C)CC1CCCN1C(C1CCCC2CC12)=O c1(N2C3CN(C(=O)Cn4cc(C5CC5)nn4)C(C3)C2)nc2ccc(Br)cc2s1 C1(C(=O)NC2CCCCC2NC(=O)COCc2nccn2C)(OC)CS(=O)(=O)C1 C1(C(N2CCCC(C(=O)NC3CC(C)(C(N)=O)C3)C2)=O)CCOC(=O)CC1 C=CCC(C(=O)N1CCCC1CC(=O)NCCc1cnn[nH]1)OC Cn1c(C(=O)NCC(C)(C)NC(C23CC(C(C)(C)C)(C2)C3)=O)cnc1S c1(C(=O)NCCC2(NC(C=CC(=O)OCC)=O)CCC2)scc2c1OCCO2 n1(CC)nc(C(N2CCC(C(C)(C)NC(=O)CC3CCCCC3O)C2)=O)cc1O C1(C(=O)NCCNC(CC)=O)CCCCC1(C)Sc1ccccc1 Nc1cncc(C(=O)NCC(C2CCCCC2)NC(c2csnc2Br)=O)c1 c1(CC(N2C(CCNC(C=NOC)=O)COCC2)=O)cn2ccccc2n1 CC(C)C(O)C(C)C(=O)NCC1(F)CCCN(C(c2ccc(CO)nc2)=O)C1 CCCC(C(=O)N(CCCCNC(=O)Cc1ccnn1C1CCC1)C)N(C)C c1(OC)ccnc(N(C(c2cc(OC(C)C)ccn2)=O)C(C2CCNCC2)C)n1 N1(C(C2(COC)CCCO2)=O)CC2CC(NC(c3ccc(NC(C)C)s3)=O)C2C1 N1(C(COCC)=O)CC2COCCC2(NC(c2nnn(C3CCOC3)c2C)=O)C1 C1(NC(C2C(OC)C2)=O)(CO)CCN(C(c2ncc[nH]c2=O)=O)C1 C1(NC(c2c(CCNC(C(C)OC(C)=O)=O)n[nH]c2)=O)CCCCCC1(C)C CN1CCC(O)(CNC(=O)CCOCCNC(=O)CC2CCC(O)C2)C1 c1(C(N(C2CCN(C(=O)C(CC)NC(N)=O)C2)CCC)=O)scc(C)c1C C(=O)(CC(C)C(F)(F)F)NCC1(C)CCN(C(CC(C(C)C)O)=O)CC1 CN1CCOc2cc(CN3CC(NC(c4cc(F)cc(F)c4F)=O)C3)ccc21 Cc1nc(C(C)C)sc1C(N1CCOC(CCNC(=O)CC2COCC2O)C1)=O C(=O)(CC(C(=C)C)OCC)NC(C(=O)N(C1C(C=C)COC1)C1CC1)C N1(C(CCC(CC)OC)=O)CC2CC1CCN2C(c1cnn(CC)c1)=O c1(C(N(CC(C)(C)CNC(C2(CC)CC2)=O)CC)=O)cc2ncc(Br)cc2o1 c1(C(N(CCCNC(C(C)OCC#C)=O)CCO)=O)ccc2c(n1)CCOC2 C12(CNC(C(c3ccc(Cl)nc3)C)=O)CCC1CCCN2 c1(C(N(C2CCC(NC(c3c(N)cnn3C)=O)CC2)C)=O)cc2sccc2[nH]1 C(=O)(C(=O)NC(C1CCCC1)CNC(C1CC1(F)Cl)=O)NCCOCC CCCC(CCC)CC(=O)NC(C)(CNC(=O)C(C)OCC)CC C1(NC(c2ncsc2Br)=O)Cc2ccccc2C1NC(C1CCC1)=O c1(C(N(CCCCN(C(CC(C)N(C)C)=O)C)C)=O)ccc(=O)n(CCO)c1 c1(NC(C2C(C(=O)Nc3c(Br)ccnc3Cl)C2)=O)cc(Cl)ccc1[N+](=O)[O-] c1(CC(=O)NC(CC(C)NC(C(CC=C)(C)C)=O)C)ccc(F)cc1[N+](=O)[O-] C1(C(=O)Nc2cccc(F)c2O)CC2CCC1N(C(c1cc(F)c[nH]1)=O)C2 C1(C(=O)OC)CCCN1N(CCNCCN(C)C)Cc1ccccn1 CC1(NC(C23CC2CNC3=O)=O)CCCCC1C(N1CC(C(N)=O)C2(CC2)C1)=O C(=O)(C1=NNC(=O)CC1)NCC(CNC(C1Cc2cc(C)ccc2O1)=O)OC C#CCCC(C(=O)N1CC(O)(C(C)C)C1)NC(=O)CN(C)CCC C1(C(C)O)CCN(C(C2CCC=CC2NC(=O)Cc2ccns2)=O)CC1 C(c1c(C)noc1C)=CC(=O)NCC(CNC(CCc1nc(C)c(C)[nH]1)=O)(C)C C1(=CCNC(=O)C(c2cccc(Cl)c2)O)CCN(C(C2(F)CCCCC2)=O)CC1 Cc1c(C(=O)NCCC(C)NC(c2cccc(C(F)F)c2)=O)nn(C)c1Br Cc1cc(C(N2CCCC2CNC(=O)C(c2ccccc2)C)=O)c(C)n1C C(=O)(C1CC(C)(C)Oc2ccccc21)N1CC(C(=O)NC2(C#C)CC2)OCC1 N1(C(C(CC)n2cccn2)=O)CC(CO)C2(C1)CN(C(c1ccoc1Cl)=O)C2 c1(N(C(CC)CC)C)nnc(N2CCOC(CCF)C2)n1CC(C)C N1(C(c2cnn(C(CC)C)c2C)=O)CC2CCC1C(CNC(=O)CNC=O)C2 c1(C(=O)NC2CCC(NC(C3CCCC(C)(C)O3)=O)CC2)cnc2nccn2c1 N1(C(C(C)N(C)C)=O)CCCC12CCCN(C(C1CC(C(F)(F)F)C1)=O)C2 c1(C(=O)NCCN(CCC#C)C)cc(C(C)C)[nH]n1 N1(C(C2C(=C)C2)=O)CCC(C2CC2)C1CNC(=O)C(c1cccc(F)c1)C C(N=c1[nH]c(C2CC2(F)F)cs1)c1cc(C(=O)OC)no1 C=CC(CCC)CC(=O)NC(CCC)C(=O)NCCC(=O)N(C)C Cc1ccc2[nH]c(C(=O)NC3CC4CCC3N4C(c3ccn(C)n3)=O)cc2c1C CC1(C)CCC(C(=O)NC(C(F)(F)F)C2CC2)CN1C(c1c[nH]c(=O)cn1)=O N1(C(C(C)OC2CCCC2)=O)CC(NC(=O)C(C)OCCN(C)C)C(O)C1 C1(C(N(CC#CC)C)=O)CC2CC1CN(C(c1coc(CC)n1)=O)C2 N1(C(C2C(C)(C)C2(C)C)=O)C(C(=O)NC23CCC(CC2)C3)C2CC(O)C1C2 c1(CC)c(C)nn(C)c1C.c12c[nH]c(n1)C(=O)N(C)CCN(C)C2=O C1(NC(C(C2(O)CN(C(CC3CCC(C)O3)=O)C2)F)=O)CC(C)(C)C12CC2 C(C(C)(C(=O)NCCSC(F)F)NC(c1ccncc1N)=O)SC C1(O)(CCNC(c2cncc(CC)c2)=O)CCN(C(=O)Cn2cnc(=N)[nH]2)CC1 C1(CNCc2cncc(Br)n2)CN2CCC1CC2 C1(CC(=O)NC2CC(CCNC(c3cnc(Cl)s3)=O)C2)CCS(=O)(=O)CC1 c1(C(=O)NC2CC(NC(C(CC)(C)COC)=O)C2)cc2cc(C)cc(C)c2[nH]1 CP(C)(=O)c1ccc(C(c2nnnn2C2CC2)NC23CCCCC2NC(=O)C3)cn1 C(=O)(N=c1[nH]nc(Cl)cc1Br)c1nc(-c2c(OC)ccs2)sc1 C1(C(C)C)(C(=O)NC2CCCC2C#N)CCN(C(C2CC(=O)C2)=O)C1 CC(C)(C)CCC(=O)NCC1CCC1NC(=O)COCc1ccccc1Cl c1(C(=O)OCC)cnc(C)[nH]c1=NCC=CCNC(=O)C(C)(O)C(C)C c1(OC)ccc(Br)cc1C(N1CCC(C)(CNC(=O)C(O)CSC)C1)=O c1(CCC(=O)N(CC(CC)NC(=O)CCNC(=O)C2CC2)C)cc(C)no1 c1(C(N2C(C)CN(C(=O)C3=CC(C)(C)C3)CC2)=O)cc(O)c2sccc2c1 CC1CC(NC(=O)Cc2cnccn2)CCN1C(c1ccc(F)nc1F)=O c1(C(=O)NC2CCCN(C(C3C(C)(C(F)(F)F)C3)=O)C2)ccnc(F)c1N c1(CCC(=O)NCC(C)(C)OCCNC(C(C)C2CCC2)=O)nnc(C2CC2)o1 c1(OCC)ccc(C)nc1C(N1CC(C(C)NC(=O)Cc2ccc(Cl)nc2)C1)=O c1(C(C2CC2)OC)cccnc1C(N1CCC(NC(=O)CC(C)(C)C)C1)=O C1(O)(CN(C(C(CCC)NC(C)=O)=O)C)CCN(C(=O)CNC(=O)OC)CC1 Cc1c(F)cc(-c2cnc(C(F)(F)F)cc2C(=O)NCC2(C)CC2)cc1F N1(CC(=O)NCC)CCN(C(=O)CC(n2nccc2C)C)CC1 c1(CC(=O)NC2CCCCC2NC(c2cc(C(F)(F)F)c[nH]2)=O)ccccc1Cl C1(C)(CC)CC(NC(C2CN(C(c3ncnc(O)c3F)=O)C(C)(C)C2)=O)CCO1 C1(CNC(c2ncc(C)nc2)=O)CC2CCC1N2C(=O)CC1CCCSC1 C1(C(=O)Nc2c(OC)ncnc2)CCN(C(c2ccc(F)s2)=O)CC1O C1(OC)CN(C(C2CCC(=O)N2C)=O)CC1NC(c1conc1C)=O N1(C(CC(C)OC)=O)CC(N(C(=O)CNC(c2ccc(F)cc2)=O)C)C2(CC2)C1 C1(C(N(CCC)CCNC(=O)C(C2CCOCC2)O)=O)CCOC(C(C)C)C1 N12CCC(C(F)(F)C1)NC2=O.C(CCC(c1ccccc1)N(C)C)N(CC)CC c1(OC)ccccc1C(C)C(=O)NCCCCNC(c1sccc1Cl)=O Cc1ccc(CC(=O)NCC(O)CCNC(c2ncoc2-c2ccon2)=O)s1 C1(C(=O)NC(CNC(C=CCOCCOC)=O)(C)C2CCC2)CCNC(=O)C1 N1(C(C=CCCC)=O)CC(C)(C)CC1CNC(=O)C(C)SCc1ccccn1 c1(C(=O)NC(C2N(C(C(C)SC)=O)CCC2)(C)C)cc2ccc(Cl)cc2[nH]1 c1(OC)ccc(C(N2CC(OC)C(NC(=O)C(F)F)C2)=O)c2ccncc12 C1(CNC(c2cc(OC)no2)=O)CC(C(=O)N2CCCCC2C(C)(C)C)=NO1 c1(NCC2CCCC(C)O2)ccc(S(=O)(=O)NCC2(CCO)CCC2)c(Br)c1 N1(C(C=C(C)C)=O)CCC2CC12C(=O)NC(c1nc(=O)o[nH]1)C c1(C(=O)NCCN(C(C(CC)COC)=O)C(C)C)ccc(C(F)(F)F)cc1SC N1(C(c2cnn(C)n2)=O)CCC2(CC1)CC2(CO)CNC(=O)C1=CCCOCC1 C(C)(C(C(C)C)NC(=O)CCc1ccc(Oc2ccccc2)cc1)NC(C)=O N1(C(c2[nH]cc(CC)c2)=O)CCC2CN(C(=O)COCCF)CCC12 C1(C(=O)NCCCCCN(C(C=C(COC)C)=O)C)CCCC(CF)C1 N1(C(C2(C)CCCC2)=O)CC2CC(NC(c3cnn(CC(F)F)c3)=O)CC2C1 C1(NC(CC(C)SC)=O)CC(NC(=O)C(C)N2CC(C)C2)CC1O c1(C(=O)NC(C)CNC(=O)Cc2ccoc2)cncn1-c1cnn(C)c1 C1(CNC(c2n(CCC)ccc2)=O)CN(C(=O)C=Cc2cnc[nH]2)CC1O C1(C(C)(C)NCc2cc(Cl)cc(Br)c2)CCc2ccccc2O1 CCCCC(O)C(=O)N1CCOC(CN(C(=O)CC(C)(C)N(C)C)C)C1 c1(CC(=O)NCC(C2CCCC2)NC(=O)C=CC2CCCO2)csc2nccn12 C(=O)(CC1=CCN(C)CC1)NCCCC(C)NC(=O)C(F)CC1CCCC1 Cc1cccc(C)c1NC(=O)C(=O)NC(CN1CCCS1(=O)=O)C1CC1 c1(OC)nc(C(=O)NC(C)(CNC(C2CC2F)=O)C2CC2)sc1C C1(NC(C(C)N(C(C)=O)C)=O)(CNC(=O)C(C)(C)c2cccnc2)CCOCC1 c1(N(CC(=O)OCC(=O)NCc2ccccc2)CCO)ccc(CNC2CC2)cn1 C1(C(=O)NCCC2CC(F)C2)(CC)CCCN1C(c1cc(CCO)on1)=O c1(C(N2CC3C(C2)N3C(c2ccc(I)cc2Cl)=O)=O)ccc(F)c(F)c1F N1(C(CC(=O)OC)=O)Cc2ccccc2C1C(=O)N1CCN(C)C(=O)C1C C(=O)(C1Cc2ccccc21)N1CC(NC(c2c(C)oc(Cl)n2)=O)CC12CCC2 C(=O)(CC(C)(C)CSC)N1CC=CC(NC(C(C2CC2)SC)=O)C1 c1(NC(c2cnc(OC(C)C)c(Cl)c2)=O)ccc2c(n1)CCCN2 C1(C(=O)NCC2(CCO)CC2)CC12CCN(C(c1cn(C3CC3)nn1)=O)CC2 Cc1cc(Cl)c(C(N2CC(NC(c3ccnn3C3CCC3)=O)CC(O)C2)=O)cn1 C1(NC(Cn2nc(C)c(Cl)c2)=O)COC2(C1)CN(C(C1(O)CCCC1)=O)C2 c1(C(=O)NCC(CC)(C)NC(=O)C(C)S(N)(=O)=O)cnc2cc(C)ccn12 n1(CCC(=O)NCC(C2CCC2)NC(C(C)NC(C)=O)=O)c(C)csc1=O Cc1ccnc2c(C(=O)NCC(O)CNC(=O)CN3CCCC3C)cccc12 C(=O)(C1CCCc2cccnc21)N(C(CNC(C1OCCO1)=O)C1CC1)C c1(CC(C)C)nnc(CN(CCNC(=O)CC2CCN(C(C)=O)C2)C(C)C)s1 C1(C(N2CC(C)C(C)(CNC(c3cnncc3O)=O)C2)=O)Cc2ccccc2O1 c1(C(N2C(C(C)NC(C3N(CCC)CCC3)=O)CCC2)=O)cccc(Cl)c1O c1(C(=O)NC2C(NC(=O)Cc3ccc(Cl)cc3)C2)ccc(O)cc1C(F)F O=C(C1=NOC2(CCC2)C1)NC1CCN(C(C23COCC2C3)=O)C12CC2 c1(OC)ccc(C(=O)NCC(C(C)C(C)C)NC(=O)CC(C)C)cc1OC N1(C(C(C)Cn2ccnc2)=O)CCCC(C2CN(C(C3(C4CC4)CCC3)=O)C2)C1 N1(C(C2C(C)C2)=O)CCN(C(=O)C(C2CCOCC2)F)CC2(CC2)C1 Cn1cncc(C(=O)NCCCCCCNC(=O)CC2(C)CC(F)(F)C2)c1=O CCC(C)(COC)C(=O)NCC1(F)CC(CNC(=O)CC2CC(SC)C2)C1.C(C)=O CCC(c1ccc(C)cc1)=CC(N1CC(N(C)C)C(O)C1)=O C1(C(C)C(=O)NC2CCS(=O)(=O)C2)CCN(C(C2CCC23CCC3)=O)CC1 C1(NC(C(=O)NCCNc2ccc(C#N)cc2)=O)CCc2nccn2C1 C1(C(=O)NC(c2cccnc2)CCOC)(CC)CCCN(C(=O)CC(=O)OC)C1 C1(CNC(c2ccsc2)=O)COCCN(C(c2cccnc2N2CCCC2)=O)C1 N1(C(C(C=C)(C)O)=O)CC2(C1)CN(C(=O)CNC=O)CCO2 C(C)(C(CC(=O)N1CC(OC(F)F)C1)NC(C1(CO)CC(C)(C)C1)=O)OC C(=O)(C(C)(C)C1CCCN1C(=O)Cn1cc(CO)nn1)NC(c1ncc(C)[nH]1)C CC1(C)C(CNC(C2(SC)CC2)=O)CCN1C(C1CCCCN1C(N)=O)=O C12(NC(c3c(C)cn(C)n3)=O)COC(C1)C(NC(c1cc(Cl)cs1)=O)C2 N1(C(C)Cc2cccc(CNC(c3c(C)cncc3)=O)c2)C(=O)NC(C)(C)C1=O c1(CC(=O)NC2C(NC(CC(CCC)(C)C)=O)CCC2)ccc(S(C)(=O)=O)cc1 c1(C(=O)OCC)c(C)[nH]c(CNC(C2CC2CNc2cncs2)=O)c1C CCCCCCC(C)C(=O)NC(COCC)C(=O)N(C)CCSC N#Cc1ccc(-c2cnn(C3CC3)c2)c2ccccc12 Cc1ccc(OC(C)C(=O)NC(C)(CNC(=O)C=Cc2ccsc2)CO)cc1 c1(C(N2CC(CNC(c3nc(Br)c[nH]3)=O)OCC2)=O)cn2ccnc2s1 C1(NC(C2(C)CCC(=O)NC2)=O)CC2CC(C1)N(c1cc(C(N)=O)ncn1)C2 C1(CC(=O)NCCC2N(C)CCC2)CC2(CC2)CN1C(C1CC2(CCO1)CC2)=O N1(C(C(CC)O)=O)CCN(C(c2cnn3ccccc23)=O)C2CCCC12 N1(C(Cc2ccc(C)s2)=O)CCOC2CN(C(=O)C(O)CCC(C)C)CC12 CCC(C)C(O)C(=O)N1CCC(CNC(=O)C(CCO)N(C)C)C12CC2 C12(C(=O)NC3CCC(N(C(CC=CCC)=O)C)C3)C(=O)C3CCC1C2C3 C#CC1(C(=O)NCC2=NOC(C)C2)CCN(C(=O)C(F)OC(F)(F)F)C1 N1(C(C2CC(CCC)C2)=O)CCC(CNC(c2cccc(OCC)n2)=O)CC1C c1(-c2nn(C(C=C)C)c(-c3ccnn3CCOC)n2)ccc(F)c(Cl)c1 CC#CC1CCN(C(=O)CC2(CC(=O)OC)CCOCC2)CC1 Cc1c(NCC(C)CO)ncnc1N1CCC(C(N)=O)C1 N1(C(CC2CC(=C)C2)=O)CC(C)(C(N2CCC(C)C(C)(C)C2)=O)CC1(C)C c1(OC)ccc2nc(C(=O)OC(C(C)C)c3ncon3)sc2c1 c1(CNC(CCN(C(C(C)(C)c2ccno2)=O)CCCO)=O)cccc(C2CC2)c1 c1(C(=O)NCCN(C(c2cc(C)c(Cl)cc2F)=O)C)cccc([N+](=O)[O-])c1Cl N1(C(c2ccc(CCC)[nH]2)=O)CCOC2(CCN(C(=O)CS(=O)(=O)C3CC3)C2)C1 C(=O)(C(F)C(C)C(F)(F)F)N1CCCC(CN(c2cc(SC)nc(SC)n2)C)C1 n1(CC(C)O)cc(C(=O)NCCCCCNC(c2ccc[n+]([O-])c2)=O)ccc1=O S(=O)(=O)(CCC(=O)N1CC2(NC(=O)CC3CCC(F)(F)CC3)CC1C2)N(C)C C1(CNC(C2(C)CC2)=O)CC(NC(c2cnc(S)nc2)=O)C1(C)C N#Cc1ccc2c(c1)CCC2OC(=O)CC(N)Cc1ccc(O)cc1 CCCC1c2ccccc2CCN1c1nc(Cl)nc2c1COCC2 Cc1cnc(C(F)(F)F)c(C(=O)NCC2(O)CCCC2C)c1 C1(NC(C(CN(C)C)O)=O)COC2(C1)CN(C(c1csc(=N)[nH]1)=O)C2 C(CC(C(C)(C)C)NC(c1cn(C)c(=O)n1C)=O)N(C)C(C1CC1C(F)(F)F)=O CCCCCCCCN(C(=O)CCC1CCCCN1C(c1ccsc1OC)=O)C N1(C(C2(C(C)(F)F)CC2)=O)CC2CC(C1)N(C(=O)CC(N1CCCCCC1)=O)C2 CN=c1nc(C(N2CCC(NC(=O)CC3CCC(=O)NC3)C(F)C2)=O)cc(C)[nH]1 N1(C(COCC)=O)CCc2sccc2C1CNC(c1ccc(Cl)c([N+](=O)[O-])c1)=O CC(C)CCCCC(=O)N1CCCC(CNC(=O)CC2CCN(CCF)CC2)C1 N1(C(CCNC(C)=O)=O)CCC(C(F)CNC(C2(CF)COC2)=O)CC1 CCC(C)(C)C(C)CC(=O)NCCC(C)(C)NC(c1cc(=O)c(OC)cn1C)=O N1(CC(COC)C)C(=O)C(CC(=O)NC2CC=CC2)SC1=Nc1ccccc1 Cc1ccncc1C(C)NC(C1CCCCN1C(c1cc(C2CC2)no1)=O)=O Cc1cccc2c(=O)c(C(=O)NC3CCN(C(=O)C(N)=O)CC3F)c[nH]c12 C1(CCC(=O)NCc2cc(OC)ns2)CCCCN(C(=O)CSC(F)(F)F)C1 c1(C(=O)NCC23C(CN(C(CSCC=C)=O)C2)C3)c(N)cc(Cl)cc1Cl N(C1c2ccccc2OCC1O)C(c1c(Br)ccc(C(C)(C)C)c1)=O c1(C(=O)NCc2ccc(CCNC(C(CCC)C)=O)cc2)scc2c1OCCO2 c1(SC)cc(C(=O)NC2CCCC2NC(c2ccc(N)c(N)n2)=O)cc(Cl)c1 N1(C(C2C(C)(C)C2(C)C)=O)CC(NC(=O)CCCNC(=O)C2CC2)CC(O)C1 C1(C(=O)NC(C)C(F)(F)F)(COC)C=CCN1C(c1sccc1Cl)=O C(=O)(CCC(=O)NCCCCN(C)C(C1CCCN(C(N)=O)C1)=O)OC N1(C(=O)N(C2CC2)CC2CC(=O)N(c3ccccc3)C2)CCOC(C(O)CO)C1 C1(C(N2C(C)CN(C(=O)C(F)(F)C3CC3)CCC2)=O)COc2cc(F)ccc2C1 c1(CCC)ccc(-c2ccc(C(N3CCOCC3C)C(=O)NC(C)C)cc2)cc1 c1(C(=O)NCC(CC(=O)NC(c2cccnc2)CC)O)ccc(O)nc1C c1(C(C(=O)NCc2nnn(C)n2)N(c2cccc(F)c2)C)cc(Cl)ncc1F C(=O)(C(F)CC(C)(C)C)NCC1(O)CCN(C(C2C(C(=O)OC)C2(C)C)=O)C1 c1(C(N(C2CCCN(C(c3ccc(CO)cn3)=O)C2)C)=O)cncc(C(N)=O)c1 C1(OC)CC2(CCC(C(=O)NCC=CCNC(C3(C)CNC(=O)C3)=O)CC2)C1 N1(C(CN(CC)CC)=O)CCC(C)C1CNC(=O)CCOc1cccc(Cl)c1 C1(NC(C(CC=CC)C)=O)CC=C(C(=O)N2CC(NC(C)=O)C2)C1 C=CCCCCCCC(=O)N1CCCC(C(=O)NC2COCC2F)C1C c1(C(N2CCCC(CNC(COCCOC)=O)(CO)C2)=O)ccc(C)c(F)c1F Cc1sc2ccccc2c1C(=O)NC(C)CCCNC(C1(C#N)CCCC1)=O c1(C(=O)NCC(C)N(c2nc(Cl)ncc2Cl)C)cnc(C2CC2)nc1O N1(C(C2C(C)(Br)C2)=O)CC2CCC1C1CN(c3nc(-c4ccccc4)ns3)CC21 N1(C(C(CCCOC)C)=O)CCCCC(CNC(c2ncoc2C)=O)CC1 n1(CCC)cc(CN(C(C(=O)NCc2cc(C)on2)C2CCOC2)C)c(C)n1 C1(C(C)C)CC(CC(=O)NCC(C)(C)CNC(=O)CCc2cnn(C)c2)CCO1 Cc1cc(N2CC3C(C2)C3(F)F)nc(N(C)CC2CCCS2)n1 Cc1nccn1CCC(=O)N(C)CCOCCC(=O)NCC1CCC1 c1(C(N2CC(C)(CNC(C3CNC(=O)N3)=O)OCC2)=O)cc(F)c(F)c(Cl)c1F Cc1nc(C(=O)NCC(C)N(C)C(c2ccc(C(C)(F)F)cc2)=O)c(C)s1 C(=O)(CCCC(F)F)NCC(CC)NC(=O)C(C)n1ccnc1 C1(C)(C(=O)NC2C(C)CCN(C(c3ccccc3O)=O)C2)CCS(=O)(=O)N1C C1(CNC(C=CC(C)=O)=O)CCCCC1NC(=O)C=Cc1ccco1 C1(CCC(=O)NC(C)C(CO)NC(=O)CCC2CCC(=O)NC2)NC(=O)NC1=O C(=O)(C(CN(C)C)C(C)C)NCC1(CCCNC(C(F)=C(C)C)=O)CCCC1 N1(C(c2cc(COC)on2)=O)CCC(NC(=O)Cc2ccc(C)cc2)C1C(C)C N1(C(C2CCCN(C(C(CN(C)C)O)=O)C2)=O)CC(C(N)=O)C2(CC2)C1 C1(NC(c2ccn(C(C)C)n2)=O)CC=CCC1C(=O)NCC1(O)CCCOC1 C(=O)(C(C)C(C)S(C)(=O)=O)NC12CC(NC(Cc3c(C(=O)OC)occ3)=O)(C1)C2 CC(CC(=O)NCC12CCC(NC(=O)C(F)=C3CCCC3)(CC1)CO2)C(C)(C)C N1(C(c2ccc(-c3nc(C)c(C)o3)cc2)C(=O)NC(C)C)CC(C)SC(C)C1 c1(CC)ccc(CC(=O)NC2CCCC2NC(=O)C(C)C(C)C)cc1F C12(NC(c3c(CC)cccn3)=O)CCN(C(c3[nH]c(C)nc3C)=O)CC1C2 c1(C(=O)NC(CC)CNC(=O)Cc2cc(C)ccc2C)n[nH]c2ccc(F)cc12 C(=O)(C1=Cc2ccccc2C1)N1CCC(CN(C(c2c(CC)nc(C)o2)=O)C)C1 O=S(=O)(c1ccc(N2CCOC(c3ccccc3)C2)cc1)C(F)(F)F N1(C(=O)NC(c2nccc(C)c2)C)CC2(C1)CN(C)C2 c1(CC(=O)NC2CN(C(CC(=C)C)=O)C(C)CC2)c(C)[nH]c2ccccc12 CCC(O)CCN=c1nc(N2CCC(CN3CCCCCC3)CC2)cc[nH]1 N1(C(CSC(C)C)=O)CC(O)CC1CO.C12CC(O)C1CC(=O)N2 C1(NC(c2onc(C)n2)=O)CN(C(C2CC(F)(CO)C2)=O)CC1C C1(NC(C=CC)=O)(CC)CCN(C(=O)C(C2CCC2)OC)CC1 NS(=O)(=O)CCC(=O)NCCC1CCC(NC(C2CC2C2CC2)=O)C1 C12(COC)CC(NC(=O)CC(C)CN(C)C)(CN1C(c1ccc(OC)s1)=O)C2 C1(=CCNC(C2(CCOC)CC2)=O)CCN(C(=O)C(=O)N(C)C)CC1 C1(CNC(C(C(C)C)(C)O)=O)CCC2(CN(C(=O)CCn3cncn3)C2)O1 c1(C(=O)NCC2(OC)CN(C(=O)C(F)(F)C3CC3)C2)cnc2nccn2c1 CC(C)C(C(=O)N1CC(CCNC(C2CCO2)=O)C1)N1CCCCC1 C1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CCN(C(C2CCC=CCC2)=O)CC1O N1(C(c2c(CC)n[nH]c2)=O)CCCCC1C(N1CC(OCC(=O)NC)C1)=O c1(C(N2CCC(C(C)(C)NC(=O)C3=C(Cl)CC3)C2)=O)cc2c(cc1Cl)OCO2 C1(CNC(C(C)N(C)C)=O)N(CC(=O)NCC2CC2)CCCC1(C)C Cc1cc(C)c(C=CC(=O)NC2CC2CNC(=O)CC(C)(C)CC(F)F)c(C)c1 C(C1=CCN(C(c2ccn(C)c2C2CCC2)=O)CC1)NC(CCSCCCC)=O C1(OC(C(c2cccc(O)n2)C)=O)CCN(c2ccc(Cl)cc2)C1=O c1(C(=O)NC2CC(NC(c3cccc(=O)o3)=O)C2)c(Cl)cncc1Cl C1(C(=O)NC(C)CCCNC(=O)COC2COC2)CNC(=O)CC12CCC2 CC1(C)CC(NC(c2ccccc2C(C)(C)C)=O)CN(c2cnc(C#N)cn2)C1 CC(N=c1[nH]c2c(c(=NC3CC(C4CC4)C3)[nH]1)SCC2)c1cc2cnccc2[nH]1 C1(NC(C=C(C)C)=O)CCCC(CNC(=O)Cc2cscc2F)C1 CC1(C)CCC(CNC(c2sc(F)cc2Cl)=O)N(C(=O)COCC2CCC2)C1 Cc1cc(C)c2c(S(=O)(=O)NCc3nn(C)c4ccccc34)n[nH]c2n1 C1(CC(C)C)CCCC1NC(C1(N(C)C(C2CCCSC2)=O)CC1)=O c1(C(N(C(C)CNC(=O)CN2CC(C)(C)C2)CC)=O)ccc(C2CC2)c(OC)c1 Cn1cnc(C(=O)NCCN2CCN(C(c3nc(Cl)ccc3N)=O)CC2)cc1=O C(=O)(CS(=O)(=O)C1CC1)N(CCn1cc(Cc2ccc(Br)cn2)nn1)CC N1(C(C(C)N(C(=O)C=CCN(C)C)CCC)=O)CCC(c2nn[nH]n2)C1 CC(C)C(CNC(=O)C=Cc1cnn(C)c1)C(=O)N(C1(C)CCCC1)C C(c1scnc1C)=CC(=O)NC1C(NC(C(C)(c2ccccc2)OC)=O)CCC1 N1(C(Cn2c(C(C)C)nnn2)=O)CCC(C)N(C(=O)CC2CCN(C)C2)CC1 N1(C(CC(C)(C)C)=O)CCN(C(=O)CSc2ccccc2O)CC1c1cn[nH]c1 C1(C(N(C)CCOCCCO)=O)(CNC(c2nnsc2N)=O)CCCCC1 c1(OC(C(=O)NC2CC(N(C(C=C(CCC)C)=O)C)C2)C)ccccn1 c1(C(=O)NCC(CCNC(Cc2cnc(C)[nH]2)=O)O)cnncc1C N1(c2nnc(CC)o2)CC(NC(C2CCC(=O)N(C(C)C)C2)=O)CC2(CCC2)C1 Cc1ncccc1CNC(=O)CCC1CCCCN1C(=O)NCC1(C)OCCO1 N1(C(C2C(C)C2)=O)CCC2(CC1)CC(NC(c1cc(Cl)cs1)=O)CO2 c1(NC(C2C3CN(Cc4cn(CC(C)C)nc4)C2C3)=O)cc(O)cc(O)c1 c1(C(N2C3CC(CNC(CS(CC)(=O)=O)=O)C2CC3)=O)c(O)nnc2c1CCC2 CCC(CC(C)C)C(=O)N1CCC(NC(=O)C(C)C(C)(F)F)C(CO)CC1 c1(COC)ccc(C(=O)NCC(=O)NCCN(C(C)C2CC2)CC)cc1 C1(NC(C(Cn2ccnn2)NC(C2C=CCS2)=O)=O)CC2CCCC(C1)C2 CC1CCN(C(c2[nH]ccc2C2CC2)=O)CC1CNC(c1cc[nH]c(=N)c1)=O c1(CC)cc(C)c(C(=O)NC2(C(=O)NC3CCNC(=O)C3)CCOCC2)o1 c1(C(=O)NCC2(F)CN(C(c3c(C)con3)=O)C2)sc(C)c(C)c1C Cc1nc2ccccn2c1C(=O)NC1CCN(C(C2C=CCCC2)=O)C1C C1(CC(=O)NCC(C)(C2CCC2)NC(C2N(CC)CC2)=O)NC(=O)NC1=O C#CC1(NC(c2ccc(CNC(=O)C(CCC)N(C)C)s2)=O)CCCCCC1 C=CCCCCCCCCC(=O)NC(CNC(=O)C(C1CCCCCC1)C)CO S(=O)(=O)(c1ccc([N+](=O)[O-])cc1CN1CCC2OCCC2C1)NCC C1(C(=O)OCCc2n(-c3c(C)cccc3)nnn2)CCCC(C)C1C C1(N=c2cc(Br)n(C)[nH]2)(c2n(CCSC)nnn2)CCC2COCC2C1 CC(C)C(CNC(C1CCN(C)C1)=O)C(=O)NCC1CCCCO1 N1(C(CNS(NC)(=O)=O)=O)CC=CC(OC)C1.C12(CC1)C(=O)N2 C(C(O)CC(=O)N1CCC(OCCN(C)C)C1)NC(C(C)=C1CCCC1)=O C(=O)(CS(=O)(=O)CC)NCCCN(C(CC(CC)C)=O)C1CC1 Cc1ccc(NC(C2CCN(c3ncc4c(n3)CCC4)C2)=O)cc1[N+](=O)[O-] N1(C(c2c(C)cc(SC)o2)=O)CC(CCNC(=O)Cn2cnnc2O)OC(C)C1 c1(CC(=O)NC2CCN(C(Cc3ccc(C)cc3Cl)=O)C2)csc2cc(C)sc12 n1(CC(N2CCC(F)(CNC(CC(CC)C)=O)C2)=O)cc([N+](=O)[O-])ccc1=O C(=O)(C(C)(C)C(C)(C)O)N1CC(CC(C(=O)NCC(C)(C)F)F)C1 c1(C(=O)NC(CCCC)CNC(=O)C(=O)N(C)C)cc([N+](=O)[O-])cnc1C c1(CC(=O)NC2CN(CS(C)(=O)=O)C2)c(F)cncc1F c1(CN(c2cc(NC(c3ccco3)C)ncn2)C)ncc(Cl)cc1F N1(C(=O)NCc2cccc(OC)c2)CCCC2C1CCN2c1ncc(I)cn1 N1(C(c2cn(CC)nc2)=O)CCN(C(=O)C=C2CCN(C)C2)CC1CF c1(C(=O)NCC(CCC)C)cc(S(=O)(=O)CC)ccc1OC N1(C(c2nnn(C)n2)=O)CCC2CCCC12CNC(c1cnc(N)cn1)=O C(=O)(CC1CNc2ccccc21)N(CCOC)CCNC(=O)C=Cc1nccs1 N1(C(CC(C)NC(=O)CCC2CCCCC2)=O)CCn2cnnc2C1C N1(C(C(F)=C(C)C)=O)CC2CCC1C1CN(C(c3c(C)noc3N)=O)CC21 C1(NC(c2nnc(O)nc2O)=O)CN(C(=O)CCCn2ccnn2)CCC1CO C1(Oc2ccc(N(C(CSCC(=O)OC)=O)C)cc2)CCCN2CCCC12 Cc1ccc(CC(=O)NCCC2(C(=O)NC3CCC(CC(C)C)C3)CCC2)o1 C1(C(=O)NCC2CN(C(C(CC)C)=O)C2)N(C(=O)COC(C)C)CCC12CCC2 S(=O)(=O)(c1cccc(Br)c1)NC(C)C(N1C2CCC1CC2)=O N1(CC(=O)NC(C)CCNC(=O)CCNC(C2CC(=C3CC3)C2)=O)CCSCC1 C1(NC(=O)CCOCc2ccccc2)COC2CN(C(=O)CCC3CC3)CC12 C12(NC(=O)CC3CCCS(=O)(=O)C3)CCC(CN(C(=O)C3=CCCC3)C1)C2 N1(C(C2C(COC)CC2)=O)CC=CC1C(N1CCC1)=O N1(C(c2nc(CC)sc2)=O)CC(O)CCC1C(=O)NC(C)Cc1cc(C)[nH]n1 N1(C(CN(CCC)C)=O)CCCC(NC(c2coc(C(=O)OC)n2)=O)C1 O=C(N=c1[nH][nH]c2c1CCCC2)C1CCCN1C(c1cccc(CCO)c1)=O CCC(CC)(CCC(=O)OC)NC(c1c(C)cc(Cl)cc1C)=O C(CN=c1nc(CO)[nH]s1)=C(CNC(C1CCC(C(C)(C)O)CC1)=O)CCCO N1(C(CCC#C)=O)CC(C2CCCN(C(C3CCCCN3N=O)=O)C2)C1 Cc1occc1CC(=O)NCC12CC(NC(C34CSCC3C4)=O)(C1)C2 CN1CCCC1C=CC(=O)NCCC1CN(C(c2n[nH]cc2Br)=O)C1 N1(CC)CCN(CCCC(N2CCC(NC(=O)C(C)=C(C)C)C2C)=O)CC1 Cc1csc(CC(=O)NCC(C2CCCC2)NC(=O)Cc2csc(C)n2)c1 C1(CC(N2C(CNC(C3(SCC)CCC3)=O)CC2)=O)COCCN1CC(F)(F)F N1(C(c2c(Br)cn(CC)n2)=O)CCC(CNC(C2CCOC(C)C2)=O)C(O)C1 C1(NC(CC)=O)CCCCC1NC(C1CC1OCc1ccccc1)=O C(=O)(CCCC(C)(C)NC(c1ccccc1OC)=O)NCC#C c1(OC)cc(C(=O)NC(CNC(C2(O)CCCCC2)=O)CC(F)(F)F)cc(F)n1 N1(C(C2C(NC(C3CC4(CCC4O)C3)=O)C3CCC2C3)=O)CCC2(CCOC2)C1 c1(COC)cccc(C(=O)NC2CCC(CC(=O)N(C)Cc3ncccn3)C2)c1 C1(C(=O)NCC(c2cccs2)C)CCN(C(C2CC2C(C)(F)F)=O)CCO1 C(=O)(C(CC)(CC)CC)NC1CCCN(C(c2nc(CC)oc2C)=O)C1 N1(C(c2c(C)coc2)=O)CCC2(CC2C(=O)NCc2cccnc2C)C1 c1(C(=O)NCCCNC(c2c(C)csn2)=O)c(C)nsc1C Cc1ccc(NC(=O)C(=O)N(C2CN(C(=O)CS(N)(=O)=O)CC2O)C)cc1C CCC(C(=O)NCC12CC(NC(c3cn(C)nc3SC)=O)(C1)C2)C(C)(C)CC c1(C(N(CCN(C(c2c(C)cn(C)n2)=O)C)C)=O)nc2ncccn2n1 C(C(C)(C(=O)N(CCCC(O)CO)C)NC(=O)CCCOC(C)(C)C)SCC Cc1nnn(CC(=O)NCCCCCN(C)C(c2[nH]nnc2C2CC2)=O)n1 CCCCC(O)C(C)C(=O)N1CCC(C2CC2)C1C(=O)NCCC1(O)CCC1 CC1C(NC(=O)COC2CCOCC2)CC2CCC1N2C(=O)CC1CCCCC1 c1(CC(=O)NCC2C(NC(C(C=C)O)=O)CC2)c(C)noc1C N1(C(C(CC)(C)O)=O)CC2(C(N3CC(O)C(N=[N+]=[N-])C3)=O)CCC1CC2 n1(CC(=O)NCC2CCC2C(N2CCCC2)=O)cnoc1=O N1(C(Cn2c(=N)scc2)=O)CC2CC(NC(C3CCCN3N=O)=O)C2C1 C1(OCC=C)CCN(C(c2cnn(CC(F)F)n2)C(=O)NCCCC2CC2)CC1 c1(-n2cc(C(NOC(C3(OC)CCNC3)=O)=O)nn2)ccc(Cl)cc1Cl C(=O)(CC(O)(C(F)(F)F)c1nccn1C)NC(c1ccc(CC)cc1)CC(=O)O c1(C(=O)NCC2(C(=O)Nc3cc(C(=O)OC)ncc3)CC2)cccc(=O)n1C c1(C(N2CCC(N(C(=O)CSc3n[nH]c(O)n3)C)C2)=O)cccc([N+](=O)[O-])c1Cl C(=O)(C(C(C)NC(c1coc(CO)c1)=O)C(C)C)NC(CC(=O)OCC)C N1(C(CC2C(C)CCO2)=O)CCN(c2ccc(NC(=O)COCCF)cn2)CC1 c1(C(=O)NC(CC)C(=O)OC)ccc2c(-c3cccc(OC(C)C)c3)n[nH]c2c1 c1(-c2n(C3CCN(N(c4nc(O)c(C)s4)CC)CC3)nc(C)n2)cc(O)nc(C)n1 C=CCCCCN(C(CC1CCC2CC12)C(=O)NC)C.C1(C)C(=O)N1 C(N=c1nc2sccc2c(N2CC(N(C)C)C(C)(C)C2)[nH]1)c1scc(C)n1 c1(C(=O)NCC(CO)NC(C2CN(c3nncs3)C2)=O)cc(F)c(O)c(F)c1 C(CC(C)C(=O)NC(C(=O)N(C(C)CC1CC1)C)C1CCOC1)=CCC N1(C(CCCN(C(C)=O)C)=O)CC2CC1CN2Cc1ncnn1C(C)(C)C N1(S(CCCC)(=O)=O)CC2CCN(C(C3CCCN3C(C)C)=O)CC2C1 C1(C(N2C(C(=O)NC(c3cc(C)on3)C)CC(C)C2)=O)CN(C)CC(C)O1 c1(NC(C=CCNC(c2ccc(OC)nn2)=O)=O)cccc(C#N)c1C C1(CNC(=O)C(C2CCCCC2)F)(NC(C2CC2C2CCCO2)=O)CCOCC1 c1(C(=O)NC2CC(NC(C(CC3CCCCC3)OC)=O)C2)cc[nH]c(=N)c1 N1(C(c2c(CNC(C3C(C)(C)C(=O)C3)=O)c[nH]n2)=O)CC(O)CC1(C)CO Cc1nc(C(=O)N(CCNC(=O)C(C)CC(C)C)C(C)C)ccc1C#N C1(NC(c2cc(C(C)(F)F)n[nH]2)=O)C=CCN(C(=O)Cc2cn[nH]c2)C1 O(N1CCC(CC(=O)NC(C)C(C)NC(=O)Cc2noc(C)c2C#N)CC1)CC c1(OC)ccc(F)c(N)c1C(=O)NC1CC(C)(NC(=O)C=Cc2ccccc2)C1 CC1CN(C(C2CCC(O)CC2)=O)CCCN1C(c1cnnc(Cl)c1)=O c1(C(=O)NCCC(C)N(C(C(C=CCCC)O)=O)C)cnc(N)c(O)c1 C(=O)(C(CCC1CCC1)NC(=O)Cc1ccncc1F)N(C1CC(OCC)C1)C c1(C(N2CCC(CNC(C3C(OCC)C3)=O)C2)=O)csc2cc(OC)ccc12 c1(C(=O)NCCOCCCNC(C2CC2Cl)=O)ccc(C(F)F)cn1 CC1CCC(CNC(c2cc(F)cnc2O)=O)N(C(=O)C2=CCOC2)C1 C1(CN(C(=O)NCc2c(OC)cnc(C(F)(F)F)c2)C)COc2ccccc2O1 C(C)(C(=O)NCC1CCC1C(=O)NCCCCO)OCC=C.C1CC1 CCCC(CCC)CC(=O)N1C(C(=O)NC2C3CCCCCC23)CCC12CCC2 C1(CNC(C2(OCC)CCC2)=O)CCCCN(C(c2ccoc2Cl)=O)CC1 CC1CC(NC(c2c[nH]ccc2=N)=O)CN1C(c1cc(C2CC2)oc1C1CC1)=O CC1CCC(C(=O)NCCc2csnn2)CN1C(=O)COCC(F)F C(CC(C)(C)C(=O)NC(C)CCNC(c1cc(Br)sn1)=O)OC C1(C(=O)NCc2cncc(SC)c2)(C(=O)NCCN(C)CCO)CNC(=O)C1 Cc1oc(S(C)(=O)=O)cc1C(=O)NCC(C)(O)CNC(=O)C(C)(F)F C1(C(=O)Nc2cccc(NC(C3C(c4n(C)nnc4)C3)=O)c2)CCOCC1(C)C c1(C(C)OC)nc(Cl)cc(=NCC2CCC(NC(c3nc(Cl)cs3)=O)C2)[nH]1 C1(CC)C(C)CCN1C(c1ccc(C2CCCC(=O)N2)cc1)=O c1(C(=O)NCC2CC(NC(C3(CC)CCC3)=O)C2)oc(CO)cc1C C(=O)(C1CCc2c[nH]nc21)N1CCCC(CC(=O)NCCn2c(CC)ncc2)CC1 c1(C(N2CC(N3CCN(C(C4(CC=C)CC4)=O)CC3)C2)=O)ccn2ccnc2c1 C(=O)(CC(CCC)NC(=O)C=Cc1cc[nH]c1)NC(CCC=C)(C)C Cc1nc(N2CC(F)(c3ccccc3)C2)sc1Br.c12ccc(cc1)o2 Cc1c(CC(N2CCCC(CNC(c3cc(Cl)no3)=O)C2)=O)sc2ccccc12 CCC(C)C(O)CC(=O)NCc1n[nH]cc1C(=O)NC1CCS(=O)CC1 N1(C(C2(C)CC(=O)C2)=O)CCN(C(C2(C#N)CC3CC3C2)=O)CC(O)C1 S(=O)(=O)(c1cccc(=NCCOc2ccccc2)[nH]1)N(C1CC1(C)C)C c1(OC)cc(C(=O)NC(C)(CNC(=O)CC(C)NC(N)=O)CO)cc(OC)c1C N1(C(c2cc(OCC)n[nH]2)=O)CCC2CN(C(=O)CN3C(=O)CCCC3=O)C2C1 C=CC(CC)C(=O)NCC1(CNC(c2cnn(C(C)(C)C)c2)=O)CC12CCC2 C1(NC(C2(N3CCN(C)CC3)CC2)=O)CN(C(=O)CC2CCC2)CC2(CC2)C1 N1(C(c2scc(C#N)c2)=O)CCCCCC1CNC(C1(F)CCCCCC1)=O CC1(O)CCC(C(=O)NC2C=CC(CNC(=O)C3=CCCCC3)C2)CC1 C(=O)(CC(F)(F)C(F)(F)F)N1C2CCC(CCNC(CCSCCC)=O)(CC2)C1 N1(C(CCC(C)SC)=O)CCCCCC1C(=O)NCCC1CCC(C)(C)O1 C1(C(N(CC(C)NC(COc2c(C)occc2=O)=O)C)=O)CCc2ncnn2C1 CC(C)CCCC(=O)NCCCOC1CCN(C(C2CCCCCN2C)=O)CC1 S(=O)(=O)(C1CC2(CC2)C1)N1CCCC(C(N2CCCC(C(N)=O)C2)=O)C1 N1(C(CCCC=C)=O)CCN(C(=O)Cc2ccc(F)cc2C)C(C)C1C CCC(CC(=O)NCC1CC1NC(=O)C(F)(F)c1csc(C)c1)C1CC1 C(CC)(CCC(=O)NCC(C)(C)C#N)NC(COCCC)=O c1(CC)ccc(C(=O)N(C)CC2CCN(C(=O)Cc3ccc(C)o3)C2)cc1F c1(CNC(CC2(C)N(C(C(C)OCC)=O)CC2)=O)cccc(CO)c1 c1(C(N(CCC2N(C(c3ccc(C)o3)=O)CCCC2)C)=O)cc2cccnc2[nH]1 c1(C(=O)NC(c2ccncc2)CC)coc(CNC(C2CC3(CC3)C2)=O)c1 Cc1cc(C(=O)N(C2CCC(NC(C3CCC(=O)C3)=O)CC2)C)oc1C C1(NC(C(C(C)C)O)=O)CCC(C)N(C(C2CCC(=O)N(C3CC3)C2)=O)C1 Cc1nn(-c2ccncc2)cc1CN(CC(O)C(C)(C)C)C C1(O)(CC(=O)NCC(C(C)C)(C)NC(c2ncc[nH]c2=O)=O)COC(C)(C)C1 CCC(CNC(c1cocn1)=O)NC(=O)Cc1cc[nH]c1 C1(NC(c2nccc(OC)c2)=O)CN(C(=O)C(C)NC=O)CC12CC2 N1(C(c2c(OC)csc2)=O)CC(CNC(=O)CC(C)CF)C2(CCOCC2)C1 N1(C(CC(C)SC)=O)CCN(CCCCCNC(=O)Cc2cc[nH]c(=N)c2)CC1 N1(C(CC(C)F)=O)C2CC1CN(C(c1ncc[nH]1)=O)C2 c1(CS(=O)(=O)Oc2ccc(CF)cc2)cc(F)c(F)cc1Cl C(C(=O)NCC(C1CCN(C(C2(C)CC2)=O)CC1)(C)O)(C(C)C)OC CC1(C)CC(CNC(c2ccccc2Cl)c2nnnn2CCC2CC2)CNC1=O C12(CNC(C(C)(C)CO)=O)CCC(CC1NC(=O)CSc1cc(F)ccc1F)C2 CCC(C)C(C(C(=O)NCC(=O)OCC)N(CCS(C)(=O)=O)CC(=O)OC)OC C1(C2CC2)(CNC(c2n(C=C)ncc2)=O)CCN(C(c2cc(C)ncc2C)=O)C1 N1(C(CCN(C(C)=O)CCO)=O)CCC(F)(CO)C1 c1(C(=O)NC(C2(O)CN(C(C3CC(OC)C3)=O)C2)C)sc(Cl)cc1Cl C1(NC(C2CC2(F)F)=O)CCN(C(=O)CCc2csnn2)C12CCC2 N1(C(CCN(C(C(C(=O)OC)C)=O)CC2CC2)=O)CCC(C)(C2CC2)C1 Cc1ccc(C(N2CC(C)(C)CC2CNC(C23COCC(C2)OC3)=O)=O)c(F)c1 CCC(CC(=O)NC(c1ccsc1)C)NC(=O)Cc1csnc1C C1(NC(CC2CCN(C(CCc3c(C)noc3)=O)CC2)=O)CCOC12CCOC2 N1(C(CN(C)C(N)=O)=O)CCC(C2CCN(C(c3cc(C4CC4)ccn3)=O)C2)C1 c1(C(=O)NC(c2cccnc2)C(=O)NCCN2CCC2)ccncc1F C12(NC(=O)CCF)CCCN(CC(F)(F)F)CC1C2.c12cccc(n1)NC2=O c1(C(N(CC(C)N(C)C(c2nnn3c2CSCC3)=O)C)=O)csc2c1CCCC2 c1(OC)nc(-c2occc2C)ccc1C(=O)NCCC#N N1(C(CCC)=O)CCCC12CCN(C(=O)C(C(C)C)n1cc(Br)cn1)C2 C1(C(=O)NC(C)CC(F)(F)F)CCN(C(C2CCCCC(=O)N2)=O)C(C)(C)C1 N1(C(CC2ON=C(C)C2)=O)CCC(N(C(=O)CC2(O)CCOCC2)CCO)CC1 N1(C(c2cc(C)no2)=O)CCC2CC(NC(c3ccncc3F)=O)CCC2C1 c1(C(=O)NC(CNC(C(C)n2ccnc2)=O)(C)C2CC2)ccc2c(c1)nnn2C c1(C(=O)NCC(CC(C)C)NC(C2(C)CC2C)=O)cnc(N)c(Cl)c1 C(=O)(C1=NNC(=O)CC1)NC1C(C)CN(C(c2sccc2C(F)F)=O)C1 c1(CC)cc(NC2CN(C(c3n[nH]cc3C)=O)CC2C)nc(C)n1 CCC(C)(CCNC(=O)Cc1ccc(O)nc1)NC(=O)C(=Cc1cccnc1)C c1(CC)ccc(NC(C2CC(OC)CN2C(=O)CN2CCCCC2=O)=O)cc1 Cc1cc(Cl)c(C(=O)NC2CC(F)(CNC(=O)Cc3cccnc3Cl)C2)cc1N CC(C)C(C)CC(=O)NC1(CNC(c2ccc(Cl)cc2Cl)=O)CCOC1 c1(C(=O)NC(CCC)CNC(=O)C(CC)OC)cnc2[nH]ncc2c1 C1(F)(CNC(C2C(C)(C(F)F)C2)=O)CCN(C(C2CCC(C)(F)CC2)=O)CC1 c1(CNC(C(C)N(C(=O)CCCNC(N)=O)CC)=O)c(F)cncc1F c1(OCC)cc(C(=O)NC(C)(C)CCNC(c2ncoc2C(C)(C)C)=O)[nH]n1 N1(C(c2c(C)nc(O)cc2)=O)CCC(C)(C)C(C(N2CCN(C)C(=O)C2)=O)C1 Cc1occc1C(N1CCCC1CCNC(C1CC1(C)C(F)F)=O)=O S(=O)(=O)(c1ncc[nH]1)NC1C(C(=O)OCC)CC=CC1 C1(NC(C2CCCN(C(CC3CCCC(C)(C)C3)=O)C2)=O)CN2CCC1(C)CC2 S(=O)(=O)(c1ccc(C(=O)OC)cc1)Nc1cccc(CN(CCCC)CCO)c1 C(=O)(C#CC1CCCCC1)N(C1CCCCN(C(C2N(C)CCC2)=O)C1)CCO c1(CN2CC3C(CN(CCOC)C)C3C2)cc2c[nH]nc2cc1C Cc1ccnc(C(=O)N(C)CC2CN(C(=O)C(n3ccnc3C)C)CCO2)n1 c12cc(C)ccc1S(=O)(=O)Oc1cc(n(C)n1)NC2=O.C1(CC)CC1 N1(C(C2CC(C)(F)C2)=O)CC2(CC(NC(C3CC3c3ccncc3)=O)C2)C1 C=CC1(C(=O)NC2CC3(CC3)C2)CCN(C(C2CCCCO2)=O)C1 N1(C(C2CCN(C)C2)=O)CC2(C(N3CCC4C(O)CC34)=O)CC1CCO2 N1(C(c2c(C)nc(Cl)cc2)=O)C2CCC1CC(CNC(c1ccnc(F)c1)=O)C2 c1(NCCC2CCCN2)ncnc2sc(Br)cc12 C1(NC(CNC(=O)OC)=O)CC2CC1CC2C(=O)NCC(F)C1CCC1 N1(C(C)=O)CC2C(C1C(=O)Nc1cc(C(=O)OC(CCO)C(C)C)ccn1)C2(C)C CC1CN(C(C2(C#N)CC2)=O)CC1NC(=O)COc1ccccc1 c1(N2C(CSC)CCC2)cc(=NC2C3Cc4c(Br)cccc4C23)[nH]c(C(C)C)n1 c1(C(=O)NC2CCCC(NC(c3cc(C(C)C)on3)=O)C2)cnc(Cl)cc1N S(=O)(=O)(c1cc(CC)c(F)cc1OC)N1CCN(CC)C(C)(C)C1 Cc1cc(O)cc(C)c1N(CC(N1CCCCC1)=O)C(C12CC1CCN2)=O c1(C(C)N(C(C)(C)C)C)cccc(N2CCOC2=O)c1.C1(=O)C(CN(C)C)N1 c1(Cn2cc(C3CN(C(C(C)CC(N)=O)=O)C3)nn2)cccc2c1ccn2C C(=O)(CCCC(C)(F)F)NC(C(C(C)C)NC(=O)COCc1ccncc1)C CCCC(O)C(=O)NCCCOCCNC(C1COC(=O)N1)=O Cc1cc(C(=O)NC2(CC(=O)NOCCCNC(N)=O)CCCCC2)c(C)cn1 CCCCCC(CC)C(=O)NCC1(C)CCCN(C(=O)CCOCC)C1 c1(C(=O)NC2(CC=C)CN(C(=O)CC(C)(C)SC)C2)ccccc1CC#N N1(C(CCSCCCC)=O)CC(F)(CNC(C2(C3CCCCO3)CCC2)=O)C1 N1(C(CCC2(C)CN(C(C(C(C)C)O)=O)C2)=O)CCCC(C)(C#N)C1 Cc1cnn(C)c1C(=O)NCC1(F)CC(NC(c2ccc(SC(C)C)cc2)=O)C1 C1(C(=O)Nc2ccc(SC)o2)CN(C(=O)CC(C)N(C)C)CCC1O c1(C(=O)NC23CC(CNC(Cc4cc(C)sc4C)=O)(C2)C3)c[nH]c2ncccc12 C=C(C)C(C)(C)C(=O)N1CC2CCC2(NC(c2ccc(=O)n(C(C)C)c2)=O)C1 c1(C(=O)NC2CC(O)(CNC(C(C)(C)C(N)=O)=O)C2)cccc2c1C1CCC2O1 N1(C(CC(C)SC)=O)CCCCC1CNC(c1ccc(CSC)o1)=O N1(C(C)C)CCC(C(=O)NC2CCCC(N(C)C(c3cn(C)nc3Cl)=O)C2)CC1 c12ccc(cc1)C(=O)N(C)C1CCC1N(NC(CCC)=O)C2.C(=O)(C(C)C)NC C1(OC)CN(C(=O)CCC2CCCOC2)CC1NC(c1ccc(CSC)o1)=O N1(C(C(CC)CC(F)F)=O)Cc2ccnn2CC(NC(=O)C=C2CCOCC2)C1 Cc1nc(C2CCCOC2)sc1C(=O)NCCN(C)C(c1cocc1C(N)=O)=O CCCCC(C)CCC(=O)NC(C)C(C)(C)C(=O)N1CCCC1C c1(C(N2CC(C)C(NC(=O)CC3CC=CCC3)C2)=O)cc2scnc2[nH]1 C12CCCC1(C)N2.c1(C(=O)NCC2CN(C(=O)OC(C)(C)C)C2)cc(F)n[nH]1 N1(C(c2c(C)coc2)=O)CCN(C(=O)CNC(c2c(C)n[nH]c2C)=O)CC12CC2 C1(NC(C2CCC(=C)CC2)=O)CCCC2CN(C(C3CC3C)=O)CC12 N1(C(C(C=C)(C)C)=O)CCCCC2(C1)CN(C(=O)C(C)(C)CC#N)C2 CCCCC(CC)CC(=O)NC1CC(NC(=O)CN(C2CCC2)C)CC1O c1(C(=O)NCC(C)NC(C2CN(CC)C(=O)C2)=O)cnc2n(c1=O)CCS2 C(=O)(CCCCN(C(N)=O)C)N(CC(O)CNC(=O)C(CO)c1ccccc1)C c1(C(N(C2CCN(C(=O)C(C)CF)C2)CC)=O)ccc(N(C)C)nc1 C#CCC(C)(C(=O)N(CCC)OC)NC(C1C2CCC(F)C12)=O N1(C(C(C)P(C)(C)=O)=O)CC2CCC(C1)N2C(c1ccn(C2CC2)n1)=O CN=c1nc(N2CCCCC(C)C2)[nH]c(=NCc2c(F)cccc2Cl)[nH]1 Cc1ccc(C(=O)NCC#CC(N2CCC(C)C2C)=O)nn1 S(=O)(=O)(c1ccc(C(=O)N(CCCNC(=O)CNC=O)C)cn1)NC c1(C(=O)NC2C(CNC(C3(CCOCC)CCCC3)=O)CC2)c(Cl)cccc1Cl C1(C(N(c2cccc(C(=O)OC(C)(C)C)c2)C)=O)CC(C(C)(C)C)=NO1 c1(N2CCN(C(C(=O)N(CCCC(=O)O)C)=O)CC2)ncc2n1CCCC2 C(=O)(C=C1SCC(=O)N1C)N1CCCC(C)(CNC(c2cnc(OCC)s2)=O)C1 C1(C(N2CC(OC(=O)NC)C2)=O)C(O)CCN1C(=O)CCc1conc1C CCCCCCCCNC(=O)C(N1CC(O)CC1CNC(C1CC1C(N)=O)=O)=O C(=O)(C1=NN(CCO)C(=O)CC1)NC(C)(C)CNC(=O)C1=CCSC1 C1(CC)CCCC2(CCN(C(c3cnn(CCC(C)C)c3CN(C)C)=O)CC2)O1 C=CCCC(F)(F)C(=O)N(C)CC1CCCN1C(=O)C=CSC c1(C(=O)NC2(CNC(c3c(C)coc3)=O)CCC2)oc2c(C)ccc(C)c2c1C N1(C(C(CCOC)C)=O)CC(C(=O)NC(C)CC(C)(C)CO)CC1(C)C C1(C(=O)NCC2(C)CC(NC(C3C(C)(C)OC3(C)C)=O)C2)CC(C2CCCC2)C1 c1(C(C)NC(c2n(CCCCCC)nnn2)c2cnc(Cl)s2)c(F)cccc1F N1(C(C2(C(C)C)CC2)=O)CCCCC(CNC(=O)C(c2ccc(Cl)c(Cl)c2)C)C1 CCCC(C)(C)C(=O)N1CCC(CN(C(=O)C(C)(O)c2ccccn2)C)CC1 C1(C(=O)NC2CC(C(=O)NCCNC(C(C)C)=O)CC2O)CC12CCOCC2 C1(NC(=O)CN(C(=O)Cc2ccc(O)cn2)C2CC2)CCOC12CCOC2 c1(C(=O)NCC2C(NC(c3cncc(OC(C)C)c3)=O)C2)ccnn2ccnc12 C1(F)(C(=O)OCC)CN(C(=O)Cc2cc(C(F)(F)F)cc(F)c2)CC12CNC2 NS(=O)(=O)C1(C(C(=O)Nc2ccccc2)N(C2CCC2)C2CCC2)CC1 c1(C(c2nnnn2CCSC)NC(C=C)(C)CC)ncn2ccccc12 C1(O)(CC#C)CC(C(=O)NC)C1.N1(C(CNC(C)=O)=O)CCC(OCC=O)C1 c1(OC)cc(F)c(F)cc1C(N1CCC(NC(C2OCCC2C)=O)CC1)=O c1(NC(N2C(CNS(N)(=O)=O)CCCC2)=O)cnc2c(c1)CNC2=O c1(CC(=O)NCC2CCC(NC(CC(=O)OCC)=O)C2)ccc(C)nc1Cl c1(COC)c(C(N2CC(F)CC2CNC(=O)C=CCOC(C)(C)C)=O)cnn1C N1(C(C2(C)CCC2)=O)CC2CCC(NC(C3(C(F)(F)F)CCCC3)=O)CC2C1 C(C(=O)NCC1(F)CN(C(=O)CCC2CCCCN2C)C1)(C(C)(C)C)SC C(C(CCC)C(=O)N1CC(C)(C)C1C(C)C)NC(C(CCC)O)=O N1(CC(=O)NC(CNC(C(C)OCC#C)=O)(C)CO)C(=O)CCC1=O Cc1nc(O)ccc1C(=O)NCCCCC1CCCN(C(c2cn[nH]c2)=O)C1 C1(=O)C2=CCCN(C2)C(=O)C2CC(C2)N1.Cc1cc(CC2CC2)cc(Cl)c1 C1(CC)CN(C(c2ccn(C(F)F)n2)=O)CCC1NC(C1(c2ncco2)CC1)=O Cc1ccccc1N1CCC(NCC2(N)CC3CC3C2)C1=O c1(C(N2CCC(C)(CNC(C3ON=C(CC)C3)=O)CC2)=O)ccc2sccc2c1 C1(OC)CCC(NCCC(=O)N2CC(NC(=O)C(F)(F)c3cccnc3)C2)C1 CC1(C)CN(C(c2ccccc2OC(F)F)=O)CCC1NC(C1CCC(F)C1)=O CC1CCCC=C1C(=O)N1CC(O)CC1CNC(c1ccc(Br)cn1)=O C=CC1CN(C(=O)C(CC)CC)CC1NC(=O)CNC(c1ccc([N+](=O)[O-])o1)=O CCC(C)CC(C)C(=O)N(C)CC1COCCN1C(=O)CCc1ccncc1 O(NC(=O)C(CNC(=O)Cc1ccon1)CC(C)C)CCCN(C)C N1(CC(N2C(CNC(c3cccn3C)=O)CC(OC)C2)=O)C(=O)CC(C)(C)C1=O c1(C(c2n(C(CC)C)nnn2)NC2(CCOC)CCCC2)noc2c1CCC2 N1(CCC(=O)NCC(=O)N(CC#N)CC#N)CCOCC1 Cc1noc(Cl)c1CCC(=O)NCC1CCCN1C(=O)CCc1ccncc1 C(C)(C(=O)NC(C(=O)NCC1(C(F)(F)F)CC1)C1CCCC1)OC(C)=O C1(CCNC(C(n2c(C)ccn2)C)=O)CN(C(c2csc(F)c2)=O)CC1C c1(CCOC)sc(C(=O)NC2CC(F)(CNC(=O)CCc3cnc[nH]3)C2)cc1C N1(C(Cc2ccc(C)o2)=O)CCC(C)(C)CC1C(=O)NC(c1cscn1)CO C=CCC(O)(CC=C)C(C)NC(=O)Nc1ccccc1CNC(C)=O CCCCS(=O)(=O)CC(=O)NC(CNC(c1cnc(C(N)=O)cn1)=O)CCOC c1(OC)cc(Br)c(F)cc1S(=O)(=O)Nc1ccc(F)c(CCC(=O)O)c1 C(CCCCCN=c1ccnc[nH]1)NC(c1c(C)nc(CO)o1)=O c1(C(=O)NC2C(C)CN(C(C3CCC3)=O)C2)ccc(-n2cncn2)c(F)c1 C(=O)(C(CCC)C(C)C)N(CC(=O)NC(CC#C)CCOC)CCOC Cc1cc(C#N)cnc1C(N1CCCC1(C)C(=O)NC(C1CCCCC1)C)=O C1(C(=O)NC2C3CN(C(=O)CCSC(F)(F)F)CC23)CCC2(CCC2)C1 C(=O)(C(=O)C(C)(C)C)N(CCC(=O)N(C)Cc1c[nH]nc1C)CC#C CC(C)(C)C(=O)CCC(=O)NC(C)(CO)C(=O)NCCC1(C)CC1(F)F c1(C(=O)NC23C(CN(C(COc4cccc(C)c4)=O)C2)C3)cscc1S(C)(=O)=O C12(NC(=O)COc3ccc(F)cn3)CCCCC1N(C(c1ccc(Cl)s1)=O)CC2 N1(C(C=CC)=O)CCN(C(c2cc(C)co2)=O)CC1C1CCCC1 c1(OC)ccccc1-n1nc(Cc2ccccc2)nc1-c1ccc(C)n1C c1(CNC(C23C(CN(C(=O)CSC4CC4)C2)C3)=O)nc2ccccc2s1 C(=O)(CCS(=O)(=O)CC(C)C)NC1C(C)(CNC(c2cccc(C)n2)=O)CCC1 C1(O)(CNC(C(CC)C)=O)CCCN(C(=O)CC2(N3CCCC3)CC2)CC1 CCC(CCC(=O)N1CC(=O)NCC1C(C)C)NC(=O)C1=CCSC1 c1(OC(C)=O)cc2c(cc1Br)C(NCc1ccc(C)c(S(N)(=O)=O)c1)CC2 N1(C(C(C=CCCC)O)=O)C2CCC1CN(C(c1cc(O)c(F)cc1N)=O)C2 C(C(=O)NCCOCCNC(c1ccnnc1O)=O)(C(C)(C)C)OC Cc1cc(Cl)c(C(=O)NCC2CCC(C)CN2C(c2cnsc2)=O)cc1F CCC(CC(=O)N1CCC(C(N2CCC23CCCC3)=O)C12CC2)C(C)C c1(OC)c(C(N2CCC23CN(C(C2CCC(C)C2)=O)C3)=O)cnc2ccccc12 c1(SCC(=O)NC(C2N(C(C(CC)NC(C)=O)=O)CCC2)C)cccc(OC)c1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CC2CN(C(C3CC(C)(C(=O)OC)C3)=O)CC2C1 c1(CC(N2C3CN(C(CCCCOC)=O)CC2C3)=O)c(C)nc2ncnn2c1C N1(C(c2c(CC)ncnc2)=O)CCC(O)C(NC(=O)C(C)C2CCCC2)C1 c1(C(N2CCC(CCNC(CCC(C)C)=O)CC2C)=O)cnc2n1CCOC2 c1(C(C(N2CCCC(Nc3cc(Cl)ncn3)CC2)=O)O)ccc(F)c(F)c1 C(c1ccsc1Br)=CC(=O)N(CC(C)NC(CCCOC(C)C)=O)C O=C(CC1=Cc2ccccc2C1)NC(CNC(c1cc2ccccn2n1)=O)CO c1(C(=O)NCC(C2CC2)NC(=O)CCCN2CCCCC2)cnc2c(c1)CCC2 CCC(C)CCCC(=O)NC(C(=O)NCc1cc(C)ncn1)C1CCC1 c1(-c2n(C(C)C3CC3)nc(-c3ccnn3C)n2)ccc2c(C)ccnc2c1 c1(C(N(C2CCN(C(c3ncc(CC)nc3)=O)C2)C)=O)cnc2cc(C)ccn12 c1(-c2cn(CC3CN(C(c4cc(C(F)(F)F)co4)=O)C3)nn2)cnc(Cl)c(Cl)c1 N=c1ncc(C(=O)NCC2(O)CN(C(C3CCCC(O)C3)=O)C2)c[nH]1 c1(C(=O)NCC23N(C(c4csc(C)c4N)=O)CCC2CC3)cc2cccnn2c1 C1(COC2CCN(C(C3N(C)CSC3)=O)C2)CCN(C(C2(F)CC2)=O)CC1 C(=O)(CCC(C)S(C)(=O)=O)NC1C2(CN(C(CC(C=C)(C)C)=O)C2)CC1 CC(C)C(CC(=O)NCC(C)(C)C(C)O)NC(=O)CC1CCC(=O)N1C C(c1ccc(C)cc1)=CCC(N1CC(SC)C(NC(=O)CN(C)C)C1)=O C#Cc1cn(C)nc1C(=O)NCC1CC1NC(C1(N(C)C)CCCSC1)=O Cc1sccc1CC(N1CC(OCCNC(C2CCCC2C)=O)C1)=O C1(C(N(C)CCNC(=O)CC2(O)CCOC2)=O)CCN(c2cc(O)ncn2)CC1 C(=O)(CC(C)(C)C#N)NCC(CN(C(C1CCC(C2CC2)C1)=O)CC)(C)C N1(C(C2=COCC(CC)=N2)=O)CCCC2(CCCCC2NC(c2ccc[nH]2)=O)C1 c1(N(C(C2(F)CCN(C(C3CCCCN3)=O)C2)=O)CCO)cc(Cl)ccc1Cl CN1CCC(n2nccc2-c2ccc(N)cn2)CC1.N12CCC(C1)CC2=O c1(OC)nc(Cl)ccc1C(=O)NC1C2CC1N(C(=O)CSCCC(F)(F)F)C2 CC(C)(C)CCC(=O)NC1CCCC(NC(=O)C(c2ccccc2F)O)C1 c1(C(=O)NCC(C)(C)CC2CN(C(=O)CC3CCC3)C2)ncnc2c1OCCO2 N1(C(CNS(CC)(=O)=O)=O)CCCC(C)(C)C1CNC(C1CCCCC1(C)C)=O C1(C(CNC(C(CC)C)=O)O)CCN(C(c2cncn2C2CC2)=O)CC1 C1(CCC)CN(C(=O)C(O)CC(F)F)CCN1C(=O)C(F)CC N1(C(C2CC(=O)C2)=O)CC(C(=O)NC2CC3(C2)CC(O)C3)C(F)(F)C1 C(=O)(C(CC)C(C)OC(c1ccccc1-c1ccccc1)=O)OCC c1(C(N2CC(C)C(CNC(c3[nH][nH]c(=N)c3Br)=O)C2)=O)cnc2n1CCOC2 C(=O)(C1=CCCN(C(c2cn3c(n2)CCC3)=O)C1)NC1CC(C)(C)OCC1 C12(C(=O)NCCOC3CCN(C(Cn4ccc(C)n4)=O)C3)CCC(CC1)C2(C)C C12(CNC(C3CC4(CC(=C)C4)C3)=O)CCCC1N(C(=O)CCC#N)CCC2 c1(C(N(CCn2cc(CSC)nn2)CC)=O)cc2ccc(OC(F)(F)F)cc2[nH]1 C(CSC)(C(=O)N1CC(F)(C(=O)NC(CC2CC2)CO)C1)OC c1(CNC(C2(F)CCCN(C(C3CC4CCC4C3)=O)C2)=O)cc(F)cc(F)c1 N1(C(c2ccn(CC)c2C)=O)CCN2C(=O)C(NC(c3cc(C)c[nH]3)=O)CC2C1 C(N(C)N1CCCN(c2ccncc2)CC1)c1c(CC)onc1C c1(C(=O)NCCN(C(CC2CCC(C(C)C)CC2)=O)C)ccc(F)c(CO)c1 c1(C(N(CCN(C(=O)CSCc2cccs2)CC)CC)=O)n[nH]c2c1CSCC2 c1(C(N2C(CN(C(C(COCC)(C)C)=O)C)COCC2)=O)c(F)cc(C)cc1F c1(OC)ncc(CN2CC(OC)CC2C(N2CC3CC2CO3)=O)cn1 C(=O)(C(O)CC(N)=O)NCC1(NC(c2nc(C)nn2C)=O)CCCC1 c1(C(C)NCCc2nc(C(C)C)sc2)cc2n(n1)CCCC2 n1(CCCOC)ccnc1CN(C(C1CCC(C)C1)C(=O)NCC(F)F)C c1(C(=O)NCCCCNC(=O)C(O)CF)ccc2c(c1)OCC2 C#CCCCCC(=O)NCCCNC(c1cc(C2CCC2)no1)=O c1(C(N2CC(CCC#C)C2)=O)ccnc(CNC(c2ccnc(CC)c2)=O)c1 C(=O)(C#CC1CCC2(CC1)OCCO2)N1CCC(O)(C(C)NC(C(C)C)=O)C1 C1(C(=O)OC)CSCCN1C(c1cccc(CSc2ccccc2)c1)=O CC(C)C(C(=O)NCCCCCNC(c1ccnnc1S)=O)NC(N)=O C(C(C)(C)CN(C)CC)NC(CCN(C(=O)CC1CC=CCC1)CC)=O N1(C(C2(COC)CCC2)=O)CCC(CN(C(=O)C(C)CF)C)CC1 C1(CNC(CC2CC(=C)C2)=O)CC(F)(F)CN1C(=O)Cc1ncc(F)cc1F CCCCCCCC(=O)N1CCCC1(C)CNC(=O)Cn1ncnn1 n1(CCCC)ncc(C(N2CCCC2CCCNC(C2(C)C=CCC2)=O)=O)c1C CN1CCC(F)(CNC(C2CN(C(c3c[nH]cc3C3CC3)=O)CCO2)=O)C1 c1(C(=O)OC)cc(C(N2CC(NC(c3cn[nH]c3)=O)C(O)C2)=O)ccn1 C1(O)(CC)CN(C(=O)C(CC2CCCC2)NC(=O)Cc2ccc[nH]2)C1 N1(CC(=O)N(c2cccc(Cl)c2)C)CCC(C2CCCN(C(c3csnn3)=O)C2)C1 C1(C(=O)NC(C(=O)NC(c2onc(C)n2)C)COC(C)C)CC(=O)CCO1 C1(COC)(CNC(=O)CCc2ccn(C)n2)CN(C(=O)Cc2cn(C)nn2)C1 C1(C(N(C2CCN(C(=O)C=CBr)C2)C)=O)CC(O)CN1CC(F)(F)F c1(C=O)cnn2c1CN(C)CC2.c1(C(=O)NCCN(CC)CC)cccc(CO)c1 C1(C(=O)OC)CCOC1C(=O)NC1CCN(CCOC)C1 n1(CC)ccc(C(=O)NC(C(=O)NCC(C)C(F)F)C2(O)CCC2)c1C c1(C(=O)NC(C(CO)NC(Cc2ncc(C)o2)=O)C)c[nH]c2cccc(Cl)c12 N1(C(C(C)SCCCC)=O)CC(CC(=O)NCc2snnc2C)C(C)C1 c1(C(N(CCCN(C)NC(=O)CCOCC(F)F)C)=O)coc(C(F)F)n1 N1(C(c2ccsc2C(F)(F)F)=O)CCCC1C1CCCN1C(c1cnns1)=O C(=O)(CC(C)(C)CC(F)F)NC1C=CCN(C(c2cc(C)nn2C2CCC2)=O)C1 C(=O)(C1=CCCCCC1)NCC(c1ccccc1)N(C)C(C1CCCC1CF)=O c1(C(=O)Nc2nnc(C)o2)ccc(-c2csc(-c3nc[nH]n3)c2)cc1 CC1(CNC(=O)C(F)(F)c2ncccn2)CC(NC(C2CCCCS2)=O)C1 N1(C(CS(=O)(=O)NCC)=O)CCCC(COC)(NC(=O)CC2C=CCC2)C1 C1(NC(c2cc(CC)no2)=O)CN(C(C2CC3(CC3)CO2)=O)CC1C n1(C(C)(C)C)cc(CNC(c2cnn3c2OCC3)=O)c(O)nc1=O C(C)(C)(CCC(=O)NCCC(O)CNC(C1C2CCCCCC12)=O)N(C)C N1(C(C=C(CCC)C)=O)CC(C(=O)NCCC(=O)N(C)C2CC2)C(F)(F)C1 C1(C(=O)NC2CCC(COC)CC2)CCC(C)NC1=O.C12(CC1)C(=O)NC2 CC1CC(N(C(=O)C(c2ccccc2)C2CCCCC2)C)CC(C)C1 c1(OC)ccn2c(C(=O)NCCC3(NC(c4cnco4)=O)CC3)cnc2c1 c1(CC)nc2c(C(N3CCCC3CNC(C3CCCS3)=O)=O)ccnc2[nH]1 C1(NC(C(c2ccc(OC)cc2)CC)=O)CCN(C(=O)CCCC2CC2)CC1O c1(C(=O)NC2CCC3C(C(=O)O)C32)ccc2nncn2c1 N1(C(c2cc(C)no2)=O)CCCC(CC(=O)NC2CC2c2ccccc2)CC1 CC(C)(C)C(C)(O)C(=O)NCC1(NC(C2CC(n3cnnc3)C2)=O)CC1 CC(C)CC(O)C(=O)NC1(CCCNC(=O)C(c2c(Cl)cccc2Cl)C)CC1 c1(C(N(CC(C)NC(C2(O)CCSC2)=O)C)=O)nnn(C)n1 CCC(C)(CCNC(=O)CC1CCCS1)NC(c1ccsn1)=O c1(C(=O)NC2CC(NC(C3CCOC3c3cn[nH]c3)=O)C2)cccc(C(F)F)c1 CCC(C(=O)N1CC(CCNC(C2CCCSC2)=O)C1)n1ccc(C2CC2)n1 c1(-c2nn(-c3c(C)cccc3)c(C3CCOCC3C)n2)ccc2ccccc2c1 c1(-c2cn(CC(C)(C)CCC(c3cc(C(F)(F)F)co3)=O)nn2)cccc(Cl)c1 c1(OCc2nnc(COC)s2)cc(N2CCCCC2)cc(Cl)c1 c1(SC(C(=O)NCC(=O)Nc2cccc(F)c2)(F)F)ccc(Br)cc1 c1(CCC)nc(=NC2CCN(C(=O)CN3CC(=O)NC3=O)C(C)C2)s[nH]1 C1(NC(C(CC)NC=O)=O)CCC(NC(=O)CSC2CC2)CC1 N1(C(Cc2[nH]c(=N)sc2)=O)CCOC(CNC(C2CCCC2(F)F)=O)C1 C1(CNC(C(CNC(CCC)=O)OC)=O)CCCCC1CC C(CCCc1ccccc1)(C(=O)OC)NC1(CCOC)CC1 C1(C(N2CC(c3nc(C)no3)C2)=O)(CNC(c2cnc(SC)s2)=O)CC12CCC2 C(=O)(C1=CCCCO1)NC(C(=O)NC(c1ccccc1)CC)CCC1CCC1 C1(NC(=O)OC)CCCN(C(C(=O)Nc2ccc(OC)cc2)C2CC=CC2)C1 c1(C(N(CC(C)NC(=O)Cn2nccc2C)CC)=O)ccc(C)c2ccccc12 C1(C(=O)O)CCN(C(c2nc(C3CC3)cs2)=O)CC1.N12CCC(C1)C2 C(=O)(C1Cc2ccccc21)N(C1CCN(C(COCCOCC)=O)CC12CC2)C N1(CC(=O)NCCC2(O)CCCN(C(CCC#CC)=O)C2)CCc2sccc2C1 Cc1nn(C(C)C)c(NCC2(F)CC(NC(C3CC(=O)N3)=O)C2)c1[N+](=O)[O-] c1(SCC(=O)N(CC(C)N(C(=O)CCc2cnn[nH]2)C)C)ccc(C(C)C)cc1 c1(C(N2C(C(=O)NCC3N(CC)CC3)C=CC2)=O)ncnc(O)c1F n1(CCC(C)C)c(C2(CN(C34CCCCC3C4)C=O)CC2)nc2ccccc12 N1(C(c2cc(OCC)n[nH]2)=O)CCC(O)(CCNC(C2(C(N)=O)CCC2)=O)CC1 N1(C(C2(Cc3ccccc3)CCOC2)=O)CCC2(CC=CCO2)CC1 c1(NC(c2c(F)cc(Br)cc2F)c2n(CCC)nnn2)ccc2nn[nH]c2c1 c1(C(C2CN(C(CC)=O)C2)C)cn(Cc2conc2C(C)(C)C)nn1 CCC(C(=O)N1CCN(C(=O)C=Cc2cn(C)nn2)C(CO)C1)C(C)(F)F Cc1cc2cc(C(=O)NCC(C)NC(=O)CC3(O)CCCOC3)c(Cl)cc2[nH]1 Cc1cccc(C(N2C(C(=O)O)CCC2(C)C)=O)c1[N+](=O)[O-] C(=O)(C(C)CCC(C)(C)C)NCC1(OC)CN(C(=O)CNC(=O)C(F)(F)F)C1 c1(NC(CC(N2CCCC23COC3)=O)c2ccccc2)ccc(I)c(F)c1 c1(CC(=O)NC(CCCNC(c2n(C(C)C)ncn2)=O)C)ccccc1O N1(C(C2CCN(C(C3CCC(C)O3)=O)CC2)=O)CCN(C)C(c2cccs2)C1 c1(C(=O)NCC(CNC(c2[nH]cc(C(=O)OC)c2)=O)OC)ncn2c1CCCC2 c1(N2C(CCCNC(c3c(CC)ncs3)=O)CCC2)ncnc2c(Br)cccc12 N1(C(CC(C(CC)C)NC(=O)C(C)N=[N+]=[N-])=O)CCN2C(=O)CCC2C1 N1(C(COCC(=O)OC)=O)CCC(C)(NC(=O)C(N2CCSCC2)C)C1 C(C(C=O)n1cc(COCCO)nn1)O.N1(CC)CCC(Cn2cccn2)C1 C1(C(N2C(C)CN(C(C3(C)CCCCC3C)=O)CC2)=O)CCC2(C1)CC2(F)F c1(C(=O)NC2CC2C(=O)NC2(CN3CCCC3)CC2)cncc(N2CCCC2)c1 CS(=O)(=O)CCC(=O)NC12CCC(CNC(=O)CC3CCCCC3O)(C1)OC2 C1(C(N(CCCC(=O)NCC(=C)Cl)C)=O)C(C)(C)C1(F)F c1(C(N2CCCC(O)(CNC(Cn3c(C)cnc3)=O)C2)=O)ncnc2sccc12 c1(CC)ccc(CC(=O)N(C2CCCN(C(C3CCCO3)=O)C2)CCO)cc1F C1(C(=O)NC(CC)CO)CC(F)(F)CN1C(c1ccnc(C)n1)=O C1(CC(=O)NC(C(=O)N(CCC=C)CC)C2CCC2)CC(C)(C)CO1 Cc1ccc(C=CC(=O)NC(CNC(C2CCC(CO)CC2)=O)C2CCC2)nc1 Cn1cc(C(=O)N(CCC(C(C)(C)C)NC(=O)C=CC=C(Cl)Cl)C)n(C)c1=O C(=O)(C(CO)C(F)(F)F)NC(c1c(C(N(C(C)C)CCN(C)C)=O)con1)C N1(Cc2c(C)coc2C#N)CCCN(CCn2ccc(O)nc2=O)C(C)C1 c1(C(N(C)CC2CCCCN2C(c2cn[nH]c2)=O)=O)cc(F)c(F)cc1O C1(C(N2CCN(CCC#C)CC2)=O)CCCCCN1C(=O)C(C1CC1)OC N1(C(CNS(CCCC)(=O)=O)=O)CC2(CCN(C(c3ccccc3OC)=O)C2)C1 C1(C(=O)NCc2cc(CC)no2)CN(C(c2cc[nH]c2C2CC2)=O)CC(C)(C)C1 O(NC(=O)CCCCC(C)C)C(C(=O)NCC(COC)(F)F)CC(C)C c1(CN2CCC(C)(NC(c3c(C)cccc3)=O)C2)cccc2[nH]ncc12 C1(C(=O)NCC(CNC(C=Cc2cn(C)nn2)=O)(C)C)CC2(C1)CC(O)C2 c1(COC(c2ccc(C(=O)OC)nc2F)=O)coc(S(N)(=O)=O)c1 c1(C(=O)NCCCOCCNC(c2cnc(C)s2)=O)cc(Cl)c(Cl)n1C Cc1cc(CC(N2CC3CC(NC(C4C(F)(F)C45CCC5)=O)C2C3)=O)cc(F)c1 C(=O)(C1COc2ccccc21)NC1CCCC(NC(c2cc(C)nc(O)c2)=O)C1 C(=O)(NNc1c(O)cccc1F)c1n(C)c(=O)n(CC(F)(F)F)c1 N1(C(c2noc(C)c2C)=O)CC2CCN(C(c3cncc(F)c3)=O)CC2C1 C(=O)(CCCC(N)=O)NCC1N(C(C2CCC(C)(CC)O2)=O)CC(F)C1 N1(C(C2(C(=O)OC(C)(C)C)C(C)C2)=O)CC2(CCCC2NC(=O)CCF)C1 C(=O)(CC(F)(F)C(C)C)N1CCC(C)(CNC(C=Cc2c(C)noc2C)=O)C1 CCCC(C(O)C(=O)NCCCC(C)CO)NC(c1cccnc1)=O c1(NC(C)CC(C)NC(c2cccn2C2CCCC2)=O)cc(-n2ccnc2)ncn1 CC1(C)OCCC1C(N1CC2C(C(=O)NCCNS(C)(=O)=O)C2C1)=O C(=O)(C1=CCCCC1C)NCC(CCC)C(=O)NCCC#CCO c1(OCCOC)ncc(C(N2CC(N(C(=O)COC)C)C2)=O)cn1 C1(C(=O)NC(C(=O)OCC)C)CC2(CCN1C(=O)OC(C)(C)C)CC2 c1(CC)ocnc1C(=O)NCCCC(C)NC(=O)CCC=CC(C)C C=CCC(CC(C)C)C(=O)NCCCCCC(=O)N(CCO)CCO CCCCC(CC(=O)NCCCC(C)(C)OC)NC(=O)C1=NOCC1 C1(C)(C(=O)NCCC(CCC)C)CCN(C(=O)CC(C)COC)CC1 C12(C(=O)NCCOCCCNC(c3occ(C)c3)=O)CCC(CC1O)C2 Cc1cc(CNC2CCC(C(=O)NCCc3ccc(Br)cc3)C2)c(C)cc1O C1(OC)CN(C(=O)CC2(C(=O)Nc3cccc(C(=O)OCC)c3)CC2)CC12CC2 N1(CCN(C)C(C2CCC(CO)CC2)=O)CCN(C(=O)CP(C)(C)=O)CC1 Cc1ccc(NC(c2ccc(NC(C34CCCC3C4)=O)nc2)=O)cc1F C#CCCCCCC(=O)N1CC(NC(C2(C)CCN(C)C2)=O)CC12CCC2 c1(CC)cc(F)ccc1C(=O)NCC1CCN1C(=O)CNC(C1CCCC1)=O N1(C(C2N(N=O)CCC2)=O)CC2CC(C1)CN(C(=O)CCc1ccco1)C2 C(c1cccc(Cl)c1)=CC(=O)NC1C2CN(C(c3n(C=C)nnc3)=O)C1C2 C1(C(=O)NC(C2N(C(CCC(C)(F)F)=O)CCC2)(C)C)CC2COCC(C1)C2 c1(OCC)ccc(Br)c(CNc2ccc(-c3cc(CO)cc(F)c3)nc2)c1 Cc1ccc(OC(F)(F)F)c(C(=O)NC2COCC2NC(c2ccc(Br)o2)=O)c1 c1(C(=O)NC(CNC(C(CC)(C)C)=O)C(C)C(C)C)cncc2c1CCNC2=O C(=O)(CCCC(F)(F)CO)N1C(CN(C(CCC(CC)OC)=O)C)CCCC1 Cc1cc(F)ncc1CN1CC2C(C(=O)Nc3ccc(Br)c(F)c3)C2C1 c1(C(N2C(C(C)NC(C3(COC)CC(=C)C3)=O)CCC2)=O)ncc(C)cc1C c1(CC(=O)NC(C(C)NC(CN(CCC)C)=O)C(C)C)ccc(F)c(OC)c1 CC1OC2CCC1(NC(=O)C=CCC(C)(C)NC(=O)CCCCC1CC1)C2 C#Cc1ccc(C(=O)NC2CC(OCC(=O)NCC3=CCCOC3)C2)c(C)c1 C1(CNC(c2c(N)c(Cl)ncc2)=O)CC2CCC1N(C(C1(F)CCOC1)=O)C2 N1(C(C2(CCOC)CC2)=O)C2CCC1C(CNC(c1scnc1Cl)=O)C2 CS(=O)(=O)c1cc(N2CCN(C(C3CCC=CCCC3)=O)CC(O)C2)ncn1 c1(C(N2CCC(CNC(C3C4CC5C(C4=O)C35)=O)CC2)=O)cc(F)cc(F)c1 Cc1cccc2c(=O)c(C(N3CCCC(CO)(NC(=O)CC(C)F)C3)=O)c[nH]c12 C1(NC(c2ccc(F)o2)=O)CN(C(=O)CCCc2cnn[nH]2)CC2(CC2)C1 n1(CC(=O)N(CCC(C)NC(C2CCC(NC(N)=O)CC2)=O)C)cnc(C#N)n1 N1(CC(=O)O)CC2(CCN(CC3CCCN3C3CCCCC3)CC2)OC1=O Cc1cc(F)ccc1C(=O)NCC1COCCN1C(C1CCNC(=O)C1)=O CCC(C)C(CNC(=O)CC(O)CNC(=O)CC(C)c1ccco1)CO C=CC(C)CC(=O)NCC(c1cccc(OC)c1)NC(=O)C1=CSCS1 C1(C(N(C(C)CCNC(=O)CCCCCNC(N)=O)C)=O)CS(=O)(=O)CC(=O)N1 Cn1c(C(N2CCC(CCNC(=O)CC(C)(C)C3CC3)CC2)=O)nnc1S CC(C)CC(=O)C(=O)NCC(=O)NCC(=O)NC1CCC(O)CC1 Cn1c(C(N2CC(F)(F)CC2CCNC(=O)CC2CC23CC3)=O)cccc1=O c1(C(C(=O)NC)N(CCC)CCOC)n[nH]c2cc(OC)c(OC)cc12 N1(C(C(CC)=CC)=O)CCCC(O)(CNC(c2cnn3c2CCC3)=O)CC1 C1(C(NOCc2cccc(C)n2)=O)CCCCCN1C(C1CN(C)C1)=O c1(C(N(CCNC(c2cncc(C)c2)=O)C)=O)c(C)nc2sc(C)nn12 C1(NC(NC(c2ccccc2)C)=S)CCC(c2ccccc2)C1 c1(NC(CC2(NCc3ccc(SC)s3)CCC2)=O)ccc(C)nc1N1CCCC1 N1(C(c2c(CNC(c3c(C)nc(CC)o3)=O)nnn2C)=O)CCC(C)CC1CC C1(C(=O)NCc2c(C(=O)NC(C)CC3CCOC3)n(C)nc2)CC(=O)OC1(C)C Cc1nn(C)cc1CNC(=O)C(c1ccco1)NC(=O)CC1CCOC1=O CC(F)(F)C(F)C(=O)NCC1CCN(C(=O)C(C)(O)C2CCC2)CC1 N1(C(c2c(COC)cco2)=O)CCN(C(=O)CC2CCC(OC)CC2)CC(O)C1 C(c1ccc(C(N)=O)cc1)=CC(=O)NC(C1CN(C(C2(C)ON=C(C)C2)=O)C1)C c1(C(=O)NCC2C(NC(C(C)O)=O)CC2)cc2c(s1)CC(C)(C)C2 N1(C(C2CC(=C)C2)=O)CCC(n2cc(CNC(C3CC(C)=NO3)=O)nn2)C1 CC(C)(CCCNC(c1coc2c1COC2)=O)C(=O)NCC(C)(O)C1CCC1 N1(C(c2c(SC)ccc(N)c2)=O)CC2(CCN(C(c3cc(Br)n[nH]3)=O)C2)C1 C1(CN(C(C(N2CCOCC2)C)=O)C)COCCN1C(C1CCCN1C1CC1)=O C1(C#CC(=O)N2CCC(CCN(C(=O)CC(C)OC)C)CC2)(CC)CC1 c1(C(=O)NCCCC(=O)N(CCC(=O)OC)CCO)ccn2cncc2c1 CC1CN(C(=O)CC2CCN(C(=O)Nc3ccc(Br)cc3Cl)CC2)CC(C)O1 C(=O)(C1=NOC(C2(O)COC2)C1)N1CCC(CCC)C1 N1(C(c2c(C)cco2)=O)CCCCC1CCN(C)C(C1CC(F)(CO)C1)=O N1(C(c2c(C)[nH]cc2)=O)C2CCC1CN(C(c1cnc(C(C)C)n1C)=O)C2 c1(-c2ccc(CN(C)C)cc2)ccn2ncc(C(=O)NCCC(C)(C)O)c2c1 N1(C(C=CCCC)=O)CC2OCC(N(C(C3CCCCC3)=O)CC)C2C1.C1(=O)CN1 CC(C)C(O)CC(=O)N1CCC(NC(=O)CCCc2cccnc2)C1C C(CC(C)(C)CN=C(NCC(F)F)NC(CS(C)(=O)=O)C(C)(C)C)SC CC1(CNC(=O)CC2(NC(=O)C3=CCSC3)CC2)CC=CCC1 c1(N2C(C)C(NC(=O)CCn3cnnn3)CC2)cc2c(cn1)C(=O)CCC2 Cc1c(C(=O)NCC(C)CCOc2cccc(F)c2)ccn1C c1(C(=O)NCC2(C)N(C)CC(OC)C2)cc(C(=O)O)c2n1CCCC2 C(c1cccc(F)c1)=C(C(=O)NCCN(C(c1c(CC)nc[nH]1)=O)C1CC1)F Cc1cnc(Cl)[nH]c1=NC1CCCOC1C1CCN(C(C2(F)CCOC2)=O)CC1 C1(CCCNC(c2n(C)ccc2)=O)CCN(C(=O)CC(O)c2cnc(Cl)s2)CC1 Cc1cncc(C(=O)NCC(C)NC(=O)COc2cncc(Cl)n2)c1Cl C(=O)(C1CCCc2c1ncn2C)N1CC(O)(CNC(c2n(CC)cc(Cl)c2)=O)C1 S(=O)(=O)(CC(=O)NCC1CCN(C(c2ccc(NC(C)=O)s2)=O)C1)NC c1(C(=O)NC(CNC(C2CCN(CC)C2)=O)C(C)C)cncn(C)c1=O N1(C(C(C=C)(C)CC)=O)CC2(CCCCN(C(=O)CC(C3CC3)C3CC3)C2)C1 Cc1nc(CC(=O)NC(C)(CNC(=O)CC(O)C2CCCC2)C2CC2)co1 C1(NC(C2CCCOCC2)=O)CC12CCN(C(=O)C=CC1CCOC1)C2 C1(NC(C2N(C)C(=O)CC2)=O)CN(C(=O)CC2C=CS(=O)(=O)C2)CCC1(C)C N1(C(C(CCC)F)=O)CCN(C(c2nnsc2C)=O)CC(C)C1 C1(C(N2C(CC(=O)NCCN(C)CC)CCCC2)=O)CC2(CCCO2)C1 C1(NC(C(C)N(CCC)C(c2coc(SC)c2)=O)=O)CC(C)N(C)CC1C C1(NC(C)=O)CCN(C(=O)COC2CC(NC(c3ccsc3)=O)C2)C1C N1(C(C2(CC=C)CCC2)=O)CC(C2(NC(c3n[nH]c(C)n3)=O)CC2)C1 C(=O)(C(C)(F)C(F)(F)F)NCCCC(C)NC(=O)Cc1ccccc1Br C1(NC(C2C3CN(C(=O)Cc4cc[nH]c4)CC23)=O)CCCC(C2CC2)C1 n1(C(C)C(=O)N(C2CN(C(=O)COc3cnn(C(C)C)c3)C2)C)cnc(C#N)n1 C1(CNC(CCN(CCC)C)=O)CCCCN1C(=O)C(=Cc1c[nH]cn1)F c1(OC)ccc(O)c(NC(C2(F)CCN(Cc3c(OC)cccc3C)C2)=O)c1 n1(C(CC)CC)nc(C(=O)NCC(C)(C)CCNC(c2cnc(O)s2)=O)cc1C c1(C(N2CC(CC)N(C(=O)C(O)C(C)(C)C)CC2)=O)cc(N(C)C)cc(C#N)c1 N1(C(CC(=O)N(C)C)=O)CC2CCC(C1)N2C(=O)C(F)n1cccn1 C(=O)(C(C)C(C)(F)F)NC1CCN(C(c2n(CC)ccn2)=O)C1C(C)(C)C C(=O)(C(O)CC(N)=O)NC(C(N1CC(C)(COC)C1)=O)(C)c1cccs1 c1(CC(=O)N(CCNC(COCCC=C)=O)C(C)C)cn[nH]c1 C1(OC)CN(C(c2sccc2-c2cn[nH]c2)=O)CC1NC(=O)CCF CC1=C(C(=O)NC(C)C(C)NC(c2c(OC(F)F)cccc2Cl)=O)CCCC1 N1(Cc2n(CCC)nnn2)CC2(CC(NC(c3c(C)nn(C)c3Cl)=O)CO2)C1 c1(C(N(CC(CC)NC(=O)CC2CCS(=O)(=O)C2)CC)=O)cncc2c1CCC2 c1(C(=O)Nc2nc(-c3c(C)ccc(C(F)(F)F)c3)sc2)cc(F)c(Br)cc1F c1(C2C(NC(c3n[nH]c(-c4cccc(C)c4)n3)=O)C2)ccc2c(c1)OCO2 CS(=O)(=O)C1CN(C(=O)CCCCc2cnn[nH]2)CC1NC(c1cc(F)n[nH]1)=O N1(C(C2CN(CC)C(=O)C2)=O)CCC(NC(=O)CSc2nc[nH]n2)C(C(N)=O)C1 c1(C(C)C)ncc(Br)c(C(N2CCN(C(c3cnn4c3CCC4)=O)CC2)=O)n1 N1(C(c2cc(OCC)ns2)=O)CC2=C(C1)CN(C(=O)CCCn1ccnn1)C2 Cc1ccc([N+](=O)[O-])cc1C(c1nnnn1C)NCCOc1cc(C)c(Cl)c(C)c1 c1(OCCCC(=O)Nc2c(CNC(=O)COCCF)ocn2)ccc(F)cc1Cl C(=O)(C1CCCc2cccnc21)N(C1CCN(c2cc(C(N)=O)nc(Cl)n2)C1)C Cc1nc(Cl)ccc1CC(=O)NCC1CN(C(=O)CN2C(=O)CCC2=O)CC1O N#CC1=C(C(=O)N2CC3CCC3(CNC(C3(CF)CCC3)=O)C2)CCC1 Cc1cc(C(=O)NC2CCCC(NC(c3cccc(Br)c3F)=O)C2)cc(C)n1 c1(SC)cc(CNC(C2CCCN2C(=O)CCCCC2CCSS2)=O)ccn1 c1(N(C)C(=O)OC(C)(C)C)ccc(NNC(=O)C2CCC(C#N)C2)cc1 N1(C(C(C)N=[N+]=[N-])=O)CC2CCCC(CNC(c3ccnc4c3CCO4)=O)C2C1 N1(C(CC(CNC(CCCOCCOC)=O)(C)C)=O)CCSC2CCCC12 CC(C)C(C)S(=O)(=O)N=c1cc[nH]c(-c2ccccc2Cl)c1 N1(CC(C)CCCO)CCc2cc(Oc3ccccc3)ccc21 N1(C(CC2(C)CC2(F)Cl)=O)CCN(C(=O)COC2CCOC2)C(C(F)F)C1 Cc1cc(C(N2CC(NC(C3CC4(C3)CC4F)=O)C(n3ccnn3)C2)=O)c(C)o1 C12(NC(C)CSC(F)F)CCOC(C)(C1)C2 O=C1CCc2cccc(C(=O)NCC3CCCN3C(=O)COCC(F)F)c2N1 c1(OC)ccc(C(=O)NCC2CC(NC(C3(OC)CCC3)=O)C2)c(OC)c1 c1(C(=O)NCCC(C)NC(c2cc(CC(C)C)[nH]n2)=O)c(C#N)cnn1C c1(-n2cc(C3CCN(C(c4c(OC(C)(C)C)coc4)=O)C3)nn2)ccc(O)nc1 C1(O)(CNC(c2n[nH]c(=O)cc2)=O)CCCN(C(=O)C(C)C(C)O)CC1.CCOC CN1C(=O)Cc2cc(C(=O)OCC3CCC(F)C3)ccc21 N1(C(c2ncc(C)c(C)c2)=O)CC2CCC(C1)C2CNC(c1cncs1)=O c1(C(N2CC(CCNC(c3c(C)nc(O)cc3)=O)C2)=O)c([N+](=O)[O-])cnn1C C(=O)(C(CC(F)F)NC(=O)CC1CCCC1)NCC1CCN(C)C1 CC(C)CC(C)CC(C)C(=O)NCc1cncc(-c2cn(C3(C(=O)O)CC3)nn2)c1 C=C1CC(C(=O)NCC(CO)OC)(CNC(=O)C(O)CC)C1 c1(CC(=O)NCC(CNC(CCc2onc(C(C)C)n2)=O)C)c(O)ncnc1O CC1CCCC(NC(c2cc(CNC(C3SCCS3)=O)no2)=O)C1 Cc1noc(C)c1CCC(=O)NCC1CC(n2cc(CNC3COC3)nn2)C1 c1(OC)cccc(F)c1CC(=O)N(CC(O)CNC(c1ccc(=O)n(C)c1)=O)C C(=O)(CCC(F)(F)F)NCCN(C1CCCCCC1)C(C1C(C)(CC)C1)=O C1(CN(C(C2CCOC2(C)C)C(=O)NC)C)CCc2nc(C)cn2C1 N1(C(CCCNC(C2CCC(C#N)CC2)=O)=O)C2CCC1CC(CO)C2 C1(C(N(CC(C(=O)OC)C)C)=O)CCN(C(C2CC3CCCC3C2)=O)CC1C C1(C(N(C)Cc2cncn2C)=O)CCC2(CC2)N1C(=O)C#CC1CC1 c1(NC(C2N(C(Cc3n4cc(C)nc4sc3)=O)CC2)=O)cnc2c(ccn2C)c1 CCCCCCC(=O)N(C)CC1CCN(C(c2cnc(C(C)=O)s2)=O)C1 C12(CNC(c3csc(C(F)(F)F)n3)=O)CC1CN(C(=O)COC1CCCCC1)C2 Cc1ccc(C(N2CC3CC(NC(c4sc(O)nc4C)=O)C2C3)=O)cc1C#N C(CC(C(=O)NCC(O)C(N)=O)NC(C1CC(O)C1)=O)=CC c1(CC)c(C(=O)NC2CC2CNC(=O)CCCn2ccnn2)cnn1CC S(=O)(=O)(c1c[nH]c2nc(F)ccc12)N1C2(CCCS(=O)(=O)C2)CC1 C1(NC(c2cc(Cl)on2)=O)CN(C(=O)CCSc2ccccn2)CCC12CCC2 c1(C(c2n(CC)nnn2)(COC)NCC2(CC)CCOC2)ncc(F)cc1F Cc1cccnc1CCCN(C1CCCC(N(C)C)C1)C C#Cc1cc(C(N2CC(NC(=O)CN(C)C(C)C)C(C=C)C2)=O)cc(Br)c1 N1(C(C2C(=C)C2)=O)CC2CC2(CNC(c2c(-c3ccccc3)noc2CC)=O)C1 Cc1ccccc1C=CC(=O)NCC(C)C(=O)N1CCCC1C(C)(C)C C(=O)(C(CC(C)C)N(C(=O)NCCOC(F)F)C)NCC1(CC=C)CC1 c1(C(=O)OC)nc(C(=O)NCC2CC2NC(=O)Cc2csc(C)n2)cs1 c1(C(=O)NCC2(CN(C(CC=CCC)=O)C)CC2)ccc(F)cc1Br C1(OC)CCC(C)(C(=O)NCCC2(O)CN(C(c3sccc3C)=O)C2)CC1 Cc1ccc(-n2ccnc2)c(C(=O)OCC(=O)NCCC2CC(=O)N(C)C2)c1 C(C1=NOC2CC12)(c1nnnn1Cc1cccc(OC)c1)NCCCC(=O)OCC CC(C)(C)C(C)(C)C(=O)N1CCCC(NC(=O)CN2CCCNC2=O)C1 Cn1ccc2cc(NC(=O)NCC(c3ccc(O)cc3)O)ccc2c1=O CC1(C)CN(C(=O)C=CC(=O)NC2CC2)CCC1CO.C12(CC1)C(=O)NCC2 N1(C(CCCc2ncc(C)o2)=O)CC(NC(c2sccc2C(C)C)=O)CC(C)C1 C#Cc1ccc(F)c(C(=O)NC(C2CN(C(c3cncc4nc[nH]c34)=O)C2)C)c1 C=CCC(CNC(=O)CNc1ccccn1)C(=O)N(CCCCC)CCO N1(C(c2c(Br)ccc(=N)[nH]2)=O)CCC(C2CN(C(=O)C3=NNC(=O)CC3)C2)C1 C#CCCCC(=O)NCC(C)(O)C(=O)N(C)C c1(C(=O)NC2(CC=C)CCN(C(C3CC(C)(O)C3)=O)C2)ccc(OCC)cc1Cl c1(C(=O)NC2C(NC(CCCOC)=O)CS(=O)(=O)C2)nn(C)c2c1CCCC2 C1(C)(CNC(CC2(OCC)CC2)=O)CCN(C(c2nocc2C2CC2)=O)C1 C(=O)(C1c2c[nH]nc2CN1C(=O)CN1CC(C)(OC)C1)N1CC2C(CC)(C2)C1 C(CCCOC)(C(=O)N(Cc1ccc(C)o1)NC=O)OCC C(=O)(C(C(C)C)C(C)C)N1CC(C)(C(N2CC(C)CC(OC)C2)=O)C1 O=C(CCC(=O)c1ccncc1)NC1CC(NC(=O)Cn2nccn2)C(O)C1 CC(C)CC(C)CN=c1nc(N(CCC(F)(F)F)C)c2c([nH]1)COC2 CCC(CNC(=O)Nc1cccnc1-n1ccnc1)C(C)C n1(C(C)C)cc(C(=O)NCC(C)(C2CCC2)NC(c2cnc(C(N)=O)s2)=O)nn1 Cc1ccccc1CCC(=O)NCC1(C(C)(C)O)CN(C(=O)C(F)F)C1 N1(C(CC(CC)C(C)C)=O)CCOC2(CCCN(C(C3CCc4cncn4C3)=O)C2)C1 C(C(C)(COC)C(=O)NC(C)Cc1cn(Cc2nc(C(=O)O)cs2)nn1)OC N1(C(C(C)=C2CC2)=O)CCN(CC2CN(C(C3CCC(N(C)C)CC3)=O)C2)CC1 C(=O)(CC(CN(C)C)C(F)(F)F)NCCC1(NC(C(C=C)O)=O)CCCC1 N1(C(c2cc(Br)cn(C)c2=O)=O)CCc2ccccc2C1CC(=O)O N1(C(c2ccc(C#C)cc2)=O)CCC2(CC(NC(c3cc(Cl)n(C)n3)=O)CO2)C1 C1(C(=O)NC(C)CC2CN(C(c3cn(C(C)(C)C)cn3)=O)C2)CCCCC1O C1(CCNC(C=CC=CC)=O)C(C)CCCN1C(c1cc(CN(C)C)on1)=O Cc1cc(C(N2CCC(CCC(N3CC(C)CC(O)C3)=O)CC2)=O)c(C)n1C N1(C(c2cccc(Br)c2C)C(=O)NCCCCCC)CCc2oc(C)nc2C1 C=CC1(C(=O)NCCOC(C)(C)CNC(=O)C(F)C(F)(F)F)CCCCC1 C(CCSC)(C(=O)NC1CCCN(C(c2n[nH]cc2Br)=O)C1)OC N1(C(c2ccnc(C)n2)=O)CCC2CCN(C(=O)C(c3ccc(C)o3)C)CC12 C1(CC)CCCC1(C)C(=O)N(CC(O)CN(C(=O)CCc1ccccn1)C)C c1(C(=O)NCC(c2ccsc2)O)ccc(C2CC2(F)F)cc1 c1(C(=O)NCC2(CC)CCCO2)coc2c1CN(C(=O)C(=O)N(C)C)C2 N1(C(c2nnn(C)n2)=O)CCN(C(=O)C(c2ccccc2Cl)O)CC1CCO Fc1nccc(CNC2(C(c3ccc(OC(F)F)cc3)N3CCOCC3)CC2)c1Cl C(C)(N=c1nc(Cl)[nH]c(C)c1C#N)C1CCC(NC(CCC)=O)CC1 c1(C(N2CC(C3(NC(C(CCC)OCC)=O)CC3)C2)=O)cn(C)c2ccccc12 c1(C(=O)NC23CN(C(CN(CC)CC)=O)C(CC2)C3)cc(C)c(F)cc1F CCCCCC(CC)C(=O)NC(CNC(=O)Cc1ccon1)CC c1(C(=O)NCCCN(C(=O)C=CC(F)(F)F)C(C)C)ccc2ncnn2n1 c1(C(N(C(C(=O)NC(c2cnnn2C)C)C)C)=O)ccc(C2CC2)cc1 c1(SC)ccc(Cl)c(C(=O)NCC2(CNC(C3(C#N)CC3)=O)CC2(F)F)c1 N1(C=O)C(CNC(C)=O)CC2COCC12.N(C1CC1)CC C(=O)(CCCC(F)F)NC1C2CN(C(C3CN(C(C)C)C(=O)C3)=O)C1C2 c1(CS(=O)(=O)NC(C)Cc2ccc(F)cc2)ccc(Br)cc1F N1(C(C2CCC(C)S2)=O)CCc2nc(CNC(C3(C(=O)N(C)C)CC3)=O)sc2C1 N1(C(Cc2cc(C)ncc2)=O)CCC(O)(C(C)NC(=O)CC2CCOC2)CC1 c1(OC)cc(Br)cc(NC(N2CCN(C3CC3)CC2)=O)c1OC C1(CC(=O)NCC(CC=C)NC(c2ccnc(O)c2)=O)CC2(CCOCC2)CO1 C1(CC)(CC)NC(=O)N(CC(=O)NCC2CN(C(=O)CNC(N)=O)CC2O)C1=O Cc1[nH]nc2ccc(C(N3CC(C)(NC(=O)CC(C4CC4)C4CC4)C3)=O)cc12 N1(C(Cc2cn(C)nc2)=O)C2CCCC1CN(C(c1ccnc3ccnn13)=O)C2 n1(CC)ncc(C(=O)NC(C)CN(C)C(C2(C(F)F)CCC2)=O)c1Cl c1(C(=O)NCC(CN(C(CC(C)N(C)C)=O)C)O)cc(F)c(Cl)cc1F c1(C(N(CC(C(=O)NCc2csc(C)c2C)C)C)=O)coc2c1COC2 N1(C(C)=O)CCc2cccc(NC(=O)NCc3ccc(-c4cncnc4)cc3)c21 N1(C(CCCCC)=O)CC2CCCC2(CNC(=O)C2=COCCC2)C1 CCC(CC)CC(F)C(=O)NC12CC(NC(c3cn(CCO)nn3)=O)(C1)C2 c1(N(CCC(=O)N(C2CCOC2)CC#C)C)cccc([N+](=O)[O-])c1 C(=O)(C(C)(Cl)Cl)NCCN(C(C1(NC(=O)NC(C)C)CC1)=O)C C1(CNC(C(C)(C)OC)=O)CN(C(c2c(C(F)(F)F)coc2C)=O)CC1O N1(C(c2ccc(OCC)cc2)=O)CCCN(C(c2ccon2)=O)C(CO)C1 n1(CC(=O)NC(C2CCCC2)CNC(C(C)OC(C)=O)=O)cnc2c1CCCC2 c1(C(=O)NCC(C)NC(c2ncc(OC)cn2)=O)c[nH]c(C)c(Cl)c1=O N1(C(C(=O)N(C)C)=O)CC(NC(=O)CCOc2ccccc2)CC12CCOCC2 C1(CNC(C2CC(=C)C2)=O)CN(C(=O)CCCC(C)(F)F)C2(CCOCC2)C1 N1(C(C=COCC)=O)C2CCC1CC(CNC(=O)CC1COC(C)(C)CO1)C2 CCCCC(C(=O)NC(CC1CC1)C1CC1)NC(c1cc(C#N)oc1C)=O CCCCCC(CC)C(=O)NCC1(NC(=O)CCNC(C2CCC2)=O)CCCC1 c1(CC2(C(=O)NCC(CNC(=O)Cc3ccon3)OC)CC2)cccc(Cl)c1 CC1CC(C)N(C(=O)CSS(C)(=O)=O)CCN1C(=O)Cc1cc[nH]n1 C1(NC(C(=O)NC(C2CCCO2)CC)=O)CCSC(c2cccnc2)C1 c1(CNC(C(C)n2ccnc2)=O)ccccc1CNC(=O)C(C)(O)C1CC1 c1(C(N2CCC(N(C(C3CC3F)=O)CC)C2)=O)cc2cc(Br)cnc2s1 C(CS(=O)(=O)N(C1CCC1)Cc1cnn(C)c1)(C1CC1)OCC C1(C(N(C(C)CN(C)C(c2ncc(F)cn2)=O)C)=O)CCCC(=O)N1C c12ccc(cc1)C(=O)NCC2SC.c1(NC(=O)C(O)C(C)C)ccccc1CO c1(C(=O)NC(c2cccc(C)c2)C(C)(C)C)ccc(Cl)c(Cl)c1 c1(C(N2C(CNC(C3(OCC)CC3)=O)CC2)=O)cc(OC)c(O)c(CC)c1 CCCC(CC(=O)N1CCCC1C(=O)OC)N(C(=O)Cc1ccc[nH]1)C1CC1 C1(n2cc(-c3ccc(OC)cc3)nn2)CON(C(=O)C(C)n2cc(Cl)cn2)C1 Cc1ccc(C(N2CCN(CC(N3CCC(N(C)C)C3)=O)CC2)=O)cn1 CC(C)(C)CCC(=O)NCC1COC(CNC(=O)Cc2cc(O)nc(O)n2)C1 C1(F)(C(N)=O)CCN(CC(=O)Nc2cccc(OC(F)(F)Cl)c2)CC1 C(=O)(C1=CCCSC1)NCC1(F)CCN(C(c2scc(C(=O)OC)c2)=O)C1 CC1CC2CN(C(c3ccc(OCC4CCOC4)cc3)C(=O)NCCCF)CC12 c1(C(=O)NCC#C)csc(N(C)C(C2CCCO2)=O)n1 c1(C(N(C2CCN(C(C(CCC)C#N)=O)C2)C)=O)cc(S(N)(=O)=O)ccc1F c1(C(=O)NCC(C)(CO)NC(c2ccnc(CO)c2)=O)ccn2nnnc2c1 N1(Cc2sc(C)c(Br)c2C)CC2CN(C)C(CO)C2C1 O=C(CCCC(c1cccs1)=O)NC1CC=CC1.C12CC1C2.C12(CC1)C(=O)NCC2 C1(N(C(N2C(CC(=O)OCC)CCCC2)=O)C2CC2)CCc2c(n[nH]c2C)C1 O=C1CCCN(C(C2C3CC2N(C(C2CC4(CSC4)C2)=O)C3)=O)C1CCO N1(C(C2(NC)CCCC2)=O)CC(n2cc(CCC(=O)OC)nn2)C(C)C1 c1(C(=O)NC2(CO)CCCN(C(C(CC)COC)=O)C2)cc(F)c(F)cc1Cl N1(C(C(CC(N)=O)O)=O)CC(O)(C2(CNC(=O)CCn3ccnn3)CC2)C1 CC(CC(=O)NC1CC2CC(C1)N(C(=O)CSc1cnn(C)c1)C2)CC(F)(F)F c1(CC(=O)N(C2CC3CC2N(C(C2CC2C2CCC2)=O)C3)C)cc(F)cc(Cl)c1 N1(C(C(C)OC2CCCC2)=O)CCC(CNC(c2ccnn2C(C)(C)C)=O)CC1 c1(C(N(CCNC(=O)CCF)CC)=O)ccc(=O)n(-c2cnn(C)c2)c1 Cc1ccc(F)c(-c2cn(CCC(=O)NC3(C)CCCCC3C)nn2)n1 CN(C)NC(=O)CCC(=O)N1CC(NC(=O)CCOC2CCC2)CCC(O)C1 c1(NC(C(=O)NCCOC2(C)CCCC2)=O)ccc(NC2CC2)cc1 CCCC(O)CC(=O)NCC1(NC(c2cc(Cl)c(Cl)s2)=O)CCOCC1 CC(C)CC(C#N)C(=O)N1CC(CO)C2(CC2)C1.C123CCC(C1C2)n1nnnc1C3 C1(CC(N2C3(C(N(CCNC(C)=O)C)=O)CC(C2)C3)=O)CCN(OC)CC1 C=CC(C)(CCOC)C(=O)NCCN(C(=O)COCc1nnc(C)s1)CCC CC1c2c[nH]nc2CCC1C(=O)NCC1CCN(C(C2CC(N(C)C)C2)=O)CC1 C(=O)(C(C)(C)C(C)(F)F)NC1C(NC(C(=O)NCCCCCCCC)=O)COCC1 C(=O)(C(O)C(C)(C)C)N1CC(CNC(c2ccc(-c3nc(C)sc3)s2)=O)C1 C1(CNC(c2cc(C(C)=O)on2)=O)CCN(C(c2ccsc2)=O)CC1 CC(N=c1ccc([N+](=O)[O-])c(O)[nH]1)C1CN(C(=O)CC2COC(=O)C2)CCO1 c1(C(N(C)CC2CCN(C(C=C(C)C(F)F)=O)C2)=O)cc2cccnc2o1 CC1CC(NC(=O)Cc2nc[nH]n2)CCN1C(c1ccc(SC(F)F)cc1)=O C1(CC)CN(C(C2(C)CCNC2=O)=O)CCC1NC(c1cnc(C)cc1Cl)=O c1(CC(=O)NC2CC3CC(NC(C(CC)C)=O)C2C3)cc(F)c(F)cc1F Cn1cc(C(N2CC3CC(NC(=O)CC4CC4(Cl)Cl)C2C3)=O)n2cncc2c1=O CCC(CC(F)(F)F)C(=O)N(CC(C)NC(=O)CCN(CC(F)(F)F)C)C c1(CCN(C)CC)ccc(O)c(C(=O)NC(C)CC)c1 N1(C(=O)CCCC2CCCCC2=O)Cc2ncsc2C1 c1(OC)nc(C)ccc1C(N1CCCN(C(=O)CC2(O)CCOCC2)CC1)=O C1(C(N2CC(NC(CCc3ccc(C)nc3)=O)(CO)C2)=O)CCCCC1C1CC1 c1(C(N2CCC(CCC)(C(=O)O)C(O)C2)=O)cn2ccc(COCC)cc2n1 N1(C(C2(C)CC3CC3C2)=O)C2CCCC1CN(C(c1sccc1F)=O)CC2 C(=O)(C(O)CC(C)C)N(C1(CC(=O)NC(CC=C)C(=O)OCC)CC1)C C(=O)(CC(=O)NC(CNC(=O)CC1CC=CCC1)CO)OCCC(C)C N1(C(c2cn(C)nc2)=O)CCC(C)(C)C(C(=O)NCc2cnc(O)c(F)c2)C1 c1(-n2cc(C3CCCN(C(c4[nH]ccc4C4CC4)=O)C3)nn2)ccccc1[N+](=O)[O-] C1(COC)(NC(=O)C(n2ccnc2C)C)CN(C(=O)CN(C)C(C)C)C1 c1(C(C)=O)ccc(C(=O)N(C2CC(NC(C3CC3C(N)=O)=O)C2)C)nn1 c1(C(=O)NC2CC(CN(C)C)C2)ccc(-n2ccnc2)cc1 c1(C(=O)NC2CN(C(C(C(=C)C)(C)C)=O)CC2O)cc2nc(Cl)ccc2s1 Cc1nc(C#N)c(COCCC(=O)N(CC(C)NC(=O)Cc2ncc(C)o2)C)o1 c1(CC(=O)NC2CN(C(c3cnc(O)s3)=O)CC23CC3)ccc(Cl)c(Cl)c1 C12(C(N)=O)CCN(C1)CCNC(=O)C(=O)N2.c1(CC)ccc(C(=O)OC(C)C)o1 CC(C(=O)N1CC=CC1(C)C(N1CCCN(C2CC2)CC1)=O)S(N)(=O)=O C1(NC(C2CC(O)C2)=O)CC2(C(=O)NC3(CN(C)C)CC3)COC1C2 c1(C(=O)OC)cccnc1C(N1CC2CC2(NC(C2CC(OC(F)(F)F)C2)=O)C1)=O C1(C(=O)NC2(CNC(=O)COCC(F)F)CCCC2)CC2(C1)CC21CCC1 CC1CN(C(c2cnn(C)c2)=O)CC1NC(c1cnc(O)n1C)=O C(CCN(C)C(C1(n2cccn2)CCC1)=O)(C(C)C)NC(C(C)NC(CC)=O)=O C(=O)(C1=C(Cl)CCC1)N1CC(C(C)NC(=O)C(Cl)=CCl)OCC1 N1(C(C(C)NC(=O)OC2CCCC2)=O)CCCC(O)(NC(=O)OC(C)(C)C)CC1 N1(C(CCC#C)=O)CCC(C)C(NC(c2ccc(OCCO)cc2)=O)C1 c1(C(N2CCC(F)(CNC(C3(OC(C)=O)CC3)=O)CC2)=O)ccc2ccoc2c1 N1(C(C=COCC)=O)CC(CNC(c2csc3nccn23)=O)C2(CCC2)C1 c1(CCCC(=O)NC(C2CCCN(C(CC)=O)C2)C)cc(F)ccc1F N1(C(COCCCCC)=O)CCC(C(C)(C)C)(CNC(c2cn(CC)nn2)=O)C1 C1(CCOC)CN(C(=O)C(=Cc2ccco2)C)CCN1C(=O)CCC1CC1(Cl)Cl N1(C(C2CCC(=O)N2)=O)CC2CCN(C(C3CC3C(F)F)=O)CC12 C(=O)(CCP(C)(C)=O)NC(C)CC1CCN(C(=O)COCC(C)(C)C)CC1 c1(C(N(CC(=O)NCC(CC)O)C(C)C)=O)cc(C(C)=O)c[nH]1 C1(CNC(CCc2ccc(OC)nc2)=O)CN(C(=O)CCS(C)=O)CCC1(F)F C1(NC(c2c(CC)csc2)=O)CC(F)CN(C(=O)C(Br)=C(C)C)C1 C1(C(=O)NCC2N(C(c3occ(C)c3)=O)CC(F)C2)Cc2nc(C)cn2C1 C(CCCC(C)NC(=O)C(CCC)OCC)NC(C1(C#C)CC1)=O CC1CC(c2ccsc2)N(C(C2CCCN(CCC(C)(C)C)C2)=O)C1 N1(C(C(CC)N(C)C)=O)CC2CCN(C(c3cn[nH]c3)=O)C2C1 C[S+](C)CCC(O)C(=O)N1CCCCC1CNC(C1CCCN1C(N)=O)=O c1(C(C(N2CCC(N(C(c3c(CC)ncs3)=O)C)C2)=O)(C)C)ccc(OC)cc1 CCC(C(=O)OC)N(CC(C1CCC1NC(=O)C1CC1)=O)C C1(C(N2C(COC)CC(O)C2)=O)CC(F)CCN1C(=O)CC(C)O C(=O)(N1CCC(C(N2CCOC(C)(C)C2)=O)O1)C1C(C)=CCS1 N1(C(C(C#C)(C)C)=O)CCOC2(C1)CN(C(c1cnc(OC)s1)=O)C2 C1(CNC(COC2CCCC(C)C2)=O)N(C(=O)CCC2CC2)CCCC1(C)C c1(SCCC(=O)NC(C(C)(C)NC(C2C(C#C)C2(C)C)=O)C)ccc(F)c(F)c1 N1(C(c2c(C)scc2)=O)Cc2nccn2CC(NC(C2Cc3nccn3C2)=O)C1 C#CC1(C(=O)OCC)CCN(C(=O)C(=O)N(c2cccc(C)c2Br)CC)CC1 c1(CNC(N2CC(C=C)(CC(=O)OCC)C2)=O)ccc2nc(O)[nH]c2c1 c1(C(N2CC(CNC(CC(C=C)(C)O)=O)C(C)(C)C2)=O)c(F)cc(C)cc1F C1(NC(C2CCN(C(C)=O)C2)=O)CN(C(=O)COCCF)CC1O C1(CCNC(=O)NCc2cc(OC)c(Cl)cc2)OCCC1CC(C)C c1(OC)nccc2c1CN(C1CC(C(N)=O)C1)CC2 CC(C)(CC1CC1)C(=O)N1CCC(CCNC(c2nn[nH]c2Cl)=O)CC1 c1(C(=O)NC2CC(C)(NC(C(C3CC3)OCC)=O)C2)cccc(-c2nc(C)cs2)c1 c1(C(N2CC(OC)(CNC(c3ccccc3C(C)C)=O)C2)=O)c(C)cncc1C N1(C(COCCC#N)=O)CCc2ccc(C(=O)NCC3CCCCO3)nc2C1 N1(CC=O)CCOC2(CCC2)C1.CN1CCC(n2ccnc2SCC)CC1 c1(C(=O)NC(C2CC=CCC2)C(=O)NC2CCN(C(=O)OC)C2)nnn(C)c1N c1(CNC(C(CC2CCOCC2)NC(c2ccc(CO)s2)=O)=O)cc(=O)cc[nH]1 c1(C(N2CCC(OCCNC(c3ccc(F)c(Cl)c3)=O)C2)=O)ncnc(O)c1F N1(C(C(C(C)C)n2cncn2)=O)CCN(C(c2ccc(C#N)[nH]2)=O)CC1CF c1(-c2cn(CCc3cccc(C(=O)OCC)n3)nn2)cccc([N+](=O)[O-])c1 C(=O)(C(O)C(C)(C)C)N1CC(CC(C)NC(C=Cc2nnc(C(C)C)o2)=O)C1 C1(NC(CC(C)OC)=O)COC2(CCN(C(=O)C(F)=C3CCC3)CC2)C1 C(C(=O)N(C1CCN(C(c2nocc2-c2ccccc2)=O)C1)C)(C(C)C)SCC Cc1nn(C)c(C)c1OC(=O)CSCC(=O)NCCNC(=O)CC1(C)CCC1 N1(C(CC2N(C(CCc3cn(C)nn3)=O)CCOC2)=O)CCC(CO)C(F)(F)C1 Cc1cc(C(=O)NC(C(=O)NC2CC3(CC3)C2)c2ccoc2)ccn1 c1(CCCC(=O)NC2CC(NC(=O)C(F)(F)C3CCCC3)C2)cc(F)ccc1F N1(C(=O)NCC2C(OC)CCCC2)C2CCC(O)C1CCC2O S(=O)(=O)(c1cc(Cl)sc1C(=O)NC1CC(C)N(C(=O)CCCC2CC2)C1)NC N1(c2ccc(C(N(C)C)=O)cc2)CC2CC(NC(=O)CCCCCBr)CC2C1 c1(C(=O)NC23C(CN(C(Cc4ccc(OCC)cn4)=O)C2)C3)cnc(O)c(C)c1 c1(C(=O)NC2CCN(C(c3cnc(OCC)s3)=O)C2)ccc(Cl)cc1[N+](=O)[O-] c1(C(N2C(CN(C)C(C3CCC=CCCC3)=O)CCC2)=O)cnn2ccccc12 CCCC(C)C(=O)N1CCCC(CCNC(=O)Cn2nc(C(F)F)cc2C)C1 c1(OC)cc(CC(N2CCC3(NC(=O)CSC)CCCC23)=O)cc(Br)c1OC C1(C(=O)NC2CCN(c3nc(OC(C)C)c(F)cn3)CC2)CCCCC(F)(F)C1 N1(C(CCCC(=O)NCC)=O)CC2=C(C1)CN(C(=O)C(C)(O)CC(C)C)C2 C1(C(=O)NCc2c(C)noc2C)CC(C)CN(C(=O)CSc2ccccc2Cl)C1 c1(NC(=O)NCC=C)ccc(C(=O)N(CC(C)CNC(=O)CS(=O)CC)C)cc1 C12(C(=O)NCC3(C)CN(C(C4(CN(C)C)CC4)=O)CCO3)CCCN(CCC1)C2 c1(C(=O)NC(CC(C)NC(c2c(CC)c(C)sc2)=O)C)cccc([N+](=O)[O-])c1 C(=O)(C1=CCCC1C)N(CCC(=O)NCC(=O)OCC#C)C(C)C C1(C(=O)NC2(CNC(c3c(C)n(C(C)C)cc3)=O)CCOC2)COCC(C)(C)O1 C(=O)(C(O)CC[S+](C)C)N1C(CNC(CN(CCC#C)C)=O)CCC1 CP(C)(=O)C1CCCCC1C(=O)NCCN(C(=O)Cc1cncnc1)C1CC1 Cc1cnn(C)c1C(=O)NCCc1cc(C(=O)NC2CC(N(C)C)C2(C)C)no1 c1(OC)ccc(C(=O)NC2CC2NC(=O)CC2(C)CCCC2)c(Br)c1 N1(C(CC(CC)C(C)(C)C)=O)CCC2(CC1)CN(C(=O)CCC(N)=O)CC2CO c1(-c2nccc(CCCCC)c2)cc(OC)c(N)nn1 N1(C(C2C(C)(CC)C2)=O)CCC(C(=O)N(C)CCc2ccccc2)=C(F)C1 C1(CNC(=O)C(O)c2ccco2)CC2CCC1N(C(=O)CC1COCCO1)C2 CCC(C)C(C(=O)NCC1C2CCCC12)N(C)C(C1CS(=O)(=O)C1)=O c1(C(=O)NCC(C)N(C(=O)C(C2CCOCC2)C)CC)cc2cccnc2[nH]1 C=CC(C)(C)CC(=O)NC1CC(OC)CN(C(=O)CN2CCCC2CO)C1 c1(C(=O)NCC(CNC(C=CCC)=O)CO)cn(C)nc1Br c1(OC)ccc2cc(C(=O)NCCNC(c3cocn3)=O)c(C)nc2c1 N1(C(c2cc(COC)no2)=O)CC(NC(C2CCS2(=O)=O)=O)CCC1C C1(NC(C=CC2(C)COC2)=O)CCCCN(C(=O)CC2CNC(=O)C2)C1 c1(CC)ncsc1C(=O)NC(C(=O)N(C)CC1CCOCC1)C1CCOC1 C1(C(=O)NC(CO)C(C)NC(C2CC(N(C)C)C2)=O)(OC)CCOC1 Cc1cc(CCC(=O)NCC(CNC(=O)C(C)Cc2ccccn2)CO)n(C)n1 N1(C(C(C)NC(=O)NC)=O)CC2CCN(C(=O)C=Cc3ccncn3)CCC2C1 c1(OC)ncnc(C)c1C(=O)NCC12CC1CN(C(=O)C(c1ccc(Cl)s1)=O)C2 C(=O)(N=c1[nH]sc2ncccc12)c1c(NC(c2ccc(C)cc2)=O)ccs1 O=C(CCCCC(F)F)NCCC1CCCCN1C(c1cc2sccc2cn1)=O N1(C(CSCCC(C)C)=O)CCOCC1C(N1CCCCC1CC(N)=O)=O CC1CCCN(C(=O)C(N2CC3CC2C3NC(=O)Cc2cccc(CO)c2)=O)C1 C1(CCC)CC1N=c1[nH]c(N(C)CCOCCN(C)C)nc2ncn(CC)c12 C1(NC(CCSc2nc(C)[nH]n2)=O)CCN(C(=O)CC=C(Cl)Cl)CC12CCC2 N1(C(CCc2cn(C)nn2)=O)CC2CCCC(NC(=O)COc3ccon3)C2C1 N1(C(C(C)SCCCC)=O)CC(C2CCCCN(C(=O)COCC3CCC3)C2)C1 Cn1ncc(C(=O)NCC(F)(F)Oc2ccc(F)cc2)c1N CC1(CNC(C2(CF)COC2)=O)CC(F)(F)CN1C(=O)Cc1nc([N+](=O)[O-])n[nH]1 c1(C(N(CCNC(C2CCC(C)S2)=O)C2CC2)=O)ccc(N)c2c1CCCC2 CCCCC(C(=O)NCCCNC(=O)CCCc1ccc(O)c(F)c1)NC(N)=O c1(C(=O)NC(C(=O)N(CCC2CC2)CC)CO)ccc(C#N)[nH]1 C1(c2nnnn2CC(F)F)(NCCC(=O)NC)CN(C)CC1C N1(C(C(C)NC(CC)(C)C)=O)CC(NC(=O)CC2(C)CCC2)CC2(CC2)C1 c1(NC(C(CC2CCN(C(N(CC)CC)=O)CC2)F)=O)cc(OC)cc(C)c1 C1(C(=O)NC(C2CCN(C(CC(C)(F)F)=O)CC2)(C)C)CCC12CCOCC2 C=C(C)CN=C(NCc1c(O)cccc1Cl)NC1CC(=O)N(C(C)C)C1 c1(CC(N2CC3C(NC(CNC(CN(C)C)=O)=O)C3C2)=O)cc(F)c(F)cc1F CC(=O)CCCC(=O)N1CC(F)CC1CC(N1CCC(CN(C)C)CC1)=O c1(CC(=O)NC2C(NC(c3c(OC)cc(CO)cc3)=O)C2)cccc([N+](=O)[O-])c1 C(C(C)(C)C(=O)NCC(C)(CO)NC(c1coc(C(F)F)c1)=O)SC C(=O)(CCN1C(=O)NCc2ccccc21)NC1c2c(ccc(C)c2)OC1 N1(C(Cc2cc(C)[nH]n2)=O)CCC(NC(=O)CSc2nc[nH]n2)C1(C)C N1(C(=O)CCCF)CCCCC(C2CN(C(c3ccc4ccsc4c3)=O)C2)C1 N1(C(C2C(OCC)C2C)=O)CC=C(CNC(=O)CCc2nc(C)no2)CC1 CCC(C)(COC)C(=O)N1CCCC(CCCCNC(=O)CN2CC3CC3C2)C1 c1(OC)ccc2nccc(C(N3CC4CN(C(C5CC(C)C5)=O)CC4C3)=O)c2c1 C(=O)(CCCCC#N)NC(c1ccccc1)CNC(CCSc1n(C)nnn1)=O c1(N2CCN(C(C(C)C)=O)CC2)nc2c(c(=NC3CSC3)[nH]1)COC2 N1(C(CCc2cc(C)no2)=O)CC2CC2(CNC(c2ccnc(CO)c2)=O)C1 CN1CC2(CCCN(CCN3C(=O)NC(C)(c4ccc(Br)cc4)C3=O)C2)CC1=O c1(C(N2CCCC(C)(NC(=O)COC3CC=CC3)C2)=O)cccc2c1OCCN2 C1(CC(c2n(CCCSCC)nnn2)NCc2ncnn2C)CCCC(C)(C)O1 C1(SC)CN(C(C2CC(C)C2)=O)CC1NC(C1(n2cccn2)CCC1)=O Cc1ccc(F)c(C(=O)NCC(C(C)C)NC(=O)CC2C(C)C2(F)F)c1 N1(C(c2ncc(C)c(Cl)c2)=O)CCC(CNC(C2(CF)CC2(F)F)=O)C(F)(F)C1 C=CC(C)(O)C(=O)NCC(CC)NC(=O)Cn1cc(C2CC2)cn1 N1(C(=O)CSC2CCCCO2)CCC(O)(NC(C23CCCC2C3(F)F)=O)CC1 Cc1nnc(CNC(c2ccn(C(C)C)c2)c2nnnn2CC2CCCO2)o1 C1(NC(C2(NC(CN(CCOC)C)=O)CCC2)=O)CCCC12CC2 N1(C(C2COCC(C)O2)=O)Cc2occ(C(N3CCC(CF)C3)=O)c2C1 c1(C(=O)NC2(CCCNC(CC(C=C)C)=O)CC2)ccc(OC)nc1Cl C(C(=O)NCC1COC1)(C(C)(C)C)NC(CCOCCOCC)=O C1(CNC(C2CCC(C)C2)=O)CCC2CN(C(c3ncccc3O)=O)CC12 C(=O)(C(F)(F)CC(C)C)NCC(CC)NC(=O)Cc1nnc(C)s1 Nc1c(F)ccc(Cl)c1C(=O)NCC1(CCNC(C2(F)CC=CCC2)=O)CC1 CC(C)CC(C(=O)NCC1(O)CN(C(C2(C)CCC(O)CC2)=O)C1)n1ccnc1 C(=O)(C(C)(C)CC(F)F)NCC(C)NC(C1(CC)CCC1)=O O=C(N=c1nc2cc(Cl)ccn2[nH]1)N1CCC(c2ccc(O)cc2)C1 c1(C(N(C)CC2CCN(C(C3(OC)CC3)=O)C2)=O)ccc(C(F)F)c(F)c1 Cc1cc(C)nc(N2CCCCC(CNC(c3sccc3Cl)=O)C2)n1 CCCCC(CC)C(=O)N1CCN(C(C2CCC(OC)CC2)=O)C(COC)C1 C1(NC(=NCCC=C)NCCCSC)COc2cc(OC)ccc2C1 N1(C(c2c(C)onc2)=O)CCC(C2CCCN(C(=O)CCn3cccc3)C2)CC1 c1(C(C#C)OC(C)CC)ccccc1 c1(CN(CCS(N)(=O)=O)C)nn(CC(F)(F)F)cc1Br c1(C(=O)OC)nc(C(=O)N(C2CC(NC(=O)C(CC3CC3)OC)C2)C)cs1 C1(CC)(CC)CN(C(c2cc(C)c(C)nn2)C(=O)NCC2CCOC2)CCO1 c1(C(N2CC(CC(C)NC(=O)CC3CCC(=O)NC3)C2)=O)cccnc1S c1(NC(C(c2csc(C(C)(C)C)c2)N(C)CC2(C)CCCC2)=O)ccccc1Cl C12(CC)CCC(C(=O)NC3CCN(C(C4CC5CCC4C5)=O)C3)(CC1)CO2 c1(CC)cccc(NC(C2CCCC2CNC(=O)C(C)(C)CCSC)=O)c1F c1(C(=O)NCC2(CN(C)C(c3cc4sccc4s3)=O)CC2)cncn(C)c1=O O(C1CCc2c(F)cc(F)cc21)C(c1ccc(C(F)(F)F)c(Br)c1)=O N1(C(c2c(CC)non2)=O)CCC(C(=O)Nc2cc(C)c(C)cc2C)C(C)(C)C1 c1(C(N(CCNC(C2CC(OC)C23CCC3)=O)C)=O)cc2c(C)ccc(F)c2[nH]1 CCC(C)CCCC(=O)NCC1CC1CNC(c1cc(N(C)C)ccn1)=O c1(CNC(C=CCN(C)CC)=O)ccc(C(C)NC(=O)C(F)=CCCF)cc1 c1(C(N(CC(C)N(C(C=CC)=O)C)C)=O)ccc(C)c(OC)c1 CC1C(C(=O)NCC(=O)N(C)O)CCN1C(=O)CCCCC1CC1 c1(OC)cnc(C(=O)NC2CCOCC2C(=O)NOCCCO)cn1 c1(C(=O)NC(C)(CNC(c2cnccn2)=O)CO)nc2c(s1)COCC2 c1(CN(CCCC)CCN2CCC(C(=O)N3CC(O)CO3)C2)ccc(OC)c(F)c1 N1(C(c2c(C)cncc2)=O)CCC2CC1CN(C(=O)CONC(=O)OC(C)(C)C)C2 c1(CCC(=O)NC2CC3CC2N(C(c2n[nH]cc2F)=O)C3)nnc(S)nc1O c1(C(N2CC(C(=O)NC(CCOC)COC)(OC)C2)=O)cccc(C)c1C c1(C(=O)NC(C(C)NC(CCC=C(C)C)=O)CO)ccc(Br)c(F)c1F C(N=c1cc(C2CC2)nc(Cl)[nH]1)C12OCC(CSC)(C1)C2.c12ccsc1NC2=O n1(CC)ccc(NC(C2(CC)CN(C(=O)Cc3cn(C)cn3)C2)=O)n1 C(=O)(C(C)C(C)NC(=O)C=C(C)CNC(c1cc(Cl)n(C)n1)=O)OC c1(OC)cccc(NC(=O)C(C)(C)C2CCCO2)c1N1CCN(C)CC1 c1(C(=O)NC2(CNC(CC(CCC)O)=O)CCCC2)cc2cnccc2o1 N1(C(C2(COC)COC2)=O)CCC2(CC2NC(=O)CC(=O)N(C)C)C1 N1(C(C(CC)C(C)C)=O)CCN(C(C2(CO)CCCO2)=O)CC(O)C1 c1(OC)cccnc1C(=O)NCC(C)(C)CNC(c1cn(CCF)nn1)=O CC1CN(C(c2ccnnc2O)=O)CC2(CCN(C(=O)CC3OCCO3)CC2)O1 Cc1cc(NC(c2ccco2)=O)ccc1NC(C1CC12CCOC2)=O CC1CCCN(C(=O)Cc2cccc(OC(F)F)c2)C1CNC(=O)COC1CC1 c1(CNC(C(CNC(=O)COC2CCCC2)N(C)C)=O)ccc(F)cc1F N1(C(CCC(=C)Cl)=O)CCCCC2(CCN(C(C34CCC(N=[N+]=[N-])C3C4)=O)C2)C1 c1(C(=O)NCCNC(CC2(C)CC2(F)F)=O)ccc(N)cc1C(F)(F)F C(C)(CCCCNC(c1ccc(F)cn1)=O)NC(CC(=C)Br)=O C1(CNC(c2n(C=C)ncc2)=O)C(O)C(O)CN1C(=O)C(c1c(C)n[nH]c1C)C CN1CCn2c(CN3CCCC3c3ccccc3[N+](=O)[O-])nnc2C1=O C(CCCC(=O)N1CCCC1CNC(c1cccnc1C1CC1)=O)OCC N1(C(C(C(=C)C)(C)C)=O)CCCCC12CN(C(=O)CCNC(=O)CO)C2 C1(CN(C(c2cc(Cl)cc(Cl)c2)C(=O)NCC2CC2)C)CCc2nccn2C1 Cc1cc(C(=O)NCC2COCCN2C(c2snnc2C)=O)cc(Br)c1 Cc1cc(C#N)ccc1C(N1CCN(C)CC1CNC(C1(F)CCOCC1)=O)=O C1(Nc2nc(OC)c(C)cn2)CCC2(C1)CN(C(=O)C(C)n1ccnc1)C2 C1(O)(CNC(C2CC(N(C)C)C2)=O)CCCN(C(c2ccc(Cl)c(N)c2)=O)CC1 c1(C(N2CCC(CNC(c3ccnc(C(F)(F)F)n3)=O)C2)=O)cc([N+](=O)[O-])c[nH]1 N1(C(c2cc(CC)n(C)n2)=O)CC2CCC(Nc3cncc(Cl)n3)CC2C1 C(=O)(CC(C)(C)c1ccc(F)cc1)OC(c1ncc(C)o1)C1CC1 Cc1cncc(C(=O)NC2CCC(F)(CNC(c3nc(Cl)c(Cl)s3)=O)C2)n1 N1(C(C(c2ccc(F)cc2)C)=O)CCCN(C(c2ccn(C(F)(F)F)n2)=O)CC1 C=CCC(CC(C)C)C(=O)NCC(C)(C)CN(C)C(c1ccc(C(C)C)cn1)=O c1(OCC(=O)NC2CC(CNC(CC(CC)O)=O)C2)ccc(C)c(C)c1 c1(CCC(=O)NCC=CCNC(C2CCC(C)CC2)=O)cc2ccccc2o1 n1(CCC(=O)OCC)ccc(=Nc2nnc(C(O)CC)n2CC(C)C)[nH]1 N1(CC)CC2CN(C(C3CN(C(=O)C=CCOC)CC(C)(C)C3)=O)CC2C1 CC(C)(C(=O)N1CC(CNC(c2ccno2)=O)C(C(F)(F)F)C1)S(=O)(=O)C1CC1 C1(NC(C(C)CCO)=O)CCCN(C(c2cc(N)cc(F)c2)=O)CC1 N#CC1CCN(C(C2CC23CCN(Cc2ccc(-c4cc[nH]n4)cc2)C3)=O)CC1 N1(C(COC)=O)CCN(CCCCC2CCCN(C(=O)CNC=O)C2)CC1 C1(C(C)NC(C2(F)CCC2)=O)CCN(C(=O)Cn2cnnc2O)C1 CCC(CC(=O)N(C)Cc1nc(C)cs1)NC(C1COCCC1C)=O C1(C)(C(N(CCc2ccc(C)s2)C)=O)CC12CCN(CC(=O)NC(C)C)CC2 c1(CC(N2C(CNC(=O)CN3CCCCC3=O)C=CC2)=O)ccc([N+](=O)[O-])cc1 CC1=C(C(=O)NC2CC3CCC2(NC(c2coc(Cn4cccn4)c2)=O)C3)CCO1 C#Cc1cccc(C(=O)NCCC(C)N(C)C(C2CCC3C(C2)C3(F)F)=O)c1F c1(CNC(c2nc(C(F)(F)F)cc(Cl)n2)=O)cn2ccccc2n1 C1(NC(C(C)N(C(c2coc(CO)c2)=O)CC)=O)CC12CC(O)C2 C(=O)(C1=Cc2cc(F)ccc2OC1)N1CCC(N(c2ccnc(C)n2)C)C1 N1(C(C(C)OCC2CC2)=O)CC(F)(F)CC1Cc1cn(CN2CCNC2=O)nn1 C1(c2noc(-c3ccc(OCC(C)C)o3)n2)(NC(C(CC)SC)=O)CCCCC1 N1(C(C(CC2CC2)NC(c2cc(Cl)cs2)=O)=O)CCCC2(C1)N=N2 N1(C(C(CC)CC2CCCC2)=O)CC2CCCCC2(CN=c2[nH]c(Cl)ncc2Cl)C1 CN1CCC(NC(C2CCCCC2(C)NC(=O)CC2CCCCC2)=O)C(C#N)C1 N1(C(CCOCCOC)=O)CCC2CCCC12C(=O)NCCC1CC(=O)N(C)C1 C1(C(=O)NC2COC3(CCC3)OC2)Cc2ccccc2S1(=O)=O N1(C(C23N(C(C(C(CC)C)N(C)C)=O)CC(C2)C3)=O)CCOC2COCC12 C1(C(=O)NCCCOC2CCCC2)C2CC(O)C(C2)N1C(=O)C1=CCCCC1 N1(CC(=O)NCC(CN(C(C2C(C(=O)NCC#C)C2)=O)CC)C)CCCNS1(=O)=O n1(CC)ccc(=NC(=O)C2=CCCN(C(=O)C(C(C)C)OCCOC)C2)[nH]1 c1(N2CCN(CC(C)O)CC2)nc2ccc(Cl)cc2c(=NCC2(C)CC2)[nH]1 CS(=O)(=O)c1ccc(C(N2CC(O)CC2C(=O)NCCc2ncc[nH]2)=O)cc1Br c1(C(C(OC)OC)C)cn(C2CCC(C(=O)NC3CS(=O)(=O)C3)C2)nn1 Clc1cccc(NC2CCC2NCCc2ccccc2I)n1 c12ccc(cc1)OCC2.C(=O)(CC(=O)OC)NCC(C)NC(COC)=O N1(C(c2nccn2CCC)C(=O)NCC(=C)C)CCOC(C)(CC)C1 CC(C)(C)CC(=O)NCC1(F)CCN(C(C2(CN3CCCC3)CCCC2)=O)C1 N1(C(CN(C(C)C)C)=O)CC2CCC(C1)C2NC(C1CCCC(=O)N1)=O C1(NC(C2(COC)COC2)=O)CCOCC1C(=O)NC1(C)CCOCC1 c1(CC)cccc(C(N2CCN(C(=O)C(n3nc(C)cc3C)C)CC2)=O)c1N CC(C)(C)[Si](C)(C)OCc1ccccc1.C12(CCC1)CCN2.C1CCOC1=O C1(C(N2CC(C)C(NC(C3CCOCC3(C)C)=O)C2)=O)CCC(=O)N(C(C)C)C1 c1(OCCCC)ccc(CNC2CCN(C(=O)C(C)CC)CC2)cc1 c1(C(=O)NC2CC(O)(CNC(C3(OCC)CCC3)=O)C2)cc(C)c(C)cn1 C1(OC)CN(C(c2conc2C2(C)COC2)=O)CC1NC(C1CC2C=CC1C2)=O N1(C(C=NOC)=O)CCOCCC1C(=O)NC(C)CN(C)C(C)C C(C)(C)(CC(=O)NC(C)CCO)N(C(=O)Cc1ccon1)C N(C1CN(C(c2ncc[nH]c2=O)=O)Cc2ccccc21)C(C(CCC)OCC)=O N1(C(=O)CCCc2cccs2)CCC2(CCCN(C(=O)CCc3cnn[nH]3)C2)C1 Cc1cnc(F)cc1C(=O)N(C)CC1CCCN1C(c1ncc(C(F)(F)F)s1)=O C12(CNC(CCc3c[nH]c(=N)[nH]3)=O)CCC1CN(C(c1ccc(Cl)cc1Cl)=O)C2 c1(-c2ccc(CC(=O)NC(=O)NCCCOC)cc2)ccc(C(F)F)c(F)c1 CCCCC(C)CCC(=O)NC1CC(C(=O)NCC2=NOC(C)C2)C1 C1(C)(OC)CCN(C(c2ccc(-c3cn(C)nc3C)cc2)=O)C1 C#CCC(C(=O)Nn1cnnc1C)NC(=O)C1=CCN(C)C1 c1(OC)cncnc1C(=O)NC1(CNC(=O)C(C2CC(F)(F)C2)O)CCC1 C1(CC(=O)OC)CCN(C(=O)C(C2CCN(C(=O)CSC)C2)F)CC1 Cc1c[nH]nc1C(=O)NC(C)CC(=O)NCCCSCCO C1(CC(=O)NCCC2(NC(=O)CN(C3CCC3)C)CCC2)(OC)CCC1 C(=O)(C(C)(C)C#N)NCC1C(C(=O)NCc2cn(CCC)nn2)CC1 C(=O)(CC(C)C(F)F)NCC(C(C)C)NC(c1cc(Cl)n(C)n1)=O C1(C(N2C(C)(C)CC(c3ccccc3)C2)=O)CCCC2(CCCCC2)O1 C1(NC(CNC(=O)OC)=O)CCC2(CC1)CN(C(=O)C1=CS(=O)CCC1)CCO2 c1(C(N2CCN(C(C3CC(SC)C3)=O)C3(C2)CC3)=O)cc2c(C)cccn2n1 c1(C(C(=O)NCc2cccs2)N(CCCC#C)C)nocc1CC CC(C)C(C)C(=O)NCC1CC1NC(c1cc(Br)cn1C)=O C(=O)(C1=CC2C=CC(C1)C2)NCCCC1(NC(C(C)C(F)(F)F)=O)CCCCC1 N1(C(c2scc(C(C)=O)c2)=O)CCC(C)(CNC(=O)C(O)CC2CCCCC2)C1 c1(OC(C(N2C(CNC(C3(OC)CCCCC3)=O)CC2)=O)C)ccc(Cl)cc1C c1(C(N2C(CNC(C=C(CCC)C)=O)CC2)=O)snc(C)c1N N1(C(c2c(CC(=O)OC)occ2)=O)CC2(CCCC2NC(=O)CCCC(N)=O)C1 Cc1ccc(CCCCC(=O)NC2CCC(NC(c3cnc(Cl)[nH]3)=O)C2)cc1 C=C(C)CCC(=O)N(C1CCCCC1NC(=O)Cc1nc(C)sc1Cl)C C(=O)(CC(C)(C)n1ccnn1)N(CC(C)CNC(C1CCCN1S(C)(=O)=O)=O)C C1(c2nnnn2CCCC2CC2)(NC(C=C)C)CCCC(C)(C)CC1 C1(CNC(c2ccc(O)nc2)=O)CC2CCC1N2C(=O)CCC1CCC1 C1(C(C)NC(=O)CCC2CC2(F)F)CCN(C(c2nc[nH]c2C(C)(C)C)=O)CC1 C1(NC(=O)CC2CC2)CCN(C(c2cnnc3ccccc23)=O)CCC1CO C(=O)(C1Cc2ccc(Cl)cc21)NCCCCN(C(C(C(=O)OCC)F)=O)C N1(C(c2c(SC)csc2)=O)CCN(C(c2ncn(C(C)C)n2)=O)C(C)C1C c1(C(=O)NC(C)(C)CCNC(C2CC2Cl)=O)cc2c(cc1N)OCO2 N1(C(CSCCCC)=O)CCC(NC(=O)Cc2ncc(C)[nH]2)C(O)C1 C12(CNC(c3cnc(CC)s3)=O)CC1CN(C(=O)C(CC)C1CCOCC1)C2 c1(C(=O)NC(CNC(C(C)OCCCC)=O)C(C)C)cccc2nc(C)cnc12 C1(C(=O)NC(c2ccnn2C)C(=O)N(CC(O)COC)CC)CC2CC2C1 C1(Nc2ccc(OC)c(N3CCOC3=O)c2)CC2c3ccccc3CCC12 CCCC(C(O)C(=O)N(C)CCc1ncon1)NC(C1CC(F)(F)C1)=O C1(NC(CN(C)C(=O)C2CC2)=O)CCN(C(c2cc(C(F)(F)F)c[nH]2)=O)CC1F c1(C(=O)NCCCN(C(=O)C(F)F)C2CC2)ccccc1C1CC1(F)F C1(C(=O)NCCC(C)(C)NC(=O)C(O)C2CC2)CCc2ccnn2C1 C(=O)(C1=NN(C(C)CN(C)C)C(=O)CC1)NC1CCCC(NC(CC(C)F)=O)C1 c1(N(C)C)ccc(C(N2CCCC(c3cn[nH]c3)C2)=O)cc1F C1(C)(C(=O)NC2CCCN(C(C)=O)C2)CN(C(=O)C(C)n2cnnn2)C(C)(C)C1 C(=O)(CC(C(F)(F)F)NC(C1C2CCCOC12)=O)NC(CC)C(N)=O C(C)(C(CC(=O)NCCC(O)CO)NC(=O)Cc1ccnn1C)OC C(=O)(C1=NOC2COCC12)NCC1CCC(NC(c2[nH]cc(CC)c2)=O)CC1 c1(CCNC(C2CCC(OC)C2)=O)ccc(CNC(C2(CO)CCCO2)=O)cc1 n1(CC)cc(C(=O)NC(C)(C)CN(C(=O)CCCCOC)C)c(C)n1 CC(C)C(CCNC(=O)CN(C)CCO)NC(c1csc(-c2ccccc2)c1)=O c1(C(=O)NCC(C2CC2)NC(CC(=C=C)C)=O)sc2cccc(F)c2c1COC C1(C(=O)NC(CN(C(c2ccc(C)c(C)c2)=O)CC)C)CC2COCC2C1 N1(C(C2CNCC(C)(C)S2(=O)=O)=O)CCOc2cccc(F)c2C1 N1(C(C2(C)C(C)CCC2)=O)CCC2(CCN(C(c3csc(S)n3)=O)C2)C1 N1(CCCC(=O)NC2CC(O)C2)C(=O)CCC1=O C(=O)(C1=C(F)CN(C(C2CCCCNC2=O)=O)CC1)NCC1(O)CCC(C)C1 c1(C(C)C)nc(NCc2cccnc2)cc(=NCC(CC2CC2)CO)[nH]1 C1(NC(C(c2ccc(-c3cnco3)cc2)N(C(C=C)C)C)=O)CCCCCC1 CC1(C(=O)NC2CCC(NC(=O)Cc3ccc(F)cc3)CC2)COC(=O)C1 n1(COC)ccc(C(=O)NCCN(C(=O)Cc2ccsn2)C(C)C)n1 S(=O)(=O)(c1cc2c(cc1Cl)OCCO2)N1C(c2c(C)cccc2)C(C)CCC1 N1(C(c2c(N)cc(OC)cc2F)=O)CCCC2(CCCN2C(C2CC23CC3)=O)C1 C(CN=c1[nH]c2c(c(=NCc3ccsc3Cl)[nH]1)SCC2)n1c(=O)nccc1 c1(CC(=O)NCC2(O)CCN(C(C3C(CC(C)C)C3)=O)C2)c[nH]c2cccnc12 N=c1[nH]cncc1C(=O)NC(C(N1CCOC(C(N)=O)C1)=O)C1(O)CCC1 C1(C(=O)NCC(C)N(C)C(C2CC3CCC(C2)C3O)=O)CC(C)(C)OC(C)(C)C1 Cc1ccc(F)cc1C(=O)NC(CNC(c1cc(O)ccc1F)=O)C(C)(C)C c1(NC(C2CN(C(Cc3nc(C)sc3C)=O)C(C)C2)=O)cc(C)c([N+](=O)[O-])cc1Br c1(OC)ccc2c(c1)CC(C)CC2NC(c1ccc(CC(N2CCC2C)=O)cc1)=O N1(C(C(CC=CC)CC)=O)CCC2CCCC12C(=O)NCCN(C)C C(CC(C)(C)C(F)(F)F)NC(CS(=O)(=O)N1CCC(C)C1)=O C1(NC(c2ccc(CC)cn2)=O)(CNC(=O)Cc2c[nH]nc2C)CCCCCC1 C(=O)(CC(C)C(F)F)NC1CC2(C(C(=O)NCC(C)NC(=O)OC(C)(C)C)C2)C1 N1(C(C(C)N(C)C)=O)CCC(C)(CNC(C2CN(C(N)=O)C2)=O)C1 Cc1cnc(C(=O)NC(C)CCNC(C2CC2CC(F)F)=O)o1 C1(CNC(C2(C(=O)OCC)CC2)=O)CN(CC(C2CCCC2)C)CCO1 C=CC(C)(CCOC)C(=O)N1CCN(C(=O)C(CN(C)C)CC)C(CCO)C1 N1(c2snc(CCC)n2)CCC(CNC(=O)C(C)OCC2CCCO2)C(C)C1 N1(C(C(CC)O)=O)CC(OC)CC1C(=O)NCC1CCCC1N(C)C N1(C(C(c2ccc(N)cc2)C)=O)CCC(CCN(C)C(C2CCOC2)=O)CC1 C1(OC)(CNC(C2CCCN2C)=O)CCN(C(=O)C(C)(C)C2CCCC2)C1 C1(CNC(CSCC(C)=O)=O)C2CN(C(C3(C)CC3c3ccccc3)=O)CC12 c1(NC(c2cn(CCNC(C3CCCS3)=O)cn2)=O)ccc(O)c(Cl)c1 C1(OC)(CNC(c2cnc(Cl)n2C)=O)CCN(C(C2OCCC2C)=O)C1 c1(OC)cc(-c2ccsc2C(=O)Nc2cc(C)cnc2Br)c([N+](=O)[O-])cc1OC C1(C(=O)OC)C2CCC1(c1nccs1)C2.C1(=O)C(NC(C)=O)CSC2CN1C2 C(=O)(C(C1=NOC2CC12)N1CCc2nc(Br)sc2C1)NCCCCCC CCC(C)(CO)C(=O)N1CCC(C)(CNC(c2cccc(OC3CC3)c2)=O)C1 n1(C(C)(C)C)nnnc1C(C1(CSC2CCCC2)CC1)NCC1CCCCC1 O=C(C1=CCCOCC1)NC1CC(O)CN(C(C2(C(F)F)CCOCC2)=O)C1 c1(C(=O)NCC(CC(=O)NC)C)n[nH]c2c1CN(C(C1(CC(C)C)CC1)=O)C2 c1(N(CC(COC)(C)C)C)nc(=NCCC(C)(C)C(F)(F)F)[nH]c2c1COC2 c1(-n2c(C)ncc2)ccc(NC(=O)C(=O)NCCc2cc(C)n(C)c2C)cc1F C(CCCC(=O)N(C)C)c1nc(CC(C)N=[N+]=[N-])on1 CCCC(C#N)C(=O)N1CCC(NC(C2CN(CC)CCO2)=O)C1(C)C C1(C(=O)NCC(C)CN(C)C)CCCN(Cc2ccc(C(C)C)s2)CC1 C(=O)(C#CC1CCOCC1)NC12CC(NC(C(C)(Cl)Cl)=O)(C1)C2 N#CC1CCN(C(c2cncc(NC(=O)Cc3cc(Br)cs3)c2)=O)C1 CC1CCCN(C(C2CCCN(C(C3CCOC3)=O)C2)=O)C1CO Cc1oc(C(C)C)cc1C(=O)NC1CC(C)(NC(=O)CCCn2cccn2)C1 Cc1cc(F)c(C(N2CC(NC(c3cc(O)nc(Cl)c3)=O)C(F)C2)=O)cc1F c1(C(=O)NC2CCN(C(c3n(CC(C)C)ncc3)=O)C2)ccc2nccn2n1 C1(CC)CN(C(=O)CS(=O)(=O)NC)CCC1NC(C1CCCCC1O)=O N1(C(C(C)OC(C(C)CC2CCCO2)=O)=O)CCc2ccccc2C1 CC12CC(C1)C(C(N1CCC(NC(=O)COc3ccc(F)nc3)CC1)=O)CO2 c1(CN2CCC(N(C)C(C3(c4ccccc4)CC3)=O)C2)c(Cl)cccc1I C1(F)(C(=O)NCC2(OC)CC2)CCCN(C(=O)Cc2c(C)cnn2C)C1 Cc1c(C(N2CCC3CC3(NC(=O)C3CC3)CC2)=O)sc2cc(F)ccc12 CCCCC(C(=O)N(C)CC1CCN(C(=O)C(C)(C)C2CCOC2)CC1)N(C)C n1(CC(=O)NCC2(F)CN(C(C3=C(C)OCCC3)=O)C2)ccc2ccc(Cl)cc12 c1(OC)cc(Cl)cc(Cl)c1C(N1CCCC(OC(C)=O)C1)C(=O)NC(C)C c1(C(=O)NC(C)CNC(c2ccn(C)c2)=O)cc2cc(F)c(F)cc2[nH]1 CC1CC(CNC(C2(Oc3ccccc3)CC2)=O)CN1C(c1ccc[n+]([O-])c1)=O C1(NC(c2cnc(C)n2C)=O)C(C)CN(C(C2(c3ccncc3)CC2)=O)CC1C C=CC1CN(C(c2c(C)nn(CCC)c2C)=O)CC1NC(=O)CCCNC(C)=O c1(C(N2C(C(C)Nc3ccnc(C4CC4)n3)CCCC2)=O)cccc(Cl)c1Cl n1(CCC#C)cc(NC(C2CC(C)(NC(=O)CC3CC(C)C3)C2)=O)cn1 C1(C(N(CCCCCCNC(C(CCC)C)=O)C)=O)CC2CCCCC12 C1(CC(N2CCN(CCNC(C3(C)CCOC3)=O)CC2)=O)CCCC2(CCC2)O1 N12CC(CC(O)C1)Sc1cccc(c1)C2=O.Cc1cccc(Cc2cnccn2)c1 C(N=c1[nH]c(=NCCS(C)=O)[nH]c2c1CSC2)C1C(C(C)C)C1 c1(CC(=O)NC2CN(C(COCCC#C)=O)CC2N=[N+]=[N-])c[nH]c2cccnc12 c1(OC)ccc(C)nc1C(=O)NC(C)(C)CNC(=O)C(C)Cc1cccc(Cl)c1 CC1(CNC(C2CC3C=CC2O3)=O)CN(C(=O)CCCF)CCO1 CCC(C(=O)NC(C)CNC(c1cc(-c2ccccc2F)[nH]n1)=O)C(C)(C)CC CC1(CNC(=O)Cn2ccccc2=O)CCC(NC(=O)CCC2CCC2)CC1 c1(C(=O)NC(CC)COC(F)(F)F)coc2cccc(Br)c12 c1(C(N2CCC(CCCC)CC2)C(=O)NCCC)cc(OC)c(Br)c(OC)c1 c1(C(N2CC(C(=O)NCCN)OCC2)=O)ccccc1[N+](=O)[O-] C1(C(=O)NC(CNC(C(n2ccc(C3CC3)n2)C)=O)(C)C)C2COCC12 c1(CC)ncc(NC(=O)CCN(C(C2SCC=C2C)=O)C2CC2)cn1 C(CNC(c1cn(C)nn1)=O)(CC(F)(F)F)NC(CCN(CC)CC)=O C1(C(=O)NCC(C)(CO)NC(C(C)C#N)=O)CN2CCN1CC2C CC(C)(C(=O)NCCCCCn1cc(CN2CCCC2=O)nn1)c1ccncc1 N1(C(C2C(OC(C)(C)C)C2)=O)CC2CC2(CNC(c2cnc(-c3ccsc3)s2)=O)C1 C=CC(C)(O)C(=O)NCC1CC(C)N(C(=O)C=Cc2cn(C)nn2)C1 N1(CC)CCN(CCC(N2CCC(C(=O)NC(C3CCCC(=O)O3)=O)C2)=O)CC1 C(=O)(C(C)(C)C1CCCN1C(c1cc(Cl)ns1)=O)N(C)CCOCCCO Cc1ncc2ccc(C(N3CCC(O)C(NC(C4CC=CCC4)=O)C3)=O)cn12 Cc1nnc(NC(C2CN(C(c3ccnc(Cl)c3)=O)CCO2)C)c(C#N)c1C N1(C(c2n(COC)ncc2)=O)CC(CCNC(C2(CO)CCCC2)=O)OC(C)C1 c1(OCCCCC)cc(NCc2cncc(CC)c2)ccc1C CC1Cc2c(C(=O)O)cccc2CN1CCn1cc(C(N)=O)nn1 c1(CCC(=O)NC(CC2CC2)C(=O)NCC#CCCO)ccncc1 n1(CC(=O)NCC2(CNC(CC=CCC)=O)CC2)cnccc1=O N1(CC)CC(NC(C2CC(O)(CNC(=O)C(C)CO)C2)=O)CC1=O C(c1cccn1C)=CC(=O)NCC1CCC(NC(C(n2cc(C)nc2)(C)C)=O)C1 C(C1=CCN(C(c2ccn(C)c2CC)=O)CC1)NC(C(CC)F)=O c1(C(N2CC3(N(C(CC(C=C)C)=O)CC3)C2)=O)ccc2cc(Cl)ccc2n1 CC1(C#CC(=O)NCCC2CCN(C(c3scc(Br)c3Cl)=O)C2)COC1 c1(C(=O)NC2CCN(C(c3cnnc(O)c3)=O)C2)cc(O)nc(O)n1 c1(CN2CC(N3CCN(C(c4c(C)nc(C)s4)=O)CC3)C2)ccc(O)c(F)c1F S(=O)(=O)(c1cc2ccccc2s1)N1CCC(CC(=O)NCc2ccsn2)C1 C1(C(=O)NCCN(C(c2cc(C(C)=O)oc2C)=O)CC)Cc2ccccc2C1C C1(C(N(C(CCNC(Cc2nc(C)sc2C)=O)C)C)=O)CCC(C)(O)CC1 C1(OC)CC(NC(=O)Cc2cc(C)n(C)n2)CN(C(C2CCC(C(N)=O)C2)=O)C1 C12(C(=O)NCC3N(C(c4nnn(CC)c4C)=O)CC3)CCC(CC1F)C2 c1(C(=O)NC2(CCNC(C=CC)=O)CCCC2)ccc2nccnc2n1 C(=O)(C(CNC(C1(C2(O)CCC2)CC1)=O)C(C)C)NC(C(=O)OC)CC1CC1 N1(c2nc(=NCc3cn(CC)nn3)[nH]c(C)c2)CCOC2(CCOCC2)C1 Cc1ccc(Br)cc1CO.C12CCC(CC1)CC(=O)N2.C123CC(C1)(C2)C(=O)N3 C(=O)(C(C)(C)CC(F)F)NCC12N(C(Cc3cccc(C)c3)=O)CCC1CC2 Cc1ncc(C(N2CC(NC(=O)CSc3ccc(C)c(C)c3)C(O)C2)=O)c(C)n1 c1(C(=O)NC2C3CN(C(C45CC(OC)C4C5)=O)CC32)cccc2cnsc12 Cc1nc2ccccn2c1C(N1CCC2(NC(C3CCC=CCC3)=O)CC2C1)=O CN=c1[nH]c(=NCCc2ccccc2OC)[nH]c(=NCCCCC(C)(F)F)[nH]1 N#Cc1cncc(C(=O)NC2CN(C(=O)CNC(c3ccccc3)=O)CC2F)c1 C1(CC)(CNC(C2CCC(CN(C)C)O2)=O)CCN(C(=O)CC2CCC(=O)N2)C1 c1(C(=O)NCCC(C)NC(C=Cc2c(C)coc2C)=O)cccc2nccn12 CCCCC(F)C(=O)N1CC2CC(C(=O)NCCc3[nH]cnc3C)(C2)C1 Cc1[nH]c(=N)sc1C(N1CCC(CN(C)C(C2CCCC2)=O)C1)=O N1(C(CCCC(CC)NC(c2c(C)nsc2C)=O)=O)CCC2CCN(C)CC12 c1(CCC(=O)NC(CC=C)CNC(C2CC(OC)C2)=O)ccc(Cl)c(OC)c1 c1(C(C)=O)cc(C(N2CCN(C(=O)CC3CC(C)=NO3)C(CO)C2)=O)ccc1O c1(C(=O)NC2(CO)CN(Cc3ccc(C)cc3F)C2)cc(F)c(F)cc1O C(=O)(C(C)CCCCCC)N1CCCCC(C(N(CCCC#C)C)=O)C1 CC1CN(C(=O)NC2C3COCC23)CC(C)C1NC(=O)OC(C)(C)C c1(C(=O)NCC(F)CNC(c2ccc(CO)s2)=O)cc(F)c2cn[nH]c2c1 c1(OCCC)ccc(N(C)C(c2[nH]cc(C(C)=O)c2C)=O)cc1 C12(C(N(CCC(C)NC(c3cnc(SC)s3)=O)C)=O)CCC(C)(C1)OC2 N1(c2n(CC)c(C)nn2)CCn2c(C(C)(C)C)nnc2C1.C(C)(C)(C1CC1)O N1(C(C(C(C)C)(C)O)=O)CCOC2(CCCN(C(C3COC(=O)N3C)=O)C2)C1 c1(-c2cn(CC3N(C(Cc4c(C)scc4)=O)CCCC3)nn2)cccc(Cl)c1Cl C1(c2n(CCC)nnn2)(Nc2cn(C)nc2CC)CCC2CN(C)CC12 CC(O)(CNC(C1(NC(C23CC(CO)(C2)C3)=O)CCSC1)=O)CCO C1(NC(C(C)SC)=O)CC(C)CN(C(c2cc(C)n(C(C)C)n2)=O)C1 N1(C(CCC(C)SC)=O)CC(CNC(c2ccnn2C2CCC2)=O)OC(C)(C)C1 O=C(CCCS(=O)(=O)c1ccc(Br)cc1)Nc1cc(OCC(F)(F)F)cc(F)c1 CCCCC(C)N(C)C(c1ccc(CNC(C2SCCS2)=O)s1)=O C1(C(N2CC(C)C(NC(=O)Cc3cc[nH]n3)C2)=O)CCC(C)(C)CC1 c1(C(=O)NCCCOCCCNC(C(C)C)=O)ccc2ccnn2c1 c1(NCc2cccc(OC)n2)nccc(=NC(C)c2ccc3c(c2)CC(C)O3)[nH]1 c1(C(C(=O)NC(CC)CNC(=O)CN2CSCC2=O)C)cc(C)cc(F)c1 C(=O)C(O)C(C)c1ccccc1F.c12n[nH]cc1C1C(C3N(CCC3)C2=O)C1.CO C1(C(N(C2CCN(C(=O)COC3(C)CCC3)C2)C)=O)CCc2nnc(O)n2C1 c1(CC(C)C)ccc(C(=O)N(CCNC(=O)C2=CCC2)C(C)C)s1 C1(C(N(C2CCCC(O)C2)C)=O)CCCN1NC(=O)c1ccn(C)n1 N1(C(c2c(C)csn2)=O)CCCC(N(C(=O)C(C)N(C)C2CC2)C)CC1 C1(CC)CN(C(c2n[nH]c(C)n2)=O)CCC1NC(C1CCCN1C1CCCC1)=O c1(N(C)C)cncc(C(N2CCCC2(C)CNC(=O)C(F)F)=O)c1 C1(C(=O)NC(C)C(=O)N(C)C)C=CCCN1C(=O)Cc1ccco1 c1(CC(=O)NCC2C(NC(C3(CC(C)C)CC3)=O)CC2)nc(C(C)(C)C)cs1 N1(C(CCN(C(C)C)C(C2CC=CC(O)C2)=O)=O)CC2C3CCC(C3)C2C1 CC1COCC(C(=O)NCc2cnn(C)c2C(=O)NCc2ncc(Cl)cn2)O1 N1(C(C(CC)NC(C)=O)=O)CCC(NC(=O)Cn2cncn2)CC12CCCC2 c1(NC(C2CCN(Cc3ccc(COC)s3)C2)=O)ccc(OC)c(OCC#N)c1 CC1CCCCC1C(=O)NCCCOCCC(=O)NCCC1CC1 C(=O)(CCCF)NC(C)C.C1(CC(NOCCCCC)=O)CCC(=O)C1C C1(CNC(C(=O)NCC)=O)CN(C(=O)C(CC)C2CCOCC2)CC1(C)C C1(C(=O)NC(CC)CN(C)C(c2nnsc2C)=O)C2CC3C(C2)C13 c1(OC)cc(NC(c2nnnn2C2COC2)(C)CC2CCCCO2)cc(F)c1 c1(C(N(CCCNC(C2(C#N)CC2(C)C)=O)C)=O)ccc(Cl)c(F)c1 CC1CN(C(=O)CN2CC3CCC2C3)CC2(CCN(C(=O)C(C)CO)C2)O1 C1(CNC(C2C(F)(C(=O)OC)C2)=O)COCCN1C(C1CCC(OC)CC1)=O CC(C)C(C)CC(=O)N1CCC(C)(C)C1CNC(C1CCCCCC1)=O O=S(=O)(c1ccc(=NCCN2CC3CC3C2)[nH]c1)N1CCC2(CC1)CC2CO Cc1cc(N)ccc1C(=O)N(C(C)CNC(c1cccc(OC(C)C)c1F)=O)C c1(C(=O)NCC2N(C(C(CC)(C)O)=O)CCC2)ccc2[nH]c(=N)[nH]c2c1 CC(C(=O)N1CC(NC(=O)COCC(F)F)C1)c1cc[nH]n1 c1(NC(C2CCC(NC(c3cc(C(C)C)nn3C)=O)C2)=O)cc(O)c(Cl)cc1Cl c1(NC)ccc(C(=O)NCC(C)(O)CNC(=O)CSc2cccs2)cc1F CC1CCC(CCNC(C23CC(NC(=O)CSC4CC4)(C2)C3)=O)O1 N1(C(C(C)N(CC)CC)=O)CCC(CNC(C2CCCC2)=O)C(O)C1 C1(NC(C=CCN(C)CC)=O)CCCC(NC(C2CCOC(C(F)(F)F)C2)=O)C1 Cc1c(CN2CCC(CNC(C3CNC(=O)O3)=O)C2)cnn1C c1(NC(C2C(NC(=O)CCCCCCBr)C2)=O)cnc2c(c1)CC(=O)N2 n1(CC2CN(C(CSC)C)C2)nc(C(=O)SC2Cc3ccccc3C2)ccc1=O c1(C(N(C2CCN(C(C3CCC4CC3C4(C)C)=O)C2)C)=O)cc2n(c1)CCOC2 N1(C(c2c(C)cc(C)s2)=O)CCC(C)(C)C(NC(=O)Cc2cn(C)nc2C)C1 Cc1cnc(C)c(C(=O)NC2CCOCC2NC(=O)CC2CCC(=O)N2)c1 N1(C(c2c(OC)c[nH]n2)=O)CC(NC(c2cnc(C)cn2)=O)CC(C)C1 C1(C(=O)NCCN(CCCC)C)CC(NC(=O)Cc2cccs2)C1(C)C N1(C(CC(=O)N(CC#C)CC)=O)CC2CC2(C(N2CC(SC(F)F)C2)=O)C1 S(=O)(=O)(c1ccc(OC(F)F)cc1)NC1(CC(=O)NC2CCC(C)C2)CCC1 C1(CC(=O)N(CCNC(=O)CC(C)C(C)C)CC)SC2=NCCN2C1=O N1(C(=O)Cc2csnn2)CCn2ncc(-c3cn(Cc4cnns4)nn3)c2C1 C(=O)(C(C)C(CC)CC)NC(CC#C)CC(=O)NCCc1ccccc1 C1(CNC(CSCC(C)C)=O)CCCCCN1C(=O)CCN1CCCC1 C=CCC(CC=C)C(=O)N1CC(C(=O)NC2CCCC2F)C(C=CC)C1 n1(CC(C)C)nc(-c2cccc(N(C)C)n2)nc1C1CCCC(F)C1 N1(C(Cc2c(C)occ2)=O)CCCC(CNC(=O)CC(C)(C)C2CCCCC2)C1 CC1(C(=O)O)CCCCC1NC(=O)CC1CC=CCC1 Cc1cccc(CCNC(=O)NC2CCCC2Cc2cnn(C)c2)c1C Cc1cc(O)c(F)cc1NC(C1(C(C)C)CCN(C(c2cc(C#N)c[nH]2)=O)C1)=O N1(C(=O)C)CC(O)(COCCC(C)C)C1.C(CCCSC)OC C(=O)(C1=CCC(C)(C)CC1)N(CC(C)O)CCNC(c1cnc2ccsc2c1)=O C1(NCc2c(C(=O)OC)ccs2)CCCC(C(=O)Nc2ccnn2CCO)C1 C(=O)(CC(F)(F)C(F)F)N(CC(C)N(C(Cc1c(OC)ccc(Cl)c1)=O)C)C Cc1csc2c(N3CCC(O)(C(=O)NCCSC(C)(C)C)CC3)ncnc12 C1(C)(C(c2nnnn2C(C)C)NC(c2n(CC)ncc2)C)CCCCCC1 C1(C2CC2)(C(=O)NC(CCCC)CC)CN(C(c2cncs2)=O)C1 c1(C(N(C(CNC(Cc2cc(C)[nH]n2)=O)C)C)=O)cc(C)c(Cl)c(N)c1 C(C(C)(C)C(=O)N1CCCC(NC(c2c(C3CC3)cnn2C)=O)C1)SC c1(C(N2CCC(Cn3cc(CN(C(C)(C)C)C)nn3)C2)=O)cc(Cl)c2c(c1)OCO2 N1(Cc2c(C#C)cccc2)CCC2CN(C(c3ccc(Br)cc3OC)=O)CCC12 Cc1cccc2cc(C(N3CCC(F)(CNC(C4CCCC4O)=O)C3)=O)nnc12 C1(C(=O)NC(C2CN(C(=O)C(F)(F)C(C)O)C2)C)Cc2cccnc2C1 Cc1nc(Cc2ccccn2)sc1C(=O)N(C1CN(C(=O)C(C)CO)C1)C c1(C(N2CCCC(CNC(C(CCC)F)=O)(CO)C2)=O)cc(C)c(F)c(C)c1 N1(C(c2n(C)c(Cl)cn2)=O)CC(NC(c2cc(F)ccc2O)=O)CC(C)(C)C1 C1(CN(C(c2scc(OC)c2)=O)C)CCCCN1C(C1COCC1(C)C)=O C1(NC(C(C)N(C(=O)CCC2OCCO2)C)=O)CC(=O)N(C2CC2)C1 C=CCC(CC)C(=O)NC1CCN(CCCNC(=O)C(C)C(C)O)C1 C1(CNC(C2(OC)CCOC2)=O)CC(C(=O)N(C)CCN2CCCC2)=NO1 CS(=O)(=O)c1cc(C(=O)NC2CC(NC(C3C=CC=CC=C3)=O)C23CCC3)cs1 c1(SC)cccc(NCCCCNC(=O)C=Cc2ncc(C)[nH]2)c1[N+](=O)[O-] c1(NC(C(c2ccc(C#N)cc2)O)=O)cccc2ccc(Cl)nc12 c1(NC(C2CC2C(N2C(COC)COCC2)=O)=O)cnc(Br)c(I)c1 N1(C(CCc2ncc(C)[nH]2)=O)CC2CC(C1)C2N=c1cc(Cl)nc(C2CCC2)[nH]1 c1(CC(=O)NC(CCN(CC)CC)C)ccc([N+](=O)[O-])c(N)c1 O=C(C=Cc1cncs1)NN1CCCC1C(=O)N(C1CC1)CC1CCCCC1O c1(C(=O)NCCOCC(C)C)ccc(CN(C)CC(=O)CN2CC3CC3C2)cc1 CCC(C)CC(C(=O)N1CCC1CC=O)NC(=O)CCCN1CCCC1 C=C(CNC(=O)Cc1cnn(-c2ccccc2)c1)CCNC(C1CCC(F)C1)=O C1(CCC#C)CCCN1C(C1OCCC1OC(C)=O)=O C1(OC)C(NC(c2cccnc2CNC(=O)C(=O)NC2CC2)=O)CC12CCC2 CC(C)CC(C)CNC(C1CSCN1C(C1CCN1C)=O)=O N1(C(C2C(C(=C)C)OCC2)=O)CC2CCC1CN2C(c1cncc(SC)n1)=O c12cncnc1CNC2=O.c1(C(N(C(C2CCCO2)C)C)=O)ccc(C(N)=O)o1 c1(C(=O)NC2(C(N(C)CC3C(C)C3)=O)CC(F)(F)C2)cncc2[nH]ccc12 c1(C(=O)NCCN(C(=O)CC(C)(F)F)C)[nH]c2ccccc2c1C1CC1 C1(NC(C2CCSC2)=O)CCC2CN(C(c3cnn4c3NCCC4)=O)CC2C1 c1(C(N2CC(NC(C=Cc3cnc(C)s3)=O)C(O)C2)=O)ccc([N+](=O)[O-])cn1 c1(N2C(C)CN(C(=O)CCC(=O)NC3CCCC3)CC2)nc2cc(F)ccc2o1 c1(C(N2CC(NC(COCC)=O)CC3(C2)CC3)=O)ccc2c(c1)CCN(C)C2 C1(C(N2CC(=CC)C2)=O)CC(OC)CN1C(C1CCCCS1)=O c1(OCCOC)cc(C(=O)NCC(F)CNC(=O)C(c2cncnc2)C)ccn1 C1(NC(CC2(C)CC2)=O)CCCN(C(c2nc(C3CC3)cs2)=O)CC1 C1(C(=O)NCc2cc(C)sc2)CC(=O)CC12CCC2 CCC(C)(COC)CNC(=O)CCC(C)NC(C1CC1(Cl)Cl)=O c1(C(N2CCC(CC=C)(NC(c3coc(CO)c3)=O)C2)=O)nc(=O)cc(N)[nH]1 N1(C(c2sc(Br)nc2C)C(=O)NC(CC)C)CC2NC(=O)C(=O)NC2C1 C(CCC1CC1)(C(=O)NC1CC1)NC(C(C)OCCCC)=O CCC(F)C(=O)N1CC(O)(CCNC(c2occc2CN(C)C(C)C)=O)C1 c1(C(=O)NCC2CCN(C(C(P(C)(C)=O)O)=O)C2)ccc(F)c2cccnc12 c1(OC)cccc2c1OC(C(=O)NC1CN(C(c3cc(F)ccc3O)=O)C1)C2 N1(C(C(CC)O)=O)CC2CC2C1C(=O)NCCc1ccncn1 N1(C(CCCOCC)=O)CC(NC(C2CNC(=O)N2)=O)C(C)(C)C1 C#CCC(CC(=O)NCc1nc(C(N)=O)co1)NC(=O)C(C)(O)C(C)C C1(NC(C2(c3ccccc3)C(C)(C)C2)=O)(CO)CCN(C(=O)Cc2cc[nH]n2)C1 N1(C(C2CC(O)(CC#C)C2)=O)CCC(NC(=O)CC2CCCN2CC)C12CCC2 C1(C(=O)NC2(C)CCCN(C(C(C)=CC)=O)C2)CCC(=C(F)F)CC1 c1(C(N(CC(N2CC(C(C3CC3)C3CC3)C2)=O)CCO)=O)ccc2c(c1)CC2 c1(NCc2cnc(C(C)(F)F)s2)nc(Cl)[nH]c2ncnc1-2 N1(C(c2c(C)nc(C)s2)=O)CCOCC(C(=O)NCC(C)(C)C2(O)CCC2)C1 C(C1OCCc2sc(C(=O)O)cc21)NC(c1c(OC)cc2c(c1)OCO2)=O CCCC(CCCNC(c1c[nH]c(C(=O)OC)c1)=O)NC(C1(F)CC1)=O c1(C(=O)NC2CCCC(NC(CC3CC(CC)C3)=O)C2)cccc2c1CCCC2 CC1CN(C(c2cncc(N(C)C)c2)=O)CCN(C(=O)CCOCC(C)(C)C)C1 C1(C(=O)NCC2N(C(C)=O)CCC2)(NC(=O)C(C#N)CC)CCCCC1 c1(C(=O)NC(C)CNC(=O)CCCc2ccc(Cl)cc2)cc(C(F)F)ccc1Cl C1(NC(C=C2CCC(C)CC2)=O)CN(C(=O)C(C)(C)N2CCCCC2)CCC1O N1(C(C(CC)c2ccccc2)=O)CCCC(c2nc(C(C)C)no2)C1 c1(C(=O)NCC(CNC(Cc2ccn(C)n2)=O)(C)O)ccc(N)c(F)n1 N1(C(c2c(CC)n[nH]c2)=O)CC2CC(NC(c3cn(CCF)nn3)=O)C(C2)C1 C1(O)(CNC(c2ccc(OC)s2)=O)CC2CCC(C1)N2C(c1cccn1C)=O CC(C)(O)C(F)C(=O)NCC1CCN(C(=O)CCCCc2ccc(Cl)cc2)C1 C1(CC)CN(C(c2sc(Br)nc2C)=O)CCN1Cc1ccc(OC(C)C)nc1 N1(CC(=O)NCC23CC2CN(C(C2CC4(CC4)C2)=O)C3)CCn2ccnc2C1 c1(C(N2CC(O)(CCNC(C(CSC)O)=O)C2)=O)noc2ncccc12 COC1c2ccccc2CC1NC(=O)NCCc1cocn1 C(=O)(C(C)(C)CCC#N)NCC#CC(=O)N1C(CC(C)C)CC1 C1(C(=O)NCCCCN(C(CCCN(C(C)C)C)=O)C)CCc2c(cnn2C)C1 C1(CNC(C2CCCC(C)O2)=O)CC2(CC2)CN1C(=O)CN1CCCCCC1 C1(C(C)C)CCC(C)CC1C(=O)NCC1(C(C)NC(C2(F)CC=CC2)=O)CC1 C1(CC(=O)N(CCCCCC=C)C)CN(C(=O)CC(C)(C)O)CC12CC2 C1(CNc2cccc(OCC(C)C)c2)CC2CNC(C1)C2 C12(C(N3CCC(N(C(=O)CCOC4CC4)C)C3)=O)CCC(C1)C(C)(C)O2 C1(NC(CC2N(C)CCC2)=O)CCCN(C(c2nnc(S)n2C)=O)CCC1 Cc1ccc(Cl)c(C(=O)NC(C)CCNC(=O)CCc2ccoc2)c1 C1(C2CCC2)(C(=O)NCC2CC(F)(CN)C2)CCC1 C(=O)(CCCCCCC(C)=O)N1CCC(C)(NC(CC=C)=O)C1 CCCC(CCC)C(=O)N1CCN(C(=O)CCCCNC(C)=O)C(CF)C1 N1(Cc2nccc(OC)c2)CC2C(C1C(=O)NC1CSC1)C2(C)C N1(C(c2ccc(CC)[nH]2)=O)CCN(C)CC1CNC(=O)C(c1c(C)noc1C)C C1(CC(=O)NCC#CCNC(C2C(CC)C2)=O)(CO)CCCC1 CC1(C)COCCC1CNC(C1CSCCN1C(=O)CCN1CCCC1=O)=O c1(C(=O)NCC2(COC)CN(C(=O)C(C)c3cccs3)C2)cn(C)c(=O)nc1O C1(F)(CNC(CC(C)CC(F)(F)F)=O)CC(N=c2nc(CC3CC3)[nH]s2)C1 C(=O)(CC1=CCCCC1)N1C2C(CNC(c3c(CC)c[nH]n3)=O)C(C2)C1 C1(F)(C(=O)NCC2CCCN(C(Cc3c(C)noc3C)=O)C2)C(F)(F)C1(F)F CC1CC(CNC(C2(C)CCC2)=O)CN1C(c1cc(C2CCOCC2)[nH]n1)=O C(=O)(C(CCC)c1nn[nH]n1)N1C(CCN(C)C)CCC1 Cc1ccc(C(=O)NC2CCCC(C(=O)N(C(C)C)Cc3cccs3)C2)cc1C c1(C(=O)NCC(C)CN(C)C(C2(CO)CC2(F)F)=O)coc(C(F)F)c1 c1(C(N(CCCCN(C(C2(CSC)CCC2)=O)C)C)=O)cc(C2CC2)cs1 CC(CCCCc1ccccc1)NCCCCF N1(C(CCCc2onc(C(C)C)n2)=O)CCCCC(NC(C2CCOC2=O)=O)C1 C(C(CC(=O)NC1(C)CN(C(C2(C)CCCS2(=O)=O)=O)C1)C(F)(F)F)N(C)C C=CC1CN(C(=O)C(CN=[N+]=[N-])NC(=O)C(CCC)OCC)CC1O CC(C(CO)NC(=O)CCCSC(C)(C)C)NC(=O)C(O)c1ccsc1 C1(CC(=O)NCC(CC)NC(=O)CCC2CCCCC2)COc2ccccc2O1 c1(C(=O)NCC(CNC(C(Cc2c(C)noc2C)C)=O)O)cnn2cnnc2c1 Cc1ccncc1C(=O)NC1CC(C(N2CCC(O)(C(C)C)C2)=O)CC1O n1(CCOC)cc(C(=O)NC2CCCCC2NC(=O)C(C)SC)c2ccccc12 c1(C(N(CC(CC)NC(c2cc(SC)c(C)o2)=O)CC)=O)cc(SC)oc1C N#CC1CCN(C(=O)C(C2CC=CCC2)NC(C2CCC3(CC3)C2)=O)CC1 O=C1CCC(NCC(N2CCC(CCC(=O)O)(C(F)(F)F)C2)=O)CN1 c1(C(N(CCN(C(c2c(C)nc(CO)o2)=O)C)C)=O)cc(S(C)(=O)=O)cnc1O CCC(C)(CCC(C)C)C(=O)N1CCC(F)C(NC(=O)CCN2CCCC2)C1 Cn1c(CN2CCOCC2CCS(C)(=O)=O)nc2ccccc12 CC1=C(C(=O)N2CC(C)(NC(c3cn4c(n3)CCC4)=O)C2)CCCO1 C1(NC(c2cccc[n+]2[O-])=O)CN(C(c2cc(F)cc(Cl)c2)=O)C2(CCOC2)C1 N1(C(CCCSC)=O)CCCCC1CCNC(c1cccc(N)n1)=O N1(C(C(=O)Nc2ccc(NCc3cccc(F)c3)cc2)=O)CCOC2(CSC2)C1 c1(C(=O)NCCC2CCC(NC(CC(=O)NCC#C)=O)C2)csc2ccccc12 c1(C(=O)NCCc2cc(C(N(CCCCCC=C)C)=O)no2)ccnc(O)c1F C1(CCCC)CN(C(=O)C(O)C2CCCC2)CCN1C(=O)CCCC#N c1(CCN(C)C(c2csnc2-c2ccccc2)=O)cn(CCCN)nn1.CCO N1(C(c2cn3c(n2)CCC3)=O)CCCC12CCN(C(C1(CO)CCOCC1)=O)C2 Cn1cc(Br)c2c(NCC(O)C(F)(F)F)ncnc12 c1(SCC)cncc(C(N2CCC(NC(C3(CC(C)C)CCC3)=O)C2)=O)n1 c1(C(N2C(CNC(c3ccn(C)c3)=O)CCCC2)=O)ccc(C(C)(C)C)cc1N C12(NC(COCC(C)C)=O)CC(NC(c3ccoc3)=O)(C1)C2 N1(C(CCCc2onc(C)n2)=O)CCN(C2CN(C(C3C(C)C3C)=O)C2)CC1 N1(C(CCCOCC)=O)CC(C)(C)OCC1CNC(=O)CCCOC N1(C(CCSCCCC)=O)CC2(C1)CN(C(C1CC1CC)=O)C2 C1(OCC(N2CCN(CCNC(C3(C(N)=O)CC3)=O)CC2)=O)C#CCCCCC1 CC(C)C(C)(O)C(=O)NCc1cccc(NC(C2CCN2S(C)(=O)=O)=O)c1 c1(C(=O)NC(CCNC(C(CC)(C)OC)=O)(CC)CC)cncc2nnn(C)c12 Cc1ccc2cc(CN3CC4(COC(=O)N4C)C3)[nH]c2c1 C1(NC(C(CCOC)NC(c2ncccc2N)=O)=O)CCN(C)CC1C CN1CCCC(CCC(=O)N(C)CCNC(=O)C(F)=C2CCC2)C1 C1(CNC(c2nc(COC)[nH]n2)=O)C2CN(C(=O)C(Br)=C(C)C)CC12 C(=O)(CC(C)C(F)F)NC(CCOCC)C(=O)NC(C)Cc1nncn1C N1(C(CN(C)C(c2cc(C(N)=O)[nH]n2)=O)=O)CC(C(N)=O)C2(CC2)C1 C(=O)(C1n2c(C)nnc2CN1C(=O)OC(C)(C)C)OC12CC(O)C1C2 C(CC(C)N=c1[nH]c(=NC)[nH]c(=NCCCOCC2CCCO2)[nH]1)SCC C1(CNC(C2(COC)CCCC2)=O)C2CN(C(c3cc(O)no3)=O)CC12 C(=O)(CC1CCCNc2ccccc21)NCC1CCCCN(C)C1 C=CCC(C)(C)CCOC(=N)O.c12cccc(c1)N(C)CC(=O)C2 C(CC(CC)C(=O)NCCOCCOCCn1cc(Cn2cccc2)nn1)=CC Cc1cc(O)nc(CN(c2cccc(NC(=O)NC3(C)COC3)c2)C)n1 N1(CC(=O)N(CCOC)CCNC(c2[nH]cnc2C)=O)CSCCSC1 N1(C(c2ccc(SC)o2)=O)CC(NC(c2cnncc2O)=O)CC1CO C=CC1(C(N2CC3CCC2C(O)C3)=O)CCN(C(=O)CCCC2=CCCC2)CC1 CC1CC(NC(C2CC(C)(C(C)(C)C)C2)=O)CN1C(C1CC(C)(C)C1)=O c1(C(=O)NC2C(NC(C(COC)OC)=O)CCOC2)cnn2ccccc12 c1(SCC(=O)NCC(C)(C2CCC2)NC(=O)C2=C(Cl)CCC2)ccc(F)cc1F c1(C(N2CC=CC(NC(c3c(C)nn[nH]3)=O)C2)=O)ccc2cn(C)nc2c1 CCS(=O)(=O)NC(C)C(=O)NCC(O)CNC(C1(CSC)CCC1)=O c1(NC(C(C)c2cc[nH]n2)=O)cn(C(C)C(=O)NCC2CC=CCC2)nn1 N1(C(c2cc(C)[nH]n2)=O)CC(C(=O)NCC(C)C(F)(F)F)OC(C)C1 c1(C(=O)NC23CN(C(C4(CC=C)CC=CC4)=O)C(CC2)C3)ccc(F)cc1C#N C(=O)(CC(C(F)(F)F)NC(C1(Oc2ccccc2)CC1)=O)NCC(COC)C c1(C(c2n(CCCOC)nnn2)NC2(C)CC2(C)C)cc(C#N)n(C)c1 Cc1c(C(F)(F)F)n[nH]c1C(=O)N(C)CC1CCN(C(C2(C)CC2C)=O)C1 c1(C(N(CC(C)NC(C2C(C)C2(F)F)=O)CC)=O)nnc2ccccc2n1 C1(NC(c2cn3ccnc3s2)=O)CCCN(C(c2cc[nH]n2)=O)CC1 Cc1cc(O)nc(C)c1C(=O)NCC(C)NC(C1(C)CCCCO1)=O Cc1sc(-c2nc[nH]n2)nc1C(=O)NCC1(NC(=O)Cc2ccsc2)CCOC1 C#Cc1ccc(CCC(=O)N(C2CC(NC(c3ccc(CO)cc3)=O)C2)C)cc1 N1(C(c2ccc(C)o2)=O)CC2CCC2(CC(=O)NCCC2CC2C)C1 c1(C(=O)NC2CN(C(CCC=C)=O)CC2(C)C)cc2ccccc2cc1F N1(C(C=Cc2c(C)ncs2)=O)CCC2(C(=O)NCC(F)(F)F)CCCC12 C(=O)(C(CC(C)C)NC(c1cnn(C(C)C)n1)=O)NC1(CCCC)CC1 C(=O)(CCCN=C1NS(=O)(=O)c2ccccc21)OC(c1ccccc1Cl)C(=O)OC C1(CC)CN(C(=O)C=Cc2ccoc2)CCN1C(=O)C(F)n1cccn1 C(C(CC)CCO)NCCCOC(C1(F)CC(C(=O)OCC)C1)=O C1(C)(C(=O)NC2C(OC)CCCC2)CC12CCN(c1ccccn1)CC2 C1(CNC(C(C)NC(C(CC)NC(C)=O)=O)=O)CCN(C)CC1 Cc1c(NC(C(C)(C)C)=O)cccc1S(=O)(=O)NN1C2CCC1(C(C)O)CC2 c1(C(N(C2CN(C(c3cc(C)sc3)=O)CC23CC3)C)=O)cc2cnccc2[nH]1 c1(CNC(C2C(NC(C3ON=C(CC)C3)=O)CC=CC2)=O)[nH]ccc(=O)c1O C#Cc1ccc(C(N2CCN(C(c3cnc(C#N)s3)=O)C(CCC)C2)=O)c(F)c1 c1(C(N2CCC(C(=O)Nc3cnc(N(C)C)nc3)C2)=O)c(O)cccc1O C1(CNC(CCC)=O)CC(NC(=O)CCSCc2ccccn2)C1(C)C CCCC(F)C(=O)NCC1(CC(=O)N(CC(F)F)CCC)CC1 C1(CC)CC(CC(=O)N(C2CCN(C)CC2)CCCN2CCCCCC2)CCO1 c1(-c2n(C(C)C3CC3)ccn2)ccc(-c2cccc(Cn3ccnn3)c2)cc1 C(=O)(C1Cc2ccccc21)NCC1C(C(=O)NCc2ccn(C)n2)CCCC1 C(CCN=c1nc2cccc(Br)c2c[nH]1)NC(=O)Cn1nc2n(c1=O)CCCC2 N1(C(CS(CC(C)C)(=O)=O)=O)CCC2CCN(C(c3cc(CO)[nH]n3)=O)CC2C1 c1(C(C(=O)NC)N(CCCCCSC)C)cc(C(N)=O)sc1C C(c1c(C)coc1C)=CC(=O)N(C1CCN(C(c2cc(CC)ncc2)=O)CC1)C CC1=NN(C)C(=O)C1CC(=O)NC1CN(C(c2sncc2C)=O)CC1CO Cc1cc(=NC(=O)C2COCCN2Cc2sccc2Br)[nH]n1C c1(C(N(CCC)CCNC(=O)CCC2CC2C)=O)nsc2ccccc12 C1(CC=C)(C(=O)NCCCC(=O)NC)CCN(C(C2CCCCS2)=O)C1 N1(C(C2CC2F)=O)CC2CCCN(C(=O)CCc3nccs3)C2C1 C1(C(N2CC(NC(Cc3c(C)nc(C)s3)=O)C(C)C2)=O)CCOCC1(C)C c1(C(=O)NCC(C)N(C(=O)CCC2CC2(C)C)CC)ccc(C(C)C)nc1 CS(C)(=O)=NCC(=O)NCCCCCNC(C1CCC2C1C2(F)F)=O C1(NC(c2nc(C)c(C)o2)=O)CCN(CCOCC(C)C)CC1C Cc1cc(C(F)(F)C(=O)NCC2(CNC(C3SCCCS3)=O)CC2)cs1 N1(C(c2cnc(C)s2)=O)CCC(C)(CNC(c2ncccc2O)=O)C1 c1(CNCc2cn(CC(O)CCl)nn2)noc2c1CCCCC2 c12nccc(n1)CN1C(=CC=CC=CC3=CC=CC=CC(CC)(C3(F)F)S2)C1C c1(-c2cc(OC)ncc2)cccc(F)c1CN1CCOCC(O)C1 N1(C(C(C)NC(=O)CN(C2CCC2)C)=O)CCCC(C)(C)C1C C1(NC(c2[nH]nc(OC)c2Cl)=O)CCCCC12CCCN(C(C1CC=CC1)=O)C2 C(=O)(C1c2c[nH]nc2CN1C(C1CC2(C1)CC21CC1)=O)NCc1ncn(C)c1 C(=O)(CC(=O)NCC1(C(=O)NCCOC(F)F)CCC1)OC C(=O)(C(CNC(=O)CCCCN(C)C)CC(C)C)NC(c1nc(C)on1)C C1(NC(CCN(C(CC(C)F)=O)CCCO)=O)CCCC1(C)C C(=O)(C1=CC(O)CCC1)N(C)CC1CN(C(c2cscc2C(F)F)=O)CCO1 CCCC(CC)C(=O)N(CC(C)(C)C(=O)NC1CCC(C2CC2)C1)C C1(NC(c2ccc(OC)c(I)c2)=O)C2CCC1CN(C(=O)C(C)=O)C2 c1(CNC(=O)Cc2ccc[nH]2)cncc(C(=O)NC2CCCC2CO)c1 c1(C(=O)NC2CCN(C(CN(CCOC)C)=O)CC2O)ccc(F)c2occc12 N1(C(C2(C)N(C)CC(O)C2)=O)CCC(C2CN(C(=O)Cc3ccsc3)C2)CC1 N1(C(c2ccc(CC)cc2N)=O)CCC2(CC1)CN(C(C1CCC(OC)C1)=O)C2 C1(C(N2CCC(C(C)(C)NC(=O)C=CC3CCCCC3)C2)=O)C2CCC(F)(F)C12 C1(C(N(C)CC2CCN(C(C(SC)SC)=O)C2)=O)CCc2nccn2C1 CC(=NO)c1cc(C(N2CCN(C(C3CCCC4CCCN34)=O)CC2)=O)cnc1O C12=c3c(n(C)nc3)=NC(=NCCN(C)C1)N2.S(=O)(=O)(CC)NCCCOC=C Cc1n[nH]c(=NCC2CN(C(C3(Sc4ccccc4)CC3)=O)CCC2C)o1 C1(NC(Cc2n(C)nnc2)=O)C2CCN(C(c3ccc4c(c3)OCO4)=O)CCC12 C1(NC(c2cnc(C(C)C)[nH]2)=O)CC(OC)CN(C(c2sccc2C(C)=O)=O)C1 c1(C(=O)NC(CCN(C(Cc2cc(C)nn2C)=O)C)C)cccc(P(C)(C)=O)n1 C1(C(=O)NCCCNC(CCNC(=O)CO)=O)C2CCCCCC12 N1(C(=O)C(c2ccccc2)O)CCS(=O)CC1c1ccccc1 c1(OCC(N2C(C(CC)C)CCC2)=O)cccc(C)c1 C1(OCC)CC(N(C)N2CCC(N3CCCC3(C)C)CC2)C12CCCC2 C#Cc1ccc(Cl)c(C(N2CCC(C3(NC(=O)C(C)CSCC)CC3)C2)=O)c1 Cc1cc(C)nc(N2CCC(C(=O)NC(=O)CCc3ncc(Br)cn3)C2)n1 C(CC(C)NC(=O)OCc1ccccc1)(c1nnnn1C)N(CC(=C)Br)C N1(C(Cc2c(C)n[nH]c2)=O)CCN(C(=O)CN2CCC(CO)CC2)CC(O)C1 C1(C(N2CCC(CCNC(c3cn(C)c(O)n3)=O)C2)=O)OCC2CCCCC12 C#Cc1cc(F)c(C(=O)NCCC(O)CNC(=O)CCC(C)S(C)(=O)=O)c(F)c1 C(=O)(C(C(C)C)NC(c1ccccc1OCc1cccs1)=O)NCC(C)OC S(=O)(=O)(c1cccc(NC(=O)C(N2CC3CC3C2)C)c1)N(CC=C)C c1(C(=O)NC2CC3CN(C(C4(C)C=CCCC4)=O)C2C3)cnn2cccc(Cl)c12 c1(C(=O)NC(C#C)(CO)CO)cnc2c(cnn2C(c2ccc(F)c(Cl)c2)C)c1 C1(C(=O)NCC(C)(C)OCCNC(c2scc(OC)c2)=O)SC2C=CC1CC2 c1(OC)cc(Br)ccc1CNCC1CCCN(C(c2cc(Br)c[nH]2)=O)C1 c1(NC(=O)NC(CC(C)=O)C)c(F)cccc1Br CC1CCC(NC(=O)Cc2cncn2C)CN1C(=O)COc1cccc(C#N)c1 N1(C(CC2ON=C(CC)C2)=O)CC2(C1)CN(C(c1ccnc(C(F)(F)F)c1)=O)C2 C12(C(=O)NC3CCC(CNC(C4CSCC(=O)N4)=O)C3)CCC(CC1)OC2 C1(CNC(c2cc(CC)sn2)=O)C(C)CCCN1C(=O)CC1CC1C(F)(F)F c1(OCC)c(F)c(C(N2CCN(C(=O)C(C)C)C3(CCC3)C2)=O)cc(F)c1F CCC(CC)CCC(=O)NC1CC1CNC(=O)CN(c1ncnc2[nH]cnc12)C C(c1ccccc1)=CC(=O)NCCOCC(=O)Nc1ccnn1CC(F)F N1(C(C2(CCNC(=O)CC(O)C3CCCC3)CCC2)=O)CC2C=CCC(C2)C1 C1(CC(=O)N(CC(C)(O)C2CC2)C)CCCCN1C(C1CC(CC2CC2)C1)=O c1(N2CC(C(C)NC(C3CCN(C4CC4)CC3)=O)OCC2)cnc(C#N)cn1 CN1Cc2ccccc2C1CNC(=O)NC1CCc2ccc(Br)cc2C1 c1(C(N2CCC(C(=O)NC3(COCC)CC3)C2)=O)ncc(N)cc1C N1(C(=O)Cc2csc(Br)c2)CCC2(CCCN(C(C3CCC4CC4CC3)=O)C2)C1 c1(CN(C(c2cnc(C3CCC3)s2)C(=O)NCCOC)C)ccc(C#N)cc1F CCC(CC)(CC)C(=O)N(CC(O)CNC(c1nccc2cc[nH]c12)=O)C c1(NC)ccc(C(=O)NC2CCC2NC(C2(c3ccc(F)cn3)CC2)=O)cc1 C(=O)(N1CCC(C(=O)NCC2CCCOC2(C)C)O1)C1CCCN(C(C)=O)C1 N1(CSC)CC(C2(NC(=O)CCNS(CC)(=O)=O)CC2)C1.c12ccc(cc1)c(=O)[nH]2 N1(CC(=O)N(CCN(C(CCOCC#C)=O)CC)CC)CCCNC1=O C=CCCN=C(NCC(C)(C)C)N1CCC(NC(c2c(Cl)cccc2Cl)=O)CC1 C#Cc1c[nH]nc1C(N1CCC(N(C(=O)C=Cc2sccc2C)CCO)C1)=O C1(CN(C)C(C23CC(C2)C(c2ccccc2)N3)=O)CCC(CO)CC1 Cc1ncc(C=CC(=O)NCC(C2CCCN(C(=O)CN3CC=CC3)C2)(C)O)s1 C1(NC(C2(CC#C)CCOC2)=O)CCN(C(c2sc(CCC)nc2C)=O)CC1C C1(C(=O)OC)CC1C1CCN(C(c2cccc3o[nH]c(=N)c23)=O)CC1 N1(C(CCCN(C(C)=O)C)=O)CC(CNC(c2cn(C)cn2)=O)CC1C C1(C)(C(=O)NCC(CCNC(C2(CC=C)CC2)=O)O)CC(C(C)C)=NO1 C=C(F)CN=C(NC1CC1C)NC1CCN(C(=O)C(CC)CC)CC1 c1(C(=O)NC2CCN(C(c3cc(C)c(O)cc3)=O)CC2F)cc(Br)cc(F)c1O C1(O)(C(=O)NC(C(=O)OC)CO)CCN(C(=O)CCCN2CCCC2)CC1 c1(OC)cc(NC(=O)CC2CC3(C2)CN(Cc2ncc(F)cc2F)C3)cc(Br)n1 C(=O)(C1=CCC(C)(C)CC1)NC(CCOC)C(=O)NCc1cncn1C1CC1 C1(C(N(C2(C#C)CC2)C)=O)CN(C(=O)Cc2ccccc2F)CC12CCC2 c1(CC)cc(C)c(C(N2CC(CC(C)(C)CNC(C3CCOC3)=O)C2)=O)o1 C1(C(N2CCN(C(c3cc(C)no3)C(=O)NCC=C)CC2)=O)CC2C(C1)C2(F)F n1(CC(=O)NC(C)C(CO)NC(C2(CCF)CCC2)=O)c(O)nc2ccccc12 C1(C(=O)NCC(N2CCCC2)C)CN(C(c2ccc3c(c2)CC3)=O)C2(CCC2)C1 N1(C(C2CCN(C(C)=O)CC2)=O)CCCC(N(C)C(c2ccc(C)cn2)=O)CC1 c1(C(=O)NC2CN(C(C3C(OC)C3)=O)CC2C)cc2sccc2[nH]1 N1(CCCNC(C2(CC#C)CC2)=O)CCN(C(C2CC(O)(C#C)C2)=O)CC1.C(C#C)O c1(NC(=O)NCCC(=O)NCCN(C(=O)Cc2cnccn2)C)cccnc1 c1(C(N(C2CCN(C(c3cncc(C)n3)=O)C2)CC)=O)cn(C)cc1C Cn1c(=O)oc2c(C(=O)NCC3CN(C(=O)Cc4ccccc4O)C3)cccc12 C#CCC(CC#C)C(=O)NC1CC(CNC(C2COC(=O)O2)=O)C1 Cn1nc(C(=O)NC2CC2NC(C2CCCN2N=O)=O)c2cc(F)ccc12 n1(CCC(=O)NCC(CC=C)NC(=O)CCC=CBr)cccnc1=O CCC(COC)C(=O)N(C(C)CN(C(=O)Cc1ccc(C)o1)C)C C1(C(C)N(C(=O)C(F)C2CCOC2)CCO)CCN(C(=O)C(=O)C2CCCC2)CC1 c1(C(=O)NC(C2CN(C(=O)C(C)Sc3ccccc3)C2)C)ccc(CO)cc1 C1(C(N2C(C)(C)C(CNC(=O)C3=CCCOC3)CC2)=O)CCC2(CCOCC2)O1 C=CCCCC(C(=O)NOCC1CC1)NC(=O)CCC(=O)N(C)C c1(C(=O)NC2C3CN(C(C4ON=C(CC)C4)=O)C2C3)ccc(C)c(S(N)(=O)=O)c1 C(=O)(CC(C)C(F)F)N1CCCC(N(C(Cc2nnc(C)o2)=O)CCF)C1 c1(NC(C2CCC(CNC(C3CC4C=CC3C4)=O)CC2)=O)c(Br)ccc(F)c1F n12nnnc1C(NCC1CC1)C1(CCC1)CC(=O)NCCC2.C(C)(COC)SC N1(C(CCCC#CC)=O)CCC(N=[N+]=[N-])(C(N2CCC(CCN(C)C)C2)=O)C1 C(=O)(C(CO)C(C)(C)C)N1C(C(=O)NC(c2nccc(C)n2)C)CN(C)CC1 Cn1cc(C(N2CCCCC2C(N2CCC(CN=[N+]=[N-])C2)=O)=O)ncc1=O CCC(C)CCCC(=O)NC1CCC(NC(=O)CC2=CCCC2)CC1 C=CCCC(O)CNC(c1ccn(CCNC(c2cnc(C)o2)=O)c1)=O C12(CNC(CC(C=C)(C)C)=O)CCC(CN(C(c3cn(C)nc3O)=O)C1)C2 C(CC(C)(C)CC(=O)N(CC(=O)NCC1(CO)CCCO1)CC1CC1)OC C(=O)(CCC(C)(C)C(=O)NCCC1CCN(C(=O)Cn2nccn2)C1)OC Cc1ccc2sc(C(N3CC(C)CCC3CNC(C3(C4CC4)CC3)=O)=O)cc2c1 C1(C(C)NC(=O)C(F)=C2CCCC2)CCN(C(C2CC2c2cncn2C)=O)C1 N1(C(CSCC=C)=O)CCC(n2cc(CNC(C3(COC)CC=CC3)=O)nn2)C1 N1(C(C(C2CCOCC2)C)=O)CCC(NC(c2ccsc2C(F)F)=O)C1(C)C c1(C(=O)NCCC(CCNC(C(C)C)=O)C)ccc(S(=O)(=O)NCCN(C)C)s1 C1(C(=O)NCC(C=C)(C)C)CCCCCC1NC(=O)C(C)(C#N)CC c1(C(=O)NC(CC#C)C(=O)NC2OCC3CCCC23)cc(C)cc(C)c1 C1(NC(C(CC)CC)=O)CCCC12CCN(C(C1CN=C3N=CNN3C1)=O)CC2 CC1CC(C(=O)Nc2ccccc2-c2ncc[nH]2)CCS1(=O)=O CCC(F)(C(=O)OC)C(=O)N1CCC(Cc2cn(-c3cccc(CO)c3)nn2)C1 CC(F)(F)CCCC(C(=O)NCCCC1CC1)N1CCC(C)(O)C(O)C1 N1(C(C(C(C)C)=O)=O)CC2(CNC(=O)C(C)CN(C)C)CC1CCO2 C1(NC(=O)CCc2ccccn2)CC2(C1)CN(C(=O)Cn1ncccc1=O)C2 C1(NC(C2(C)CC2)=O)CC2(C1)CC(NC(C1CC1c1ccc(Cl)s1)=O)C2 N1(C(C(C)=CC)=O)CCCC(C2(NC(c3noc4c(F)cccc34)=O)CC2)C1 C1(CNC(C(CC)=CC)=O)(CNC(C2CCC(C(=O)OC)C2)=O)CCOCC1 C1(F)(CNC(c2cc(CC)sn2)=O)CCN(C(=O)C(C)C2CCCC2)CC1 CCC(C(=O)OC)C(=O)N1CCCC(CO)(NC(=O)C=Cc2c(C)coc2C)C1 C(=O)(C(F)C(F)(F)F)N1C(CNC(Cn2c(C)cnc2)=O)C(C)CC1 C1(C(=O)NCC2N(C(CSc3c(OC)cccc3)=O)CC2)CC2(CCC2O)C1 CCC(C)(CNC(=O)C(C(C)O)N(C)C)C(=O)NC(C)CC(N)=O CN1CCc2ccc(C(=O)NC3CC4CC(C3)N(C(c3ccn(C)c3)=O)C4)cc21 N1(C(C(CN(C)C)(F)F)=O)CCC2CCC(C1)N2C(C1(CO)CCCO1)=O N1(C(C2(COC)COC2)=O)CCC(C(=O)NCC(C)C(C)(C)C)CC1 C(=O)(C(CCC1CC1)NC(=O)Cc1c(C)noc1C)NCC(C)SC C1(C(=O)NCC2CCN2C(=O)CCOc2ccc(F)cc2)CCC2(CCC2)CO1 C(=O)(CC(C)C(C)(C)C)N(CC(C)N(C(CC(CC)CC)=O)C)C c1(C(C)NC(=O)OC(C)(C)C)cc(NC(=O)OCCC(F)(F)Cl)nn1C c1(OC)cc(CC(N2CC(CNC(c3cc(Br)ccn3)=O)C2)=O)ccc1F C1(C(=O)Nc2cccc(NC(CCCCC#N)=O)c2)CCC2(CC1)CC2(F)F C(=O)(C(C(C)(F)F)c1ccccc1)N(CCC(C)NC(C1CCCCC1)=O)C N1(C(C(C)(F)F)=O)CCC2(CCC(NC(C3CNC(=O)N3)=O)C2)CC1 c1(C(N(CC(C)O)CCNC(=O)Cc2cnsc2)=O)ccnc(OC2CC2)c1 CC(F)(F)C(F)C(=O)N1CC(O)CC1CC(=O)NCC1CCCOC1 N1(C(c2cc(CSC)no2)=O)CCCC(CO)(NC(=O)CCc2ncccn2)C1 C(=O)(C(C)(C)C(O)CC)NCCCOCCC(=O)N(C(CC)C)CC1CC1 C1(NC(C(C)=C(C)C)=O)CCN(C(c2ccc(-c3ccccc3)nc2)=O)C(C)C1 C1(OC(C(=O)NCC2(F)CC(CNC(c3c(C)con3)=O)C2)C)CCCCCC1 c1(C(N2C(COCC)CC(F)C2)=O)cc(OC)cc(OC)c1N.CCC(=O)NC c1(C(=O)NCC2(C(C)(C)C)CCN(C(C(C)=CC)=O)C2)cc(C#N)ccc1C CC(C)C(C(C)NC(=O)C(=O)NCc1ccc(F)cc1)NC(=O)CCCC#N n1(C2CC(NC3CCOCC3C(=O)CC(=O)C=CBr)C2)ccc([N+](=O)[O-])n1 Cc1ccc(-c2cnc(NC(=O)C(c3ccccc3)C)c(O)c2)c([N+](=O)[O-])c1 Cc1nc(CO)oc1C(=O)NCC1CC(F)(CNC(C2(C)CC2(F)Cl)=O)C1 CC(N=c1cc(Cl)c2ccc(Br)cc2[nH]1)c1ccc2ccccc2c1 c1(C(N2CCC(C)(NC(Cc3cc(CC)no3)=O)C2)=O)cccc2oc(=N)[nH]c12 c1(NC)ccc(C(=O)NC2CCCN(C(=O)CCN3CCCCC3C)C2)nc1 Cc1cccc(NC(=O)CN(C(C)C(=O)N(C)C)C)c1 C(=O)(CS(C)(=O)=O)NC(C(=O)NCCNC(COC)=O)C1(C)CC1 c1(C(N2C(CNC(COc3cn(C)nc3)=O)CCC2)=O)cnn(C)c1C#N S(=O)(=O)(c1cccc(Br)c1F)N1CCN(Cc2c(OC)ncc(F)c2)C2C1C2 Cc1nc(Cl)[nH]c(=NC2CCCCC2NC(=O)CC(F)(F)C(F)F)c1Cl N1(C(C=CC2(C)COC2)=O)CC2(CC(NC(C3CC4C=CC3O4)=O)CO2)C1 C1(C(=O)Nc2c(OCC)nccc2)CC(O)CCN1C(=O)C(O)C(C)C c1(NCC(CCCC)NC(c2nnn(C(C)(C)C)n2)=O)ncn(C)c(=O)c1Br C=C(C)CN=C(NCc1ccnn1CCC)N1CCc2ncsc2C1 c1(CC(=O)N(C2CC(NC(c3c(C)ncs3)=O)C2)C)ccc(F)cc1Cl c1(OC)cccc(NC(=O)C(C2(C)CC2)NC(=O)CCCN=[N+]=[N-])c1F C(N=C(NCC(=O)NC(C)C)NCC(C)(C)F)C1(OC)CC1 N1(C(c2cnc(C3CC3)s2)=O)CCC2C(CCCN2C(=O)CCC2CCCO2)C1 c1(NCCN(CCNC(C)=O)C)ncccc1S(=O)(=O)NC(c1ncnn1C)C c1(C(N2C(CCC(=O)N(C3CC4CC4C3)C)CCC2)=O)ccc(O)cn1 CC(C)CCC(=O)C(=O)N1CCC1CNC(c1cccc(CF)c1)=O N1(C(CC(C)CF)=O)CC(C2CN(C(c3ccc(C4CCC(=O)N4)cc3)=O)C2)C1 CS(=O)(=O)c1cc(C(N2CC3(CC(NC(=O)COCC4CC4)C3)C2)=O)cs1 N1(C(C2(C)COC2)=O)CCOC(CCNC(c2cccc(C(C)(C)C)c2)=O)C1 C1(C(N(C2CCS(=O)(=O)C2)CCC)=O)CC=CC(n2ccnn2)C1.C(C(C)(C)CO)N C1(NC(=O)C=C2CCSCC2)CCCN(C(=O)Cc2c(Cl)cccc2Cl)CC1 C1(C(=O)NC(c2ccccc2)CNC(C2(C#C)CC2)=O)CCOCC1C c1(C(=O)NCC(CN(C(C(N2CCNC2=O)C)=O)C)O)cc2sccc2s1 C1(C(=O)NCCC(C)CCNC(=O)C(C)(C)CC(F)F)CCCC2(CCC2)O1 C1(CNC(CN(C2CCC2)C)=O)CN(C(=O)Cc2cncs2)C2(CCC2)C1 c1(NC(NNC(=O)c2scc(OC)c2)=O)c(C)nc2n1CCCC2 C(=O)(CC(CC)NC(=O)C=CCN1CCCC1)NC(COCC)C C(=O)(C(C)(C)C)NCCC(=O)NCC1C(NC(CC2CC(=C)C2)=O)C1 S(=O)(=O)(c1cccnc1NCC(c1ccccc1Cl)O)NCC1(C)CCC(C)C1 c1(-c2cnc(C(N3C(C(N)=O)CC(F)(F)C3)=O)nc2)ccc2c(c1)OC(F)(F)O2 c1(OC)nc(OC)nc(N2CCC(F)(C(N3CCCC(O)C3C)=O)CC2)n1 c1(C(N2CCCC(NC(C(=O)NCC)=O)C2C)=O)cc(C)c(F)c(C)c1 c1(C(=O)NCC2CC(NC(C3C(C)(C(C)C)C3)=O)C2)ccnc(CO)c1 C1(CN2CCC(C(N(C3CCCCCC3)CC)=O)CC2)CC2OC1CC2O N1(CC)CCOC(C(=O)NCC(CNC(c2ccnc(C(F)F)c2)=O)CO)C1 C(=O)(C(O)(CN(C)C)C(F)(F)F)NC1(CNC(CC(CC)CC)=O)CCOCC1 c1(SC)cc(C)c(C(=O)NCC(C2(O)CCN(C(=O)CCc3cnoc3)C2)C)o1 C1(COCCCN(C(CCNC(=O)OCC)=O)C)CCCOC1.C1(=O)CN1 c1(C(N2CCC(F)(CNC(C(P(C)(C)=O)O)=O)C2)=O)c(F)ccc(F)c1F c1(C(=O)NC(C(C)NC(CS(=O)(=O)NCC)=O)C)cccc(C)c1N CC1CCN(CC(=O)NCc2c[nH]nc2C2CCN(C(=O)CSC3CC3)C2)CC1 C1(NC(Cn2nnc(C)n2)=O)CC(C2CCN(C(c3ccc(F)cc3O)=O)C2)C1 Cc1[nH]nc2ncnc(N3CCC(CCNC(=O)C(F)Cc4ccccc4)C3)c12 c1(NC(=O)NC2C3CCC4C(C3)C24CO)cnc2c(c1)CS(=O)(=O)CC2 c1(CC2N(C(=O)NC3C(=O)N(CCF)CC3)CCCC2)ccc(Cl)cc1F C1(C(N(C(C(=O)OC)C(C)O)C)=O)CCN(S(=O)(=O)N(C)C)CC1 C1(NCCCOCCCO)COCC1n1cc(Br)cn1 C(CN=c1[nH]c(=NCc2ccc(C3CC3)cc2Cl)[nH]c2c1CCC2)C1C(F)(F)C1 c1(C(N2CCCC(CN(C(c3cc(OC)ncc3)=O)C)C2)=O)cccc(C)c1C c1(C(N(C2CCNC2c2ccccc2)CCCOC)=O)ccccc1C N(C1CC2(CCCC2)c2ccccc21)C(C(=O)NC1CCCN(CCO)C1=O)=O c1(C(N(CC(C)NC(c2cc(CC)oc2C)=O)C)=O)cc(F)cc2nccnc12 C1(CC(N2CC(=C(CNC(C3CCCC3(F)F)=O)F)C2)=O)CC2(CCC2)C1 c1(CC)cncc(CNC(=O)C(C2CCC2)NC(c2cc(Cl)cn2C)=O)c1 CCCCC(O)C(=O)NCC12CC(CC)(CN1C(=O)CN(CC(C)(C)C)C)C2 c1(C(N2C(C(=O)NCCCC(C)(C)C)CCCC2)=O)cccc(Br)c1F CN1CCN(C(=O)Cn2cc(C3COCCN3)nn2)C1=O CC1(NC(C2CCC(NC(=O)C=Cc3cncs3)CC2)=O)CCSCC1 c1(C(N(CC(CCC)C)C)=O)oc(CNC(c2ccncc2)=O)nc1C C(=O)(C(CCC1CCC1)NC(C1CC=CCC1)=O)N(CC(C)C)C(C)C C(=O)(C(Cc1ccc(O)cc1)C(F)(F)F)NCC(C)NC(CC=C=C)=O N1(C(C(C2CCOCC2)C)=O)CCC(NC(=O)Cn2cc(Cl)cn2)C(F)C1 Cc1ccc(C(=O)NCC(C)(C)C(=O)NCC2(CO)CC(C)C2)c(C)n1 N1(C(C#CC(C)C)=O)CC2CCC(C(=O)NCCCC3CC3C)(C2)C1 C1(=O)CC(CC#C)N1CCO.c1(C(NOCCCC#C)=O)oc(C)nc1CC CS(=O)c1cccc(C(=O)NC2COCCC2NC(c2nocc2C2CC2)=O)c1 C1(C(=O)NC(C)CN(C)C(c2occ3c2CCC3)=O)COC2CCCCC12 C#Cc1cncc(C(N2CCN(C(=O)C(C)OCC3CCCO3)C(C)C2)=O)c1 N1(C(C(C)OCC=C)=O)CCC2CCCC(C1)N2C(=O)CSc1ccccc1 C1(C)(CNC(C(C2CN(C(c3n(C)ccn3)=O)C2)O)=O)CC(C)(C)C1 c1(NC(c2c(C)scc2)=O)cncc(C(=O)NC(C)C(=O)OC(C)(C)C)c1 c1(SCC(=O)NC(C2OCCN(C(CC(C)OC)=O)C2)C)ccc2c(c1)CCC2 C1(NC(CC(=O)N(C)C)=O)CC2CC1N(C(=O)CCc1nncs1)C2 C(=O)(C(C)C(O)C(C)C)NC.c12ccc(cn1)C(=O)NCCN2CCC CC1CC(CNC(=O)COc2ccccn2)CCS1 C1(C(=O)NCC2CC(OC)CN2C(C2CCCC2(C)C)=O)CS(=O)(=O)CC12CC2 C1(C(N(CC(COC)C)C)=O)(CNC(c2cnc[nH]c2=N)=O)CC12CCC2 Cc1cccc2[nH]cc(CC(N3CC(NC(=O)CCC(C)C)C4CC34)=O)c12 C12(C(=O)NCC3(NC(c4c(N)nccc4)=O)CC3)CCC(CC1)CC2 C(=O)(C(C)(C)C(C)(F)F)NCC1C(CC(N2CCC(OC(=O)NC)C2)=O)C1 C1(C2CCCO2)(C(N(CCCNC(c2cccc(C#C)c2Cl)=O)C)=O)CCCO1 c1(-n2c(-c3csc(CO)n3)nc(CCCCC)n2)cc(C)nc(C)c1 C1(C(C(=O)NCCCSCC)C)CCN(C(=O)Cc2ncc(CC)[nH]2)C1 Cc1cccc(C(N2CC(O)(C(C)NC(C3CCN3S(C)(=O)=O)=O)C2)=O)c1C C12(C(=O)NCC3(F)CC(CNC(c4csc(Cl)n4)=O)C3)CC(CF)(CO1)C2 c1(NCc2cc(C(=O)O)cc(Cl)c2)c(Br)cc(C(F)(F)F)cc1Br c1(C(N2CCN(C(C(C)(C)C)=O)CC2CC(F)F)=O)ncn2c1CCCC2 C(=O)(CS(=O)(=O)CCO)N1CCCC(N(C(=O)C2CC2)CC)C1 N1(C(c2scc(C)c2C)=O)CC(CC(=O)NC2CC(C)(O)C2)CC1(C)C c1(CC)[nH]c(=N)sc1C(=O)NCC1(CNC(c2cnc(C)nc2)=O)CC12CCC2 c1(OCC(=O)NCC=C2CCN(C(C3C(C(C)C)C3)=O)CC2)ccc(F)c(F)c1 C=C(C)CCC(=O)NC1CCCC1N1CCN(C(C2CC3CC3N2C)=O)CC1 N1(C(CN(C)C(c2ccsc2)=O)=O)CC2(CCCN(C(=O)CC3CNC(=O)C3)C2)C1 C=CCN=C(NCC1COCCN1CC)N1CCC(O)C(C)(C)C1 CC(C)C(C)CCNC(C1C2CN(C(=O)C(c3cncnc3)C)CC12)=O N1(C(CCC=C)=O)CCC2(CC1)CN(C(=O)CCCC1CCCC1)C2C(C)C N1(CC(=O)N(CC(=O)NCc2cc(C)on2)CCC)CCOCC1=O N1(C(c2ccc(C)cc2)=O)CCC2(CCCC2C(=O)Nc2ccc(C#N)cc2)C1 CC(C)C(O)C(=O)N1CCC(CN(C)C(C2CCN(C(=O)C3CC3)CC2)=O)C1 Cc1cc(C(=O)NC(CNC(c2nscc2Br)=O)C2CC2)nc(O)c1 C1(CNC(C2CC3(C2)CC3F)=O)CC2(CCC2)CN1C(=O)COCC(F)(F)F C1(CC)CCN(C(C2CCCC(=O)C2)=O)C(C(=O)NCc2ccsn2)C1 C#CC12CCC(C(=O)N(CCCN(C(=O)C(C)OCC)C)C)(CC1)CC2 Cc1cc(P(C)(C)=O)oc1C(N1CCOCC1c1cn(-c2ccc(F)c(Br)c2)nn1)=O C1(C(N2CCN(C3CN(C(CCC4CC(OC)C4)=O)C3)CC2)=O)CCCCCCC1 C(c1ccc(SC)cc1)=CC(N1C2C(CNC(C(C)N(CC)CC)=O)C(C2)C1)=O N1(C(C2(C(C)C)CCC2)=O)CC(C(=O)NC2CCN(C)C(=O)C2)CC(C)(C)C1 c1(Nc2ccc(C(=O)Nc3cnc(C)s3)nc2)ncnc2cc(C(=O)O)ccc12 CC1C(=O)CCC(C(N2CC3C(CNC(C4(CO)CCCO4)=O)C3C2)=O)C1(C)C CCCC(CNC(c1oc(CNC(c2[nH]ccc2C)=O)cc1C)=O)CCO C(CC(C(C)C)NC(=O)C(CNC(=O)COCCCCC)CC1CC1)OC C1(CNC(C2(F)C(C)C2)=O)COCC2(CCN(C(=O)CC3CC=CC3)CC2)O1 C1(CNC(c2cn(C3CCC3)nn2)=O)COC(C(=O)NCC2CC2)C1.C12CC(C1)C2 CC1=NOC(C(=O)NCC(O)CCNC(=O)COC2(C)CCCC2)C1C C1(=O)C(CNC(C)=O)NC(=O)N(CC)CCN1.c1(OC(C)(C)C)nnsc1N CCCCCC(=O)N1CC=CC1C(N1CCC(C(=O)NCc2ccsc2)CC1)=O c1(OCC)nc(NC(C)(C)CCNC(=O)C(C2CCC(=O)N2)C)ncc1C O=C1OC(C(=O)Oc2cccc(C3CCCC3)c2)Cc2cc(C(F)(F)F)ccc21 C(CCC)(C(=O)N1CCC(=CCNC(C2(n3cnnn3)CC2)=O)CC1)=CCC c1(CC(N2CCC(NC(CC(C)SC)=O)(CF)C2)=O)ccc(Cl)c2cccnc12 C(=O)(C#CC1CCCCC1)NC(CC=C)CNC(=O)Cc1cncnc1 C12(CNC(CSC)=O)CCC(CC1NC(=O)Cn1cnccc1=O)C2 C(CCCCC(=O)NCc1cccc(C(=O)N(C2(c3cc[nH]n3)CC2)C)n1)SC CC1CC(C(=O)NCC(C)N(C)C)N(C(=O)CCCn2cncn2)C1 C1(NC(COCCCCC)=O)CCN(C(c2cnn3c2CCCC3)=O)CC(O)C1 C1(O)(C(=O)NCC2C(NC(c3c(OC)cc(C)cc3)=O)CC2)CCC(C)(C)CC1 Cc1cc(CCCC(=O)NC2CCCC2NC(=O)CC(C)c2ccccc2)on1 c1(C(N2C(C)(CNC(=O)C(O)CF)CCC2)=O)ccc(F)c2ccccc12 C1(CCC(=O)NCc2cc[nH]c2C(=O)N(CCCO)C2CCC2)CCCOC1 CC(C)(C(=O)NCc1ncco1)C1=CCN(C(c2ccc([N+](=O)[O-])o2)=O)C1 C=CCCC(C)(C)C(=O)NCC1C=CC(NC(=O)CCOCC2CCCO2)C1 c1(CC(C)NC(=O)C(=O)NCC(=O)Oc2ccc(Cl)cc2)csc2ccccc12 Cc1cc(C)c(C(=O)NCC(C)(O)CNC(=O)C(C)N(C)C)c(O)c1 c1(C(=O)NC(C(CO)NC(CC2CCN(CC)C2)=O)C)cccc(OC(F)F)c1 Cc1cnc(NCCCC(C)CO)c(S(=O)(=O)NCC2CC(=C3CC3)C2)c1 c1(CN(C(CCN(C(=O)C(O)C=C)CC#C)=O)C)cccc(C)c1 c1(N2CC(CN(C)C(c3csnc3Cl)=O)OCC2)ncc([N+](=O)[O-])cc1C(N)=O CCCC(C(=O)N1CC2(NC(C3CC3c3ccncc3)=O)CC1C2)NC(N)=O c1(C(=O)N2CC(n3cc(-c4cccnc4)nn3)CO2)nccc2c(Cl)cccc12 C(=O)(C(C(C)(C)O)NC(=O)CC1CCSCC1)NC(C#C)CC1CCC1 N1(CC(=O)NCC2C=CCN2C(C2CC2(F)F)=O)CCCC2(CC2)S1(=O)=O N1(C(C(C#N)C2CC2)=O)CCC(O)(CNC(c2ccc(OCCF)cn2)=O)C1 c1(C(=O)OC)ccc(CN2CCN(C(=O)Cc3ccccc3)CC2)cc1C C1(C(=O)Nc2cccc(C(N)=O)c2)CC12CCN(C(=O)CC1CCNC1)CC2 C1(CNC(CSCC#C)=O)CN(C(c2cccc(C(=O)NC)c2)=O)CCC1(F)F N1(c2ncc(C)c(C)n2)CC2CCCN(C(c3ccccn3)=O)C2C1 Cc1nn(-c2ccccc2)cc1C(=O)NCCNC(=O)COCCCF N1(C(c2n(COC)ncc2)=O)CCC(F)(C(=O)NCC(c2ccccn2)O)CC1 N1(C(C=Cc2c(C)ncs2)=O)CCCC(NC(C2(O)CC2)=O)C1C C=C(Br)CN=c1[nH]c(=NCc2ccccc2S(C)(=O)=O)c2ccccc2[nH]1 c1(C(=O)NCC2(NC(c3c(C)c[nH]n3)=O)CCCCC2)cc([N+](=O)[O-])nn1C C1(CC(=O)NC)CCN(C(=NCCC2CCOC2C)NCCCF)CC1 CCC(C)(C)CC(=O)NCC(C)(C(C)C)NC(=O)Cc1ncc(Cl)s1 C(CC(C)C)(C(=O)NC1(C)CC1)N1CCC(n2c(C)ccn2)CC1 c1(C(=O)NCC(C)(CNC(C2(CO)CCOC2)=O)OC)cc(C)c(C)c(C)c1 N1(C(CCc2onc(C)n2)=O)CC2CC1CN2C(C1CCC(=O)N1)=O c1(CC(=O)NC(CCCNC(C2CC(C)C2)=O)C)cccc([N+](=O)[O-])c1 c1(OC)ccnc(OC)c1S(=O)(=O)N1CCC(S(N)(=O)=O)CC1 c1(C(=O)NC2CN(C(CCOC(C)=O)=O)CC(O)C2)[nH]c2ccccc2c1Cl c1(C(=O)NC2C3OCC(NC(CS(CC)=O)=O)(C3)C2)cc(S(N)(=O)=O)c[nH]1 C1(C(N2C(CNC(=O)CC(O)C3CCCC3)CCC2)=O)CCc2cncn2C1 C1(F)(CNC(C2(C)C=CCC2)=O)CCCN(C(C2CC3(C2)CC(O)C3)=O)C1 N1(C(C2N(C(C)=O)CCCC2)=O)CCC(NC(=O)CCSCC(C)C)C(F)C1 C1(NC(C2C=CCC2)=O)CCC2(CC1)CN(C(C13CCCC1C3(F)F)=O)CCO2 N1(C(COCCC)=O)CCC(C)N(C(=O)CC(O)C(C)CC)CC1 c1(C2CCN(C(C(=O)NC(c3nncn3C)C)=O)C2)ccccc1Cl N1(C(C(F)=CCC)=O)CC(NC(c2ccc(CN3CCOCC3)cc2)=O)C(F)C1 C1(C(=O)NCc2ccc(C(=O)NC3(CO)CC3)nc2)CN2CCC1C2 C1(C(=O)NC2C(CCC)CN(C(=O)OC(C)(C)C)CC2)CC1C1CC(F)(F)C1 C12CCCC1OCCNC2=O.C(=O)(C(F)(F)F)NCC#N c1(C(=O)NCCCC(C)(C)NC(CC2CC(OC)C2)=O)cc(C)cc([N+](=O)[O-])c1N C1(NC(c2c(C)nco2)=O)CC(O)CN(C(=O)CCOCC2CC2)C1 c1(NC(c2cc(C(C3CCOCC3)C3CC3)on2)=O)cccc(N2CCC2=O)c1 c1(C(N2CCC(Cn3cc(-c4ccc(C)cc4)nn3)C2)=O)cccc(C#N)c1F N1(C(CCc2nc(=N)[nH][nH]2)=O)CCOC(CCNC(=O)Cc2ccnnc2O)C1 Cc1cc(C(=O)NC2COCCC2NC(C2CC2C)=O)nn1-c1cccc(Cl)c1 CCC(CCCC(=O)N1CC(C)=CC(C)C1)NC(c1cn(CC)nn1)=O Cc1cc(C)cc(C=CC(=O)NC(C)C(C(C)C)NC(c2ncccc2F)=O)c1 C1(C(N(CCN(C)C(c2ncccc2N)=O)C)=O)CC2CCC(C1)S2(=O)=O c1(C(=O)NCc2nc(CNC(=O)C=C3CC3)nc(O)c2)cnn2cc[nH]c(=O)c12 c1(C(=O)NCC2C(NC(C(C)Cn3cccn3)=O)CC2)cc([N+](=O)[O-])n[nH]1 C#CCC(C)C(=O)N1CC(N2CC(NC(=O)CCc3c(C)n[nH]c3C)CC2=O)C1 C1(N(C(C2N(CCC)CCC2)=O)C)CCC(CNC(c2ncccc2Cl)=O)CC1 c1(C(N(C2CCN(Cc3ccn(C)n3)C2)CC)=O)c(F)cccc1F C1(CNC(CN2CC(=O)NCC2)=O)CC2CCC(C1)N2C(=O)Cc1ccno1 N1(C(c2c(CC)c[nH]c2)=O)CC(C(=O)N(C)CCc2cccs2)CC(C)C1 CCC(C)(C(=O)NCCC1CCCCN1C(=O)COCc1ccncc1)C(F)F CONC(=O)C(=O)N1CC(=O)CC1C(=O)NCc1c(F)cncc1F C1(OC)CCC2(CCN(C(C3CC=CCC3)C(=O)Nc3c(C)cccc3C)C2)C1 S(=O)(=O)(c1cccc(Br)n1)N1C(C(=O)Nc2cncc(Br)c2Cl)CC2(CC2)C1 N1(C(C(C)C2CCC2)=O)CC(NC(c2ccn(C)c2)=O)CC12CCC2 C(N=c1[nH]cncc1OC)C1C(NC(CNc2ccc(C#C)cc2)=O)CCCC1 CCC(CCCC(=O)NC1(c2ncc[nH]2)CC1)NC(=O)C=CC1CCOC1 c1(C(N2CCC(F)(C(=O)NCC=CCCC)CC2)=O)ccc2c[nH]nc2c1 C1(C(=O)NCCCOCCC(=O)NCC2CC2CO)CCC(=O)O1 C1(CNC(c2sc(C(=O)OC)c(N)c2)=O)CN(C)CCN1C(=O)C(C)OCC(C)C c1(COC(c2cc(OCC)c(Br)cc2)=O)c(C)nc(C(C)CC)nc1C C(=O)(C(F)CC1CN(C(C2CCCOC2)=O)C1)NC(C(=O)OC)C1CC1 C(=O)(C1(C)CCn2c(C)nnc21)N(CCCCN(C(C(C=C)O)=O)C)C N1(Cc2ccc(OC)nc2)CCC2CN(C(c3cccnc3)=O)CCC12 C1(C(C(=O)N(CCOCCC(=O)NCC(COC)O)C)C)CCC(=O)N1 c1(-c2n(CC=C)c(N(CC(C(C)C)OC)C)nn2)cnn2c1CCCC2C Cn1ccc(C(N2CCN(CCNC(=O)C(C)(C)CCl)CC2)=O)c1C1CNC1 CC1CC(NC(=O)Cn2[nH]cnc2=N)CN(C(C2(N(C)C)CCCCC2)=O)C1 C(c1cccc(Cl)c1)=CC(=O)NC(CC)CNC(=O)CCC(=O)NC n1(CC(=O)NCC(CC)NC(=O)C(C)OC(C)=O)cc(C(=O)O)cn1 N1(C(C2CCC(=C)CC2)=O)CC2(CNC(=O)C(CC)C(F)(F)F)CC(F)(C1)C2 c1(C(=O)NCCCCCN(C(C2(COC)CC2)=O)C)cnc(O)c2ncccc12 N1(C(C(CCOC)OC)=O)CCC2CCC(C1)N2C(=O)CC1CC(F)(F)C1 C(=O)(C(CNC(=O)CCC1CC1C)CC(C)C)N(CCCO)CC c1(C(=O)NC(CNC(C2C(C(=O)OC)C2)=O)C2CC2)cc2ccncc2[nH]1 CCCCC(CC)CC(=O)N1CC2CC(C(=O)NC3C(C)CCC3C)CC2C1 N1(CC(C2COC(=O)N2)ONC(C2CCCCC2)=O)CCCCC1C1CC1n1cncn1 CC12CCC(C(=O)NCC3(CNC(c4[nH]ccc4C4CC4)=O)CCC3)(C1)OC2 N1(C(C(CC)COC)=O)CCC2(CCC2)C(NC(c2cccc(CF)c2)=O)C1 CC(CN(C)C)C(=O)NCC1(CNC(c2cnc(C3CCOC3)s2)=O)CCC1 c1(CC)ccc(C(=O)NC(CO)CCCCNC(C2CC(C3CC3)C2)=O)c(C)c1 C(=O)(CC(C)(C)COC)N(C1CCCN(C(=O)CCCCc2cnc[nH]2)C1)CC Cc1cn2nc(C(N3CCC(NC(c4coc(Br)n4)=O)C(F)C3)=O)cc2c(=O)[nH]1 CC(C)C(C(=O)NCc1cscn1)NC(C1CN(C)C1)=O c1(OCC)nc(C)c(C(=O)NC2CCN(C(=O)CCC(C)OCC)C2C)s1 C(CC)(CC)(CCNC(=O)C(C)(C)Oc1cccc(Cl)c1)NC(C(F)=CCC)=O N1(C(C2C(C)=C2)=O)CCC(N(C(=O)CC2CC2)C)C1 c1(C(N(C(C(C)C)CO)C)=O)ccc2c(c1)N(C)C(=O)CO2 C(N=c1cc[nH]c(C(C)C)n1)C1(c2c(C)cccc2)CCC1 N#Cc1nc(Cl)ccc1NC(C1CC(F)CN1C(=O)CCN1CCCCC1)=O C1(C(N2CCCC(O)CC2)=O)CCN(C(=O)C2(C3CC3)CCCC2)O1 C(C(C)C(=O)OC)SC.C1(=O)C(=O)NCCOCCN1 c1(C(=O)NCC2(OCCNC(C3C(C)C3C)=O)CCOCC2)ccc2cncn2c1 c1(OC)cccc(F)c1C(N1C(C(=O)Nc2cc(Cl)cc(Cl)n2)CC2CC12)=O C(=O)(C1Cc2ccccc21)NCC1OCCN(C(C2(S(N)(=O)=O)CCCC2)=O)C1 O=C1CC(C(=O)NC2(CO)CCN(C(C3CC(N4CCCC4)C3)=O)C2)CN1O Cc1nc(C(N2CCC=C(C(=O)N(C)C[Si](C)(C)C)C2)=O)ccc1C#N c1(CN(CCCNC(=O)CO)C(=O)Cc2csc(S)n2)cccnc1 N1(C(C(C2(O)CCC2)NC(C=CCOC)=O)=O)CCC1(C)COC C1(NC(C2(C3CCCCC3)CC2)=O)CC1C1CCCN(C(c2ns[nH]c2=O)=O)C1 c1(C(=O)NC(CNC(c2[nH]cc(C)c2C)=O)C(C)C)nnc(O)nc1O c12sc(nc1-c1ccccc1)[nH]c2=O.C(=O)(C(C)N(CC(F)(F)F)C)OC CC(C)CC(C(=O)N(C)CCNC(c1ccc(-c2ccncc2)cc1F)=O)C(N)=O CC1OCCC1CC(=O)NCC(=O)NCC1CCCS1 c1(SC)ccc(O)c(C(=O)NC(C2CN(C(c3n[nH]c(C)c3C)=O)C2)C)c1 Cc1cc(Cl)cc(C)c1OCC(N1C2CCC1CC(NC(=O)CCC(C)C)C2)=O c1(CCC(=O)NC(C(C)C)(C)CNC(c2cc[nH]n2)=O)ccc2cnn(C)c2c1 N1(C(C(CCC)C)=O)CCC(NC(=O)CNC(c2cccc(F)c2)=O)C1(C)C Nc1cc(C(N2CCCCCC2CNC(=O)C=C2CCOCC2)=O)cc(Cl)n1 C(=O)(CCCCc1ccc(F)cc1)N1CC(CC(C)NC(C2COC(=O)O2)=O)C1 c1(C(=O)NCC2CC(OC)CN2C(c2ccsc2)=O)ccc([N+](=O)[O-])[nH]1 c1(OC)nc(C)ncc1C(=O)NC1CC2CCC1(CNC(c1cc(Cl)no1)=O)C2 C1(CC)CCN(C(=O)C(NC(C2CC(C)C2)=O)SC)CCO1 c1(C(C(=O)N2CC(CNC(C(=O)NCC)=O)C2)(C)C)ccc(Cl)c(Cl)c1 C1(C(=O)NC2(CC)CN(C(=O)Cc3ccc(C)cc3)C2)(OC)CCCCC1 C1(C(N2CC(OC(=O)NCC)C2)=O)CCCCCCN1C(c1cncs1)=O c1(OCC)nc(N(CC(C)CNC(C2CCCN2CC)=O)C)ncc1C Cc1cnc(C)c(C(=O)NCCC2CN(C(=O)COC3CCOCC3)CCO2)c1 C(=O)(CCC(CF)CF)NC(C(=O)N(C)Cc1snc(C)n1)(C)C1CCC1 c1(CN(CC(=O)N(CCNC(c2cn(CC)nn2)=O)C)C)cccc(C#N)c1 N#Cc1cccc(OCC(=O)NC(=O)C=Cc2ccco2)c1.C(CN(CCO)CCO)N c1(C(N2CC(C)C(CNC(=O)CN3CCOCC3)C2)=O)cc(C(N)=O)cc(F)c1 C#CC1CN(C(C2CCC(C(C)C)N2C(=O)CNC(=O)CN(C)C)=O)CCO1 n1(CC(=O)NC2(CCNC(CCC)=O)CC2)ccc(O)nc1=O C1(NC(COCCC#C)=O)CC(CO)N(C(=O)Cc2ccccc2)C1 CC1CCCC(C)N(C(C2CCCO2)=O)C1.C1(C=O)CC12CCCCC2 c1(OC)ccc(C(c2nnnn2C2CCOCC2)NCC2COC(=O)O2)c(C)c1 C1(C(=O)NC2CCC(F)(CNC(c3cnn(C)n3)=O)C2)CCC(=C(F)F)CC1 C#CCC(CC(=O)N(C)Cc1ccco1)NC(=O)CC1CC2C=CC1C2 c1(OCCC)cc2c(cc1CNC1CCN(c3nc(O)n[nH]3)CC1)OC(C)C2 CN1N=CC(CC(=O)NCC2CC(C(=O)NC3CCCC(CO)C3)CO2)C1=O Cc1cc(C#N)sc1C(N1CCC(N(C(=O)C(c2ccccc2)F)C)C1)=O C(=O)(C1CCCc2nncn21)N(CC(C)N(C(Cc1cccc(OC)n1)=O)C)C c1(OC)ccc(C(=O)NC(CNC(c2csnc2C)=O)C2CC2)c(F)n1 N1(C(C(C)=CC2CC2)=O)CC(CNC(c2nccnc2N)=O)C2(CC2)C1 CC1(C)OCC2CC12C(=O)NC1CCN(c2ccccc2Cl)C1 Cc1nc(N)cnc1C(=O)NCC1CCCC(CNC(c2csc(O)n2)=O)C1 N1(C(C(C#N)=CC(C)C)=O)CCC(C)(C)C(CNC(C2CCOC(C)C2)=O)C1 C#CCC(CC#C)C(=O)N1C2CCC1CC(NC(C1COC(=O)C1)=O)C2 N1(C(c2n(C(C)C)ccn2)=O)CC(C(=O)NCC(O)CO)CC(C)C1 CC1(C#CC(=O)N2CC(O)CCC2C(=O)NCCCn2ccnc2)COC1 CC(C(=O)NCC1CCC1NC(=O)CCC1CCC1)c1cncs1 c1(N2CCN(c3c([N+](=O)[O-])cccc3)CC2)ccc([N+](=O)[O-])cc1Cl N1(C(C(C2CCCC2)OC)=O)CC(NC(c2cc(Cl)ns2)=O)C(F)C1 N1(C(C(C)CC(N)=O)=O)CCC(C(=O)N(C)C(C2CC2)C2CC2)C(C)(C)C1 C1(CC(=O)N(c2cnc(Cl)s2)C)CCN(CCN(S(C)(=O)=O)C2CC2)C1 c1(C(N2CCC(NC(CCC=C(C)C)=O)C2(C)C)=O)cc(O)cc(C#N)c1 C#CC(C1CCc2ccccc21)NC(=NCC=C)NCC(=C1CCOCC1)F C1(CNC(C(C)OCC)=O)C2CN(Cc3ncnn3C)CC12 C1(C(=O)NCC(COC(C)C)O)C2CCN(C(=O)Cn3ncnn3)CC12 C12(C(=O)NC3C(C)OCC3)CC(CO1)N(C(=O)CCCC1CC1C)C2 c1(OC)ncnc(OC)c1C(=O)NCC1CN(C(c2ccc(Cl)cn2)=O)CC1C c1(C(=O)NC(C(c2ccccc2)NC(C=NOC)=O)C)ccc2nccnc2n1 c1(C(N2CCC(C3N(C(c4c(OC)scc4)=O)CCC3)C2)=O)cc(Br)n(C)c1 Cc1cccc(C(N2CC=CC(NC(=O)Cc3ccoc3C)C2)=O)c1N C(=O)(C(F)(F)C(F)F)N1C(C(=O)NC2CC(Cl)(Cl)C2)CC2CC21 n1(CC)cnc2[nH]c(=NC(C)c3cncs3)nc(N3CCCOC(CCO)C3)c12 O=C(C1=CC2(CCOCC2)C1)N1CC2(CCN(C(c3ncoc3C3CC3)=O)C2)C1 C1(COC)CN(C(c2cc(N)ccn2)=O)CCN1C(c1sncc1C)=O c1(NC2(c3n(CC=C)nnn3)CC(C(C)C)C2)cnc2ncccc2c1 c1(NCC2C(C)CN(C(c3cnc[nH]3)=O)C2)nc2c(cc1C#N)CCC2 C1(NCCCn2c(C(C3CC3)NCCC=C=CC)nnn2)COCCN1S(C)(=O)=O N1(C(C(CC)=CC)=O)CCC(O)(C(C)CNC(C2CN(C(N)=O)C2)=O)C1 C1(C(N2CCC(NC(=O)CCN3CCCCC3=O)(CO)C2)=O)CC2OC1C1CC21 C1(CC)CN(C(C2CCS(=O)(=O)C2)=O)CCN1C(C1CN(C(N)=O)C1)=O N1(C(C(C)CC2CCC2)=O)CCC2(CCCN2c2ncnc(=N)[nH]2)C1 C12(C(=O)NCC3CN(C(c4c(C)ncs4)=O)C3)CCC(CC1)C(C)(C)O2 c1(C(N2CCC(O)(C(C)NC(c3c(C)csc3)=O)C2)=O)ccc2ncn(C)c2n1 C1(O)(C(C)NC(=O)C2=CCSC2)CCN(C(c2cc(C3CCOC3)[nH]n2)=O)CC1 CCCC(CC)C(=O)N1CCN(C(c2cc(F)ccc2NC)=O)CC1C C#CCCN=C(NCC1(OCC)CCOCC1)NC1CCC(C#C)CC1 c1(C(N2CC(COC)N(C(C3CNC(=O)C3)=O)CC2)=O)cc(C)c2n[nH]cc2c1 C(=O)(C1=C(Cl)CCC1)NCC(C)CNC(=O)C(CN(C)C)N(C)C Cc1[nH]nc(C(=O)NCC2CCN2C(C2(c3ccn(C)c3)CC2)=O)c1C Cc1c(C(=O)NC(C)CCNC(=O)Cc2ccsc2Cl)sc2cncn12 c1(OC)ccc(C(=O)NC2CCN(C(C34C=CC(CC3)C4)=O)C2)c(F)c1 N1(C(C=NOC)=O)CC2(CCCC2NC(=O)C2=CCCCC2)C1 N1(C(C2(C)CCC2)=O)CC=C(CNC(C2Cc3nnsc3S2)=O)CC1 CCCC(CNC(=O)CC1COCCN1C(c1cccc(F)c1N)=O)CCC CC1(C)COCCC1C(=O)C(CC1CC(C(=O)NN)C1(C)C)=O.c1(C2CC2)cc(C)n[nH]1 C(=O)(CC(C)(C)CCC)NCCOCCOCC(N1C(C)CCC(OC)C1)=O C1(NC(C2(C)CC=CCC2)=O)CCN(C(c2cc(O)ccc2Cl)=O)CC1F C(=O)(CCCCC(N)=O)NCC1CCCC(NC(C(CN(CC)CC)F)=O)C1 N1(Cc2cc(C(=O)O)cc(Cl)c2)CCC2CN(C(c3ccno3)=O)CC2C1 C1(N(C)C(c2cc(C3CC3)ns2)=O)CN(C(C2(N(C)C)CCOC2)=O)CC12CC2 C1(OCC)CCC(c2nc(-c3nc(C)cs3)nn2C2CCCC2)CC1 c1(C(=O)NC2C(CNC(c3ccc4snnc4c3)=O)C2)cc2c(Cl)ccnc2s1 c1(C(=O)NCC2(O)CN(C(c3cnc(CC)s3)=O)C2)ccc([N+](=O)[O-])o1 S(=O)(=O)(c1ccc(-c2cnc(C(=O)NCC3CNCCO3)cc2C)cc1)NCC C(=O)(C(C)(O)C(F)(F)F)NCC1N(C(C2CCN(CC)C2)=O)CCCC1 c1(C(=O)NCC#CCNC(C(CC=C)C)=O)cc2c(=O)[nH]c(C)cn2n1 N1(C(CC(=O)NCC)=O)CCC2(NC(=O)Cc3cc(F)ccc3O)CC2C1 C1(NC(c2cccc(C(=O)NC)n2)=O)CCCN(C(=O)C(F)n2ccnc2)CC1 C12(OC)CCC(C(=O)NCCCN(C)C(C3CC4(C3)CC4(F)F)=O)(CC1)C(=O)C2 N1(C(c2cnc(COC)s2)=O)CCC2(C1)CN(C(C1CCOC1C)=O)CCO2 C1(CC(=O)NC2(CCC)CCNC2=O)CN(C(c2c[nH]nc2CC)=O)CCC1C N1(C(C(C)CC2CCCCC2)=O)CCC(NC(c2cc(Cl)cc(Cl)c2)=O)C12CC2 C(=O)(CCCS(=O)(=O)N1CCCC1)N1C2CCC(NC(C3=CCCC3C)=O)(C2)C1 C1(NC(C(CCC)NC(C)=O)=O)CCCC12CN(C(c1cnn(CC)c1Cl)=O)C2 C1(CNC(CC)=O)CC(F)(F)CN1C(=O)C(C)C(F)(F)F Cc1ccnc(C(N2C(C(=O)NCCc3cccc(O)n3)CCC2C)=O)c1F n1(CCNC(C2(C)CCC2)=O)ccc(C(F)F)n1 N1(C(C2CC(=C)C2)=O)CC(C)(C)OCC1CNC(=O)COc1ccc(C)c(C)c1 C(CCC(=O)NC(CNC(c1ccc(C(F)(F)F)o1)=O)C1CC1)SC CC1CCN(C(=O)NCCc2cc(C(F)(F)F)ccc2Br)C(C(=O)N(C)C)C1 CC(C)C(C)(CNC(c1cc(C2CCC2)no1)=O)NC(C1CC(F)(F)C1)=O C1(C(N2C(CNC(c3cc(C(F)F)cs3)=O)CC(O)C2)=O)CC2C=CC1C21CC1 c12cccc(c1)N(CCNC(c1cc(C)cs1)=O)C2=O.c1(CC)ccc(C)cc1 C1(NC(C(CCC)C#N)=O)C2CCCN(C(=O)C3=CCSC3)C2C1(C)C c1(C(N2CCCC(C(C)NC(c3cc(CC)nn3C)=O)C2)=O)c(C)cncc1C C1(c2n(CC(=C)C)nnn2)(NCC2CCC3(CCC3)O2)CC2OC(C)(C)OC2C1 Cc1cccc(CC(=O)NC2CCC2NC(C23CC(F)(C2)C3)=O)c1Br C=CC1CN(C(c2cnc(OC)c(C(F)(F)F)c2)C(=O)NC2CCC2)CC1O C(=O)(C#CC1(C)CCCO1)NCCOC1CC(NC(C#CC(C)(C)C)=O)C1 C(CCC(C(=O)NC1CCCCCC1C)NC(=O)CC1CCOC1C)OC c1(N(C)C)ccc2c(c1)C1CN(C(=O)CN3CCOCC3)CC1NC2=O c1(CC)cccc(C2CCOC2C(=O)NS(=O)(=O)Cc2ccc(C)cc2)c1 Cc1ccc(CCNC(c2nnnn2C)(C2CCOC2)C)c(F)c1 C1(CN2CC(CC(Cc3c(C(=O)OC)ccnc3)=O)C2)C2Cc3ccccc3C12 Cc1nc(N2CCC(NC(c3cnoc3C3CC3)=O)C2C)c2c[nH]nc2n1 CC1CCN(N2CCCC2c2ccccc2)CC1C(N)=O c1(OC)cc(C(N2CCC(C)C2c2cn(CC(C)O)nn2)=O)ccc1C(F)F C1(C(=O)NC2CN(C(c3c(OC)scc3)=O)CC2F)CC2(C1)CC(CO)C2 C#CC1(O)CCCN(C(=O)CNC(=O)CN(C(=O)CCC2CCCOC2)CC)C1 c1(C(N2CC(NC(C3(CCCC)CC3)=O)C(C)(C)C2)=O)cc2c(C)n[nH]c2cn1 C1(C(N2CCCC(NC(c3n(CC)c(O)nc3)=O)C2)=O)COC(C)(C)CO1 Cc1cnc(COC(=O)Cn2cnnc2-c2ccccc2)nc1 N(C(=NCCCn1cncn1)N1CCC(Oc2ccncc2)C1)CCF c1(C(=O)NC(CC)(C)CNC(=O)CCCNC(N)=O)ccc(C(F)(F)F)cc1C CCC(CC(=O)N1CCCCC(N(C(=O)C=C2CCOCC2)C)C1)CC(F)(F)F c1(C(c2nnnn2C)NCC)cn(C)c2cccc(C)c12.N12CCN(CC1=O)CC2 C(C(C)(C)C#CC(=O)NCC1CCCNC1=O)NC(C(C(C)C)OCC)=O C1(N(C(=O)Nc2c(C(=O)OCC)oc(Br)c2)CCO)CC(C)CC(C)(C)C1 N1(C(C2CC(C(F)(F)F)C2)=O)CCN(C(=O)CCC2CC2(F)F)C(CO)C1 C1(N(CCNC(C(C)C)=O)C(c2ccsc2)=O)CCCCC1 C1(CNC(C2C(C)(C)C2CNC(=O)Cn2[nH]cnc2=N)=O)CCC(O)CC1 c1(C2C(C(N(CCC)CCNC(C3C=CCC3)=O)=O)C2)ccc(Cl)cc1 N1(C(CCN(C(CC2C(OC)CCCC2)=O)CCO)=O)CC2C=CCC(C2)C1 C(=O)(C1=Cc2ccccc2C1)NC1C=CC(CNC(CCCS(N)(=O)=O)=O)C1 S(=O)(=O)(c1scc(Br)c1Br)Nc1nn(C)c(C(F)(F)F)c1 c1(CNC(c2nc(C)oc2)=O)ccc(C(=O)NCCc2cn(C)nc2C)nc1 c1(C(N(CCC(=O)NC(CSC)C)C)=O)cc(O)cc(F)c1 c1(C(=O)NC(C2CCCN(C(c3c(OC)c[nH]n3)=O)C2)C)c(C)ccc(Cl)c1F C1(C(=O)NCC(C)(CO)NC(CC(CC)C)=O)CCN(OC)CC1 C(C(=O)NCCC1CCCN1C(c1cc(C)c(Br)o1)=O)(C(C)(C)C)OC C1(C)(C(=O)NCC(C)CNC(C2(O)CC3CC2C3)=O)CC(C#N)C1 N1(C(c2cc(C)ncn2)=O)CCC2CN(C(=O)Cn3cc(C4CCC4)nn3)CC12 N1(C(CC2(C=C)CC2)=O)CCC(F)(CNC(=O)C(F)(F)c2cccnc2)C1 C(=O)(C1c2c[nH]nc2CN1C(=O)CC(CC)SC)N(CCOCC)CC C=CCN=c1[nH]cc(C(N2CC=CC2CNC(=O)C(CSC)c2ccccc2)=O)s1 N1(C(CN(C2CC2)CC)=O)CCC(NC(=O)Cc2csc(C)c2)C(CO)C1 c1(CC(C(=O)N2CC(CNC(N)=O)C2)NC(C)=O)ccc(Br)cc1 O=C(NN1CCCC1C(N1CCC2CC1C(=O)O2)=O)c1nccs1 Cc1cc(C(=O)OC2CN(Cc3cnn(-c4ccccn4)c3)C2)c(Cl)cc1F C1(NC(Cc2cccc(COC)c2)=O)CN(C(=O)CC2CSC2)CCC1C C(CCC(=O)NC(CNC(N)=O)CO)NC(C1(NCC2CC2)CCC1)=O.CC(=O)NCC C#CCCC(C(=O)NCCCN1CCC1)NC(=O)CCOC(C)C CCC(C(C)(F)F)NC(c1conc1C(C)NC(=O)C(c1ccccc1)C)=O c1(C(=O)NC(CNC(CCCCC#C)=O)(C)CC)cc2cc(F)ccc2[nH]c1=O c1(OC)ccc(Cl)c(C(N2CC(O)(CCNC(=O)C(C)CN(C)C)C2)=O)c1N C(=O)(CS(=O)(=O)CCO)N(C1CCCN(C(CC(n2ccc(C)n2)C)=O)C1)C C12(NC(c3c(COC)noc3)=O)CCCC1N(C(=O)CCS(C)=O)CC2 C12(C(=O)NC3(CC=C)CCN(C(C4C5CC(=O)CC45)=O)C3)CCN(CC1)CC2 N1(C(C2CC(N(C)C)C2)=O)CC(C(=O)NCCC(O)CO)CC1(C)C c1(C(N(CCCNC(C23CC(C(C)C)(CO2)C3)=O)CC)=O)cc2ncccc2s1 Cc1cc(C)c(C(=O)NC(C)C(C(C)C)NC(c2[nH]nnc2C)=O)o1 C1(NC(C2(N(C)C)CCCC2)=O)CC(NC(C23CCCC2C3)=O)C(O)C1 c1(C(=O)NC2C(C)CCN(C(c3cc(COC)[nH]n3)=O)C2)ccc2cnsc2c1 CCC(CC(=O)N(CCNC(=O)Cn1nc(C)cc1C)CC1CC1)CC(C)C C1(C(=O)NC2C(NC(COCC(=O)OC)=O)COCC2)Cc2nccnc2C1 Cc1cccc(C(O)C(=O)NC(C2CCN(C(C3(C4CC4)CC3)=O)CC2)C)c1F N1(C(C=C(CCC)C)=O)CC(NC(c2[nH]c(=N)sc2C(F)(F)F)=O)CC1C N1(CC(=O)NC(C2CN(C(=O)CCC3(C)CC3)CCO2)C)CCC(C)(C)C1 C1(NC(c2c(CC)occ2)=O)CCCCC12CCN(C(C1CCSCC1)=O)C2 CCCC(O)CC(=O)NC(C)(CNC(=O)C=CC=C(Cl)Cl)CO Cc1ncnc(C)c1-c1cn(CC23CCCC2(CO)C3)nn1 c1(Nc2cc(C(=O)OC)cc(Cl)c2)ccc2c(c1)CC(=O)N2C C(c1cc(Cl)sc1Cl)=CC(N1CCCC1c1ccc(F)c(F)c1)=O C#CCCCCCC(=O)NCC1CC(C)CN(C(=O)CC2CCC(=O)CC2)C1 CCC(C)(CC)C(=O)NC(C1CCCN(C(=O)C(C)Sc2ccccn2)C1)C c1(N2CCC(NC(C3CC(C#C)(O)C3)=O)C(C)(C)C2)ncnn2c(Br)ccc12 C(=O)(CCC(C)(C)F)N1CCC(C)(CNC(C=CC=CC)=O)C1 N1(C(C(C(C)C)NC(CC(=O)NCC)=O)=O)CCC2(CCC2)CC1 C1(O)(C(=O)NC2CCC(CNC(C(C(=O)OC)C)=O)C2)CCCCCC1 c1(OC(N(C2CC23CC3)CCCN(S(C)(=O)=O)C)=O)ccccc1 c1(NCCN(C(=O)C(c2c(C)n[nH]c2C)C)CC)cc(C)ccc1[N+](=O)[O-] CCC(C)(CNC(=O)C(C)(C)CCNC(c1cn(C(C)C)cn1)=O)C(C)O C(=O)(C(F)(F)C1=CCOCC1)N1CCCN(CCNC(C(C)(C)C(N)=O)=O)CC1 S(=O)(=O)(CC(C#N)C1CCOCC1)NC1CCC(CCC(=O)OC)C1 N1(C(COCCOCC)=O)CC(NC(=O)C(c2ccc(F)c(Cl)c2)C)CC(F)C1 c1(C(N)=O)ccccc1C(=O)NCC1CN(Cc2ccncc2Cl)CCO1 C(=O)(C1=C(C2CC2C)N(C)C(=S)NC1c1c(C(=O)OC)cncc1F)OC c1(C(C(N2CC(O)(CN(C(C3CN(C(C)C)C3)=O)C)C2)=O)C)cccc(Br)c1 CCCC(C)(C)CC(=O)N1CCOC(CNC(c2cc(Br)cnc2O)=O)C1 c1(CNC(c2cnc(OCC)s2)c2nnnn2C2COC2)nc(Cl)cc(C)c1Br O=C(CC1=NNC(=O)C1)NCCC1CCCN(C(C2(C3CCOCC3)CC2)=O)C1 c1(C(=O)NC(C(=O)N(C(CC(=O)OC)C)C2CC2)C)cncc(OC)c1 c1(C(C)(C)CNC(=O)NCCN(CCO)Cc2ccccc2)cccc(Br)c1 C1(COC)(CNC(=O)CC2(O)CCCC2)CN(C(=O)CSc2nncn2C)C1 C1(NC(Cc2cc(C)sc2C)=O)CC2CC(NC(=O)CC3COC(=O)N3)C1C2 c1(C(=O)NCC2(O)CN(C(c3c(CC)n(CC)nn3)=O)C2)ncc(F)cc1F C1(C(N2CC(CC(C)NC(CNC(C)=O)=O)C2)=O)CC2(C1)NC(=O)NC2=O C1(NC(CCCCCC=C)=O)CCC2CCN(C(=O)CCC(C)(C)C)C1C2 C1(NC(C(C)C)=O)CC2CN(C(=O)C(c3cc(F)cc(F)c3)C)CC2C1 C1(CNC(c2n[nH]c(C)c2C)=O)CC2(CCC2)CN1C(=O)C=Cc1cscn1 C1(CC(=O)NCC2(CN(C(c3c(C)nco3)=O)C)CC2)CC(C)CC(C)(C)C1 C1(NC(COC(CC)(C)C)=O)CS(=O)(=O)CC1NC(=O)C(F)(F)c1cscn1 CC(C)(CCCNC(c1cc[nH]c(=N)c1)=O)NC(C1CCC12CCC2)=O c1(C(=O)NCC2N(C(Cn3nc(C)oc3=O)=O)CCC2)ncc([N+](=O)[O-])cc1C Cc1cc(S(=O)(=O)N2CCC(n3cc(C)nn3)CC2)c(C)cc1[N+](=O)[O-] C=C1CCN(C(c2ccc(C3CC3)cc2)=O)C(C(N2CC(F)CC2C)=O)C1 C1(C)(CNC(C2C(CC)C2)=O)CCN(C(=O)CC2CCCC2)C1 C1(C)(C(=O)NCCCCCC#C)CC(O)CN1C(c1c[nH]c(=S)cn1)=O c1(OCCCOC)ccc(-c2ccc(NC(=O)C(C)CSC)cn2)cc1 c1(CC)onc(C(=O)N(CC(O)CN(C(=O)C(c2ccc(C)s2)C)C)C)c1C CC1(CNC(C2(C3CC3)CCC2)=O)COCCN(C(c2cccc(Cl)c2F)=O)C1 c1(NC(NC)=S)nc2ncccn2n1 N#Cc1c[nH]c(C(=O)NCCOCCCNC(=O)CSc2nncs2)c1 C1(F)(CNC(c2c(CC)ncs2)=O)CCN(C(C2CCC23CCCO3)=O)CC1 c1(-c2cn(C(C(=O)OCC)C)nn2)ccc2[nH]ccc2c1 C12(Cc3ccc(C(=O)N(C4CC4)Cn4cccn4)o3)COCCN1C(=O)COC2 C1(CCOC)(NC(C(F)=CCC)=O)CCN(C(C2COC(C)C2)=O)CC1 C(C(C(=O)N(CCO)CCO)NC(C1CCNC1=O)=O)OCC N1(CS(CCN(CCC)C)(=O)=O)CCC2NC(=O)OCC2C1 C(=O)(CC1=NN(C)C(=O)C1)NC(CSC)(C)C(=O)NC1CSC1 C1(OC(=O)C(C2(C)CC2)NC(=O)OCC)CC2(CCCO2)C1 C1(C(=O)NCCN(C(=O)C(C2CCCCC2)C)CC)COCCC1(F)F C(=O)(C(O)CC(N)=O)NC(C1(O)CCN(C(c2conc2C2CCCC2)=O)C1)C C1(NC(COCC(=C)C)=O)CN(C(C2(CN(C)C)CC2)=O)C2(CCCOC2)C1 C(C(=O)N1CC(CNC(=O)CCc2cncs2)CC1C)(C(F)(F)F)OC(C)=O C1(NC(c2cnc(C)o2)=O)CCC(CN(C(=O)C(F)n2ccnc2)C)CC1 Cc1cc(C(=O)NC2(CCNC(C3CCOC(C)C3)=O)CCCC2)c(F)cc1N c1(C(=O)NCC(CC(C)C)NC(c2c(CCC)n(C)nn2)=O)cc([N+](=O)[O-])n[nH]1 Cc1nccc(C(=O)NCCCN(C(=O)C(O)C(C)C)CCO)c1N C(C)(CC(C)C(F)F)NC(C1(C(C)C)N(C(c2ccc(OC)nn2)=O)CCC1)=O C(=O)(CS(=O)(=O)N(C)C)N(CC(CC)NC(=O)C=CC1CCCC1)CC c1(OC)ccnc(C(N2CCC(N(C(=O)C(C)(C)SC)C)C2)=O)c1 Cc1cc2[nH]c(C(N3C4CCC3CC(NC(C3C=CCCC3)=O)C4)=O)cc2o1 c1(C(=O)NCC2=CCN(C(C(C)SC)=O)CC2)cccc2c1OC(C)C2 C(CCC(C)C(=O)NC(C)(C)CNC(c1cnc(C)c(C(F)(F)F)c1)=O)OC N1(C(c2ccc(SC)s2)=O)Cc2ccnn2CC(NC(=O)COC2CCOC2)C1 C1(NC(c2nn(C)c(O)c2)=O)CN(C(c2scc3c2CCCC3)=O)CC2(CC2)C1 Cc1ccc2c(c1)SC(C(N1CCC(NC(C34CC(C)(C3)C4)=O)C13CC3)=O)C2 c1(CC)cc(F)ccc1C(=O)N(C1CCCN(C(=O)C(C)NS(C)(=O)=O)C1)C c1(C(N2CC(C(C)NC(c3ccccc3O)=O)OCC2)=O)cnn2c1CCC2 c1(C(N2CC3C(C(=O)Nc4ccncn4)(C3)C2)=O)cc([N+](=O)[O-])cs1 Cc1[nH]c2ncccc2c1C(=O)NC(C)CNC(=O)CN1CC2CC2C1 CCCCCC(C)(CC)C(=O)NC1CCC(CN=c2[nH]cnc(Cl)c2CC)CC1 C1(CC=C)(NC(=O)CNS(C)(=O)=O)CN(C(=O)C(F)(F)c2cccnc2)C1 C(=O)(C(C)CC(C)C)NC1C(CC(=O)N(CC=C)CCOC)CCCC1 C1(C(=O)NC2CN(CC)C(=O)C2)CCCCCCN1C(c1ocnc1C)=O c1(-c2onc(-c3cc(C(F)(F)F)cc(N)c3)n2)cccc2nc(O)ccc12 N1(C(C(CCCCC)O)=O)CCC2CCCC(C1)N2c1cc(C(=O)OC)ncn1 Cn1c(C(=O)NCC2CN(C(C3(c4ccsc4)CC3)=O)CCO2)cccc1=O N1(C(c2nc(COCC)sc2)=O)CCCN(C(=O)C(=O)NCC(F)F)C(CO)C1 n1(NC(N2CCC(N(C)C(c3ccccc3)=O)CC2)=O)ncc(C(N)=O)c1N C1(CC(=O)NCC(CC)NC(c2cc(C(C)=O)cs2)=O)CCC(C)CO1 C1(NC(CCCc2cc(C)sc2C)=O)CCCC(NC(c2cnccn2)=O)CC1 c1(CC)ccccc1-n1nnnc1C(c1cnsc1)NCC1CC12CC2 C1(N(C(C(OC)OC)=O)C)CCC(NC(c2n[nH]cc2C2CC2)=O)CC1 N1(C(C2(CNC(C3(C)CCCOC3)=O)CC(=C)C2)=O)CC(C)CCCC1C N1(C(c2nc(C)oc2)=O)CCOCC1CNC(C1CC(=C2CC2)C1)=O CC1CCc2ncc(C(=O)NC3CCC3CNC(=O)CC3(n4cccn4)CC3)n2C1 C1(C(=O)NCCC(C(=O)NCc2ncn(C3CC3)n2)OC)CCCCC1(C)C N1(Cc2c(C)cccn2)C(=O)CCN(Cc2cccc([N+](=O)[O-])c2)C1=O CC1C(NC(=O)C=Cc2ccncn2)CCN1C(=O)CCOc1ccccc1Cl CCCCC(O)C(=O)N1CCC(C(C)(C)NC(=O)CC2(C(=O)OC)CCCC2)C1 c1(CN(CCOC)CCNC(C23CCCC2C3)=O)cccc(OCC#N)c1 Cc1cc(C(N2CCC(C(C)CNC(c3ccsn3)=O)CC2)=O)cc2ccoc12 CCC(C(=O)NCC1CCC(NC(=O)CCC=C(C)C)C1)C(F)(F)F c1(CSCCn2cc(CNC(C(C=C)OC)=O)nn2)cccc2c1NCCC2 C1(N(C)C)CCC(N=c2[nH]c(NC3CC4C=CC3CC4)nc3ncn(C)c23)CC1 N1(C(C(CCCC)CC)=O)C2CCC1C(CO)N(C(c1cc(OC)ncn1)=O)C2 N1(C(C(CCC)F)=O)CCC2CN(C(C3CCc4ncnn4C3)=O)C(C)C12 N1(C(C(C(=O)OC)C)=O)CCC(CNC(c2cc(CO)[nH]n2)=O)C(F)(F)C1 c1(NC(C2(CC=C)CN(C(=O)CNC=O)C2)=O)ccc(CO)c(F)c1 C1(C(=O)NC2CCC(C)(C)C2)(NC(Cn2ncc(C)c2)=O)CCCCC1 CC1OCCC1(F)C(=O)NCCC1CSCCN1C(=O)CC1CCC(=O)N1 C(C(=O)NNC(=O)CCCOCCCSC1CC1)SC(C)(C)C c1(CC(=O)NC2C(NC(c3c(C)cn(C)n3)=O)CC2)ccc2n[nH]cc2c1 n1(C(C(=O)NC(C(=O)OC)C2CCCC2)C)cc(CCOC(=N)O)nn1 Cc1noc2nc(C(N3CCN(C(c4cccnc4S)=O)C(C)C3)=O)ccc12 C1(NC(C(C2CC2(Br)Br)N(CCCC)CCOC)=O)CCOCC1 C1(NC(C(C)=CC)=O)CC2CCC1C(NC(=O)CC(C)CN(C)C)C2 Cc1nsc(N(C(=O)C2=CSCCO2)Cc2ccccc2)c1C#N c1(NC(=O)CCCC2CCCC2)cccc(NC(=O)C(C2CCCO2)C2CC2)c1 CC1(C)CN(C(C2(CC(F)F)CC2)=O)CCC1NC(=O)CN1CSCC1=O N1(C(C2N(C(C(COC(C)=O)C)=O)CCC2C)=O)CCCOCC1C c1(C2C(C(=O)NCC(C)NC(=O)Cc3cnn(C(F)F)c3)C2)ccc(F)c(Cl)c1 C1(NC(C(c2cc[nH]n2)N(C)CCC2CC2)=O)CCN(c2ccccc2)C1 C(CCCCCC(=O)NCC1CCOCC1)NC(c1c(C)c(F)cnc1)=O c1(C(=O)NCCC2OCCN(C(CC(CC)C)=O)C2)c(O)cc(Cl)cc1F C=CCCC(C(=O)NCCCSC)N1CCOC(CC(=O)OC)C1 c1(C(N2C(CNC(C(C(C)C)(C)C)=O)C(C)(C)CC2)=O)ccnc2cc[nH]c12 C1(C(=O)NCC(CC)CO)CN(C(c2cc(CO)oc2C)=O)CC1CC1CC1 C1(C2CCN(C(C3(C(N)=O)CC3)=O)C2)(NC(Cn2c(C(C)C)ncc2)=O)CC1 c1(OC)ccccc1C(C)C(=O)NC(c1nc[nH]n1)C1(C)CCC1 C1(NC(COc2cccc(C)c2)=O)CC2CC1CN(C(C1(C)CCC1)=O)C2 C1(CCCNC(c2n(CC=C)nnn2)c2cnn(CCOC)c2)CCC(C)(C)O1 CCCC(C)(O)CNC(C1CCC1NC(c1cc(CO)ccn1)=O)=O c1(C(=O)NC(C2N(C(CC3CC(=C)C3)=O)CCCC2)C)cccc2[nH]c(=N)oc12 c1(OC)cccc(C(C)=O)c1NC(C1CN(C(c2ncccc2C)=O)CCS1)=O c1(C(N2C(C)(C)C(NC(=O)CNC=O)CC2)=O)cnc(O)c2cccnc12 c1(NC(c2c(C)n[nH]c2)=O)ccc(Cl)cc1[N+](=O)[O-] CCC(C)CCCC(=O)NC1CC2(C1)CN(C(C1CCC1c1nncn1C)=O)C2 C1(C(=O)NC(CC)CNC(C2CC2C2CCCO2)=O)CC(=O)NC(=O)C1 C1(C(=O)NC(C)CCSC)(OC)CCN(C(c2nccnc2N)=O)C1 c1(OC)ccc(C(=O)NC2C3CC2N(C(C2(C)CC(=O)N(C)C2)=O)C3)nc1OC n1(CC)nnc2c1C(C(=O)N1CCc3cccnc31)CN(c1ncncc1I)C2 c1(C(=O)NCCC(C)NC(c2cnccc2C(F)F)=O)snc(O)c1Cl C1(CC(=O)N(CCC(=O)NCC2CSCCO2)CC)CCCN(C)C1 c1(CCOCC(=O)N(C2CCN(CC3CCCCC3)C2)C)cccc(Br)c1 N1(C(C(C)(C)CC#N)=O)CC2CS(=O)(=O)CC2(NC(=O)C2=NOC(C)(C)C2)C1 C(C(=O)NC1CCCC1CNC(=O)Cn1cccnc1=O)(C(C)C)SCC N1(C(c2nc(CC)oc2)=O)CC2CCC(CNC(=O)CCc3cnccn3)C2C1 C(C(C)(CC)C(=O)NCC(C)(O)C(F)F)NC(C1C(=C)C1)=O N(C)(C1CCc2ccccc21)C(c1n[nH]cc1C)C(=O)NC(CC)(C)C N1(C(C(CC)(C)O)=O)CCCC(F)(Cc2ccccc2)C1 c1(C(=O)NC2CCN(C(C(C)(C(C)C)NC(C)=O)=O)CC2)cnc2scnc2c1 N1(C(c2cnc(CC)o2)=O)CC(C)CCC1CNC(c1nccn1C)=O c1(OC)ccc(C(=O)NC(C)(C)CNC(C2SC3C=CC2CC3)=O)cc1C c1(N(C)CC2N(C(C(CC)(F)F)=O)CCC2)cc(S(C)(=O)=O)ncn1 C12(CNC(C(CC)CN(C)C)=O)CN(C(C3CCN(C)CC3)=O)CC1CCO2 N1(C(c2c(C(C)C)noc2)=O)CCC(C)(CNC(=O)CC2CCC2C)C1 C(=O)(C1=C(SC)CCCC1)N(C1CCN(C(C(CC)(C)OC)=O)C1)C CC1(C)CCC(C(=O)NC2COCCN(C(=O)CCCn3ccnc3)C2)OC1 C1(NC(c2c(C)cc(C3CC3)cc2)=O)CN(C(=O)C(C)O)CC2(CC2)C1 N1(C(c2ccc(OC)o2)=O)CCC(C)(C(=O)NCC2CC23CCC3)CC1 c1(C(N(C2CCCC(NC(c3cnccc3Cl)=O)C2)C)=O)ccnc(S)c1 c1(C(N2CC(O)(CN(C(C(c3cnn(C)c3)OC)=O)C)C2)=O)cncc(Cl)c1C C(=O)(C1CCCn2nccc21)N1CCN(C(CNC(=O)C2CC2)=O)CC1 C=C(C)CC(C(=O)OC)NC(C1CC(F)(CNC(=O)CCNC(N)=O)C1)=O CCCC(CC)C(=O)NC1C=CCN(C(=O)CSc2ccc(OC)cc2)C1 C1(C(=O)OCc2nc(C)sc2C)COC2(C)CC1C2 CCN=c1cc(-c2nc(C(O)CC3CCC3)n(CCc3ccccn3)n2)cc[nH]1 c1(CN2CCCC(NC(c3ccccc3I)=O)C2)ccc(Br)cc1CO c1(CC(=O)NC(CNC(CCc2ccc(C(=O)OC)[nH]2)=O)C)cnc(C)nc1O C1(C(=O)NC(C=C)COC)CCCCN(C(=O)C(C(C)C)SC)C1 C(CN=c1ccc(C)c[nH]1)NC(C(N1CCCC(COC)C1)=O)=O c1(C(N2CC(C(C(=O)NCCCn3cncn3)O)C2)=O)cc2cccnn2c1 c1(SCC)ccc(CC(=O)NC2(C)CCN(C(=O)C(O)Cc3cnc[nH]3)C2)cc1 C1(NC(C2C(C)(C)CCN2C(C2CC=CC2)=O)=O)CCCOC12CCC2 c1(C(N2C(C(c3cccnc3)Cc3cn(OC)nn3)CCC2)=O)n[nH]c(C)c1Br N1(C(C2(CC)CN(C(c3ccc(C#N)o3)=O)C2)=O)CC(C)CC(O)C1 CCCCCC(C)CC(=O)N1CCC(CCNC(c2c(C)ccc(Cl)c2N)=O)C1 C1(C(=O)OC)(CC)CCN(C(=O)C(C)N(C)C(C2(C)CC2)=O)C1 C(CN=c1nc(N2CCCC(c3cccnc3)C2)c2c([nH]1)COC2)(C(C)(C)C)SC C1(C)(NC(CC2(N(C)C)CC2)=O)CCN(C(=O)C=CC2CCOCC2)CC1 c1(C(=O)NCC(C)NC(C2(C)CC2c2ccccc2)=O)coc2cccc(O)c12 N1(C(COCC=C)=O)CC2CCCCC2(NC(c2cc(C3CC3)nn2C)=O)C1 c1(OC)ccncc1C(=O)NCC1CC(F)CN1C(C1CC1(C)C)=O c1(C(=O)NC2(C(N3CCC(CC=C)C3)=O)CC2C)cc(O)cc(F)c1 C(=O)(CC(C)(C)COC)NC(CNC(c1[nH]cc(CC)c1)=O)C1CCC1 C(=O)(C(O)CCNC(C1CCN(CCO)CC1)=O)NCCC(=O)NO c1(C(=O)OC)cc(C(c2nnnn2C2CCC2)NC(C)C(C)(C)OC)n(C)n1 N1(C(c2cccc(OCC=C)c2)C(=O)NCCC2CC2)CCC(C)(C#N)CC1 C1(N(CCCNC(C2CC2F)=O)C(C2CC2F)=O)CCCC1 c1(OC)cc(C(=O)NC(C)CN(C)C(C2CCOC2C2CC2)=O)cc(N)c1OC C12(C(N3CCC(NC(c4cccc(=S)n4O)=O)(CF)C3)=O)CCC(=O)N1CCS2 C1(C)(OCC)CN(C(=O)CNC(c2cncnc2)=O)C1.C12(CCC1)C(=O)N2 N1(C(C2CCCC(C(=O)OC)C2)=O)CCCC(C)(CNC(C2CCC(F)C2)=O)C1 C1(C(N2CCN(CCC)CC2)=O)COCCN(C(C23CC(COC(C)=O)(C2)C3)=O)C1 c1(NC(c2cc(Cl)cc(I)c2)=O)cc(Br)cc(Br)c1O c1(NC(CCC)c2nn[nH]n2)ccc(C(=O)NC(=O)C(C)(C)C)cc1 N1(C(C2(c3cc(C)no3)CC2)=O)CCC2(CCC(NC(C3CCC(C)C3)=O)C2)C1 N1(C(C(CC)=CC)=O)CCC(C(C)(C)C)(CNC(=O)Cc2nncs2)C1 C(=O)(CCCCCSC)NCC(C1CCCCC1)NC(c1ccc(COC)[nH]1)=O C1(NC(c2c(CC)ccs2)=O)CN(C(=O)C=Cc2c(C)coc2C)CCC1F c1(C(=O)Nc2cc(O)c(Cl)cc2Cl)ccn2c(C3CC3)cnc2c1 C1(NC(C(C=C)CC)=O)CN(C(=O)C(CC)N(C)C)CCC1(C)C c1(C(=O)NC(C(C)NC(C2CCC(CC)O2)=O)CO)cccc(N(C)C)c1 Cc1ccc(C(=O)NC2CCCN(C(=O)C(C)(O)C3CC3)C2)c(C)n1 C(=O)(C(C)P(C)(C)=O)N(CCCCCC#C)CC(N1CCOCC1)=O C(CC(C)C)(C(=O)NC(C)CS(C)=O)NC(CNC(CCC)=O)=O C1(C(=O)NCC2CC(C(=O)NCC3(C(=O)NC)CCC3)C2)CS(=O)(=O)CC(=O)N1 C1(C(C(=O)NC2(C)CC2)N(CCOC)CC#N)CC12CCOC2 C1(C(N(C(CNC(=O)C(F)(F)CC2CC2)C2CC2)C)=O)CCCC12CCOCC2 n1(CC(=O)N(C2CC(NC(C3C(CCC)CCC3)=O)C2)C)cc(C#N)cn1 CCC(C)CC(=O)N1CC2CC2(NC(=O)C(C)(C)COC2CCCC2)C1 N1(C(C2=C(C)OCCS2)=O)CCC2CCCN(C(=O)C=Cc3ncc[nH]3)C2C1 Cc1cc(C#N)cnc1C(=O)NC(C)C(C)NC(=O)CS(=O)(=O)N(C)C Cn1cc(Cl)c(C(N2CCOC(CCNC(=O)CC3CCCC3O)C2)=O)n1 C1(CNC(CC2(C)N(C(CC3CN(C(C)=O)C3)=O)CC2)=O)CCC(=O)NC1 C(CC(=O)NNc1nc(C(C)(C)C)no1)c1nc(C#N)cc(C)n1 N1(C(CCCCC)=O)CC2(CCC2NC(c2ccc(Cl)c(F)c2)=O)C1 CCCCC(O)C(=O)NCC12CC(CC)(CN1C(=O)C(CC)N(C)C)C2 c1(C(=O)Nc2ccc(C3CCN(S(=O)(=O)C4CC4)CC3)cn2)cnn2ccccc12 N1(CCCC(=O)NCC2C(CNC(C3CC(C)(C)C3)=O)C2)C(=O)CNC1=O C1(CC(=O)NCC2CC(O)CN2C(c2ccc(F)c(Cl)c2)=O)CCC(F)(F)CO1 N1(C(C(C(C)C)C)=O)CCN(C(=O)CCC2CC2(Cl)Cl)CC1C C1(C(=O)OC)(C(=O)NC2CCC(N(C)C(c3cnsn3)=O)CC2)CCOCC1 c1(C(N(CC(CC)NC(c2c[nH]nc2C2CCOC2)=O)CC)=O)nnccc1C c1(-c2c(C(=O)OC)scn2)ccnc(N2CCN(Cc3csc(Br)c3)CC2)c1 N1(C(C(C2CN(C(C3C(C)CCOC3)=O)C2)O)=O)CCC(F)(F)CC1 c1(NC(C(C)OCCC(C)C)=O)cccc(NC(=O)CC2CCC23CCC3)c1 N1(C(CCC(=O)OCC)=O)CCC(CNC(C2CC(O)C2)=O)C12CC2 N1(C(COc2cccc(C)c2)=O)CCN(C(=O)C(C)NS(C)(=O)=O)CC12CC2 c1(C(N2CCC(N(C(=O)C=C3CCOCC3)CCC)C2)=O)cc2sccc2n1C N1(C(C(OC)OC)=O)C(C(=O)NCC(C)(F)C(C)C)CC2CC12 Cc1cc(C(N2CC(CNC(C3(c4ccc(Cl)c(F)c4)CC3)=O)C2)=O)ccc1Cl Cc1[nH]c2ccccc2c1CC(=O)NC(C)CCCNC(C12CC(C)(CO1)C2)=O CC1=CC(O)CN(C(C2(CNC(=O)OC(C)(C)C)CCC2)=O)C1 Cc1cc(C)n(CC(=O)NC2CC(CCNC(C3CCCCS3)=O)C2)n1 C(=O)(C#CC1CCOC1)NC1(C(N2CC(=C)C2)=O)CCC(C)(C)C1 c1(OC)c(C(=O)N(C2CCCN(C(=O)CCC3CC(C)(C)CO3)C2)C)csc1C CCC(C)C(CO)NC(=O)C(C)N(C)C(C1CC2CCC2C1)=O N1(C(c2nccc(C)c2N)=O)C2CCC1CC(CNC(c1ccnc(F)c1)=O)C2 c1(C(=O)NCCN(C)C(c2cc(CC3CC3)[nH]n2)=O)c[nH]cc1-c1ccc(Cl)s1 C(=O)(C1CCCc2c1ncn2C)NCC(CNC(Cn1c(C)ccn1)=O)CO O=C(CC(CC1CC1)NC(C1CCC2(CC2)C1)=O)NC(c1ccco1)CO C#Cc1ccc(F)c(C(N2CC(OC)CC2CNC(=O)CC(C)CCC)=O)c1 c1(C(=O)NCCC(C)NC(=O)CC2CC(=O)NC2=O)oc2ccccc2c1CO C(CS(=O)(=O)CC(=O)NCCNC(C1CCC1C(N)=O)=O)OC c1(C(=O)NCC2CCC(C(=O)NCCCCCCO)CC2)cnc(O)nc1O C1(C(=O)NCc2cc(C)oc2)Cc2ccc(F)cc2C(=O)O1 c1(C(N2CCN(CC3CN(C(C(C)OCC#C)=O)C3)CC2)=O)nnc(O)cc1C c1(OC)ccc(F)cc1CCC(=O)NC1(CCNC(=O)CNC(C)=O)CCC1 C(CS(=O)(=O)C1CC1)NCC.C(CC=O)N(CC)CC c1(N2C(C)CCN(C(c3cc(O)nn3C)=O)CC2)cc(=O)n2cc(Cl)ccc2n1 c1(OCC(C)N(CCOC)C(C2CC(n3cc(CO)nn3)C2)=O)ccccc1Cl O=C1OCc2c(NC(C3(F)CCN(C(C4CCNC(=O)C4)=O)CC3)=O)cccc21 C=CCN=C(NCC#Cc1ccccc1)NCc1cc(C)oc1C N1(C(C=C(C)C2CC2)=O)CCCC(C2CN(C(=O)C(F)=C3CCC3)C2)C1 S(=O)(=O)(CC(=O)NC1CCC(C(=O)N(C(C)C(=O)N(C)C)C)C1)NC C1(CNC(C(C)=C2CC2)=O)CN(C(C2(N(C)C)CCC2)=O)CCC12CCOC2 c1(C(=O)OC)cnc2c(Br)cncc2c1NCC1CC2CCC1(C)C2(C)C O=S(=O)(c1cc(Cl)cc(Cl)c1)N1CC2(CCN(c3nccc(C(F)F)n3)CC2)C1 C1(F)(C(N(C2CCN(C)CC2)C)=O)CCCN(C(C2CC3(C2)CC32CC2)=O)C1 CCCCC(O)C(=O)NC(C)(C)CN(C)C(c1sccc1C(=O)OC)=O CC1=C(C(=O)NC2(C3CCN(c4cc(F)ncn4)C3)CC2)SCCO1 c1(C(=O)NC2C(C(=O)NC(C(=O)NC)C(C)(C)C)C2)cccc([N+](=O)[O-])c1Cl Cc1ccc2c(c1)SC(C(=O)NCC(C1CC1)NC(c1cc(C(F)F)no1)=O)C2 C=CC1(C(=O)NC2CCC(CCC(N3CCC(COC)C3)=O)C2)CCCCC1 C1(CC(N2CCOCC(NC(C3(COC)CCC3)=O)C2)=O)CCC2(CCC2)CO1 C1(C(=O)NC2CN(C(CCC(=O)N(C)C)=O)CC2O)CC(c2ccccn2)=NO1 CC(C)C(O)C(=O)NC(C)(C)CNC(=O)CCC1CCCC(=O)N1 n1(CCC)nnnc1C(c1csc(Cl)n1)NCC(C1CCCCC1)OC n1(CC(=O)NCC)cc(C2CC2)nn1.N12CCCC1C2.C1(C)C(=O)N1CC C1(CNC(=O)CC(F)F)CN(C(=O)Cc2csc(-c3ccc(F)cc3)n2)CCO1 c1(C(=O)NCc2ncn(C)c2)ccc(-c2ccc3ncsc3c2)c2c1OCO2 C1(CNC(C(COC)n2cc(C3CC4(CCC4)C3)nn2)=O)C2CC3C1C3C2C(=O)O Cc1cc(NC(=O)NCC2CCN(C(=O)OC(C)(C)C)CC2C)c(Br)nc1C c1(CC(=O)OCCS)cn(CC)nn1.CC(C)(C)OC(=O)CC1CC1 c1(NC(C2N(C(CCOC)=O)C3C(C2)C3)=O)cc(F)c(Cl)cn1 CC1CN(C(c2sc(N(C)C)nc2Cl)C(=O)NCC2CCOC2)CCS1=O Cc1c(C(=O)NC2CCCC(NC(=O)C(c3ncccc3F)(F)F)C2)cnn1C CCC(C)CC(C)C(=O)NC(CNC(=O)Cc1ccc(F)nc1)C1CC1 c1(CC)ccc(C(=O)N(CCC(C)NC(=O)C(c2ccc(Cl)nc2)(C)C)C)nc1 C1(C(=O)NCC(=O)OCC)C2CCCC2CN1C(=O)CC1C=CCC1.C1CC1 C1(CNC(=O)Cc2cnn(C(F)F)c2)CC2(CCC2)CN1C(C1CC2CC1C2)=O C#Cc1ccc(C(N2CC(O)(CNC(c3cc(OC)cs3)=O)C2)=O)nc1 CCCC(O)CC(=O)N1CC(CNC(c2cc(CC3CCC3)c[nH]2)=O)C(O)C1 C(=O)(C1=NN(C)C(=O)CC1)NCCN(CCOC)C(C1CCCC1(F)F)=O C(=O)(CCC(C)(C)C#N)NC(C(=O)N(C)Cc1ncc(C)o1)Cc1ccco1 Cn1nc(C(=O)NC2(CNC(=O)CC3CCNC(=O)C3)CC2)cc1C(N)=O C1(CCN(C)C(C23COC(CF)(C2)C3)=O)CCN(C(=O)CCC2CC2(Cl)Cl)CC1 C12(C(=O)NC(CNC(CCc3onc(CC)n3)=O)C3CC3)CCC(CC1)O2 CN1CCCC(O)(CC(=O)NCC2C3CN(C(c4cncn4C)=O)CC23)C1 N1(C(Cn2c(C)cnc2)=O)CCOC(C(C)NC(c2ccn(CCC#N)n2)=O)C1 CC(C)(CS(C)(=O)=O)C(=O)N1CCN(CC(C)(C)NC(C2CCOCC2)=O)CC1 N1(C(c2cnc(COC)s2)=O)CC(C2CCCCN(C(C3(C)CC3(C)C)=O)C2)C1 CCC(O)C(C)C(=O)N1CC(C)(NC(c2cccc(C(N)=O)n2)=O)C1 N1(C(CNC(CC(C)C)=O)=O)CCC(C)(NC(=O)C(C2CCCCC2)F)CC1 Cc1ccnc(O)c1C(=O)N(C)CCN(C(=O)CC1(C)CCCC1)C N1(C(CSC)=O)CC2(CCN(C(=O)C=CCNC(=O)OC(C)(C)C)CC2)CC1C C=C1CC2(C1)CN(C(=O)C(C1CCN(C(=O)C(CCCC)N(C)C)CC1)C)C2 C1CC(O)CC(=O)N1C.c1(COC2CCO2)ccccc1.CN(C)CCO N1(C(C(CC)CO)=O)CCCCC12CC(NC(c1ccc3nc(C)cn3c1)=O)C2 C1(N(C(=O)CCn2ccccc2=O)C(c2ccc(Cl)s2)C)CC2CCC(C1)N2 N1(C(C)C)CCC(NC(C2CC(=O)CN2C(=O)CC2CC(N(C)C)C2)=O)CC1 c1(C(=O)NC2CCCN(C(C(C)CC3CCC3)=O)CC2)cccc([N+](=O)[O-])c1Cl Cc1cc(F)ccc1N1CCN(C(C2(C)CCN2C(=O)CCC2CC2)=O)CC1 C1(CC)CCCC1(C)C(=O)NCC1CC(F)CN1C(c1cc(C(=O)OC)co1)=O c1(C(=O)Nc2nc(C(=O)Nc3cc(C)cc(C)c3)n(C)c2)cc(C)c(C)cc1C c1(C(N2CCN(C(CCC)=O)C(Cc3ccccc3)C2)=O)c(Cl)ccc(F)c1N N1(C(c2ncc(N(C)C)nc2)=O)CCCC2(CCN(C(C3(C)C=CCC3)=O)C2)C1 N(C(=NCCC(C)C1CC1)NCCc1cc(Cl)ccc1Br)C(C)C1CC1 N1(C(CCN)=O)CCC(O)C(C)C1.C1(NC(COC(C)=O)=O)(O)CCC1 C(=O)(C(F)(F)C(C)(C)O)NCCCCC(C)NC(C1C=CCCC1)=O c1(CC(=O)NC2(CC=C)CN(C(=O)C(F)(F)CSC)C2)c(C)nc2ccccn12 c1(OC)ccccc1CC(=O)N(CCNC(c1ccnn1C1CCC1)=O)C1CC1 N(C1CCCc2ccoc21)C(C1CC(O)(CNC(CN(C)C(N)=O)=O)C1)=O c1(NC(C2C3CN(C(C4CC(=O)NCC4)=O)C2C3)=O)cccc(Br)c1[N+](=O)[O-] C#CCCCCC(=O)N1CCCC(C)(NC(=O)CSCC(N2CCCCC2)=O)C1 CCCCC(CNC(C1C(Cl)(Cl)C12CC2)=O)NC(c1cnn(CC)c1)=O N1(C(CCN(CCCCC)C)=O)CCOCC12COCCN(C(=O)C=NOC)C2 c1(C(=O)NC2CCCC(NC(C3CN(C)C3)=O)C2)cc(N)c(Cl)cn1 c1(C(=O)NC2CCN(C(c3[nH]c(=NCC)sc3)=O)C(C)C2)cc(C)c(Cl)cc1C N1(C(C(COC)C)=O)CC2CCC(C1)N2C(=O)CCN1CCOCC1=O N1(C(CC2CC(CC)C2)=O)CC(NC(=O)CNC(=O)OC(C)(C)C)C(C(F)F)C1 c1(C(=O)NC(CN(C(=O)C2=CCCOC2)CC)C)cc(OC)ccc1Cl N1(C(c2c(C)nn[nH]2)=O)CCCC2C1CCN2Cc1ccccc1I N1(C(=O)Nc2c(C)cc(C)nc2)CCCC2C(C(=O)OC(C)(C)C)C(C)(C)C12 C(=O)(CC(CC)C(F)F)NC(CC=C)CNC(c1cc(C(C)(F)F)on1)=O CCCCC(O)C(=O)N1CC(CNC(c2sc(C(C)OC)nc2C)=O)C1 c1(C(N2CCC(N(C(=O)C(CC)CC=C)CC#C)CC2)=O)cc(C)c(C)cc1Cl Cc1[nH]nc2c1C(N(C)C(c1cn(CC3CCOC3)nn1)=O)CCC2 c1(C(C(=O)NCC(C)N(C(C2COCCO2)=O)CC)C)ccc(C(N)=O)cc1 Cc1ccc(C(=O)NC2CC(C)N(C(C3CC(=O)CO3)=O)C2)c2c1CCC2 C1(NC(C(CC)=CC)=O)CC2(CCC(NC(=O)CCS(=O)(=O)NC)CC2)C1 C1(OCC=C)CCN(C(=NCCc2ccccc2)NCc2cc(C)on2)C1 CCC(CC(=O)N1C2CCC(C2)C1CNC(c1ccncc1C(F)F)=O)C(C)C Cc1cccc(C(=O)NC(C(C)NC(C2(CF)CC2)=O)C(C)C)c1 N1(C(C=CCOC)=O)CC2CCC(C1)N2C(c1cc(C(C)(C)C)n[nH]1)=O C(C(C(=O)OC)NCc1ccc(CC)o1)SCC=C Cc1nn(C)c(C)c1CN1CCC(O)(C(=O)Nc2ccc(CC#N)cc2)C1 CC1(C)CC(C(=O)NC2(C)CCN(C(C3CC4(CSC4)C3)=O)CC2)CC(C)(C)O1 N1(C(c2cc(F)c(I)c(F)c2)=O)CCC2(CCN(C(C3(F)CC3)=O)C2)C1 C1(NC(CN(C(=O)CCc2cc(OC)no2)CC#C)=O)CCC(C)C1 C1(C(=O)NCC2C(C)(C)C2)CN(C(=O)CC#N)C(C)(C)C1 c1(CC)ccc(C(=O)NCc2csc(CNC(C3CCC3C)=O)n2)cn1 c1(-c2ccc(C(=O)NC(CN(C(=O)COCCCF)CC)C)s2)cccc(F)c1 c1(C(C(=O)NC2C(CNC(C(c3cn(CC)nc3)=O)=O)C2)C)ccc(C)cc1 N1(C(c2n(CC#C)ccc2)=O)CCCC(NC(c2ccc(Cl)cc2Cl)=O)C(F)C1 CCCC(C(=O)N1CCOC(CCNC(=O)C(F)CC2CCC2)C1)NC(C)=O C1(CC=CC)CCCN(C(=O)C(C)CN(C(=O)C(C)COCC)C)C1 Cn1ncc2c(O)nc(=NNC(=O)NCc3ccc(N4CCCCC4)c(F)c3)[nH]c12 c1(NC(C2CCCN(C(C(C)C(F)(F)F)=O)C2)=O)cnc2c(c1)CCC2 N1(C(CN(C(c2cc(CC)[nH]n2)=O)C(C)C)=O)Cc2cc(O)nnc2C1 C1(NCc2nc(CCC(=O)NC)on2)CCC(N2CCCC2=O)CC1 CC1(C)CC(CNC(=O)CCc2cnco2)N(C(C2CCC2(C)C)=O)C1 C1(C(=O)OC)CCC(C(N2CC(CNC(=O)CNC(N)=O)C2)=O)C1 N1(C(C2CC(C(C)C)C2)=O)CC(O)CC1C(=O)NC1CCCCC1F C(=O)(C(C(=O)N1CCOC(CC(=O)NCC(C)O)C1)OC)OCC Cn1cc2ccc(NC(=O)NCC3COCCC3c3ccccc3)cc2n1 N1(C(=O)CCc2cccc(O)n2)CC2(CCN(C(=O)C(F)CC3CCCC3)C2)C1 Cc1cc(Br)c2c(c1)CN(C(c1ccc(OCc3nn[nH]n3)c(F)c1)=O)CCO2 C1(CC=C)OCCC1(c1nnnn1C(C)(C)CC)NCCCC1CCC1 C1(C(=O)NC2C=CC(C(=O)NC)C2)CC(NC(=O)C(C)(C)OC)CCO1 C1(C(=O)NCCC(C)NC(=O)Cc2cncc(Br)c2)CCCC(=O)N1C CC(C)CC(C(=O)N1CCOCC1CO)NC(=O)CCC(N)=O c1(OCC=C)ccc(CC(N2CCC(NC(c3nc(=O)n(C)[nH]3)=O)C2)=O)cc1 c1(C(=O)NC2CCC(NC(C(C)NC(C)=O)=O)C2)cc(C)nn1-c1ccccc1 N1(C(C(CC)C(C)O)=O)CCC(C2(NC(=O)C=Cc3ccc(C(F)F)o3)CC2)C1 c1(C(N2CC(C)C2C)=O)cc(N)ccc1-n1cc(CCCCCO)nn1 C1(CC(=O)N(C)CC2CC(F)CN2)SC2=NCCN2C1=O.c1(C(=O)N)cn[nH]c1 C(C(=O)NOCC1CCCC1)(C1CCC1)NC(Cn1ccc(C)c1)=O C1(NC(c2c[nH]cc(C)c2=O)=O)C2CC3CN(C(c4cnc(C)n4C)=O)C1C3C2 C1(C(=O)NCC(CNC(c2c(CC)ocn2)=O)CO)CC(=O)N(C(C)(C)C)C1 N1(C(CCCC(N)=O)=O)CCCC2(CNC(=O)C(F)C3CCCC3)CCCC12 C12(CNC(CCC(C)OC)=O)CCC(C1)N(C(c1ncc(OC)cn1)=O)C2 C1(C)(CNC(C=C(C)C(C)C)=O)CN(C(=O)Cn2cc(F)ccc2=O)C(C)(C)C1 n1(CCNC(CCN(CCCO)C(C2C(C(C)(C)C)CC2)=O)=O)cccnc1=O C1(CN(C(CNC(=O)OCC)=O)C)COCCN1C(=O)C(C#N)CC1CC1 Cc1cccc(C(N2CCC(NC(C3CC3c3cccc(F)c3)=O)C2)=O)c1 c1(N2CC(C)=C(C)CC2)nc(=N)[nH]c(=NC(C)Cc2nncn2C)[nH]1 c1(C(=O)NCC23CC(NC(CSCCOC)=O)(C2)C(C)O3)c(Cl)ccc(F)c1N c1(-c2cc(F)c(OC)c(Cl)c2)ccc2nccc(C(N3CC4(CCC4)C3)=O)c2c1 C1(NC(c2n(CC#C)ccc2)=O)CS(=O)(=O)CC1NC(=O)C=CC(=O)N(C)C C=C=CC(C)C(=O)NC(C)(C)CCNC(c1cc[nH]n1)=O Cc1nc(C(C)(C)C)nc(O)c1C(=O)NC(C)C(CO)NC(=O)C#CC1(C)CC1 C1(C(=O)NC(COC(C)C)C(=O)NC(C)C(O)C(F)F)Cc2nccn2C1 N1(C(Cc2c(C)noc2)=O)CCC(NC(c2ccc(C(C)C)c(Cl)c2)=O)CC1C C1(C(=O)OC(C(CC)=CC(=O)OC(C)(C)C)(C)C)CC(C)(C)C12CCC2 O=S(=O)(c1cccc(=NCCN2CCCC2)[nH]1)NCC1CCC2CC12 C(c1ccc(C)cc1)=CC(N1C(CCNC(c2n(CC)nc(C)c2)=O)CCC1)=O N1(C(CC(CCC)O)=O)CCC2C(CCN2C(=O)CCCOCC2CC2)C1 C=C=CCC(=O)NCCCC(=O)NC(C)(C)COCC C1(NC(C(CCOCC)NC(C2COCOC2)=O)=O)CCCCCC1OC CCCCCCC(C(=O)NC(C)(C)C)N(C1CCN(c2c(F)cccc2F)C1)C C1(NC(CCC=C)=O)CS(=O)(=O)CC1NC(c1cnc(N(C)C)c(Cl)c1)=O Cc1cccc(C(C)C)c1C(=O)NC(CO)C(C)NC(=O)CCC1CCC1 C(CC(=O)N=c1ccn(C)[nH]1)N(C(=O)C(C1CCCCC1)=O)CC#C C(=O)(C1CCCc2nccn21)NC1(CNC(C2(SCC)CC2)=O)CCCCC1C c1(OC)cc(NC2CC(NC(C3(C)CC3Br)=O)C2)ccc1[N+](=O)[O-] C1(C)(NC(C(C)O)=O)CCN(C(c2ccccc2Oc2ccccc2)=O)C1 C(=O)(C(O)(C(F)(F)F)c1cn[nH]c1)NCCCN(C(c1ccc(C)nn1)=O)C Cc1nc(C2CC2)ncc1C(=O)NC1CC2(C1)CC2NC(=O)C1CC1 c1(C(N(CCN(C(c2c(C)cc(CC)o2)=O)C)C)=O)nccc2ccccc12 c1(CC(=O)NC2CC(NC(C(C)C(F)(F)F)=O)C2)cccc2c1CCC2 c1(C(N2C(CN(C(C(CC)N(CC)CC)=O)C)CCC2)=O)cc2c(ccn2C)[nH]1 CC1CCCN1CC(=O)NC1(CCNC(c2nocc2-c2ccccc2)=O)CC1 N1(C(C(=O)Nc2ccc(OCC)cc2)C)CC2(CCC2)C1c1ccco1 Cc1nnc(CNC(=O)CC2(C)CCN2C(=O)CCCC2CCCC2)n1C c1(CNC(CCCSC(C)(C)C)=O)ccccc1-c1cn(C2CC(C#N)C2)nn1 C1(NC(CC2C(NC(c3cnc(C(C)C)o3)=O)CCCC2)=O)CCC(C2CC2)C1 CCC1=NOC(CC(=O)NCC=CCC(=O)NCCOCC(F)F)C1 C(=O)(CC1=CCCC1)N(CC(C)NC(=O)C(c1ccc(O)cc1)C)CC CC1Cc2c[nH]nc2CC1NC(=O)N(C)Cc1ccc(CO)o1 C(c1ccc(F)cc1)=C(C)C(=O)N(CCC(O)C(C)(C)C)Cc1nn[nH]n1 Cc1coc(C2CCCN2C(c2cscc2Br)C(=O)NCCCOCC2CC2)n1 C1(C(=O)NCC(C)(O)CNC(=O)C(CO)c2ccccc2)C(F)(F)C12CCCC2 N1(C(C2CC(C#N)C2)=O)CC2CC(NC(=O)Cc3cc(F)cc(F)c3)C1C2 c1(OCOC)ccc(C(=O)NC2CC(F)(CNC(c3cnc(S)[nH]3)=O)C2)cc1 C(CC(=O)NC1CC(NC(C23CCC2C3)=O)C1)N(CC)CC CC1CC(C(=O)N(C(C)CCNC(=O)C=CC2CCCC2)C)CCS1(=O)=O N1(C(C(C)(C)c2ccns2)=O)C2CCC1CN(C(=O)COC1CCC1)C2 c1(C(=O)NCc2c(C)csc2)ccc2cc(O)ccc2n1 CC(C)C(C(=O)N(CCCCN(C)C(c1cnc(Cl)[nH]1)=O)C)c1cnn(C)c1 C1(CCN(C(C(C)OC)=O)C)CCN(C(c2ccc(C(F)(F)F)cn2)=O)CC1 Cc1cc(C(N2CCC3(NC(c4c(F)cccc4Br)=O)CC3C2)=O)c(C)n1C Cc1cnn(CCN(C)C(C2CCN(C3COC3)C2)=O)c1.C12CCC1NC2=O C#Cc1ccc(C(=O)NC(C)CCNC(=O)C#CC2CCCC2)c(C)c1 c1(C(N(CCN(CC(O)CO)C(C)=O)Cc2ccc(F)cc2)=O)nc(Cl)oc1C C#Cc1ccc(F)c(C(=O)NCC(CNC(=O)C(C)OC)S(C)(=O)=O)c1 N1(C(c2cc(C)sc2C)=O)CCC(NC(=O)C2=CSCS2)C(F)C1 C(=O)(C(=O)CC(C)CC)NC1C(C(N2CCCC(CC)CC2)=O)OCC1 C12(C(=O)NC(c3nc(=O)o[nH]3)C)CC(CN1C(=O)CC(C)N(C)C)C2 C1(C(C)C)CCC(C)CC1(O)CNC(=O)C(N1CCCCC1CO)=O CC1C2CCC(C2)C1C(=O)N(CCC(=O)NC1CC1)C.C1CCC(=O)N1 C1(C(C)C)CCC(NC(=O)C(C)Cc2ccccc2)CC1.N1CC(O)C1 C1(C(CNC2(c3onc(C(C)C)n3)CCC2)C)OCCCC1(C)C c1(C(N2CCC(CC=C)(NC(=O)C(C)C3CCCO3)C2)=O)c(C)ncnc1C C(C)(C(=O)N1CCC(O)(CN(C)C(c2cc(C)co2)=O)CC1)(C(C)C)NC(C)=O CC(C)CC(C)CC(=O)NCC1COCCN(C(=O)C#CC(=O)N(C)C)C1 C(=O)(C1=CCOCC1)N(C)CC1CCN(C(c2nn(CC)c(C3CC3)c2)=O)C1 N1(C(c2c(C)ccc(C)n2)=O)CC2(CC(C(=O)NCCN(C)OC)CO2)C1 C1(OC(C)C(=O)NC2CCC2NC(c2ccc(=N)[nH]n2)=O)CCCCCC1 Cc1cccc(CCC(N2CCCC2CNC(C2CC3CCC2O3)=O)=O)c1 c1(CC(CO)NC(C2CCN(Cc3cnccc3Cl)C2)=O)ccc(Cl)cc1 N1(C(C2N(C=O)CCC2)=O)CCC2(CC1)CC2NC(c1cccc2ccoc12)=O c1(CN2CCN(C(=O)C(Cl)(Cl)Cl)C(C(F)(F)F)C2)c[nH]c2c([N+](=O)[O-])cccc12 CC(C(=O)NCCC1(NC(C2CC=CC2)=O)CC1)N1CCCC1 N1(C(C2(C)COC2)=O)CCC2CCCN(C(=O)CS(C)(=O)=O)C2C1 C(c1ccccc1C)=CC(=O)N(C1CCN(C(C(C2CC2)OCC)=O)C1)CC c1(OCC)ccc(C)cc1C(=O)N(C)CCNC(C1C2CCC12)=O c1(C(N2C3(CNC(c4ccn(C(F)F)n4)=O)CC(C2)C3)=O)ccc(CO)c(Cl)c1 c1(CCCC(=O)NCC2N(C(C(CC)NC(N)=O)=O)CCC2)ccc(Br)cc1 N1(C(C2(OC)CCSC2)=O)CC2(CC(NC(=O)Cn3nnnc3C3CC3)CO2)C1 C(N=c1cc(NCCCCN(C)C)nc[nH]1)C1(OC(C)C)CCSC1 CCCCCCCCNC(=O)C(C1(O)CN(C(c2n[nH]c(=N)[nH]2)=O)C1)F C(=O)(CCC(C)C)NCC(=O)NCC(C1CCOC1)NC(C(C)(C)SC)=O CC1(C)CCC(CN=c2nnn(-c3ccccc3)[nH]2)(NCc2ccccc2)CC1 N1(C(CCS(=O)(=O)N(C)C)=O)CCC2(CC(NC(C3C=CCCC3)=O)C2)C1 N1(C(CC(C)(C)C2CC2)=O)CC2CCCC(C1)N2CCN1C(=O)CCC1=O C(=O)(CC(O)CCCCC)N1CCC(C(=O)NC(C#C)C(C)(C)C)(CF)C1 C1(NC(C2C3CNCC23)=O)CCN(CCNC(C2CCCO2)=O)CC1 Cc1cc(Cl)c(C(=O)NC2CCN(C(=O)Cc3ccc(C)o3)CC2O)cn1 c1(C(N2CCN(C(c3cn(C(C)C)nn3)=O)C(C)C2)=O)cc2cccc(Cl)c2s1 C1(C#N)(c2ccccc2)C(C#N)C1(C)C.C1(O)(c2c(C)cncc2)CCN(CSC2C3N2C(=O)C3C)CC1 C12(C(=O)OC)CCC(C(=O)NCC3(C)CCOC3)(CC1)CC2.C(CO)O c1(C(=O)NCCC2(C(=O)N(CCCNC(N)=O)CCO)CC2)nc(Cl)cs1 C1(F)(C(N2CC(OC)C(NC(=O)C(C)n3cccn3)C2)=O)CCN(C)CC1 c12ccc(cc1)Cn1cc-2nn1.Cc1cc(CNC(=O)CC2CCCO2)on1 N(C1Cc2ccccc21)C(C(=O)Nc1cncc(C#C)c1)=O C1(C(N(CC(C)(C)NC(C2CC(=O)NC(=O)N2)=O)C)=O)CCc2cnnn2C1 N(C1CCCc2c1cnn2Cc1ccccc1)Cc1ccc(CN)cc1 C(=O)(CC(C)(C)C1CCCCC1)N(C1CC(NC(=O)C=Cc2ccncc2)C1)C c1(C(N2CCC3CN(C(C4C(CN(C)C)C4)=O)C3C2)=O)cc([N+](=O)[O-])cnc1O C(C(=O)NCCCn1cncn1)(C(C)C)SCC.C1(C2CCC2)C(=O)N1 N1(C(C2CN(c3ccc(C)cc3)C(=O)C2)=O)CCC2(CC1)NC(=O)C(C)O2 c1(NC(C(c2cc([N+](=O)[O-])sn2)N(c2nncs2)CC)=O)ccc(OC)cc1C C1(C2CCN(C(=O)CCP(C)(C)=O)C2)(NC(CCOCC)=O)CC1 N1(C(C(C)(C)CO)=O)CCC(O)(CCNC(C2(C(N3CCCC3)=O)CC2)=O)CC1 CCCC(C)(C)C(=O)N1CCC(O)(CNC(=O)Cn2c(C)c(C)sc2=O)C1 N1(C(Cc2nc(C)sc2)=O)CCCC(C)(C)C1CNC(C1(C)CCNC1=O)=O Cc1nc(C)c(C(=O)NC2CCC(NC(C3CC34CCCC4)=O)CC2)s1 c1(C(=O)NC2C(NC(c3ccc(C)c(C)c3)=O)CCC2)cc(N)cc(O)c1C C1(N(C(COCCOCC#C)=O)CC)CCCN(C(C2CC3CC3C2)=O)C1 N1(C(c2scc(C)c2)=O)CC2(CCNC(c3ccc(Cl)cc3)=O)CCC1C2 Cc1nocc1C(=O)NC1(C(=O)N(C)CC2(N(C)C)CCC2)CCCC1 C(CC(C(=O)NCc1ccccc1COCC)NC(=O)CC(C)C)=CC CCCCC(CN=c1[nH]c(C)nc(C)c1F)NC(c1ccncn1)=O Cc1ccc(C(N2CC(C(N3CC4CC4C3)=O)C(F)(F)C2)=O)cc1C#N N1(C(C(Cn2ccc(C)n2)C)=O)C2CCC1C(C)C(NC(=O)CC1CN(C)C1)C2 c1(C(=O)OCC)ncc(CNC(C)C(C)O)cn1 Cc1cc(Br)sc1C(=O)NCC(C)NC(=O)CCc1ccco1 CCCC(CCC)C(=O)NCc1nc(C(N2CC(COC)C2(C)C)=O)co1 N1(C(c2c(C)cccn2)=O)C2CC=C(C(=O)N3CC(O)(c4nn[nH]n4)C3)C1CC2 c1(NC(NCCNC)=S)cc(C(F)(F)F)cc(C(F)F)c1.c1c(C)noc1C NS(=O)(=O)c1coc(C(=O)NCCC2CCN(C(c3cnc4sccn34)=O)C2)c1 c1(CC(=O)N(CC)CC2CCN(C(=O)CC(C)OC)CC2)cccc(F)c1Cl c1(C(N)=O)cocc1C(=O)NC1CCCC1CC(=O)NCC(N1CCOCC1)=O c1(C(N(C)Cc2c(C)ncs2)=O)c(-c2ccccc2)nn(C)c1Cl c1(OC)cccc(Cl)c1C(N1CCC(NC(c2nc(C)ncc2Br)=O)C1)=O C12(OC)CCCC(CC(NC(=O)N(C3CCC3)C(C)C)C1)C2 N1(C(COC(CC)(C)C)=O)CCC(NC(c2c(Br)nnn2C)=O)CC1 N1(C(c2c(NC)cnnc2)=O)CC(C)CN(C(c2cncnc2C)=O)CC1C C=CCCC(C)N=c1[nH]c2c(c(=NC(C)c3ccc4ncccc4c3)[nH]1)CCC2 C1(CNC(CCN(CCC)C)=O)CC2CCC(C1)N2C(=O)C(C(C)OC)N(C)C C1(NC(c2cn(CC=C)nn2)=O)C2CC1N(C(=O)CN(c1ccc(Cl)cn1)C)C2 c1(C(C(=O)NC2CCC2)N(C(CCSC)C)C)cc(S(C)(=O)=O)c(C)o1 c1(-n2ccc(C)c2)ccc(C(N2CC(NC(c3cc(C)co3)=O)CC2C)=O)cc1 c1(NC(C2(C(=O)Nc3nc4ccccc4o3)CC2)=O)ccc2c(c1)CCNC2 N1(C(c2cn(CC=C)nc2)=O)CCN(C(c2csc(Cl)n2)=O)CC(O)C1 C=C1CCC(C(N2CC=CC(NC(=O)C(C)CSc3ccccc3)C2)=O)CC1 C1(NC(C(COC)COC)=O)CCCCN(C(=O)C=Cc2ccccc2)C1 c1(C(=O)NC2C=CCN(C(C3CCC(C)(C)CC3)=O)C2)ccc2cnoc2c1 C1(C(N(C(C)C)C)=O)CCN(C(=O)C(N2CCN(c3nccnn3)CC2)=O)CC1 C1(C(=O)NCC2OCCN(C(c3ccc(=N)[nH]c3)=O)C2)Cc2ccc(F)cc2O1 Cc1cc[nH]c1C(=O)NCCCCCNC(=O)C(=O)NCCc1ccccc1 N1(C(C2(NC(CCn3c(C)nnn3)=O)CCC2)=O)CCC(C(C)CO)CC1 CCC(CC(=O)N1CCCC(NC(c2c(Cl)nn(C)c2C)=O)CC1)C(C)C C1(C(=O)NC2CC(NC(C(C)NC(=O)C3CC3)=O)CC2O)CCCC12CCC2 c1(C(N2CC3C(CNC(C4CCC(C(N)=O)C4)=O)(C3)C2)=O)cc(O)ccc1F Cc1nc(C(=O)NCC(O)CN(C)C(c2ccc(-c3ccccn3)o2)=O)c(C)s1 n1(CC)nc(C)c(CC(N2CCOCC(NC(=O)CC(C)O)C2)=O)c1C N1(c2ncc(C#C)cn2)CC2(CN(C(c3cccnn3)=O)CC(C)(C)O2)C1 CC(CF)C(=O)NC(C)CCNC(=O)CCNC(c1ccco1)=O c1(C(=O)NC2C(C)CN(C(=O)Cc3ccn(C)n3)C2)ccc(O)c(C(=O)O)c1 C1(C(=O)OCc2n(-c3cn(C)nc3)cnc2)CCCCC(P(C)(C)=O)C1 C=CCC(C)(CC)C(=O)NCC1(C)CC(C(=O)NC2(c3ncccc3Cl)CC2)C1 C(=O)(C(CCC)NCC(C1CC1)OC(C)=O)NCC=C CCCCC(CC(=O)NCCC1CC=CCC1)NC(c1cccc2ccoc12)=O N1(C(C2CC(O)(CNC(C3(COC)COC3)=O)C2)=O)CC2CC2C2CC12 N1(C(CC)C(=O)NCCOC2CN(C(c3cnn[nH]3)=O)C2)C(=O)CCC1=O CCC(C)C(C(=O)N1CCCC(CCNC(=O)CCCCSC)C1)OC N1(CC2CC(OC(C)(C)C)C23CCC3)C(=O)C2CCCCN2C1=O Cc1onc(-c2ccc(F)cc2)c1C(=O)NCC1(CO)CCCNC1 c1(C(N2CCC(CN(C)C(C3(F)CC4(CCC4)C3)=O)C2)=O)cncc2sccc12 C1(NC(c2cnc(SC)s2)=O)CCC(C)(CNC(=O)CCc2cccn2C)C1 N1(C(c2c(C)[nH]nc2C(F)(F)F)=O)CCCOC(CCNC(C2CC2(C)C)=O)C1 Cc1ccc(C(N2CC3C(CNC(C4(C)CCC(=O)NC4)=O)C3C2)=O)c(F)c1C c1(NC(C2(F)CCN(C(Cc3nc(CC)on3)=O)C2)=O)cc(C)cc(Br)c1F N1(C(c2c(CC)ocn2)=O)CCN(C(=O)C(C(C)(C)C)NC(N)=O)C(C)C1 C(CN=c1c([N+](=O)[O-])c[nH]c2c(Cl)cccc12)=CCNC(=O)CCN1CCC1 C1(C(N(CCNC(C(C)C(C)(C)C)=O)C2CC2)=O)C2(CCC2)C12CCC2 C1(C(=O)NCC(CC(C)C)C)C2CC(O)C(C2)N1C(=O)C(C)CC1CCC1 C1(NC(c2ncc[nH]c2=O)=O)CN(C(=O)C2=CCOCC2)CC(F)(F)C1 c1(OC)cccc(C(C(=O)N2CCC2C2CC2)OC)c1.C1(=O)C(C)(C)CN1C C(CC(F)F)(C(=O)NC1CC(C)(C)C12CC2)N(C(Cc1c(C)n[nH]c1)=O)C Cc1ccc(C(=O)NCCC2CCC(NC(=O)C(=O)NCC(F)(F)F)C2)s1 c1(C(N2CCC(CCNC(C34CC(O)C3C4)=O)C2)=O)cc(-c2ccco2)[nH]n1 N1(C(C(CC)COC)=O)CCN(C(C2CC3(CC(OC)C3)C2)=O)C(C)C1 CC1(C)CCCCC(C(N2CCN(C(C3C4COCC34)=O)C(CCO)C2)=O)C1 CCC(C)C(C(=O)N1CC(CNC(c2cc(C)cs2)=O)C(F)(F)C1)N(C)C C1(NC(C(C)O)=O)CC1C1CCCN(C(c2cn(C)nc2C2CCC2)=O)C1 N1(CC(COC)NC(=O)NC(c2csc(=N)[nH]2)C)CCOCC1 c1(C(=O)NCC2(CNC(C34CC(C)(C3)C4)=O)CCCC2)cc2n(n1)CCNC2=O c1(COC)cc(C(=O)NCC(=O)NCC(=O)NCC2CCOC2)n[nH]1 c1(C(=O)NCCCCNC(c2cnc(C)[nH]2)=O)cccc(-n2cncn2)c1 N1(C(C2C(COC)CC2)=O)C2CCC1C(F)C(NC(C1CC=CCC1)=O)C2 CC1(CC(=O)NCC(O)CCNC(=O)CCSc2ccccn2)OCCO1 C(CC(O)C(=O)N1CC2CC2(C(=O)NCCCc2ccccn2)C1)SC CC(C)(F)C(C)(F)C(=O)NCC1CC(NC(=O)CCc2ccc(Cl)nc2)C(O)C1 Cc1cc(CC(=O)NCc2cn(CCCC#N)nn2)on1 c1(N(C)Cc2ccc(=N)[nH]c2)ccc(S(=O)(=O)NCc2ccncc2)cc1F C1(OC)CCN(CC(=O)NC(CNC(=O)CN2CCC(C)C2)C(C)C)C1 CC(O)C(C(N)=O)NC(C1CCC(NC(=O)Cn2cc(Cl)cn2)CC1)=O N1(C(CC(C(=O)OC)C)=O)CC(CNC(=O)Cc2ccccc2Cl)C2(CCC2)C1 N1(C(C(C)CN2CCOCC2)=O)CCC(N(c2ncncc2I)CC2CC2)CC1 CCC(CC)C(C)C(=O)N1CC2CCCC2(NC(c2cnc(Cl)[nH]2)=O)C1 c1(CNC(N2CCCC2CO)=O)ncccc1S(C)(=O)=O.CCCCCN c1(CC)cccnc1C(N1CCCC1(C)CNC(=O)C(C)(C)c1ccccn1)=O C(=O)(C1=NOC(C)C1C)N1CCC(CC=C)(C(N2CC=CC2)=O)C1 C1(CCOC)(NC(=O)C=C(C)Cl)CCN(C(=O)CCC2C(=O)NN=C2C)C1 C(=O)(CC(O)C(C)C)N(C)CC1CCN(C(C2(CCOCC)CCC2)=O)CC1 C1(CNC(C(C(C)C)O)=O)CCC2(CO1)CC(NC(=O)Cc1cc[nH]n1)C2 c1(C(=O)NC(C2CCN(C(C3ON=C(C)C3)=O)CC2)C)c(Cl)ccc2ccoc12 c1(C(N2C(C(C)C)COCC2)C(=O)NCc2ccccc2)cccc2c1CCC2 C(=O)(CS(=O)CCC(F)(F)F)NCC1CCN(C(Cc2cn(C)nc2)=O)C1(C)C c1(CC(=O)NC2C(NC(C=CC=CC(C)(C)C)=O)CC2)ccc(Cl)cc1Cl N1(C(C2CCN(CC)C2=O)=O)CC2CCC(CNC(C3(CN(C)C)CC3)=O)C2C1 C(=O)(C(CCC)CC(C)C)NCC1(OC)CN(C(c2cn(CCCC)nn2)=O)C1 c1(OCC)ccccc1CN(CCCNC(=O)C(O)CC1CCCCC1)C(C)C C1(CC)C(NC(=O)Cc2c(C)noc2Cl)CCCN1C(C1CC2CCC1O2)=O N1(C(c2ccc[n+]([O-])c2)=O)CCC2(CCNC2)CC1 c1(C(N2C(C)(CC)CC(NC(=O)C=CSC)C2)=O)cc2c(nc1O)CCCC2 N1(c2ncn(C)c(=O)c2)C2CCC1CN(C(c1ccc3c(ccn3C)c1)=O)CC2 CC(C)C(C)C(CNC(c1nocc1Cl)=O)NC(=O)COCCc1cccs1 C(=O)(C1CCc2cc(F)ccc21)NCC(CO)NC(c1c(C)n2c(n1)scc2)=O N1(C(C23CCC(OC)C2C3)=O)CC(C)C(C)(C(=O)NCC2CC(=O)N(C)C2)C1 Cc1noc(CNC(c2ncsc2Br)c2nnnn2CC2CCCO2)n1 C(c1ccccc1OC(F)F)=CC(=O)NCC#CCNC(C1CC(C)(F)C1)=O C(C(=C)c1ccccc1)NC(C1(CCNC(CC2(CC)CCC2)=O)CCC1)=O c1(N(C2CCNCC2F)C(c2ccc(C)cc2Cl)=O)ccn2nccc2n1 c1(C(N2CC(NC(C(N3CCCC(O)C3)C)=O)C2)=O)cc2scc(Cl)c2[nH]1 CC1CC(NC(=O)C2=CCC2)CN(C(c2ccc(Cl)c(N)c2)=O)C1 Cn1nccc1C1CC1C(N1CCC(N(C(=O)COCC(=O)OC(C)(C)C)CCO)C1)=O N1(S(CC)(=O)=O)CCCCC1C(N1CCOC(CNC(c2csc(Cl)c2)=O)C1)=O N1(C(CCC)=O)CCCCC1C1(CCOc2ccc(CNS(C)(=O)=O)cc2)CC1 C1(NC(CC2(C)CC2(Cl)Cl)=O)CCN(C(C2Cc3cscc3C2)=O)CC1F C=CC1CC(N=c2[nH]c(N(C)Cc3cccc(C(C)C)c3)nc(=N)[nH]2)C1 C1(N(C(CC(c2cccc(F)c2)C)=O)C)CCC(NC(=O)COCC(F)F)CC1 CN1CCCC(O)(CC(=O)NCCN(C)C(C2(CCO)CC2)=O)C1 C(=O)(C(C)CS(C)(=O)=O)NCC(c1cccc(C)c1)NC(C1(O)CCCC1)=O CN1C(=O)CCC1CC(=O)NC(C(=O)NCCC(=O)NC(N)=O)C1CCOC1 c1(CN2C(CO)CC3OCCC32)cc(F)ccc1[N+](=O)[O-] CCC(CC(=O)NC(C(=O)N1CC(C(N)=O)(OC)C1)C(C)C)SC CC1(C(N2CC(NC(c3cccn4nncc34)=O)C2)=O)COc2ccccc2O1 N1(C(C(N2CC(CCNC(=O)C(C)CO)(OC)C2)=O)C)CCc2ccccc21 S(=O)(=O)(c1ccc(NC(CC)CC(F)(F)F)c(F)c1)NCCC(CC)O C1(NC(c2cccc(CNC(C(C(C)C)(C)O)=O)n2)=O)CC2CCC(C1)C2O c1(C(N2CCCC(CC=C)(NC(=O)C3=NOC(C)C3)C2)=O)cccc(S(C)=O)c1 C(CC(=O)N1CC(O)C(O)CO1)c1c([N+](=O)[O-])nccc1 S(=O)(=O)(c1cccc(C(=O)NC2CCN(C(c3ccoc3)=O)C2CC)c1)NCC C#CCCCN=C(NCC1CC1)NCC1CC2(C1)CC21CC1 N1(C(c2c(OCCOC)nccc2)=O)CC2CN(C(C3CC(O)C3)=O)C2C1 C1(NC(C2(CC)CC2)=O)(Cc2ccccc2)CCCN(C(=O)CC(C)C(F)F)C1 C12(CC(F)(F)C1)CN2.C1(C(=O)OC(C)(C)C)(COC)CN(C(=O)OC(C)(C)C)C1 c1(C(=O)NCC2C(NC(c3cc(CC)on3)=O)COC2)ncccc1S(C)(=O)=O C(=O)(CC(C)(C)OC)NC1CCC(NC(C2(CC=C)CCOC2)=O)C1 CCCCC(F)C(=O)N1CCCC(C(C)(C)C(=O)NCC2CCC2OCC)C1 C1(NC(C2N(CC)CC2)=O)CC2CN(C(C3CCCN3C)=O)CC12 c1(C(N2CCN(CC#CC)CC2)=O)ccc(Br)c(OCc2ccc(Cl)cc2C)c1 N1(C(C(F)=CC)=O)CCN(C2CCCN(C(c3nncs3)=O)C2)C(=O)C1 C12(CC(=O)OCC(=O)Cc3ccc(O)cc3)CCC(CC1)OC2 C1(COC)CC(O)CN1Cc1ccnc(-c2ccccn2)c1 c1(CNC(CCC)=O)cn(C2CCN(C(=O)C(C)Cc3cnc[nH]3)C2)nn1 C1(NC(Cc2c(C)ocn2)=O)CCC(CNC(c2cnc(O)s2)=O)CC1 C1(NC(c2cnn(CC)c2Br)=O)CCCC12CCN(C(C1CSC1)=O)CC2 c1(C(N2CCCCC(NC(C3CC(=O)N(O)C3)=O)C2)=O)cc2cnccc2[nH]1 c1(OC)cc(F)ccc1CC(N1CC(O)CC1C(=O)Nc1cccc(CO)n1)=O c1(SC)cc(C(N2CCCC2CN(C)C(C2CCO2)=O)=O)c(Cl)cc1Cl CC(CNC(=O)C(C1CCC1)NC(c1ccns1)=O)CCCO Cn1c(C(=O)NC2COCC2C(=O)Nc2cnccc2CO)nnc1S c1(OC)ccc(F)c(CC(=O)NC2CC3CC2CN3C(=O)C2=CCOCC2)c1 N1(C(C2C(OCC)C2)=O)CCN(C2CN(C(=O)C(C)Cc3c(C)noc3C)C2)CC1 C1(C)(C(=O)NCc2cn(CC(CC)C)nn2)CC2CCC1CC2=O c1(OC)ccc(-c2ccc(-c3nccn3C(C)CCO)s2)cc1F N1(C(C(=Cc2cccs2)C)=O)CCC(C)C(NC(c2cn(C(C)C)cn2)=O)C1 C1(C(=O)NC2(CCCC)CC2)C(C)CCN1C(c1cccc(C)n1)=O C12(C(=O)NCC3(C)CCCN(C(C=CC)=O)C3)C3C4C1C1C2C3C41C(N)=O C1(NC(CSC(C)C)=O)CCN(C(=O)C(C)(C)C(F)(F)F)CC12CCC2 Cc1cc2ncc(C(N3CC(C)(C)CCC3(C)C)C(=O)NC3CC3)cn2n1 C(=O)(C1CCSc2ccccc21)NC1C2CN(C(C(C)CC(N)=O)=O)CC1C2 Cc1c(F)ccc(Br)c1C(N1CC(N(C(=O)C=Cc2cncnc2O)C)C1)=O C1(CC(=O)NCC(C2CC2)NC(c2coc(C(F)F)c2)=O)C=CS(=O)(=O)C1 C1(C(=O)NCCC(C)NC(=O)CCc2csc(Br)c2)NC(=O)OC1C N1(C(C(C)=CC)=O)CCCCC(C2CN(C(=O)C(C)(C)CC(C)C)C2)C1 n1(CC)ccc(C(=O)NC(C2CN(C(=O)CNC(=O)OCC)CCO2)C)cc1=O C1(C(N(C2(CO)CC2)C)=O)CC2(CC(NC(=O)CN3CC4CC4C3)C2)C1 N1(C(CCNC(N)=O)=O)CCC(C#N)(C2(C#C)CCCC2)CC1 Cn1ncc2c1CN(C(c1cc3c(s1)CCC(C(C)(C)C)C3)=O)C2C(=O)O c1(C(=O)NC(C2N(C(C(CCC)C#N)=O)CCC2)C)c(Cl)sc2nnsc12 N1(CC)CC(NC(=O)COC(C)(C)C)CCC1=O.C12CC1CN2 C(=O)(C1CCc2cc(OC)ccc21)NCC(CN(C(c1n(C=C)ncc1)=O)C)O C(c1cc(C)cc(C)c1)=CC(=O)NCC(C1(O)CN(C(CSCC)=O)C1)(C)C C1(CNC(c2cc(F)c(Cl)cc2)c2ccccn2)COCC2(CCNC2)O1 C(=O)(C1=C(C#N)CCC1)NC1C(CNC(CC(C)N(C)C)=O)CCCC1 c1(OC)c(C(=O)NCC2CCCN2C(c2nnc(C)s2)=O)oc2ccccc12 N1(C(C(=O)NCC)=O)CCN(C(C)C(N2CCCCC2)=O)CC1 c1(C(=O)NC2C(NC(CCC)=O)CCC2)cc(NC(=O)C#CC2CCC2)ccc1Cl c1(N2CCC(N(C(=O)CCCCCF)CCC)C2)ncn(C)c(=O)c1Br c1(C(=O)NC2CCC3(C(NC(=O)C=C4CCC4)C3)CC2)coc2c1C(=O)NCC2 c1(C(N2C(CN(C(=O)CNC(=O)C(C)(C)C)C)CCC2)=O)ccc(N)cc1F C1(C(=O)NCC2CC3CN(C(c4ncncc4Cl)=O)CC23)CCc2nc[nH]c2C1 N1(C(C(CC#C)O)=O)CCC(C(=O)N(CCCN(C)C)C)C1(C)C C1(NC(C2C(C)CCN2C(c2nc(=N)cc[nH]2)=O)=O)CCCC(O)C1O C12(NC(=O)COCC3CCCC3)CCC(C1)N(C(c1c(N)cccc1F)=O)C2 Cc1ccn2c(CC3C(F)(F)C34CCC4)cnc2c1.C12CCCN(C1)C2=O N1(C(C(C2CCOC2)OCC)C(=O)NCC(F)F)CC(CO)CC(C)(C)C1 C#CC1(C(=O)NCCCCN(C(=O)CCC2CCC(=O)N2)C)CCC1 CCCCC(O)CC(=O)NC1(CO)CN(C(c2ncc(C(=O)OC)cc2Cl)=O)C1 N1(C(C23CN(C(c4ncc(F)cc4F)=O)C(C2)CO3)=O)C2CCC1CC(CO)C2 N(C(=NCC(C(F)(F)F)N1CCOCC1)NC1CC(OC)C1(C)C)C1CCOC1 c1(C(N2CCCC(C(C)NC(c3cn(CC=C)nc3)=O)C2)=O)nc(C)ccc1C C1(NC(C2(C)CCCC2)=O)CS(=O)(=O)CC1NC(c1ncc(F)cc1N)=O C1(C(=O)NC(C2CCCC2)CO)CC=CCN1C(=O)CC1CNC(=O)O1 Cc1nc(NCC(C)Cc2ccccn2)cc(=NC(C)c2cccc(F)c2)[nH]1 C1(NC(CCCCCCC)=O)COC2(CCN(C(=O)CC3CCOC3=O)CC2)C1 c1(OC)cc(C)sc1C(=O)NCC1CCCC1NC(=O)C=CSC Cc1ccc2cc(C(=O)NCC(C)NC(c3cc4ccsc4[nH]3)=O)ccc2c1 N1(C(CCn2ncc(C)c2)=O)CCC2(CCC(NC(=O)C(C)S(N)(=O)=O)C2)CC1 c1(CN2CCC(CNC(=O)CCCCl)C2)cncc(OC(F)F)c1 N1(C(c2c(C)noc2)=O)CC2CCC1C1CN(C(=O)CSCC(N)=O)CC21 C(=O)(C1=C(Cl)CC1)NCCN(C(C(n1ccc(C)n1)C)=O)CC1CC1 N1(C(c2cc(C)no2)=O)CCc2cccc(C(=O)NCc3ccc(F)nc3)c2C1 c1(C(N(CCN(C(c2c(CCC)nns2)=O)C)C)=O)cccn2cc(C)nc12 c1(CC(=O)NCC(c2cccc(Cl)c2)OC)cn(C)nc1I c1(NC(C2C(C(C)NC(C=C(C)C(F)F)=O)C2)=O)ccc(OCF)cc1 C1(CN(C(=O)COC2CC(NC(c3cn(C)nc3O)=O)C2)C)CCCC12CCC2 n1(CCC(=O)NCC2CCC2NC(C2CCC(F)CC2)=O)ccc(O)nc1=O C=CC1(C(=O)NC2(C)CC(N(C)C)C2)CCN(C(=O)CC2CC(OC)C2)C1 N1(C(C=C(C)C2CC2)=O)CCC(C(=O)NC(C)CC(F)(F)F)CC1(C)C Cc1cc(C(=O)N(C)CCNC(=O)CSc2nnnn2C)nc(C(F)(F)F)n1 c1(CCN(C)C(C2CCCC(O)C2)=O)ccc(C(=O)OC(C)(C)C)cc1 CCC(C)C(C(=O)N(C1CC2CCC1O2)C)N(C(=O)Cc1nocc1C(C)C)C c1(NC(CC(CC(C)C)O)=O)nc(Cl)nc2cc(Br)cnc12 C1(CNC(c2ccn(C)c2)=O)CCCCN(C(=O)Cc2cccnc2N)C1 CC1CN(C(c2cc(C(F)F)nn2C)=O)CC(C)C1NC(=O)Cc1csc(=N)[nH]1 C(=O)(C(C(C)C)n1cncn1)NCC1(OCC)CN(C(=O)C(F)OC(F)(F)F)C1 CCCCCCCCC(=O)NCC1(C)CCCN(C(c2cnccc2CC)=O)C1 Cc1ncnc(C(=O)NCc2ccc(C(=O)NCC(c3cnc[nH]3)C)cn2)c1C CC(C)C(C)C(=O)NC1CN(C(c2csc(C(F)F)n2)=O)CC1C N1(C(c2cccc(C)c2Br)=O)CCC2CCNCC12 Cc1c(C(N2CC(CO)(NC(C3CC4(CC4)CO3)=O)C2)=O)nn(C)c1N Cc1cc(O)ncc1C(N1CCCC(C(=O)NCCOc2ccncc2)C1)=O C1(CNC(c2c(OCC)nc(C)cc2)=O)C2CCC1CN(C(=O)C(CC)CC)C2 CC1CC(NC(=O)CC2CCCCC2)CN(C(c2ccnc(C(F)(F)F)c2)=O)C1 N1(c2nnc(COCC)n2CCc2cccc(C)c2)CCn2nccc2C1 C1(C(=O)NC(CCC)C2CC2)(NC(c2ccco2)=O)CC1(C)C C(C)(CCCC(=O)N(CC(=O)OCc1ccc(O)cc1)C)c1ccc(OC)cc1 Cc1nn(C)c(=O)c(-c2nc(CCc3ccccc3)nn2CC2CC2)c1C c1(CC)cncc(CNC(C2CC23CC(NC(c2cnc(OC)cn2)=O)C3)=O)c1 c1(C(N(C2CCN(c3snc(CC)n3)C2)C)=O)cnn2c1CCC2 C(C(C)(C(=O)NC(C)Cc1nn[nH]n1)NC(c1cccc(O)n1)=O)SC CN1CCC(C(=O)NC2CC(N(C(=O)C=Cc3cscn3)C)C2)C1 C#CCC(CC(F)F)C(=O)NCC1C2CN(C(c3nccn3C)=O)CC12 c1(C(N2CC(NC(c3ccc(O)nn3)=O)C3C2C3)=O)cc2nccnc2cc1F c1(CN(C)C(=O)NCC2CC2c2cccs2)cnc(N(C)C)s1 C12(NC(C(CNC(C(C=C)C)=O)N(C)C)=O)CCC(CC1)C2(C)C c1(C(=O)NC2C(NC(C3CCC(CC)CC3)=O)CCCC2)cc(F)c(F)cc1O C1(C#N)(C(=O)NC(C(C)NC(C2CCC=CCC2)=O)CO)CCS(=O)(=O)CC1 C(=O)(CCCN(C)N=O)NCCCC1CCN(C(C2CC(C#C)(O)C2)=O)CC1 c1(C(C2CC2)NC(C2CCCCCC2)CC)ccnc(C)n1 C1(OCCn2cc(CNC(C3N(C(C)=O)CCC3)=O)nn2)CCCN(C(N)=O)C1 c1(CC)ccc(S(=O)(=O)NC2CCN(S(=O)(=O)c3cnn(C)c3)CC2F)cc1 C12(CNC(=O)C=Cc3ccco3)CCCCC1CN(C(c1cnsn1)=O)C2 n1(CCC(N2CCC3CN(C(=O)COCC4CC4)C3C2)=O)ccc2ccccc12 C(=O)(C(CO)NC(=O)C(c1cccnc1)N)OC c1(NC(c2ccc(C(C)CC)cc2)c2n(CCCC)nnn2)cccc(C#N)c1 c1(C(=O)NCC(CO)NC(CCCOC)=O)cnc(C2CCC2)nc1O N(C1CCCn2ccnc21)C(CC(CNC(C1(C)CC(F)(F)C1)=O)OC)=O c1(OC)cc(C(c2nnnn2CCN2CCOCC2)NCC=CBr)cc(Cl)c1 C1(NC(Cc2nc(=N)[nH][nH]2)=O)C2CC(O)C1N(C(=O)Cn1nc(Cl)ccc1=O)C2 C12(CNC(C3(CC)CC3)=O)CC(CO1)N(C(=O)Cc1ccccc1SC)C2 C(CO)(C(=O)N(C1CC1)CC1CCCN1C(c1cnsn1)=O)NC(=O)OC(C)(C)C C(=O)(CCN(OC)C(=O)C1(C)CCCN(C)C1)NCC#CC CC(C)CS(=O)(=O)CC(=O)NCCN(CC(C)O)C(c1ccc(=O)n(CCF)n1)=O C(=O)(C#CC1(C)CCCO1)N1CCC(N(C)C(c2ccc(CO)cc2F)=O)CC1 C1(C(N2CCC(O)(C(C)NC(C3CC(F)C3)=O)C2)=O)CCc2ccnn2C1 C1(C(=O)OC)CCC(C)N(C(=O)CCNc2cc(C(N)=O)nc(Cl)n2)C1 C1(NC(C(CCNC(C23OCCC(C)(C2)C3)=O)O)=O)CCCCC12CCC2 c1(C(C(=O)NCCN(C(=O)C=Cc2ncc[nH]2)CC2CC2)O)ccccc1Br N1(CC)C(=O)CCC1CC(=O)NCCCC(C)NC(=O)CCNS(C)(=O)=O c1(N(CCCC)C2CC2)nccc(N2CCC(c3nc[nH]n3)CC2)n1 N1(C(CCN(c2ccccc2)C)=O)CC2CC1C2NC(c1c[nH]c(C(N)=O)c1)=O C(=O)(C(CC(C)C)c1ccccc1)NCC(C)N(C(c1c(OC)csc1)=O)C C=CCC(C)(C)CC(=O)NC1CC(OC)CN(C(=O)C(C)N(C)C)C1 CN(C)NC(=O)CCC(=O)NC1CCCCC1N(C)C(c1cc(C(N)=O)c[nH]1)=O C1(NC(CC2CCN(C(c3cncc(CC)c3)=O)C2)=O)CC2CCC(C1)N2CC C(=O)(CC(CC)C(C)(C)C)N1CCC(OCC2CCN(C(C(F)=CC)=O)CC2)C1 C(CC(C)(C)C)(C(=O)NCc1ccc(F)cc1)NC(CCCOC(C)=O)=O Cc1nnc(CCC(=O)NC(CO)C(C)NC(=O)CC2CC2(C)C)n1C C1(CNC(C2N(C)C(=O)NC2)=O)CC2COCC2N1C(c1csnn1)=O CCCCCC(O)C(=O)NC(CNC(c1nc(C2CC2)cs1)=O)Cc1ccccc1 c1(C(C)NCCc2ccccc2Cl)ccc2nc[nH]c2c1 Cc1cnc2n1CC(C(=O)NCC(C)CNC(C1CCC(C(N)=O)CC1)=O)CC2 Cc1cc(C(=O)NCCC(C)NC(=O)CCCN(C)C(=O)OC(C)(C)C)sc1Cl Cc1cccc(Br)c1OCC(=O)NC(CNC(C1CCOC1C)=O)CC(C)C c1(C(=O)NCCC2N(C(C=CSC)=O)CCC2)cccc(Br)c1F Cc1ccnc(C(C)NC(=O)C(c2ccccc2F)(F)F)c1 S(=O)(=O)(CCC(=O)NC1(C)CC(NC(=O)CC2CC3CC3C2)C1)NC C1(C#N)(NC(c2c(C)n(CCC#N)nc2)=O)CCOCC1 S(=O)(=O)(c1ccc(NCC2CCCSC2)cc1Br)N(CCC#N)CC1CCCO1 c1(COC)ncc2c(n1)CCN(c1ccccc1C(c1cccs1)=O)C2 C1(C)(C(=O)NCC2(CC(=O)NC3(C(COC)O)CC3)CC2)CC=CCC1 C(CC(C(=O)NCCCC1(O)CC1)NC(c1cnc(S)nc1)=O)N(C)C N1(C(c2c(C)non2)=O)CCN(C(C2C3CCCOC23)=O)CC(C)C1 c1(C(N2CC(CNC(c3ncc(CC)s3)=O)C(C)C2)=O)c([N+](=O)[O-])c(C)nn1C c1(C(=O)NC(CC)(C)CCC(=O)O)nc2ccccc2n1C1CCN(C)CC1 N1(C(C(C)(C)CF)=O)CCC=C(C(=O)NCC2CCOC2C(C)(C)C)C1 C(=O)(C(CNC(=O)C(CN(C)C)N(C)C)CC1CC1)NCCNC(C(C)C)=O C(=O)(CC(C)CC(F)(F)F)NC1C2(CN(C(c3c(C)cccc3F)=O)C2)CCC1 C#Cc1cccc(C(=O)NC2CC(C)(NC(c3cc(C)nc(C)c3)=O)C2)c1C N1(CC)CC(C(=O)NCC(C)(C)NC(=O)CC2CCC(C(F)(F)F)O2)CCC1=O c1(OC)ccccc1CC(C)CC(=O)NCC1(NC(=O)CCNS(C)(=O)=O)CC1 c1(C(N2C3CN(C(c4cc(NC(C)=O)ncc4)=O)CC32)=O)c(F)cc(Cl)cc1F c1(C(c2n(CCCOC)nnn2)NCC(C)(CC)CO)ccc2occ(C)c2c1 C(=O)(C(CC(N)=O)NC(=O)CC1(C)CC1)NC1CCC(C(=O)OC)C1 N1(C(CC(CC)C)=O)CCCC2(C1)CN(C(=O)C(C1CCC1)OC)C2 C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCCCCCNC(=O)CCCCC1CC1)C S(=O)(=O)(c1cccc2c(Cl)nccc12)N1C2CCN(C(CC)=O)CC2CC1 C1(NC(Cn2cc(CNC(c3ncccc3Cl)=O)nn2)=O)CC2CCC1O2 c1(C(=O)NC2(C(N(CCc3nc(C)on3)C)=O)CC2(C)C)cccnc1S c1(C(C(F)(F)F)NC(c2cc(-c3ccccn3)[nH]n2)=O)ccc(C2CCC2)cc1 c1(C(=O)NC2(C)CC(NC(c3ccncc3)=O)C2)cccc(Cc2nc[nH]n2)c1 C(CCNC(C1CCCCC1n1ccnc1)=O)(C(C)C)NC(c1cc(C)[nH]n1)=O N1(C(C(COC)(F)F)=O)CCC(C)(C)C(CNC(C2(SC)CC2)=O)C1 c1(C(=O)NCC(CCCC)NC(=O)C(CC)CCC)nc(Cl)ccc1N C(=O)(C(F)C(F)(F)F)NC(c1nc(C(F)(F)F)cs1)C(=O)OC N1(C(C2(C(C)C)CC2)=O)CCCC(NC(=O)CCC2(C)CC2)C1 c1(CC)ncc(Cl)c(C(=O)NCC2CC3(CC(NC(=O)CC(C)(C)CC)C3)C2)n1 Cc1ccc(CC(N2CCOCC2C(C)NC(c2coc(CO)c2)=O)=O)c(Cl)n1 C1(C)(NC(C(C=C)O)=O)CCN(C(c2cc(C(C)C)nn2-c2ccccc2)=O)C1 c1(C(=O)NC2C(OC)CN(C(=O)C(c3cnn(C)c3)O)C2)cc2c([nH]1)CCOC2 CN=c1nc(N2CCC(C)(N(C)C)C2)[nH]c(=NCC2(F)CCOCC2)[nH]1 N1(C(=O)OC(C)(C)C)CC2CCCC2(c2nc(CNC(C3(CF)CC3)=O)no2)C1 c1(C(=O)NC2(C)CC(NC(C(C)O)=O)C2)ccc(=N)[nH]c1 CCCCC(CNC(=O)CN(C(=O)C(c1cccn1C)=O)CC)CCC C(=O)(CC1OC(=O)c2ccccc21)N1CC(C(C)C)N(C(c2cnsc2)=O)CC1 C(=O)(C1=CCS(=O)(=O)C1)N1CCN(C(C2CC3C(C2)C3(F)F)=O)CC1CCO N1(C(c2c(C)c(Br)cnc2)=O)CCN(C(=O)Cc2ccnn2C)CC2(CC2)C1 N1(C(=O)NC2C(C)COC2)CCc2nc(O)ccc2C1 C(=O)(C1=CC2(CCN(C(=O)C(C)n3ccnn3)C2)C1)Nc1ccc(C(C)C)nc1 C(C(C)(C)C(=O)NCC1(C)CCC(NC(c2ccc(C(C)C)cc2)=O)C1)OCC C(=O)(C(O)C(C)(C)C)NC1C=CC(CNC(c2nc(OC)oc2)=O)C1 O=S(=O)(NCC(O)COc1ccc(Br)cc1)N1CCc2ccccc2C1 N1(C(c2cnc(C(C)OC)s2)=O)CCN(C(C23CC(F)(C2)C3)=O)C(CO)C1 N1(C(CCC=C)=O)CC2(COC(CNC(=O)Cc3nocc3C(C)C)C2)C1 C(C(C)C(C)(C)C)N(C(c1ccccn1)C)Cc1ccc(OC)o1 c1(C(N2CC(NC(c3cc(O)cc(F)c3)=O)C(F)CC2)=O)ccc2nc[nH]c2c1 C1(NC(C(CC)OC)=O)C=CCC(C(=O)NCCS(=O)(=O)NC)C1 C(C(=O)N1CCOC(CN(C)C(c2cnoc2C(C)C)=O)C1)(C(C)C)SCC Cc1cn2c(CC(N3CCN(C(=O)C4=CCOCC4)C(C)C3C)=O)csc2n1 c1(C(=O)NCC2(C)CCN(C(=O)Nc3cc(F)ccc3F)C2)ccc(O)cc1Cl C(=O)(CCCCN(C)C(C)=O)N(CCNC(c1cnc(CC)s1)=O)C c1(C(N(C2CCN(C(c3cc(Cl)c(Br)c(Cl)c3)=O)C2)C)=O)ccc2c(c1)OCO2 N1(C(C(C)=C(CC)C)=O)CCCOC(CNC(=O)CC2CCN(CCF)CC2)C1 C1(=O)CCCCN1.c1(CONC(CC2N(CC)CCC2)=O)ccccc1F c1(C(N2CC(CNC(c3ccoc3Cl)=O)C2)=O)cc2ccc(F)cc2nc1O NC1CN(C(c2cc(Cl)ncc2F)=O)C2(CCCCCC2)C1 Cc1ccc(C(N2CCCN(C(=O)CC3(CO)CCCC3)CC2)=O)cc1CO N1(C(C(CC=C)C(C)C)=O)CC2(C1)CN(C(=O)COCc1ccccc1)CCO2 N1(CC)CCCC1C(=O)N(C)CC1(NC(=O)CC2CCCO2)CC1 C(=O)(CCC(C)(C)C#N)NC(CN(C(C1CC1c1ccncc1)=O)CC)C C(C(=O)NCc1cc(Cl)ccn1)(C(C)O)NC(C(C)=CC=C)=O C1(NC(c2c(C)nc(C)[nH]2)=O)(CNC(=O)C(C)(C)C(C)O)CCCCC1C N1(C(c2c(C)con2)=O)CC2CN(C(c3cc(Br)ccc3N)=O)CC2C1 C(CC(C(=O)N(CC(O)CN(C)C(c1ccc(CN(C)C)cc1)=O)C)OC)OC Cn1c(C(N2CC3CC2CN3Cc2c(Cl)cncc2Cl)=O)cccc1=O Cc1c(C(N2CCCC2CN(C(=O)C#CC(C)(C)C)C2CC2)=O)cncc1Cl N1(C(C2C(COC)CC2)=O)CCC2(CCCN(C(=O)CSc3cccnc3)C2)C1 C#CC1CN(C(c2cn3ccnc3cn2)=O)CCN1C(C1CC1C(C)C)=O CC1(CC(=O)NC2(CCO)CN(C(C3(C(N)=O)CCC3)=O)C2)OCCO1 Cc1cc(C(=O)NC2COCCC2NC(C2CC23CC(F)(F)C3)=O)c(Cl)cc1N c1(NCC2CC(C)NC(=O)C2)nc(N(C)Cc2ccccc2Br)nc2sccc12 CCC(C)CCCC(=O)NCC(C)(C)NC(c1cn(CCOC)nc1C)=O c1(C(=O)NCCNC(CC(=C=C)C)=O)ccc2c(c1)C(=O)CCC2(C)C C12(C(N(CC(=O)N(CC)CC)C)=O)CCCC1CN(C(C1(C)COCCO1)=O)C2 N1(C(C2C(CC)CCC2)=O)CC(F)(F)CC1(C)CNC(c1snnc1C1CC1)=O C(=O)(C(C)(C)C(C)NC(=O)C(c1ccn(C)c1)C)N(CC(C(C)C)OC)C c1(C(N2C(CNC(C(C)NS(C)(=O)=O)=O)CC2)=O)cc2sccc2cn1 C1(NC(C2(OC)CS(=O)(=O)C2)=O)CC2CCC(C1)N2C(c1snc(O)c1Cl)=O c1(OC)cc(C(=O)NC(c2cccnc2)C(=O)N2CC(c3ccccn3)C2)nn1C n1(C(C)C)ncc(Cl)c1C(N1CCC(CCN(C)C(C2(C#N)CC2)=O)CC1)=O c1(C(N2CCC(CNC(C(CC)OC)=O)C2)=O)nc2nccc(C)n2n1 C1(CC)C(NC(=O)CN(C)S(N)(=O)=O)CCN1C(c1cn(C2COC2)nn1)=O C1(C(=O)NCC(C)(O)C2CC2)(SC)CN(C(=O)C(F)OC(F)(F)F)C1 c1(CC(=O)NC2CN(Cc3cccc(OC)c3)CC2(F)F)cnc2ccccn12 c1(OC)ccc(C2CC2C(=O)NC2CCCC2Oc2ccc(Cl)cc2)cc1 N1(C(C(CC)(C)O)=O)CCC(NC(=O)C(C)(C)CCOC)C(CO)CC1 N1(c2nc(NCC(=C)Br)c3c(n2)scc3)CCc2c(Cl)cc(F)cc2C1 Cc1coc(C(=O)NCC(=O)NCc2cn(-c3cnn(C)c3C)nn2)c1C C1(CC(=O)NCc2ccc(C)s2)CC(NC(c2cc(O)nn2C)=O)C1(C)C C(=O)(C1=NOC(C)(C)C1)NC(CN(C(c1scnc1Br)=O)CC)C C12(NC(Cn3c(C)cc(C)n3)=O)CCCC1N(C(c1ccc(F)cc1Cl)=O)CC2 c1(CC(C)C)ccc(C(=O)N(c2ccc(N(C)C)nc2)C(C2C=CC(N)C2)=O)cc1 c1(C(=O)NCC2CCN(C(C(C)N(C)C)=O)C2)c[nH]c(=NCC(F)(F)F)cn1 c1(C(=O)NCC(CO)NC(C=CSC)=O)cnn(C)c1C(F)(F)F C1(NC(CONC(CNC(=O)OCC)=O)=O)CN(C)CC1(F)F C1(CNC(C(CCO)N(C)C)=O)CC2(C1)CN(C(=O)CC1(C)CCOCC1)C2 c1(C(=O)NC2C(NC(c3nc(C(=O)OC)oc3)=O)CCCC2)c(C)[nH]c(C)c1C c1(C(=O)NC2CCN(C(C(CC)CCOC)=O)C2(C)C)cn2c(C)cccc2n1 Cc1nc(NCC23CC(CN2C(C2CCCCN2C)=O)C3)cc(O)n1 c1(C(N2CCC(NC(=O)CCC3OCCO3)(CO)C2)=O)ccn2c(O)nnc2c1 c1(CCC)ccc(NC(C2CC(C)N2C(=O)CC2(O)CCC2)=O)cc1 Cc1cccc2oc(C(N3CC(NC(=O)CCc4ccoc4)C4(CC4)C3)=O)cc12 C1(C(=O)NC(CCNC(C(C=C)OC)=O)(C)C)CCOC1C=C C1(C(=O)NCc2scc(C(=O)NCC3(C)CC3C(F)(F)F)c2)OCCC1(C)C CC(c1ccc(C(F)(F)F)cc1)=CC(N1CC(NC(=O)CC(C)(C)N(C)C)C1)=O c1(N(C)Cc2nc(C)[nH]n2)nc(NCCc2cc(F)cc(Cl)c2)c2ncsc2n1 c1(CCC(=O)NC(CNC(C2(CCOC)CCCC2)=O)C)ncc(F)cn1 c12cccc(c1)N(CC)C(=O)CCNC2.N1(CC(=O)OC(C)=O)CCCC1 C1(C(=O)NC2CC(CNC(C(C)Cc3cnco3)=O)C2)CC12CCCCC2 N1(C(c2ccc(C)c(OC(F)F)c2)C(=O)NCCC2CC2)CC2CCN(C)CC2C1 N1(C(Cc2ccc(OC)cc2F)=O)CCCC12CCN(C(=O)C(C(C)C)OC)C2 c1(NC(C2(Cc3nc[nH]n3)CC2)=O)nc(C2CC2)cs1.CC(C)C(=O)N1CCO1 c1(C(=O)NC2C(NC(C3N(CC)CCOC3)=O)CCC2)n[nH]c2ccc(Cl)cc12 NC1CS(=O)(=O)C2CN(C(=O)C(=O)Nc3c(F)cc(F)cc3Br)CC12 C#CC1(NC(=O)C(C)C(C)NC(c2cc(C)nc(C)n2)=O)CCCCCC1 C1(NC(CC2N(C(c3nc(C)sc3)=O)CC2)=O)CCCC2(CC1)CC2 c1(SC)ccnc(N2CCC(NC(c3ccnc(O)c3)=O)C2)n1 C(=O)(C(O)C(C(C)C)OC)N(C(CC)CC(=O)N1CC(C)(C(=O)NC)C1)C N1(C(C2(c3c(C)cccc3)CC2(F)F)=O)CCN(C(c2cnns2)=O)CC(O)C1 c1(C(N(CC(CC)NC(=O)CSc2cccc[n+]2[O-])C)=O)cn2nc(C)sc2n1 Cn1cncc1C=CC(N1CC(F)CC1C(=O)NCC1CC2(CCC2)C1)=O N1(C(C=CC2(C)COC2)=O)CCC2CN(C(=O)CCC3CCCO3)CC12 CCC(N=c1[nH]c2c(c(=NCCCC#N)[nH]1)SCC2)c1ncc[nH]1 C1(C(=O)NCC(CO)NC(CCC#C)=O)CCC(=O)N(C(C)C)C1 C1(CNC(c2c(C)n(C3CC3)nc2)=O)CCN(C(=O)Cc2cn[nH]c2)C12CCC2 c1(OC)ccc(O)cc1-c1csc(NC(=O)CCSCc2ccccc2)n1 CC1(C)CC(C(=O)NCc2csc(CNC(c3cc(C4CC4)no3)=O)n2)CO1 N1(C(C2C(OC)CCCC2)=O)CC2(C1)CN(C(c1coc(C)c1)=O)CCO2 C1(C(=O)NCC2(C(C)NC(c3c(C)csc3)=O)CC2)CCC(C(F)F)CC1 C1(NC(c2ccc(C3CC3)o2)=O)CCCCCC1NC(C1CSCCS1)=O C1(NC(CCS(=O)(=O)NC)=O)CCC2(CCCN(C(c3cc(OC)n[nH]3)=O)C2)C1 c1(CN2C(C(=O)NCCC(N3CCN(C)CC3)=O)CC(O)C2)cccc(F)c1Cl C(c1ccccc1)=CC(N1CC=CC(NC(C2(CF)CC(F)(F)C2)=O)C1)=O c1(CN2C3CC(NC(C4CCCO4)=O)CC2CC3)cccc2c1CCCC2 N(C(=NCCCC(C)(C)C)N1CCC(OC)C(C)C1)C(CC)CC c1(CC(N2CC(O)CC(NC(C3(N=[N+]=[N-])CC3)=O)C2)=O)ccc2c(c1)CCOC2 c1(C(=O)NC2CC(O)(CNC(c3c(C)n(C)cn3)=O)C2)ccc(O)nc1Cl c1(C(N2CC(F)CC(C(=O)NC(C#C)C)C2)=O)cc(O)cc([N+](=O)[O-])c1 c1(C(=O)NC2C(CNC(c3ccnnc3)=O)CC2)nc2ccc(Br)cn2n1 C1(NC(Cn2cc(-c3ccc(C)c(C(F)(F)F)c3)nn2)=O)CC12CCCCCC2 C(C(C(F)(F)F)N1CCN(C(C2CCCCS2)=O)CC1)NC(COC)=O c1(COC(C)=O)cccc2c1cnn2C.c1(C2C(=O)N2C)cccc([N+](=O)[O-])c1 C1(CNC(C2C(=C)C2)=O)CCC2(CCN(C(c3cnc4n3CCS4)=O)CC2)CO1 N1(C(c2c(OC)ccnc2F)=O)CCCN(C(=O)COC(C)=O)C(C)C1 C1(C)(NC(c2c(CNC(Cc3cc(CC)no3)=O)noc2)=O)CCCC1O N1(C(c2c(C)cns2)=O)CCC(C)(CNC(c2ccc(O)c(N)c2)=O)CC1 c1(C(=O)NCCC(CNC(C2(CCC)CC2)=O)O)[nH]cnc1C#N N1(S(=O)(=O)c2cccc(Cl)n2)CCc2cc(-c3ccc4nonc4c3)cnc2C1 c1(C(N2C(CNC(C3C(C)=C3)=O)CC3(CC3)C2)=O)cnn2c1NCC(C)C2 C1(CNC(c2ncnc(OC)c2F)=O)(CO)CC12CCN(C(=O)C=C(C)C)CC2 N1(C(C2(OC)CCC2)=O)CCCCC(C2CN(C(C34CC3CCC4(F)F)=O)C2)C1 CCCS(=O)(=O)C(C)C(=O)N1CC(NC(c2cccc3[nH]ncc23)=O)CCC1C CC(C)(C)C1=NOC(C(=O)NCCCNC(=O)CCCN2CCCC2)C1 C1(C(=O)NC2(C)CCOC2=O)(CC)CCN(C(C2CN(C)CCO2)=O)CC1 CCC(COC)C(=O)N1CC(CCNC(C2(O)CCC2)=O)(OC)C1 c1(C(N2CC(C)C(NC(C3CCC(=O)N3)=O)CC2)=O)cccc(N=[N+]=[N-])c1 CCCCC(C(=O)NCc1csc(CNC(=O)COC(C)C)n1)ON=C(C)C CC1CCC(F)(C(N2CCN(C(c3sccc3F)=O)C(CC3CC3)C2)=O)CC1 C#CCC(C)(CNC(=O)NC1(Cc2ccccc2)CCOC1)CO N1(Cc2nnn(C)n2)CCCCC1CNC(=O)CC(=O)Nc1ccccc1 c1(C(C)C(=O)NCC(=O)N(C(C(N)=O)C2CC2)C)ccn(C)c1 c1(C(N2CC3CN(C(=O)C(Cl)(Cl)Cl)C3C2)=O)cc(I)c(F)cc1F N1(C(C(C)O)=O)CCC(C2CC2)C1CNC(=O)CCC(C)(F)F C1(NC(=O)Cc2ccco2)CCCN(C(=O)CCc2cccc(F)c2)CC1 c1(C(N2C(C)CC2C(N2CC(F)(F)C2C2CC2)=O)=O)cn2ccccc2n1 C1(NC(c2coc(CO)c2)=O)CN(C(c2ccoc2C2CC2)=O)CC12CCC2 c1(N2CC(CCCCNCc3ccc(N(C)C)cn3)C2)nc2cccc(F)c2o1 c1(C(=O)NCCCC(=C)C)ccc(C)c2c(C#N)c[nH]c12 N#Cc1ccc(Br)cc1CN1CC(C(=O)Nc2ccc(F)c(I)c2)C1 c1(C(=O)NCc2cccc(CNC(CC)=O)c2)cnc2nc(C)ccc2c1O c1(C(N2CCC(OCC(=O)N(C(CC(C)C)CO)C)C2)=O)cnn2ccccc12 c1(-c2cn(C3C(C(C(=O)C(C)(C)c4ccn(C)n4)C)C3)nn2)cc(Cl)c(Cl)cc1Cl Cc1cncc(CC(=O)NC(C)CCNC(c2onc(C)c2C)=O)c1 C=C1CCN(C(C2CN(C3CCC3)C2)=O)C(C(=O)NCCc2cccc(C)c2)C1 C(=O)(C1=NN(CC)C(=O)CC1)N(CC(CC)NC(c1ccn(C)c1)=O)C C12(CC(=O)N(CC(F)F)CCC)CCC1CN(C(C1C3CC(=O)CC13)=O)C2 CC1OC2(C(=O)NCC3(c4ccc(C(=O)O)cc4)CC3)CCC1C2 C1(C)(COC)C=CCN1C(=O)CC(CNC(c1ccnc(CO)c1)=O)C1CCC1 C1(NC(c2nnn(CC)c2C)=O)(CNC(=O)C(F)=C2CCC2)CCCCC1C CCC(C)CCCC(=O)NCC1CC(NC(=O)CCOc2ccc(Cl)cc2Cl)C1 C1(CCC)CN(C(c2sc(OC)nc2Cl)=O)CCN1C(=O)CP(C)(C)=O CC1(C)CN(C(=O)C2=CCCO2)CC2(CN(C(=O)CC3(O)COC(C)(C)C3)C2)O1 N1(C(C(C)NS(C)(=O)=O)=O)CC2CCCN(C(=O)CCC3CCCC3)C2C1 c1(CC)cncc(CNC(=O)CN(CC(C)C)C(=O)CC23CCCC2C3)c1 c1(OC)ncc(C(N2CCC(NC(c3cc(C)co3)=O)C23CC3)=O)nc1C C1(C(N2C(CNC(c3c(OC)ccc(C)n3)=O)CCC2)=O)CCn2ccnc2C1 c1(C(=O)OC)ccc(Cl)cc1S(=O)(=O)NC(c1nc2ccccn2c1Cl)=O c1(N2C3(CN(c4nc(SC)nc(C)c4Br)C3)CC2)ncc2cccc(Br)c2n1 C1(CC(=O)NCC(C)(C(C)C)NC(CCCC(C)C)=O)CCc2sccc2C1=O c1(C(=O)NC2CN(C(c3cc[nH]c3)=O)CCC2CO)cc2c(=O)cc[nH]c2s1 c1(CCNC(CCC=C)c2nnnn2C)cnn(-c2ccc(C)cc2)c1C C1(CC(N2CCC(N(C(=O)CN(C(=O)C(C)C)C)CCC)C2)=O)CC(=O)NC1=O c1(CN2CCCC(N)(CC)C2)nc2cccc(C)c2o1 C=CC(CC)CC(=O)N1CCC(OCC(N2CC(SC)C2)=O)C1 CCCC(C)(C)C(=O)N1CC2C(CNC(=O)CCc3ccccc3OC)C2C1 c1(C(N2CC(NC(C(C)(C)C3CC3)=O)C3C2C3)=O)ccc(C(F)F)c(Cl)c1 CCC(C)CC(=O)C(=O)N1CCOCCC1C(=O)Nc1cn(C)c(=O)nc1O CCCCN=C(NCc1ncnn1CC)NC1CC(C)CC(C)C1 c1(C(C(=O)NC)N(C(C)C(=O)OC)C2CC2)ccc2c(c1)OC(C)(C)O2 C1(C(=O)NC(CO)CCF)(NC(C(c2ccnn2C)C)=O)CCCCC1 C1(C(=O)NCc2c(C)ccs2)CCCN(C(c2noc(C3CCCO3)n2)=O)C1 CC1(C)C(NC(=O)C=Cc2cccc(F)c2)CCN1C(c1n[nH]c(=N)s1)=O CC(CN(C(=O)Cc1ccc([N+](=O)[O-])cc1F)C)N=c1ccnc(CO)[nH]1 C=CCCCC(C(=O)Nc1cccnc1)NC(=O)CCNC(=O)CO CN1C2CCC1CC(C(=O)NC1CC(CNC(=O)CN3CC(=O)NC3=O)C1)C2 c1(OCC(=O)NCC(C)(CC(C)C)NC(CSCC)=O)ccc(S(N)(=O)=O)cc1 N1(C(CCCc2onc(CC)n2)=O)CCCC(NC(c2cn(C)nn2)=O)C1 C(=O)(CCCCCCC(C)C)N1CCC(C)(Nc2ccnc(C(CC)C)n2)C1 C(=O)(C(C)(C)C(C)(C)C)NCCOCCNC(C(C1CC(F)(F)C1)OC)=O c1(CCC(=O)N(C(CNC(c2cccnc2O)=O)C2CC2)C)ccc(O)nc1 c1(C(N2CCN(C(CCOCC#C)=O)CC2)=O)cnc2n1CCCC2C c1(NC(C(c2ccc(C(C)=O)cc2)CC)=O)ccc(C)c(CO)c1 c1(OC)noc(C(N2CC(CNC(=O)Cc3n[nH]c(C)n3)C(C)C2)=O)c1Br c1(OCCC(=O)NC(CC)CNC(=O)CSCCC#N)cccc(C)c1 c1(-c2cn(C)nc2)nc(=NC(=O)C2(C)CNC(=O)N2)s[nH]1 CC(C)CCC(=O)NC(C)(C)COCCCNC(c1cnn(C2CC2)c1Cl)=O n1(CCCC)ncc(C(=O)NC(CO)C(C)NC(C2(C)CCCOC2)=O)c1C c1(N(C)Cc2cccnc2)nc(N2CCC3(CC2)CC3)nc2c(F)cccc12 c1(C(N2CC(CNC(CCCC#C)=O)C(C)C2)=O)cc(C#N)ccc1C C12(CNC(C(c3ccccc3)SC)=O)CN(C(=O)CCC3CC3)CC1CCO2 C=C(C)CN=C(NCc1ncnn1C(C)(C)C)NCC1CCCN1CC C1(C(=O)Nc2ccc(OC)c(C)c2)CN(C(C2(CO)COC2)=O)CC1C1CC1 c1(OC)cccc2c1OCC2NC(c1ccc(C(F)F)cc1)C(=O)NC1(C)CC1 C(=O)(CC1=CCCCC1)O.c1(N(C(C)C)C)nnc(C2CCS(=O)(=O)C2)n1CC1CC1 C12(C(=O)NC(C)(CNC(c3cc(Cl)cs3)=O)Cn3cccn3)CCCC1C2(F)F c1(C(=O)NCC(C)CNC(c2nocc2Br)=O)cnc(C2CCOCC2)s1 N1(CC)CCC(c2nnnn2C2CC2)(NCCN(C2CCCC2)C)C(C)C1 c1(N(C2CCNC2)C(c2nccc(C)c2)=O)ncnc2cccnc12 C(=O)(CC(O)Cc1ccccc1)N1CC(NC(CN(C)C)=O)C1 C(=O)(C#CC1CCOC1)NC1CC(C)(NC(c2cc(C(F)(F)F)c[nH]2)=O)C1 CC1CCC(NC(c2cc(Br)cc3c2OCCO3)=O)c2ccccc21 C(C)(C(=O)NCCCN(CC(C)C)C)(C1CN(C(C)=O)C1)NC1CC1C(N)=O c1(C(=O)NC2CC3(CC(C(=O)NC(C(C)C)CO)C3)C2)cc2ccccc2n1C C(C(=O)NC1CC(C(=O)NCCc2cn(C)cn2)C1)(C(C)C)SC Cc1ccc(=O)n(CC(N2CCC(N(C(=O)C(C3CCCCC3)F)C)C2)=O)n1 C1(NC(c2ccnn2C(F)F)=O)CCN(C(C2CCC=CCC2)=O)CC1 c1(OC)c(F)cc(C(N2CC3C(C(=O)NC(C)CF)C3C2)=O)cc1F C#CCCCC(=O)NC1CCOC(CNC(C2(c3ccc(Cl)cc3)CC2)=O)C1 c1(OC)c(C(=O)NCC2CCN2C(=O)C(C(C)O)NC(N)=O)csc1C N1(C(c2c(C)nc(C)o2)=O)CCC(F)C(c2ccccc2)C1 CC(C)CC(C)(O)C(=O)NC1CCN(C(c2c(O)cc(Br)cc2F)=O)C1 c1(C(=O)NCC2N(C(C(CC)C(C)C)=O)CC(O)C2)cc(C)nc2c1cnn2C c1(C(N2CCCC(NC(=O)CC3CCCCO3)CC2)=O)nc[nH]c2ncnc1-2 Cc1nc(C2CC2)oc1C(=O)NCCOCCN(C)C(C1C(C)C1C)=O C1(C(=O)NCC2(CNC(C(C=C=C)C)=O)CC2(F)F)CC2(CCOCC2)C1 c1(C(N2C(CNC(C3CCCN(CC)C3)=O)COCC2)=O)ccnc2ccnn12 C1(O)(C(C(=O)N(CCNC(=O)CC2CCOC2)C2CC2)F)CCCC1 c1(OCC(=O)NCCCC(CO)NC(=O)CC2CCCSC2)ccc(F)nc1 C1(CC(=O)N(CCCNC(=O)C=C2CCC2)C)CC(=O)c2ccccc2C1 Cc1cc(O)cc(C)c1CC(=O)NC1CCC1NC(=O)C(C)C CCC(C)C(C(=O)N(CCCCN(CC)CC)C)N(C(=O)C=Cc1cc[nH]n1)C Cc1cc(=O)ccn1CC(N1CC(O)CC1CNC(C1(C)CC=CC1)=O)=O C1(CC(N2CC(NC(C3CCN(C(=O)OC)CC3)=O)C2)=O)CCN(OC)CC1 C1(OC)CC(NC(C2CC3C=CC2C3)=O)CN(C(c2cn(CCO)nc2C)=O)C1 c1(CCC(=O)NCC2CC2CNC(C2(CC(F)F)CC2)=O)ccc(F)c(F)c1 N1(C(CC(C)C(F)F)=O)CCC2(CCN(C(=O)CCC3CC3(Cl)Cl)CC2)C1 C1(CNC(C2N(C(C)=O)CCC2)=O)CC2CCC(C1)N2c1cc(F)ncn1 CC(Cc1cnn(C)c1)C(=O)NC(CNC(C1(C#N)CCC1)=O)C1CC1 C(=O)(C(C)(C)C(C)(C)O)NCCC(C)CCNC(=O)C=C1CCCCC1 N1(C(CNC(CC)=O)=O)CCC2(CC(NC(=O)C(C)(C)N(C)C)CO2)C1 N1(C(C=C(C)C(C)C)=O)CCC(O)(CN(C(=O)C(C)CC#N)C)C1 c1(N2CCC(C)(C(=O)NC)C2)nc(N(C)Cc2cc(Br)cn2C)nc2c1COC2 C=CCC(C)(C)CC(=O)N(CC(=O)NCC(CO)OC(C)=O)CC(C)C C1(n2cc(CCC(=O)Nc3ccsc3)nn2)CCCN(C(C2CCOC2)=O)C1 N1(C(C2CCC=CO2)=O)CCCC12CCN(C(C13CCCCC1C3)=O)CC2 C1(CCNC(COCCC)=O)CC(F)(F)CN1C(=O)Cn1cccnc1=O c1(CC)ccc(CCC(=O)NCC(CNC(C2C3CCN2CC3)=O)OC)cc1 N1(C(c2ccc(C(F)F)c(F)c2)=O)CC2CCC1C(Nc1ncnc(Cl)c1Br)C2 c1(C(Cc2cnc(NC(=O)CSc3ccc(C)cc3)s2)O)nc2ccccc2[nH]1 N1(C(C(C)O)=O)CCN(CCC2CCN(C(=O)C(F)C3CC3)CC2)CC1 C(=O)(CC1COc2cc(OCC)ccc21)N1CCC(NC(CCC)=O)C1 N1(C(=O)NC(c2ccc(Cl)cc2)COC)CCOC2CCCC12 c1(C(=O)NCC(CC)NC(=O)CCNC(C)=O)oc(Br)nc1C c1(C(=O)NCC2N(C(C)C(=O)N(C)C)CCC2)ccc2ccn(C)c2c1 c1(C(N(CCCNC(Cc2ncc(CC)[nH]2)=O)C(C)C)=O)ccc2ocnc2c1 C12(C(=O)NCCC3N(C(c4ccc(Cl)s4)=O)CCSC3)CCC(CC1)CO2 CN1C(=O)OCC1C(=O)NCC(CC(=O)N1CCCC1C1(C)CC1)N(C)C c1(OCC)c(CC(=O)NCC2(CNC(=O)CC#N)CCCC2)cccc1Cl n1(C(C)C)cc2c(n1)C(C(=O)N1CC(C(C)NC(=O)CC3CC3(Cl)Cl)C1)CCC2 N1(C(CN(C(CC(C)OC)=O)C)=O)CCN(C(=O)CSc2ccc(O)cc2)CC1 c1(COC2(CF)CC(OC)C2)c(F)cc(Br)cc1[N+](=O)[O-] C(=O)(CC1=CCN(C)CC1)N(C)CC1CCC(NC(=O)COC(F)F)CC1 C1(CN(C(=O)CCC2NC(=O)NC2=O)C)C2CN(C(c3csnn3)=O)CC12 C1(C(=O)NC2CCCC(NC(c3ccncc3O)=O)C2)CC2CCC(C1)S2 c1(C(C)=O)cccnc1N1CCCC(C(C)NC(c2ccccn2)=O)C1 c1(CC(CNCC(CO)O)O)cccc2ccccc12 C1(CNC(C23CC(CC)(OC2)C3)=O)CC(C)(C)CN1C(c1[nH]nnc1C)=O C1(CCC(N2C(C(C)C)CCC2)=O)CCCN(C(c2scnc2Cl)=O)C1 C(c1ccc(Cl)cc1)=CC(=O)NCCC(=O)NC(C1=CC=CC(O)=NC=C1CCl)C c1(C(C(=O)NCC(C)(C(C)C)NC(CC=CC)=O)C)ccc(F)cc1F N1(C(C=C(CC)C)=O)CC(NC(=O)C(C)=C2CCCC2)CC2(CC2)C1 C12(C(=O)NC3C(C(=O)OC)CC3)CC(C)(CN1C(=O)Cc1ccoc1)C2 c1(CSC)c(C(=O)NCC2(CNC(C3CC=CCC3)=O)CC2)sc2ccccc12 c1(C(C)C)ccc2c(c1)C(NC(c1nc(CN(c3ccccc3)C)n[nH]1)=O)CC2 Cc1c(Br)ncc(F)c1CNC(C)C(c1ccccc1Cl)C c1(C(=O)NCC(CNC(C2ON=C(C)C2C)=O)O)c([N+](=O)[O-])cnn1C Cc1cccc2c(C(N3CCN(C(=O)CC4CC(C)(C)CO4)CC3C)=O)c[nH]c12 N1(C(C(C)OCCCC)=O)CC(O)(CCNC(=O)CCc2cc(Cl)cs2)C1 O(NC(=O)C1=CCN(C(C2CC=CC2)=O)C1)C(CC)CC N1(C(CC(C)OC)=O)CCOCC(F)(CNC(=O)CCc2cnc(O)[nH]2)C1 C1(C(=O)NC(c2n(CC)ncc2)C)N(C(c2cc(O)ccc2F)=O)CCC1(C)C c1(N2CCC(SCCl)C2)nc(NC(=O)OC)nc(=N)[nH]1.C1CCC(=O)NC1C Cc1c(NC(=O)CCC(C)(C)NC(c2cc(Cl)n(C)n2)=O)cccc1C#N Cc1ccc(C)c(OCC(N2CC3(CCC3NC(C3CCCC(=O)O3)=O)C2)=O)c1 N1(C(c2cc(C(C)(C)C)no2)=O)CC(NC(c2nccnc2N)=O)C2(CC2)C1 C1(CNC(COCCCCC)=O)CC(NC(c2cc(C)ccc2N)=O)C12CCC2 N1(C(Cc2c(C)scc2)=O)CCOC(C(=O)NCCc2ccc(O)cc2)C1 c1(C(C(=O)NCC2(c3ccccc3)C(C)C2)=O)cc(F)c(F)cc1F c1(C(N(C2CCCC(NC(C3CCOCC3)=O)C2)C)=O)cnc2cccnc2c1 c1(C(=O)NCC2(CNC(=O)CC(F)(F)F)CCC2)cc2cc(Br)ccc2[nH]1 C12(NC(C(CSC)OC)=O)COC(C1)C(NC(C1(CO)CCC1)=O)C2 C1(NC(C(c2c(CC)cccc2)(F)F)=O)CCCCCC1NC(c1cnc[nH]1)=O N1(C(C(C)c2ccsc2)=O)Cc2ccccc2C1CNC(=O)C(F)OC(F)(F)F CCC(C(=O)N1CCC(CN(C(c2ccnc(CO)c2)=O)CC)CC1)C(C)C C1(OC)CN(C(=O)C(n2ccc(C)n2)C)CC1NC(c1cnc[nH]1)=O c1(C(=O)NC(CCOC)C(=O)N(C)Cc2nc(C)no2)ccc(C)c(O)n1 C1(C(=O)NC2CC(NC(CSc3c(C)n[nH]c3C)=O)C2)CC2(C1)CC(C)(C)C2 c1(C2CCN(c3n(CCOC)c(C4CCC4)nn3)C2)cc(OC)c(F)c(F)c1 c1(C(=O)NCC(CNC(C2C(C=C)C2)=O)(C)O)n[nH]c2ccc(F)cc12 Cc1nc(NC2CC3CC(C2)N(C(=O)CCC2CCCCO2)C3)c(C)c(O)n1 N1(C(c2ccc(OC)cc2)=O)CC(=O)NC2CN(C(c3ns[nH]c3=O)=O)CCC12 c1(NC(CNC(c2[nH]c3cc(C)sc3c2)=O)=O)c(C)ccc2c[nH]nc12 Cc1ccc(F)c(C(N2CC(C(N3CCCC(CCO)C3)=O)OC(C)C2)=O)c1 N#Cc1cc(F)ccc1C(N1CCC=C(C(=O)Nc2cccc3nsnc23)C1)=O C=CC1CCCN(Cc2coc(-c3ccc(Br)cc3)n2)C1 Cc1ccc(CN=c2[nH]cc(-c3cnn(-c4ccccn4)c3)s2)cc1Cl C1(C(=O)NC2CCN(C(c3c(C)cns3)=O)C2)(CN(C)C)CCCCC1 N1(C(C)=O)CCC2(CC1)CN(C(c1cccc3c1OCO3)=O)C2C(C)C C(C(C)(C)C1=CCCC1)NC(c1c(C)cn(C)n1)c1nnnn1CC1CC1 C1(N(C(C(C)N(C(C)=O)C)=O)C)CCC(CNC(C2(C)CC=CCC2)=O)CC1 O=S(=O)(CCCS(=O)(=O)NC12CCN(CC1)C2)NC(c1ccccc1)CF c1(C(=O)OC(C)C)ccc(C(N2CCC(CNC(C3CC3(C)C)=O)C2)=O)cc1 c1(CCC)nnsc1C(=O)NCCC(C)NC(=O)Cn1nnc(C)n1 CN1CCN(C(c2ccc(-c3ccon3)cc2)=O)C(CNC(C2CC2(Cl)Cl)=O)C1 CCC(C(=O)Nc1coc(-c2ccccc2Cl)n1)C(C)O.C12CC(C)(C1)NC2=O C1(C(=O)NC2(COC)CC=CC2)CCC(c2cn(C3CCCC=C3Br)nn2)CC1 C12(C(=O)NCC3C(NC(CCc4cc(C)sc4C)=O)COC3)COCC(C1)OC2 c1(NC(C23CC(C(=O)Nc4ncc(F)c(Cl)n4)(C2)C3)=O)c[nH]c2c(Cl)cccc12 C(=O)(C1=CCCCCC1)N1CCC(O)(CCNC(C2CC3CC2C3)=O)CC1 c1(CNC(C(C(C)O)(C)C)=O)nnc2ccc(C(F)(F)F)cn12 c1(CC)ccc(CN(C(c2ccncc2)C(=O)NCCCOC)C)cc1C CCCC(C)CC(C)(c1nnnn1C(C)(C)C)Nc1ccc(-c2cnco2)cc1 Cc1cc(C(=O)N(CCCNC(C2CCCCC2F)=O)C(C)C)cc(C)c1 CC1CN(C(c2ccc(-n3cc(CN)nn3)cc2)=O)CCO1.C12CCCCN1C2 c1(C(N2CCC(N(C(=O)CSC(F)F)C)C2)=O)cc(F)c(F)c(O)c1F c1(C(N2CC(CC=C)(NC(=O)CCn3cc(Cl)cn3)C2)=O)cc(C)cnc1Cl C1(C(NOC(CC)CC)=O)CCc2ccnn2C1 C12(CNC(C(C(C)(C)O)F)=O)CC(CCO1)N(C(c1ccc(CO)cn1)=O)C2 c1(C(=O)NCCC(CCNC(c2cncc(OC)c2)=O)C)ccc2oncc2c1 C(C1CCc2ncnn21)N1CC(NC(C2(c3cc(C)no3)CCCC2)=O)C1 N1(C(C2(CC#C)CC2)=O)CC(NC(C2(C(F)F)CCC2)=O)C(c2ccccc2)C1 CC(C)C(F)(CNC(=O)CNC(C)(C)C)C(=O)NCCCN(c1cccnc1)C c1(C(=O)NC2CCC(C(=O)NC3C(C)(COC)CCC3)C2)ncc2ccccn12 CC(C)CC(C)(CNC(=O)COC1CC(F)(F)C1)NC(=O)CCC(=O)N(C)C C1(C(=O)NC(C)C(C)(C)NC(=O)CC2OCCO2)CCc2ccccc2C1 O=C(C(F)(F)C(O)C1CC1)NCC1C2CN(c3ccc(Cl)nn3)CC12 Cc1cc(F)c(C#N)cc1NC(C1CCCC1NC(c1ccc(CO)o1)=O)=O CCC(C(=O)N(CC(C)(CC)OC)C)N(C)C(c1cn(C)cn1)=O C1(C(N(C)CC2CCN(C(C(C)OC)=O)C2)=O)CCC2CC1C2(C)C C1(CCC)(NC(=O)Cn2c(C)csc2=O)CCCN(C(=O)C=CSC)C1 O=C1CN(C(c2cc(N3CCOCC3)ccn2)=O)C2(CCC2)C1 C1(C(N(CC(C)NC(=O)CSS(C)(=O)=O)CC)=O)CCC(CCO)CC1 C1(C)(C(=O)NCC(N(C(CCCOCC)=O)C)C2CC2)CCN(C)C1 c1(C(=O)NC2(CCOC)CCN(C(CC=CC=C)=O)C2)cc2n(c1)CCSC2 Cc1c(C(N2CCCCC2CCNC(=O)COCCO)=O)cnn1C1CCCC1 c1(C(=O)NCCC(C)NC(=O)C(c2ccc(Cl)nc2)(F)F)ccc(N)c(F)c1F CC(C)(CC(=O)NC1CC(NC(c2coc3c(Br)cccc23)=O)C1)C(F)(F)F c1(C(=O)NCC(CN(C(c2cn(CC(CC)O)nn2)=O)C)O)cc(=O)n(C)o1 CC1CCC(NC(=O)C(N2CCOCC2=O)C)CN1C(=O)Cc1cc[nH]n1 C(=O)(CCC1=CCCCC1)NCC(C)(F)CNC(C1(CO)CCCO1)=O C=CCCC(O)CN(C(=O)CN(C)C(c1nonc1CC)=O)C c1(C(N2C(CO)CC(NC(C3CC34CCOCC4)=O)C2)=O)ncc(Cl)cc1F CC1NC(=O)CCC1Cn1cncn1.c12nnc(s1)NC2 CC(C)CC(F)(F)C(=O)NCC1(C)CCCN(C(=O)CC2C(C)C2(F)F)C1 CCCCS(=O)(=O)CC(=O)NC(C1CCCC1)CNC(=O)CC(C)N(C)C c1(CC)ccc(C(=O)N(C)CC2COCCN2C(c2oncc2C)=O)nc1 N1(C(C)=O)CCC(NC(=O)C(O)Cc2ccccc2)c2ccccc21 CC(C)S(=O)(=O)C(C)C(=O)NCC1(C(F)F)CCN(C(C2(C)CC=CC2)=O)C1 c1(C(=O)NCC(CNC(CC2C(C)=NNC2=O)=O)(C)F)nc[nH]c2nccc1-2 c1(CN2CCOCC(C(=O)NCCOC(C)(C)C)C2)c[nH]c2ncc(Cl)cc12 N1(C(CC2CN(C(=O)N(C(C)(C)C)CCO)C(C)(C)C2)=O)CCSc2ccncc21 C1(C(C)NC(CC2(COC)CC2)=O)CCN(C(=O)CC2CCOCC2)C1 C1(NC(CCCCC)=O)CC12CCN(C(C1CCC(=O)N1CCC)=O)CC2 C1(CC)C(NC(c2nccc(C)c2N)=O)CCCN1C(=O)C=Cc1ccoc1 C(CN=c1[nH]c2c(c(=NCCC=CBr)[nH]1)CC(C)CC2)c1cc(C)sc1C c1(C(N2CC3C(CNC(C=C4CCN(C)CC4)=O)(C3)C2)=O)cc2ccccn2c1 N1(C(CCCOC)=O)CCC(C)C(NC(=O)COCC2CC2)C1C C(=O)(C1=NNC(=O)C1)N1CC(CCNC(c2c(C)nc(CO)o2)=O)C(C)C1 c1(C(C)C)noc(CCC(=O)NC(CNC(C2COCCO2)=O)CO)n1 CC(C)(O)C(F)C(=O)NC1CCCC1NC(=O)Cn1cc(F)ccc1=O Nc1cc(N2CCC(C(=O)NC3CCN(C(=O)C4CC4)C3)CC2)ncn1 CC1OC(C)C(C(N2CCOCC(NC(C3(S(C)(=O)=O)CC3)=O)C2)=O)C1C N1(C(CCC(N)=O)=O)CCC2(CCOC2)C(CNC(=O)CC2CCNC2=O)C1 c1(NCC(CC)NC(=O)OC(C)(C)C)nccc(=NCC2(O)CCC2)[nH]1 c1(OC)nc(C)ccc1C(=O)NCC1CCCN1C(=O)Cc1ccc(C)nc1 c1(CCCONC(c2c(OC(C)C)cccc2)=O)ccc2c(c1)OCO2 Cc1cncc(C(=O)NC(c2ccccc2)C(=O)NCCCS(N)(=O)=O)n1 c1(C(N2CC3C(CNC(c4ccc(COC)cc4)=O)C3C2)=O)ccc(N)cc1F c1(OC)cc(F)ccc1C(=O)NC1CN(C(c2cc(C(F)F)no2)=O)CC12CC2 N1(C(CC(C)C)=O)CCCN(C(C2CC(=O)N(C)C2)=O)CCC1 C1(C(=O)NC(c2cnn(C)c2)CC)(NC(=O)C(O)C2CC2)CC(F)(F)C1 C=Cc1cnn(C)c1C(=O)NCCC(O)CNC(c1ccc(C)cn1)=O C1(c2cccnc2)(C(=O)NCC2C(NC(=O)CCOC3CCOC3)C2)CCCC1 C(=O)(C(C)CCC(C)(C)C)NCC(CC(=O)NCC(F)(F)CO)OC N1(C(c2sc(C)c([N+](=O)[O-])c2)=O)CC(C)CN(C(c2cscc2F)=O)CC1C C(c1cccc(-c2cc(F)cnc2F)n1)=CO N1(C(C(CC(C)=O)(C)C)=O)CC(C2CCCN(C(=O)Cc3cnsc3)C2)C1 N1(C(CNC(C(n2c(C)ccn2)C)=O)(C)C)CCN(C(=O)C(C)CN(C)C)CC1 N1(C(C(CC#C)C)=O)CCC(C2CCN(C(=O)C(O)Cc3cnc[nH]3)CC2)CC1 N1(C(C2CC(SC)C2)=O)CC2CCC1CN2C(=O)CC1CC2CC2C1 C(c1ccc(F)cc1)=C(C)C(=O)NC1C=CCN(C(=O)Cc2ccc(Cl)cc2)C1 CC1=C(C)CC(C(N2CCCCC2CC(=O)NCC(=O)OC(C)C)=O)CC1 C1(CC(=O)NCCCN(C(=O)Cc2csc(C)c2)CCC)CCCC(C)(C)C1 Cc1coc(C2CC2)c1C(=O)N(CC(C1CCCC1)=O)C(c1coc(Br)n1)=O Cc1[nH]nc(Cl)c1C(=O)NCC1(F)CC(NC(=O)CC2(C)CCCO2)C1 C1(C(=O)OCc2ccccc2N2CCOCC2)CCC(C2CCCO2)O1 C1(O)(OCCOC(C=C(C)C)=O)CCCN(C)C1=O C(CC(C(C)(C)C)NC(=O)Cn1ncc(O)nc1=O)N(C)C(C1CC1(C)C)=O CC(CC(=O)N1CCCC1CN=[N+]=[N-])C(C)(C)NC(=O)CN(C)C c1(OCC)ccc2c(c1)CC(C(=O)NC1CCC1NC(=O)C(C(C)C)SC)CO2 c1(C(N2CCCC(OC)C2C)=O)c(Br)nc2n1CCC2 C1(NC(c2ccnn2CCF)=O)CN(C(=O)CN2CC=CC2)CC1C(F)(F)F C(C(CC(C)C)C(=O)NCC1CC(NC(=O)CCCF)C1)OC C1(CC(=O)NC2CC(N(C)CCO)C2)CC(O)CN1C(C1CC1(C)OCCO)=O O(N(C(=O)C1COCC1NC(C1C=CC1C(=O)OC)=O)C(C)C)CC C(CCC(=O)NC1(C(=O)OC)CC(O)C1)(C(C)C)NC(C1N(CC)CCOC1)=O Cc1ncsc1CCC(=O)NCC(C)(C)Cn1cc(C)nn1.C(CC#N)O C1(C(C(=O)NC(C(=O)NCCC2(CO)CCC2)c2cccs2)=O)CCCCC1 c1(C(=O)NC2C(NC(c3cccc(SC)c3)=O)CCC2)ccc(=N)[nH]c1Cl C1(NC(c2n(CC)cc(Cl)c2)=O)COCCN(c2nccc(C#N)n2)C1 CC(C)C(C(=O)NCc1ncsn1)C(C)NC(C1CC2CC(=O)C1O2)=O N1(C(CC=CCC)=O)CCC(O)(CNC(c2coc(N(C)C)n2)=O)C1 CC1(C)COCCC1C(=O)NC1CC(CCC(=O)NC(c2ncc[nH]2)(C)C)C1 c1(OC)c(CN(C(C(=O)NC2CC(F)(F)C2)C2CCC2)C)cccc1F C(=O)(C(F)CCC(C)C)NC1(CNC(c2cc(CC)c(Cl)cc2)=O)CC(OC)C1 N1(C(C)(C)C)CCN(C(c2n[nH]cc2NC(C2CNC(=O)C2)=O)=O)CC1 C(=O)(C(C)(C)CCC#N)NC1(C(N2CCC(CC(C)C)C2)=O)CC(O)C1 c1(CC(=O)N(C)Cc2n(CCC)cnn2)ccc(OC2CCCCO2)cc1Br c1(OC)cc(NC(C2CC(O)CN2C(c2cc(C)ccc2F)=O)=O)nc(Cl)c1 C1(C(=O)NC2(CC=C)CN(C(C3CC(CF)C3)=O)C2)CCCNC1=O N1(C(c2nnn(C(C)(C)C)n2)C(=O)NC2(C)CC2)CCC(C2CC2(F)F)C1 C(=O)(CCCCC(F)(F)F)N1CC(O)(CCNC(C(CC)C(C)(F)F)=O)C1 c1(NC(c2c(OC)cc(C(F)(F)F)cc2)=O)cc(O)nc2cccnc12 N(C1CCc2cc(F)cc(Br)c21)C(C1(N)C(C)CCC1)=O c1(C(N2CCC(NC(C3N(C(=O)OCC)CSC3)=O)C2)=O)nccc2n[nH]cc12 n1(CC(C)C(N2CCCN(C(C34CC(C)(C3)C4)=O)CC2C)=O)ccc2ccccc12 c1(CNC(=O)NC(CC=C)CO)cc(C)ccc1C(F)(F)F C(=O)(CCC(=O)NC1(CNC(C2CCC(F)C2)=O)CCC1)N(CC)CC C(c1ccc(O)cc1)=CC(=O)N(CCCCNC(C(=O)NCCOC)=O)C(C)C C1(C(=O)NCC=CCNC(=O)C(O)CN2CCCC2)OCCOC12CCC2 C12CCC(C1)N(C)C(=O)C2.n1(C2CN(C(C)=O)C2)cc(Br)cn1 CCCCCC(=O)NC1CCOC(CNC(=O)CCc2cc(C)[nH]n2)C1 c1(C(=O)NCC(CNC(CSc2n(C)ccn2)=O)F)ccc(C2CC2)cn1 C1(C(N(CC(C)SC)C)=O)CCN(C(c2cccnc2S)=O)C1C N12CCN(CC1)C(=O)C2=O.c1(C(Cc2ccccc2)N)ccc(Cl)cc1.CSC c1(C(=O)NCC2OCCCN(C(c3c(SC)ccs3)=O)C2)c(C)ncn(C)c1=O c1(C(N2CCC(CNC(C(C(C)C)O)=O)C2(C)C)=O)ccc2cccc(O)c2c1 C1(C(=O)OC)CN=C2N=C(CSC3CCC(C(N4CCCCC4)=O)O3)NN2C1 CC1CN(C(C2COCCO2)=O)CC1CNC(=O)CSCC#N c1(C(=O)NC2(CC=C)CN(C(=O)Cc3cncnc3)C2)ccn2cc(C)nc2c1 N1(C(c2n(CC)nnc2)=O)CC2(NC(=O)C(C)CN(C)C)CCC1CC2 C1(C(=O)NC(C(c2c(C)cccc2)C)=O)CCN(C(=O)CCCC2CC2)C(C)C1 C1(C(N2C3(CNC(C(CC=CC)C)=O)CCC2CC3)=O)CCc2nc[nH]c2C1 Cc1c(C(=O)N(C)CC2CCCN2C(C2(C)CC(O)CN2C)=O)cc(O)cc1N c1(SC)c(C(=O)NCC2CC(NC(c3cnc(C)[nH]3)=O)C2(C)C)cnn1C c1(-c2cn(CCC(=O)NCC3(C)N=C(C)SC3)nn2)ccc(C#N)cc1 CC(C)(C(=O)N1CCC(OCC(=O)NC2CCCNC2=O)C1)C(F)(F)F CC(CC(=O)NCC(O)C(N)=O)NC(=O)C=C1CCC1 c1(C(N(C(C)C)CCNC(c2ccnc(C(F)(F)F)c2)=O)=O)csc2nccn12 C(=O)(CCCCCO)N1C(CN(C)C(C2(CO)CCCO2)=O)CCC1 c1(C(=O)NCCN(C(CCC2CCC(C)O2)=O)C2CCCC2)nccc(Cl)c1O C(=O)(C(O)(C(F)(F)F)C1CC1)NCC(C1CCCC1)NC(C1(OCC)CCC1)=O N1(C(c2ccn(CC(C)C)n2)=O)CC(NC(C2CC3(CCC3)C2)=O)CC12CCC2 c1(C(=O)NCC2CCC(NC(C=CC(C)C)=O)C2)ccc2c(c1)NC(=O)C(C)S2 C1(CCC(C)C)C(=O)N=C2C=C(C)N1N2.Cc1c(CN)cccc1F N1(C(c2cc(OC)ns2)=O)Cc2ccccc2C(NC(c2c(C)n[nH]c2C)=O)C1 c1(N(C)C)noc(CNC(=O)CN(C(=O)CC23CCCC2C3)C2CCC2)n1 C1(n2c(-c3c(C)nc(Cn4cccn4)s3)nc(C(C)C)n2)CCS(=O)(=O)CC1 C1(CC#C)(C(=O)NCCN(C)Cc2csc(-c3ccc(C)cc3)n2)CCCCO1 c1(C2C(CNC(c3nc4cccc(Br)c4[nH]3)C)C2)ccc2c(c1)OCCO2 CCCC(C(=O)NCC(CC)(CC)NC(=O)CCOC)c1ccccc1 C(=O)(CC(C)CC(C)(C)C)N1CCC(OC)(CNC(C2C(C)C2C)=O)CC1 Cn1ncc(NC(=O)Cc2cc(Cl)sc2Cl)c1-c1cn(CCC(C)(C)C)nn1 Cc1ccc(C2CCN(C(C3CCOCC3)C(=O)NC3COC3)C2)c(C)c1 N1(C(c2c(C)ncnc2)=O)CCC2(NC(c3cn4c(n3)CCC4)=O)CC2C1 N1(C(C=CC)=O)CC2(CCN(C(=O)Cc3ccc(OC)cc3I)CC2)C1 c1(CCC(=O)NC2CCN(C(C3=C(C)CCC3)=O)C2C)nc2ccccc2s1 c1(C(=O)NC2(CC)CCCN(C(C3(O)COC3)=O)C2)cnc2ccc(C)cn12 N1(C(c2ccc(C(C)(C)C)cn2)=O)CCC2C(C1)CN2C(c1ccncn1)=O Cc1cc(C2CC2)ncc1C(N1CCCC1CNC(=O)CC1(C)CC1(F)F)=O C1(C(N2CC(OC(CC)=O)C2)=O)CC2CC1CN(C(c1oc(C)nc1CC)=O)C2 C1(NC(C=COCC)=O)CCN(C(=O)CC(C)(C)C2CC2)CC12CCC2 CC1CNC(C)(C)CN1Cc1ccc(Br)c(Br)c1 C1(S(C)(=O)=O)(C(N2CCC(C(CNC(C(CC(C)C)O)=O)F)CC2)=O)CCCC1 CCCC(CCC)CCCC(=O)NC(C)C(CO)NC(C1(COC)CCCC1)=O C1(NC(C2(NC(C3CCCCC3(F)F)=O)CSC2)=O)C2CCCCCC12 CCC(CC)C(C)C(=O)N1CC(O)(CNCc2cc(C)ccc2NS(C)(=O)=O)C1 C1(C(=O)NCCCNC(c2cn(CC(=O)N(C)C)nn2)=O)CC(S(C)(=O)=O)C1 C1(NC(c2c(CC)nc[nH]2)=O)COC2CN(C(=O)C3=CCCCO3)CC12 C12(NC(c3cccc(OC)c3F)=O)CCCN(C(c3scnc3Cl)=O)CC1C2 CN1CCOCC1C(N1CCC(C)(CNC(=O)CSC(F)F)C1)=O CC1CC(CC(N2CCC(F)(F)C2)=O)CN1C(c1c[nH]c(=N)o1)=O CCC(C)C(O)CNC(c1coc(CNC(c2ccc(C#N)o2)=O)n1)=O Cn1ccc(C(=O)NCC2OCCC2C(N2CC(CC3CC3)C2)=O)n1 c1(CC)cccc(NC(=O)C(C)N(C(c2c[nH]c(=S)cn2)=O)C2CC2)c1F c1(OC)cc(OC)c(CN2CC3CC2C3C(=O)N(CC#N)CC#N)c(OC)c1 N12CCC3C1CCN3CCC2=O.Cc1ccccc1NC(C1(C(F)(F)F)CC1)=O CN1C(=O)CSC1=CC(=O)NCC1CCC(CNC(=O)CC2CNC(=O)C2)CC1 c1(C(=O)NC2C(CNC(c3ccoc3)=O)CCC2)nnn2c1C(=O)NCC2 c1(C(=O)NCC2(O)CN(C(CC3CCCC(C)C3)=O)C2)cnc2c(c1)COCC2 c1(C(C)O)ccc(C(=O)NCCCC(CO)NC(=O)Cc2ccc(O)nc2)cc1 C(=O)(C(F)CC(C)(C)NC(C12C(=O)C3CC1C2C3)=O)NC1CC(C)(C)OC1 c1(NC(=O)NCC(CC)CO)cc(N2CCN(C(C)=O)CC2)ccc1F c1(C(=O)NCCC(C)NC(=O)C(C)(C)Cc2cnn[nH]2)c[nH]c2cccc(F)c12 N1(C(CCc2onc(COC)n2)=O)CCC(C)OC(C)C1 c1(C(=O)NCC2OCCC(NC(C(C=C=C)C)=O)C2)ccc2c(O)ncnc2c1 CC1CCN(C(C2CC(C)CC(C)C2)=O)CC1CNC(=O)CCNS(C)(=O)=O N1(C(COCCCCC)=O)CC(NC(=O)CCc2cccc(O)n2)C(CC)C1 C1(C(C)NC(=O)COc2ccsc2)CN(C(=O)COCP(C)(C)=O)CCO1 N1(C(=O)CSc2cccc[n+]2[O-])CCC2CCN(C(=O)CC3CCCOC3)C2C1 c1(OC)cnnc(C(=O)NC2CCN(CC(=O)NCc3ccc(C)cc3)C2)c1 C(C(O)C(C)(C)C)N(C(=O)CC1(NC(=O)C(=O)NC2CC2)CCC1)C c1(SC)cn(C)nc1C(=O)NC1CC(C)(NC(=O)C(N2CCCC2)C2CC2)C1 C1(O)(CN(C(C(C)NC(=O)NC)=O)C)CN(C(=O)C(O)Cn2cncn2)C1 C1(C)(C(=O)NCCN(CC(C)O)C(c2ccc(C(C)(F)F)cc2)=O)COCCO1 C1(C(CNC(C(C)=CC)=O)(C)C)CCCN1C(=O)C(CC)NC(c1ccco1)=O C(C)(CC(=O)NCCCOCCNC(=O)CCCN1CCCC1)SC N1(C(c2nccc(OC)c2C)C(=O)NCCC)CCC2(CC1)C(=O)NCCN2C Cc1ccc(C=CCC(=O)NCCCCC(C)NC(=O)C=Cc2cscn2)cc1 N1(C(c2csc(C(C)(C)C)n2)C(=O)NC)CCc2cccc(C(F)(F)F)c2C1 c1(C(=O)NCC2(F)CN(C(CC)=O)C2)ccc(C)c(S(=O)(=O)CCO)c1 C1(C(N(CCCNC(c2cc(COC)[nH]n2)=O)CC)=O)CNC(=O)C(C)(C)C1 Cc1cc(C(N2CCN(C(=O)C(C)NC(C)(C)C)CC2C2CC2)=O)ccc1Cl C(=O)(CC1OCCc2sccc21)N1CCCC(CNC(=O)CCn2ccnn2)C1 Cn1nnc2ccc(C(N3CCC4CCC(C3)N4C(c3cnc[nH]3)=O)=O)nc12 C1(C(=O)NC(C2CCN(C(c3cccs3)=O)CC2)(C)C)(CC)CCNC1=O C12(C(N(CC(C)N(C(=O)C(C)S(N)(=O)=O)C)C)=O)CCN(CC1)CC2 N1(C(C(C)OCCC=C)=O)CC2CC(NC(=O)C=CSCc3ccco3)C(C2)C1 c1(C(=O)OCC)noc2c1CN(C(c1cc(C3CCOCC3)no1)C)CC2 C1(NC(COC2(C)CCC2)=O)CCCN(C(=O)CCCc2ccc(Cl)cc2)CC1F c1(C(=O)NC)ccc(CC(=O)NCCCN(C)C(C2CC3CCC3C2)=O)cc1 Cc1cccc(OCC(=O)NC2(C)CN(C(C3CCC(=O)C(C)C3)=O)C2)c1C C1CC(C(C)C)N1C(C(CC)n1cccn1)=O.C1(OCC)CCCOC1.C1(=O)CO1 c1(C(=O)NC(CC)(C)CNC(c2nn(C)cc2C)=O)ccc(N)cc1S(N)(=O)=O c1(NC(C2CCC(CNC(=O)NCCCl)O2)=O)ccccc1F.C12CCN1C2=O C12(NC(C(CC#C)C)=O)CCC(CNC(c3ccc(C(C)O)cc3)=O)(CC1)OC2 c1(C(=O)NC2CCN(C(CS(=O)(=O)NC)=O)C23CC3)cnc2cnn(C)c2c1 N1(C(c2c(C)c[nH]c2)=O)CCN(CC2CCN(C(=O)C(O)C3CCC3)CC2)CC1 C(=O)(CCCCCC(C)C)NCCN(c1ccc(C)cc1)CCC c1(C(N(CCNC(CC(C)C2CC2)=O)C)=O)ccc(S(C)(=O)=O)cc1 c1(C(=O)NCCC2(O)CCN(C(C3(C#N)CC=CC3)=O)C2)nc2ccccc2[nH]1 C(=O)(C1Cc2ccc(Cl)cc21)NC1CC(C)(C)N(C(=O)CCc2cncnc2)C1 C1(CC(=O)N(CCCCCNC(c2c(C(C)C)con2)=O)C)COCC1(C)C c1(CN2CC(NC(c3c(OC)ccs3)=O)C(F)(F)C2)cc(Cl)c(Cl)nc1Cl C1(C(C)C)C(=O)NCCN1C(=O)CC(O)CNC(=O)C1=CCCSC1 Cc1nc(-c2ccccc2)sc1C(C)NC(=O)Cc1cc(-c2ccco2)on1 c1(C(=O)NC2CCN(C(C(C)(C)C)=O)CC2F)ccc2c(Cl)ccnc2c1 CS(=O)(=O)c1sccc1C(N1CC(CCNC(=O)COCC(F)F)C1)=O Cc1ccc(CNc2csc(-c3ccccc3)c2)cc1C#N.N12CC=CC1C2=O Cc1nc2nc[nH]n2c(=O)c1CCC(=O)N1CC(NC(C2(C)CC3CC3C2)=O)C1 C1(CCCC)CN(C(=O)C(C(C)C)OCC)CCN1C(=O)CCc1scnc1C C1(C(NOC(CC)C)=O)(N(C(=O)CN(C2CCC2)C)C)CCC(C)(C)C1 C(=O)(CC(C)C(F)F)N1C(CNC(Cn2ncc(CC)c2)=O)CC(COC)C1 c1(C(=O)NCc2nc(C)[nH]n2)ncccc1NCc1cccnc1C(F)(F)F N1(Cc2c(CC)cnn2C)CC(C(=O)OC(C)(C)C)OC(C)C1 Cc1ccc(S(=O)(=O)NC2(c3ccc(F)cc3)CCCCC2)c(C)c1 O=C1NCCCCC1C(=O)NC(c1ccccc1)c1cccnc1 c1(C(=O)NCC2(O)CCN(C(COCCC=C)=O)C2)c(C)sc2ccc(F)cc12 N1(C(c2cc(C)on2)=O)CCCC2CN(C(C3CC(=O)NC3(C)C)=O)CC12 C1(NC(C(Cc2ccco2)NC(C(C=C=C)C)=O)=O)CC2CCC(C1)N2C Cc1cccc(CC(=O)NCC(C)(O)CNC(=O)Cc2ccn(C(F)F)n2)c1Cl n1(CC(N2C(CNC(=O)C(O)C3CCC3)CCC2)=O)nnc2ccccc12 N1(C(C2N=C(C)SC2)=O)CCC(CNC(c2n[nH]cc2Cl)=O)C(F)(F)CC1 C=CC(C)(O)C(=O)NCCN(CCC)C(C1CC(C)CCO1)=O c1(C(=O)NC(C)CCNC(=O)CN(C)C(N)=O)cn(C)nc1-c1ccnn1C c1(NC(C2C3C(=O)OCC23Br)=O)cc2c(s1)COCC2 C(=O)(C(C)S(N)(=O)=O)NC1(CF)CCN(C(C2CC(C(=O)OC)C2)=O)C1 c1(C(=O)NCc2cn(CCNC(CCOC)=O)nn2)cc(C)n(C(C)(C)C)n1 N1(C(C(=O)Nc2c(OC)ccc(Cl)c2)C)CC2CCCC2(N)C1 N1(C(C(C)C)C(=O)NCCc2c[nH]c3ccccc23)C(=O)C2CCCCC2C1=O c1(C(=O)NC2CCN(C(C(C)c3cc[nH]n3)=O)CC2)ccnc2[nH]ncc12 c1(C(C(=O)NC(CNC(C(C)SCC)=O)C2CC2)(F)F)ccc(F)cc1F c1(C(=O)OCC)c(NC(=O)C(=O)NCCCc2cn[nH]c2)sc2c1CCC(C)C2 c1(C(N2CCCC(CCNC(C3COCCO3)=O)CC2)=O)ccc2cccnn12 C1(CNC(C=Cc2ccc(CC)o2)=O)COCCN(C(C2CN(C(N)=O)C2)=O)C1 Cc1sc(=O)n(CC(=O)NCCCN(C(C2C(C)(C)OC2(C)C)=O)C2CC2)c1C c1(-c2nc(CC(CC)C)nn2CCC2CC2)cccc(S(=O)(=O)CCO)c1 C1(C(=O)NC2(CC=C)CCN(C(C3CCC(OC)CC3)=O)C2)COCCC1(F)F C1(C(=O)NCCNC(=O)CO)(CC)CN(C(=O)C(n2ccc(C)n2)C)C1 C1(CC(=O)NCc2n(C(C)C)cnc2)N(C(=O)C(C)C2CCOC2)CCC1(C)C N1(C(c2nnc(SCC)s2)=O)CCN(C2CCCN(C(=O)C(C)OC)C2)C(=O)C1 CCCCC(O)C(C)C(=O)NCC1CCN(C(c2ccc(COC)o2)=O)C(C)C1 N1(C(c2c(C)n(C)nn2)=O)CCC2(CCCCC2NC(=O)Cn2cc(Cl)cn2)C1 N1(C(C2CC(OC)C2)=O)CCC(F)(CNC(c2nc(=N)cc[nH]2)=O)C1 C(CC(C)C(=O)NCc1cncc(C(=O)NCC2(F)CN(C)C2)c1)=CCC c1(N(C)CCn2ccnc2)nc2cc[nH]c2c(=NC2CC(NC3CC3)C2)[nH]1 S(=O)(=O)(c1cc(C)cnc1NCCOC(F)F)NCC(c1ccc(OC)cc1)O S(=O)(=O)(c1cnc2ccsc2c1)NC(c1ccc(SCC)cc1)=O c1(C(N2CC(C)C(NC(c3c[nH]nc3F)=O)C2)=O)ccc(C#N)c(C(F)(F)F)c1 CC1CN(C(=O)C=Cc2cn(C)nn2)CC1(C)CNC(C1(CCF)CCC1)=O C12(C(N(c3c(C)cccc3)C)=O)C3C(=O)C4C5CC(C14)C2C35 N1(C(C2(OC)CCC2)=O)CC2CC1CN2C(c1cccc(Cl)c1Br)=O c1(OCC)ncc(NC(C2CC(NC(c3nccs3)=O)C2(C)C)=O)cn1 N1(C(c2cc(C)c(C)[nH]2)=O)CC(C2CN(C(=O)C=Cc3cnc[nH]3)C2)C1 N1(C(C2(OC)CCS(=O)(=O)C2)=O)CCC2CC(NC(=O)C(C)(C)CO)CCC2C1 O=C(N=c1ccn(C2CN(N3CCn4cnnc4C3)C2)[nH]1)C12CC(CO)(C1)C2 c1(C(N2CCCC(N(C(=O)C(C)C)CC)C2)=O)ncc(Br)cc1C N1(C(c2nccc(OC)c2)=O)CCN(C(=O)C(=Cc2ccccn2)C)CC1CO c1(C(=O)NCC(C)N(C(=O)C#CC2CC2)C)ccc2c(c1)OC(C)(C)OC2 CC1CN(C(c2ccnn2CCF)=O)CCCN1C(=O)CCC1CCC(=O)NC1 N1(C(C(C=C)(F)F)=O)CC(NC(=O)CCSC(F)(F)F)C2(CCC2)C1 Cc1cc(C)c(C(N2CC3(CNC(C4CCNC4=O)=O)CC2CO3)=O)c(C)c1 CS(=O)(=O)c1ccccc1CN1CC2C(Nc3ncnc4sc(Br)cc34)C2C1 C1(C(=O)NCCC(C)N(CCC)C)C=CCN(C(c2cnsc2)=O)C1 C(c1ccnc2ccccc12)=CC(=O)NC1CCCC(NC(C(F)=C(C)C)=O)C1 C1(NC(=O)C(F)=C2CCC2)CCOC(C2CCN(C(=O)CSC(F)F)CC2)C1 c1(CNC(C(CC)C(C)C)c2nnnn2C2COC2)cccc2c1NC(=O)CO2 c1(C(N(C)CC2CCN(C(=O)COC(F)F)C2)=O)cccc(O)c1 C(=O)(CCC(=O)N1CC(NC(=O)C(C)(COC)OC)C(O)C1)OC C1(NC(C2C3CN(C(C(CCC)NC(N)=O)=O)CC32)=O)CC2CC(O)C1C2 c1(COC)nc(C)c(C(=O)NCCC2CC(NC(=O)C(C3CCOCC3)F)C2)s1 C12(C(=O)NCC3CC(NC(CN=S(C)(C)=O)=O)C(O)C3)CCC(O)(CC1)CC2 C1(C(N2CCC(CNC(c3c(SC)csc3)=O)C2)=O)CCC(=O)NC1 c1(C(N2C(CCNC(Cc3cnc(C)s3)=O)CCC2)=O)cccc2ncccc12 C#CC1CCCCN1C(=O)CCCNC(=O)Cn1nccn1 C(CCOC)(C(=O)N(C(C)C(C)C)C)NC(c1cc(COC)on1)=O c1(C(N(C)CC2CCN(C(C=C(C)C(C)(C)C)=O)C2)=O)cc(=N)[nH]cc1Br c1(OC(CC)C)ccc(O)cc1.c12ccc(cn1)CNC(=O)N(CCO)CC2 CCCC(C(=O)N1CCCC1(C)C(C)(C)C)NC(c1cc(CO)[nH]n1)=O C(c1ccccc1C#N)=CC(N1CCC(CCNC(c2c(C)nccc2)=O)C1)=O C1(CNC(c2cnc(Cl)[nH]2)=O)CC2(CCC2)CN1C(=O)CCc1nncnc1O N1(C(C2CN(C(C(C)=C(CC)C)=O)CC(C)C2)=O)CCC(F)(F)C(F)C1 C#Cc1ccc(C(=O)NC2CCC(NC(=O)C(c3cscn3)N(C)C)C2)cc1C N1(C(C(C)c2cccs2)=O)CCCC(NC(=O)CCOCC(F)F)CCC1 S(=O)(=O)(c1cc(C)cnc1NCc1occc1C)NCC(CC)(CC)SC c1(C(=O)NCCC2CC(NC(=O)C=Cc3nccs3)C2)c(F)cc(O)cc1F CC(C)C(C)C(C)CC(=O)N1CC(CNC(C23CC=CC(C2)OC3)=O)C1 c1(C(=O)NC2COCCN(c3cc(N(C)C)ncn3)C2)cc(F)ccc1[N+](=O)[O-] C1(C)(CNC(c2cnc(CC)s2)=O)CN(C(C23CCC(C2)OC3C)=O)CCO1 n1(C(CC)C)ncc(C(=O)NCC(C(C)(C)C)NC(c2coc(Cl)n2)=O)c1C N1(c2nc(Cl)c(C3CC3)cc2)CC=CCC2(CCOCC2)C1 C(=O)(CCC(=O)NC1CCN(Cc2cccc(F)n2)C1)NCCC c1(CCC(=O)NCC(C)NC(c2ncc[nH]c2=O)=O)ccc(Cl)c(F)c1 C1(C)(CNC(C=CC)=O)CCN(C(c2ccc(-c3ncc[nH]3)cc2)=O)C1 N1(C(=O)NC(C2CCCO2)COC)CCC(O)(c2nn[nH]n2)C1 C1(C2CCN(C(=O)CS(N)(=O)=O)CC2)(NC(c2c(C)n(CCO)cc2)=O)CCC1 C(CC(=O)NCC(CO)NC(C1(n2cccn2)CCC1)=O)OCCN(C)C c1(C(=O)NCCC(CNC(C2(CC)CCCC2)=O)O)ccc(O)c([N+](=O)[O-])c1 CCCC(C)(O)C(=O)NCc1ccc(C(=O)NC(c2ccccc2)CO)cn1 C1(C(C)N(C(C2CCC2NC(COC)=O)=O)C2CC2)(OC2COC2)CCCC1 c1(CCC)nc(C)c(C(=O)NCCN(CCC)C(c2sc(C(C)C)nc2C)=O)o1 C(C(C(=O)NCCCCC1CC1)NC(=O)COC)OCC.C1CCO1 N1(C(C2C(C=C)C2)=O)CCN(C(c2cc(-c3ccco3)[nH]n2)=O)C(CO)C1 N1(C(C(C)OCCC=C)=O)CCC(OCCNC(=O)C(O)Cc2cnc[nH]2)CC1 C1(C(NNC(C)=O)=O)CCN(CCNC(C(C)(C)C)=O)CC12CCC2 c1(OC(C)C)ccc(S(N)(=O)=O)cc1C(=O)NC1CN(C(C2(CO)COC2)=O)C1 CC(CC#N)C(=O)NCC1CCCN(C(=O)C(C)(F)F)C1 C(=O)(C1=NOC(CNC(=O)CC(C)(C)C#N)C1)NCC(CC)(C)O N1(C(c2cn(C)nc2O)=O)CCCC2(CCN(C(C3CC4CCC3O4)=O)CC2)C1 C12(CNC(C(C)(F)F)=O)CCCC(CN1C(=O)CCCc1cccc(Cl)c1)C2 C(=O)(C1(C)CCn2ccnc21)N1CC(C(C)NC(c2oc(CC)c(C)c2)=O)C1 C1(C(N2C(C)CCC2)=O)CN(C(c2cn(C)ccc2=O)=O)CCN1C c1(C(N2C3C(NC(C4CC5CC5C4)=O)C(CC3)C2)=O)cccc2nn[nH]c12 S(=O)(=O)(c1c[nH]c(C(N2CC(NC(C3CC3OC)=O)CC(C)C2)=O)c1)NC c1(OC)cccc(F)c1NC(C1CCCN(C(c2oc(C)nc2C)=O)CC1)=O N1(C(c2nccc(N)c2)=O)CC2CCC(NC(=O)C(c3ccccc3)O)CC2C1 N1(C(C2C(OCC)CC2)=O)CCC(C2CC2)C1C(=O)NCc1ccc[n+]([O-])c1 N1(C(CCCCC#C)=O)CCCC(C)(C)C1C(N1CCC(n2ccnc2)C1)=O n1(CCSC)nnnc1C(c1occc1C1CC1)NCc1cc(C)no1 CC(C)CC(CNC(=O)CC(C)C1CC1)NC(c1[nH]nnc1C1CC1)=O c1(C(N2CC(C(=O)NCC(C)(C3CC3)OC)C(C)C2)=O)cc2ncccc2[nH]1 C(=O)(C1=CCCCO1)N(C1CCCC1)CCCNC(C(n1cc(C)nc1)(C)C)=O c1(CN2C(CC(=O)N(CCO)C3CC3)COCC2)ccc(F)c([N+](=O)[O-])c1 N1(C(CC(C)c2ccncc2)=O)CCN(C(C2CN(C)C2)=O)CC1CC(F)F N1(C(C(c2cccs2)SC)=O)CC2CC2(CNC(=O)CN2CCC(C)CC2)C1 C#Cc1cncc(C(=O)NC2(CNC(=O)C(O)(C(C)C)c3ccccc3)CC2)c1 c1(CC)ccc(C=CC(=O)NC23CC(NC(=O)C=CCOCCOC)(C2)C3)s1 C1(c2nnnn2C2(C)CC2)(NC(CSC)(C)C2CC2)CCCCC1CCCO c1(C2(C(=O)NC(CC=C)CNC(=O)C=Cc3cncs3)CCC2)cccc(C)c1 c1(CC(=O)NCCC2CCCCN2C(=O)C(F)=CC2CC2)ccc(C(F)F)cc1 N1(C(CCCC(=O)NCC)=O)CCC2CCCC12CNC(c1cc(C)ns1)=O C1(C(=O)NCc2cn(CCC)nn2)N(C(=O)OC(C)(C)C)CC12CCOCC2 c1(C(N(CCCCNC(c2ncc(OC)cn2)=O)C)=O)ncccc1S(C)(=O)=O c1(C(=O)NC(CC(C)C)CNC(=O)CCCN(C)C)ccc2c(c1)C(=O)NCC2 N1(C(Cc2cccc(OC)c2)=O)CC2CCCC(C1)N2C(C1CCC(C)CO1)=O N1(C(c2ccnc(C(C)C)n2)=O)CC2CCC1CN(C(=O)CCC1OCCO1)C2 N1(C(CNC(C=C)=O)=O)CCOC(c2cn(C3CCOCC3)nn2)CC1 Cc1cc(C#N)cc(CCNC(CCCC2CCC(C)(C)CC2)=O)c1N c1(OC)ccc(C(=O)NCC2CC2NC(c2cccc(N)c2)=O)c(OC(F)F)c1 c1(C(=O)NC(C(C)NC(=O)C=CC2CCOC2)(C)C)cc(N)ccc1Br N1(C(CCNC(C2C(C)C2)=O)=O)CCCN(C(=O)C(O)c2cnc[nH]2)CC1 C1(C(C2CCCC2)NC2(C)CN(Cc3cccc(NC)n3)C2)Cc2nccn2C1 c1(C(C(=O)N(CCCN)C)NC(N(C)CCO)=O)ccc(F)cc1 CC1C(C(=O)NCC(CC(N2CCC3(CC2)CSC3)=O)C2CCC2)=NOC1C c1(N(C)C)cc(NC(N)=O)ncn1.N12CCC(CC1)N(C)C1CCN(CC1)CCC2 c1(C(c2ccccn2)NC(N(C(CC)CO)CC)=O)cc(Cl)ccc1Cl N1(C(C(=O)NCC)=O)CC2CN(C(c3ccc(C4CC4)nc3C)=O)CC2(C)C1 C1(NC(CCN(CC)CC)=O)CCCN(C(c2n[nH]c(C)c2Cl)=O)C1 c1(C(N2C3C(NC(CC(C)NC(N)=O)=O)CC(C3)C2)=O)cccc(C#CCO)c1 N1(C(c2cnn(CC)n2)=O)CCCC(C2CC2NC(=O)CCc2cc(C)on2)C1 N1(C(COCCOC)=O)CC(C)(C)CC1CNC(=O)C(F)(F)c1nccs1 Cc1nc2ccc(C(N3CCN(C(=O)CC4(C)CC4)CCC3C)=O)cn2n1 C1(CN(C(c2cc(C)sn2)=O)C)COCCN1C(c1ccc(O)nc1)=O N1(C(=O)COC2CCC2)CCC2(CC1)CN(C(=O)CC1C=CCC1)CC2CO N1(C(c2n(CC)ncc2Br)=O)CC2CC(C1)N(C(=O)C=CC(C)(C)SC)C2 O=C1N(Cc2ccc(OC(=O)N3CCC3)cc2)C(=O)C23CC(CN12)C3 N1(C(c2cn(C)nn2)=O)CC2(C1)CN(C(=O)C(CO)C(C)(C)C)CCO2 CCC(C)(CC)C(=O)N1CCC(C)C(CC(N2CCC(NC(C)=O)CC2)=O)C1 CC1(C)CC(C(=O)NOC2CC3CCC2C3)CN1C(=O)CCc1cccs1 c1(C(N2CCC(N(C(c3nc(COCC)sc3)=O)C)C2)=O)ccc(C)nn1 C1(c2nnnn2C(C)(C)C)(NCc2cc(C)sc2C)CCC2CCC1C2 C1(NC(C(C)CC2CC2)=O)CC(F)(F)CC1NC(c1cc(C2CC2)on1)=O C(CC(CNC(C1(C(=O)NC2(NC(C)=O)CCC2)CCCO1)=O)OC)OC.C=O N1(C(C2CNC(=O)N2)=O)CC2(C1)CN(C(C1CCc3ccnn3C1)=O)CCO2 c1(SCC(=O)NCCCN(C(=O)CCc2ccsc2)CC)ccc(C)cc1F N1(C(c2ccc(C)nn2)=O)CC2CCC(N(C(=O)C(N)=O)C)C2C1 C(c1ccccn1)=C(C)C(=O)NC1CC1NC(c1cccc(SCC#N)c1)=O Cn1nc(C(=O)OC2CCCN(C(C3(C)CCOCC3)=O)C2=O)c(Br)c1Cl N1(C(CC(C)(C)F)=O)CC(CNC(=O)C#CC2CC2)CC12CCC2 C1(CNC(c2cc(CNC(=O)CC3CSCCO3)oc2)=O)CC2(CCCO2)C1 CC1CN(C(=O)CC2(C)OCCO2)CC1CCNC(c1cnc(C(C)(C)C)o1)=O c1(CCC(=O)NC(C)CNC(=O)CSCc2cscn2)ccnc2ccccc12 C12(NC(c3c(Cl)cn(CCC)n3)=O)CCC(CC1)N(C(c1cccc(Cl)c1)=O)C2 C1(CNC(Cn2c(C)ccn2)=O)CCC(F)(CNC(C2(C#N)CC2C)=O)CC1 C1(C(N2CCC(O)(CC)C2)=O)CN(C(=O)C(C)(C)CO)CC12CCC2 c1(-c2cn(CC3C(CNC(CNS(C)(=O)=O)=O)C3(F)F)nn2)ccc(F)c(F)c1 N1(C(=O)CCc2cnc(O)o2)CCCCC1C1CCN(C(c2ccccc2)=O)C1 C(=O)(CC(O)C(Cl)(Cl)Cl)N(CCNC(=O)CC1COCCO1)CC1CC1 Cc1nc(-c2cccs2)sc1C(=O)NCCN(C(C1CCN(C)C1C)=O)C1CC1 N1(C(c2n(CC)ccc2)=O)CC2C(NC(C3CCN(C)C3=O)=O)C2C1 C(=O)(C(C(C)C)n1ncc(N)n1)N(C(CNC(CCc1cnc(C)s1)=O)C)C C(CCC(N)=O)(C(=O)N1CC2CC1C2NC(C1CCS(=O)(=O)C1)=O)N(C)C Cc1ccc2nc(N(C3CCN(C(C4C(C)C4C)=O)C3)C)sc2n1 CCCCCC(O)C(=O)NC1CC(C(N2CCC(C(C)CC)CC2)=O)C1 c1(-c2cn(C(C(=O)NC(C=C)COC)C)nn2)cc(Cl)c(Cl)cc1Cl C1(C(N2CC(C(C)C)OCC2)=O)CC2CCCCC2N1S(=O)(=O)c1ccccn1 Cn1cc(C(=O)NCC2=CCN(CC(F)(F)C(F)F)CC2)c(O)nc1=O NS(=O)(=O)C1CCN(c2cc(NCc3nnc(Br)n3C3CC3)ncn2)C1 C(CCCCCNC(C1(c2cc[nH]n2)CC1)=O)NC(CC=C)=O CCCC(CC)(c1nnnn1Cc1ccccc1OC)NCCP(C)(C)=O N1(C(c2cc(C)n(CC)c2C)=O)CC(C2CN(C(=O)CC34CCC(CC3)C4)C2)C1 CN1CCCC(C(N2CC3C(CNC(=O)C=CCn4cncn4)C3C2)=O)C1 N1(C(CCn2ccc(C)n2)=O)CC(C)CN(C(c2csc(F)c2)=O)CC1C N1(C(c2n(CCCC)ncc2)=O)CC(NC(=O)Cc2cnnn2C)CCC1C N1(C(C2(CC=C)CC2)=O)CCC(CN(C(=O)CSCC(=C)C)C2CC2)CC1 N1(CC(=O)NC(C(C)C)CNC(C2CC2c2cncn2C)=O)CCCNC1=O Cc1ccc(NC(C2(NC(=O)C(C)CC#N)CC2)=O)c(C)n1 CC1CCC(C)(C(=O)NCCCNC(c2ccc(CO)cn2)=O)C1 N1(C(C(C(CC)C)OC)=O)CC2CC(C(=O)NCC(=O)NCC3CC3)CC2C1 c1(C(=O)Nc2n(C)nc(-c3ccccn3)c2)cccc([N+](=O)[O-])c1O O(NC(=O)C(C1CCC1)NC(=O)C(C1CCCCC1)O)C(C(C)C)CO CC1(NC(c2[nH]ccc2C2CC2)=O)CCCCC1C(=O)NCc1nc[nH]n1 N1(C(CNS(NC)(=O)=O)=O)CC(NC(=O)C=Cc2cccs2)C(C)C1 c1(C(N(CCC)CCNC(C2CCC2C)=O)=O)cc(C)c(Cl)cc1OC N1(C(CSc2cn(C)nc2)=O)CC2CCC1C1CN(C(=O)Cn3ccnn3)CC21 c1(CNCCCN(C)C2CC2)ccc2c(c1)C(=O)NCC2 C1(OC)CC2(C1)CC2NC(=O)C=CC.C1(NC(=O)CC2(OC)CCC2)CCCO1 Cc1cc(C(=O)N(C2CN(C(=O)CC(C)NC(N)=O)C2)C)c(N)cc1F C1(CC(=O)OCC)OCC2CN(C(c3occc3Br)=O)CCC12.C12CCN(C1)C2 c1(C(=O)NC2CCCC2CNC(C2CCCC3(CC3)C2)=O)cc2ncccn2n1 c1(C(C(=O)NC2CC(CNC(=O)CC3(CSC)CC3)C2)N(C)C)ccc(Cl)cc1 C(=O)(C(CC)C(C)(C)CC)NCCC(CNC(c1c(C)nc(CC)s1)=O)O N1(C(CC(=O)NCC)=O)CCC2(CCN(C(C3(C)CC(=O)N(C)C3)=O)C2)C1 c1(CCC)cc(C(=O)NCCn2cc(CN)nn2)no1.C(CN1CCCC1)CO N1(C(CSCC=C)=O)CCC(CNC(=O)CC(C=C)c2ccc(OC)cc2)CC1 CCCCC(C(=O)N1CCCC1CCNC(=O)C(C)N(C)C(C)=O)NC(N)=O Cc1ccc(NC=O)c(C(=O)NC2CC(CNC(c3snnc3CC3CC3)=O)C2)c1 c1(C(N2CC(CNC(C(CC=C)C)=O)CC2(C)C)=O)ccc2c(C)noc2c1 CCCC(C)(CC)C(=O)NC1CCN(Cc2nnn(C)c2C(=O)NCC)CC1 C1(C(=O)NCCN2CCC(NC(c3scnc3C)=O)CC2)(OC)CC2CCC1C2 C=C(C)CCC(C)NC(c1cnc(CNC(=O)C(C)(C)Cl)nc1)=O c1(C(N2CC(C)(C)C(NC(=O)C=C3CCC3)C2)=O)ccc2cccnn12 Cc1cccc(C2(C(=O)NCC3CC3NC(c3cscc3C)=O)CCCCC2)c1 C(=O)(C1=CC2(CN(C(=O)CNC(C3CC3C)=O)C2)OC1)N1C(CC)C(=O)NCC1 C1(C(=O)Nc2ccc(OC)c(F)c2)CN(C(=O)C2=CCOCC2)C2(CCC2)C1 c1(C(N(C(CNC(C2CCCO2)=O)C2CC2)C)=O)cccc(S(C)=O)c1 C1(NC(CCc2ncc(C)[nH]2)=O)CN(C(=O)C(C)NC=O)C2CCCC12 C1(NC(C2C3CC2N(C(c2cc(C(N)=O)[nH]n2)=O)C3)=O)CC(O)C12CCC2 S(=O)(=O)(c1ccc(Cl)s1)NCC(=O)N(CCCNC(C(C(C)OC)O)=O)C1CC1 c1(C(=O)NC(CN(C(CC2C(CC)C2)=O)C)C)ncc([N+](=O)[O-])n1C C(CNC(c1cccn1-c1cnn(C)c1)=O)(C(C)C)NC(COCCCCC)=O N#Cc1cc([N+](=O)[O-])ccc1NC(C1CC(O)CCN1C(=O)Cc1cscn1)=O C(c1ccc(F)c(Cl)c1)=CC(=O)NCC(CN(C)C(c1cn2c(n1)SCC2)=O)O C(c1cc(F)cc(F)c1)=CC(=O)NC1CC2(CN(C(C3CC(=O)NC3)=O)C2)C1 C#CCCCCCC(C(=O)NCCC)N1CCN(c2ncccc2Cl)CC1 C(=O)(C1CCCc2sccc21)N1CC2CC(CNC(C(C)(C)C)=O)C2C1 C(=O)(C(F)CCC(C)(C)C)NC(C(C(=O)N1CCC(OC)C1C1CC1)C(C)C)C CCC(C(=O)N1CCCC1CC(N)=O)N(C(=O)Cc1sccc1C)C C1(CCCC)CCC(C(=O)NCC2CC(O)CN2C(C2CCC(=O)N2)=O)CC1 c1(OC)ccc(F)c(C)c1.N1(C(CC2C(=O)N2)=O)CC(n2ccnn2)C(O)C1 C=CCCCC(C(=O)NCC=Cc1ccccc1)NC(c1cc(C#N)n(C)n1)=O N1(C(C2CN(C)C(=O)C2)=O)CC(C(=O)NC2CC2C(C)(C)C)CC1(C)C c1(CNC23CC(C(=O)NCC)(C2)C3)nccnc1C n1(CC)ncc2c(NC(CNC(C3CC34CCOC(C)C4)=O)C(C)C)ncnc12 C1(C(C)NC(=O)CC2(C)CC2)CN(C(c2ccc(C(F)(F)F)cc2)=O)CCO1 N1(C(=O)NCC(CC2CCCO2)OC)CCN2C(CNS2(=O)=O)C1 C(=O)(C(C)C(C)O)NCCN(CCOC)C(c1sc(Cl)cc1Br)=O c1(COC)c(C(=O)N(CCNC(=O)CNC=O)CC2CC2)sc2ccccc12 C12(CC=O)CC3CC(C1)CC(O)(C3)C2.C1(N)CC2(CC2)CN1c1ncc(O)cn1 C1(NC(c2c(CC)non2)=O)CC2CN(C(c3cccc(OC)c3F)=O)CC2C1 C1(C(=O)NCCCN(C(C(C)NC(C)=O)=O)C)CCON1C(=O)OC(C)(C)C c1(C(C)NC(CN2CCC(c3c(C(=O)OCC)c[nH]n3)C2)=O)c(F)cccc1F C1(C(=O)NCC(C2CC2)NC(c2cc(-c3cn(C)nc3)on2)=O)CCCCCC1 c1(C(N2C(CNC(CCc3c(C)ncs3)=O)CCCC2)=O)cc(C#N)ccc1Cl N1(C(c2ccc(CC)s2)=O)CC2CC3CC2C1C3NC(c1cc(F)c[nH]1)=O N1(Cc2ccn(CC)n2)CCCC(NC(c2cc(C)on2)=O)C1 C1(C(=O)Nc2cn(CCOC)nc2)CN(C(C2(C)COC(COC)C2)=O)CCO1 CC(CO)CCCNC(=O)CC1CCCN(C(C2C(C#N)C2(C)C)=O)C1 c1(OCC#N)ncccc1C(=O)NCC(=O)NCCNC(=O)C1CC1 c1(CC)oc(C(N2CCCC2CN(C)C(C2C3CCN2CC3)=O)=O)cc1C C(=O)(CC(=O)NC(Cn1cccn1)C(=O)NCCCc1n[nH]c(C)n1)NCC C1(C(=O)Nc2c(C)ccnc2C#N)CC1N=c1[nH]cnc2cnn(C)c12 C=CC(C)(CC)C(=O)NCC1(OC)CN(C(=O)C(C)N(C)C(=O)OC(C)(C)C)C1 N1(C(C2CC23CCOCC3)=O)CCC2(CC(NC(C34CCC(CC3)C4)=O)CO2)C1 c1(C(=O)NC2C(NC(c3cc(CC)nn3C)=O)CCOC2)cccc2nsnc12 c1(OC)cc(N)ccc1C(N1CCC(C)(NC(C2CC(N(C)C)C2)=O)C1)=O Cc1nc(N)c(CC(=O)NC(C)(C)CN(C)C(C2(F)CCOC2C)=O)c(O)n1 N1(C(C2(NC(C3ON=C(C)C3)=O)CCCCC2)=O)CC(CO)OC(C)C1 CCC(CC)C(C)C(=O)NCC1CN(C(c2ccc(C(C)(C)C)cc2)=O)CC1O C=CC(CCC)CC(=O)NCC(O)CCNC(c1cc(CO)n(C)n1)=O C#CCC(CC(=O)OC)NC(=O)C(C)N(CCC)C(C1CCCOCC1)=O C(C(C)(C)C(C)(C)O)C(N1CCCC1CC(=O)NC1ON=C(CC)C1)=O C(=O)(CC(C)(C)C1CCCCC1)NC1CCC(NC(CC2(C)CCCO2)=O)C1 c1(N(C)Cc2c(C)cc(Br)cc2)ncc(S(=O)(=O)NC2(C)CC2)cc1Cl C(=O)(C1=NOC(C(C)(C)C)C1)N1CCC(C)(NC(=O)CC2CCCC(=O)N2)C1 c1(C(=O)NCC(C)CNC(=O)CNC(N)=O)cccc2[nH]ccc12 Cc1oc(CNC(C2(CN(C)C)CCC2)=O)nc1C(=O)NC(c1nc[nH]n1)(C)C C1(CNC(CCNS(CC)(=O)=O)=O)COC(CNC(=O)Cc2n[nH]c(C)n2)C1 c1(C(N(CC(C)CNC(c2cc(N)cc(O)n2)=O)C)=O)cccc2c1CC(=O)N2 N1(C(CC(C=C)C)=O)CCC2CN(C(=O)CCS(C)(=O)=O)CCC12 c1(OC)cc(Cl)cc2[nH]c(C(N3CCC(NC(=O)C(C)OC)C(O)C3)=O)cc12 C(CCCC(=O)N(C)CCOCCNC(c1cccc(C2CCOC2)c1)=O)=CC CCCC(C)CC(=O)N1CC2CC1CN2c1ncc(C)c(O)n1 N1(C(C23C(CN(C(c4cc(I)c(F)cc4Cl)=O)C2)C3)=O)CCC2(CCCNC2)C1 c1(CNC(=O)NC(c2ccc(Cl)s2)C)cccc(S(C)(=O)=O)c1 C1(C(=O)NCC2C(C)CN(C(=O)COC3(C)CCCC3)C2)CCCCC12CC2 C1(CC)(NC(C2CCC(F)C2)=O)CCN(C(=O)CC2=CCCC2)CC1 N1(C(Cn2ncc(C(=O)OC)c2)=O)CCC2CC1CN(C(=O)C(O)C1CC1)C2 CC1CN(C(=O)CC2CC=CC2)CC1NC(C1CCC(CN(C)C)O1)=O C=C(C)C1OCCC1C(=O)NCC(=O)NCC(=O)NC1CCCN(C)C1=O n1(CC(=O)NC2(CCC(=O)NC3C(C)(C)CC3)CCC2)cc(C#N)cn1 C(=O)(C(C)(C)S(C)(=O)=O)NCC(CN(C(C1CC(CC)OCC1)=O)CC)(C)C N1(C(c2c(OC)cncc2)=O)CCC2CN(C(=O)C(C)CC(C)C)C2C1 N1(Cc2nc(C)sc2)CC(C(=O)NCCNC(c2ccccc2)=O)CC(F)(F)C1 CC(C(=O)NC1CCC1NC(c1csc(C(F)F)c1)=O)C(C)(C)C c1(C(=O)NC2CCC(CNC(c3ccsn3)=O)CC2)ccnc2ncccc12 N1(C(c2scc(C)c2Cl)=O)CCCCC2(CCN(CC=C(Cl)Cl)C2)C1 N1(C(Cc2c(C)n[nH]c2C)=O)CC(O)(C2(CNC(=O)C3=CCCCC3C)CC2)C1 c1(C(=O)NC(C2CCN(C(C=Cc3ccc(C)o3)=O)CC2)C)cc(O)cc(O)n1 C=CC(CCC)CC(=O)NCC1(NC(c2nocc2Cl)=O)CCOC1 N1(C(C2N(CC)C(=O)CC2)=O)CCC(C)N(C(c2cc3ncccc3o2)=O)CC1 N1(c2n(Cc3cncc(C)c3)nnn2)CC2C(CC1(C)C)C2(F)F C1(OC)CCN(C(=O)C(=O)NCC(CSC)OC)CC1 c1(OC)ccc(C(=O)NCC=C2CCN(C(C3CC(O)C(F)C3)=O)CC2)c(F)c1 O=S1(=O)CCN(C(=NCCF)NCCC2(CN3CCOCC3)CCCCC2)CC1 CC1(C)C(=O)CC1C(=O)NCC1CCCCN1C(C1C=CCC1)=O c1(C(N(C)CC2COCCN2C(=O)C(O)C2CC2)=O)c(F)cc(F)cc1Cl N1(C(C(c2c(C)scc2)N)=O)CCC(C)(N)C1.N(C)(CCSC)N(C)C C1(C(=O)NCCCC(C)NC(c2c(C)c(Br)no2)=O)CCC(N=[N+]=[N-])CC1 c1(CNC(C2C(OC)CC2)=O)ccnc(N2CCN(C(c3cc[nH]c3)=O)CC2)c1 c1(SCC#N)cccc(C(=O)NC2CC(NC(c3c[nH]nc3F)=O)C2)c1 c1(CC(=O)NC2C=CCN(C(c3cnc(CC4CC4)s3)=O)C2)cccnc1Cl C(=O)(C(F)(F)C(C)O)N1CCN(C(c2c(C)nsc2I)=O)CC1 C1(CC=C)(C(=O)NC(CN(C)C(C2CCCCN2CCC)=O)CC)CCOCC1 N1(C(C(C)P(C)(C)=O)=O)CCCN(C(c2ccc(N)c(N)n2)=O)CCC1 N1(C(c2cc3sc(Cl)cc3s2)=O)CCC2CN(C(c3ccon3)=O)CC2C1 C1(CNC(C2(COC)CC2(F)F)=O)CC(F)CN1C(c1cc(C(C)(C)C)no1)=O N1(C(CC2(CN)CCC2)=O)CCCCC1C1(C(F)(F)F)N=N1 N1(C(c2ccc(OC)nc2C)C(=O)NC2CC(CC)C2)CCC2(CCOC2)CC1 c1(C(N2CC(CC)C(C(=O)NOCC(O)CO)C2)=O)cnc(C)[nH]c1=N c1(C(N2CCCC(CNC(c3n[nH]c(C)c3Cl)=O)C2)=O)ccc2[nH]c(=N)sc2c1 N1(C(C(C)(C)CF)=O)CC2(CCC(NC(C3CC34CC4)=O)CC2)C1 n1(CC)nc(C)c(C(=O)NC2CCOC(SC)C2)c1C(F)(F)F c1(C(=O)NCC)cccc(C(N2CCCC(NC(=O)C(COC)N(C)C)C2)=O)c1 C(CC(=O)N(CCF)CC)(C(F)F)NC(C=C(CCC)C)=O N1(C(C(C)C)=O)CCC2(CCCC2CNC(C2CCCCN2C(N)=O)=O)CC1 C1(NC(C(C2CN(C(=O)OC(C)(C)C)C2)O)=O)CCCCC1 c1(C(=O)NC2CCCC(NC(C3CC34CCOCC4)=O)C2)cc2c([nH]1)CCOC2 c1(C(N2CC3C(CNC(C4CCN(C)C4=O)=O)C3C2)=O)ccc(S(N)(=O)=O)o1 c1(C(=O)NCC(CNC(c2cnn(CC)c2C)=O)CO)c(F)ccc(O)c1F C1(NC(c2cc(COC)[nH]n2)=O)CN(C(C2C=CC=CC=C2)=O)C2CCCC12 C(=O)(C(C)S(=O)(=O)C1CCOCC1)NC1CC(CNC(c2occ(C)c2C)=O)C1 C(=O)(CC(F)(F)F)NC1CN(C(C2CCN(C(C)=O)C2)=O)C1 c1(CC)c(C(=O)NC(C)CCN(C(=O)C=Cc2cn(C)nn2)C)nnn1CC C1(C(N(C2CCCN(C(c3c(C)coc3C)=O)CC2)C)=O)C2CCC3C(C2)CC13 CCC(CC)(CC)C(=O)N1CCC(NC(C2CC(=O)N(O)C2)=O)C1 c1(CCC(=O)NCCC(O)COC)ocnc1C(=O)NC(CC)CNC(=O)CO C#CCC(C)(C(=O)N1CCC(C)(O)C1)NC(=O)CCN(C)CCC C=CCC(CC)C(=O)NCC(C1C2CC1N(C(=O)C=C1CCCCC1(C)C)C2)=O n1(CC)cnc2c(N3Cc4[nH][nH]c(=N)c4C3)nc(=NCCN(C)C3CC3)[nH]c12 C1(O)(CNC(CCCOC(C)C)=O)CCN(C(C2CC2C(C)C)=O)CC1 C(c1ccc([N+](=O)[O-])s1)=CC(N1CCN(C(C=NOC)=O)C(CCOC)C1)=O c1(C(N)=O)ccoc1C(=O)NCC1(F)CC(NC(C2CCNC2=O)=O)C1 C1(NC(CCc2n(C)ccn2)=O)CC=C(C(=O)NCC2CCCC(C)(C)C2)C1 C1(C(=O)NCC(=O)Nc2ccc(F)cc2)COCCN(CC2CCS(=O)(=O)C2)C1 n1(CCC(N2CC(C)C(O)CC2)=O)cnc2ccccc12 C1(CCNC(C=CC(C)(C)NC(=O)Cn2cc(CO)nn2)=O)CCCCC1O C(=O)(C1=COCCO1)N1CCC(COC)(NC(c2ccc(C(C)=O)c(O)c2)=O)C1 CN=c1nc(N(C)CCc2ccccn2)[nH]c(=NCCC(=O)OC)[nH]1 C(=O)(C(C)(C)C(C)(F)F)N1CCN(C(C(CC)OC)=O)C(CCOC)C1 c1(CC)nc(C(C)NC(=O)C(=O)NCCC(C)(C)c2ccccc2)n[nH]1 CN1CCOC(C(=O)NCC2CC3CC3N2C(=O)COc2ccc(F)nc2)C1=O Cc1ccc(C(N2CC(NC(C3CCn4nnnc4C3)=O)C2)=O)c(Br)c1F Cc1cc(C(=O)N(C2CN(C(=O)CCCn3ccnc3C)CC2F)C)oc1C C12(CNC(=O)C=CCO)CCC1CCN2C(c1ccc(-c2cccs2)o1)=O C1(F)(CNC(c2c(C)nc(-c3nc[nH]n3)s2)=O)CCCN(C(=O)C(Cl)=CCl)C1 CCCCS(=O)(=O)CC(=O)NCC1C(C)CCCN1c1ncnc(C)c1F c1(CN2CCN(C)C(CC3CC3c3ccccc3)C2)n[nH]c2ccc(F)cc12 C(=O)(CCCCCN(C)C(C1(C)CC1)=O)N(C)Cc1nnc(CC)o1 Cc1ccc2sc(N3CC(CCCCNC(=O)C(O)CC(C)(C)C)C3)nc2c1 N1(C(c2cnccn2)=O)CC2(CCN(CC3CC(C(=O)O)CO3)CC2)C1 C1(NC(c2cnn(-c3ccccc3)n2)=O)CCCCN(C(C2CC2(F)F)=O)CC1 c1(C(=O)NC2CCN(C(C(COC)COC)=O)C(C)C2)cnc2c(c1)CCCC2 CC1CC(NC(c2cc3n(c2)CCC3)=O)CCN1C(=O)C=Cc1ccncn1 c1(C(N(C2CCN(C(=O)Cc3ccccc3CC)C2)CCC)=O)ccc(N)cn1 Cc1cnc(C(=O)NCC2CC2C(=O)NC(CO)C(C)C)c(C)c1 C1(C(N2C(C=C)CC2)=O)CC(C)CN(C(=O)C=Cc2ccc(C)o2)C1 CC1CCCN(C(c2ccc(CNC(C3CC(F)(F)C3)=O)o2)=O)C1CO CC1(CNC(=O)CCC(N)=O)CN(C(c2cn(C(F)F)cn2)=O)CCO1 C(=O)(CC(C(F)F)C(C)(C)C)N1CC(CNC(C2=C(C)OCC2)=O)C(O)C1 C1(NC(CC2ON=C(C)C2)=O)CN(C(c2cc(F)cc(Cl)c2N)=O)CC12CCC2 CCCCCCCCC(=O)N(CCNC(C1CCC(O)C1)=O)Cc1ccccc1 c1(C(N2C(CNC(C3(OCC)CCSCC3)=O)CCCC2)=O)ccc(=O)n(C)n1 c1(SCC(N2C(CC(=O)NC)C(=O)NCC2)=O)ccc(CO)cc1[N+](=O)[O-] N1(C(C)CC(N2CC3(C2)CN(C(=O)Cn2cccc2)C3)=O)CCc2ccccc21 N1(C(c2ccc(CC)[nH]2)=O)CCN(C(c2cccc(CS(C)=O)c2)=O)C(CC)C1 C(=O)(CCS(C)=O)N(C(CNC(=O)C(C)(O)c1ccccc1)C1CC1)C Cc1ccn2c(C(=O)NC3CCCN(C(C4(CCF)CCC4)=O)CC3)cnc2c1 c1(NC(=O)NC)ccc(C(=O)NCC2CCC2NC(C2CNC(=O)N2)=O)c(Cl)c1 c1(C(=O)NCC(C)NC(c2c(C)cnn2C(C)C)=O)cc(F)c(F)c(Cl)c1F c1(C(N2CCC(CC)C2CNC(=O)CN2CCSCC2)=O)n[nH]c2c1CCC2 C(=O)(C1=CCCCC1C)NC1C(NC(c2snc(C)c2N)=O)CCC1 Cc1c(C(N2CCCC(C(C)NC(c3cn4c(n3)SCC4)=O)C2)=O)cccc1N c1(C(=O)NC(C)(C)CCNC(C2(c3cc[nH]n3)CC2)=O)cc(Cl)cc(Cl)c1F N1(C(CC=C)=O)CCC(C2CCN(C(=O)CC(F)(F)Br)CC2)C1 Cc1ccncc1C=CC(=O)NC1CN(C(=O)CO)CCC1c1ccccc1 c1(OC)cc(C)c(NCCCCSC)c(C)c1 c1(C(=O)NCCCCNC(C2C(C)(Br)C2)=O)ccc2c(c1)C(=O)OC2 c1(C(N(CC(C)NC(Cc2ccc(C(C)=O)nc2)=O)C)=O)nccc(Cl)c1F CC1(C#CC(=O)NC2CCN(C(c3cc4n(n3)CCO4)=O)C23CC3)CCCO1 Cc1snnc1C(=O)NCC1C=CC(NC(=O)CNC(=O)C(F)(F)F)C1 C(CC(C)C)(C(=O)NC1CC2(C1)CN(c1ccnc(-c3ccccc3)n1)C2)OC c1(C(=O)NCC2CCCC(CNC(c3n(C)ncc3Cl)=O)C2)cccc(F)c1N c1(CCC(=O)NC2CN(C(c3ccc(Br)o3)=O)C2)cncc(O)c1 Cc1ccc(C(=O)NC(C(=O)N2CCCCC2C)C(C)O)n1C C1(CNC(CC=C)=O)CC(C)N(C(=O)C=Cc2cc(C)no2)C1 C1(N(CCOC)C=O)CCN(C=O)CC1.C1(OC)CN(C(=O)CCOC2CC2)C1 N1(C(C(CC)(C)CC)=O)CC2CC(C1)N(C(c1ccnn1COC)=O)C2 c1(CC(N2CC(CCNC(C3(CCOCC)CCC3)=O)C2)=O)c(O)ncnc1O c1(C(N2C(CNC(C3=NOC(C)C3)=O)COCC2)=O)cnc2cc(O)ccc2c1 N1(C(C=C(NC(C)=O)C)=O)CCCC12CCN(C(c1cc(O)ccc1C)=O)C2 C1(C(N(CCN(C)C)Cc2nccs2)=O)(C(=O)N(C)C)CC2(CCC2)C1 Cn1ncc(S(C)(=N)=O)c1C(C1CCN2CCOCC12)N N1(C(c2c(CC)ocn2)=O)CCC(C(C)NC(=O)C(=O)NCCC(N)=O)CC1 Cc1cc(C(=O)NCC(O)CNC(=O)CC2CCSCC2)nn1C(C)C c1(OC)csc(C(N2CCC(CNC(c3ccnc(S)c3)=O)C23CC3)=O)c1OC c1(C(=O)NCC(CC)NC(=O)CCc2nncs2)ccc(F)c(Cl)c1 N1(C(CC(=C)C)=O)CC(N(C(=O)CCc2ccc(CO)cc2)C)C2(CC2)C1 C1(CNC(c2n(CC)ncn2)=O)CC2(CC(NC(=O)CCN(C)CCO)C2)C1 c1(C(N2CCC(NC(=O)Cc3cc[nH]n3)C(F)C2)=O)ccc2c(c1)S(=O)(=O)NC2 C(=O)(C1CCCc2cncn21)NC(C)CCN(C)C(c1cc(Cl)ccn1)=O c1(CC)cccnc1C(=O)NCC1(C)CCN(C(c2cc(C)nn2C(F)F)=O)C1 n1(CCNC(c2ccoc2C(F)(F)F)=O)cc(CNC(c2nncs2)=O)nn1 N1(C(c2ccc(CCC)cc2)=O)CCN(C(=O)C(C)NC(C)=O)CCC1C c1(C(=O)O)cc(CO)cc(S(=O)(=O)NCCc2ccc(Cl)cc2F)c1.CCO C1(C(N2CCC(c3cnccn3)CC2)C(=O)NC(CC)(C)C)CCC(C)(C)CC1 N1(C(CN(C(=O)CCC2CC2)CC=C)=O)CC2CC(NC(=O)CO)C(C2)C1 C1(NC(C)=O)CCCN(C(C2CN(C(C3CN(C)CCO3)=O)CC2C)=O)C1 c1(NC)ccc(C(N2CCC(NC(C3CCC3(F)F)=O)C(O)C2)=O)c(Cl)c1 Cc1cc(C(F)(F)C(=O)NCCN(C(=O)CCCn2ccnc2)C)cnc1Cl c1(C(=O)NC(C)CCCNC(=O)C(=O)N(C)C)cc2ccccc2cn1 C(=O)(CCCCC(N)=O)NC(C(=O)N(C1CCC(F)(F)C1)C)C1CC1 C1(C(N2CCC(CN(C)C(c3ccncc3)=O)CC2)=O)Cc2cccnc2C1 c1(C(=O)NCC2OCCCN(C(C=C(C)C)=O)C2)cnn2ccccc12 c1(C(N(C2CC(NC(=O)C(F)CC3CC3)C2)C)=O)cc(Br)ccc1Cl C=CC(C)(O)CC(=O)NC1CCN(C(=O)CCC(=O)NCC)CC1 N1(C(C2(C(C)NC(=O)C(F)(F)F)CC2)=O)CCCCC1c1nc(C(N)=O)no1 c1(C(=O)NC2C(C)(C)C(CNC(C3(C)CC=CC3)=O)C2)cc2ccc(Cl)nc2s1 c1(C(N(CC(C)NC(=O)CCc2cnn(C)n2)CC)=O)ccc(F)cn1 C1(NC(=O)C(c2ccc(F)cc2)O)C=CCN(C(c2ccc(Br)s2)=O)C1 N1(C(CNC(=O)OCC)=O)CCCC(C2CCCCN2C(c2nocc2C)=O)C1 c1(CC)ccc(OC)cc1C(=O)NC1CCC12CN(C(c1cccc(N)n1)=O)C2 c1(C(N(C)CCN(C)C(C2CC(O)CN2C)=O)=O)ccccc1[N+](=O)[O-] N1(C(C(C)(C)OCC)=O)CCCC(Cn2cc(C(C)(C)OCC(=O)NC)nn2)C1 CC(CCNC(=O)C#CC(C)(C)CNC(c1nn(C)cc1Cl)=O)CC(C)(C)C c1(C(CNC(C)=O)NC(=O)C(Cl)=CCl)ccc(C)cc1 C(CC(C)CCNC(=O)CN1CCC(C)(C)C1)NC(C(C)C1(O)CCC1)=O N1(C(CC2(C=C)CC2)=O)CCCCC2C1CCCN2C(C1CCC(F)(F)C1)=O C1(NC(CN2CC(CC)C2)=O)CCN(C(=O)CCN2CCCCC2=O)CC(O)C1 c1(NC2CC3(CN(C(=O)OC(C)(C)C)C3)C2)cccc2oc(O)nc12 C1(C(N2C(C3CCN(C(CC#N)=O)CC3)CCCC2)=O)CC2CC1C1CC21 c1(C(N(CC(O)CNC(c2cc3c(s2)CCC3)=O)C)=O)nc(O)nc(O)c1F CC1CN(C(c2nccnc2Cl)=O)CCC1CNC(c1ncc(Cl)cc1Cl)=O c1(C(=O)NC(C2(O)CN(C(CN(CCOC)C)=O)C2)C)cnc(O)cc1OC Cc1cc(F)c(Oc2ccc(SCCC(=O)Nc3ccc(Br)cc3)cc2)cc1Cl c1(CC)ccc(Br)cc1C(N1CCC(NC(=O)C2=NOCC2)C(O)C1)=O c1(C(N2C3CC(NC(CCC(CC)CC)=O)(C3)C2)=O)cc2ccc(OC)cc2s1 Cc1nc(C(C)C)cc(=NCC2CCCCC2NC(=O)CSC(F)(F)F)[nH]1 Cc1cc(C)n(C(C)C(=O)NCC2CCCN2C(c2cnn(C(F)(F)F)c2)=O)n1 c1(OC)cccc(C(N2CC(CNC(=O)C(C3CC3)OC)C2)=O)c1F c1(C(=O)NC2CCC(C(=O)Nc3ccc(CC)cc3)C2)cccc(OC)c1O N1(C(C(C)C)=O)CC(CNC(C2CC2F)=O)C2(CCOCC2)C1 C1(CC(N2CC(NC(c3c(C)nccn3)=O)C(F)C2)=O)CC(C)(C)CCO1 C1(NC(c2n(CC=C)nnn2)(C)CSC)CC2(C1)CC(C)C2 C1(CNC(C2(COC)CCOC2)=O)CN(C(c2cn(C3CC3)nc2C)=O)CC1O C(=O)(C(C)S(C)(=O)=O)NCC(CC)OC.c12ccc(cn1)c(=O)n2CC c1(CNC(=O)NC(c2nc(C3CCCCC3)cs2)C2CC2)ccc2sncc2c1 C=CCC(CC(F)F)C(=O)N1CC2CN(C(=O)C(CC)n3nccc3C)CC2C1 C1(NC(c2c(C)noc2)=O)CC(NC(C2(O)CCCCCC2)=O)C12CCOCC2 c1(-c2nc(OC(C(N3CCN(C(=O)OC)CC3)=O)C)sc2)ccc(C)c(F)c1 S(=O)(=O)(c1cccc(C(=O)OCC23CC(C)(CO2)C3)c1)NC(CC)C C#Cc1ccc(F)cc1C(=O)NC1CN(C(c2cc(CC)ccc2F)=O)CC1O C1(NC(c2cc(O)nc(O)n2)=O)C2CCC(C2)C1C(=O)NC1CCCCC12CC2 C1(C(=O)NC2CCN(C(C(c3ccc(OC)nc3)(F)F)=O)C2)CCCC12CCC2 C=CCCN=C(NCc1ccc(C)cc1OC(C)C)NCC(C)(O)C(F)(F)F N1(C(C(C=C=C)C)=O)CC2(CC2)CC1CNC(=O)COCc1ccccc1Cl c1(C(=O)NCCCNC(c2cc(C#C)c(Cl)cc2)=O)nc(CC)n2ccccc12 C1(OC(c2cnn(-c3ccncc3)c2C(F)F)=O)CCC(F)(F)CC1 CC1CCN(C(=O)C(=O)Nc2ccccc2)C1c1cn(C2C=CCCC2)nn1 N1(C(=O)CC2CC2C2CC2)CCC2(C1)CN(C(C1(c3cc[nH]n3)CCC1)=O)C2 CN1N=C(C(=O)NCC2(C(=O)NC3CCSC3)CC23CCC3)CCC1=O C=CCCC(C)(C)C(=O)NC1CC2CCC1N(C(=O)C(F)(F)C(F)F)C2 c1(-c2cncc(C#N)c2)ccc2c(c1)CCN(S(=O)(=O)c1cn[nH]c1)C2 c1(OC(C)(C)C)ccccc1CC(=O)NCC1CC(NC(C2(C)CC2F)=O)C1 N1(C(c2c(C)nsc2)C(=O)NC2CCCC2)CCN(C)CC1C(C)C c1(CC)ncccc1C(=O)NC1CCN(C(c2cc[nH]c2CC)=O)C1C1CC1 c1(C(=O)NC2CC(NC(c3ccc(NCCO)cc3)=O)C2)cc(F)cc(F)c1 C1(CNC(C(C)Cc2ccnn2C)=O)(CNC(C2(C)CCCC2)=O)CC12CCC2 Cc1cn2nnc(C(=O)NCCCN(C(C3C4CC(=O)CC34)=O)C3CC3)c2c(O)n1 c1(C(c2n(CCCSCC)nnn2)NCC2CCCOC2)cc(S(C)(=O)=O)co1 C(=O)(CC(CC(C)C)NC(c1ccnn1C1CC1)=O)N1CCOCC(=C)C1 C1(NC(C(C)OCCC)=O)CC2CCC1N(C(c1cc(C(=O)OC)nnc1C)=O)C2 C(=O)(C(C(C)C)Nc1ccccc1)NCC(C)(C1CC1)NC(C(F)=CC=CC)=O C(=O)(C(CNC(c1ccsc1Cl)=O)N(C)C)N(C1CCN(C)C1)CCC C12(NC(=O)CCN3CCCCC3=O)CCC1CN(C(C1CCCCC1)=O)C2 C(=O)(C(F)CC(CC)CC)NC(CCCC)CNC(=O)CCc1ccccc1F C(=O)(C(C)(C)N=[N+]=[N-])NCCC1C(C)CN(C(c2cc(O)ncn2)=O)C1 C1(C(=O)NCC2CCC(NC(c3cn(C)nc3O)=O)CC2)CN=C2N=CNN2C1 c1(C(=O)NC(C)CNC(=O)CCc2ccccc2)cc2c(nc1O)CCSC2 CC1CC(C)CN(CCNC(=O)C(O)CCn2cc(C3CCC3)nn2)C1.C(C)(C)O c1(-c2cn(C(C(=O)NCC(C)C)C)nn2)ccccc1OCC(=O)O C1(CNC(c2c(CC)cco2)=O)CC(NC(C2(O)CCOCC2)=O)CC1O N1(C(CCCC(=C)C)=O)CC2CC(C)N(C(c3ccc(N(C)C)cc3)=O)C2C1 N1(C(c2ccc(CNC(C3N(C)CC3)=O)o2)=O)CC(CO)CC12CCC2 C1(C(N2CCC(C(C)C(=O)NCC=C(Cl)Cl)CC2)=O)CN(C)CCN1C CC1CCc2nc(Cl)nc(N3CC(CN(C)C(C4(C)CC4)=O)C3)c2C1 c1(CC(C)C)c[nH]c(C(=O)NCC(C)CNC(=O)CN2CCC2C)c1 c1(OC)ccc(C(=O)NCC(C)NC(=O)Cc2cc(C)ccc2F)n2nccc12 c1(C(N(C(C)CCNC(c2cc(C(F)(F)F)cs2)=O)C)=O)cccnc1F n1(CC(C)C)ccc(C(=O)N(C2CCCC2)CCNC(=O)C=Cc2ccsc2)n1 CC1(C)CCCCCC1NC(c1csc(CNC(C2C=CCS2)=O)c1)=O c1(C(=O)NC2CCN(C(c3cnc(CCC)s3)=O)C2)ccc2c(c1)CCN(C)C2 C1(c2nnnn2CCCC2CC2)(NCc2ccn(C(C)(C)C)c2)CCC2CC12 N1(c2nnn(C)n2)C2CCCC1CN(C(=O)Cc1c[nH]c3cc(Cl)ccc13)C2 Cc1cccnc1CN(C)CC1CCN(C(=O)CNC(=O)Nc2cccs2)C1 CC(=O)CCCC(=O)NC1CC2CC1CC2C(N1CCC(C2CC2)C1)=O C(=O)(CCCN(C)N=O)N(CCOCCNC(C(CC=C)C)=O)C C(=O)(C1=C(CC)OCCS1)N1C(CCCC)CN(C(=O)C(F)C2CC2)CC1 C1(C(N(C(CC)C2CC2)C)=O)CCN(C(=O)NC2CCCO2)CC1 C(C(C)(C)CCCO)NC(C(c1cn(C)nn1)N(C(C1C(C=C)OCC1)=O)CC)=O Cn1nccc1CCNC(c1cc(CNC(=O)C=CCN2CCCC2)no1)=O N1(C(CC(COC)COC)=O)CC2(C1)OC1(C)CC2(NC(C2CCCOC2)=O)C1 CC(CS(C)=O)C(=O)NCCCC1CCN(C(C2CC=CC2)=O)CC1 c1(C(N2CCC(CNC(C3(C#N)CC4CC4C3)=O)CC2)=O)nnn2c1COCC2 N1(C(c2ccc(C)nc2O)=O)CCC2CCCN(C(c3cc(Cl)n(C)n3)=O)C2C1 N1(C(c2cc(C)cc(O)c2)=O)CCCC1C1CCCN1C(=O)CN(C)S(N)(=O)=O c1(C(=O)NCC2CC(NC(c3cc(C)ncn3)=O)C2)ccc(N)c2ncccc12 N1(c2c(C#N)cncn2)CCOC2CN(C(c3cc(Br)ccn3)=O)CC12 C(CC(C)(C)CC(=O)N(C(C)CN(C)C(C12CCC(CC1)C2)=O)C)OC c1(C(N2CCCC2c2cn(Cc3cnoc3)nn2)=O)ccc(-n2cnnn2)cc1 c1(C(=O)NC(C(C)NC(c2c(OCC)cccn2)=O)CO)nsc2ccccc12 C(=O)(CCCC(C)=O)N1CC2C(CNC(c3c(CC)nc[nH]3)=O)(C2)C1 c1(NCCOCCNC(CC2CCC(C)O2)=O)ncnc2c1ncn2C1CC1 N1(CC)C(=O)NC(c2ccc(N)c(Br)n2)C2=C1C(C)CN(C)C2=O N1(C(Cc2c(C)noc2)=O)CCC2CCN(C(c3ccc4c(c3)CCN4)=O)CC12 C=CCC(CC(C)C)C(=O)N1CCN(C(c2cccc(N)c2O)=O)C(COC)C1 CCC(C(=O)NC(CNC(C1SCCS1)=O)C1CC1)SC C1(NC(C=C(C)C)=O)COCCN(C(c2cccc(-c3ccncc3)c2)=O)C1 c1(C(=O)NCC2COCCN(C(C(=O)N(C)C)=O)C2)cc2n(n1)CCNS2(=O)=O CC(C)C(CC(=O)N1CCCCCC1)NC(=O)C(CO)N(C)C O=C1NC(=O)CN1.N1(C(C2CC2)C2CC2)CCC(n2ncc(=O)[nH]2)CC1 CC1C2C(CCN2C(=O)COCC(F)(F)F)CN1C(=O)C1CCc2c[nH]nc21 C1(CNC(=O)NCc2c(C(=O)OC)scc2)CC2CCCCC2O1 C1(CCC=C)(C(N2CCC2(C)CC)=O)CN(C(=O)Cc2cc(C)on2)C1 N1(C(C2C(C(=O)OCC)CC2)=O)CCC(O)C(NC(c2ccc(Cl)cn2)=O)C1 N1(C(c2ccsn2)=O)CCC2(CC1)CC(n1cc(CCO)nn1)CCO2 C(=O)(C(CC(C)C)NC(C1CC(=O)OC1(C)C)=O)NCC(CC(=O)OC)O c1(OC)ccc(F)c(CN2C(C(=O)N(C)CCC3OCCO3)CC3CC23)c1F N1(C(C2CN(C)C(=O)C2)=O)CC2CCCC2(CNC(=O)COc2ccsn2)C1 CN1CC=C(CC(=O)N2CCC3CCC(C2)N3c2nc(CC3CC3)ns2)CC1 N1(C(Cc2scc(C)c2)=O)CCCC(O)(CN(C(=O)Cc2ccns2)C)C1 C(=O)(C1=CCC(NC(C2CCCN2C)=O)C1)NC(C(=O)OC)C CC1CN(C(=O)CC2CN(C)C2)CC1CNC(c1csc(C(F)(F)F)n1)=O CON(CCC(=O)NC(C(=O)NC)C1CCOC1)C(=O)C(C)N1CCCC1=O C1(C(N2CC(OC)C(NC(=O)CC(Cl)Cl)CC2)=O)CC12CCC(=O)CC2 c1(OCC)ccc(C(N2CCCC(CNC(=O)C(C)COC)C2)=O)cc1C c1(CNC(C2C(CC)NCC2)=O)cc(C)ccc1C C1(O)(CCC)CCN(C(C2CN(C)CCN2C(C2CCSC2)=O)=O)CC1 c1(C(=O)NCC2(O)CCN(C(CCC(=O)OCC)=O)C2)ccc(C)c(C)c1Cl c1(CC(=O)NCCOC2CN(C(C3CCOC3=O)=O)C2)ncn2ccccc12 C(=O)(C(C)CC(C)C)NCC1CN(C(c2c(CC)n(C)nc2)=O)CC1C c1(N(C)C)ccc(C(=O)NCC2CC2NC(c2cnc(C(F)(F)F)s2)=O)cn1 CC(CCN=c1[nH]c(N2CCc3ccccc3CC2)nc2cc[nH]c12)c1cn[nH]c1 C1(CC)C(C(=O)NC2CC3(CC(OC)C3)C2)CCCN1C(=O)C1=COCC1 N1(C(c2cc(CNC(CCCCN(C)C)=O)sc2)=O)CCOC2CCC12 C(=O)(N=c1[nH][nH]c2ccc(C(=O)O)cc12)N1C(C(C)C)C2(C1)CCOCC2 C1(NC(C2C(COC)C2)=O)CCC(CNC(=O)COCO)CC1.c12cn(nn1)C2 c1(NC(C2C3CN(C(c4c(CC)occ4C)=O)CC32)=O)cc(O)ccc1C N1(C(CSC)=O)CC(NC(c2ccc(Br)c(F)c2N)=O)CC12CCOC2 C1(C(=O)NC2CCC(NC(c3cnn[nH]3)=O)C2)(CN(C)C)CCCC1 Cc1cc(C#N)ccc1C(=O)NC1CN(C(=O)CCc2nc[nH]n2)CC1C N1(C(C(N2CCSCC2)C)=O)CC=CC(NC(=O)C(c2ccnn2C)O)C1 N1(C(C(COC)N(C)C)=O)CCCC(CC(=O)Nc2cnn(C)c2C)C1 N1(C(C(C)n2ccnn2)=O)CC2CCCC(C1)N2C(=O)CC1CCN(C)CC1 N1(C(c2c(C)scn2)=O)CCC(O)(C(C)NC(=O)CC(C)C(F)F)CC1 c1(C(N2CCC(F)(CNC(CC(C=C)(C)C)=O)C2)=O)ccc(N)c([N+](=O)[O-])c1 C1(C)(CNC(C2(SCC)CC2)=O)CN(C(=O)CC2CCCOC2)CCO1 C12(NC(C(C)(C)c3ccns3)=O)CC1CN(C(=O)CN1CCCCC1=O)C2 C12(NC(c3cc(Cl)ccc3F)=O)CCN(C(c3conc3C3CC3)=O)CC1C2 N1(c2ncnc(NC(CCC)c3ccco3)c2C)CCCN(C)C(=O)C1 c1(C(CNC(C=CC(C)C)=O)NC(c2cccn2C)=O)ccc(F)cc1 N1(C(c2cc(C)oc2C)=O)CCC(NC(=O)Cc2cc(F)ccc2O)CC1C c1(C(C(=O)NC(C)(CNC(=O)C=CCF)C2CCC2)=O)ccc(F)cc1 Cc1[nH]c2ccc(C(=O)OCc3ccc(C(F)F)c(F)c3)cc2c1C C(CC1=CCN(C(=O)CC2CCCCC23CC3)CC1)NC(C1(C)CCOCC1)=O CC(C)(C)C(C(=O)Nc1cccc(Cl)c1)NC(c1cncnc1)=O C1(O)(C(N(CCCNC(c2ccc(CCF)cc2)=O)C)=O)CC2CCC1C2 C1(C2CCN(C(c3nn[nH]c3Cl)=O)C2)(NC(=O)CC2(CO)CC2)CC1 c1(OC)ccc(Cl)c(CC(N2CC3C(NC(C4CC4C)=O)C3C2)=O)c1F c1(SCC)nc(C)c(CC(=O)NC2C=CC(CNC(=O)CCC3CCCC3)C2)s1 C(=O)(CC(C)(C)C)N(C(C)CNC(c1cnn(C2CCC2)c1)=O)C C(=O)(C(O)CC(N)=O)N1CCC(COC2CN(C(C3(OC)CCOCC3)=O)C2)CC1 N1(C(C(C2CC(NC(c3ccc(OC)nc3)=O)C2)F)=O)CC2(CCCCCC2)C1 c1(CC(=O)NC2C(CNC(CN(C3CC3)CC)=O)CC2)c(Cl)cccc1Cl C=CCCCC(C(=O)NC)N(C)CCc1cnc(OC)nc1 c1(N(C)C)ccnc(C(=O)OCC(=O)CC2(C)CC2)c1 N1(C(c2c(C)noc2)=O)CC2(C1)CN(C(C1CC1c1cccs1)=O)CC(C)(C)O2 CCC(CC)C(F)C(=O)N1CCN(C(c2ccc[nH]2)=O)C(c2ncc[nH]2)C1 c1(OC)n[nH]cc1C(=O)NC1CC1NC(=O)Cc1c[nH]nc1O C(C(C(=O)NCC(O)C(=O)N(C1CCCC1)CCO)OC)OC c1(OC)ccc([N+](=O)[O-])cc1CNC(c1ccc(I)cc1)(C)C c1(C(C)(C)C)n[nH]c(=Nc2cccc(F)c2C(=O)NCC(C)(C)O)o1 c1(COC2CCCN(C(C)C)C2)cccc(C(F)(F)F)c1O.C12CCN(C1)C2=O c1(CC)ncc(C(=O)NC(C)CNC(=O)CCCCc2ccc(F)cc2)c(C)n1 c1(COC)nc(C)c(C(=O)OC)c(O)n1.C12CC1N(C)C2.C(=O)(CC(C)C)O N1(C(=O)NCc2c(C)nc(C)s2)CC(NC(=O)OC(C)(C)C)C(C)(C)C1 Cc1cc(C(F)(F)F)c2cc(C(N3CCSCC3(C)C)=O)oc2n1 C1(NC(C(CC)N(CC)CC)=O)COC2(C1)CN(C(=O)CC1OCCO1)C2 c1(NC(C(c2nc(C(C)(C)C)cs2)N(C2CCOC2)CC)=O)ccccc1 Cc1cn(C)nc1CNC(=O)N(C1CC(c2ccccc2)C1)C c1(C(N2CC(NCc3cccc(C(=O)OC)c3)C2)=O)ccc2c(c1)CCCC2 c1(C(N2CCC3(CC(OC)C3)C2)=O)cc2cc(Cl)cnc2o1 Cc1ccc(-c2ocnc2C(N2CCOC(CN(C(=O)C3=CCC3)C)C2)=O)cc1 N1(C(C2CCC(C)O2)=O)CC2(C1)CN(C(=O)Cc1cn(CCO)nn1)CCO2 C(=O)(CCC(C)C#N)N1CC2C(CNC(CCc3cncc(OC)n3)=O)(C2)C1 c1(C(=O)OC)ccc(NC(C2CCN(Cc3scnc3Cl)C2)=O)c(F)c1F CS(=O)CCC(=O)NC(C)(C)CNC(c1cc(C2CCOCC2)[nH]n1)=O C1(NC(C2CC3(CCC3)CO2)=O)CC2(CCCN(C(C3CCCCC3O)=O)C2)C1 c1(C(=O)NCC=CCNC(CC2C(C)(C)C(O)C2)=O)cc2ccc(O)cc2[nH]1 C1(Nc2cc(C)nc(N3CCC(c4coc(=N)[nH]4)CC3)n2)CCCCC(F)(F)C1 c1(C(N(C(C)CNC(c2cnccc2OC)=O)CC)=O)[nH]nc([N+](=O)[O-])c1Cl Cc1cc(F)c(C(=O)NC2CC3CC2N(C(=O)CCN2CCCCC2)C3)c(F)c1 c1(OC)cncnc1N(C)CC1CCN(C(=O)Cn2ccc(C)n2)CC1 C1(C(=O)NC(=O)COC(C)(C)C)CCCC(CN(C(CN(CCOC)C)=O)C)C1 C1(NC(c2c(N)nccn2)=O)CCC12CN(C(=O)C(c1cc(F)cc(Cl)c1)=O)C2 c1(C(=O)NCC2(OCC)CN(C(=O)C=Cc3ccccn3)C2)cc(C#N)c[nH]1 C1(C(N(CCCNC(CS(CC)=O)=O)C)=O)CCc2nc(C3CC3)ncc2C1 C(=O)(CC(C)C(C)(C)C)N(C(C(N1C(CC#C)CCCC1)=O)C)CC C(N=c1[nH]nc(CO)s1)C1C2CN(C(c3c(OCC)cccc3)=O)CC21 c1(C(=O)NC2CC3CN(C(C(=O)NC(C)C)=O)CC32)cccc2ncnn12 C1(NC(c2c(C)nccc2)=O)CC2CCC1N2C(C1(C(C)(C)C)CCCCC1)=O c1(OC)cc(C(=O)NC2CN(C(=O)Cc3cccc(F)c3)CC2C#N)cnc1Cl C1(C(=O)OCC)CN(C(C23CCC2CCN3)=O)c2cccc(Br)c2O1 N1(C(C2C(C)(C)C2)=O)CCC2(C1)CN(C(C13CCC(C1)C(C)(C)O3)=O)C2 C(=O)(C(F)CCC(C)(C)C)NCC(C(=O)NC(C)C1CC1)CC1CC1 C1(CCNC(C(C2N(C(Cn3ccc(C)c3)=O)CCC2)(C)C)=O)CCCCCC1 C(CS(=O)(=O)N(CCCOc1cccc(Cl)c1)C)(C1CCOCC1)OC C(N=c1[nH]c(=NCc2nncs2)[nH]c2cccnc12)C1CCn2c(C)nnc2C1 C12(CCC(=O)N(C)CC)CCC(CC1)C2.CCC(O)C(=O)NCC1(CO)CC1 N(C1c2ccccc2CC1NC(C1(n2cnnn2)CC1)=O)C(C(C)n1cncn1)=O c1(OC)ccc(Br)c(C(N2CCOC(CNC(=O)CC(O)C(C)C)C2)=O)c1 O=C(C(CO)C(F)(F)F)NC1(C(=O)NCC2CC23CCOCC3)CC1 N1(C(c2c[nH]c(=N)o2)=O)CCN(C(C2CCCS2)=O)C(c2ccc(F)cc2)C1 C(=O)(C(C)(C)CNC(=O)Cn1cc(Cl)cn1)NC1C(OC)COC1 C(=O)(C(C)CC(C)CC)N1C2CC(NC(Cc3c(C#C)cccc3)=O)C2CC1 CC1CC(C)(C(=O)NC2(CO)CC2)CC(C)O1.c12ccccc1CNC(=O)CN2 C1(CNC(C(C(C)C)NC(=O)OC(C)C)=O)CCN(C(c2ccoc2)=O)CC1C n1(C(C)C)nnc2c(NCCC3CCN(C(=O)C(C)CN(C)C)C3)ncnc12 C1(CC)CN(C(C2CC23CCOCC3)=O)CCC1NC(c1ccncc1F)=O n1(CC(=O)N(CC#C)C(C)C)cc(CNC(C2CCCC2C)=O)nn1 C1(c2cccs2)(C(=O)NCCC(C)NC(C2C(F)(C(=O)OCC)C2)=O)CCCC1 CC1CCC(O)C(NC(=O)CC2CC(NC(=O)CC3CC(C4CC4)C3)C2(C)C)C1 C1(C(=O)NC2CC(CNC(C3C(CC)N(C)CC3)=O)C2)CC2CCC(C1)C2 N1(C(CC(CC)C2CC2)=O)CC2CCC(C1)N2NC(=O)C(C(C)C)NC(N)=O C1(C2CC2)(C(=O)NCCCOCCCNC(C=CC(CC)C)=O)CCOCC1 c1(C(N2CCC(OC)(CNC(C)=O)C2)=O)cc2c(Br)ccc(F)c2[nH]1 N1(C(c2cccc(NC(C)=O)c2)=O)CC(NC(c2occc2F)=O)CC(F)C1 CC(C)CS(=O)(=O)CC(=O)N1CCC(CNC(c2cc3c(ncn3C)[nH]2)=O)C1C c1(CC)cc(C)nc(NC2(CC)CCN(C(C3CCOC(C(C)C)C3)=O)CC2)n1 C(CC1CC1)(C(=O)NC(Cn1cncn1)C(=O)NC1CC(OC(C)C)C1)OC c1(C(=O)NCCC(C)N(C(c2c(CC)ccs2)=O)C)ccc(C(C)C)c(C)c1 c1(C(=O)NCCN(C(CCC(=O)NC)=O)C)nc(C(C)C)ncc1Cl CCS(=O)c1ccccc1C(N1CCC(C)(NC(=O)C2=CS(=O)(=O)CCC2)C1)=O C(C(C(=O)N1CC(n2ccnc2)C1)n1cc(C2(C)CCCO2)nn1)OCC C1(CN(C)NC(C2CC3(CCCC3)C2)=O)CCOCC12CCC2 C(=O)(C1=C(C(F)Cl)N(CC2CC2)C(=O)NC1c1cc(I)c(Cl)cc1F)OCC C(C1CCOCC1)=CC(=O)NCC(CC=C)NC(c1cc(C)nn1CC)=O N1(C(CC(CC)C)=O)CCC(C)(C)C(NC(c2cc(C(C)C)[nH]n2)=O)C1 N1(C(c2c(NC(C(C)NC(CC)(C)C)=O)ccs2)=O)CCCCCCC1 c1(OCC)ccc(C(N2CCCCC2CN(C(C)C(N)=O)C)=O)cc1OC C1(C(=O)NC(CCC)CNC(=O)COC2CC=CC2)CCCCC1CC CCCC(CCCNC(=O)C(C1CC1)OC)NC(=O)C=CC(F)(F)F C(=O)(N=c1c(Br)c[nH]cc1Br)c1cc(-c2ccc([N+](=O)[O-])cc2)cn(C)c1=O C1(NC(C2C(CNC(c3c(CC)n[nH]c3)=O)C2)=O)CCC12CCCC2 C#CC1(C(=O)NCC(CC)N2CCCC2)CCN(C(=O)C(C(C)C)SC)CC1 CC1CN(C(c2ccon2)=O)CC2(CCN(C(C3CCC=CCC3)=O)CC2)O1 C(CC1=CCN(C(c2ccc(Cl)s2)=O)CC1)NC(C1OCC(C)C1)=O c1(OC)cc(C)c(NC(C2CC(O)CN2Cc2sccc2Cl)=O)cc1OC N1(C(c2cnc(C)s2)=O)CCc2cc(C(=O)Nc3cnc(Cl)c(Cl)c3)cnc2C1 CN1CCC(NC(C2(CNC(C3OCCC3(C)C)=O)CCCC2)=O)CC1 N1(C(C2N(C(C)=O)CCCC2)=O)CCC2C(C1)CN2C(c1ncc[nH]c1=O)=O N1(C(C(n2c(C)cc(C)n2)C)=O)CCc2ccccc2C(O)C1 CCC(CC)(C(=O)NC1CC(NC(=O)CN2CCC2C)C(O)C1)c1ccccc1 c1(N(CCOC2CCN(C(C3(N)CC3)=O)CC2)C)ccc(OCC)nc1.C(C)(C)O Cc1cn2cccc(C(=O)NC(C)CNC(c3ccc4c(c3)N(C)CC4)=O)c2n1 c1(CC(N2C(CNC(=O)CCC(=O)c3ccccn3)CC2)=O)ccc2c(c1)CCO2 c1(N(CCCCCC=C)C)[nH]c(=NCC2(NC(C)=O)CCOCC2)nc2sccc12 N1(C(CC2(COC)CCOCC2)=O)CCC2(CC1)CC(NC(=O)C(C)C(C)C)C2 c1(N2C(C)CC(NC(=O)C=CBr)C2)nc(C2CC2)nc2c1CCC2 c1(C(=O)OCC)nc(C(=O)NOCC2CC2)cs1.C1(C2CC2)CNC(=O)N1 CC1(CS(=O)(=O)Nc2ccc(C(N3CC(S(C)(=O)=O)C3)=O)cc2)CCC(=O)CC1 C#Cc1cnc(NC(C2CC23CCN(C(C2CCCC(C)C2)=O)C3)=O)cn1 c1(CC(=O)N(CC(=O)NC(C)C(=O)NC2CC2)CC2CC2)ccn(C)c1 Cc1cc(C2CC2)ncc1C(=O)NC(C)CCNC(=O)Cc1csc(Cl)n1 C1(NC(CS(C)(=O)=O)=O)CC2(C1)CN(C(=O)Cn1nccc1-c1ccccc1)C2 C(CO)(CCCNC(=O)C(C)Cn1ccnc1)NC(C1CC(=C)C1)=O CCCCCC(O)C(=O)NCC1(O)CCN(C(c2cc([N+](=O)[O-])sn2)=O)C1 c1(C(N2C(CNC(=O)Cc3ccnn3C)CC(OC)C2)=O)ccc2n[nH]cc2c1 C1(NC(C(CC=C)NC(=O)CC2CCC(C)(C)O2)=O)CC2C=CCC(C1)C2 CCC(C)C(O)CC(=O)N1CC(CCNC(=O)CCC(=O)c2ccccc2N)C1 c1(C(N(C(c2ccccc2OC(F)(F)F)CC)C)=O)ccc(C(=O)OC)cc1 C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CN(C(C2CC(C)(O)C2)=O)CC12CC2 c1(C(=O)NC2(CNC(C(CCC)(C)O)=O)CCOC2)ccc(C)c(OC)c1F C1(C(=O)N(CCCN(C)C(C2(C)CCOC2)=O)C)(COC)CCOC1 N1(C(C2(C(=O)OC)CC2)=O)CCC(CCNC(C2CC2C(N)=O)=O)C1 c1(OCC)ncc(C(N2CC(NC(c3ccoc3)=O)C(O)C2)=O)cn1 C1(C(=O)NC(CCNC(CC(C)C(F)(F)F)=O)C)CCC2(CC1)CC(N(C)C)C2 Cn1nccc1C(C(=O)NC1(CO)CCC1)NC(C1CC1(F)F)=O C(=O)(CCC(CC)OC)N(CC(C)NC(c1cnc(CC)[nH]1)=O)CC CCCC(C(O)C(=O)N1CC(CO)CC(C)(C)C1)NC(=O)COC C1(C(=O)NC)Cc2ccccc2CN1C(=O)C(=O)NCC1CCC(F)(F)C(=O)N1 N1(C(c2cn(CCC)nc2)=O)CCN(C(c2cc(C#N)cn2C)=O)C(C2CC2)C1 C(=O)(C(F)CC(C)(C)NC(=O)C(F)n1ccnc1)NC(c1c(C)ncs1)C C1(CC)CN(C(C2COCCN2C(=O)CCn2ccnc2)=O)CC(=O)N1 C(=O)(C(C(C)(C)C)N1CCCC1=O)NC(C(C)(C)NC(c1c(C)onc1)=O)C N1(C(COCCC(C)C)=O)CCOC(CN(C)C(C2(N(C)C)CCC2)=O)C1 c1(C(=O)NC2C(C(=O)Nc3c(C)scc3)CCC2)cc(O)nc(O)n1 c1(C(=O)OCC)nc(C(=O)NCC2CCN(S(C)(=O)=O)C2)nn1C C1(C(=O)NCCC(C)N(C)C(c2csc(-c3cnn(C)c3)n2)=O)CC12CC(O)C2 C(C)(C)(C(C)CC(=O)N(C(C)CN(C)C(C)=O)C)NC(c1c(C)cc(C)o1)=O C1(C(=O)NCC(CO)NC(C=NOC)=O)CCC(O)(C(F)(F)F)CC1 C12(C(N3C(CNC(C4CN(C)C(=O)C4)=O)CCCC3)=O)CCOC(C)(C1)C2 C=CC(C)(O)CC(=O)NCC(CC1CC1)C(=O)N(C)C(C1CCOCC1)C N#Cc1csc(C(N2CCN(C3CCN(C(c4ccncc4Cl)=O)C3)CC2)=O)c1 C12(C(=O)OC)CC(N)CC1CN(C(=O)CCOc1ccccc1)C2 C(C(CC(C)C)NC(=O)C(F)(F)c1cnn(C(C)C)c1)NC(c1ccc(C)s1)=O C(CN=c1nc(N2CCC(CN(C)C)CC2)c2sccc2[nH]1)c1ccc(C)s1 CC1CCNCCC1N(c1cccc(C(F)F)n1)C(C12CC(CO)(C1)C2)=O C(=O)(C#CC(C)(C)O)NC(COC)CC(=O)NCc1nc(C)sc1C C1(CNC(CN(C(=O)C(N2CCOC2=O)C)CC)=O)CCOC1(C)C c1(C(N2CCC(NC(CC3(COC)CC3)=O)CC2)=O)csc2c1C(C)(C)CCC2 C(=O)(CS(=O)(=O)CCO)NC1CN(C(c2c(CC)nn(C)c2)=O)CC1(C)C C(=O)(N1CCCc2ccnn21)C1(NC(=O)Cc2cscn2)C(C)CCC1 C(=O)(C(C)(C)C(C)NC(C1CCC2CC1CO2)=O)N(CCC)C C1(C(N2CC(CNC(CCC=C(C)C)=O)C2)=O)CCCC(N2CCCC2)C1 C1(NC(C(C)(C)NC(CCCN(C(=O)OC)C)=O)=O)CCCC2(CCC2)C1 C1(CC(=O)Nc2ccon2)(NC(CN(CC(C)(C)C)C)=O)CCC1 c1(C(N2CCC(N(C(c3ccc(C(C)C)o3)=O)C)C2)=O)cc2occc2s1 C1(C(N2CC(C(C)NC(C3(C#N)CCCC3)=O)C2)=O)CCCC(C)CC1 c1(C(=O)NC(C2CCCC2)CNC(C2CC2C(F)(F)F)=O)ncn2c1CCC2 C1(C2(OC)CCC2)(NC(C2N(C(C(C)=CC=C)=O)CC2)=O)CC1 c1(C(=O)NC2CC(N(C(C(C)SCCCC)=O)C)C2)cnn2c1OCC(C)(C)C2 O=C(C1=CS(=O)(=O)CCC1)N1CC2CCC(C1)N2C(C1Cc2ccncc2N1)=O C1(CNC(c2ccc(SC)cc2)=O)CC2CN(C(=O)CCC3(C#N)CCC3)CC12 c1(C(C)NC(C2CCOC2CNC(=O)C(=O)NC2CC2)=O)cncc(F)c1 CC1CC2(CC(C(=O)NC(CCF)C(=O)NCC3CCC=CO3)C2)C1 N1(C(C2(C(=O)OCC)C3CCC23)=O)CCC(NC(c2ccns2)=O)C1C(C)(C)C N1(C(C2N(C(c3ccc(C#C)nc3)=O)CC(F)(F)C2)=O)CC2(CCOC(=O)N2)C1 c1(CN(CCN(C(CC2C(OCC)COCC2)=O)C)C)ccc(C)c(Br)c1 CC#CCCC(=O)NCC=CCC(=O)NCC(O)C1CC1 C1(NC(Cc2cn(C(C)C)nc2)=O)CN(C(=O)CCn2ccnc2)CCC1CO c1(C(=O)NC2C(CNC(c3cnn(C)c3Cl)=O)C2)cc(Cl)cc(F)c1N c1(OC)ccc(C)c(C(=O)NCCC(C)(C)NC(=O)CN2CCP(C)(=O)CC2)c1 c1(OCC(=O)NC(C)CC(C)NC(c2cc(C(N)=O)c[nH]2)=O)ccccc1C#N O=C1CN(C(=O)C2=COCCC2)C2CCN(C(=O)COC3CCC3)CC2N1 C1(C(C)NC(=O)C(O)C2CCCC2)CCCN1C(=O)CC1(N(C)C)COC1 CCCC(CNC(c1cncs1)=O)C(=O)NCC1(O)CC(O)C1 C1(C(N2CCC(c3ccc(Br)cc3)C2)=O)CNCCN1C(c1sccc1Cl)=O CCC(C(=O)N1CC2CC(C1)CN(C(C1CC3(C1)CC31CCC1)=O)C2)C(C)(C)CC c1(C(=O)NCC2N(C(C3(OC(C)=O)CC3)=O)CCC2)ccncc1Br C(=O)(C1CCCc2sccc21)N1CC(C)CN(C(c2ccnc(C)n2)=O)C(C)C1 C(=O)(CC#Cc1ccccc1)NCC1C(C)(C)CC1O N1(C(CC2C=NN(C)C2=O)=O)CCCC(C2(NC(c3ccc[n+]([O-])c3)=O)CC2)C1 C1(CCCC)CN(C(c2cc3n(n2)CCC3)=O)CCN1C(c1cnc(C)nc1)=O C1(CC=C)(NC(C2CCOC2)=O)CCCN(C(=O)CC=CC)C1 C(C(CC(C)C)C(=O)NC1CN(C(c2ccc(C)s2)=O)CC12CC2)OC N1(C(c2c(C)onc2)=O)CC(C)C(NC(=O)CCC2CCC(=O)NC2)C(C)C1 n1(CCC)ncc(C(N2CCCC2CN(C)C(c2ccn(C3CC3)n2)=O)=O)c1Cl CC(F)(F)C(=O)NC(CNC(c1coc(C2CC2)n1)=O)C1CCC1 CC1(C)CCC(CCNC2CC3CC3(COC)C2)CC1 C(C(C(C)C(C)C)Nc1nccc(-n2ccnc2)n1)NC(c1ccc(C)cc1)=O C1(OC)(CNC(=O)C(O)CN(C)C)CCN(C(=O)CSCc2ccc(Cl)s2)C1 C#CCCCCC(=O)NCCC1CCC(NC(C2(O)CCCC2)=O)C1 CCC(C(=O)NC1CCC(CC(=O)N(CC(C)OC)C)C1)C(F)(F)F c1(C(=O)NCCN(C(C2CCN(C(C(C)C)=O)CC2)=O)C)ccc(O)c(F)c1F c1(OC)cc2c(cn1)N(C(=O)CSc1c(C)oc(C)c1C)CC2 N1(C(=O)OC)CCCC(N=c2nc3c(ncn3C)c(NCc3cc(Cl)no3)[nH]2)C1 c1(C(C)(C)C)ncc2c(n1)CCN(CC1OCCC1CCCl)C2 N1(C(CCC=CC(C)C)=O)CCN(C(=O)C2=CCCCC2)CC1CC1CC1 C(=O)(C#CC1CCCC1)NC(C(=O)N(CC(=O)NC)C)CC(N)=O c1(C(=O)NC)cc2ncc(-c3ccc(C#N)c(OC(F)(F)F)c3)cc2[nH]1 C(CCCC(=O)NCC12CC1CN(C(c1cccn1C1CCCC1)=O)C2)OC CC1CCCC(C)N1CC(N1CCOCC(NC(c2cnoc2)=O)C1)=O N1(C(C(n2ccc(Br)n2)C)=O)CC2CCC1CN2C(=O)CN(C)CCO C[Si]1(C)CCCCN(C(C2N(C(=O)COc3ccccc3)CC23CCCC3)=O)C1 Cc1cccc(-c2cccc(Nc3nccc(N4CC(CO)C5(CC5)C4)n3)c2)c1 c1(C(=O)NCC2(F)CC(CNC(C3CCC(CC)C3)=O)C2)ccc(F)cc1N C1(CC)CN(C(c2nsnc2O)=O)CCC1NC(=O)Cc1cc(O)nc(O)n1 N(C(=NCC1CCOC1)NCC1C(C)(C)C1(C)C)CC(c1ncccc1F)(C)C c1(N(C)CCSc2ccccc2)nc(=N)nc(N2CC3CCC3(C(F)(F)F)C2)[nH]1 c1(-c2nnc(C3(COC)CCN(C)C3)o2)cc2occc2[nH]1.C12CCCN(C1)C2=O CN1N=C(C(=O)N2CCCC(O)(CNC(=O)CCCC(F)(F)CO)C2)CCC1=O c1(C(=O)NCc2ccc(CN(C(=O)CCC3(C)CC3)C)cc2)c(Cl)cccc1Cl N1(C(C(c2ccccc2)NC(C2CC23CCCCC3)=O)=O)CCc2sccc2C1 CC1CC(CNC(C2(C)CCN(C)CC2)=O)CCN1C(c1cnc(N(C)C)s1)=O Cc1cc(C(=O)NCC2CN(C(C34CCC3C4)=O)C(C)(C)C2)cc2c1NCCC2 C1(CNC(c2c(C)occ2)=O)CCCC12CCN(C(=O)CC1COCCO1)CC2 c1(C(=O)NC2CC(C)(C)N(C(=O)CC#N)C2)occ2c1CCOC2 C1(NC(CCCC#C)=O)CC2CCC1N(C(=O)CCc1cnoc1)C2 c1(C(=O)NCCCOC)cc(CNC(=O)Cn2cnnn2)ccn1 c1(NC)cc(=NCCN2CCN(C(C3CCN(C)C3=O)=O)CC2)[nH]cc1[N+](=O)[O-] O=C(C1=CCC(NC(C2CCCCO2)=O)C1)NCC1COC(=O)N1 Cn1ccc(C(=O)NCC2COC(CNC(=O)CC3(N4CCCC4)CC3)C2)n1 CC1(C2CC2C(=O)NC2CCC(CC(=O)NCc3ncc(F)cn3)CC2)COC1 CCC(C)CCCCC(=O)NC1C2CCN(C(=O)C=C(C)C(C)(C)C)C12 C=CCCCCCCC(=O)N(C1CN(C(=O)C(C2CCOCC2)C)CC1(C)C)C C1(CCCNC(=O)C2CC2)CCCCN1C(C1CN(S(=O)(=O)C(F)(F)F)C1)=O C(CCC(=O)NCC1(CNC(=O)COC2(C)CC2(F)F)CCC1)NS(C)(=O)=O C1(C(=O)Nc2cnn(CCF)c2)CCN(C(=O)c2cc3n(n2)CCO3)O1 N1(C(CCN(CC)CC)=O)CCC(C(N2CCC2(C)C(=O)OC2CC2)=O)C12CC2 Cc1cc(OCCC(=O)NCC2CCN2C(C2COC(=O)O2)=O)cc(C)c1 C=C=CC(C)C(=O)NC(C1(C(=O)NC(C)CO)CC1)C c1(SCC(=O)NCC2C(C(=O)NC(c3cn[nH]c3)C)CC2)ccncn1 C1(OCC)(CNC(=O)C(F)(F)C=Cc2ccccc2)CCCCC1 C#CC1(C(N2CCC(NC(c3cc[nH]c(=N)n3)=O)C2)=O)CCCC1 Cc1nc(N(C)CCN(C)C(c2ccnc(CO)c2)=O)c2cnn(C)c2n1 c1(C(N(C2CCCC(NC(CC(C)C)=O)C2)C)=O)ccn(C)c(=O)c1 C1(NC(CN2CCN(C(C(COC)(C)C)=O)CC2)=O)COCC(C)(C)C1 C1(OC)CN(C(=O)CSC2(CO)N(C(c3cccnc3)=O)CC2)CC1CO C1(CNC(Cn2c(C)ncc2)=O)CCC12CCN(C(=O)C(C1CC1)C1CC1)CC2 c1(C(CC)NC2CCCN(C(=O)N(C)C)CC2)nc2ccccc2[nH]1 N1(c2cc(CC(C)C)ncn2)CC2(C)CN(C(c3cccc(F)c3)=O)CC2(C)C1 n1(CC)ncc2c1CC(C(=O)NCC1CN(C(=O)Cc3cn[nH]c3)CC1O)CC2 c1(C(=O)NCC(CN(C(c2c(CC)c[nH]n2)=O)C)C)cc(Cl)cnn1 CC1C(NC(c2ccncc2C(F)F)=O)CC2CCC1N2C(=O)CC1CC1(Cl)Cl CCCCCCCCNC(C1CC2CC2N1C(=O)CCn1cc(C)cn1)=O c1(C(=O)NC2(CNC(CC3CCC(C)(C)O3)=O)CCC2)cnc2[nH]cnc2c1 Cc1nc(N(C)CC2CCN(C(C3CCCN3C(C)C)=O)C2)c(C)c(C)n1 Cc1cc(C(N2CCSC(C(=O)Nc3ccc(F)cc3Cl)C2)=O)cnc1F c1(CC(N2CC(N(C(C3C(C(=O)OC)C3(C)C)=O)C)C2)=O)cn(C)nc1C CN1CCN(C(c2ccccc2CNC(=O)CN2CCCCC2)=O)C(CCO)C1 C1(F)(C(=O)NC(c2ncnn2C)CC)CCCN(C(=O)C2=C(C)CC2)C1 CCC(CC(=O)NCC(F)CNC(=O)CC1CCOCC1)C(C)C C(=O)(C#CC(C)(C)C)N1CCC(CC)C1CNC(c1ncn2c1CCC2)=O N1(C(COC)=O)CCC(CN(C(=O)CC2NC3CCC2C3)C2CC2)CC1 N1(C(c2cc(CCOC)on2)=O)CCCCC1CC(C)NC(=O)C(Cl)=CCl C1(C(C(=O)NCCCC)N(CC)Cc2ccc(C)cc2)CCOC1(C)C C1(NC(C2CCc3c[nH]nc3C2)=O)CC2CN(C(c3cscc3Cl)=O)CC2C1 C1(C(=O)NCCC(C)O)(CO)CCN(C(=O)CCc2ncccn2)C1 c1(C(=O)NCC2(CNC(C=CSC)=O)CCC2)cnc2cc(O)ccc2c1 C1(NC(c2c(C)cc(N)cc2)=O)CCN(C(C2C(C)C2C)=O)CC12CCC2 CCC(C)(C)C(O)C(=O)NCCC1=CCN(C(=O)CCC2CCC(=O)NC2)CC1 C1(NC(CSCC(C)C)=O)CN(C(c2cnn(C3CCCCC3)c2)=O)CC1(C)C c1(C(=O)NCC(C)CNC(C2(C)COCCO2)=O)ccc2c(ccn2C)c1 c1(C(=O)NC(CSC)C)cc2c(-c3cc(OC(C)C)cc(C)c3)cccc2s1 CN1C(=O)Cc2ccc(C(N3CCC(NC(=O)CS(N)(=O)=O)C(O)C3)=O)cc21 CC1C2CCC(C2)C1C(=O)NCC(O)CC(=O)N(C)Cc1cccnc1O CC1(C(=O)NC23CCC(NC(C4CCC=CCC4)=O)(CC2)C3)CCCCNC1=O CCC1=NOC(CC(=O)NCCCNC(c2ccncn2)=O)C1 c1(C(N2C(C(=O)OC)CCCC2)C(=O)NC(C)C)cc2cccc(OC)c2o1 CC(=O)CCCCC(=O)NCC(O)CC(=O)NCC(C)(C)C1(O)CCC1 N1(C(C2(C=C)CCC2)=O)CCCC(N(C)C(C2CCC(CCC)CC2)=O)C1 c1(OC)cccc(C(=O)NCC2CCCN(C(C3C(C)CC3C)=O)CC2)c1C C1(C(C)C)CN(C(c2ccc(N)c(F)c2)=O)CCN1C(=O)C=CC1CCOC1 C12(C(N3CC(CC)(OCC)C3)=O)CC(C)(CN1C(C1CCC(C3CC3)O1)=O)C2 C1(C(C(=O)NCCN(C(Cn2c(CCC)ncc2)=O)CC)C)CCC(C)(C)CC1 C1(C(=O)NC(CC=C)CNC(c2ccon2)=O)CCCCN1C(C)=O C1(CC(=O)NCCOCC(=O)NCC2CC2CO)CCCCCC1 CC1(C)CCN(C(C2CC(=O)NC(=O)N2)=O)C1CC(=O)NCCc1nncs1 N1(C(C=CC=CC)=O)CCCC(C)C1CNC(c1cn(C)nc1C(F)(F)F)=O N1(C(C2CC(OC)C2)=O)CCC(CNC(=O)CCOC2CCC2)CC1(C)C S(=O)(=O)(c1ccc(=NCCCNC(c2cnc(C(F)F)nc2)=O)[nH]c1)N(C)C Cc1c(C(N2CCCC(NC(C3(C)CCCN3C)=O)C2C)=O)cnc2ncnn12 c1(C(=O)NCC(CC)NC(c2cccc(C)c2)=O)nc2n(c1C(C)C)CCCC2 CC1CCN(C(C2CC(O)C2)=O)CC1CNC(c1cccc(C(N)=O)n1)=O C1(CCNC(C2C(C(=O)OCC)C2)=O)CN(C(=O)CCOC)CC1C c1(NC(=O)NCC(=O)OC)nnc(COC)s1 c1(C(C)=O)cn(C(=O)NCC(C2CC2)NC(C2(C(N)=O)CC2)=O)nn1 Cc1cc(CCNC(C2(CO)CCN(C(=O)CCN=[N+]=[N-])C2)=O)nn1C N1(CCC(=O)NC2CCN2C(=O)C=CCN2CCC2)C(=O)c2ccccc2C1=O N1(C(CCN(C(=O)C(n2ccc(C)n2)C)CC)=O)CCCN(C)CC1C N1(C(c2c(C)noc2C(C)C)=O)CCCC2(CC(NC(=O)C(C)N3CCC3)C2)C1 N1(C(c2ccn(CC)c(=O)c2)=O)CCC(CNC(=O)COCC(F)F)C(F)(F)C1 N1(C(C2CN(C(c3cc(C)cc(O)c3)=O)C2)=O)Cc2cccc(Cl)c2C1 C=CC(CC)C(=O)NC1(CF)CN(C(=O)C(C)=C2CC2)C1 c1(-n2cc(C(N3CCOCC3)C)nn2)noc2ccc(F)cc12 N1(C(CSC(C)(C)C)=O)CCC2CN(C(C3(C)CC4CCC3O4)=O)CC2C1 C(=O)(C(C)C(O)CCCC)NCc1ncc(C(N(CCCCCC=C)C)=O)cn1 N1(C(CC2C(C)CCO2)=O)CCC2(C1)CN(C(=O)CCC1(C)CCC(=O)N1)C2 CN=c1cc(C(=O)NC2(C)CN(C(=O)Cc3cccnc3)C2)c(Br)c[nH]1 c1(C(N2CCN(C3CCCN(C(=O)C4CC4)C3)CC2)=O)c(F)cccc1Br C(=O)(C(C)(F)C(C)(C)F)N1CCCC(CN(C(C(CCC)NC(N)=O)=O)CC)C1 CC1CCN(CC(=O)NC(C(=O)NCCCS(C)(=O)=O)C2CC2)CC1 Cc1cc(F)c(C(N2CCOC(C(C)NC(=O)CCCC(F)F)C2)=O)c(Cl)c1 C1(C2CC2)(CNC(c2ncc(C)c(Cl)c2)=O)CCN(C(=O)CCCC2CC2)C1 C(=O)(C(C)CC(C)(C)C)NC(CN(C(C1CC(C(F)(F)F)(OC)C1)=O)C)C Nc1cc(C(=O)NC2(CCNC(C3CCCC34CCC4)=O)CCC2)cc(F)c1 C1(CNC(=O)C(N2CCCC2c2ccc(Cl)cc2Cl)=O)CCC2(CCOCC2)C1 c1(NC(COC)=O)cccc(N2CCN(CC(CO)CO)CC2)c1 CCCC(CC(=O)NCCN1CCC(O)C1)NC(C1CCCC1OC)=O C1(NC(CC2C(NC(C3(CN(C)C)CC3)=O)CCC2)=O)C2CCCOC12 CC(CS(C)(=O)=O)C(=O)NC1CCN(c2nc(C(F)F)nc(=N)[nH]2)C12CCC2 N1(C(c2cn(C)nn2)C(=O)NCCCC)CCCC(C)C1C(=O)OC Cc1nc(N2CC(CNC(C3CCCOCC3)=O)CC2C)cc(C(F)(F)F)n1 c1(CC(=O)NC(CCNC(C(CC)N(CC)CC)=O)C)c(Cl)cnn1C CC(C)CC(C(=O)NC1CCC(=O)NC1)ONC(=O)CN1CCSCC1 N1(C(CC2(C#N)CCC2)=O)C2CCC1C(C(N1CCCCC1C1CCC1)=O)C2 c1(CC)ccc2cc(C(=O)NC34CC(C3)N(C(C3(F)CCOCC3)=O)C4)[nH]c2c1 C(CCCCC(=O)NCc1cccc(OC)c1)N(C(C(C=C=C)C)=O)C C1(C(=O)NCC(CC)C#N)CCC(C)CN1C(c1nccs1)=O C#Cc1cccc(CC(=O)NC(CCF)C(=O)NCCCOCC)c1 C=CCC(CC(F)F)C(=O)N1CCN(C(=O)C(C)n2cncn2)C2(CCC2)C1 c1(NC(C(C)N(CCC)C(c2ncccn2)=O)=O)cccc(F)c1O C1(NC(CCCNC(=O)OCC)=O)CC(C)N(C(c2ncncc2F)=O)C1 S(=O)(=O)(c1cnc(N2CCC3(CCSC3)C2)c(Cl)c1)NCc1c(=N)cc[nH]c1 c1(C(=O)NC2C(NC(c3[nH]nnc3C(F)F)=O)CCCC2)cccc2cc[nH]c12 c1(N2CC(CC=C)(NC(c3ccc(NCC)cc3)=O)C2)cc(=O)n(C)c(=O)n1C N1(C(c2cc(C)[nH]n2)C(=O)NCCCC)CCC(CCC(F)(F)F)CC1 c1(C(=O)NCC(C2CCC2)NC(C2CCCOCC2)=O)ccn2c1CCCC2 C1(C)(CC(=O)OC)CCN(C(=O)NC(c2ccc(Cl)c(Br)c2)C)CC1 CON=C(C(=O)NC(C1CN(C(c2cc(C)c(C)o2)=O)C1)C)c1ccco1 N1(C(C(C)NC(CC)=O)=O)C(C)CC2CN(C(C3OCCC3C(C)C)=O)CC12 c1(C(C)=O)cccc(CN(C(=O)COC2(C)CCC2)C)n1 C#CCC(CC(F)F)C(=O)NCC(C)N(C)C(c1ncn2ccccc12)=O C1(C)(C(=O)NCC(C(=O)NCCN(CCOC)C)OC)CC(=O)N(C)C1 C1(CNC(C2N(C(=O)C(C3(O)CCCC3)F)CC2)=O)(CO)CCCCO1 C(=O)(CC(O)C(C)C)N1CCC(F)(CNC(C2CC(CC)C2)=O)C1 C1(NC(C(CCC)OC)=O)CCN(C(c2ccc(C3COC3)cc2)=O)CC1CC c1(C(=O)NC23C(CN(C(c4cnc(OCC)nc4)=O)C2)C3)ccc2cc[nH]c2n1 N1(c2snc(C(=O)OC)n2)CCCC2CN(C(=O)CCC3CC3(C)C)CCC12 c1(COCCOCCOC)cc(NC(C2CC(O)C2)=O)ccc1Cl Cc1cnc(C(=O)NCC(C2CC2)N(C)C(C2(C)CCNC(=O)C2)=O)cc1C N1(C(C(C)c2cc[nH]n2)=O)CCC2(C1)CN(C(=O)CCC(F)(F)F)CCO2 C1(O)(CC(=O)NCC(CNC(C(C)NC=O)=O)(C)O)CCOCC1 N1(C(C2(CNC(C34CCC(C3)C4)=O)CC2)=O)CCC(C(C)(C)OC(C)C)CC1 c1(SC)cccc(C(=O)N(C)CC2CCN(C(=O)C=NOC)C2)c1 CC1CCCC(OCC(=O)NC2CC(O)(CNC(=O)CN3CCCCC3)C2)C1 C=CC1CCCCN1C(C1CC(F)CN1C(c1ccc(F)cc1C)=O)=O C(=O)(Nn1cnc2ccccc12)C1CC(CNC(C2C(C(C)N(C)C)C2)=O)C1 c1(C(=O)NC(Cc2cnc[nH]2)C(=O)N2CC(OC(F)F)C2)ccc(O)nc1 CCC1=C(C(=O)NCC(O)CNC(c2cc(C)c(F)cn2)=O)CCCO1 C1(C(=O)NC23CCCC2CN(C(c2ccc(F)o2)=O)C3)CCc2nnc(O)n2C1 N1(C(C2(OCCC3(COC)CC3)CCCC2)=O)CC2CCC(C1)N2C(=O)C1CC1 C(=O)(C#CC1(C)COC1)NCC1(O)CN(C(c2c(C)ccc(C)n2)=O)C1 c1(C(N(C)CC2N(C(C3(C=C)CCC3)=O)CCC2)=O)cnc2[nH]ccc2n1 c1(C(N2CCCC(N3CCN(CC(=C)Cl)CC3=O)C2)=O)cnc2n1CCOC2 Cc1ccc(C(C)NC(=O)CC2CCCN2C(c2coc(C)c2)=O)nc1 C1(NC(C(C2CC2)SC)=O)CCCCCC1NC(C1CCC(F)(F)CC1)=O CCCC(C)(O)C(=O)N1CC(N(C(=O)C(F)=C2CCC2)C)C2(CC2)C1 Cc1cc(N2CCC(NC(=O)Cc3nc4ncccn4n3)C2)n2nc(C)nc2n1 N1(C(Cn2c(C(=O)OC)cnc2)=O)CCCC2(CNC(=O)C2)C1 c1(NC(N)=O)ccc(C#N)cc1[N+](=O)[O-].CC(C)CC1CNC(C(C)C)C(=O)N1 c1(OC)ncc(F)cc1C(=O)NCC1CCCCN(C(=O)Cn2cnnc2)C1 N(C(=NCCc1ccccc1)N1CCC(Br)=C(C)C1)Cc1ccc(CC)s1 C(=O)(C(C)(C)C1=CCN(C(c2ccc(CC#N)cc2)=O)C1)NC1C(C#C)CCC1 c1(CC)c(C(=O)N(CC(C)O)CCNC(=O)CC2(C)CC2)cnn1C C12(NC(CN(S(N(C)C)(=O)=O)C)=O)CCCC1CN(C(C1CC3CC3C1)=O)C2 CC1(C)CCCN(C(=O)Cc2cnsc2)C1CNC(=O)C(F)C(C)(C)O c1(C(N2CCC(OCCNC(CC(C)SC)=O)CC2)=O)cncc(P(C)(C)=O)c1 n1(CCOC)cc(C(c2nnnn2C)NCCC2(C)CCOCC2)c(C)n1 C12(NC(CC(C)(C)OC)=O)CCCC1(F)CN(C(C1(C)CC(C3CC3)=NO1)=O)C2 c1(CCC(=O)NC(CCNC(c2nc(C)nn2C)=O)(C)C)cnc2ccccn12 C1(C(=O)NCCC2(NC(CCCCCCC)=O)CCC2)CN2CCCCC2CO1 Cc1cc(=NC(=O)CC(O)c2ccccc2)[nH]n1-c1ccc(Cl)c(Cl)c1 Cn1ncc(C#N)c1NC(C1CC1NC(c1ccc(F)c(Cl)c1)=O)=O c1(OC)nc(C(=O)NCCCNC(C2(C)CC=CCC2)=O)sc1C C1(NC(=O)CNC(C2CCOCC2)=O)CC2CC(C1)N(C(C1CCCCO1)=O)C2 c1(NC(N(c2nccc(OC)n2)C2CCCNCC2)=O)cccc(Cl)c1F C(C(F)(CO)c1ccccc1)N(C(C(N1CCOCC1)C)=O)C1CC1 C(=O)(C(C)CC(C)(F)F)NCC(CC)NC(c1ccc(Br)c(N)c1)=O C(=O)(C1(C)COc2ccccc21)NCC1C(C)(C)CCN(C(C2(O)CCC2)=O)C1 S(=O)(=O)(c1ccc(C#N)cc1)NC1CCCN(C(=O)OC(C)(C)C)C1 CCCCC(O)C(=O)N1CC(C)(OCC(=O)NC(C)C(=O)OCC)C1 C=C(C)C(O)CC(=O)NCC1(CCNC(c2nc(CC(F)(F)F)sc2C)=O)CC1 Cc1cc(CC(=O)NC2(CNC(C3CCCCCC3)=O)COC2)cc(Br)c1 C1(C(N2C(CCC)CN(C(=O)CN3CCSCC3)CC2)=O)CCC2(CCCC2)C1 C1(C(=O)NCCC(=C)C)CCCCCC1NC(c1cc(C(C)C)[nH]n1)=O C1(CNC(C2C(C=C)OCC2)=O)CC2(C1)CN(C(=O)C(C)NC(C1CCC1)=O)C2 C12(CCCNC(C3CCN(C(CN(CC)CC)C)CC3)=O)CCCC1OCC2 N1(C(C2CCCN2C)C)CCCCCC1C=Cc1cccs1 C(=O)(CC(C)(CN(C)C)C(F)(F)F)NC1CN(C(c2c(COC)noc2)=O)CC1C CC1CCC(Cl)=C(C(=O)NCC(C)N(C(=O)CCN2CCCC2)C)C1 c1(C(n2ccnc2)(n2nccn2)C)nc(-c2cccs2)nn1Cc1ccccn1 c1(C(C)C)nnsc1C(=O)NC(CNC(=O)Cc1ccon1)C1CC1 N1(C(C(C)NC(C)=O)=O)CCC2(CCC(NC(C3CN4CCN3CC4)=O)CC2)C1 CCC(C)(O)C(=O)N1CCC(O)(CNC(=O)CCCc2cncs2)C1 CCCCCCCCC(C)C(=O)N1CCN(C(=O)C2=CCOC2)CC1C1CC1 CN1CCn2ncc(C(N3CCCC(N(C(=O)C(Cl)=CCl)C)CC3)=O)c2C1 c1(CNC(C2(CCC=C)CN(C(=O)C(C)C3CCCO3)C2)=O)ncccc1Cl CC(C)CC(C)C(=O)N1CCOCC1CN(C)C(c1cc(F)c[nH]1)=O O=C1NCC2(CN(C(c3c[nH]nc3CNC(=O)C=Cc3cscn3)=O)C2)N1 C(=O)(C(C)(C)CC1CC1)NCC(CCNC(CN(C)C(=O)OC(C)(C)C)=O)O C1(C(C)NC(=O)Cc2csc(Br)c2)CCN(C(=O)C=CCF)CC1 c1(CN(C2COC(=O)C2)C(C(c2ccn(C)n2)C)=O)ccc(F)cc1 Cc1ccc(Cl)c(F)c1C(N1CCC1CNC(C1CCC2CC12)=O)=O c1(NC(C(C)N(CCC)C(C2CC(O)C(F)C2)=O)=O)cc(C)c(F)cc1C c1(OC)ccc(C)c(OC)c1C(=O)NCC1CC(F)CN1C(=O)C1=CC(C)(C)C1 CC1CCN(CC(=O)NCC2(O)CN(Cc3cccc(Cl)c3)C2)CC1 O=C1NCC2(CCCN(CC3CCC(O)C3)CC2)N1 c1(COC)nn(C)cc1C(=O)NCCC1(CNC(c2ccsc2Cl)=O)CC1 C1(CNCc2c(-c3ccc(F)cc3)n[nH]c2)COC2CCCC2O1 c1(C(=O)NC(C2CCCN2C(=O)CCC2CCCOC2)(C)C)n[nH]cc1Br N1(C(CCCN(C)C)=O)CC2C3CCC(C2C1)N(C(c1cnc(O)s1)=O)C3 N1(C(c2on(C)c(=O)c2)=O)CC(NC(c2cnn(CCO)c2)=O)CC12CCC2 c1(C(=O)NCC(C2(O)CN(C(C(C)C(C)O)=O)C2)(C)C)c(N)cccc1F C(=O)(C(C1=C(C)C=CCC1(C)C)N1CCC(CC(N)=O)C1)NCC N1(C(c2c(C(=O)OC)cco2)=O)CC(NC(=O)Cc2ccccc2)CCC1C c1(NC(N2CC(C(N3CC(=O)NCC3)=O)(OC)C2)=O)cc(I)ccc1OC(F)F C(=O)(N=c1ccn(C2CC2)[nH]1)C1C(CC)N(C(C2CCC=CCCC2)=O)CCC1 N1(C(C2N(S(C)(=O)=O)CCC2)=O)CCC(O)C(NC(=O)CN2CCCCC2)C1 c1(C(C)C)cc(NC2(C3CN(C(=O)CCc4cc[nH]n4)C3)CC2)n2ncnc2n1 c1(C(N2C(C)CCC(CNC(CCCCC#C)=O)C2)=O)n[nH]c2ccc(Cl)cc12 c1(OC)c(CN2CCOC(COC)C2c2ccnn2C)cc(C)cc1C C1(NC(c2nnnn2C2CCC2)C2(c3occ(C(=O)OC)c3)CC2)CCCNC1=O C(CN=C(NCc1ccccc1Cl)NCc1cncn1C)OCC c1(C(=O)NC2(CNC(C=CC3N(C)CCC3)=O)CCC2)cc(S(C)(=O)=O)co1 C1(C(=O)NCCCN(C)C(c2ccccc2OC(F)F)=O)C2CCN1CC2 O=S1(=O)CC2CC(NC(c3nnnn3-c3ccccc3)c3ccoc3)CC2C1 CCCCC(C(=O)NC1CCC(F)(CNC(c2csc(C)n2)=O)C1)C(C)C C(COC)(CC(=O)NCC1CCCOCC1)NC(C1CCN(CC)C1)=O N1(C(c2n(C)nc(O)c2)=O)CC2OCCN(C(=O)C3=CS(=O)(=O)CCC3)C2C1 C1(C(=O)NCC2(F)CC(CNC(c3ccc(Br)o3)=O)C2)CCCCNC1=O N1(C(c2cc(OCC)n[nH]2)=O)CC(CCNC(=O)COCCF)C(C)C1 c1(CC)ncc2c(n1)CCC(C(=O)NCCC1CN(C(C3CSC3)=O)CCO1)C2 N1(C(C2C(CNC(C(COC)CC(C)C)=O)CCC2)=O)CCC2(COC(=O)N2)C1 c1(C(=O)NCCC(C)N(C)C(c2occc2F)=O)cccc2ncnc(O)c12 n1(CC(=O)NCC=CCNC(Cc2cc(C)sc2)=O)cnc([N+](=O)[O-])n1 CCC(C)C(C(=O)NCCn1cc(CO)nn1)N(C)C(c1ccoc1)=O CC(C)(C)S(=O)(=O)CC(=O)N1CCC2CN(C(c3cccc(F)c3Cl)=O)CCC12 N1(C(Cc2cc(C)ns2)=O)CCC(C2CCN(C(C34CCCC3C4)=O)CC2)CC1 N1(CC2(C(=O)OC)CCNCC2)CCc2c(NC(C(=O)NC)=O)cccc2C1 c1(C(=O)NNC(=O)c2ccc(Br)cc2)ccc(Br)c(Cl)c1F CCCCCC(=O)NC(c1cccnc1)CNC(C1CC(OC)C1)=O C1(C(=O)NC(C#CC)(C)C)CCCCN(C(=O)CCc2ccco2)C1 CCC(CC)CCC(=O)NCC(O)CCNC(c1cc(C#N)ccc1N)=O S(=O)(=O)(c1ccc2c(c1)OCCCO2)N1CCCC(C(=O)NC(COC)C)C1 c1(C(=O)OC)cc(NC(C2CC2NCc2ccc(C)nc2Br)=O)cc(C#N)c1 C12(CNC(COC(C)C)=O)CCC(CC1)N(C(=O)CC1CCCNC1=O)C2 C(=O)(C1=CCC(C)CC1)NCC1(OC)CCN(C(=O)Cn2nc(C)cc2C)CC1 C1(COC)CCN(C(=O)CC2(N(C(=O)C(F)=C(C)C)C)CC2)CC1 C1(C(=O)OC)COC2(CCN(S(=O)(=O)c3cc(C(=O)OC)sc3Br)CC2)C1 c1(C(=O)NCCCC(C)(C)NC(c2c(CC)c[nH]c2)=O)cc(F)ccc1C C1(C(N(CCCNC(=O)C=Cc2cccs2)C2CC2)=O)CCc2nnnn2CC1 C1(C)(C(N(C)CC2N(C(CCOCCCOC)=O)CCC2)=O)CCCN1C C1(C(N(C(c2cccnc2)C)CC)=O)CC=CCC1C c1(C(N2CCC(C(C)NC(c3c(C)ccn3C)=O)C2)=O)cnc2onc(C)c2c1 C(=O)(C(C)(C)CC(F)F)NC1CC(C)N(C(C2CCC(C(C)(C)C)CC2)=O)CC1 C(CCCC(=O)NC(CC1CC1)C(=O)NCC1(CO)CC(C)C1)OC C1(NC(=O)COCC(F)(F)F)CCCN(C(C2(F)CCOCC2)=O)C1 C1(NC(c2sccc2Cl)=O)CC2(C(=O)NCc3ccc(O)nc3)COC1C2 CCC(C(=O)NCCCOCCC(N1CC=CC1(C)CO)=O)C(C)(C)CC C(CCC(C)(C)C(=O)NCC(CC(=O)N1CC(CC(=O)OC)C1)C1CCC1)OC C(C(CNC(=O)CCSC1CCCC1)C(F)(F)F)NC(C1CC(OC)C1)=O CCC(C(=O)NC1CC2(C1)CN(C(=O)C(=O)Nc1cc(F)ccc1C)C2)C(C)C C(=O)(CC(C(C)OC)NC(=O)CCC1CCCCC1)NCCC(CCC)C c1(C(=O)NC(C2CCCCC2)C(=O)NCc2cnsc2)cc(F)ccc1O CN=c1[nH]cc(C(=O)NCC2(C(F)F)CCN(C(=O)C(CSC)OC)C2)s1 CN1CCC(c2ccccc2)(CNC(=O)Nc2cncnc2NC2CC2)C1 N1(C(Cc2cn(CC)nn2)=O)CC2(CCC(CNC(=O)C(C)c3cccs3)O2)C1 c1(C(N2C(C(=O)OCC)(CNC(C=COCC)=O)CCC2)=O)ccc(C)c(Cl)c1F C1(C2CCN(C(c3cscn3)=O)C2)(NC(c2c(C)cc(C)s2)=O)CC1 c1(C(F)(F)F)ccc(C2CCC2)cc1.N1C(=NCC2CC2)NCC2CCC(O2)C1 CC1(CO)CN(C(C2CC(NC(=O)CCc3cncnc3)C2)=O)CCC1O C1(CC)(NC(=O)CC(F)(F)F)CCCN(C(=O)COC)C1 Cc1oc(C(=O)Nc2cccc(NC(=O)NC3CCC(=O)N3C)c2)cc1Br C1(C(N(CCCOCCN(C(=O)Cn2cccn2)C)C)=O)CCC12CCCO2 N1(C(C2C(NC(CCCCCC)=O)CCOC2)=O)CC2(CCC(=O)N2)C1 c1(C(=O)NCC2(NC(C(C)CCN(C)C)=O)CC2)ccc2nc[nH]c2n1 C1(C(N(CCC(=O)NCC(c2cccs2)O)C)=O)COCCO1 N1(c2ccc(C(=O)OCC)cn2)CCC(C)C(NC(=O)C(c2cccnc2)C)C1 c1(C(=O)NC(CCCC)CNC(c2cc(C)oc2C)=O)c(C)nc2sccn12 Cc1cn(C(C)C)cc1C(=O)NC1CC(CNC(=O)CCN2CCCCC2C)C1 N1(C(CCC)=O)CCOCC1CC1CCN(C(c2oncc2C)=O)CC1 Cc1nn2c(c1CNC(=O)CCCn1cncn1)CN(C(=O)C(O)C(C)C)CC2 N1(C(C2(C(=O)OCC)CC2)=O)CCC2(CC1)CN(C(c1ccc(Cl)cc1O)=O)C2 C(C)(C)(CCCCNC(=O)CCC1CCCCC1)NC(C(CSC)O)=O C=CCC(C)(C)CC(=O)NC(C)(C)CN1CCN(C(=O)Cc2c[nH]nc2O)CC1 N1(C(CC(CC)O)=O)CCC2(CCN(C(=O)C=Cc3ccncn3)CC2)C1 C1(CNC(C(C)(C)SC)=O)N(C(=O)C(F)n2ccnc2)CCC1(C)C c1(C(=O)NC(C)CNC(c2cn(C(F)F)cn2)=O)ccccc1N1CCOCC1 c1(SCC)cc(Cl)ccc1C(=O)NC(CO)C(C)NC(C1CCCN1C(C)C)=O CN(OC1CCCC1)C(=O)C(CC1CC1)NC(C1CC2(C1)CC2(F)F)=O C1(C(N2C(C(C)NC(CCOCC#C)=O)CCC2)=O)COc2cc(F)ccc2O1 C1(NC(CCC2(NC(CC3CCCN(C)C3)=O)CCC2)=O)CCCCNC1=O N1(C(C2C(C)CC=CC2)=O)C2CCC1CC(CNC(C1CC13CCOCC3)=O)C2 CC1=C(C(=O)NCC2CCN(C(C3(CCN(C)C)CC3)=O)C2)CCS1(=O)=O c1(C(N2CC=CC(C(=O)NC3CCCN(C)C3)C2)=O)cc(F)cc(F)c1 c1(N(Cc2cn(C3CCN(C(C(CC)O)=O)C3)nn2)CC)ccc(C(C)C)cc1 CCC(C)C(C(=O)NC(C)C(=O)N(C)C)NC(=O)CCc1nc(C)no1 N1(C(C(CC(=C)C)NC(C)=O)=O)CCCN(C(c2sc(OC)nc2Cl)=O)CC1C N1(C(c2c(C)nccc2)=O)CC2CC(C(N3CC(F)CC3C#N)=O)C(C2)C1 CC(C)CC(F)C(=O)NC1(C2CCCCN2C(=O)CCC(=O)N(C)C)CC1 c1(N2C3CN(C(C4C(C)(C)C4)=O)C(C3)C2)ncnn2cccc12 c1(OCC(=C)C)ccc(CCC(=O)OCCN2CCCC2CC(=O)O)cc1 c1(C(=O)NC2(C(=O)NCCCCCC3CC3)CC(F)(F)C2)cnn2ccccc12 Cc1cc2c(C(=O)NC3(C)CC(NC(=O)Cn4cncn4)C3)cccc2o1 C(=O)(C1=CCC(C)(C)CC1)NC(C1CCCN(C(=O)CSCc2cscn2)C1)C CC1CC(=O)CCC1c1nc(Cc2ccccc2Cl)nn1C(CC(N)=O)C(=O)O c1(OC)nc(C)ncc1C(N1CCC(NC(c2cc(CC(C)C)on2)=O)CC1)=O c1(CNC(c2cccc(Cl)c2Br)c2n(C)nnn2)ccc2occc2c1 N1(N(C)C)CCCN(C(=O)NCc2ccc(Cl)cc2Cl)CC1 Cc1cc(C)c(CN2CCCC(NC(C34CCC(CC3)CC4)=O)CC2)c(C)c1 C(=O)(CN1C(=O)CCCc2sccc21)NCC(CC)NC(C1(C)CC=CCO1)=O N1(C(C(=O)NCC)=O)CCCN(C(c2ccc(F)cc2C#N)=O)C(C)C1 N1(C(c2nc(CC)oc2C)=O)CC2CCC2(CCNC(=O)CCC#N)C1 C1(CN(C(Cn2cc(CC(=O)OCC)nn2)=O)CC)CN2CCC1(C)CC2 C1(OC)CC(CNC(C2CC(O)C2)=O)N(C(=O)CC(F)F)C1 c1(C(N2C(CNC(c3cnc(C)[nH]3)=O)CC(C)(C)C2)=O)ccc(S(C)=O)cc1 N1(C(=O)OC(C)(C)C)CCC2(CCC2C(=O)NCC(=O)NC2CCC2)CC1 c1(NC(C)=O)ccccc1C(F)(F)C(=O)NC1CN(C(=O)C(C)=C(C)C)C1 c1(C(=O)NC2CCC(NC(CCC(C)C)=O)CC2)ncn2cccnc12 c1(CC(N2CCC(NC(c3c(C)cco3)=O)(CF)C2)=O)coc2cc(O)ccc12 c1(OC)cc(Cl)ccc1C(=O)NC(C)(CNC(c1ccns1)=O)CC(C)C Cc1[nH]c2c(NC(=O)NCC3OCCC3F)cccc2c1C c1(CC(=O)NCC(CNC(C(C)C2CCC2)=O)F)ccc(OCC#N)cc1 C(C1=CCCOC1)N(C(=O)C(Cc1ccco1)NC(=O)CCC1(C)CC1)C CC1C(=O)N(C(c2nc(Br)cn2C)=O)CCN1CC1CCOC1 C1(C(=O)NC2COCCC2O)CC2CCN(Cc3c(I)ccnc3O)CC12 C1(c2cn(Cc3ccc(CNC(C4C(C)CC4)=O)cc3)nn2)CCC(C)(C)CC1 C(=O)(C1SCCc2ccccc21)NCCN(C(=O)CC1COCCO1)CC1CC1 C1(C(N2CC(NC(c3c(C)nsc3NC3CC3)=O)C(C)C2)=O)CN2CCC1CC2 C1(CC(=O)NCC(F)CO)C(NC(C2CCCSC2)=O)CC1O C1(NC(=O)CSc2nnc(S)s2)CC(CNC(C2COC2)=O)C12CCC2 c1(CNC(C(c2ccnn2COC)N(C(CC)CC)CC)=O)nnn(C)n1 Cc1cccc2c1ccn2CC(=O)NC1C=CCN(C(=O)C=CC(F)(F)F)C1 C1(C)(CC(=O)N(CC(CC)NC(=O)C(c2ccccc2F)C)CC)CC(F)(F)C1 C1(F)(CNC(C=C(C)C(C)C)=O)CCN(C(c2c[nH]ccc2=O)=O)C1 N1(C(c2c(NC(=O)OC)cccc2)=O)CCC(F)(F)C(CNC(=O)CC(F)F)C1 N1(C(C2(CC)CCOC2)=O)CCN(CCNC(=O)C(F)C2CC2)CC1 N1(C(C2=C(C)CC2)=O)CC(NC(=O)CC2(O)CCCN(C)C2)C(S(C)(=O)=O)C1 N1(C(CCCC=C)=O)CCN(C(C2CC(F)CN2C)=O)CC1CCO N(C1CC2(CCCC2)Oc2ccc(Cl)cc21)C(=O)NC1(C(F)F)CCCC1 C1(NC(C=CC=CC)=O)CC(F)(CN(CC)CC)C1.C1(=O)C(CC)N1 Cc1cnc2ccccc2c1C(=O)NCCC(C)NC(=O)C(C)CF S(=O)(=O)(c1ccc(NC(C)COc2ccccc2F)cc1Br)NCC(C)OC C1(CNC(c2c(F)ccc(OC)c2)=O)CC2(C1)C(F)(F)C21CCC1 c1(C(=O)NCCN(C(c2c[nH]c(=N)s2)=O)CC)sccc1C(C)(C)C CC1=NOC(C(=O)NC2(C)CC(NC(c3nocc3Br)=O)C2)C1 Cc1ccn2ncc(C(=O)NC(C)CC3CN(C(C4(C)CCCC4C)=O)C3)c2c1 C(C(=O)N)(C(C)C)n1cc(C(c2nn[nH]n2)C2CC2)nn1.C(C1CC1)(C1CC1)SC N1(C(=O)OC)CCCN(C(c2ccnc(-c3ccco3)c2)=O)CC1 CC(C)S(=O)(=O)C1CCN(N2CC(CCn3cc(-c4cnn(C)c4)nn3)C2)C1 N1(C(C(CC)c2ccccc2)=O)CCC(C)(C)C1CNC(c1c(O)noc1C)=O N1(CC(=O)NCCC(CNC(CC2C(C)C2)=O)(C)C)C(=O)c2ccccc2C1=O C1(C(N2CC(O)(CCc3cn(CCC=C=C)nn3)C2)=O)(OC)CCCSC1 N1(C(C(C)(C)OC)=O)CCC(CNC(=O)C(c2ccccc2Cl)(C)C)C(C)C1 c1(C(N2CC3(C(NC(C(CCC)OCC)=O)CC3)C2)=O)nc(O)nc(O)c1F C#CCCC(C(=O)OC)NC(=O)CCCCCBr C1(C2CN(C(c3csc(C4CC4)n3)=O)C2)(NC(c2nnn(CC)c2C)=O)CC1 CC1=NOC(CNC(C2(NC(C3CC(C)(C)C3)=O)CC(CO)C2)=O)C1 c1(C(N(CCCNC(C2(C(F)F)CCC2)=O)C(C)C)=O)ccc(F)cc1Cl N1(C(C2(CC)CC2)=O)CC2(CCN(C(=O)C=CCN3CCCC3)C2)C1 CC1CN(C(C23CCCC(C2)OC3)=O)CC2(CCN(C(=O)CCC(N)=O)CC2)O1 CC(C)(C(=O)NCc1cn(-c2cc(C(=O)O)cc(F)c2)nn1)S(C)(=O)=O C1(NC(=O)NCCOC2COC2)CCCN(C2CCCC2)C1 c1(C(N(CCC#C)CCCOC)=O)ccc(OC(c2ccccc2)=O)cc1 c1(C(N2CCC(O)(CNC(C(C)CF)=O)C2)=O)ccc(=O)n(CC(F)(F)F)c1 c1(OCCN(C(=O)C(N2CCC(OCCO)C2(C)C)=O)C)ncc(Br)cc1F C12(NC(C(CCCC)O)=O)CCC(CC1)N(C(c1cnnn1C1CC1)=O)C2 C(=O)(C(CC(F)F)C1CCC1)N(CC(CNC(c1cn(CC)nc1)=O)C)C C#CCCC(C(=O)NC(C(=O)OC)C1CCC1)NC(C1C2CC3C(C2)C13)=O CN1CCN(C(C2CC2CNC(=O)C=CC(N)=O)=O)CC1CC1CC1 N1(c2ncc(C(N3CCOCC3)=O)s2)CCS(=O)C2(CCC2)C1 O=S(=O)(c1ccc(NC2CC3(CCC3)C2)c(F)c1)NC1CCOC12CCCC2 CC1CCNCCC1N(C(C1(C(F)(F)F)CC1)=O)CC1CCCCO1 C(=O)(C(C)(C)C(C)(F)F)NCCN(C)CCF.c12cccc(c1)C(=O)N2 C1(NCC)CCN(CCC(=O)NC(=O)C(C)CSc2ccc(F)cc2)CC1 C1(C(N2CCCC(n3cc(CNC)nn3)C2)=O)COc2c(OCC)cccc2C1 c1(C(=O)NC(C(C)C)CNC(C2CCCCN2C(C)C)=O)ncnc2ccsc12 C1(F)(CNC(CCOC(C)C)=O)CC(NC(=O)CC2CC(F)(F)C2)C1 C1(CNC(c2cccc(C(N)=O)c2)=O)CN(C(c2cscn2)=O)CCCO1 N1(c2nc(NC(CCSC)C)nc(C)c2)CCn2c(nn(C)c2=O)C1 c1(C(=O)NCCCCCNC(C2(C#N)CC3CC3C2)=O)nccc2ncncc12 c1(C(N2CC3C(NC(Cc4c(C)ncs4)=O)(C3)C2)=O)cnc2ccsc2c1 c1(C(=O)NC2COCCN(C(C(CC)C(C)(F)F)=O)C2)oc2ccccc2c1C C1(C#N)(C(=O)NCC(CC)NC(=O)C(C)C(C)C)CC2(CC2)C1 C=CCCCC(C(=O)NC1(C)CC1(C)C)NC(=O)Cc1c(C)noc1C c1(CNC(c2c(CC)cc[nH]2)=O)nc(C(=O)C2CC2)c(C)o1.C1C(C2CCC2)N1 N1(C(C2C(C)N(C)CC2)=O)CC(C(N2CCN(C)CC2CO)=O)C(F)(F)C1 c1(C(=O)NCC#CCNC(C2CCC(C)(CC)O2)=O)cc2ccccc2nc1O CCCCCCCC(=O)NCC1COCC1NC(c1ccc(Br)o1)=O c1(C(N2CCC(C(C(=O)N(C3CCOC3)CC)C)C2)=O)ccncc1NC CCCCC(C)CCC(=O)N1CCC(NC(c2cccc(N(C)C)c2)=O)CC1C C1(C(=O)NC2C(NC(C3CSC3)=O)COCC2)Cc2nnsc2S1 C1(OC)CNC(=O)C1.c1(C(N2CC=CC2CF)=O)cc(CO)nn1C CN1CC(O)CC1C(=O)NCc1csc(C(=O)N(CCO)CCO)c1 c1(C(Cc2ccccc2)SC)nc(-c2ccc(C)o2)nn1Cc1ccc(F)cc1 C12(CNC(c3cn(CC)nc3)=O)CCCC1N(C(=O)CN=S(C)(C)=O)CCC2 c1(C(N)=O)ccoc1C(=O)NCC=CCNC(=O)C=C1CCC1 C1(NCC2(C(=O)NCC(C)(C)C(=O)OC)CC(=C)C2)CCCC(F)C1 C1(CCOC)CN(C(c2ncoc2C2CCC2)=O)CCN1C(=O)CP(C)(C)=O c1(C(=O)NC2COCCN(C(=O)C=Cc3ccoc3)C2)cn2ccc(Cl)cc2n1 CCCCC(CNC(c1cncc(COC)c1)=O)NC(c1cc(C)n(C)n1)=O C(=O)(C1Cc2ccccc21)NCC1(CNC(c2c(C)nn(C)c2)=O)CCOCC1 c1(SC)cc(C(N2CCC(O)(CNC(c3ccc(F)o3)=O)C2)=O)ccc1F O(NC(=O)C(O)CNC(=O)CC1CCCC1O)CC(CC)C Cc1cc(Br)ncc1NC(C1CCN(C(c2ccc(F)cc2)C)C1=O)=O Cc1cnc(N(C)Cc2cscn2)c(S(=O)(=O)NC(CO)C2(C)CC2)c1 N#CC1(C(=O)NC2CCC(NC(C3(C(F)F)CCCO3)=O)CC2)CCOC1 C(C)(CNC(C1(C)CC1(C)C)=O)(CC(C)C)NC(CCc1ccc(C)cc1)=O C1(C(C)NC(C2(C(=O)OCC)CC2)=O)CCN(C(C2(F)CC2)=O)C1 c1(C(=O)NCC(CNC(c2ncc(Br)cn2)=O)OC)cnc(O)n1C C(C(C)(C)CC(=O)NCCC1CC(NC(c2ccc(Cl)nc2OC)=O)C1)OC Cc1ccc(C(C)C(=O)NC2CC(NC(c3ncncc3Br)=O)C2)cc1 N1(C(CC(=O)OC)=O)CCCN(C(c2ncnc(OC)c2OC)=O)C(C)C1 C12(NC(COCCC)=O)CCCC1N(C(=O)Cn1cc(C)cn1)CC2 c1(-n2cc(C3(C)CCCC3)nn2)cccc(C(=O)NCCc2cccnc2F)c1 C(CC(C(=O)N1CCC(C#N)C1)NC(=O)CCCOC)OCC C12CCC3(CC1)CC(C3)CN2.C1(C(=O)OC)CN(C(=O)OC(C)(C)C)C2CC12 S(=O)(=O)(c1c[nH]ccc1=NCc1ccc(Cl)s1)NC(C)C(C)CO CCC(CNC)CC(=O)N(CC)CC1CCN(C(c2cc(CC(C)C)c[nH]2)=O)C1 c1(OC)ccc(CCCC(=O)NC2COCC2NC(=O)C(C)C(C)O)cc1 N1(C(C)=O)CC2(C1)CN(C(=O)Cc1cn3c(C)cncc3n1)CC2C(O)C1CC1 C1(CNC(c2cc(CCCO)on2)=O)CN(C(=O)C(F)F)CC1C(F)(F)F N1(C(C(CC=C)C)=O)CC2CCC1CC2NC(=O)C(F)(F)C1(O)CCC1 c1(NC(N(CCC(=O)NCC(=O)N(CC)CC)C)=O)cn(C)cc1C C(CCCCC(=O)NC(c1cn(C)nn1)C(=O)NCc1ccc(F)c(F)c1)OC N1(C(C(Cc2ccc(C=C)cc2)N)=O)Cc2c(OC)ccc(C(=O)OC)c2C(O)C1 N1(C(CCN(C)CC)=O)CCC2(CC1)CCN(C(=O)CC1CCC(C)O1)C2 c1(C(=O)OC)c(C(=O)NCC(C2CCOC2)NC(C2CCCCC2)=O)n[nH]c1C C(=O)(C1=C(F)CN(C(C2C3CCC(C3)C2C)=O)CC1)NCCCCCC C1(CNC(C2(C)CCC2)=O)CC2CC(C1)N(C(c1cnn(CC(F)(F)F)n1)=O)C2 C1(CC)(NC(=O)CC2(O)CCC2)CCCN(C(=O)C(C)CC2CCCC2)C1 C(=O)(C(C)(C)CSC)OC.c12ccccc1Cn1cc(nn1)CN(O)C2=O C(=O)(CCCCC(C)C)NC(C(C)NC(c1n(CC)cc(Br)c1)=O)C C(=O)(C(CCCOC)NC(c1c[nH]c(C(N)=O)c1)=O)NCC=C c1(N2C(CCNC(C(CCC)(C)O)=O)CSCC2)nc(C)c(C#N)cc1Cl c1(CCCC(C)SC)nc(CCN(C)C)nn1-c1cnn(C)c1 c1(C(N2CCC(C)(CC(=O)NCC(c3ccco3)O)C2)=O)cc2occc2[nH]1 O=C1NC(Cc2ccc(F)c(Cl)c2)C(=O)N1Cc1cccc(-n2cncn2)c1 C(=O)(C(C)(CO)NC(c1nc(CO)oc1C)=O)N1CC(C)(CC)C1 CCC(C(=O)N(CCN(C)C(c1cnn(C2CC2)c1)=O)C(C)C)OC1CCCC1 N1(C(C2CCC(OC(C)C)CC2)=O)c2ccccc2CC(C)C1C c1(C(=O)NCCc2ccncc2)ccc(C2CC2)cn1.O=C1NCCN1 c1(C(=O)NCC2N(C(C(C(CC)O)C)=O)CCC2)c(Cl)ccc(C)c1O c12ccc3c(c[nH]c3c1)CN2.c1(-c2ccc(SC)s2)ccc(C(=O)O)c(C#N)c1 C1(N2CCC(CNC(C3C(C)(C)C3)=O)C2)CC2CCCCC2NC1=O c1(C(=O)NC2CN(C(C=CC=CCC)=O)C(C)C2)c(Br)c(C)nn1C C1(C(=O)NC(C)CCC(F)F)CC2(CCCCC2)C1 N1(C(c2ccc(CCCCC)cc2)=O)CCC(NC(=O)C(C)C2CC2)CC1C CC(C)CCCC(=O)NCCC1CN(C(=O)CCCn2ccnn2)CC(C)O1 C1(C2CN(C(=O)CCCC(N)=O)C2)(NC(Cc2c(C(=O)OC)csc2)=O)CC1 C(=O)(C(C(C)(C)C)n1ccnn1)N(CC(CNC(CN1CCC(C)CC1)=O)C)C c1(OC)ncc(Cl)cc1C(N1CCCC(N(C(=O)C(C(C)C)OC)CCO)C1)=O C=C(C)CC(C)C(=O)N(C1CN(C(c2oc(C)nc2CC)=O)C1)C c1(C(N2C(C#N)CN(C(=O)Cc3ccncc3)CC2)=O)ccc([N+](=O)[O-])c(F)c1 C1(NC(C(C2CC2)OCC)=O)CCCC1CNC(=O)Cn1cnnc1C1CCC1 C1(C(=O)NC2(CC=C)CCC2)CC2CN(C(=O)C(C)(C)C(=C)C)CC2C1 N1(c2cc(C(=O)OC)nc(Cl)n2)CCC(NC(c2csnc2C)=O)C(CO)CC1 C1(C(=O)NC2C(NC(Cc3c(C)non3)=O)CCC2)Cc2ccccc2S1(=O)=O c1(C(N2CCC(NC(CC3(C)CCC3)=O)C2)=O)cccc2ncsc12 N1(C(C=C(CC)CC)=O)CCC(C)C(CNC(=O)CCCCCN(C)C)C1 c1(N(CC(F)F)C)nc(=NCCc2ccsc2Cl)[nH]c2c(F)cccc12 c1(C(=O)OCC)cccc2c1CCC2NC(=O)Nc1c(Br)nn(C)c1Br c1(C(=O)OCC)cc(=NCC2CC(n3ncn4cccc4c3=O)C2)[nH]cc1C#N C1(NC(c2c(C)nc(C)s2)=O)CN(C(c2cnc(Cl)[nH]2)=O)CC1C1CC1 c1(OC)cncc(CC(=O)NCC2CCC(NC(C3CCS(=O)CC3)=O)CC2)c1 CC1(NC(c2cc(O)nc(C3CC3)n2)=O)CCN(C(C2CCCCS2)=O)CC1 c1(C(=O)NC2C(NC(C(C(C)(C)C)O)=O)COCC2)cnc2ccccn12 c1(C(N(C2CCC(NC(C3(COC)CCCC3)=O)C2)C)=O)ccc(P(C)(C)=O)o1 C(=O)(CCC(C(=O)O)NC(c1ccc(F)cc1C(F)(F)F)=O)N(C)C C(=O)(C(=O)C(C)(C)CC)N1C(CCC)CN(C(=O)Cn2cc(C)ccc2=O)CC1 c1(C(=O)NC2(C)CN(C(Cn3ncc(C)c3)=O)C2)cn(C)c2ccccc12 C12(CNC(C(C)(c3cccs3)OC)=O)CCC(CC1)N2C(C1CN(C(N)=O)C1)=O C1(C(=O)NC2(CCOC)CCC2)(CC)CCCN(C(=O)CC2CCCC2O)C1 c1(OC)cc(O)cc(OC)c1C(=O)NCCC1CC1.c12cccc(F)c1CN2 C1(CC(=O)NCC(C)N(C(c2ccccn2)C(N)=O)C)COC(=O)C1 c1(CC(N2CCC(NC(C(C)OCC)=O)C2C2CC2)=O)ccc(C(C)C)cc1Cl Cc1cccc2c(C(=O)NC3CN(C(c4cnc(Cl)c5ccsc45)=O)C3)cnn12 C1(C(=O)NC2CCN(C(c3ncn(C(C)(C)C)c3)=O)CC2)CCCC1S(C)(=O)=O C(=O)(C(C(C)O)N(C)C)NCC1(OC)CN(C(c2cc(C3CCCC3)[nH]n2)=O)C1 N1(C(CNC(CC(C)(C)C)=O)=O)CC(NC(c2cnn[nH]2)=O)Cc2ccccc21 N1(C(C2C(C(N(c3nccc(F)c3F)C)=O)C2)=O)CCc2ccc(C#N)cc2C1 N1(C(C2=NNC(=O)CC2)=O)CCC2C(CCCN2C(=O)CCCC(F)(F)F)C1 c1(C(N(CCOC)CCNC(=O)CC2CCOC2=O)=O)cc2ccccc2o1 N1(c2nnc(CCOc3cccc(C)c3)n2C)CC(C(=O)N(C)C)C2(CC2)C1 C1(OC)CC2(C1)CC(C(N1CCN(C(=O)C(c3cnccn3)C)C(CF)C1)=O)C2 C1(NCC(N2CCC(F)(F)CC2)=O)CCCCC2CN(Cc3ccccc3)CC12 C1(C(=O)NC(C(=O)OCC)CO)CSCCN1C(=O)CN1CCCC1 c1(CC)ccccc1C(=O)NC1CCOCC1NC(=O)CCCn1ccnc1 CC1CCC(CC(=O)NCC(C)N(C)C(C2CCC(CC#N)CC2)=O)OC1 CCC(C)C(O)C(=O)NCCCC(C)NC(c1c(OC)nsc1OC)=O c1(C(N2C(CNC(=O)C=Cc3ccccc3)CCCC2)=O)n[nH]c2c1CC1CC21 Cc1nc(C(C)(C)C)ncc1C(N1CCCCC1CNC(c1cnoc1C)=O)=O C(C(=O)NCC1(C(N)=O)CN(C(=O)C(c2ccccc2)C)C1)(C(C)C)SCC N1(C(CNC(CCCCC)=O)=O)CCC(C2CCN(C(=O)C(F)=C3CCC3)C2)C1 N1(C(CS(CC)=O)=O)CC(CNC(c2ccc(OC3CCC3)cc2)=O)C(C)(C)C1 CC1=NN(C)C(=O)C1CC(=O)NCCOCCNC(=O)CC1CCOC1C N1(C(c2c(OC)nsc2)=O)CCC(NC(=O)C(=Cc2c[nH]cn2)F)C(F)(F)CC1 N1(C(c2c(Br)c(C)n(C)n2)=O)CC(CNC(=O)CC(C)F)CC(C)(C)C1 C1(C(=O)NCC(CNC(CN(CCC)C)=O)C(F)(F)F)CCn2ncnc2C1 CS(C)(=O)=NC(=O)C(=O)NCC1CN(C(c2c[nH]nc2C2CCOC2)=O)CC1O c1(OC)cc(C(N2CC(F)CC2CN(C(=O)C(F)OC(F)(F)F)C)=O)ccc1Cl c1(OCC=C)ccc(CNC2CC2C(=O)Nc2cn(C)nc2C)cc1 N1(C(c2ccc(C(C)(C)C)s2)=O)CC(NC(C2CCCO2)=O)CC(O)C1 c1(C(C)NC(=O)CCNC(=O)C(=O)N(C)C)ccccc1NC1CC(=O)N(O)C1 Cc1ccc(F)cc1CC(=O)NC1CN(C(=O)C(O)c2ccsc2)CC1C N1(C(CC(=O)NC)=O)CCC(C)N(C(C2CC(C)CO2)=O)CC1 c1(SCC)ccc(C(=O)NCCOCCN(C)C(C2CNC(=O)N2)=O)cc1 c1(C(=O)NC2CCN(Cc3cccc(CC(=O)OC)c3)CC2)ccc(C)cc1C N1(C(C(C(=O)OCC)F)=O)CCCC(CCNC(=O)C(C(C)CC)N(C)C)CC1 c12ccc(cc1)NC(C(C)C)CNC2=O.c1(C(C)=O)cccc(NC=O)c1 C1(CC(=O)NCC2CCCN(C(C3CC4CCC3C4)=O)C2)CCCC(F)(F)C1 c1(NC(CC2(O)CCN(C(C=CC)=O)CC2)=O)cc(Cl)cc([N+](=O)[O-])c1 C(=O)(C1=Cc2ccccc2OC1)N1CC2N(C(c3csc(C)c3C)=O)C(CC2)C1 N1(C(c2c(CC)ccs2)=O)CCN(C(C2(CO)CCCC2)=O)CC1CS(C)(=O)=O CC1(C)COC(C(=O)NC(CNC(c2ccccc2OCCF)=O)C2CCC2)C1 C(=O)(C1=NOC2(CNC2)C1)N1C(CC)CN(C)C(=O)C1 CCCCC(CCCC)(c1nnnn1CCSC)NCC1CCC2(CC2)C1 C1(NC(c2ccc(C)s2)=O)C2CC3CN(C(C4CC(C)OC(C)C4)=O)C1C3C2 C(=O)(C(F)(F)C(O)C1CC1)NCC1N(C(c2ccc(C(C)C)cc2)=O)CC(F)C1 C1(C(=O)NCCOCCNC(CCN(C)C2CC2)=O)CC2C=CC1C2.OC(F)(F)F CC(C)(C)CCC(=O)NCC12CC(NC(C3CCCCC3(F)F)=O)(C1)C2 Cc1cn2c(n1)CCC(C(=O)NCC1CN(C(=O)CCOC3CC3)CC13CC3)C2 c1(NC(=O)NC23N(C(=O)OC(C)(C)C)CCC2C3)ccc(F)c(Cl)c1F C(C(=O)Nc1ccccc1)(C(C)(C)C)NC(C=Cc1c(C)n[nH]c1)=O C1(NC(C(=O)NCC)=O)CCN(C(=O)OC)CC1OC1CSC(C(F)(F)F)C1 C#CCC(C)(C(=O)NC1CCN(C)C1)NC(C1CCCC1)=O C1(CC(=O)N(C)CC2(F)CCC2)C(NC(c2ocnc2C2CC2)=O)CC1O CC1(C)CC(CC(=O)N(C2CCCC2)CCCc2ccn(C3CC3)n2)C(=O)O1 C1(C(=O)NCC2N(C(C=CSC)=O)CC(C)(C)C2)CCc2nnn(C)c2C1 c1(C(=O)NC2CCCCN(C(C3(C)CCCO3)=O)C2)cccn2nncc12 C(=O)(C(=O)N=c1cc(C)o[nH]1)NC1CN(C(CC(C)OC)=O)C2C1CCC2 c1(C(=O)NC2CC(F)(CNC(C3CC4(CSC4)C3)=O)C2)[nH]c2ccccc2c1Cl c1(C(=O)NCC2CC3CC3N2C(C2CC(F)(F)C2)=O)cc2cccn2cn1 C1(C)(C(=O)NC(CC)C(C)(C)O)CCN(C(c2ccc[n+]([O-])c2)=O)CC1 CCCCCC(C(=O)N1CCC(C)(CNC(C23CCOC(C)(C2)C3)=O)C1)C(C)C c1(OC)cc2[nH]ncc2cc1NC(C1CC(NCc2cnc(Cl)nc2)C1)=O C1(NC(C(C2CCN(C(c3cc(C)sn3)=O)C2)C)=O)C2CCC(C2)C1CO Cc1cncc(S(=O)(=O)NC(c2cc3cnccc3o2)C)c1 c1(C(N2CCOCC(NC(C(C(C)C)C3CCC3)=O)C2)=O)ccc2c(c1)CCO2 N1(C(C=CCCC)=O)CCCC(C(C)(C)C(=O)NCC(O)C(F)F)C1 C#Cc1ccc(C(=O)NCC2(OC)CCN(C(c3c(Cl)noc3C)=O)C2)nc1 C(=O)(CC(C)CCC(=O)Nc1cnn(CSc2ccccc2)c1)OC c1(OC)ccc(N)c(C(=O)NC23CC2CN(C(c2nncn2C2CC2)=O)C3)c1 Cc1cnc(C(=O)NCCOC2CN(C(C3(C)CCCCC3C)=O)C2)cc1C#N c1(OC)ncc(C(=O)NC23CCC(C(=O)O)(CC2)O3)cc1Cl C(CN=c1[nH]c(=N)[nH]c(=NC2CC3CCCCCC23)[nH]1)c1scc(C)n1 N1(C(c2cc(SC)c(N)cc2)=O)CCC2(CC(NC(=O)C(C)(F)C(C)(C)F)C2)C1 Cc1ccc2[nH]c(C(=O)NCC3(F)CN(C(c4cnsn4)=O)C3)cc2c1F N1(C(C(C(=O)OC)C)=O)CC2CCC2(CC(=O)NCC2(C#N)CCOCC2)C1 C1(F)(CNC(C(c2cncn2C)N(C)C)=O)CCC(NC(=O)Cc2cc[nH]n2)C1 O=C(C1=Cc2c(ccc3ccccc23)OC1)OCC1CCC2(CC1)COCCO2 N1(C(C2(NC(C(C)NC(CC)=O)=O)CCC(C)(C)C2)=O)CCC(=O)N(C)CC1 C(C(C)(C)CCCC(=O)OC)NC(=O)NC(CC(CC)C)CC FC1(F)CC(n2nnnc2C2CC(NCC3CC(c4ccccc4)C3)C2)C1 C1(NC(C2C(C)CCC2)=O)CCN(C(=O)Cn2ccccc2=O)C1(C)C c1(CC(=O)NCCC2CCCN2C(=O)C(O)C(F)F)ccc(F)cc1 N1(C(C2ON=C(C)C2)=O)CC=C(CCNC(C2CC2(F)F)=O)CC1 Cc1cc(Cl)c(O)c(NC(c2ccc3nnnn3c2)=O)c1F N1(C(C2(C(=O)OCC)CC2)=O)CCc2cc(Nc3cc(CC)nn3C)cnc2C1 c1(C(N2CCC(C)(C)C(CNC(c3cn[nH]c3)=O)C2)=O)cnc2ccnn2c1N CC1CCCC1(C)C(=O)NC1C2CC(NC(=O)Cc3cn[nH]c3)CC12 c1(NC(c2n(CC)ccn2)c2nnnn2C2CC2)cncc(C(F)(F)F)c1 C(CCCC(CO)NC(=O)C(c1ccccc1)N(C)C)NC(c1scc(C)c1)=O Cc1noc(C)c1CN(C1CCC(COC(C)C)O1)C c1(C(N(CCCNC(C2CC23CC3(F)F)=O)CC)=O)nccc2ccsc12 c1(C2C(C(N(CC(CNC(COCC(=C)C)=O)C)C)=O)C2)ccncc1 C1(SCC2CC(C)OCC2)CC2CC3(CC2C1)OCC(C)(C)CO3 C(C(CC1CC1(F)F)C(=O)N(C)CC1CCC1)NC(C(C)OCCOC)=O C(CCCCCNC(C1(C)CC1C)=O)N(C(CCCOCC=C)=O)C N1(C(c2c(N)ccc(F)c2)=O)CCN(C(=O)CC2CCC2)CC(O)C1 C1(N(CC(=O)NC(CN(C(C(C)OCC=C)=O)C)CC)C)CCCCC1 C1(NC(COC(C)C)=O)CC2CC1CN(C(=O)CCc1cccc(C(N)=O)c1)C2 C(=O)(CCCC(F)(F)CO)NCC1CCC(NC(C(C)(O)c2ccccc2)=O)CC1 c1(C(N(C(C)C)CCNC(C2COC(C)C2)=O)=O)cc(F)cc2nn[nH]c12 C(CC(C(=O)NCCc1ccc(F)cc1)NC(C1CC(C#N)(OC)C1)=O)OCC c1(N(C)C)cc(C(=O)NC2(CO)CN(C(C3COC(C)(C)C3)=O)C2)cc(Cl)n1 C1(CNC(c2n[nH]c(C)c2C)=O)CC(C)CN(C(=O)C=CC2CCOC2)C1 CS(=O)(=O)CCCC(=O)NCC1COCC1NC(c1cccc(C(F)(F)F)c1)=O N1(C(C(C)n2ccnn2)=O)CC(NC(=O)CC(F)(F)Cl)C(N=[N+]=[N-])C1 C(=O)(C1CCCn2nccc21)N(CCCCCCNC(C1(OC)CCSC1)=O)C CCC(CNC(=O)CCc1nc(=N)[nH][nH]1)(CC)C(=O)NCC1CCC(O)C1 C(=O)(C(=O)C(C)(C)C)NC(CCNC(C(C)SC(C)C)=O)(C)C C1(CC)CCCN(C(=O)CC(C)CC)C1C(=O)NCC1COCC(C)O1 Cn1nc(C(=O)NC2CCC(NC(=O)NC3CC3)C2)c2ccccc12 C(=O)(C(F)(F)C(O)CC)N(CCCNC(c1nc(CC)sc1)=O)CC CC1(C)CC2(CC(C(=O)NCCC3=CCN(C(=O)C(C)CC(N)=O)CC3)C2)C1 c1(OC)ccc(F)c(NC(C2(C)CN(C(c3cccc(Br)c3)=O)C2)=O)n1 N1(C(COC)=O)CCOCC(F)(CNC(C2CCCN(c3nccs3)C2)=O)C1 C(=O)(CC(C)CC(C)C)NCCCN(C(c1c(CC)cccc1F)=O)C N1(C(C2(CS(C)(=O)=O)CCNCC2)=O)CC=C(c2cccc(F)c2)CC1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCC(C(C2CCC(C)(C)O2)C2CCCN2)CC1 N1(C(COCC=C)=O)CC2(C1)CN(C(c1ccc(-c3ccncc3)o1)=O)C2 N1(C(c2scc(C)c2)=O)CCC(C)(C)C1CNC(C1(C)CCN(C)C1)=O C1(NC(c2ccc(C#C)o2)=O)CC2CCC(C1)N2C(=O)CC(C)CC(C)C C(=O)(C1=CC2CCC(C1)C2)NCC1C(CC(=O)NCC(C)CN(C)C)C1 CCC(C)C(C(=O)N(CCCNC(c1cnncc1O)=O)C(C)C)NC(=O)OC c1(OCC)ccc(C(C(C)C)NC(=O)NC2(CCF)CCC2)cc1F N1(C(C2(C#C)CN(C(=O)CCCCC)C2)=O)CC2(CCC2)C12CCC2 C(C(O)CC(F)(F)F)NC(C1C2(CC(NC(CCCOCCC)=O)C2)C1)=O c1(C(N2CCC(NC(c3cnc(O)c(F)c3)=O)C2)=O)cccc(S(=O)(=O)CF)c1 c1(C(N2C(C)CN(C(C3CCSCC3)=O)CCC2)=O)cc2c(nn1)CCCC2 c1(C(=O)NC2CN(C(CC3CCCN(C)C3)=O)C(CO)C2)cc2cccnn2n1 c1(C(C)NC(C(=O)N(C2CCC(C)C2)CCO)=O)ccc(Cl)cc1 c1(CC(=O)NC2(C)CC(NC(COCC(=O)OC)=O)C2)nc2c([nH]1)CCCC2 c1(C(N2CCC(NC(C3CCN(C)CC3)=O)C(F)C2)=O)ccc(I)c([N+](=O)[O-])c1 C1(CC(=O)NCC2(CC(N3C(C=C)CC3)=O)CC2)CC2(CC2)CO1 N1(C(C2(COC)CC=CC2)=O)CC(N(C)C(c2nnc(C)s2)=O)C2(CC2)C1 c1(CC(=O)NC2C3CN(C(C(C(C)O)C)=O)CC2C3)cc(Cl)ccc1[N+](=O)[O-] C1(C)(C(N2CC(CNC(CCc3c(C)noc3C)=O)C(O)C2)=O)CCCNC1=O Cc1nc2cnn(C)c2cc1C(=O)N(C)CCN(C(=O)CCc1cscn1)C Cc1cnc(C(=O)NC2CCC(CCNC(C3(F)CCCOC3)=O)C2)cn1 N#Cc1ccc(CN2CCC2C(=O)Nc2cccc(CCO)c2)cc1Cl CCC(CC)C(C)C(=O)N1CCCC(CC)(NC(c2cn(C3COC3)nn2)=O)C1 N1(C(CCOCC#C)=O)CC2=C(C1)CN(C(c1occc1COCC)=O)C2 c1(C(=O)C2CC2)ccc(NC2CC2)nc1.C1(N)CC(NC(C2(C=O)CC2)=O)C1 N1(C(c2n(CC)nc(C)c2)=O)CC2CC1CN2C(=O)COc1c(C)cccc1C c1(C(=O)NCC2COCCN2C(=O)CC(O)C2CCCC2)ccnc2ncnn12 c1(C(=O)NCCCN(C(C2C(C(=O)OCC)C2)=O)C)nc(C)c(C)[nH]c1=O c1(C(=O)NC2CCN(c3nccc(C)n3)CC2F)cccc2c1CC(=O)N2 C1(C)(CNC(CC2CCN(OC)CC2)=O)COCCN(C(=O)C(C)(CC)CO)C1 C(=O)(CC(C)C(=O)NCC(C)C(=O)NCc1ccnc(CO)c1)OCC N1(C(C2C(C=C)OCCC2)=O)C2CCC1CC(CNC(=O)CCOCCOC)C2 C1(C)(C(=O)NC(CC)CC)CN(C(C2CCCN(C)C2)=O)C(C)(C)C1 C(N=c1[nH]c(=NC(C)c2ncnn2C)c2[nH]ccc2[nH]1)c1ccc(SC)nc1 Cc1noc(C)c1NCC1CCCC1Oc1cccc(CO)c1 c1(C(N(CCOCCN(C)C(c2cc(CO)[nH]n2)=O)C)=O)c(O)cc(Cl)cc1F Nc1ccccc1CNC(=O)Nc1cnn(-c2cccc(C(F)(F)F)c2)c1 C1(NC(c2n(CC#C)ccc2)=O)CCC(C)(CNC(c2csc(Cl)c2)=O)C1 c1(C(=O)NCCCC2N(C(C3CC(N(C)CC)C3)=O)CCC2)cc(Cl)ccc1F C=CC(C)CC(=O)NC(CO)C(C)NC(=O)CC(=O)N(C)C O=C1CCCC(C(=O)NC(CCC2CC2)C(=O)N2CC(F)C(F)C2)CC1 C1(C(=O)NC(CC(C)NC(=O)CN(C)C)C)CCN(c2nccs2)CC1 c1(C(N2CCC(N(C(C(F)=CC)=O)CC3CC3)CC2)=O)cc(C)cc(OC)c1O N1(C(C(CC=C)c2ccccc2)=O)CC2CN(C3CCN(C(C)C)C3=O)CC2C1 Cc1ncccc1-n1nc(C(C)C)nc1CC1CCCC1(F)F C(=O)(C1=CCCOCC1)N(C(C)C)CCNC(C1CC(=O)C1C(C)(C)C)=O N1(C(C2(C)CCN(C)C2)=O)CC2CN(C(c3ccn(C4CC4)n3)=O)CC2(C)C1 N1(C(C(CC)CCOC)=O)CC(NC(=O)CC23CCC(CC2)C3)CC12CCCC2 N1(C(CN(C2CC2)CC)=O)C(CNC(c2cncs2)=O)CC2CC12 N1(C(CONC(=O)CCC2CC2)=O)CCc2n[nH]cc2C1 CCCCC(CC)CC(=O)NC1(C)CCCC1NC(=O)CCC1CCCC1 c1(CC)cccc(C(N2CCOCC(CNC(c3ncncc3F)=O)C2)=O)c1N Cc1cc(C(=O)NCC(C)CN(C)C(c2cnccn2)=O)co1 CCN=C(NCc1ccn(-c2ccccc2)n1)NC1Cc2ccccc21 Cc1nc[nH]c(=NCC2CN(C(=O)Cc3nc(C(C)(C)C)cs3)C2)c1Br C1(F)(C(=O)NCCN(C(c2cn(C(C)C)nn2)=O)CC2CC2)CC=CCC1 C1(C(=O)NCCCOCC#C)CCC2(CC2)N1C(=O)C(C)S(N)(=O)=O C1(NC(CCCOCC)=O)CCN(C(C2CCC(=O)N2)=O)C1C(C)C CCCC(C(=O)NCc1ncoc1C1CN(C(c2ccn(C)c2)=O)C1)OC C1(CC=C)(NC(=O)CCc2ccccc2)CCCN(C(=O)C(C)NS(C)(=O)=O)C1 C1(CNC(c2n(C=C)nnc2)=O)CC12CCN(C(C1COCC(C)(C)O1)=O)CC2 c1(C(=O)NC2CCC(NC(=O)CNc3cccnc3)CC2)cnn2ccncc12 CC(CSc1ccccc1)C(=O)N1CCC(N(C(=O)CN(C)C(N)=O)C)C1 C1(C(=O)OCC)CC2(CCN(C(=O)CNc3cccn4ccnc34)C2)C1 C1(NC(c2cc(C)sc2)=O)CC(C(=O)NC2C3CCC2CC3)C12CCC2 C(=O)(C(O)C(F)(F)F)N(CC(CN(C(c1cccc(OCC)c1)=O)C)O)C c1(Nc2c(NC(=O)OCC)ccc(C)n2)ccc(N2CCCC2)c(C#N)c1 c1(-c2nc(CC)nn2C)ccc(Cc2nc(C3CCC(=O)N3C)n[nH]2)nc1C c1(CNC2C(O)CC(CC=Cc3ccccc3)C2)ccc(I)c(Cl)c1 c1(C(=O)NC(C(C)NC(C(CCOC)C)=O)(C)C)ccc2[nH]c(=N)n(C)c2c1 N1(C(C(F)=CCC)=O)CC(NC(C2CC(C)(C)CO2)=O)CC1(C)C N1(C(C(C)C)=O)CCC(O)(C2CCN(C(C3CN4CCN3CC4C)=O)CC2)C1 Cn1ncc2c1CCCC2N=c1[nH]c(=NCC2CC(F)C2)[nH]c2c1CCCCC2 N1(C(c2nc(C(C)(C)C)oc2)=O)CC2CN(C(c3ccccc3Cl)C)CC2C1 C1(C(=O)NC(CCCCC)C)CC1C1CN(C(C2CC3CC2CC3O)=O)C1 c1(C(N2CC(CNC(c3ccnc(OC)n3)=O)C2)=O)n[nH]c2c1CC1CC21 N1(C(C=Cc2nc(C)c(C)[nH]2)=O)CC2CCN(C(=O)CC3(O)CCC3)CC12 c1(C(=O)NC(CC=C)CNC(=O)C(C)c2ccsn2)cc(C)c(F)cn1 C1(CNC(C(C)C2CC2)=O)CN(C(=O)CC2CCC(F)(F)CC2)CCC1(F)F Cc1cc(N2CCn3nncc3C2)nc(=NCCOCCOCCO)[nH]1 C1(OC)CCCCC1n1nnnc1N1CCCC(c2n[nH]cc2OC)C1 Cn1ccc2[nH]c(C(=O)NCCC3CCCN3C(c3cccn(O)c3=O)=O)cc12 c1(OCC)ccc(CC(N2CC(O)(CCNC(C3CC(C)OC3C)=O)C2)=O)cc1 C12(NC(c3cncc(C(C)(C)C)c3)=O)CCCC1CN(C(=O)CN1CCCC1)C2 C(C)(CCC(=O)NCCN(C)C(c1cc(OC)cnn1)=O)OC C1(CNC(C(CSC)O)=O)COC(C)(C)CN1C(c1ccc(OC(C)C)nc1)=O C1(NC(C2CC(C)(NC(=O)CCc3csnn3)C2)=O)CC2(CCC2)C1O O=C(C1=CCOC1)NCC(CNC(c1cscc1C1CC1)=O)CO c1(C(=O)NCCCN(CCCNC(C2CCC(O)C2)=O)C)[nH]nc2ncccc12 C(C(CC(=O)Nc1ccc(OC)nc1)OC)NC(c1cnc(CC)s1)=O N1(Cc2ccc(COC)cc2)CCC(=O)N(NC(=O)CC2(n3cccn3)CC2)C1 C1(NC(CN(C2CC2)CC)=O)CCCN(C(=O)CC2CCOC2=O)CCC1 c1(-c2c(C(=O)NC(C(C)(C)O)c3ccccc3)c[nH]n2)ccc(F)c(Cl)c1 C1(NC(Cc2c(C)con2)=O)CC2CCC(C1C)N2C(=O)CC1(C)CCCO1 C1(c2n(CC(=C)C)nnn2)(NC2CCN(C(N)=O)CC2)CCCOC1C(C)(C)C N1(C(C(=O)NCC)=O)CCC2CCC(C1)N2C(=O)Cn1nc(C)c(Cl)c1C Cc1c(CNc2cccc(C(=O)NC3(c4ccccc4Cl)CC3)c2)cccc1O N1(C(CNC(CC)=O)=O)CC2CC2C1C(=O)NCC1CCOC1 CN1CCCCC1CCC(N1CCOC(CNC(=O)CSc2ccncc2)C1)=O c1(C(N(CC(CC)NC(C2(n3nccn3)CC2)=O)C)=O)cc(C)nc(O)c1 C1(C(=O)NCc2c(C(N(CC(F)Cl)C)=O)con2)C2CC3C(C2=O)C13 c1(OC)cc(NC(C23CC2CN(C(C2(C)CCCN2)=O)C3)=O)cc(F)c1 Cc1nc(N)cnc1C(=O)NCC1CCN1C(=O)C=CC1CCC1 N1(C(C2CCN(Cc3ccc(C)o3)C2)=O)CCCC(O)(CC(N)=O)C1 c1(CC(=O)NC(CC=C)CNC(c2ncoc2C)=O)ccc2c(c1)OCCCO2 c1(SC)cncc(NC(C2CC(C)N2C(=O)CC2CCC(C)(C)C2)=O)c1 CN1CCN(C(=O)C(O)(c2ccccc2)C2CCCCC2)CC1 c1(C(=O)NCC2(OC)CCS(=O)(=O)C2)cc(Cl)c(Br)c(OC)c1N c1(CC)noc(C(=O)NCC2(NC(=O)C(N3CCSCC3)C)CCOC2)c1C N1(C(CCc2nc(=N)[nH][nH]2)=O)CCC2(CC2C(=O)NCCC(F)(F)Cl)C1 c1(N(C)C)ncccc1C(=O)NC(C)(C)CCNC(C1CCC(C(N)=O)C1)=O CCC(CC)C(C(=O)NC12CC1CN(C(C1(n3cccn3)CCC1)=O)C2)OC c1(OCCC)cccnc1C(=O)NC(C)CN(C)C(C1(CN(C)C)CCCC1)=O c1(C(=O)NCCCN(C(C(c2c(C)cccc2)C)=O)C)cncc(S(C)(=O)=O)c1 C(=O)(C1=CCN(C(C2(O)CCC2)=O)CC1)N(C)CCOCCCO C1(NC(CN(CCOC)C)=O)COC2(C1)CN(C(=O)C(C)(C)C(C)C)C2 N1(C(c2ccc(OC)nn2)=O)CCC2CCN(C(=O)CC3CS(=O)(=O)C3)CC12 c1(C(N(CCN(C(CC=CCC)=O)C(C)C)C)=O)cnn(C2CCC2)c1C c12ccc(c(C(=O)OC)c1)[nH]c2=O.N1(C(=O)NC)CCC(C)C(C(=O)OC)C1 Cc1cc(Cl)nc(N)c1C(=O)NCC(C)CNC(=O)CCc1cncs1 c1(OC)cc(NC(C2CC(C)CN(C(=O)Cn3nc(C)oc3=O)C2)=O)cc(F)c1 c1(CNC(C2SCCCS2)=O)cc(C(=O)NCc2ccncc2)n[nH]1 c1(C(=O)NCC2CC(OC)CN2C(C2COC2)=O)cn2cc(Cl)cc(Cl)c2n1 C1(N2C(=O)NC(c3c(OC)nc(Cl)cc3)C2=O)CCCC2(CCOC2)O1 c1(C(=O)NCC(CC)NC(c2cc(-c3cccs3)on2)=O)noc(C)c1CO CCC(C)C(C(=O)NC(Cc1ccco1)C(=O)NCC(CC)C(C)C)N(C)C N1(C(c2cc(C(C)C)nn2C)=O)CCCC2(CCN(C(=O)Cc3cc[nH]n3)C2)C1 C1(NC(CCC=C(C)C)c2nnnn2C2CCOCC2)COC(C)(C)C1 C(=O)(CC1OCc2ccccc21)NC(C)CNC(c1coc(CO)c1)=O c1(CC(=O)N(CCCNC(C(CCC)OCC)=O)C)c(C)cc(C)nc1O N1(C(=O)NC(c2ccccc2)C=C(C)C)CCC12CCCOC2 C1(C(=O)NC2C(NC(c3ccoc3)=O)COC2)CCCN(c2cc(O)ncn2)C1 C1(NC(C2C(C=C)C2)=O)CN(C(c2ncc(Cl)s2)=O)CCC12CCC2 N1(C(CC2(OC)CN(C(C3CCC(=O)C3)=O)C2)=O)CC(C)(C)CCC1CO CC1(NC(=O)C(N)CC2CC2(F)F)CCCCCC1 CC1CCCN(C(=O)C(=O)NC(C)C(=O)N(CCCN(C)C)C)C1 N1(C(CCCC#CC)=O)CCC2CN(C(=O)CCC3CCCO3)CC12 C1(C(=O)NCc2cc(C)ncn2)C(C2CC2)CCN1C(c1cc(C(N)=O)co1)=O C(=O)(C#CC1(C)COC1)NC1CCN(C(COCCCCCC)=O)CC1C c1(-c2cn(CC(C)C)nc2)cc(C(=O)N(CC(F)(F)F)C)c2nccn2c1 c1(C(=O)OCC(=CC(C)OC)C)cnn(-c2ccccc2F)c1N C(=O)(C1Cc2ccccc21)N1CC(C2(NC(c3scc(C(N)=O)c3)=O)CC2)C1 N1(C(CCN(CCC)C)=O)CC(O)CC1CNC(C1CCN(CC2CC2)CC1)=O CC(Cc1ccncc1)C(=O)NCCC(O)CNC(c1sccc1CO)=O Cc1cn(C)cc1C(=O)NC(C)(C)C=CC(=O)NCC1(O)CCN(C)C1 n1(C(C(=O)NC(C(C)C)C(=O)N(C2CCCCC2)C)C)c(=O)oc2ccccc12 C1(CNC(c2n(C)ncc2Cl)=O)CCCN(C(=O)CC2(C)CC2(Cl)Cl)CC1 c1(N(C)CC2N(C)CCC2)ccc(S(=O)(=O)NCc2nccc(=N)[nH]2)cn1 C(=O)(C(C)(C)CCCc1ccccc1)NCC(CNC(C1COC(=O)N1)=O)OC C1(CNC(C(N2CCNC2=O)C)=O)COCCN(C(=O)CCc2ccccc2)C1 Cc1ccc(F)c(CC(N2CCC(C(C)(C)NC(c3cc[nH]c(=N)n3)=O)C2)=O)c1 c1(C(=O)NCC23N(C(c4c(C)nccc4)=O)C(CC2)CC3)c(Cl)sc2nnsc12 C1(CC(=O)NCC(C2N(C(CN(C)C)=O)CCCC2)(C)C)CC2(CCC2)CCO1 n1(CC(N2CC(C(C)NC(=O)C(F)n3cccn3)C2)=O)nc2n(c1=O)CCOC2 c1(C(N2CCC(NC(c3cn(C(F)(F)F)cn3)=O)C2)=O)ccc(O)cc1F Cn1cc(C(=O)NCc2cc(C(=O)NCC3(O)CCCOC3)co2)n(C)c1=O C1(CNC(c2cc(C)[nH]n2)=O)CC(C)CN(C(=O)CN2CCOCC2)C1 C1(C)(C(=O)NC2C(C)CN(C(c3ncccc3CO)=O)C2)CCCCCC1 C(C)(C(C)C(=O)NC1C2CCCC12)NC(c1cc(OCC)n[nH]1)=O c1(CC)nc(C(=O)NCC(C(C)C)NC(c2cc(CC(C)C)on2)=O)co1 C1(O)(CNC(C2(CCN(C)C)CCCC2)=O)CCN(C(=O)CCc2ccoc2)C1 c1(C(=O)NC2CN(C(C(C)CC3CCCC3)=O)CC2C)ccc(P(C)(C)=O)cc1 C12(C(=O)NCC#CCNC(c3cn(CC(C)C)nc3)=O)CCCCC1CCC2 c1(C(=O)NCCC(CNC(C=C(C)C(C)C)=O)O)ccccc1SC(F)F C1(NC(CCNC(C)=O)=O)CN(C(C2CCN2C(C)(C)C)=O)CCC1(C)C c1(C(=O)NCC(CNC(=O)C=CC2CCCC2)OC)ccc(Br)cc1O CC1(CNC(c2cc(O)cc(O)n2)=O)CC(F)(F)CN1C(=O)CC1COC(=O)C1 C1(C#CC(=O)N2CCCC(CN(C(=O)C(F)(F)C(F)F)C)C2)(CC)CC1 N1(C(c2cccc(C)c2C)=O)CCCN(C(=O)CC(F)F)C(C)C1 C(C1c2ccccc2CN1C(c1cnc2[nH]cncc1-2)=O)NC(COCCC)=O C(=O)(C(CO)C(C)(C)C)NCC1CN(C(Cc2ccc(C)cc2)=O)C1 N1(C(c2ccc(Cl)c(Cl)c2)=O)CCOC2(CCN(C(C3(O)CCC3)=O)C2)C1 N1(C(CC2(CCC#C)OCCO2)=O)CCCCC1CNC(=O)CC1CC2CC2C1 C1(C(C)C)N(C(=O)CC2CCCN(C(=O)CN(C)C(N)=O)C2)CC12CCCC2 CC(C)(C)C(CNC(C1(C(N)=O)CC1)=O)NC(c1coc(-c2cccnc2)n1)=O C=C1CC(C(=O)NC(C)CNC(C2CCCN2Cc2ccccc2)=O)(C(F)F)C1 C12(C(=O)NCC(CCNC(c3c(COC)cccc3)=O)O)CCCCN1CCC2 O=C(N=c1ccn(C2CC2)[nH]1)C1CCCCCN1C(=O)Cc1cccc(F)c1 C(=O)(C1=CCCSC1)N1CCC(N2CCC(NC(C(CC)C#N)=O)CC2)C1 c1(C(=O)NCC2CC(NC(c3c(CC)noc3C)=O)C2)cccc(C=C(F)F)c1 Cc1cc(C(N2CC3CCC3(CCNC(c3cc(F)c[nH]3)=O)C2)=O)cc(O)n1 Cc1ccc(SCCC(=O)NCC2(c3cc[nH]n3)CC2)cc1 n1(C(C)C)cc(N(C(=O)CC2CCC(NC(=O)Cc3cccnc3)C2)C)cn1 c1(NCC(=O)NC2C3CCC2CN(C(=O)COC(F)F)C3)ccccc1[N+](=O)[O-] C1(C2CCN(C(c3ccc(Cl)c(C(F)(F)F)c3)=O)C2)(NC(C2C(C)(C)C2)=O)CC1 C(CN=C(NCC1CC1C1CCC1)N1CCCC(CN(C)C)C1)OCC=C N1(C(c2cnc(CC)[nH]2)=O)CCC2(CC1)CN(C(c1c(Cl)csc1Cl)=O)C2 N1(C(c2c(CCC)[nH]cc2)=O)CCCN(C(=O)CCF)CC1CO C1(C(=O)NCC(C)(C)C(=O)NCCCn2cnnn2)CCCC12CCC2 Cc1cc(CN2CCC(O)(C(=O)Nc3cc(Br)ncc3C)C2)ccc1O CC(C)C(O)CC(=O)NC1CC(OCC(=O)NCC23CCC(CC2)O3)C1 c1(C(=O)NC(CN(C(=O)C=NOC)CC)C)cc([N+](=O)[O-])c(N)cc1F Cc1nc(NC(C2CC3CC3N2C(=O)CCc2ccco2)=O)ccc1Cl N#Cc1cnc(C(=O)NCC2CCN(C(C3CCCCC3O)=O)C2)c(Cl)c1 c1(CNC(=NCC=C)NCCOCCN(C)C)nnc2c(=O)[nH]ccn12 N#Cc1ccc(F)c(C(=O)NCC2CCCCN(C(C34CSCC3C4)=O)C2)c1 C1(CCC(=O)NC(CC)CN(C)C(C2(CCN(C)C)CC2)=O)NC(=O)NC1=O N1(C(c2cc(C)[nH]n2)=O)CC2CCCCC2(CNC(=O)CCc2ccccc2)C1 N1(C(c2cc(CC)no2)=O)CCC2C(NC(=O)CCC(=O)N(CC)CC)C12 C1(CNC(C2(CCC)CC(=O)C2)=O)CCCN(C(=O)C=Cc2cncs2)CC1 N1(C(C2(OCC)CCCCC2)=O)CCC(C)C(NC(c2cccc(C)c2)=O)C1 c1(OC)ncnc(C)c1C(=O)NCC1CCN(C(C2C(F)(F)C23CC3)=O)C1(C)C C1(CNC(=O)COCCF)CN(C(c2cc(C(O)C(F)(F)F)ccn2)=O)CCO1 C(=O)(CCCCCF)N1CCC(N(C(C=CC(CC)C)=O)CCO)CC1 C12(NC(CC3(N(C(CCC(C)CN(C)C)=O)C)CC3)=O)CC1COC21CCC1 CC1CC(NC(c2nc(Cl)c(Cl)s2)=O)CCN1C(C1CNC(=O)N1)=O CS(=O)(=O)CCCC(=O)N1CCCC(CO)(NC(=O)CCN2CCCC2)C1 c1(OC)cc(C)c(C(N2CCC(C)S(=O)(=O)CC2)=O)cc1S(N)(=O)=O c1(C(=O)NCC2CCC(NC(C3CCCCC3F)=O)CC2)ccc2c(c1)OCC2 C(=O)(C(Cc1cnc[nH]1)NC(=O)C=Cc1ccco1)NC1C(C)(C)C1 C1(NC(C2CCN(C)C2=O)=O)CC2CC1CN(C(=O)C1=C(Cl)CCOC1)C2 C1(C(N(C)Cc2cc(CC(C)C)on2)=O)CCCN(c2cc(C=O)ccn2)CC1 c1(C(=O)NCC2(OC)CN(C(C3CC(C(C)C)C3)=O)C2)cnc(N)c(N)c1 CC1CN(C(=O)C(CC2CC2)NC(=O)CC2C(C)(C)C2(C)C)CCN1C1CC1 CC1(C)C(C(=O)NCC2CCCCC2)CCN1C(C1CC(F)(CF)C1)=O N1(C(C(c2cn(CC)nc2)=O)=O)CCN(C(c2cccc(F)c2Cl)=O)CCC1C Cc1cc(CCC(=O)NCC2CC2NC(c2c[nH]cc2C)=O)c(C)s1 N1(C(CC2(NC(CCCOCC=C)=O)CC2)=O)CCC(=O)N(C)CC1 N1(CC(=O)NCC2(C)CC(NC(c3c[nH]cc(Cl)c3=O)=O)C2)CCP(C)(=O)CC1 c1(C(=O)OC(C)(C)C)cccc(O)c1F.C12CC(C(CO)C1)NC(=O)C(=O)N2 C1(NC(CC)=O)CC2CC1CN(C(c1c[nH]c(C(N)=O)c1)=O)C2 C1(CCNC(C2CN(C)C2)=O)CCCCN1C(=O)Cn1cc(CO)nn1 C12(OC)CCN(C(=O)CC3(C)OCCO3)CC1C2 n1(C(CC)C)ncc(C(=O)NC2COCCC2NC(c2ccncc2O)=O)c1C C1(NC(CCC=C(C)C)=O)CCC2CCN(C(c3c(CO)n[nH]c3C)=O)C1C2 N1(C(c2cc3cccc(C)c3[nH]2)=O)CCCC(C2CN(C(=O)C(C)C(C)O)C2)C1 c1(C(=O)NCC2C(C)CN(C(C3(C(F)(F)F)CCC3)=O)C2)ccn2ccccc12 C1(NC(CC2(CSC)CC2)=O)(CO)CCCN(C(=O)C(F)(F)CC2CC2)C1 CC1(CNC(C2(NS(=O)(=O)C3CC3)CCCC2)=O)CC2(C1)CC(F)(F)C2 C(CC(CC)C(=O)NCCCNC(=O)C(C)NC(c1cc(F)cc(F)c1)=O)=CC C1(NC(C=CCOC)=O)CC12CCN(C(c1ccc(OC)cn1)=O)CC2 c1(OC)ccc(C(=O)NCCC(C)N(C(=O)CCCC2CCC2)C)cc1N Cc1cc(Cl)ccc1OCC(N1CCC(NC(=O)C2=CCC2)C(C(C)C)C1)=O CC(F)(F)CCC(=O)NCc1ccc(C(=O)NCc2nccn2C2CC2)o1 C=CCN=c1[nH]c(C(N2CC3(CCCC3NC(C3CC4CCC3C4)=O)C2)=O)cs1 c1(CN(C(=O)CCC2CCCN2C(c2ccoc2Cl)=O)C)cccc(F)c1 Cc1cnc(CNC(C2CC23CCN(C(=O)Cn2ncnn2)C3)=O)c(C)c1 c1(OC)ccc(OC)c(C(=O)NCC2C=CCN2C(c2csc(C(F)F)n2)=O)c1 N1(C(c2ncccc2Cl)=O)CCC2(CC1)CN(C(C1CC13CC3(F)F)=O)C2 c1(C(N2CCCN(C(c3c(C)ncc(F)c3)=O)CC2)=O)ccc2c(=N)[nH][nH]c2c1 C1(C(N2CCC(CC(=O)O)C2)=O)C2CN(CCC3CCS(=O)(=O)C3)CC12 C12(OC)CCC(C(=O)NC(C)(C)C(C)NC(c3ccc(Cl)cc3C)=O)(CC1)C2 c1(C(=O)NCC2CCC(NC(c3nc(CC)sc3)=O)C2)ccn2ccccc12 C(=O)(CC(C)CCC)NC1C(C(N(C2(C#C)CC2)C)=O)CCOC1 CC1CC(F)(F)CCN1C(C1(CCNC(=O)COCC2CCCC2)CCCC1)=O N1(C(c2cc(C)[nH]n2)=O)CC2CC1(c1cn(CC3CCC3)nn1)CO2.N1CCCC1 c1(C(=O)NC(C)CCC(=O)N(C)C(C2CCOCC2)C)cccc(F)c1N c1(CNc2cc(-c3scc(C)c3)ncc2)cccc(S(C)(=O)=O)n1 C1(OCC)CCN(C(=O)CCC2CCN(C(=O)C(C)N3CCCC3)C2)C1 C1(C(=O)OC)CC(NC(C2CC2CNC(C2CNC(=O)O2)=O)=O)CCO1 c1(C(N(C2CCC(NC(C3(OCC)CCC3)=O)C2)C)=O)ncccc1F C1(C(=O)NCC(c2ccco2)O)(CC)CCCCN1 O=C(C1=NOCC1)NC1CCCC(NC(c2cc(C(F)(F)F)ns2)=O)C1 C1(C)(CNC(CCOC)=O)COCCN(C(=O)CC2CN3CCC2CC3)C1 C(=O)(CC(C)(C)C(F)F)NCCC(CNC(c1ncc(C)cc1F)=O)O C1(CC(=O)N(CCC(=O)NCCCN(C)C)CC=C)C=NN(C)C1=O N1(C(c2ccc(C)[nH]2)=O)CC(C)CN(C(c2ccc3c(c2)COB3O)=O)CC1C Cc1ccc(C=CC(=O)NC2CCC(CCNC(=O)Cc3ccccc3)C2)s1 Cc1ccccc1N=c1[nH]c(COC(=O)CC2CCc3ccccc32)nc(=N)[nH]1 C1(NC(CN(C2CCSC2)C)=O)C=CCN(C(C2CCS(=O)CC2)=O)C1 C1(CC)(CO)CCCN1CC(C)Cc1nn[nH]n1 C(=O)(C(C)(O)C(C)(C)C)N1CCC(n2cc(CC(COC)O)nn2)CC1 O=C(C1=NOC2(CCC2)C1)NC1CCCC1CNC(C1CC(F)(CO)C1)=O C1(NC(CCC#C)=O)CCN(C2CCN(C(C3(CC(C)C)CCC3)=O)C2)CC1 c1(C(N2CCC(NC(C(CC)CC)=O)C2)=O)cc(=O)oc2ccc(O)cc12 N1(C(C2(C)CCCCCC2)=O)C2CCC1C1CC1(NC(=O)CC1(CO)CC1)C2 c1(OC)cc(C(=O)NC(C)C(C)NC(C23CC(C)(CCO2)C3)=O)cnc1O CN1CCC(C(N2CC(C(N)=O)(CNC(c3n[nH]c(C(C)(C)C)n3)=O)C2)=O)C1=O Cn1ccc2cc(C(N3CC4CC(C3)N4C(c3cc(O)ccc3Cl)=O)=O)ccc12 c1(C(=O)NC(CNC(C(COC)N(C)C)=O)C)cc(Cl)nnc1O N1(C(Cc2cc(C)[nH]n2)=O)CC2CCCC(NC(=O)CN3CSCCSC3)C2C1 C1(NC(c2ncc(C)c(Br)c2)=O)CN(C(C2(F)CCC2)=O)C2(CCCC2)C1 C1(C(=O)NCC(C)CC(=O)NCC2CC2C2CCC2)CC2(CCO1)CC2 C(C1=CCCOC1)NC(=O)CCC1(NC(C2CN(C3COC3)C2)=O)CCC1 c1(CC)c(C(=O)NCC2(O)CCN(C(C3CC4CCC3CC4)=O)C2)cccc1F S(=O)(=O)(c1cnn2ccc(N3Cc4ccccc4C(C)(C)C3)nc12)NCC(C)O c1(C(=O)OC)c(C)[nH]c(C(=O)C(C)OC(=O)CC23COC(CF)(C2)C3)c1C C(=O)(C1=COCCC1)NCCNC(=O)Nc1n(C(=O)OCC)ncc1 N1(C(C(CO)NC(C(C)C)=O)=O)CCC2CN(C(C3CN4CCN3CC4)=O)C2C1 n1(CC(=O)NC2CCC(NC(C3(C(F)(F)F)CCCCC3)=O)C2)cnccc1=O C1(CC(=O)NC2CCN(C(CC(C)F)=O)CC2)CCc2ncc(Br)n2C1 CC1=NOC(C(=O)N(C2CCN(C(=O)Cc3csc(-c4ccco4)n3)C2)C)C1C C(C(C)(O)C(C)(C)C)NC(C1(n2cc(CCCC(C)=O)nn2)CC1)=O C(C)(CNC(=O)C(CO)NC(N)=O)(C(C)C)NC(Cc1cc(C)on1)=O O=C1COC(NC2CCC2)=C1C(=O)N1CC(c2ccccc2Br)(O)C1 C(=O)(C(CC(C)C)NC(=O)CC(F)(F)F)N(CCN(C(CC(=O)OCC)=O)C)C N1(C(C)=O)CCCC(C2CN(Cc3ccc(Br)c(C(F)(F)F)c3)C2)C1 C=CCC(CNC(=O)CC1COCCO1)NC(C1(COC)CCC1)=O C(CN1C(=O)C(C)Oc2ccccc21)NC(C(c1cn(CC)nc1)=O)=O Cc1cccc(N)c1C(N1CCCC(NC(c2c(Br)cnn2C)=O)C1)=O C#Cc1c[nH]nc1C(=O)NC1CC1CNC(=O)C(C)(C)SC N1(C(C(C=C)CC)=O)CC(C)CN(C(=O)CCCc2nncn2C)CC1C N1(C(c2c(C(=O)OC)cccc2)=O)CCC(F)(F)C(CNC(=O)C(C)N(C)C)C1 C(=O)(C(CC)C(C)O)N(CC(C)NC(CC(CC)O)=O)C C=Cc1cnn(C)c1C(=O)NCCCCC(C)NC(=O)CCCOCCC c1(C(=O)NC2CN(C(c3cnc(N(C)C)s3)=O)CC2C(F)F)ccc(F)c(N)c1 c1(C(N2CCN(Cc3nnn(C)n3)CC2)C(=O)NCCSC)cc(C)cc(C)c1 C1(C(CNC(C(C)OCC)=O)(C)C)CCN(C(=O)C(F)=C2CCCC2)CC1 C(=O)(C(C(F)(F)F)C(F)(F)F)NC1CC(NC(CNC(c2cc(C)nn2C)=O)=O)C1 C(=O)(C(CC(C)C)NC(c1csc(CNC(=O)CCn2ccc(C)n2)c1)=O)NC N1(C(c2nc(CC)oc2C)=O)CCCN(CCNC(=O)Cc2csc(S)n2)CC1 c1(NCCC(=O)NC)[nH]c(=NC2COC3(CCCC3)C2)nc2c1ncn2C(C)C C1CC(=O)N(C2CCS(=O)(=O)C2)C1.c1nccs1.C(CN1CCNC1=O)OC C12(CNC(c3c(C)nns3)=O)COC(CNC(c3cc(C(C)(C)C)n[nH]3)=O)(C1)C2 Cc1nccn1C(C)C(=O)N(C(C)C(=O)NCCCC(F)F)C C1(NC(=O)CCn2cnnn2)CC(NC(=O)Cn2cnnn2)C12CCC2 C=CC1CN(C(C2CN(C(=O)CCC#CC)CCN2C)=O)CC1O C1(NC(CCC#C)=O)CCC2(CC1)CC(NC(=O)C(C)C(F)(F)C(F)F)C2 c1(C(=O)NC(C)CN(C(=O)CSC(F)(F)F)C)cc2c(F)cc(F)cc2o1 N1(C(C(C)NC(C)=O)=O)CCC2(CC1)COC(CNC(c1[nH]ccc1C)=O)C2 C12(C(=O)NC3CCN(C(C(C=CCCC)O)=O)CC3)CCC(C(F)F)(CC1)CC2 C12(CNC(N(c3ccc(C(F)(F)F)cn3)C)=O)CC=CCN1CCC2 c1(C(N2CC(NC(CCC(C)(F)F)=O)C2)=O)cc(C(F)(F)F)ncc1[N+](=O)[O-] c1(C(=O)NC2CN(C(C=C(C)c3cccs3)=O)C3C2C3)c(C)cccc1F c1(N2CCC(CNC(C3(C)CCC(C)C3)=O)CC2)ncccc1C#N C1(NC(=O)Cn2ccccc2=O)CCCC12CN(C(C1CC=CC1)=O)C2 c1(C(N(CC(C)NC(CC(C(C)C)OCC)=O)C)=O)cnc2ccncc2c1 C=C1CCC(C(=O)NC2COCCC2NC(=O)C(C)NC(c2ccoc2)=O)CC1 c1(C(N2CC(NC(C(CC)C3CCOCC3)=O)C2)=O)[nH]c(O)nc1C N1(C(CCc2ccc(=N)[nH]c2)=O)CCCCC(CNC(c2nc(Cl)c(Cl)s2)=O)C1 CCC1=NOC(CC(=O)NCC(CNC(=O)CCc2ccc(Cl)cc2)CO)C1 C1(C(=O)NCCC2CCSC2)CC2(CCC2)CN1C(=O)C(O)C(F)(F)F c1(C(N2C3C(NC(C4(SCC)CC4)=O)CC(C3)C2)=O)nccc2c(F)cccc12 c1(C(=O)OC)ccc(S(=O)(=O)N2CCC(NS(=O)(=O)CCc3ccccc3)C2)n1C N1(C(C=NOC)=O)CCC2(NC(C3CCN(C4CC4)CC3)=O)CCCCCC12 C1(CNC(C2(OC)CCCOC2)=O)CN(C(C2CSCC(=O)N2)=O)CCC1C C1(F)(CNC(C2C(CC)C2)=O)CCN(C(c2c(Cl)nsc2Cl)=O)CC1 CC(C)(CCCC(=O)NC1CC1F)NC(C1CC(C2CC2)=NO1)=O O(S(=O)(=O)c1ccc2nc(Cl)ccc2c1)c1ccc(CC(=O)OC)c(Cl)c1 C=CCC(Cc1ccccc1)C(=O)NCC(C1CC1)NC(C1(CO)CCCC1)=O Cc1cc(NCC2CC(F)(F)CO2)ncc1S(=O)(=O)NC(C)(C)C(C)O c1(Cn2c(C(C3CCOC3)Nc3cn(COC)nc3)nnn2)ccc(OC)cc1 C1(O)(CS(=O)CC2CCCN(c3ccccc3Cl)C2)CCOCC1 c1(OC)ccccc1CNC(C1C(C)CCN1C(=O)C=CCN1CCCC1)=O C1(O)(CCNC(C(C)OCC(C)C)=O)CCN(C(=O)CN2C(=O)CNC2=O)CC1 c1(CNC2C(CC)CCCC2)cc(C)c2nccn2c1 C(C(CC(F)(F)F)NC(=O)C(C)NS(C)(=O)=O)NC(CC1(OCC)CC1)=O N1(C(C2C(C)CCOC2)=O)CCCN(C(=O)CSc2nccn2C)CC1 c1(CC(=O)NC2CCN(C(c3c(CC)[nH]cc3)=O)CC2)ccc(C)c(Cl)c1 c1(C(N(C2CCN(C(=O)Cc3csc(CC)n3)C2)CCC)=O)ncccc1N c1(OC)ccc(-c2cnccc2CN2CCCC2c2cccc(Br)c2)c(F)c1 c1(NCC2(NC(C3C(COC)C3)=O)CCCC2)cc2nnc(C(C)(C)C)n2cn1 CCCCC(C)CCC(=O)N1CC(NC(c2cnn3c2CCCC3)=O)C(OC)C1 N1(CCCNC(c2cnc(Cl)[nH]2)=O)CCN(C(C2CCOC2C(F)(F)F)=O)CC1 c1(C(=O)NCC(CC)NC(=O)C#CC(C)C)cc(S(N)(=O)=O)ccc1O CCCC(C(O)C(=O)N1C2CCC1(CO)CC2)NC(c1nnn(C)c1CC)=O N1(C(c2nc(CC)oc2)=O)CCCN(C(C2CCCN2C(C)C)=O)C(C)C1 CC1CCCCC1C(N1CCN(C(C)CNC(=O)C(F)F)CC1)=O C(=O)(C1=CCCCC1)NC1CC(C)(NC(CC2(C)CC2)=O)C1 C(=O)(C1=C(C)CCCC1)N1C(CO)CC(NC(c2ccc(OC)cc2C)=O)C1 N1(C(c2c(C)ocn2)=O)CC(F)CC1C(=O)NC(c1cccnc1)CO c1(C(N2CCN(CC(=O)NC(C#C)C(C)(C)C)CC2)=O)cccc(F)c1F CC(CC(C)NC(=O)C=Cc1cn[nH]c1)NC(=O)C(C)(C)Nc1ccccc1 c1(C(N2CC(CNC(CN3CCC(OC)C3)=O)C(C)C2)=O)ccc2c(c1)CCO2 CC1CCN(C(c2cnnc(O)c2)=O)CC1NC(C1(CN(C)C)CC1)=O c1(C(=O)NC2CCCC(NC(CCCC=C)=O)CC2)cc(C)cc([N+](=O)[O-])c1 c1(C(CN2CC3C(CC)(C3)C2)=O)cc2cc(F)c(F)cc2[nH]1 C1(C(=O)NCCC2(NC(CCCC(N)=O)=O)CCC2)Cc2ccc(F)cc2O1 N1(C(CC(=C=C)C)=O)CC2(CNC(C3(C4CCCCO4)CC3)=O)CC1CO2 N1(C(C(C)NC(C)=O)=O)CCCC12CCN(S(=O)(=O)c1cc(Cl)ccc1Cl)CC2 CC(C(C)(C)C(=O)NOCC(C)(C)O)NC(C1CCCN1C1CC1)=O CC(C)C(O)CC(=O)NC1CN(C(c2ccnn2CCN(C)C)=O)CC1C c1(C(=O)NC(CCC)CCCNC(=O)C(F)n2cccn2)cc(F)c(F)cc1O c1(C(=O)NCC(C)(CO)NC(c2n[nH]c(C)c2O)=O)cc2n(n1)CCN(C)C2 C(C)(C(C(C)C)NC(=O)C=Cc1ccn(C)c1)NC(CNC(=O)NC)=O c1(C(=O)NC(CNC(C(CC)N(C)C)=O)(CC)CC)ccc(OC)c(N)n1 C(CCN=c1[nH]nco1)OCC(C)C.c12cccc(n1)C(=O)N2 Cc1cn(C)cc1C(=O)NC(C)(C)CNC(=O)C(c1ccc(CC(C)C)cc1)C C1(C)(CC(=O)NC2(C(C)Cn3cncn3)CC2)CCN(C(=O)Cc2ccccn2)C1 Cc1noc(Cl)c1CC(=O)NC(C)C(C(C)C)NC(=O)C=Cc1ncco1 Cc1ccc(C2(C(=O)NCC(C)NC(=O)CCC(C)(C)C)CC2)cc1Cl c1(C(C(=O)NCC=C)N(CC(c2cccc(C)c2)(C)C)C)ccc(OC)cc1 c1(C(N2CCC(O)(CNC(C3CC34CC4)=O)C2)=O)cc2c(s1)CCCCCC2 S(=O)(=O)(c1cc(C(=O)NC2CCN(C(c3ccc([N+](=O)[O-])cc3)=O)C2)co1)NC C12(CNC(CN(C3CC3)CC)=O)CC(CN1c1ncns1)C2 c1(COC)n[nH]c(CNC(C2(Nc3ccccc3)CCC2)=O)n1 c1(C(=O)NCCn2cc(C(=O)NCC3(OC)CC3)nn2)cc(C)n(C)n1 C(C)(CO)(C(=O)NCc1cc[nH]c1C(=O)N(C)CCc1ccncc1)OC C1(CNC(C(C)O)=O)(CNC(=O)C(C2CCCCC2)N(C)C)CC=CC1 c1(C(=O)NC2CC3CN(C(C4CCCC(OC)C4)=O)CC32)ccc2c(c1)COC2 CC(C)C(O)CC(=O)N1CC=CC1CNC(=O)C(C)(C)Sc1ccc(Cl)cc1 c1(C(=O)NC(C2CN(C(C3(C)CCCC3)=O)C2)C)cc(N2CCCC2)ncn1 c1(C(N2C(C(=O)Nc3cn(C)nc3)CC(F)C2)=O)cc2cc(Br)ccn2n1 C1(C(=O)NCC=CCOC)C2CC3C(C2NC(C2CC2C(N)=O)=O)C13 c1(SC)cccc(C(=O)NCC(C)N(C)C(C2CCC(C(C)(C)O)CC2)=O)c1 c1(CC)ccccc1CC(=O)N(C1CCCCC1NC(C1(C)CC1)=O)C c1(C=O)ccc(CO)c([N+](=O)[O-])c1.CC(C)(CO)C(=O)OCc1csc(C)n1 c1(C(N2CCN(C(C=CCOC)=O)CC2C)=O)ccc(S(N)(=O)=O)cc1Cl Cc1ccc(F)c(C(=O)NC2C3CC2N(C(c2cc(C4CCC4)nn2C)=O)C3)n1 Cc1cc(C(N2CCN(C(c3ccncc3Cl)=O)C(CF)C2)=O)c(C)n1C C12(NC(=O)Cc3cc[nH]n3)COC(C1)C(NC(c1cnc(C3CC3)s1)=O)C2 S(=O)(=O)(c1ccc(F)cc1)N1C(CNC(c2cc(Br)cs2)=O)COCC1 c1(Nc2c(NC(=O)NC3C(OC)CC3)cccc2)cccc([N+](=O)[O-])c1 N1(C(C(C=C)C)=O)CC2(CCCC2CC(N2CCn3nccc3C2)=O)C1 C1(C(N(C)Cc2nncs2)=O)CN(C(c2ccn(C(F)F)n2)=O)CC12CC2 Cc1cc(Br)c(F)cc1NC(=O)NC(CC1CCCO1)C(F)(F)F C1(OC(C)(C)C)CC(F)CN(c2nnc(-c3ccc(Br)s3)n2CC2CC2)C1 n1(CC)cc(C(O)CNC(=O)C(=O)N(C)C2CC2)cn1 c1(OC(C)C)ccc(Cl)cc1C(=O)NCC(C)(O)CNC(=O)CCCCC#N C1(O)(CNC(CC2(N(C)C)CC2)=O)CCCN(C(=O)CCc2cnco2)CC1 N1(C(CCCC#C)=O)CC(C)CN(C(=O)Cc2nccs2)CC1C Cc1cc(C)n(CC(N2CC3C(NC(=O)C(C(C)C)N(C)C)C3C2)=O)c(=O)n1 C(=O)(C1CCCc2cncn21)N1CC2(CCN(C(CC(C=C)CC)=O)C2)C1 S(=O)(=O)(c1ccc(C#N)c(NCc2nc(Cl)cs2)c1)N1CCCC(C=C)C1 CC(CN=c1nc2scnc2c(NCC(C)(F)F)[nH]1)C(C)(F)F N1(C(C2(c3ccccc3)CCN(C)C2)=O)CCN(C(=O)CC2(C)CC2)C(CO)C1 Cc1ccnc(C(=O)NC2(CCNC(=O)CC(C)(C)C3CC3)CCCC2)c1F C(=O)(CCC1=NNC(=O)CC1)N(C)CC1(C)CCCCN1C(=O)OC(C)(C)C CC(C)(C)C(=O)C(=O)NC1CN(C(c2c(O)cccc2F)=O)CCC1C(F)(F)F Cn1ncc2ccc(C(N3CC(NC(=O)C=CBr)C4CCCC34)=O)cc12 c1(CNc2cc(NC(C3CCCOC3)CC)ncn2)cc(F)ccc1F C1(O)(CNC(=O)C(O)C2CCC2)CCN(C(C2CC2(Br)Br)=O)CC1 Nc1ncc(C(N2CCCC2CNC(c2ns[nH]c2=O)=O)=O)cc1CO C1(CCNC(=O)NC2CC2)CN(C(C2CCC3CC2C3)=O)CCCO1 C1(NC(=O)C=C2CCC2)CCCN(C(c2ccncc2)=O)CC1F C1(CN(C)C(C2CCC(O)C2)=O)CCCN1C(=O)CN1CC(F)(F)C1 C1(C(=O)NC2CCN(C)C(=O)C2)C(C2CC2)CCN1C(=O)CCC(N)=O C1(C(N(CCCN(CC)Cc2cnc[nH]2)C)=O)CCC1(CSCC)OCC Cc1sc(N)c(C(=O)NC2CCC2NC(=O)C=Cc2cccs2)c1C c1(C(=O)NCc2c(CCNC(c3n(C)cnc3)=O)ocn2)ccc([N+](=O)[O-])cc1 N1(CC(=O)N(CC(N)=O)C)CCC(N2CC=CC2)C1 c1(C(=O)NCc2cc(O)ns2)ccc2c(=O)cc[nH]c2c1 c1(-c2noc(C)c2C(N2CCC(=O)NC2=O)=O)cccc(S(C)(=O)=O)c1 C1(CN(C(=O)CS(N)(=O)=O)C)CCCN(C(C2CCS(=O)(=O)C2)=O)C1 C(=O)(CCCC(F)F)N1CC(NC(C2(C)C=CCC2)=O)C(n2cccn2)C1 C1(CNC(C(CC)(C)OC)=O)Cc2ccccc2CN1C(C1CC(SC)C1)=O N1(C(C(C)NC(C)=O)=O)CC=CC1C(N1CC(CN=[N+]=[N-])C1)=O C(=O)(C1=NNC(=O)CC1)NC(C1CCCN1C(c1cccnc1)=O)(C)C c1(OC)ccc(C(=O)NC2(CCCNC(=O)C(F)CC(C)C)CC2)c(O)c1 c1(NCC2C(C(F)(F)F)CN(C(C(CC)OC)=O)C2)nc(Cl)nc(CC)c1C#N C(=O)(CCC(F)(F)CN=[N+]=[N-])N1CCN(C(CC(COC)C)=O)CC1.C1(=O)CN1 C12(C(=O)NCCC(C)NC(C3C4CCC3CC4)=O)CCCC1CC(=O)C2 CC(CCCNC(=O)CC1(O)CCCC1)NC(C1(C2CC2)CCCO1)=O CCCC(CCCO)C(=O)NCCOC1CN(C(C2CCCCC2(C)C)=O)C1 N1(C(CC(C)F)=O)CCN(C(c2cccnc2O)=O)CC1c1ccccc1 CCCS(=O)(=O)C(C)C(=O)NCC1CC2(CC2)CN1C(=O)CNC(=O)CN(C)C C12(CCNC(=O)CC3CSC3)CCC1CN(C(c1ccncn1)=O)C2 CC1(C)CC(NC(C2(C)CCCN(C(C3CC(=O)CCO3)=O)C2)=O)CCO1 N1(C(CCOCCN(C(c2c(CC)cco2)=O)C)=O)CCS(=O)C(C)C1 CC#Cc1cncc(-c2csc(-c3nccn3C3CCCC(C)C3)c2)c1 C#CC1CN(C(=O)CC2CCCCC2)CCN1C(c1cc2nccnc2[nH]1)=O n1(CCCC)cc(C(=O)NCC2CC2NC(=O)COCC2(F)CC2)nn1 c1(C(N2C(Cn3cc(C(COC)(C)O)nn3)CCCC2)=O)c[nH]nc1S(N)(=O)=O N1(C(C(CCCC)C)=O)CCC2(CC1)CC(C(=O)Nc1cc(Cl)nc(C)n1)CO2 c1(C(N(CCCCNC(c2ccncc2)=O)C)=O)cccc2c1CCC2 C1(CC)(CC)CN(c2cc(NCc3c(Br)nnn3C)ncn2)CCS1=O c1(C(N2C3CN(C(C4(C)CCN(C)C4)=O)C(C3)C2)=O)nccc2ccccc12 c1(C(=O)NCCN(C(C2CCC(C)(CC)O2)=O)C)cc(C)c(C)nc1C c1(CC(=O)N(CCCNC(=O)CC2C=CCCC2)C2CC2)ccc2nn[nH]c2c1 N1(CC(=O)N(C(c2ccccc2)C)C)CCC(NC(=O)CC2CC2C)CC1C c1(C(=O)NC2(CNC(C3(C)CC3(Cl)Cl)=O)CC2)nn(C(F)F)cc1Cl N1(C(C(CC)NC(N)=O)=O)CC2(CCN2C(C2CCCC2C(F)(F)F)=O)C1 c1(N2CCC(CC=C)(NC(c3cc(OC)ns3)=O)CC2)ncc(C#N)cc1F Cn1ccc2cc(CN(c3nc(C)ncc3Br)C3CCCCNC3)ccc12 N1(C(CC(=O)OCC)=O)CC2C(CNC(c3cccnc3CO)=O)C2C1 n12cc(nn1)CN(C(c1coc(C3CCC3)n1)=O)C21CC1.C1(C)CCOCC1 c1(OC)ccc(F)cc1C(=O)CSC1(O)CCN(c2nc(CO)cc(C)n2)CC1 N1(C(CC(C(F)F)NC(C2(CC=C)CC=CC2)=O)=O)CCOCC(C)(F)C1 c1(C(=O)NC2CC(NC(c3cc(Cl)c(Br)[nH]3)=O)C2)cccc2c1CCOC2 CC(C)(Cn1cc(CC2CCCC2)nn1)CC(F)F c1(C(N(CCN(C(=O)CC(C)F)CC)CC)=O)ccc(O)c(C(C)C)c1 CCC(C)(CO)C(=O)N(CCCN(C)C(c1ccsc1C(F)F)=O)C CC1(Br)CC1C(=O)NCCCN(C(=O)CSc1cccs1)C1CC1 C(=O)(CCCC(F)F)N1C(C2(NC(=O)CCc3cnccn3)CC2)CCC1 C(=O)(CC1OCCc2sccc21)NC1(C)CN(C(CSc2c(C)cccc2)=O)C1 c1(C(=O)NCC2(O)CCN(C(C(CCSC)N(C)C)=O)C2)cc(F)c(C)cc1F c1(C(=O)NCC2CN(C(CC(=C=C)C)=O)CC2C(F)(F)F)cnc(C)nc1OC C1(C(=O)NCC(CC)NC(C2CN3CCC2CC3)=O)CC1C1CCCC1 c1(C(N(C2C(C)CN(C(C3CCCCC3)=O)CC2)C)=O)ncc2n1CCCC2 C1(NC(C(C)Oc2ccccn2)=O)CC2CCC(C1C)N2C(C1SCCS1)=O C1(C)(CNC(CC2C(C)(C)CC2)=O)CCN(C(c2c[nH]nc2C2CCCO2)=O)C1 C(CS(=O)(=O)CC(=O)NC(C(N1CCC(OCCO)C1)=O)C1CC1)OC c1(C(=O)NC2CC(C)(NC(C(n3cc(Cl)cn3)C)=O)C2)ccc2snnc2c1 C1(C)(CC)C=C(C(=O)N2CCCC(NC(C3CCCO3)=O)C2C)C1 c1(C2CCN(C(=O)Nc3c(CN(C)C)cccc3)CC2)nnc2cnccn12 CCCCCCCC(=O)N1CCCC(C)(CNC(=O)CC2(C)CC2(F)F)C1 C1(C(=O)OC)CC2(CCCC2)CCN1C(=O)Cc1ccc(OC)cc1OC C(CCC(=O)N1CC(O)(CN(C(=O)COC2CCOCC2)C)C1)OCCOC C1(F)(CNC(c2ccccc2Oc2nccs2)=O)CCCN(C(=O)CC2CCN(C)C2)C1 C(N=c1[nH]c(-c2ccccc2)nc(=NCC=C(Cl)Cl)[nH]1)C1CC2S(=O)(=O)C(CC2)C1 N1(C(C2N(CC)CCC2)=O)CC(CO)C2(C1)CN(C(c1cc(C(C)=O)c[nH]1)=O)C2 c1(C(N2CCC(C)(NC(C(C)SCC)=O)C2)=O)cc(C)c(C)c(F)c1 c1(C(=O)NCC(C)N(C(C2CC2(C)C)=O)CC)ccc2cccc(OC)c2n1 C1(NC(CCN(C)CC)=O)CC2(C1)CC2NC(C1C(C#N)C1(C)C)=O c1(OC)ccc2c(n1)NC(C(=O)NC1CCCCN(C(C3CC=CCC3)=O)C1)C2 C1(C(=O)NC(c2nc(C)[nH]n2)C)CCN(C(c2ccc(CC#N)cc2)=O)C12CC2 C1(C(=O)NCC(COC)NC(c2n[nH]cc2Cl)=O)CCC(OC)CC1 N1(C(c2c(C)noc2)=O)CCC(C2CC2)(CNC(=O)C=Cc2cnccn2)C1 n1(CCCN)cc(C)ccc1=O.CSC CC1CCC(NC(C2CN3CCC2CC3)=O)CN1C(c1ccc(CO)nc1)=O C1(C)(NC(CC2(CNC(c3c(C)ccc(O)c3)=O)CC2)=O)CC(C)(C)OC1=O C1(CNC(CSCCCC)=O)(NC(c2ccn(C(C)(C)C)c2)=O)CCCCCC1 c1(C(=O)NC2CCCN(C(C3C=CCCC3)=O)C2)nccc2c(Cl)cccc12 Cc1cc(C(=O)NC2CCCC(C(N3CCCC(OC4CC4)C3)=O)C2)cn1C c1(C(=O)NC(C(=O)N(CCC(=O)OCC)C)Cn2ccnn2)ccccc1O c1(COC(C2CC3CC(N(C)C)C3C2)=O)c(-c2ccc(F)cc2)cc(F)cc1F C1(C)(C(=O)NCC(=O)N(CCCOCCOC2CC2)C)CCCO1.C1C(=O)O1 Cc1ccc(C2(C(=O)NC3CCN(C(=O)CCC4CC4)C3C(C)C)CC2)c(F)c1 n1(CCC(=O)NC(CNC(C2N(C)CCC2)=O)C2CCC2)ccc2ccccc12 c1(C(=O)NCC(CNC(c2cc(O)nc(C3CC3)n2)=O)O)cnc2ncccn12 N1(C(c2scc(CNC(CNC(N)=O)=O)c2)=O)CCC2(CCOCC2)C1 C1(CNC(CNC(C)=O)=O)CCCN(C(c2cccc(C3CNC(=O)C3)c2)=O)C1 C12(C(N3CC(CCNC(CC4CCC(C)CC4)=O)C3)=O)CCC(C(F)F)(CC1)C2 c1(SCC)cc(C(=O)NC2(C)CC(NC(c3sccc3OC)=O)C2)ccn1 N1(C(c2c(OC)con2)=O)CCC(c2ncncn2)CC1 C1(CNC(=O)COc2ccsn2)(CO)CCN(C(c2cc[n+]([O-])cc2)=O)C1 CC1(C)CCN(C(=O)C=C(C2CC2)C2CC2)CC1C(N1CC(c2nn[nH]n2)C1)=O C(CCCCO)(C(=O)NCC(N1CCOCC1)O)NC(=O)CN1CCCCC1 C1(CN(CC)Cc2ccccc2)CCCN(C(=O)CC2CC(O)C2(C)C)C1 c1(C(C)C)nc(CC(=O)N(C(C)CNC(c2ncoc2C2CCCO2)=O)C)cs1 N1(Cc2c(OCC)cccc2)CCCC(F)(CNC(c2coc(C(C)C)n2)=O)C1 N1(CCC)CC(NC(N2CCC(CCc3ccccc3)CC2)=O)CC1=O c1(NC(CCC2(C)CN(C(C3CC4(CCCO4)C3)=O)C2)=O)cccc2c1OCC2 C(=O)(C(C(C)C)n1ccnc1)N(C1CCCN(C(C2CCC(CO)CC2)=O)C1)C N1(C(CCNC(C)=O)=O)CCCC(C(C)NC(c2csc(-c3ccco3)n2)=O)C1 C(=O)(CCCCCC#N)N1CCC(NC(c2cnc(N(C)C)s2)=O)CC1 c1(OC(C)C)ccc(C(=O)NCC(C)(O)CNC(=O)C(C)(C)C2CCCO2)cn1 c1(C(=O)NC(C)CCN(C(=O)C(F)=C2CCC2)C)cc(F)c(F)c(F)c1F C(CCC(C)(C)C(=O)NCC(=O)OC(C)C)NC(C1OCCC(C)C1)=O Cc1nccc(C(N2CCOCC2CN(C(=O)CSc2cn[nH]c2)C)=O)c1O CCCCC(C)C(=O)NCc1nocc1C(=O)NC1CC1CN(C)C C1(C(=O)NC(C(=O)OC)C2CCC2)CC2(CCN(C(C3CNC(=O)N3)=O)C2)C1 c1(OCCC(=O)N(CC(C)NC(C2CC2(C)C)=O)C)cc(F)ccc1F c1(C(N(CC(C)N(C(C2CN(CCC)C(=O)C2)=O)C)C)=O)cnc2n1CCOC2 c1(CNC(CC#N)=O)cc(C(=O)Nc2cncc(Br)c2)ccn1 C1(NC(C(=O)NC(C)C)=O)CC2CC(NC(C3(NCC(F)(F)F)CC3)=O)CC12 C1(C(C)NCCCOCCOC)CCN(c2nccs2)CC1 Cc1cccc([N+](=O)[O-])c1C(=O)NCC(O)CNC(=O)C(c1ccccc1Cl)O C1(CCC)CN(C(C)Cc2cn[nH]c2)CCN1C(=O)NCCC CC(C)CC(C)CC(=O)N1CC=CC(NC(c2cc(O)nc(N(C)C)n2)=O)C1 C1(C(=O)NCCCN2C(=O)C=CC2=O)CC12CN(C(=O)C=CC1CCCC1)C2 C(C)(CCCNC(C1CCC(Oc2cccnc2)C1)=O)NC(C1CC(OC)C1)=O C(C(=O)NCC(F)F)(C1=NOC2CC12)N1CCCC(OC(C)=O)C1 c1(C(=O)NC2CCC(CNC(C3(n4cccn4)CC3)=O)C2)ccn2ccnc2c1 C1(CNC(c2ccc(CCC)s2)=O)CCCCC1NC(c1cnc(C)nc1)=O C1(CNC(C2N(C(CNC(=O)OCC=C)=O)CC2)=O)CC1[N+](=O)[O-] c1(N(CCC)C(C2CC(F)CN2CC(O)CC)=O)ccc(CC)cc1 CC1CCCC(C2=NOC(C(=O)Nc3c([N+](=O)[O-])ccc(F)c3F)C2)C1 C=CC(CC)C(=O)N(C)Cc1cccc(C(C)(C)C)c1 N1(C(C(C)n2cccn2)=O)CCC(C)(C)C(C(=O)NCc2cnns2)C1 c1(CC)nn(C)cc1NC(=O)CC1(CNC(=O)CC2CCC(=O)N2C)CC1 c1(C(=O)NC(c2ccco2)C)cnn(CCO)c1.C12CC(C1)N2 c1(CC(=O)NCCC(C)(C)NC(C2C(C#C)C2)=O)coc2cc(CC)ccc12 CC1CCCC1(C)NC(c1c(CNC(c2cc(Cl)cn2C)=O)cnn1C)=O N1(C(C2(C(C)NC(=O)CNCc3cnnn3C)CC2)=O)CCC2(CC=CCO2)C1 C1(NC(CC2C(C)CCO2)=O)CCC(C)N(C(c2cc(F)ccc2O)=O)C1 CCCC(CC)CCC(=O)N1CCC=C(C(=O)N2CC(C)(CSC)C2)C1 n1(CC)ccnc1CNC(c1cccn1C)c1nnnn1CC1CC1 C1(CCC)CCCCC1N=c1[nH]c(N(CCCC(C)C)C)nc2cc[nH]c12 N1(C(c2nc(OC)c(C)s2)=O)CC(C)(C)OCC1CNC(=O)C(C)NC(C)(C)C c1(C(N2CC(NC(CC(C)n3cc(Br)cn3)=O)C2)=O)cc(F)c(Cl)cc1F C1(NC(c2c(N=[N+]=[N-])cccc2)=O)CS(=O)(=O)C12CCCC2 c1(C(C)C)ccc(C(=O)NCC2CC(F)CN2C(=O)CCCCO)nc1 CCC(C)(F)C(=O)N1CC(n2cc(CNC(C3CC(=O)N(C4CC4)C3)=O)nn2)C1 C1(C(=O)NCC(CC=C)NC(=O)Cc2ccc(C)nc2)Cc2ccc(F)cc2C1 C1(C(N(C)CCOCCC(=O)NCC(C)(C)C#N)=O)CCCCC(=O)N1 N#CC12CN(C(=O)Nc3ccc(Cl)cc3)CC1CS(=O)(=O)C2 C1(CNC(=O)NC(C(=O)OC)(C)C)CCCCC1O N1(C(=O)CC2CC(NCc3ccc(Cl)c(O)c3)C2)Cc2ccc([N+](=O)[O-])cc2C1 C=CCC(F)(F)C(=O)NCC(C)CNC(=O)C(C)(O)CSc1cccc(F)c1 N1(C(C)=O)CCCC1CC(N1CC(C)(C(N2CC(n3cc(C)cn3)C2)=O)C1)=O Cc1cscc1C(=O)NCC1CCN1C(=O)C(C1CCCCC1)O Cn1cnc2c(N(c3ncc(Br)cc3Cl)CC3CNCCOC3)ncnc12 Cc1ccc(C(N2CC(C(=O)NCC3(C#N)CCC3)C(F)C2)=O)c(F)c1 C1(C(N2C(C(=O)OC)CC2)=O)N(C(=O)CC2CCC(=O)NC2)CC12CCCC2 Cc1cc(CC(=O)N(C(C(=O)N(C2CCCC2C)C)C2CC2)C)no1 c1(C(=O)NCC2(CC)CCCN(C(=O)C(C)SC(C)C)C2)cnc2ccnn2c1 c1(-c2cccc(C(=O)OCC)n2)cc2n[nH]cc2cc1C n1(CC)ccc(CC(=O)NC2C(C(=O)NCCCCSC)C2(C)C)n1 CC(CC(=O)OCC(C(F)F)n1cccn1)n1cccn1 C1(N(C(c2cnn(C(C)C)c2)=O)CC)CCN(C(C2CC(C)(C)CO2)=O)CC1 Cc1c(C(=O)N(C)CC2COC(=O)O2)sc2[nH]cnc(=S)c12 N1(C(=O)CN2CC3CC3C2)CCC2(NC(C34CC(CC(F)F)(C3)C4)=O)CCCC12 C=CCCCCCCCCCNc1ccc(N2CCN(C)CC2)c(Cl)c1 C1(O)(C(C(=O)NCC2=C(C)CCC2)(F)F)CCN(C(=O)OC(C)(C)C)CC1 C1(C2(O)CN(C(=O)CSC3CC3)C2)(CNC(C2CC(=O)N(C3CC3)C2)=O)CC1 C1(CCC(=O)N(CCCCNC(C2(CCOC)CC2)=O)C)NC(=O)NC1=O CCCC(CC)C(=O)NCCC(C)(C)CNC(=O)COCC=Cc1ccccc1 N1(C(COCC(=O)OC)=O)CCCC(C(=O)NOC2CC3CCC2C3)(CC)C1 C(=O)(C(CC)C(=O)NCC(C)C(=O)N(C)Cc1cocn1)OCC CP(C)(=O)C(O)C(=O)NCC1COCC1NC(=O)CC1CCC2(CC1)CC2 C12(CNC(C(C3(O)CCC3)NC(C=C(C)C)=O)=O)CC(C)(CCO1)C2 C1(CC(=O)NC2(C)CC(NC(c3c(C)nco3)=O)C2)CN2CCN1CC2 CCC(CC)(CN=C(NC1CCS(=O)(=O)C1)N1CCC(F)(F)C1)c1ccccc1 c1(CNC(c2ncccc2F)CC)cc(F)cc(I)c1 C1(C(=O)NCC2(NC(COc3ccc(C)cc3C)=O)CC2)CCn2nnnc2C1 C1(NC(c2c(C)nc(-n3cccc3)s2)=O)CN(C(=O)Cc2cnoc2)CCC1C CC1=CCSC1C(=O)N(CCCNC(=O)CCCC1CC1)C1CC1 C1(CC=C)(NC(c2ccnc(Cl)c2)=O)CCCN(C(=O)C2=C(C)OCC2)C1 N1(C(=O)COC(F)F)CC2CC1CN2C(C1CCN(S(=O)(=O)C(F)(F)F)C1)=O S(=O)(=O)(c1cccnc1N1CCCC(C)(C)C1)NCC(C)(C)OC N1(c2cc(NCC(n3cccn3)C)nc(COC)n2)CCOCC(C)(F)C1 Cc1ccc(F)cc1CNC(=NCCc1ccc(F)cc1)NCc1cccnc1 c1(C(=O)Nc2cncc(-c3ccc(-c4ccccc4)s3)c2)cnc2ccccn12 c1(OC(CC)CN(C(C2CCOC2(C)C)C(=O)NCCC#N)C)cccc(Cl)c1 O=C(C#CC1CCC1)NCC1CC(NC(=O)COc2ccccc2F)C12CCC2 CC(CC(=O)NC1CC(=O)N(C)C1)C(C)(C)NC(=O)CC(C)(C)C(F)F C1(C(=O)NCC(C)(C)OC(C)C)CCN(C(=O)CN2CCC(C)C2)C12CC2 c1(C(=O)NCCc2c(OC)cccc2)nc2c(C)cccc2s1 N1(C(C2CCC(=O)C2)=O)CCN(C(c2cc([N+](=O)[O-])n[nH]2)=O)CC1CC1CC1 N1(C(C(=O)NC2CCC(NC(C(C=C=C)C)=O)CC2)C)CCP(C)(=O)CC1 CC(C(=O)N1CCCC1CCCNC(=O)CCC(C)(C)NC(C)=O)S(N)(=O)=O C=C(C)C1OCCC1C(=O)NCC(C)CN(C)C(c1sccc1C#N)=O Cc1nn(CC(=O)NCC(C)(C)C(=O)NCCCCCF)c(=O)o1 C1(NC(C2(CCC=C)CN(C(C34CC(CO)(C3)C4)=O)C2)=O)CCCCC1(C)C C1(NC(c2c(CC)n(C)nc2)=O)CN(C(c2ncnn2CC)=O)CCC1CO CC1=C(C(=O)N2CC(CC(=O)NCC(Cl)C(C)(F)F)CC2(C)C)CCCO1 C1(CNC(=O)C(O)C2CCCC2)CC2(CO1)CN(C(C1(C3CC3)CCCO1)=O)C2 N=c1ccc(C(N2CCC(OC3CC3)C2)=O)c(Cl)[nH]1 c1(CC(=O)NC2C(NC(CC=CC)=O)COCC2)cc(C)cc(F)c1 N1(C(CC(CC)CC)=O)CC(C)CN(C(c2coc(Br)n2)=O)C(C)C1 c1(OC)nc(Cl)ccc1C(=O)N(C(C)CCNC(=O)CC(=O)N(C)C)C C(C(C)(C)C(=O)N1CC(O)CC1C(=O)NCCC1CCCCO1)OCC C1(C(C)C)N(C(c2cscn2)=O)CC12CCN(C(=O)CCC1CCC(C)O1)CC2 c1(C(=O)NCC2CCC(NC(=O)COc3ccc(F)cn3)C2)cncc(F)c1Cl N1(C(CCC(C)O)=O)CC2CCC1CN2C(c1coc(C2CC2)n1)=O CCCC(C#N)C(=O)NCCCOCCN(C)C(c1cc(C)nc(C)n1)=O C(=O)(CC(C)C(F)(F)F)NC1(CCC(=O)Nc2cccc(OC)c2O)CCCC1 C1(NC(C(C)(C)n2cncn2)=O)CC2CC1N(C(=O)CCCCCF)C2 C1(NC(CCc2cc(C)no2)=O)CCC(N(C(=O)Cn2ncccc2=O)C)CC1 Cc1cc(CNC(=O)C(C2CCC2)NC(c2cccnc2C)=O)cc(C)n1 C(CC)(C(=O)N(CCC(C)(C)NC(C1CCCC1C)=O)C)=CCCC C(CC(C)(C)C(=O)N(CC(O)C(C)(C)C)CCC(=O)N1CCCC1)NC(C)=O C1(C(=O)NC2(CCNC(CCC(=O)NCCC)=O)CCCC2)CNC(=O)CC1C N1(C(CC2(CC)CCC2)=O)CCC(C(=O)NC2CCN(C)C2=O)C(O)C1 C1(N(C(c2cc(COC)sc2)=O)C)CN(C(=O)C(C)(C)N2CCCCC2)CC1O O=C1CNc2ncc(C(N3CC(NC(C45CCCC4C5)=O)C(O)C3)=O)cc2N1 C(=O)(CC1OCc2ncccc21)NCC1CC(C)(C)CN1C(=O)C(F)C(F)(F)F N1(C(c2cc(C)c(O)nn2)=O)CCC(C)(C)C(C(N2CC3CC2(CO)C3)=O)C1 CC(N)(CS(C)(=O)=O)C(=O)NCc1nc2cc(F)ccc2s1 c1(C(=O)OC(COC)C2CC2)c(-c2ccccc2)coc1C C1(C(=O)NCCC2CCCN(C(C3CC(SC)C3)=O)C2)(CC)CCCCO1 c1(OC)ccc(C)c(C(=O)NCC2CCC(C)CN2C(=O)C=CC(C)C)c1N C1(NC(C2C(C)C2)=O)CC2CCC(C1C)N2C(=O)CCC1CC(C)(C)CO1 N1(C(COC(C)C)=O)CC2(CCC(NCc3cc(F)cc(Br)c3)C2)C1 CC(C)CC(C)C(=O)NC1(CC=CC(=O)NC(C)Cc2cn[nH]c2)CCC1 c1(C(=O)NC2CC(NC(c3c(CC)cccc3CC)=O)C2)cc(S(N)(=O)=O)c[nH]1 CC1CN(C(=O)CN(C)C(N)=O)C(C)CN1C(c1ccc(Cl)c(Br)c1)=O N(C(=NCCc1ccccn1)NCc1ccsn1)C1C(C)(C)SC1 C(=O)(CC(CN(C)C)CC)N1CC(C#C)(C(=O)NCC(O)CCC)C1 C1(N=[N+]=[N-])(C(=O)NC(C)CCNC(=O)CCCC2CC2C)CCOCC1 N1(C(CC2C(=O)NC(=N)S2)=O)CCCC2(NC(=O)CCc3cccnc3)CC2C1 C(C(CCC)C(=O)N(C1CCN(C2CC2)C1)C)NC(C1(CCC=C)CC1)=O c1(C(N2CCC(C(=O)NC(CSCC)CO)C2C)=O)ccc2cc[nH]c2n1 c1(CC)nocc1C(=O)NCC1C=CCN1C(C1CC1C(C)C)=O c1(CC(N2C(CNC(Cc3nnc(C)s3)=O)CC2)=O)csc2ccccc12 C(CC(CC)C(=O)NCC1CN(C(=O)CCC(=O)NCC)CC12CC2)=CC N1(C(CCC2CCC(=O)C2)=O)CCOC(CCC(=O)NC2(n3nccn3)CC2)C1 c1(CC(c2n(C(CC)C)nnn2)NC2CN(c3cnccn3)C2)cccc(Br)c1 Cc1cc(Cl)cc(NC(C2CC(F)CN2C(c2ccc(Cl)s2)=O)=O)c1Cl CCC(F)(F)CC(=O)NCC1(F)CCC(NC(c2cccc(CF)c2)=O)C1 N1(C(c2c[nH]c(=NC)s2)=O)CC2(CCN(C(C3CCCN3C(=O)NC)=O)C2)C1 C1(C(N2C(COC)CN(C(=O)CCC(C)(C)F)CC2)=O)CCCCC12CCC2 Cc1ncc(C(=O)NCCC2CC(NC(C3(n4cccn4)CC3)=O)C2)n1C CCC(C)(CCC(C)C)C(=O)N(CCCCNC(c1c[nH]cc1Br)=O)C C1(C(=O)NCCN(CCC)C(C2CC3(CC3)C2)=O)(COC)CCCCO1 C(CCC(O)C(=O)NCc1cn(C)nn1)NC(C=CC)=O C1(NC(c2[nH]cc(OCC)c(=O)c2)=O)CC2CC(C1)N(c1nc(C#N)c(Cl)s1)C2 Cc1c(C(=O)NC(C)CNC(c2scnc2C(C)(C)C)=O)ccn1C1CC1 c1(NC(C23CC(NC(C(CC(C)C)O)=O)(C2)C3)=O)cccc(Cl)c1C#N Cc1nc(O)[nH]c1C(=O)N(CCNC(C1CCC(C(F)(F)F)C1)=O)C1CC1 c1(C(N2CC(NC(CC(C)F)=O)CC2(C)C)=O)ccnc2ccc(F)cc12 N1(C(CCCC(=O)OC)=O)C(CNC(=O)Cn2cnnc2)CC2COCC12 CCCCC(C)CCC(=O)N1CCC(NC(c2cc(C#N)ccn2)=O)C1 C1(CNC(CCOCCOC)=O)C2CN(C(c3c[nH]nc3CN)=O)CC12.C(C)(C)C c1(C(=O)Nc2c(C)ccc(C(=O)N(C)C)c2)cc(S(=O)(=O)NCC(C)O)c[nH]1 c1(NCC(N2CC3C(NC(c4c(CC)[nH]nc4Cl)=O)C3C2)=O)oc(C)nc1C#N C(CCCCC(=O)NC1C2CCC(C2)C1C(=O)NCc1nnn(C)n1)OC C(=O)(CC(CC)C(F)F)N1CCCC(N(C(CCC#CC)=O)C)CC1 CCCCCC(O)C(=O)N1CCCC(C)(NC(C2CCC(C3CC3)CC2)=O)C1 c1(OC)cnc(C(=O)NC2(CCO)CN(C(=O)C=C(C)C)C2)c(F)c1 N1(C(C2C(COC)(COC)C2)=O)C2CCCC1CN(C(=O)CC#N)C2 N1(C(CCCN(C)C)=O)CCC(C)(NC(=O)Cc2ccsc2Br)CC1 N1(C(C(CCC)C)=O)CC2(CCC(CNC(=O)CCCOC(C)C)O2)C1 c1(OC)nc2ccc(C(N3CC(C)CN(C(=O)CSC4CC4)C(C)C3)=O)cc2[nH]1 C(CCN=C(NCc1cccnc1)NCc1nc(C(C)C)cs1)(C(F)(F)F)OC c1(CCC)ccccc1C(=O)NC(C(=O)NC(C)CCN(C)C)C(C)C Cc1cc(CC(=O)NCCC2CCCN(C(=O)C(F)(F)C(C)O)C2)ccc1CO c1(C(N2CCN(C(=O)CC3(O)CCCCC3)C(CF)C2)=O)cc([N+](=O)[O-])n[nH]1 c1(C(N2CCN(C(C)C)CC2C)=O)ccc2ncc(C3=CCCC3)n2c1 Cc1ccc(NC(C2CCN(C(=O)CCCCCl)CC2O)=O)cc1O N1(C(C2CCN(C(=O)COc3ccccc3)CC2)=O)CCC2(CCCCO2)C1 C1(C(=O)NC(CNC(CS(=O)(=O)NCC)=O)C2CC2)CC2(CCC2)CO1 c1(SC(C(N2C(C(=O)OC)CC(O)C2)=O)C)cc(-c2ccccc2)sc1SC n1(CC(N2CC3C(CNC(C4CC(SC)C4)=O)(C3)C2)=O)cnc([N+](=O)[O-])c1 c1(Cn2cc(C(N(CCCCN(C(CCSC)=O)C)C)=O)nn2)cccc(Cl)c1 N1(C(C2(CF)COC2)=O)CCCOC(CNC(C2(CO)CCCO2)=O)C1 C1(C(N(OC)Cc2cccnc2)=O)CCCN(C2CCCCC2C(=O)N)CC1.OC c1(C(N2CC(NC(c3n(C)ccn3)=O)C3C2C3)=O)cc2c(cn1)OCCC2 Cn1nc(CNC(=O)CCNC(C2CC2OC(C)(C)C)=O)oc1=O CCC(C(=O)NCC1CCC(F)(CNC(=O)CCn2ccc(C)n2)C1)C(C)C C(=O)(CCCC(=O)NC1CCCCC1CC1(C(=O)NCC)CC1)N(CCC)CCC N1(C(C(C)NC(C)=O)=O)CCCCC1CN(C)C(c1cocn1)=O CC1CN(C(=O)CCCC#N)CCN1C(=O)Cc1ccon1 C1(NC(c2ncn(C(C)C)n2)=O)CN(C(=O)CC#N)CC1C C(=O)(C(C)CC(=O)NC(c1ncc(F)cn1)C)ONC(C1(NC(N)=O)CC(F)C1)=O C1(NC(c2cncc(SCC)n2)=O)CCN(C(C2CC(=O)N(C)C2)=O)C(C)C1 N1(C(C(=O)Nc2ccc(OCCC)cc2)=O)CCC12CCS(=O)(=O)C2 C12(CNC(C3CCCO3)=O)CC(C1)C(NC1(C(=O)OCC)CCCC1)CO2 Nc1cc(C(=O)NCC(C2CC2)NC(=O)CCC2CCCO2)c2ccccc2c1 Cn1cc([N+](=O)[O-])c(CC(N2CCN(C(=O)COC3CCOC3)C(CF)C2)=O)n1 C1(C(=O)NCC2(COC)CN(C(C3CC(F)(CF)C3)=O)C2)CCNC(=O)C1 C1(NC(=O)CC(C2CC2)C2CC2)CCN(C(c2cc3sccc3[nH]2)=O)CC1F C12(CCCC1OC)c1nnnn1-c1ccccc1N2.CCCC=CCC Cc1cc(C(=O)NCC2CCCN(C(C3(C)CCCC3(F)F)=O)C2)c(C)cc1Cl n1(CC)cc([N+](=O)[O-])c(C(=O)NCC2CCC(CN(C)C(C3CC3F)=O)CC2)n1 C1(NC(CC2N(C)CCC2)=O)C2CCCN(C(C3CCCCN3C)=O)C2C1(C)C C(C)(c1ccco1)=CC(=O)NCCOCC(N1C(C)(CCC)CC1)=O Cc1nc(C=CC(=O)NCCN2CCC(NC(c3c(C)csc3Cl)=O)CC2)cs1 N1(C(C2C(C)OCC2)=O)CCC(O)(Cc2cn(-c3ccccc3Cl)nn2)CC1 CCC(C#N)(CC)C(=O)NC1CN(C(=O)CSc2ccc(Cl)cc2)C(C)(C)C1 C1(=CC(=O)NCCN(C(=O)C(C2CCOC2)OC)CC)CCC(C)(C)CC1 N1(C(c2nc(CC)sc2)C(=O)Nc2c(C)csc2Cl)CCCN(C2CC2)CC1 N1(C(CC2CCC(C)CC2)=O)CC2CCCC(CNC(c3cscn3)=O)C2C1 N1(C(C)C)C(=O)CCC1C(=O)N(C1CCN(C(c2ccc(C(N)=O)nc2)=O)C1)C Cc1ccncc1C1CCN(C(=O)NCc2ccoc2C(F)(F)F)C1 C1(C(=O)NC(C2CCCC2)CNC(C2CCC(COC)O2)=O)CC2CCC1CC2 CC(C)C(O)C(C)C(=O)NC(CC1CCC1)C(=O)NC1CC2(C1)CC(C)(C)C2 C1(NC(C2OCCN(C(Cc3ccn(C)c3)=O)C2)=O)CCC2(CCC2)CC1 c1(CC(=O)NC2CC3CN(C(CCC(=O)OCC)=O)C2C3)nsc2ccccc12 c1(N(C2CN(C(C(C)(C)C)=O)C2)C(Cn2ncc(C#C)c2)=O)ccc2ccn(C)c2c1 C(=O)(C1=CCC(C)(C)CC1)NC1C2(CC(NC(c3cc(OC)n(C)n3)=O)C2)C1 c1(C(N(C)CC)=O)ccc(NC(c2cnc(C(C)=O)s2)=O)cc1 Cc1cc(OCCN(C)CC2CCC(C)N(c3ncccn3)C2)cc(C)c1 c1(C(=O)NC2CN(C(CC(C)c3ccco3)=O)CC23CC3)cc2ccccc2o1 CC(C)CCCCC(=O)N1CC(O)CC1c1n[nH]c(CC2CCC(O)C(O)C2)n1 c1(C(N(CC(C)C(=O)N(CCC(F)(F)F)C)C)=O)cccnc1S N1(C(c2c(O)ncc(CC)c2)=O)CC(C)CN(C(=O)CCCOC(C)C)C(C)C1 CC1(CC(=O)NCCCN(C(c2ccn(CC(F)(F)F)n2)=O)C2CC2)CCCO1 C(c1cnccn1)=CC(=O)N(C1CCN(C(C2CC(C#N)C2)=O)CC1)CC Cc1cnc(CC(=O)NC(CNC(=O)Cc2cnc(C)o2)C2CC2)[nH]1 C1(CSC)CCN(C(=NCCc2c(C)nn(C)c2C)NCCc2cccs2)C1 C1(CC(C)NC(=O)Cc2ccno2)CC2CCC(C1)N2C(c1ccc(O)cn1)=O C=CC(CC)CC(=O)N(CC(=O)NCCc1noc(=O)n1C)CC N1(C(C(CC)C)=O)CC2(CNC(C3CSCCS3)=O)CC1CO2 CC1CCC(C(N)=O)CN1C(=O)CSc1cccs1.c12ccccc1CNC2=O C1(NC(C(C)=C(C)C)=O)CCN(C(=O)CCC(=O)c2cccc(N)c2)CC1F c1(C(=O)NC2CC(F)(CNC(c3cnco3)=O)C2)csc2ncnc(O)c12 N1(C(C2N(CCC)CCC2)=O)CCC(C)N(C(c2nnc(S)n2C)=O)CC1 Cc1cc(C(=O)NC2CC3(C2)CC3NC(=O)C=Cc2cncc(O)c2)cc(O)n1 C1(OC)CCN(C(C2(NC(=O)CCCCSC)CCC(C)(C)C2)=O)C(C)C1 C=CC(C)(O)CC(=O)N1CC(NC(=O)Cc2cnsc2)C(n2ccnn2)C1 c1(CCC(=O)NCCNC(C2(CC(F)F)CC2)=O)cc2ccccc2[nH]1 N1(C(C(c2ccn(C)n2)C)=O)CC(NC(=O)CN2CCC(O)CC2)C2CCCC12 N1(C(N2CC(C(=O)NC(CC)C(=O)c3ccccc3)C2)=O)CCCCC1C(C)C C1(C(=O)NC(C2CCN(c3ncnc4[nH]ccc34)C2)C)CC(C)(C)CC(C)(C)C1 C1(NC(c2nc(C)[nH]n2)=O)CC=CCC1C(=O)NCCC(C)C c1(CNC(c2n(CC)nnn2)c2cc(C(N)=O)cs2)c(F)cccc1I N1(C(c2nc(COC)sc2)=O)CC(CNC(=O)CC23COCC(C2)C3)CC1(C)C c1(CC(N2CCC(O)(CN(C(C(C=C)O)=O)C)CC2)=O)ccc2sccc2c1 c1(C(=O)NC2CC(C)(NC(C(C)=C3CC3)=O)C2)cc2c(O)cccc2[nH]1 C1(N(C)C)CCCC(C(N2CC(N3CCN(C(C4C5CCCC45)=O)CC3)C2)=O)C1 c1(C(=O)NCC2N(C)CCN(C(CCC#C)=O)C2)ccc(F)c(C(F)(F)F)c1Cl Cc1c(F)cc(C(=O)NC2CN(C(=O)CNS(C)(=O)=O)CC2C#N)cc1Br Cc1ccc(CCNC(=O)CCCc2cnccn2)cc1F C(=O)(C(CC(C)C)ONC(C1CC(=O)C1(C)C)=O)N(c1ccccc1)CC Cn1cnc2c(NC3CCCC3C3CC3)[nH]c(=NCC34CCCN3CCC4)nc12 C(=O)(C1c2ccccc2CN1C(=O)C(C)(C)O)N(C1CCCC1)CCCC c1(COC)nc(N2CCCCC(NC(C3CCN3C3CCCC3)=O)C2)cc(C)n1 C12(OC)CCC(C(=O)N(CC(C)O)CCNC(=O)C(F)OC(F)(F)F)(CC1)C2 N1(C(C(CC)(C)CO)=O)CC2(C=C(C(=O)NCCC(C)F)CO2)C1 c1(C(N2C3(CNC(CCC)=O)CCC3CC2)=O)ccc2[nH]ccc2c1 C(=O)(C(C)(COC)OC)NCc1cc(C(=O)NCCC#C)on1 c1(C(N2CCCC(O)(CNC(c3cnon3)=O)C2)=O)ccc(Br)c(F)c1F N(C(=NCCC(C)=O)NC1CCC(SC)C1)C1CCN(C(=O)OCC)CC1 C1(CC#C)(C(=O)NCC(C2CCOC2)NC(=O)Cc2nonc2C)CCCC1 C(=O)(C(CC1CCCC1)NC(=O)C(O)CN(C)C)N(CC(C1CC1)OC)C C1(CNC(C(N2C(CC)CCC2)=O)=O)CC2CN(C(=O)CC(C)(C)C#N)CC12 C#CC1CN(C(C2CN(C(=O)COCCCF)CCO2)=O)CCO1 N1(C(C2CCC(C)(CC)O2)=O)CCC2(C1)CN(C(C1(F)CC3(CCC3)C1)=O)C2 C(C1c2ccccc2CCN1C(C1(O)CC(F)(F)C1)=O)NC(C(CCC#C)O)=O c1(C(=O)NCCCCC(C)NC(c2cc(C(N)=O)n(C)n2)=O)ncc(Cl)cc1Cl C(CN=C(NCc1ccsc1)N1CCC(N2CC(C(F)(F)F)CC2=O)CC1)OC C1(C(=O)NC(CC(C)NC(c2c(C)nn[nH]2)=O)C)CCCCC(=O)C1 C=CCC(F)(F)C(=O)NCC(c1ccccc1)NC(c1ccnn1CC)=O C1(NC(CN2C(C)CC2)=O)CN(C(=O)C=CC(c2ccc(Br)cc2)=O)CC1C C(=O)(C(C)(C)C(F)(F)CC)NC(CC=C)CNC(c1noc2c1CCCC2)=O c1(NC=O)ccc(C(=O)NC2CCC(F)(CNC(C3CC4CC4C3)=O)C2)cc1 c1(N2C(C)COC3(CCC3)C2)[nH]c(=NCc2nnc(CCO)s2)nc2sccc12 c1(CC(=O)N(CCC(C)NC(=O)CNS(=O)(=O)C2CC2)C)cc(F)cc(C#N)c1 N1(C(C2N(C(C3C(C)C4CCC3C4)=O)CC3CC32)=O)CC(C)(C)C12CCC2 c1(-n2cc(CC3CCN(C(C(C)O)=O)C3)nn2)ccc(Cl)c(Cl)c1 C12(CNC(c3cc(C)oc3)=O)CN(C(c3cnc4ccsc4c3)=O)CC1CCO2 C12(C(=O)OC)CC1CN(CC)C2.c1(N(C(=O)O)C)ccc(N2CCCCCC2)cc1 N12CC(O)C(O)C1C(=O)NCCC(O)CNC2=O.CC(C)(C)O.C(=O)(C1CC1)N c1(CC(=O)NCC(CC)NC(C2CCCC(C(C)(C)C)C2)=O)nnc(S)n1C c1(C(N2CCC(N(C(C3C(C)C3)=O)C)C2)=O)nc2ncc(Br)cc2[nH]1 c1(SC)nc(C(=O)NCCCNC(C23CCCN2CC(O)C3)=O)c2ccccn12 Cc1ccc(F)c(C(=O)NCC2(CNC(c3c(F)cccc3Cl)=O)CC2)c1 c1(-c2scc(NC(C3CCC(O)CC3)=O)n2)c(Cl)cccc1Cl Cc1cc(C(N2CC=C(C(=O)NCCCCCO)C2)=O)nnc1C C1(NC(C2CC(C)OCC2)=O)CC2CC1CN(C(c1ccsc1C(F)(F)F)=O)C2 CCC(O)C(F)(F)C(=O)NC1CC1NC(=O)CCSc1ccc(F)cc1 c1(OC)ccc(O)cc1C(=O)NC(C)(C)CCNC(c1ccc(CCO)cc1)=O c1(CCN2C(C(N3CC(NC(CCC#C)=O)C3)=O)CCC2)ccc(Cl)cc1F CCN=c1[nH]cc(C(=O)NCC2CN(C(=O)C(O)P(C)(C)=O)C(C)(C)C2)s1 N#CC1CCC(NC(=O)CCCCc2ccc(I)cc2)C1 C(C(CNC(=O)Cc1cnc[nH]1)C(F)(F)F)NC(=O)CN1CCSCC1 c1(NC(C(=O)NC(C(C)NC(CC=C)=O)CO)=O)nc(C(C)C)c(C)s1 C1(COC)CCCN(C(c2ccn(CCNC(c3cc(C)nn3C)=O)c2)=O)CC1 C=CCCC(C(=O)N(CC(C1CC1)OC)C)NC(c1cc(C)[nH]c1C)=O C1(NC(Cc2cc(C)on2)=O)CCCCC1NC(C1CCCCS1)=O N1(C(c2c(F)ccc(C(C)C)c2)=O)CC2CC(C1)C2(F)F C=CC(CCC)CC(=O)N1CC(O)(CNC(c2cc(C3CC3)ncn2)=O)C1 Cn1nc(Br)nc1C(N1CCC(c2ccc(Cl)cc2)C1)C(=O)NC1COC1 c1(C(=O)NCC(CC)NC(=O)CN2CCC(CO)CC2)c(C)nn(CC)c1Cl c1(C(=O)NCC2C(NC(C(C)NC(C)=O)=O)CCC2)cccc2c1OCCCO2 c1(C(N2C(CNC(C(C)OCC=C)=O)CC2)=O)coc(C(C)OC)n1 Cn1nc(C(N2CC3CN(C(c4ccsn4)=O)CCC23)=O)c2c1CCSC2 Cc1cccc(C(N2CC(CC(C)NC(c3cnc(Cl)c(Cl)c3)=O)C2)=O)c1O N1(C(C(CCCC)C)=O)CCC2(CC1)CC2NC(C1CCC(=O)N(CC)C1)=O C1(C)(C(=O)NC(C)CCN(C)C(C2CCC(C)O2)=O)CCS(=O)(=O)CC1 Cc1cc(C(N2CCN(c3cccc(C)n3)C(C)C2)C(=O)N(C)C)nc(C)c1 CC1CC(C)(C(=O)Nc2cnc(Cl)c(CNc3cnc(F)cn3)c2)CCO1 Cc1cc(C)c(C(=O)NCC(C)(C(C)C)NC(c2cc(C#N)c(C)s2)=O)c(O)c1 Cc1cccc(C(=O)NC(C)C(=O)NC23CC(C2)N(C(C2(O)CCC2)=O)C3)c1 N1(C(c2c(CC)nns2)=O)CCC2(CC1)CC2NC(=O)C(CC)SC CCC(C)CCC(=O)N(C1CCN(C(=O)CCOC2CCCCC2)C1)C N1(C(Cn2cnc(C)c2C)=O)CC(C)(C)C(O)C1(C)C C1(C(N2CC(O)(C(C(N3C(CC(N)=O)CCCC3)=O)F)C2)=O)CCOCC1(C)C c1(CN2C(C(=O)NCC3(N(C)C)CCOCC3)COCC2)c(Br)cc(F)cc1Br c1(CNC(C)CCC2CC2(Cl)Cl)nncn1CC1CC1 C(=O)(C(C(C)C)NC(c1ccccc1F)=O)N1CC(C)(OC)C1 c1(OC)ccc(Cl)cc1OS(=O)(=O)CC1CCOCCCC1 C(CC)(C(=O)NC1(C(=O)NC(C)(C)CCN(C)C)CC1(C)C)OCC C1(C)(C(N2CCN(C(C3=CC(C)(CC)C3)=O)C(CO)C2)=O)CCS(=O)(=O)CC1 C1(CC(=O)NC23CC(NC(c4cnn(C)c4Cl)=O)(C2)C3)CCC(=O)NC1=O C(=O)(C1CCc2c(Cl)cccc21)NC1CC(N(C)C(c2cn[nH]c2)=O)C1 N1(C(C)C)CCN(CCC(=O)NCC(O)CN(C)C(C2CCCS2)=O)CC1 O=C1OC2CON(C(=O)c3cc(-c4ccncc4)[nH]n3)CC2O1 c1(C(=O)NCCN2CCN(C(C3(O)CCC(CC)C3)=O)CC2)cc(F)ccc1O CC(C)CC(C(=O)N1CCN(CC(=O)N(C2CCOC2C)C2CC2)CC1)C(C)C S(=O)(=O)(c1cnc(C)c(C#N)c1)Nc1c(NC(CC)C)cc(Cl)cc1 c1(N2CCCC(NC(c3ccnn3CC3CCOCC3)=O)C2)ccc(Cl)cc1 C1(CN(C)C(C2CC23CC3)=O)CCN(C(c2csc(Br)c2)=O)C1 C1(CNC(CCNC(C)=O)=O)CC2CCC1N2C(C1(C)CC2CCC1C2)=O CC(CC(=O)N(CCCN(C(=O)C=C1CCSCC1)C)C)C1CCCO1 c1(OC)cccc(-c2nc(C(C)C(C3CC3)OC)n(CCCO)n2)c1 C1(NC(=O)COCc2ccccn2)CC2(NC(=O)Cn3cnnn3)COC1C2 C(C)(C)(CCC(=O)N1CCCC(CO)(COC)C1)OC(c1c(CC)oc(C)c1)=O c1(CC)ocnc1C(N1CC(CF)(NC(c2csc(=N)[nH]2)=O)C1)=O C1(NC(c2ccc(C)nc2)=O)CC(NC(C2C=CC=CC=C2)=O)C12CCC2 C1(NC(c2c(CC)nn[nH]2)=O)(CNC(C2CCCC(CC)C2)=O)CCCCCC1 c1(CC)ccc(C(=O)NCCC2(O)CN(C(c3cc(Cl)nc(=N)[nH]3)=O)C2)c(O)c1 N#Cc1ccc(=NCC(=O)N2CC=CC2CNC(=O)C=CC2CCC2)[nH]c1 c1(C(=O)NC(C2CCN(C(=O)C(C)OCC(F)(F)F)CC2)C)occ2c1CCCC2 n1(CC)nc(C)c(C(=O)NCC2CC(NC(C3NC(=O)CC3C)=O)C2)c1C C(=O)(C1=CC2CCCC12)NCC(C)(C)NC(=O)C1=CCCOC1 c1(C(N(CCN(C(CCC=C=C)=O)CC)CC)=O)ccc(C(F)(F)F)c(N)c1 C1(CC)CN(C(c2ccccc2Cl)=O)CCC1NC(=O)CSc1cccc(C)c1 n1(CC)nnc(C)c1C(=O)NCC(C)NC(c1cnoc1-c1ccccc1)=O C1(CCC)CN(C(=O)C(C)CC(N)=O)CCN1C(=O)CCc1ccc[nH]1 C(=O)(C(F)(F)C(F)(F)F)NCCCN(C(C(C)(C)NC(=O)OCCC)=O)CC c1(C(=O)NCC2(NC(C3C(C)CN(C)C3)=O)CCC2)csc2cc(Cl)cnc12 C(=O)(CC(C(C)C)c1ccon1)NCC(=O)OC.c1(O)ccc(NCCCC)cc1 C1(CCOC)CN(C(=O)CC#N)CCN1C(c1cncc(OCC(F)(F)F)c1)=O CCC(CCC(=O)NC(C)(CNC(c1cc(C)cc(C)n1)=O)C1CCC1)OC CCC(C)(CCC(C)C)C(=O)N1CCCC(CNC(=O)CC(C)(C)COC)CC1 C1(CCOC)(NC(=O)Cn2ncc(CO)c2)CCN(C(=O)Cn2ncnn2)CC1 S(=O)(=O)(c1ccc(C#N)c(NCCn2ccnn2)c1)N1CCC(CC(C)O)CC1 CCC(C)(C)C(=O)NCCC(Cc1ccccc1)NC(=O)COCC1CCOC1 C1(CNC(=O)CCCc2nccs2)CCN(C(=O)C(=O)NC2CC2)CC1 C=CCC(C(=O)NCC=CCNC(c1occc(=O)c1OC)=O)C(C)C Cc1ccc2c(=NCN3CCC(OCCF)C3)[nH]c(=NC3CCCC3C)[nH]c2c1 C1(C(N(CCN(C(CC=CC)=O)C(C)C)CCC)=O)CCCCN1CCC C(=O)(CCS(=O)(=O)N1CCOCC1)N(C(C)CN(C)C(C1(C2CCC2)CC1)=O)C c1(C(C(=O)NCCOCC2CC2)N(CCN(C)C)C)ccc2ccc(Cl)cc2n1 N1(C(CC=CCC)=O)CCC2CCCC12C(N1CCC(CN(C)C)C1)=O CC(C)CC(=O)NC(C(=O)NCC1C2COCC12)C1CCC1 C1(NC(CSCCC(C)C)=O)CC(O)CN(C(c2ccnc(OC(F)F)c2)=O)C1 S(=O)(=O)(c1ccc(NCCc2cn(CC)nn2)c(Cl)c1)N(C)CC1CC(=C)C1 Cc1cc(C(=O)NC(C2CCCN(C(=O)C=CCO)C2)C)cc(O)c1 c1(C(N2CC(N(C)C(c3ncn(C)n3)=O)C(F)C2)=O)cc(Cl)cc([N+](=O)[O-])c1 C1(CNC(C2(C(N)=O)CC2)=O)CCN(C(c2nn[nH]c2Cl)=O)C12CC2 c1(NC(c2nnnn2CCC2CC2)(CC)C2CC2)cccc2c1OC(C)(C)C2 CC(C)C(O)C(=O)NCC1(C)CC(NC(=O)CSc2cn[nH]c2)C1 Cc1cc(C)c2c(C)c(C(=O)NC3CCC3NC(c3cc(C)oc3C)=O)[nH]c2c1 Cc1c[nH]c(CC(N)=O)c1C(N1CCC(CNC(c2n[nH]c(C)c2Cl)=O)C1)=O O=C(C(O)C(F)(F)F)NC1CN(C(c2nncs2)=O)C1 n1(CCCOCC)c(N2CCC(N(S(C)(=O)=O)C)CC2)nnc1-c1ncn(C)n1 c1(C(=O)NC(CC=C)CNC(=O)C(F)OC(F)(F)F)nc(-c2ccsc2)oc1C Cc1noc2cc(C(N3CC(CNC(C4C(C)(C)C4(C)C)=O)C4CC34)=O)ccc12 C1(N(C(C2C(=C)C2)=O)C)CN(C(C2(c3ccc(F)cc3)CCCC2)=O)CCC1C C1(CNC(C(C)NC(=O)NC)=O)CCN(C(c2cnn(CCO)c2)=O)C(C)C1 C(=O)(C(O)C(C)(C)C)N(CCNC(C1(C(=O)OCC)CC1)=O)C CCCC(CC(=O)NCc1ncccc1O)NC(=O)C(O)CC N1(C(C2C(C)C2C)=O)CCN(C(=O)Cn2nc(-c3cccs3)oc2=O)CC(O)C1 c1(C(=O)NCCCC2N(C(c3c(C)nn[nH]3)=O)CCC2)ccc2nc(O)cn2c1 C(=O)(C1CCOc2ccccc21)N1CC(NC(c2csnn2)=O)CC12CCCC2 c1(CC)ccc(C(=O)NCCCn2cc(-c3ccc(C(C)C)cc3)nn2)cn1 N1(C(CN(C(C)=O)C)=O)Cc2nccn2CC(NC(c2cnc(Cl)cn2)=O)C1 N1(C(C(CC)N(C)C)=O)CCC(CNC(c2ccc(-c3ccco3)[nH]2)=O)C12CC2 c1(C(N2CC(F)(C(N3CC(CC#C)OCC3)=O)C2)=O)ncc(N)cc1C c1(C(=O)NCC2(NC(C3C(C)N(C)CC3)=O)CCCC2)cc2n(n1)CCCC2O N1(C(C(=Cc2cnc[nH]2)C)=O)CCN(C(c2nc(C)ccc2F)=O)CC1C1CC1 N1(C(C(CC)=CC)=O)CCC2(CC1)CC(NC(=O)Cc1cncn1C)CO2 N1(C(C(C)OCCOC)=O)CC2CCOC2(CNC(=O)C(C)(C)CC(=O)OC)C1 c1(C(=O)NCC(C)(C)OCCNC(C(F)=C(C)C)=O)ncc2ccccn12 C=CC(CC)CC(=O)C(N1CC(C(=O)ON2CCCCC2)C(O)C1)=O N1(CC(=O)N(C2C(C)CCCC2)C)CCC2(CC1)CN(C(C1(C)CC1)=O)C2 n1(CCC(=O)NCC(C)NC(=O)CN2CCSCC2)ncc2ccccc12 C(=O)(C(C)S(N)(=O)=O)N(C)CC1CCN(C(C=C(CC)CC)=O)C1 CC(C)CC(C(=O)N1C2CCC(C2)C1CNC(C1CC1C)=O)n1ccnc1 C1(C)(NC(CC2C(OC)COCC2)=O)CCCN(c2nccc(CO)n2)C1 c1(CN=c2c(C#N)cc3c([nH]2)CCSC3)nccc(=NC2CCOC(CO)C2)[nH]1 N1(C(C2(C)CC2(F)F)=O)CC(C2CCN(C(C3COC(=O)C3)=O)CC2)C1 C(=O)(C1Cc2c(Cl)cccc21)NC(CNC(c1ccc(OC)cc1)=O)(C)CO c1(C(N2CCN(CC3CCCC3)CC2C)C(=O)NC(C)C)cccn(C)c1=O N1(C(C2CCC(n3cc(C4CCN(C)CC4)nn3)C2)=O)CCc2cccc(O)c2C1 N1(C(c2c(Cl)nc(Cl)n2C)C(=O)Nc2cccc(OC)c2)CC(C)CC(O)C1 CCCCC(F)C(=O)NCc1cc(C(=O)NCC2CCCC2O)n(C)n1 CC(C(=O)NC(CNC(=O)CC1CC2(CCO1)CC2)C1CCC1)C(C)(C)C c1(OC)cccc(SCC(N2CC(N(C(=O)CSC(F)F)C)C(O)C2)=O)c1 N1(C(C(COCC)n2cc(Cn3cc(C)cn3)nn2)=O)CCC2(C=CCO2)C1 C1(CNC(c2c[nH]nc2-c2ccncc2)=O)(NC(C2CCC2(F)F)=O)CCOC1 c1(OC)ccc(F)c(C(N2CC(CNC(C3C(C)C3(F)F)=O)CC2(C)C)=O)c1 CCC1=NOC(CC(N2CC(CC(F)C(=O)NC(C)(CC)CC)C2)=O)C1 C(=O)(C1=CCOCC1)NCC1(C(N2C(CC(=O)OC)CCC2)=O)CC2(CC2)C1 C1(CNC(C2(c3cc(C)on3)CC2)=O)C(C)CCCN1C(c1cnnc(O)c1)=O c1(C(N(CCCCC)C)=O)occc1CNC(c1ccncc1)=O N1(C(CSCC(=O)Nc2ccoc2)=O)CCn2c(cnc2C(F)(F)F)C1 C1(C(=O)OC)CN(C(c2ccnc(OC(F)F)c2)=O)c2ccc(F)cc2O1 c1(CC)cnccc1CNC(=O)NOCCF CCCCCC(O)C(=O)N1CC2(NC(c3coc(C(C)=O)c3)=O)CCC1CC2 C#CC1CN(C(=O)C(CNC(=O)CC(COC)COC)CC(C)C)CCN1C C1(O)(CCNC(C(C)=C(CC)C)=O)CCCN(C(=O)CC2(NC(C)=O)CCC2)C1 N1(C(CC2CC(=C)C2)=O)CCC2(CC1)CN(C(c1ncncc1Cl)=O)CC(C)O2 C1(C)(CNC(C(C)Cc2cnn(C)c2)=O)CCCN(C(=O)C2=CCSC2)C1 C1(NC(C(C)OCC)=O)CC(F)CN(C(c2cc(Cl)n(C)n2)=O)C1 C=C1CCN(C(=O)CCN(C(=O)C(CC)n2cncn2)CCN(C)C)C1 c1(C(=O)NC23CCCN(C(C4N(CC)CC4)=O)CC2C3)cnc2ncnn2c1O c1(C(=O)NCCC2CN(C(C3CN(C)C3)=O)CC(C)O2)cccc2nccnc12 c1(C(N2C3CC(CC(NC(C(C)S(N)(=O)=O)=O)C3)C2)=O)cn2cc(F)ccc2n1 CCCC(C(=O)N1CCC(CNC(=O)CC2CCC3(CCC3)O2)CC1)S(N)(=O)=O N1(C(c2nc(C(C)=O)sc2)=O)CC(NC(=O)C(F)(F)c2ccnn2C)CC1C Cc1[nH]c2ncccc2c1C(=O)N(CCNC(=O)Cc1cc(C2CC2)on1)C1CC1 C1(NC(c2ccc(OC)nc2)=O)CC12CCN(C(=O)C(O)CSC)C2 c1(C(N(C)CCNC(c2cc(F)c(Br)cc2N)=O)=O)cc2c(=O)[nH]ccn2c1 Cc1nc(C(=O)NCC2(O)CN(C(C3CC4OC3C3CC43)=O)C2)c2ccnc-2[nH]1 C1(NC(c2nc(CC)oc2)=O)CC2CCC(C1)N2C(c1cc(CC(C)C)[nH]n1)=O N(C(=NCCSC)NC1CCOC1)CC(c1cccc(C)c1)OC CC1C(C(=O)N(CC2=CCSC2)C)CCN1C(C1CCC(C)(C)C1)=O C(=O)(CC(C)(C)CNC(C1CC(C)(O)C1)=O)NC(CCOC)CO CC(C)(C#N)C(=O)NCCC(O)CNC(=O)C1=C(Cl)CC1 Cc1cc(NC(=O)CC2COCCN2C(=O)C(O)C(C)C)cnc1Cl C=CC(C)(CCOC)C(=O)NCC1(C)CC(NC(c2csnc2OC)=O)C1 N1(c2cc(CC)ncn2)CCOCC(NC(c2c(C(F)(F)F)coc2C)=O)C1 c1(C(=O)NC2CC3CN(C(Cc4ncc(C)s4)=O)C2C3)cnc2snc(C)c2c1 c1(C(=O)NCC2=CCN(C(C3C(C)(C)C3(C)C)=O)CC2)ccc2c(c1)C(=O)NC2 C1(O)(C(CNC(C2(CC(=O)OC)CC2)=O)C)CCN(C(=O)C=NOC)C1 c1(CC)nncn1NC(=O)C1(NC(=O)CN(C)Cc2cccnc2)CCC1 C1(NC(C(C(=C)Cl)(C)C)=O)CC1C1CCN(C(C2CC3(C2)CC(F)C3)=O)CC1 c1(C(N2CC(NC(c3n(CC)ncn3)=O)C(O)C2)=O)c(O)cccc1Cl C=C(C)CC(C(=O)N1CC(c2nc(=O)o[nH]2)C1)NC(=O)C(C(C)C)SCC N1(C(c2scc(C)c2)=O)CC(F)CC1CN(C(=O)C(N1CCOCC1)C)C c1(CC)oc(C)cc1C(=O)NC(CNC(c1cnc(C(N)=O)s1)=O)CCOC C(C(CC(=O)N1CCC(Cc2ccn(C)n2)C1)C1CCCCC1)OC N1(C(C2C(CC)C2)=O)CCC2(C(=O)NC3CC3C(C)C)CCCC12 C1(CCNC(C)=O)CCC(C(=O)COC(=O)C=CC2CCOC2)CC1 C1(N(C(c2[nH]cc(C)c2)=O)C)CN(C(=O)COC2CC2)CCC1C CC1(C)CN(C(C2CCc3nc[nH]c3C2)=O)CCC1NC(=O)C1=CCCC1 N1(C(C(C)(C)C2CCOC2)=O)CC2(C1)SCCC2NC(=O)COCc1nc[nH]n1 CCC(CCOC)C(=O)NCC1CN(C(c2ccnn2COC)=O)CCN1C N1(C(c2c(OC)scc2)=O)CC(NC(C2(n3cccn3)CC2)=O)C2CC12.C1C(=O)N1 c1(OCC(N2CCN(C(C(=O)NCC)=O)C(CO)C2)=O)c(C)cc(Cl)cc1C C(=O)(C(O)(C(F)(F)F)C1CC1)NCCOCCCNC(c1c(C)ccnn1)=O N1(C(C(C(C(C)C)O)C)=O)CCN(C(c2cc[nH]c2)=O)C2CCCC2(C)C1 C1(=CC(=O)NCCN(C(=O)COC2(C)CCCC2)CCC)CN2CCC1CC2 N1(C(c2cccc(O)n2)=O)CC2CCCC2(CNC(C2(c3ccccc3)CC2)=O)C1 Cc1cc(C(=O)Nc2ncccc2OC(C)C)n2ncnc2n1 CCCC(C#N)C(=O)N1CCN(C(=O)CN(CC)CC)CC1C c1(C(N2C(CC)CN(C(=O)CC3CC(F)C3)CC2)=O)cc2c(s1)CCCNC2=O N1(C(Cn2c(C)ccn2)=O)CCN(C(=O)C(C(C)C)NS(C)(=O)=O)CC1CCO Fc1cccc2c1OCC2N=c1nc2scnc2c(NCCC=CBr)[nH]1 C(=O)(C(C)(CO)CO)Nc1c(C(=O)Nc2ncn(C)c2)scc1 C1(NC(CNC(C2(OC)CC2C)=O)=O)C2CC3C1C3C2C(=O)OC(C)C c1(C(N2C3CN(C(=O)Cc4ccsc4Br)C(C3)C2)=O)n[nH]c2c1CCCC2 C(Cc1ccccc1)(CC(=O)O)NC(c1n(C)cnc1)c1nnnn1C C1(C(=O)NC2CC(NC(C(C)(C)F)=O)C2)CC(=O)CC(=O)C1 c1(N2CCC(N(C(c3cc(C)[nH]n3)=O)C)C2)cc(CC(C)C)ncn1 C1(C(=O)NCC(C(C)C)NC(c2csc(-c3ccsc3)n2)=O)CC(C)(C)CN1C C(=O)(CC(CC)CC)NCC1(CNC(c2ncc(OCC)nc2)=O)CC(F)(F)C1 Cc1cccc(C(N2CC(N(C)C)C(CNC(C3(O)CC3)=O)C2)=O)c1Cl c1(NCC(=O)NC2CN(C(C(COCC)C)=O)CC2C)ccc(C#N)cc1 c1(C(=O)NCCCC(C)NC(C(CC(=O)OC)(C)C)=O)ccc2c(c1)SCCN2 c1(C(=O)NCC(C)(CO)NC(C(C)OCCOC)=O)ccc(-c2cn[nH]c2)cn1 N1(C(CCn2ccc(C)n2)=O)C2CCCC1CN(C(C1CCCNS1(=O)=O)=O)C2 c1(C(N2CCC(O)(C(CNC(C=CC)=O)C)C2)=O)cn(C(F)F)c(C)cc1=O C1(COC)CN(C(=O)Cc2ccc(C)o2)CCN1C(c1occc1F)=O C1(CSC)CCN(C(C2C=CCN2C(=O)CC2C=CCCC2)=O)C1 c1(C(=O)NC2C3CN(C(CC=C)=O)CC2CC3)nc2ccc(C(F)(F)F)cn2n1 C1(C=C)(C(=O)NCCC2CCCN(C(C3(C#C)CCCC3)=O)C2)CCOCC1 N1(C(C(CC)C)=O)CC2CCCN(C(=O)CCc3ccsc3Cl)C2C1 C(C)(CCCCNC(C1(CN(C)C)CC1)=O)NC(COCC(C)C)=O c1(C(=O)NC(C(=O)NC(CCCCC)C)C(C)(C)C)c[nH]c2ccccc12 N1(CCC(=O)N(CC(C)NC(C2(CC(C)(C)C)CC2)=O)C2CC2)CCCCC1 N1(C(Cc2nc(CC)sc2)=O)CC(NC(c2ccc(Cl)cn2)=O)C(C)(C)C1 c1(C(N2CCC(COC)(NC(=O)COC3CC3)C2)=O)c2c(nn1C)CCCC2 N1(C(CCc2c(C)nccc2)=O)CCN(C(=O)C(C2CCOCC2)C)CC1CO c1(C(N2CCCN(C(CC(CC(C)C)C)=O)C(C)C2)=O)cccc2oc(O)nc12 C1(C(N(CCC(=O)NC(CC(=O)OCC)C)CCO)=O)C2CC3C(C2)C13 CCC(O)CC(=O)N1CCC(O)(C(C)NC(C2CC2(Cl)Cl)=O)C1 CC(C)(CCCNC(=O)CC1(n2cccn2)CC1)C(=O)NCC1CNC(=O)CO1 N1(C(C(OC)OC)=O)CCC(C2CC2)C1CNC(C1CC(N=[N+]=[N-])C1)=O N1(C(c2nc(C)oc2)=O)CCC(NC(=O)CC2CCC2)C(C)C1 c1(COC(NOCCCOCC)=O)cc2sc([N+](=O)[O-])cc2s1 c1(C(=O)NC2CCN(C(C(C(CC)O)C)=O)C2C)ccc2nc(C)nc(O)c2c1 c1(C(=O)NC2(C)CN(C(CN(CCCCCC)C)=O)C2)cnc(C(C)C)n1C C(=O)(C1=NOC2(CCC2)C1)N1CCCN(C(CC(CCSC)O)=O)CC1 C(=O)(C(C(C)C)c1cccnc1)NCC(C1CC1)NC(c1n(CC)ccc1)=O c1(C(N2CCN(C(c3c(C)cns3)=O)CC2CO)=O)cnc2[nH]nc(O)c2c1 c1(C(=O)OC)cc(OC)c(S(=O)(=O)NC(c2ccccc2)C2CCOC2)s1 C1(C)(C(=O)NC23CCC(CN(C(CCC#C)=O)C2)C3)C2CC3CC(C2)CC1C3 c1(C(N(C2CCN(C(C3(OC)CCC3)=O)C2)C)=O)ccc(Br)c(C)n1 N1(C(C2CN(C)C2)=O)CC2(CC(C(=O)NCC(O)C(F)F)CO2)C1 c1(OC)ccc(C(N2CC3CC(C2)N3C(=O)CC2CCN(C)CC2)=O)c(Br)c1 C(C(C)(C)CC(=O)OCc1ccc(C(C)(C)C(F)(F)F)cc1)OC N1(C(C(C2CCC2)OC)=O)CCC(F)(C(N2CCCCC2C2CCC2)=O)CC1 C1(O)(CN(C(CCN(C(C)=O)C)=O)C)CCCN(C(c2ccccc2CO)=O)C1 N1(C(c2cccc(C#C)c2)=O)CCC2CN(C(=O)C=Cc3cn(C)cn3)CC2C1 N1(C(C=CC)=O)CCC2(COC(CNC(c3cccn3C)=O)C2)C1 N1(C(C(COC)N(C)C)=O)CC2(C1)CN(C(c1ccnc(C3CCC3)c1)=O)C2 c1(C(N2CCCC(O)(CNC(CCCC=C)=O)C2)=O)cncc2cc(Cl)ccc12 N1(C(C2CC(=C)C2)=O)CCC(NC(=O)C(F)Cc2ccccc2)C1(C)C c1(-c2cc(NC(c3c(O)cccc3F)=O)sc2)ccc(B(O)O)cc1 N1(C(c2cc(CC)no2)C(=O)NCC2CCOC2)CCCC(c2ccn(C)n2)C1 C1(CNC(c2c(NC)scn2)=O)CC(O)(CNC(C2CCN2C(C)(C)C)=O)C1 C1(C(=O)NCC2(O)CN(C(C3(SC)CCSC3)=O)C2)(N(C)C)CCCSC1 C1(OC)(CNC(=O)C(C)Sc2ccccn2)CN(C(=O)C(c2ccn(C)n2)C)C1 Cc1n[nH]c(C)c1CC(=O)NCC1C=CCN1C(c1cc(C2CCC2)[nH]n1)=O CCCC(CC(=O)N1CCCC(C2OCCO2)CC1)c1ccccc1.C1CSS1 c1(COCCN(S(Cc2c(C)ocn2)(=O)=O)C)ccccc1Br c1(C(N2CC(C(=O)NC(c3c(OC)cccc3)C)C2)=O)ccc(C)nc1C C1(C(N(C)CC2CCC(=O)N2)=O)CCC2(CC2)N1C(C1CC2CCC1CC2)=O C1(F)(C(=O)NCCOCCNC(C(CC(C)C)OC)=O)CS(=O)(=O)CC12CCC2 N(S(=O)(=O)N(C)Cc1csc(CO)n1)CC(C)N(C)C(=O)OC(C)(C)C c1(C2(CNC(C(c3ccccn3)C)=O)CC2)ccc(Cl)nc1 c1(OC)cc(C(N2CC(NC(=O)CCC(C)C)CC2C)=O)c(N)cc1F CC1COCC(C(N2CCOCC2CC(=O)NC(c2ccccc2F)C)=O)O1 c1(SCCC(=O)NCC2(COC)CN(C(=O)CSC)C2)ccccc1Cl Cc1cc(Cl)ccc1NC(C1CCCCC1NC(=O)CCC1CCC(=O)C1)=O c1(C(N2CC(OC)C2)=O)coc(CNC(c2ocnc2C)=O)c1 c1(C(N2CC(CNC(CCNC(=O)NC)=O)C2)=O)cnc(O)n1CC N1(CC(COC)(C)O)CC(C(=O)OC)CC(CNC(=O)OC(C)(C)C)C1 c1(C(N2CC=C(CNC(C3CCC4(CC4)C3)=O)CC2)=O)cnn2c1CCCC2 N1(C(CCNC(COC)=O)=O)CC(NC(C23CCCC(C2)OC3)=O)CC(O)C1 C1(CCC=C)(C(=O)NC(CC(=O)OC)C2CC2)CN(C(c2ncsc2NC)=O)C1 C=CCC(C)(C)CC(=O)NC1CC2CC(C1)N(C(c1cn3ncccc3n1)=O)C2 N1(C(CC)=O)CCC(C2CCN(C(c3cnn(CC(F)(F)F)c3)=O)C2)C1 C1(NC(CSC)=O)COC2(CCN(Cc3scnc3C)CC2)C1 CCC(CC(=O)N1CCCCC1C1(NC(c2oc(C)nc2C)=O)CC1)C1CCC1 C1(NC(COCCNC(C(COC)(C)O)=O)=O)CCCCNC1=O N1(C(C2C(OC)(OC)CC2)=O)CCC(C)(CCNC(C2CCCS2(=O)=O)=O)CC1 C(CC(CC)(CC)NC(C1CC(OC2CC2)C1)=O)NC(c1c(OC)cnnc1)=O C1(CC(=O)NC(C(C)NC(CCCN(C(C)C)C)=O)CO)C=NN(C)C1=O CN1CCC(C)(C(N2CC3CC(NC(C4CC(=O)NC(=O)N4)=O)C3C2)=O)C1=O C1(S(C)(=O)=O)(CNC(NC2C(C)C2)=NCCc2cnco2)CCCC1 Cc1conc1C(=O)NC(C(=O)NC1(C(C)C)CC1)C1CCCO1 N1(C(C(CC)(F)F)=O)CC(C2CCN(C(C3(CO)CCCCO3)=O)CC2)C1 c1(C(N(C2CC(NC(c3ccc(F)o3)=O)C2)C)=O)ccn(CC(F)F)c(=O)c1 c1(CC(=O)NCC(C)N(C(=O)CN(C)C)C)csc(-c2ccccc2)n1 C(=O)(CCCCN1CCCCC1)NCC1CC(CNC(c2n(C)ccn2)=O)OC1 N(C(=NCCSC)NCC(c1c(F)cccc1Cl)(C)C)C1CCN(C(=O)OC)C1 CC1CCCCC1OCC(=O)NC(C)(C)CCCNC(=O)CC1(C)CC(F)(F)C1 CC1CN(C(c2nncs2)=O)CC(C)CN1C(c1cc2ncccc2[nH]1)=O N1(C(C2CCCCN(C(C(CCSC)O)=O)C2)=O)CCc2nc(O)[nH]c2C1 C1(OC)CC(C(=O)N(C)CC2CCCN2C(c2cnns2)=O)CC1OC C1(C(F)(F)F)(C(N2CC(CCCCNC(COCC#C)=O)C2)=O)CCCCC1 CC1(C)CC(C(=O)NCC2(C)CCCN(C(=O)Cn3ncnn3)C2)CC1(C)C c1(C2N(C(c3scnc3Cl)C(=O)NCCCCCC)CCC2)cc(F)ccc1F c1(C(=O)NC2(CNC(C(CC)C#N)=O)CCCC2)cccc2c1CCCC2 c1(OCCCNC)cccc(COC2(CN)CCOC2)c1 N1(C(C(COCC)C)=O)CCN(C(=O)C=Cc2ccccc2C#N)CC(O)C1 C(=O)(CS(=O)(=O)CC(=O)OC)N1C2CCC(NC(C(C=C=C)C)=O)(CC2)C1 O=C(C#CC1CCOC1)NC1CC2CC1N(C(=O)C1=CCCC1)C2 C1(F)(CNC(C(CC)CC)=O)CCN(C(=O)CC2CCC(F)(F)CO2)CC1 c1(C(N2C(c3cccc(C)c3C)CCCC2)=O)ccc(S(=O)(=O)CCN(C)C)cc1 C1(CNC(C2N(C(C)(C)C)CC2)=O)C=CCN1C(c1cc(C(N)=O)c[nH]1)=O Cc1ccc(S(=O)(=O)NCCC(=O)N(C)CCNC(=O)C(C)CN(C)C)cc1 Cc1ncc(C(N2CCCCC(CNC(C3CCCC3C3CC3)=O)C2)=O)c(=N)[nH]1 CCC(CO)N(C(=O)C=C(C)CNC(=O)CC1CC(N(C)C)C1)C1CC1 C1(Cn2cc(C(C)NC)nn2)CCN(C(c2nc[nH]c2C(F)(F)F)=O)CC1 C1(C(=O)NC2(CCOCC)CCCC2)CN(C(=O)C=C(C)C(C)C)C2(CCC2)C1 N1(C(CNC(=O)NC)=O)CCCC(O)(CNC(C2(CF)COC2)=O)C1 N1(C(C2CCC(C)O2)=O)CC2(NC(=O)CCC(C)(C)F)CCC1CC2 C1(NC(c2c(C(=O)OC)[nH]cc2)=O)CCCC(NC(C2CCCS2)=O)C1 c1(C(=O)NC2C(C(=O)NC(C)(CO)C(F)F)CC=CC2)cccc2ccoc12 C1(NC(=O)CC2CC(C)(C)CO2)CCCCN(C)C1=O.C1(CC)CCN2C1C2=O Cc1csc2ncnc(NC3CN(C(=O)Cc4ccc(Br)cn4)CC3C#N)c12 CC1(C)CCCN(C(C2CN(C(C3(F)CC=CCC3)=O)CCN2C)=O)CC1 CC(C)C(CC(=O)N(C1CCSC1)C)NC(c1cc(C#N)cn1C)=O C1(CC=C)(NC(=O)CCC#CC)CCN(C(=O)CSC2CCOC2=O)C1 C1(C(=O)NCc2nc(C)c(Br)s2)CC(N)CC(C)(C)O1 c1(C(N2C(C)CCC(NC(C3CC4(CSC4)C3)=O)C2)=O)cnc2cccnc2c1 C1(CN(C(=O)CCC(=O)NC2CCSC2)C)CCC(C(=O)Nc2nccs2)CC1 c1(C(=O)NC2C(CNC(CN(C(=O)OC)C)=O)CC2)cncc(C(C)(F)F)c1 C(c1ccccc1)=CC(=O)NC1CC(C(N2CCCC(CCCO)C2)=O)C1 Cc1c(C(=O)NCC2CCCN(C(=O)CC3CCC(C)(C)C3)C2)ncn1C C1(C(=O)NCCC2(OCC)CN(C(C(CC(=C)C)C)=O)C2)Cc2ccccc2S1 C1(C(=O)NCCCNC(c2ncc(C(F)F)s2)=O)CC2CCCCN2C1 c1(OC)sccc1C(=O)NC(C)CN(C)C(c1cnc(Cl)[nH]1)=O N1(C(c2ccc(CNC(CC(COC)C)=O)cc2)=O)CCC(OC)C(C)(C)C1 c1(OC)ccc(SCCC(=O)NC2COCC2NC(C2CSC2)=O)cc1 c1(C(N2CCC(NC(c3cncc(CC)c3)=O)C2)=O)ccc(F)c(Br)c1 C(=O)(CCCC(=O)NCCCCCNC(=O)Cc1ncc(Cl)s1)OC(C)(C)C c1(CNC2C(C(=O)NC(CC)C)CCC2)cccc(-c2cccc(Cl)c2)c1 C#CCC(CC#C)C(=O)N1CCCC(CCNC(=O)CCOc2cccnc2)C1 C(=O)(CS(=O)(=O)c1ccccc1C)NC1C(F)CCN(C(CNC(CC)=O)=O)C1 CS(=O)(=O)c1cc(C(N2CC3CC2(CNC(=O)COC2CCCOC2)C3)=O)co1 c1(NC(CC)=O)cncc(C(N2C(CN(C)C(C3COCCO3)=O)CCC2)=O)c1 c1(C(N2CCC(N(C)C(c3cnsn3)=O)C2)=O)cc(Br)cc(F)c1F c1(CC(=O)NCCCNC(C2C=CC=CC=C2)=O)cc2nc[nH]c2cc1Br C1(NC(CCc2cccc(C)c2)=O)CC2CN(C(C3(O)CCCC3)=O)CC2C1 C1(C(N(C(CC)CC)CCO)=O)CN(C(c2nc(C)sc2C)=O)C(C)(C)C1 CC1N(C(c2c(CNC(=O)CN3CCCC3=O)nnn2C)=O)CCC1(C)C C(=O)(C1CCCc2scnc21)NCCC(CNC(C1CC2(CC2)C1)=O)O c1(NC(C2(C(=O)OC)CCNC2)=O)ccc(CC2(O)CCNCC2)cc1 CC1(C)CCc2nc(C(N3CCCC(O)(CNC(=O)CC(F)F)C3)=O)ccc2C1 C(=O)(C1c2c[nH]nc2CN1C(c1cccc(CO)c1)=O)NCC(CC(=O)OC)O c1(C(c2nnnn2Cc2ccccc2)NC(CSC)(C)C)nc(C(F)(F)F)cs1 C(C)(CNC(C1(O)CCC1)=O)(C(C)C)NC(c1cnc(C(C)OC)s1)=O C(=O)(C(CC(C)C)C(C)C)NCC(N(OCCC(=O)NCCSC)C)=O C1(N(CCCC)C(c2cc(OC)n[nH]2)=O)CCN(C(=O)C(C)NC(C)=O)CC1 C(=O)(C(O)Cc1cnc[nH]1)NC(CN(C(CCC)=O)C)CC N1(C(C2C(OC)CC2)=O)CC2CCN(C(=O)C=C(C)C)CC12 c12cccnc1CS2.CC1CCC(NC(c2cn(CCn3cccn3)nn2)=O)O1 CC1(C)CC(NC(=O)C(C)(F)C(C)(C)F)CN(C(c2ccccc2)=O)C1 c1(C(=O)NC2CN(C(C(C)C3CCCC3)=O)CC(F)C2)cnc2[nH]cnc2c1 N1(C(c2c(C)scc2)=O)CC(NC(c2cc(C3CC3)cs2)=O)CC12CCC2 C1(C(=O)NC2CC(NC(C3C(C(=O)OC)CC3)=O)C2)CCCCC12CCC2 Cn1[nH]c(C2CC(CNC(=O)CNc3ccccc3Cl)C(O)C2)nc1=O C(C)(CCCN=c1[nH]c(=NC2CCC(C)C2)[nH]c2cc[nH]c12)c1ccc(OC)cc1 C1(C(=O)NCc2ncc(C)nc2)CN(Cc2ccc(O)cc2)CCC1O c1(OC)cccc(C(=O)NCc2ccc(N(C)C)c(F)c2)c1OOC(F)F C1(NC(C2N(CCC)CCC2)=O)CN(C(=O)C(C)(C)n2cccn2)CC1F C1(CNC(C(CC=C)NC(C)=O)=O)CC2CCC1N(C(c1cc(Cl)no1)=O)C2 Cn1oc(C(N2CCC(c3cn(C(c4ccccn4)CCO)nn3)CC2)=O)cc1=O C(=O)(C1CCCc2ncccc21)N1CC2C(CNC(C3C(C)OC(=O)N3)=O)(C2)C1 c1(C(=O)NC(C)CCNC(C2CCCCO2)=O)ccc(F)cc1OC(F)F N1(C(C2C(CCC)C2)=O)CC2CCC2(CNC(c2cnc(S)n2C2CC2)=O)C1 N1(C(C=CCOC)=O)CC2CCC(Nc3nccc(C(=O)OC)n3)C2C1 C(=O)(C1COc2ccc(Cl)cc21)NCCC1CCCN(C(CSC)=O)C1 c1(C(N2CCC(NCc3ccc(C)c(F)c3)C2)=O)c[nH]c2cc(C#N)ccc12 CCCCC(C(=O)N(CCNC(c1ccnc(OCC)c1)=O)C(C)C)C(C)C C1(C#N)(CCC(=O)NCC(CC)NC(=O)C(CO)N(C)C)CCC1 c1(C(=O)NC(CNC(C(CCC)CC)=O)(C)CO)ccc(S(=O)(=O)N(C)C)o1 N1(Cc2nnc(C)s2)CCC2(CC1)CN(C(c1ncn(C(C)C)n1)=O)CC(C)O2 C12(NC(C=CCN(CC)CC)=O)CCC(CC1)N(C(=O)C(CCSC)OC)C2 CCCCCC(F)C(=O)NCC1CCCCN(C(c2cc(CO)[nH]n2)=O)C1 C(C(C)(CNC(c1cncc(CNC(=O)CCCn2cccn2)c1)=O)CO)OC Cc1nc(=NCC2C(C)CCCN2C(=O)Cc2ccc(F)cc2F)c(C#N)c[nH]1 C1(NC(C(COC)O)=O)CN(C(C2(OC)CC2)=O)CC1CC(C)(C)C N1(C(CCOCCN(C)C)=O)CC(CC(=O)NCc2n[nH]cc2CO)C2(CC2)C1 N1(C(c2ccc(C)cn2)=O)Cc2ccccc2C(NC(=O)CC2COC(=O)C2)C1 C1(NC(C2CC3C=CC2C32CC2)=O)CN(C(=O)CC2(O)CCC2)C2(CCOC2)C1 CC1=C(C)CC(C)(NC(c2[nH]ccc2CNC(=O)C(C)(C)CO)=O)CC1 O=C1CCN(CC2C3CCCC23)C(=O)N1CC12CCC(CC1)O2 C1(CC(=O)OC)CCC2(CCN(C(=O)C(=O)NCC(=C3CCCCC3)F)C2)C1 Cc1ccc(NC(C2(CNC(C3CC(=O)C3)=O)CC23CCC3)=O)cc1O c1(C(=O)NCC2OCCC(NC(C3N(N=O)CCC3)=O)C2)cc2n(n1)CCCN2 C(=O)(CCCCCC#N)N1CCCC(C)(CNC(c2ccc(C(C)C)nc2)=O)C1 c1(CNC(C2(OC)CC2)=O)cc(O)nc(CNC(c2cccn2C2CC2)=O)n1 C(CCC(C)(F)F)C(N1CCC(C2N(C(C(c3ccccc3)C)=O)CCC2)C1)=O CC1(C)CN(CCC2=CCCCCC2)CCC1NC(c1ccc(C(F)(F)F)s1)=O n1(CC)ncc(C(=O)NC(C)CNC(=O)CCC2CC(C)(C)CO2)c1C1CC1 N1(C(Cn2cc(C(C(=O)O)N(C)C)nn2)=O)CCN(CCC2CC2)CC1.NCC N1(C(C(C(C)C)O)=O)CCCC2(C1)CN(C(c1ccnn1-c1ccccc1)=O)C2 C(=O)(C1CCOc2c(F)cccc21)C(CC)CN(C(c1cc(F)n[nH]1)=O)CC.N Oc1ccc2c(c1)C(Nc1ncc(Cc3ccccc3)s1)CCC2 c1(CC(=O)NCCCC(CCC)NC(C(CC=C)C)=O)noc2ccccc12 c1(C(N2CC(F)(C(=O)NCc3cn[nH]c3)C2)=O)cc(F)c(F)c(F)c1F N1(C(C=CCOC)=O)CC2CCN(C(c3cnc(C(C)C)nc3C)=O)CC(C2)C1 C1(NC(C2N(CC#C)CCC2)=O)CN(C(=O)C(C)OCC2CC2)CC1C N1(C(C(CCC)C)C(=O)NC)CCn2c(nc(C(F)(F)F)c2Br)C1 C(=O)(CC(C)(C)C(C)=O)N1C(c2cn(CC3CCCCN(CC)C3)nn2)CCC1 C12(N)CC3CC1C2C3.C1(CC=O)CCC1NC(=O)C(=O)NCC1CC1 C1(NC(C(c2n(C)ccc2)=O)=O)CC2CC(NC(C3CCC(=O)N3)=O)CC2C1 CCC(C)(C)C(O)C(=O)NC1CCN(C(c2ccc(S(=O)(=O)N(C)C)o2)=O)C1C N1(C(=O)Cn2ncnn2)C2CCC1C(F)C(NC(C1(CCO)CC1)=O)C2 O=C(C(c1cccs1)=Cc1ccco1)c1ccccc1.C1(N)CCC1O C1(CNC(C=C=C(C)C)=O)CCN(C(=O)CCCC2CCC2)CC1(F)F C1(C(=O)NCCCN2CCC(NC(=O)C(Cl)=CCl)C2)OCCOC12CCC2 CC1(C)CN(C(=O)CC2(O)CCOC2)CC(CNC(=O)CCn2cc(Cl)cn2)O1 C1(C(N2CCCCC(NC(C3CCC(=O)C3)=O)C2)=O)CC2CCCC(C1)C2 CC1CC(NC(c2cc(-c3ccncc3)on2)=O)CN1C(C1CCCCO1)=O CN1CCC(C#N)(C(=O)NCCC(O)CNC(C2CCn3cncc3C2)=O)CC1 C12(CC(=O)NCC3(O)CN(C(CNc4cn(C)nc4)=O)C3)CCCCC1C2(F)F C1(NC(C2(C)CCCCC2)=O)Cc2ccccc2C1NC(C1(C)CC1Br)=O N1(C(c2nc(CCCCC)sc2)=O)CC=CC(NC(=O)C(C2CCC2)OC)C1 C(C(CC1CC1)C(=O)NCC(=O)NCC(F)F)NC(c1ccc(C)o1)=O c1(OC)cccc(-n2nc(-c3cncs3)nc2-c2cnc(SC3CCCC3)s2)c1 N1(C(CC)=O)CCC(CF)(NC(=O)C(C)n2ccnc2)C1 Cc1cc(C)n(CC(=O)NC(C2CC=CCC2)C(=O)NC(C2CSC2)C)n1 c1(C(N(CCN(C(c2cnn(C)c2OC)=O)CC)CC)=O)cncc2c1CCC2 c1(C(N2C3C(NC(CC4(C=C)CC4)=O)C(C3)C2C)=O)cc(F)c(Cl)cc1F c1(C(=O)NC2CC(CCNC(C3(n4cnnn4)CC3)=O)C2)cc(Cl)c[nH]1 c1(C(=O)NCc2c(CCNC(CC(COC)C)=O)ocn2)cc(C)c(Cl)cc1F c1(C(=O)NC2C(CNC(C(CCOC)C)=O)CC2)ccc2c(c1)C(=O)NCC2 C1(C(N2CCC(C(=O)OC)C2)=O)CCC2CCC1N2C(=O)C=CCO NS(=O)(=O)CCCC(=O)NCC(F)CNC(=O)CSCc1ccncc1 CCC(C)C(C(=O)N1CC(n2cc(-c3ccn(C)n3)nn2)C(SC)C1)OC C1(C(N2CC(NCc3c(OC)ncc(F)c3)C(C)C2)=O)CCC2CCC(=O)N2C1 Cc1scc(C(=O)NCC(C(C)C)NC(c2ccc(C(F)(F)F)o2)=O)c1C c1(OC)cnc(Cl)cc1C(N1CCOC(CNC(=O)CC2CCCOC2)C1)=O N1(C(c2cnc(CC)o2)=O)CCCC2C(NC(=O)Cc3cncn3C)C(C)(C)C12 N1(C(C2CCC(NC(c3c(C)cns3)=O)CC2)=O)CC2OCCN(C)C2C1 CCC(C)(CO)C(=O)NCC1(CNC(c2ccc[n+]([O-])c2)=O)CCCCC1 C1(N(C(c2c(CC)csc2)=O)C)CCN(C(=O)CCN(S(C)(=O)=O)C)CC12CC2 C#CC1(NC(=O)COC(=O)Cc2cc(C(C)C)nc(O)c2)CCCC(C)(C)C1 CC(C(=O)C(=O)C(C)N(CC(F)(F)F)C)=CCNCC(C)NC N1(C(CC(C)(C)SC)=O)CC2(CNC(c3cnc(C)nc3)=O)CC1CCO2 CCCC(CNC(=O)C=Cc1cccnc1)C(=O)NOCCOCC C12(C(=O)NCC(c3cccc(Br)c3)(C)C)CC1CN(C(c1nc(Br)cs1)=O)C2 N1(C(=O)NC(c2cc(Cl)cnc2F)CC)CCSC2COCCC12 C(=O)(C#CC1CCOC1)NCC1(NC(c2c(CN(C)C(N)=O)nccc2)=O)CC1 c1(C(=O)NCC2C(NC(C(Br)=C(C)C)=O)CCC2)cc2c(nc1N)CCC2 c1(C(N2CC(CCNC(C(CC)C(=O)OC)=O)C2)=O)ccc(Cl)c2ncccc12 c1(C(N2CCC(CCNC(Cc3ccn(CC)n3)=O)C2)=O)cnncc1NC c1(NC(C2(NC(C(F)=CCC)=O)CC2(C)C)=O)ccc[n+]([O-])c1 c1(C(=O)Nc2c(C(=O)NC(c3ccccc3F)C)n[nH]c2)cc(Cl)nc(Cl)c1Cl C#CCC(C)(CC)C(=O)NCCSCC(N1CCCC(OCCC)C1)=O C1(CC(N2CC(NC(C(=Cc3cnc[nH]3)C)=O)C(C)C2)=O)CCC(C)(O)CC1 c1(OC)cccc2c1OCC(C(=O)NCCCc1cn(C3CCOC3)nn1)C2 C1(C(=O)NCC(CNC(C2C(CCC)CCC2)=O)(C)C)(COC)CC2(CCC2)C1 N1(C(c2scc(C)c2Cl)=O)CCC(CNC(c2ccn(CCO)c2C)=O)C(C)C1 N1(CC(=O)NCC(C)NC(=O)CNc2cccc(O)c2)CCS(=O)(=O)CC1 N1(C(C(C)C2CC2)=O)CC2CCC1C(CNC(c1coc(S(C)(=O)=O)c1)=O)C2 CC1(C)CC(C(N2CCC3C(NC(=O)CSC(F)(F)F)C23)=O)CCO1 N1(C(=O)CCc2cnc(O)[nH]2)CC2CCCC(C1)N2C(=O)C(CO)C(F)(F)F N1(C(c2ccncc2O)=O)CCC2CCN(C(c3c[nH]cc3Br)=O)CC2C1 C(CCCC(CO)NC(C1CC2CC2C1)=O)NC(CCc1c(C)nn(C)c1)=O c1(COC)c(C(=O)NC2COCCC2NC(c2ccsc2C)=O)cnn1C c1(C(=O)NC(C)CCCNC(=O)Cc2cncs2)ccc2nc(CO)[nH]c2c1 N1(C(C(c2ccncc2)C)=O)CCCC2(CCN(c3ccnc(C#N)n3)C2)C1 c1(C(N2CC(C(C)NC(c3nnc(S)n3C)=O)C2)=O)c(F)ccc2[nH]ccc12 N1(C(C(F)OC)=O)CC(NC(C2(C)CNC(=O)C2)=O)CC2(CC2)C1 C12(CNC(C(CC=C)(F)F)=O)CCCCC1CN(C(C1CCC1(C)C)=O)C2 C(=O)(C1CC(=O)Nc2ccc(Br)cc21)N1Cc2c(ccc(C(=O)OC)c2)C1 CC1(C)C(C)(C(=O)NC2CC2CNC(=O)C2=C(Cl)CC2)C1(C)C C1(OCC)(CNC(=O)CC2CCC(O)C2)CN(C(c2coc(Cl)c2)=O)C1 c1(NC(C(CNC(c2[nH]cc(C(C)=O)c2)=O)O)=O)cc(CO)cc(C)c1 N1(C(CCOCC#C)=O)CC(C)(C)CC1CC(N1CCN(C)CC1CO)=O C1(CNC(C(C)NC(N)=O)=O)CN(C)CCN1C(=O)CNC(c1cccs1)=O Cc1ccc(F)c(CN2CC=CC2C(=O)Nc2ccc(Cl)c(O)c2)c1 CCCCCCC(CC)C(=O)NC1(C)CC(NC(=O)C(F)C(C)(C)O)C1 CC1(CC(=O)NCC2CCOC2C(N2CCC(C(F)F)C2)=O)CCOC1 N1(C(C2CC3(CC3)C2)=O)CC(C2CC2)(C(N2CC3CC3C3CC23)=O)C1 n1(CC(=O)NC2C(NC(=O)COCc3ccncc3)C2)ccccc1=O C(C(C)(O)CNC(=O)CC1(C2CC2)CC1)NC(CN(C1CC1)CC)=O CC1CC(n2nc(-c3ccccn3)nc2C(C)CCc2cccc(Cl)c2)CCO1 C12(C(N(C3CCC(NC(c4cccc(C)c4)=O)C3)C)=O)CCC(CC1)C2(C)C c1(C(=O)NCC2(C)CCC(NC(=O)CCc3cnn[nH]3)C2)cn2ccsc2n1 C1(CNC(COCCCOC)=O)CN(C(C23CC=CC(C2)OC3)=O)CCC1(C)C c1(CC(=O)Nc2cc(CO)ccn2)cccc2ncccc12 CC1(C)CCC(NC(=O)C(N)CC2OCCO2)C1 c1(NC(C2CC(C)(N=c3[nH]ncs3)C2)=O)ccc2c(c1)NC(=O)C1CCCN21 c1(C(N2CCC(CC(=O)N(C)Cc3nc[nH]n3)C2)=O)cnn(C(C)(C)C)c1N Nc1c(C(N2CCOCC2c2nc(C(F)(F)F)n[nH]2)=O)cccc1I C1(C(=O)NC(CC=C)CC)CCN(C(C2CC(CF)C2)=O)C12CCC2 c1(C(=O)NC(C2CCN(C(=O)C(C)(C)CN(C)C)CC2)C)ncc2[nH]ncc2n1 C1(C(=O)NC2CC(C)(C)N(C(c3cccc[n+]3[O-])=O)C2)CCCC2(CCC2)O1 Cc1scc(C(=O)N(C)CCNC(=O)CCC2CCC(=O)N2)c1Br S(=O)(=O)(c1ccc(N2CCC(CN(C)C)C2)c(F)c1)NCCN(CCC)CCC Cc1ccc(CC(=O)NC(C)(CNC(C2CCC2(C)C)=O)CO)s1 C1(C(N2C(C=CC(=O)NCCC3OCCO3)CCC2)=O)CC2(CCCO2)C1 C1(NC(Cc2c(C)ccs2)=O)CCN(C(=O)Cc2cc(C3CC3)no2)CC1O C(C(C)(C)CN(C(=O)CC(C)O)CC)NC(C1(CC#C)CCC1)=O C1(NC(c2nc(CC)sc2)=O)CCN(c2nc(Cl)ncc2C)CCC1CO c1(C(=O)NC2CCN(C(=O)CCc3cccnc3)CC2F)cnn2ccccc12 c1(OC)ccccc1NC(=O)C(c1ccc(C(N)=O)s1)N1CCC(C(F)F)C1 C1(NC(=O)C2=CCC2)CC2CCC(C1)N2C(c1c[nH]nc1C1CCCCC1)=O N1(CC(=O)NC(c2ccc(F)cc2)CC(=O)NCC(C)OC)CCN(C)CC1 Cc1c(NCC(C)CC(C)C)nc[nH]c1=NCC1CC2(C1)C(F)(F)C21CC1 C1(C(=O)NCC(CNC(c2c(OC)nccc2)=O)O)CCCN1S(=N)(=O)N(C)C C1(C(N2CCC(C(=O)OC)C2C)=O)CN(C(=O)Cc2cc(C)cs2)CC12CCC2 C1(C(N(C)C)=O)CC(F)(F)CN1C(c1cccc(N(C)C)c1)=O c1(C(N2CCC(CNC(CC(C(=C)C)O)=O)CC2)=O)cc(F)c(Cl)c(N)c1Cl C(=O)(C1=C(Cl)CCCC1)NCC1(F)CCC(CNC(C(=O)N(C)C)=O)CC1 C1(C)(C(N2CCCC(CCC(=O)NC(CC)C(=O)NC)C2)=O)CCC2CC2C1 N1(C(C(CCC)C)=O)CCC(C(C)C)CC1CNC(c1ncoc1C(C)(C)C)=O C12(C(=O)NC(CC)C3CC3)CC(CN(C(=O)C(C(C)O)N(C)C)C1)C2 C(N=c1cc(C#N)nc(C2CC2)[nH]1)C1(NC(C2CCCC(C)C2)=O)COC1 Cc1ccc(C(N2CCC(C(N3CC4CCC3C4)=O)C2)=O)cc1I Cc1ccc(-c2nc(NC(=O)C(=O)NCC3CC(=C4CC4)C3)sc2C)c(C)c1 N1(C(C)=O)CC(C)CN(Cc2cccc(C(F)F)c2C)CC1C C1(NC(=O)Cc2cc[nH]n2)C2COCC1CN(C(=O)C=CCN1CCOCC1)C2 N1(C(C=CCOC)=O)CCN(C)C(CNC(c2ccc(C)c(F)n2)=O)C1 C(=O)(C(O)C1=CCCCC1)NCC(CC(=O)NC1C2CCC(F)(F)C12)O Cc1cncc(C(=O)NC(C(=O)N(C)Cc2occc2C)C(C)C)c1 CC(C)C(CC(=O)N1CC(C)=C(C)C1)NC(c1nc[nH]n1)=O CC(C)(C#N)C(=O)NC1CCN(C(c2cnc(-c3cnccn3)s2)=O)C1 CC(N=c1nnn(C)[nH]1)C1CCCCN1C(=O)Cc1cccc(Cl)c1F Cc1c(C(=O)NCC2CCN2C(=O)CCCCC(F)(F)F)oc2c1C(=O)CCC2 C#Cc1ccc(Cl)c(C(=O)NCC2(F)CCN(C(=O)C(CCOC)OC)C2)c1 CC1N(C(C2CC(O)CN2C(C2CC(F)CN2C)=O)=O)CC(C)OC1(C)C N1(C(c2c(C)onc2)=O)CCC(CNC(=O)Cc2ccc(Cl)c(Cl)c2)C(C)C1 C(=O)(CCC=CC(C)C)NC1C(NC(C2(C(=O)NC)CC2)=O)C1 C1(NC(C)(C)C(=O)NC2(c3ccccc3)CCOC2)CCC(F)(F)CC1 c1(C(=O)NC2CCN(C(c3c(C)cc(C)o3)=O)CC2C)c(F)ccc(F)c1F N1(C(Cc2cc(C)on2)=O)CC2CC(C(=O)NCc3ccc(O)cc3C)C(C2)C1 C#Cc1ccc(C(=O)NCCC2CC(NC(=O)C(O)C3CCCC3)C2)c(OC)c1 C1(C(=O)NC(C)CC2(O)CCC2)CC2(C1)CC21CC1.C12(CCCC1)CCC(=O)N2 C1(CCC)CN(C(=O)CCc2cccc(OCC)n2)CCN1C(=O)C(C)C1CC1 C1(C(N2CCC(CCNC(C(C)NC(C)=O)=O)C2)=O)CCc2cnn(C)c2C1 c1(C(N2CC(CCCNC(C(C)N(C)C)=O)OCC2)=O)c(O)cccc1F S1(=O)(=O)c2cccc(c2)C(=O)N1.C(CCCC(=O)OC)N(C(CC)C)C(C)(C)C C#CC1(C(=O)NC(c2nocc2C(=O)OC(C)(C)C)C)CCN(C(C)=O)C1 N1(C(c2on(C)c(=O)c2)=O)CCC2C(C1)CN2C(=O)C1=CCCOC1 C1(c2n(C(C)(C)C)nnn2)(NCCCn2cncn2)CCC2C3CCC(C3)C12 N1(C(C(C(C)C)F)=O)CC(NC(=O)CSCc2ccc(F)cc2)CC12CCCC2 C(=O)(C(C)(O)C(C)C)N(CCNC(=O)C(=O)Nc1ccccc1SC)CC CC1(C)C(CNC(c2cc(Cl)sc2Cl)=O)CCN1C(=O)C=Cc1nccs1 CON(CCC(=O)NCc1cccc(C)c1)C(=O)c1n[nH]c(=N)[nH]1 N1(CC)CC(c2ccc(Cl)cc2)N=C1N1CCN(CCN(CC(F)(F)F)C)CC1 c1(C(=O)NCc2cc(-n3ccnc3)ccn2)ccc(CF)cc1 C(=O)(C(C)C1=CCCC1)NC(CC=C)CNC(c1ccn(C)c1C)=O C(=O)(C1=C(F)CN(C(C2CCCCC(=O)C2)=O)CC1)Nc1c(C(=C)C)cccc1 Cc1ccc2ncc(C(=O)NCC(C)CNC(=O)CC3CC3C3CC3)n2c1 C(=O)(C(CC(F)F)N(C(=O)C=CC1CCCN1C)C)NC(C)CC(C)(C)C N1(C(C(C2CC2)SC)=O)CC(C(=O)N(C2CSC2)C)CCC1(C)C c1(NC(C2N(Cc3ccc(C(C)(C)C)[nH]3)CCSC2)=O)c(Br)ccnc1Cl N1(C(C2C(C)(C)C2)=O)CCCC2(CC(NC(c3c[nH]ccc3=O)=O)C2)C1 C1(NC(C(COC)C)=O)CCCCC12CCN(C(C1CSCCS1)=O)CC2 C1(NC(CCOCCN(C(c2n(CC#C)cnn2)=O)C)=O)CN2CCC1(F)CC2 N1(CC)CC2(CCN(C(c3cc(C(F)(F)F)ccc3O)=O)CC2)CNC1=O C1(C(=O)NCCN(CC(C)O)C(=O)CSc2ccccc2O)CC12CC(C)(C)C2 C(S(=O)(=O)c1ccc(Cl)cn1)C1CN(C(c2n(C)c(-c3cccnc3)cc2)=O)C1 C1(C(=O)N(CCO)CCC2CC2)(N(C(=O)COC(C)CC)CC)CCOCC1 C1(C#N)(COC)CN(C(=O)CC2CCC(NC(=O)C(C)OC)C2)C1 CC1(CNC(C2(C)CCCOC2)=O)CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1 CCCCC(C)CCC(=O)N(CCN(C(C1CCC(N(C)C)CC1)=O)CC)CC N1(C(CCc2ccn(C)c2)=O)CC2C(CNC(c3ccc(CF)cc3)=O)C2C1 N1(C(CN(S(CC)(=O)=O)C)=O)CCC(C)C(CNC(c2cc(C#N)n(C)n2)=O)C1 C1(CC(N2CC(CCNC(c3nnn(C)n3)=O)C2)=O)CC2COCC12 N1(C(CCCN(C(C)C)C(c2ccc(=O)oc2)=O)=O)CCOC(C)C1 C(=O)(CCCC(N)=O)NCCCNC(C(N1CCCC(O)C1)C)=O C12(NC(CCC=C)=O)CCC1CN(C(c1cc(-c3cccc(Cl)c3)no1)=O)C2 C(F)(C(=O)N(C)CCOCCCNC(=O)Cc1cnoc1)OC c1(NCC(=O)Oc2ccccc2C2CC2)ccc(N2CCOCC2)cc1C(=O)O C1(C)(NC(CCNC(COC)=O)=O)CCCCC1C(N1CCCCC1C)=O N1(C(c2scc(C#N)c2)=O)CC2OCC(NC(=O)CCn3cncn3)C2C1 c1(OC)ccc2c(ccn2CC(N2CCC(NC(=O)C=CS(C)=O)CC2)=O)c1 O=C1CC(C(=O)NC2(CCNC(=O)C(F)(F)c3cnccn3)CCCC2)CCN1 C1(C(N(CCCCN(C)C(C2(c3cccc(Cl)c3)CC2)=O)C)=O)CC(C2CC2)C1 C1(NC(C2C(OC)C2)=O)CN(C(c2coc(OCC(F)(F)F)n2)=O)CC1(C)C C1(C(N2CC(F)(C(=O)NCC3(F)CC(CO)C3)C2)=O)CCNC1=O N1(C(C(CC)SC)=O)CCCC(NC(c2ccc(OC(C)C)nc2)=O)C1 C1(NC(=O)CSc2ccncc2)CC2CN(C(=O)CCc3ccncc3)CC2C1 CC(CBr)C(=O)N1CCCC1Cc1cn(Cc2cnoc2C2CC2)nn1 C#Cc1ccc(C(N2CCCC(C)(C)C2CNC(=O)C(O)CCCC)=O)cc1F Cc1cc(C)n(CC(N2CCC(C(C)C(N3CCC(CN=[N+]=[N-])C3)=O)CC2)=O)n1 c1(NC(C(CNC(CCNC(COC)=O)=O)CC2CC2)=O)cnc(Cl)c(C)c1 c1(SC)ccc(Cl)c(C(N2CCC(N(C(=O)Cc3nncn3C)CCO)C2)=O)c1 c1(NCC2(O)CN(C(c3c(OC)noc3C)=O)C2)ccc([N+](=O)[O-])cn1 CCCCC(=O)C(=O)NCCCCNC(C1CCCC(C2CC2)O1)=O N1(C(C2C(C(=O)OC)C2(C)C)=O)CC2CC2(NC(=O)Cc2scnc2C)C1 c1(C(=O)NCC(C)NC(C(F)=CC)=O)cc(Cl)c2c(c1)OCO2 C(C(CC(C)C)C(=O)N(C)C)c1c(OC)c(F)ccc1.C1(C)C(=O)OCCO1 CC1=C(C(=O)NCCCC(C)NC(C2CC3C(C2)C3(F)F)=O)SCCO1 c1(C(=O)NCC=CCNC(c2cnn(C)c2Br)=O)ccc2c(c1)CCC2(F)F CCCC(C)C(=O)NC1CC1NC(C1(Cl)CC1C(=O)OC)=O N1(c2nc(C)nc(Cl)c2)CC(NC(C2OC(C)CC2C)=O)C2(CCOCC2)C1 c1(C(=O)NC(C2CCCN2C(C2CC(=O)N(O)C2)=O)(C)C)cn2ncccc2n1 N1(C(C)=O)CCC(N=c2[nH]c(C(C)(C)C)no2)C1 C1(NC(Cc2c(C)noc2C)=O)CN(C(c2ccnn2C)=O)CCC1C C1(CNC(CCCC(C)C)=O)CCC2CN(C(=O)CCN(C)C)CC12 c1(C2C(C(=O)NCc3ccccc3CC(F)(F)F)CC2)cccc(F)c1 c1(C(C)=O)cc(C(=O)NC2CCC2NC(C2(C3CC3)CC2)=O)ccc1Br N1(C(CC2(CC)CCC2)=O)CCCC(C(=O)N(C2CCC(O)CC2)C)CC1 C(C(CNC(c1cc(C2CC2)nn1C(C)C)=O)C(C)C)OC c1(C(=O)NCC(C(C)C)NC(C(C=C)(C)O)=O)cnc2onc(C)c2c1 c1(C(=O)OC)cc2c(N(CC(O)CN(C)C(C3CC(C)(C)C3)=O)C)[nH]cnc-2n1 C(=O)(C(F)CC(C)(C)NC(=O)C(CO)C(F)(F)F)NCC(CC)CC(C)C C1(C(c2nnnn2C)NC2C(c3cn(C(C)C)nc3)OCC2)(CCl)CCOCC1 N1(C(c2ccc(OCC)nc2)=O)C2CCCC1CC(N(C)C)C2 C1(CC)CN(C)C(=O)CN1C(=O)CCCCCN(C)C(C1CC(=O)N(OC)C1)=O CCS(=O)CC(=O)NCCCN(C(c1cccc(-c2noc(C)n2)c1)=O)C1CC1 C1(C)(C(=O)NCCC2(C)OCCO2)CC12CCN(c1nccc3occc13)CC2 Cn1ncc(C(=O)NC2CCCC2(C)C)c1F N1(C(CCCN(C(C)=O)C)=O)CCC(C)C(CNC(=O)CNc2cnn(C)c2)C1 C(CCCCC(=O)NCC1CCO1)N(C)C(c1coc(C(N)=O)c1)=O c1(CC)c(C(=O)NCCC(C)NC(=O)C(C(C)C)c2cnn(C)c2)csc1C C1(NC(C(c2ccccc2F)OC)=O)CC2(C1)CC2NC(c1cncc(C)n1)=O c1(OC)ccc(C)cc1C(=O)NCC1CC(NC(=O)C=C2CN3CCC2CC3)C1 c1(OC)ccc(C(N2CCCC2CC(=O)NCC2C3CCCOC23)=O)nn1 CN1CCOc2ccc(C(N3CCC(CCNC(=O)C(F)=C4CCC4)C3)=O)cc21 C1(CNC(C(C)C2CCCC2)=O)CCN(C(c2nnn(C)c2N)=O)C(C)C1 Cc1[nH]c(C)c(C(=O)NCC2CCC2NC(c2nc(Br)c[nH]2)=O)c1C Cc1cc(C)n2nc(C(=O)NC3(C)CCC(NC(C45CCC4C5)=O)CC3)nc2n1 N1(C(C(CC)C)=O)CCC2(CC1)CC2NC(c1cc(F)ccc1C)=O C=C(Br)CCC(=O)NC(C1CCN(C(=O)C(C)n2ccnc2)CC1)(C)C C1(NC(C(CCOC)NC(=O)CCC2OCCO2)=O)CCc2nncn2C1 N1(C(CCS(=O)(=O)NC)=O)CCC(C2CC2)(CNC(c2cn3c(n2)SCC3)=O)C1 C1(C(=O)NCC(c2ccccc2)F)COCCN(C(c2c[nH]cc2C2CC2)=O)C1 c1(CCNC(c2nc(C)nn2C)c2nnnn2C2CC2)c[nH]c2cccc(F)c12 N1(C(C(C)SC)=O)CCCC(NC(=O)CN(CC(=O)NCCOC(C)C)C)C1 CC1CN(C(=O)CCOCC(F)F)CC1CC(=O)N(CCO)CCn1cccn1 C1(C(=O)NCC(C)(C)CNC(=O)C(O)C(C)SC)(CC)CCC(O)CC1 c1(C(N2CC3(CCC(C(=O)NCC(C)(C)C)O3)C2)=O)cc2ccc(Br)cc2s1 CC1(C)OCCC1CC(=O)NCC1CC(NC(=O)CSCc2cscn2)CC1O N1(C(CC(C=C)CC)=O)CC2CC3CC2C1C3NC(=O)C(CO)C(C)(C)C N1(C(c2cn(CCCC)nn2)=O)CC(NC(=O)C(CC)SC)C2CC2C1 Cc1noc(C)c1C(CC1CCCC1)NSC[Si](C)(C)C Nc1nn2ccccc2c1C(=O)NC1CN(C(C2C3CCCCC23)=O)CC2CC12 Cc1ccc2occ(C(N3CCC4CCN(C(=O)C=CCF)CC34)=O)c2c1 c1(OC)ccc(F)cc1C(N1CCCC(N(C(=O)COCC(F)F)C)C1)=O c1(NC(C(N2CCC(C(=O)NCCC)C2)=O)=O)c(OCC)ccc2c1CCC2 C1(C(=O)NC)(CF)CCN(C(c2ccc(OC)nn2)=O)C1 N1(C(CCN(C)C)=O)CCCC1CC(N1CC(C)(CN(C)C)C1)=O c1(C(=O)NCCC(C)NC(CCc2cnc(C)o2)=O)cnc(Br)c(N)n1 Cc1ccc(CCC(=O)NC(C(=O)NCCOCC(N)=O)C2(O)CCC2)o1 N1(C(C2N(C)CC2)=O)CC2CC(C1)CN(C(C1(C)CCCO1)=O)C2 c1(OC)cccc2[nH]c(=NC(CN3C=CS(=O)(=O)C=C3)C(C)C)sc12 C=CC1(C(=O)OC)CCN(CCCCO)C1 N1(C(CCCSC)=O)CC2(CNC(=O)CCc3nccn3C)CC1CCO2 c1(C(N2CC(C)CC(NC(C(C#C)(C)C)=O)C2)=O)ccc(F)c2c1CCC2 C1(NC(C(C(C)C)OCC)=O)CCC2(CCN(C(=O)Cc3ccco3)C2)C1 C1(C(=O)NC2CC(CNC(=O)CC(C)c3cccnc3)C2)(OC)CCCCC1 C#Cc1ccc(C(=O)NCCC2CC(NC(C3C=CCC3)=O)C2)cc1C Cc1ccc(Cl)c(O)c1C(N1CC2(COC(CNC(c3cocn3)=O)C2)C1)=O c1(C(=O)NC(C)CCN(C)C(C2COC(=O)O2)=O)cnc2n(c1=O)CCS2 c1(NC2(C3CN(C(C(C)(C)N4CCCCC4)=O)C3)CC2)ncc2c(n1)CCOC2 c1(C(=O)NCC(CCNC(=O)CCCn2cncn2)OC)cccc(F)c1 c1(CC)cnc(C)c(NC(=O)C(C)(C2CC2)N(C(=O)CSCCC(C)C)C)c1 C1(C(N2CC(C(=O)NC3(C=C)CCCCC3)C(C)(C)C2)=O)CC(C)(C)OC1(C)C Cc1cc(NC(=O)C(C)C(=O)O)ccc1-n1cc(C2CCCC2O)nn1 CC(C)(C)C(C)(C)C(=O)N1CCC(C)(CNC(C2CN(S(N)(=O)=O)C2)=O)C1 N1(C(c2cc(C)cc(F)c2)=O)CC(NC(C2C(C)C2C)=O)CC12CCCC2 C1(C(N(C(CNC(Cc2nc(CC)sc2)=O)C)C)=O)CC(C)(C)CCO1 CCCC(CCNC(=O)C1=NOC(CNC(C2CC=C(C)CC2)=O)C1)CCC S(=O)(=O)(c1c[nH]ccc1=NCC1CCCOC1)NC(c1ccc(Cl)cc1)C C1(CNC(C(=O)NC(C2CCCC2O)C)=O)CCN(c2ccccc2)C1 C1(CC(=O)NC2CCN(C(=O)CC3(C)CC3(F)Cl)CC2)(CN(C)C)CCOCC1 Cc1oc(CNC(=O)CC2CNC(=O)O2)nc1C(N1CCCC1(C)C(C)(C)C)=O N1(C(C2(OC)CCCC2)=O)CCC(C)C(CNC(C2(F)CCCC2)=O)C1 C1(OCCC)CCCN(C(=O)NCCCCCCN(C)C)C1 c1(OC)cc(OC)c(C(N2CCN(C(=O)Cc3ccsc3)C(C(F)F)C2)=O)cn1 c1(OC)ccc(CC(N2CC3(NC(=O)CC4CC(OC)C4)CCC2C3)=O)c(C)c1 C=CC(CCC)CC(=O)N1CCC(C)(NC(=O)CC2C=CCC2)CC1 C(=O)(CCC(=O)N1CCC(C(C)C(=O)NCC(C)(CC)OC)C1)OCC C1(C(=O)NCC(CC)(CC)NC(=O)C#CC(C)(C)O)CCc2cncn2C1 c1(COCCOC)ccc(C(=O)NCC(C)N(C)C(C2(C)C=CCC2)=O)cc1 C(CC(=O)Nn1ccnn1)(C(C)(C)C)NC(c1c(C)cc(C)s1)=O c1(C(N2C(C#N)C3CC3C2)=O)cc(-c2cc(F)cc(F)c2CO)c2[nH]ccc2c1 c1(C(=O)NC(C)C)cccc(NC(=O)NCCC(O)C(=O)O)c1 C(CCC(O)C(=O)NCC1(CO)CCOC1)NC(C1(OC)CCCCC1)=O N1(C(c2c(C)ccc(C)n2)=O)CCN(C(=O)Cn2cnnn2)C(C)C1C N1(C(=O)NCC(=O)OCC)CC2CN(C(c3ccnnc3C(F)(F)F)=O)C2C1 c1(CN(C2CCN(CC)C2)C(=O)CCn2cc(C(C)O)nn2)ccccc1Br CC1CCC=C1C(=O)N1CC(NC(c2ccc(OCF)cc2)=O)C2(CC2)C1 Cc1cc(C(N2CCC(C)N(C(c3nnsc3C)=O)CC2)=O)c(C)c(C)c1 N1(CCC(=O)NCC(CNC(c2c(CC)nccn2)=O)(C)O)CCP(C)(=O)CC1 c1(CC)cc(C(N2CCOCC(NC(c3csc4cncn34)=O)C2)=O)cc(O)n1 N1(C(C23CCC(OC)C2C3)=O)CCC(C(=O)NC(C(C)C)C2CCC2)CC1C C1(C2CCN(C(C3(CC=C)COC3)=O)C2)CCCCN1C(=O)CN1CCOCC1 c1(CCNC(C=CC(C)NC(=O)C=CC(C)(C)C)=O)noc(=O)n1C c1(C(N2CCC(NC(c3n(C)cnc3)=O)C(F)C2)=O)c(F)c(F)c(F)c(F)c1F c1(C(C2CC2)(Cn2cc(C3N(C(=O)CO)CCCC3)nn2)C)ccc2c(c1)OCCCO2 C(=O)(CCCC(=O)NCC)N1CC(CNC(COCC(=C)C)=O)C(C)C1 c1(C(N2CC(C)C(CNC(=O)C(O)C(C)(C)C)C2)=O)cc(F)c(CO)c(F)c1 c1(C(=O)NCC(CNC(C2(OC)CCCOC2)=O)O)cc2ccccc2nc1O Cc1nc(NCc2ccc3c(c2)CN(C)C3)cc(=NC(C)C2CCCC2O)[nH]1 N#Cc1c[nH]c2cccc(C(=O)NC3CC3NC(=O)C=Cc3ccc(F)cc3)c12 C(=O)(C(CC(C)C)C(N)=O)N1CCC(C(=O)NCC2C(OC)CC2)(CCl)CC1 C1(NC(=O)Cc2ccn(C(F)(F)F)n2)(CF)CCN(C(=O)CC2CSC2)C1 N1(C(c2ccc(SC)o2)=O)CC(NC(=O)CCC2CCCN(C)C2)CCC1C N1(C(c2c(CC=C)cccc2)=O)CC(C)(C)CC1CNC(C1CCCOC1)=O C(=O)(CC(C)(C)C(=O)N(CC(C)CNC(c1ccc(F)s1)=O)C)OC C12(C(=O)O)CCCC1(C(N1CCCC1Cc1ccc(Br)cc1)=O)C2 C=CCC(CNC(C1CSCCN1C(=O)C=C(C1CC1)C1CC1)=O)CC(C)C c1(NC(C)=O)ccc(Cl)c(CNC(N2CC(Oc3cccnn3)C2)=O)c1 Cc1ccc(CC(N2CC3C(C(=O)N(CC(C)C)C)C3C2)=O)cc1 c1(C(=O)NCC(C2(O)CCN(C(c3c(CC)scc3)=O)C2)C)cc([N+](=O)[O-])c[nH]1 c1(C(=O)NC(C2CC2NC(=O)COC2(C)CCC2)C)ccnc(Br)c1F n1(C(CC)(C)C)nnnc1C(c1ccncc1)NCCc1ccnn1C C(C(C)C(=O)N1CC(CNC(=O)Cc2ccc(C(C)=O)s2)C1)OCC c1(C(=O)NC2(CNC(c3cc(Cl)c[nH]3)=O)CC3CCC2C3)ccnc2ncnn12 n1(C(C)C(=O)O)cc(CN(CCCCC2CC2C)C(c2ncn(C)n2)C)nn1 C1(C(=O)NCCOCC(=O)NC)(CO)CCN(C(C2CC(C(C)C)=NO2)=O)CC1 Cn1cnc(C(N2C(C(=O)NCC3CC(C)(C)C3)CCC2C2CC2)=O)cc1=O c1(CC(N2CC(NC(C3N(C)CCCC3)=O)CC2(C)C)=O)c[nH]c2cccnc12 Cc1occ(C(F)(F)F)c1C(=O)NC1CCC(NC(=O)C=CC2CCCO2)C1 CC1OCCCC1C(=O)N(C)CCOCCN(C(=O)Cc1cccnc1)C C(C1=CCCCC1)NC(CC1(C)N(C(CC=CCCCCC)=O)CC1)=O c1(C(N(C(C(=O)OC)C)C)=O)ccc(C2CC2)s1.C12(CCCO1)C(=O)NC2 N1(C(C(=O)NCCC)C2CC2(C)C)CCCC2(CCCC2)C1 C(C(CCC)CCC)NC(C1C(NC(CCOCC#C)=O)CC1)=O C=CCCCC(C(=O)NC(c1nc[nH]n1)C)NC(c1ccc(C=C)cc1)=O CC(F)(F)C(=O)NC1(CO)CN(C(=O)CN2CCCC2CO)C1 c1(C(=O)NC2(C)CCN(C(c3ncsc3C3CC3)=O)C2)cc2ccccc2[nH]1 C(=O)(C(F)CCCC)NCC(CCCC)NC(c1cc(C)oc1CC)=O C(=O)(CCC(CC)CCC)NC(CC#CC)C(=O)NCC(O)C(=O)NC c1(C(N2CCOC(COC)C2)C(=O)NCCC(=O)OCC)cncc2ccccc12 C#CCC(CC#C)C(=O)NCCC(C)N(C(=O)Cc1cn(CC)nn1)C C(=O)(C(C)(C(C)C)OC)NC(C1CCN(C(CN(CCC#C)C)=O)CC1)CO c1(OCC=C)ccccc1C(=O)N(c1nnc(Br)n1C)CC C(=O)(C(CC(C)C)N(C)C(c1coc(C)c1)=O)N1CCC(OCC=C)CC1 c1(CC)ccc(C(=O)NC2CC(NC(=O)CCC=CCC=CO)C2)cc1Br c1(NC(C)=O)cccnc1C(=O)NCC(C)NC(=O)C(c1ccc(F)cc1)(C)F C(=O)(CC1=CCOCC1)N1C(C(=O)NCCCC2CC2)CC(O)C1 C1(CCNC(C2CC(=C)C2)=O)CN(C(c2ccc(-c3cnco3)cc2)=O)CCO1 CN=c1ccc(C(=O)N(C)CC2CCCN2C(=O)CSC(C)C)c[nH]1 CN1CCC(NC(=O)C2=CCCO2)C12CCCN(C(=O)C(C)(C)C(C)(F)F)C2 C1(Nc2ccc(NC(C(NS(NC)(=O)=O)C)=O)cc2)CC2CCC(C1)N2C(C)=O C(=O)(CCCCCC#N)NC(C(=O)NC1C(SC)CCC1)CCSN(C)C C1(CNC(c2cc(C)c(Cl)s2)=O)CCC(C)CN1C(c1cn2ccnc2s1)=O c1(C(N(CC(C)NC(CCCC(=O)OCC)=O)C)=O)ccc2c(c1)COCC2 C1(C(N2CCC(C(C)NC(=O)CCC3CCCOC3)CC2)=O)C2C3CCC(C3)C12 C(CC(C)(C)CC(=O)NCCC(C)NC(c1cnn(C2CCC2)c1C)=O)OC c1(CC)sc(=N)[nH]c1C(=O)NCC(C)(O)CNC(=O)Cc1cnccc1Cl c1(C(=O)NCCC(C)NC(=O)Cc2n[nH]cc2Br)ccc(F)c2ccncc12 N1(C(C2(C#N)CC3CC3C2)=O)CCOC2(CCN(C(C3CC(=O)N3)=O)C2)C1 n1(CC)nccc1C=CC(=O)NCCC1(NC(c2ccoc2Br)=O)CC1 C=Cc1cc(C(=O)NCC(C)CNC(c2cccc(F)c2C)=O)cc(F)c1 N1(C(C=C(C)C(C)(C)C)=O)CCC(O)(C2CCN(C(C3(C)CCC3)=O)CC2)CC1 CCCCC(C)(F)C(=O)N1CCN(C(C2CC2(Cl)Cl)=O)C(C)C1 C1(COC)(NC(=O)CCCn2ccnn2)CCN(C(=O)CC2C(=O)NN=C2C)C1 C1(NC(c2cncc(CC)c2)=O)CC(O)CN(C(c2ccc(CC)cc2)=O)C1 CCC(C)(C)CC(=O)NCC1(O)CC(NC(=O)CCc2ccoc2)C1 c1(CCC(=O)NC23CC(CNC(C(CC)NC(N)=O)=O)(C2)C3)ccc(Cl)c(C)c1 c1(C(=O)NCCNC(COc2cc(C)c(Cl)cc2)=O)ccc2c(c1)C(=O)NCC2 c1(-c2cc(C(N3CC(C)N(C)CC3)=O)sc2)ccc(O)c([N+](=O)[O-])c1 Cc1cc(C)c(C(=O)NC2(CO)CCCN(C(C3CCC(C)O3)=O)C2)cc1N c1(CC)ncc(C(=O)N(CCCN(C)C(C2CC3CC2C2CC32)=O)C)c(O)n1 NS(=O)(=O)CCCC(=O)NC1COCCN(C(C2CC2C2CC2)=O)C1 c1(OC)cc(C(=O)Nc2ccc(C)c(C)c2)cc(Br)c1OC c1(NC(C)(C)CCNC(=O)C(O)CCSC(C)(C)C)c(F)cc([N+](=O)[O-])cc1F C#Cc1ccc(C(N2CCN(C(=O)C(CC3CCCC3)C(C)C)C(C)C2)=O)nc1 N1(C(c2nc(C(C)C)sc2)=O)CCC2OCCN(C(=O)C#CC3CC3)C2C1 CC1CCN(C(c2cc(F)cc(Cl)c2)=O)C(CNC(=O)CNc2ncccn2)C1 C=CCCCC(N)C(=O)N1CCCC(O)(C(F)(F)F)CC1 N1(C(C2(C#N)C(C)(C)C2)=O)CCN(C(C2CCCCC(F)(F)C2)=O)C2(CCC2)C1 C1(C)(CC)CCCN(C(c2ccc(CNC(=O)CC3(NC(C)=O)CC3)nc2)=O)C1 C1(CN(C(c2cn(CC=C)nn2)=O)C)CCCCN1C(=O)Cn1nc(C)cc1N C1(CCC)CCC(O)(C(=O)NCCCC(C)(C)NC(=O)C(O)C(F)(F)F)CC1 C#CCC(C(=O)NC)NC(=O)C(Cc1cnc[nH]1)NC(c1cc(CC)ccn1)=O c1(CN(CCCN(CC(CCCCC)CC)C)C)cc(=O)oc2cc(C)ccc12 C(CCC(CCC)NC(=O)CC12CC(C1)C2)NC(C(C)SCCCC)=O c1(C(N2CCCC(C3N(C(COCC)=O)CCC3)C2)=O)cc2cc(Cl)ccc2[nH]1 c1(CC(=O)N(CCNC(C2COC(=O)N2)=O)CC)ncccc1F N1(C(C2C(CC)OCC2)=O)CCC2CN(C(c3cnccn3)=O)CC12 N1(C(c2c(C)c(Br)cs2)=O)CCCC(O)(CNC(c2cncn2C)=O)C1 CC(O)(C(=O)NCCCCNC(=O)CCC1CCCC1)c1ccccn1 c1(OC)cc(CNC(=O)NCc2ccccc2N(S(C)(=O)=O)C)ccn1 c1(NC(CC)CNC(C2(C)CCOCC2)=O)ncnc2sc3ccccc3c12 c1(C(=O)NC(C)CN(C)C(C2(n3cnnn3)CCOCC2)=O)cnc(O)cc1O C(=O)(C(O)CNC(C1CC(C)(F)C1)=O)N(C)Cc1cncs1 c1(C(=O)NCC2N(C(c3ccn(CC)c3C)=O)CCCC2)ccc2c(c1)OCO2 C1(COC(c2cccn2C(F)F)=O)CCC(Cc2ccncc2)C1 CCC(CCOC)C(=O)N1CC2CC2C1C(=O)CCNc1cccc(OC)c1 c1(C(C(=O)NCCOC)N(CCCO)C2CC2)nccc(Cl)c1Cl C12(CN(C3CC4CNC3C4)C(c3cnn(C)c3Cl)=O)CC1COC2(C)C C(=O)(C(C)CC(C)(F)F)NC1CCN(C(c2c(C)c(Br)cs2)=O)C12CC2 Cc1ccnc(C)c1C(=O)NCC(C)CNC(=O)CCn1ncn(C)c1=O C(=O)(C(C(C)(C)C)N1CCCC1=O)NC1C(NC(c2c(C(C)=O)nccc2)=O)C1 c1(CNC(C2C3CCCC23)=O)ccc2c(c1)CN(C(c1ccoc1)=O)C2 c1(N(C)C)nc(C(N2CC3(NC(=O)CCC4CC4(F)F)CCC2C3)=O)cc(O)n1 C1(NC(C(c2c(C)n[nH]c2C)C)=O)CC(C)CN(C(c2ccc(CO)nc2)=O)C1 CC(CCCCNC(=O)COC(F)F)NC(=O)CCC(=O)C1CC1 CC1CC(C(=O)NCCC2CC(NC(c3coc(Br)c3)=O)C2)CO1 C(O)(CN=c1cccc(S(=O)(=O)NCCCN2CCCCC2)[nH]1)c1n(C)ncc1 CCC(C)(C)C(=O)NCc1ncccc1NC(=O)C(CNC(=O)OC(C)(C)C)SC C1(CNC(CSc2c(C)n[nH]c2C)=O)CC(F)(F)CN1C(c1ncn(C)c1C)=O N1(C(c2n(CC)ccc2)=O)CCC(C)(C)C(C(=O)NCC(C)CC(C)C)C1 C1(C(=O)NCC(c2ccccc2)CNC(C(F)=C(C)C)=O)CCCN1CC(C)C Cc1cnn(C)c1C(=O)NC(C)(CNC(=O)CC1CC1(Cl)Cl)C(C)C N1(C(C(=O)NCC(C)C(=O)O)=O)CCCC(OCc2cn(C3CCCC3)nn2)C1 C(C(C)(C(=O)NCC1(F)CC(NC(c2cc(N)ccn2)=O)C1)OC)OC Cc1nn(C)cc1C1=NOC(C(N2CCCC2C(C)NC(=O)C=C(Cl)Cl)=O)C1 c1(C(N2CC(NC(C(COCC)C)=O)C3C(C2)C3)=O)noc2c1CCCC2 C1(CC)CN(C(C2COC3(CCC3)C2)=O)CCN1C(=O)CS(=O)(=O)N(C)C(C)C C=CCC(C)(C)CC(=O)N1CC=CC1CNC(=O)CCC(C)OC CC(CC(C)(C)C)C(=O)NCCC1CCN(C(=O)C(F)(F)CN(C)C)C1 c1(C(N2CC(CNC(CCCOCC=C)=O)C(O)C2)=O)coc2ccc(F)cc12 C1(NC(C2CC3CCC2CC3)=O)CC2CC1CN(C(c1c[nH]nc1C(F)F)=O)C2 c1(CC)nc(N(C2CCN(C(c3cnc(C)cc3Cl)=O)C2)CCO)c(C)c(Cl)n1 N1(C(C(C)OCCC#C)=O)CCC(N(CCC)C(c2cc(C(C)(C)C)on2)=O)C1 CC1CN(C(=O)CC(F)F)CC1CCNC(=O)C(C)NC(=O)OC(C)(C)C c1(C(N2CCC(N3CC(C)(C(=O)O)C3=O)CC2)=O)cc2ccc(F)cc2s1 C(=O)(CC(C)C(F)F)N(CCC(=O)NC(C)CCN(C)C)CCCO c1(CCNC(C(C)OC(c2cc(C(F)(F)F)n[nH]2)=O)=O)ccccc1 Cc1ccc(NC(=O)C(N2CCC(CNC(C3(C(N)=O)CCC3)=O)C2)=O)cc1C C1(NC(c2coc(C(F)F)n2)=O)C2CC1N(C(=O)Cc1cccnc1Cl)C2 C(CC(=O)NC1(c2ncc(C)o2)CC1)(C(F)(F)F)NC(c1nc(COC)oc1)=O c1(C(=O)NC2CN(C(C3C(C=C)C3)=O)CC2C)cc2cnn(C(C)C)c2nc1C C(=O)(C(CCc1ccccc1)OC(=O)COCC1CCC1)OCC c1(CC)cccc(CN2CC(C(C)NC(c3cnc(CC)s3)=O)C2)c1 N1(C(C(c2ccnn2C)C)=O)CCOCC(CNC(c2cncc(F)c2Cl)=O)C1 Cc1cc(C(=O)NC2CCC(CNC(=O)C(C)NC(N)=O)CC2)ncn1 c1(CCC(N2CCC(N(CCC)C(c3nocc3C)=O)C2)=O)ccc(C)c(C)c1 C1(C)(C(=O)Nc2c(CC)cccc2)CN(C(C2C3CC4C(C3)C24)=O)C(C)(C)C1 Cc1cc(NC(C2C3CC2N(c2cc(-c4ccccc4)ncn2)C3)=O)nc(C)n1 Cc1nn(CC(=O)NCC2CCN2C(C2CC3CC3CC2C)=O)c(=O)n1C C(C(N=[N+]=[N-])C(=O)NC(C(N1CCC(F)(C#N)C1)=O)C1CC1)OCC N1(C(C=CCC)=O)CCC2(CCCCN(C(=O)Cc3csc(C)n3)C2)C1 C(=O)(N=c1[nH]onc1C1CC1)c1cnc(NC(C2C(C(=O)OC)C2)=O)nc1 c1(-c2cnc(C(N(CC(C)C)CC(C)C)=O)nc2)ccccc1C#N c1(NC(C(CCSC)NC(c2cccc(F)c2Cl)=O)=O)cccc2c1CCO2 C12(CN3CCCC(COC(C)=O)C3)CNCC1COC2 N1(C(C(C)=O)=O)CCC2(CCC2NC(C2CCC(F)(F)C2)=O)CC1 c12cc(Br)ccc1C(=O)N2.N1(C(C2N(C(C)=O)CCC2)=O)CC(O)C(F)C1 Cc1cc(C(N2CCCC2CCCNC(=O)C(C(C)C)NC(N)=O)=O)c(C)s1 c1(NC(=NC)NCc2cccc(F)c2)cccc(S(=O)(=O)N2CCN(C)CC2)c1 C12(CNC(C(C)OC)=O)CC1CN(C(=O)COC1CCCOC1)C2 CCCCCC(O)CC(=O)N(CCN(C(=O)CC(CC)C(F)F)C)C(C)C c1(C(=O)NC(CN(C(c2nc(O)c(C)s2)=O)CC)C)ccc(F)c(F)c1C CC(C)C(CN(C)C)C(=O)NC1CCN(C(=O)C(N)=O)CC1O C1(C(=O)NCCC2(C(N(CC(O)CO)CC)=O)CC2)CCCCS1 Cc1cc(F)cc(Cl)c1NC(=O)CC1CCN(C(=O)Cc2cccc(Cl)n2)CC1 N1(C(C(C2CC2)SC)=O)CCC2C(C1)CN2C(=O)Cc1nocc1C C1(C(N2CCC2c2cn(C3CCCC=C3Br)nn2)=O)CN(C2CC2)CC2(CCC2)C1 N1(C(c2ccnc(Cl)c2)C(=O)NC2CCOCC2)CCOC2(CCSCC2)CC1 Cc1nnc2c(C(=O)NCC3(F)CC(CNC(=O)Cc4cnoc4)C3)cccn12 Cc1ccc(CN(C=O)Cc2ccc(O)c(Cl)c2)cc1C(F)(F)F N1(CC(=O)N(CC(C)NC(=O)C(C)n2ccnc2)CC)CCP(C)(=O)CC1 C#Cc1ccc(CC(N2CCCC2CN(C)C(C23CCC(CC2F)C3)=O)=O)cc1 N1(C(CC=C)=O)CC2(C1)OC1(C)CC2(NC(c2cc(C(F)(F)F)ncc2F)=O)C1 S(=O)(=O)(c1ccc(=NCC2CC2)[nH]c1)NC(c1cc(C)cc(C)c1)CC c1(C(C)C)cc(CC(=O)N(CCC(C)NC(=O)CCc2cnn(C)n2)C)on1 N1(C(C2C(=C)C2)=O)C2CCC1CC(c1cn(-c3cnn(C)c3C)nn1)C2 C(=O)(C(CNC(=O)C1=CCC(C)CC1)(CC)CC)N(CC#C)C c1(C(=O)NCC2(OC)CN(C(C3CN4CCN3CC4C)=O)C2)c(F)cc(F)cc1Cl c1(C(C)NC(=O)C(N)=O)ccc(CNC(=O)C(F)(F)CNN(C)C)cc1 Cc1c(Br)cc(Cl)c(NC(=O)CC2CCCN2C(c2ncccn2)=O)c1Cl C1(CNC(C(CC)=CCCC)=O)CCC(CNC(=O)C(C)Cc2cnc[nH]2)CC1 C1(C(=O)NC2COCCC2NC(C23CCC(CC2)C3)=O)CC2CCCC(C1)C2 C1(CNC(c2c(COC)scc2)=O)CCCCN1C(C1C(C(F)F)C1(C)C)=O N1(C(c2c(C(C)C)onc2)=O)CCCN(C(=O)CCSCC2CCCO2)CCC1 c1(C(C)=O)cnccc1C(=O)NCC(C)CNC(C1OCCOC1C)=O N1(C(c2c(N)c(F)ccc2F)=O)CCC2CC(NC(=O)CC3CSC3)CCC2C1 Cc1cc(C(N2CC(O)CC2(C)C(=O)NC2(c3ccsc3)CC2)=O)nc(O)n1 N1(CC(=O)NC2(C)CC(NC(CC(C)O)=O)C2)C(=O)NC2(CCOCC2)C1=O c1(C(=O)OC)csc(C(N2CC(OCCNC(=O)COC3CCOC3)C2)=O)c1 N1(CC(=O)OCC(c2c(OC)c(Cl)ncc2)=O)CCC(N=[N+]=[N-])CC1 CCS(=O)(=O)CC(=O)N1CCCC1(C(=O)NC1CC2(CCC2)C1)CC N1(C(CCCNC(CCSCCCC)=O)=O)CCC(C)C1(C)C C1(C(N(C)CCN(C)C2CC2)=O)CC(=O)CN1C(c1ncc[nH]1)=O N1(C(C(C)(Cl)CCl)=O)CC2(CC(C(=O)NC3CC3(F)F)CO2)C1 N(C(=NCCF)NC1CCN(C2CC2)CC1)Cc1cccc(C(C)O)c1 Cc1cc(C(=O)NCCn2cnc(C(=O)NCC(F)Cl)c2)nc(O)c1 C1(N2CCOCC(C(=O)OC)C2)CCN(S(=O)(=O)c2ccccn2)CCC1C N1(C(C(N2CCOCC2)C)=O)CC2CCCC2(Nc2nccc(C(C)(C)C)n2)C1 Cc1cc(C(N2CCCN(C(=O)C(C)NC(N)=O)CC2C(C)C)=O)c(O)nc1C CC1(C)CN(C(C2(F)CCNC2)=O)CCN1Cc1c(F)cccc1F N1(C(C(C)OCCOC)=O)CCC(NC(C23CCC(CO)(CC2)C3)=O)C(CO)C1 c1(CCC(=O)NCC23CC(C(=O)NC4C(C)(C)C4(F)F)(C2)C3)ccc2c(c1)OCO2 c1(OCC)cc(C(C)NC2CCCC(C)C2)c(F)cc1OC C1(C(=O)NC2CC(NC(c3csc(C(F)F)c3)=O)C2)CCCCS1(=O)=O CC1CCCN(C(=O)COC(c2cc(C3CCOCC3)nn2C)=O)CC1 N1(C(C2(COC)CCCCC2)=O)CCC2C(CCCN2c2cc(C)ncn2)C1 C1(CC=C)(C(=O)NCCC2CCC(NC(C3OCCO3)=O)C2)CCCCC1 c1(CC)cccc(C(=O)NC2CCC(NC(=O)C(C)(C(C)C)OC)CC2)c1N C(=O)(C1=Cc2ccccc2OC1)N1CC(N(C(=O)C#CC2CC2)C)C(C)(C)C1 C1(NC(c2cccc(SC)c2)=O)CCN(C(C2CC(=O)NC2(C)C)=O)CC1CO c1(CC(=O)NCC2(NC(Cc3n(C)ncc3)=O)CCC2)cc(C(F)(F)F)cc(Cl)n1 c1(C(N2CC(OCC)C(c3cn(C4CCCCC4)nn3)C2)=O)cc(F)cc(Cl)c1 N1(C(C(C)=C(CC)C)=O)CCOC(C(=O)NCC(C)(C)C(C)O)C1 N1(C(CSC)=O)CC2CC2(CNC(C2CCC2C(C)(C)C)=O)C1 C1(C2CC2)(CNC(=O)CCC2CCCO2)CCN(C(c2cnc(C(F)F)s2)=O)C1 c1(C(N(CCCNC(C(C=CC)O)=O)C2CC2)=O)nccn2nccc12 N1(C(CN(S(CC)(=O)=O)C)=O)CC(F)(F)CC1CNC(c1nocc1C(C)C)=O c1(C(=O)OC)c[nH]c(=NCC2CN(C(C3COCCO3)=O)CC2C)cc1[N+](=O)[O-] C(=O)(C1CCc2c[nH]nc21)NC1CCCCN(c2nc(C)cc(CSC)n2)C1 CCC(O)C(C)C(=O)NC1CC(F)(CNC(c2cnn3ccsc23)=O)C1 c1(C(=O)NCC2CCC(C(=O)OCC)C2)ccc(OC)c2cnccc12 c1(C(=O)NC(CNC(c2ccc(COC)s2)=O)C)cn2c(n1)CCC2 C1(NC(CCCC)=O)CCN(C(C2CCOC2C)=O)CC1 N(C1CN(C(=O)C=Cc2cccs2)Cc2ccccc21)C(C1C(C)C1C)=O N=c1[nH][nH]c2cc(C(N3CCC34CN(C(=O)OCc3ccccc3)C4)=O)ccc12 Cn1nccc1C(C(=O)O)NC(=O)CCNc1ccccc1 c1(N(C(C2CC(S(C)(=O)=O)CN2)=O)CC)cc(F)c(C#N)cc1C C1(NC(c2c(C)cco2)=O)C2CN(C(=O)CC3CCCC3C)CC12 C(=O)(C(O)CC(N)=O)NCC1CC(NC(CCN(C)C(=O)OC(C)(C)C)=O)C1 N1(C(c2ccc(C(OC)OC)o2)=O)CCC(NC(=O)C(O)CC(N)=O)C(C)C1 Cc1nc(C)c(C(=O)NCC2(C(=O)NC3CCCC3C)CC2)s1 CC(C)CC(F)(F)C(=O)NCCC1CCCCN1C(c1cccc(F)c1N)=O C1(C(N(C(C)C)CCNC(=O)CCC(N)=O)=O)CCC2CC1CO2 C1(C(=O)NC(CC)Cn2cncn2)(CNC(=O)COCC(=O)OC)CCCCC1 N1(C(C2(CCOC)CC2)=O)CCC(CCNC(C2CCC2C(N)=O)=O)CC1 c1(NCC(CC)CCO)ncnc(NCC(C(C)CC)OC)c1C C1(NC(=O)CCc2nncs2)CC2(C1)CC(NC(=O)C(=CC1CCCCC1)F)C2 c1(-c2cccc(C(C)=O)c2)cncc2sc(C(=O)Nc3ncc(F)cc3Cl)cc12 N1(C(CSSC)=O)CC23CCCC2(C1)CN(C(=O)C(C(C)C)NC(N)=O)C3 c1(C(C(=O)NCC(CO)NC(C2N(CCC)CCC2)=O)(C)C)ccc(C#N)cc1 N1(C(C2(OC)CCOC2)=O)CCC(C(=O)NCCCCCCF)CC1 c1(CC(=O)NC2(CC=C)CN(C(C3CNC(=O)N3C)=O)C2)nccc(OC)n1 c1(-c2cn(C(COCC)C(=O)NC(C)(C)C(N)=O)nn2)cccc(O)c1 C(=O)(C#CC1CCOC1)NC1CN(C(C(C)CSc2ccccc2)=O)CC(F)C1 C(=O)(C(C)CS(C)(=O)=O)NCCCC1CCN(C(C(n2c(C)ncc2)C)=O)CC1 C1(OC)C(NC(=O)CC2(N(C)C(C3OCCC3(C)C)=O)CC2)CC1(C)C C12(CC(N3CC(CCC)OCC3)=O)CCC1CN(C(C1(CO)CCCC1)=O)C2 N1(C(C(C)(C)c2ccno2)=O)CCCN(C(=O)C(c2cccnc2)O)CC1 C(=O)(C(O)CC(F)F)NC(CCCC)CNC(=O)C=Cc1cc(C)no1 Cc1cccc(C(=O)NCC(C)(C)CNC(c2cnc(O)c(Cl)c2)=O)c1Cl N1(C(C(c2n(C)ccc2)=O)=O)CCC(C=CC(N2CCCC(C)(C)C2)=O)CC1 C1(CN=C(NC(C2CC2C(F)(F)F)C)NCc2ccco2)CC2C=CC1CC2 N1(c2cccc(C(C)C)n2)CCS(=O)(=O)C(C)(C)C1 c1(CC(=O)NC2CC(NC(=O)CC34CCC(CC3)C4)C2)cc(O)nnc1O c12ccc(cc1F)-c1cscc1N2C(=O)NCCC.c1(NC)ccc(C)cc1Br C(=O)(CC(O)C(=O)NC1CC1NC(C1CCC1)=O)OC(C)(C)C c1(C(N2CCN(C(CSCCC#N)=O)C3C2C3)=O)ccc2nc(O)oc2c1 c1(C(=O)NCC(C)(CO)NC(=O)CC2CCCN2CCF)cc(Cl)c(Br)[nH]1 CC(CC(=O)N1CCCC1)N(C(=O)CCN(C(=O)C(C)Cn1ccnc1)CCO)C C1(CC(N)=O)(NC(CCOCCC)=O)CCN(C(=O)C(CO)N(C)C)CC1 C(=O)(C(CC)(CC)CO)NCCC(C)NC(C=CC(CC)C)=O C1(C)(NC(C2CN(C)C2)=O)CN(C(=O)C=CC(=O)N(C)C)C1 CC(C)CC(C(=O)N1CCOC(C(C)C)C1)NC(=O)CCCn1cccn1 C(=O)(CS(=O)(=O)c1ccc(C2CC2)cc1)N(C1COC2(CCNC2)C1)C c1(CC(=O)N(C2CCN(C(c3nnnn3C)C)C2)CC)cncn1C c1(NCc2n(C)cnn2)cnc(Cl)c(Cl)c1.N12CCN(CC1)C1(CC1)C2=O Cc1ccc(C(=O)NCC(C)(C)CCNC(=O)CC2CCC(C)C2)c(C)c1 c1(CC(=O)NCC2(F)CC(NC(CSCCC)=O)C2)cccc2ccccc12 N1(c2ccc(CN(CC=C)CCO)cc2)C(=O)c2ccccc2C1=O c1(CNCC(O)Cc2ccccc2)ccc(OC(F)F)c(F)c1 C1(CC(=O)N(CC(C)CNC(=O)CC2(C)CC2)C)CC2CCC(C1)N2C CC1(CNC(=O)Cn2ccccc2=O)CCCN(C(C2(Cl)CCCCC2)=O)C1 CCC(Cc1ccccc1C)C(=O)NCC(C)(CO)NC(=O)CC1CCOCC1 C1(C(=O)NC2CC(C)(NC(C34CC(F)(C3)C4)=O)C2)CC2(CCOCC2)CO1 c1(CC)cc(C(N2CC(CN=c3[nH]nco3)C(CCO)C2)=O)ccc1C C1(CCC)CN(C(=O)CC23CC(C2)C3)CCN1C(c1ncoc1-c1ccon1)=O N1(C(C2N(C(c3c[nH]c(=NC)o3)=O)C3C(O)CC2C3)=O)CC(=O)N2CCCC2C1 c1(CC)ccc(OC)cc1NC(=O)C(N1CCOC(c2noc(C)n2)C1)=O Cc1cccc(C(=O)NCC2CC(CNC(=O)CCC3CC3)CO2)c1O c1(C(=O)NC2(CCOC)CCN(C(c3nc(Cl)c(Cl)s3)=O)C2)cc(C)nc(C)c1 C1(CCNC(C(c2cn(C)nc2)(F)F)=O)CCCCN1C(c1ccc(O)nn1)=O C1(CN(C(c2coc(Cl)n2)=O)CC)CCN(C(c2ccc(Cl)cn2)=O)CC1 N1(C(C(C(COC)C)C)=O)CC2CCCC(C1)N2C(C1(Cl)CCCCC1)=O c1(C(C)C)n[nH]cc1C(=O)NCC1CCCC1NC(=O)CC(=O)Nc1nccs1 c1(C(=O)NC2CN(C(CCSCCC)=O)CC3C2C3)[nH]c2ccc(C)cc2c1Cl c1(CC)nc(-c2cccc(-c3ccc(C)nn3)c2)n(CCc2ccncc2)n1 CCC(CC)(CO)NC(=O)C=CCCSc1ccccc1 c1(OC)cc(OC)c(NC(C2CC(F)CN2C(C2CC(=O)N2)=O)=O)cc1F C1(C(=O)NCCC(=C)CNC(=O)C=C2CCOCC2)CCCC(F)C1 C1(NC(c2ccc(Cl)cc2)=O)CCCC(C(=O)NC2(c3cccnc3)CC2)CC1 Cc1cnc(CNCC23CC2CN(C(c2cncn2C)=O)C3)nc1 C1(NC(C(C)(C)C(F)F)=O)CN(C(c2cccc3nc[nH]c23)=O)C2(CCOC2)C1 CCCCC(CC)CC(=O)N1CC(NC(c2conc2C)=O)CC12CCCC2 N1(C(Cn2c(C)nnn2)=O)C(CNC(=O)C=CC2CCC2)CC2CCCCC12 Cc1c(Nc2cc(O)ncn2)cnn1CC1CC1 c1(C(N)=O)ncccc1NC(C1CC(F)CN1Cc1ccc(I)o1)=O C(CC(C)(C)NC(C1CNC(=O)O1)=O)=CC(=O)NCCN(C)CCF C12(OC)CCCC1(C(N1CCC(C)C(N(C(=O)Cc3ccoc3)C)C1)=O)CCO2 C(=O)(C(C(F)(F)F)C(F)(F)F)NC1(CO)CN(C(c2c(CC)c[nH]n2)=O)C1 N1(C(C2CCC(OC)C2)=O)CC2(CCN(C(c3cccc4nsnc34)=O)C2)C1 Cc1nn(C)c(F)c1C(=O)NCc1ccc(C(C)NC(=O)C(C)C(C)(C)C)cc1 C1(COC)CN(C(=O)C(N2CCCCC2c2ncno2)=O)CC(C)(C)O1 Cc1cc(C(=O)NC(C)CC2CCN(c3cc(C)nc(C)n3)CC2)nc(Cl)c1 c1(SC)ccc(CC(=O)NCCC(CNC(C2(O)CC(F)(F)C2)=O)OC)cc1 N1(C(C(C(C)C)O)=O)CCC2(CC1)CN(C(=O)C=Cc1ccco1)CCC2O c1(OCC)ccc2nc(N3CC4CC(NC(=O)CCCC(N)=O)C4C3)sc2c1 C(=O)(CCCCC(=O)NC12CC(NC(=O)CCCSC(C)(C)C)(C1)C2)NC c1(C(=O)NC2C(C)CN(C(c3ncc[nH]3)=O)CC2)ccc2nc(O)n(C)c2c1 C#Cc1ccc(C(=O)NC2CC3CC(NC(C4(O)CCSCC4)=O)C2C3)c(F)c1 CCCCCC=CCC(=O)NCc1ocnc1-c1cn(CC2(C)CC2(Cl)Cl)nn1 CC1(C)CCCC(C(=O)NC2C3CC(NC(c4ccnc(C5CC5)c4)=O)CC23)C1 c1(OC)ccc(C(N2CCN(C(c3nccc(C)n3)=O)CC2C)=O)c(F)c1 Cc1ncc(C(N2CC3CC(NC(C4CN(C(N)=O)C4)=O)C2C3)=O)cc1N n1(C(C(=O)OC)C)nnnc1C(c1cc(C(C)C)on1)NC1CC1C(F)(F)F Cc1cc(C(=O)NCC(C2CC2)N(C)C(C2CC3(CCC3O)C2)=O)cc(F)c1 C1(C(N2CC(N(C(COCc3ccc(OC)cc3)=O)C)C2)=O)CCCC(C)(C)C1 C(CC(C)(C)CC(=O)N1CC(OC)C(NC(c2ccn(C3CCC3)n2)=O)C1)OC N1(C(C(C)C)=O)CCC(F)(F)C(CNC(=O)COC(F)(F)F)C1 C1(CC(=O)NC(CN(C(CSCC)=O)C)(CO)CO)CSc2ccccc2O1 C(CCCCC(=O)NC1CC(C)N(C(c2cc(N(C)C)ccn2)=O)C1)OC C1(C(=O)NCC(C2CC2)OC)CCCN1C(C)=O.c1(C2C(C(=O)NC)C2)ccccc1 Cn1nnc2c1C(C(=O)NCC1CCCN(C(=O)C(F)(F)C3CC3)CC1)CCC2 C=CCCC(C(=O)NCC(CC)OC)NC(C1CCN1C)=O N1(C(=O)CC2CCCCN2C(C2C3CCCC23)=O)CCC(CO)C(O)C1 N1(C(CC=CC)=O)CC2CCC1C(NC(=O)C1=C(C#N)CCC1)C2 C(=O)(C(C)(C)CO)NCC(C)N(C)C(c1cccc(C(F)(F)F)n1)=O N(C1COCc2ccccc21)C(N(C)CCOc1ccccc1)=O.C1CC1 N1(C(C#CC(C)(C)O)=O)CCC2(CCOCC2)C(NC(C2CCNC(=O)C2)=O)C1 c1(N(CC(=O)NC)C)nc(NCC23CCC(CC2)C(C)(C)O3)c2ncsc2n1 c1(OC)cc(F)c2c(C(=O)NC(C)(CNC(C3(F)CC3C)=O)C(C)C)n[nH]c2c1 N1(C(C2(C)CCN2C(=O)C(F)(F)F)=O)CCC(CC(c2cc(Cl)c(Cl)[nH]2)=O)CC1 CN1N=C(CC(=O)N2CC(O)(CCNC(c3cn(C)nc3C(F)F)=O)C2)CC1=O N1(C(c2c(OC(C)C)n[nH]c2)=O)CCC(CO)C(NC(=O)CS(N)(=O)=O)C1 c1(OC)cccc(C(N2CCCCC2CN(C)C(c2ncc(Cl)s2)=O)=O)n1 c1(COC)cc(C(=O)NCC2(NC(=O)C(C3CCCCC3)F)CCOC2)cs1 c1(C(=O)NC2CC(C)CN(C(c3cnn(C4CC4)c3)=O)C2)ccc2n[nH]cc2n1 C1(NC(C2(CC#C)CCCO2)=O)CCN(C(c2cnc(C(C)C)nc2)=O)CC1O C(=O)(C(O)C(CCC)N(C(=O)CN(C(=O)C(C)C)C)CC=C)N1CC(C#C)OCC1 C12(CF)CN(C1)C(=O)N2.C1(COC)(COC)CC(C(=O)OC)C1 c1(C(N2CCC(n3cc(C4(C)CSC4)nn3)C2)=O)coc2c1CCCC2 C1(NC(C2C(C)(C)C2)=O)CC(C)(CNC(C2(N3CCCCC3)CCCC2)=O)C1 N1(C(C2CC(SC)C2)=O)CCCC(C(N2CCCC3(C2)N=N3)=O)CC1 c1(C(N2CC(OCC)(CNC(c3[nH]c(O)nc3C)=O)C2)=O)cccn2nnnc12 c1(C(N2CCC(CCNC(c3c(C)[nH]cc3)=O)C2)=O)cnc(O)c([N+](=O)[O-])c1 C1(NC(C(C)(O)C2CCCCC2)=O)CCN(C(c2cn(CC3CC3)nn2)=O)CC1 c1(C(N(C(C(=O)OC)C)C)=O)ccn(CCNC(=O)C(C)n2cnnn2)c1 C12CCCC1N(C(C1CC=CCC1)=O)C2.c1(C(=O)O)ccc(-c2ccncc2)s1 CCN=c1[nH]c(C(=O)NC2CCN(C(c3csc(Cl)n3)=O)CC2C)cs1 N1(C(C(C)(C)OC)=O)CCC(C)(CC(=O)NC2CCOC2(C)C)C1 C1(NC(c2c(C(N)=O)csc2)=O)CCN(C(c2coc(C3CCC3)n2)=O)CC1F C1(CNC(C(C)O)=O)Cc2ccccc2CN1C(c1ccc2ccn(C)c2c1)=O C#Cc1cccc(C(=O)NC(CO)C(C)NC(C2(CC(F)F)CCC2)=O)c1F C(=O)(CCCC(=O)NCC(C)CNC(c1oc(CC)nc1C)=O)NCC c1(C(=O)NC2CC(C)(NC(C3CCCN3S(C)(=O)=O)=O)C2)cnn2c1CCCC2 N1(C(Cn2c(C)ccn2)=O)CCC(NC(C2CCN(C)S2(=O)=O)=O)CC(O)C1 C1(CNC(c2ccnc(S)c2)=O)CCN(C(=O)C(O)C2CCCC2)CC1O Cc1ccccc1C(=O)NC(c1cccc(C(C)O)n1)c1nnnn1C1COC1 N1(C(C2C(CC)C2)=O)CC(NC(c2cncc(C)n2)=O)CC2(CCC2)C1 c1(C(=O)NCC(C)(C(C)C)NC(c2nc(C)oc2)=O)cccc(F)c1C#N C(=O)(C(C(C)(C)C)C1CCCCC1)N1CCCC(CN(C(CCC(=C)Cl)=O)C)C1 Cn1cc(C(=O)NCC(=O)NC23CCCCC2C3)ccc1=O C1(NC(c2n(C)nc(CNC(=O)C(F)CC3CCC3)c2)=O)CCCC2(CC1)CC2 C1(C(=O)NCC(CC(=O)N(C2CCN(CC)CC2)C)C)CC(=O)OC1(C)C C(c1c(C)noc1C)=CC(=O)NC1CC(C(C)NC(C2(COC)C=CCC2)=O)C1 CC1(C)C(CNC(c2coc(Cl)c2)=O)CCN1C(=O)CCC=CBr C1(NC(=O)Cc2cnn(C(F)F)c2)CCN(C(=O)C2=CCCSC2)CC1F N1(C(CC2CCN(C(C3(C)CCCC3O)=O)C2)=O)CCCC(F)CC1 C(CC(C(=O)N(C)C)NC(CC(C)SC)=O)NC(=O)C(C)N(C)C c1(N(C)C)ccc(CNC(C2C3CC3CN2C(C2CC2(Cl)Cl)=O)=O)cn1 N1(C(c2cc(C)c(Br)s2)=O)CC2CC1CN2C(=O)COCC1(F)CC1 C1(C(=O)NC2(C(=O)O)CC(O)C2)CNc2ccccc2O1 Cc1cccc(C)c1C(=O)NCC1CC1C(=O)NCC1CN(C)CCN1C c1(CCC(=O)NC2COC3(C2)CN(C(=O)C=CCO)C3)cccc2ccccc12 C(=O)(C(F)(F)C(F)F)NCC(CN(C(C(c1ccccc1)OC)=O)C)O N1(CC)CC2CC1CN2c1cc(N(C)Cc2ncc(C)o2)nc(C(F)(F)F)n1 c1(OC)nc(C)c(Br)cc1C(N1CCOC(CF)C1)C(=O)NC1CCC1 CC1(F)CCN(C(C2CC(O)CN2C(c2ccncc2Cl)=O)=O)C1 c1(CC)cc(C)c(C(=O)NCC2CN(C(C34CC(CO3)C4)=O)CC2C)o1 CC(C)C(O)CC(=O)NCc1occc1C(=O)N(CC(=O)NC1CC1)C C=CC(C)(O)CC(=O)N1CCC(OCCNC(=O)C(C)(C)C2CCCO2)CC1 CC1CC(NC(c2nc(Cl)ccc2Cl)=O)CCN1c1ncc(Br)c(O)n1 C1(C(N2CC(OC)C(NC(=O)C(C)(C)C)CC2)=O)Cc2nc(C)cn2C1 N1(C(C#CC(C)C)=O)CCC2(CNC(=O)Cc3ccc(F)c(F)c3)CCCCC12 CCCS(=O)(=O)CC(=O)NC1CN(C(c2cnccc2Cl)=O)CC1C C1(N(C(C(N2CCCC(O)C2)C)=O)CCO)CCN(C(C2CCCN2C)=O)CC1 c1(OC)ccc(CNC(=O)CC2CCCN(C(=O)CN3CC(=O)NC3=O)C2)cn1 O=C(CC(F)(F)C(F)(F)F)NCC1(C2CC2)CCN(C(=O)CCn2cncn2)C1 c1(CC)ccc(C(=O)NCC(O)CN(C(=O)Cn2nc(C)oc2=O)C)nc1 N1(C(c2n[nH]c(C)c2O)=O)C2CCC1CC(CNC(=O)CNC(=O)C(F)(F)F)C2 CC(CCN=c1cc(Cl)nc(-c2cccnc2)[nH]1)NC(c1csc(Cl)c1Cl)=O C1(C)(C(=O)NC(c2ccccc2)C)CCCN1C(C1CCCSC1C)=O Cc1nc(CN(C(=O)C(n2cc(-c3cn[nH]c3)nn2)C)C)nc2ccccc12 C(=O)(CCCS(C)(=O)=O)NC(C1CCN(C(C2(C(C)(C)O)CCC2)=O)C1)(C)C Cc1cccc2c1CCOC2C(=O)NC1(CNC(=O)C(C)O)CCC1 c1(NC2CC(C)(C)OCC2)nccc(=NCc2ncccc2CO)[nH]1 C1(CC(N2CC(SCC)C2)=O)C2CCCC2N1C(c1ccc(C)nc1)=O N1(C(C2ON=C(C)C2)=O)CCC(O)(CN(C(=O)CCc2c(C)noc2Cl)C)C1 N1(C(C(COC)NC(C)=O)=O)CCC(=CCNC(c2coc(C(F)F)c2)=O)CC1 c1(N2CCCC(CC=C(C)C)C2)nc(=N)[nH]c(=NCCc2c[nH]nc2O)[nH]1 C1(c2onc(C(N)=O)n2)CCCN(C(=O)N(C2CCCC2)CC2(O)CCNCC2)C1 C1(CNC(c2c(C)c[nH]n2)=O)CN(C(C2CCCCO2)=O)C(C)(C)C1 c1(OC)ccc(C2(C(=O)NCCCCCCN(C(=O)C(C)OC)C)CCC2)cc1 Cc1ccc(F)c(C(N2C3CCC(C3)C2CNC(=O)C(C)OCC2CC2)=O)c1F C1(CN(C(C2(NC(C(CO)NC(=O)OC)=O)CCC2)=O)C)CCC(C)CC1 c1(OC)cc(NC(C2COCCN2Cc2ccc(F)c(C#N)c2)=O)c(Br)cc1Br c1(C(N2CCC(N(C(=O)CC3CCC(=O)NC3)C)C2)=O)ccc(C#N)n1C C1(NC(c2ccc3nn[nH]c3c2)=O)CCSC12CN(C(=O)C=Cc1cccs1)C2 c1(C(=O)NCc2c(CNC(C3C(COC)C3)=O)cccc2)ccc2n[nH]cc2c1 c1(N2CC(CN(c3cnc(C4CCN(CC)C4)s3)C(C)=O)C2)ccc(N)cc1C C1(C(N(CC(CCC)C)C)=O)C=CCN(C(C2(OC(C)=O)CC2)=O)C1 c1(C(=O)NC2CN(C(C3C(OC)CCCC3)=O)C2)c(C)nc(C(C)(C)C)nc1O C12(C(=O)NC3CC(NC(c4nc(C)nn4C)=O)C3)CCCC1C2(F)F C1(F)(CNC(c2cccc(CCC)c2)=O)CCCN(C(C2C=C(C)CS2)=O)CC1 c1(N(CC(=O)N(CCCCCC)C)C)ccc(C)c(C)c1 c1(C(N2C3CN(C(Cc4c(C)noc4)=O)C(C3)C2)=O)ccc2nc[nH]c2c1 C(C)(C(C)NC(=O)CC1CC(NC(c2c[nH]nc2C2CC2)=O)C1)(C1CC1)OC C1(C(N2CCCC(NC(Cc3ncc(C)s3)=O)C2)=O)Cc2c(F)cccc2O1 c1(NC(=O)NC2C(CCC)N(C(=O)C3=CCCC3)CC2)cnn2ccccc12 c1(CNC2CC(F)(C(=O)Nc3ccc(F)c(Cl)c3)C2)cc(F)c(Cl)cc1Cl C1(COCC(=O)NCCN(CCC)C(C2(CC)CCCC2)=O)CCCCO1 C1(N(C(c2cnn(C(C)C)n2)=O)CCO)CCCN(C(=O)COCCOCCO)C1 CC1CC(C(N2C(CNC(c3ccnnc3)=O)CC3CCCC23)=O)CC(C)(C)C1 N#Cc1c[nH]c(C(=O)NCc2ccccc2CNC(C2CC2[N+](=O)[O-])=O)c1 C1(NC(C=Cc2ncn(C)c2)=O)CC2CC1N(C(C1(C)CC1(F)F)=O)C2 c1(C(=O)NC2CN(C(C#CC(=O)O)=O)CC(F)C2)n[nH]c2cccnc12 CCC(CC)C(=O)N(C1CCC(NC(=O)CC(c2cccs2)NC(N)=O)CC1)C c1(OC)nscc1NC(C1OCCC1CNC(C1(NC(N)=O)CC1)=O)=O C(C(C)(C)C(=O)NCC1(F)CCN(C(C2CC(=O)N(C)C2)=O)C1)OCC C1(C(=O)NC(C2CCOCC2)C)(CC)CCN(C(=O)C(C)SC(C)C)C1 C(=O)(CC(C)C(=O)N(CC(C)N(C(=O)Cc1ccc(C)nc1)C)C)OC c1(C(C(=O)NC)N(C2CC2)Cc2cccc(C(C)C)c2F)cc2ccccc2o1 C1(CNC(C(Cc2c(C)nc[nH]2)O)=O)CC12CCN(C(=O)Cn1cnnc1)CC2 CC1(C)CC(NC(c2nnnn2Cc2ccc(F)cc2)c2cn[nH]c2)C12CCC2 c1(COCC)nc(N2CCC(C)(NC(=O)Cc3ccon3)C2)cc(C)n1 N1(C(Cc2c(C)cco2)=O)CC(C)CN(C(c2n[nH]c(=N)[nH]2)=O)C(C)C1 N1(C(C2C(C)C2)=O)CCC(CNC(c2ccc(S(C)=O)cc2)=O)C(F)(F)C1 N1(C(C(CC=CC)NC(=O)CNC(=O)OCC)=O)CCOCC(CO)C1 C12(NC3(C(=O)O)CC(CS(=O)(=O)NCc4ccccc4)C3)CC(CN1)C2 C(C(COC)CC(=O)NC1COCC1C(N1CCC1CN=[N+]=[N-])=O)OC N1(C(=O)CCn2cncn2)CC2CCN(Cc3cc(Cl)c(Cl)c(Cl)c3)CC2C1 C1(CC(=O)NCCC2CN(C(C3CCC(=O)NC3)=O)C2)CC2(CCC2)CCO1 N1(C(c2ccc(CO)nc2)=O)CCC(C2CCCN(C(C3CCC(O)C3)=O)C2)C1 Cc1nc(NC(C)Cc2ncccc2C)cc(NC2CCCCCC2)n1 c1(CNC(C(=O)NC(c2ccnn2C)CC)=O)cccc2c1OCCCO2 C(N=c1[nH]cnc2c(Cl)cc(Cl)cc12)C1(C)CCN(C(c2ccno2)=O)CC1 c1(C(N2CC3(CNC(C45CSCC4C5)=O)CC2CO3)=O)ccc(F)cc1F C(=O)(CC(C1CC1)NC(C)=O)NCCN(C(C(c1cnn(C)c1)OC)=O)C N1(C(CC)=O)CCC(CNC(=O)C(C)OCC)(OC)C1 c1(COC)ccccc1C(=O)N(C)CC1CCCN1C(=O)CCc1cnn(C)c1 CCCCCC(O)CC(=O)NC1CC2CN(C(c3cc4n(n3)CCC4)=O)CC2C1 C1(C(=O)Nc2cccc(NC(C34CCCC3CCC4)=O)c2)CCc2c[nH]nc2C1 N1(C(C(C=C)OC)=O)CCC(C2CC2)C1C(=O)NC(COCC)C(C)C CC1(C(=O)NC2CC(F)(F)C2CO)COCCN1 n1(CC)ccnc1C=CC(=O)NC(C1CCCC1)CNC(c1ncoc1C)=O c1(C(=O)NC(C2CCC(F)(F)CC2)CC)cn2c(n1)CCC2 C(CCC(CO)NC(C)=O)NC(CC(C)=C(C)C)=O.C(=O)(C(C)(F)F)N CC1(CNC(c2cc(CNC(C3CCOC3(C)C)=O)cs2)=O)NC(=O)NC1=O CC1(CNC(=O)C(=O)NCC2CC2)COCCN(C(=O)C=Cc2ccc(Cl)s2)C1 N1(C(=O)COCC(F)F)CCCCC1C1CCCN1c1cc(CC2CC2)ncn1 N1(C(C(COCC)(C)C)=O)CCN(C(=O)CCC=CBr)C(CF)C1 Cn1cnnc1C1CCN(CC(O)Cn2cccn2)C1 c1(C(=O)NS(CCCC)(=O)=O)cc(Cl)ccc1C.C12C3CN(CC13)C2 c1(NC(CC)C(C)C)ccc(S(=O)(=O)N(C2(COC)CCC2)CC)cc1Cl C=CCCC(CC(C)C)C(=O)N1CC2CC(N(C(=O)CNC(N)=O)C)C1C2 CCC(C)C(CC(=O)N(C)CC1CCCN(C)C1)NC(=O)C(C)(C)n1cccn1 C(CC(C)CC(C)(C)C)NC(CN(C1CCC1)C(c1c(CC)nco1)=O)=O c1(C(=O)NC(C2(CNC(c3ccc[nH]3)=O)CC2)C)ccc(F)c(Cl)c1F N1(C(c2n(CC(C)C)ncc2)=O)CCCC2(CCN(C(C3(C)CCCO3)=O)C2)C1 c1(NCCC2(O)CN(C(CCSCCCC)=O)C2)ccccc1[N+](=O)[O-] c1(CSCC)ccccc1C(=O)NCC1CC1NC(=O)CNS(=O)(=O)NC N1(C(CNC(c2ccoc2)=O)=O)CCCCC(NC(C2CCCS(=O)(=O)C2)=O)C1 C1(NC(CNC(=O)NC)=O)CCN(C(C2CC2F)=O)CC1c1ccccc1 Cc1c(NCCCCC(C)C)ncnc1NCCc1cccc(C(F)(F)F)n1 C1(C(=O)NC2CN(C(c3ncn4ccccc34)=O)C2)CCC2(CCOCC2)C1 c1(CCC)nc(C)c(C(=O)N(CC(C)(C)NC(=O)CN(C)C(C)=O)C)s1 C=CC1CN(C(C23CC2CCN3C(=O)CCc2cnn(C)c2)=O)CC1O C=CCC(C(=O)N1CCC(C=CC(N2CCC(C3(C)CC3)C2)=O)CC1)C(C)C c1(OC)ccc(C(N2CCN(C(=O)C(C)C(C)C)CC2CF)=O)cc1F N1(C(C(C)(C)C2CCCO2)=O)CCC2(CCCN2C(C2CC3(CCC3)C2)=O)C1 N1(C(CNS(CC)(=O)=O)=O)CCC(F)C(NC(c2csc(C(=O)OC)c2)=O)C1 n1(CCCNC(CN(C(=O)CSCCC#N)C(C)C)=O)cnc(=N)[nH]1 n1(CC)nc(C(=O)NC2(C)CC(NC(=O)Cc3ccnn3C)C2)c2c1CCOC2 c1(C2N(C)C2)ccc(N)cc1Cl.C12CC(=O)N(C1)C1CC1CC1(F)CN(C1)C2=O N1(C(C(C)OCCN(C)C)=O)CC(F)(F)CC1CNC(C1CCCCN1N=O)=O c1(OC)ccc2[nH]c(=NCc3csc(C4CC4)n3)[nH]c(=NC3COCC3F)c2c1 N1(C(CCC(C)C)=O)CCCC2(CCCN2C(=O)CC2CCC(C)(C)CC2)C1 c1(NC(C(c2ccc(F)cc2)OC)=O)csc(C2=C(C)CCCC2)n1 Cc1cccc2c1CN(C(C1(C3CC3)CN(C(=O)C(C)CC(C)(C)C)C1)=O)C2 c1(OC)ccc2nc(N3CCC(CCNC(C4CC4(F)F)=O)C3)c(C#N)cc2c1 N1(c2nccc(OCC)n2)CC(NC(=O)C=CBr)CC12CCOCC2 c1(C(=O)NC2C3CN(C(CNS(CC)(=O)=O)=O)CC32)cc2cccnc2nc1C C1(CNC(=O)NC2CCN(C(C34COC(CF)(C3)C4)=O)CC2)CCCC1C1CC1 c1(CCC(=O)N(CCCNC(c2c(CCC)n[nH]c2)=O)CC)ccc(OC)nc1 N1(C(CC2C(C)(C)OCC2)=O)CCC(F)(C(=O)NCCN2CCC(CO)C2)CC1 c1(C(N2C(C)CN(c3nccc(Br)n3)CC2)=O)cc(F)c(F)cc1[N+](=O)[O-] N1(CCN(C(=O)C(CNC(=O)CC2CC(C3CC3)C2)CC2CC2)C)CCNC(=O)C1 N1(C(C23N(C(C4CCSC4)=O)CC(C)(C2)C3)=O)CCCC2(C=CCO2)C1 c1(C(=O)NCC23CCC2CN(C(c2ccc(Cl)cn2)=O)C3)nccn2nccc12 C(=O)(C(C)S(C)(=O)=O)NCC1(COC)CCCN1C(C1CCC(F)C1)=O Cc1cccc(C)c1OCC(O)CN(CC(F)(F)F)Cc1nnc(C(C)C)s1 N1(CC)CC(NC(=O)CC(C)(C)NC(C2OCCC2C(C)C)=O)C(C)C1 C(=O)(C(CNC(=O)C(=O)NC)C(C)(C)C)NC1C(CC)C1 c1(CC(=O)NCCCCCNC(C2(C)CC(=C)C2)=O)cccc(C(C)C)c1 CONC(=O)C(=O)N(C1CCCN(C(=O)CCN2CCCCC2)C1)CC1CC1 C(CCCCC(=O)NC(C)(CNC(c1ncn2c1CCC2)=O)CO)OCC N1(C(Cc2cccc(OCC)n2)=O)CC(NC(=O)C(F)CC2CC2)CCC(O)C1 N1(C(C2C=C(C)CS2)=O)CCC(C(CO)NC(=O)C(C)Cc2cnc[nH]2)CC1 N#Cc1cc(NC(=O)CC2CN(C(c3cc(O)c(O)c(Cl)c3)=O)C2)ccc1Br C(=O)(C(C)(O)CCN(C)C)N1C2(CNC(C3CCN(CC)C3)=O)CC(C1)C2 c1(CN2CC(O)(CNC(c3ccc(F)c(Br)c3)=O)C2)cc(F)c(O)cc1F C1(COC)(NC(=O)CCC(C)(C)C)CCCN(C(C2CC2c2ccccc2)=O)C1 C(=O)(CCC(C)(C)N(C)C)NCC(C)(CNC(=O)C(C)C(C)(C)C)OC C1(OC(C(=O)NCC2CN(C(CNC(C)=O)=O)C2)C)CCCCC1 C1(NC(c2[nH]cc(C(C)=O)c2)=O)CS(=O)(=O)CC1NC(c1coc(C(F)F)c1)=O c1(C(C)(C)C)cccc(CC(N2CCC(CCO)(CCC(=O)O)C2)=O)c1 C1(C(N(C)CC2COCCN2C(C2(C)C=CCC2)=O)=O)CCCC(F)(F)C1 N1(C(COCC)=O)CCCC(C)(C)C1C(=O)Nc1ccc(N(C)C)nc1 C(=O)(CC1=CCN(C(=O)COC(C)CC)CC1)NCCc1nc(CC)on1 C(CC1=CCN(C(=O)CNC(C2CC2C)=O)CC1)NC(c1c(C)ncn1O)=O N1(CCC(=O)NC(C)CC(C)NC(=O)CN2CCCC2=O)CCCS1(=O)=O c1(OC)cccc(C2CNC(=O)CC(=O)N2)c1.c1(COC(C)=O)ccc(F)cc1 CCCC(CN=c1[nH]c(N2CCC(Br)=C(C)C2)nc2c1SCC2)OCC C#Cc1nc(C(=O)N(C(CNC(C2CSCCS2)=O)C2CC2)C)cs1 C1(C)(C(=O)OC)CCN(C(c2cccc(I)c2)C(=O)NCc2ccccc2)C1 Cc1c(CC(=O)NCc2cc(C(=O)NCC3CCCC(O)C3)cs2)ncn1C N1(C(CNS(N(C)C)(=O)=O)=O)CC(NC(=O)C=Cc2cnccn2)C2(CC2)C1 C1(CNC(C(C)Cn2cccn2)=O)CCCCCN1C(C1CC2(CSC2)C1)=O N1(C(CCCCNC(C)=O)=O)CCC2(NC(C3CCC(C)C3)=O)CCCC12 N1(C(C(C)=C2CCC2)=O)CCCCC(N(C)C(c2ccc(F)s2)=O)C1 Cc1cc(C(N2CCC(F)C(NC(c3cn(C)c(=O)cn3)=O)C2)=O)nc(O)n1 C1(C(N(CCN(C(C)C)C(c2ccc(F)cc2)=O)C)=O)CCCCC(F)(F)C1 c1(C(=O)NC(C)CNC(c2cccc(=S)n2O)=O)cc2n(n1)CC(F)C2 N1(C(C2CC(S(C)(=O)=O)C2)=O)CCC2CCCC12CNC(c1ncccn1)=O C(=O)(CCCC(=O)N1CCC(NC(c2csc(C3CCCCC3)n2)=O)C1)OC N1(C(c2c(C)cc(Cl)cc2)=O)CC2C(C1C(N1CC(O)C1)=O)C2(C)C Cc1coc(C=CC(N2CC3CC3(NC(=O)CCCCN(C)C)C2)=O)n1 c1(C(N2C(C)(C(N3CC(O)C(O)C3)=O)CC2)=O)cccc2c1CC(=O)N2 CCCC(CNC(c1ccsc1)=O)C(=O)N(C1CCOCC1)CCC C1(NC(COCCC#C)=O)CC(O)CN(C(c2ccc(O)c(CC)c2)=O)C1 CC1CC(=O)NCC1C(=O)N(CC(C)(C)NC(=O)CN1CCOC1=O)C C1(CCNC(c2c(C)onc2)=O)CC(F)(F)CN1C(=O)COCc1cccnc1 C#CCC(CC#C)C(=O)NCC1(C(N)=O)CN(C(=O)C(COC)N(C)C)C1 CC(O)(CNC(=O)C(C1(O)CCCC1)F)CNC(C1(C(F)(F)F)CCC1)=O c1(C(=O)NC2C3CN(C(CCOCC)=O)C(C3)CC2)csc2c(C)cccc12 C1(O)(CN(C(=O)CC2CCCSC2)C)CCN(C(=O)COC2CC2(F)F)CC1 c1(CN(C)Cc2ccnc3[nH]ccc23)nc2c(s1)CC(C(F)(F)F)CC2 c1(C(=O)NC(C2CCOC2)CNC(C(=CC2CCCC2)C)=O)ccnc(C)c1C CCC(F)(F)C(C)(C)C(=O)NCC1C=CC(NC(c2ccc(=N)[nH]c2)=O)C1 CN1CC2(CC2)CC1C(N1CC(O)(C(C)(C)CNC(c2cn[nH]c2)=O)C1)=O N1(C(CC)CC)CCC(C(C(=O)NCCC#N)N(C)CC2CCCO2)C1 C(=O)(Nn1cnnc1C)C1(F)CCN(C(C(C(C)(C)C)OC)=O)C1 N(C1C(=O)Nc2c(C)cccc21)C(C1CCN(C(c2scc(C)c2)=O)CC1)=O C12(C(N3CCC(C)(N(C)C)C3)=O)COCC1CN(CC13CCCNC1CCC3)C2 c1(C(=O)NC2(C(=O)Nc3cc(CC)c(C)cc3)CC2C)cccc2nccn12 N1(C(=O)OC(CC)C)CC(C(F)(F)F)OCC1(C)C C1(CNC(c2c(C)cnnc2O)=O)CCCC2(CN(C(c3ccsc3C)=O)C2)O1 c1(NC(=O)NC(c2cccc(Cl)c2Cl)CO)cnccc1[N+](=O)[O-] N1(C(C(c2scc(C)n2)C)=O)CCOC(C(C)NC(c2nccn2C)=O)C1 O=C(CCC(=O)N1CCOCC1)OCC(=O)NCCc1csc(N2CCCC2)n1 C1(C(=O)NCC2C(C)(C)CCO2)CC2CN(C(=O)CC3CCC(=O)CC3)CC2C1 CON(C(=O)C1CCCN(C(=O)CCn2ccnc2C)CC1)C1CCC1 N1(C(CC(C)F)=O)CCOC(CNC(=O)C(N2CCOCC2=O)C)C1 C(c1c(C)coc1C)=CC(N1CCC(C(CNC(C(CC)=CC)=O)C)CC1)=O C1(N(CC(N)=O)C)CCN(C(=O)C(=O)NCC2CC2(C)C)C1 C1(CCC)CCCCN1C(C1C2CCCCC12)C(=O)NC1CC(F)(F)C1 c1(C(=O)NC(CC)CNC(C2CC=CC2)=O)csc(=NC2CCCCC2)[nH]1 C1(C(C)C)CN(C(C2CCOC2CNC(c2ccc(O)nn2)=O)=O)CCCO1 c1(C(=O)NC2CC(CNC(C(C)(C)CF)=O)C(O)C2)cc2c(cc1Cl)NCC2 CCCCCCC(C)C(=O)NCc1ccc(CN(c2nc(COC)ns2)C)cc1 N1(S(=O)(=O)CC2CCCO2)CC2OCOC2C1 N1(C(CC(C(=O)OC)C)=O)CC2(C1)SCCC2NC(=O)Cc1ccn(C(F)F)n1 C#CCC(C(=O)NC(C=C)C(F)(F)F)NC(c1cnn(CC)c1)=O CC(CC(=O)NCC(C1CC1)NC(=O)C(C)(C)O)C(C)(C)C C1(NC(COC2CCC(C)CC2)=O)CN(Cc2cccnc2F)CCC1C N1(C(COC)=O)CCC2(C1)CN(C(=O)CN(C)S(=O)(=O)N(C)C)CCO2 c1(CC(=O)NC2C(SC)CN(C(C3(C)COC3)=O)C2)cccc2cnccc12 N1(C(=O)OCCCC)CCCC(c2n[nH]cc2C(=O)OCC)C1.OCC N1(C(c2c(CC)ncs2)=O)CCCCC(CNC(=O)Cn2nnnc2C2CC2)C1 N1(C(C2CCc3n(cc(C)n3)C2)=O)CCc2cc(Br)c(Cl)cc21 CCC(C)CCC(O)CC(=O)NCC1CCCCN(C(=O)C(C)(C)C(C)C)C1 C(=O)(C1=C(C)CCCC1)N1CC(CNC(c2c(CCC)n[nH]c2)=O)C2C1C2 C1(NC(Cc2c(C)cccn2)=O)CCCCN(C(=O)C(C)OC2CCCCC2)C1 c1(NC(Cn2cc(-c3nc(C)nc(O)c3)nn2)=O)ccc2ccoc2c1 c1(C(N2C(CNC(C(C)SCC)=O)C3CCC2C3)=O)cncc2ccsc12 C1(CC)C(C(=O)NC2CC2c2cncs2)CCCN1C(c1scc(C)c1C)=O C(C(C)(C)C)=CC(=O)NCC1(CN(C)C(C2CC(N3CC(O)C3)C2)=O)CC1 O=C1NCCN(C(c2cnoc2-c2ccc(Cl)s2)=O)C1c1cc(F)cc(F)c1 C1(C2(O)CCOCC2)(C(=O)NC2C(NC(c3cc(C(C)C)on3)=O)COC2)CC1 C(CC(C)(C)CN)N(C(C(C)n1cccn1)=O)CCO Cc1cc(C(=O)N(CCCNC(=O)C(N2CCOCC2)C)C)cc2c1CCC2 N1(C(c2c(C)oc(C)c2Br)=O)CCC2CCN(C(=O)CCCN(C)C)C2C1 c1(C(=O)NCCCCC(C)NC(COCC=C)=O)ncn2c1CCCC2 N1(C(C2N(C(Cn3c(C)ncc3)=O)C(C)C2)=O)CCC(C)(N(C)C)CC1 CC(C)CS(=O)(=O)CCC(=O)N1CCCC1(C)CNC(=O)C(CO)NC(N)=O N1(C(CCCNC(=O)OC)=O)CC2OCCN(C(=O)C(C)CC3CCCCC3)C2C1 N1(C(CCc2n(C)ccn2)=O)CC2CC1CCC2NC(=O)COCC1CC1 CC(CCC(C)(C)C)C(=O)NCC1CNCCC1C c1(N2CC(CC(C)NC(c3n[nH]c(C)c3Cl)=O)C2)ncc2c(n1)CCOC2 C1(CN(C)C(C2CCCCC2n2cc(C(O)C3CC3)nn2)=O)CC2(CCC2)C1 c1(CCC(=O)NC2CCC(NC(C(=O)N(C)C)=O)C2)ccc(NS(C)(=O)=O)cc1 C(CC(CC)C(=O)N1CC(O)(CCNC(=O)C(C(C)C)NS(N)(=O)=O)C1)=CC c1(CNC(CC2C(C)(C)C2)=O)cccc(CNC(C2CC23CCC3)=O)c1 Cn1ncc2c(C(=O)NC3C4CCC3N(C(C3CC35CCCC5)=O)C4)ccnc12 C1(CNC(C(C)N(C)C)=O)CN(C(=O)C(C)n2cccc2)CCC1C c1(C(=O)NCc2cncc(OC3CC3)c2)cc2cccn2c(O)n1 CC1=CCC(C(=O)NC2CN(C(c3ccccc3-n3ccnc3)=O)CC2F)CC1 Cc1c(C(=O)NCC2CCN2C(=O)C(C)CC2CC2)cncc1Br C12C=CC(C1)CC(=O)N(NC(C(C)OC1CCCC1)=O)CC(=O)N2.C1(CO)CC1 CC1CCN(C(c2cnc(O)n(C3CC3)c2=O)=O)C(C)C1NC(=O)CC1CC1 C=CCC(F)(F)CN(C(C1CCCCC1)C(=O)NCCC1(C)CC1)C Cc1cnc(C(=O)NC2CCC(CCNC(=O)C(C)(C)c3ccnn3C)C2)nc1 C1(C(=O)NCC2N(C(c3c(CC)ncs3)=O)CCOC2)CCc2nnnn2CC1 C1(C(N2CC3COCC3(C(N3CC(F)C3)=O)C2)=O)CCc2ccccc2C1 c1(C(C(=O)NC(C)C(C)NC(c2cnc(C(N)=O)s2)=O)=O)cc(F)cc(Cl)c1 c1(C(N2CCC(C)(NC(C(C)CC3CC3)=O)C2)=O)cc(S(N)(=O)=O)c[nH]1 C1(NC(C=COCC)=O)CCN(C(=O)CC2CC(CC)=NO2)C1C C#CC1CC2CCC1N(C(C1C3CCN(C(=O)C=Cc4ccncn4)CC13)=O)C2 C12(C(=O)NCCC(C)NC(=O)CCCC3CCCCC3)CC3CC(C(=O)N1)C2C3 C1(OC)CC(NC(=O)CC(C)N(C)C)N(C(=O)C#CCN(C)C)C1 C12(NC(N3CCCC(Cc4nnc5ccccn45)C3)=O)CCCC1CC(F)(F)CC2 CCCCC(CO)NC(C1(C(C)NC(C2C(C)(C)C2(C)C)=O)CC1)=O c1(-c2ccc(C(N(CCN(C(=O)CC3CCCSC3)C)C)=O)o2)cccc(F)c1 Cn1ccn2ncc(C(=O)NC3CCN(C(=O)CNC=O)C(c4ccccc4)C3)c12 CN1CCN(C(=O)C(CNC(c2ccnnc2O)=O)N(C)C)C(CCO)C1 N1(C(c2c(C)nncc2)=O)CC2CCC(N=c3[nH]c4cc(Cl)cc(Cl)c4o3)C2C1 c1(C(N2CC(CNC(=O)C(O)C3CC3)C(C(F)(F)F)CC2)=O)nccn2ccnc12 N1(C(=O)C(F)(F)C2CCNC2)CC(O)CC1c1cccc(F)c1 c1(CN2CC(C(=O)NCC3CN(C)C3)C2)ccc(C(N2CCOCC2)=O)nc1 c1(C(N(CCN(C(CC(C)N(C)C)=O)C)C)=O)c(Cl)cccc1Br C1(CNC(C(C)=CC)=O)CC2CCC1N2C(=O)C1=C(C)OCC1 N1(C(C(C)(C)SC)=O)C2CCC1C(C)C(NC(c1cc(C)oc1C)=O)C2 C(=O)(CC(F)(F)C(F)F)NC1CN(C(C2CC(N3CCN(C)CC3)C2)=O)C(C)(C)C1 C(CCNC(c1cccc(Cl)n1)=O)(C(C)C)NC(CC1(COC)CC1)=O C1(CCNC(C2CC(SC)C2)=O)CC(F)(F)CN1C(C1CC2(C1)CC(C)C2)=O c1(C(=O)NC(CC)C(N2CCCC(F)(F)C2)=O)cc2ccccc2[nH]1 CC(CCCCNC(C1CCCCN1S(C)(=O)=O)=O)NC(C1C(C)(C)C1(C)C)=O c1(OC)cncc(C(=O)NC(CNC(=O)C(F)C(C)(C)O)C2CC2)c1C c1(OCC(C)C)ccc(C(N2CCC(NC(C3(C(N)=O)CCC3)=O)C2C)=O)cc1 c1(N2CCC(OC(C)(C)C)CC2)nc2c(c(=NCC3C(C)(C)C3(F)F)[nH]1)COC2 c1(C(=O)NCC(O)CNC(c2coc(CC3CC3)n2)=O)csc([N+](=O)[O-])c1 C1(C(=O)NCC(C2CCC2)OCC)CNC(=O)CN1C(=O)C(=O)CC(C)C C(=O)(CCC1CCc2ccccc21)N1CCCCC(NC(C2CC(=O)N2)=O)C1 C1(NC(c2nc(C)nn2C)=O)CN(C(=O)C=C2CC2)CCC1C C1(CC=C)(NC(c2cc(COC)[nH]n2)=O)CCCN(C(C2CCCN2C=O)=O)C1 c1(C(N2C(C)CC(NC(c3ccc(OC(F)F)nc3)=O)C2)=O)cc2ccsc2s1 C(CC(C)C(=O)NC1CCC1C(N1CC(OCCF)C1)=O)=CC C1(C(N2CCN(C)CC2)=O)CN(CC(O)CC(F)(F)F)CCC1O C1(N(C(C(C2CC2)OC)=O)CC2CC2)CCN(C(c2cc(Cl)cs2)=O)CC1 c1(C(N2CCN(C(C3N(CC)CC3)=O)CC2)=O)ncsc1S(N)(=O)=O c1(C(=O)NC(CC(=O)NCCC(C)N2CCCC2)C(F)F)cc[nH]c2nccc1-2 C1(OC)C2CCN(C(c3cc(-c4nn[nH]n4)ccc3OC)=O)C2C1(C)C N1(C(c2ccnc(-n3cncn3)c2)=O)CCCN(C(C2CC2CF)=O)CC1 O=S(=O)(c1ccc(COC)cc1Cl)N(CCC1CCCO1)Cc1ccsc1.C(CCO)N C1(CN(C(CC2(C=C)CCC2)=O)C)CN(C(C2CSCCS2)=O)CCO1 C#CC1COCCN1C(=O)C(O)C1CN(C(=O)Cc2cnsc2)C1 CC(C)S(=O)(=O)c1ccc(C(=O)NCCC(C)NC(C2CC(C3CC3)C2)=O)cc1 n1(CCC(C)C)nc(-c2ccnc(Cl)c2)nc1C1CCCN(C2CC2)C1 N1(C(CC2COCC(C)O2)=O)CCN(C(c2cn(C3CC3)nn2)=O)CC(C)(C)C1 C1(C(C)(C)C)(NC(C2CCC2)=O)CCN(C(=O)CC2CCC3CC23)CC1 c1(NC(=O)NC(C(=O)NCC)C2(C)CC2)ccc(OC(F)F)c(Cl)c1 C(=O)(C(CC(C)C)OC(c1ccccc1C#N)=O)N1CCC(C(CC)(C)C)C1 Cn1cc2c(n1)CC(C(N1CCC(F)(CNC(c3ccncc3)=O)CC1)=O)CC2 c1(CC)ccc2c(c1)C(CC(=O)N(CCCN(C)C(c1ccsn1)=O)C)C(=O)N2 c1(CC)cnc(O)c(C(N2CC(CNC(=O)CCCCc3ccccc3)C2)=O)c1 c1(C(=O)NCC(CC=C)NC(c2nnn(CCOC)c2N)=O)cc2occc2n1C c1(NC(C2CCCN(C(CCc3c(C)cccn3)=O)C2)=O)ccc(F)cc1Cl C(N=c1[nH]c(N(CCCN2CCOC2=O)C)nc2ccsc12)C1(CCO)CN(C)C1 c1(C(=O)OC)cnc(NC(C2C3CN(Cc4sccc4OC)CC23)=O)c(Br)c1 c1(C(C)C)nsc(NC(=O)C(=O)NC2(n3cc(Br)nn3)CC2)n1 c1(C(=O)NC23C(CN(C(CC(=C=C)C)=O)C2)C3)cc(OC)cc2c1OCC2 C(CCC(=O)N1CCC(Cn2cc(C3(C)CCCO3)nn2)C1)CC(CC)N C(c1cccc(CO)c1)=CC(N1C(CO)CCC1c1ccccc1)=O C1(NC(C(C)CCO)c2nnnn2CC2CCCO2)CC2(COCCO2)C1 C12(NCCN(CC(=O)N(C)C3CC3)C(C3CC=CCC3)=O)CC1CNC2=O N1(CC)CCC(C(=O)NC23CC(NC(=O)C(c4ccccc4)F)(C2)C3)CC1 C1(C(=O)NCC2(F)CN(C(c3occc3F)=O)C2)(CC)CCC(O)CC1 n1(CC(=O)NC2C(NC(CC3CC(OCC)C3)=O)CCC2)cc([N+](=O)[O-])cn1 C1(CC(=O)NCC(c2ccccc2)NC(C2(C)CC(F)C2)=O)(OC)CCOCC1 N1(C(C23CCC(OC)C2C3)=O)CCC(NC(C2CCCCN2C(C)=O)=O)C12CC2 N(C(=NCCCCl)N1CCC(C)(OC)C1)C.c1(OCCOC)cc(C)ccc1C CCC(C)(CNC(c1cscc1Cl)=O)NC(=O)C(C)OCCOC C1(OC)CN(C(=O)Cc2nnc(C)s2)CC1NC(C1CCOC1CCOC)=O C(=O)(C(C)C(=O)NC1CCCC1NC(C1(c2cccc(Br)c2)CC1)=O)OC Cc1ccnn1CC(=O)NC(C)CCCNC(c1cc(C2CC2)no1)=O n1(CC)nc(C(C)C)cc1C(=O)N(C(CNC(=O)CC1(C)CCCO1)C1CC1)C c1(C(=O)NCCC2(OC)CN(C(c3ccccc3C)=O)C2)c(C)ncn(C)c1=O Nc1ccc(Cl)c(C(=O)NCC2CCCN2C(c2cc(CCO)on2)=O)c1 CC1=NOC(C(=O)NC2CC(NC(=O)C)C2)C1.C1(C2CO2)CCCC1.C1CC1 C12(C(NOCCCOC)=O)CC(CO1)N(C(C1CCC1(F)F)=O)C2 c1(CC(N2C(C(C)NC(C(=O)NC(C)C)=O)CCCC2)=O)ccc2c(c1)COC2 C(C#CC(=O)NC(C)C(C)(C)OC)NC(COC(C)=O)=O c1(C(=O)O)sccc1CN(Cc1ccco1)CC12CCCC1C2 C(C)(CCC(=O)NCC1CCCCC1C(=O)NCCS(C)(=N)=O)OCC C1(CC(=O)NCCCOCCNC(CNC(=O)OC)=O)CCC2CC12 N1(c2nccc(C#N)n2)CC2(CCC(NC(=O)CN3CCCCC3)C2)C1 Cc1ccc([N+](=O)[O-])cc1NCc1ccncc1CN1C(=O)CCc2ccccc21 c1(C(N(C)CC2(O)CCCN(C(CC(C)SC)=O)C2)=O)n[nH]c2ccc(F)cc12 C=CC(CC)CC(=O)N1CC(CNC(c2cnc(COC(C)(C)C)s2)=O)C(C)C1 N1(C(C(C)CC2CC2)=O)CCN(C(=O)CSc2nncn2C2CC2)CC1 CCCC(C(=O)NCC1(CC(N2CCC(CC)(CC)C2)=O)CC1)OCC n1(CC)ccc(C(=O)NCC(C2CC2)NC(=O)CN2CCCC2C)cc1=O CCCC(CC(C)C)C(=O)NCCN(C)C(C1COCCO1)=O CC1C(NC(=O)CCOCCNC(=O)C=C2CCC2)CCN1C N1(c2ncnc(=N)[nH]2)CC2CC1CN2C(c1cc(C(N)=O)c[nH]1)=O C1(C(N(CC#C)CC=C)=O)CCCCC1(C)NC(=O)CCc1nccn1C c1(CC)ccc(C(=O)NCC2CCN(C(=O)C(O)CC(F)F)C2(C)C)cc1N N1(C(c2c(C)nc(C)s2)=O)CCC2C1CCN2C(c1ccc(F)c(F)c1O)=O N1(C(CC(CN(C)C)O)=O)CCOCC(CNC(c2cn(CC3CC3)nn2)=O)C1 c1(C(=O)NC2C(CC)N(C(c3ccsc3)=O)CC2)nn(C)c(C(F)(F)F)c1Cl N1(CCNC(C(C)Oc2cccnc2)=O)CCC(NC(=O)CC2CCOC2)CC1 Cc1cc(C)n(CCNC(C2C(O)CCN2C(=O)CNC(C2CC2C)=O)=O)n1 Cc1ccc(C(=O)NC(C2CN(C(=O)CC3CCC(C)(C)CO3)C2)C)nc1C C1(NC(c2cc(CO)[nH]n2)=O)CCN(C(=O)CN2CC(CO)C2)C1 c1(CCC)cccc(NC(=O)C(CC)N(C(=O)C(CN(C)C)CC)C)c1 N1(C(CCCCC)=O)C(CNC(C2(CN(C)C)CCCCC2)=O)CC2COCC12 C1(C(=O)NCC(CNC(CCCc2nc(C)sc2)=O)F)CC2C=CCC(C1)C2 N1(C(C2CC(C)CN2C(c2ccc(N3CCCC3)nc2)=O)=O)CC2C(C1)C2(F)F N1(C(=O)CCCCc2ccc(Br)cc2)CC2CN(C(C3CC(O)C3)=O)CC2C1 C(CCCCC(=O)N1CCC(CC)C1C(=O)N(CC(C)C#N)C)OCC C(C1CCc2ccccc21)NC(=NCc1ccc(SC)s1)NC1CC1 c1(C(=O)NC(CCOC)C(=O)N2CCC(COC)C2)cc2n(n1)CCC2 Nc1ccc(C(N2CCC3C(NC(C4C=CCC4)=O)C23)=O)cc1F C1(NC(C2(C)N(C(C)=O)CCC2)=O)CC2CC1N(C(c1cc(C)cnn1)=O)C2 N1(C(C2(C)CCCC2)=O)CC2C(C1)N2C(=O)CCOc1ccccc1 c1(C(C)C)cc(C(=O)NC2CC(NC(C3CC4(CCC4)C3)=O)C2)n(C)n1 Cc1ccc(-c2cn(C3CC(C(=O)O)C3)nn2)c(C(=O)Nc2cccc(I)n2)c1 C1(CC(=O)N(C)CC2(NC(c3nc(C(C)C)oc3)=O)CC2)CC2COCC12 C1(N(C(C2(C(=O)N)CC2)=O)C)CCC(CNC(c2[nH]c(=N)sc2)=O)CC1 C1(C(=O)Nc2nnc(C)o2)CC(F)CN(C(C2CNC(=O)C2)=O)C1 C1(NC(c2c(C)ocn2)c2nnnn2C2COC2)CCN(S(N)(=O)=O)C1 C#Cc1ccc(C(N2CC3CC3(C(=O)Nc3c(C)cccc3F)C2)=O)cc1 c1(C(N(C)CC2CCCN2C(c2cnc(C3CC3)s2)=O)=O)ccc(N)cc1[N+](=O)[O-] NC1CC2(C1)CC1(CC(NCC(C3CCCCC3)=O)C1)C2 C1(C(C)C)CN(C(c2cc(C3CC3)[nH]n2)=O)CCN1C(=O)CC1CCC(=O)C1C C1(CC)C(=O)NCCN1C(C1C2CN(Cc3cc(F)ccc3C)CC12)=O c1(CNC(=O)C(N2CCOC(Cc3ccccc3Cl)C2)=O)cccc(F)c1F C1(CNC(C(C)CNC(c2cccn2C)=O)=O)CC12CC2(F)F c1(CCC(=O)NC(CNC(CC2(OC)CC2)=O)(C)C2CCC2)cccnc1 c1(OC)cc(C(N2CCC3CN(Cc4ccsc4)CC32)=O)cc(CN(C)C)c1O C(=O)(N=c1[nH]c(Cl)cnc1Br)C1C(NCc2c(OC)ncc(Br)c2)C1 CCC(CN(C)C)C(=O)NC1CC1NC(=O)C(c1ccccc1)N(C)C(C)=O C(CC1=CCCCC1)N(C)C(C1CN(C(c2cccc[n+]2[O-])=O)CC1F)=O c1(NC2C(C(F)(F)F)CCN(Cc3n[nH]c(C)c3C)C2)c(F)cccc1[N+](=O)[O-] C1(C(N(C(CC)C)C)=O)CN(C(c2cn(CC)cn2)=O)CCC1(C)C Cc1nc(C)n(CC(=O)N(C2CC(NC(=O)C=Cc3ccoc3)C2)C)n1 c1(OCCOC)ccc(Cl)cc1C(=O)NC1CN(C(c2n[nH]cc2C)=O)CC1O c1(C(=O)NC(CN(C(=O)C(C2CC2)OC)CC)C)cc[nH]c(=N)c1 CC1OC2CCC1(C(=O)NC1CC1NC(C1C(C)C1C)=O)C2 C(=O)(C(C)(C)S(C)(=O)=O)NCC1N(C(CCc2c(OC)cccc2)=O)CCCC1 O=S(=O)(c1ccc(N2CC3CC3C2)cc1Cl)NCc1cccc(F)c1 N1(C(COC2(C)CCC2)=O)CC(NC(c2cc(=N)[nH]cc2Br)=O)C2(CC2)C1 CC1(CNC(=O)C(F)(F)C2CC2)CCCN(C(=O)Cc2cc(F)ncc2Br)C1 c1(C(N(CCN(C(=O)CCC=C(C)C)CC)CC)=O)nnc2ccccn12 C(=O)(CC(COC)NC(C1CC2(CC2)CO1)=O)N(C(CC)CO)C c1(CCC)nc(C)c(C(=O)NC(C2CCCC2)CNC(c2c[nH]c(Br)c2)=O)o1 N1(C(c2cnc(C)nc2C)=O)CCC(NC(C2(C)CC2)=O)CC(C)(C)C1 C1(NC(CCc2c(C)n[nH]c2C)=O)C2CC1CN(C(c1ccc(=O)n(C)c1)=O)C2 N(C(=NCC1CC1)NCC1CCC(C)CC1)C(C#C)CCC N1(C(C(CC)(CC)CO)=O)CC(C)(C)OC2(C1)CN(C(=O)CC1(C)CC1(F)Cl)C2 C1(CC)CN(C(c2c(C)cccc2O)=O)CCN1C(=O)C(C1CC1)SC Cc1cc(CC(=O)NC(C2CCCCN2C(=O)COC(F)F)C)cc(C)c1 Cc1nn(C)c(C)c1C1OCCC1NC(C1CC2(C1)CC(CNC(=O)C(C)C)C2)=O C(c1cnccn1)=CC(=O)NCC(CNC(C(Br)=C(C)C)=O)(C)O Cc1cc(=NC2CN(C(=O)CN3CCCCC3=O)CC3(CCC3)C2)[nH]cc1C#N CC1CCCN(CCc2nc(CCc3cccn3C)n(-c3cccnc3)n2)C1 C1(C(=O)NCC2(CN(C)C(c3csc(O)n3)=O)CC2)CCCC2(CCOC2)O1 c1(C(N2CCCCC(NC(c3c(C)cc(F)s3)=O)C2)=O)cnn2c1OCC(F)C2 N1(C(C2CC=C(C)CC2)=O)CCN(C(=O)CC(O)C2CC2)C(C)C1 N1(C(c2c(OC)c[nH]n2)=O)CCCCC(CNC(=O)C(C(F)(F)F)OC(C)=O)C1 CN1CCN(CC(N2CCN(C3CCCC3NC(C3CC=CC3)=O)CC2)=O)CC1 c1(C(NOCC(=O)NC(C)CCC2CCCC2)=O)ccccc1 c1(C(=O)NC(CCNC(c2n(C=C)nnc2)=O)(C)C)cc(Cl)c(Cl)n1C C1(N(C(c2[nH]cc(C)c2C)=O)C)CN(C(=O)C(C(C)O)N(C)C)CCC1O C1(O)(CNC(=O)N(C2CC2)Cc2ccccc2)CCN(N2CC(O)C(F)C2)C1 C(C)(C(C)(C)NC(=O)C(O)Cc1ccccn1)NC(CN(CCC#C)C)=O O=C(N=c1[nH]ncs1)NC(CCc1ccccc1)C(F)(F)F N1(C(CC(C(C)C)C)=O)CC2CCC1CC2NC(=O)Cn1cnnc1O N1(C(COCCOCC)=O)CCN(C(=O)Cc2cc(Cl)ccc2Cl)CC1COC CN(C1CCc2ccccc2C1)N1CC(C)(C)C1C1CCN(C(=O)C2CC2)CC1 c1(CC(C)C)cc(C(=O)NCC2CCN2C(=O)CSC2CCOC2=O)n(C)n1 N1(C(C2ON=C(CC)C2)=O)CCCC2CN(C(c3cc(=O)n(C)o3)=O)CCC12 C(=O)(C(C)(C)C(N)=O)NCC(CC(=O)N(C(C)COC)CC=C)C1CCC1 C1(N(C(C2C(=C)CC2)=O)C)CCC(NC(c2ccncc2N)=O)CC1 c1(C(N(C2CCN(C(CC3(C(=C)F)CCC3)=O)C2)C)=O)nc[nH]c2ncnc1-2 N1(C(c2cc(CCOC)on2)=O)CCC(NC(C2CCCC(F)(F)C2)=O)CCC1 c1(OC)ccc(C(=O)NCCN(C(C2OCCOC2C)=O)C2CC2)nc1Cl CC12CN(C(c3cnc(O)o3)=O)CC1CN(C(c1ncccc1OC(F)F)=O)C2 C(=O)(CCCCC(C)CC)N1CC(O)(CNC(COCCSC)=O)C1 N1(CC)CC(C(=O)NCC2(Nc3nccnc3F)CCC2)CC1=O c1(C(N2CCCC(CC(=O)NC3(CO)CCC3)C2)=O)cccn2nccc12 c1(C(N2CCOCC(CNC(C(C)NC(=O)NC)=O)C2)=O)ccccc1S(C)=O CC1(C(=O)NC2CCC2NC(c2ccc(F)s2)=O)CC=CC1 c1(C(=O)NC(CCCCNC(CC(=C)C)=O)C)cc(OC)ccc1F CC(C)CC(CNC(=O)CCCOC(C)C)C(=O)NCC(C)(F)C(C)C C1(CC#N)(NC(C2(C(N(C)C)=O)CC2)=O)CCC(F)(F)CC1 CCC(C(=O)NCC1=CCN(C(C2(c3ccsc3)CC2)=O)CC1)C(C)(C)CC C1(CC(=O)NCCC2(NC(c3cc(COC)no3)=O)CCCC2)CCCCN1C c1(CN2CCOCC(NC(c3ccoc3)=O)C2)n[nH]c2cc(Br)ccc12 Cc1cc(C#N)cc(NC(C2CCCOC2)C)n1 CC1(NC(=O)OCc2ccccc2)CCCN(C(=O)CCCC(F)F)C1 C(=O)(CC(C)(C)SC)N(C1CCN(C(C2CCC=CO2)=O)C1)CC C(=O)(C1=CCCC1)NC(C(=O)NCCCC(=C)Cl)(C)C1CCC1 N1(C(CCS(=O)(=O)N(C)C)=O)CCC(C)(C)C(NC(c2cc(F)cs2)=O)C1 C(CO)(C(=O)NOCC1CCC1)NC(CCn1ncc(C)c1)=O O=C1CCC(c2cn(CC3CCN(C(=O)Cc4cscn4)C3)nn2)CC1 c1(OC2CCN(C(=O)NCCCC(C)OC)CC2O)ccc(Br)c(C)c1C C(CS(=O)c1ccccc1F)Nc1c(C)c(N2CCC(C3CCCC3)C2)ncn1 C1(C)(C(N(C(C(=O)OC(C)C)C)C)=O)C2CC3CC(C2)CC1C3 Cc1cccc(C(C)C(=O)NC2CC23CC(NC(C2(c4cccs4)CC2)=O)C3)c1 CC1(NC(=O)Cc2csc(Cl)n2)CC(NC(C2CC2Cl)=O)C1 Cc1cc(N(C2(C)CC(C)C2)C)ncc1S(=O)(=O)NC1CC(C(F)F)C1 CCC(CC)C(F)C(=O)NCCOCCC(=O)NCC1CCN(C(N)=O)C1 CCC(C)CC(C(=O)NC(C)C(=O)N(CC)CC)NC(=O)C(O)CCC(C)C C1(NC(COCC=C)=O)CCC2(CCCN(C(c3cocc3Br)=O)C2)C1 N1(CC(=O)NC2CCC2c2ccccn2)C(=O)C2CC=CCC2C1=O C#CCCC(N)C(=O)N1CC(C(=O)NCCCO)CC1(C)C Cc1ccc2cccnc2c1C(=O)NCCC(C)(C)NC(=O)CC1CCCC1C C(=O)(C1CCc2ccc(OC)cc21)NCCCN(C(C1C(=C)C1)=O)C Cc1ccnc(F)c1-c1cnc(CNC(c2cc(O)ccc2F)=O)nc1 C1(C(N(CC)CC2CC2)=O)N(C(C2CCC(O)CC2)=O)CC12CCCC2 c1(CN(C=O)Cc2n(C(C)(C)C)ncc2)ccc(N2CCCCC2=O)cc1 C1(C(N2CC(CNC(C3(F)CCCN(C)C3)=O)C2)=O)CC2(C1)CC(C)(C)C2 C(CC(C)C)(C(=O)Nc1ccc(SC)cc1)NC(C=CC(CC)C)=O C1(CCC)CN(C(=O)C=CC=C(Cl)Cl)CCN1C(=O)CC1CCCC(C)(C)C1 c1(C(=O)OC(C)CC)ccc(OC)nn1.C1CCC(C(=O)NC2CN(C(CC)=O)C2)O1 CC1C(NC(c2cc(C3CC3)nn2C)=O)CCN1C(c1ccc(C2CC2)cn1)=O C1(NC(c2cc(OC)cc(Cl)c2)=O)CC2(CCN(C(C3CCC3(C)C)=O)C2)C1 C1(NC(C=NOC)=O)CN(C(C2(c3cccc(C)c3)CC2(F)F)=O)CC1(C)C CC(CC(=O)NC1CN(C(c2cc(F)c(O)c(F)c2)=O)CC1(C)C)C(C)(C)C c1(C(=O)NC(C)CN(C)C(c2ccc(Cl)cc2C(F)F)=O)ccc2ccnn2c1 N1(c2nc(C)cc(OC)n2)CCN(C(=O)C(C)C2CCCC2)CC(O)C1 Cc1ccc(Br)c(F)c1C(=O)NC1(C)CCOC1C1CC1 C#Cc1ccc(C(=O)NC(CN(C)C(C2(CC(C)(C)C)CC2)=O)CC)c(F)c1 N1(C(c2cnc(C3CC3C)s2)C(=O)NCCCC(=O)OC)CCNC(=O)C1(C)C C1(C(N2CSCC2C(=O)NCC(C)C(F)F)=O)(OC)CCC(C)C1 c1(N2CCCC(C(C)NC(c3c(C)c(I)ccc3)=O)C2)ncnc2cc(I)sc12 c1(C(N2CC(NC(C(CC#C)O)=O)C(C=C)C2)=O)cc(Br)ccc1[N+](=O)[O-] c1(OC)cnc(F)c(C(=O)NCC2(OC)CN(C(C3CCCN(CC)C3)=O)C2)c1 c1(CC(=O)N(CCC(N2CCC(NC(=O)NC)CC2)=O)CC)cccc(C)c1Cl c1(OC)ncc(CN2CCCC(NC(c3nccnc3C(N)=O)=O)CC2)cc1C N1(C(CNC(C)=O)=O)CCCC(O)(CNC(C2CC(C3CCC3)C2)=O)CC1 N(C(=NCc1ccccc1)N1CCC(Cc2cc(C)ccn2)C1)C(COC)C c1(C(N(CCNC(c2cc(C(CC)CC)no2)=O)C)=O)ccc2[nH]c(=N)[nH]c2c1 C(CCC(C(=O)NCC(C)C)N1CCC(CCS(C)(=O)=O)CC1)=C(C)C CCCC(CCC)C(=O)NC1CCC(N(C)C(c2onc(Br)c2C)=O)C1 c1(CC)cc(C(F)(F)C(N2CC(NC(=O)OC(C)(C)C)CC2C(=O)OC)=O)n(C)n1 CC12COCC1CN(C(C1N(C(=O)C3=NNC(=O)C3)CC13CCCC3)=O)C2 c1(C(=O)NCCC(C)N(C)C(C2CNC(=O)N2)=O)ccc2c(n1)CCC2=O CC(C)C(O)CC(=O)NCCCN(C(C1(C)CC(OC)(OC)C1)=O)C1CC1.N(C)C Cc1cc(C(N2CC3CC3(NC(=O)CCCc3ccsc3)C2)=O)c(C(F)(F)F)o1 c1(CN(C)CC2CN(C(=O)CC34CCCN3CCC4)C2)cc([N+](=O)[O-])ccc1F N1(C(c2c(C)nn[nH]2)=O)CCC(C)N(C(c2cc(Cl)cnc2O)=O)CC1 C(=O)(C(CCN(C)C)N(C)C)NCCC1N(C(C(=C(C)C2CC2)F)=O)CCC1 C(C(O)C(=O)N(CC(=O)NCCN1CCCC1)C)N(C)C c1(C(N(CCC)CCNC(=O)CC2COCCN2C)=O)cc(F)c(CO)c(F)c1 Cc1ccc(C(=O)NC2CC3CCC2N3C(=O)C(C)(O)C(C)C)cc1C C#Cc1ccc(NC(=O)C(=O)Nc2cnn(CC(N3CCCCC3)=O)c2)cn1 C(=O)(C1=CCC2CCC1N2C(C1(C)CCC(F)(F)CC1)=O)OC(C)(C)C N1(C(C=CSC)=O)CC(NC(=O)C(CC(C)C)NC(=O)OC(C)C)CC12CCC2 N12CCC(C)(CC1)C2=O.C1(C(C)=O)CC=CC(n2cc(C3C4COCC34)nn2)C1 Cc1cc(C(N2CC(C(C)NC(C3COCCO3)=O)C2)=O)cc(Cl)n1 N1(C(CCN(CC#C)C(C2CC2C(C)(C)C)=O)=O)CC(F)(F)C1 c1(CCNC(c2n(C)nnn2)CCc2ccsc2)ccccc1[N+](=O)[O-] CCC(C)(C(c1nnnn1C1CCCCC1)NCCCc1ccco1)OC c1(CC(C)C(=O)NC2CC(NC(=O)Cc3ccco3)CC2O)cccc(Cl)c1 C1(CNC(C2(C(C)(F)F)CCC2)=O)C=CCN1C(=O)Cn1cnc(C(N)=O)n1 N1(C(=O)CNc2nccs2)C2CCC1CC(NC(C1(O)CCOC1)=O)C2 c1(NC2CC(CNC(C3CC(OC)C3)=O)C2)csc(CC(c2ccccc2)=O)n1 N1(C(C2(F)CCN(C(Cc3ccc(C)s3)=O)C2)=O)CCCC(C)C1CO N1(C(C(=O)Nc2cc(C(C)(C)C)no2)=O)CCOCC1C1CC(F)(F)C1 c1(C(N2CC(=C(CNC(C3C(C)C3C)=O)F)C2)=O)nccc2[nH]ccc12 C1(CC=C)(N(C(C)=O)C2CC2)CN(CCn2nnc(-c3ccsc3)n2)C1 c1(C(C)=O)cccc(CCn2cc(CC3CN(C(=O)CCC(F)F)C3)nn2)c1 c1(C(C(=O)Nc2cc(C(=O)N(CC)CC)c(Cl)cc2)O)cc(F)c(F)c(F)c1 C(=O)(C#CC1CCCC1)N(C1CCC(NC(c2c(OC)c(Cl)sc2)=O)CC1)C c1(C(=O)NC2C(C=C)COC2)ccc(OC(F)F)c(OC)c1 n1(CC(=O)NC(C)(CNC(c2nccnc2O)=O)C2CC2)cnc([N+](=O)[O-])n1 C(c1ccc(F)cc1F)=CC(=O)NCC1CC(NC(=O)CCN2CCCC2)C1 c1(C(=O)OCC)cn(CCC(=O)N2CC(Cc3nnc(OC)s3)C2)nn1 CC1CCN(C(C2CC(CNS(C)(=O)=O)C2)=O)CCN1C(=O)Cc1cccnc1 C(=O)(C(C)CCCC(C)=O)NC(CCC)C(N1CC(O)CC1(CC)CC)=O c1(C(C(=O)Nc2ccn(CC(=O)N(C(C)C)CC)n2)N(C)C)c(F)cccc1Cl c1(CC(=O)NCC2CN(C(C34CC(C3)S(=O)(=O)C4)=O)C2)ccc(F)c(Cl)c1F C(CCS(C)=O)(C(=O)NC1CCC(NC(c2ocnc2C2CC2)=O)CC1)N(C)C C1(CNC(CSC)=O)CC(C(C)C)CCN1C(c1cnccc1Br)=O Cc1ccc(F)cc1CN1CCCCC(NC(=O)C(C)(O)Cc2ccccc2)C1 N1(C(C2(C=C)CC2)=O)CCCCC1C(C)NC(=O)CCn1cc(C)cn1 c1(C(=O)OC)ccc(C=CC(N2CCCCC2CNC(C2CCCSC2)=O)=O)o1 C1(CNC(c2c(F)ncc(C)c2)=O)CC2(CCC2)CN1C(c1ccnc(Cl)c1)=O N1(CCCC)C(=S)NC(c2cccc(OC(C)=O)c2)C(C(=O)OC)=C1C1(C)CC1 c1(C(N2C(CC(=O)N)COCC2)=O)cncn(C)c1=O.C(C(CO)n1cccn1)OC C1(N(C(=O)Cc2ncc(C)s2)CC)CCN(C(C2CC2F)=O)CC1 C1(C)(NC(CCC(=O)OCC)=O)CCN(C(C2(C)CCCC2C)=O)CC1 Nc1c(C(=O)Nc2ccc(N3CCCCC3)c(F)c2)cc(Cl)nc1Br CC1=C(C(=O)NCC2CCOC2C(=O)NCC2CC2c2ccoc2)CC1 c1(C(N2CC3C(N(C(CC4CCCC(C)O4)=O)C)C3C2)=O)c[nH]c2nccc-2c1 N1(C(CC(=O)NCC#C)=O)CCN(C(C2(c3ccc(F)cc3)CC2)=O)CC(O)C1 N1(C(C2CC(OC)C2)=O)CCC(NC(=O)Cc2ccc(SC3CC3)cc2)C1(C)C C1(C(=O)NC(CC(=O)OC)C2CC2)C(C)CCN1C(c1cncc(NC)n1)=O CCC(O)C(F)(F)C(=O)NC1CC(NC(=O)CN2CC(C)(C)C2)C(O)C1 C1(C)(CNC(c2cnc(COC)s2)=O)CC(F)(F)CN1C(=O)Cc1ccc(Cl)s1 CN=C(NC1CCN(c2ccc3cc[nH]c3n2)CC1)N1CCCCCCCC1 c1(C(=O)NC(CC=C)CNC(=O)C(c2ccnn2C)OC2CC2)ccccc1Cl C(=O)(CC(C)(C)O)NCC1(C(N)=O)CN(C(c2c(CC)[nH]cc2)=O)C1 N1(C(C=CCN(C(=O)CC2CCSC2)C)=O)CCN2CCCCC1C2 c1(CCC(=O)NCC2CN(C(=O)C=Cc3cocn3)CCO2)cc(F)ccc1F C1(NC(c2ccc(OC)nn2)=O)CC(F)CN(C(c2cc(C)nc(C)c2)=O)C1 C=CCC(CNC(c1[nH]ccc1C1CC1)=O)C(=O)N1CCC(CC)C1 C12(C(=O)NC(C3CCOC3)CNC(=O)CSc3ccccn3)CC1CNC2=O CN(CCCC(=O)NC(c1ccc(F)cc1)CNC(=O)Cn1cncn1)N=O c1(C(C)C)cc(C(=O)NCC2CCCCN2C(=O)Cc2cncs2)ccc1F C1(NC(=O)CC2(O)CCCCC2)CCCN(C(=O)CCc2ccsc2)CC1F C12CCCCCC1C(=O)N2.Cc1ccc(C(N2CCCC2C2(C)CC2)=O)s1 CCC(CC(=O)N(CC(C)NC(=O)C(C)=C(C)C)C)NC(N)=O c1(C(=O)NC2CCCC(NC(CC=CC)=O)CC2)cc(C)c(Br)c(Cl)c1 C1(CCC)(NC(=O)COCC)CCN(C(=O)C(C(C)(C)C)NC(N)=O)CC1 C(=O)(C1Cc2ccccc21)NCC1(F)CCN(C(c2ncn(C(C)(C)C)n2)=O)C1 N1(C(C2CC(C#C)(O)C2)=O)CC2CC1CCN2C(c1cccc(C2CC2)c1)=O C1(NC(C(C(CC)O)C)=O)CCN(c2nc(C(F)F)nc(=N)[nH]2)CCC1CO Cc1ccnn1C(C)C(=O)NC(C)(C)CNC(=O)C(C)Cc1ccccn1 C(=O)(C(CCC1CCCC1)N(C(C)CCNC(=O)OC(C)(C)C)C)NCC CCCCC(C(=O)NC(CCN(C)C(C1CC2CC1C2)=O)C(C)(C)C)NC(N)=O c1(C(=O)OCC)cccc2c(NC(=O)COc3ccccc3C)c[nH]c12 N1(C(CC)=O)CCC2(CCCN2C(=O)C(C)CC(=O)c2ccc(F)cc2)C1 c1(C(=O)NCC2CC(OC)CN2C(C2COCCOC2)=O)cc(O)ccc1Cl c1(CC=C)cc(C(=O)NCC(C(C)C)NC(=O)C(O)CSC)cc(OC)c1OC c1(CC(=O)NCCN(C(=O)Cc2ccccc2SC)CCOC)nn(C)cc1Cl c1(C(=O)NCC(C)CN(C(=O)CCC2CC2)C)n[nH]c2c1CCCC2 C1(CC)CN(C(c2cccc(C3(O)COC3)c2)=O)CCN1C(c1ccc(C)o1)=O C(=O)(C(C(C)C)C(C)C)NC1C2CN(C(c3ccc(C(CC)C)cc3)=O)C1CC2 C1(CNC(C=C(CC)C)=O)CN(C(c2ccc(O)c(F)c2)=O)CCC12CCOC2 CC(CC(C)(C)CO)NC(=O)CC1N(C(c2nc(Cl)cs2)=O)CCC1(C)C C#CCC(CC(F)F)C(=O)N1CC(NC(c2cnoc2CC)=O)C2CCCC2C1 O=C(C1=CS(=O)(=O)c2ccccc21)N1CC2CCN(C(c3ccsn3)=O)C2C1 C(=O)(C(C(C)(F)F)c1ccccc1)N=CCCCN(C(=O)C=CC(C)C)CCOC C1(C(=O)NCCOCCCN(C(=O)CSc2nc[nH]n2)C)CC12CC(O)C2 c1(C(=O)NC(c2cc(Br)c(F)cc2F)C)cc(F)c(N)c(F)c1 N1(C(=O)CC2CC=CCC2)CC2CCCC2(Nc2ncncc2Cl)C1 N1(C(c2cccc(Cl)c2C)C(=O)NCCCCCC)CC(=O)NC2(CCCC2)C1 c1(OC)cc(C)c(Cl)cc1C(N1CCN(C(c2cc(F)c(C)c(F)c2)=O)CC1)=O N=c1[nH]cc2c(c1C(N1CCC3(CCC3)C(NC(=O)C3=CCSC3)C1)=O)CCC2 N1(C(Cc2nnc(C)o2)=O)CC2(C)CN(C(C3CC3C)=O)CC2(C)C1 C(=O)(C(C)(C#N)CC(=O)NCCCSC)NCCNC(CCCOCCOC)=O Cc1onc(Cl)c1C(=O)NC1CN(C(C2SCCS2)=O)CC1CC1CC1 CC(C(=O)NC(C)CSC(C)(C)C)OC1CCCC1 C1(NC(=O)Cn2cncn2)CN(C(c2cnn(C3CCC3)c2)=O)C2(CCOC2)C1 c1(CC(=O)NCC2(C)CCN(C(=O)CN3CC=CC3)C2)cccc2ccccc12 c1(CCC(=O)NCC(C(C)(C)C)NC(C(COCC)C)=O)cc(F)cc(F)c1 C12(C(=O)NC3C(CNC(C4N(C)CCCC4)=O)COC3)CCC(CO)(CC1)C2 C1(NC(CCn2ncc(C)c2)=O)C2CCCN(c3ncnc(O)c3Br)C2C1(C)C N1(C(C2CCC(C)(CC)O2)=O)CC2CCC1CN2C(=O)C(C(C)(C)C)NC(N)=O c1(C(N2C(C)(C(N3CCC(C(=O)OC)C3)=O)CCC2)=O)ccc(F)cc1C c1(C2CC(=O)NC2)cccc(NC(c2cnn(CC(N3CCOCC3)=O)c2)=O)c1 c1(C(N2C(CCNC(CC(=C)C)=O)CCCC2)=O)cc2nccc(Cl)c2s1 c1(NC(CC#C)COC)cnc(Cl)c(C2CC2)c1 C(C(C)C(C)C(=O)N(C)CC1(NC(c2ncoc2C2CCC2)=O)CC1)OC C(=O)(C1=COCCO1)NCC1CC(N(C)C(c2sccc2OC(F)F)=O)C1 CCC(CC)(CCNC(=O)CCc1cncnc1)NC(c1nccc(N)c1Cl)=O C(C)(C(O)C(=O)NC(C)(C)CCNC(c1cccc(N(C)C)c1)=O)SC N1(C(C23CN(C(C4CC(C#C)(O)C4)=O)C(C2)CO3)=O)CC2(C1)CC1(CCC1)C2 C#CC(C(C)OC)NC(C1(C)CC(NC(c2cc(O)cs2)=O)C1)=O N1(C(C(CC)C)=O)CC2CCN(C(=O)CC3CCC(O)C3)C2C1C c1(C(n2cc(C3(C)CN(C(c4c(C(C)C)cco4)=O)C3)nn2)C)ccccc1Br c1(C(=O)NCC(CNC(=O)CCc2cn[nH]c2)OC)cnc(S)n1C1CC1 CC(F)(F)C(F)C(=O)NCC1CC(C(=O)NCC2CCC(O)CC2)=NO1 N1(C(CN2CCC(C)(C)C2)=O)CC2(C1)CN(C(C1CC3CCC1C3)=O)C2 N1(C(c2ncn(C)c2)=O)CC2COCCC2(NC(=O)C=Cc2cc[nH]n2)C1 c1(OC)ccc(COC(c2cc(C3C(C)(C)C3(C)C)[nH]n2)=O)nn1 N1(C(CS(=O)(=O)NC)=O)CCCC12CCN(C(=O)Cc1ccc(O)cc1C)CC2 C1(C(N2C3CC(NC(CC=CC=C)=O)CC2CC3)=O)CC(c2ccncc2)=NO1 c1(CN2C(C(=O)NC3CN4CCC3CC4)CC3CC32)c[nH]c2cccc(Cl)c12 C(CCC(C)(C)C(=O)NCCOC(C)(C)C)N(C(CC1CC1)C(=O)O)C c1(C(CN(C)C)NC(=O)Cn2cc(CC3CCNC3=O)nn2)ccc(Cl)c(Cl)c1 N1(C(C=CCC(C)(C)NC(=O)Cn2[nH]cnc2=N)=O)CCCC2(C=CCO2)C1 C=CCC(CC(=O)Nc1cnc(CC)nc1)NC(=O)C(CO)NC C1(C(C)C)OCCC1CNC(C1OCCC1NC(=O)C(C)(C)OC(C)(C)C)=O C1(NC(C2N(C(C)C)CCCC2)=O)CC12CCN(C(=O)CCP(C)(C)=O)CC2 c1(CC(=O)N(C)CC2N(C(CC(=O)OC)=O)CCCC2)nsc2ccccc12 C(C)(C)(CCC(=O)NC(CC)CCC)NC(C1C(=C)C1)=O N1(C(CNC(CN(C)C)=O)=O)CCN(C)C(C(=O)NCC2(CO)CCCO2)C1 C(=O)(C1CCc2c(Cl)cccc21)NCCC1(NC(C2=CC(C)(C)C2)=O)CCC1 c1(CN(c2c(C)nn(C)c2C)C2CC3CNC2C3)ccc2oc3ccccc3c2c1 c1(C(=O)NCC2CCCN(C(C3(C#N)CCOC3)=O)CC2)nccc2cc[nH]c12 c1(C(N2C(C)(C(=O)NCc3ccnc(OC(F)F)c3)CC2)=O)c(F)cncc1Br C(=O)(CC(CC)SC)NCC(CCNC(c1cnc(CC)s1)=O)O c1(CC)cnoc1C(=O)NC(C)CCCNC(=O)C=CCCC(C)C C1(C(=O)NCCCN(C)C(C2CC3(C2)CC3F)=O)(N(C)C)CCCCC1 C1(CNC(C=C(C)Cl)=O)CN(C(C23CC2COC3(C)C)=O)CC12CC2 C1(O)(C(=O)NC2C(NC(C3CC3C(F)(F)F)=O)CCOC2)CCOCC1 C1(NC(CCC2N(C)CCC2)=O)CCCN(C(=O)CC(C)(O)c2ccccc2)C1 Cc1cc(CO)oc1C(=O)N(C)CC1CCN(C(=O)CC2COCCN2C)C1 N1(C(CC(CC)O)=O)CCC2(CCCN2C(c2cc(CO)oc2C)=O)C1 N1(C(CC2(CSC)CC2)=O)CC(OC)CC(NC(=O)CC2C=CCCC2)C1 C(=O)(C(C)C(F)(F)F)NC(C)CCCNC(C1(C(C)(F)F)CC1)=O C12(C(=O)NCCC3C(C)(C)C3)CCC(CN(C(C34CC(C#N)(C3)C4)=O)C1)C2 O=C(C1CSc2ccccc21)NC1(CCNC(C2(C(F)(F)F)CC(O)C2)=O)CC1 C1(C(=O)NCC(CCC)NC(=O)Cc2cc[nH]n2)(CC)CC(C)(C)C1 C1(C(N2CC(OCCNC(C(C)n3cnnn3)=O)C2)=O)CC=CCC1C(F)(F)F c1(C(N(C(CNC(C(C(C)C)(C)C)=O)C)C)=O)nc2ncc(Br)cc2[nH]1 C1(NC(c2c(C#C)c[nH]n2)=O)CN(C(C2COCCN2C)=O)CCC1(C)C S(=O)(=O)(CC(=O)NC1(C)CN(C(=O)CC(c2ccccc2C(F)(F)F)C)C1)NC c1(CN2C3(CNC(c4n(CC)nc(C5CC5)c4)=O)CC(C2)C3)ccc(C)cc1Cl c1(C(=O)NCC2N(C(C3N(CC)CC3)=O)CC2)cc(N)cnc1C c1(NC(CC(=O)N2CC(CNC(COC(C)=O)=O)C2)=O)cccc2ccccc12 CCCCCCCCS(=O)(=O)N1CC2CN(C(c3cc(Br)ncc3Br)=O)CC12 O=C1CCN(C(=O)CCc2ncccn2)C(C(N2CC=CC(O)C2)=O)C1 CC1CCOCC1C(=O)N(C1(C(=O)NCCc2cccc(F)c2)CC1)C C1(CC#C)(C(=O)NCC23COC(CNC(=O)C(C)(C)COC)(C2)C3)CC=CCC1 C1(CNC(c2cc3c[nH]nc3s2)=O)CCCCN(C(C2CC23CC(F)(F)C3)=O)C1 N1(C(c2ccc(C)c(N)c2)=O)CCN(C(=O)CSC2CCS(=O)(=O)C2)CC12CC2 CC1C(NC(=O)C(C)(C)N2CCCC2)CCCN1C(c1cc(C2CCC2)[nH]n1)=O CC(C(C)C(=O)N(CCCCNC(C12CC(CCO1)C2)=O)C)C(C)(C)C C1(C(=O)NCC2CC(NC(C(CCSC)NC(N)=O)=O)C2)CCC2CC2CC1 N1(C(C2(C)CCCNC2=O)=O)CC2CCC(C1)N2C(c1cccc(N)c1O)=O N1(c2cc(COC)ncn2)CCC(CNC(C2CCCSC2)=O)C(C)C1 c1(C(=O)NC(C(C)C)C(C)NC(C2C3CCC2CC3)=O)ccc2nc[nH]c2c1 Cn1ccc(C(=O)N(C2CC2)CC2CCCN2C(=O)C=CC(F)(F)F)cc1=O c1(-c2nc(C)c(N(C)C)s2)cc(C(N2CCCC(CO)(CO)C2)=O)c2c(c1)CCO2 N1(C(c2ncc(C(F)(F)F)[nH]2)C(=O)NC)CCOCC1C1CCOCC1 C1(NC(CCCOCC)=O)CN(C(C2(COC)CC=CC2)=O)CC1C c1(C(=O)NC2CCCN(C(CC(C(C)C)O)=O)C2)cc2c(cc1N)OCCO2 CC(O)C(C(N)=O)NC(=O)CC1(C)CCN1C(C1CCCNC1=O)=O c1(C(=O)NC2C(NC(C3C(C(N)=O)C3)=O)CCC2)cccc(C(F)(F)F)c1 C(N=c1nc(N2CCc3nc(Br)sc3C2)c2[nH]ccc2[nH]1)C1CC(OCC)C1 CCC(C)CC(C)C(=O)N1CC2CC1(c1cn(-c3ccncc3)nn1)CO2 N1(C(c2c(CC)ccs2)=O)C2CCC1CN(CC(N1CCCCC1=O)(C)C)CC2 CCCC(O)C(CO)NC(=O)CCN(C(C1CCCCC(=O)N1)=O)C(C)C N1(C(C2CSCCN2C(c2cnccn2)=O)=O)C2CCC1COC2 c1(C(N2C3CN(C(CC(C(C)C)C)=O)C(C3)C2)=O)ccc2cncn2c1 C1(CCNC(CN(C)C2CC2)=O)CCCCN1C(C1CCCCC1O)=O Cc1ccnnc1C(=O)NCCC1CN(C(=O)Cc2nonc2C)CC1C N1(C(c2n(CC)nnc2)=O)CC(C(=O)NCC2(C)CCOCC2)C2(CCC2)C1 S(=O)(=O)(c1cnn2ccc(N3CCC(C)(F)C3)nc12)NC1(CC(C)C)CC1 C(CC1CCC1)(C(=O)NC(C1CN(C(=O)C(c2ccccn2)O)C1)C)OC C(=O)(C1=C(F)CN(C(C2CNC(=O)C2)=O)CC1)NC1C(C#N)CCCC1 N1(C(COC(C)=O)=O)CCC(C)(CNC(c2ccc(C(F)(F)F)nc2)=O)CC1 C(=O)(CC(C)(C)CNC(C12CCCN1CCC2)=O)N(CCCSC)C N1(C(C(CC(C)C)NC(C)=O)=O)CC2(C=C(C(=O)NC3CC(=O)N(C)C3)CO2)C1 C1(C(=O)NC(CO)(CO)CO)CN(C(=O)Cc2cccnc2)CC1F c1(C(=O)NCC2CC(NC(C3C(C)(C)OC3(C)C)=O)C2)cc2n(n1)CCCC2 C1(C)(NC(CCCn2c(C)ncc2)=O)CCCN(C(=O)CC(=O)N(C)C)C1 c1(CC)ccccc1CC(=O)NC1CCCC1NC(=O)C(C)(C)c1ccsc1 n1(CC)nc(C)c(C(C)NC(N2CC(Sc3ccccc3)C2)=O)c1C c1(C(N(C(C)CNC(=O)Cc2ccn(CC)n2)CC)=O)cc(C(N)=O)no1 C(CC(C(=O)NC(CNC(c1sccc1C(F)F)=O)CO)OC)OC CC1CC(C(=O)NCC(Cl)Cl)CN(C(=O)CNC(=O)NC2CC2)C1 N1(C(C2N(CC)CCC2)=O)CCC2(C1)CN(C(=O)C=Cc1ncccc1C)C2 CC1(C)COCCC1C(N1CCC(=CCNC(C2CC3(C2)CC3(F)F)=O)CC1)=O c1(C(N2CC(CC(C)NC(=O)CSc3n[nH]c(=N)s3)C2)=O)n[nH]c2c1COCC2 CCC(CC)(CC)C(=O)N1CCC(C)(NC(c2ccc3nc[nH]c3n2)=O)C1 N1(C(=O)OCC)CCN(C(=O)Cc2cnccc2C)C(CC(F)F)C1 C1(O)(C(=O)NCC(C)NC(CCOCCOCC)=O)CCOC1(C)C N1(C(C2CCN(C(c3n[nH]c(C)c3Br)=O)CC2)=O)CC(C)NC(=O)C12CC2 C(C(C)C(F)C(=O)NOC(C)CC)NC(c1c(CC)n(C)nc1)=O OCC(CO)(CO)CCCNC1CCNC(c2cccc(C(F)(F)F)c2)C1 CC1CN(C(=O)C(O)c2ccsc2)CC1CNC(=O)CCCOc1ccccc1 C1(NC(C=CC(C)C)=O)CCN(C(=O)CCC2CCC(=O)N2)C12CC2 C1(NC(Cc2cc(C)c(F)cc2)=O)CC2CC(NC(=O)CC3(C)CC3)CC2C1 Cc1cccnc1CC(=O)NCC(C)NC(=O)C(C)n1cccn1 c1(OC)cccc(C(C)C(N2CCCC2CN(C(=O)C(C)OCC(C)C)C)=O)c1 c1(OC)ccc(N2CC(C(=O)NCC=CCOC(=O)CC3CC3)CC2=O)cc1 C1(OC)CS(=O)(=O)CC1NCc1cnn(CCc2ccccc2)c1 c1(OC)ccnc(C(=O)NC2(C)CCN(C(C3CCCS(=O)(=O)C3)=O)C2)c1C c1(NC(C(=O)N(CC(C)CNC(c2cscn2)=O)C)=O)ccccc1 C1(NC(=O)CC2CCS(=O)(=O)C2)CCCCN(C(=O)CCC2CCOCC2)C1 N1(C(c2ccccn2)=O)CCCCC(NC(c2cn(CC(=O)OCC)nn2)=O)C1 C1(C)(C(=O)NCCCN(C)C(C2(C3CCCO3)CCOCC2)=O)CCCCO1 CC1CC(=CC(=O)N(C)CCOCCCNC(=O)CN(C)C(=O)OC)C1 N1(CC(=O)NCC2CC2CNC(c2ccc[nH]2)=O)CSCC1=O N1(C(C(CC=C)C)=O)CCC2(CC1)CC(NC(=O)CCNC(=O)COC)CCO2 C#CCC(CC(=O)NCc1nc(CC)cs1)NC(=O)CNC(C1CC1C)=O c1(C(N2CCN(Cc3n(C(C)C)ccn3)CC2)=O)nccc2ccncc12 C1(C(=O)OCC=C(CC)C)CCC(c2ccccn2)CC1 C1(C)(CC)CC(C(=O)NCCCCCCN(C(=O)C(C)CSC)C)CCO1 N1(Cc2ccc(-c3c(C#N)ccc(C(F)(F)F)c3)s2)C2CCCC1CC(N)C2 C1(OCC(=O)NCC2(C(N(C(C(C)SC)C)C)=O)CSC2)CCN(C)CC1 c1(CNC(NC2C(C)C2)=NCCNCCS(C)(=O)=O)cc(CO)n2c1COCC2 N1(C(c2c(OC)nsc2)=O)CC2CC2(CNC(c2nc(C(F)(F)F)cn2C)=O)C1 c1(N2CC(Cc3sccc3)OCC2)nccc(=NCC2C3CCC(F)(F)C23)[nH]1 c1(C(=O)NC(CN(C(C2CCOC2)=O)CC)C)ccc2c(c1)N(C)C(=O)CC2 C1(C(=O)NC23CC(CNC(C4(CC)CC4)=O)(C2)C3)CC(OC)C(OC)C1 c1(OC(C)C(=O)NC2CCNC2=O)cccc2ccccc12 N1(C(c2cnn(CC)c2C2CC2)=O)CCC(CNC(C2CC2(C)Br)=O)C(C)C1 N1(C(C=CCOC)=O)CC2(CC(NC(c3snnc3C)=O)C2)C1 C#Cc1ccccc1CN1CC(CC(C)C)C1 c1(COC(c2n[nH]c(C)c2C)=O)nc(O)c2cc(Cl)ccc2n1 CC(CN=c1nc(N2CCOCC2)[nH]c(=NC2CC2N(C)C)[nH]1)C(C)(C)C N1(C(C(C)C)=O)CCC2(CCCC2NC(=O)CCCn2ccnc2)C1 c1(C(=O)NC(CNC(C(C)=C2CCCC2)=O)(C)C(C)C)ncc(Cl)cc1F N1(C(c2c(C(C)(C)C)noc2)=O)CCC(NC(=O)CC2CCC23CCC3)C(F)C1 [N-]=[N+]=NC1(C(=O)NC2CCC2)CCN(C(=O)CCC2CC2(F)F)C1 c1(N2CCC(NC(C3(O)CCOCC3)=O)C2)ncc2cc(Br)cnc2n1 Cc1nnc(Oc2cccc(NC(=O)NNC(=O)CSc3ccccc3)c2)nc1C N1(C(C2N(C(C)=O)CSC2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)CC(O)C1.COC NS(=O)(=O)CC(=O)NCCC1CCCN(C(c2cncc(O)c2)=O)C1 N1(C(C2CC(NC(c3c(OC)ccnc3)=O)C2)=O)CCC2(CCNC2=O)CC1 CCCC(C(=O)NCC(C)(CC(C)C)NC(c1sc(C)nc1C)=O)C(C)C Cc1sc2ccccc2c1CNC(c1cccc(-c2cnc3cncn3c2)c1)=O CCC(C)CCC(=O)N1CC(CNC(c2cccnc2N)=O)C(C)(C)C1 c1(CC)cc(C(=O)N(C2CCCN(C(C3(OC(C)=O)CC3)=O)CC2)C)c(C)nn1 C(c1cn[nH]c1)=C(C)C(=O)N1CCC1C(=O)NC(C)COC(F)(F)F C(=O)(CC(C)(C)C(F)(F)F)OCc1c(OCC=C)cccc1 C1(C(=O)OCC)C(C2CC2)CCN1C(=O)Nc1cc(OC(C)(C)C)cnc1F N1(C(c2ccc(CC)cn2)=O)CC(C(=O)NCC(C)(O)C2CCC2)C(F)(F)C1 c1(C(N)=O)ccc(F)nc1NC(C1CN(C(=O)CN2C(=O)C=CC2=O)C1)=O C1(C(N2C(C(=O)NCCC(C)C)C=CC2)=O)CCCC(C#N)C1 C1(C(=O)NCC2N(C(C(F)OC)=O)CCCC2)Cc2cscc2C1 C1(CNC(=O)CNC(=O)C2CC2)(CNC(C2CC(O)CN2)=O)CC1(F)F c1(C(=O)NC(C)C#N)cc2c(s1)CCN(Cc1ccc(Br)c(Cl)c1Cl)C2 C1(O)(CNC(=O)C(O)c2cnc[nH]2)CC(NC(=O)CCOC2CC2)C1 C1(C(=O)NCCCCC2CN(C(C(C)(C)F)=O)C2)C2Cc3ccccc3C12 C(C(CNC(c1nc(=N)cc[nH]1)=O)C(F)(F)F)NC(C1N(CC)CCC1)=O C1(C(CNC(C=C(C)Cl)=O)F)CCN(C(c2cc(C(F)(F)F)on2)=O)CC1 C1(C)(CNC(CC(CN(C)C)O)=O)CN(C(C2CCCCC2)=O)CCO1 C1(CC(=O)NCC(CNC(C(c2c(OC)cccc2)O)=O)C)CC(=O)NC(=O)C1 C(=O)(CCCC(=O)N1CSCC1C(=O)NCC1CCCC1N(C)C)OCC c1(NC(N2CCC(C(N)=O)C2)=O)ccc(-c2cncnc2)cn1 c1(C(=O)NCCC2(O)CN(C(c3cc(N)c(Cl)cc3)=O)C2)cc(F)c(O)c(F)c1 S(=O)(=O)(c1ccc(Cl)cn1)NC1COCCN(C(c2sccc2F)=O)C1 CC1(C)CC(N=c2[nH]c(=NCCC3(CS(C)(=O)=O)CC3)c3ncccc3[nH]2)CCS1 Cc1nc(C)n(C2CCCN(C(=O)Nc3cc(N4CCCC4)ncn3)C2)n1 C=C(C)C1OCCC1C(N1CCC(CCOC)(C(N2CC=C(C)C2)=O)CC1)=O CCC(CC(=O)N1CCC(C)CC1C(=O)NCC1CC2(CC2)C(=O)O1)C(F)F N1(C(c2n(C(C)C)nnc2)=O)CCCC(NC(=O)C(O)(C2CC2)C2CC2)CC1 C1(C(=O)NCC2(C)CC(NC(=O)C3=CCCSC3)C2)CCc2ccccc2O1 c1(NCC2(C)CCN(C(=O)CCn3cc([N+](=O)[O-])cn3)C2)ncnc2scnc12 c1(OC)cc(CC(N2CC3C(CNC(c4nnc(C)s4)=O)C3C2)=O)ccc1O c1(C(=O)NCC2CN(C(Cc3cn(C)nc3)=O)CC2(C)C)nc[nH]c2nccc1-2 C1(OC)CN(C(c2ccc(C(C)=O)cc2)=O)CCC1NC(c1ccc(C)cn1)=O c1(OCC(=O)NCC2CCCN(C(=O)CCn3cccn3)C2)cccc(Cl)c1 CC1(C)CCC(CNC(c2ccc(F)o2)=O)N(C(c2c[nH]c(=N)s2)=O)C1 N1(C(C(C)OC(C)=O)=O)CCC(C(N2CC(C(=O)N(C)C)C2)=O)C(O)C1 C12(c3nn(-c4ccc(C)c(F)c4)c(-c4coc(Cl)n4)n3)CC3CC(CC(C3)C1)C2 C1(N(C)CCOCCN=[N+]=[N-])CC2CCC(C1)N2C(=O)C(N)=O c1(C(=O)NCCCCC2CN(C(C(C)C(C)(F)F)=O)C2)cncc2ccccc12 N1(C(C(CCC)NC(N)=O)=O)C2CCC1CC(NC(C1OCC1(C)C)=O)C2 c1(OC)ccc(C#N)c(NC(=O)Cc2csc(=NCc3c(O)cccc3F)[nH]2)c1 CC1(CNC(=O)C(F)(F)CN2CCCC2)CN(C(=O)CCN2CCCC2)CCO1 c1(CC=C)cccc(C(=O)Nc2cccc(CNC(=O)C(C(C)C)OC)c2)c1 C(=O)(C1CCCc2n[nH]cc21)NCC1N(C(=O)C=Cc2ncc[nH]2)CCN(C)C1 C1(C(=O)NCCC2CC(NC(C(CCC)C)=O)C2)CSc2ccccc2O1 CC(C)(C)C1=NOC(C(N2CC(CNC(c3ccsc3)=O)C3(CCC3)C2)=O)C1 c1(C(=O)OC)cc(C(C(=O)Nc2nnn(C)n2)N(CCCO)C)oc1C N1(C(CCCC(=O)OC)C(=O)NC2CCOC2)CCn2c(nc(C)c2C)C1 CCCC(CCCNC(C1COC1)=O)NC(=O)CCOc1ccc(OC)cc1 C=C(Cl)CC(C(=O)N(C1CC2CCC1O2)C)NC(=O)C(CC)n1cncn1 C12(C(=O)NC(C)(C)CF)CCN(C(c3c[nH]cc3C3CC3)=O)CCC1C2 c1(C(=O)NCC(C2CC2)NC(C2(CC(C)C)CCCC2)=O)nn(C(F)F)cc1Cl C1(N(CC#C)C(C2CCCO2)=O)CCN(C(=O)C(C)SCC2CC2)CC1 CN1CCOC(C(=O)NCCN(C(=O)Cc2ccn(C)n2)CCOCCO)C1=O C1(CNC(c2c(C)snn2)=O)CC2(CCN(C(c3cccc(CO)c3)=O)CC2)C1 C1(C(N(CCOOCC)C)=O)CC(=O)C12CCCC2.C1(C)C(=O)N(C)CC1 CC1CNCCC1CNC(C1CCN(c2ccc(C(F)(F)F)cc2)C1)=O c1(C(N2C(CNC(C(C)CF)=O)CCCC2)=O)cc2n(n1)C(C)CCC2 C(=O)(C=C1SCC(=O)N1C)NC1C2CN(C(CCC)=O)C1C2 C(=O)(C1Cc2ccc(F)cc21)NCC(C)NC(C1CCCN1CC(F)(F)F)=O c1(C(N2CCCC(CC(=O)NC(c3cnc[nH]3)C)C2)=O)cc(Cl)ccc1Cl c1(N(C(N(c2cc(C)ccn2)C(C)=O)=O)C)cccc(C)c1.c1(C)ccco1 CCCCCCCCOCC(N1CCN(C(c2sccc2COC)=O)C(C)C1)=O c1(C(=O)NC(CNC(C2CN(CC)C(=O)N2)=O)(C)C)cc(Cl)c(F)c(Cl)c1 C1(O)(C(C(=O)NC(C)CC2CCCCC2)NC(CC2C(CC)C2)=O)CCCCC1 c1(SCc2cn(CC3CN(C(C(CO)OC)=O)C3)nn2)cc(C(=O)O)ccc1Cl c1(CC(N2CC3C(CNC(C(C)(C)F)=O)C3C2)=O)cncc2ccccc12 CC1CC(C(=O)NCC(C)(F)CNC(c2cc(C3CC3)no2)=O)CC(=O)N1 c1(-c2c(C(=O)NC3CN(Cc4ccccc4)CC3F)csc2)ccc2c(c1)OCC2 C1(O)(CCNC(C2C(C)C2)=O)CCN(C(=O)CCC(C)C#N)CC1 C#CCC(C)(CNC(=O)COC1CCN(C(c2cnco2)=O)C1)CO CC1CN(C(C2(P(C)(C)=O)CC2)=O)CCCN1C(=O)COc1cccc(O)c1 c1(OC)c(C(=O)N(C(C)CCNC(c2cncc(C(N)=O)c2)=O)C)ccnc1Cl Cc1cnc2c(C(=O)N)cccn12.N1(C(C2CC23CC3)=O)CCN(C)CC1CCO c1(OC)ccc2c(c1)C(C(=O)N1CCN(C(=O)CC3(C)CC3)CC1C(C)C)CC2 CN1C(=O)CSC1=CC(=O)N1CCCOC(CNC(C2CC(F)(F)C2(C)C)=O)C1 S(=O)(=O)(c1ccc(NC(CO)C2CC2)c(Br)c1)N(CCC(C)C)Cc1ccccc1 C(C)(C1OCCc2sccc21)NC(C(=O)NC(c1c(C)nc(C(C)C)s1)C)=O CCN(OC)C(=O)CNC(=O)C(Cn1cccn1)NC(C1CC(C)(C)CO1)=O c1(CCC(N2CCC(F)(CNC(C(CCC)(C)O)=O)C2)=O)ccc2ncsc2c1 C#CCC(CC#C)C(=O)NC1(C)CC(NC(=O)CN(C)C(C)C)C1 Cc1ccc2c(c1)CN(C(C1CC1NCc1cccc3ccncc13)=O)CC2 C1(NC(c2c(CC)cno2)=O)CCC(CNC(=O)C(C)CN2CCOCC2)CC1 C1(NC(c2nc(COCC)sc2)=O)CN(C(=O)C(F)=C(C)C2CC2)CCC1C N1(C(CCC(C)O)=O)CCC2(CCCCN(C(C3(CO)CCC3)=O)C2)C1 Cc1nc2n(n1)CC(C(=O)N(CCNC(c1coc(C#N)c1)=O)C(C)C)CC2 c1(NC(C(C2CCN(C)CC2)NC(C23CC(C2)C3)=O)=O)cn2cc(Cl)ccc2n1 C1(NC(C2CCCCC23CCC3)=O)CCN(C(C2CCSCC2)=O)CCC1CO c1(-c2cn(C(C)(C)C(=O)O)nn2)ccccc1CC(=O)NC1(C2CCCO2)CC1 N1(C(CCc2ccc(C)o2)=O)CCN(C(c2csc(-c3cnc[nH]3)n2)=O)C(C)C1 C1(C(N2CC(CCC)C2)=O)CCC(C)(C)N(C(C2CC2Cl)=O)C1 CCC(C)CC(C(=O)NCC(C(C)C)C(C)C)NC(=O)CC1OCCO1 c1(C(=O)NCC=CCNC(CC2CCC(C)O2)=O)cccc(C2(C#N)CC2)c1 C1(NC(=O)CCC2CCOCC2)CN(C(c2coc(Cl)c2)=O)C2(CCCCC2)C1 C(CCCCNC(C1OCCO1)=O)N(C(C1N(CC)CC1)=O)C c1(CC(N2CCCC(C(=O)NC3CCOCC3)C2)=O)c(F)ccc(Cl)c1Br c1(C(N2CCC(C3(NC(CCC#C)=O)CCC3)CC2)=O)cc(C)ccc1[N+](=O)[O-] C1(C(=O)NCC(C(C)(C)C)NC(CC(C)(C)O)=O)CCC(=C(F)F)CC1 C(=O)(C1CCc2nccn21)NCCC1CCN(C(c2c(CC)noc2)=O)C1 c12ccc(cc1)c(=O)oc2=O.C1(CN(CCC)CC)(NC(=O)C2CC2)CCC1 C(=O)(C1=CC2CC=CCC12)N(C1CCCCCC1)CC C1(NC(C2N(C(C(CSC)C)=O)CC(=O)NC2)=O)CCC2(CCC2)CC1 C1(C(=O)NCC(C(C)C)(C)O)CC(F)CCN1C(c1cc(O)nc(O)n1)=O c1(C(N(C2CN(C(CC(CC)C)=O)C2)C)=O)[nH]nc2ncc(Br)cc12 S(=O)(=O)(c1ccc(C#N)cc1)N1CC2CN(C(c3ccc(CCC)cc3)=O)C2C1 Cc1nc2n(n1)CCN(C(=O)CC(C)CNC(c1cc([N+](=O)[O-])c[nH]1)=O)C2 n1(C(CC)C)ncc(C(=O)NCC2CCN2C(c2cccc(C3CC3)n2)=O)c1C C(=O)(CC(C)CC(C)C)N(CCC(=O)NC(c1nc(CC)[nH]n1)C)CC c1(C(=O)NCC2CN(C(C(C)SC(F)(F)F)=O)CC2(F)F)cccc2nc[nH]c12 C1(CC(N2C(C(NOCCCC=C)=O)CCC2C2CC2)=O)C=NN(C)C1=O Cc1ccc(C(=O)N2CCC(C(=O)NC(Cc3ccccc3)CO)O2)cc1C#N C1(C(=O)NCCC(=O)OC(C)(C)C)CCCCN1Cc1cncs1 N1(C(CCCN(C)C)=O)CCC2(CCCN2C(=O)CC2CC(O)C2(C)C)CC1 c1(NC(N(C)Cc2cccc(SC)c2)=O)cc(S(N)(=O)=O)ccc1Cl N1(C(=O)NC2C(C)OCC2)CCC2(CC(=O)c3ccccc3O2)C1 c1(C(N2CC(NC(C(C)(C)OC)=O)C(OC)C2)=O)ccnc(C)c1C C1(C(=O)N(C)CCOCCOC)(CC)CCN(C(=O)CN2CCC(=O)CC2)C1 c1(C(N2CCCN(c3nccs3)CC2)=O)cc2c(s1)CCC2=O N1(C(C(C)(C)O)=O)CCCC2(C1)CN(C(=O)CC1OCCCC1(C)C)C2 N1(C(C(=O)OC)=O)CCC2(CO)CN(C(c3ccccc3C3CCC3)=O)CC2C1 CCCCC(O)C(=O)N1CCC(N(C(=O)C=C(C)C)C)C(C(N)=O)C1.N1(CC=C)CCC1 c1(C(C)OC(c2cn(-c3cccc(Cl)c3)cn2)=O)ncccc1Br N1(C(c2ncn(C(C)C)n2)=O)CC(CNC(=O)Cc2cnoc2)OC2(CCC2)C1 C1(N(C(CSCCC)=O)C)CC2CC1N(C(C1CCCC(C)(C)C1)=O)C2 c1(C(C(=O)NCCN(C(=O)CCSC(F)(F)F)C)(C)C)c[nH]c2ccccc12 C1(CCNC(c2cc(C)n(C)c2)=O)CC(F)(F)CN1C(=O)C(C)C1CCC1 Cc1nn(CC(=O)NC2(C)CC(NC(=O)CS(C)(=O)=O)C2)cc1[N+](=O)[O-] c1(NCCCC(C)NC(c2ccoc2Br)=O)snc(Cl)c1C#N C1(CC(=O)NC2(CO)CN(C(C3(OCC)CCCCC3)=O)C2)CCCCC(=O)N1 C(N=c1[nH]c(=NC)[nH]c(=NCc2cccc3c2NC(=O)CO3)[nH]1)C1N(CC)CCC1 N1(C(C(C)SCC)=O)CCOC2CN(C(c3csc(C(=O)OCC)n3)=O)CC12 N1(C(Cc2ccc(C)o2)=O)CCN(C(=O)C2=C(Cl)CCOC2)C(C)CC1C c1(N2CCC(NC(C(CCCC)C)=O)C2(C)C)ncnc2c(Br)nn(C)c12 C#Cc1ccc(C(=O)NC(C)C(C)CC(=O)NC(C)(CC(C)C)C(N)=O)c(C)c1 C1(C(=O)NC2CCNC2=O)(OC)CCN(C(=O)CC2CCCCO2)CC1 C1(CC(N2CC(C)(CSC)C2)=O)CC(O)CN1C(=O)C(C)O C(=O)(C1=NOC2(CCC2)C1)N(C1CCN(C(c2cnsc2C)=O)CC1)CCC CCCC(O)CC(=O)NC(CNC(c1cc(C2CC2)nn1CC)=O)CCOC C1(C(=O)NC(C(C)NC(=O)Cc2csc(-c3cccs3)n2)C)OCCOC1(C)C c1(C(=O)NCC(CNC(C(CCC)C)=O)F)nn(CC)c(=O)c2ccccc12 c1(OC)cc(F)c(S(=O)(=O)NCC(C)(C)O)cc1Br N1(C(c2n(CC)nc(C)c2)=O)CCC2(C=C(C(=O)NCCSCCO)C2)C1 C1(CN(C)C(c2ccn(C3CC3(F)F)n2)=O)COCCN1C(c1csc(O)n1)=O Cc1cc(C(=O)NCC2CCCN2C(=O)COCc2ccnn2C)ccc1F C1(CNC(C(C)OCCOC)=O)CCN(C(=O)CC2CCC(=O)N2C)CC1 N1(C(CN(C(=O)OC(C)(C)C)CC)=O)CCC(CC2CC2)C1.c12nnnn1C2 Cc1nc(C(=O)NC2CCN(C(=O)CCC3(C)CC3)C2C(C)C)cn1C N1(C(C(CC2CC2)NC(CCC2C(C)C2)=O)=O)CCc2n[nH]cc2C1 N1(C(c2cc(C)c(-c3nn[nH]n3)cn2)=O)CC2(COC(=O)N2C)C1 c1(OC)cc(C(N2CC(C(F)(F)F)CC2CNC(=O)C(C(C)C)SC)=O)ncn1 C(C)(C)(CCCNC(c1ccc(-c2cccs2)cn1)=O)NC(CN(C)CC)=O Cc1cc(C(N2CC=CC(NC(=O)C(c3ccncc3C)C)C2)=O)c(C)cn1 c1(OC)cccnc1CC(=O)NCCN(C(=O)CC1(C(F)F)CC1)CC1CC1 c1(OC)noc(C2CC2)c1C(=O)N(CC(C)CNC(c1ccnc(S)c1)=O)C C=C1CC(C(=O)NC2CC2c2cncs2)(CNC(C2CC(CCC)C2)=O)C1 N1(C(CC2ON=C(C)C2)=O)CCC(NC(c2cc(Br)sn2)=O)C(C)(C)C1 C1(CNC(c2c(C)n(C3CC3)cc2)=O)CN(C(C2CC(O)C2)=O)C2CCN1C2 CCCCC(CNC(=O)C=Cc1cnc[nH]1)NC(c1cc(Cl)c(Br)[nH]1)=O Cc1c(C(=O)NCC2(C(=O)O)CCOCC2)oc2ccc(Br)cc12 Cc1cc(C(N2CC(NC(c3c(C)noc3C(F)(F)F)=O)C(C)C2)=O)cc(Cl)n1 c1(C(N2CC(C(=O)NC)C2)=O)n[nH]cc1CNC(C1CCC1C)=O C1(C(N2CC=C(C)CC2)=O)CCN(C(c2c(C)noc2N)=O)CC1(C)C C12(C(N3CCC(NC(c4c(C)nncc4)=O)(CF)C3)=O)CCC(O)(CC1)CC2 CC(CS(C)=O)C(=O)NCCCNC(c1cnc(O)c(Cl)c1)=O C1(OC)(OC)CC2(COC(CNC(=O)C(CO)C(C)(C)C)C2)C1 N1(C(C2C(C(C)=O)C2(C)C)=O)CCN(C(C2CCCC3CC23)=O)CC1C c1(OC)cccc(C)c1-c1ccc(CNC(C2CCN(CCF)C2=O)=O)nc1 C(=O)(C(F)(F)CCn1cc(-c2ncoc2C)nn1)N1CCC(OCCOC)C1 C1(CC(=O)NC(c2ccn(C)n2)CC)(NC(=O)CC2CCC(=O)C2)CC(F)(F)C1 N1(C(C(C)(C)SC)=O)CC2(C1)C(NC(=O)CC1CCS(=O)(=O)C1)CCS2(=O)=O N1(C2CCCN(C(C(C(C)C)NC(=O)C(F)(F)F)=O)C2)CCC2COCC2C1 C1(NC(C(C)Cc2cnn(C)c2)=O)CC(NC(c2cccnc2Cl)=O)C(O)C1 C=CC(CCC)CC(=O)NC1CC(C)(CNC(c2cnoc2CC(C)C)=O)C1 N1(C(C(C)(C)N2CCCCC2)=O)CCCC(O)(NC(=O)COc2cn[nH]c2)C1 O=C(CCN=c1[nH]ccs1)NC1(CO)CN(C(C2(C(F)F)CCCO2)=O)C1 C1(O)(CN(C(COCC=C)=O)C)CCN(C(=O)CN(C)Cc2ccccc2)C1 C1(NC(C(COCC)C)=O)CCC(NC(=O)Cc2ccc(C(F)(F)F)nc2)CC1 N1(C(C2(C3CC3)CN(C(C3C(C(=O)OCC)C3)=O)C2)=O)CCC2OCCC2C1 N1(C(CCC(N)=O)=O)CCC(C2CC(NC(=O)Cc3ccc4sccc4c3)C2)C1 N1(CCCN2C(CCCNC(=O)C=Cc3cnc[nH]3)CCC2)C(=O)CNC1=O C12(C(=O)NC(C)CCNC(=O)CCCCc3ccccc3O)CCC(F)(CC1)C2 N1(C(COCC)=O)CCC(O)C(N(C(=O)C=C2CCC(C)CC2)C)C1 C(C(=O)NC1CC2CS(=O)(=O)CC2C1)(C(C(C)C)OC)OC C1(CCC)CN(C(c2cncc(F)c2)=O)CCN1C(c1ccnc(CO)c1)=O C1(CC)C(C(=O)NCc2cc(OC)ncn2)CCCN1C(c1[nH]cc(C)c1C)=O N1(C(CCCn2cc(CCCC#N)nn2)=O)CCC(F)(C(=O)OCC(F)(F)F)CC1 CN1CC(O)CC1C(=O)NC1CC(NC(=O)Cc2ncc(Cl)s2)C1 C1(CC=C)CCCC1N=c1nc2sccc2c(NCc2nc(C(C)(C)C)cs2)[nH]1 C1(CN(C)C(C2CCC(=O)O2)=O)CCN(C(c2ccnn2CC2CCC2)=O)CC1 c1(CCC(=O)NCCOCCN(C(=O)CCSc2cccnc2)C)nccn1C Cc1ccc(C(=O)NC2CC(CNC(=O)COCC3CCOC3)C2)c(Cl)n1 C1(NC(c2c(C)nsc2)=O)COCCN(c2nccc(N3CCCCC3)n2)C1 Cc1cc(=NC(=O)C2CC(O)CCN2C(=O)Cc2ccc(O)c(O)c2)[nH]n1C c1(C(C)C)nn(C)cc1C(=O)NC1COCC1NC(C1(c2cc[nH]n2)CC1)=O c1(CC(N2C(CN(C)CCC3CCOC3)CCC2)=O)ccccc1Br N1(C(C(C)OCCC#C)=O)CCC(C2CC2)(CNC(c2cccc(F)c2)=O)C1 CCCCCC(O)C(=O)NC(C1(CNC(c2cn(C)c(=O)c(C)n2)=O)CC1)C c1(OC)ccc(C(=O)NC(C2CN(C(=O)C=Cc3cn(C)nn3)CCO2)C)nc1 N1(C(C#CC2(C)CC2)=O)CCC2C(CCN2C(=O)Cc2nc3c([nH]2)CCCC3)C1 C(=O)(C1CCC(=O)c2cccn21)NC(C1CCN(C(C2CCC(=O)N2)=O)CC1)C N1(C(CN2CCC(C)CC2)=O)CCC2CN(C(=O)C(F)F)C(C)C12 c1(C(N(C(C2CCNCC2)C(=O)OC)C)=O)ccnc2c(I)cnn12 C=CCC(CC(C)C)C(=O)N1CC2CCC(C1)N2C C(=O)(C(C)Cc1ccco1)N(C(CC)CNC(=O)CNC(=O)NC)C c1(CNC(C(=O)Nc2n(C)nc(-c3ccccc3)c2)=O)ccc(F)cc1O c1(C(=O)OC)oc(C(=O)NC2CCC2NC(C2(C)CCCO2)=O)cc1C C12(NC(C=NOC)=O)CCCC1N(C(=O)C(=C1CCCCC1)F)CC2 Cc1cccc2cc(C(N3CCC(NC(c4cn[nH]c4)=O)C(C)(C)C3)=O)cnc12 C(=O)(C(C(C)C)C(C)C)N1CCC(OCCNC(C=Cc2c(C)cccc2)=O)C1 c1(SC)ccc(OCC(N2CC3CC2C3NC(=O)CCCCN2CCCC2)=O)cc1 CC(C)CC(C(=O)N1CCCOC(CNC(C2C=CCC2)=O)C1)C(N)=O c1(C(=O)NC(CC2CN(C(C=CC)=O)C2)C)cc(F)c(CO)c(F)c1 c1(C(=O)NCCC2CC(NC(=O)C(Cl)=CCl)C2)c(Cl)ccc2ccncc12 C1(C)(C(=O)NCc2cnc(C(C)C)[nH]2)CC(O)CN1C(C1CC(=O)CCO1)=O Cc1ccc(NC(C2CCC(O)CN2C(c2cnn(C)c2Cl)=O)=O)c(F)c1F CC1CC(NC(=O)CNC(=O)C2CC2)CN(C(c2occ3c2CCC3)=O)C1 C1(C(=O)NC(C)CC(C)NC(=O)CCc2ncc(F)cn2)C2Cc3ccccc3C12 CON(CCCO)C(=O)C(CC(F)F)NC(C1CCCN1C(C)C)=O c1(C(N2C(C(=O)NCCCC=C)CC2)=O)cccc2c(O)ncnc12 N1(C(Cc2cn(CC)nc2)=O)CCCN(C(C23CC(N=[N+]=[N-])C2C3)=O)C(C)C1 c1(CN(C)C(c2cccc(C(C)(C)C(F)(F)F)c2)=O)ccc(Cl)cn1 N1(C(c2c(C)ccnc2C)=O)CCC2C(CCCN2C(c2cn(C)c(C)n2)=O)C1 N1(C(c2c(C)ccc(F)c2)=O)CCc2cc(C(=O)NCCC(N)=O)ccc2C1 N1(C(C2CC=CC2)=O)CCC(C2CCCN(C(C3CC=CC3)=O)CCC2)CC1 C1(CNC(CC(CN(C)C)O)=O)CC(C(C)(C)C)CN(C(C2(O)CCC2)=O)C1 CC1CCC(CC(=O)NC2CC(NC(c3ccccc3OCC(N)=O)=O)C2)CC1 N1(C(C23CC(C)C2C3)=O)CC2C(NC(=O)CC3C(C)(C)C3(C)C)C2C1 C1(CNC(CNC=O)=O)(NC(=O)CCc2nnc(C3CCCC3)o2)CCOC1 CC1CC(=O)NCC1C(=O)NCCCOCCCNC(=O)C(C)(F)F C(=O)(C1(C)CC(=O)N(C)c2ccccc21)NC(C(C)C)CCNC(=O)CC(F)F c1(C(=O)NC(C(CO)NC(C=CC=CCCCCC)=O)C)cccc(=O)n1C N1(C(C(C(C)(C)C)O)=O)CC(C(N2CC(O)CC2CO)=O)CC12CCC2 C1(C(=O)NC2C(NC(c3c(C)nncc3)=O)CC2)CC(C(=O)OC(C)(C)C)=NO1 C=CC1CN(C(=O)COCc2scnc2C)CC1NC(c1ccnc(C)c1)=O c1(OCCCC)ccc(C(=O)NCC2(C)CCCN(C(=O)CSCC)C2)c(Cl)c1 N=c1[nH]c(C2CC2)ncc1C(=O)NC(Cc1ccccc1Br)C(=O)O n1(CC)ccc(C(=O)NC2CN(C(=O)CC3CC4(CC4)CO3)CC2(C)C)cc1=O C1(NC(C(C)c2cccs2)=O)CCSC12CN(C(=O)CC1CC3CC3C1)C2 N1(C(C(CSC)(C)C)=O)CC2(CCCCN2C(=O)CCC=C(C)C)C1 N1(C(CC2CCN(OCCNC(C(C)(C)C)=O)C2)=O)CCc2cccc(Cl)c2C1 N1(C(CCC)=O)CCC(CCC(=O)N(C)CC2(O)CCOC2)C1 C(=O)(N=c1ncc(C#N)c[nH]1)NC(c1ccnn1C)C(=O)OC CC(C)C(C(=O)NCc1ccn(CC(F)F)n1)N(C)C Cc1nc(NC2CCN(C(=O)CSc3ccncc3)C(C)C2)c2ccsc2n1 Cn1cc(C(=O)NC2CCC(CCNC(C3(N4CCCC4)CC3)=O)C2)cn1 C1(C(=O)OC)CC(O)CCN1C(=O)C1=C(Cl)CC1.C1(C)(C2CC2)CSC(C)=N1 C1(NC(c2c(CC)nc(C)nc2)=O)CCC2CCN(C(C3CCCC3O)=O)C1C2 C=CCC(C)(C)C(=O)N1CC2(C(=O)NCCc3ccccn3)CC1CO2 c1(C(N2CCC(N(C(C=C(CC)CC)=O)C)C2)=O)ccccc1NCC(F)(F)F CC(=O)CCCCC(=O)N1CCCC1C=CC(=O)N(C)CCO C1(C(CC(C)(C)O)CC)CCCCC1.C(=O)(C=O)NCCC(=O)N(C1CCC1)C1CC1 C(C)(C)(CC(C)N=c1ccnc(NC2C(C3CC3)C2(C)C)[nH]1)OC N#Cc1c[nH]c2ncnc(N3C4CN(Cc5ccc(-c6ccc(Br)s6)s5)CC34)c12 C1(CNC(c2csc3nnsc23)=O)(NC(C2CCOC2)=O)CCC(F)(F)CC1 c1(OCC)cc(C(=O)NCCCC(C)NC(=O)CC2COCCO2)cc(F)c1 c1(C(N(CC=CC(=O)N(CC)CC2(O)CCC2)C)=O)cc(C)ccc1O c1(C(N2CCCC2C(=O)OC)C(=O)NC)cc2cc(C)ccc2s1 c1(C(=O)NC(CNC(C2(Oc3ccccc3)CC2)=O)C2CC2)cc(CF)on1 C(=O)(CCCCN=c1nc(N2CC3C(C(N)=O)C3C2)c2ccccc2[nH]1)NC CC(CNC(=O)CN(C)CC1CCC1)CN(C(=O)CCC1(C)CC1)C N1(C(c2n(C)c(=O)ccc2)=O)CCCC2(CCN(C(=O)CC3CSCCS3)C2)C1 Cc1ccc2occ(CC(=O)NC3CC3CNC(=O)Cc3sc(O)nc3O)c2c1 C#CCCC(O)C(=O)N1CCC(NC(=O)CCCN=[N+]=[N-])C1 c1(C(=O)NC(CCCNC(c2ccn(CC(C)C)n2)=O)C)csc(S(N)(=O)=O)c1 Cc1c(O)ccc(C(=O)NC2CC(C)(NC(=O)Cc3csc4nccn34)C2)c1C c1(C(=O)NC2CCCC(C(=O)NC(CC=C)CC)C2)nnc(O)nc1O N1(C(CC(C)CF)=O)CC2(CCN(C(c3ccnn3CCN(C)C)=O)CC2)C1 C(=O)(C(CCC)C(=O)OC)C(CCN(CC#C)C(C1CCC(C2CC2)C1)=O)=O C(CC(C)C(=O)N1CC2CC2(CNC(=O)CNC(C)=O)C1)OC N1(C(C=CCCC=C(C)C)=O)CCC(C2(O)CCN(C(=O)C(C)(Cl)Cl)C2)CC1 C(=O)(C(CC1CCCCC1)N1CCC(n2cccn2)C1)NC(C)C C12(C(N3CC(CNC(c4cc(O)cs4)=O)OCC3)=O)CCCCC(F)(C1)C2 C12(C(N3CC(C#N)C3)=O)CC(CN(C(=O)C=Cc3ccsc3)C1)C2 CCC(CC)(CN=c1[nH]c(C(C)C)nc(C)c1Br)NC(c1cccc(OC)n1)=O N1(c2nccc(C)n2)CCOC2(CCN(C(=O)CCC3CC3(C)C)CC2)C1 C(C)(CCS(=O)(=O)NC1CCN(Cc2ccc(F)cc2)CC1)OC CC1(NC(=O)CN2C(=O)CNC2=O)CCC(NC(C2(Cl)CC23CCC3)=O)CC1 N1(C(C)=O)CCC(NC(=O)Nc2ccc(Cc3ccccc3F)s2)C(C)C1 c1(C(=O)NC(CCNC(c2c(C)n(C)cc2)=O)C)cnc2ccccc2c1 C1(O)(CN(C(=O)CC2(O)CCCCCC2)C)CCCN(C(C2(C)CCCCC2)=O)C1 CC1CCN(C(=O)COCc2ccccc2)CCN1C(c1ncncc1Cl)=O N1(c2nccc(OC)n2)CCN(C(c2cc(C(F)(F)F)[nH]c2C)=O)CC1C C(C(=O)NC1CN(C(=O)Cn2cc(CN(C)C)nn2)CC1C(F)F)(C(C)C)SC Cc1c(C(=O)Nc2cccc(F)c2CNC2CCC(=O)NC2=O)ccc(Br)c1F C1(C(C)C(=O)N(C)CCOCCN(C(=O)CCOC2CC2)C)CCCOCC1 C#CC1(C(N2CC(CN(C(=O)C(C)(C)OC)C)C2)=O)CCCC1 Cc1cncc(C)c1C(=O)NCC1CCN(C(=O)Cc2cccnc2)CC1O c1(-c2scc(C(=O)NNC(=O)c3cn[nH]c3)n2)ccc2cncn2c1 C1(CN(C(c2scc(OC)c2)=O)C)CCCCN1C(c1cc(C2CC2)ncn1)=O c1(CC(=O)N(CCC(C)NC(=O)C2=NOCC2)C)cccc(C(F)(F)F)n1 c1(OC)cc(F)cc(C(=O)NCCNC(c2sc(F)cc2Br)=O)c1N C(=O)(CS(=O)(=O)CNC(=O)C(CCN(C)C)N(C)C)NC1C(CCC)CCC1 C1(C(N2CCC(N(C(CS(CC)(=O)=O)=O)C)C2)=O)CCCN(S(N)(=O)=O)C1 CC(C)(C)CC(=O)NNC(=O)NC1CCCCC1S(C)(=O)=O c1(C(c2n(C(C)C)nnn2)NC2CC(Cl)(Cl)C2)cc(F)ccc1Br c1(C(N2CCC(O)(NC(N)=O)C2)C)ccc(Br)cc1F Nc1cc(C(N2CC=C(CCNC(=O)CC(F)(F)F)C2)=O)ncc1F CC1CN(C)C(=O)CN1N1CCC2(CC1)CN(C(=O)OC(C)(C)C)C2 CC(C)CCC(C(=O)NC1CC12CCOCC2)NC(c1cnn(C(C)C)c1)=O c1(C(=O)NCc2ccc(OCC(F)(F)F)cc2)cccc2ccc(O)nc12 c1(OC)cc(OC)nc(N(C2CNCC(F)(F)C2)C(=O)CCSC)n1 C=CC1(CC(=O)N(CCN(C(=O)Cc2cc(Cl)n(C)n2)CC)CC)CCCCC1 c1(OC)cnn(C)c1CNC(c1nncs1)C C1(CN(C(=O)C=Cc2ccn(C)c2)C)CN(C(=O)C(O)CC(N)=O)CC12CC2 c1(OC)cc(C(=O)NCC2CCC2NC(=O)Cc2c[nH]nc2O)sc1S(N)(=O)=O c1(CN2CC(c3ocnc3CNC(c3n(C)ncc3)=O)C2)cc2ccncc2[nH]1 c1(OC)ccccc1CC(=O)NCC(O)CNC(c1oncc1C)=O c1(C(=O)NC(CCCCNC(COCCCOC)=O)C)ccnc(Cl)c1Cl C1(C(=O)NC(C(C)(C)C)CNC(C2(C#N)CC3(CC3)C2)=O)CCc2cnnn2C1 N1(C(CN(C(CC(CC)C)=O)CC)=O)CCOC(C)CC1 N1(C(C2CN(CCC)C(=O)C2)=O)CCCC(C)(CNC(c2nnc(C)s2)=O)C1 N1(C(C(c2cccnc2)C)=O)CCC(NC(C2CCCCS2)=O)C(O)C1 Cc1cc(CCC(=O)NC(C)CCCNC(C2(C)CCCC2C)=O)nn1C C(=O)(CCC(F)(F)F)N(CCCNC(C1(OC)CC(C(F)F)C1)=O)CCO C1(COC)(CNC(C2CCC(C)(C)C2)=O)CCN(c2cc(O)nc(C)n2)CC1 C1(CC=C)(C(=O)NCCc2[nH]cnc2C)CCCN1C(=O)CC1CC(CC)=NO1 c1(NCC(=O)NCC(CNC(=O)C=CCO)O)ccccc1Br C1(C(=O)NCC2(OCC)CCCC2)C=CCN(C(C23C=CC(CC2)C3)=O)C1 C(F)(C(=O)NCCC(C)NC(=O)CCSCC(C)C)=CC CS(=O)C1(CNC(=O)COC2CCN(C(c3cscc3Cl)=O)C2)CC1 c1(C(N(C(C)CNC(C2(C)CC(C)(C)C2)=O)C)=O)ncn2c1CCC2 CON1CCC(C(=O)NCCC2CCCN(C(=O)Cn3cccc3)CC2)CC1 n1(CC(=O)NC2CN(C(CSCCC(C)C)=O)CC2O)ncn2cccc2c1=O N1(C(C(C)C)C(=O)NC(C)(C)CNC(=O)C(O)C(C)C)Cc2ccccc2C1=O CCC(CC)C(C)C(=O)N1CC(CNC(=O)C(c2cccc(C)c2)O)C1 C(CCCCC(=O)N1CCCC1C)N(C(c1cc(CC)[nH]n1)=O)C CC1CN(C(c2cc(Cl)c(Br)cn2)C(=O)NCCC2CC2)Cc2c[nH]nc21 C(c1cncnc1O)=CC(=O)NC1(C2N(C(c3c(C)scn3)=O)CCC2)CC1 Cc1ncc(C=CC(=O)NC(C2CCCN(C(=O)C(O)CC3CCCC3)C2)C)s1 N1(C(C2CC(C)(C)C2)=O)CCC2CN(C(C3(C)CCCC(F)(F)C3)=O)CC2CC1 C1(C)(NC(C=C(C)CN2CCOCC2)=O)CCN(C(C23CC(C2)C(C)O3)=O)C1 C(=O)(C(C(C)Sc1ccc(C2(C(F)(F)F)N=N2)cc1)C(C)C)OCC c1(C(=O)OC)cc(CNC(=O)NC2CCC(N(C)C)C2)ccc1C C1(CCNC(C(C)N(C(CNC(=O)NC)=O)C2CC2)=O)COCCO1 C(=O)(C1=CNC2=NCCCC2=C1)NCC1C(C)CN(C(=O)CSc2cn[nH]c2)C1 C1(CC)CN(C(=NCCF)NCCc2ccc(OC)nc2)CC(C)S1(=O)=O Cc1c(C(=O)NCC2CC(F)(CNC(c3cocn3)=O)C2)cc(C(C)C)n1C c1(CCC(=O)NC2CC(O)(CNC(C(C)=C3CCCC3)=O)C2)ccc(F)c(F)c1 c1(C(=O)NC2(CNC(C3CCC(OC)CC3)=O)CCOC2)ccc(F)c(Cl)c1N C1(c2ccccc2)(CNCCCCCOCC)CC2(CC2)C1 c1(C(=O)NC2CN(C(c3cc(C4C(C)C4)on3)=O)C2)c(F)ccc(Cl)c1N N1(C(CSCCCC)=O)CCC(NC(=O)CCn2ccnc2C(C)C)C1C(C)C C(=O)(N1OC2CCC1CC2)C1(F)CCN(C(c2ccnc(O)c2)=O)C1 c1(C(=O)NC2CN(C(c3[nH]n(C)c(=O)n3)=O)CC2(C)C)cc(F)c(F)cc1Cl C(=O)(C#CC1(C)COC1)NC1CCC(C)N(C(=O)C(O)Cc2cnc[nH]2)C1 N1(C(C=CCCC)=O)Cc2ccccc2C(NC(=O)Cn2nnc(=O)[nH]2)C1 CC(CC(=O)NCc1ccc(CNC(=O)Cc2cc[nH]c(=N)c2)cc1)C(F)F c1(CC)cc(C(=O)NC(C2CCOC2)CNC(c2cnns2)=O)ns1 C1(C(=O)NC2(C)CN(C(c3cc[nH]c3C3CCC3)=O)C2)CCCC(F)(F)C1 C1(NC(c2ccccc2)=O)CN(C(c2cnsn2)=O)C2CCCCC12 C(=O)(C1CCc2nccn21)N1CC2CN(C(c3cc(OC)c(F)cc3)=O)CC2C1 c1(C(N2C(c3cccc(C)c3)C(C)C2)C(=O)NC(C)(C)C)ccc(F)c(F)c1Br N1(C(c2ccc(CCC)cc2)=O)CC2(CC(NC(=O)Cc3nnc(O)s3)C2)C1 C1(C(N2CCC(CC=C)C2)=O)CN(C(C2OCCC2C)=O)CC1(C)C CC1CCC(CC(N2CC(CN(C)C(C34CCCN(CC3)C4)=O)C2)=O)CC1C N1(C(C2(CCOC)CCC2)=O)CC2CC(C1)N(C(c1cnc(SC)s1)=O)C2 Cc1cccc(C(CNC(C2NC(=O)C3CC23)=O)NC(=O)C=CC2CC2)c1 C1(C(=O)NC2CCCC2C(=O)NCc2cccc(C)c2Cl)(OC)CCC(C)(C)C1 C(N=c1nc(NC2CCN(C)C2)c2c([nH]1)c(C)nn2C)c1cnn(CCC)c1C N1(C(C2(C(C)C)CC2)=O)CC(NC(c2cnoc2-c2ccc(F)cc2)=O)C(C)C1 c1(CC)cc2c(cc1OCCCC1CCCO1)OC(C)C2.c1(=O)c(=O)[nH]1 c1(C(N2CCC(NC(C3CCCN(CC)C3)=O)C2C)=O)cc(C)c(C#N)cn1 CCCC(C(=O)NC(C)CN(C)C(C1(NC(C)=O)CCC1)=O)NC(N)=O c1(OC(C)C)ccc(S(=O)(=O)N2CCC(N(CC(C)C(=O)N(C)C)C)CC2)cn1 C1(NC(N(C)C)=O)CCN(C(=O)C(=O)NCC2CC23CC3(F)F)CC1 N1(C(C=CCCC)=O)CCC(C2CCN(C(c3ccnc4[nH]nnc34)=O)C2)C1 c1(C(=O)NCC2N(C(CC(=C)C)=O)CC=C2)cc(-c2ccccc2)oc1C CC1CCCCC1N(C)C(=O)NC1(c2csc(Br)n2)CC1 Cc1cccc(CNC(C2CCN(CC3(C4CCCCO4)CCC3)CC2)=O)c1 c1(C(=O)NC(C2CCN(C(CC3C(C)(C)C3)=O)C2)(C)C)cccc(Cl)c1N Cc1ccc(C(=O)N(C2CN(C(c3cnnc(O)c3)=O)CC2(C)C)C)cc1Cl C1(C(=O)NCc2c(OC)cccc2)CCCCN(C(=O)CCc2nc(O)n[nH]2)C1 C(C(C)C(F)C(=O)NCCSC(C)C)NC(C(C(C)C)SCC)=O Cn1cc(C2CCN(C(C(=O)NC(=O)CSC3CCCO3)c3cnsc3)C2)cn1 N1(C(CCSCCCC)=O)CCOC(C(C)NC(C2CCC2C)=O)C1 CC1(C)C(C(N2CCC(O)C2)=O)CCN1C(=O)C(=O)C1CC1 C1(CNC(c2cccc(SCC)c2)=O)CCN(C(=O)C2=COCC2)CC1(F)F C=CCCC(C)NC(C1(C(C)NC(=O)Cc2sccc2C)CC1)=O C(CC(C(C)C)NC(c1cc(N2CCCCC2)ccn1)=O)N(C(COC)=O)C N1(C(c2cn(CC)nc2)=O)CC(C)N(C(C23CCC(CC2F)C3)=O)C(C)C1 CCCCC(CNC(=O)Cc1coc(-c2cccs2)n1)NC(=O)CNC(=O)NC N1(C(CC(C(C)C)NC(C(C(=O)OC)(C)F)=O)=O)CCC(C)(C2CC2)C1 N1(C(c2c(SC)ccs2)=O)CCC2C(CCCN2C(=O)CCc2cnccn2)C1 N1(C(c2c(C)nsc2N)=O)CCOCC(NC(=O)C(C)OCCC(C)C)C1 CC(C)CC(CNC(c1cccc(I)c1)=O)NC(c1ccon1)=O Cc1cc2ccc(C(=O)NCC(C)(C)CCNC(=O)CCNC(N)=O)cn2c1 C1(F)(CNC(c2c(COC)ccs2)=O)COCCN(C(=O)CNC(=O)C2CC2)C1 CC1CN2CC1(C)C2=O.C1(NC(=O)CNC(=O)C(F)(F)F)CCC2CC2CC1 C1(O)(C(C)NC(c2cnc(O)s2)=O)CCN(C(C2CCOCC2)=O)CC1 c1(CC(=O)NC(CNC(c2ccc(N(C)C)cn2)=O)CO)cccc2c1OCO2 c1(C(=O)NC(C)C(CO)NC(c2ccc(CF)cc2)=O)cccc(=O)n1C N1(C(c2cc(CC)oc2C)=O)C2CCCC1CC(NC(C1CC(=O)CCO1)=O)C2 c1(OC)csc(S(N)(=O)=O)c1.CN1CCC(C)(C2c3nnnn3CCN2)CC1 C(=O)(NN1CC(C(=O)OCC)CC1=O)NCCCC(c1ccccc1)N(CC)CC N1(C(CC(C)C)=O)C(CNC(=O)CC2SC(=N)NC2=O)CC2CCCCC12 Cc1nc2c(N3CCCC(NC(c4cc(I)c(O)c(I)c4)=O)C3)ncnc2[nH]1 C1(CNC(C(C(C)C)NS(C)(=O)=O)=O)C2CCC1CN(C(c1ccon1)=O)C2 CC(C)CCCC(=O)NC(CNC(C1(C)CCC2CC2C1)=O)Cc1ccccc1 N1(C(CC=C(C)C)=O)CCC(N(C(=O)CC(c2ccc(F)cc2)C)CCO)CC1 c1(CC(C)C)cc(C(=O)NCC2(NC(=O)C(C(C)C)NS(C)(=O)=O)CC2)n(C)n1 C1(C(=O)NC(C)(CNC(c2ccsc2C(F)(F)F)=O)C2CC2)CC2OC1C1CC21 Cc1nnc2n1CCC(C(=O)NC1CCC(NC(=O)CC3COC4CC3C4)C1)C2 c1(COC)cc(C(=O)NCCO)ccn1.C12(COC(C)(C)C)CCN1C(=O)N2 c1(SCCC)cccc(C(=O)NCCC(O)CNC(C2(O)CCSC2)=O)c1 c1(C(=O)NC2(CC(=O)NC(C(C)C)CO)CCC2)cc2c(s1)CSC2 c1(C(=O)NCC(CNC(C2CC(F)(F)C2)=O)OC)c[nH]c2cc(F)ccc12 c1(OC)ccc(NC(=O)Cc2sc(C3CCC3)nc2C)cc1[N+](=O)[O-] C1(CNC(N(CC(C)(C)O)Cc2ccsc2)=O)CN2CCN1CC2 C1(C(=O)NCCOCCC#C)COCCN(C(=O)CCCCCC)C1 N1(CC2N(C(c3cc([N+](=O)[O-])sn3)=O)CCC2)C(=O)C2CCCCC2C1=O C1(C(=O)Nc2cccc(CSC)c2)CCC12CCN(C(=O)COCC(C)C)CC2 N1(C(=O)Cc2ccc(C(F)(F)F)cc2)CC2CC1CN2C(c1cc[nH]n1)=O C(CC(C(=O)N1CCCC(CF)C1)NC(C1C(C#N)C1(C)C)=O)OCC C(C(C)C(F)C(=O)NCCc1nc(C)no1)NC(C(CO)OC)=O C#CC1CC(NC(=O)C(C)=CCNC(=O)Cc2ccc(C)s2)C1 c1(NC=O)cccc(NC(=O)C(=O)NCc2cnn(C(F)(F)F)c2)c1.C1CCOC1 C1(C)(CC)CC(NC2CC(C)(CC(=O)OC)C2)CCO1 c1(OCCCC(N2CC(NC(C(CC=C)C)=O)C(C)C2)=O)ccc(Cl)c(C)c1 C1(OCCC)CCN(c2nnc(-c3ccoc3C)n2CC(C)C)CC1 N1(C(CCN(C)CC)=O)CC(NC(c2sc(F)cc2C)=O)CCC1C C(C)(CO)(C(=O)NCC1CCCN(C(C2CC(Cl)(Cl)C2)=O)C1)NC(C)=O CC(C)CC(C)CC(=O)NCC1CCCN(C(=O)C2=CCOCC2)CC1 CC(C)CCC(O)C(=O)NC(Cc1ccc(Cl)cc1Cl)C(=O)NCC(C)N=[N+]=[N-] C1(NC(C2C(C)(Br)C2)=O)CCC(NC(c2cnc(O)o2)=O)CC1 C1(CC(N)=O)(NC(CC(COC)C)=O)CCN(C(C2CC(OC)C2)=O)CC1 Cc1cc(CNC(=O)C(C)CN(C)C)oc1C(N1CCCCC1CC(C)C)=O c1(CC)nc2c(C(=O)N(CCC(C(C)C)NC(=O)C(C)(C)CF)C)ccnc2[nH]1 n1(CC(N2CCN(C(c3ncc(Br)cc3F)=O)C3CC23)=O)ccc2ccccc12 C(=O)(C1=NNC(=O)CC1)NC1(C)CC(NC(c2cn(CC)nc2C(C)(C)C)=O)C1 c1(OC)ccc(CC(N2CCNC(C(=O)NCCn3cccc3)C2)=O)cc1O c1(C(N(C2CCCN(C(=O)NC3CC3)C2)C)=O)ccc(CNC(N)=O)cc1 c1(CC)cc(C(=O)NCC(=O)NCC(=O)Nc2c(C)noc2C)n(C)n1 c1(C(N2CCC(CCC(=O)NC(C(=O)OC)CO)CC2)=O)cc(C)cc(O)n1 N1(C(Cn2cc(C(C)=O)nn2)=O)CCCC(CNC(c2nnc(S)n2C)=O)C1 n1(CC(=O)Nc2cc(CC)cc(Br)c2)ccc2ccc(-c3ccoc3)cc12 c1(OC)nscc1C(=O)NCCN(C(C1C(OC)C1C)=O)Cc1ccccc1 Cn1ccnc1C(=O)NCCCN(C(=O)CC1CCOC1)Cc1ccccc1 N1(C(C(C2CCCO2)OC)=O)CC(C)(NC(=O)Cc2cc(C)[nH]n2)C1 C12CCCN(C1)CCC(O)N2C(=O)CN(S(=O)(=O)Cc1ccccc1)C.CO.SC CCCC(C)CC(=O)N1CC(F)CC1CNC(=O)CC1CC1(Cl)Cl C(C(C(F)(F)F)OCC)N(C(C(=C)C)C)Cc1ccccc1 N1(C(C)C(=O)NCc2ccc(C3CCC3)cc2)C(=O)c2ccccc2C1=O c1(CC)nc(=N)[nH]cc1C(=O)NC(C1CCN(C(=O)CCC2CCC(=O)N2)C1)C N1(C(C(C)(C)CC2CC2)=O)CC2CN(C(C3CC4CCC(C3)O4)=O)CC2C1 C=CCCC(F)(F)C(=O)NCC1(CCNC(C2CN3CCCN2CC3)=O)CC1 C(=O)(C(C)(C)C(O)C(C)C)NC(COC)CC(=O)Nc1ccc(C)nc1 C1(C(N2C(CNC(COCc3ncc(C)o3)=O)CCC2)=O)COCCC1(F)F c1(C(N2C(C(=O)NCCCC=C)CSCC2)=O)cccn2cncc12 N1(C(CC(=O)OCC)=O)CCCC2(CCCCN2C(=O)Cc2ccc(C)o2)C1 CCC(C)(C)C(C)NC(=O)CC=CCNC(=O)C(C(C)OC)N(C)C C(CCCOC)(C(=O)OCC(C)=CC)ONC(C1CC=CCC1)=O C1(CC(=O)NCCc2c(C(N3CC(CCOC)C3)=O)c[nH]n2)CCCC12CC2 c1(C(=O)NCC(C)(C2CC2)NC(C2C(F)(F)C23CC3)=O)ccc([N+](=O)[O-])cc1N c1(CC(=O)NCC(CO)NC(c2cnc(C(C)(C)C)[nH]2)=O)ccc2nc[nH]c2c1 C1(CNC(C(C)CO)=O)CCN(C(=O)C(=Cc2cccnc2)F)C12CCC2 N1(C(C2OCCCO2)=O)CCN(C(C2(n3cccn3)CCOCC2)=O)CC1 c1(CC(=O)NC(CC)CN(C)C(C2(c3cccs3)CC2)=O)c[nH]nc1O c1(CNC(c2ccc(SC)o2)=O)ccc(CNC(C2(C(F)F)CC2)=O)cc1F C1(C(=O)NCCC(CC)(F)F)N(C(C2OCCCC2(C)C)=O)CC12CCCC2 N1(C(C2CC(C)OCC2)=O)CCCCC12CC(NC(=O)C=CC(=O)N(C)C)C2 CC(C)C(C)(O)C(=O)NC1CCN(CC(C)OCc2ccccc2)C1 Cc1cc(C(=O)NCCN(C(=O)C(c2cncc(F)c2)C)CC2CC2)ccc1CO N1(C(Cn2cc(CC)nn2)=O)Cc2ccccc2C(NC(=O)Cn2cnnc2)C1 c1(NC)nc(C)nc(N(C)C)c1C.C12CCC(C)(CC1)N2 CC(C)CCCCC(=O)NCC(O)CCNC(c1c(C2CCC2)cnn1C)=O C#CC(C)(C)C(=O)N(CCC(C)NC(c1nc(Cl)c(Cl)s1)=O)C Cn1cc(C(N2CCC(C)(NC(=O)CC3CCNC3=O)C2)=O)c(-c2cccs2)n1 C(=O)(C1c2c[nH]nc2CN1C(=O)C(C)c1ccco1)N(CCC(=O)OC)C c1(C(=O)NC(CN(C(=O)C(N)=O)CC)C)csc(C(C)(C)C)n1 Cc1ccc(C(N2CCN(C(=O)CN(C)C(N)=O)C3CC23)=O)c(N)c1F c1(C(N2CCC(n3cc(C4CCCOC4)nn3)CC2)=O)ncc(Br)cc1C(F)F N1(C(CCC(C)OC)=O)CCC2(CCCN2C(c2cc(C)c(Cl)cc2F)=O)C1 c1(C(=O)NC(C(C(=O)OC)O)C)nc2ncccc2cc1C N1(C(C2C(NC(C3C4CCC(F)C34)=O)CCCC2)=O)CCc2cncnc2C1 N1(C(c2c(C)nc(O)s2)=O)CCCC2(NC(=O)CSCC(F)F)CCCC12 C12(CNC(C(C)NC=O)=O)CC(CO1)N(C(=O)CNC(=O)C1CC1)C2 N1(C(CC(C(C)C)O)=O)CC2(C=C(C(=O)NCC3OC(=O)CC3(C)C)CO2)C1 c1(-c2cccc(C)c2)nc(SC(F)F)n(C2CCc3ccccc32)n1.C12CC(C1)C2 c1(CCC(=O)NC(CC)CNC(=O)C=Cc2cscn2)ccc(Cl)nc1 N1(C(C(C)OCC)=O)CCC(CNC(=O)CCN2CCC2)(COC)C1 N1(C(C2(C)CCOC2)=O)CC2CC1CN2C(c1sc(Br)cc1F)=O C(=O)(C(=O)C(C)(C)CC)N1CCN(C2CN(C(CC=CC)=O)C2)CC1 C1(CNC(=O)CO)CCCCN1C(c1cc(-c2ccco2)on1)=O C(=O)(C(F)(F)C(F)F)NC(C1CCN(C(c2c(C)nncc2)=O)CC1)C N1(C(CC(=C)C)=O)CC(O)CC1CNC(C1(Cc2cnn[nH]2)CCCC1)=O c1(C(=O)NCc2n(C)cnc2)cnc2n[nH]c(-c3cc(CO)cc(F)c3)c2c1 N1(C(C2(C(CC)=O)CC2)=O)CCC2CCN(C(C3C=CC3C(=O)OC)=O)C2C1 CC1CCCN(N(C)CCc2ccccn2)C1 C1(C2(O)CCC2)(CN2CC2=O)CC1.C(c1cc[nH]c1)=CC(=O)N(C1CC(C#N)C1)C c1(C(=O)NC2CCCN(C(CC(C)SC)=O)C2)c(OCC2CC2)cccc1Cl c1(NC(N2CCC(CN(C(C)=O)C)CC2)=O)ccc(S(=O)(=O)C2CC2)cc1 C(c1ccncn1)=CC(=O)NCCCN(C(C)C)C(C1CCCN(C(N)=O)C1)=O C(CC(C)(C)CC(=O)N1CCC2(CC(NC(C3CC4CCC3C4)=O)C2)C1)OC N1(CCN(CC(=O)OC)Cc2sncc2Br)CCOCC1 N1(C(C2C(C(=O)OC)CC2)=O)CCCCC(NC(c2cnc3n2CCC3)=O)C1 c1(C2N(C(C3N(C(=O)Cc4ccsc4)CCC3)=O)CCC2)ccc(Cl)cc1 C(CCC(C)C(=O)N(C1CCCNCC1)Cc1ccccc1)OCC c1(C(=O)NC2CN(C(=O)C3=CCCC3)CC23CC3)cc(=O)c2ccc(Cl)cc2o1 c1(CN2CCC(C)C(NC(c3cccc(Cl)c3)=O)C2)nnc(S(C)(=O)=O)s1 N1(C(C(CC)(O)c2ccccc2)=O)CCC(NC(=O)CC2C=CCC2)C(F)C1 C1(C)(OCC(=O)NC(C(=O)N(CC(C)C#N)C)C2(O)CCC2)CCCC1 N1(C(c2c(C)ncc(N)c2)=O)C2CCC1CC(CNC(c1c(C)noc1C)=O)C2 N1(C(COC(C)C)=O)CC2CCC(C1)N(C(=O)C=Cc1cncc(F)c1)C2 N#CC1(C(=O)NCCOCCNC(c2cnsc2)=O)CCOC1 Cc1cccc(C(CNC(C2CCN(C)CC2)=O)NC(=O)CCCF)c1 N1(C(C2(C)N(C)CC(O)C2)=O)CCC(C)(C)C(CNC(C2CCCCO2)=O)C1 C(=O)(CC(=O)N(C(C)(C(=O)NCCCC1CCOC1)C1CC1)C)N(C)C C1(NC(C2(CC)CCN(C(=O)CCCN(C)C(C)C)C2)=O)CCN(C)CC1(C)C C(c1cncnc1O)=CC(=O)NCC1(O)CN(C(C2CC2F)=O)C1 c1(CN(C(C)C(=O)Nc2c(CC)cccc2C)CC)ccc(S(C)(=O)=O)cc1 CCC(C)C(C)C(=O)NC1CC(OCC(=O)NCC23CCCC(CO2)C3)C1 C12(C(=O)NCCN(C(=O)CCc3cncc(F)c3)C)CC(C#N)(C1)C2 c1(C(=O)NC(CNC(CCSCC)=O)C(C)C(C)C)cc(S(N)(=O)=O)n(C)c1 c1(NC(C(C(C)C)NC(C2(SC)CC2)=O)=O)cc(C)cc(C)c1 c1(NC(c2nccn2-c2cccc(F)c2)=O)ccnc2cc(Br)ccc12 C1(C(N2CC(OCC(=O)NC3C(CC)C3)C2)=O)CC12CCCCC2 C1(C(N2CCCC(C(=O)OC)C2)=O)CN(C(=O)C(=O)N(C)C)CCC1O c1(C(C(=O)NC(CC)CN(C)C(c2cn(C)c(O)n2)=O)C)ccc(F)c(F)c1 CN1CC2CC1CN2C(C1CCC(NC(=O)C2=CCCC2C)CC1)=O C(=O)(C(F)(F)C(C)O)NCc1c(CCNC(c2nc(C(C)C)sc2)=O)ocn1 N1(C(C2OCC(C)(C)OC2)=O)CCC2C(CCCN2C(c2cnc[nH]2)=O)C1 c1(C(N(CCNC(C2(C)CNC(=O)C2)=O)CC)=O)ccc(F)c(S(C)(=O)=O)c1 Cc1ccc(Br)c(C(N2CCCC(NC(=O)COc3cccnc3)C2)=O)c1F N1(C(c2ccc(C)nc2)=O)CCN(C(=O)C(C)(C)C2(O)CCC2)CC(C)C1 CC1(C)OCCCC1CNC(=O)CC(O)CNC(C1CCC(=O)O1)=O Cc1ccc(C(=O)NC(C)CNC(=O)CC2CCC(=O)NC2)cc1C#N C1(C(N2CCC(CNC(CC(C)c3ccccc3)=O)C2)=O)COCCN1C(C)=O Cc1cc(Cl)ccc1C(=O)NC1CC12CC(NC(c1oc(C(C)C)nc1C)=O)C2 c1(CC)cc(C(N2CC(CNC(c3ccc(Cl)nc3N)=O)C(C)C2)=O)ccc1F N1(C(CC=C(C)C)=O)CCC(=CCNC(C23CC(C2)C(C)O3)=O)CC1 N1(C(Cc2c(C)n(C)nc2)=O)CCC(NC(C2(C3CCCO3)CC2)=O)C(F)C1 Cn1nnc2cc(C(=O)NC3COCCC3NC(=O)CCc3ccccc3)ccc12 c1(OCC)cc(CNC(C2CCCN(CCC(=O)O)C2)=O)ccc1F C1(C(N2CCC(N(C(c3coc(C(F)(F)F)c3)=O)CC)C2)=O)CCC(=O)N(C)C1 CC(=O)CC(C)(C)C(=O)NC(C)CC(C)NC(c1c(C)coc1C(C)C)=O N1(C(c2cnn(C)c2F)=O)CCC2C1CCCN2C(c1cc(C(C)(C)C)on1)=O C1(CNC(CC2CC(CC)C2)=O)CCCC2(CCN(C(=O)CC(C)C)CC2)O1 C1(CC(=O)NCC(C(=O)NC)C)N(C(=O)CCc2cc(C)[nH]n2)CCC1(C)C Cc1c(CC(=O)NC(C)(C)C(C)NC(=O)C=C2CCCCC2)cccc1[N+](=O)[O-] c1(CNC(N(C2CC(OC)C23CCC3)C)=O)cn(C)c(=O)nc1O C1(C(N2CC(OCC)(CNC(c3ccc(CO)cc3)=O)C2)=O)CCC12CCCO2 CC1CCC(C(=O)N(CCCCCNC(c2scnc2C(F)(F)F)=O)C)C1 CC(C)CC(C(=O)NC(C(=O)NCC1CC2(CCC2)C1)C1(O)CCC1)C(N)=O C(=O)(CCN(OC)C(=O)C=C(CC)CC)NC(CCCCC)C1CC1 Cc1cc(C(=O)NC2CC2CNC(=O)Cc2cnn(C)c2C)c(F)cc1N N1(C(C(F)=C(C)C)=O)CC2CCN(C(C3CC4(C3)CC(C)C4)=O)C2C1 c1(C(C(=O)NCC(CC=C)NC(C23COCC(C2)C3)=O)C)ccc(Cl)cc1 c1(CCNC(N(CCC(=O)OC)Cc2nnc(C)s2)=O)cn2c(C)cccc2n1 C1(CSC)CCCC2CN(C(=O)OC(C)(C)C)CC12.C12CC3CCC1C3NC2=O C(C)(C(C)C(=O)Nn1cnn(C)c1=S)NC(CSCC#C)=O c1(CN(C(C(CC)C)C)C)cc(F)c(N2CCOCC2)c(F)c1 CN1C(=O)c2ccccc2C1C(=O)N(C1CCCC1)CC1(O)CCN(C(=O)CN)C1 N1(C(C2C3(CCN(C(Cc4n(C)ncc4)=O)CC3)C2)=O)CCc2c(cnn2C)C1 Cn1cc2ccc(C(=O)NC34CCN(C(C5(C)CC(F)(F)C5)=O)CC3C4)cc2n1 C1(CC)CCCCC1OCC(N1CC(NC(=O)CSC(C)C)CC1C)=O CCCC(C#N)C(=O)NC1CCCC1NC(c1ccnc(S)c1)=O C(=O)(C(C(C)(C)C)NC(N)=O)N(C)CC1CCN(C(CC)C(=O)OC)C1 Cc1cc(C(=O)NCC2(C(=O)N(CC(C)C#N)C)CCCO2)nc(O)n1 c1(C(=O)NC2C(NC(C(CC)C)=O)CCC2)ccc2nnc(S)n2c1 c1(OC2(CC(=O)NC(C3CCCCC3)CNC(C3C(C)C3)=O)CC2)ccccc1 CCCC(C(=O)NCC(C)NC(C1CCSCC1)=O)S(N)(=O)=O c1(C(=O)OCC)cc(C)nnc1NCC1CCCN1C(c1cc(C)cs1)=O c1(C(N(C2CCN(C(C=C(C)C3CC3)=O)C2)C)=O)cc2ccc(Br)nc2[nH]1 C1(CC)CN(C(=O)C(=Cc2cccs2)C)CCC1NC(C1CC2(CCC2)C1)=O C1(NC(COCCC)=O)CN(C(c2sc(C)cc2Br)=O)C2(CCOC2)C1 C1(CNC(c2cc(Cl)n[nH]2)=O)(CO)CCCN(C(=O)COCC2CCCO2)C1 c1(C(CC)C)ccc(C(=O)NC2CCN(C(C3CC(SC)C3)=O)C2)cc1 CCCCCC(C)C(=O)N1CCCC(C(=O)Nc2cc(C(F)(F)F)ncc2F)CC1 C1(NC(c2ccc(C#C)o2)=O)CC2CCC1N2C(C1CCCO1)=O c1(C(=O)NC(C)CCN(C(=O)CC=CC(C)(C)C)C)ccccc1C1(C)CC1 C1(C(N2CCC(C(C)NC(=O)Cc3cnccn3)C2)=O)CCCC(F)C1 C(=O)(C(C(C)CC1CC1)N(C)Cc1ccc(N(C)C)cc1)C1CC(C(=O)OC)C1 c1(C(=O)NC(C)CN(C(=O)C(CO)NC(=O)C(C)C)C)cc(C(F)F)cc(F)c1 c1(C(=O)NCC2N(C(c3c(F)cccc3Cl)C)CC2)n[nH]c2c1CCCC2 c1(N2CCC(=CC(=O)Nc3cc(Cl)c(Cl)cc3Br)CC2)ncnc2n[nH]cc12 c1(N(C(c2ccc(Oc3cccc(OC)c3)cn2)=O)C)nc2ccc(Cl)cc2s1 C(C(CCN=c1nc(N2CCOCC2)[nH]c(=NC(C)C)[nH]1)OC)OC C(=O)(C(CC(=C)C)NC(=O)CCC=C(C)C)N1C(C=C)CC1 CCC(C#N)C(=O)NCCC1CN(C(c2csc(C3CC3)n2)=O)CCO1 c1(CNC(C(C2N(C(=O)OC(C)(C)C)CCC2)(C)C)=O)ccc2c(Cl)n[nH]c2c1 N1(C(C(C)NC(C)=O)=O)CC2CN(C(C3CCC=CO3)=O)CC2C1 O(P(=O)(CCC1CCN1C(=O)C(=O)NC(N)=O)OCc1ccc(F)c(C)c1)CC CC12CN(C(c3ccsn3)=O)CC1CN(C(c1ccccc1Br)=O)C2 C1(NC(=O)Nc2nncs2)CCN(CC(O)COc2ccccc2F)CC1 N1(C(C(CCCOC)NC(C2CC(O)C2)=O)=O)CC2(CCC1CO)CC2 c1(C(=O)NCC(CNC(c2c(C)cc(Cl)cc2N)=O)C)cc([N+](=O)[O-])ccc1Cl C(CNC(CC(=O)NOC1(CO)CCSC1)=O)(CCOC)NC(CCC)=O C(CCOC)(C(=O)NC1(C(O)CO)CC1)NC(C(CC)=CC)=O C#Cc1ccc(C(=O)NC(CCCOC)C(=O)NCC(=C)C(F)(F)F)nc1 Cc1c(NC2(c3nnnn3C(C)C)CC3(C(N)=O)CC23)cccc1C#N C(=O)(C(O)CC(F)(F)F)N1CCCC(CC)C1C(=O)NC(c1ncc[nH]1)C C1(CC(=O)NCC(C(C)C)NC(C2(c3cccnc3)CC2)=O)CCC(C)C(C)C1 C1(Cl)(C(=O)NCC(c2ccccc2)N(C(COCCC)=O)C)CC1(C)C Cc1c(C(=O)NC(C)C(C(C)C)NC(=O)Cc2ccsn2)ccn1CCO CCCCC(F)C(=O)N(C(C)CN(C(=O)CC1CCCNC1=O)C)C c1(C(N2CCCC(n3cc(CCO)nn3)C2)=O)ccc2nncn2c1 N1(C(C(F)=CC)=O)CCC2C(CCCN2C(c2n[nH]cc2Br)=O)C1 c1(C(N2CCCC(C(C)(C)C(=O)OC)C2)C(=O)NC)cccc2cc(OC)ccc12 N1(Cc2c(OC(C3N(Cc4scc(C)c4)CC3)=O)cccc2)CC(C)OC(C)C1 Cc1cc(=NCCCCN(C)C2CC2)[nH]c(N2CCC(C)S(=O)CC2)n1 N1(C(c2c(CNC(c3cc(O)cs3)=O)nccc2)=O)CC2(CCC(O)CC2)C1 C1(NC(CCCC(CC)C)=O)CCN(C(c2cnc(S)[nH]2)=O)CC(C)(C)C1 C1(NC(C(C(C)C)NS(C)(=O)=O)=O)CCC2(CC1)CN(C(c1cnnn1C)=O)C2 CC(C)CCCC(=O)N1CC2(Cn3cc(-c4nn(C)cc4Cl)nn3)CC1C2 N1(C(C2CCN(C(C3(CN(C)C)CC3)=O)C2)=O)CCC2CCC(C1)S2 C1(CN(C)C(C2CCS(=O)(=O)N2)=O)CCCN(C(=O)CN2CC(F)(F)C2)C1 C1(CNC(C2N(S(CC)(=O)=O)CCCC2)=O)COCCN(C(C2(OC)CC2)=O)C1 C1(C(=O)Nc2ccsc2)C2CC1N(C(=O)CCc1ccncc1)C2 c1(C(=O)NCC2(OCC)CN(C(=O)C(C)C#N)C2)ccc(NC(C)=O)cc1F C=CC(CC(=O)NCC1CCC1NC(=O)C1=CCSC1)c1ccc(OC)cc1 N1(C(CCC)=O)CCCC(C2(NC(c3n[nH]c(C)c3Br)=O)CC2)C1 S(=O)(=O)(c1ccc(NCC2CCC(CO)O2)c(F)c1)NCC(C(C)(F)F)(C)C C1(C)(C(N2CC3(N(C(C4(OC)CCOCC4)=O)CC3)C2)=O)CC(C(C)C)=NO1 C(c1ccccc1Cl)=CC(=O)NCC1CN(C(c2cc(F)ncc2Br)=O)CCO1 c1(C(=O)NC(C)CNC(C2CC(C#N)C2)=O)ccccc1C(=O)N(C)C C1(C(=O)NC2(C)CCN(c3nc(Cl)c(C#N)s3)C2)CC2CCCCN2C1 C1(C(N2CCN(C(C(C)(O)C3CC3)=O)CC2)=O)CCCN(c2ccccc2)C1=O Cc1nc(CNC(=O)Cc2ccccc2F)oc1C(=O)NC1CSCC1C C(CCC(C)(C)C(=O)N1CC=CC(C(N2CCCC(CO)C2)=O)C1)OC c1(C(=O)NC(CC)CNC(=O)CC2CCCCO2)cc(O)n(CC)n1 C12(NC(c3ccn(C(CC)CC)n3)=O)CCCN(C(c3cc[nH]c3)=O)CC1C2 c1(CN(C2(CCC(=O)NC3CCOCC3)CCC2)C(=O)C=CCO)cccc(Cl)c1 N1(C(Cc2c(C)noc2C)=O)CC2CCN(CCOc3ccccc3C#N)C2C1 N1(C(C(C)c2ccco2)=O)CCCN(C(c2cccc(C(F)F)c2F)=O)C(C)C1 CCCC(C)(C)CC(=O)NCCCN(C)C(c1sccc1C(C)=O)=O c1(C(=O)NCCc2ccc(C)s2)c(NC2CCOC2)sc2c1CCC2 C1(CC(=O)N(C2CCCC2)CC=C)CN(C(C2CC(O)C2)=O)CCC1C C12(C(=O)NCc3cnc(C)o3)C(NC(=O)CCC3CC3(F)F)C3CC1C2C3 CCC(CC(=O)NCC(O)CCNC(c1cnn(CCO)c1)=O)C(C)(C)C C1(C(N2C(CNC(c3cn(C)cc3C(F)(F)F)=O)C=CC2)=O)CCCCC1(F)F N1(C(c2cncc(-c3cn[nH]c3)c2)=O)CCC2(CCCC2)C1 N1(C(C(C)OCCOC)=O)CC2C3CCC(C(NC(c4cscc4Cl)=O)C3)C2C1 C=CCC(C)(C)C(=O)NC(CN(C(=O)Cn1nc(C)cc1C(F)F)C)CC c1(OCC)ccc2sc(CN3CCCOC(CC)C3)c(C)c2c1 C(CCC)(C(O)C(=O)N1CCCC1CN=[N+]=[N-])NC(C(C=C)O)=O Cc1nc2nccc(NC3CC(C)N(C(=O)C(C)(F)F)C3)n2n1 c1(C(N(CC(C)(C)C)CCC#C)=O)ccc2occ(C)c2c1 N1(C(Cc2c(C)cccc2)=O)CCN(C(c2cc(CO)[nH]n2)=O)C(C)C1C N1(C(C(C)=CCC)=O)CCC2CCC(NC(c3ccccc3NC(N)=O)=O)C1C2 C1(NC(c2c(C)n(C)nn2)=O)CCN(C(c2cocc2C(N)=O)=O)CC1F N1(C(Cc2cc(C)cc(C)c2)=O)CC(NC(c2coc(Cl)n2)=O)CC12CCC2 c1(C(N2CCC(NC(CC3CCCC(C)O3)=O)(CF)C2)=O)cc(F)cc(F)c1N C1(NC(C2(C)CC2)=O)CC2(C1)CN(C(C1CCCN1Cc1ccccc1)=O)C2 C1(CC(=O)OC)CN(CC23CC(C#N)(CO2)C3)CC2(CCC2)O1 CC1(C(=O)NCCCCNC(=O)Cc2cccc(C(F)F)c2)COCC1(F)F Cc1c(O)ccc(C(N2CCN(C(C34CC(C)(CO3)C4)=O)CC2)=O)c1C C1(F)(C(=O)NCc2cccc(CC)c2)CCCN(C(C2(CO)CCCO2)=O)C1 C(CCCC(C)NC(=O)Cn1nnc(C)n1)NC(C1(COC)CCOC1)=O c1(C(N2CC3(C(NC(CC(CCC)C)=O)CC3)C2)=O)cn(C)c2ccccc12 C1(CNC(C(C)(C)OCCC)=O)CN(C(C2CCOC2CC)=O)CCN1C C(=O)(C(C)(C)C#N)NC(C1CCCN(C(=O)CCSc2ccccc2F)C1)C C1(O)(CNC(c2c(C)nc[nH]2)=O)CCN(C(=O)CC2OCCC2(C)C)C1 c1(C(N2CCOCC(NC(C=COCC)=O)C2)=O)cnc(O)c([N+](=O)[O-])c1 N1(C(COCC(=O)NC)=O)CC2CC(C(=O)NC(CO)CC(F)(F)F)(C2)C1 N1(C(CCCCOCC)=O)CCN(C(=O)C(C)N2CC(C)C2)CC12CCC2 CCCCCC(O)C(=O)NCC1CCCN1C(c1oc(C2CCC2)nc1C)=O C1(NC(C2CC(NC(CCCC=C)=O)C(O)C2)=O)CCCC(O)CC1 c1(C(=O)NCC2N(C(C(C)SCC)=O)CC2)cccc(F)n1 c1(C(N(C)CC2N(C(C(C)OCCC=C)=O)CC(F)C2)=O)cccc(N)c1Br N1(C(C2CC(=C)C2)=O)CC2CS(=O)(=O)CC2(CNC(C2(CCN(C)C)CC2)=O)C1 N1(C(COC(C)C)=O)CC2(CC(CNC(C3CC4(C3)OCCO4)=O)C2)C1 C(c1cccc(O)c1)=CC(=O)NC1(CN(C(=O)C(C)(C)CO)C)CC1 C1(O)(C(N2CC(NC(c3occc3F)=O)C2)=O)Cc2ccccc2C1 N1(C(CC(OCC)OCC)=O)C2CCC(C(=O)NC(CC)CCO)C1CC2 CCS(=O)(=O)C=CC(=O)N1CC(F)(F)CC1CNC(=O)C(C)(O)c1ccccn1 N1(C(c2n(C=C)ncc2)=O)CCN(C(c2coc(S(=O)(=O)NC)c2)=O)CC(O)C1 C1(C(=O)NC(CN(C(C(C)OCCOCC)=O)C)C)CCC(=C(F)F)CC1 Cc1ccc(OCCC(=O)NCC2CCN(C(=O)C=CC3CC3)CC2)cc1C c1(C(=O)NCC2(NC(c3ccc(C(F)F)cc3F)=O)CC2)ccc(O)c(F)c1 c1(C(=O)NC(C(C(C)C)NC(C2SCCCS2)=O)C)cc2cccnc2cc1F c1(C=CO)ccc(C2(Oc3ccccc3F)CC2)cc1.c1(N(C)CC)nnc(C2CC2)o1 N(C(=NCCF)N1CCCC2(CC2)C1)C1CC(NC(=O)NCc2ccccc2)C1 c1(C(C)C)nn(C)cc1C(=O)NC1CCN(c2nn[nH]n2)C1 CC1(C(=O)NCC(CO)NC(c2csc(C(F)F)c2)=O)CC(C2CC2)=NO1 C(=O)(C1c2ccccc2OCC1(C)C)NC1CN(C(C(C)CCC(C)(C)C)=O)C1 N1(C(c2ccc(OCC(C)C)cc2)=O)CCN(C(=O)C(O)C(F)F)CC(C)(C)C1 C1(C(=O)OCCn2cc(-c3nccs3)nn2)CCCN(C(c2cnn(CF)c2)=O)C1 CC1CCCC(C(=O)NCC2CCN2C(=O)Cc2ccnc(C(F)(F)F)c2)C1 C1(NC(c2c(CC)c[nH]n2)=O)CCCC(N(C)C(C2CC(O)C2)=O)C1 c1(C(C(=O)N(CC(C)NC(=O)C(C)(C)C2CCOCC2)C)C)cccc(C#N)c1 c1(C(N2CCC(C)(N3CCCC3)C2)C(=O)NCC=C)n[nH]c2ccccc12 N1(CC)CCC2(CC1)CC(C(N1CCC(c3nc4ccc(C)cc4[nH]3)CC1)=O)C2 N1(C(C2(OCC)CCCC2)=O)CCC2(CCC(NC(C3(C)CC(F)C3)=O)C2)C1 CN1CCN(CCCNC(=O)NC(C2CCC(O)C2)C(=O)O)CC1 CS(=O)(=O)C(CN=c1[nH]c(N2CC3CCC3C2)nc2c1SCC2)C1CC1 C1(CNC(=O)C(c2ccccc2)F)CNCCOC1 CON1CCC(C(=O)N(C2CN(C(c3cn(CC(F)F)cn3)=O)CC2F)C)CC1 N1(C(C=CC(=O)OCCCC)=O)CCCC(NC(=O)C(C)NC(=O)NC)C1 C1(C2CC2)(NC(C=CCN(C(C(CC(C)C)=O)=O)C)=O)CCCCC1 CC1CC(NC(=O)CN2CCS(=O)(=O)CC2)CCN1C(=O)CCc1ncccn1 c1(C(=O)NCCCN(C(C(=O)NCC)=O)C2CCCC2)c(C)nc2sccn12 c1(NC(c2c(C)cccn2)C)cc(Br)ccc1S(=O)(=O)N1CCN(C=O)CC1 N1(C(CCCCCOCC)=O)CCC2(CNC(c3ncccc3Cl)=O)CCCC12 c1(NC(C2(C(=O)OCC)CCC2)=O)nc(NS(C)(=O)=O)sc1C1CC1 CCCC(CC)C(=O)NC(CCSC)C(=O)NCCN1CCCC1 c1(C(=O)NC2CCCN(C(C=CCC)=O)CC2)ccccc1S(C)(=O)=O C1(C(=O)NCCOCC#C)CN(C(=O)C=CC)CC12CC2 c1(CC)ccc(N)c(C(=O)NC2CCCC2NC(=O)C=CC2CCOCC2)c1 C1(C(N(CCCCCNC(C2(SC)CCC2)=O)C)=O)CC2C=CCC(C1)C2 C1(C(N2CCC(C(C)NC(=O)C(F)C3CCOC3)C2)=O)(CC)CCOCC1 C1(NC(C2N(C(CCN=[N+]=[N-])=O)CSC2)=O)CCn2nccc2C1 N1(CCOC)CC2COCC2(C(N2CCCC(OC3CC3)C2)=O)C1 c1(OC)nccc(C(=O)NC2CC(CC(=O)NCC(C)O)C2)n1 c1(C(N(CCNC(C2C(C(C)C)CCO2)=O)C)=O)cnc(Br)c(N)c1 CC1=CCC(C)(C(N2CC3C(CNC(c4cnn(C5CC5)c4)=O)C3C2)=O)CC1 C1(N(C)C(c2cc(-c3ccc(F)cc3)[nH]n2)=O)CC2CC1N(C(=O)C(N)=O)C2 N1(C(CCOCCN(C)C)=O)CC(O)CC1(C)C(=O)NCc1nccn1C(F)F N1(C(CC2CC(OC)C2)=O)CCC(NC(c2cnc(S)[nH]2)=O)C(F)(F)CC1 CCCCC(C(=O)NC(C)CC1CN(c2cc(C(=O)OC)nc(C)n2)C1)C(C)C CCC(C)CCCCC(=O)N1CCOCCC1C(=O)NCCCc1ccccn1 N1(C(c2onc(C)n2)=O)CCCCC(C2CN(C(=O)CCC3CC(F)(F)C3)C2)C1 C#Cc1ccccc1CC(=O)NCC12CC1CN(C(C1C3CC4C(C3=O)C14)=O)C2 c1(C(N2CC3CC(NC(C4CC=CC4)=O)CC3C2)=O)cnnc2ccccc12 N1(C(CCCN(C(=O)CCC(=O)C2CC2)C)=O)CCCNC(=O)C1 N1(C(c2cc(C)c(C)s2)=O)C2CC=C(C(=O)N3CCC(F)(CF)C3)C1CC2 C(c1cncc(O)c1)=CC(=O)NCCCOCCNC(C1CSCCS1)=O c1(C(=O)NCC23CC(NC(C=C4CCC(C)CC4)=O)(C2)C3)cnc2c(c1)CCC2 N1(C(CCN(CCC)C)=O)C2CCC1CC(C(=O)NCc1ccnc(OC)c1)C2 c1(C(c2nnnn2Cc2ccc(F)cc2)NCC(C)(C)OC)cnn(C)c1Cl C1(NC(C(CC)n2ccnc2)=O)C(C)CCN(C(c2cnc(O)n2C)=O)C1C Cc1c(C(N2CCOC(C(C)NC(=O)C3=CC(C)(C)C3)C2)=O)cncc1Br C1(N(C(C(CC)O)=O)CC(C)C)CCN(C(C2CN(C(C)=O)C2)=O)CC1 C1(NC(c2ccc3c(c2)CC3)=O)CN(C(=O)COCC2CCOC2)CCC1F c1(OC)ccsc1C(=O)NCc1cccnc1.C1(C)C=CC(=O)N1C1CC1 C1(C)(C(=O)NC(Cn2cc(CNC(C#CC(C)C)=O)nn2)C)CC(C(C)C)=NO1 C#Cc1cccc(C(=O)NCC(O)CNC(c2cnccc2C(C)(C)C)=O)c1 N1(C(C(C)(C)Oc2ccccc2)=O)CCCCC1CCCNC(c1cocn1)=O C1(C(N2CC(O)(CNC(=O)CCOc3ccc(F)cc3)C2)=O)CC2C=CC1CC2 CCCCCC(O)CC(=O)NC1CCCC(NC(=O)CCCc2nncn2C)C1 c1(OC)ncnc(OC)c1C(=O)NCC(C)(C)CNC(=O)C=Cc1cn(C)nn1 c1(C(=O)NC(C2CCCN(C(C34CCC(C3)C4)=O)C2)C)ccc2occc2c1 c1(C(c2n(CC(=C)C)nnn2)NC2(C(=O)N(C)C)CC2)nc(C)sc1C c1(-c2occ(Cc3nnn(C(C)(C)C)n3)n2)ccc(I)cc1 C(=O)(C1CCCc2nncn21)NC1(CO)CCCN(C(CCSCC(C)C)=O)C1 Cc1nc(C(=O)NCC2(NC(=O)CSc3nccn3C)CCC2)c2ccnc-2[nH]1 c1(NC(C(Cc2cc[nH]n2)NC(c2cc(Cl)cs2)=O)=O)ccccc1Cl N1(C(c2c(OCC#C)nccc2)=O)CC2CC1CN2C(c1cn(C)c(=O)n1C)=O c1(C(=O)NC2(CNC(=O)CC3COCCO3)CC2)sc2cccnc2c1Cl C(CC(C(C)(C)C)NC(c1ncnc(O)c1Cl)=O)N(C(C(CC)(C)O)=O)C N1(C(C(CC)Oc2ccccc2)=O)CC2CC2(NC(c2cnc(OC3CC3)s2)=O)C1 c1(NC(C2CC3(CC(NCc4cncc(C)n4)C3)C2)=O)ccn2cnnc2c1 N1(C(C2(OC)CCC2)=O)CCC(O)(CCNC(C2CC2C(C)C)=O)C1 C(C(C)C(C)C(=O)NC1(CNC(C2CCCN(C)C2)=O)CC1)OC N1(C(Cc2c(C)nccc2)=O)CCC(C)C(NC(=O)CCC2CCCCC2)C1 C1(C(N(CC(C)(C)NC(c2c[nH]nc2C2CC2)=O)C)=O)CCCCC(F)(F)C1 C1(CC(=O)N(C)CC2N(C(COCC(=O)NC)=O)CCC2)CCOC1(C)C N1(C(C(C)Oc2ccccc2)=O)CCCC(C)(NC(C2(C#N)CC2)=O)C1 N1(C(c2nc(NC(C)=O)sc2)=O)CCOCC(F)(CNC(C2(CO)CC2)=O)C1 C(CNC(=O)CP(C)(C)=O)(CC(F)(F)F)NC(Cc1nnc(C)o1)=O CCCCC(C)(F)C(=O)NC1CC2CC(C1)N(C(=O)Cn1cnc([N+](=O)[O-])n1)C2 N1(C(CN(C2CC2)CC)=O)CC2CCC1CN2Cc1c(C)noc1COC C1(C(=O)NCC2(O)CCC(C)C2)(NC(C2CCO2)=O)CCc2cc(Br)ccc2C1 C(C)(CNC(C1CC(C(F)F)(OC)C1)=O)(C(C)C)NC(C(C1CC1)OC)=O C1(C)(C(=O)OCC)CCC(C(F)(F)F)CC1.C1(C)C(=O)N1C1CC1 CC1=C(C(=O)N2CCN(C(=O)CC3(n4cccc4)CCOCC3)CC2)CCO1 c1(OC)cc(C)c(CN2CCC(NC(C)C)C2)cc1OC(F)F c1(OC)cc(C(=O)NC2CC(CC(=O)NCC(N)=O)C2)ncn1 c1(OC)ccc(C(=O)N(C2CCC(NC(=O)CSCC3(F)CC3)C2)C)nn1 N1(C(c2ccc(-c3n(C)ncn3)cc2)=O)CCCC(NC(=O)CC(F)(F)F)C(F)C1 c1(C(=O)NCCNC(C2(C)CCSCC2)=O)ccn2ccnc2c1 C(CCCCC(=O)N1CC(COC)CC1CNC(c1cccc(Cl)c1)=O)=CC C1(C(=O)NC(C(=O)NCC(C)C(C)(C)C)CCF)CC2(CCC2O)C1 Nc1cc(C(=O)NC2CC(NC(c3ccc(OCC4CC4)cc3)=O)C2)ccc1Cl c1(C(=O)NCCCNC(c2c(C)n(CCO)cc2)=O)nc(Cl)c(Cl)c(N)c1Cl c1(C(N2C(CC(=O)NC(CC)CO)CC2)=O)cccc(NC)n1 CC1CCCn2c(C(N3CCN(C(C4CCC(C)(C)C4)=O)CC3C)=O)cnc21 C1(C(N2C(C)(C)C(CNC(=O)CC3CCCC3)CC2)=O)COC2(CCC2)CO1 c1(C(=O)NC2CC(NC(C3CCC(C)O3)=O)C2)[nH]c(=N)sc1C(F)(F)F C(C(C)(C)CC(=O)N1CC(O)CC1(C)C(=O)OC)OCC.C12CC(C)(C1)NC2=O c1(C2OCCN(C(C(CCO)N(Cc3ccccc3)OC)=O)C2)ccc2c(c1)OCO2 Cc1nc(CO)sc1C(=O)NC1CCOCC1NC(C1CC(O)C1)=O CC1CN(C(=O)CC2CCSC2)CC1CNC(c1cc(Cl)ccn1)=O c1(C(N2CC(CC(C)NC(c3ncccc3F)=O)C2)=O)cc([N+](=O)[O-])nn1C N1(C(c2ccc(C)n2C)=O)CC2OCC(NC(C3CCN(C)CC3)=O)C2C1 N1(C(C(CCSC)O)=O)CCC(O)(C(C)NC(=O)C(C)CC(C)C)CC1 C(=O)(CCS(N)(=O)=O)NC(C(C)C)CCN(C)C(c1cc(C(C)(C)C)n[nH]1)=O c1(C(N2CC(O)(CCNC(C3CCCC(C)O3)=O)C2)=O)ccc2[nH]ccc2c1 CCCCCC(O)CC(=O)NC(C)CN(C)C(C1CCOC(CCC)C1)=O N1(C(C(C)Cn2cccn2)=O)CC2(CNC(C3CCCC(F)C3)=O)CC(F)(C1)C2 C1(Sc2c(C(=O)OCC)[nH]nc2Cl)CCc2cc(OC)ccc2C1=O c1(C(N(C)CC2CCCC(NC(=O)CCC(C)(C)F)C2)=O)ccc([N+](=O)[O-])n1C c1(OC)ccc2c(C(=O)NC3CCN(C(=O)C#CC4CC4)CC3F)csc2c1 c1(C(=O)NC(CC2CN(C(C(CC#C)O)=O)C2)C)ccc2ccn(C)c2c1 N1(C(=O)NC(C(C)(C2CC2)OC)C)CCCSC1C c1(OC)cc(C(=O)NC(CCN(C(=O)C(O)C2CCCC2)C)C(C)C)cc(C)n1 C(CS(=O)(=O)c1ccc(C)cc1)NC(c1cc(F)ccc1F)CC=C c1(OC)cc(C(N2CCC3(NC(=O)C4=CCCC4)CCCC23)=O)cc2c1OCC2 C(=O)(C1=CC2C=CC(C1)C2)NC12CC(NC(c3cnc4ccsc4c3)=O)(C1)C2 c1(CC(=O)NCCN(C(=O)C=CCOCC)CCC)nc2ncccn2n1 CN1C(=O)Cc2ccc(C(=O)NC3CC(C)(NC(=O)CCn4ccnn4)C3)cc21 N1(Cc2cccc(CC)c2)CC(NC(c2ccc(OC)nc2OC)=O)C(C#N)C1 c1(C(N(C(C)C)CCNC(c2ccn(C)c2)=O)=O)ccc(Cl)c(Cl)c1N c1(CNC2CCC(NC(C3(C(F)(F)F)CCC3)=O)C2)cc(Br)ccc1OC(F)(F)F Cc1ccc(C(C2(CF)CCC2)NC(C(=O)O)c2cccs2)cc1 N1(C(C2CN(C(C)C)C2)=O)CCCC2CC3(CCC3)C12 c1(NC)cncc(C(=O)N(C(C)C(N2CC(N(C)C)C(C)C2)=O)C)c1 c1(C(N2CCC(C)(NC(c3cccc(N)c3F)=O)C2)=O)cc2cc(F)ccc2s1 c1(CSCC(=O)NCC2N(c3snc(CCC)n3)CCC2)ccc(Cl)cc1 C(CC1CCC1)(C(=O)NCC(F)CO)NC(CSCCCC)=O Cc1conc1C(=O)NC(C(=O)NC1CC1F)c1ccoc1 Cc1ccc(NC(=O)C(CC(C)C)ONC(C2CCC(C3CC3)C2)=O)cc1F c1(C(CC)(C)C)n[nH]c(=NCC2(NC(=O)Cc3cccc(COC)c3)COC2)o1 C=CC(CCC)CC(=O)N1CCCC1CN(C(=O)COc1cc(F)cc(F)c1)CC Cc1n[nH]cc1NC(c1nc(C(=O)NCc2ccoc2)cs1)=O C1(CCNC(c2n(CC)ncc2)=O)CC(OC)CN1C(c1cocn1)=O Cc1c(C(=O)NCC(C)CNC(c2cnc(C3CCOC3)s2)=O)cccc1C#N N1(C(CCN(C(C2CC2F)=O)CC)=O)CC(F)CC(F)C1 N1(C(CCC(=O)N(C)C)=O)CCCC2CCN(C(=O)C=Cc3cncn3C)CC12 C(=O)(C(CC1CC1)Nc1ccc(C(F)F)s1)NCC(OC)OC N1(C(C2C(=C)C2)=O)CCCC2(CCN(C(c3ncoc3CC)=O)C2)C1 CC(CCNC(=O)Cn1ccc(C2CC2)n1)CCNC(c1cnc[nH]c1=N)=O CC(C)=C=CC(=O)NC(Cc1cc[nH]n1)C(=O)NCC1CCC=CCC1 c1(C(N2C(CNC(CC3C(OC)CC3)=O)CC2)=O)nc(C)ns1 CCC(CC)CCCNC(=O)C(Cc1cc[nH]n1)NC(=O)C=Cc1cc(C)no1 c1(NC(C2(C)CCCN(C(Cc3c(C)cccc3)=O)C2)=O)nc(Cl)c(Cl)cc1Cl C1(C(N2CC(C)(CC)C2)=O)CC2CC1CN(C(C1(CO)CC1)=O)C2 C1(CNC(CCC2CC(NC(COCCCOC)=O)C2)=O)CC2(CC2)C1 C12(CNC(C3C(C)(C(F)F)C3)=O)CC(CN1C(C1(C)CCCO1)=O)C2 C(N=c1nc2ncn(C)c2c(NCc2cc(C(F)F)no2)[nH]1)c1nnn(C)n1 N(C(=NCCCSC)NC1CCN(c2nccs2)CC1)CC1(OC)CCSCC1 C(=O)(CC(C)CC(C)C)N1C(CCOC)CN(C(c2ncc(N)cc2Cl)=O)CC1 C1(N(C(=O)CCSC(C)(C)C)C)CCCCN(C(CC(N)=O)=O)C1 C=C1CC(C)(NC(c2ccccc2)C(=O)N(C)C)C1 Cc1cccc2c(C(=O)NC3CCCC(NC(C4CC4C)=O)C3)cccc12 N1(C(C=CC=CCC)=O)CCC(CNC(c2cn(C3CCOC3)cn2)=O)C12CC2 c1(C(N2C3CN(C(C(=O)N(C)C)=O)C(CC3)C2)=O)cc2cc(Br)cnc2[nH]1 c1(C(C(=O)NC)N(C)Cc2cnn(C)c2)ccc(N(C)C)cc1OC CC(C)(C(=O)NCC1CCCN1C(=O)CC1CC=CCC1)N1CCOCC1 N1(C(CCC2CCN(C)CC2)=O)CC(NC(=O)CC2CSCCS2)C(C2CC2)C1 c1(CC(=O)NCC2C(NC(c3n(C)nnc3Br)=O)CC2)ccc2occc2c1 C1(C)(CNC(CSSC)=O)CN(C(C2CCC2c2nncn2C)=O)C1 N1(C(CC2N(C(C(C)(C3CC3)OC)=O)CCOC2)=O)C2C=CCC1CCC2 C1(NC(C2(CO)CCC2)=O)CCCC(NC(C2(C(F)F)CCCO2)=O)C1 c1(C(N(CCCCCNC(c2nn[nH]c2Cl)=O)C)=O)cc2nccn2c(O)n1 C1(CNC(C=CC(C)C)=O)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CCC1C c1(CC(=O)NCCC(C)(C)NC(C(C(C)(C)C)SC)=O)ccc2oc(O)nc2c1 CC1(C)CN(C(c2ccn(C(F)(F)F)n2)=O)CCC1NC(=O)Cc1ccno1 C12(C(=O)NC(C)(C)CNC(C3CC34CCC4)=O)CCCCC1NC(=O)CC2 c1(CNC2CCC(=O)NC2c2ccccc2)nc2cccc(Cl)c2s1 c1(C(N2C(C3CCN(CC)C3)CCCC2)=O)ccc(N2CCOCC2)cc1C c1(OC)ccc(C)c(C(=O)NC(C)(C)CCN(C)C(C2CCOC(C)C2)=O)c1 CC(C)C(O)CC(=O)N1CC(CNC(=O)C(C(C)C)NC(N)=O)CC(C)C1 c1(C(N2CCC(NC(CCCC=C)=O)C(F)C2)=O)ccc2[nH]c(=N)sc2c1 CCC(O)C(C)(C)C(=O)NOCC(=O)NCCC1(C)CC1(F)F C1(CNC(CN(CCC)C)=O)CC(F)CN1C(=O)Cn1nnnc1-c1ccsc1 C1(CC)CN(C(=O)C(F)(F)c2ccnn2C)CCC1NC(c1cccc(O)n1)=O c1(CO)cccc(CN=c2[nH]nc(Cl)s2)c1F CCCCCC(C(=O)NCC1CCCN(C(=O)C(C#N)CC)C1)C(C)C N1(C(C(c2cccs2)NC(C(C)=C2CC2)=O)=O)CCC(C2(C)CC2)CC1 C1(NC(c2n[nH]cc2F)=O)CCN(C(=O)C=CC2CCOC2)CC1F O=C1NC(=O)c2ccccc2C1=CNCC1(O)CCc2ccccc21 C(=O)(C1=C(Cl)CCOC1)NCCC(CNC(c1cc(CC(C)C)on1)=O)O CC1(C)COCCC1C(=O)Oc1ccc(OCc2ccccc2)cc1 C1(NC(CSSC)=O)CC1C1CCCN(c2ncnc3c2nnn3C(C)C)C1 Cc1ccc(C2(CN3CC(F)(CNC(=O)COc4ccc(F)cc4)C3)CC2)nc1 C(=O)(C(CN(C=O)CO)CC1CC1)OC(C)(C)C.C1(O)(CSC)CCSCCOC1 C1(NC(C2C(C)C2)=O)CCCCN(C(=O)CCSc2ccc([N+](=O)[O-])cc2)CC1 N(C(=NCCF)NCC(C1CC1)C1CC1)C1CC(OC)C1 c1(C(C(=O)NCC2CC(n3cc(C4CCCC(O)C4)nn3)C2)O)ccc(Cl)c(Cl)c1 C1(C(=O)NC(CSCC)C(=O)NC(C)Cc2cccnc2)CCC(=O)N(C)C1 C(C)(C(C(C)C)NC(=O)CSCCC(F)(F)F)NC(c1cc(COC)no1)=O C1(C2(NC(C3CCC3(F)F)=O)CC2)CCCN1C(c1ccsc1Br)=O C1(C2CCCCO2)(C(=O)NCCNC(=O)C(c2ccccc2F)O)CCOCC1 C1(N(C(c2c(CC)n(C)nn2)=O)C)CCN(C(=O)Cc2cc(C)nn2C)CC1C CC1CC(CNC(=O)C=CC2CCC2)CN1C(C1CCN(CC(F)(F)F)CC1)=O c1(C(=O)NC2(CC=C)CN(C(C3CCC(=O)C3)=O)C2)cc(Br)c2[nH]nnc2c1 C1(N)COC2CN(C(=O)OC(C)(C)C)CC12.c1(CNC(C)=O)c(Br)noc1C1CC1 C1(CNC(C2C(CCC)CCC2)=O)CN(C(=O)CNc2ccccc2)CCCO1 N1(C(c2c(OC)nccc2)=O)CC(CC(=O)NCCCc2nccs2)CC1(C)C N1(C(C2(SC)CCC2)=O)CCCCC(CCC(N2CC(O)(c3nn[nH]n3)C2)=O)C1 c1(C(=O)NCCN(C(C2(CC)CCCO2)=O)C)cnn(C)c1C(C)(F)F c1(C(=O)NCC(C)NC(C(C)OCCC=C)=O)c(C)nn2c1CCCC2C C1(OC)CC2CCC1N2C(=O)CC1N(C(=O)CC2(OC)CCC2)CCC1(C)C Cc1cc(C2(NC(=O)C(Cn3ccnn3)NC(C3CC(C)(C)C3)=O)CC2)no1 N1(C(C2C(C(C)C)C2)=O)CC(CNC(=O)CCc2ccsc2)C2(CC2)C1 CC1CCC(NC(=O)C(c2cccc(Cl)c2)O)CN1C(=O)CN1CCCS1(=O)=O N1(C(C2(CC=C)CC2)=O)CCCC(CC)(NC(c2ccnn2CCOC)=O)C1 N1(C(CCOCCOC)=O)CCN(C(C2(C(F)(F)F)CC2)=O)CC1CC(C)(C)C O=C1CCC2CN(C(=O)NC(c3cccc(OC(F)F)c3)C(F)(F)F)CC2N1 C1(NC(c2ccn(C)c2CC(=O)O)=O)CN(Cc2cnc(Cl)nc2Cl)CC1(F)F N(C1CCc2cc(Cl)ccc21)C(=O)NC(c1ccc(Br)cc1)CC N(S(=O)(=O)N1CCCCC1)Cc1nc(C(=O)OC)c(C)o1 N1(C(c2c(C)nc(C)[nH]2)=O)CCC(C2CN(C(=O)C(O)C3CC3)C2)CC1 CC(C)(CCS(C)(=O)=O)C(=O)N1CC(CNC(=O)COC(C)(C)C)C2(CC2)C1 C1(CCC(=O)NCC=CCNC(c2ccc(C3CCC3)cc2)=O)NC(=O)NC1=O O=C(C#CC1CC(F)(F)C1)NCC12CC1CN(C(=O)CCSC1CCCC1)C2 C1(c2cn(CCCOC)nn2)CC2CCC(C1)N2C(C1CCCCN1C)=O N1(C(C=C(CC)C)=O)CCOC2(CCN(C(=O)CCOC3CCCCCC3)C2)C1 C1(C(N(C)Cc2c(C)cccc2)=O)CCCN(C(C2CC3(C2)CC3(F)F)=O)CC1 C(=O)(C(F)CCC(C)C)NCC1CCCN(C(c2cncc(C#C)c2)=O)C1 N1(C(COCCCCC)=O)CCCCC1C(=O)Nc1[nH]ccc1CC C1(C(=O)NCC2C(CNC(c3cc(C(C)(C)C)on3)=O)C2)C2(CC2)C12CC2 C(=O)(C(C(C)C)c1cnn(C)c1)NCC1(NC(c2c(SC)csc2)=O)CCOC1 N1(C(C(C)OC(C)(C)C)=O)CC(NC(=O)C(F)(F)C(F)F)CCC(O)C1 Cc1cc(F)cc(C(=O)NC23CCCN(C(=O)C(C)NS(C)(=O)=O)CC2C3)c1N Cc1cc(F)c(C(=O)NCC2(CCNC(C3C4CS(=O)(=O)CC34)=O)CC2)cc1F CCCCS(=O)(=O)NCC(=O)N(CCCCCN(C)C(C1CC1F)=O)C(C)C C1(C(=O)NC2C3CN(C(c4c[nH]c(=N)o4)=O)C2C3)CC2(C1)CC(F)C2 N1(C(CCC=CC)=O)CCN(C(=O)C(C)NC(C2CCCC2)=O)CCC1C C=C=CCCC(=O)NCCn1cc(C(=O)NCc2nc(C)cs2)cn1 c1(CCNC(C(CC2CC2)NC(C(CC2CCC2)OC)=O)=O)ncccc1F O=C(C1=Cc2ccccc2C1)NCCC1(C(=O)NC2C3CC4C(C3)C24)CCCC1 N1(C(c2c(C)n(C)cn2)=O)CC2CC(C1)N(C(=O)Cn1ncccc1=O)C2 CC1CC(C(=O)NCC(O)CNC(C2(CC(=O)NS(C)(=O)=O)CCC2)=O)CN1C Cc1cnc2c(C(=O)NC3CC4CC3N(C(C3(C#N)CC3)=O)C4)cnn2c1 C12(NC(Cc3cccc(C)c3F)=O)CCN(C(c3nn(C)cc3N)=O)CCC1C2 N1(CC)CC(C(N2CCCCC2CN(C)C(c2ccon2)=O)=O)CC1=O Cc1cc(C2CC2)ncc1C(N1CCOCC1CCNC(c1ncn(C)n1)=O)=O CCC(CC)(CN=c1[nH]cnc2c1CCCC2)NC(c1c[nH]nc1C)=O C1(NC(CCCCSC)=O)CCN(C(=O)CCc2c(N)cnn2C)CC(C)(C)C1 c1(SC)cccc(C(=O)N(CC(C)N(C(=O)C(O)CN2CCOCC2)C)C)c1 Cc1cc(N2CCC3(CC(C(F)F)=NO3)C2)nc(=NC(C)Cc2cccnc2)[nH]1 C1(C#N)(NC(c2c(CC)cccc2)=O)CCN(C(c2csc(Br)c2)=O)C1 C1(C(=O)NC2CC3CC(NC(CCC)=O)CC3C2)CC2CCC1CC2(F)F c1(NC(=O)N(c2ccc(SCc3ccccc3)cc2)N2CCCC2)ccc(Cl)cc1 c1(C(=O)NCC2CN(C(CNS(CC)(=O)=O)=O)CC2C)cncc(C)c1C c1(C(N(CCCNC(Cc2scc(C)c2)=O)C2CC2)=O)ccc2c(n1)OCCO2 C1(C(N2CC(CCNC(c3cc(CC)no3)=O)C2)=O)CC2CCCC(C1)C2(F)F CCC(O)C(C)(C)C(=O)N(CCNC(=O)C(c1ccccc1)SC)CC C(=O)(C(F)C(C)(C)O)NCc1ccc(CN(C(=O)CCC2CCN(C)C2)C)cc1 Cc1cc(F)ccc1C(=O)NCC1CN(C)CCN1C(=O)CCCc1cnn[nH]1 NS(=O)(=O)c1ccc2c(c1)CCCC2NC(c1ccccc1Cl)C1CCCO1 C12(CNC(CC3C(COC)C3)=O)CCC(NC(c3cnns3)=O)(CC1)CO2 C1(NC(c2n(CC=C)ccn2)=O)(CO)CCCN(C(c2ccc(C)s2)=O)C1 C1(CCOC)CN(C(c2cnc(C3CCC3)s2)=O)CCN1C(=O)C(O)C1CCC1 N1(C(C2(C#N)C(C)(C)C2)=O)CCCC(CO)(CNC(=O)CCc2cccnc2)C1 C12(NC(c3cc(CC)c(F)cc3)=O)CCCC1N(C(=O)C1=C(Cl)CCOC1)CC2 CC1(C)CCCC1CNC(C1(CO)CN(C(c2n[nH]c(=N)[nH]2)=O)C1)=O N1(C(c2cc(C)[nH]c2)=O)CCCC(C2CN(Cc3ccc(C(C)(C)C)cc3)C2)C1 c1(C(=O)NCC(C#C)OC)[nH]ccc1CNC(=O)Cc1cc[nH]c1 N1(C(C(CC)Sc2ccccc2)=O)CCC(CNC(C2(CO)CC2)=O)C(F)(F)C1 c1(CNC(C(OC)OC)=O)cc(C(=O)N(CCCCO)C2CC2)co1 c1(C(=O)NC2C(NC(C(=O)NCC)=O)CCCC2)nn(C)c2c1CSCC2 CC(C(=O)NCC1CN(C(=O)C=Cc2ccncn2)C1)C(C)S(C)(=O)=O c1(NC(CC2C=CC(NC(=O)CCC3CCCC3)C2)=O)ccc2ncnn2c1 N1(C(c2c(O)nnc(C)c2C)=O)CCCCC2(C1)CN(C(=O)CCCC#N)C2 c1(C(N2CCC(CCNC(C(C)C#N)=O)C2)=O)ccc(C2CC2)nc1 c1(C(N(CCCNC(CC(CC)C)=O)C)=O)cccc(C)c1N N1(C(Cc2cccc(SC)c2)=O)CCC12CCN(Cc1cc[nH]n1)CC2 C1(O)(C(C)NC(c2nnc(C)s2)=O)CCN(C(=O)CCCc2cccs2)C1 C1(C)(CC(=O)OC)CCN(C(=O)Cc2csnn2)CC1.C1CC(=O)N1CCO c1(CC(=O)NCC(CN(C(C2CC(O)(CC#C)C2)=O)C)C)ccccc1C(C)C N1(C(CC(CN(C)C)O)=O)CCC(C)(C)C(CNC(=O)CCSCC(N)=O)C1 N1(C(c2ccc(C(F)F)cn2)=O)CCN(C(=O)CO)C(c2ccccc2Cl)C1 C(=O)(C(C)(C)CCC#N)NCC(Cn1cc(CNC(C(C)O)=O)nn1)(C)C C1(C(=O)NC23CC(NC(=O)C4=COCCO4)(C2)C3)CCOC2(CCCC2)C1 Cc1cnc(C(=O)NCC2CCC2NC(c2sncc2Br)=O)c(F)c1 Cc1ccncc1CCNC(C1CC(NC(=O)CCCCC2CC2)C1(C)C)=O C1(NC(CC(C)C)=O)CCN(C(=O)C(C(C)C)n2ccnc2)CC1 CC1(C)COC(C(=O)NC2COCC2C(=O)NCC2CCC(C)(C)O2)C1 n1(C(CC)C)nccc1C(=O)N(C)C(c1cn(CC2CCC2(F)F)nn1)C Cc1[nH]nc2c(C(=O)NC34CCC(CC3NC(c3ccoc3Cl)=O)C4)cccc12 Cc1nc(CO)ncc1C(=O)NC(CNC(=O)CN1CC(C)(C)C1)C(C)C(C)C CCC(CC(F)(F)F)C(=O)NCC1(CNC(=O)C(C)c2ccsc2)CC1 C1(=CC(=O)NCC=CCNC(CC2C(C)CCO2)=O)CCCCC1(C)C C1(C(=O)NCc2cccc(C#C)c2)CCC(C)(C)N(C(=O)C=CCCC(C)C)C1 c1(CC(=O)N(C2CC2)CC)ncc(-c2ccc(OC)nc2)cn1 c1(COC)ccnc(C(=O)NCC2(F)CN(C(c3coc(C)c3)=O)C2)c1 C1(C(N2CC(C3OCCN(C(C4C(CC)CCC4)=O)C3)C2)=O)CC(C)(C)CCO1 c1(C(N2C(C(C)C)(C(=O)NCCC3(C)CC3(F)F)CCC2)=O)cc(O)nc(O)n1 Cc1ncccc1CC(=O)N(CCC(=O)NCC1CC1C)C c1(C(N2CCCC(CNC(C(CCC)NC(N)=O)=O)C2)=O)ncc2ccccn12 c1(C(=O)NC2CC(C)N(C(c3ccc(Cl)[nH]3)=O)CC2)cncc2ccccc12 N1(C(CC(=O)NCC)=O)CCC(CNC(C2(Cl)CC2)=O)C(C)C1 c1(CNC(c2cc3ccccn3c2)=O)nc2c(s1)CN(C(c1cscn1)=O)CC2 c1(C(=O)NCC2C(NC(C(C)NC(C)=O)=O)CC2)ccc(O)c(Cl)n1 C(C1=NOC2CN(C(=O)CCCS(N)(=O)=O)CC12)NC(c1noc(CC)c1C)=O C1(C(=O)NCC2C(C)CN(C(=O)CC3(O)CCOCC3)C2)CC2(CCCC2)CO1 C1(C(N(CC#C)Cc2ccco2)=O)CCC(C(C)C)N1C(C1CCCC(=O)N1)=O N1(C(C(CC)CC)=O)CCN(C(C2(C#N)CCCCC2)=O)C2(CC2)C1 c1(C(=O)NC2CN(C(CSCC(C)C)=O)CC(C)C2)cc(C#N)c(O)nc1N c1(OC)ccc(Cl)c(F)c1C(N1CC(CNC(=O)CCOC(C)=O)C(O)C1)=O n1(CC(N2CC(CNC(C(CC)SC)=O)C2)=O)ccc2cc(Br)ccc12 C#Cc1cnc(C(=O)NCCN(C(=O)C(C(C)C)C(C)C)CC)c(C)c1 N1(C(C=C2CCC(C)C2)=O)CCCCC2(CCN(C(=O)Cc3cnn(C)n3)C2)C1 C1(NC(CCSCC)=O)CN(C(=O)Cc2cnns2)C(C)(COC)C1 C(=O)(C1=NOC(C2(O)COC2)C1)NC(CNC(c1cc(C)ncc1)=O)C1CC1 N1(C(c2nc(CC)oc2)=O)CC2CC1C2CNC(=O)CC1(O)CCC1 Cc1cc(C)c(C(N2CC(CCCCNC(c3nccnc3N)=O)C2)=O)s1 CC1(C)C(NC(c2ccc(-c3cc[nH]n3)s2)=O)C(C)(C)C1NC(c1cnn[nH]1)=O c1(CCNC(C(C2(C)CC2)NC(C2C(CC)OCC2)=O)=O)cnn(C)c1C C1(C)(CC)CC(C(=O)NCCC=Cc2ccc(OC(F)(F)F)cc2)CCO1 N1(C(C=C(C)C(C)C)=O)CCCN(C(=O)CCOc2cccc(C)c2)CC1 c1(C(N(CC(CC)NC(c2cc(Cl)c[nH]2)=O)C)=O)csc(Br)n1 CCC(O)C(C)(C)C(=O)NC1CCC1CNC(c1ccnn1C)=O Cc1cc(C(=O)NC2CN(C(=O)C=CS(C)=O)C2)c(F)cc1F C1(C(=O)NCC2(NC(=O)Cc3nc([N+](=O)[O-])n[nH]3)CCC2)CCN2CCOCC12 C(=O)(C(F)(F)C(F)(F)F)NCC(CNC(c1cccc(N2CC=CC2)c1)=O)O c1(C(N2C3C(NC(CCCOCCC)=O)CC(C3)C2)=O)ccc2oc(=N)[nH]c2c1 c1(N2CCN(C)C(CO)C2)nc(N2CCCC(CCF)C2)nc2ccc(Cl)cc12 c1(CC)onc(C)c1C(=O)NC(C)CC(C)NC(C1(CC)CC(C)(C)C1)=O C1(C(N(CCCNC(c2nc(C)sc2)=O)Cc2ccccc2)=O)CNC(=O)N1C C(C(C(C)C(C)C)NC(c1cnc(C(C)(C)C)[nH]1)=O)NC(C1CC(=C)C1)=O C1(C(=O)NCC(CC)(CC)NC(CC)=O)CCc2c(n[nH]c2C)C1 C1(C(C)(C)C)CCN(C(=O)C2=NOCC2)C(CNC(C2(C3CC3)CC2)=O)C1 C=CCCCCCCCC(=O)N(CC(C)NC(c1cn2cc(C)ccc2n1)=O)C N1(C(C2(C#N)CC3(CC3)C2)=O)Cc2nccn2CC(NC(C2CC23CCC3)=O)C1 C(=O)(C(C)(F)C(=O)NCC(C1CCN(C(C2CCOC2)=O)CC1)(C)C)OCC C(C)(CO)(C(=O)N1CCCC(C(C)NC(=O)CCCOC(C)C)C1)OC n1(C(C)C)nc(Br)cc1S(=O)(=O)N(C)CC1CCNC1 Cc1ccc(C(=O)NCC(C(=O)NC2CC3CCC2CC3)C(C)C)c(C)c1 c1(C(=O)NC2C=CCN(C(Cc3ccc(C)s3)=O)C2)ccc2ccnc(O)c2n1 C(C(C)(C)NC(=O)C(F)C1CCC1)CCNC(COCCOC)=O C1(CC(N)=O)(NC(C(C)OCC#C)=O)CCN(C(C2CCCC(C)(C)C2)=O)CC1 Cc1cc2[nH]c(C(=O)OC(C(F)(F)F)C3CC3)cc2o1 Cc1cccc(C)c1CC(=O)NCCCCCNC(=O)CCc1cncc(F)c1 c1(OC)cccc(Br)c1C(N1CC2(CC(C(N3CCC(C)C3)=O)C2)C1)=O c1(NC(CCN(C(c2c(C)c[nH]n2)=O)C)=O)cccc2ccncc12 c1(C(=O)NC(C2(CNC(c3cncs3)=O)CC2)C)c[nH]c2ccc(Cl)cc2c1=O Cc1cc(NC(C2CN(Cc3ccccc3C(=O)O)CCO2)=O)cc(F)c1 N1(C(CCOC(C)C)=O)CCC(O)(CNC(C2C3CCC2(c2ccco2)C3)=O)C1 C1(C#CC(=O)N(CC(C)CNC(=O)CC2(C)CCCC2)C)(CC)COC1 N1(C(C2C3(CCN(C(C(CCCC)=O)=O)CC3)C2)=O)CCCC2(C=CCO2)C1 N1(C(CC(=O)OC(C)(C)C)=O)CCN(C(C2CCC(O)C2)=O)C(CC(F)(F)F)C1 C1(CC(=O)NCC2N(C(C3C(C)(C)C3)=O)CCCC2)CCCCCC1(F)F Cc1ccc(CC(=O)NC(CC(=O)N(C2CCC2)C2CCC2)C2CC2)cn1 C#CCC(C(=O)N1CC(C)(O)C1)NC(C1CCCCCC1)=O C(=O)(CC(C(C)CC)NC(C1(OC)CCOC1)=O)NCCCCCCC=C C1(C(N2CCC(C)(CCC)C2)=O)CCCCN(C(c2snnc2C)=O)C1 Cc1cc(C#N)ccc1-c1nc(C(=O)NCc2cnc(Cl)s2)c(C)s1 N1(C(C2CCC(CCCC)CC2)=O)CC2CC(NC(C3CCC(C)(C)O3)=O)C2C1 c1(C(N2CC=CC2Cn2cc(-c3cn[nH]c3)nn2)=O)c[nH]c2cc(Cl)ccc12 Cc1c(F)ccc(N)c1C(=O)NCC(C)CNC(C1CCCN(CC(F)F)C1)=O c1(C(N(CCCNC(=O)CC2CC(n3cnnc3)C2)C)=O)csc(C2CC2)n1 C(CCC(C)NC(=O)C(n1ccc(Br)n1)C)NC(CN(C(=O)OC)C)=O C1(NC(c2cc(C)cc(O)n2)=O)CC2CC1CN(C(c1cc3occc3s1)=O)C2 Cc1cc(=NC2CC(C(N)=O)C2)[nH]c(N2CCC(C)(CN3CCCCC3)C2)n1 CCCC(CCCO)C(=O)NC1CCN(C(=O)C(C(C)C)c2ccccc2)C1 c1(C(=O)NC(CNC(CCCC=C)=O)(C)C)noc2c1CC(C)CC2 CC1(C(=O)NCC2CCC2NC(c2cnoc2C2CCC2)=O)CC(F)C1 N1(C(CCNC(Cc2n(C)ncc2)=O)=O)CCSC2CCCC12 c1(C(C)NC(=O)Sc2ncc(C(F)(F)F)cn2)ccc(Cl)c(Cl)c1 Cc1cc(C)n2cnc(C(N3CCC(NC(C4(C)CCCOC4)=O)CC3)=O)c2n1 N1(C(c2cc(C)on2)=O)CCC(C(=O)NCC(=O)NC(C)(C)C)C12CC2 c1(SC)ccc(C=CC(=O)NC(C)CCNC(=O)Cc2ccc(C#N)cc2)cc1 c1(CC)[nH]nc(C(=O)NC2C3CN(C(C4(O)CCOCC4)=O)CC23)c1[N+](=O)[O-] c1(CC)nc(C(=O)NCC(O)C(=O)N2CCCC2c2ncc[nH]2)co1 c1(C(N2CC(n3cc(NC(C4CC5CCC45)=O)cn3)C2)=O)ccc(O)cc1 N1(C(C2C(C)OCC2)=O)CCOC2(CCN(c3nnc(C(F)(F)F)s3)CC2)C1 c1(C(CC)=O)cc(C(F)(F)F)ccc1CC1CCCN(C(=O)COC2CCC2)C1 C1(C(N2CCC(CF)(NC(C3(CCF)CC3)=O)C2)=O)CCCCC1C1CC1 C1(C(C(=O)N2CCC2C(N)=O)NC(=O)C(c2ccccc2)=O)CCCCC1 c1(CC(C(=O)NCCN(C(=O)Cc2ccon2)CC)O)ccc(OC)cc1 C(CC(C)CC)(C(=O)N1CC(C2=NOCC2)C1)NC(C(=O)NCC)=O c1(CN2CCC(CC(=O)NCc3n(C)nnc3)C2)cc(F)cc(Cl)c1O O=C(CC(C(F)F)n1cccn1)NC1CC2(C1)CC(NC(C13CCC1C3)=O)C2 C#CCC(CC(=O)NCCOC)NC(C1CCCC(=O)CC1)=O C(=O)(N1OC2C=CC1CC2)C1N(C(C(C(C)(C)C)CO)=O)CC(=O)NC1 Cn1c(NC(=O)CC23CCCC2C3)cnc1C(=O)OS(C)(=O)=O CC(CCN(C)C)C(=O)N1CCOCC1CC(=O)NCCCc1ncc[nH]1 CS(=O)(=O)C1(C(=O)NCC2CN(C(=O)C3=C(Cl)CC3)C2)CC1 CC(=O)C(C)(C)CC(=O)NCC(O)C(N1CCCC1(CO)CO)=O C12(CNC(CCc3cncc(C)c3)=O)CC(NC(=O)CC3=CCCC3)(C1)C(C)O2 C1(C)(C(=O)NCC2(NC(CCc3ccc(C)s3)=O)CC2)CCCCO1 C(=O)(C(CC)C(C)O)NC(CNC(c1n(CCC)ncc1)=O)C CCCCCC(C)(C)C(=O)Nc1ccc(CCC#N)cc1 N1(C(c2c(C)ncc(Cl)c2)=O)CC2CCCC2(NC(=O)C=C2CCC(C)C2)C1 CC1COC(C)(C)CN1C(=O)CN(C(=O)C(C1CCCCC1)C)C1CC1 CCCC(C(N)=O)NC(=O)C(CCC1CC1)NC(=O)CN1CCC(OC)C1 NS(=O)(=O)c1cccc2c1CCN(N1CCCC1C1CCCCC1)C2 N1(C(C2CC(OC)C2)=O)CCCCC(NC(=O)C(C)C(C)O)C1 c1(NC(CC)=O)cncc(C(=O)NC(C)CN(C(=O)Cn2cnnn2)C)c1 n1(CCOC)cc(CC(=O)NCC(C)N(CC(=O)NCC2CC2)C)cn1 N1(Cc2nc(CC)on2)CC(NC(c2conc2C(F)(F)F)=O)CCC1C C(C(=O)NC(C)COC)(C1CCCO1)OCC.C1(C2CCC2)C(=O)N1 N1(C(C2C(C)C2)=O)CCCC(C)(C)C1CNC(C1(C)CNC(=O)C1)=O c1(C(N2CC3C(C(=O)NCCC(F)(F)F)(C3)C2)=O)cc(F)ccc1I c1(C(=O)NC(C2CCN(C(Cn3ccc(C)n3)=O)C2)C)cc2c(F)cccc2[nH]1 c1(C(N2CC=C(CNC(c3c(C)scc3)=O)CC2)=O)n[nH]c2c1CSCC2 c1(OC)cc(NC(C(C2CCN(C)CC2C)NC(=O)OC(C)(C)C)=O)nc(Br)c1 c1(CN(CCC#C)C(=O)CNC(C)CC)ccncc1 N1(C(c2c(C)cc(O)nc2)=O)CCC2CCCC12C(=O)NCCCN1CCC1 N1(C(CC2(OC)CCC2)=O)CCCC(F)(CNC(=O)Cc2ccc(C)cc2)C1 CCC(CC(=O)N1CC2CC1CN(C(=O)C(C)SC)C2)C(C)C CC(CCNC(=O)CC(C)NC(c1ccc(C2CC2)o1)=O)C(F)F c1(C(=O)NC(CNC(C(CC=C)OC)=O)(C)C)nc(OC)ccc1C CCC(CC(=O)NC1CC(CO)N(C(=O)CC2(C)OCCO2)C1)C(C)C c1(C(N2CC(CNC(CN(C(C)C)C)=O)C(C)C2)=O)cc(F)c(F)cc1F C1(CN(C(COCc2c(C)ncs2)=O)CC)CCN(C(=O)CCC(C)C)CC1C N1(C(c2c(CC)nc(C)s2)=O)CCN(C)C(CNC(=O)C(F)C2CCC2)C1 C(C(=O)N(C1CCN(C(=O)C(C2(C#N)CCC2)=O)C1)C)(C(C)C)CCC#C C12(CNC(=NCc3ccc(OC)cc3)NC3CC(SC)C3)CCC(C1)C(C)(C)O2 C#CC1(O)CN(C(C2CSCN2C(c2coc(C(C)C)n2)=O)=O)C1 C1(OC)CC2(C1)CC(NC(C1CN(C(=O)CSC(C)C)CC1C(C)C)=O)C2 N#Cc1c(Br)cccc1S(=O)(=O)Nc1cccc2c1ccn2CC(=O)O C12(CCSC1)C(=O)N2.C1(CCNC(C2CCCN2C2CC2)=O)CCCOC1 C#CCCC(O)C(=O)N1CCC(CNC(c2ccncc2Br)=O)(OC)C1 C#CC1(C(N2CC(O)(CCNC(=O)Cc3cnccc3C)C2)=O)CCCC1 n1(CC)nc(C)c(NC(=O)CC(CC)S)c1C.C(C)(C)(C)OC(=O)NCCS N1(C(C(C)=CC(C)(C)C)=O)CC(C)CC1C(=O)NCC(C)(C)C#N c1(CC(=O)N(CCNC(CSC(C)C)=O)C(C)C)cnn2c1OCCC2 C(=O)(C1=CC2CCCCCCC12)N1CC(CNC(CCNC(=O)C=CCl)=O)C1 C(=O)(C(F)(F)C1CC1)NC(CNC(CCN(CCCCC)C)=O)C N1(C(COCC)=O)CCN(C(C2CCCOC2C)=O)C(c2cccc(Cl)c2)C1 C1(NC(c2c(OC)cccc2)=O)CC12CCN(C(=O)Cc1cc(C)no1)C2 C1(CC)CC(C(=O)NCC2(F)CN(C(C3CCCCCC3)=O)C2)CC(=O)N1 c1(CCC(=O)NC2C(NC(C(C=C)c3ccccc3)=O)COC2)ccnc(C)n1 Cc1ccn(C)c1C(=O)NC(C)CCN(C)C(C1CCS(=O)(=O)N1)=O S(=O)(=O)(c1cccc(=NCc2ccco2)[nH]1)NCc1scc(C(N)=O)n1 C=CC1(CC(N2CCC(COCC)CC2)=O)CN(C(=O)CC2CC2)C1 Cc1ccc2c(CC(C)NC(c3ccc(OC(C)C)nc3)=O)c[nH]c2c1 C1(CNC(c2ccc(OCF)cc2)=O)CCCCCN1C(=O)Cn1nnc(=O)[nH]1 C(C)(N=c1nc2scnc2c(NC(c2ccc(Cl)c(Cl)c2)C)[nH]1)c1nnc(C)s1 N1(C(CC2CCC(=O)N2)=O)CC2(NC(c3ccnnc3)=O)CCC1C2 N1(C(c2c(CC)cno2)=O)CCC2CC12C(=O)N(CCOC)CC C(=O)(CC1=CCCCC1)N1CCC(CN(C(C(C)N(C)C)=O)C)C1 C(=O)(CCCC(N)=O)NCCOC1CN(C(C(CC)C)=O)C1 C(=O)(CS(=O)(=O)C1CC1)NCC1(CNC(C(C2CCCOC2)OC)=O)CCC1 CCC(CC)CCC(=O)N1C(C)C2CC1C2NC(=O)Cn1ccnc1C(C)C C12(CNC(CCOC)=O)CCCC(CN1C(c1ccccc1CS(C)(=O)=O)=O)C2 C1(CNC(C2ON=C(C(C)C)C2)=O)(NC(=O)C=CCO)CC2CCC1CC2 N1(C(C2C(C)C2)=O)CCc2sccc2C1CNC(=O)CCc1ccnc(Cl)c1 C(=O)(CCCC(F)(F)CO)N1CCC(CCNC(c2c(C)cc(C)[nH]2)=O)C1 c1(CNC2(NC(C(=O)N(C)C)=O)CCCOC2)cc2cncc(Br)c2o1 C(=O)(C1CCc2ccccc21)N1CC2CC(NC(c3c(Cl)ncc(C)c3)=O)C2C1 C(c1ccc(Br)o1)=C(C)C(=O)NC1CC=CCC1C C(=O)(CCCSC)NCCN(C(C1(SC)CC1)=O)CC CCCCC(O)C(=O)N1CCOC(C(C)NC(=O)CNc2ccc(Cl)cc2)C1 C1(NC(c2cn(C)c(=O)n2C)=O)CCCCC12CCN(c1cncc(Cl)n1)CC2 N1(C(C(N2CCOCC2)C)=O)CCOCC1CC(=O)Nc1cccc(CO)c1 CC(C(=O)NCCCOCCNC(C1CSC1)=O)NC(N)=O S(=O)(=O)(c1nc(N(CC(C2CCCCC2)(C)C)C)ccc1Br)NCC1CN(C)C1 C1(C2(O)CCN(C(=O)CC3CCCN3CC)CC2)(NC(C=CCCC)=O)CC1 c1(C(N2CCN(C(N3CCN(C(N(C)C)=O)CC3)=O)CC2)=O)cc(Cl)ccc1I CCCCC(CC)C(=O)N(C1CCCN(C(=O)CCn2cnnn2)CC1)C N1(C(C(CSC)C)=O)CCC(CNC(C2CCCN2C)=O)C(F)(F)CC1 C1(C(=O)NCCOC(C)C)CC(O)CN1C(=O)Cc1cn(C)nn1 N1(C(C2CCCC2(F)F)=O)CC(S(=O)(=O)N2CCN(C(C3CC3(F)F)=O)CC2)C1 CC1CC(C(=O)N(C)CCN2CCN(C(=O)C=C3CCCCC3)CC2)CC(C)C1 CCCC(C#N)C(=O)N1CC(O)CC1CNC(=O)COCCCF N1(C(C(C(C)O)N(C)C)=O)CCCCCC1C(=O)N(C1CC(C(N)=O)C1)C c1(C(CCC)=O)ccc(OCC(=O)Nc2cnn(C)c2-c2cn(CC)nn2)cc1 C1(C(N2CCN(CC(C)NC(c3n(C=C)ncc3)=O)CC2)=O)CC2C(C1)C2(F)F N1(C(C2(CSC)CC(F)(F)C2)=O)CCCC(CO)(NC(=O)C(C)n2cncn2)C1 c1(C(=O)NC(C2CCN(C(c3c(CC)cco3)=O)C2)C)cc(CC)c(=O)n(C)c1 C1(CCOC)(NC(c2csnn2)=O)CCN(C(=O)CC(C)F)C1 C(CN=C(NCc1ccc(Cl)o1)NC1CCS(=O)(=O)C1)c1cc(C)sc1C S(=O)(=O)(c1cc2sc(=NC(C)C3CCC3)[nH]c2cc1Cl)N1CCC(C(C)C)CC1 N1(C(Cc2c(C)noc2C)=O)CCC(C2CC(NC(C3(O)CCSC3)=O)C2)CC1 c1(OC)nc(C)ccc1C(=O)NCCCCCCNC(C1(CO)CC1)=O c1(NCC)ccc(C)cc1C(N1CC(NC(=O)CS(=O)CC)CC(F)C1)=O CC(C)CC(C(=O)NCc1cnco1)NC(=O)CCC1CC1C N1(C(c2cccc(OC)c2O)=O)CCC2C1CCN2C(=O)CNC(=O)O C(C(C)C(C)C(=O)N(CC(=O)NCC(C)(C)c1cccs1)C(C)(C)C)OC CCCCC(C(=O)NC1CCN(C)CC1C)NC(=O)CCCCC1CC1 Cc1cccc(C)c1-n1nnnc1C(C1CC1(Br)Br)NCc1csc(C)c1C c1(C(N2C(CNC(C3N(C)CCOC3)=O)CC2)=O)cc(S(N)(=O)=O)ccc1Cl CC1=C(C)CN(c2nnc(-c3ccc(OC(F)F)cc3)n2C)CC1 C1(N(C)C)CCCN(C(C2(NC(C3SCCS3)=O)CC(CO)C2)=O)CC1 c1(C(=O)NCC2(C)CCN(C(C3CCN(C)C3)=O)C2)cc(O)nc2c1CCCC2 c1(CNC(=O)NCC(C)NC(c2ccc(C(C)=O)o2)=O)cc2c(s1)CCC2 C12(CO)CCCN(C1)C(=O)OC2.n1(COC)nccc1C(=O)OC(C)(C)C C(c1ccccc1)=CCC(=O)NCC(C(=O)NC(c1cccs1)CC)C Cc1cccc(C(F)C(=O)NCC2(CNC(C3CCSC3)=O)CC(F)(F)C2)c1 CCC(CN(C)C)CC(=O)NC1C2CN(C(C3(COC)CC=CC3)=O)CC12 c1(C(=O)NC(Cn2cc(C(CC)N(C)C)nn2)C)ccc(OC(F)F)c(O)c1 C(CCN(C)C(c1cc(-c2ccccc2)nn1C)=O)(C(C)C)NC(C(F)OC)=O C(=O)(C(F)CC(C)(C)OC)NCC(C(=O)Nc1cnc(F)cc1C)OC c1(OC)cccnc1C(F)(F)C(=O)NCC1CC1(C)c1cccs1 c1(C(c2n(CC(=C)C)nnn2)NCCc2ocnc2CO)ccc2c(c1)CCC2 C(C(=O)NNC(=O)Nc1ccc(OCCO)cc1)C1CC(OCC)C1 c1(C(=O)NC2CCCCN(C(COCCOCC#C)=O)C2)cc(C)c(Cl)cc1F N1(C(c2ncn(C)c2C(F)(F)F)=O)CC2CCN(C(=O)CNC(N)=O)C2C1 C#CCCC(C(=O)NC1(CCF)CC(O)C1)NC(=O)CCC(C)N(C)C C1(C2(C=C)CCC2)(C(N2CC(C=C)C(NC(=O)C(C3CC3)SC)C2)=O)CCC1 c1(OC(C(=O)NCCC(CNC(C(CC)C)=O)O)(C)C)cccc(C(C)C)c1 C1(C(=O)NC(CNC(C(C)SCC)=O)(CC)CC)CCC2(CCC2)C1 c1(C(N2CC3C(NC(c4ccc(F)cc4F)=O)C3C2)=O)cc(Cl)cc2cc[nH]c12 N1(C(COC)(C)C)CCN(C(=NCCSC)NCc2cnc3n2CCOC3)CC1 n1(C2CN(C(=O)OC(C)(C)C)C2)cc(CN(CCCO)C2CC2)nn1 C1(CC(N2CC(NC(CNC(CC)=O)=O)(CC)C2)=O)CCCCN1C CC1CN(C(=O)CC(O)CN(C)C)CCN(C(C2CCCCC2N=[N+]=[N-])=O)C1 C1CCC(CCC)NC(=O)C(CCC)OC(=O)C=CO1.CCCCCCCOC N1(C(c2ncn(C(C)C)c2)=O)CCN(C(C2CC(O)CN2C)=O)CC2(CC2)C1 C=CC(C)(O)CC(=O)N(CCC(C(C)(C)C)NC(=O)C=Cc1ccc(C)cc1)C C1(NC(C(C)OCC=C)=O)(CNC(=O)C=Cc2cnc[nH]2)CCC(C)(C)CC1 Cc1cc(C(=O)NC2(C)CC(NC(c3coc(C(F)F)c3)=O)C2)n2ncnc2n1 C1(NC(C)=O)CCN(C(=O)CC(c2cccs2)NC(C23CCCC2C3)=O)C1 c1(OC)ccccc1CCNC(=O)NC1CCC(c2ccccc2)C1 C1(CNC(CP(C)(C)=O)=O)CN(C(=O)Cc2ccc(O)cc2Cl)CC1(C)C CC(C)(C)C(C(=O)N1CCCC(NC(=O)C=CC2CC2)CC1)C1CCCC1 C1(NC(C(C)NC(c2ccco2)=O)=O)CCC(NC(C2CN(C)C2)=O)C1 c1(CN2CCC(CNC(c3cccnc3)=O)C2)cccc2cccnc12 C#Cc1ccc(OCC(=O)N(CCNC(=O)CCc2cnc[nH]2)CCOC)cc1 C1(C(N(CC)CC2CCCCO2)=O)CC2CC2N1C(c1cc(CO)[nH]n1)=O c1(N(CC(C)N(C(C)=O)C)C)nc2ccsc2c(=NCc2cn3ccsc3n2)[nH]1 C(=O)(C(C)(O)C(F)(F)F)NC1CN(C(c2c(OCCC)cccc2)=O)C1 c1(C(=O)NC(C)CN(C)C(C2OC(C)(C)OC2(C)C)=O)cnn2c(=O)cc[nH]c12 Cc1cc(C(=O)NC2CCOC(CNC(C3C4CCCC34)=O)C2)ccc1C(C)C C1(C(NOCC=C)=O)C=CCN(C(=O)CC(C)(C)OC)C1 N1(C(=O)COC2CCOCC2)CCC2CC1CN(C(C1(CCF)CCC1)=O)C2 C1(C(N2CC(NC(CCCC(=C)C)=O)C(C)(C)CC2)=O)CCN(S(N)(=O)=O)CC1 CC1=CCC(NC(=O)CCC2CCCN2C(=O)C#CC2CC2)CC1 N1(C(=O)NCC2C3COCC23)CCCc2c(F)c(F)cc(F)c21 c1(COC)ccc(C(=O)N(CCCCN(C(=O)CN2CC3CC3C2)C)C)cc1 Cc1ccc(-c2cc(C(=O)NCCCC(C)NC(c3cncs3)=O)n[nH]2)c(C)c1 N1(Cc2cccc(CCC=C)c2)C(=O)NC(c2ncc[nH]2)C1=O N1(C(C(=O)NC(CC#C)CC)=O)CCCC(O)(C(C)C)C1 C12(C(=O)NCC(C)NC(c3c(OC)noc3C)=O)CC3CC(F)(C1)CC(F)(C3)C2 C(=O)(C1=CN=C2N=CNN2C1)N1CCC(CNC(C2CC=CCC2)=O)C1 N1(C(c2nccn2C)C)CCC(CN)CC1.C(=O)(CCSC)C(=O)CO c1(C(N2CC(C(C(=O)NC(COCCOC)C)OC)C2)=O)ncnn1C1CC1 C1(C(=O)NCC(C)(CO)NC(C2(C(F)(F)F)CC(F)(F)C2)=O)CCCCCC1 CCCCC(F)C(=O)NC(Cc1cn[nH]c1)C(=O)N(C(C)CC(=O)OC)C c1(C(N(CCCNC(C(CCC)NC(N)=O)=O)C(C)C)=O)ncc2n1CCCC2 C1(NC(c2c(C)cc(C)s2)=O)CS(=O)(=O)CC1NC(=O)CN1CC=CC1 Cc1coc(C2CC2)c1C(N1CC(NC(C2NC(=O)OC2C)=O)C(C)C1)=O CCC(F)(F)CC(=O)NC(C)(CNC(=O)CC1CCC(C)CC1)C1CC1 C1(C(N2C(C)CC(CNC(=O)Cc3nnc(O)s3)C2)=O)C(C)(C)CCCC1(C)C C1(C(=O)NCC2CC23CC3)CC2(CCN1C(=O)CCc1ccco1)CC2 C1(C)(C(N(CCOCCCNC(C2CC(SC)C2)=O)C)=O)C=CCC1 c1(C(=O)NC2CN(C(C3N(CC)C(=O)CC3)=O)CC2C)csc2cncn12 C1(NC(C2C(OC)CC2)=O)CCN(C(c2ccc(C(F)(F)F)o2)=O)CC1(C)C n1(CC(=O)N(C2CCN(C(c3n[nH]cc3C)=O)C2)CCC)cc2ncccc2n1 CCC(C)CCCC(=O)N(CCNC(C1OCC2CCCC1C2)=O)CC c1(OC(C)C)ccc(C(=O)NC2(CNC(=O)Cc3cnnn3C)CCCC2)cc1 C1(NC(Cc2cc(C)no2)=O)CCCC(N(C(=O)CCCF)C)C1 CC(C)C(C)C(C)CC(=O)N1CCN(C(=O)CC(C)(C)C)CC1c1cccnc1 CCCCC(C(=O)NC(CC(=O)N(C)Cc1cc(C)nn1C)C(C)(C)C)C(C)C C1(C(N(C2CCN(C(c3cnc(C)c(N)c3)=O)C2)CC)=O)CC2CC(C1)C(=O)N2 C(=O)(CCCN(C)C(C1CCCO1)=O)NC(c1ncc[nH]1)C C(=O)(C1CCCc2nc[nH]c21)NC1CCC(C)N(C(c2cnc(C3CC3)o2)=O)C1 C1(C(=O)NCC2CN(C(C#CC3(C)CC3)=O)C2)Cc2cccc(F)c2O1 c1(C(CO)NC(C2(C)CN(C(C3CC3C3CC3)=O)C2)=O)cccc(F)c1 NS(=O)(=O)c1cc(C(=O)NC2CCCC2CNC(c2csnn2)=O)cs1 c1(C(=O)NCC(CNC(C(C)SC)=O)(C)C)c(N)c(F)cc(F)c1F c1(C(N2C(CNC(C(C)O)=O)C=CC2)=O)ccc2ccccc2c1F N1(C(C(=CC2CCCC2)C)=O)CC2CC2(CNC(c2nc(C)oc2C)=O)C1 N1(C(C2(C)C(C)C2)=O)CCC2(C(=O)NC(c3ccc(O)cc3)CO)CC2C1 C1(OC)CN(C)C(C)(C(=O)N(C(CNC(c2nc(Cl)sc2C)=O)C2CC2)C)C1 c1(OCC=C)ccc(C(=O)NCCC(C)NC(=O)OC(C)(C)C)cc1 c1(CC(=O)NC(CC)(C)CNC(=O)CCN(CCO)CCO)cc(Cl)n(C)n1 Cc1ccc(CN(C)Cc2c(C)nn(C)c2-n2cccn2)cc1Br C1(C(N(C(CN(C(Cc2c(C)cccc2)=O)C)C)C)=O)Cc2ccccc2O1 N1(C(C2CC(CNC(C(CC)=CC)=O)C2)=O)CCCCC1C(C)(C)C C12(CNC(c3cc(C)c(C)o3)=O)CCC1CN(C(=O)C(F)(F)CN(C)C)C2 c1(COC)cccc(C(=O)NCC#CCNC(c2ccncc2Cl)=O)c1C c1(OC)cccc2c1CN(C(C1Cc3cccc(F)c3O1)=O)CC(C)(C)O2 c1(NC2CCC(N(C(C(C(C)O)(F)F)=O)C)CC2)ncnc2c1CCC2 c1(C(=O)NC(C)CNC(=O)CCc2ccc(F)nc2)cccc2c(C#N)c[nH]c12 c1(C(=O)NCC(CO)NC(C2N(CCC)CCC2)=O)cnn(C)c1N C(C(C)CN=c1cc(C)nc(CCC2CC2)[nH]1)NC(C(C(CC)CC)C)=O C=CCCCCCC(=O)N1CC(=O)NCC1C(=O)NCCC(C)C(C)C N1(CC(=O)N(C2CCCC2)CCNC(c2cocc2C(N)=O)=O)CCSCC1 c1(C(N(C2CCN(c3nc(C4CC4)ns3)CC2(C)C)C)=O)ccc2nn[nH]c2n1 N1(C(C2CN(CC)C(=O)C2)=O)CCCCC(NC(=O)C(F)F)C1 c1(C(N2C3CN(C(c4c(OC)cnnc4)=O)C(C3)C2)=O)c(C)ccc(C)c1C CCCCC(C(=O)NC1CN(C(c2ccc(O)cc2O)=O)CCC1C)C(C)C C1(C(=O)NCC2(S(N)(=O)=O)CC2)(NC(CC(C)C)=O)CCc2cc(Br)ccc2C1 CC(C)C(F)C(=O)NCC(C)(C)CNC(=O)Cc1ccc(Cl)cc1 C12(CNC(CSc3nc(C)[nH]n3)=O)CN(C(=O)CN(C)C(N)=O)CC1CCO2 C1(NC(Cc2c(C)n(C)nc2)=O)CCN(C(c2cc(N)ccn2)=O)CCC1CO C1(C(N2C3CN(C(C4CCCN(C(C)C)C4)=O)C(C3)C2)=O)CN2CCN1CC2C C(=O)(CS(=O)c1ccc(Cl)cc1)N(C1CCN(C(=O)C#CC2CCC2)CC1)C N1(C(Cc2nc(C)[nH]n2)=O)CCC(F)(F)C(C(=O)CCNc2ccccc2Cl)C1 Cc1ccc(F)c(OCC(N2CCCOC(CNC(c3ccsc3C)=O)C2)=O)c1 N1(C(C(CC)(C)OC)=O)CCOC2(CCC(NC(c3cc(OC)ns3)=O)CC2)C1 c1(C(N2CCCC(N(C(=O)CC3(COC)CC3)CC)C2)=O)c[nH]c2ncccc12 N1(C(c2onc(C)n2)=O)CCC2(CC1)CC2C(N1CCC2(CCOC2)C1)=O c1(C(=O)NC(C)C(C)NC(c2sccc2CN(C)C)=O)cccc(O)c1F c1(C(=O)NC2CC(CCNC(Cc3c(C)n[nH]c3)=O)C2)ccc2c(c1)C(=O)OC2 c1(OC)cc(C(N2CC(CNC(c3ncnn3C)=O)CC2C)=O)nn1C O(NC(=O)C=Cc1nccs1)CC(=O)NCCNC(=O)C1CC1 C1(CC(N2C(CNC(=O)CN(C3CCSC3)C)CC3CC23)=O)(OC)CCCCC1 N1(C(CC2(C)CN(C(N)=O)CCO2)=O)CCOC2CC(NOC(=O)OC(C)(C)C)CC12 N1(C(C2(C)CCC2)=O)CC2CN(C(c3ccc(CC#N)cc3)=O)CC2C1 C1(C(N(C2CC3(CC3)C2)C)=O)N(C(C2CC2C2(C)COC2)=O)CCCC1(C)C C(=O)(C1COCc2ccccc21)NCC1(CNC(c2cc(C)sc2)=O)CCC1 c1(C(=O)NCc2nnn(C)c2C(N2CCC(CC(F)F)C2)=O)cccc(F)c1O n1(CCC(=O)NC2CCOC2c2ccco2)cc(-c2nccs2)nn1.N1CCOCC1 C1(NC(Cn2c(C)ccn2)=O)CCN(C(=O)CC(O)CN(C)C)CC(C)(C)C1 C(C)(C)(CC(=O)NCC1(F)CN(C(=O)CSc2cccc(Cl)c2)C1)N(C)C CC1(NC(c2ncccc2Cl)=O)CCN(C(C2(C)CC=CCC2)=O)CC1 CCCC(CC)CCC(=O)NC1(C(=O)NCc2cnn(C)c2)CCCC1 C12(CNC(C3C(=C)CC3)=O)CCCC1N(C(C1CC=CC1)=O)CCC2 C1(CCNC(C(c2cccc(Cl)c2)(C)C)=O)COCCN1CCOCC(F)(F)F Cc1cc(=NC2CCN(CC(N)=O)CC2)[nH]c(N2CC(C)OCC(C)(C)C2)n1 C1(C)(CNS(C)(=O)=O)CCCS1(=O)=O.n12cc(nn1)C(CC(N)=O)NC(=O)C2C C1(NC(c2c(C)nc(CO)s2)=O)CCN(C(c2c(C)nc(C)n2O)=O)C1(C)C c1(C(=O)NCC(C2CCN(C(C3(SC)CC3)=O)CC2)F)ccc(C)c(Cl)c1 c1(CC(N2CC3C(NC(C4C(F)(C(=O)OC)C4)=O)C3C2)=O)ncn2c1CCCC2 c1(C(=O)NCC(C)(C)NC(C(C)SC)=O)cc(C)c2ncccc2c1C c1(C(=O)NC2CN(C(C(CC)F)=O)CC2F)cc(S(=O)(=O)NC2CCC2)c[nH]1 c1(NC(c2ccc(OC(F)(F)C(F)Cl)cn2)=O)cccc(F)n1 N1(C(=O)Nc2cc(C(=O)OC)nnc2C2CC2)CCC(C2CCOCC2)C1 c1(C(C(=O)NC2(C=C)CC2)N(C(=O)OC(C)(C)C)CC)ccccc1F C1(NC(c2c(CC)cccc2)=O)CCN(C(=O)CC2(C)CC2(Cl)Cl)CC1F N1(C(C(CCC)C(C)C)=O)CCC2CN(C(C3CC(C)OC3C)=O)CC2CC1 C(C)(C(CCC(=O)O)CCCC(=O)O)NC(CC(=O)OC)C(=O)N1CCN(C)CC1 CCC(C)(CC(=O)N1CCC(CN(C)C(c2cc(C)no2)=O)CC1)C(=O)OC N1(C(CCCc2[nH]c(=N)sc2)=O)CCCC(CNC(C2CC3(CC3)CO2)=O)CC1 N1(C(Cn2nc(C)c(Cl)c2)=O)C2CCCC1CN(C(c1cc(=O)cc[nH]1)=O)C2 c1(C(=O)NC2CC(N(C(CCC=CC(C)C)=O)C)C2)cc(Cl)c(Br)[nH]1 C(=O)(C(O)C(F)(F)c1ccccc1)NC(C)(C)Cn1cc(CCOCCO)nn1 C1(CNC(CN(C(=O)C2=CCCC2)C)=O)CCCC(F)C1 C1(C(=O)NC2(CCC(=O)N3CC(c4ccncc4)C3)CCC2)CC12CCOC2 N1(C(c2cc(OC)ccc2Cl)C(=O)NCCCC)CCCC(O)(COC)CC1 C(C(C(C)(C)C)NC(=O)NC(Cc1ccnnc1)=O)NC(=O)OC(C)(C)C C1(CC(=O)NC2CC(CCC(=O)NCc3n(C(C)C)ccn3)C2)CCCC(=O)N1 C1(CC(=O)N(C2CCC(NC(c3sccc3C3CC3)=O)CC2)C)CCCCCO1 CC1CC(NC(C2CC2C)=O)CN(C(c2cnn(CC(F)(F)F)c2)=O)C1 c1(C(=O)NC2C(NC(C(c3c(C)noc3C)C)=O)COCC2)cccc(Cl)c1F N1(C(CCC)=O)CCC(C(F)CNC(c2ncoc2Br)=O)CC1 N1(Cc2n(C(C)C)nnc2)CCc2cc(F)cc(F)c2C1 N1(C(C2(CC)CCC2)=O)CCCCC(N(C)C(c2cc(C)cs2)=O)C1 C1(NC(C2C(C=C)C2)=O)CCC(C)(CNC(c2cccnc2N(C)C)=O)CC1 C1(CCC)(NCCOC)CN(C(=O)C=CCF)C1.C1CO1.C1COCCO1 c1(C(=O)NCC2(NC(CCN(CCCCOC)C)=O)CCC2)n[nH]cc1[N+](=O)[O-] c1(OCOC)ccc(CNC2CN(C(c3ccsc3C)=O)CC2C)cc1 c1(OCC)cc(C(=O)NC(C)(CNC(=O)C(C2CCCC2)OC)CC)[nH]n1 c1(CCC)n[nH]cc1C(=O)NCc1cc(C(=O)N(CCCO)CCCO)cs1 n1(CC(=O)NC2CN(C(C(CC)F)=O)CC(C)C2)c(C)nc2ccccc2c1=O c1(CC)nn(C)c(C(N2CCC(NC(c3cc(CC)c[nH]3)=O)C(F)C2)=O)c1Cl C1(C2(C(=O)N(c3ccsn3)CCO)CC2)CCCN1C(c1ccsc1Br)=O c1(CN(C(c2cccc(Cl)c2Cl)C(=O)NC)C)ccc(C(C)C)c(F)c1 c1(OC2C(C#N)CCC2)cccc2c(Cl)c(Cl)sc12 Cc1nnc2n1CC(C(N1CCC(CNC(c3csc4nccn34)=O)CC1)=O)C2 C1(CNC(=O)CC2C=CCC2)CC2CCCCC2N1C(c1ccnn1C(F)F)=O c1(C(N(C2CC2)CC2C(C)C=C(C)CC2)=O)occc1C1=CCNCC1 c1(C(=O)NC2CCCN(CC(=O)NCC3CCCO3)C2=O)cc(F)cc(F)c1O c1(COC)c(C)csc1NC(C1C2CN(Cc3ccccc3OC)CC12)=O c1(C(=O)NC2CCN(C(c3cnn(C)c3Br)=O)C2)ccc2c(c1)CCC=C2 c1(C(C)C)cc(C(=O)NC(C(C)NC(c2cccc(Cl)c2)=O)C(C)C)ccc1F c1(CNC(C2(C)CCCN(C(=O)CN3CCCCC3)C2)=O)ccc2c[nH]nc2c1 Cc1cc(=O)c(C(=O)N(C2CCN(C(=O)CSC3CC3)C2)CCO)cn1C1CC1 c1(CN2CCC(NC(c3cnco3)C)C2C)cccc([N+](=O)[O-])c1 C1(C(N2CCOC(C(F)(F)F)C2)=O)CN(Cc2c(Br)ccnc2Cl)CCC1(F)F c1(C(=O)NCC(C)N(C(=O)CC2CC2c2cnc[nH]2)C)ccccc1CC#N CC1CCCCC1(C)C(N1CC(C)(NC(=O)CCC(=O)c2cccc(N)c2)C1)=O N1(C(c2n[nH]c(C(C)C)c2Br)=O)CC2CC(NC(=O)CC3(N(C)C)CC3)C1C2 c1(OCC(=O)NCC(CCCC)NC(C2C(C)C2C)=O)ccc(C)cc1OCC c1(OC)cc(F)ccc1CC1CCCN(C(c2cnccc2N(C)C)=O)CC1 C1(NC(COC(CC)CC)=O)CCN(C(=O)CN2CC(C)C2)CCC1CO N1(C(C2CC(CN(C)C)C2)=O)CCOC(CNC(=O)Cc2cncn2C)C1 N1(C(C(C(C)C)SCC)=O)CCCCCC(NC(c2cn(C3CCC3)nn2)=O)C1 C1(C(=O)NCc2cc(C(=O)NC(C)C(N)=O)n[nH]2)CCCC(CF)C1 Cc1nccc(Br)c1NC(c1ccnc(CNC(=O)C=Cc2cnccn2)c1)=O C1(C(=O)NC2(CN(C(=O)C(F)OC(F)(F)F)C)CC2)C2CC3C(C2)C13 C=CCC(C)(C(F)F)NC(=O)CCC1CC(NC(=O)C(C)CC=CC)C1 c1(C(=O)NC(C)CNC(c2cnn(CC(F)(F)F)n2)=O)c(F)ccc2c1OCC2 C(=O)(C(O)CC(F)F)NC1C(NC(c2ccc(CCC)s2)=O)COCC1 c1(SCC)ccccc1C(=O)NCC(C(C)C)NC(=O)CCCC1CC1 Cc1nnc(C(=O)NCC2CC(F)(CNC(=O)C=C3CCSCC3)C2)s1 c1(OC)ccc(CC(=O)N(CCN(C(=O)Cc2csnn2)C)C(C)C)nc1 Cc1ccc(Br)c(F)c1C(N1CCCC1C(=O)Nc1c(Cl)cccc1C#N)=O CC1N(C(C2COC3(C2)CN(C(=O)CC(O)C(F)(F)F)C3)=O)CCCC12CCC2 c1(C(N)=O)ccc(C(N2CC(O)(CCNC(C3COCCO3)=O)C2)=O)[nH]1 O=C(CCS(=O)(=O)C(F)(F)F)NC1C=CCN(C(c2nn(C(F)F)cc2Cl)=O)C1 c1(CNC(=O)C(c2cccc(F)c2Br)F)cc2c(o1)CCCC2 C1(C(=O)NC2(CC=CC(=O)NC3C(C)CC3)CCC2)CNC(=O)N1 CCC(C)(COCc1ccccc1)C=O.C1(COC)CCN(c2ccccc2)C1 c1(CC(=O)NC2CCN(C(=O)CC3CCC(O)C3)C2)c[nH]c2cc(Br)ccc12 C(=O)(CC1=CCCC1)N(C1CCCCN(C(=O)C(c2ccc(F)c(F)c2)=O)C1)C c1(C(=O)NC2CC(CNC(c3cc(C)nnc3)=O)C2)cc2occc2[nH]1 c1(CSCC(=O)NCCN(C(=O)CC2CCCO2)CCC)ccc(Cl)cc1 CC1=C(C(=O)N2CC(N3CC(NC(c4[nH]c(O)nc4C)=O)CC3=O)C2)CCO1 c1(C(=O)NCCC(=C)CNC(=O)CCOC(C)C)ccncc1C(F)F c1(C(N2CC(CNC(c3nc(OC)oc3)=O)C(C)C2)=O)cc2cnn(C)c2s1 CCCC(C)(C)CC(=O)N1CC(NC(c2cc(C#N)cs2)=O)C(C)C1 c1(NC(C2C(COC)C2)=O)cn(C2CCN(C3(CNc4nccs4)CC3)C2)nn1 c1(C(=O)NC(C(C)NC(c2c(CCC)occ2)=O)C)onc(Br)c1C c1(SC)ccccc1NC(=O)C(CCN(C)C)NC(=O)CCc1ccn(C)n1 Cc1nc(C)c(CC(=O)NCC2(NC(c3c[nH]nc3Cl)=O)CCOC2)s1 CN1CCCCC1C(N1CCCC1C(C)(C)C(=O)NCCOC1CCCC1)=O C(CCN=c1[nH]cc2ccnc-2[nH]1)N(C(c1c(C)coc1C(C)C)=O)CCO C(=O)(C(C)(C)CCCF)N1CCN(CC(C)NC(=O)CN2CC3CC3C2)CC1 N1(C(=O)CCCCc2cnn[nH]2)CCCCC2(CCN(c3nccnc3F)C2)C1 Cc1c(Cl)ncc(F)c1CNCc1cncc(-c2cn[nH]c2)c1 c1(C(N2C(C3CCN(C(C4C(OC)CC4)=O)C3)CCC2)=O)[nH]c(C)cc1C C(=O)(C(O)(C(F)(F)F)C1CC1)NCCN(C(=O)CC1CN(C)CC1O)C C1(N(C(C=NOC)=O)C)CCCC2CN(C(=O)CSC(C)C)CC12 c1(C(N2CCC(CN(C(=O)C=C3CC3)C)C2)=O)csc2ccccc12 C(=O)(C(C(C)C)C(C)C)N(C1(C(=O)NC(C(=O)OC)C)CC1)C C1(C(N(C(C)C)CCNC(C2(C(N)=O)CC2)=O)=O)C2CCC12c1ccccc1 C1(CNC(=O)Cc2ccc(C(F)F)cc2)CN(C(=O)C(O)CC2CC2)CCCO1 C1(CC(=O)NCC(CC)(C)C)CCCN(C(=O)CC2CC=CC2)CC1 N#Cc1cnc(NC(C2CC23CCN(C(C2CC(O)CN2)=O)C3)=O)c(Cl)c1 C(=O)(C(C(=O)N(C)CC1CCCN1C(=O)CCCc1cccs1)C(C)C)OCC c1(CC(N2CC(NC(C(CCSC)O)=O)(CO)C2)=O)c[nH]c2nccc(Cl)c12 N1(C(C2C(NC(CC(=O)OCC)=O)CCCC2)=O)CC2(COC(C)C2)C1 C=C1CCN(C(c2ccc(C)[nH]2)=O)C(C(=O)NC(C(=O)OC)C2CC2)C1 C1(=O)C(OC)CN1.C1(O)(C(C(=O)NC(CC)(C)C)F)CN(C(C)=O)C1 c1(NC(C(=O)NC(CC)CCOC)=O)cc(I)c(Br)cc1C c1(C(N2CC(CN(C(=O)Cc3ccoc3)C)OCC2)=O)cccc2c1OCCC2 Cc1cc(=O)n(C)cc1C(N1CCC(NC(=O)C2=CCCOC2)C(C)(C)C1)=O Cc1cc(=NC(C)CCCO)[nH]c(=NCc2nnc3c(=O)[nH]ccn23)[nH]1 c1(C(N(C)CC2CCN(C(c3c(C)onc3)=O)C2)=O)nccc2c1CNC2=O c1(C(N2CCC(C)(CNC(=O)CCN3CCC3)C2)=O)ccc2cc(F)ccc2n1 C(C)(CO)(C(=O)NCCCC(C)(C)NC(=O)CSc1[nH]c(C)nc1C)NC(C)=O C1(C(N2CCCC(NC(C3CC4CCC(C3)C4)=O)C2)=O)CC2(C1)CC2(F)F Cc1cc(O)cc(O)c1C(=O)NC1(CNC(C2CCCCO2)=O)COC1 C1(NC=O)CCC(F)(F)C1.C(=O)(CCC#N)OC(C)(C)C.C1CCNC(=O)N1C C(=O)(C1=CCCCC1)N1CCC(N(C(c2ccc(CC)s2)=O)CC)CC1 CCC(C)(C)C(c1ccccc1)NC(c1ccc(C2(F)COC2)cc1)=O CCCS(=O)(=O)CC(=O)NC1CC(CCNC(C2CC(=O)NC2(C)C)=O)C1 C1(CC(=O)NCC(C)N(C)C(C2CC23CC(O)C3)=O)CCCOCC1 C(=O)(C1=CCC(C)CC1)NC(CCCNC(C1(CC#C)CCOC1)=O)(C)C N1(C(c2cn(CCC=C)nn2)=O)CCCC(NC(c2cccnc2N)=O)C1CC N1(C(c2cc(N)c(Cl)nc2)=O)CCC2CN(C(=O)CC3CC4C=CC3CC4)C2C1 c1(C(N(C(C)CNC(=O)CC2(O)CCC2)CC)=O)ncnc2c1CCCC2 CC1CC(C(=O)N2CCN(C(c3cnn(CCO)c3)=O)CC2CC2CC2)=NO1 Cc1cocc1C(=O)N(CC(C)CNC(c1c[nH]nc1-c1ccoc1)=O)C CC(CC(C)NC(c1c[nH]nc1I)=O)NC(=O)C(=O)N(C)C c1(C(=O)NC2CC(NC(CC3C=NN(C)C3=O)=O)C(O)C2)cccc(Cl)c1O C(=O)(C#CC(C)(C)CNC(C1(CC)CCCC1O)=O)NC(C=C)C1CC1 c1(CN2CCC(C)(NC(c3coc(C4CC4)n3)=O)CC2)c[nH]c2ccccc12 N1(C(c2ncn(CC)c2)=O)CCOC(C)(CNC(C2CCCCN2C(C)C)=O)C1 C1(C(=O)NCC2(CCC)CCC2)CN(C(c2cnnc(C)c2)=O)CC12CCC2 c1(OC)cc(C)ccc1C(C)Nc1nccc(N(C)CC2CC2)n1 CCC(CC)C(C)C(=O)NCC(C)(C)CNC(C1CCC(O)CN1C)=O c1(C(N2CC3C(CNC(=O)CC4(CO)CC4)C3C2)=O)cc2ncccc2o1 C1(C)(CNC(C(C=C)(F)F)=O)CCN(C(C2CC2c2ccnn2C)=O)CC1 C1(NC(NCc2n(CC)nnc2)=NCCN2CCOCC2)CCCCC12CCC2 C12(NC(C(C(=O)OCC)OC)=O)CCCC(NC(=O)CCCN(C)C)(C1)C2 C(=O)(C1=CC2C=CC(C1)C2)N(CCOCCC(N1CC(C#C)(F)C1)=O)C C1(C)(CC)CC(NC(=O)CCCn2cncn2)CN1C(=O)C=Cc1ccncn1 c1(NC(c2nc(CC(=O)NCC(CN(C)C)OCC)sc2)C)ccc(C)nc1 c1(Cc2cn(C3N(C(N)=O)CC4CCC3CC4)nn2)cccc2cc(F)ccc12 c1(C(N2CC(CNC(C(CCOC)OC)=O)C2)=O)cc(Cl)c(F)cc1C N1(C(CC2(OC)CCCCC2)=O)CC(C)CCC1CNC(=O)CCC(F)(F)F C1(NC2CCC(CC(=O)O)C2)CNCC(F)(F)C1 N1(C(C)(C)CO)CCN(C(=O)C(C2(O)CCC2)NC(c2cccnc2)=O)CC1 c1(CC(=O)NCCC(Cn2cc(C(CC)CC)nn2)(F)F)ccc2occc2c1 c1(C(N2CCC(NC(c3coc(O)n3)=O)CC2)=O)c[nH]c2c(F)cccc12 c1(C(=O)NCC(CNC(c2cc(OC)c(Cl)cc2)=O)(C)O)ncc2[nH]ncc2n1 N1(C(C(C)NC(C)=O)=O)CCCC(O)(CCNC(C2(N(C)C)CCOCC2)=O)C1 N1(C(CSCCCC)=O)CC2(CCN(C(c3ncc(F)cn3)=O)CC2)CC1C CCCC(CC(=O)Nc1ccccc1C)NC(=O)CC1(COC)CC1 N1(CC=C)CCC(N=c2[nH]c3c(c(=NCc4nn(C)cc4Cl)[nH]2)COC3)CC1 c1(SCC(=O)NCCn2cc(C(CC)(C)O)nn2)cc(C)ccc1C O=C(C1CCSc2ccccc21)NC(CNC(C1C2CC3C(C2)C13)=O)C1CCC1 c1(N(C)C)cnccc1C(=O)NC1CC(F)(CNC(=O)CCc2nccn2C)C1 n1(CC(=C)C)nc(-c2cccc(OCC)c2)nc1CC(C)C C1(C(=O)NC2CCN(C(CCC(C)N(C)C)=O)CC2)CCN(C)S1(=O)=O CC(C)C(O)CC(=O)NCC(C1CCN(C(C2(C)CC(F)(F)C2)=O)CC1)C c1(N2C(C(N3CC(NC(c4cnsn4)=O)C3)=O)CCC2)nc2ccccc2s1 CN1C(=O)c2ccccc2C1CC(=O)NCCSC(C)(C)C C1(Cn2cc(C(CC)(C)O)nn2)C(C2CC2)CCN1C(=O)CCSC(F)(F)F NS(=O)(=O)c1cc(C(=O)NCC2(C(N3CCCC(F)C3)=O)CC2)c(O)cc1Cl c1(C(=O)NCC2CC(C)N(C(=O)CCC#N)C2)cccc2nccn12 N1(C(COc2c(C)cccc2)=O)CCC(CNC(C2C(C)C2C)=O)C12CCC2 C1(NC(c2nc(CCC)oc2)=O)COCCN(C(C2(C(=O)C3CC3)CC2)=O)C1 c1(C(C)C)[nH]ccc1C(=O)NCC1(F)CC(NC(=O)CCCc2ccccc2)C1 c1(C(N2CC(NC(c3cnn[nH]3)=O)CC3(C2)CC3)=O)ccc2c(c1)CCC=C2 N=c1nc2cc(C(=O)NCCOC3CN(C(=O)COc4ccccc4)C3)ccn2[nH]1 C(N=c1cc(C)nc(-c2ccccn2)[nH]1)c1ccc(OC)c(C)c1 Cn1c(=O)sc2cc(S(=O)(=O)NCc3cnc(-c4ccccc4)nc3)ccc12 N1(C(c2cc(OC)c(Cl)nc2)=O)CC(C2CCN(C(c3cc(Cl)ncn3)=O)CC2)C1 C1(OC)CC2CCC(C1)N2C(=O)CCCOC1CCC(OC)CC1 N1(C(CCCCC#C)=O)CC(NC(=O)COCC2CCCOC2)C2CCCC2C1 C(c1nc(C)c(C)[nH]1)=CC(=O)NCC1CC(CNC(C2CC(C#C)(O)C2)=O)OC1 C1(NC(C2(NC(c3cccc(CC)c3F)=O)CC2)=O)CCn2nnnc2C1 c1(C(=O)NCC(C)(C)NC(CCCc2n(C)cnn2)=O)cc(Cl)c(Cl)[nH]1 C12(NC(C3(SC)CN(C(C4(C)CCC(=O)CC4)=O)C3)=O)CCCN(CCC1)C2 CC(CC(=O)NC1CC(F)CN(C(=O)CCCc2cc(F)ccc2F)C1)C(F)F C(=O)(C1=CCCCC1)N1CC(COCC)(CNC(=O)CC2(C)CC(F)(F)C2)C1 C=CC(O)C(C)(C)C(=O)N1CCC(O)C(C(=O)NC(C)COCC)C1 c1(C(N2CC(NC(C(CC)OC)=O)C3(C2)CC3)=O)ccc(COC)c([N+](=O)[O-])c1 C(=O)(C1=CC2C=CC1C2)N1CCC(CC)C1C(=O)NOC CCCCC(C)C(=O)NC1CCCN(Cc2cn(Cc3cc(C)on3)nn2)C1 C(=O)(C1=NOC(CNC(C2CC3(CCC3O)C2)=O)C1)NC(C(N)=O)CO c1(C(N2CCC(NC(Cc3c(C)cnn3C)=O)C(O)C2)=O)cc2cccnc2[nH]1 CCCCCCC(CC)(CC)C(=O)OCC1CCNC(=O)CC1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CN(C(C2C(C)C2)=O)CC1N=[N+]=[N-] C1(NC(C(CC)N(CC)CC)=O)CN(C(=O)Cc2nonc2C)CC1C Cc1cc(F)ccc1C(F)(F)C(=O)NCCC(C)NC(c1cc(CF)on1)=O c1(CC(N2CCC(C(C)NC(C3CCCC3F)=O)CC2)=O)nc([N+](=O)[O-])n[nH]1 c1(C(N2C(CNC(C(N)=O)=O)C=CC2)=O)ccc2c(c1)OCC2 N1(C(C#CC(C)C)=O)CCC2(CCCCC2NC(c2cc[nH]n2)=O)C1 N1(C(c2c(C)nn[nH]2)=O)CCCC1(C)C(=O)Nc1cccnc1C(F)(F)F c1(C(=O)NCCN(C(c2ccc(CC)cc2)=O)C2CC2)c2c(nn1C)CCSC2 C(CNC(=O)C(C)NC(=O)CC1C=CCC1)(CC(C)C)NC(CC=C(C)C)=O N1(C(c2[nH]c(CC)c(Cl)n2)=O)CC2CC1CCC2NC(C1(CCO)CC1)=O c1(NC(=O)OC)sc(C)c(C)c1C(N1CC(NC(=O)CC2CCCS2(=O)=O)C1)=O C12(C(=O)NC3(C(=O)OCC)CCC3)CCCC1CN(C(c1n[nH]cc1Cl)=O)C2 n1(CC)cnc(C(=O)NC(C(=O)N(CCC(=O)NC(C)C)C)C2CC2)c1 CC1CN(C(=O)Cc2cn(C)nn2)CCC1Nc1cc(C(C)(C)C)ncn1 N1(C(CCCC)=O)CC(NC(c2nc(-c3ccccc3)oc2C)=O)C2(CCC2)C1 c1(CC)nc(C)c(C(N2CC(F)CC2CNC(=O)C(c2ccccc2)C)=O)o1 c1(C(=O)NC2CCN(C(c3c(C)c(Br)no3)=O)C2)cc2c(nn1)CCCC2 N1(C(c2ccc(NC)cn2)=O)CCC(O)(C(C)NC(c2ncn(C)n2)=O)CC1 C1(CNC(C=CCCC)=O)CC2(CC2)CN1C(C1C2CC3C(C2=O)C13)=O N1(C(C2C(C)SCCC2)=O)CC2(CC(CC(=O)NCC3CCC(=O)NC3)C2)C1 N1(C(C2(Cl)C(CC#C)C2)=O)CC(C=C)(CC(=O)NCC2(CC(=O)OC)CC2)C1 Cc1ccccc1CN1CCN(C(=O)C(=O)NC(C2CC=CCC2)C)CC1 N1(C(C(C2CN(C(c3c[nH]c(=N)o3)=O)C2)OC)=O)CC(COC)C1(C)C c1(CC(=O)NCCC(C)NC(COC)=O)cc(F)cc([N+](=O)[O-])c1 C1(CC(C)CN2CCC(CCN3CCC(F)(F)CC3)CC2)CC2(CC(=O)C2)C1 c1(C(=O)NCC(CNC(Cc2cccc(OCC)c2)=O)O)csc(=NCC=C)[nH]1 c1(C(=O)NCC(=O)NC(C2CCCN2C(C2C(C)C2C)=O)C)cc2ccccc2[nH]1 C(=O)(C(F)C(C)C)N(C(CNC(c1ccn(CCCC)n1)=O)C)CC C1(CCOC)(NC(=O)CCC(F)F)CCN(C(=O)CC2CCC3CC23)CC1 C(=O)(C1=NOCC1)NCCCOCCO.c1(N2CCC(=O)NCC2)ccccc1 c1(CCC(=O)N(CC(C(=O)OCC)O)C2CC2)cc(C)nc(C)c1 C=CCCCC(C(=O)NCC(COC)OC)NC(c1ccc(C(F)F)o1)=O c1(N(CCNC(=O)CSC(F)F)C(C2CCCC2)=O)cccc(Br)c1Cl Cc1cc(C(N2CCOC(C(C)NC(=O)CNS(=O)(=O)C3CC3)C2)=O)cn1C N1(C(c2cc(C)cc(F)c2)=O)CCCC(NC(c2ccn(C)c(=O)c2)=O)C(F)C1 N1(C(c2cc(C)cc(C)n2)=O)C(C)CC2CN(C(=O)C(F)(F)C(O)C3CC3)CC12 C12(NC(=O)COc3cccc(F)c3)COCCC1CN(C(c1nsnc1O)=O)C2 c1(CCCC)cc(C)c(NC(C2CCCN2Cc2cccc(Br)c2)=O)cn1 N1(C(c2ccc(O)nn2)=O)CC2CC(C1)N(C(=O)CCN1CCOC1=O)C2 C1(C)(CC)C=C(C(=O)NCC2(C)CCCN2C(=O)Cc2c(Cl)cnn2C)C1 Cc1nnc2n1CCC(C(N1CC(CNC(=O)CCc3cccnc3)C1)=O)C2 C1(NC(=O)CC2C=CCCC2)CCC(O)CN(C(=O)Cc2csc(C3CC3)n2)C1 C12(C(N3CC(C)N(C(c4ccc(N)cn4)=O)CC3)=O)CCC(CC1)C2(C)C c1(N2C(=O)CC(C(N(CCC)CCc3nccs3)=O)C2)ccc(C)c([N+](=O)[O-])c1 C1(NC(CN(C2CC2)CC)=O)C(C)CN(C(C2(OC)CCC2)=O)CC1C C=C(C)C1OCCCC1C(=O)NCCC(C)N(C(=O)CC12CCC(CC1)CC2)C C1(C(=O)Nc2cnc3cc[nH]c3c2)CCCC12CCN(Cc1ccncc1F)C2 N1(C(COCC)=O)CCC2(CCCN(C(=O)C(c3cnc(O)nc3O)(F)F)C2)C1 Cc1cc(C)c2c(c1)C(N(C)C(c1nccnc1-n1ccnc1)=O)CCO2 C(=O)(C(C)(C)CC1CCOCC1)N1CC(O)(CNC(CC2C(C)OCC2)=O)C1 S(=O)(=O)(c1cccc(N2CCSC3(CCC3)C2)n1)NCC1CCCN(C)C1=O C(=O)(C(CC(N)=O)NC(c1cc(C)cc(O)n1)=O)NC(C(CC)CC)C CN1CCCC12CCN(C(C1CC(F)CN1C(=O)CC1OCCO1)=O)C2 c1(C(=O)NC2COCC(C)(C)NC2)ccc2nc(CCN)[nH]c2c1 c1(CC)nn(C)c(CC)c1C(=O)NC1CCCC1NC(=O)CC1CCN(C)C1 C=C(C)C(C)(O)C(=O)N1CC2(C1)CN(C(c1ccc(C(F)(F)F)nc1C)=O)C2 N1(C(c2c(CC)con2)=O)CCCC(F)(CNC(=O)C=COCC)C1 Cc1nc(NCCC2CC(C)(C)NC2=O)cc(N2CCC(N(C)C)CC2)n1 C(C(=O)N1CCCc2nncn21)N1CCN(C(CC(C)C2CC2)=O)CC1 N1(C(CSC)=O)CCN(C(=O)C(Cc2ccccc2)NC(C)=O)C2CCC12 N1(C(c2ccc(C)s2)C(=O)NCC(C)C)CCOCC1C1CCCO1 c1(C(=O)NCCC2(C)CCN(C(C3(C#N)CC4CC4C3)=O)C2)cc2c(s1)CCC2 C(=O)(C1=COc2ccccc2O1)NC1CC(C)(NC(C(CCC)O)=O)C1 N1(C(=O)NC(C2CCOC2)C)CCn2c(nc3c2CCCCC3)C1 N1(C(c2c(C)ccc(F)c2)=O)CCC(NC(C2(F)CCOC2)=O)CC(C)(C)C1 c1(OCC)cccc(CC(N2CC=CC(NC(=O)CC3(CO)CCCC3)C2)=O)c1 N1(C(C(C)(C)C2CC2)=O)CCC2(CC(NC(=O)C(c3ccc(Cl)s3)=O)C2)C1 CC1(CNC(C2CNC(=O)C2)=O)CCCN1C(c1ccsc1-n1cnnn1)=O Cc1cccc(C(=O)NCC(N2CCN(C(C3(CC(C)C)CC3)=O)CC2)C)c1O N1(C(C(C=C=C)C)=O)CC(=O)NC2CN(C(=O)CCc3nc(C)cs3)CCC12 C1(CCNC(CCCNC(=O)OC)=O)(NC(c2csc(F)c2)=O)CCOCC1 N1(C(CCCN=[N+]=[N-])=O)CC(CO)C2(C1)CN(C(c1nc(=O)cc(N)[nH]1)=O)C2 C1(S(N)(=O)=O)(C(N(CCCN(C)C(C23CCC2C3)=O)Cc2ccccc2)=O)CC1 C1(C)(CNC(CC(COC)NC(C23CCCN2CCC3)=O)=O)CCCCCC1 c1(C(=O)NC(c2ccc(Br)c(Cl)c2)C)n[nH]c2ccc(C#N)cc12 CC1(C)COC(CC(=O)NCC2CCN(C(=O)CCc3cnoc3)CC2)C1 c1(C(=O)NCC2CC(NC(c3n(CC)ncn3)=O)C2(C)C)ccc(C#N)cc1C C1(CC)CCCCC1C(=O)NCCCC(C)NC(c1cnc(C(C)(C)C)nc1)=O c1(C(=O)NCC(CNC(c2cnn(CC)n2)=O)(C)C)cccn2c(C)nnc12 c1(CC)cncc(C(N2CC(C(C(=O)NC(c3[nH]c(C)nc3C)C)OC)C2)=O)c1 N1(C(CN(CCC)C)=O)CCC(NC(=O)C(C)(C)C2CCCO2)C(CC)C1 C1(C(=O)NC(CNC(C(C(C)C)OCC)=O)C)CCc2cc(C)ccc2O1 C=CCC(CC(C)C)C(=O)NCC(C)(C)CC(=O)NC(c1ccnn1CC)C CCC(C)C(C(=O)N1CC2(CC(NC(=O)CN(C(=O)C3CC3)CC)C2)C1)NC(N)=O c1(C(N2CC(NC(Cn3c(C)cc(C)n3)=O)C3(C2)CC3)=O)ccc2c(c1)CCO2 c1(OC)ncccc1CC(=O)NC(C)(C)C(C)NC(=O)C(n1cc(C)cn1)C CCC(F)(F)C(C)(C)C(=O)NC1CCC1CNC(c1[nH]cc2c1CCS2(=O)=O)=O Cn1ncc(C(=O)NCC(C)(C2CC2)NC(=O)C(C2(O)CCCC2)F)n1 C1(NC(c2c(C)cco2)=O)C2CCC1CN(CC(F)(F)F)C2 C1(CC(N2CC(CC(C(=O)NCC(C#C)CC)F)C2)=O)CCCN(C)C1 c1(C(N2CCCC(NC(C3(OC)CCC3)=O)CCC2)=O)nc2cc(F)ccc2s1 c1(C(=O)NC(CNC(C(C)n2ccnn2)=O)C(C)(C)C)ccc(F)c(F)c1O C1(CC(N2C3C(NC(c4c(C)nc(C)[nH]4)=O)CC(C3)C2)=O)CCC2(CCC2)CO1 O=S(=O)(c1ccc(NCCSC(F)F)cc1Cl)NCC(c1ccc(F)cc1)CO c1(C(=O)NCCCN(C(C(COC)(C)O)=O)C)csc2nnsc12 N1(C(C(CC#C)(C)NC(C2C(C#N)C2(C)C)=O)=O)CCC2(CCSC2)C1 c1(CC(=O)NC(C(C)NC(C23OCC(COC)(C2)C3)=O)CO)c(C)cccc1C Cc1cc(C)c(C(N2CCC(O)(CCNC(c3coc(Cl)n3)=O)CC2)=O)cn1 CC1CN2CCCCC2CN1C(=O)CCc1cccc(F)c1Cl c1(SC(C)C(N2CCCCC(NC(C3CC3F)=O)C2)=O)ccc(C#N)cc1 CCCCC(C(=O)NCCNC(=O)CC1C=NN(C)C1=O)C(C)C C1(NC(C(N(C(C(C)=C2CCC2)=O)C)C2CC2)=O)CNC(=O)C1(C)C N#CC1CN(C(=O)CC2(NC(C3C4C5CCC(C5)C34)=O)CCCCC2)CCO1 C(=O)(CCS(=O)(=O)N1CCOCC1)N1CC(NC(C(C=C=C)C)=O)C(O)C1 c1(C(=O)NC2CCC23CN(C(c2nn[nH]c2Cl)=O)C3)ccc2cc[nH]c2c1 CCCC(C1CC1)NC(=O)N(CCC)CC1CC1 CCC(CCOC)C(=O)NC(C1CN(C(c2c(C(F)F)nn(C)c2C)=O)C1)C c1(SCC(=O)NC(CNC(C(c2ccc(OC)cc2)O)=O)C)cc(C)ccc1C C=C=CCCC(=O)NC1CCC1NC(=O)C=CC(C)C C1(N(C(C=CCOC)=O)CCOC)CCN(C(=O)CCc2cnoc2)CC1 N1(C(CC(=C)C)=O)CC2CC1CC2NC(c1nc[nH]c1C(C)(C)C)=O C(=O)(C1=CC2CCCCC12)N(CCCNC(CC(C(=C)C)OCC)=O)CC c1(C(N=c2[nH]n(C)c(Cl)c2)=O)cnc2n[nH]c(C3=COCCC3)c2c1 c1(C(=O)NC2(CNC(C(CC)OC3CCCCC3)=O)CCOC2)cncc(N)n1 c1(C(=O)NCCCCN(C)C(C23CSCC2C3)=O)cnc2sccn12 C(=O)(CCCC(CC)CC)N1CC(C(C(N2CCC(CC=C)C2)=O)OC)C1 C1(C(N2C(C(C)(C)C(=O)NC3CCOC3CC)CCC2)=O)CCCC2(CCC2)C1 C1(NC(C(C)=O)=O)CCCC1CNC(=O)C=C1CCCC1 c1(C(=O)NC2(CNC(CC3C(C)CCO3)=O)CCC2)cc(F)cc2c1NCCC2 c1(C(N2C3(CNC(c4c(C(C)C)ocn4)=O)CC(C2)C3)=O)cc(F)cc(N)c1F c1(C(=O)NCCCCNC(C(C)NC(=O)C(C)(C)C)=O)cnn(C)c1S(N)(=O)=O c1(C(N2CC3C(N(C(c4c(C)nccc4)=O)C)C3C2)=O)cncn(C)c1=O c1(C(=O)NC2C(NC(C3(NC(N)=O)CC3)=O)CC2)ccc(-c2cnccn2)cn1 Brc1ccc2c(c1)C(NC1CCNCCC13CCC3)CCO2 N1(Cc2ncn(C)n2)CC(NC(c2cc(Cl)cc(Br)c2)=O)C(F)(F)C1 C(=O)(C1=NOC(CNC(=O)C=C(C)c2ccccc2)C1)NC(CCCC)COC N1(Cc2c(CC)onc2C)CC2CC1CN2C(c1coc(C(C)C)n1)=O C(=O)(C1CCCc2nccn21)NCC1(C)CCN(C(c2cnnc(O)c2)=O)C1 C1(CC(=O)NC2(C3CCCN3C(=O)Cc3nc[nH]n3)CC2)C=CS(=O)(=O)C1 Cc1ccc(C(N2CCCN(C(c3cscc3C(F)(F)F)=O)CC2)=O)cc1C CC(C)(C)CC(F)C(=O)N1CCC(C)(CNC(=O)C(O)Cn2cncn2)C1 CC1CC(C(N2CC(CF)C2)=O)N1C(c1ccoc1)=O S(=O)(=O)(c1[nH]c(=NC2CCN(C)C2)ccc1Br)NCC1C(C)CCNC1=O C#Cc1cc(C(N2CCCCC2CNC(C2C3CCC(F)(F)C23)=O)=O)cc(F)c1 C(=O)(C(CNC(C1CC=C(C)CC1)=O)C(C)(C)C)NCCS(CC)(=O)=O C1(CC(=O)NCC(C(C)C)NC(c2cc(COC)on2)=O)CCC2CC2C1 CC1(C)CN(C(C2(CF)CC2)=O)CC1CNC(C1CCCNC1=O)=O CC(C)(CC(=O)N(CCC1CC1)CC1CC1)NC(=O)C(F)=CC1CC1 C1(OC)CCC(C(N2CC(F)(C(=O)NOCC(C)(C)O)C2)=O)C1 c1(CC(=O)NC2C(CNC(c3cnc(SC)s3)=O)CCC2)cnn(C)c1C C12(C(N3C4(C(=O)NCCC(C)CO)CC4CC3)=O)CCC(CC1)CC2 n1(CC(=O)NCC2CN(C(C(C)C)=O)C(C)(C)C2)nc2n(c1=O)CCCCC2 c1(OC)ccc(O)c(C(=O)NC2(C3CN(C(=O)C(O)C(F)F)C3)CC2)c1 N(C(=NCCF)N1CCC(c2ncccc2OC)C1)CC(N(CC)OC)=O CC(CN=C(NCC1C=CCC1)NC1CCCC1)Oc1ccc(Br)cc1 c1(C(=O)NCC(CNC(CCC)=O)CO)ccc(-n2ccnc2)c(F)c1 N1(C(CNC(CC)=O)=O)CC(C)(OCC(=O)NC(c2cnn(C)c2)C)C1 C=C(C)C(CC(=O)NCC1CCC(C(=O)NCc2cnccc2Cl)CC1)OCC N1(C(c2c(CC)n(C)nn2)=O)CCCC(C)(CNC(=O)C=CCF)C1 N1(CC(=O)N(C)CCc2ccccc2)CCOC(CCO)C1 c1(C(N2CC(NC(C=CC(CC)=CC)=O)CC2(C)C)=O)cc(S(N)(=O)=O)oc1Cl N1(C(CCOC(C)C)=O)CCC(CO)C(NC(c2nn(C(F)F)cc2Cl)=O)C1 C1(NC(c2ccc(CNC(C)=O)o2)=O)CCCC(CNC(C2CC3(CSC3)C2)=O)C1 c1(C(=O)NC(C(N2CCC(C)(COC)C2)=O)(C)C2CCC2)cc(C)ccc1C N1(C(C(CC(C)C)ONC(c2c(OC)cncc2)=O)=O)C2CCC1CC(=O)NC2 CC(CC(=O)NC(C)(CN(C)C)CO)N(C)C.C1=CC(=O)NC1(C)C c1(C(=O)NC2(CF)CCN(C(C(C(C)C)(C)O)=O)C2)ccc(P(C)(C)=O)nc1 C(=O)(C(C)C(O)CC(C)C)N(C1CN(C(c2sc(C)c(C)c2Br)=O)C1)C c1(C(=O)NCc2ccc(CNC(Cc3cc(C)ns3)=O)cc2)cnc(Cl)cc1N N1(C(=O)CCOCC2CC2)CC2(CCN2C(=O)Cc2ccnn2C2CCCC2)C1 c1(C(C(=O)NCC(=C)C)N(C2CC2)C2CC2)cccc(F)n1 O=C(C(O)C1=CCCCC1)NC1(C(N2CC3CCC2C3)=O)CCSC1 N1(C(C(CC)SC)=O)CCC(C)N(C(=O)CN(C)C(c2ccc(F)cc2)=O)CC1 C1(COC)(NC(c2ccc(OC)nn2)=O)CCN(C(=O)CC2CC3(CC3)CO2)C1 N1(C(Cn2c(C)cc(C)n2)=O)CCN(C)CC1CNC(=O)C#CC(C)(C)O CC1CN(C(c2cc(O)ccc2Br)=O)CCN1C(c1ccc(CO)s1)=O c1(C(=O)NC(CNC(COC)=O)(C)C2CCC2)csc(C(F)F)c1 Cc1c(C(=O)NC2(C)CCN(C(C3COC(=O)O3)=O)CC2)oc2ccc(Cl)cc12 N1(C(c2c(C)noc2)=O)CC2CCC1CN2C(=O)C(C)CC1CCCC1 C1(OC)CC2(C1)CN(C(=O)C(CNC(c1cccnc1C)=O)CC1CCCC1)C2 c1(CC(C(=O)N2CC(CNC(C(C)OCC#C)=O)C2)C)ccc(OC)cc1 N1(C(c2cnc(SC)s2)=O)CCOCC1CN(C(=O)CC1(C)CC1)C Cc1cccc(N)c1C(=O)NC1CCN(C(c2cnn(C3CC3)c2Cl)=O)C(C)C1 C1(NC(C=Cc2n(C)ncc2)=O)COC2(CCCN(C(c3cccs3)=O)C2)C1 C1(N(C(C(c2ccccc2)SC)=O)C)CC2CCC(C1)N2C(=O)C1=CCCO1 CCC(C#N)C(=O)N1CC(N(C)C(c2nn(C)cc2C)=O)C1 Cc1cc(F)c2cc(C(=O)NCCCN(C)C(C3CC3c3ccsc3)=O)[nH]c2c1 N1(C(CCN(C(C)=O)C)=O)CCCN(C(c2nocc2Cl)=O)C(C)C1 c1(C(N(CCNC(c2c(C)csc2)=O)C2CC2)=O)cc(N)ccc1Br N1(C(C(CC(C)C)ONC(C(C)=CCC)=O)=O)CCc2c(C#N)cccc21 Cc1nnccc1C(N1CCCCC1CCNC(=O)CC1CN(C)C1)=O c1(C(C(=O)NCC(=C)C)N(C)Cc2ccc(C)s2)ccc(C(N)=O)cc1 n1(C(C)(C)C)nnnc1C(c1csnn1)NCC1(Br)CC1(F)F c1(N(C(c2c(C(C)C)scn2)=O)C)cc(-n2ccnc2)ncn1.C12CCCN1C2 c1(C(=O)NC2CC(NC(c3cc(OCC)n[nH]3)=O)C2)ccc2cnnn2c1 C1(NC(COCC)=O)CCCCC1CNC(C1(NC(c2ccc[nH]2)=O)CCC1)=O N1(CCN(C(=O)CCCc2cccs2)C)CCN(C(=O)Cc2cnn(C)c2)CC1 c1(C(=O)NC(CCN(C(C(CC)OC)=O)C)C(C)(C)C)cn2cc(C)sc2n1 C1(CNC(c2ccc[nH]2)=O)COCCN(C(=O)CC2C=CCC2)C1 c1(CC(=O)NCC(C)(CO)NC(COCCC)=O)cccc(Cl)c1O.SCC C(=O)(CC(C)(O)COC)NCC(NOCC)=O.C12CCCN(C1)C(=O)C(CC)NC2 CCCC(C#N)C(=O)N1CCCC(CNC(=O)CCn2ccccc2=O)CC1 C1(CNC(C(CC)N(C)C)=O)CC2(CCC2)CN1C(c1cc[nH]c2nccc1-2)=O C1(C(N(C(c2cc(C)on2)C)C)=O)CC12CCN(C(c1cc[nH]c1C)=O)C2 C1(C(N2CCC(C(C)C(=O)N(CCO)CCO)CC2)=O)CCC=CCCC1 Cc1ccc(OC(C)C(=O)NCC2CC(F)(F)CN2C(=O)CC(C)(C)O)c(C)c1 C1(c2ccc(CF)o2)CN(Cc2ccc(OCC(F)(F)F)cc2)CCO1 C=C(C)CCCC(=O)N1CCC=CC1C(=O)NCC=CCl N1(C(C=C(C)C(F)F)=O)CCOC(CN(C(=O)CC2CCC3CC23)C)C1 Nc1c(C(=O)NC2CC(CCNC(=O)C(F)(F)C(O)C3CC3)C2)cc(Cl)cc1F C(c1ccc(Cl)c(Cl)c1)=CC(N1CC(CC(=O)N(C)Cc2cccnc2Cl)C1)=O Cc1cnn(C)c1C(=O)NCCc1cc(C(=O)NCCCCCCO)no1 Cc1cccc(CSCC(=O)NC2CN(C(=O)C(C3CCCCC3)F)CC2O)c1 C1(F)(C(=O)NCCc2c(Br)ccc(C)c2)CC2CCC(C1)N2C(=O)OC(C)(C)C C(=O)(C(O)CCS(C)=O)NC1C2CN(C(CCCOc3cccc(C)c3)=O)C1C2 C1(C(=O)NC2C(C#C)N(C(=O)OC(C)(C)C)CC2)CCn2ncnc2C1 c1(CC(=O)NC(C2CCN(C(C3C(=C)C3)=O)CC2)C)cc(O)cc(Br)c1 C(=O)(C1COc2ccc(Br)cc21)NC1(C)CCN(C(C2(C#C)CCC2)=O)C1 C(C1CCCN1C)=CC(N1CC(CCNC(C(c2cccc(F)c2)C)=O)C1)=O N1(C(C(C2CCCN(C(C(C)(C)SC)=O)C2)C)=O)CCC2(CO)CCCC12 C=CC(C)CC(=O)NC(CCSC)C(=O)NCC1CC(C)(C)C1 c1(N2C3CN(C(c4cc(C)nc(C)n4)=O)C(CC3)C2)nccc(C)c1[N+](=O)[O-] C1(N(C)C(c2cnn(CCNC(=O)Cn3ncnn3)c2)=O)CCOCC1F C(C(C(=O)N1CCCC(NC(c2sc(F)cc2C)=O)CC1)C(C)(C)C)OCC=C c1(NC(c2csc(Cl)n2)=O)cccc2c1CN(C1CC1)C2=O C#Cc1ccc(C(=O)N(C)CC2COCCN2C(=O)CCSCC)c(F)c1 n1(CC)cc([N+](=O)[O-])c(C(N2CC(O)(CNC(c3sc(F)cc3C)=O)C2)=O)n1 c1(C(N2CC3C(NC(C4C(C)(C)COCC4)=O)(C3)C2)=O)csc(S(N)(=O)=O)c1 C(=O)(CCCC(F)(F)F)N(CC(=O)NCC1CCC=CCCC1)CC Cc1ccsc1C=CC(=O)NCC1CCC1NC(=O)C(C)C1CC1 C1(C(=O)OC)CC(C)N(C(=O)C(C2CCC(C)(C)CC2)C)CC1C C1(C2CCN(C(=O)CC3CCCCC3O)C2)(NC(C2CCCO2)=O)CC1 c1(C(N(CCN(C(C(C)OCC)=O)C)C)=O)sc(C2CCCCC2)nc1C c1(OC)cc(C(N2CCC(NC(=O)C=C3CC3)C(CO)C2)=O)ccc1Br N1(C(C(=O)N(C)CC2CC23CCOC3)=O)CCC2CC(O)CCC2C1 CCCCCCC(C)C(=O)N1CCC(CC)C1C(=O)NCCCC(C)C C(=O)(CCCC(C)(C)CC)NCC(CNC(c1n(CC)cnn1)=O)C CC1CN(C(c2cc(C#N)n(C)n2)=O)CCN1C(=O)Cc1ccc(Cl)c(Cl)c1 CC1(C)CC(CNC(C2(C)CCCS2)=O)CN1C(=O)Cc1cccnc1 C1(CC)C(C(=O)NC(C)Cc2nc[nH]n2)CCCN1C(c1coc(C)c1)=O CCCCCC(C)CC(=O)N1C2CCC1CN(C(=O)Cn1ncnn1)C2 c1(C(=O)NC(CC(C)NC(c2cncc(C)c2)=O)C)cc(N)nc(Cl)c1 CCC(CC(F)(F)F)C(=O)NC(CNC(=O)CC1CCC1)C1CCC1 C=C1c2ccccc2C(=O)N1CCC(=O)NCC1OCCC12CCNCC2 Cc1c[nH]c2ncnc(N3CCC(C(N4CCCC(CO)CC4)=O)C(O)C3)c12 c1(C(C)Nc2c(C)ccc(OC)c2)oc2ccccc2c1C C1(NC(C2C(CC)CN(C(C3CCS(=O)CC3)=O)C2)=O)CCOC12CCCC2 C12(CCNC(CC3(C=C)CC3)=O)CCC1CN(C(C1(C)CS(=O)(=O)C1)=O)C2 c1(C(N2CCC(C3N(C(C4CCC(CC)O4)=O)CCC3)C2)=O)cccc(OC)c1 C(=O)(C(COC)NC(C)=O)N(CCC(=O)NC(COC)(C)C1CC1)CCCO c1(C(=O)NC(C)CCNC(=O)CCC2CCN(C)CC2)c[nH]c(=O)c2ccnn12 C1(CC)CN(C(C2(CCOC)CCC2)=O)CCN1C(=O)CCn1ccnc1 c1(C(N2CC3C(NC(C4CCC(=O)C4)=O)(C3)C2)=O)cc2nc(Cl)ccc2s1 N1(C(=O)OCC)CCC(C(=O)Nc2cn(Cc3cnn[nH]3)nn2)C1C(=O)O C1(NC(C(C(C)C)SC)=O)CC2(C1)CN(C(c1occc1C(C)C)=O)C2 Cc1cc(C(=O)NC2(C)CC(NC(=O)C(C3CCC(=O)N3)C)C2)co1 C1(C)(NC(C(c2ccc(OC)cc2)C)=O)CCCN(C(c2c(Cl)cnn2C)=O)C1 c1(C(=O)NC2C(C)CCN(C(C(CNC(C)=O)(C)C)=O)C2)cc(S(N)(=O)=O)co1 Cc1cc2ccc(C(=O)NCCC3CCCN3C(C3CCCCCC3)=O)cc2o1 C1(CCNC(CCC2(NC(c3c(CC)ncs3)=O)CCC2)=O)CCCC2CC12 C1(CNC(C2C(C)C2)=O)CCCCN(C(=O)C(C)(C)COC2CCCC2)C1 n1(CC)nnc(C(=O)NC2(CCNC(C3(COC)CC3)=O)CCCCC2)c1C C(=O)(CCCC(C)CO)OC(C)C(C)(C)CNC(c1c[nH]nc1OC)=O c1(C(=O)NCCC(C)NC(C2C3(CC(OCC)C3)C2)=O)c[nH]c2c(C)cccc12 N1(C(C(C)C2CC2)=O)CCC2(NC(c3ccc4ocnc4c3)=O)CCCC12 C1(NC(c2n(Cc3sccc3)nnn2)C2CCSC2)CC2CCCC2C1 CCC(C#N)C(=O)NC1CCCC1NC(c1cc(C(N)=O)cs1)=O Cc1ccc(C(C)(CNC(=O)N(C2CC(O)C2)C)CO)cc1 C1(NC(C(C)C(C)O)=O)COC2(C1)CN(C(c1ccc(O)c(F)c1F)=O)C2 c1(CC(=O)NCC2C(NC(CCC(=C)C)=O)CC2)ccc2nc(O)[nH]c2c1 c1(N2C(=O)CC(NC(CC)Cc3ccc(Cl)cc3Cl)C2)cc(F)c(C)c(F)c1 N1(C(c2nc(C)nc(O)c2)=O)CCC2(CC1)OCCC2NC(C1CCC1(C)C)=O C1(NC(N(CCC#N)CCOC)=O)(OC)CCCC(C(C)(C)C)CC1 C1(NC(=O)C(=O)NC2CCN(c3ccccc3)CC2)CCNC2(CC2)C1 CC1CCC(CC(=O)NCc2cc(C(=O)NCc3nccs3)cs2)O1 C1(NC(Cn2nc(C)c(Cl)c2)=O)CC2CCC1N2C(c1snnc1C)=O N1(CC)CCCCC1C.c12ocnc1C(=O)NC2.n1(CCN)cc(C2CC2)cn1 c1(CN2CCC(=CC(=O)N(C)CC#N)CC2)ccc(F)cc1C(=O)O N1(C(C2(C#C)CCN(C(=O)C(C)C)C2)=O)CC2(CNC(=O)OC2)C1 C1(NC(=O)CCn2cnnn2)CC2CC1N(C(C1(COCCO)CC1)=O)C2 C1(CC)C(C(=O)NCC2(CCO)CC2)CCN1C(c1c[nH]c(C#N)c1)=O C(C(C(=O)NCC(O)CC(=O)OC)C(C)(C)C)NC(c1cc(COC)on1)=O C1(C(N(CC(C)NC(=O)C(C)n2cncn2)CC)=O)CC(CC(=O)OC)C1 c1(C(=O)NC(CNC(C(CC#C)C)=O)(C)C2CCC2)cnc(O)c2cnccc12 CC(CC(=O)NC1CCC12CN(C(c1cc(CS(C)(=O)=O)on1)=O)C2)C(F)(F)F CC1CCN(C(c2cnc(N)c(Cl)c2)=O)CC1CNC(C1CCCN1C1CC1)=O N1(Cc2cc(OC)ns2)CC(NC(c2occc2Br)=O)CCC1C N1(C(C2CC(OC)C(OC)C2)=O)CCC(F)(CNC(=O)C(F)C(F)(F)F)CC1 Cc1n[nH]c2cnc(C(=O)NC3CN(C(c4ccc(Cl)cn4)=O)CCC3C)cc12 c1(-c2nc(CC(CC)C)nn2CCCOCC(F)(F)F)ccc(Cl)c2occc12 c1(C(=O)NC2CCN(C(CCCCOC)=O)CC2F)cc(C)c(C)nc1C C1(CN(C(=O)CC2CC2C)CC)CCN(C(c2cc(C3(C)CC3)on2)=O)CC1 N1(C(C(CC#C)O)=O)CCCC(C)(C)C1CNC(=O)CSC(C)(C)C c1(C(=O)NC2(CNC(C(C)n3cnnn3)=O)CCOC2)cc(Cl)ccc1N C1(CCNC(CCC)=O)CN(C(c2cnc(C)cc2Cl)=O)CCS1(=O)=O Cc1nc(NC2CCCN(C(C3CCc4cncn4C3)=O)C2)c2ccsc2n1 c1(C(N(C2CCCN(C(C3CCN(C)C3=O)=O)CC2)CC)=O)nccc(Cl)c1F C(=O)(CC(CC)C(C)(C)C)N1CC(O)(CCNC(C(CC)=CC)=O)C1 c1(NCCC2CCN(C(C3(C)CC3)=O)CC2)nc2c(cc1C#N)CCC2 C1(NC(c2ccn(C(F)F)n2)=O)(CO)CCCN(CCN2CC3CCC2C3)C1 c1(C(N2CCC(F)(C(=O)NCC(c3cc(C)sn3)=O)C2)=O)c(F)cc(F)c(F)c1F C1(N(CCC)C(C23CCC2C3)=O)CCN(C(=O)CSc2nncs2)CC1 Brc1ccc2ncc(CN3CCCC4(CCO4)C3)n2c1 C(C)(CCCNC(c1ccnn1CC(C)C)=O)NC(C1(C#C)CC1)=O c1(NC(C(C2CC(C)OC2)N2CCC(CN(C)C)C2)=O)ccccc1Cl c1(C(N2C(CNC(C(C)(C)OC(C)C)=O)C=CC2)=O)c(Cl)cccc1Cl c1(NC(C(c2ncc(Br)s2)N(C(C(=O)NCCOC)C)C)=O)ccc(F)cc1C C1(NC(CC2N(C)C(=O)CC2)=O)CC2CCC1(NC(=O)COC1CCOC1)C2 C1(NC(=O)CN(C(=O)C(F)F)C2CC2)CCOCC1O c1(C(N2CCN(C(CC3C(CC)C3)=O)CC2CF)=O)cc(N)c(Cl)c(O)c1 Cc1cc(C(=O)NC2CN(C(=O)Cc3cncc(O)c3)CC2C)n2ncnc2n1 C1(NC(=O)Cc2noc3ccccc23)CN(C(=O)CC(F)F)C2(CCCCC2)C1 C(=O)(C(C(CC)=Cc1cccnc1)N(C)Cc1ccncc1)NCC c1(C(=O)NC(C(C(C)C)NC(CCSCCC)=O)C)cc(Cl)ccc1C Cc1cc(Cl)cc(Cl)c1OCC(N1CC2CC(NC(=O)C=C(Cl)Cl)CC2C1)=O c1(CC(C)NC(C2C(NC(=O)C=CC3CCC3)C2(C)C)=O)cnn(C)c1 C1(N(C(C(C2CCCOC2)OC)=O)CC2CC2)CCN(C(=O)C(C)(C)CO)CC1 c1(NCCC(=O)N(C)C)ccc(S(=O)(=O)NCC2CCN(CC(F)F)C2)c(Cl)c1 C1(CSCCOC)(OC2(n3cc(CC(=O)OC)nn3)CN(C(C)=O)C2)C=CCC1 N1(C(CCSCCCC)=O)CCCC2(CCN(C(=O)CCn3cnnn3)CC2)C1 c1(C(=O)NCC2N(C(COC(CC)(C)C)=O)CCC(C)C2)nnn2c1CCCC2 C#CCC(C)(C)C(=O)N1CCC(C)C(CNC(C2(CC(C)C)COC2)=O)C1 CC1C(NC(c2ccc3c(c2)CC3)=O)CCCN1C(=O)C(C(C)(C)C)NC(N)=O CC1=C(C(=O)N2CCC(F)C(NC(=O)CC3CC(C)(C)CO3)C2)CCCO1 c1(C(N(CCNC(C(C)(C2CCC2)OC)=O)C)=O)nccc2occc12 N1(C(C2(OC)CCSCC2)=O)CCC(NC(=O)C=Cc2ncc(C)[nH]2)C(CO)C1 C1(NC(CC(C=C)C)=O)CCC2(CC1)CC2NC(c1cc(O)cc(Cl)c1)=O c1(C(=O)NCC2N(C(C3C(C)C3)=O)CC(F)(F)C2)cn(C)cc(Br)c1=O C1(NC(c2n(C=C)nnc2)=O)CN(C(c2scnc2Cl)=O)CC1C1CC1 N1(c2nc3c(N4CCCC4)cccc3s2)C2CC3C4CC(C3C2O)C4C1 N1(C(CN(CC)CC)=O)CCN(C(=O)C(C)(Cl)Cl)CC1c1cccc(OC)c1 CS(=O)(=O)C1CCC(CC(c2ccccc2)CNC(=O)OCc2ccccc2)CC1 C1(NC(C(CC)(C)OC)=O)CCC2(CC1)CC(NC(=O)C=Cc1cn(C)nn1)C2 c1(C(=O)NCC(Cc2ccccc2)NC(C(C(C)C)F)=O)cccc2ncoc12 N1(C(c2nc(C)sc2C)=O)CCC2CC(CNC(=O)CNC=O)CCC2C1 CC1(C(=O)NCC2(C(N)=O)CN(C(c3ccnc(Cl)c3N)=O)C2)CCCCCC1 c1(C(=O)NCC(C)N(C(c2ccc(C)cn2)=O)CC)cc(OC)cc(C)c1 N1(C(=O)N(C)C)CCC2CN(C(=O)COC(c3cc(C)c(F)nc3)=O)CC12 N1(C(C2COC(C)(C)O2)=O)CCCC(C2(NC(=O)CN3CCNC3=N)CC2)C1 c1(C(=O)NC2(CCNC(C3(CC)CC3(F)F)=O)CCCC2)ccc2sccc2c1 n1(CCCC(=O)NCC2(CNC(C(C)N(C(C)=O)C)=O)CCC2)cnc(C#N)n1 C1(C2CN(C(=O)CCc3cn(C)nn3)C2)(NC(CC2N(C)CCC2)=O)CC1 c1(C(C(=O)NCC2(F)CC(NC(c3cc(C)n(C)n3)=O)C2)O)ccc(Cl)c(F)c1 C(=O)(NNc1oc(CC(C)C)nc1C#N)N1C(CC)CCC(C)C1 c1(CC(=O)NCC(CC2CC2)C(=O)OC2(C(=O)OCC)CC2)ncc(F)cc1F c1(C=O)ccc(CCN)cc1.C(=O)(CCC1CC1)N(C1CCSC1)C N1(C(C(P(C)(C)=O)O)=O)CCC2(CCC2)C(CNC(=O)CC2(O)CCCC2)C1 C12(CNC(C3CCS(=O)CC3)=O)CCCC1N(C(c1ccccc1F)=O)CCC2 N1(C(CC2N(C(C3C(C(C)C)CCO3)=O)CC2)=O)CCC(N(C)C)(CO)C1 C#CCC(CC(=O)N1CC(C)(C)CC1CO)NC(=O)C=CCO C(CCCCCNC(C1CC12CC(NC(=O)CC1CCOC1(C)C)C2)=O)N(C)C C(C1CCCN1C)=CC(=O)NCCN(C(c1nc(Cl)cs1)=O)CC CCCCS(=O)(=O)NC(C)C(=O)NC(C)CNC(c1cn(C(F)(F)CO)nn1)=O c1(C2CC2)ccc(N)c(C(=O)NCCNC(C2(C(C)(F)F)CCC2)=O)c1.COC CC(N=[N+]=[N-])C(=O)NC1CCCC(CNC(C2CCC(CCO)CC2)=O)C1 C1(NC(Cn2c(CCC)ncc2)=O)(CC)CCN(C(c2cc(CC)no2)=O)CC1 O=Cc1sc(CNCCC2CC3C=CC2C3)c(Br)c1Br CN1C(=O)CCN(C(=O)Nc2c(Cl)ccnc2C(=O)OC(C)(C)C)c2ccccc21 C(=O)(C1=CCS(=O)(=O)C1)N1CCCC(NC(C=Cc2ncn(C)c2)=O)CC1 c1(C(N2C(C)CC(NC(C3(c4ccc(F)cn4)CC3)=O)C2)=O)ccc(N)c(F)c1 N1(C(CN2CCN(CC)CC2)=O)CC(C)N(C(=O)CNC(=O)NC2CC2)CC1C C(=O)(CC(C)CC(C)C)NCC1N(C(c2cccc(CC)c2)=O)CC(O)C1 CC1(C)C(NC(=O)CSC2CC2)CC1CN=c1[nH]nco1 CC1(NC(c2cccn(O)c2=O)=O)CCCN(C(=O)CCn2ccnn2)C1 C(CC(C)C)(C(=O)NC(CNC(=O)C=CC=C(Cl)Cl)CC(C)C)NC(C)=O N1(C(CC(CC)(C)C)=O)CCCN(C(c2coc(-c3ccccc3)n2)=O)C(C)C1 N1(C(C)=O)CCc2c(sc3nc(CNCC(O)C(C)C)nc(O)c23)C1 c1(C(C(=O)NCCCN(C(C(C)(C)SC)=O)CCO)F)cccc(C)c1 Cc1ccc(Cl)c(C(=O)NCC23CC(CNC(=O)C4=COCCC4)(CO2)C3)c1 C(=O)(C1=CC2(CCOC2)C1)N1CCC(NC(=O)C=Cc2ccc(Cl)cc2)CC1 Cc1ccc(NC(=O)C(C2CC2)NC(c2cccc(Cl)c2)=O)c(C)c1O CC1(C)C(CNC(=O)CN2CCN(C(c3ccc(O)cn3)=O)CC2)C1(C)C N1(C(CCCSC)=O)CCC(C(=O)NCC2CC3(CCCO3)C2)C(C)(C)C1 c1(C(CNC(=O)CCC2CC(C)CS2)OC)ccccc1C(F)(F)F C1(CC=C)(NC(c2ccc(C)c(C)n2)=O)CCCN(C(=O)C(N)=O)C1 N1(C(c2ccc(O)cc2OC(F)(F)F)=O)CCOC2CN(Cc3cscn3)CC12 c1(C(C(=O)N(CC(O)CNC(=O)CCc2ccccc2)C)OC)ccccc1Cl C#Cc1c[nH]nc1C(=O)NCC1(CC(=O)NCCC(C)C=C)CC1 Cn1ncc(C(=O)OC)c1CN(CC(=O)O)C(C1CSCCN1C(=O)CCCC#N)=O c1(CC)cc(C)[nH]c(=NCC2CCC(NC(=O)C(C)S(N)(=O)=O)CC2)n1 C1(C(N(C2CCN(C(=O)CC3CCC(C)CC3)C2)CC)=O)CC(=O)NC(=O)N1 N1(C(C(C)N(CC)CC)=O)CCC(C(=O)NCC#CC#CCO)C12CC2 c1(COC)ccc(C(=O)NCC(=O)N(C)Cc2nnc(C)o2)o1 N1(C(C(CC=C)N(C)C)=O)CC(NC(=O)CCCC(OC)OC)CC1(CC)CC c1(C(C)C)cccc(NC(C2CCCC2NC(=O)CN2C(=O)CSC2=S)=O)c1 CCC(F)(F)C(=O)NCCCN(C(=O)CC(n1nc(C)cc1C)C)C N1(C(c2cccc(CC)c2)=O)CC(F)(F)CC1C(=O)NCC(c1cnn(C)c1)O c1(NC2(c3n(CC=C)nnn3)CC2)ccc(NCc2ccccc2)cc1 CCCC(CCCNC(=O)CC1(O)CCCCC1)NC(=O)C(CCSC)OCC C=CC(C)(C)CCNC(=O)N(C)Cc1ccncc1C Cn1ncc2c1CCN(C(C1N(C(c3cncnc3)=O)CCCC1(C)C)=O)C2 CC1(C(=O)NC2CCC(CNC(=O)CC(F)(F)F)CC2)CCC12CCC2 C(CO)(C(=O)NCc1cc(C(=O)NC2(c3nc[nH]n3)CCC2)cs1)OC C(=O)(C(F)CC(C(=O)OC(C)(C)C)NS(=O)(=O)c1ccc(I)cc1)OC c1(C(=O)OC)ccc(C#CC=O)cc1.c1(CCCC2CCCC2)cccnc1 C1(C(=O)NCC2CCC(=O)N2)CN(C(=O)CCc2cn[nH]c2)CC12CCC2 c1(CN2CC(CC(=O)Nc3cc(C(F)(F)F)no3)C2)ccccc1Br C(=O)(C1=COc2ccccc2O1)N1CC(CNC(c2cn(C)[nH]c2=N)=O)OCC1 N1(C(C(COCC)C)=O)CCCCCC1CNC(=O)CC(F)F c1(C(=O)NC2C(NC(C(C)OCCOCC)=O)C2)c(N)ccc(F)c1C C1(CNC(COCC(=C)C)=O)CC(C(=O)NCc2ncn(C(C)C)n2)CO1 n1(CC)nnc(C(=O)NC2(COC)CCN(C(c3conc3C(C)C)=O)C2)c1C C(=O)(C1CCCc2nccn21)NC1CCN(C(c2ccc(C#N)o2)=O)CC1CO C(=O)(CS(=O)(=O)c1ccccc1Cl)N(C(=O)CC1CCCC(F)C1)CC(F)F Cc1oc(C#N)cc1C(N1CCC(CNC(=O)C(C2CCC(=O)N2)C)C12CC2)=O c1(CC(=O)NC2(CNC(=O)C=Cc3ncc[nH]3)CCCC2)ccc(Cl)cc1 C1(NC(c2ccnc(C)c2C)=O)CN(C(=O)CC2CCC2)CC(F)(F)C1 C(=O)(CCCN(C)C(c1cscc1OC)=O)NCC(C1CC1)SC C(=O)(C(C(C)(C)C)SC1CC=CCC1C)NC1C(c2cn(-c3nc(C)sc3)nn2)C1 Cc1nc2c(CC(=O)OC3CCCCCCC3)cccc2o1 CC1CN=C2NC(C(=O)N3CC4(C3)CN(C(c3ccc(Br)o3)=O)C4)=NN2C1 n1(CC(N2CC(NC(COCC#C)=O)C3C2C3)=O)ccc([N+](=O)[O-])n1 C12(CCCCC1)CC(=O)N2.CC(C(=O)NC1CC1)N1CCCC1 C1(NC(C(N2CCC(Cn3c(C)ncc3)C2)=O)=O)CC2CCC1O2 c1(C(N2CC=CC(NC(c3cncs3)=O)C2)=O)[nH]nc2ncnc(O)c12 C1(NC(CCCSC)=O)CC(C2CCN(C(c3cc(C)nc4ccnn34)=O)C2)C1 N1(C(C(c2ccc(N)cn2)C)=O)CC2(C)CN(C(C3CC(O)C3)=O)CC2(C)C1 C1(NC(=O)CSC2CCOC2=O)CN(C(c2ccnc(C3CC3)c2)=O)CC1O N1(C(c2scc(OC)c2)=O)CC2(CCC(CNC(C3CCC(C)C3)=O)O2)C1 C1(=CC(=O)NC2(C)CN(C(C3(CC)CC3(F)F)=O)C2)CN2CCC1CC2 c1(C(N(C(C)CNC(c2cn(C)nc2C2CCC2)=O)C)=O)ccc(Cl)c(C#N)c1 C(=O)(C1Cc2ccc(Cl)cc21)NC(C1CCCN(Cc2nccc(C)n2)C1)C CC1CC2(CCO1)CC2C(=O)NCC1C2CN(C(=O)CCCc3nccs3)CC12 c1(C(=O)NC2CC(n3cc(-c4cn(C)nn4)cn3)C2)ccc2nnn(C)c2c1.CC CC1CCC1N=c1[nH]c2ccc(S(=O)(=O)N(CC(C)(C)CO)C)cc2s1 c1(C(N(c2nc(C)cc(OCC)n2)C2CC(N)C2)=O)c(F)cc(C#N)cc1F c1(C(N2C(C)CC(NC(c3c(NCC)scn3)=O)C2)=O)cc(C)cc(Cl)n1 C1(CNC(=O)C(=O)NC2CC2)CCN(C(=O)CN2CCOCC2)C1 Cn1ccc(-n2cnc(C(=O)NCCNC(=O)CCN(c3ccncc3)C)c2)n1 Cc1cc(C)n2ncc(C(=O)NCCC(C)N(C)C(C3COC3)=O)c2n1 C1(NC(C(C)(C)n2cc(Cl)cn2)=O)COCCN(C(C2COCCC2(F)F)=O)C1 c1(C(C(=O)N(C)Cc2ccccn2)NC(=O)Cn2cccc2)ccc(F)cc1 C1(C(=O)NCCCNC(c2cc(C(F)F)[nH]n2)=O)CC2CC1CC2O N1(C(CC(CC)OC)=O)CC(C2CN(C(=O)C(CC)CCOC)C2)C1 CC1CNc2c(C(=O)NC3CCCCC3CNC(c3csnn3)=O)cnn2C1 C1(C(=O)NCC(C)N(c2nc(COC)nc(O)c2)C)Cc2ccccc2O1 N1(C(C(CC)(C)F)=O)CCCCC2(CCN(C(c3cc[nH]c3C)=O)C2)C1 N#Cc1ccc(CN2CCC=C(C(=O)NCCc3ccc(Cl)cc3)C2)c(Cl)c1 Cc1nc2ncnn2cc1C(=O)NC1CC(O)CN(C(=O)CC2CC=CCC2)C1 C(=O)(CCCC(=O)NC1CCCN(C(c2n[nH]cc2Br)=O)C1C)NCC c1(OC)cc(C(=O)NCCOC(C)(C)CNC(C2(N=[N+]=[N-])CC2)=O)ccc1F C(=O)(N=c1cc2n([nH]1)CCCC2)C1C(CC)N(C(C23C(=O)C4CC2C3C4)=O)CC1 c1(C(=O)NC2CC(C)(NC(C(CC)OC)=O)C2)n[nH]c2c1COc1ccccc1-2 n1(CC)ncc(C(=O)NCC2(C(N)=O)CN(C(=O)C(C)(C)SC)C2)n1 C1(CNC(C(CC)F)=O)CN(C(c2[nH]cnc2C)=O)CC(C)(C)O1 c1(SN2CC=C(C)C2)nc(C)cc(=NC(C)c2ccc(-c3cc(F)cc(F)c3)cc2)[nH]1 N1(C(c2cc3n(n2)CCO3)=O)CC2CCN(C(=O)Cc3cccc(Cl)c3F)C2C1 N1(C(CCN(C(c2c[nH]c(=N)o2)=O)C2CC2)=O)CCC(O)CC1 N(C1CCCc2n[nH]cc21)C(=O)NC1C(C2ON=C(C(=O)OCC)C2)CCCC1 C1(NC(C(C)SCC)=O)CCCCN(C(c2nc(C)c(N)cc2C)=O)CC1 N1(C(CC2CCC(NC(C(C)(C)N3CCCC3)=O)C2)=O)CCC=C(F)C1 C12(C(=O)NCCCNC(C3(C)CC3C(F)(F)F)=O)CC(C(F)(F)F)(C1)C2 C1(C(=O)NCC=CC(=O)N(C)Cc2occc2C)(CC)CCCCO1 C12(NC(C(C)O)=O)CC(CNC(c3cnn(-c4ccncc4)c3)=O)(C1)OC2(C)C C=CCC(C)(CC)C(=O)N1CCC(CCNC(=O)CCC2(C#N)CCC2)C1 C(=O)(CC(O)C(Cl)(Cl)Cl)N1CCC(NC(c2cc(C(C)C)c(N)cc2)=O)C1 CN1CCN(C(C2COCCO2)=O)C(CNC(c2cc3occc3[nH]2)=O)C1 O=C(N=c1cc(C(F)(F)F)[nH][nH]1)c1cnc(-c2cnn(C(F)F)c2)cn1 N1(CC)CCN(C(c2ccc(OC(F)F)cc2C)C(=O)NC2CCOC2)CC1C C(c1cc(C)no1)=CC(=O)N(CC(=O)NC(C)C(C)F)CCOC CCC(CCC(=O)N1CC(SC(F)F)C1)NC(=O)CCCCCOC C(=O)(C(CCc1cc[nH]n1)NC(=O)OC(C)(C)C)N1CC(O)(NC(=O)NCC)C1 C1(C)(CC(=O)NCCOCCN(C)C(C2CCCCO2)=O)CC(F)(F)C1 CCC(O)(CC)c1cn(CCCC(=O)N(CC(=O)OC)CCOC)nn1 c1(C(=O)NC(CN(C(c2cccc(OC)c2F)=O)C)C)coc2c(C)cccc12 N1(C(COC2(C)CCC2)=O)CCC(C2CC2)C1C(=O)Nc1cnc(C2CC2)[nH]1 N1(C(c2c(SCC)cncc2)=O)CCC2(CCC2NC(C2CCCO2)=O)CC1 N#CC1(C(=O)NCC2(C(F)F)CCN(C(c3ccn(CCF)n3)=O)C2)CC=CC1 N1(C(=O)OC)CCCC(N(C(CNC(=O)C=C2CCC2)=O)C)C1 C#Cc1ccc(Cl)c(C(=O)NC2(CNC(=O)C=Cc3sccc3C)CC2)c1 c1(C(=O)NC(C2CCN(C(=O)COCCCF)C2)C)cccc(-n2cncn2)n1 Cc1oc(C(=O)NC(C)CCNC(C2CCCCC2O)=O)cc1-c1ccccc1 Cc1cccc2c1OC(C(=O)NC1CC3(NC(=O)C4=CCCCO4)COC1C3)C2 C1(OC)CC(CNC(C2(CC3CC3)CCCO2)=O)N(C(=O)CC2CC3(CC3)C2)C1 c1(C(=O)NCCC(C)NC(c2c(OCC)oc(C)n2)=O)cccc2c1COCC2 c1(C(N2C(C)(CNC(c3cc(C)on3)=O)CCC2)=O)ncn2cc(Cl)ccc12 c1(C(=O)NC(CN(C(=O)C(C)CC(F)F)CC)C)cc(O)ccc1OC c1(C(C)NCc2ccc(OCC)cc2)ccccc1[N+](=O)[O-] N1(C(C2(Cl)C=CC(OC)=C2)=O)CCN(C(C2(CF)CCCOC2)=O)CC1C c1(C(=O)NC2CC(C)N(C(c3ccns3)=O)C2)c(F)cccc1Cl C1(NC(c2c(C)nsc2)=O)CCN(C(=O)C(C)NC(C2CCC2)=O)C1(C)C c1(C(=O)NCCOCCN(C(C(C)OCC)=O)C)cn2cc(C)nc2s1 C1(CC)C(NC(=O)C(F)CC2CCOC2)CCCN1C(C1CCOC1)=O N1(C(=O)C=C(Cl)Cl)CC2CCCN(C(=O)C3=CC4(CCOC4)C3)C2C1 NC1CC(CNC(=O)CCNC(=O)C=CCl)C12CCC2 N1(C(c2cc(O)c(F)cc2N)=O)CCC(C=O)=C(F)C1.CO C(C)(N(C)N1CCCN(C(C)C)CC1(C)C)c1c(C)c(Cl)ccc1 CC1CCN(C(=O)CCS(C)(=O)=O)CC1CC(=O)NOCC(C)(C)O C(=O)(C(C)(C)C(=O)N1CCC(NC(c2cc(O)ncn2)=O)C1)OCC S(=O)(=O)(c1cccc(C2(C(F)(F)F)N=N2)c1)NC(C1C(C)CC(=O)N1)=O CN1CCn2nccc2C1=O.C1(F)(n2c(=O)c2=O)CCOC1C.C(C)(C)(C)OC=O c1(C(N2C3CN(C(c4cc(N)c(F)cn4)=O)C(C3)C2)=O)cnc2ccnn2c1 N1(C(c2c(CNC(C(C)O)=O)cco2)=O)CC2(C1)CN(C)CCO2 Cc1c(C(=O)N(C)CC2CCCCN2C(c2ncccn2)=O)cccc1Br N1(C(COc2c(OC)cccc2)=O)CC(NC(c2cnnn2SC)=O)CC1(C)C CC(C)(CO)C(CO)NC(=O)C1=CCN(C(=O)C=CC(=O)NC2CC2)C1 C1(C(N2CCC(CN(C(CCSC)=O)C)CC2)=O)Cc2ccccc2S1 C=CCCCCCCCC(=O)NC1CS(=O)(=O)CC1NC(C1CCCCC1)=O C(=O)(CC(C)(C)Cc1cn(-c2ccc(Br)c(C)c2)nn1)OCC N1(C(c2cc(C)c(C)nn2)=O)CCC(NC(C2CN(C(C)C)C2)=O)CC(O)C1 Cc1ncc(CC(=O)NCCOC2CCN(C(=O)CC(C)N3CCCC3=O)C2)s1 Cc1cc(N)cnc1C(=O)N(CCCN(C)C)CCNC(=O)CC1CCCOC1 N1(C(C2CC(C)(CC)C2)=O)CCN(C(=O)C(C)SC(F)(F)F)CC12CC2 C1(CCC)(Nc2ncnc(O)c2Br)CCN(C(c2cc(Cl)ccc2C)=O)CC1 C1(CNC(CC2CC(N(C)C)C2)=O)N(C(=O)Cc2ccccn2)CCCC1(C)C c1(C(N(C2CN(C(=O)C(C)(C)c3ncco3)CC2F)C)=O)cc(Cl)cnc1O C1(C(=O)NCc2c(C(=O)NC(C(C)C)CO)occ2)C2CCC(C2)C1C C1(CNC(CCC(=C)Br)=O)C(C2CC2)CCN1C(c1cnc(C)c(N)c1)=O c1(N2CCCC(OCC)C2)ccc(Br)c(S(=O)(=O)NC(c2cc(C)nn2C)C)n1 n1(CC(=O)NC2(COC)CCN(C(c3c[nH]cc3C)=O)C2)cc(P(C)(C)=O)cn1 C1(C(N(CC#C)CC=C)=O)(CC)CCCN(C(=O)CC(C)C(=O)OC)C1 c1(OC)cc(C(=O)NC2CCN(C(c3cnns3)=O)C(C)C2)cc2c1OC(C)C2 Nc1c(C(=O)NC(CNC(c2cc(F)ccc2F)=O)C2CC2)cc(Cl)cc1Cl C(=O)(CCCC(=O)NCCC1CCCN(C(=O)C=CBr)CC1)NCCC c1(C(=O)NCCN(CCC)C(C)C)cnc2ncnn2c1C C1(NC(c2cnc(C)n2C)=O)CCN(C(C2(CN(C)C)CC2)=O)CC12CCC2 c1(C(C)NC(CNC(C)C(c2ccccc2)O)=O)cnn(C)c1 c1(C(CNC(C(C)(C2CCOCC2)OC)=O)O)ccc(Cl)cc1 C(=O)(C1=NOCC1)N1C(C(=O)NCC2CCCCC2)CCC1 N1(C(c2c(C)c3c(s2)ccc(F)c3)=O)CC(C)OC2(CCN(C(=O)C(C)C)C2)C1 c1(CC)cccc2[nH]c(C(N3CCC(CNC(C4CCO4)=O)C34CCC4)=O)cc12 C(N=c1[nH]c(-c2cc3cscc3s2)cs1)C1C(O)CC1 Cc1ccccc1OCCC(N1CCC(CNC(C2CCC(F)(F)C2)=O)C1)=O C1(C(=O)CC2(C(=O)NC3CC(C(=O)OC)C3)CCCC2)CN(C(C)C)CCO1 C12(N(C)C(C3CCCS(=O)(=O)C3)=O)CCCC1N(C(=O)CSS(C)(=O)=O)CC2 C1(C(=O)Nc2cccc(NC(C(c3n(C)cnc3)O)=O)c2)CCCC(C)(C)CC1 N1(C(C(C)OC)=O)CC2(C1)SCCC2NC(=O)CN(C)C(C)C c1(CC(N2C(C(=O)NC(C=C)CO)CC(F)C2)=O)cc(Cl)cc(Cl)c1 c1(C(=O)NCC2(CNC(CC(=C=C)C)=O)CCOCC2)cc(C2CC2)nc(O)c1 C1(C(=O)NC(c2cnn(C)c2)C(=O)N(CC(F)Cl)C)CC(C)(C)C1 C(=O)(CC=C(Cl)Cl)NC(C(=O)NCC1(CCC)CC1)C C(C(F)(C(=O)NCCc1nncs1)C(C)C)NC(C(C)(C)NC(=O)OC)=O N1(C(=O)C(c2cccc(Cl)c2)O)CCC2(CC1)CC2C(N1CCCCCC1)=O CC(CC(F)(F)F)C(=O)NCC1CCN1C(C1CCC(C)(C)C1)=O N1(C(C2N(N=O)CCC2)=O)CC2(CC(NC(C3(F)CC3c3ccccc3)=O)C2)C1 C1(NC(c2cnc(C3CC3)[nH]2)=O)CN(C(C2(Br)CC2)=O)CC1C1CC1 N1(C(C=CC(C)=O)=O)CCC2(CCN(C(=O)C(C)(C)S(=O)(=O)C3CC3)C2)C1 N1(C(c2n(CC)ccn2)=O)CCN(C(C2(C(=O)NC)CCC2)=O)CC1CO N1(C(N2C(c3c(C(=O)O)c[nH]n3)CCCC2)=O)CC2(CC(O)C2)C1.c1ccns1 c1(C(=O)NCCCCCN(C(C(C)NC(C)=O)=O)C)cc(Br)cnc1C c1(C(=O)NC2CC(NC(c3nn(C)c(O)c3)=O)C2)cc2cccn2c(O)n1 C(=O)(CC(C)(C)C(F)F)NCC1(O)CCN(C(C(=Cc2ccccc2)CC)=O)C1 c1(Cc2cn(C3CCCNC3=O)nn2)cc2ccccc2s1.C(C(=O)O)N(C)N c1(OC)c(C)cc(-c2csc(NC(=O)C(C)(C)C(N)=O)c2)cc1C C1(NC(CCc2nnc(C)n2C)=O)CC12CCN(C(C1COC(=O)N1C)=O)CC2 CC1CCCc2c(C(N3CCCCC3CN(C)C(C3(CO)CC3)=O)=O)cnn21 c1(C(C(=O)NC2(CC3CCC3)CC2)(F)F)ccc(F)cc1Cl c1(C(N2C(C(N(CC=C)CC=C)=O)CC(F)(F)C2)=O)cc2ccccn2n1 C1(CNC(C(C2CCN(C(C3(F)CC=CCC3)=O)CC2)C)=O)CC2CCCC2C1 S(=O)(=O)(c1cc(C(F)(F)F)cc(Br)c1)NC(CCCC)(C)C(N)=O N1(C(c2cc(CC)ncn2)=O)CC2CC(O)C1C2NC(c1coc(C)n1)=O C1(CC)CN(C(=O)CCc2cc(C)no2)CCC1NC(=O)Cc1n[nH]c(=N)s1 c1(OC)cc(C(C)Nc2cc(C(=O)O)c(C)c(Br)c2)c(F)cc1F C1(NC(C=CC)=O)CCCCC1CNC(=O)CCCN1CCCC1 C(=O)(C1CCCn2cc(C)nc21)NC(CNC(Cc1cn(CC)nc1)=O)C1CC1 c1(C(=O)NC2CN(C(c3cnc(CCC)s3)=O)C(C)C2)cc(CC)ccc1N N1(CC)CCCCC1C(N1CC(OC)C(C(=O)NCCOCC(C)(C)O)C1)=O CC1(C)CC(C)(C(=O)NCCOC(C)(C)CNC(=O)CCC2CC2(Cl)Cl)C1 C(C)(CC(=O)NCC(C)(C)CNC(=O)C(F)(F)c1cnn(C)c1)OC Cn1[nH]c(C(=O)NCC(C(C)(C)C)NC(=O)CC2CNC(=O)C2)nc1=O c1(C(=O)NC2CCCN(C(c3c(C)noc3)=O)C2)n[nH]c2c1CCSC2 C#CC1CCCN(C(=O)C(F)CC2CN(C(C3C(=C)C3C(=O)OC)=O)C2)CC1 c1(NC(=O)NC2CN(C(C)=O)CC2N=[N+]=[N-])c(Cl)nc2ccccn12 N1(Cc2n(C)c(NS(=O)(=O)C(F)(F)F)cn2)CC(=O)N2CCCC2C1 N1(CC(CCOC)(C)C)CC2(CCCC2)CC1CO C1(C(=O)NC2CN(C(CCc3ccc(CC)cc3)=O)CC2C)CC(C)(C)CN1C c1(C(=O)NC(C(C)NC(C(CCCC)C)=O)C)cc(C)c2ncccc2c1 Cc1cc(C)c(CNCC2CN(C(C3(c4ccccc4)CC3)=O)C2)c(O)n1 c1(N(CC)CC2CCN(C(C3CC(O)C3)=O)CC2)cc(C(C)C)nc(Cl)n1 CC1(C(N2CCC(CNC(=O)C(F)F)C2)=O)CCCCCC1 CC1CCCN(C(c2n[nH]cc2CNC(C2CCNC(=O)C2)=O)=O)C1CO C(C)(C(CO)NC(C1CCS1(=O)=O)=O)NC(CCC1CC(OC)C1)=O c1(OCC)cncc(C(N2CCC(CCNC)C2)C(=O)NC2CC2)c1.C1CCO1 c12nc(=N)[nH]cc1C(=O)N1CCCC1C1CC1NC2.C(=O)(CCOC1CC1)OC C(=O)(C(C)(C)N)NCCN(C(=O)CN(S(=O)(=O)CC)C)C(C)C.CC Cc1ccc(O)cc1NC(=O)CCN(C(=O)C(C)C(C)(C)C)CCCO CCC(CNC(=O)Cc1cnn(C)c1)(CC)C(=O)NCC1CC(=O)N(C)C1 N1(C(C=C(CC)C)=O)CCC(CO)(NC(C2CCC(C(=O)OC)C2)=O)C1 c1(C(=O)NCC(CNC(C(CC=C)OC)=O)(C)F)cccc(O)c1F C1(C(N2C(CN(C(c3nc(CC)sc3N)=O)C)CCC2)=O)CCCCC12CCC2 c1(C(C(=O)NCC(=C)C)N(CC(C)CC)CC)ccc(Cl)cc1Br c1(NC)cccc(C(=O)NC(C2CCCN2C(c2csc(C(F)F)n2)=O)(C)C)n1 C12(C(N(C(CC)CNC(c3ccc(C)c(C)n3)=O)C)=O)CCCCC1C2(F)F c1(C(=O)NC2CN(C(C3(OC)CCSC3)=O)C2)ccnnc1C n1(CC)nncc1C(=O)NC1CCC(CCNC(=O)CCc2n[nH]c(=N)s2)C1 C1(CNC(C(C)n2ccnc2)=O)CCC12CN(C(=O)Cc1nc([N+](=O)[O-])n[nH]1)C2 c1(CNC2C(C(=O)NCCC#C)CCC2)cc(Cl)cnc1OCC Cc1ncncc1C(N1CC=CC1C(=O)NCC(C)O)=O C12(C(=O)NCCC(C)NC(c3cnccn3)=O)CC(CC(F)F)(C1)C2 C1(C(N(CC(=O)N(C2CCC2(F)F)C)C)=O)CCCCC1 C(CN=c1nc2sccc2c(NCC2CCC(O)CC2)[nH]1)(C1CCCCC1)OCC c1(CC(=O)Nc2cc(C(F)(F)F)cc(Cl)c2)cc2ccccc2o1 CCCC(CC)C(=O)N1CCN(C(c2cn(C)nc2C)=O)C(c2ccnn2C)C1 C1(NC(CC(=C)C)=O)CC(C2CCN(C(c3cc(O)ccc3F)=O)C2)C1 C1(C(=O)NC(C2N(C(C(CC=C)NC(C)=O)=O)CCC2)C)CC2(CC(OC)C2)C1 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CC2(C(NC(=O)Cc3cccs3)CCC2)C1 CC(C)C(O)C(F)(F)C(=O)NCC(C1CC1)N(C)C(C1(CCF)CCC1)=O C1(CC)CN(C(=O)CCCCN(C)C)CCC1N=c1[nH]nc(C2CC2)s1 CN1CCN(CC(=O)NCC2(CO)CCN(C(c3cnc(Cl)s3)=O)C2)CC1 N1(CCNC(c2csc(Cl)c2)=O)CCN(C(C2(C(F)(F)F)CC2)=O)CC1 N1(C(C2CC(=C)C2)=O)CCCC(CO)(NC(c2cc(C#N)oc2C)=O)C1 C1(N(C(c2c(C)cc(C)nc2)=O)C)CCN(C(C2C3CCCC23)=O)CC12CC2 C1(NC(CSc2c(OC)cccc2)=O)CN(C(=O)CCC2CC2(F)F)C(C)(C)C1 C1(NC(C2CCC(C)C2)=O)CC1C1CCCN(C(c2cc3sccc3s2)=O)C1 C1(CNC(c2scc(C)c2)=O)CCCCN(C(c2ccnc(Cl)c2O)=O)C1 Cc1nc(NCC(O)CNC(=O)Cc2ccc(O)nc2)c2c(C)csc2n1 C1(CC(=O)N(CCNC(c2csc(COC)n2)=O)CC)CCC(=O)N1C C1(CNC(C(C)=C2CC2)=O)CCC(C)N(C(c2csc(O)n2)=O)C1 C12(COC)CC(CNC(c3cccc(O)n3)=O)(CN1C(C1CC1CF)=O)C2 c1(C(N2CC=CC(NC(C3(CC#C)CCCO3)=O)C2)=O)cncc2sccc12 C1(C#N)(C(N(CC(C)(C)NC(C(CC)NC(C)=O)=O)CC)=O)CC2CC2C1 c1(C(=O)NCCn2cc(C(C)(C)O)nn2)ccc(SCC(=C)C)cc1 C(=O)(C1=CS(=O)CCC1)N(C1CCCN(C(=O)CCC2CCC2)C1)CC C1(CNC(C=C(C)C(F)F)=O)CC2CCC1N2C(c1cc(C(F)F)[nH]n1)=O Cc1nc2ncc(C(=O)NC3CCN(C(c4cc(F)c(N)c(F)c4)=O)C3)cc2o1 C1(NC(C(CC)N(C)C)=O)CN(C(=O)Cn2ccc(=O)cc2C)CC12CCCC2 C1(CCCNC(c2c(CNC(C3CC3C(C)C)=O)cco2)=O)(COC)CCCC1 CC1CNCC(CN2CCC(F)(C(=O)N(C)C)C2)C1 c1(OCCC(=O)NCCC2CN(C(C(CC#C)C)=O)CC2C)ccc(F)cc1F N1(C(c2c(C)onc2C2CC2)=O)CC(NC(=O)CCc2nc[nH]n2)C2(CCC2)C1 Nc1ccc([N+](=O)[O-])c(C(N2CC(OCCNC(=O)CCC3CC3(F)F)C2)=O)c1 C1(NC(C2(C)CCCOC2)c2nnnn2CCOCC2CC2)CC1C1CCOCC1 N1(C(C(C)=CC2CC2)=O)CCCC(C)(C)C1CNC(C1CC12CCCCC2)=O CCCC(C(=O)N(CC(C)C(C)C)C)NC(=O)CC1(O)CCOC1 CC(C)C(C)(O)CNC(C1(C(C)NC(C2COC(=O)N2)=O)CC1)=O C(=O)(CC(F)(F)C(F)(F)F)NCCC1CCN(C(C(C)(CO)OC)=O)CC1(F)F Cc1ncc([N+](=O)[O-])n1CC(N1CCC2(NC(=O)Cn3cnnn3)CC2C1)=O C(=O)(C1=CCOCC1)N(CC)CC1CCCCN1C(=O)CCCN(C)C n1(-c2n(C)nnc2)nc(Cn2nccn2)nc1C1CC(C)(C)C1 c1(C(=O)NC(CC)CNC(=O)COC(C)(C)CC)nc(OC)cc(OC)n1 C1(C(CC)NC(c2cnc(C3CCCC3)nc2)c2nnnn2C)CCCCCC1 c1(OCC(=C)C)ccc(-c2nn[nH]n2)cc1OCCNC(=O)CN1CCCCC1 Cc1nn(C)c(-n2cncn2)c1C(=O)NCc1n[nH]c(-c2cccc(F)c2)c1C N1(C(C2N(C(C)C)CCC2)=O)CCN(C(c2c[nH]cc(Cl)c2=O)=O)C(CF)C1 C(=O)(C(C)(C)CCNC(c1ccnc(O)c1)=O)NCC=CC(C)(C)C C(=O)(C(F)C(F)(F)F)NC(C(=O)NC1(C2CC2)CC1)Cc1ccco1 c1(OCC)ncnc(OCC)c1C(N1CCC(NC(C2(F)CCCOC2)=O)C1)=O